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c1(C(=O)OC)ccc2nc(=NCCN3CCc4sccc4C3)[nH]n2c1 Cc1ccc(Br)c2[nH]c(C(=O)NCC(C)NC(c3cnn(C)c3N)=O)cc12 c1(C(=O)NC(C(C)NC(=O)C=CCN2CCOCC2)C)cc(Cl)ccc1O CC(c1cccnc1)=CC(N1CC(CNC(c2ccc(CO)s2)=O)CC1(C)C)=O N1(C(CCC#C)=O)CC(NC(=O)CNC(=O)CCNC(C)=O)CC1(C)C c1(CNC(C(=O)O)Cc2cccs2)cnc(-c2ccc(F)cc2)nc1 COCN1C(=O)CCc2cc(NC(c3cc4cc(C(C)=O)ccn4n3)=O)ccc21 c1(C(N2CCC(C(C)NC(C3(C)CC(F)(F)C3)=O)CC2)=O)ccn2c1CCCC2 Cc1csc2ncc(C(=O)NCC3CC4CCC(C3)N4C)n12 [SH](=O)(=O)c1ccc([N+](=O)[O-])c(F)c1.c1(C(=O)OC)cnc(NC(=O)C)cn1 c1(C(=O)NC2C(CNC(c3onc(C)c3C)=O)C2)nccc2c1NCCC2 N1(C(C2(OC)CCC(C)C2)=O)CCCC(CC(=O)N(C(C)C(N)=O)C)CC1 c1(NC(N2CCC(c3n(C)c(S)nn3)CC2)=O)ccc(CNC(N)=O)c(O)c1 c1(C(=O)NCc2cc(C(=O)NCCn3c(C)nnc3)no2)ccncc1O C(=O)(C(C)C1=CCCC1)NCC1(NC(C(C)OCC=C)=O)CCCC1 C1(C)(NC(C(C)N(C(=O)Cc2cncnc2)C2CC2)=O)CCCC1O C1(NC(c2ccccc2O)=O)CN(C(c2cc3n(c2)CCCC3)=O)CC2(CC2)C1 CCC(C(=O)N1CCCC1C(C)(C)C(=O)NCCN1CCCC1=O)NC(N)=O C1(C(=O)NCc2c(C)ncs2)CN(C(C2(C(F)(F)F)CC2)=O)CCC1(C)C C(=O)(CCCN(C(=O)C(C)n1cncn1)C)N1CC(CCOC)C1 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c1(C(N2CCC(NC(c3n(CC=C)ccc3)=O)C2)=O)ccc(CCC)cc1 Cc1nn(C)c(Cl)c1C(N1CCCN(CC(C)O)CC1)C(=O)NC1CCC1 Cc1csc(CC(=O)NC2C(C(=O)NCc3nncs3)C2(C)C)c1 C1(NC(c2c(CC)scc2)=O)CN(C(C2CC3(CCC3)CO2)=O)CC12CCC2 Cc1nc(Br)sc1C(=O)NCCC(C)NC(=O)C(C)NC(C1CCC1)=O N1(C(c2c(C)cc(F)cc2)=O)CCC(C2(NC(C3NC(=O)CC3C)=O)CC2)CC1 C(=O)(C1=CC2(CN(C(=O)Cc3cccs3)C2)OC1)NCc1c(C)c(C#N)ccc1 C1(OC)CCCCN(CC(=O)NC2CC23CC(NC(=O)C(C)(F)F)C3)C1=O C(C)(CCC(=O)NCCN(C1CCCCC1)C(=O)CCn1cnnn1)SC c1(C(c2n(CCSC)nnn2)NCC(C)(C)CCCO)cc2cccc(OC)c2o1 Cc1ccc(F)c(C(=O)NC2CN(C(C3CC3C(C)(F)F)=O)CCC2O)n1 CC1CC(C#N)(C(N2CCCC(CNC(C3CCC(C)CC3)=O)C2)=O)C1 N1(C(c2c(CC)cccc2C)=O)CCC=C(C(=O)Nc2ccc(C#N)s2)C1 c1(CC)ccnc(C(=O)NCCC(O)C(=O)NC(c2cnn(C)c2)CC)c1 C1(CC=O)CCOC1(C)C.C1(CC(=O)NC(C2(C)CC2)C)CCCC1O.N c1(C(NNC=O)=O)cc2c(cc1Cl)OCO2 c1(CN(C(C)C(C)N)CC)cc(Br)ccc1[N+](=O)[O-] C=CCCCC(C(=O)NOCC=CC)NC(=O)CCc1ncccn1 C1(C(C)NC(=O)Cc2ccnnc2)CCCN(C(c2ccc(CO)o2)=O)C1 C(N=c1[nH]c2cccc(F)c2o1)C1(O)CCCN(C(C(c2cnn(C)c2)C)=O)C1 c1(CC)cc(N)ccc1C(=O)N.C1CN(C(=O)C)CC1C(F)(F)F.C(C)C c1(OC)ccc2c(c1)C(C(=O)NC1CCCN(c3ncccn3)C1)CCC2 Cc1cccc(F)c1NNC(=O)C1(CN)CC2(C1)CC(F)(F)C2 N1(C(c2ccc(C)c(N)c2)=O)CCCN(C(=O)CC2CCCC23CC3)CC1C c1(C(C)OC)nc(C)c(C(=O)N(C(c2ccc(OC)cc2)C(=O)O)C)s1 C1(C(=O)NC(CCC(=C)C)C)CC12CCN(C(c1csc(C)n1)=O)C2 c1(C(=O)NC(CC)CN(C)C(C2CN(C)CC(C)O2)=O)cc2cc(Cl)ncc2[nH]1 C12(CNC(C(c3ccc(C)s3)C)=O)CC(C1)C(C)O2.c1(C(=O)N)cnn[nH]1 C1(C(=O)NCCC2N(C(CC3(C=C)CC3)=O)CCSC2)CCC2(CCC2)O1 c1(C(C)C(=O)N(CC(=O)NCCCNC(=O)N(C)C)C)ccccc1 c1(CCC(=O)O)cn(C2CCC(NC(C3(c4ccsc4)CC3)=O)C2)nn1 C1(CC(N2CCC(C)(C)C(NC(=O)C(N)=O)C2)=O)Cc2ccccc2NC1=O c1(C(=O)NC2CCCC(NC(c3ccc(O)cc3)=O)C2)cc(Cl)c([N+](=O)[O-])[nH]1 c1(C(N2CCCC(CNC(C(CC#C)C)=O)C2)=O)cc(C)n(C)c(=O)c1 N1(C(CC(C(C)C)O)=O)CCC(NC(=O)C(C)Cc2ccccc2)C(C)(C)C1 c12cc(ccc1F)C(=O)OC1CCN(C)CC1Sc1nncn1-2.CS N1(C(C(C)OC)=O)C2CCC1C(CO)N(C(c1ccc3nnn(C)c3c1)=O)C2 Cc1nc(C(=O)NC2C3CC2N(C(c2cccc(O)c2C)=O)C3C)c(=O)[nH]c1C C(=O)(C(C(C)C)C(C)C)NC1C(C=C)CN(C(=O)Cc2cncc(C#N)c2)C1 C(=O)(C(CCN(C)C)N(C)C)NCC(C)NC(c1ccc(NC=O)cc1)=O c1(C(N(C)CCN(C)C(C2CC2(C)C(F)F)=O)=O)ccnn1CCF c1(CC)ncc(C)cn1.C(CC1CCC1)(C=O)NC(C1CN(C(C)=O)C1)=O.N c1(C(=O)NC2C3CN(C(CC(C)C)=O)CC2COC3)ccc2cc(O)ccc2n1 C1(C(=O)NOCc2ccc(Cl)cc2)(NC(c2c(C)ocn2)=O)CCC(C)(C)C1 N1(C(C2(COC)CCOC2)=O)CCC2(CC1)CCCO2.C1(CC(=O)N)CCCC1 C=CC1(CC(=O)NCC23COC(C)(C2)C3)CCOCC1.C(=O)CC(O)CCC.N c1(OC)cc(C=CC(=O)N)cc(Cl)c1.c1ccc(C(=O)O)o1.c1cccs1.C c1(C(=O)NC2CN(C(CC3N(C)CCC3)=O)C2)c[nH]c2c(F)cc(F)cc2c1=O C(=O)(C(CC)C(F)(F)F)N(CC(C(=O)NCC(CCC)OC)(C)C)C N1(C(N2C(C)C(C)OCC2)=O)CCOc2ccc(Br)cc21 c1(NC2CCCN(C(C3(C)CCCOC3)=O)C2)ccc([N+](=O)[O-])cc1C(F)F Cc1ccc(C(C)(C)C(=O)NCCCN(CCC2CCS(=O)(=O)C2)C)cc1.O N1(C(c2nc(C)sc2)=O)CC=C(CNC(c2csnn2)=O)CC1 N1(C(CCS(C)=O)=O)CCC2(CCCN2C(c2ccc(Cl)cc2)=O)CC1 C1(CC=O)CCCC(C)C1.Cc1n[nH]cc1C(=O)NCCOCCO.CC O=C(N=c1ccn(C2CCSCC2)[nH]1)c1ocnc1S(=O)(=O)N1CCOCC1 CCCCCCC(C)NC(=O)CC(C)(C)N(C)C(C1(C)CCCC1)=O NC(CC1CCCC1)CC(=O)NCCCCn1cc(C2CCCCC2)nn1 CC1CC(O)CCN(C(c2cc(Br)c(F)cc2O)=O)C1 c1(C(N2CCCCC(CNC(c3cnsc3)=O)C2)=O)c(O)cnc2ccccc12 c1(CNC(C2C(CNC(=O)CCC3CCC3)CCC2)=O)cccc(O)c1F C1(CCNC(=O)CC2CCC(F)C2)CCCN(C(C2CN3CCC2CC3)=O)CC1 C1(NC(CC(C)(F)F)=O)CC2CCC(C1)N2C(c1ccc(N2CCCC2)cc1)=O N1(C(C(C)CC2CC2)=O)CCOC(C(=O)N(C)Cc2nnnn2C)C1 N1(C(C)=O)CCCC2CN(C(C3(C)CC(O)CN3C)=O)CC12.C1CCS(=O)(=O)C1.N CC1(C)CN(C(C2CCC(CN)C2)=O)CCO1.C(=O)CC1CC1C(F)(F)F c1(C(CNC(=O)C(C)(C)CF)NC(C(CCOC)C)=O)ccc(F)cc1F C1(C=O)C2CCCCC12.CC1(C(=O)NCCO)CCC1.CC.C(C)OC C(=O)(C(CO)C(C)(C)C)N(CCCNC(C(C)(CO)OC)=O)C(C)C C1(CNC(C2(CC#C)CCCO2)=O)CN(C(c2ccc(N)cc2C)=O)CCC1C C1(C(N2C(CCNC(=O)C3=CCCCO3)CC(OC)C2)=O)CCOCC12CCC2 C(=O)(C(C)(C)C(=O)N(C(C)C(=O)NCCCc1cn[nH]c1)C1CC1)NC C(C)(C(=O)N=c1cc(Br)[nH][nH]1)c1cc(C)c(Br)cc1C Cc1nc(C(=O)NCC2CCCC(CC(=O)NCC3CCCOCC3)C2)c(C)o1 C1(CC(=O)N(C2CCCN(C(=O)C=Cc3cccnc3)C2)CC)COCCN1C CC1CCCn2c(C(=O)NC34CC(C)(C3)C4)cnc21.c1(C(=O)N)ccncc1F c1(C=O)cc2c(cn1)NC(=O)CO2.C1(C(=O)NCC(O)CC)(CC)CCCO1.N CCC(C)(C)C(C)CC(=O)N(C)CCNC(c1noc(C)c1Br)=O c1(CC(=O)NCC(CNC(CCCOCC)=O)(C)C)ccc(O)cc1 c1(CN(C)C)cc(NC(=O)Cn2ccc(C(F)(F)F)n2)ccc1Cl c1(OCOC)ccc(C(=O)NC(C2CCN(c3nnc(O)s3)CC2)C)cc1 C1(C2CCCCC2)(C(N2CCC(C)C2)=O)CC1.C1(C)(CC)C=C(C(=O)N)C1.C Cc1cn2c(n1)CC(C(N1CCN(C(=O)C=C(C3CC3)C3CC3)C3CC13)=O)C2 N1(CCNC(C(CN(C(C(C=C)C)=O)C)C)=O)CCOCC1=O N1(C(CC(CC#C)NC(=O)C(COC)N(C)C)=O)CCC(C#C)(CC)CC1 C1(CC(=O)NC(c2cnc(C)s2)C)CN(C(c2cc(Cl)n(C)n2)=O)CC1C N1(C(C2CCN(C)C2)=O)CC2CC1CN2C(c1c[nH]c(=N)nc1C(F)(F)F)=O N1(C(C2N(C(C)C)CCCC2)=O)CC2CC(NC(c3ccccc3)=O)C1C2 c1(OCC)cc(Br)ccc1C(c1nnnn1C)Nc1ccc(Cl)c(C)c1 c1(C(=O)NCC(C)NC(=O)C(O)CCc2ccccc2)cnc2c(Cl)cccn12 CC1(C)CCCC(CN2CCCN(C(c3ccccn3)=O)CC2)O1 c1(CC(=O)NC(CN(C(c2c(CCC)occ2)=O)C)C)ccc(O)cc1C c1(OCC(C)(C)C)ccc2c(c1)CCN(C1CCN(CC(F)(F)F)C1=O)C2 N1(c2ccnc(OC)n2)CCSC2CCC12 N1(C(c2cc(OC)cc(Cl)c2)=O)CC2CN(C(c3ccc(Cl)cc3F)=O)CCC12 C1(C(=O)NCC2(CO)CCN(C)C2)CCN(C(C2CCCC2O)=O)C(C)(C)C1 c1(C(=O)NCCN(C(C)C)C(c2cnnn2C)=O)cccc2nc(O)ccc12 N1(C(C=C(C)C(C)C)=O)CC2C3CCC(C2C1)N(C(C1(CC(C)C)COC1)=O)C3 n1(CC)ncc(C(=O)NC2CCOCC2NC(=O)C(N2CCNC2=O)C)c1C C1(CC(=O)NC(C#C)C)CC(C)N(C(c2cc(OC)no2)=O)C1 CC1(C)CC(C(=O)NCCCCCCNC(=O)C=Cc2cccnc2)=NO1 c1(C(N2CCN(C(CC(=C=C)C)=O)CC2CC)=O)csc2c1CCCC2 c1(CC(C)C)nc(-c2cncc(C3CC3)c2)n(C2CCOC2(C)C)n1 Cc1ccc(C=CCC(=O)NC2CCC(NC(=O)CC(C)C)C2)cc1 C1(NC(CN(C(C)=O)C)=O)CC(C)(NC(=O)CC2C=CCC2)C1 Cc1cn(C)nc1C(=O)NCC#CCNC(C1CCOC1C(F)(F)F)=O C(=O)(C(C)(C)n1cc(-c2ccc(CCO)s2)nn1)N(CCOC)C(C)C1CC1 c1(C(=O)NC(CNC(CCCCCC)=O)(C)CO)ccc2c(c1)C(=O)CCN2 CCCCCC(O)CC(=O)N1CCC(CNC(=O)CC(=O)NCC)C1(C)C Cc1cncc(CCC(=O)NCC(C2CCCC2)NC(=O)CCn2cncn2)c1 C=CCC(C)(CC)C(=O)NCC1(F)CCCC1.c1(C(=O)N)c[nH]nc1C(F)F C1(C)(C(=O)NCc2ncn(CC)n2)CCCN(C(C2(C)CCN(C)C2)=O)C1 S(=O)(=O)(c1cc(Cl)ccc1Cl)Nc1cn(C)c(C(=O)NCCc2cccnc2)n1 C1(C(N(C)CC)=O)(NC(C2CC2C(C)(C)C)=O)CCCC1 Cc1ncc(C(N2CC(C)CC2(C)C)=O)c(=N)[nH]1.c1(C=O)coc(C(F)F)c1.N c1(CC(=O)Nc2c(OC)cc(Cl)c(Cl)c2)cccc(C2=CCC(C#N)CC2)c1 Cc1cc(NC(C)CCc2ccc(Br)cc2)ccc1F CC12CCC(C(=O)NC3CN(C(=O)CCCF)CC4(CCC4)C3)(CC1)C(C)(C)O2 c1(CC#N)cc(C(C(=O)NCC2CCCO2)N(C)C2CC2)cc(Br)c1 N1(C(C23N(C(CCC(CC)OC)=O)CC(C)(C2)C3)=O)CCC(O)C(F)(F)C1 N1(CC(=O)NC(CNC(c2c(C)c[nH]n2)=O)CC(C)C)CC(=O)Nc2ccccc21 N1(C(C2(CCOC)CCC2)=O)CC(CCNC(C2CCCC2F)=O)OC(C)C1 N1(C(C(C(C)C)=O)=O)CCC(C2CN(Cc3c(Cl)cccc3Br)C2)CC1 N1(C(C2(C=C)CC2)=O)CC(C)(CN2CCCCC2)C1 CCCCC(CNC(c1cn(C)nn1)=O)NC(C1(CF)CC(F)(F)C1)=O C12(C(N(CCC)C3CC3)=O)CC3CC1C2C3(F)F.O=NN1CCCCC1C=O.N c1(CNC(=O)Nc2sc(C)c(C3CCOC3)n2)cccc2c(Br)cccc12 CC1=NC(C)(CNC(C2(CC)CC2)=O)CS1.C1(CC(=O)N)CC(C)C1 Cc1ccc2sc(NC3(CF)CCN(C(=O)C(C)O)C3)nc2c1 C1(NC(=O)C2=CCOC2)(CO)CCN(C(C2CN(C3CCOCC3)C2)=O)CC1 c1(NC(CCCn2cc(C3N(C)CCC3)nn2)=O)cnn2cc(Br)ccc12 Cc1nc(C)c(C(=O)NC(C2CN(C(c3cccc(Cl)c3)=O)CCO2)C)c(C)n1 c1(N2CCC(CCOC)(NC(=O)CC(C)(C)C(F)F)C2)ncc([N+](=O)[O-])cc1F c1(C(C)NC(N2CC3(C)CC2(C(=O)O)C3)=O)nc2c(s1)CCCC2 N1(C(C(COC)NC(=O)Cc2ncoc2C)=O)CC2CC=CCC2C1 c1(SC)cc(C(C(=O)NCC2CC2)N(C2CCC(C)CC2)C)c(C)o1 N1(C(C(C)n2cncn2)=O)CCCCC1CN(C)C(C1(C(F)F)CCOCC1)=O c1(CC)sccc1C(=O)NCC(C1CC1)N(C(=O)C(C)n1ccnc1)C CC(C)(C(=O)NCC(C)(F)CNC(=O)C=CC1CC1)C1CCCO1 c1(C(C)C(=O)N(CCCCCNC(C2CC2C(F)F)=O)C)ccc2c(c1)OCO2 C(=O)(C(C)S(N)(=O)=O)NC(c1ccccc1)CNC(C=CCCC)=O c1(C(N2CCC(C)(CNC(Cc3cnc(C)s3)=O)C2)=O)coc2c(C)cccc12 C(=O)(CCCCC(F)(F)F)NC1CN(C(C(c2ccc(OC)cc2)=O)=O)C2C1C2 C(=O)(C(C)CC(C)C)NC1C(C(N(CCNC(C(C)C)=O)C)=O)CCOC1 C1(O)(CNC(c2cc(CNC(COCC)=O)sc2)=O)CCCC1(C)C C1(C(=O)NC2CCCN(C(c3nccc(N)c3)=O)C2)CCc2cncn2C1 C1(CNC(c2cn(CCNC(c3cc(C)ns3)=O)nn2)=O)COCCN1C Cc1cccnc1C(=O)N(CCNC(c1scnc1C)=O)CC1CC1 N1(C(C2(CNC(CNC(N)=O)=O)CC=CC2)=O)CCC(O)C(C(=O)O)C1 c1(C(N(C2CC(NC(=O)C=CC(C)(C)C)C2)C)=O)ccc2c(c1)CC2 N1(C(c2cc(OC)ns2)=O)CCOCC(C(N2CC(C(C)(C)C)C2)=O)C1 N1(C(CC(C)C)=O)CCC2(CC1)CC(C)N(C(=O)COCCCF)C2 Cc1cc(OCC(N2CCC(C)(c3ccccc3)C2)=O)ccc1-n1cncn1 CCCC(C(=O)N1CCC(C)C1C(=O)NCC)CC.CC(N)=O.C(N)(=O)N N1(C(c2scc(C)c2)=O)CC=C(C(=O)Nc2cnn(C)c2C(N)=O)C1 C1(O)(C(C)C)CCCN(C(=O)C(=O)N(C)CC2OCCC2(C)C)C1 c1(C(N(CCC)C)=O)c(Cl)ccc(F)c1N.c1(SCC)cncc(C(=O)N)n1 C1(C2CC2)CCN(C(=O)CCc2cscn2)C1.C1(C(=O)N)(CC)CC1(F)F.C CC(C)CC(C(=O)N1CC2(CCCCN2C(=O)CCNC(N)=O)C1)C(N)=O C(=O)(C(CCS(C)(=O)=O)OC)N1CCCC(CNC(C(C=C)(F)F)=O)(CO)C1 CCCCC(CC)C(C(=O)NCCCSCC)N1CCOCC1c1nc[nH]n1 CCCCC(C)C(=O)NCCC1CCCN(C(c2ccc(C(F)(F)F)cc2)=O)C1 NS(=O)(=O)N1CC(C(=O)NC2CC3CC2N(C(=O)Cc2ccc(Cl)cc2)C3)C1 C=C(C)CC(C(=O)N(CCCCCNC(C1CCC(CCO)CC1)=O)C)OC C1C(O)C(=O)N1Cc1ccccc1.C(CC)(CC)NC(COCC=C)=O c1(-c2ccc(CC(C)C)cc2)cc(C(=O)NC2CONC2=O)cc2[nH]ncc12 C1(CC=O)CC2(C1)CN(C(C1CC3(CCC3)C1)=O)C2.c1(CCCC)nn[nH]n1 C1(CC)CCN(C(=O)C(C)(CO)NC(=O)Cc2cncn2C)C1C c1(C2CCCN(C(N(CC)Cc3ccccc3C)=O)C2)ccc([N+](=O)[O-])cc1 C1(CNC(CCC(=C)C)=O)CCCN(C(=O)C(C)CSC(F)(F)F)CC1 C1(NC(=O)Cn2cc(Br)cn2)CCC(C(=O)NCC2CCCOC2)CC1 N1(C(C2(C)CCN(Cc3c(C)nccc3)C2)=O)CCC(C(N)=S)CC1 N1(CCC(=O)N(C2CCN(C(C3CCN(C)C3=O)=O)CC2)CC)CCCCC1=O C1(C(=O)N)CCC(c2ccccc2)CC1.O=C(C(F)C1CC1)NCCOCCC c1(C=O)cn(C)nc1C(C)(F)F.c1ncoc1CC.CC(C)C=CC(=O)N C1(CNC(c2c(C)nsc2)=O)CCC(C(=O)NC(c2ncc[nH]2)CO)CC1 C1(CC)CC(c2nnnn2CC)(NCCCc2nncs2)CCO1 O=C(C1CCCc2c[nH]nc21)NC1CCCN(C(=O)C(F)(F)CC2CC2)C1 CC(C(=O)N(C)CCC1CCN(C(=O)CCc2cn[nH]c2)CC1)C(C)C(C)(C)C c1(C=O)ccc2c(n1)CCC2=O.N1(C(CCNC(=O)NC)=O)CC(C)C(C)C1 c1(C(N(CC(CN(C(=O)CCCF)C)O)C)=O)cn2cccnc2n1 c1(C(=O)NC2CC(C(F)F)(NC(CC3CCC(=O)N3)=O)C2)cc2nccnc2[nH]1 C12(C(=O)NC(CN(C(CCC(=O)OCC)=O)C)(C)C)CCC(O)C1CC2 Cn1cnn(CC(N2CCC(CF)(NC(C3CSCCS3)=O)C2)=O)c1=O N1(C(C2(CCC)CCC2)=O)CCCC(C(=O)NC2CC(O)C2O)C1 CC(C)CCCCC(=O)NC1(CC(=O)NC(CC2CC2)CO)CC1 c1(C2(CN3CC(CCC)C(C=O)C3)CC2)cccc(F)c1C.C1(C)CC1 CC(CC1CCCC1)C(=O)NC1C=CC(CNC(=O)C(C)C2CCCC2)C1 C1(C2CC2)CCN(C(=O)Cc2cc(C)[nH]n2)C1.C1(OCC)CC(CC=O)C1.N Cc1cc(C(N2CCC2(C)C(=O)NCc2ccc(Br)cc2Cl)=O)ccc1[N+](=O)[O-] C(=O)(C(=O)N=S(C)(C)=O)N1CC(C)C(NC(C2CCC(=O)N2)=O)CC1 N1(C(=O)C#CC2CC2)CC2CC1CN2C(=O)CCCC1CCCO1 c1(C(C)=O)cccc(C(=O)N(C)CC2CCCN2C(=O)Cc2c[nH]nc2O)c1 C(=O)(C(C(C)C)NC(C)=O)NC(CN(C(C(CSC)O)=O)C)C C(=O)(C#CC1(C)CC1)N1CC(C)C(CCNC(=O)C(C)(C)c2ccccc2)C1 c1(C(=O)NCC2C(NC(=O)Cc3ccc(O)nc3)CC2)cc(F)cc(Cl)c1 c1(C(=O)NCCCCn2cc(C3COCC3O)nn2)c[nH]c2nc(Cl)ccc12 c1(C(N2CC(CCC)N(C(=O)C(F)CC)CC2)=O)ccc2oc(C)nc2c1 c1(OC)cc(C(=O)N(C2CN(C(=O)C(c3cccnc3)C)CC2O)C)n(C)n1 c1(OCC)cccc(C(=O)NC2CC2)c1N.C1(CC=O)SC(=N)NC1=O.C c1(-c2cc(C(=O)NCCNC(c3cc(CCC)[nH]n3)=O)on2)cccc(O)c1 C1(C(=O)NCCN(C(C2CCCN2C=O)=O)CC)CN(C)C(=O)N1 N1(C(c2cc(C)nc(C)c2)=O)CCC2CCCN(C(=O)C(=O)NCC3CC3)C2C1 N#Cc1cc(C(=O)NC2CCC2CNC(C2(F)CC=CC2)=O)cc(O)c1 C1(C(N2C(C(C)C)CN(C(c3ccc[nH]3)=O)CCC2)=O)CC2(CCCCC2)CO1 C(=O)(C1=NOC2COCC12)N1CC(C(=O)NC(COC)C)C2(C1)CCC2 c1(OCCC(=O)N(C2CN(C(CN(C(C)=O)C)=O)CC2O)C)cc(F)ccc1F N1(CC(=O)NCCC2CCN(C(C3CC(C)(O)C3)=O)CC2)CCCCC(O)C1=O c1(C(=O)NC2CC(NC(C(C)(C)C3CCCOC3)=O)C2)cc2nc(F)ccc2o1 C=C(C)CCC(=O)NCC1CC(NC(c2ccoc2C)=O)C1 N#CC1CN(Cc2cc([N+](=O)[O-])cs2)CCN1C(c1cc(Cl)c(O)c(Cl)c1)=O C(=O)(C(CC)C(C)O)NC12CC(CNC(c3cc(CCC)n[nH]3)=O)(C1)C2 N1(C(C(C)(CO)NC(=O)CCc2ccco2)=O)CC2C(C1)C2(F)F C1(NC(c2cc(C)c(C)o2)=O)CC=C(C(=O)NCC2CCCC(C)(C)O2)C1 C1(C(=O)NCCNC(c2c(C(F)(F)F)nc(C)s2)=O)CCc2ccnn2C1 N1(C(C2CCC(=C)CC2)=O)CCCC12CCCN(C(=O)CN(S(=O)(=O)CC)C)C2 c1(C(=O)NC23CCCC2CN(C(=O)CCC2CC2)C3)cc(O)ccc1[N+](=O)[O-] c1(C=O)ccc(C(=O)N(C(C)CC)C)cc1.C1(CC(=O)N)(OCC)CCC1 N1(C(Cc2cc(CC)no2)=O)CC=CCC1C(N1CCC(SC)C1)=O C=CC(C)(CCOC)C(=O)N1CCCC(CN(C)C(c2ccc(C)cn2)=O)C1 C(=O)(CCCCC(C)(C)C)N1CCOCC(CNC(C2(C#C)CCCC2)=O)C1 C1(C(=O)NCC2C(NC(c3ccc(C#N)cn3)=O)C2)COc2ccccc2O1 c1(C(=O)NC2CCN(C(C3C(C)CN(C)C3)=O)CC2)coc2c(Cl)cccc12 c1(CC)cnn(CC(=O)NCc2nc(C=O)co2)c1.c1(CC)ccc(C)s1.N C1(C2CCCOC2)(NC(CC2(C)N(C(C3N(CC)CCCC3)=O)CC2)=O)CC1 c1(C(=O)NC2C(CNC(=O)CCCC(F)F)C2)cc2cccnc2cc1F N1(Cc2cccc(OC)n2)CC2(C(N3CCC(C(C)(C)C)CC3)=O)CC2(CO)C1 c1(C(N2C(CNC(Cc3c(Cl)cn(C)n3)=O)CC2)=O)ccnc2ccc(Cl)cc12 C1(C(C)C)CN(C(C2(NC(=O)C(O)CCN(C)C)CCCC2C)=O)CCO1 c1(CC(=O)NC(CCCNC(C(C)(C)SC)=O)C)c[nH]c2ccc(Cl)cc12 N1(C(C(C)=C2CCC2)=O)CC2C3CCC(C2C1)N(C(=O)C(O)C(C)C)C3 C12CC1CN(C(=O)CC1CCC(C)(C)C1)C2.C(C(=O)N)NC(=O)NC.C N1(C(C2CNC(=O)N2)=O)CC2CCCC(C1)N2C(c1cc2ccc(Cl)cc2o1)=O N1(CCC(=O)NCCC(C)NC(=O)C(c2ncccc2F)(F)F)CCNC(=O)C1 c1(CC(=O)NC(C)CCNC(C23CCC(CO2)C3)=O)ccc2c[nH]nc2c1 c1(C(=O)NC(CN(C(c2n(OC)cnc2C)=O)C)C)ccc(N)c(C)c1C CC1=C(C=O)S(=O)(=O)CCO1.C12CCN(C(c3ccc(C(C)C)o3)=O)CC1C2.N C1(NC(c2ncn(CC)n2)=O)CN(C(=O)COc2ccc(O)cc2)CC12CC2 c1(OC)ccnc(CN(C2CCSC(C)C2)C=O)n1 CCC(CC(=O)N1CC(NC(c2c(OC)nsc2OC)=O)C(O)C1)C(C)(C)C c1(C(N(C)CC2(NC(C(C=C)O)=O)CC2)=O)cc(C2CC2)nn1CC c1(CNC(C2(F)CN(C(C(c3ccccc3)C)=O)C2)=O)ccc(F)nc1 C=CCN=C(NCCC(C)(C)OC)NCC1CCOC(C)C1 CCCC(C(=O)N1CC(CNC(C2CC2COC)=O)CC1C)OC C=CCC(CC)C(=O)N1CC(OC)C(CNC(C2(n3ccnn3)CC2)=O)C1 N1(C(c2cnc(C)nc2)=O)CC2CN(C(c3cccnc3C)=O)C2C1 S(=O)(=O)(c1cccc(=NCCC(=O)N2CCCC2)[nH]1)NC1CC(C)CC(C)C1 C1(OCC)CC2(C1)CC2.c1(C=O)cnc(C)cn1.C1(CC(=O)N)CCCC1 N1(C(C)=O)CC(CNC(=O)C(c2ccc(F)c(F)c2)(C)C)C(F)(F)C1 C1(NC(=O)CCCn2cccn2)(CNC(=O)C2=CCOC2)CCC(F)(F)CC1 n1(CC)ccnc1C(=O)NC1CC(CNC(=O)C(O)CSC)C1 C1(C(=O)NC(Cn2ncc(C)c2)C)CC(NC(c2ccon2)=O)C12CCC2 N1(C(CCCCCC)=O)CCC2CN(C(=O)C(=Cc3cn(C)nn3)F)CCC12 C1(NC(c2c(C)nn(C3CC3)c2)=O)CN(C(C2CC2C#N)=O)CC1C1CC1 N1(C(c2cc(CC)oc2C)=O)CCC(CC)(NC(=O)C(CC(C)C)OC)CC1 C(=O)(C1=CC(C)CC1)NCC(CCOC)NC(c1cc(OC)nn1C)=O c1(C(=O)NCC(C)(C)NC(C2CC(=C(F)F)C2)=O)cc(F)ccc1F c1(NCc2c(C)con2)ncc(C)cc1O C(=O)(C1CCc2nnc(C)n21)N(CC(C)O)CCNC(C1C(CCC)C1)=O CC1CCC(CC(=O)NCCCCCNC(=O)C(C)(C)c2cc[nH]n2)C1 c1(C(=O)NCCC(=C)CNC(=O)COCCF)cnc2sc(C)c(C)n12 N1(C(CSC)=O)CCCC(N(C(c2ncsc2C)=O)Cc2ccccn2)CC1 Cc1c(-c2ccc3n[nH]cc3c2)cccc1N=c1[nH]ccn1C C1(C(NC)=O)C2CS(=O)(=O)CC12.Cc1cnn(C)c1C(N1CC(O)C1)=O.C N1(C(C(CCCC)C)=O)CCC2(C)CN(C(=O)CC(=O)N(C)C)CC12 C(=O)(C1CC(=O)Nc2ncn(C)c21)N.C(C(=O)NC(C)C1CC1)NC(C)=O C(=O)CCC1=CCCCC1.c1(C(N2CC(COC(C)=O)C2)=O)cnc(C)nc1.N C1(NC(CN(C2CCC2)C(c2c(C(C)C)nco2)=O)=O)CCCCC1(C)C N1(C(C(C)O)=O)CCC2(CCCN(C(c3cnc(Cl)cc3N)=O)C2)C1 C(=O)(C(CCOC)NC(=O)CC1CC(C)(C)CO1)NC(C=C)C c1(OCCC)ccccc1C(C)NC(=O)C(n1cc(C)nn1)C.CC(N)=O.O c1(C(N2CCC(C(F)F)(CNC(C(CC)O)=O)C2)=O)cc2c(C)c(F)ccc2[nH]1 CC1OCCCC1C(N1CCC(NC(=O)CC2(c3ccccc3)CCC2)CC1)=O CC1CC(c2nnnn2Cc2cccs2)(NCc2nccn2C)CC(C)S1 c1(NC(C#CCNC(C(C2CCC(=O)N2)C)=O)=O)ccc(CO)c(F)c1 c1(C(=O)NC2(CNC(C3CC3(F)F)=O)CC(CO)C2)cccn2nnnc12 C(=O)(C(F)(F)C(C)(C)O)N1CCN(C)C(CNC(=O)C(c2cnn(C)c2)O)C1 C(=O)(CS(=O)(=O)C(C)(C)C)OCc1cnc2ccc(-c3c(OC)ccs3)cn21 C1(c2cn(CCC(=O)NCCc3nnc(O)o3)nn2)CCC(F)(F)CC1 C1(NC(c2c(C)cns2)=O)CN(C(c2ccc(C(N)=O)[nH]2)=O)CCC1(C)C N1(C(C(C)OC2CCCCC2)=O)CC2(C1)CN(C(C1CCNC(=O)C1)=O)CCO2 CCCCC(C)CCC(=O)N(C)CCNC(=O)C(C)Cc1ccc(Cl)cc1 C(C(C(=O)N(C(C)CC(C)C)C)N(C)C)NC(C(C)NC(=O)OC)=O c1(C(=O)N)c[nH]c(=NCC)s1.C1(COC)(C)CCCN1C(=O)C.C1CCC1 c1(C=O)c(N)cc(C)cc1F.C(=O)(C(F)C(=O)N1CCCC1)OCC.C(C)O C=CC1(C(N2CCN(C3(C)CC3)CC2)=O)CCN(C(=O)C(C)CC(C)(C)C)CC1 c1(CN2CCC(F)(C(=O)Nc3ccc(F)cc3Br)C2)cccc2cc[nH]c12 N1(C(c2c(CNC(C3CCC=CCC3)=O)cco2)=O)CC2CCCCCC2C1 N1(C(C2CCCO2)=O)CC2C3CCC(C2C1)N(C(C1CCCOCC1)=O)C3 c1(N2CCN(C(CN(C)C)=O)CC2)nc(C(F)(F)F)cc(-c2ccccc2)n1 C1(N(CC(=O)NCC2=CCSC2)CC)CCS(=O)(=O)C1 C1(C(N(CC(C)NC(c2ccnc(N(C)C)c2)=O)C)=O)COC2(CCC2)C1 N1(C(C(CC#C)C)=O)CC2(CCC2NC(c2cc[nH]n2)=O)C1 C1(C2CN(C(=O)C(c3cccc(C=O)c3)C3CCCC3)C2)(C(=O)NC)CC1.O C(=O)(CC(F)(F)C(F)F)N.c1(SC)cccc(C(=O)NCC2(C)CC2)c1 C1(NC(c2c(CSC)cccn2)=O)CCCN(C(C2CCCC(C)CC2)=O)C1C c1(C(N2CCC(C)(NC(=O)CC3CC=CCC3)C2)=O)ccc2c(n1)NC(=O)CO2 c1(CC(=O)NCC(CC=C)NC(C)=O)cccc2c1NC(=O)CC2 C(=O)(N1CC2COCC2O1)C1CCCN(C(CCS(=O)(=O)N(C)C)=O)C1 C(c1ccc(F)cc1F)=CC(N1CC(C)CC1)=O.C(C)(C(=O)N)N(C(C)=O)C CC1CCC(O)CN1C(c1ccnc(CNC(=O)CCc2cccs2)c1)=O C(=O)(C(CNC(=O)COCC(C)C)C(C)C)NC(C(=O)NC)CC c1c(C)nn(C(F)F)c1C.Cc1ccc(NC(=O)C(N2CCC(CN)C2)=O)cc1 S(=O)(=O)(c1ccc(NC)c(Cl)c1)N1CCC(N(CC)CC)C1.C1CN(C)C1 C1(C)(NC(c2c(OC)nccc2)=O)CCN(C2CCNC2=O)CC1 C(=O)(C(CC(C)CC)NC(c1cnnn1CC)=O)N1CC2(CC(=C)C2)C1 c1(C(C(=O)O)NC(N2CCN(CC)CC2)=O)cc(Cl)ccc1Cl C1(C(=O)NC(C(CO)NC(c2ncn(C(C)C)n2)=O)C)CC(C)(C)CO1 CON1CC(C(N2CCN(C)C(CNC(=O)C(C)(F)F)C2)=O)CC1=O N1(C(C2(Oc3ccccc3)CCCNC2)=O)CCCc2n[nH]cc21 c1(OC)ccc2oc(C(=O)NCC(C)CC3CCCO3)cc2c1 c1(C(=O)NC)ccc(C(=O)NC(C)C(C)NC(c2cncs2)=O)cc1F.C C(=O)(C(CCc1ccco1)N1CC(F)(F)C1C1CC1)NCCC#N O(NC(=O)C(CC(F)F)N(C)C(c1ncccc1N)=O)CC(=O)OCC C1(C(C)CO)CCN(C(=O)CN(C(=O)CN(C2CCC2)C)CC2CC2)CC1 c1(NC(C2CC(NCc3c(C)c(Cl)ncc3)C2)=O)nc(Cl)cc(Cl)c1[N+](=O)[O-] C1(NC(C(COC)C)=O)CN(C(c2cc(-n3nnnc3C)cc(F)c2)=O)CC12CC2 Cc1cocc1C(=O)NC(Cc1ccco1)C(=O)NCCC12CCCC1C2 c1(CN(C(C2(F)CC(NC(=O)C(Cl)Cl)C2)C2C(C)C2)CC)ccccc1 N1(C(C=CC(C)(C)SC)=O)CCC(C)(CNC(c2nn(C)cc2N)=O)C1 CCC(CC(=O)NCC(=O)OC(C)(C)C=CC(N1CC=CC1)=O)C(C)(C)C c1(C(N(C(CCNC(Cc2c(C#C)cccc2)=O)C)C)=O)cc(Cl)cc(C)c1O CCC(CC(=O)N1CCN(C2CCN(C(c3ccc(C)[nH]3)=O)C2)CC1)C1CCC1 C=CCCCCCCC(=O)NC(CC(C)CC)C(=O)NCC(=O)NC1CCCC1 CC1c2cc(Br)ccc2OC1C(=O)NCCC(C)NC(c1cccnc1)=O CN1N=C(C(=O)NC(C(=O)NCCc2cnco2)C2CCOC2)CCC1=O Cc1coc(C)c1C(=O)NC1CCCN(C(c2cccnc2C(F)F)=O)C1 N1(C(C2C(NC(C(C)CN(C)C)=O)CC2)=O)C(C)CC1(C)C N1(C(C2N(C(C3OCCC(C)C3)=O)CCN(C)C2)=O)CC2NC(=O)OC2C1 C1(NC(CC(COC)(C)O)=O)CCCCC12CCN(C(=O)CC(C)C)CC2 C(=O)C1=NN(C)C(=O)CC1.CC1CCCCC1(C)C(=O)NCCC1(C)CC1.N CC1CCN(C(c2ccc([N+](=O)[O-])[nH]2)=O)CC1NC(=O)COc1ccccc1F c1(C(C)C)nc(NCC2CC23CC3)cc(=NC(CS(C)(=O)=O)CS(C)(=O)=O)[nH]1 C(=O)(C(C)C(F)(F)F)NC(C(=O)NCC(CC)(CC)OC)CC1CC1 C(=O)(C#CC1CCCOC1)N1CC(CCC)N(C(=O)CP(C)(C)=O)CC1 CCC(CC)CC(F)C(=O)NC1CCCC1CNC(=O)C(F)(F)C(F)(F)F CC(C)(O)C(F)C(=O)NC1(CC(N2CC3(CC(O)C3)C2)=O)CCC1 N1(C(c2cnc(C(C)C)o2)=O)CC2C(NC(c3ccccc3O)=O)C2C1 C1(CNC(CC(C)c2ccco2)=O)CC2(CCC2)CN1C(=O)C=C(Cl)Cl c1(OC)ccnc(COCC(=O)NCCC2(C(=O)O)CCNC2=O)c1 c1(C(=O)NCC2CCCN(C(C3(OC)CCCOC3)=O)C2)nc2ccccc2s1 N1(C(c2cn(CC=C)nn2)=O)CC2CCC1C1CN(C(=O)C(C)CCC)CC21 Cc1cc(C)c(C(N2CCC(NCCO)C2)=O)c(C)c1.C(C(C)(C)C)C1CC1.C C1(CC(N2CCC(NC(CCS(C)=O)=O)C2)=O)CN2CCC1CC2 N1(C(CCC(=C)Cl)=O)CCOCC(NC(C23CC(CO2)C3)=O)C1 c1(C(N2CCC(CC=C)(NC(c3cnoc3C)=O)C2)=O)ccnc(OCC)c1F CCC(C)C(O)C(=O)NCC(C)CNC(=O)CSc1nncn1C(C)C c1(C(=O)NCCN(C(C2C(C)C2C)=O)C)cc(C(F)(F)F)cc(N)c1 c1(C(N(C2CCN(C(c3cnc(CCC)s3)=O)C2)C)=O)ccc(F)cc1 C(=O)(CCCC(=O)N1CCOCC1)N1CC(NC(CCC(C)N(C)C)=O)C(C)C1 c1ccc(F)cc1F.C=CCC(CNC(C1(C(=O)NC)CC1)=O)NC(=O)C c1(C(=O)NCC(CO)NC(C2(C)C(C)C2)=O)onc2ccccc12 CC(C)CC(CC(=O)N1CCCSCC1C)NC(=O)C(CO)C(F)(F)F CC1CCC(NC(c2cnc(-n3cccn3)cn2)=O)CN1C(=O)Cc1ccon1 c1(OC)cc(OC)c2[nH]c(C(N3CC4CC3C4C)=O)cc2c1.C(=O)(CC(C)C)N c1(C(=O)NCC(C2CC2)NC(c2sccc2Br)=O)cncnc1C1CC1 C1(C)(CCNC(C(C(=O)OC)OC)=O)CCN(C(=O)CCC2CCCC2)CC1 c1(C(N2CC(CC(C)NC(C3CCC(C)C3)=O)C2)=O)nc2ccccn2c1F CN1CC(O)CC1C(=O)NCCC(C)(C)NC(c1ccc(N(C)C)nc1)=O N1(C(C=CC(C)(C)NC(c2c(C)[nH]cc2)=O)=O)CCOCC1CO N1(C(c2nc(C)nc(O)c2)=O)C(C(=O)NCCOC(=N)O)C2CC(O)C1C2 CCCC(C)C(=O)N1CCOCC1CC(=O)NC1CC1C1CC1C CCCCCC(CC)C(=O)NCCCCCNC(c1ccn(C)c1CC)=O c1(CNCC(CSC)O)ccc2c(c1)C(=O)NC2 C1(C(N2CC(NC(CSCCCC)=O)C2)=O)CC(=O)N(CCOC)C1 c1(C(=O)NCC(CC(C)C)NC(c2ccon2)=O)cncc(F)c1Cl.N(C)C.C CCC(c1ccccc1)=CC(=O)NC(C)CCNC(c1cnc(=N)[nH]c1)=O c1(CC)cc(C(N2CCC(CNC(=O)C(C3CC3)N(C)C)C2)=O)ccc1Cl N1(C(c2c(C)ccn2C)=O)CC23CCCCC2(C1)CN(C(C1CCC(C)O1)=O)C3 CN1CCC(CCNC(=O)CCOCC)C1=O.c1(CC=O)ccc(O)nc1.N C=CCC(C(=O)Nc1n[nH]c2c1CN(C(=O)C(CC)N(CC)CC)C2)C(C)C c1(CN2CCC3(C(C(=O)NCCC4CCCC4)C3)C2)c(Cl)cc(Cl)cc1Cl C(C(F)(F)C(F)(F)F)NC.N1(c2[nH]c(C3CCCCC3)nn2)CCC2OCC2C1 C1(F)(CNS(=O)(=O)Cc2c(Oc3ccccc3)cccc2F)COCCOC1 C1(C(=O)NC2C(C)CC=CC2)CCC2(CC2)N1C(=O)C(O)c1ccsc1 C1(COC(Cc2c(Br)cn(CC)n2)=O)CC(S(C)(=O)=O)C1 C(=O)(C(CC)(CC)c1ccc(Cl)cc1)NC1CCCC(SCC(=O)OC)C1 CCCC(CC)CC(=O)NC12CCC1CN(C(=O)CCC(N)=O)C2 c1(CC(N2CC(O)CC(NC(=O)CSCC(F)F)C2)=O)cc2ccccc2o1 C12(C(=O)Nc3ccc(-n4cc(CCN(C)CC)nn4)cc3)CCC(CC1)C(C)O2 N1(C(C=C(CC)CC)=O)CCN(C2CCC(NC(C3C=CC=CC=C3)=O)C2)CC1 N1(C(C2(C(=O)OC)CC2)=O)Cc2ccnn2CCC1.C(=O)CCC1CC1(Cl)Cl.N C=CC1(C2(C(=O)NC(C)C(C)NC(=O)C3=C(C)OCCS3)CCC2)CCC1 C(C(C(C)C(C)C)NC(c1ccnc(O)c1)=O)NC(CCc1ccc(C)cc1)=O N1(CCNC(C(c2cnn(C)c2)C)=O)CCN(C(=O)CC2CC3CC3C2)CC1 CC1(C)CCCC(C(=O)NC(C)(C)CC(=O)NCCCCC2CCCC2)C1 C1(C)(C=O)COCCO1.n1(CC(=O)N(C)CCO)ccnc1C(C)C.CCC CC(C)CCC(C)NC(=NCC1CCCN1Cc1nccnc1C)NCC1CC1 c1(C(=O)OCC)cc(Cl)n[nH]c1=NC1CN(c2nnc(C(N)=O)s2)CC(C)(C)C1 N1(C(C2CC(CCC)OCC2)=O)CCC(CNC(C2(CS)CCC2)=O)CC1C C1(NC(=O)C=CC2CCCO2)CN(C(=O)CCN2CCC2)CC12CC2 N1(C(=O)C=CC2CCCC2)CCN(C(C2CC=CC2)=O)C2CCCCC2C1 c1(C(=O)NCC(C)(O)CNC(c2cccn2C2CC2)=O)cnn2ccncc12 C(=O)(CCC(=O)CC)N(C(CC)CC(=O)N1CCCC1COC1CC1)C C=C(F)C1(CC(=O)NCc2ocnc2-c2cn(CCN(C)C)nn2)CCC1 C1(C)CCN(C(C2([SH](=O)=O)CCC2)=O)CC1.C(C)C=O.C(C)(C)C.CC.O c1(CCC(N2CCCC2)=O)cccc(N2CCOCC2)c1.O=C1C(=O)N2CC(C2)O1 N1(C(CCOCCOCC)=O)CCC(NC(c2[nH]cnc2C)=O)C12CCC2 C12(CNC(C3CCN(C(CC(C)n4cccc4)=O)C3)=O)CCCC(CO1)C2 c1(N2CCCC(CC)(CC)CC2)[nH]c(=NC2CCCC2CF)nc2scnc12 C1(C(N(CCN(C)C)C)=O)CC(F)(F)C1(C)C.c1c[nH]nn1.C1CC2CC2C1 C1(C)(CNC(C(C)(C2CCC2)NC(c2c(C)non2)=O)=O)CCC(=O)N1C CCC(CC(=O)NCC(CNC(c1cn(C(C)C)nc1Br)=O)OC)SC CC1CN(C(c2csnc2Cl)=O)CC1CNC(=O)CSCc1ccccc1 CN1CC2(C1)CN(C(=O)C=CC(F)(F)F)c1ccccc12 N1(C(CN(CCC)C(c2ccc(C(C)=O)o2)=O)=O)CCCC(C(C)(C)O)C1 N1(CCN(C(=O)C(F)F)C)CCN(C(=O)CN(S(C)(=O)=O)C)CC1.C CCCC(C(=O)NC)NC(=O)C(C)NC(=O)CC(C)COC C1(C(=O)NC(CCO)C2CC2)CCC(O)CN1C(=O)C(O)Cn1cncn1 C(=O)(C1=COCCO1)N1CCC(NC(CCCn2cnc(C#N)n2)=O)C1 N1(C(CN(C)CC)=O)CC2(C1)C(NC(=O)C1=C(C)CCC1)CCS2(=O)=O CC1CCNC(=O)C1CNC(=O)CCN(C(=O)CCc1cccnc1)CCCO c1(NC(=O)NC2CC(N3CCOCC3)C2)cnn(C2CC2(F)F)c1 C12(C(N3CCCCC3)=O)CCC(n3ccnc3)(CC1)CC2.CN(C(C1CC1)=O)C N1(C(C(C)CO)=O)CC2(CO)CC1(C(=O)NC(c1ccn(C)n1)C)C2 c1(C(N2CC(CNC(c3ccc(O)cc3)=O)C2)=O)cc(Cl)ccc1Br C(=O)(C(CC(F)F)NC(C1CC12CCCCC2)=O)NCCSC C1(NC(C2(C)N(C)CCC2)=O)CC2CCC1CN(C(c1ccncc1)=O)C2 CC1(C)CCCC1NC(C1(F)CN(C(C2CC2(F)F)=O)C1)=O Cc1cc(Cl)ccc1Nc1nccn1-c1ccccn1 c1(C(=O)N(Cc2ccccc2)CC2CCCO2)c(F)ccc(Cl)c1F c1(C(N2CCC(NC(CC(COC)(C)C)=O)C2C)=O)ccc(S(N)(=O)=O)s1.O c1(C=O)cnc2c(c1)CCOC2.CC1CCCCC1CNC(=O)C=CC(N)=O C(=O)(CCc1ccoc1)NCC1(OC(C)C)CCC1.c1(CC=O)ccon1 CCCCCCN(CCNC(=O)CSC1CCCCO1)C(C1(CC)CC1)=O C1CCC(C)N(C(c2cn(C3CCC3)nn2)=O)C1.Cc1csc(Cl)c1C(=O)NC C12CCC1CCN2C(=O)Cn1c(C)csc1=O.c1(CC)oncc1C(=O)NC C(c1cccn1C)=CC(=O)NCCCN(C(=O)CCCc1ccccn1)C C1(NC(CC(CN(C)C)O)=O)CCCCN(C(c2cnn(CC(F)(F)F)n2)=O)C1 N1(C(CCOCCNC(C(CC(CC)C)C)=O)=O)CCc2ccc(C#N)cc21 N1(Cc2c(OC)cccn2)CC(NC(c2csc(C)c2C2CC2)=O)CCC1C c1(OC)cc(C)cc(C=O)c1C.C1(CC=O)CCC(C)O1.C(C)(C)C1CC1.N N1(C(C(COC)OC)=O)CC(NC(C2Cc3ccccc3N2)=O)CC2(CC2)C1 C1(C(=O)NCc2cc(C)sc2C)CC2CC(=O)C1C2.C1(C=O)(C)CC1.N C(=O)(C1=CCCCC1)N(C1CC(NC(c2csc(C(F)F)n2)=O)C1)C N1(C(C(CC=CCC)C)=O)CC2CCC2(CNC(c2occ3c2CCC3)=O)C1 C(=O)(C#CC1CCOCC1)NC1COCCN(C(c2cnc(C)[nH]c2=N)=O)C1 c1(C(N2CCC(C(=O)OC)CC2)C(=O)NC2CCOC2)nc(OC)ccc1F c1ccc(C(=O)N(C2(C(=O)NCC3(CSCC)CC3)CC2)C)nc1 C1(C(=O)NC2CC(NC(C(c3cccc(Cl)c3)C)=O)C2)CCCC2(CC2)C1 c1(OC)ccc(NC(c2[nH]ccc2C)=O)c(C)n1.c1(CC=O)cncnc1O.N C(=O)(CCCCCF)NCC(C(N1CCOC(CC(C)C)C1)=O)OC c1cn2ccccc2n1.C(CCO)NC(C1(NC(=O)OC(C)(C)C)CC1)=O.N CC1CCC(C(N2CC(O)C2)=O)N1C(c1ccncc1O)=O C#Cc1cccc(C(N2CC(O)(C(F)C(=O)N(C3CC(=C)C3)C)C2)=O)c1C c1(C(=O)NC2(CNC(C(C)SC)=O)CCCC2)nc2ncc(Br)cc2[nH]1 Cc1cc(C(=O)NCC2(CNC(C3(F)CCOC3C)=O)CCCC2)ccc1Cl C(=O)(C1COc2ccccc21)NCC(c1cccc(Cl)c1)NC(C(C)(C)CF)=O CC1(O)CC2(CN(C(C3C4CCN(C(C5CNC(=O)O5)=O)CC34)=O)C2)C1 c1(CNC(C(C)CS(C)=O)=O)nnc2n1CCN(C(=O)Cn1ncccc1=O)C2 c1(-c2nc(CC(C)OC)nn2C(C)C(C)(C)C)c(Cl)sc2nnsc12 CCCC(CN1CCN(C(=O)Nc2cc(Br)ncc2F)CC1)C(=O)OC C1(CCNC(c2ncc(C)nc2)=O)CN(C(=O)CCc2cn(C)nn2)CC(C)O1 C(=O)(C(C(C)(C)C)NCc1cn(-c2cccc(C#N)c2)nn1)OC c1(C(=O)N)ccc2ccncc2n1.C1(OCC(=O)NC(C)C2CCC2)CC=CC1 Cc1nn(CCO)cc1C(=O)NC(C)C(C)NC(=O)CCc1cccn1C N1(C(CC(=O)NCC)=O)CC2CCCC(NC(=O)C(C)(C)CC(=O)OC)C2C1 C1(C)(CCCC(=O)NCCCCNC(C2C3CN(C)CC32)=O)NC(=O)NC1=O N1(C(C(C(C)C)C#N)=O)CCCC12CCN(C(c1ccc(C(N)=O)c(Cl)c1)=O)C2 C(=O)(C(F)(F)C(C)(C)O)N1CC(C)N(C(=O)C=C(Cl)Cl)CC1 C1(C)(CC(=O)NC(C2(C(=O)N(C)CCC3CC3)CC2)C)OCCO1 C=CCCC(C(=O)N1CCC(C)(C)C1)c1ccccc1.C1(=O)COCCCN1C C1(NC(C2=C(C)CCC2)=O)CC12CCN(C(=O)Cc1ccn(C(F)F)n1)CC2 c1(C(C)C)cccc(C(=O)NCC2(C)CCCN2C(=O)CCC2CCOC2)c1 C1(CC(N2CC(CCNC(c3cncc(C)n3)=O)C(C)C2)=O)CCCC(F)(F)C1 Cc1nccc(C(=O)NC2(C)CCN(C(=O)C(C)(C)C3CCC3)C2)n1 CC1(C)CCC(O)(CNCc2cc(Cl)ccc2Br)C1 c1(C(=O)OC)ccc2[nH]c(=NC(C)CC(C)NC(=O)C(C)CO)oc2c1 C1(N(C(C(CC)OCC)=O)C)CN(C(c2cc(C)cc(Br)c2)=O)CC1(C)C N1(C(C)=O)CCCc2ccc(S(=O)(=O)NC3CCCNCC3)cc21.C(C)(C)C C12(CCNC(c3c(CC)nc[nH]3)=O)CCC1CN(C(c1ccc(OC)nc1)=O)C2 N1(C(c2ccc(C(N)=O)cc2)=O)CC2CCC1C2NC(c1cc(Cl)ncc1O)=O Cc1cc(Cl)cc(C)c1C(=O)NC1CC1.c1(C=O)cn(C)nc1C1CCC1.N CC1CCN(C(C2CCCSS2)=O)CC1NC(c1cccc(CCN(C)C)c1)=O C1(CC)CCCCC1C(F)(F)F.C(CC=O)NC.C(C)(C)C.C=O.C(C)C.C c1(C=O)cnc(O)c([N+](=O)[O-])c1.C(C)(CC(=O)NC(C1CCCCC1)C)OC.N C1(C(=O)NCC2CCC(F)C2)CCN(C(c2cccc(Cl)c2)=O)CC1 C1(C(N2CCC(O)(CN(C(CSCCOC)=O)C)C2)=O)CC2(C)CC1CO2 c1(NCC2C(NC(C=NOC)=O)CCC2)ncnc(O)c1Br c1(OC)ccc(-c2nc(C(O)CC(C)(C)C)n(CCS(N)(=O)=O)n2)cc1 c1(C=O)coc2c1CS(=O)(=O)C2.Cc1nsc(N)c1C(=O)NC1CCCC1.C C(c1ccccc1)=CC(N1CC(N(C(=O)Cc2cscc2Br)C)C1)=O CC1CC(NC(=O)C=Cc2ncc[nH]2)CCN1C(c1ccc(Cl)s1)=O CC1OC(C)C(C(N2CCCC(CSc3ccc(F)cc3)C2)=O)C1C N1(C(=O)CSC2CCCCO2)CC2CCC1C(CNC(=O)C(F)(F)C1CC1)C2 c1(CC)cc(NC(c2cccc(Br)c2O)=O)cc(N)c1 c1(C(=O)NC(CN(C(c2ccn(CCCC)n2)=O)C)C)ccc(SC)cc1Cl C1(C(=O)N)OCCN(C)C1=O.c1(OC)c(C(=O)NC2CCC(C)CC2)csc1C C1(CC(=O)N(c2cccc(C)c2)CCO)CN(C(c2cc(Cl)n[nH]2)=O)CC12CC2 c1(C(=O)NC2C(C)CCN(C(CSC(C)C)=O)C2)cc2cc(F)ccc2cn1 N1(C(c2cc(NC)nc(Cl)c2)=O)CC2CC1CCC2NC(C1OCCC1C)=O C1(COC)(COC2CCCNC2)CCCN(CC(=O)Nc2ccccc2Cl)C1 N1(C(CC(C)OC)=O)CC=C(CCNC(C2(P(C)(C)=O)CC2)=O)CC1 Cc1sc(C(=O)NC2CC2CNC(=O)CC2CCN(C)C2=O)c(C)c1Br CCCCCCCCn1ccc(=NC(C)(CCNC(N)=O)n2ccnn2)[nH]1 CC1(F)CN(C(C2(CO)CC2)=O)CCN(C(=O)CCc2ccc(CO)cc2)C1 CC#CCCC(=O)N1CC(O)(CCNC(C2(C(F)F)CC2(F)F)=O)C1 c1(C(C(=O)NCCCC2(NC(CCC(=C)Cl)=O)CC2)C)cccc2ccccc12 C1(C(N(C(CC)C)CC)=O)CCCN(C(C2CN3CCC2C3)=O)C1C c1(C(=O)N)cnc(O)c([N+](=O)[O-])c1.N1(C(c2cnc(C)[nH]2)=O)CCCC2(C)CC12 Cc1nc(C(=O)NC2CCC(C)C2)cc(O)n1.C1(C=O)CC2(C1)CC2(F)F.C N1(C(c2c(OC)cc(Cl)c(Cl)c2)=O)CCC2(CC1)CN(C(=O)C(C)(CO)OC)C2 N1(C(c2c(C)c[nH]c2)=O)CCN(C(=O)C(C)Nc2ccccc2)CC1 c1(C(N2CC3N(C(C4(C#N)CC4)=O)C3C2)=O)cc(Br)cnc1Cl c1(C(=O)NC2CC(CCOCC)C2)cc(OC)c(C)c([N+](=O)[O-])c1 C(=O)(CC(C)C(C)(C)C)N1CCC(NC(C(=Cc2ccco2)C)=O)(CF)C1 N1(C(C2N(C)C(=O)CC2)=O)CCC(C2CC2)(NC(=O)Cc2csc(S)n2)C1 C(CC)(C(=O)NC(CCCNC(=O)C(C)c1ccco1)c1ccccc1)=CC C1(C)(C(=O)NC2(CCNC(C(C=C)C)=O)CCC2)CCN(C)C1=O Cn1ncc(C(F)(F)F)c1CNC(=O)NNC(=O)c1cccc(Br)c1 C1(Nc2c(CC)ncnc2CC)CCCC2CN(C(=O)OC(C)(C)C)CC12 N1(C(CC(=O)OCC)=O)CC(CCNC(C2CCCC2)=O)C(C)C1 C1(CNC(C(c2ccccc2)OCC)=O)CCCN(C(=O)Cc2ccon2)CC1 N1(C(CC(C)C)=O)CC2CC(C1)N(C(c1cc(C(C)C)nn1C)=O)C2.CC(=O)N Cc1nn(CC(=O)NCC(C)(C)CNC(C2(CO)CCCC2)=O)c(C)c1C c1(C(=O)NCCCCCCNC(c2nc(OC)oc2)=O)cc2ccncc2[nH]1 Cc1[nH]cc(C(N2CCCCC(N(C(=O)C#CC3CC3)C)C2)=O)c(=O)c1Br N1(C(CC(C(C)C)NC(C2C(C)=CCS2)=O)=O)CC(C2CCCC2)C1 N1(C(C(CCC(C)C)NC(CCCOCC)=O)=O)CCCCCCCCC1 Cc1[nH]c(C(N2CCOC(CNC(C3CC3(F)F)=O)C2)=O)c(C)c1[N+](=O)[O-].C C1CN(C(=O)CC2CS(=O)(=O)C2)CC1c1nccn1C.CCCC(C)=CC=O.N C1(C(N(CCN(C)C(C2CCCOC2)=O)C)=O)CCCCC1 c1(C(N2CC(C)(NC(C3N(C)C(=O)CC3)=O)C2)=O)cc(N)c(O)c(F)c1 CCCCCCCCNC(=O)Nc1ccc(CCC(=O)NCCC2CCCC2)[nH]1 C1(C2CC2)(CNC(CCC2C(C)(C)C2)=O)CCN(C(c2ccnc(F)c2)=O)C1 c1(C(N(C(C)CN(C(=O)CC(F)F)C)C)=O)ccc(-n2cccn2)nc1 N1(C(C(CC)C(=O)OC)=O)CC(NC(=O)CN2CCCC2=O)CC12CCOCC2 c1(C(c2n(CCCC(=O)OCC)nnn2)NCCCCO)coc2ccccc12 c1(C(N2CCC(C)(NC(c3ccnc(C)n3)=O)C2)=O)cc([N+](=O)[O-])cnc1O CC(C(=O)NCC1CCN(C(=O)CN(C)CCO)CC1CO)C(C)(F)F CC(CS(C)(=O)=O)C(=O)NCC(C)(C)NC(C1CN2CCC1(C)CC2)=O C1(C(N2CC(F)(C(=O)NCc3cn(CC)nc3)C2)=O)CC2CCC2C1 c1(C(=O)Nc2cnc(I)c(Cl)n2)csc2c1CCN(C(C1CCCC1)=O)C2 N1(C(CC2(COC)CCOCC2)=O)CCC2(CC1)CC2.C1(C=O)CC(C)=NO1.N N1(c2nc(N3CCC(c4n[nH]c(C)n4)C3)cc(C)n2)CCc2nc(O)[nH]c2C1 N1(C(C(CC(C)C)OC)=O)CCC2(CCN(C(C3CC3(C)C)=O)C2)C1 C1(C(=O)OCC)CCC(C2C(C(=O)OC)C2)N1C(=O)OC(C)(C)C CC(C)CC(O)CC(=O)NC1COC2(C)CC1C2.C1(C(=O)N)C(C)(C)C1(C)C C1(C(=O)NCC(CC(=O)NCCc2scc(C)n2)O)CN(C)CC(C)O1 N1(C(c2cncc(C)n2)=O)CCCC(O)(CNC(=O)C(C)S)C1.C1CCCO1.C c1(CC)c(C(=O)NCCc2ccc(C)cc2)cccc1C.C(=O)C(F)C1CC1.N c1(SCC)cnccc1C(=O)NCC1CC1NC(=O)C(C)(O)CC N1(C(C(C)c2ccsc2)=O)CCC(CNC(=O)CCc2ccsc2)C(F)(F)C1 c1(C(N2CCC(NC(CC(C)C)=O)C2(C)C)=O)ccc2c[nH]nc2c1 c1(C(=O)NC(CC(C)NC(=O)CSC(F)F)C)cc[nH]c(=N)c1[N+](=O)[O-] C1(NC(C(N(C(=O)C(=O)C(C)(C)C)C)C2CC2)=O)CCc2ncnn2C1 CCCC(CC)C(=O)NC1CCCC1NC(=O)Cn1c(C)ccc1C C1(C(=O)NCC2(CNC(C(C3CC3)SC)=O)CC2)CCC(C)O1 Cc1cc(=O)oc(C)c1C(N1CC2CC(NC(=O)C=O)C1C2)=O.c1ncc[nH]1.N C#Cc1cccc(C(N2CCOCC2CNC(c2cnsc2)=O)=O)c1F N1(C(CN(c2ccccc2)CC)=O)CC2CC(C1)C2NC(c1ccccc1O)=O C(=O)(C(=O)NC1(COC)CCC1)NC(C)C.C(C=O)=CC.N(C)C.N C=CCC(C(=O)N(CC(=O)NC(C)(C)CCCO)CC1CC1)NC(C)=O CC1CC(NC(c2ccc([N+](=O)[O-])[nH]2)=O)CN(C(=O)Cc2cc(Cl)cs2)C1 C(CC(=O)N)(C(F)(F)F)OC.C1(C(C)C)CCCN1C(=O)CC1CC(=O)C1 N1(CC(=O)N(C(C)C)CC)C(=O)c2ccccc2C1=O.C(=O)C(F)(F)CCC N1(C(C(C)OCC=C)=O)CC(C(N2CCC(F)(C(N)=O)C2)=O)C2(CC2)C1 Cc1cc(C(=O)NC2CN(C(C3CC4(C3)CC4F)=O)CC2C)c(N)c(C)c1 Cc1ccc(C)c2[nH]c(C(=O)N(C3CN(C(=O)C(=Cc4c[nH]cn4)F)C3)C)cc12 N1(C(c2cccc(OC(C)C)c2C)C(=O)NCCSC)CCC2CCCCC2C1 CCC(CC(=O)NC1CCN(C(C2CCC(C(=O)OC)CC2)=O)C1C1CC1)OC C(C(C)C(=O)N1CCC(N(C(C2CC2c2csc(Br)c2)=O)CC)C1)OCC O=S(=O)(c1ccc(NCC2CC3CCC(C2)O3)c(F)c1)N1CC2CCC(C1)C2O N1(C(CCNC(N)=O)=O)CCC2CC(CNC(c3n[nH]c(O)n3)=O)CCC2C1 N1(C(C(C(CC)C)=O)=O)CCC(C(N2CC(OC)CC2CO)=O)CC1(C)C C(=O)(N=S(C)(=O)c1cnn2c1CN(C(C1(Cl)CC1)=O)CC2)c1ccc(C)c(O)n1 C1(SC)CCCC1NC(c1cc(C)[nH]n1)=O.c1(C(=O)N)cocn1.C1CC1 C(CCCCC(=O)N1CC(NC(=O)C=Cc2ccc(Cl)cc2)C(O)C1)NC(C)=O C1(CNC(c2n(C=C)nnc2)=O)CN(C(C2(C#N)CCCC2)=O)CC2(CCC2)O1 Cc1cc(C(=O)NCC2CC(C)CN(C(=O)CC3CCCC3)C2)cc(C)c1 Cc1ncc(Cl)cc1CC(=O)NCC(C)(O)CNC(=O)CSC(F)F C(C)(C(C(=O)NCCc1noc(C)n1)C(C)C)NC(COCCCC#C)=O N1(C(c2c(C)c[nH]c2)=O)Cc2n[nH]cc2C1C(=O)NCC1C(C)(C)C1(F)F c1(CNC(C2(N(C(C(C)NC(CC)=O)=O)C)CC2)=O)nccn1C C(=O)(C1CCNc2ccccc21)N1CCC(CCNC(C2=CC(C)(C)C2)=O)CC1 c1(C(=O)O)ccnc(-c2cnn(CC)c2)c1.c1(NCc2cccs2)ccccc1 c1(C(N(CC(CC)NC(=O)C(F)OC(F)(F)F)C)=O)nn(C)c2c1CSCC2 c1(OC)cccc(SC(CNC(=O)C(C)O)CO)c1.c1cccc(C(C)=O)c1 N1(CC(CC)OC)CCC2(CC1)CC(C)N(C(c1ccc(C)c(Cl)c1)=O)C2 c1(NC)cc(C(N2CCC(C)(NC(c3nc(C)c(C)s3)=O)C2)=O)cc(Cl)n1 C1(CNC(C2C(CC)C2)=O)C(C2CC2)CCN1C(C1CCc2cncn2C1)=O N1(CC(=O)NC2(CO)CN(C(C3(C)CCCO3)=O)C2)CCN(C)CC1.C1CC1 CC(C(=O)NC1(C2CCCCN2C(=O)CC)CC1)C(F)F.c1(C=O)ccoc1.N C1(NC(c2cc(O)ncn2)=O)CC2CC1N(C(C1CCCCS1)=O)C2 N1(C(c2ccc(OC)nc2)=O)CC=C(CC(=O)N2CC(C3(C)CC3)C2)CC1 C1(CC(=O)NC2CC(NC(c3c(C)nccn3)=O)C2)CC2CCC1CC2 C1(Sc2n(C)nnn2)CCN(C(c2cccc(C3CCC34CCC4)c2)=O)CC1 N1(C(c2c(C)scc2)=O)CCC(NC(=O)CC(C)C)C1C(C)C.[SH](C)(=O)=O C1(C(N(CC(=O)NC(C)(C)C)C)=O)CC(=O)NC1(C)C N1(C(C(C)OC)=O)CC(C(=O)N(C)Cc2ccccc2F)C2(CC2)C1 N1(C(C2C(C)OCCC2)=O)CCCC2(CC(NC(C3CC(=O)N3)=O)C2)C1 C(C)(C(CC(=O)NC1C(C)C1C)NC(c1cc[n+]([O-])cc1)=O)OC n1(CC)ccc(C(=O)NCCCCCCNC(c2cccc(NCC)c2)=O)c1C c1(CC(=O)NC2CC2NC(=O)CC2CCC3(CCC3)O2)ccnc(Cl)c1F CCCCC(C)C(=O)NC1(CO)CCCN(C(=O)C=CSc2nc[nH]n2)C1 Cc1sccc1CC(=O)NC(C)CN(C)C(c1occc1Cl)=O CC1(C)C(C#N)C1(C#N)C(N1CCC2(CCC2)C1)=O.C(=O)(CCn1cncn1)N C(=O)(C(F)C(F)(F)F)N1C(CN(C(C(c2cccc(Cl)c2)C)=O)C)CCC1 Nc1cc(F)c(O)cc1C(=O)NC1CN(C(=O)C(=O)NC2CC2)CC12CCC2 c1(NC(C(CCOCC)NC(=O)CCOCCC)=O)cnc(OC)c(C)c1 C1(C(=O)N)CCCC2C1C2(F)F.Cc1ccc(C)c(C(=O)NC2CCC(C)C2)c1 C1(C(N2C(CNC(c3c(C)cc(N)cn3)=O)CCC2)=O)CCc2ncc(C)n2C1 N1(C(CC2N(C(COCCC)=O)CC2)=O)CCCCC1CC(C)C C(=O)(C(N)CCC(=O)O)NC1CCN(C(N)=O)CC1 N1(Cc2cnc(C(=O)OCC)nc2)CCN(c2ccc(C)cc2)C(=O)C1 N1(C(C(=C)C(F)(F)F)=O)CC2(CCN(C(C3(Br)CC3)=O)C2)C1 CCC(C)CCC(=O)N(C)CC1C(C)(C)C1(C)C.C(=O)C(C)Cn1cccn1.N N1(C(CN(C(=O)OC)C)=O)CCC(NC(c2coc(C)c2)=O)C(C)C1 C1(C(=O)NC2C3CCC2N(C(c2ccc([N+](=O)[O-])s2)=O)C3)CCOCC12CCC2 N1(C(CCCCC)=O)CCCC2(CCCN2C(=O)CC2OCCCO2)C1 N1(C(C(C2CC2)SC)=O)CC(C2CCCN(C(=O)C(c3ccccc3)C)C2)C1 c1(C(=O)NC(C)CCNC(=O)C(C)(C)c2ncco2)cccc(CC#N)c1 C(=O)(CCCCCC1CC1)NCC(C(=O)N(CC(CCC=C)O)C)C c1(C(=O)NCCC2CCCN2C(C2CCC3(CC3)C2)=O)cc2cccn2c(O)n1 c1(C(N2CC(NC(C(OC)OC)=O)CC2(C)C)=O)cc(F)c(F)c(F)c1 c1(C(=O)NCC=CCNC(C(CCCC)(C)F)=O)cc2c(Cl)cc(F)cc2[nH]1 c1(C(=O)NCC2CC2)cccc(C=O)c1.C1(C=O)CCCCC1.C1CC1.N c1(NC(=O)CN2CCNC(c3cccc(C(=O)O)c3)C2)cccc2c1CCCO2 CN1C(=O)CN(CC(=O)NC2CC(O)CN(C(=O)C(C)(C)CCF)C2)C1=O C(=O)(C(CC)(CC)CO)N(CC(CC)NC(=O)CCn1ncn(C)c1=O)C O=C1CC2(CCC2)C(C(N2CCCC2Cc2cn(CC3CC3)nn2)=O)N1 C1(NC(C(CC)C)=O)(COC)CCCN(C(=O)C(=O)Cc2ccc(F)cc2)C1 C1(NC(c2ccsc2Br)=O)CCN(C(=O)CCF)C1 Cc1nn(C)c(F)c1C(N1CCCCC(NC(c2cnc(C(C)(C)C)[nH]2)=O)C1)=O c1(C(=O)NCC(CN(C(CCNS(CC)(=O)=O)=O)C)C)cccc2ccncc12 N1(C(C(C)SC)=O)CC(CO)C2(C1)CN(C(=O)CSc1cnn(C)c1)C2 CCC(O)C(F)(F)C(=O)N1CC(NC(c2ccc(Cl)c(C)c2)=O)C(CC)C1 C12(CC(F)(F)C1)CS(=O)(=O)NCC2.N1(CC)CCN(C2CCCCO2)CC1 c1(C(N2CC(CC)(NC(C3CN(C4COC4)C3)=O)C2)=O)ccnc(CO)c1 Cc1[nH]c(C)c(C(=O)NC2CCCC2NC(C2CCS(=O)(=O)CC2)=O)c1C N1(C(CC(CNC(CCCC(C)C)=O)C2CCC2)=O)CCCC2C(O)CC12 CC1CCC(=CC(=O)N(CCCNC(=O)C(F)OC(F)(F)F)C2CC2)C1 N1(C(c2ccc(OC)cn2)=O)CCCC(C)C1CNC(c1ccon1)=O c1(C(N2CC3(CN(C(C(P(C)(C)=O)O)=O)C3)C2)=O)cc2ncccn2n1 c1(-n2cc(COC3CCN(C(CC(O)C(F)(F)F)=O)C3)nn2)ccc(Cl)cc1Cl Cc1ccc(C)c(CNC(=O)CC2CN(C(c3c(Br)cnn3C)=O)C2)c1 CC1CCC(NC(C2CCCCC2C(N)=O)=O)CN1C(=O)CC#N C1CC2CC1CN(C(=O)Cn1nc(C)cc1C(F)F)C2.C(F)(C(=O)N)=C(C)C c1(C(=O)NCC2(CNC(CCC(C)N(C)C)=O)CCC2)cccc2c1nnn2C Cc1nc(C2CN(c3ccncn3)C2)no1 c1(C(N2CCN(C(c3ccncc3)=O)C(CCO)C2)=O)ccc(=O)n(CCO)c1 C1(NC(c2scnc2Cl)=O)CN(C(c2cnn3c2CCC3)=O)C2(CCC2)C1 c1(OC)ncccc1CCNCc1oc(C2CC2)nc1C c1(NC(C(N2C(C)CC(N3CCOCC3)C2)=O)=O)ccc(Cl)c(Cl)c1 CCCC(C)CCCC(=O)NC1CCC(NC(=O)C(=Cc2c[nH]cn2)F)CC1 C12(C(=O)NCC3(OC)CN(C(C(C=CC)O)=O)C3)CCCN(CC1)C2 C(N=c1cnc(F)c[nH]1)C1OCC(CNC(CCOCC2(C)CC2)=O)C1 Cc1coc(-c2ccccc2)c1C(=O)NCC(O)CNC(c1c[nH]nc1F)=O C1(NC(c2cc(Br)sn2)=O)CC2CC(C1)N(C(=O)CCc1cncnc1)C2 C(=O)(C1CCc2nccn21)NCC1C2CN(C(C(C(CC)O)C)=O)C1C2 C(=O)(C(Cc1cn[nH]c1)NC(=O)C1CC1)NC(C)CCC1CC1 N1(C(CCc2ncc(C)[nH]2)=O)CCC(NC(=O)C(c2ccc(C)s2)C)C1C(C)C C1(CCNC(c2cccs2)=O)CSCCN1C(=O)CCc1nccs1.C1CC1.C c1(C(C(=O)NCC)N(C)CC2CC3CC2C2CC32)oc2ccccc2c1Br c1(OC)ccc(Cl)cc1C(=O)NCCC(C)CCNC(=O)COCCF C=CCCCC(C(=O)Nc1cncnc1O)NC(=O)CC(C)CC C(=O)(C1=NOC(C)C1C)NC(C(=O)N(CCC=C)CC)CC#CC CCC(CC)CC(C(=O)NC1CCOC1)N1CCCCC1C(C)(C)C C(=O)(C(C)(C)CC(=O)NCC1CN(C)CCN1C(=O)CCCN=[N+]=[N-])OCC c1(OC)cccc(C(c2cccs2)NCC(Cl)=CCl)c1 C1(C(=O)NC(C2(O)CN(C(=O)CC(F)(F)C(F)F)C2)C)CC2CCC1C21CC1 c1(NCc2ccc(C)o2)c(C)[nH]c(C(N2CC(C)(O)C2)=O)c1C C(CC(=O)NC(CO)C(C)(C)C)(C(C)(C)C)NC(C=CCCC(C)C)=O CC1(C)CCCC(C)(C)C(NC2CCSC(C)(C)C2)C1 CC(CC(C)(F)F)C(=O)NC1(C)CC(NC(c2ccn3nccc3n2)=O)C1 N1(C(c2ccn(C(CC)CC)n2)=O)CC2(CCCCN(C(=O)C#CC3CC3)C2)C1 CC1=NS(=O)(=O)NC(C)=C1CCC(=O)NCC1CC1.C(=O)CCC.C(N)=O N1(C(C(C)OC(C)(C)C)=O)CCCCCC1C(=O)N(C)CCc1ccccc1 CCCCCC(C)C(=O)N1CC2CN(C(c3ccc(OC)s3)=O)CC12 C12CCCN(C1)C2=O.c1(CC)occc1C(=O)NC1CCC(NC(C)=O)C1 C1(OC)Cc2ccc(C(=O)OCc3cc4ccncc4[nH]3)cc2C1 CC(N=c1[nH]c(=NCCc2nc[nH]n2)[nH]c2ccc(Cl)cc12)C1CCCCCC1 C1(C2CN(C(=O)C=CC3CCCCCC3)C2)(NC(=O)CC2CCNC2=O)CC1 C1(C(N2CCC(N(C(C)=O)C)C2)=O)CCCN(C(c2ncccc2F)=O)C1 N1(C(COC(CC)C)=O)CC2CC1(C(=O)NCCN1CCCCCC1)C2 N1(C(C(CC(F)F)N(C)C(c2c[nH][nH]c2=N)=O)=O)CC2CC(F)CC2C1 N1(C(C2C(OCC)CC2)=O)CCSCC1C(N1CCOC(CC2CC2)C1)=O S(=O)(=O)(CCC(=O)N1CCC(N(C(=O)C(C)(F)F)CC2CC2)CC1)NC Cc1cc(C)c(C(=O)NCC(O)CN(C)C(C2CCn3ncnc3C2)=O)c(C)n1 C1(CNC(CN(C)CC)=O)CCC(NC(=O)CCC2CCOC2)CC1 N1(C(C2CC(C)(C)OC2(C)C)=O)CCC2CN(Cc3ccccc3)CC2C1 N1(S(c2ccn(C)n2)(=O)=O)CCC2(CCOCC2)C(CNC(C2CC=CC2)=O)C1 c1(C=O)cc(C)cc(C)n1.c1(OC)cccc(OCC(N2CCCC2C)=O)c1.N c1(N2CC(N(C(C(CN(C)C)c3ccccc3)=O)C)C2)nc(Cl)nc2sccc12 C1(C(=O)NCC(C)(CO)NC(C2OCCC2C(C)C)=O)(CC)CCOCC1 Cc1c(C(=O)N(C(C)CNC(=O)C(C)(O)C2CCOCC2)C)ccn1C1CC1 C1(NC(c2cccc(C)c2)=O)CC2CN(C(=O)C3=CC(C)(C)C3)CC2C1 c1(C(=O)NC(C(=O)NC(C(CC)CC)C)Cn2cncn2)ccc2c(c1)CCC2 CC1CC(NC(=O)CC2CCCCCC2)CN1C(=O)COCC(C)(C)C n1(C2CCN(C(C(CC)NC(C)=O)=O)C2)cnc2c1c(=O)n(C)c(=O)n2C C1(NC(C(C)S(N)(=O)=O)=O)CN(C(c2cc(N)cc(O)c2)=O)CC(C)(C)C1 c1(C(=O)NCC2N(C(CN(CCC#C)C)=O)CCC2)c[nH]c(=O)cn1 C(=O)(C1CCCc2nn[nH]c21)NCCC1CN(C(Cc2ccn(C)n2)=O)C1 c1(C(N(CCC(c2cccs2)NC(C=CC=CC)=O)C)=O)c[nH]nc1F C1(NC(c2n(C)ccn2)=O)CN(C(=O)Cn2cnnc2O)C2(CCCC2)C1 C1(C(N(CCCC#C)CC)=O)CN(C(=O)COCC(=C)C)CC1(F)F C(CC1=CCN(C)CC1)NC(C(C(C)CC)N(C(c1cncc(CC)c1)=O)C)=O C(CCO)(C(=O)NCC(C)(O)CNC(C1(CN(C)C)CC1)=O)N(C)C C1(NC(CC2(C#N)CC2)=O)CN(C(=O)COc2nc(O)nc(O)n2)CCC1O c1(C(N(C(C)C)CCNC(C2C=CC=CC=C2)=O)=O)cncc2c[nH]nc12 C1(N(C)C(C2CSCCS2)=O)CCCCN(C(=O)CNC(N)=O)C1 C1(c2ncc(C(=O)NCc3sc(O)nc3O)s2)CC12CCOc1ccccc12 Cc1cc(CCC(=O)NC2CC(CNC(C3(F)CCOC3C)=O)C2)cc(C)c1 C1(NC(CC)=O)CCCN(C(C2CCN(C(C3(F)CC=CCC3)=O)CC2)=O)C1 C1(NC(C2CC3CCC2O3)=O)CC12CCN(C(c1ccc(I)c(Cl)c1)=O)CC2 N1(C(C2C(C#C)C2)=O)CC2=C(C1)CN(C(c1cccc(N3CCCC3)n1)=O)C2 c1(C(=O)NCC(CC)NC(=O)CC2CCCC2(F)F)cnn2cccc(OC)c12 c1(C2N(C(C(=O)Nc3csc(CC4CC4)n3)=O)CCC2)cc(Cl)cc(Cl)c1 C(C(C(=O)N(C1CC2CC2C1)C)NC(c1ccc(C)s1)=O)OCC Cc1ncc(C(=O)NC(C)CNC(=O)CCCC2CCC2)c(C(C)C)n1 C(=O)(C1=CCN(C(=O)C(C)CC(F)F)CC1)NC(C)C(=O)NC(C)(C)C c1(C(=O)NC(CCN(C(CC(CC)C)=O)C)C)c[nH]cc(Cl)c1=O C(=O)(C(CN(C)C)C(C)C)NCCCCNC(C(C)NC(=O)NC)=O C(C(C)(O)CC(=O)NC(c1ccnn1C)C(=O)NCCC(C)(C)CO)OC C1(CNC(C2C(CC)CCCC2)=O)CN(C(=O)C(=O)NCC(F)F)CCCO1 CCCC(CCCO)C(=O)N1CCCC(NC(=O)CC2CC3(CC3)C2)CC1 Cc1cc(C)c(NC(=O)COC2CC(NC(=O)Cc3ncc(C)o3)C2)o1 N1(C(CCSC)=O)CCCC(C(C)C(=O)N(C2CC3(CC3)C2)C)C1 CC(C)CC(C)CC(=O)N1CCC(C(C)(C)NC(=O)Cc2nccn2C)C1 Cc1cccc(C(=O)NCC2CCN(C(=O)C(C)(C)CF)CC2C)c1C#N N1(C(C(C)NC(CC)=O)=O)CC2(CCN(C(c3cccc(C4CC4)c3)=O)CC2)C1 C1(O)(C(=O)NC(C)CCCCNC(c2cncs2)=O)CCCC(C)(C)C1 C=C=CCCC(=O)N(CC(CC)NC(C1CC1c1ccc(OC)cc1)=O)C c1(C(=O)NC2CC(NC(C(CCCOC)C)=O)C2)nc(O)nc(O)c1OC C(CN=c1[nH]cnc(Cl)c1C(=O)Nc1ccn(C)c(=O)c1)C1CCCC(C)C1 N1(C(CC(=O)OCC)=O)CCCC2(CC(NC(c3nnc(O)nc3O)=O)C2)C1 c1(C(=O)NCC2CN(C(=O)Cc3ccncc3)C2)c(Cl)ccc2c1OCO2 N1(C(C(C)OCCC(C)C)=O)CCCC(C)(C)C1C.c1(CC=O)ccsc1.N C1(C(=O)NC2(C#C)CC2)CC2CC1CN(C(=O)C(C1CCOCC1)=O)C2 C#CCC(C(=O)NC1CC(NC(=O)C=CC=C(Cl)Cl)C1)C1CC1 c1(CNC(C(=O)NC(CC)C)CC2COC(C)(C)O2)nc(O)c2ccccc2n1 N1(C(C)C(=O)N(C)C)CC(NC(=O)CCN2CCCC2=O)CCC1C CC1(NC(=O)C2=CCCCO2)CCCN(C(C2CCCNS2(=O)=O)=O)C1 C1(NC(c2ccccc2)=O)CCC2(C1)CN(C(c1cc3ncsc3[nH]1)=O)C2 CCCCC(C)(F)C(=O)NC1C2CC(NC(C3CCC(C)(C)C3)=O)CC12 c1(N(C(C(C)N(C(=O)C=CC(F)F)CC)=O)CC)cc(OC)ccc1F N1(C(C(=O)Nc2c(CC)cccc2)C)CCc2nc(C(=O)O)[nH]c2C1 c1(C(N2CCN(c3cnnc(Cl)c3Cl)CC2)=O)ccc([N+](=O)[O-])o1 O=C(CCC(=O)c1cccs1)NC1(CO)CN(C(=O)C=Cc2ccncc2)C1 Cc1cccc(C(C(=O)NC2CC2)N(C)Cc2ccc(C(C)(C)C)cc2)c1 C1(NC(c2cncnc2)=O)CN(C(C2OCCC2C2CC2)=O)CC1n1cccn1 C1(O)(CCNC(=O)COc2cccnc2)CCN(C(=O)C(F)C2CCC2)C1 c1(-c2c(NC(c3ccc(OCC)c(F)c3)=O)cccc2)c(OC)cccc1C#N c1(OCC)ccc(-c2noc(CNC3CCCC3C#N)n2)cc1 c1(CN(C(NC(C#C)C(C)(C)C)=NCC2CCCO2)C)cccc2ccccc12 C1(C(=O)NCC2CCC(C(=O)NCC(=O)N(C)C)C2)COCCOC1 C1(CC)CCOCCN1C(C1C=CCN1C(=O)C(=O)C(C)C)=O c1(C(C)=O)cc(NCCC2(O)CCN(C(=O)C(C)C(C)O)CC2)ccc1[N+](=O)[O-] C1(C(N2C(C)CCC(NC(c3c(C)[nH]c(C)c3C)=O)C2)=O)CCCCCS1(=O)=O c1(OC)ccc(C(C)C(=O)NCCN(C)C(c2nc(Cl)ccc2N)=O)c(C)c1 C(CCOCCO)(C(=O)Nc1cccc(Cl)c1)NC(C(C)=CCC)=O c1(CN(C(=O)CC2CCN(C(=O)CN3CCOC3=O)C2)C)nnc(O)o1 c1(NC(C2C3CN(C)CC23)=O)ccc(F)cc1O.c1ccc(C(F)(F)F)c(Cl)c1 CC(CC(=O)NC1CC(CNC(c2ccc(O)nc2)=O)C(O)C1)C(F)(F)F C1(C(=O)OC)CCCC(C(=O)OCC2CCCC2OC(C)(C)C)C1 C(CCCC(=O)NC1CN(C(=O)C(C2CCCCC2)NC(C)=O)C1)OC c1(C(=O)N)cc(F)c2nc(O)ccc2c1.C(=O)(CC(C)C(=O)NC1CCC1)OC Cc1cc(C(=O)NC2COCC2CNC(=O)C)nc(C)n1.c1ccc(O)cc1 C1(C)(NC(C(c2coc(C)n2)N(CC(C)C)CCC)=O)CCS(=O)(=O)C1 N1(C(C2(C)CC3CC3C2)=O)CC2CC(NC(=O)C=C3CCC3)C(C2)C1 c1(CC(N2CCC(C)C2C(=O)NCC=Cc2ccco2)=O)ccc2c(c1)CC2 C(=O)(CS(=O)(=O)CC(C)C)N1CCCC(N(C(CC(C)C)=O)C)C1 CN1CCC2CCN(C(=O)C(C)(CO)NC(=O)C3=CC4(CCOC4)C3)C2C1 c1(C=O)cc(S(N)(=O)=O)sc1C.Cc1cc(C(N2CC(C)C(C)C2)=O)c(C)[nH]1 CN1CCc2[nH]nc(C(=O)N(C)CCNC(c3cn(C(F)(F)CO)nn3)=O)c2C1 Cc1cc(C)c(C(N2CCN(c3ccnnc3)CC2)=O)c(O)n1 N1(C(c2c(CC)nc(C)[nH]2)=O)CCCC12CCN(C(=O)C(C)c1cccs1)C2 c1(C(N2CCCC(CN(C(=O)C3=CCOC3)C)C2)=O)ncnc(O)c1F c1(C(=O)NC2(CNCc3cccc4c3OCO4)COC2)cn2cccc(Br)c2n1 C1(COC)CN(C(=O)C(C)(Cl)Cl)CCN1C(=O)CC1CC(=O)NC(=O)C1 N1(C(C(N2CCSCC2)C)=O)CC(NC(=O)CSc2ccccn2)CC12CCC2 C1(NC(C2CC=C(C)CC2)=O)Cc2ccccc2N(C(C2CCCCC2O)=O)C1 N1(C(C(CCOC)C)=O)CCCCC(C(N2C(CO)CC2CO)=O)C1 N1(c2c(C)c(NC(C)Cc3nccn3C)ncn2)CCc2ncncc2C1 C(C)(C)(CCC)NC(C(C)OCCOC)=O.c1cccc(O)c1.C(=O)C.N C(C(CC(C)C)C(=O)N)OC.N(S(=O)(=O)NC)CC(=O)N(CCC)C1CC1 N1(C(CC2(OC)CCC2)=O)CC2(CCCC(C)O2)C1.C(=O)C(C)CC(F)(F)F.N C1(C(=O)NC2C(C)COCC2)CC(C)(C)CN1C(=O)CC=C(Cl)Cl C(C)(CCCCNC(=O)CCC(C)c1ccc[nH]1)NC(C(C)SCC)=O c1(CN(C(c2ncccn2)C)C)ccc(C)cc1.C1(C=O)CCCO1.N(C)C.N N1(C2CCCN(CC(C)(C)C)C2=O)CCC2(CC1)OCc1ccccc12 c1(C(N(C(C)CCNC(=O)CC2CCC23CCC3)C)=O)ccnc2ccncc12 CC1C(NC(C2CCC(C)(C)C2)=O)CC2CCC1N2C(c1cc2c[nH]nc2s1)=O C1(C(N2CCC(C#C)C2)=O)CC2(CC(NC(c3nc(Cl)cs3)=O)C2)C1 C1(NC(c2c(C)nc[nH]2)=O)CC(F)CN(C(c2cc(Cl)ccc2Cl)=O)C1 Cc1n[nH]c(C)c1CC(N1CCC(C(C)C(=O)NCC2(C#N)CC2)C1)=O C(=O)(C(C(C)(C)C)C1CCCC1)NC(C)CCCNC(c1cc(O)cs1)=O C(=O)(C(C)CCCC(C)C)N(CC(=O)NC(C#C)(C)C1CCCC1)CCOC C1(C(=O)NCC(CC)(CC)NC(=O)Cc2cnccc2C)CCCCC(C)(C)C1 c1(C(=O)NCC(C(C)C)NC(c2c(C)nsc2)=O)cccc(NC(C)C)c1 C1(CCNC(=O)C(O)C2CC2)CSCCN1C(c1cc(C2CCCC2)ncn1)=O c1(C(N(CC(C)CNC(c2ccnn2C)=O)C)=O)cccc(C(F)(F)F)c1F N1(C(C(COC(C)C)NC(c2cnc(CC)nc2)=O)=O)CCC(O)C(C)C1 Cc1c(C(=O)NCC(F)CNC(=O)Cc2ccc(Cl)cc2)sc2cccc(F)c12 C1(C(=O)NC2(c3nc(C)on3)CC2)CCN(C(=O)CCO)C12CCC2.CC(F)F CCC(CC(F)(F)F)C(=O)NC1C2CN(C(C3C4CN(C)CC34)=O)CC12 N1(C(C2CC(NCc3c(C)cc(Cl)nc3)C2)=O)CCn2cncc2C1 c1(C(=O)NCC2CC(NC(c3c(C)n(C)cn3)=O)C2)nnc(O)nc1O C#CCCCC(C)C(=O)NCCCCC(=O)NCC(C)(O)CCO c1(C(C)NC(C(C)CC(N)=O)=O)ccc2c(c1)CN(C(=O)C(F)=C1CCCC1)C2 C#CCC(CC(F)F)NC(c1sccc1CNC(C1CC2C=CC1CC2)=O)=O c1(OCCCC(=O)NCC(CN(C(C(C)CF)=O)C)(C)C)ccc(F)cc1 C1(C(C)C)CN(C(=O)Cc2cccc(N(C)C)c2)CCC1NC(=O)C1=CCC1 C1(COC)CCCN(C(=O)CN2CC3CC3C2)C1.C1(C=O)CCNC(=O)C1.C CCC(C)CC(C)N(C)C(C1C(C)CN1C(c1cccnn1)=O)=O Cn1cc(C(C(=O)NC2CC2)NC(=O)COC2CCOC2)cn1 C(=O)(C(O)C1=CCCCC1)N1CCC(C)(CC(=O)NCC(=C)C(F)(F)F)C1 C1(CNC(c2c(C)ncc(C)c2)=O)CC2CC(C1)N(C(=O)CCC(F)(F)F)C2 Cc1cc(Cl)cc([N+](=O)[O-])c1C(=O)NC1CCC(NC(=O)C)C1.C1CCCC1 c1(C2(C(=O)NC(C3CCN(C(c4c(C)[nH]cc4)=O)C3)C)CC2)cccc(Cl)c1 c1(NCCC=C=CC)nc2ccccc2nc1NC(c1ccco1)C c1(C(=O)NC2CC(C)N(C(=O)CC3CCCC3)CC2)cc(S(N)(=O)=O)co1.C C(CCC(C)C)(C(=O)N)NC(C)=O.C1(O)(CC)CN(C(=O)C=C(C)Cl)C1 C(=O)(CCC(=O)NCCCO)NCCC.c1(C(=O)N)cc(-c2cnn(C)c2)on1 N1(C(C(CCC)CC)=O)CC2(CCN(C(C3CN(C(N)=O)C3)=O)C2)C1 N1(C(c2cc(-c3ccc(C(C)C)cc3)[nH]n2)=O)CC2CCCC1CCC2 N1(C(CCc2ccc(C)s2)=O)CC(C)CC1C(=O)NCC(c1ccccc1)O c1(OCC)cc(OC2CC2)ccc1C(=O)N.C(=O)(C(C)(F)F)N1CCC1 CC1CN(C(c2nncs2)=O)CC1CNC(c1c[nH]ccc1=O)=O C#CC1CCC(CN(CC(=O)NC2(CSC)CC2)CCC)CC1 c1(CC(N2CCC(OCCNC(C(C(C)(C)C)O)=O)C2)=O)n[nH]c2ccccc12 C=CCC(CC)C(=O)NC(C)C(=O)N(C(C)CC1CC1)C N1(C(C2CC(OCC)C2)=O)C2CCC1CN(C(=O)C(C)(C)C(C)(C)OC)C2 C1(NC(c2n(CC)nc(Br)n2)c2nnnn2C2CCOCC2)CCOC(C)(C)C1 c1(CNC(C(C)O)=O)ccc2c(c1)CCN(C(=O)Cc1ccc3n[nH]cc3c1)C2 C(=O)(CC(C)(C)C(=O)NCC(C(=O)N(C1CCOC1)C)C(C)(C)C)OC c1(NCC2CN(C(C(C(CC)CC)C)=O)CC2C)nc(Cl)nc2nc(Cl)n(C)c12 C1(C(=O)N)CCC(C)(C)C1.C=C1CC(C=O)(C(F)F)C1.CC(C)N(C)CCC c1(CNC(CN(C2CCC2)C(C2(C)CC2(F)F)=O)=O)ccnc(F)c1F N1(C(c2c(CC)[nH]cc2)=O)CC2C(CNC(=O)CC(=O)NC3CC3)C2C1 Cc1ccc2nc(NC3CN(C(c4cnc(CC5CC5)s4)=O)CC3C)sc2n1 c1(C(=O)NCC2CCN(C(C(C)OCC)=O)CC2O)ccc2cnccc2c1 C1(O)(CCNC(C(C)OC)=O)CCN(C(c2sc(C3CCCCC3)nc2C)=O)C1 C(=O)(C(CC(C)C)C(N)=O)N1CCN(C(C2C(=C)C2)=O)C(CO)C1 O=C(C(O)CC(F)F)NC1CCC(NC(c2sccc2-n2cccc2)=O)C1 c1(C(C)(C)C)c[nH]nc1C(=O)NCCCN(CCO)C(C1(C)CCCO1)=O CCC(CC)(CO)C(=O)N1CC(NC(c2cc(Cl)ccc2OC)=O)C1 CC1(CC(=O)NCC2CC2)CCN(C(=O)CCC2CCC2)C1 C1CCC12CCC2.c1(C=O)ccc(O)nc1C.C(=O)(C(C)N)NCC(=O)OC c1(-c2cn(CC(C)Nc3ncc(Cl)cn3)nn2)cccc2c1C(=O)NC2=O C(=O)(CC(C)N(C)C(C1COC(=O)N1)=O)NCCCCOCC C(=O)(C1=CCC(F)(F)CC1)N(C1CCN(C(=O)CCC2CC2)CC1)C N1(C(c2[nH]cc(C)n2)=O)CCCC(Cc2cn(CC3CC3C(F)(F)F)nn2)C1 C(CC(=O)N1CC(C)(NC(=O)CCNc2cncnc2)C1)(C(C)C)OCC c1(C(=O)NC(C(=O)NCCC(CCC)C)CCN(C)C)c[nH]c2ccccc12 C1(NC(=O)NCC2N(S(CCCC)(=O)=O)CCC2)CC2CCC1CC2 N1(C(C2N(C(CSCCOC)=O)CC(O)CC2)=O)CCn2nc(C)cc2C1 Cc1ccc(Cl)cc1OCC(=O)NC1CCC1NC(c1coc(O)n1)=O N1(c2nc(N3CCCC(CS(C)(=O)=O)C3)cc(C)n2)CC2CCC1C(O)C2 CCCC(CC(=O)O)NC(=O)CCCn1cc(CC(O)Cc2ccccn2)nn1 CP(C)(=O)C1(O)CCN(CCOc2ccc([N+](=O)[O-])cc2)CC1 N1(c2nccc(C)n2)CCC(C)C(CNC(=O)CC2CC3CCC2CC3)C1 N1(c2nc(C)nc(O)c2C)CCC2(CCC2)C(NC(=O)CC2CCNC2=O)C1 N1(C(C(C)C2CC2)=O)CCC2CC12C(=O)NC1CC2(CCC2)C1 N=c1[nH]c(=NCC2CC2)[nH]c(=NCC(CO)c2ccc(Cl)cc2)[nH]1 c1(C(N(C2CCN(C(=O)CNC)C2)CCC)=O)cccc(Nc2ncccn2)n1 N1(C(C2(C)CCC2)=O)CCN(C(C2CC(n3ccnc3)C2)=O)CC1CS(C)(=O)=O c1(C(=O)NCC(c2ccccc2)NC(CCN(C)CC)=O)nc(OC)ccc1F c1(CNC(CC2(N(C)C)CC2)=O)nocc1C(=O)N.C(C(N)=O)C1CC1 c1(C(=O)NC2COCCN(C(C3(CC#C)CCC3)=O)C2)c(C)ccc(F)c1O c1(C(N2CC(C(C)NC(CCCCCC)=O)C2)=O)ccc2c(c1Cl)OC(F)(F)O2 C(=O)(CC(C)C(C)(C)CC)N1CC2N(C(c3c(CC)ocn3)=O)C(CC2)C1 C(=O)(C1=CCCCC1)N(C1CCN(C(C2(O)CC(CF)C2)=O)C1)CCC N1(c2n(CCC#C)c(C(CC)CC)nn2)CCC2(CCCCC2)C1 c1(C(N2CCC(O)(CNC(CC(C)O)=O)C2)=O)ccc(C(F)F)cc1F CCC(CNC(=O)CCc1cccs1)NC(=O)C(C)SC(F)(F)F N1(C(CCC(C)(C)C)=O)CC(C(=O)NC2(C(N)=O)CCOC2)CC(C)(C)C1 C=CCCCCCC(=O)N1CCC(O)(CCNC(=O)CCc2nccn2C)CC1 C1(CC)(NC(C2(NC(N)=O)CC2)=O)CCCN(C(=O)CC)C1.CC(C)C C1(NC(c2ncc[nH]c2=O)=O)CC12CC(NC(C1(C(F)F)CC1)=O)C2 N1(CC(C)C)CCCC(CNC2CCCC2C(=O)Nc2nc(Cl)cs2)C1 c1(C(=O)NCCC(C)NC(CCCCC#C)=O)cnn2c1NCCC2 c1(C(=O)NC(C)(C)C=CC(=O)NC2CC23CCC3)ccc(F)cc1 N1(C(C(CN)N)=O)CCC2(CCC2NC(c2cc(I)ccc2O)=O)CC1 C1(NC(C2(CC3CC3)CC2)=O)CCCCN(C(=O)C(F)F)C1 N1CC(C)c2ccccc21.C1OCCC1C=O.C1(C(=O)NC)(C(=O)N)CC1.C C1(CC(N2C(C(C)NC(=O)C(=O)N)CCC2)=O)CCC(=O)N1C.CC(F)F O(C=CC(O)(CNC(=O)NCC1(CO)CCCOC1)C(F)(F)F)CC C=CCC(C)(C)C(=O)N1CCOCC(NC(=O)CCNC(=O)NC)C1 C1(OC)CC2(C1)CC(NCc1cccnc1N1CCCCC1)C2 C1(NC(C(C=C=C)C)=O)CN(C(=O)C(C)(C)CC)CC(C)(C)C1 Cc1cc(C)c2[nH]c(=NC3CCN(C(=O)CS(=O)(=O)CC(C)C)C(C)C3)sc2c1 C1(C(=O)NCCC2N(C(c3c(C)nsc3)=O)CCCC2)CCC(O)CN1C N1(c2nnc(CCOC)s2)C2CCCC1CN(C(=O)CN1CCNC(=O)C1)C2 CC1(C)CN(C(C2CC(=O)NC2(C)C)=O)CCN(C(C2CCCCC2(C)C)=O)C1 N1(CC(=O)NCC(CNC(C(CCC)OC)=O)(C)O)OC(C)(C)CC1=O C1CC(=O)N2CCC(O2)C(=O)NOCCN1.C(=O)(C1CC1)OC C(C)(C(=O)NC1(CCC=O)CCC1)(C1(C)CC1)OC.c1(CC)nc(=O)o[nH]1 Cc1ccc(O)c(CC(=O)NC(C)CC(C)NC(C2(C)CCCC2)=O)c1 c1(C(=O)NNC(=O)c2ccc(O)nc2)c[nH]c2nccc-2c1 c1(C(=O)NCC(CC)NC(=O)C=C(C)C(F)F)ccc2nnc(C)n2c1 c1(OCCC)ccc(C(=O)NC(CNC(=O)CCC(C)SC)CC)cc1CC O(NC(=O)C(CC1CCOCC1)NC(=O)C(CC)OC)CCOCCOC C1(O)(C(C)NC(=O)C(O)C(F)F)CCN(C(c2ccc(C(N)=O)s2)=O)CC1 c1(CNc2c(F)c(Cl)ccn2)c(F)ccc2c1OCO2 C1(CC(=O)N(C)CC2COCCO2)N(C(=O)C=C2CCOCC2)CCC1(C)C C(C(CC(C)C)C(=O)NC12CC1CN(C(=O)CCc1c[nH]c(=N)[nH]1)C2)OC N(C1CCOc2cc(F)cc(F)c21)C(c1cc(C)nn1C)=O c1(CN2C(C(=O)NCCC(C)CO)CNCC2)cc(Cl)c(Cl)cn1 C#CCC(C(=O)N1CCC(CCN(C)C(c2ccc(C(C)C)o2)=O)CC1)C1CC1 C=CC1(CC(N2CCC(CCO)CC2)=O)CN(C(=O)C(N2CCOCC2=O)C)C1 c1(C(C)C)nc(Cl)cc(=NCC(C)(C)NC(C2CCC3CC3C2)=O)[nH]1 N1(C(CSCC)=O)CC(NC(=O)C(C)(C)OC(C)C)CC1(C)C CCC(C(=O)N1CC(C(N)=O)(CNC(=O)C=Cc2ccncc2)C1)C(C)C C(=O)(CC(F)(F)C(C)C)NC1(CNC(c2c(CC)[nH]cc2)=O)CCC1 N1(C(C=CCOC)=O)Cc2ccccc2CC1CNC(C1(OC)CC1)=O C12(N(C(Cc3cc(NC(CC)C(=O)O)no3)=O)C)CC3CC(CC(C3)C1)C2 C1(C(N)=O)CN(C(c2cncs2)=O)CCC1NC(C1CS(=O)C1)=O c1(C(=O)OC)c(C(=O)NC(C)CC)cnn1C.c1(C=O)nn(C(F)F)cc1Cl Cc1c(C(N2CC(CC(C)NC(=O)CN3CC4CC4C3)C2)=O)cccc1CO C12(C(=O)NC(c3c(C)nccn3)C)CC(CO1)N(C(=O)C(C)NC=O)C2 Cc1cnc(NCc2cnoc2C)c(S(=O)(=O)NC)c1.C1CCCN(C(C)C)C1 c1ccc(F)cc1.C1(C(=O)NC)(CC)CCCC1.C1CC1.C(=O)C=CC C1(C(N(CCN(C(C)=O)C)C)=O)CCN(C(c2cc(Cl)cn2C)=O)C1C c1(C(N2C(C)(C(=O)Nc3ncccc3C#N)CC2)=O)ccc(Cl)c2[nH]ccc12 C1(CNC(C(CC=CC)C)=O)CN(C(c2cnc3ccccn23)=O)CC12CCC2 C=CCCCC(C(=O)N1CCCOC(C)(C)C1)NC(c1ccc(=O)n(C)c1)=O c1(C(=O)N)c2c(nn1C)CCC2.CC(C)C(C)CNC(=O)CC12CCCC1C2 C(=O)(CC(C(F)(F)F)N(C)C)NC1C(C(=O)NCCc2scc(C)n2)OCC1 N1(C(C(C)N(C)CC)=O)CC2(C1)CN(C(=O)C(C)CC(C)=O)C2 c1(C(c2nnnn2C2CCC2)NCC2(C)COC(=O)N2)nc2ccccc2s1 CS(=O)(=O)CC(=O)NC1CCCC(NC(=O)Cc2cscn2)C1 n1(CC)ncn(NC(=O)CC(O)CNC(c2n[nH]c(C)c2C)=O)c1=O S(=O)(=O)(c1cc(C(C)(C)C)c(OC)cc1C)N(C1CC(F)(F)C1)CC Cc1cnc(C(=O)N(CC(C)(C)NC(=O)CCC(=O)c2ccncc2)C)c(C)c1 C1(OC)CCCCC1C(=O)NCc1ccc(C(=O)NCCc2ncc[nH]2)s1 N1(CC(=O)NC2CCCC2)CCNC(=O)C1.c1(CC=CCC=O)ccccc1.N C(=O)(C(O)Cc1cn[nH]c1)NCC(C)(C)OCC(=O)OC O=S(=O)(c1ccc(N2CCOC(C3CC3)CC2)c(F)c1)NC1CC2(CCC2)C1 c1(C(N(CC(C)NC(c2cccc(OC(F)F)n2)=O)C)=O)ccc(Cl)nc1O C12(C(=O)NC(CCC)CCC)COCC1CN(C(=O)C(CC)CCOC)C2 C1(CNC(c2cc(C)cc(F)c2)=O)C2CCCC1N(C(C1CC(C)CO1)=O)C2 c1(C(N2CC(OC)C(NC(=O)Cc3scnc3C)C2)=O)cnc(N)c(N)c1 Cc1nc(-c2ccsc2)sc1C(=O)NC1CN(C(c2cc(=O)cc[nH]2)=O)C2CC12 C1(CNC(c2c[nH]c(=NC)o2)=O)COC(C)(C)CN1C(=O)C(O)C(C)C N1(C(c2n(CC(C)C)ncc2)=O)CC2CC(C1)C2.C1(=CC(=O)N)CCSCC1 CC(C)(C)CCCC(=O)N1CCCC1CC(=O)NC1CC1C1CC1 c1(C(C(N2CCCC(N(C(C=NOC)=O)C)CC2)=O)C)cccc([N+](=O)[O-])c1 C1(CNC(C(=O)NCC)=O)CC2(CCN(c3ncc4ncn(C)c4n3)CC2)CO1 C#CCCCCCC(=O)NC1COCCC1NC(C1(C(O)C(F)(F)F)CCC1)=O c1(C(N2CC(OCCNC(=O)C(F)=C3CCCC3)C2)=O)ccc2nc[nH]c2c1 N1(C(C2C(C)C2)=O)CCOC(C(N2CCCCC2C)=O)C1.c1cn(CC(=O)O)nn1 N1(C(CCC(=C)Cl)=O)CC(NC(C2(c3ccc(C)cc3)CCC2)=O)C(C2CC2)C1 c1(C(N2CC(C(C)NC(C(C)N3CCC3)=O)C2)=O)cnc(C(N)=O)cn1 CC1CCCN(C(c2ccc(Cl)nc2)=O)C1CNC(c1ccc(F)o1)=O C#Cc1ccccc1CC(N1CCC(C)C1C(N1CC(N(C)C2CC2)C1)=O)=O C(=O)(CC1=Cc2ccccc2C1)NC(C(C(C)C)NC(c1ncc[nH]c1=O)=O)C C1(NC(C(=O)NC(c2ccccc2)C2COCCO2)=O)CCC(C(F)F)CC1 Cc1ccc(C)c(CNC(C2CCCN(S(=O)(=O)CC#N)CC2)=O)c1O N1(C(C2(C)CCCOC2)=O)CCC(C2(NC(C34CCC(CC3)C4(C)C)=O)CC2)C1 CCCC(C(O)C(=O)NC(C)(CO)CCF)NC(=O)Cc1ccnn1C C1(NC(C(CC#C)C)=O)CN(C(C2CC2C)=O)CC2(CC2)C1 C1(NC(c2cc(OC)no2)=O)CC2CC1CN(C(C1CCCCCC1)=O)C2 c1(OC)cc(O)ncc1C(=O)NCC1(O)CCN(C(=O)C(C)C(C)C)C1.O N1(C(CCN(C(c2conc2C(C)C)=O)CC)=O)CC2(C)COCC2(C)C1 c1(C(=O)NCC2CN(C(CC)=O)C3(C2)CCC3)cccc2occ(Br)c12 C1(C(=O)NCC2CSC2)CC(NC(C2CC23CCCC3)=O)C(O)C1 C1(C(=O)NCC2CC(NC(C3(C#C)CC3)=O)C2)CCC(CC)C1 C(=O)(CC(O)C(C)CC)NCCn1cc(C(NOCC(=O)OCC)=O)nc1 C1(CNC(CN(CCC#C)C)=O)CCC(C)(C)CN1C(C1CC2CC2C1)=O c1(NC(C2N(C(Cn3c(C)cc(C)n3)=O)CC=C2)=O)cnc2cc(F)ccc2c1 C12(CC(N3CC(NC(c4cccc(C5CCCOC5)c4)=O)C3)=O)CCC(CC1)C2 c1(N(C(C(CCCC)O)=O)C2CC2(F)F)ncc2ccc(F)cc2n1 C(CC(C=O)NC(C1CCOC1C(C)C)=O)OCC.C1CCC1.C(N)=O.N C1(C(=O)NCC2C(NC(Cc3c(C)n[nH]c3C)=O)C2)CCCCCCC1 C(=O)(C(Cc1ccccc1)S(C)(=O)=O)N(C(CN(C(C=C(CC)C)=O)C)C)C C1(CNC(CC(=O)OCC)=O)CC2CCC1N2C(=O)C(C)(C)C(F)F C1(NC(=O)CCc2nncn2C)CCN(C(C2(CC(=O)N(C)C)CCCC2)=O)C1 c1(C(N2CCC(O)(C(C)NC(c3cc[n+]([O-])cc3)=O)C2)=O)cc(O)ccc1O Cc1cc(Cl)c(C(N2CCN(C(=O)CC3C=CCCC3)C(C)C2)=O)cc1N Cc1ccc(C(=O)NCC23CC2CCN3C(C)C)cc1.C1CCCO1.C(=O)N C(=O)(C(C)(C)C(=O)NCC1CCC1)OCC.C(C1CCOC1)=CC=O N1(C(c2cc(C)cc(O)n2)=O)Cc2n[nH]cc2C1C(=O)N(C)Cc1ccccc1 Cc1cnc(Cl)c(S(=O)(=O)N2CCC2(C)C(N2CCC(C)(CO)C2)=O)c1 c1(C(=O)NC(CNC(c2cccnc2S)=O)C2CC2)ccn2ccccc12 C1(C(=O)NCC2C(C)(C)CCC2)CC2CCC(C1)N2C(c1ncccc1O)=O n1(CC)ncc(C(=O)NCC(C)(C2CC2)NC(c2scc(C)c2Cl)=O)c1C c1(CNC(CC(C)(C)NC(c2ccc(Cl)cc2)=O)=O)cccc(O)c1F c1(C(N(CC)CCNC(=O)CC2CC(C)C2)C)ccc(Cl)c(Cl)c1.C N1CCNC(=O)C1C.c1(C(N2CC(F)CC2C(=O)N(C)C)C)ccc(F)cc1 N1(C(Cc2ccc(S(C)=O)cc2)=O)CCC2CCC(C1)N2C(=O)Cc1cnns1 N1(C(=O)CC2OCCO2)CC2(C(=O)NCCCCO)CC1CCO2 N1(C(c2cnc(C)o2)=O)CCC2CCC12CNC(c1cc2ccsc2s1)=O C(C(=O)NCCc1ccccc1)(C(C)O)NC(CCSCCOC)=O C12(C(N3CC4N(C(=O)CN5CCSCC5)CC(C4)C3)=O)CC3CC(C(=O)N1)C2C3 CC(C)C(C)(O)CNC(=O)C#CCNC(=O)COC(C)(C)C c1(C(C2CCOCC2)CNCC(C)C2CC2)ccccc1 c1(OC)cccnc1C(=O)NC(C)C(C)NC(c1cncc(-n2ccnn2)c1)=O C1(COC)CN(C(=O)CC(C)O)CCN1C(=O)CNC=O.c1ccccc1.N CC1(C)CC(CNC(=O)CCc2ccccn2)N(C(=O)CCN2CCC(F)C2)C1 C12(C(=O)NC3C(C(N)=O)COC3)CCC(CC1)N(C(=O)C=Cc1cocn1)C2 n1(CC(=O)N(C2CCN(C(=O)C(F)CC)C2)CCC)cc([N+](=O)[O-])ccc1=O N1(C(CCOCCOC)=O)CC(C)CN(C(c2cc(C)c(Cl)cc2C)=O)C(C)C1 c1(C(=O)NCC=CCNC(c2cscc2F)=O)nc(O)nc(O)c1F C1(CNC(c2c(C)cccc2)=O)CCC2(CCC2)C1NC(c1ccco1)=O c1(CC=O)c(F)cccc1C#N.c1(CSC)ccc(C(=O)NC2CC2)cc1.N C1(C(=O)N)CN(C)CCN1C.C1(NC(c2cnc(OC)s2)=O)CCC(C)(C)C1 C(=O)(CS(=O)(=O)CCCC)NCC(CC=C)NC(c1ccc(C(F)F)cn1)=O C1(NC(C(C)N(C)C(C2(C)COC2)=O)=O)CC2(C1)CC(O)C2 C1(C(=O)NCC(C)(F)C(C)C)CCCC(=O)N1C.C(C1C(=O)N1)OCC C1(NC(c2n(CC=C)nnn2)C2(c3ccncc3)CC2)CC=C(C)CC1 c1(C(=O)NCC(N(C(c2[nH]cc(C)c2)=O)C)C2CC2)cc2c(Cl)nccc2o1 c1(SCOC2CCN(C(C(=O)NCC)=O)C2)c[nH]c(C(N)=O)c1 Cc1c(C(=O)NCCC2(C)CCN(C(=O)C(C)O)CC2)sc2nnc(S)n12 N1(C(C2CCC(C)(CC)O2)=O)CC=C(C(=O)N)C1.C1CCN1C(C)(C)C.C C(CCCC(C)NC(c1ccc(OC(C)C)cc1)=O)NC(C(C=C)O)=O C(C)(C)(CCC(=O)NC(C)C(C)(C)C(=O)N1CCC(F)C1)OC C1(CC)CN(C(=O)CC2(C)CCCC2)CCN1C(C1C2COCC12)=O c1(Sc2cccc(-c3nc(C)c(C(=O)NC4CC4)cc3)c2)cc(F)cc(F)c1F C(=O)(CC(C)(C)CC(F)(F)F)NC1C(C)CCN(C(CCCCC(C)C)=O)C1 C(=O)(C(CO)C(C)(C)C)N(C)CC1CCCCN1C(=O)CC1CCCSC1 N1(CCCC(=O)NCC(C)NC(c2nc(Cl)cs2)=O)C(=O)CN(C)C1=O C(=O)(CCCC(CC)NC(=O)C=CC1CCOCC1)NC(CCC)(C)CC C(=O)(C1CCc2nccn21)N1CC(C#C)(C(=O)N(C(C)C(=O)OC)CC)C1 CC(C(=O)NCc1cn(CC)nn1)C(C)(F)F.c1cnn(C)c1.C(=O)(C)N CN1CCC(=CC(=O)N(C)CC2CCN(C(c3ccc(C4CC4)cc3)=O)C2)CC1 C(=O)(C(C)C(O)CC)NCc1ccc(C(N(CCOCC)C)=O)cn1 Cc1[nH]nc(C(C)C)c1C(N1CC(n2cc(CCO)nn2)C1)=O.C1CCCC1 c1(C(N2CCC(F)(C(=O)OC(C)(C)C)C2)=O)cccc2c1NC(=O)C21CC1 c1(CC(=O)NC(C)CCNC(C2(C)CCN(C)C2)=O)c[nH]c2ccc(F)cc12 N1(CC=C)CCC(N(C)C(=O)Nc2ccccc2CCN=[N+]=[N-])C1=O CCCC(O)CCN(c1ccc(Cn2cccn2)o1)Cc1ccncc1Cl C1(CC(=O)NC2CCC2(C)C)(NC(c2c(CC)ccs2)=O)CCCCC1 C1(CNC(=O)CC2(CO)CC2)COCC1NC(c1scnc1C1CC1)=O N1(C(Cc2cc(C)no2)=O)C2CCC1CN(C(=O)C1=NOC(C)C1)C2 c1(C(=O)N)ccc(C#N)c(Cl)c1.CC1CCC(C(N2CC(C3CC3)C2)=O)C(=O)N1 C1(CNC(c2cnc(OC)s2)=O)CCN(C(c2c(Cl)cccc2Cl)=O)C12CCC2 Cc1nc(C(=O)NCC2(CNC(=O)C)CCC2)c(C)o1.c1ccccc1Cl c1ccc(Cl)cc1C.C1(CC=C)(C(N2CC(CNC(=O)CC)C2)=O)CCC1.O C(=O)(C(C)C(F)(F)C(F)F)NC(CN(C(c1cc(OC)cc(C)n1)=O)C)C C1(C(=O)NC(CC)(C)CCO)CN(C(c2cc(F)cc(F)c2)=O)CC1(F)F c1(C(N2CCC(NC(C(=O)NCCOC)=O)CC2)=O)c(N)sc2c1CCSC2 Cc1cccc(OCC(=O)N(CCC)C(C)C)c1C.C1(C=O)CC12CC2(F)F.N C1(NC(c2cc(C)no2)=O)CC2(C1)CC(NC(=O)C=CCF)C2 C(=O)(CC(C(C)OC)NC(=O)C(=O)Nc1ccc(OC)cc1)OC c1(C(=O)N)ccnc(C)c1N.C(=O)(C(C)N(C)C)NC(C(=O)N(C)CC)C N1(C(C(CCCC)C)=O)CCC(C2(O)CN(C(=O)C=Cc3ccn(C)c3)C2)CC1 CC(F)(F)CCCC(=O)NCC(O)CNC(C1(C)CC1)=O c1(CC(N2C(COC)(C)CCC2)=O)cc(C)ccc1.C(=O)(CC=C(Cl)Cl)N C1(CC(=O)NCc2coc(CO)n2)CCCN(C(C2(CO)CCCO2)=O)CC1 C1(NC(CCC2CCC(=O)N2)=O)CCC(O)CN(C(c2cnn[nH]2)=O)C1 C1(C(=O)NCC=CCC=O)(CC)CC(C)(C)C1.C1(CC)CCOC(C)C1.N c1(C=O)cnc2c(c1)CNC(=O)N2.C(C)(C)(C(=O)NC1CCC(CC)C1)OC C1(CCNC(=O)C(F)C2CCC2)(NC(C(C)n2cncn2)=O)CCCC1 C12CCCN(C1)C(=O)c1cc(on1)CNC(=O)C2.C1(CCO)CC1.C1CC1.C c1(C(C(=O)NCc2ccco2)N(CC)CC2CCC2)ccc2c(n1)CCC2 N1(C(CC(C)C2CCCC2)=O)CC(C)(C)CC1C(=O)NCCN1C(=O)CNC1=O CC(C)C(O)C(C)C(=O)N1CCCC(C(=O)N(CCO)C2CC2)CC1 CC(C)C(F)C(=O)NCCCOC1CCN(C(c2coc(Cl)n2)=O)CC1 CC(C1=CCN(C)CC1)NCC(=O)N(C)Cc1ccc(OC(F)F)cc1 CCC(CCCO)N=c1nc2c(ncn2C(C)C)c(NCc2ccc(N)cn2)[nH]1 C=CCCC(C)C(C(=O)Nc1ccc(C(=O)OC)cc1)N1CCC(NC)C1 C1(NC(=O)CCc2ncccn2)CN(C(C2CCCCCCC2)=O)CC12CC2 C1(N(C(C=C(CC)CC)=O)CCF)CCCN(C(C2CC2C(C)(C)O)=O)C1 c1ccccc1Cl.c1(C(=O)NCC(C)CN(C(=O)C)C)ccc(C(C)(C)C)[nH]1 CCC(C)CC(C)NCCOc1ccc(C(F)(F)F)cc1 N1(C(c2cc(C)cc(N)c2)=O)C2CCC1CN(C(=O)CCc1cc(Cl)no1)C2 CCC(F)(F)CC(=O)NCC1CCC(NC(c2cn[nH]c2)=O)C1 Cc1cc(-c2cn(CCCN(C(=O)C(C)C3CCCO3)C)nn2)ccc1N CCCC(C)CC(=O)NCC(CC(F)(F)F)NC(c1cccc(O)c1Cl)=O N1(C(c2sccc2F)=O)CC2CCC(C1)N2c1ccc([N+](=O)[O-])cc1 c1(C(=O)NC2CCCN(Cc3n(C(C)C)ncn3)CC2)ccc2c(c1)CCO2 C1(CC(=O)N(C2CCCC2C)C(C)CO)(CN(C)C)CCCCC1 c1(C(=O)NCC2=CCN(C(c3c(OC)c[nH]n3)=O)CC2)nc2cnccc2s1 c1(CN(C(=O)NCC(C2CCCC(C)C2)(C)O)C2CC2)ccc(F)c(F)c1 c1(C(N2CCC(C)(NC(c3ccnc(C4CC4)c3)=O)C2)=O)cc(Cl)ncc1Cl N1(C(CCOC(C)C)=O)CCCC(NC(C2(C)CCCC2C)=O)CC1 c1(C(=O)NCCCC(C)NC(C2CCC(=C)CC2)=O)cnn2c1OCCC2 N1(C(C2(NC(C3CC(CC)C3)=O)CSC2)=O)CCCC(CF)C1 c1(C(=O)NC(CCCNC(COC(C)C)=O)C)cnc2ccc(C#N)cn12 c1(C(=O)NC2(C(NOCC(C)O)=O)CC(O)C2)cc(=O)n(C)cn1 C1(C(=O)Nc2c(C)ncnc2)CCN(C(c2cncc(O)c2)=O)CC1O C(C(CC(C)C)C(=O)NC(c1ccccc1)C(=O)NC1CCC(O)C(O)C1)OC c1(C(C(=O)NCCCN(C(C(CSC)OC)=O)C)O)cc(Cl)cc(Cl)c1 N1(C(CCSC)=O)CCC(NC(c2sccc2OC(F)F)=O)C(F)(F)CC1 C(=O)(C(C)(C)CC#N)N1C(CN(C)C(C23CC4CC2C3C4)=O)CCC1 C#CCCCCC(=O)NC(COC)CC(=O)NCC(C)(C)N1CCCC1 C1CCCCCC1.C1(O)(C(C=O)F)CCCC1.C(C=CC(=O)N)(CC)=CC.C c1(C(N(C(C)C)CCNC(C2CCCCO2)=O)=O)ccc2ccc(O)nc2n1 c1(C(N(CC)C2CC2)=O)ccc(Cl)nc1.c1(COC)ccc(C=O)cc1.N CCC(C(=O)OC)C(=O)N1CCC(CCCCNC(=O)C(N)=O)CC1 c1(C(=O)NC(CC)(C)CNC(=O)CC2=CCOCC2)cnc2c(c1)C(=O)CCC2 c1(C(NCCC)=O)c[nH]c(=N)c2[nH]ccc12.C(C=O)NC(=O)OC.C1CC1 c1(C(=O)N)ccc([N+](=O)[O-])s1.c1(NC)ccc(C(=O)NCC2CCC2)cc1 C1(NC(=O)CCc2ccccn2)CCN(C(=O)CCCF)C12CC2 c1(C(=O)NCC(C)N(CC#N)C)ccc(F)c(S(=O)(=O)N2CCCC2)c1 c1(CN(CCC(NOC)=O)C(c2ccc(C3CC3)cc2)=O)cccc(C)c1C Cc1ccc(C(C)NC(=O)CC2(C)CCN(C(=O)CC(C)(C)C)C2)cc1F N1(C(C(C(CC)O)C)=O)CC2CCN(C(C34CCC(C3)OC4)=O)CCC2C1 c1(CC(CC)NCC(F)(F)C2CC2)ccccc1 N1(C(C(C=C)CC)=O)CCC2(CCC2)C(NC(=O)C=CC2CCOC2)C1 C1(NC(CCCc2ccc(C)s2)=O)CC2(CCN(C(C3(O)CCSC3)=O)C2)C1 C(=O)(C1=CCCOCC1)NC1(C)CCN(C(CC2CCN(C(C)C)CC2)=O)CC1 C1(C(=O)NC(C)C(F)(F)F)C2CC2CN1C(=O)CC1CCCCO1 C#CCCCCCCC(=O)N1CCN(C(=O)CC2OCCO2)C(CC)C1 C1(c2cn(Cc3ccc(C)s3)nn2)C2CCCC1N(C(=O)CCC1CC1(F)F)C2 c1(OC)cccc(C(N2CC(NC(c3ncccc3C3CC3)=O)C(C)C2)=O)c1F c1(C(=O)NCC2(C)CCCN2C(=O)CCC2CCCOC2)noc2ncccc12 c1(C(=O)NC(C2CN(C(c3c(C#C)cnn3C)=O)C2)C)ccn2ccccc12 c1(C(=O)NCC(CN(C)C(c2cnn(C)c2N)=O)O)coc(S(N)(=O)=O)c1 N1(C(c2nn(C)c(=O)cc2)=O)CCC(C)(C)C(CNC(C2(F)CCOC2)=O)C1 C1(C(N2CCC(CC=C)(NC(c3ccoc3C)=O)C2)=O)CCOC2(CCCC2)C1 C(C(=O)N1CCC(NC(c2c(C)ncn2O)=O)C1C1CC1)(C(C)C)OC N1(C(c2nc(CNC(C3(CC#C)CCOC3)=O)oc2)=O)CCCCCCCC1 Cc1c(Cl)cnn1CC(=O)NC1CC(F)(C)C1.C(=O)C(O)Cn1cncn1.N C12(C(=O)NC3CN(C(CC(C)c4ccco4)=O)CC3O)CC(C)(C1)OC21CCC1 C1(CN(C(CSCC#C)=O)CC)CN(C(c2cc(O)n(CC)n2)=O)CCO1 n1(C(C)C)ccc(C(=O)NCC(C)N(C(=O)COC2CCOC2)C)cc1=O N1(C(C2(CC)CCC(=O)N2)=O)CCCC(COC)(NC(=O)CC(CC)CC)C1 CCCC(CCc1ccccc1)C(=O)N(C(C)CCC(F)F)CC CCCC(O)C(=O)NC1CC(NC(c2cccc(C3COC3)c2)=O)C1 C1(CC(=O)NC2CCN(C(=O)C(C)SC(F)(F)F)CC2)CCC2(CCC2)O1.C c1(C2(C(=O)NC3C(CNC(C(CC)C)=O)COC3)CC2)cccc(C#N)c1 c1(C(Cc2ncc[nH]2)NC(=O)CCc2cscn2)ccccc1 O=C(C1CCc2nccn21)OCc1nc2cc(Cl)ccc2s1 CC1(C)CCCC(C(=O)NCC2(C)CCC2)O1.C(C1CCCC1)=CC=O.N Cc1cc(C(N2CCSCC2CCNC(c2cc(F)c[nH]2)=O)=O)c(O)cc1F C(CC(C)C)(C(=O)NCCC(O)CCNC(=O)CO)OCC.c1ccccc1 C1(O)(CC)CCCN(C(C2(C)CCC(=O)N2)=O)C1.c1(OC)nn(C)cc1C=O C1(CC)CC(C(=O)N(CCCN(C(=O)CO)C)C)CCO1 Cc1cc(C(=O)N(CCCN(C)C(C2(C)CC(C)(C)C2)=O)C)c(N)s1 C1(NC(C2COCCO2)=O)CC(NC(C23CSCC2C3)=O)C(O)C1 N1(C(=O)NCc2cccc(OC(CC)C)c2)CCOCC2(CCSCC2)C1 C(=O)(CC(CNC(C)=O)C(F)F)NCCCCC(C)NC(CC(=C=C)C)=O C(=O)(NNc1ccc(C(=O)O)cc1)c1cccc(-c2cccc(C)c2C)n1 Cc1nc2ccccn2c1C(=O)NCCN(C(=O)CC(C)C(C)(C)C)C c1(SC)cc(C(=O)NCC2CC(C(=O)NC(c3csnn3)C)C2)oc1C C1(=C(C(=O)N)F)CCCCC1.C1(C(C)NC(C2CC(CC)C2)=O)CCCCC1 C1(CNC(=O)Nc2cnc(C(=O)OCC)nc2)CCCC(C)(C)CC1 c1(C(=O)NC(C(C)NC(C2CCCCN(C)C2=O)=O)(C)C)ccc(Cl)c(Cl)c1O c1(N2CCC(NC(C(CCOCC)O)=O)CC2)ccc(C(=O)OC)c(C)n1 c1(C(=O)N)cncc2nc[nH]c12.CC(C)C(C)C.C1(CC=O)C=CS(=O)(=O)C1 C1(CNC(C2(C)CCNC2=O)=O)CCCC12CCN(C(c1occc1Br)=O)CC2 C(=O)(C(C)(C)C)N(CCCCNC(=O)CCc1cc[nH]n1)C Cn1ncc(Cl)c1C(=O)NCC(C1(O)CCN(C(=O)CCCCC2CC2)C1)C O=C(C1=COCC1)NCC(O)CCNC(c1ccnc(-c2ccco2)c1)=O N1(C(CCC(C)(F)F)=O)CCC2(CC1)CC(NC(=O)CSCC(N)=O)CO2 Cc1ccncc1C(N1CCC2CC12C(=O)NC(C)C(C)C)=O C(=O)(CCCC(C)(C)C#N)NC1CCC(C(N2C(CC)CN(C)CC2)=O)C1 N1(C(C(C)SCCCC)=O)CCCCC1CN(C)C(c1scnc1C1CC1)=O CC1CCc2c(C(=O)N(CCNC(=O)CSC(F)(F)F)C3CC3)csc2C1 CC(C)CCC(F)C(=O)NCC1(C(=O)NC2CNC(=O)C2(C)C)CC=CC1 c1(N2CCC(NC(c3ccc(C(C)(C)C)[nH]3)=O)C(F)C2)nccn2nnnc12 n1(CC)c(N(CCCOC(F)(F)F)C)nnc1-c1ccc(OC)cc1.C1CCCS1 C=CC1(C(=O)N(C)CC2COCCN2C(C23CC(F)C2C3)=O)CCOCC1 c1(C(=O)NCC2(C)CCN(C(c3c(OC)ccs3)=O)C2)cc(O)ccc1F O=CC1=CC=CN2CCS(=O)(=O)N=C12.C1(CC)CCCN1C(=O)C=C1CCC1 N1(C(CCCc2ccc(C)s2)=O)CC(CNC(=O)Cc2cscn2)CC1C N1(C(C(CCC2CCC2)NC(C2C(C)(C)COC2)=O)=O)CCC(C2CCCC2)C1 C1(NC(c2ccc(CCC)s2)=O)CCN(C(=O)Cc2sc(O)nc2O)C1C N1(C(c2cc(C)[nH]n2)=O)CCN(C(=O)CCC2CCCN(C)C2)C(CF)C1 c1(-c2cn(C)nc2C(N2CCC(CCF)C2)=O)ncc(O)c(=N)[nH]1 c1(OC)cc(CC(N2CC(NC(=O)Cc3nn(C)cc3Br)C(C)C2)=O)ccn1 C(N=c1[nH]c(=N)[nH]c(=NC(C)CS(C)(=O)=O)[nH]1)c1c(CC)ccs1 CCCCCCCCCN(C)C(C1(C)CCCN(C(=O)CCC2CC2)C1)=O C#Cc1ccc(CC(=O)NC2CCCN(C(c3cc(F)cnc3O)=O)C2)cc1 c1(CC)ccc(O)c(C(N2CCCC(NC(=O)NC)C2)=O)c1 Cc1ccnc(C(N2CCC(CC(C)NC(C3CC3(F)F)=O)CC2)=O)c1F c1(OC(C)(C)C)ccc(OCC(=O)NC2CCCC2c2cccc(F)c2)cc1 c1(OC)cccc(CN2CCCC(F)(CNC(c3c(F)cncc3Br)=O)C2)c1O N1(C(CC(c2ccc(OC)cc2)C)=O)CCC2C(CCCN2c2nnn(C)n2)C1 N1(C(C(CNC(c2c(CC)ncnc2)=O)C)=O)CC2(C1)CN(C)C2 C1(CNC(c2ccc(F)cc2F)=O)CC2CCC1N2C(=O)CCC1CCCOC1 c1(C(=O)NC23CN(C(C4C(C)OCC4)=O)C(C2)C3)c[nH]c2ccc([N+](=O)[O-])cc12 c1(NCC2(CNC(c3ccc(OC)c(C)c3)=O)CC2)nccn2nnnc12 N1(CC(C)NC(C)(C)CC2CCOC2)CCOC1=O N1(C(C2(NC(c3nccc(OCC)c3)=O)CCCC2)=O)CCS(=O)C(C)C1 N1(C(C=C(C)C(C)C)=O)CCCC1C1CCCN1C(c1ccc(Br)cc1O)=O C(=O)(C(O)C(F)(F)F)N(CCC(=O)NC(CO)C1CC1)CC#C c1(C(=O)N)cnc(C(F)(F)F)nc1.Cc1ncsc1C(N1CCC(C(C)C)C1)=O c1(C(=O)NCCN(C)CC2(C)CCC(OC)CC2)ccc([N+](=O)[O-])c(Cl)c1 C(=O)(N1CCC(C(=O)NCC(N2CCOCC2)=O)O1)c1cc(C)[nH]c1C c1(C(=O)NCC(C)(CO)NC(C(C)n2ccnc2)=O)cc(F)c(F)cc1Cl C#CCCCCCC(=O)NC1CC2(C1)CN(C(C13CCCC1C3(F)F)=O)C2 CCC(CC)C(F)C(=O)NC1CC(C(=O)NC(CC2CCCC2)CO)=CC1O c1(CC)ncc(C(=O)NCC(CCOC)NC(c2ccnn2CCO)=O)[nH]1 c1(C2C(C)C2)cc(C(N2CC(C)(c3cn(C4CCCC4O)nn3)C2)=O)on1 c1(CN2CC(CC(=O)Nc3c(C)cc(Br)nc3)C2)ccc(C#N)c(Cl)c1 n1(CCOC)cc(C(=O)NC2CCC2NC(=O)CSc2cn[nH]c2)cn1 c1(CNC(=O)CCCn2ccnn2)nc(C)cc(O)n1.c1(CC=O)cnc[nH]1.N C1(NC(=O)CNc2ccccn2)CC=C(C(=O)N2CC3CCC3C2)C1 Cc1[nH]nc2cc(-c3ccc4c(c3NC(=O)CCc3ccco3)OCO4)ccc12 CC(O)C(C(=O)N1CCCC(NC(c2cncnc2)=O)C1)NC(=O)C1CC1 CC(C)(C)C(CO)NC(C1CCCCC1NC(=O)Cc1ncccn1)=O c1(C(=O)NC(C2CCN(C(C3CC4CCCC34)=O)CC2)C)cccc2cncn12 C1(CNC(C=CCCC)=O)CCN(C(c2cc(N(C)C)ccc2N)=O)C12CC2 c1(C(N(CCNC(CCCC(C)=O)=O)C)=O)cnc2ncnc(O)c2c1 C(=O)(C1=CC2CCCCCC12)N1CCC(CCCNC(c2ccc(Br)o2)=O)CC1 CC(C(=O)N1CC(NC(=O)Cc2cccnc2Cl)CC(F)C1)C(C)(C)C n1(CC(=O)Nc2ccccc2)cccc(OCC2CC3(CCOC3)C2)c1=O c1(C(=O)NCC23CCC2CN(C(C2(O)CCSC2)=O)C3)c(F)ccc(F)c1O c1(C(=O)NCCN(C(=O)C2=CCCS2)C)ccc(-n2cc(Br)cn2)cc1 C(=O)(CC(=O)NC(C)CNC(=O)C(c1cscn1)N(C)C)OC C1(C(N(CC(C)=O)C)=O)CC(=O)N(C2CCNCC2)C1 C1(CNC(C2(C)CC2)=O)CN(C(=O)C2CC2)CC1c1ccc(F)cc1 c1(C(=O)NC(C)C(C)(C)NC(C2CC(=O)NC(=O)C2)=O)ccc(Br)cc1F c1(C2(C(c3nnnn3CCCOCC)NCC(CC)O)CC2)cccc(Cl)n1 N1(C(Cc2ccc(C#C)cc2)=O)CCC2(NC(=O)COC3CC=CC3)CCCC12 c1(C(=O)NCC(C)N(C(C(Cc2c(C)n[nH]c2C)C)=O)C)cnn2c1OCCC2 Cc1cc2nccnc2cc1C(=O)OC1CCN(c2ccc(F)cc2)C1=O CC(C)N=c1nc(N2Cc3cccc(Br)c3C2)c2c(F)cccc2[nH]1 CC1CCn2c(C(=O)NC3(C)CN(C(c4cncnc4)=O)C3)cnc2C1 CON(C)C(=O)C(C)(C)NC(=O)NCCCc1ccc(O)cc1 C1(C(=O)NC2CC(NC(C(C)c3cccs3)=O)C2)COc2ccccc2O1 C(CC(C)C(=O)NC1(C(=O)NCCn2cnccc2=O)CCSC1)=CCC Cc1[nH]c(C)c(C(=O)NCC2=CCN(C(c3cccc(=O)o3)=O)CC2)c1C CCC(F)(F)CC(=O)NCC1(NC(c2ccnc(S)c2)=O)CCC1 c1(NC(C2(F)CCN(C(CCC(C)C)=O)C2)=O)cc(F)ccc1C#N C1(CNC(C2CCC(=C)CC2)=O)CN(C(=O)CC(=O)NC)CCC1(C)C c1(C(C)C)cccc(C(=O)N(CCC(C)NC(C2(C)CCCO2)=O)C)c1N CN=c1[nH]cc(C(N2CC(CCCCNC(c3cc(C(C)(C)C)on3)=O)C2)=O)o1 CCC(COC)C(=O)N1CC=CC(C(=O)NCCN(C)CCOC)C1 CC(CCC(C)(C)C)C(=O)N1CC2=C(C1)CN(C(=O)CSC(F)F)C2 CC1(C)CCCC(C(=O)NCC2CN(C(c3c[nH]c(=N)nc3O)=O)CCCO2)C1 C(=O)(C1=Cc2ccccc2C1O)N(CCCNC(C1CC(O)C1)=O)C CCCC(C(=O)OC(C)(C)C)S(=O)(=O)NCCCCN(C)C(C)=O c1(NC(=O)CNC(=O)C(F)n2ccnc2)cccc2c1OCC2 c1(NC(=O)NCCC2COCC3(CCC3)O2)ccc2c(c1)OCCO2 CC1CN(C(=O)C=Cc2ncc[nH]2)CCC1NC(C1(c2ccncc2)CC1)=O N1(Cc2ncc(CC)o2)CCC(C2(NC(c3cc(C)nc(O)n3)=O)CC2)CC1 CC(C)CC(C)(O)CNC(=O)Cc1cn(C)nn1.c1(C(=O)N)n[nH]c(=N)[nH]1 Cc1cc(=NC(=O)NNc2ccccc2C)[nH]o1 Cn1cncc1C1CC1C(=O)NCCCNC(c1nc[nH]c1C(C)(C)C)=O c1(CC(C2NCCN(C(c3c(C)cc(F)cc3)=O)C2)=O)cc2ccccc2o1.CC C#CC1(F)CCN(C(C2CCN(C(C3CC3(C)C(F)F)=O)CC2)=O)CC1 C1(NC(C2C(C)=C2)=O)CC2CCC(C1C)N2C(=O)Cc1c(C)cnn1C c1(C(=O)N)cnn2ccsc12.Cc1cnn(C)c1CC(=O)NC(C)(C)C1CCC1 Cc1c(C(=O)NC(C2CN(C(=O)Cn3cccc3)C2)C)[nH]c2ccccc12 c1(C(=O)NC(CC=C)CNC(=O)Cc2cncc(F)c2)c[nH]c2cccc(O)c12 c1(CC)cccc(C(=O)NCCC2CC(Nc3cc(C4CCCC4)[nH]n3)C2)n1 CCC(C#N)(CC)C(=O)NCC1CN(C(c2n[nH]cc2Br)=O)C1 C(=O)(CC1COCc2ccccc21)NCC(CNC(c1ncn(CC)n1)=O)OC c1(C(C(N2CCCC(N(C(=O)C=CCO)C)C2)=O)O)cc(F)c(F)cc1F C1(NC(COCC)=O)CCC2(CC1)CCN(C(=O)C(C)NS(C)(=O)=O)C2 c1(N2C3C(CNC(=O)CCc4cccc(Cl)c4)C(C3)C2)cc(Cl)c(O)nn1 CC1=NOC(C)(C(=O)NC2CC(N(C)C(c3cccnc3)=O)C2)C1.C1CC1.O C(=O)(CC(O)C(C)C)N1CC2C(CNC(CN3CCC(C)C3)=O)(C2)C1 c1(NCC(=O)NC)ncnc(NCCCCNC(C)C(N2CCOCC2)=O)c1C C1(CNC(C(c2ccc(CC)s2)=O)=O)CCN(C(=O)CC(C)C)CC1O C(=O)(CS(=O)(=O)C1CCCC1)NC(CCNC(Cn1ccc(C)c1)=O)C N1(CC(C(=O)N(C)Cc2c(C)ccs2)(C)O)C(=O)c2ccccc2C1=O Cc1cc(=O)n(C)nc1C(=O)NCC(C)CO.c1(C=O)cnn(CC(F)F)c1.N C1(C(=O)NCCC(C)NC(c2c(C)nc(C)[nH]2)=O)CC1C1(C)CCOCC1 c1(CC(C)C)ccc(C#N)c(N(C2CCN(C(c3cc4c[nH]nc4s3)=O)C2)C)n1 c1(C(N(CCNC(CC(C)(C)OC)=O)C)=O)cc(Cl)nnc1O Cc1sc(C(=O)NC2CC3(C2)CC3NC(=O)C(C)N2CCC2)c(Br)c1C c1(OC)nc(C)c[nH]c1=NNC(=O)c1ccc(-c2ccc(SC)cc2)cc1C#N C(=O)(C1=CC2(CCOC2)C1)N(CC(=O)NC(CC#CC)C)C(C)C N1(C(C(C)N(C(=O)CN2CCCC2=O)CCC)=O)CC(C)N(C)C(C)C1.CC C1(NC(CCOCCCOC)=O)CCCCC1CC(=O)NCc1ccno1.O N1(C(C(CCCC)F)=O)CC2N(C(c3ccc(CCC)cc3)=O)CCC2(C)C1 CCCCCC(C)CC(=O)N1CCCC(NC(=O)CN2CCc3sccc3C2)C1 c1(CC)cc(C(=O)NC(CNC(c2ccc(Cl)o2)=O)CC)c(C)o1 N1(C(C2CCCN(C(C)=O)C2)=O)C2CCC1C(C)C(NC(=O)CCC(C)(C)C)C2 N1(C(CCn2c(C)csc2=O)=O)CCC(C)(CCNC(=O)C(C)C2CC2)CC1 CCCCC(C)C(=O)NC(C)Cn1cc(CNC(c2ccncc2)=O)nn1 c1(C(N2CCC3(C(NC(C(CSC)O)=O)C3)C2)=O)cc2n(n1)CCCC2=O c1(C(=O)NC(CC(C)NC(CCC(C)OC)=O)C)cc2c(C)cccn2n1 C(=O)(CCC(F)(F)F)N(CCN(C(c1cc(Cl)c(C)cn1)=O)CC)CC C12CCCCCCC1CN2.C(C(C(=O)OC)NC(=O)OC(C)(C)C)OC C1(CC(N2C(C)(C)CCC2)=O)Cc2ccccc2O1.C1(C(C)(C)O)(C=O)CC1.N C1(NC(C=CC)=O)CCC2(CC1)CC2.C1(C=O)CCN(c2cnn(C)c2)C1=O c1(C=O)ccc(C#N)cc1.CC1(NC(=O)C)CCC1.C1(C=O)CCC(F)C1.N CC1CCC(NC(=O)CC2CCCC2)CN1C(c1csc(O)n1)=O Cc1ccc2[nH]c(C(=O)NC3CC(NC(C4CCCCC4C(N)=O)=O)C3)cc2c1 n1(CCC)ncc(C(=O)N(CC(C)N(C)C(C2CCN2C2CCCC2)=O)C)c1Cl C#CCC(C)(C)C(=O)NC(C1CCN(C(=O)CCCOC(C)=O)C1)C c1(OC)ccn2cc(C(N3CC4CC3C4NC(=O)CCc3ccon3)=O)nc2c1 c1(CC=O)cc(F)cc(Cl)c1.c1(C(C)C)occc1C(=O)NCC1CCCC1 CC1CCC(CC(N2CCC(N(CCC(F)(F)F)CCO)CC2)=O)CC1C C(=O)(C1CCc2nccn21)N1CCC(CN(C(C23OCC(CC)(C2)C3)=O)C)C1 c1(C(CO)NCc2c(OC(C)(C)C)cccc2)cc(Cl)cc(Cl)c1 c1(C(=O)NCC(C)NC(=O)CC(C)(C)C)ccnc(C2CCC2)c1 c1(C=O)cnc2n1CCOC2.N1(C(c2cc(OCC)n[nH]2)=O)CCC(O)(C)C1.N C1(C(=O)NCC2(NC(C(C)O)=O)CCCC2)CNC(=O)CC12CCC2 c1(C(=O)NCCC(N2CCOCC2)C)cccc2cc(Br)cnc12 C1(COC(CNC(C2CCCOC2)COCC)=O)CCCC2(CCC2)O1 Cc1onc(C2CC2)c1C(=O)NC(C)CCCC.C1(C(=O)N)CC(N(C)C)C1 C1(C2CCN(C(c3csc(C4CC4)n3)=O)CC2)(NC(C(COC)O)=O)CCC1 N1(C(c2ncn(C(C)C)n2)=O)CCN(C(=O)C#CC2CC2)CC1CO N1(C(c2c(CCNC(C3CCCN(CC)C3)=O)n[nH]c2)=O)CCCC[Si](C)(C)C1 C(=O)(C1CCCc2nn[nH]c21)N1CC(NC(=O)COCC2CCOC2)(CO)C1 C(=O)(C1CCc2c[nH]nc21)NC(C1CCN(C(C23CCC(CC2)C3(C)C)=O)C1)C C1(OC)CCCCC1C(=O)NCC12CC1CN(C(=O)C(C)(C)C#N)C2 c1(OC)ccc(F)c(C(=O)NC2CC(CNC(c3occc3Cl)=O)C2)c1Cl C(N=C(NCC1CCC(C)(C)C1)NC(CC)CC)c1n(CC)ncc1 C(=O)(C(CC(C)C)N(C)C)N(C1CCN(C(=O)C(C)OC)CC1)CCOC C#Cc1ccc(CC(=O)NCC2CC2NC(=O)Cc2cc(C)no2)cc1 C(=O)(C1CCc2nccn21)NC1C(C)CN(C(=O)C(c2ccccc2F)(C)C)C1 C1(CNC(c2c(SC(C)C)cccc2)=O)CCN(C(c2cc[nH]n2)=O)C12CC2 c1(SC)sccc1C(=O)NCC1CCC1NC(C1CCCO1)=O S(=O)(=O)(c1ccc(C(=O)NC2CC(C)N(C(=O)CCCF)C2)cc1)NC(C)C c1(C(=O)OC)cc(C(=O)NCC2CCCC2)ns1.C1(CC=O)CCOC1.C CS(=O)(=O)c1cccc(CN2CCC2C(N2CCCC2)=O)c1 C(=O)(CCC(F)(F)F)N1C(CCC(=O)NCC2(CC)CCOC2)CCC1 CS(=O)(=O)CCCC(=O)N1CCCN(C(c2ccc3occc3c2)=O)CC1 Cc1oc(CO)cc1C(=O)NCCC1CC(C(=O)NCCN(C)C)C1 C12(CNC(CC(=C)Br)=O)CCC1CN(C(C1CCN(c3ccccc3)C1)=O)C2 O=C(CC1CC1(F)F)NN=c1[nH]nc(-c2ccsc2)s1 C1(CCC(=O)N(CC(O)C)C)NC(=O)NC1=O.O(CP(C)(C)=O)CC(=O)N Cc1[nH]c(C#N)cc1C(N1CCC(CC(C)NC(=O)C(C)S(C)(=O)=O)CC1)=O C1(C(=O)NCC2(COC)CN(C(c3cncc(F)c3)=O)C2)CN(C)CCO1 O=C1CCCCC(C(N2CC3CC2C3C(=O)NC2CC3(CC3)C2)=O)C1 c1(C(=O)NC2C(CNC(C=CC=CC)=O)CCC2)ccc(Cl)cc1C N1(C(C(=O)NCC)=O)CCN(C(C2CC2C2CC2)=O)C2CCCC2(C)C1 N1(C(C2(OC)CCCC2)=O)CCC2CCC(NC(C3CCCCC3(C)C)=O)C1C2 C1(NC(CCCN(CCOC(F)(F)F)CC)C)CC2(CCC(F)(F)CC2)CO1 N1(C(CC)=O)CC2CC(C1)C2CNC(=O)Cc1ccc(Cl)nc1C.c1ccccc1 c1(C(N(C)CCNC(c2csc(CO)n2)=O)=O)cc(-c2cccs2)on1 N1(C(C(CC)C2CC2)=O)CCCCC(N(C(=O)CCCc2cccnc2)C)C1 C1(NC(C2(OCC)CCC2)=O)CC2CC(NC(=O)C=C(Cl)Cl)C2C1 C(=O)(C1CSc2ccccc21)N.C1(OCC)CN(C(c2cnc(O)s2)=O)CC1C C1(CCC)(NC(=O)C(C)NC(=O)OC)CCCN(C(c2cccs2)=O)C1 Cc1nccn1CCNC(=O)Cc1cnn(C)c1.c1(CCC=O)csc(=N)[nH]1 c1(C(N2C3CC(NC(c4c(C)cns4)=O)C(C3)C2)=O)cc2cccc(F)c2o1 C1CC2CCCC(C1)N2C(=O)CCN1CCC1.c1(NC(C)=O)nc(C=O)cs1.N C1(NC(CCC)=O)CCN(C(C2(SC)CC(=O)C2)=O)CC1C(N)=O C(=O)(C1Cc2ccc(F)cc21)NC1C2CC(NC(c3c(C)nccn3)=O)CC21 c1(CNC)nc(N2CCC(CCN(C)C)C2)nc2ccsc12 C(=O)(C1CCCn2cnnc21)N1CC2C(NC(c3cnns3)=O)(C2)C1 Cc1nc2c(s1)CN(C(c1ccncc1Br)C(=O)NCCCOC(F)F)CC2 c1(C(C)=O)cc([N+](=O)[O-])ccc1NCC1CN(C(c2ccno2)=O)C1 N1(C(C2N(C(c3c(CC)nns3)=O)CSC2)=O)CC(OC)CC1C(=O)O CC(C)CC(C)C(=O)NCC(CC1CCCC1)C(=O)NC1(C)CC2(CC2)C1 N1(C(c2cc(OCCN(C)C)ncc2)=O)C(C)C2CC1C2.C1(C=O)CCOC1.N C12(C(N3CCC(F)(CNC(=O)Cn4cnnc4O)CC3)=O)CCCN1CC(O)C2 C12CCCC(C1)NC2=O.C1(CC)(CO)CCN(C(=O)CCCN(C)C(C)=O)C1 c1(C(N2CC(CNC(C3(C)N(C)CCC3)=O)OCC2)=O)cc(=O)n2nccc2[nH]1 C(=O)(C1=C(C)C(C)(C)OC1=O)N1CCC2(CCN(c3c(Cl)cnc(OC)n3)C2)C1 C1(COCC(=O)NC)CCCCO1.C1(F)CN(C(=O)C(C2CCOCC2)O)C1 c1(C(=O)NCC=CCNC(=O)C(F)CC2CC2)cc(Cl)c(Cl)[nH]1 C1(C#N)(CCC(=O)N(CC(CC)NC(C2(O)CCC2)=O)CC)CCC1 N1(C(c2c(C)ccnn2)=O)CCC2CCN(C(C3CCC=CCC3)=O)C2C1 N1(C(C(C)=C(C)C)=O)CC2(C1)CN(C(C1CC3(CCC3)CO1)=O)CCO2 C=CCCCCC(=O)N1CCC2CC12C(=O)N(C1CCCCC1O)C Cc1c(Cl)ccc(C(N2CCC(O)(CN(C)C(C3COCCO3)=O)C2)=O)c1O N1(C(C(C)C#N)=O)CC2(CCC(CNC(c3cc(C(F)(F)F)ncn3)=O)O2)C1 C(=O)(C1CNC(=O)c2ccnn21)OCC(=O)N(C1CC1)Cc1ccc(C)cc1 Cc1c(NC(=O)N(C)CC2CCCS2(=O)=O)cnn1-c1ccccc1F c1(NC(CNC(c2nc(CC)sc2)=O)CC)ncnc2ccc([N+](=O)[O-])cc12 c1(C(N(C2CN(C(c3nc(Cl)c(=O)[nH]c3N)=O)C2)C)=O)cccc2c1CCO2 c1(C(=O)OC)ccc(C(O)CN2CCOC(c3nnn(C)n3)C2)cc1 N(C1c2ccccc2OC1C)C(c1c(C)onc1-c1cccs1)=O C=C(F)C1(CC(=O)N(C2CCCN(C(C3(N4CCCC4)CC3)=O)C2)CC)CCC1 CC(C)(C(=O)Nn1ccnn1)NC(c1c[nH]c2cccnc12)=O c1(C(N2CCN(C(CCN(CCC)C)=O)C(CC)C2)=O)c(F)c(F)cc(F)c1F C1(CCNC(CC2C(C)OCC2)=O)CCCCC1C=O.C(CCC1CC1)CC.N CC1CC(C(N2CCOCC(NC(c3n[nH]c(=N)[nH]3)=O)C2)=O)CC(C)O1 N1(C(c2cn(CC)nn2)=O)CCOC2(CCC(NC(C)=O)CC2)C1 Cc1ccc2c(C(N3CC4CN(c5cc(C(F)F)ncn5)CC4C3)=O)c[nH]c2c1 C(=O)(C1=COCCC1)N.C1(C(=O)N(CCC)C2CC2)(OC)CS(=O)(=O)C1 c1(SC)nc(O)c(CN2CCCC2C(=O)C2=NOC(C)(C)C2)cc1C#N N1(C(C(C)N2CCCC2)=O)CC(O)CC1CC(=O)NCC(C)(C)CCO C1(C(N(CCC(=O)N(CC(C)SC)C)CC)=O)OCCC1(C)C c1(C=O)ccccc1-n1cnnn1.C(=O)(C(F)=C(C)C1CC1)N(CCC)CC c1(OC)ccc(C(=O)NCC2CCN(C(=O)C3=CCCOC3)CC2)cc1C(C)C N1(C(C2CC(=O)OC2)=O)CCCC(F)(CNC(c2c[nH]cc2C2CC2)=O)C1 C1(CCCC)CN(C(C2(CC)CCOC2)=O)CCN1C(=O)CC(C)(C)COC CCCS(=O)(=O)C(C)C(=O)NC(CNC(=O)COCC(C)C)CC Cc1cnc2nccc(C(=O)NCC3CCCC(NC(c4cnc[nH]4)=O)C3)c2c1 CC1(C)CN(C(=O)CCOC2CC2)CCC1NC(=O)CCC[N+](=O)[O-] c1(N2CCCC(C(C)NC(C3(CC)COC3)=O)C2)cc(O)nc(O)n1 C1(C)CN(C(=O)CC2CCCS2(=O)=O)CCO1.C1(SC)CC(CC(=O)N)C1.C c1(C(=O)N)cc2n(n1)CCC2.N1(C(CC)=O)CCC(C(=O)NC(C)(C)CC)C1 C(=O)C(C)P(C)(C)=O.c1(CC(=O)N(CCC)CC)ccnc(C(F)(F)F)c1 C1(NC(COC(CNC(CC(CC)OC)=O)(C)C)=O)CCOC12CCCC2 N1(C(C(C)(C)NC(C=COC)=O)=O)CCC(C)C(O)C1.c1(C(=O)N)ccncn1 CCCCCC(C)CC(=O)NC1CCN(C(=O)C(C)(C)C(=O)OC)CC(O)C1 c1(OC)ncccc1CC(=O)NCC(C(C)(C)C)NC(=O)CCC(C)OCC CCCC(C(=O)NCc1cccnc1Cl)NC(=O)CCC(C)C C(=O)(C(CC(C)C)C(N)=O)NCC1CN(C(c2c(C)c(N)cnc2)=O)CC1(F)F C1(c2n(C)cnc2)CN(C(=O)CNC(N)=O)CC1.C(=O)C(O)CC1CC1.N C1(NC(Cc2ccn(CC)n2)=O)CCN(C(c2ccc(C)c(C)c2)=O)CC1CO CC1CCC(NC(=O)Cc2ccc(O)nc2)CN1C(C1CCCC1(C)C)=O c1(C(=O)NC2CCC(NC(c3cc(CCC)oc3C)=O)CC2)cc(C#N)[nH]c1C N1(C(C2(O)C(C)(C)OCC2)=O)CC2CCC(C1)C2NC(c1cc(F)ccc1F)=O Cc1cc(NCC(=O)Nc2ccccc2C(=O)O)c(C)cc1Br C1(C(=O)NC(C(=O)N(CC#C)C)(C)C2CCC2)C2CN(C)CC12 C1(CNC(=O)C=CC2CCOC2)(NC(=O)Cc2ccno2)CCCCCC1 C(CC1CC1)(CC(=O)NC)NC(COc1cc(C)on1)=O.c1cc(C)oc1C CCCC(CCCO)C(=O)NCCC1CN(C(=O)C(F)CC2CCCC2)C1 c1(C=O)cccc(N2CCCC2=O)c1.C(C)(C)OC.O(C(F)(F)F)CC(=O)N N1(C(c2ncn(COC)n2)=O)CCC(C(C)(C)C)(C(=O)OC)C1 N1(C(Cc2cc(OC)c(C)cc2)=O)CCCN(C(=O)C2=CC(O)CCC2)C(C)C1 N1(C(CNC(C(C)(C)C)=O)=O)C(C=O)CC2CC12.C1(C(N)=O)CCCOC1.N c1(C(=O)NCCN(C(C2CCC(C)O2)=O)CC)cccc2c1CCCC2=O C1CC(S(C)(=O)=O)C1.C1(C(N(CC)C)=O)CCS(=O)(=O)C1.C(CC)NC C(C(=O)Nc1cccc(NC(C2(Br)CC2(F)F)=O)c1)(C(C)C)OC C=C(C)C1OCCC1C(=O)NC1C=CC(CC(=O)NCCc2ncccn2)C1 C1(C(=O)NCCN(C(C2C(C)C2C)=O)C2CC2)C=CCCC1 C1(C(=O)NCC2C(NC(=O)CCN3CCCC3=O)CCC2)C(Cl)(Cl)C12CC2 CC(C)C(CCC(F)F)NC(C1CCCOC1c1ccccc1)=O N1(C(c2cc(C)oc2)=O)CC2CCC1CC2NC(=O)CCCC(C)C C(C)(C)(CCC(=O)N1CC2CC1CC2NC(=O)CCN1CCNC(=O)C1)OC C1(CNC(C(N2C(C)CCC2C)C)=O)CCN(C(=O)C=Cc2cncs2)CC1O n1(CC(N2C3CC(OC(C)(C)C)(C3)C2)=O)ncc2ccc(OC(F)F)cc2c1=O c1(C(N(C2CCN(C(=O)CC3CC34CC4)CC2)CC)=O)c[nH]c2nc(Cl)ccc12 CC1CN(C(c2cc(F)c(Cl)cc2Cl)C(=O)NC2(C)CC2)C(C)(C)CO1 C1(O)(CC)CCN(C(=O)CN(C)C(c2ccsc2)=O)C1.C(=O)CCN(C)C C(=O)(CC(O)C(Cl)(Cl)Cl)NCCN(CCC)C(c1cn2c(n1)SCC2)=O C(=O)(C(O)C1=CCCCC1)NCC1CCC(C(=O)NC2CC(O)C2)CC1 C1(CNC(=O)C=CCN2CCC2)CC(C)CO1.n1(CC=O)cnnc1.N C(=O)(C(O)CCCNC(=O)CC1COCC(C)O1)N1CC(NC(C)=O)C1 c1(CNC(C2N(C(C(C)n3cnnn3)=O)CCOC2)=O)ccc(=O)n(C)c1 N1(C(c2cc(CNC(CCC(=O)NC)=O)[nH]n2)=O)CC(N(C)OC)C1 c1(OCC#C)cccc(C(N2CCC(C(O)C(F)F)C2)C(=O)NCCCC)c1 c1(NC(C2CC(F)(F)CN2Cc2nccs2)=O)ccnc(O)c1[N+](=O)[O-] C(=O)(C(C)CC(C)(C)C)NC(CC)CNC(C1COCCN1C(C)=O)=O C1(CNC(=O)Cc2cc(F)cc(F)c2)CN(C(=O)CC2CSC2)C2COCC2O1 Cc1nc(CNC(=O)Cn2cnnc2O)oc1C(=O)NCCN1CCCC1 C(CN=c1[nH]c(=NC(C)C2CCC2)c2c(ncn2C)[nH]1)(c1cccc(F)c1)OC c1(OC)ccc2c(c1)CCC(C(=O)NCC(O)CCc1ccccc1)N2 c1(CCCC(=O)N(C)CC2CCCN2C(=O)CC(F)(F)F)ccc(F)c(F)c1 c1(CC(N2C(CCCNC(C3(C)C(C)(C)C3)=O)CCCC2)=O)cc(F)cc(Cl)c1 c1(C(N2CC(O)(CNC(C3CC(F)C3)=O)C2)=O)ccc2sncc2c1 C1(C(=O)OC)CC(NCc2ccc(NC(C)=O)nc2)CCO1 N1(C(CCn2c(C)nc(C)n2)=O)CCC2CC1CN2C(=O)CC1(O)CCOCC1 c1(OC)ccc(C(=O)NCC(=O)NCC(=O)NC(C)CC(C)O)o1 CCC(C(=O)NCCN(CC(=O)Nc1cc(C)no1)CC)c1ccccc1 C1(C(=O)NCCC2N(C(C(=O)NCC)=O)CCOC2)CCc2nc(C)nn2C1 C1(C(N2CC(C)(CC=C)C2)=O)CN(C(=O)C(O)CC(F)(F)F)CC12CCC2 c1(CC(=O)NC(CNC(c2csnc2Cl)=O)C2CCC2)nc([N+](=O)[O-])n[nH]1 CCC(CCCC(=O)N1CCN(C(C)=O)CC1)NC(=O)C(O)CC(C)C Cc1coc(C2CC2)c1C(=O)NCC1CN(C(=O)C#CC2CC2)C2CC12 C12CC1CN(C(=O)C(c1ccncc1)C1CCCC1)C2.C1(C(=O)N)(SC)CCC1 c1(C(N2CC3(OCC(NC(C(C(C)C)CO)=O)C3)C2)=O)ccc2c(c1)COCC2 C(=O)(CC(F)(F)Cl)N(CC)CC1CCCN1C(=O)CCCC1CCCO1 c1(C(N2CC(C)(NC(=O)CN3CCCC3CO)C2)=O)cnc(S)nc1 c1(CC(C)NC(c2c(C(=O)N(C)C)cc(F)cc2F)C)cc(F)c(F)cc1F CCCCC(C(=O)NCCN(C(=O)CCC1CCOC1)CCOCCO)C(C)C Cc1cc(CN(C(=O)C(C2CCCCCCC2)O)C)cc(F)c1 C1(C(=O)NCCCOC2CC2)COCCN1C(C1(n2cccn2)CC1)=O C=CC(C)CCN=c1nc(-c2ccc(C(=O)N(CC)CC)cc2)cc(C)[nH]1 n1(CC=O)ccc(O)nc1=O.C1CC2CCC(C1)O2.C1CC(O)CN1C(=O)C1CC1 c1(C=O)cc2ncccc2[nH]1.c1(OC)cc(C(=O)NCC2CC2C)n(C)n1 N1(C(c2nc(C(C)C)oc2)=O)CCC(C(F)F)(C)C1.c1(C(=O)N)ncc[nH]c1=O C1(C(=O)Nc2ccc(CO)o2)(NC(C(N2CCOCC2)C)=O)CCN(C)C1 C1(NC(c2cnc(OC)nc2)=O)CCCN(C(C2(C)CC2(F)F)=O)CC1 c1(CN2CCC(C(=O)OC)C2)c(OC)cncc1OC N1(C(c2cnn(CCC)c2C)=O)CCN(C(=O)CC2CCCCC2C)C(C)C1 Cc1cn2cc(C(N3CC=C(C)CC3)=O)nc2s1.[SH](=O)(=O)C1CC1.C(=O)(C)N O=C(CCC(F)(F)CCO)N(CCCO)Cc1ccc(Cn2ccnn2)o1 CC1C(NC(C2(C)CCC2)=O)CC2CCC1N2C(=O)CC1CCCC2(CCC2)O1 c1(NC(c2c(-c3nc(CC)on3)nccc2)=O)ccc(F)cc1S(C)(=O)=O C=CCCCC(C(=O)NCC1CCOCC1(C)C)NC(=O)CCCCCOC C(CN=c1[nH]c2c(c(=NCC3CCSC3)[nH]1)SCC2)NC(COC)=O C1(C(NOCC(C)(C)O)=O)CC=CCC1NC(=O)C1=C(Cl)CC1 [SH](=O)(=O)CCN(CC(CC1CCC1)CO)C=O.CC(C)(C)C=O.CCO.O n1(CCC(=O)NC2CCCC(C(C)C)C2)cc(C2(O)CCc3ccccc32)nn1 N1(C(CC2N(C(CCc3n(C)cnc3)=O)CC(O)C2)=O)CCCC2(CCOC2)C1 N1(C(C23CC(C)(OCC2)C3)=O)CC(CNC(C2C3CCCC23)=O)CC12CCC2 C1(NC(C(CC#C)(C)C)=O)CCCCCN(C(c2cc(C(C)C)cnc2O)=O)C1 C(=O)(CCC(F)(F)C(F)F)NCCC(C)NC(CCCCCOCC)=O CC12CC(NC(C3CC3F)=O)(C1)C1(CCN(C(c3ncc(F)cc3F)=O)CC1)O2 C(C)(CCC(=O)N1CCOCC1C1CC1)NC(C1(CC)COC1)=O N1(C(Cn2c(C)cc(C)n2)=O)CC(CNC(c2coc(N(C)C)n2)=O)CCC1C C=CCC(CC=C)C(=O)NC1CCN(C(c2ccc(F)c(CC)c2)=O)CC1CO N1(C(C=CC(C)(C)SC)=O)CCCC(CCCCNC(C2CC3CC3C2)=O)C1 N1(C(c2ccc(CC)cc2N)=O)CCCC2CN(C(=O)CNS(N)(=O)=O)CC12 CC1OC2CCC1(C(N1CC(C)C(F)(F)C1)=O)C2.C(=O)(CC(C)(C)C1CC1)N C1(NC(c2scc(C)c2C)=O)CCCCCN(C(c2cnc(O)o2)=O)C1 Cc1cccc(C(=O)N(CCCNC(=O)CC2(C)CC2(F)F)C)c1O c1(C(=O)NCC2(F)CCC(NC(=O)CCC(F)F)C2)cnc2ccc(F)cn12 C1(NC(C2(CN(C)C)CCC2)=O)CCCN(CC(=O)OC(C)(C)C)C1 C(=O)(CS(=O)C(F)(F)F)N1CCC(O)(CNC(c2c(C)nc(N)cn2)=O)C1 C1(CNC(COC(C)C)=O)CC(C)N(c2ncns2)C1 C1(NC(c2c(C#N)csc2)=O)CN(C(=O)CC23CCC(CC2)CC3)CC12CC2 C1(C(N2C(C=CC(=O)NCCC(F)=C(F)F)CCC2)=O)CCCC2(CC2)C1 c1(C(=O)OCC)cnc(C(=O)N(C)CCN2CC=CC(OC)C2)cn1 Cc1[nH]nc(C(=O)NCCC(C)NC(C2CCCOC2)=O)c1Br C1(NC(C=C(C)C(F)F)=O)C(C(=O)NCCCCNC(N)=O)C1(C)C c1(OC)cccc(NC(=O)CC2CCCCC2)c1O.c1(C(=O)N)cc(C)n(C)n1 C1(NC(c2c(C)csn2)=O)CCCC1(C)CN(C)C(C1C=CCS1)=O N1(C(C(C)=CC=C)=O)CC2CC(C(=O)Nc3cnccc3C)C(C2)C1 N1(C(=O)NC(C)CCn2cncn2)CCC2(CNC(=O)OC2)C1 c1(NC2CC(NC(c3cc(C4CC4)on3)=O)C23CCC3)ncc([N+](=O)[O-])cc1Br C(N=c1nc(C)c([N+](=O)[O-])c[nH]1)C1OCCN(C(c2c(C)cc(=O)oc2C)=O)C1 CC1(CC(=O)NCCC2CCN(C(C3CC=CCC3)=O)C2)CCOC1 N1(C(c2c(C)ncs2)=O)CC2C=CC1C2.C12(CCC1)N(C)C2=O C1(CC(=O)N(C(C)C(=O)N(C)CCC2CCCN2C)CCC)CSCCO1 CC(C)CC(F)C(=O)NCC1CC(F)(CNC(=O)CC2CC=CCC2)C1 O(N1CCC(CC(=O)NCCNC(=O)C(Cc2ccccc2)C2CC2)CC1)CC C(=O)(CCCC(=O)NC1CCC1)OCC.c1(C(=O)N)cnc(C(C)(F)F)s1 c1(C(=O)N)cc(C(F)(F)F)cc(O)c1.c1(OC)cc(CCC(=O)NCC)on1 Cc1ccc2c(c1)CCC(C(=O)NCc1ccc3c(c1)CN(C(=O)N(C)C)C3)O2 C(=O)(C#CC1CCOC1)N1CCC(CN(C(=O)C(CO)C(F)(F)F)C)C1 C(C(C)(O)CC(=O)N1CC2C(CC(=O)NCC(O)C(C)O)C2C1)OC Cc1cc(=O)n2nc(N3CCC(O)(C(N4CCCCC(C)C4)=O)CC3)nc2[nH]1 C(=O)C1=NOC(C)C1C.c1(OCC(=O)OC)ccc(C=O)cc1.C1CCC1.N c1(OC)cccc2c1OC(C(=O)NC1CCC(O)CN(C(=O)C3=CCCS3)C1)C2 c1(CC)nc(=N)[nH]cc1C(N1CCC(C)C1C)=O.c1(CCC=O)ccncn1.N N1(C(C(N(C(COCC(=O)OC)=O)C)C2CC2)=O)CC(C)C12CCOCC2 CN1CC(C)(C)CC1NC(N1CCC(Oc2cc(O)nc(=N)[nH]2)C1)=O C1(O)(CNC(COC(C)=O)=O)CN(S(=O)(=O)CCc2ccccc2)C1 N1(C(C(C)=C2CCC2)=O)CCN(C2CCC(NC(c3ncccc3O)=O)C2)CC1 CS(=O)(=O)C1(CO)CC(NC(=O)NCc2ccc(-n3cncn3)cc2)C1 c1(NC23C(NC(=O)CCCC4CC4)CC(CC2)C3)ccc2nnnn2n1 c1(C(=O)NCC2OCCC2C(=O)NCC2CCC2CO)cc(Cl)cs1 Cn1cccc1CCNc1ccn(Cc2ccccc2)n1.c1(C)nnnn1C C(=O)(C1=CCCC(C)(C)C1)NC(C1(O)CN(C(CC(COC)(C)O)=O)C1)C c1(C(N2CCC(CNC(C(C)SC)=O)CC2)=O)c[nH]c2nc(Br)ccc12 Cc1ccc(C(=O)NC2CCCC(C(=O)NCCP(C)(C)=O)C2)c(C)n1 Cc1cc(C(N2CC(O)(CNC(=O)C(O)C3CCCC3)C2)=O)cc(N)c1O C(=O)(C1CCc2ccccc21)NC(CC)(CNC(=O)CC(C1CC1)C1CC1)CC CCCCCCC(C)(CC)C(=O)NOCC1CCN(C)CC1 n1(C(C)C)cc(NC(C2(C(F)(F)F)CCOC2)=O)cn1 C(=O)(C1=CC2(CN(C(=O)CC3C=NN(C)C3=O)C2)OC1)NC(CC#C)C=O.O N1(C(C(COC)O)=O)CCC2(NC(C3CC34CC(O)C4)=O)CCCC12 C1(N(C(C(CC)OC2CCCCC2)=O)CC)CCCN(CC2CCCCC2)CC1 c1(N(CCNC(C)=O)C)nc(=NCC(C)SC(F)F)[nH]c2c1COCC2 c1(C=O)ccc(O)c(C(C)(C)C)c1.CNS(=O)(=O)NCC(N1CCCC1)=O.C c1(C(=O)NCC(CNC(COCCCC#C)=O)F)ncc(COC)s1 CC1CN(C(c2cncn2C)=O)CC(C)N(C(C2CCC2C#N)=O)C1 C(=O)(C#CC1(CC)COC1)NC(C=CC(=O)NCC1CCN(CC)C1)C N1(CCCNC(C2CCN(Cc3c(C)ccs3)C2)=O)C(=O)C=CC1=O c1(C(N2CC(NC(Cc3nc(C)sc3)=O)(CO)C2)=O)cncc(C)c1C c1(C(N(CC(C)N(C(CSCC#C)=O)C)C)=O)cc(Br)c(C)o1 c1(SC)nc(NC23CC(C(=O)NCC4CCCCNC4)(C2)C3)cc(O)n1 C1(CNC(c2cc(C)c(C)o2)=O)CCCCC1N=c1nc(C#N)[nH]cc1C C1(C2(O)CCOCC2)(C(=O)NC2C(CC)CN(C(=O)Cc3cc[nH]n3)CC2)CC1 N1(CC(=O)OCCOC)CCN(C(=O)CCO)CC1.c1ccc(F)cc1.CC N1(C(C2C3CN(C(c4nc(CC)sc4)=O)CC32)=O)CC2CCN(C)CC2C1 N1(C(c2cc(OC)ncn2)=O)CCC(C2CC2)(CNC(c2cnccn2)=O)C1 C1(F)(C(N2CCC(C)(C(=O)OCC)C2)=O)CCCN(C(=O)C#CC(=O)O)C1 n1(CC(N2CC(CNC(C3C(=C)C3)=O)OCCC2)=O)cc(P(C)(C)=O)cn1 CC1(C)CN(C(=O)C=C2CN3CCC2CC3)CC1NC(=O)CC1CCC1 C(=O)(CC(F)(F)C(C)C)N1CCN(C(CCCc2ccc(C)c(C)c2)=O)CC1C c1(C(N2CC(C)(CC(=O)NCC(F)F)C2)=O)cnc(O)c(Cl)c1 C1(NC(CCCN(C(=O)OCC)C)=O)CN(C(C2(C(F)F)CC2)=O)CC1O N1(C(C(CCCCC)O)=O)CCC2(C=C(C(=O)Nc3cc(CC)cc(F)c3)C2)C1 CC1(c2nc(C(F)F)no2)OCCO1.C1CCCCc2noc(n2)C2CCC1C2 C1(NC(CCC(C)C)=O)CN(C(C2CC23CCC3)=O)CCC1C(F)(F)F C1(NC(C(C)C)=O)CC2CCC(C1)N2C(c1ccc(C(F)F)cc1F)=O C1(NC(c2c(C)noc2)=O)COCCN(C(=O)C(n2ccc(C3CC3)n2)C)C1 c1(C(=O)NC2C(NC(c3[nH]cc(C)c3)=O)CCCC2)cnc(O)c2ccsc12 c1(CN(c2cc(N)ccn2)C)nc(CO)nn1-c1ccc(Br)nc1 C1(NC(CC2(OC)CCC2)=O)CCC(C)(CNC(=O)C2=C(C)CC2)C1 C(=O)(C1=CC(C)(C)C1)N(C1CCCN(C(C2CCN(C3CCSC3)CC2)=O)C1)C c1(C(N2C(CCNC(CCN(C)CC)=O)CC(F)(F)C2)=O)cccc2sncc12 C1(NC(c2ccn(CC)n2)=O)CCC(O)CN(C(=O)C=Cc2cccc(Cl)c2)C1 N1(C(c2c(N=[N+]=[N-])cccc2)=O)CCCC(C2(NC(c3csc(O)n3)=O)CC2)C1 Cc1ccc(CNC(C2CCCC2NC(c2ccn(C)c2)=O)=O)c(O)c1 N1(C(c2c(C)nc(C3CC3)o2)=O)CC2CC1CN(C(c1ccc(C#N)cn1)=O)C2 C(CCC(O)C(=O)NCC=CBr)NC(=O)Cc1cccnc1 Cc1nonc1CNC(=O)C(C1CCCC1)NC(=O)C=CC1CCOC1 c1(COCC(N2CCCC2Cc2ccc(Cl)cc2)=O)ccc(Cl)cc1 N1(C(C2CC(CC)C2)=O)CCC2CN(C(C3(CC4CC4)CC3)=O)CCC12 c1(C(N2CC3CN(C(C(CCCC)(C)F)=O)CC3C2)=O)ccc2c(c1)B(O)OC2 C1(NC(C2CCN(C)C2=O)=O)CCC2(CCN(C(C3CC34CCCC4)=O)CC2)C1 N1(C(CC(COC)NC(=O)CNC(N)=O)=O)CC(C)(C)OC(C)(C)C1 c1(C(C(=O)NC2CCOC2)N(C)CC2CCCSC2)ccncc1Br C1(C)(C(=O)NCCCC(C)NC(c2coc(-c3ccccn3)n2)=O)CC(C#N)C1 c1(N(C)Cc2c(C)ccs2)ccc(S(=O)(=O)N2CCC(O)C2C)c(Br)c1 Cc1ccc(Cl)cc1S(=O)(=O)NC(=O)CC1COC1.N(C)C C=C(C)CC(C(=O)NCC1CC2(C1)CN(C(=O)C(C)c1ccsc1)C2)OC N1(C(c2nnc(C(C)C)s2)=O)CC23CCCC2(C1)CN(C(=O)C=CI)C3 CCC(O)C(C)(C)C(=O)NCC1CC2(CO1)CN(Cc1c[nH]nc1)C2.CC.O C1(N(C(=O)CC=CCC)CC#C)CCN(C(c2sccc2SC(F)F)=O)C1 Cc1c(C(N2CC(N(C(=O)C(c3ccccc3Cl)C)C)C2)=O)cnc2nncn12 CC(CC(=O)N1CC2(C1)CN(C(C1(C)CCCO1)=O)C2)C(F)(F)F c1(C(=O)NC2CCC(NC(=O)C3=CCC3)CC2)cc(F)c(Br)c(F)c1 N1(C(CC2N(C(CC(OCC)OCC)=O)CCC2)=O)CCc2nocc2C1 C(C(C)(O)CC(=O)N1CCN(C(c2ccccc2C2CC2)=O)CC1CO)OC c1(OC)cc2c(cc1C(=O)NC1(C)CCCCC1)CCC2.c1(C=O)ccsn1.N N1(C(c2ccnc(C)c2)C(=O)NCCCSCC)CCc2cccc(Br)c2C1 N1(c2nc(CC)nc(Cl)c2CC)CC2(CCN(C(C3CCCN3CC)=O)CC2)C1 C1(C=O)CC2CCC(C1)C2.c1(CC)nn(C)cc1C(=O)NCCC1CC1.N c1(C(C(N2CCC(O)(C(C)C)C2)=O)(C)C)c(F)cccc1F.C(=O)CC1CC1.N CC1(C)CCN(C(=O)C(F)C(F)(F)F)CC1NC(C1CCCN1C1CCCC1)=O Cc1cc(Cn2nccn2)ccc1NC(=O)CC1CCCN1C=O.C(C)(C)C C1(NC(=O)C2=CCOC2)CN(C(C2(n3cccn3)CCOCC2)=O)CC1C1CC1 N1(C(C(C)C(F)F)=O)CC(NC(c2ccc(F)cc2Cl)=O)CC12CCCCC2 CC(C)C(C#N)C(=O)NC1CCC(CNC(c2cc[nH]n2)=O)C1 C1(C)(NC(C(C)OCC(F)(F)F)=O)CCN(C(=O)C(C)(C)c2cnsc2)CC1 N1(C(C(C)NC(c2ccoc2)=O)=O)CCC(N(C)C(C2CCCS2(=O)=O)=O)CC1 CC1CCCCC1OCCN(C(C)=O)C(C)C.C1(CC=O)COC(=O)N1 C(=O)(C1=CCC2CCC1N2C(=O)C(C)C=C=C)NC1(C#C)CC1 C1(C(N2CCC2)=O)C2CC(=O)CC12.C1(C(=O)OC)COC(C(=O)N)C1.C C(C(=O)N(C1(CC(=O)Nc2cnc(O)nc2)CC1)C)(C(C)C)OC C1(C(=O)NCC(=O)Nc2scc(CC(=O)OCC)n2)CCC2CC2CC1 O=C(C1=CCCN(C(C23CCC(CC2F)C3)=O)C1)NC1CC2CCCCC12 C(=O)(CC(C(F)F)NC(=O)C(O)CN(C)C)NCC(C(C)C)C c1(C(=O)NC2CCCCC2NC(C2CC(Cl)(Cl)C2)=O)ncnc2ccsc12 N1(C(c2cc(C(C)C)sn2)=O)CCN(C(C2COC(C)C2)=O)CC(C)C1 N1(C(=O)OC(C)(C)C)CCC2(CC1)CC2CNC(=O)C.c1ccccc1.N C1(C(=O)NCc2n(C)ncn2)CC2(CC2)CN1C(=O)CCC=O.c1nccs1.N C1(O)(CN(C(C(C)OCC=C)=O)C)CCN(C(c2cscc2CC)=O)C1 c1(NCC(=C)Br)[nH]c(=NCC(CO)C(C)CC)nc2c1ncn2C(C)C C1(NC(c2ccc(C(C)C)o2)=O)CCC12CN(C(=O)CCn1cnccc1=O)C2 Cc1cccc(C(N2CCCC(CCC(=O)NCC3CCC3C)C2)=O)n1 C(CCN(C)C)(C(=O)NC(c1nnnn1C)C)NC(C(CC)=CCCC)=O C1(C(N(C)Cc2c(C)ncs2)=O)C(C)CCN1C(=O)CCC(C)N(C)C N1(C(COCc2c(C)ncs2)=O)CC2(CNC(=O)C=C(Cl)Cl)CCC1C2 CCCCC(O)CC(=O)NC1CC=C(C(=O)N2CC(O)CC2(C)C)C1 N1(C(Cc2c(C)scc2)=O)CCC(C)(C)C(C(=O)NCC(C)(O)CC(C)C)C1 C1CCOC2(CCC2)C1.c1(CNC(C2(COC)CC2)=O)ncc(C=O)cn1 NC1COc2c(C(=O)Nc3cccc4nsnc34)cnn2C1 c1(CNC(=O)C(=O)NC2CCCCC2)c(F)cccc1F.C(=O)(C1=NOCC1)N Cc1cccc(Cl)c1C(=O)NC(CNC(c1ccc(F)c(N)c1)=O)CO c1(C(=O)NC2CC(C)CN(C(=O)Cc3ccccc3Br)C2)cccn2cncc12 C1(NC(=O)CCc2ccsc2)CCCCC1NC(C1CCCNC1=O)=O C1(C(=O)NC(C2CCN(C(c3nn[nH]c3Cl)=O)CC2)(C)C)CCC(F)(F)C1 C(c1ccccn1)=C(C)C(=O)N(C(CNC(=O)C(C)N(C)C)C1CC1)C CC(CS(C)=O)N=c1cc(NCCc2c(F)cccc2Br)nc(C(F)(F)F)[nH]1 C(=O)(C1=NOC(C)C1)N(CCC)CCNC(c1c(N(C)C)cnn1C)=O C(=O)(CCC(F)(F)F)NC(CCOCC)C(N1CCOCC(C)C1)=O C1(CC(=O)NC(C)CCN(C(=O)CC(=O)N(C)C)C)CCCC1(F)F CC(C)(C)C(C(=O)N1CCCC(CCC(=O)O)C1)n1cc(C2CCCO2)nn1 CS(=O)c1ccc(C(=O)NCC2CN(C(=O)CN3CCS(=O)CC3)CC2O)cc1 c1(C(N2CC(F)(CNC(C3(C=C)CC3)=O)C2)=O)nc(C)ccc1O S(=O)(=O)(CC(=O)NC1CN(C(C2CCOC2C2CC2)=O)CC1SC)NC C#CC1(C(=O)NC(C2CCCCC2)C)CCN(C(=O)C#CC2CCCC2)CC1 Cc1nnc2cc(N3CCC(CF)(NC(C4CC5C=CC4C5)=O)C3)ncn12 C1(CNC(C(C)=C2CC2)=O)CC(NC(=O)CNC=O)C12CCC2 C(C(CCC)C(=O)NCc1nc(C2CC2)n[nH]1)NC(CC=CCC)=O C1(CNC(C(=O)NC2CCC(C)(C)CC2)=O)CC2(C1)C(F)(F)C21CCC1 C(N=c1nc(C(F)F)[nH]s1)C1C(C)CN(C(=O)CCCN(C)C(N)=O)C1 c1(CC(=O)N(C(c2nccs2)C)C)c(F)cc(C#N)cc1Br C1(C)(C(=O)NCC2CC(COC)OC2)Cc2cc(OC)c(OC)cc2C1 Cc1cc(C)n2cnc(C(=O)NCCOCCCNC(=O)C(C)CO)c2n1 C(C)(CCCN=c1[nH]cc2ccnc-2[nH]1)NC(CCc1c(C)nc(S)nc1C)=O N1(C(c2c(C)nccc2)=O)CC2CCN(C(C3CC3(C)C)=O)C2C1 O=S(=O)(c1cc2cc(Cl)ccc2s1)NC12CCC(CC1)C2 N1(C(c2c(C)ccnc2)C(=O)NCC2CCC(F)(F)CC2)C2CCC1CN(C)C2 c1(C(N2CC(C(=O)NCC(CC(C)C)C)C(F)(F)C2)=O)cc2ccccc2o1 C1(NC(CCCC2C(C)C2)=O)C2CC3C1C3C2C(N1CC(CN=[N+]=[N-])C1)=O c1(CN2CCCC(C(N3CCc4sccc4C3)=O)C2)cc(Br)c2c(c1)OCO2 c1(C(N(CCC)CCNC(C2(F)CCOC2C)=O)=O)ccn(C(C)C)c1C C1(O)(CCNC(CCC2CCC(C)O2)=O)CCN(C(C2(C)COC2)=O)CC1 Cc1c(C(=O)NC2CCCCN(C(=O)C(C)C#N)C2)cnc2ccccc12 C1(C(=O)NC2C=CC(CC(=O)NCC3CCC(=O)O3)C2)CCCC(=O)C1 C1(CNC(c2ncc(Cl)cc2F)=O)(C)CC2CCCC2C1.C1(C=O)OCCO1.N Cc1cnc2c(C(=O)NCCC(C)CCNC(=O)C3=CCCC3)c(C)nn2c1 Cn1cncc1C(C)(C)C(=O)NCc1ccno1.C1(C=O)C(C)(C)C1(C)C C1(CCNC(c2c(C)n(C)nc2)c2nnnn2CCCF)CC2(CCC2)CO1 Cc1cc(C(N2CCC(NC(C3CCCCN3C(=O)C3=CCC3)=O)C2)=O)[nH]c1C C1(O)(CN(C)C(c2ns[nH]c2=O)=O)CCN(C(C2CC3C=CC2O3)=O)C1 CCCCCCC(C)CC(=O)NC1CN(C(c2[nH]ccc2COC)=O)CC1C1CC1 C(C(C)(C)CC(C)O)NC(C(c1cnn(C)c1)NC(CCc1onc(C)n1)=O)=O CN1CC(O)CCC1C(=O)NCC1CCN(C(c2cn[nH]c2)=O)C12CC2 C(c1cccc2cccnc12)=CC(=O)NC1C(NC(C2ON=C(CC)C2)=O)CC1 C1(CNC(C(C)c2ccsn2)=O)CCCCN1C(=O)C(C(C)O)N(C)C C1(C(=O)NCCC(C)N2CCC2)CC(N=[N+]=[N-])CN1C(c1ns[nH]c1=O)=O C1(OC)CC(NC(=O)CCSc2ccc(C#N)cc2)CN(C(C2CCCC2)=O)C1 C1CN(C(C2(CCN(C)C)CC2)=O)CC(C)(C)O1.CC1=NOC(CC(=O)N)C1 c1(C(N2CC(Cn3cc(C4CCCN(C)C4)nn3)C2)=O)nccc2ncncc12 c1(C(N2CCC(COC)C2)=O)c(C)cc(C)oc1=O.C1(C=O)CC(C)OC1C.N c1(C(=O)NC(C)CCNC(C23CC(CO2)C3)=O)ccnc(O)c1Br C1(CC(N2C(C)C(NC(c3cscc3C(F)F)=O)CC2)=O)CCCC2(CCC2)O1 C1(OCCC(=O)NC2CC(N(C(=O)C=CC3CCC3)C)C2)CCCOC1 C1(NC(c2cc(SC)oc2)=O)CC2CCC(C1C)N2C(c1ccc(Cl)cc1O)=O n1(C(C)(C)C)cc(Cl)c(C(=O)NCC2(O)CN(C(c3sccc3F)=O)C2)n1 N1(C(C2CCC(F)(F)C2)=O)CCC2C(CCN2Cc2c(Cl)cc(O)cc2Cl)C1 C(F)(F)(C(F)(F)c1ccc(CNC2CCCCC2c2ccccc2)cc1)OC CC1CC(N(C)C(C2CSCN2C(=O)CCc2cncs2)=O)CC(C)C1 c1(C(N2C(CNC(Cc3c(C)n(C)nc3)=O)CC2)=O)ccnc2ccc(O)cc12 N1(C(CC(=C=C)C)=O)CC2(C1)CN(C(=O)C(C)P(C)(C)=O)CC2CO c1(C(N2CCC3C(C(N(C4CCC(O)CC4)C)=O)C3C2)=O)cc2ncccc2[nH]1 CC(C)(CCCO)C(=O)NCC1CCCCN(C(C2CC3CCC2O3)=O)C1 c1(C(N2CC(O)(C(C)NC(CN3C(C)CC3)=O)C2)=O)ccc2c(c1)COCO2 C1(CNC(C(C(C)C)C)=O)CC2(CCN(C(=O)CC3(C)CC3(Cl)Cl)C2)CO1 N1(C(c2ccc(OC)c(C)n2)C(=O)NCC2CCCO2)CC2CCC1C(O)C2 Cc1sc(C(N2CC(NC(=O)CNC=O)CC23CCOC3)=O)cc1S(N)(=O)=O C1(CNC(c2ccno2)=O)CCCC1NC(c1cc(C2CC2)on1)=O Cc1nc(NCc2cc3n(n2)CCCO3)cc(=NC(C)CC2CCC2)[nH]1 N1(C(c2cnc(OC)s2)=O)CCC(O)(C(N2CCC(C(C)(C)O)CC2)=O)C1 CC1CN(C(c2cc(CNC(=O)C(CO)C(C)(C)C)[nH]n2)=O)CC(C)N1C c1(C(N2CC(NC(C3CCCC(C)C3)=O)C(O)C2)=O)cc(Br)cc(Br)c1 N1(C(c2nc(C(C)C)oc2)=O)CCOCC1CC(=O)N(C1CN(C)CC1O)C c1(C(C)C)nn(C2CC2)cc1CCCO.C1(N(C(CCNC)=O)C)CC(F)(F)C1 C1(CC)CN(C(c2cn3ccnc3s2)=O)CCC1NC(c1ncncc1F)=O N1(C(C(=O)NCc2cc3cscc3s2)=O)CCCC2CCNC(=O)C12 C=C(C)CCC(=O)N(CC(C)NC(=O)C(c1ccccc1F)C)CC Cn1cccc(C(N2CCC3(NC(=O)Cc4cnns4)CC3C2)=O)c1=O CC(C)C(C(=O)NCC12CC(CO1)C2)N1CCCC1=O.C(=O)C=C1CC1 C12(CNC(c3cccc(OCC)c3)c3nnnn3C)CC(C1)NC(=O)O2 N1(C(C(Cc2c(C)cccc2)C)=O)CCCN(CCCCNC(=O)C2CC2)CC1 Cn1nc(C(=O)NC(C2CCCC2)CNC(C2(Cl)CC2(C)C)=O)c(Br)n1 C(=O)(CCC(F)(F)F)N1CCCC(C(C(=O)NC2CC(OC)C2)C)C1 C12(C(N(CC(C)N(C)C(c3ccncc3)=O)C)=O)CCC(CO1)C2.N(C)(C)C C(=O)(C#CC1CCCO1)N.N1(C(CCNC(=O)OC(C)(C)C)=O)CCCC1C C(C(C)CC(C)C)NC(c1c(OC)noc1C)=O.C12(C=O)CC3CC1C2C3.N C1(NC(=O)CC2CC=CC2)CCCC12CN(C(C1Cc3cccnc3C1)=O)C2 c1(CC2CN(C(c3cn(C)nc3C(F)(F)F)=O)C2)ccc(S(C)=O)cc1 Cc1nn(C)cc1C.n1(N(CCCCO)C)cnnc1CC(C)C Cc1nc(-c2csc(CN(C)C)n2)cs1.c12ccc(s1)C1CCCN1C(=O)C2 c1(C(N(CCC(C)NC(C(CC=C)C)=O)C)=O)cc(F)c2nc(C)cn2c1 Cc1c(N(C(=O)CCCNC(C2CCN(C(C)C)C2)=O)C)cccc1F CCCC(C)(C)CC(=O)N1CC(NC(c2ccc(C)c(F)c2)=O)C(C)C1 c1(OC)ccncc1C(N1CC(O)CC1C)=O.c1(C2C(C(=O)N)C2)cnc[nH]1 C1(NCc2ccc(OCCC)cc2)CCN(c2ncc(Br)c(C)n2)CC1O C(=O)(CC(C)C(C)(C)NC(c1cscc1OC)=O)NCc1cccc(C#C)c1 N1(C(C(C2CCCC2)NC(C2N(C)CCC2)=O)=O)CCC2(CCOC2)CC1 C1(NC(=O)C2CC2)CC2(C1)CC2NC(=O)Cc1cscc1F C1(C(=O)N(CCO)CCOCCO)C2Cc3ccc(Br)cc3C12 c1(OC)ccc(CN2CCC(C(=O)Nc3ccn4cnnc4c3)C2)c(Cl)c1OC N1(C(C(C)C2CCCC2)=O)CC(F)(F)CC1C(=O)NCCc1ocnc1CO C1(NC(c2c(C)cccn2)=O)COCCN(C(C23COC(CF)(C2)C3)=O)C1 C1(C(N2CC(NC(Cc3ccc(C(C)C)cc3)=O)C(O)C2)=O)COCC(C)(C)O1 N1(C(=O)NCc2c(OCCCOCC)cccc2)CCC2(CCCC2)CC1 C1(CCC(=O)Nc2cn(CC#C)nc2)CCCN(C(=O)CN(C)C)C1 C(C(=O)NCCCN(C)C(C1CCCC1(C)C)=O)(C(C)C)NC(=O)OC CCCC(CC(C)C)C(=O)NCC1(NC(c2cc[nH]c(=N)c2)=O)CCOC1 N1(C(C2CC(C)(O)C2)=O)CCOCC(CNC(=O)CC(F)F)C1 C(=O)(CS(=O)(=O)CC(F)(F)F)N1CC2CCN(C(C(C)O)=O)C2CC1 C1(C(=O)NCC23OCC(CNC(CCCCC)=O)(C2)C3)CCCC12CCOCC2 c1(C(N(CC(=O)NCCOCCCO)CC)=O)cnn(C)n1 C1(NC(C2CCN(CC(C)C)CC2)=O)CC2CC(NC(=O)C3=CCCCC3)C1C2 C1(CNC(c2n(CC)ccn2)=O)CN(c2nc(C3CCCC3)ns2)CCC1(C)C C12(NC(c3c(C#N)cccc3)=O)CCC(C(=O)N)(CC1)CC2.N1(CC)CCOCC1 c1(OC)ccc([N+](=O)[O-])c(CN2CCC(O)C2)c1.C(=O)C(C)(O)C(F)(F)F.N c1(C(=O)NC(CSC)(C)C(=O)NC(c2cccnc2F)C)cc(C#N)oc1C C1(CN(CC(c2ccc(F)cc2)=O)CC(=O)OC)CC2CCC1CC2.CO N1(C(C(COCC)C)=O)CCN2CCOCC2(CNC(=O)CCn2cccn2)C1 c1(C(=O)OC)cc(Br)cc2c1ccn2CC(N1CC2(C1)CN(C)C(=O)C2(F)F)=O C1(C(N2CC(C)N(C(=O)COCc3nc[nH]n3)CC2)=O)CC2CC(O)C(C1)C2 c1(C(=O)NCC2(NC(Cc3nc(=N)[nH][nH]3)=O)CCC2)cnc2n1CCC2 C(C1CCCC1)=CC(=O)NC1CC(N(C)C(c2ccco2)=O)C1 CC(CC(F)(F)F)C(=O)NCC1CCCN1C(=O)C.c1ccc(C(N)=O)cn1 C=CCCC(CO)NC(=O)C(CO)NC(=O)CC1CCCN1C C(c1ccccc1Cl)=C(C)C(N1CCN(C(C2COCCOC2)=O)C2CC12)=O c1nc(=N)[nH]cc1C(=O)N(C(C)C)C.c1(C=O)cncn1C(F)(F)F.CO CC1(C)CC(C(=O)NC2CCN(C(c3coc(C(F)F)c3)=O)C2(C)C)CCO1 C=CC(O)C(=O)N(CCCNC(C1(Cl)CC1(F)F)=O)CC CC(C)CCCC(C)C(=O)NC1CCC12CN(C(=O)COCC1CCOCC1)C2 Cc1csc(C(=O)N(CCCCCNC(=O)CSCc2cscn2)C)c1C c1(N2CCC(CC(C)C)C2)nc(NC2CCc3ccccc32)c2ncsc2n1 Cc1nc2c(s1)C(NC(C1CSCN1C)=O)CCC2 CC(O)(CC(=O)N1CC2(CCN2C(=O)CC2(CO)CC2)C1)C(F)(F)F n1(CC)cc(Cl)c(C(N2CCCC(CN(C(=O)CC3CCCC3)C)C2)=O)n1 C(=O)(CC(C)CC(=O)N1CC(C(N)=O)C1)OC.n1(C2(C=O)CC2)cccn1.C c1(N2CC(CC)OC(C)C2)nc(=NCCCC(N)=O)[nH]c2c1CCCCCC2 Cc1cc(Br)ccc1CC(=O)NC1CN(C(C2(C(C)C)CC2)=O)CC1O C1(CNC(C2C(C=C)C2)=O)CC(NC(c2cn(CCF)nn2)=O)CCO1 c1(C(N2CCC(N(C(CC(C)n3cccn3)=O)C)C2)=O)ccnc2[nH]cnc12 c1(C(=O)NC2C(C)CN(C(c3[nH]ncc3C#N)=O)C2)cc2ccccc2n1C Cn1nc([N+](=O)[O-])c(Cl)c1C(=O)N.N1(C(CC2CCC2)=O)CCC(N(C)C)CC1 C1(CNC(C(CC)SC)=O)CC2CCC(C1)N2C(C1(C)CCC(=O)N1)=O c1ccc(C2(C=O)CC2)cc1.C1(OC)C(NC=O)CC1O.C(C)(C)C.CC C(=O)(C(C)(C)C(N)=O)N(CCCCCCNC(c1cnnn1C)=O)C N1(C(C(C)=CC2CC2)=O)CCC2CCN(C(c3ncc(Br)cc3O)=O)CC12 C1(C)(CNCC(C=C(C)C)(O)CO)CCCCCCC1 c1(C(CNC(=O)C=Cc2cn[nH]c2)NC(c2csnn2)=O)cccc(Cl)c1 CCCCCCC(C)CC(=O)NC(C)CCCNC(=O)Cc1cc(F)ccc1O c1(C(=O)NCC23N(C(C(C(CC)C)OC)=O)CC(C2)C3)onc2c1CCCC2 N1(C(CS(CC)(=O)=O)=O)CCOC2(C1)CN(C(c1onc(OC)c1Br)=O)C2 C#CCCCCC(=O)N1CCN(C(=O)CSc2nncn2CC2CC2)CC1CO c1(C(N2CC3CN(C(C)C)CC3C2)C(=O)NC2CC2)ccc2c(c1)oc(=O)n2C C1(C(=O)NC(C)C(=O)N(c2cccnc2)Cc2cccs2)CC2CCC(C1)N2 [N-]=[N+]=NC1CCC(C(N2CC(=O)CC2C(=O)NCC2CC3(CC3)C2)=O)C1 O=CCCC(=O)N1CCCC(N(C(=O)CSCC(F)F)CC2CCCO2)C1.C Cc1cn2nc(N(C)CC3CCCN(C(=O)CC4CC4C)C3)sc2n1 Brc1cccc2c1CCCC2NC1CC12CCNC2 c1(C(=O)NCC2CN(CCn3cncn3)CCCO2)ccc2cc[nH]c2c1 C(=O)(C1CCCc2scnc21)NCCCN(C)C(c1cccn2nnnc12)=O Cn1cc(CCNC(C2CCCC2NC(c2ccn(CCF)n2)=O)=O)cn1 c1(OC)cncc(CCC(=O)NCC(CNC(=O)C(=O)N(C)C)CO)c1 N1(C(C(CC#C)(C)CC)=O)CCN(C(c2cc(N)ccc2F)=O)CC(C)(C)C1 c1(C(N(C2CN(C(C3(C(C)C)CC3)=O)CC2F)C)=O)ccc2nc(S)[nH]c2c1 c1(Cc2nnnn2C2CCCC2)nc(C(F)(F)F)c(Br)s1.Fc1cscc1CN c1(CN(C(c2ncc(C)[nH]2)C)C)cc(F)cc(C#N)c1 CN1CCCC(F)(C(=O)NCCOC2CCN(C(c3c(Cl)cnn3C)=O)C2)C1 C1(NC(=O)NC2COCC2N2CCOCC2)CCCCC1C(F)F N1(C(c2c(C)c[nH]c2)=O)CCC2(CC2C(N2CC(S(C)(=N)=O)C2)=O)C1 c1(C(c2nnnn2CCCS)NCc2n(CC)nnn2)ccncc1C1CC1 c1(C(=O)NC2CCC(CF)CC2)nc2ccccc2[nH]1 CC(C)C(C)(O)C(=O)N1CC(C)(NC(=O)C(O)P(C)(C)=O)C1 c1(OC)ccc(F)cc1C(N1CCN(CCc2ccnn2C)CC1)=O N1(C(c2ccc(CC)cn2)=O)CC2CCN(C(=O)C3=CCC(C)CC3)C2C1 N1(C(C2CCN(C)C2)=O)CC(C(=O)NCC2CCCN(C)C2=O)C2(CCC2)C1 c1(C(N2C(C3(C(=O)N)CC3)CCC2)=O)csc(C#N)c1.C1(CCC)CC1C C1(CNC(c2cccc(C(C)=O)c2)=O)CCC(C)N(C(c2cnnc(C)c2)=O)C1 c1(N(C(C)CNC(=O)CCCC2CCCCC2)C)ncncc1C#N C(C(C)CC(=O)N(C1CCSCC1)C)NC(Cc1ccc(C)s1)=O c1(CC(C(=O)O)NC(CCC)C)cccc(Br)c1 c1(CN(CC=C)C)cccc(NC(=O)NC(C23CC(CC)(CO2)C3)C)c1 C1(C(C)C)CCc2ccccc2C1NC(C1(C)CCOC1)=O C(=O)(C1=CCCN(C(=O)CN2CCOCC2)C1)NC1(C)CCOC1 N1(C(C2CC(C)(C(C)(C)C)C2)=O)CC2CC1CN2C(=O)CC12CCCC1C2 C1(NC(CC2C(C)(C)C(O)C2)=O)CCC2(CC1)CN(C(C1CC1(C)Br)=O)CCO2 C1(CNC(C(C)CN(C)C)=O)CCCN(C(c2ccccc2C2CCC2)=O)CC1 Cc1nc2cccc(C(=O)NCC3CCCN3C(C3C4CCCC34)=O)c2[nH]1 C1(C(=O)Nc2c(C)noc2)CC12CCN(Cc1nccn1C)C2 N1(CCC(=O)N(C2CC(NC(C3(C)CC3)=O)C2)C)CCOC1=O.C1CCC1 N1(C(c2c(CNC(C(CC)n3ccnc3)=O)noc2)=O)CCCCC(C)(F)C1 C1(N(C(=O)C2=CCC2)CC)CCCN(C(c2c[nH]c(C(N)=O)c2)=O)CC1 N1(C(c2cccc(OCCCC#N)c2)C(=O)NC(C)(C)C)CC2C(C1)C2(F)F Cc1cc(Cl)c(C(N2CC(F)CC2CNC(C2(O)CCCC2)=O)=O)cc1C CN1CCCC(CCNC(=O)C(C2(O)CN(C(C3(C)CC(=O)C3)=O)C2)F)C1 C1(C(=O)NCCC(C)(C)CSN)CC2(C1)CC(CN)C2 c1(OC)cc(C)c(C(c2nnnn2CCCSC)NCCc2ccc(I)s2)cn1 N1(C(c2c(C)cncc2)=O)CCC2C(CCCN2C(C2(C)CC2(Cl)Cl)=O)C1 C(C(C)(C(C)C)C(C)C)NC(C1CC(CNC(C=C(CC)C)=O)C1)=O C1(NC(CC(CC)O)=O)CN(C(C2CCC(=O)C(C)C2)=O)Cc2nccn2C1 N1(C(CCC=C(C)C)=O)CCN(C(c2cc3ccsc3n2C)=O)CC(O)C1 c1(C(N2CCN(C(C3CCN(CC)C3)=O)C(C(F)F)C2)=O)nc2cnccc2s1 c1(C(C)(C)C)cc(N2CCC(NC(c3cnc4sccn34)=O)C2(C)C)nc(Cl)n1 N12CCC(C(C)(C)C1)OCCC(=O)NCCCOCCC2=O.CC1CC1CC c1(OC)c(C(=O)NCC(C)CNC(=O)Cc2cnc(C)[nH]2)cccc1Br CC(C)CCCCCCNC(C1CC2(CCN1C(=O)C(C)OC(C)(C)C)CC2)=O C=C(Cl)CCCNC(=O)Cn1cc(CNC(=O)CN)nn1.c1cccnc1 Cn1cc(C(=O)NC2CC3(C2)CC3NC(C2CCCCCC2)=O)nc1O Cc1cc(N(CC(F)F)C)nc(N(C)CCc2ccccn2)n1 c1(CC(=O)N(CC(F)(F)F)C(C)C)ccc([N+](=O)[O-])cc1F c1(C(=O)NC23CC(NC(C4C(C)COCC4)=O)(C2)C3)ccc(CO)cc1F CC(CC(=O)NCC1CC(NC(=O)CCN2CCCCC2)C1)N1CCCC1=O C(=O)(CCCC(C)(C)NC(c1nc(=N)cc[nH]1)=O)NCC1CCC(C)C1 N1(C(CC=CC)=O)CCC(N(C(c2cncc(-n3cccn3)n2)=O)CC)CC1 c1(CC(=O)NC(c2ncco2)CC)cc(-c2cncc(OC)n2)ccc1F c1(NC(c2ccc[nH]2)C)[nH]c(=NCCc2cc3ccccc3[nH]2)nc2scnc12 c1(C(N2CCC(O)(CNC(C(c3cccc(C)c3)O)=O)C2)=O)cc(F)cc(F)c1 N1(C(C(C)(C2CC2)OC)=O)CC(O)CC1CNC(=O)CCc1cnc[nH]1 C(=O)(C(F)CC(C)(C)NC(=O)CN1CCCCCC1)N1CC(C)OCC1C c1(NC(C23N(C(C4N(C)CC4)=O)CCC2C3)=O)cccc(C#N)c1 N1(C(C2(C)C(C)C2)=O)CC2CS(=O)(=O)CC2(NC(C23CCCN2CCC3)=O)C1 C1(CC(C)O)CCCCN1C(C12CC1CCN2)=O c1(OCC)nc(C)ccc1C(N1CC(CO)C1)=O.C1(C(=O)N)CCCC(C)C1 Cc1ccc(CNC(=O)C(F)C2CC(NC(=O)CCOCCO)C2)cc1 CCC(COC)C(=O)N(C)CC1CCCCN1C(=O)CSCC1CCCO1 C1(NC(CCN(C(=O)C(O)Cn2cncn2)CC#C)=O)CC1C1CCOCC1 C(c1cccc(F)c1F)=CC(=O)N(C)CCNC(C1COC2(CCC2)C1)=O C#CCC(C(=O)NC(CNC(c1sncc1C)=O)CO)C1CC1 C1(C(C)(C)C)CCCCN1C(=O)C=O.S(C[Si](C)(C)C)CCNC(C(C)O)=O.N c1(CN2CCC(C(N(C(C(=O)NC)C)C)=O)CC2)cc(C)n(-c2nccs2)c1C CC1(C)CCN(C(C2CCC3(CC3)C2)=O)CC1C(N1CCCC(C)(O)C1)=O Cc1ccc(F)c2[nH]c(-c3nc(CSC4C(C)(C)C4(C)C)no3)cc12 C1(C(=O)NC(C)CC)C2(CCC2)C12CCC2.C(=O)C(C)(C)C.C(=O)(CC)N N1(C(C=C(CCC)C)=O)CCC(F)(C)CC1.c1(C=O)ccc(=O)n(C2CC2)c1.N c1(C(N(C2CN(C(CC3CCC(C)C3)=O)C2)C)=O)sc(NC2CC2)nc1Cl C1(C(=O)NCC(CC=C)NC(=O)CCC(=O)NC)CCC(O)CC1 Cn1ncc(C(=O)NC2CC(CC(=O)NCC3COCC3O)C2)c1N C(C(C)(C)[N+](=O)[O-])n1cc(C(c2cncc(C(=O)O)c2)C)nn1.N12CCCC1C2 c1(C(N2CC(C)C(NC(=O)CN3CCN(C)CC3)CC2)=O)ccc2nonc2c1 N1(C(CCNC(C2(C#N)CCCC2)=O)=O)CC(O)C(O)C1CO N1(C(CCSCC)=O)CC(CNC(C2(c3cccc(Cl)c3)CC2)=O)C(O)C1 N1(C(c2n(C)ncc2C(F)F)=O)CCCC(N(C(C2CCC(O)C2)=O)CC)CC1 C1(CCOC)CCCCN1C(c1ccc(Cl)o1)=O N1(C(c2cn(C(C)C)c(=O)cc2)=O)CC2CC(NC(c3cscc3Cl)=O)CC1C2 C(CC)(CCC(=O)NC(CCOC)C(N)=O)NC(C=CC(CC)C)=O CC(C)(C)C#CC(=O)N(CCC(=O)NCCC1CC2CCC1O2)CCCO c1(C(CNC(CCn2cc(-c3ccn(C(C)C)n3)nn2)=O)=O)ccccc1F Cc1nc2cncc(C(N3CCCC(NC(=O)C(C)CC(C)(C)C)CC3)=O)c2[nH]1 O(N=C1CCCCCC1)CC(=O)N(CCNC(C(C)CN(C)C)=O)C1CC1 c1(CN(C(C)(C)C(O)c2ccccc2)C=O)cc(Cl)ccc1O c1(C(=O)NC(C)(C(=O)N(CCCO)CCCO)C2CCC2)ccc(F)c(F)c1 C(CN=c1ccnc(CO)[nH]1)(C1CC1)NC(C12CCCN(CCC1)C2)=O n1(CCC(=O)NC2CCC(NC(C(C)C3CC3)=O)CC2)cnc2ccccc12 C(CC(F)F)(C(=O)NCc1ccc(C(N)=O)o1)NC(CCOCC)=O C1(NC(CNS(CC)(=O)=O)=O)CN(C(c2cncnc2C)=O)CC2(CC2)C1 CC1CN(C(=O)COc2ccc(F)cn2)CCC1NC(=O)C(N1CCOCC1)C CCC(CC)CC(=O)NCC(C)(CNC(=O)CC1CCC(=O)NC1=O)OC c1(NCC(N=S(C)(C)=O)=O)nc2c(c(=NCC3COc4cscc4O3)[nH]1)SCC2 N1(C(CSSC)=O)CC(NC(=O)Cc2cnn(C(C)(C)C)c2)CC1CO C1(n2cc(C3CCCN3C(C34CCCC3(C(=O)O)C4)=O)nn2)(OC)CCCOC1 c1(C(N2C3CC(NC(C(C)n4cncn4)=O)C(C3)C2)=O)cc(Br)c2cn[nH]c2c1 C(C(C)C(=O)NCC(F)Br)N(C(C1C(C(C)C)C1)=O)C C1(CNC(C=CC(C)NC(c2c[nH]nc2C(F)F)=O)=O)OCCC1C c1(NC(CN(CCC)Cc2nc(-c3ccc(C)cc3)cs2)=O)ccccc1C c1(C(N2C(C(C)NC(C3CCC(C)(C)CC3)=O)CCC2)=O)cc(Cl)c(F)cc1F c1(C(N(C(C)CN(C)C(C2CCSC2)=O)C)=O)cc(C(F)(F)F)ncn1 C=CC1(O)CCN(C(=O)CCC2CC(NC(=O)CC3OCCC3C)C2)C1 Cc1cn2c(n1)C(C(=O)N1CCC1CNC(c1cc(C3CCC3)no1)=O)CCC2 CON=CC(=O)NC1CCCC1NC(C1CCC1(F)F)=O CCC(CCOC)C(=O)N1CCCC1(C(=O)NCC(C)Cc1cn[nH]c1)CC C(CC(C(C)(C)C)NC(c1cc(=O)n(C)o1)=O)N(C)C(c1scnc1Cl)=O c1(C(=O)NC2(CCCNC(Cc3cc(C)no3)=O)CC2)ncc(F)cc1F N1(C(C(NOC)=O)=O)CCCC2(CNC(=O)Cc3cccc(C)c3C)CCCC12 C1(CC)CN(C(=O)C(=Cc2cccs2)C)CCN1C(=O)Cc1cn2ccsc2n1 C1(NC(N(CC(CC)C)CC)=O)CCN(c2cccnn2)CC1 C1(F)(C(=O)NC(CC)CNC(C2(O)CC(C)(C)C2)=O)C2CCCCC12 N1(C(C(COCC)C)=O)CCC(C)(CNC(C2CC2c2sccc2C)=O)C1 C=CCC(C(=O)NC1(COC)CC1)NC(=O)CC1CCC(=O)N1 c1(C(F)(F)F)ccc(-c2nc(-c3ccc(Br)cc3)no2)nn1 N1(C(C(c2ccccc2)NC(=O)OC)=O)CC(C)(N2CCOCC2)C1 c1cccc(N2C(=O)CCC2=O)c1.c1(C(=O)OC)csc(C(C)NC(C)=O)n1.N N1(C(C(C=C)(C)CC)=O)CC2(C1)CN(C(C1CC13CCOC(C)C3)=O)CCO2 Cc1cc(C2(C(N3CC(O)C3)=O)CC2)cc(C)c1.C(=O)C(C)(C)C1CCC1.C C=CCCC(=O)N(C)CCOCCNCC=O.C(=O)(CC)NC(=O)OC c1(C(N2CC(O)CC(NC(=O)CC3CC4(CC4)C3)C2)=O)cncc2sccc12 C1(NC(=O)NC(C2CCCCC2)CO)CCCC(CC(F)(F)F)C1 C1(C)(C(=O)NCc2snc(CC)n2)CCCN1C(C1CC2CC2C1)=O c1(C=O)nc(C)[nH]c2nccc1-2.N1(C(C2(OCC)CCC2)=O)CCC(C)CC1.N C(=O)(C1=C(F)CN(C(C2CCC(C)(C)CC2)=O)CC1)N1C(C(=O)OC)C=CCC1 c1(C(=O)NC2C(OC)CN(C(=O)CCc3cncs3)C2)nccc(Cl)c1F C1(C(=O)N)(OC)CS(=O)(=O)C1.C1(C(N2CCCC2)=O)CCC(C(C)C)CC1 c1(OC)ncccc1C(N1CCN(C(=O)C)CC1)=O.C12(C=O)CC(C1)C(C)O2 C1(CC=C)(C(=O)O)CN(C(C2(N(C)C)CCCC2)=O)CCO1 c1(C(=O)NC(CC)CNC(=O)C(C)(O)C2CCC2)cc(Cl)c(C(F)F)cc1F O=C1CSC(C(=O)NC23CC(C(=O)NOCCOCCO)(C2)C3)C1 N1(C(c2csc(O)n2)=O)CCN(C(C2COCCO2)=O)CC(CO)C1 C12(CNC(c3c(C)con3)=O)CCCC1N(C(=O)CC1CC=CC1)CCC2 c1(C(=O)NCC2CN(C(C3C(C)(C)CO3)=O)CC2O)cc2cccc(Cl)c2s1 CCC(CC)C(C(=O)NC(C1CCCN1C(=O)CCCC(=O)NC(C)C)C)OC Cc1cc(C(N2CC3(CC3)CC2C)=O)cc(C)n1.C1(CC=O)CCC2CC2C1.N C(C(CC(C)C)C(=O)NCC(O)CNC(=O)C(F)(F)CCc1ccccc1)OC Cc1nsc(NC(C)Cc2ccccc2)c1C#N.C1(CC=O)CCS(=O)(=O)C1.N c1(C(N2CCC=C(C)C2)=O)cc2n(n1)CCO2 Cn1ncc2ccc(CC(N3CCC4(C3)CN(C(C3CC=CCO3)=O)C4)=O)cc12 C1(NC(c2cnc(C3CC3)[nH]2)=O)CCC2CN(C(=O)Cc3csc(Cl)c3)CC2C1 c1(C(=O)NC(C(=O)NC(CC=C)C2CC2)C2CCC2)ccoc1C C1(N(C)CC)CCN(C(c2cc(CCNC(C3(CO)CCCO3)=O)on2)=O)C1 N1(c2ccn(C)n2)CCC(NC(=O)C(C)(C)c2cnn(C)c2)C1=O CC#CCC(C(=O)NC(CC1CCCC1)CO)NC(=O)CCC(C)CC C1(O)(CNC(=O)CCC2CCCCN2C(c2ncccc2O)=O)CC2CCC1O2 N1(C(CCN(C(C2(CC(C)C)CCC2)=O)C2CC2)=O)CCC(OCCCO)C1 c1(C2(C(NC)=O)CCC2)ccc(F)c(Cl)c1.c1(C=O)cc(C#N)cs1.C1CC1 N1(C(c2c(C)onc2)=O)CCCC(NC(C2(C(F)F)CC2(F)F)=O)C1 c1(CN(C)C(c2ccc(C(=O)O)nc2)=O)cnc(-c2ccccn2)nc1O C(=O)(C(CC(C)C)C(N)=O)NCC1(C)CCN(C(CCC(C)=O)=O)CC1 C(C1=NOC2CN(C(=O)CSc3nnnn3C)CC12)NC(c1cc(CC)[nH]n1)=O C1(NC(CC=C(C)C)=O)CCCN(C(c2sccc2OC(F)F)=O)C1C Cc1cn2cc(C(N3CCN(C)CC3CNC(=O)C(C)C(C)(C)C)=O)sc2n1 CC1CCN(CC2CCCCCC2)CC1NC(c1cccc(C(N)=O)n1)=O c1(NC(C)CC2CCC2)ccc(S(=O)(=O)N2CC(C)CC(C)(C)C2)cc1F N1(C(C(CC=CC)C)=O)CCOCC(C(=O)NCC2(COC)CC2)C1 C1(C=O)CCC(C(C)(C)O)CC1.N1(C(C(=O)N(CC)CC)C)CCCCCC1.N C=CC1CN(C(C23CC(NC(c4n[nH]cc4C)=O)(C2)C3)=O)C1 C1(C(=O)NCC2(NC(C3CC34CCC4)=O)CCCCC2)CC1C1CCCCC1 N1(Cc2c(OC)nccc2)CCC(c2ccccc2)C12CC2 c1(C(=O)NCCC2CCCN2C(=O)Cc2c[nH]nc2O)ccc2c(c1)COC2 C(=O)(CCCCCCS(N)(=O)=O)NC(C(C)NC(c1cnns1)=O)CO c1(OC)ccc(C(=O)NCCCNC(=O)CC2CC2(C)C)c(O)c1F c1(C(=O)NCCC2N(C(CC3(C=C)CC3)=O)CCSC2)c(OC)ccnc1O Nc1ccc(C(N2CC3CC2CN3C(c2nc[nH]c3ncnc2-3)=O)=O)c(O)c1Cl C1(C(=O)NCC(CNC(C(=Cc2cnc[nH]2)C)=O)(C)O)CC2(CCC2)CO1 c1(C(=O)NCC(CC)NC(=O)C(O)COC)sc(Cl)c(Cl)c1N c1(OC)ncc(C(N2CCC(CNC(=O)CC3(C)CCC3)C23CC3)=O)cc1Cl C1(C2CC2)(NC(C2C(C=C)C2)=O)CCN(C(c2ncccc2COC)=O)C1 N1(CC(N2CCC(C(=O)NCCn3ccnc3)C2)=O)CCCCCC1 C1(C)CC(F)(F)CN1C(c1cccc(C(C)=O)c1)=O.CCCCC(O)C(=O)NC N(C(=NCCOC1CCC1)N1CCCC(C(F)(F)F)C1)CC(CC)(C)CO c1(C(N2CC(N3C(=O)CC(NC(CCC(C)C)=O)C3)C2)=O)cnc(N)c(N)c1 c1(C(N2C(CNC(C(CC#C)C)=O)CC3(CC3)C2)=O)cn(C)c2ccc(Cl)cc12 N1(C(CC2C3CN(c4ncc(C(=O)OCC)cn4)CC32)=O)CCOC2COCC2C1 C(=O)(C1=C(C)OCC1)NC(C(=O)NC(CC#C)CC)C(C)OC C1(OCC)CCCN(c2ccn(C)n2)C1=O.C12CCN(CC1)C(=O)C1CCCN21 C(C)(CN=c1[nH]c2c(c(=NC3CCCC3C(C)C)[nH]1)CCCCCC2)OC CC1CN(C(c2cnccc2Cl)=O)CC(C)N(C(c2cc(C#N)ccc2N)=O)C1 C1(CC)CC(F)(F)CN1C(c1cccc[n+]1[O-])=O.C1(C(=O)N)CC(CC(F)F)C1 Cc1nnc2n1CC(C(=O)N)N(C)C2.C12CN(C(=O)C(C)C#N)CC(F)(C1)C2.C C(CCC(=O)OC)NC(=O)NCC(=O)NCCCC CS(=O)(=O)c1ccc(F)c(C(=O)COC(=O)C=Cc2cncc(O)c2)c1 C(=O)(C1CCCc2nncn21)N1CC2(CN(C(C(C(CC)O)C)=O)C2)OCC1 N1(C(C2(C)N(C(c3cc(=NC)[nH]cc3)=O)CC=C2)=O)CC2CC(C)(C)C2C1 C#CCCC(O)C(=O)N1CCN(C(c2ccc(F)c(C(C)C)c2)=O)C(C)C1 c1(C(N2C3C(C(=O)Nc4cc(O)ccn4)C(C3)C2)=O)cccc(Cl)c1F c1(C(=O)OCC)ccc(C(=O)OC(C(=O)NC2CC2)C(C)C)c(Cl)c1 N1(C(C2N(C(C(C)NC(=O)NC)=O)CCCCC2)=O)CCC2CC1C(=O)N2C Cc1cc(C(N2CCN(C(c3ccoc3C)=O)CC23CCC3)=O)c2occc2c1 C(CO)(CC(C)(C)C)c1cn(C(COCC)C(=O)N(CC(F)F)C)nn1 N1(C(CC2C(OC)COCC2)=O)CCC2CN(C(=O)C)CC12.C(=O)CN(C)C.N c1(C(N2CCC(F)(CNC(=O)CCC3CC3(Cl)Cl)CC2)=O)cccc2c1CCO2 C(=O)CCC(=O)N(C)C.c1(NC(C2(COC)CC=CC2)=O)ccc(C)cc1 c1(C(=O)NCC2CN(C(CC3(CC)CCC3)=O)CC2C)cccc(C)c1Br Cc1nc(CNC(=O)C(CCN(C)C)NC(C2CCCOCC2)=O)c(C)s1 CCCCC(C(=O)NCc1ccnc(C)n1)NC(=O)C(C1CCC1)OC Nc1cccc(-n2cc(CCNC(=O)CC3CC(F)(F)C3)nn2)c1 CC1CN(C(c2nc(O)[nH]c(=O)n2)=O)CCN1C(=O)CC(C)c1ccco1 c1(OC)ccc2c(c1)CCC2(C)CNC(=O)NCCC.C(C)(C)C.C(C)=O c1(NC2(CNC(CCCC#C)=O)CCCCCC2)cc(C)nc2ncnn12 CCCC(CCCO)C(=O)NCC(C)(C1CC1)NC(=O)CCC(=O)NC N1(C(COCC)=O)CC(NC(c2ccccc2-n2cnnn2)=O)CC12CCCC2 c1(C(N2CCC(O)(CCNC(CCSC)=O)C2)=O)cc(S(N)(=O)=O)ccc1O N1(C(CCC)=O)CCC2C(NC(c3csc(COCC)n3)=O)C12 Cc1nn(C)c(C)c1CC(=O)N(c1nccc(C(C)C)n1)C1(C#N)CCNC1 N1(C(C(CC)N(C)C)=O)CCC2(CCCCC2NC(=O)CSc2nncs2)C1 c1(CC)nccnc1C(=O)NC(Cc1cn(C(c2ccccn2)C)nn1)C(=O)O C12(CNC(c3nc(CC)sc3)=O)CCCC1CN(C(C1SCCCS1)=O)C2 c1(C=O)cncc(S(C)(=O)=O)c1.N1(C(c2n(C)ncc2)=O)CCC2CCC12C.N C=CCC(C)C(=O)NCCNC(=O)CSc1nncn1C1CC1.C1CC1 c1(C(N(CCC)CCNC(c2cnnn2C)=O)=O)cc2cc(F)cc(OC)c2[nH]1 c1(OC)cc(CN2CC(C(F)(F)F)CC(C)C2)cc(Cl)c1 N1(C(C2(CCC=C)CN(C(=O)C(C)c3ccco3)C2)=O)CCC(C=C)C1 Cc1nc(CC(=O)NCC2(C(=O)NC(c3ccnn3C)C)CC2)co1 Cc1ccc2cc(C(=O)NC(CNC(=O)C(C)CN(C)C)C(C)C)[nH]c2c1 n12nc(C)c(c1C)C2.N1(CC)CCCC(C(=O)NCCC(C)N(C)C)C1 C1(OC)CCC2(C(=O)NCC3CN(C(=O)CCCCN(C)C)C3)CCC12 c1(C(N2CC(NC(CCC=C(C)C)=O)C(N=[N+]=[N-])C2)=O)cn2c(n1)CCC(C)C2 C(CCC(C)(c1nnnn1C(C)C)NC1(CCO)CCCCC1)=CCC c1(SCC=CCc2ccc(OC)cc2)cc(OC(F)F)ccc1OC(F)F N1(C(C2CCN(CC)C2)=O)CCC(C)(C(=O)NCc2cc(CO)n(C)n2)C1 N1(C(C(C)OC(C)=O)=O)CC2(C1)CN(C(=O)Cc1sc(S)nc1C)CCO2 CCCC(C(C)(C)C)NC(C1C(CC)CCN1C(=O)CCc1cc(C)[nH]n1)=O C12(C(N3CCC(F)(CNC(C4(O)CCOCC4)=O)CC3)=O)CCN(CC1)CC2 C(=O)(CC(C)(C)C)N1CC(O)(CCNC(CN2C(C)CC2)=O)C1 c1(C(=O)NC2CC(C)N(C(=O)Cn3cc(CO)nn3)C2)c(O)cc(O)cc1O C1(CNC(c2c(C)ncnc2)=O)CC(C)(C)CN1C(=O)CCC=CBr O=C1CCC(C(=O)NC2CCCC(NC(C34CCC(CC3)C4)=O)C2)CCN1 C#Cc1ccc(C(=O)NCC2CC(NC(=O)C=CSC)C(O)C2)c(F)c1Cl N1(C(c2c(CC)nns2)=O)CCC2(C1)CN(C(=O)C(O)C(C)SC)CC(C)O2 CCC(C)(O)C(=O)N1CC2C(CNC(c3ccc(-c4cn[nH]c4)cc3)=O)C2C1 C(C(C(C)(C)C)NC(=O)CCC1CCC1)OC.C1(CC=O)CC(C)=NO1.N C1(C=O)CCCC(O)(C(F)(F)F)C1.O=C1CCC(CC(N2CCC(C)C2)=O)N1.N C1(n2cccc2)(C(=O)NC(C2CC(NC(=O)CC(C)C)C2)C)CCCC1 c1(C(=O)NCC2CC(C)N(C(=O)CC(C)(C)C)C2)sccc1S(N)(=O)=O C1(SC)CC(CC(=O)NCC2CCC2NC(C2(Cl)CCC2)=O)C1 N1(C(CC=CCCCCC)=O)CC(C(N2CC3CCC(O)C3C2)=O)CC(C)(C)C1 C=CC1(NC(=O)C(CC#CC)NC(=O)Cc2ccnc(O)c2)CCCCC1 CN1CCOCC1C(=O)NCC1(C(=O)NC2CCCC2F)CC=CC1 C1(NC(C(N2CC(C)C2C)=O)=O)CCCCN1C c1(CC#N)ccccc1C(N1CCC(C(F)C(N2CC(F)(C(N)=O)C2)=O)C1)=O c1(C(=O)NC2CC(F)(CNC(CNC(CCC)=O)=O)C2)cncc(O)c1 c1(CC(N2CCN(C(c3ccc[nH]3)=O)C(CO)C2)=O)cc(Br)ccc1Br CC(C)(C)C1=NOC(C)(C(N2CC3CCC(C2)N3C(=O)Cc2nc[nH]n2)=O)C1 C(CC(=O)NC)N(C)C=O.C1CCC1.C(=O)CCc1cnn[nH]1.C(C)(C)C c1(C(N2CC3CC3C2)=O)cc(F)c(O)c(Cl)c1.C1(C(NC)=O)CCC2(CC2)C1 c1(C(=O)NCC(N(C)C(C2CCC(F)C2)=O)C2CC2)c(Cl)ccc2ccoc12 N1(C(C2N(C(C(CC)(C)C)=O)CC2)=O)CC2COCC2(C(=O)O)C1 O(N=C1CCCCCC1)CC(N1CC(NC(C(C(C)C)F)=O)CC1(C)C)=O CC1(F)CN(C(=O)CSc2cccs2)CCN(C(=O)C(=O)Nc2ccccc2)C1 CC(C)CC(C)(O)C(=O)NCC(O)CNC(=O)CCCOc1ccc(F)cc1 C1(C(=O)NC(C#C)CC2CC2)COCC1NC(c1sccc1F)=O n1(CC)ccc(C(=O)NCCC2CCC2)cc1=O.N1(CC=O)CCS(=O)CC1 c1(-c2nc(-c3c4c([nH]n3)C(C)CCC4)on2)cc(Cl)c(Cl)cc1[N+](=O)[O-] c1(N(C)C)cccnc1C(=O)NCC1CCN1C(=O)Cc1ccc(Cl)nc1 c1(C(N2CCC(CN(C(C(CC=C)C)=O)C)C2)=O)cc(S(=O)(=O)NC)c[nH]1 C(C(CC(C)C)C(=O)N1CCCCCCC1C)NC(C(OC)OC)=O C1(C(=O)NCCCCCN(C)C(c2nnn3c2CCC3)=O)CC2OC(=O)OC2C1 C=CCC(CNC(c1cocn1)=O)C(=O)NCC1CCCC1O C1(CNC(c2ccco2)C)CCCCN1C(=O)Cc1cocn1 C1(NC(Cc2c(C)n[nH]c2)=O)CCCC(NC(c2nnn(C(C)C)c2C)=O)C1 C1CCS(=O)(=O)C12CN(C(=O)C1CC1)C2.Cc1nc2ncc(C=O)c(=O)n2[nH]1.N CC(CNC(=O)C(C)(C)CF)CCC(=O)NCCNC=O.C(C)(C)C.O C(=O)(CCCCCC(C)C)NCC1N(C(c2c(C)ccnn2)=O)CC1 c1(C(C)(C)C)ncncc1C(N1CC(=C(F)C)C1)=O.C1(C=O)CCC(F)C1.N n1(CCC)nc(C)cc1C(C(=O)NCc1ccccc1)N(C1CCCC(C)C1)C CC1CCC(C(=O)NC(C2CN(Cc3ncoc3C3CCC3)C2)C)O1 C1(NC(CC=C)=O)CCCCCC1NC(=O)CCOc1ccccc1F CC(C)(C)CCCC(=O)NC1CC(F)(C)C1.c1(C=O)nn[nH]c1C(F)(F)F.N N1(C(CCNC(C)=O)=O)CC2C3CCC(C2C1)N(C(C1CC=C(C)CC1)=O)C3 C1(C(N2CCC(CNC(=O)COCc3ccccc3)C2)=O)CC12CCCC2 c1(C(N(C)CC2CN(C(C3(O)CC3)=O)C2)=O)ccc2nonc2c1 N(C1c2ccccc2CC1NC(=O)CCCF)C(C(C(CC)C)OC)=O N1(C(CC2C(C)OCC2)=O)Cc2occ(C(=O)NCC3(O)CCOC3)c2C1 c1(OC)cccc(Br)c1C(=O)NC1CN(C(=O)C(F)(F)c2ccccc2)CC1F c1(C=O)n[nH]c2ccccc12.C1(C2CC2)CCCCN1C(C12CC(F)(C1)C2)=O.N c1(CNC(=O)CC2CCCN2C(=O)C(F)(F)F)ccc2c(c1)CNC2=O CC1CCN(C(=O)CC(F)(F)F)CCN1C(=O)C(=Cc1cn(C)nn1)F c1(C2c3nnnn3CCCN2)cc(F)ncc1F.C(C)(C(=O)NO)CC(C)C N1(C(c2c(NC(=O)Cc3c(Cl)cccc3Cl)c[nH]n2)=O)C2CCC1CC(O)C2 C(C(CC(F)(F)F)NC(C1CC2CC2C1)=O)NC(c1ccccc1F)=O c1(C2CCC(=O)N2)cccc(C(=O)NCC(F)CNC(=O)Cc2cccnc2)c1 c1(SC)ccccc1-c1ccc(NC(c2cc(C(=O)O)on2)=O)cc1 C1(C(N2CC3C(CNC(C4CCC(=C)CC4)=O)C3C2)=O)CC(C)CC(C)(C)C1 c1(C(N2C(CCNC(CCCNC(=O)OC)=O)CCCC2)=O)cc2occc2[nH]1 c1(C=O)cc2n(c(=O)c1)CCS2.C(=O)(CCC=CC(C)C)NC(C)C.CC N1(C(C(C(COC)C)C)=O)CC2CC(C1)N(C(c1n[nH]cc1C)=O)C2 N#CC(S(=O)(=O)c1ccc(C(F)(F)F)cc1)=C1CCCCCC1(F)F C(=O)(C1CCCn2cnnc21)N1CC(C(C)NC(C2(C#N)CC3CC3C2)=O)C1 C1(CC(=O)NC(C=C)C2CCC2)CC(C)N(C(c2ccccc2O)=O)C1 c1(C(C)C)ccc(CN2CC3(CC(C(=O)NC)C3)C2)c(Br)c1.c1cnn(C)c1 N1(C(C(C)=CC2CC2)=O)CCC(CCC(=O)NCC(CO)C(C)C)CC1 CCCCCC(C)(C)C(=O)N1CCCCC1.c12cc(C#N)nc(n1)CN2C C1(NC(c2c(C)coc2)=O)CCC12CN(C(=O)Cc1cccc(F)c1F)C2 N1(C(c2ccc(CSC)o2)C(=O)NCCCC)CCC(N2CCC2)CC1 C1(CCC=C)(C(=O)OC)CN(C(c2cnn(C3CCCC3)c2)=O)C1 C(CC(CC)C(=O)NC(CCSC)C(N1CC2(CC(O)C2)C1)=O)=CC N1(C(CC(CC)OC)=O)CCC(C2CCN(C(C3OC(C)CC3C)=O)CC2)C1 C1(C(=O)NC2CCN(CC)C2=O)N(C(=O)CC2CCCC(=O)C2)CCCC1(C)C C1(CCOC)(NC(=O)CCSC)CCN(C(=O)CCC2CCCCN2C)CC1 Cc1c(CNC(c2ncnn2C)C)ccc(OCC(F)(F)F)c1Br CC1(C)C(C(N2CCC(C)(C)C2)=O)CC1(F)F.C1(C=O)CCCN1C1CC1.C n1(CCNC(c2nc(C(C)NC(=O)Cc3cn[nH]c3)oc2)=O)cccnc1=O c1(C(=O)OC)nn(C)nc1C(=O)NCCCCCNC(C1CCCOC1C)=O c1ccc(Cl)c(Cl)c1.Cn1cc(C(N2CC(F)(C(=O)N)C2)=O)c(C(F)F)n1.C c1(C(=O)NCC(CN(C(C(C=CC)O)=O)C)O)c(OC(F)(F)F)cccc1F CCC(C)CC(=O)NCCC1CC(NC(=O)Cn2cnc(=N)[nH]2)C1 C1(C(=O)NC2CCCCC2F)C2CCC(C2)N1C(c1cc(F)ccc1O)=O c1(C(=O)NC(CCC)CCCNC(C2(C)CC2C)=O)cccc2oc(C)cc12 N1(C(CC(=C)C)=O)CC(NC(C2CCC(NC(C)=O)CC2)=O)C2(CCOCC2)C1 C(=O)CC(O)C(C)C.c1(NC)cncc(C(=O)NCc2ccc(CC)cc2)c1.N C(=O)(CC(C)C(C)(C)NC(C1CCC(C)CC1)=O)NCCn1c(C)cc(C)n1 N1(C(C2N(C(c3c(OC)ncnc3OC)=O)CCC2)=O)CC2CCCCC2C1 c1(CN(C(c2cnn(-c3ccc(F)cc3)c2)C(=O)NC)C(C)C)ccccc1Cl c1(C(=O)OC)cnc(C(C)(C)C)nc1N1CCC(c2cnc(Cl)s2)C1 c1(NC(=O)NCC(c2ccc(Br)cc2)C)snc2ncccc12 CC(C)CCC(=O)N1CCCC1CN(C)C(C1CCCC2CC12)=O C1(NC(C(CCCCC)O)=O)CCCC12CCN(C(=O)C(=O)C1CCCC1)CC2 N1(C(C2N(C(CC=C=C)=O)CCC2C)=O)CCCC(C2CC2)CC1 Cc1cc(CC(N2CCC(c3ccc(N4CCC4)cn3)C2)=O)cc(C#N)c1 C=CC1CN(C(c2nccnc2N)=O)CC1NC(C1(C)CC1(C)C)=O Cc1cccc(Cl)c1C(N1CC2CC(NC(=O)CCCCN(C)C)C2C1)=O c1(C(=O)NCCC(C)NC(CCCC(=O)NC(C)C)=O)nc2cnccc2s1 C1(C(=O)NC(c2nccn2C)CC)CCN(C(c2ccc(O)cc2)=O)C1C C1(CNC(N2CCCS(=O)(=O)CC2)=O)CCC2(CCCCCCC2)O1 c1cc(CSCCOC2CCCC2)cc(-c2cn(C3CCC4CC34)nn2)c1 n1(CCC=C)cc(C(=O)NC2CC2NC(C2CSCN2C(=O)CC)=O)nn1 c1(NCCc2cc(OC)c(Cl)cc2)c(Cl)cc(C#N)cc1C#N N1(C(c2c(CC)onc2)=O)CC(NC(c2cnnc(Cl)c2)=O)C2CCCCC12 C(=O)(CC1CN(C(c2cnc3[nH]ccnc2-3)=O)Cc2ccc(OC)cc21)OC CCC(CC(C)C)C(=O)NCC(O)CNC(C1(c2cc(C)cc(C)c2)CCC1)=O C1(C(=O)NCC(Cc2ccccc2)NC(COCC=C)=O)(C)CC=CC1 Cc1c(C)cccc1F.C1(CC=O)CC2(CC2)CN1C(=O)CN1CC(C)(C)C1 c1(OC)cc(CC(=O)N(C)CC2CCN(C(C3(C)CCCO3)=O)CC2)ccc1F C1(C(=O)NC(C2CCCN2C(=O)CSCCC#N)(C)C)CCC(=O)N1 C(=O)(CC(C(F)(F)F)NC(c1nccn1C)=O)N1CC(CC)SCC1 C1(C(N2C(C)C(NC(c3csc(=N)[nH]3)=O)CC2)=O)CS(=O)(=O)CC12CC2 C(=O)(C1=CCC(C(F)(F)F)OC1)NC1(C)CCN(C(c2cc(C#N)on2)=O)C1 C(=O)(CCC(F)(F)C(F)F)NC(CNC(CCCNC(C)=O)=O)(C)C1CC1 c1(C(N2CC(NC(CSC(C)=O)=O)C(F)(F)C2)=O)ccc(O)c(F)c1F C(=O)(CCCN(C)N=O)N1CCC2(NC(CCCN(C)C)=O)C(C1)C2 c1(CC)nn(C)cc1NC(C1(C)CC(C)=NO1)=O.C1CCCN1C(=O)C.N C(C)(C)(CCCC(=O)NCCOC(F)F)NC(CNC(CC(C)C)=O)=O c1(OC)cc(C(=O)NC2CN(C(=O)C3=COCCC3)C3CC23)ccc1F C1(NC(C=C(C)C)=O)(CO)CCCN(C(=O)C(C)=NOCC#N)C1 c1(C(C(=O)NC2CCOC2)N(C(C(CC)C)C)CC)cc(C(C)(C)C)n(C)n1 Cc1cc(C(N2CCC(CNS(=O)(=O)CCBr)CC2)=O)ncc1Br C1(NC(c2cnc(C)[nH]2)=O)CCC(C)N(C(c2ccnn2C(F)F)=O)C1 C#CCCCC(C)C(=O)N1CCC(C)(CNC(=O)CCc2cnn(C)c2C)C1 N1(C(C(CC(C)C)ONC(=O)CN2CCCC2)=O)CCCC(C)(O)CC1 c1(N2CC(C)OC(C3CC3)C2)nc(N(CCCF)C)c2ncn(C)c2n1 N1(C(CCS(=O)(=O)NC)=O)CCOC2CN(C(=O)C(C)(C)CC(F)(F)F)CC12 N1(C(CC2CCN(CC3C4CN(C)CC43)C2)=O)CCC2(CC1)CNC(=O)C2 CP(C)(=O)C(O)C(=O)NCCN(C(C1SCCCS1)=O)Cc1ccccc1 O=C(CC(C(F)F)N1CCOCC1)NC1CCC1CNC(=O)COCCF.O C1(C(=O)NCC2CN(C(COC(C)C)=O)C(C)C2)SC2C=CC1CC2 c1(C=O)[nH]c(C)c(S(N)(=O)=O)c1C.C=CC(CC)CC(=O)N(C)CCOCC c1(CC)ccc(C(=O)NCC2CCCC2NC(C2CCSC2)=O)s1 c12cc(Br)c(Cl)cc1SC(C)COOP(=O)(OOC)O2.C(C)(C)OC c1(C(=O)NC(c2ccccc2)CNC(c2c(C)noc2)=O)ncnc2sccc12 CC(C)C(C)CC(=O)NC1CN(C(=O)Cc2ccc(Cl)cc2Br)CC1C c1(C(=O)NC2CCCN(CCOCC)CC2)cn2cc(Cl)cc(Cl)c2n1 C(CCC(C)(C)NC(c1cc(Br)no1)=O)NC(CC(C)N(C)C)=O N1(C(C)=O)CC2(C1)CN(C(c1ccc(Br)o1)=O)C2.C(C(=O)N)N(C)C(N)=O CC(C)(CC#N)C(=O)N1C2CCC1C(NC(C1CC3CCC1CC3)=O)C2 C=CCCCCCC(=O)NC1CCCC1NC(=O)C(COC)COC N1(C(C(CCC)(C)O)=O)CCC2(CC1)CN(C(=O)CSCC(C)C)C2 c1(C(CCSC)NC(=O)NCC2CCC2c2ccccc2)ncc(F)cc1F N1(C(CC)=O)CCCC(C(=O)NC(C)CCNC(c2ccn(C)c2CC)=O)C1 N1(C(C=C(C)C(C)C)=O)CCCC(C)C1CNC(c1cc(Br)n(C)c1)=O N1(C(CC(C(C)C)NC(C2CC2c2ccccc2)=O)=O)CCC(C)(C#N)CC1 c1(CC)ncc(C(=O)NC2CN(C(C3CN(C)CC(C)O3)=O)C2)c(O)n1 c1(OC)ncnc(C(N2CC(CNC(c3cc(O)n(C)n3)=O)CCC2C)=O)c1F N1(C(CC2N(C(C(C=C)O)=O)CCC2)=O)CC2CC1CN2C(C)=O c1(-c2ccc(CN3CC(C(=O)OC)C(N)C3)s2)nc[nH]c2ncnc1-2 c1(C(N2CCN(CC#C)CC2)=O)n[nH]c2c1CN(C(=O)CCN1CCCC1)CC2 c1(-c2ccc(OC)cc2)csc(=Nc2cccc(Br)c2)n1CC1CCOC1 C1(CC)(CC)NC(=O)N(CC(=O)NC(C)(C)CO)C1=O.c1(C=O)occc1Cl C12(C(N(C(C3CCOC3)C)C)=O)CC(CO)(CN1C(=O)CCC1CCCO1)C2 c1(CC)nc(CCNC(=O)C=CCC)n[nH]1.C(c1cc[nH]c1)=CC(=O)N C(=O)(CCCCN=[N+]=[N-])N(C(C(=O)NCC1(O)CCC(C)CC1)C)C N1(C(c2ccn(CCCC)n2)=O)CC2CC2(C)C1.C(=O)(C(C)(C)n1cnnn1)N N1(C(c2cc(C)c(O)nn2)=O)CC2CCN(C(=O)C(F)n3cccn3)CC12 C1(NC2C(SC)CCC2)CNCC2(CCC2)C1 N1(C(C2C(CNC(c3cc(O)cs3)=O)OCC2)=O)Cc2c[nH]nc2C1 CCCCCC(O)CC(=O)NC1CC(CO)N(C(c2cc(C)c(CO)cn2)=O)C1 S(=O)(=O)(c1ccc(N2CCN(CC(C)C)CC2)c(F)c1)N1CCC(C)C1 c1(N(C)CC2N(C(C3CC4(CC(OC)C4)C3)=O)CCCC2)ncc2ccsc2n1 C1(CC)CCCCN1N1CCC1COCCO C(=O)(C(=O)N1CCC1CNC(=O)C(C)SC(F)(F)F)NCC Cc1ccncc1CN(C)C(C1(C)C=CCN1C(c1cc(O)cs1)=O)=O c1(C(=O)NC(c2ccccc2Cl)CC(=O)O)cc2ccc(Br)cc2c(=O)o1 N#Cc1cnc2c(C(=O)NC3CN(C(c4cc(Cl)ns4)=O)CC34CC4)cnn2c1 N1(CCC(C)NC(COC(CC)(C)C)=O)CCN(C(C2(C#N)CCCO2)=O)CC1 C(=O)C1=CCS(=O)(=O)C1.Cc1nn(C)cc1CCC(=O)N.C(C)(C)C1CCC1 c1(C(=O)OC)nc(NC(C2(CNC(C3CCCCC3C)=O)CC2)=O)sc1C CCC(N)(C(=O)NCc1nc(C#N)cs1)c1ccccc1 c1(N(C(CC2CC2)=O)CC)cccc(C(C)C)n1.C1(C=O)CC(C#N)C1.C N#Cc1nccnc1N1CC2C(NC(=O)CC3CC4(CC4)CO3)C2C1 c1(C(N2C(C)(CNC(C3CCCOC3)=O)CCC2)=O)ccc(=O)n(O)c1 c1(C(=O)OCCN(C)C)ccccc1C(=O)NCC(N1CCCCC1)(C)C c1(C(N(C2CCCN(C(c3nncs3)=O)C2)CC)=O)cncc(Cl)c1Cl c1(C(C(=O)NCCSC)N(CC(C)C#N)C2CC2)ccc(CC(C)C)cc1 c1(OC)ccnc(C(=O)NC2CCCC2NC(=O)C=Cc2ccsc2)c1F C1(C(=O)OC)Cc2c(C)cccc2CN1C(=O)CC1CC2C=CC1CC2 c1(C(N2C(C)CC(NC(=O)Cc3ccc(Cl)s3)CC2)=O)nccn2ccnc12 c1(C(=O)Nc2c(C(=O)OC)scn2)cccc(C2CCOCC2)c1 c1(C(=O)NC2C(CC)N(C(c3ccco3)=O)CC2)ccc2n[nH]c(C)c2c1 c1(C(=O)NC2CCN(c3nc(CC)oc3C)CC2F)cccn2c(O)nnc12 CCC(CC)(CO)C(=O)N1CCC(CO)C(NC(C2CCC(C)(C)CC2)=O)C1 c1(C(=O)NC(C(C)(C)NC(C2N(C(C)=O)CCC2)=O)C)ccc(F)cc1.C c12cccc(F)c1SCOC(=O)Cc1cc-2ccn1.c1(CO)ccc(Br)nc1 Cc1c(CCNC(=O)C(N2CCNCC2C)=O)cccc1Cl CC1CN(C(=O)C(O)C2CC2)CC2(CCN(CC(O)CC(F)(F)F)C2)O1 N1(C(=O)CCc2cncs2)CC=CC(C(=O)N(C2CC2)C2CC2)C1 C1(C(N2CC(CNC(C(F)OC)=O)C2)=O)CCc2ccnn2C1 c1(C(=O)NC2CCC(N3CCN(C(CC)=O)CC3)C2)ccc2oncc2c1 Cc1nncn1NC(=O)C1C=CCN1C(c1ccc(O)nc1)=O c1(C(=O)NC(CNC(C2C(C(=C)C)OCC2)=O)(C)C2CC2)cccc2nonc12 Cc1cc(C(N2CCC(N(C)Cc3ncnn3C(C)(C)C)C2)=O)ccn1 c1(C(=O)NCC2CN(C(CCCc3ccc(C)s3)=O)C3C2C3)cc(Cl)ncc1O c1(C(CN(C)C)NC(N(C)Cc2cnco2)=O)ccccc1 N1(CC(=O)NCC(CNC(C2(C#N)CCOCC2)=O)O)CCc2ccccc21 N1(C(CC2CCN(OCC)CC2)=O)CCCCC1C1CC(N)CCO1 Cc1ccc(C(C)C)c(Oc2nc(C3CC34CC4)nn2-c2ccnc(O)c2)c1 Cc1nn(C2CCC2)cc1C(=O)NCC(C1CCCC1)NC(c1ccnn1C)=O Cc1cc(C(=O)N(CC(=O)NC(c2ccco2)CO)CC2CC2)co1 C(=O)(CCCC(C)=O)N1CCC(N(CCC)C(c2cc(Cl)ns2)=O)C1.NC C1(C)CC(F)(F)CN1C(c1cn(CCO)nc1C)=O.C(C(=O)NC)N(C)CC C(CC(C)C(=O)NCC(C)N(C)CC1CCCC12CC2)OC CC(c1ccccc1F)=CC(N1CCN(C(=O)CC2(C)CC2(Cl)Cl)CC(O)C1)=O CC1(O)CCN(Cc2ncc(C(=O)O)cc2F)CC12CCOCC2 c1(C(N2CC(C)(C(=O)NC(c3cc[nH]n3)C)C2)=O)ncccc1Cl N1(C(CCc2c(C)ncs2)=O)CCCC2(NC(c3ccc(F)s3)=O)CCCC12 c1(C(N2C(CNC(CC(C)O)=O)CC2)=O)cccc2[nH]nc(O)c12 S(=O)(=O)(c1ccc(C)nc1)N1CCCC(CNC(C(CC)(C)C)=O)C1 C1(NC(c2cncn2C2CC2)=O)CC2(C1)CC(C(=O)NCC(O)CF)C2 c1(CC(=O)NC(C)(C)CNC(C2CC3CCC(C2)O3)=O)cccc2[nH]ncc12 C1(C(=O)NC(c2nc(C)sc2)C)CN(C(C2CCC(O)CC2)=O)CC1C1CC1 c1(N(C)Cc2ccoc2)nc2c(c(=NCc3ccc4[nH]ccc4c3)[nH]1)CCC2 C1(NC(c2c(C(N)=O)nccc2)=O)COC2C(NC(c3sccc3F)=O)COC12 N1(CCN(C)C(c2ccc(O)nn2)=O)CCN(C(C2CCC2(F)F)=O)CC1 C1(C(N(C2CCN(C(C(CSC)C)=O)CC2)C)=O)CCOC(=O)CC1 N1(C(Cc2cc(C)on2)=O)CCC(CCCCNC(C2CCC=CCC2)=O)CC1 C1(CN(C)Cc2c(CC)csc2)CN(C(=O)CC2C=CCCC2)CCO1 C1(NC(C2(CSC)CC2)=O)CCC(C)(C)C1.C(=O)C.C(=O)C1CC1 N1(C(c2ccc(SC)cc2Cl)=O)CCC(C2CC2)(NC(C2CC3CC3C2)=O)C1 CC1CCCC1(C)C(=O)NCC1(CO)CCN(C(=O)COCC(C)(C)C)C1 C(=O)(CCCCC(F)(F)F)N1CC(O)(C(C)NC(c2[nH]cc(CC)c2)=O)C1 c1(CC)nocc1C(=O)NC(c1ccnn1C)C(=O)NCCCc1cnn(C)c1 C#Cc1cnc(C(=O)NC2(C)CN(C(C3CC3C(C)C)=O)C2)c(C)c1.O N1(C(c2c(C)ncs2)=O)CC(=O)NC2CN(C(=O)CSC(F)(F)F)CCC12 C(CCCCC(=O)NC1CN(C(=O)Cc2ccc(C)c(Cl)c2)CCC1C)=CC C(=O)(N=c1cc[nH]cc1C(C)C)N1C(CC(=O)OC)CC2(CCC2)C1 c1(C=O)ccc(C2CC2(F)F)cc1.C(C(C)CC)NC(CC1CC(OC)C1)=O.N C(=O)(CC1=NNC(=O)C1)N1CCN(C(C2C(C)(C)NC(=O)C2)=O)CC1CC(F)F C(C(C)(CC)C(=O)N)NC(c1nc(OCC)oc1)=O.C1CC2CC3C(C2)C13 C(=O)(C1CCCc2sccc21)N(C)CCNC(C1(C)CC(C2CC2)=NO1)=O N1(CC(N2CCN(C(C3CC(F)(CO)C3)=O)C3CC23)=O)CCCNS1(=O)=O C12(C=O)CC=CC(C1)OC2.Cc1ccsc1C1CC1C(=O)N(CCC)CCC Cn1c(O)nc2ccc(C(=O)NC3CC(C(=O)O)CC3O)cc12 c1(N(C)CC2CCN(C(c3cc(CC)nc(O)c3)=O)C2)nnc(C)c(C)c1C#N CCC(C)C(C(=O)NCCC(C)CO)N(C)C(c1cc(C)cc(O)n1)=O N1(C(c2c(C)cc(OC)nc2)=O)CCC2(CC1)CCN2S(=O)(=O)c1cccs1 CC1CN(C(=O)C2=NOCC2)CC1CNC(=O)CCOCC1CCC1 Cn1ncc2c(Nc3cccnc3N3CCCC3)[nH]c(=NC3CSCCSC3)nc12 C1(CNC(C2(C)CN(C(C(C(C)C)=O)=O)C2)=O)CC2(CCO1)CC2 C(=O)(C1=CC2CCCCC12)NCC(C)(C)CCNC(C1C2(CC2)C12CC2)=O c1(C(=O)NC2CC(C)(NC(C(C(CC)C)OC)=O)C2)cnc2cc(O)ccc2c1 CC(C)CCC(C(=O)NCC1(C)CC1(F)F)NC(=O)C=Cc1cocn1 N1(C(C23CCC(OC)C2C3)=O)CCC(CC(=O)NC)C1(C)C.c1cncc(C)n1 c1(C2(CN(C)C(C3CC(=O)CC34CCC4)=O)CCCC2)ccc(F)cc1Cl C1(NC(CCN(C)CC)=O)CC(NC(c2c[nH]nc2-c2ccsc2)=O)C12CCC2 C(=O)(C(C)CC(C)(C)C)NCC(C)NC(Cn1ccc(C)n1)=O Cc1nc[nH]c1CC(=O)NCCCCCNC(C1CC1Sc1ccccc1)=O S(=O)(=O)(c1ccc(N2CCCCCCCCC2)c(C#N)c1)NC1C(C)CN(C)C1 C1(OCC)CCN(C(=O)CC2CC(NC(=O)Cc3cnn(C)c3)C2)CC1C C(CC(C)(C)CC(=O)N(C(C)CCNC(=O)C(C)(C)COC)C)OC Cc1cccc(C(=O)NC2(CN(C)C(C3CCCC34CC4)=O)CC2)c1Cl C1(OCCNC(N2CCC(N(C)C)C2)=O)C#CCCCCC1 CCC(CC)C(F)C(=O)NC1(C(=O)N(C)CCc2cnn(C)c2)CC1C N1(C(CN(C(COC)=O)C)=O)CC2CCC2(CC)C1.c1(C(=O)N)c(C)cnn1C c1(C(=O)NCC(CC)(C)NC(=O)Cn2nnc(C)n2)cc(Cl)cc(C)c1C c1(OC)ccc2c(c1)N(C)CCN2Cc1ccccc1C(F)(F)F c1(C(=O)Nc2cc(C)nn2C)ccc2c(-c3cncc4cc[nH]c34)cccc2n1 c1(C(N2C(CC)CN(C(c3ccncc3Cl)=O)CC2)=O)ccnc2ccncc12 C1(CS(=O)(=O)NCCNC)(C(=O)OCC)CC(F)(F)C1.c1ccoc1C CC(CCCCNC(C1C=CCCC1)=O)NC(=O)CC1CC(c2ccccc2)C1 C1(NC(C(CC(N)=O)O)=O)CN(C(c2cnc3scnc3c2)=O)CC2CCCC12 N1(C(C)C)CCC(N2CCN(Cc3coc(C(N)=O)c3)CC2)CC1 CC1(NC(C2CC2C#N)=O)CCCCC1C(=O)NCCn1cncn1 C(=O)(C(C)(CNC(C1CC(F)(F)C1)=O)CC)NCC1CCCN(CC)C1 C1(C(=O)NCC(C(C)C)NC(c2cnn(C)c2Cl)=O)CCCCCCC1 C1(CNC(C2CC(CC)(CC)C2)=O)COCCN(C(c2cnc(C)cn2)=O)C1 C(=O)(CCC(C)(C)S(C)(=O)=O)N1CCC(CC)C1.C(=O)C(C)S(N)(=O)=O.N c1(N(C2CC3CNC2C3)C(c2cc(C(=O)OC)n(C)n2)=O)cccc(Br)c1Cl C1(C)(CNC(N2C(C)CC2)=O)CCCC1C C#CC1CCCCN1C(c1c(C)nn(CC(C)C)c1Cl)=O C(CC1=CCN(C(C)C(=O)NC)CC1)NC(c1cc(OC(CC)C)ncc1)=O C1(OCC(CCCC)CC)CCC12CCN(c1ccnc(NCC3CC3)n1)CC2 N1(C(C2CCC(C(=O)OC)C2)=O)CCCC(F)(C)C1.c1(C=O)coc(C)n1.N c1(CCC(=O)NC(CNC(C2CSCCS2)=O)C2CCC2)ccccc1F N(C(=NCCCOc1ccc(Cl)cc1)NCC1(CN(C)C)CCCC1)C1C(C)C1 Cc1cncc(C(N2CCN(C(C3(C)CCCCC3)=O)CC2C)=O)c1Cl C(=O)(CN=c1[nH]c(C)cs1)N1CC(C)CC(NC(C=CCOC)=O)C1 Cn1cc(C=CC(N2CCOCC2C)=O)nn1.C1(C=O)CC(=O)N(C(O)C)C1 C(=O)(C1=CC(O)C(NC(C2CC(=O)C2)=O)C1)NC1C(CC=C)CCC1.C C1(N(C(c2cc(CC)n(CCO)n2)=O)C)CCCN(C(=O)C(C)=C2CC2)CC1 c1(CCNC(CCCOC(COCC(C)C)=O)C)ccc(Br)cc1 C(CC1CCC1)(C(=O)NCCc1ccccn1)NC(=O)CCC1CCCO1 C1(CNC(C(C)CF)=O)(CO)CCN(C(=O)C(=O)NCC2CC2)CC1 C1(C(=O)Nc2c(C)sc(O)n2)CC12CCN(C(c1ccccc1)=O)C2.C1(O)CC1 C(=O)(CCS(=O)(=O)C1CCCC1)N.C1(C(N(CC(C)C)C)=O)C2CNC(=O)C12 C1(NC(c2n(CC)ccn2)=O)CCC2CCN(C(=O)C=CCN3CCC3)C1C2 C1(NC(CCCCC(=O)NC)=O)CCCC2CN(c3nc(Cl)ncc3OC)CC12 c1(C(N(CCC(C)NC(C2CC2C)=O)C)=O)c[nH]cc1-c1ccc(Cl)s1 N1(C(CCC(C)C)=O)CCN(C(C2OCCOC2(C)C)=O)C(c2cnn(C)c2)C1 C1(O)(C(=O)NCc2c(C(=O)NCCc3cc(C)on3)scc2)CCSCC1 N1(C(c2ccc(NC(=O)C3CC3)cc2)=O)CC23CCCC2(C1)C(=O)NC3=O Cn1ncc2c(C(=O)NC3CN(C(C4CC5CCC5C4)=O)C(C)(C)C3)ncnc12 CCCC(C(=O)N1CCN(C(=O)C(C)CCCOC)C2(CC2)C1)C(C)C C1(OC)CC2C1CCN2C(C1(C)CC(O)CN1C(c1nccc(C)c1F)=O)=O c1(CC)cc(C(=O)NCc2ccsc2C(N2CCCC2CO)=O)c(C)o1 c1cc(-c2ccco2)n(C)n1.C(=O)(C(C)CNO)OCCOC C(=O)(CN=c1nc(N2Cc3c[nH]nc3C2)c2cnn(C)c2[nH]1)NC(C)C C1(NC(CCCOC)=O)CCCCC1NC(C1CC1c1ccsc1)=O Cc1[nH]c(C)c(C(=O)NCC(F)CNC(c2scnc2C(F)(F)F)=O)c1C C1(C=O)CC(F)(F)CCC1(C)C.c1(C(C)=O)c[nH]nc1C(=O)NC.C1CCC1 c1(OCC)nccc(C)c1C(=O)NCC1CCCCN1C(=O)CCC(C)C.O C1(NC(C2CCc3nnnn3C2)=O)CC2CC1CN(C(=O)C(O)C(F)(F)F)C2 n1(CC)ncc2c(O)nc(N(C(C)C)Cc3cnn[nH]3)nc12 C(=O)(CC1=CCN(C(c2cccc(F)c2)=O)CC1)NC(CC)C(C)CN(C)C C1(CN(C(C=NOC)=O)C)CC(F)CN1C(c1cc(C)ns1)=O N1(C(c2ncn(C(C)(C)C)n2)=O)CC=CCC1.c1(C=O)ncn(C(C)(C)C)n1.N c1(CN2CCCN(CCN)CC2)c[nH]c2cnc(Cl)cc12 C1(C(=O)NCc2ccc(C)nn2)CCCN(C(c2n[nH]c(=N)[nH]2)=O)CC1 n1(CC)nc(C(=O)NCCN(C)C(C2CC(C)N(c3ccccc3)C2)=O)cc1O C#CCC(CC(=O)NC1CCN(C(=O)C(C)OCC2CCCCC2)C1)OC C1(C=O)CNC(=O)CC1C.C(=O)(CCC(=O)NCC1COC(C)C1)NCC Cc1cc(C=O)cc(O)n1.C1(CC(=O)N(CC)C2CC2)C=CS(=O)(=O)C1 S=c1n(CCN2CCSCCC2c2ccccc2)nc2ccccn12 C1(CN(C)C(C2C3CN(C(=O)OC(C)(C)C)CC23)=O)CN2CCCC1C2 c1(CC)ccc2c(Cl)c(C(=O)NCC3CC3)sc2c1.C(=O)C(C)N(C)C.N C1(C=O)CC(=O)CN1C(C1CCOC1C1CC1)=O.C=CCCC1(C)CC1.N C1(C(C(=O)NC(C)COC(F)(F)F)NC(C=C(CCC)C)=O)CCCCC1 C1(SC)CN(C(=O)C=Cc2cccnc2)CC1NC(C1CC12CC2)=O NS(=O)(=O)c1cc(C(N2CC=CC2CNC(=O)CCCn2cccn2)=O)co1 C1(OC)CCC(C(=O)NC2CC(NC(=O)CC3CCCC3C)C2)C1 c1(C(N(C(C)C(=O)NCCC2CCC(=O)N2)CCC)=O)ccn(C)c1C c12ccc3[nH]c(cc3n1)C(=O)NCC(=O)N2.N1(CC)CCC(CO)CC1 c1(C(=O)NCC(C)N(C)C(C2CCN(C)C2=O)=O)cccc(Cl)c1[N+](=O)[O-] N1(C(c2cnc(SC)nc2)=O)CC2(CCN2S(=O)(=O)c2cn[nH]c2)C1 c1(CC(C)NC(=O)CNC(=O)CNC(C2CC2(Cl)Cl)=O)nc[nH]n1 N1(C(COCC=C)=O)C(C(=O)NC2CC2c2ccnn2C)CCC12CC2 c1(C(N2CC3C(NC(C4OCCN(C)C4=O)=O)(C3)C2)=O)ccnc2ncnn12 S(=O)(=O)(c1nc(N2CC(C)OC(C)C2)ccc1Br)NCC1(COC)CCCC1 C(=O)(C(C)C)OCC.C1(O)(C(C=O)F)CN(C(=O)CC2CSCCO2)C1.N C1(C(=O)NCC(CNC(CC(CC)CC)=O)OC)CCC2(CCOCC2)O1 C(c1c(Cl)c2ccccc2n1C)=CC(N1CC(C)OCC1)=O.C1CO1 c1(NC)nccc(=NCC(C2CCCCC2)NC(Cc2ccccc2)CO)[nH]1 Cc1nc(Br)ccc1C(N1CC2CN(C(C3C=CC(=O)N=N3)=O)C2C1)=O N=c1ncnc(NCC2CCCN(C(=O)CC3COCCO3)C2)[nH]1 c1(C(C)NC(Cc2cc(C)sc2)=O)ccc(N2CCCC2=O)cc1 Cc1cc(C(F)(F)F)ccc1-c1cn(CC(N2CCOCC2CC2CC2)=O)nn1 C1Cc2nccn2C1.C1(C(=O)NC2C(C)(C(F)F)C2)C=CCN(C(=O)CO)C1.C CC1CCC(C)(C(N2CC(OCC(=O)NCCC(C3CC3)C3CC3)C2)=O)C1 C#CC1(F)CCN(C(c2cc(CNC(=O)CC3CCC(=O)N3C)ccn2)=O)CC1 N1(C(c2c(CC)nn(C)c2)=O)CCCCC(CNC(c2cc(N)ccc2Cl)=O)C1 C1(CC(=O)NC(c2ccc(OC)cc2)CNC(C(CC)O)=O)OCCC1(C)C c1(CN)cn(C2COCC2NC(=O)CC(c2cccs2)NC(N)=O)nn1 c1(C(=O)NC(CCNC(C2N(C(C)C)C(=O)CC2)=O)C)ccc2n[nH]cc2c1 C1(CC)C(NC(C2CC3(CCC3)C2)=O)CCCN1C(=O)CC(C)C1CC1 C(=O)(C(C)(C)CNC(C1CN(C)C1)=O)N(C(C)CO)C C1(C(=O)NCC(C)N(C)C(c2cccnc2NCCO)=O)CCC(F)CC1 Cc1nn(C)c(C)c1C(C)C(=O)NC(C)C(C)C.C(=O)(CC)N.CCC(C)C Cc1cc(CCCC(=O)N(C)CCNC(=O)C(C)Nc2ccccn2)c(C)s1 C(=O)(C1=CSCCO1)N1C(C)CC(CNC(c2ccccn2)=O)C1 CCC(C(=O)N1CC(NC(=O)CCC2CC(OC)C2)C(F)C1)C(F)(F)F N1(C(c2nc(C)cs2)C(=O)NCCCCCC)CCC2(COC(=O)N2C)C1 CC1(C)CCN(C(C2(F)CC2)=O)CC1NC(C1(C2CCCO2)CCOCC1)=O C1(C(=O)NCCC(c2cccs2)NC(c2cnn(C)n2)=O)CCC(C)(C)O1 c1(CNC(=O)NC(C)COC(F)(F)F)ccc(C#N)s1 C(C(=O)N1CC(O)(CC)C1)(C(C)C)SCC.c1(C=O)sccc1-n1ccnn1 C(C(C(=O)N1CC(C)C1)N(C)C)OC CCC(CC)(CC)C(=O)NC(CC(=O)N1CC(Cc2ccoc2)C1)C1CC1 C(CC(C)(C)C)(C(=O)N1CCC(C)(C)CC1C(=O)N)OC.c1cccc(C)c1.C N1(C(COCCC=C)=O)CCC(CNC(c2ccc(O)c(F)c2)=O)C(C)C1 C1(C(=O)NC(C(C)NC(Cc2cc(C)ns2)=O)C)CCC(=O)N1C(C)C N1(c2ccc(OCCCCN(C)C)c(I)c2)C(=O)C2CSCCN2C1=O C=CCCCC(=O)NC(C)(C)CCNC(C12CCC(C1)C2C(=O)O)=O CCCC(CCNCC1CC2CCCCC12)CCC CP(C)(=O)c1cccc(C(=O)NCCCN(C(=O)CC)CCO)c1.C1CC1.O CCC(C)C(CO)CN=c1nc(N2CCc3c[nH]nc3C2)c2ccc(C)cc2[nH]1 CC(C(=O)NC1CC(C)(CNC(c2nnc(O)cc2O)=O)C1)P(C)(C)=O C(CC(F)F)(C(=O)N1CC(C)(CF)C1)NC(CCc1cnc(C)o1)=O Cc1nc(C(C)C)ncc1C(N1CC(CNC(=O)C2=CCCC2C)C1)=O N1(C(C2CC(=O)NC2)=O)CCCCC1CCC(N1CCC(O)CC1)=O c1(C2N(C(C3NCCC3c3ccccc3)=O)CCC2)ccc(Cl)c(Br)c1 CCS(=O)(=O)CC(=O)N1CCN(C(c2ccnn2C)=O)C(Cc2ccccc2)C1 C1(N(C(C2C(CC)OCC2)=O)C)CCCCN(C(=O)CCP(C)(C)=O)C1 c1(C(N2C(CC)C(NC(C3CC34CC4)=O)CC2)=O)cc2[nH]ccc2s1 N1(C(CC=CCC)=O)CC(F)CC1CN(C)C(c1cccc(SCC)n1)=O N1(C(C(C)OCC)=O)CCC2CN(C(=O)CCc3nnc(C(F)F)o3)CC2C1 c1(C=O)cn(C2CC2)nc1C(F)(F)F.CC1(C)CC1(O)C(N1CCC1)=O.C C1(CC(N2CCC(COC)(NC(c3cnc[nH]3)=O)C2)=O)CN2CCC1CC2.S C1(C(=O)OCC)CCCCN1C(=O)Nc1ccc(N2CC(O)C2)cc1 CN(C1CCc2c(Cl)cccc21)C(C1C2CCC(F)(F)C12)C(=O)NCCOF CC1(C)CC(CNC(C2CCC(F)C2)=O)N(C(=O)CCn2cncn2)C1 N1(C(c2c[nH]nc2C2CCCO2)=O)CCOCC1(CO)CO Cc1ccc(SCC(=O)NCC(C)NC(=O)CCc2nnc(C(C)C)o2)cc1 c1(C(N2CC=CC(NC(c3c(C)onc3)=O)C2)=O)ccc2ncsc2c1 N1(C(c2c(CC)cc(F)cc2)=O)CC2OCC(NC(=O)CC3CC(O)C3)C2C1 c1(CCC)ccc(CCCC(=O)NCC2CCN2C(c2snnc2C)=O)cc1 CC(CCC(C)(C)C)C(=O)N1CCC2CCN(C(c3csc(S)n3)=O)CC12 c1(OCC#C)ncccc1C(=O)NC1COCC1NC(=O)CCSCCC CCCC(C)(CCCNC(C12CC1COC2(C)C)=O)C1OCCO1 c1(OC)ccc(Br)c(CNC2CC2C(=O)NCc2cccc(Cl)c2Cl)c1 n1(CC(=O)OC)nccc1.C1(Cc2nnnn2C2CCCCC2)CC(C)(C)C1.N N1(C(c2ccc(C)s2)=O)CC(NC(c2ccc(C3CC3)s2)=O)C(C2CC2)C1 CC1CN(C(=O)CCCn2cc(C(C)(N)C3CCC3)nn2)CCCO1 c1(C(=O)NC(CN(C(C(C)N(CC)CC)=O)C)C)sncc1CO C1(OC)CC(O)CN(C(C23CC(NC(=O)C(C)(C)CO)(C2)C3)=O)C1 Cc1nn(CCO)cc1C(=O)OCC(=O)NC1CCC(C)CC1 C1(F)(CNC(CC(C)C2CC2)=O)CCC(NC(=O)COC(F)(F)F)C1 CCC(C)C(C(=O)NCCN1CC(CF)C1)N(C(=O)CC1CCC(C#N)C1)C c1(NC(c2ccc3n[nH]cc3c2)=O)ccc2c(c1)CN(C(=O)C1CC1)CC2 N1(C(Cn2c(C)ccn2)=O)CCC(C2CC2)C1C(=O)NCCC(F)(F)Cl C#Cc1cnn(C)c1C(=O)NC1(C(=O)NCCc2ccncc2C)CCN(C)C1 c1(OCC)ccc2[nH]c(C(=O)N(CC(C)NC(=O)CC(F)F)C)c(C)c2c1 C1(NC(C(C)OC)=O)CCC12CN(C(c1ccc(O)cc1Cl)=O)C2 N1(C(c2c(O)cc(OC)cc2Br)=O)CCCC12CCN(c1nccc(C)n1)CC2 C1(CNC(C(CC)(C)CC)=O)CCC2CN(C(=O)CC3(N(C)C)CC3)CC12 CC1Cc2ccccc2N1C(=O)CC1CC2(CCOCC2)CN1 c1(C(C(=O)NC)N(C)CCc2cccc(C#N)c2)oc2ccccc2c1C c1(C(=O)NC(CC)CN(C)C(C2CCCCO2)=O)ccc(Cl)c(O)c1N C1(NC(c2cc(C)sn2)=O)CCCCC1NC(c1cc(C2CCCCC2)on1)=O c1(CC)cncc(C(N2CC(N(C(=O)Cc3cncs3)C)C(F)C2)=O)c1 C=C(Br)CC(C)(C)C(=O)NC1CCN(C(C2CC2CC(C)(C)C)=O)C1 N#Cc1cc(CC(N2CC(F)(C(N3CCS(=O)CC3)=O)C2)=O)ccc1F N1(C(CC2C(C)CCC2)=O)CCCCC1CN(CCCCc1ccccc1)C N1(C(c2c(C)ocn2)=O)CC(NC(C2(C#N)CC23CCC3)=O)CC(C)C1 CCC(C)C(O)C(=O)NCc1nc(C2CCN(C(c3ccc(C)n3C)=O)CC2)n[nH]1 C(=O)(N=c1cc(C2CC2)n(C)[nH]1)C1(NC(C=Cc2cccc(C)c2)=O)CCSC1 c1(C(C2CCCC2)NC(=O)NC2CCN(S(C)(=O)=O)CC2)c(F)cccc1F C1(NC(C(c2ccccc2F)OC)=O)(CNC2CCCN2C(C)=O)CCCCC1 Cc1nc2c(N3CCC(C)(NC(c4cc(C(F)(F)F)on4)=O)CC3)ncnc2s1 C1(C(=O)NCC(c2ccc(C(=O)O)cc2)O)CC2CC3(CC3)CC2C1 C1(NC(C(C)(C)OCC)=O)COC2(CCN(C(c3cccnc3)=O)C2)C1 c1(C(=O)OCC(F)C2CCC2)ccc(OCc2ccccc2)cc1Cl C(=O)(CC(C)CC(=O)NC1CC(F)CN(C(=O)CCNC(=O)C)C1)OC.O C=C1CCC(C(=O)NCc2cccc(C(=O)N(C(C)CC(C)C)C)n2)CC1 c1(C(N2CCCC(NS(CC(=O)OCC)(=O)=O)CC2)=O)cc2ccccc2[nH]1 Cc1[nH]ccc1C(=O)N(CC(=O)NC(CN(C)C)CO)CCO O=C(CCc1cn(C2CC(Nc3cnccc3N3CCOCC3)C2)nn1)CCO C1(OC)CC2(C1)CC(C(=O)NC1(CO)CCN(C(=O)C(C)SC)C1)C2 C12(C(=O)NCC3CCN3C(=O)CCCCCc3ccccc3)CCCC(C1)OC2 C(c1cncc(O)c1)=CC(=O)NCCC1(O)CN(C(C(C(C)SC)O)=O)C1 N1(C(C)=O)CC2CCC(C(=O)N(C)CCNC(=O)Cc3ncccc3C)C2C1 C1(=O)CC(CC(C)C)CN1.C(F)(C(=O)NCCNC(C)=O)=CC.C c1(CCC)ccc(C(=O)NC(C)(C)CN(C)C(c2cc(Br)n[nH]2)=O)[nH]1 C1(C(=O)NCCCCC2C(C)C2)CCCCN(C(C2(C)COC2)=O)C1 c1(-c2cccc(NC(C)=O)c2)cc2ccc(CN(C3CCC(O)C3)C)cc2[nH]1 c1(OC)ccc(Br)cc1C1(NC(c2cc(C(C)(C)C)oc2C)=O)CC1 N1(C(CC(C)C(F)(F)F)=O)CCOC2(C1)CN(C(c1conc1C(C)(C)C)=O)C2 c1(C(=O)NC2CCCC(CNC(C3CCC(C)(C)O3)=O)C2)nc2cnccc2s1 CC(=O)C(C)CC(C)C(=O)NC(C)C(=O)NCCC1CCCC12CC2 CC(C)C(C(=O)NC1C2CN(C(=O)CS)CC12)c1ccn(C)n1.C1CCOC1=O c1(OCC)cc(C(=O)N)sn1.c1(CCC=O)ncccn1.C1(C=O)CC1.C c1(OCCC)cccnc1C(N1CCOC(CN(C)C(C2CC3CC2C3)=O)C1)=O c1(CCC(N2CCCC(N(C(C(C(C)C)F)=O)C)C2)=O)nc2ccccc2[nH]1 c1(CC(N2C(CNC(C(n3ncc(C)c3)C)=O)CCC2)=O)cc(C)sc1C c1(OC)c(Cl)ccc(C(N2CCC(NC(c3nc(C)c(C)s3)=O)C(O)C2)=O)c1N C1(C(N(C2CCN(C)C2)C)=O)(NC(=O)CN2CSCC2=O)CCC(C)(C)C1 CCCCCCC(CC)C(=O)N(C(C)CNC(c1cc(Cl)c[nH]1)=O)C C(=O)(C1=CC(C)(C)C1)NC(C(=O)NCC(CCC)C)CCF N1(C(C23C(C)(C)C(CC2)CC3)=O)CCCC2CN(C(=O)COC(F)(F)F)CCC12 C1(C)(C(=O)NC(c2occ(C(N(CCCO)CCC)=O)n2)C)CCCCC1C c1(CN(CC(=O)O)C(C(CC(F)F)C2CCC2)=O)c[nH]nn1.c1ccccc1.C c1(OCC)cc2c(cc1CN1CC3CC3(CC)C1)OC(C)C2.C(C)(C)C C(=O)(C(C)(C)CC(=O)OC)NC1CN(C(CC(=O)NCC)=O)CC1(C)C Cc1sc(C(=O)N)cc1S(N)(=O)=O.C1CN(C(C2CC=CC2)=O)C(C)(C)C1.C c1(C(=O)NC2C(CNC(C3(CC=C)CC3)=O)C2)ccnn1C.C1CC1 c1(C(N2CCN(C(=O)CC3(O)CC3)C(CO)C2)=O)cc2ncccc2o1 c1(C(=O)NCC(CNC(Cc2ccc(C)o2)=O)O)cnc(S(C)(=O)=O)s1 C1(CCC)CCCN(C(=O)C=CC2CC2)C1.C1(C=O)CCC(=O)N(C2CC2)C1 C1(NC(CCC)=O)CN(C(=O)C(C)CC(=O)Nc2ccccc2)CC1S(C)(=O)=O CC(C)C(CCNC(c1ccccc1-c1ccncc1)=O)NC(c1cc[nH]n1)=O c1(C(=O)NCC=CCNC(C2CCC(C)C2)=O)cnc2ncccn12 c1(C(=O)NCCN(C(C)C)C(C2CCC3CC23)=O)ccnn1CC1CC1 c1(CN(C(C2ON=C(C)C2)=O)C)cnn2c1CN(C(C13CC(CO1)C3)=O)CC2 C1(CC)CC(C(N2CC(O)(CNC(=O)C(c3cccc(F)c3)C)C2)=O)CCO1 N1(C(CCCSC)=O)CCN(C(=O)C(F)C(C)C)C(c2ccccc2)C1 CCCCC(O)CC(=O)N1CC(C)(NC(=O)C=Cc2ncc(C)[nH]2)C1 c1(C(=O)NCC(c2ccccc2)NC(C2(CC#C)CC2)=O)cc(C)ccc1C CC1(C)CN(C(=O)C=Cc2ccc(Br)s2)C1CNC(=O)C1=CCCC1 c1(C(=O)NC2C3CN(Cc4c(F)cc(Cl)cc4Br)CC23)ccnc2c1OCO2 C12(C(N3CCCC(NC(c4cc(C)sc4C)=O)C3)=O)CCC(CC1F)C2 C1(C)(C=O)CCCS1(=O)=O.C1(O)(CC)CCN(C(c2cc(O)ncn2)=O)CC1.N n1(CC)ccc(C(=O)N(CCNC(C2CCO2)=O)CC2CCCC2)cc1=O c1ccc(C)cc1Cl.C1(OC)(CNC(c2c[nH]nc2F)=O)CN(C(=O)CC)C1.O c1(C(=O)NCC(C(=O)NCCC#C)C)nccc2[nH]ccc12 CCS(=O)(=O)CC(=O)N(C(CC(C)C)C(=O)NC1(CO)CCC(C)(C)C1)C C(CC(C)CCO)NC(C(C1(C)CC1)NC(c1nc(COC)oc1)=O)=O N1(CCNC(=O)CCc2ccncc2)CCN(C(=O)CC2CCCC2)CC1 C1(C)(NC(C(C(C)C)F)=O)CCN(C(=O)CN2CC=CC2)CC1 C(=O)(CC1COc2ccccc21)NC1CN(C(CCC=CC)=O)CC1C C1(C(C)C)(CC)CC1C=O.C1(N(C(=O)C)CC)CCCC1.C1(F)CC1 Cn1cnc2c(N3CC4CC(NC(C5(C)CCOCC5)=O)CC4C3)ncnc12 C1(CC(=O)NCC(COC)NC(C2OCCCO2)=O)CCCCC1 c1(C(N2CCC(CCOC)(NC(=O)C(O)C(C)C)C2)=O)c(C)cccc1Br C(CCC(O)C(=O)NCCC1(O)CCOC1)NC(c1c(OC)cccc1)=O C=CC(C)(O)C(=O)NCC(CC(C)C)NC(=O)C(F)(F)c1cnn(C)c1 N1(C(c2cnc(CC)s2)=O)CCC(CO)(CNC(c2nnc(Cl)cc2N)=O)CC1 c1(-c2nc(C3CCC(C)CC3)nn2CC(F)(F)F)ccc2n[nH]cc2n1 N1(C(COC)=O)CCC(O)(C2(NC(=O)C(=O)N)CC2)CC1.C1CC(F)(F)C1 c1(C(=O)NCCC(CCNC(COC)=O)O)ccc(-n2cccn2)cc1Cl CCS(=O)(=O)c1cccc(CC(=O)NCCNC(=O)CSC2CC2)c1 N1(C(C(C)N(C(C)=O)C)=O)CC(C)(OCC(=O)NC2(C(C)O)CC2)C1 C(=O)(C1=NOCC1)NC(C)C(CO)NC(=O)CCCCN1CCCC1 N1(C(COCCC)=O)CCN(C(C2(Oc3ccccc3)CC2)=O)CC1C(F)F C(CCN(C(=O)C)C)C(C)(C)C.c1(CC)cccc(OCC(=O)N)c1.CCF C=CCCC(F)(F)C(=O)N1CC2CCC2(CCNC(c2ccc(SC)s2)=O)C1 c1(OC(C2(c3cccs3)C(C)C2)=O)cc(F)c(F)cc1F C(C(CC(F)(F)F)NC(C1(c2cccc(OC(F)(F)F)c2)CC1)=O)NC(C)=O N1(C(Cc2c(CC)con2)=O)CCC(C)C1C.n1(CC(=O)N)c(C)csc1=O c1(C(N2CCCC(CNC(COCC(=C)C)=O)C2)=O)n[nH]c2c1CCCC2 C1(CNC(c2c(COC)cc[nH]2)=O)CCCC1O.C12(C=O)CCC(CC1)C2 c1(OC(C(=O)OC)CNC(=O)C(Cc2ccc(C)cc2)OC)ccc(Br)cc1 N1(C(C(C(C)C)O)=O)CC2CCC(C1)N2Cc1cc2n(n1)CCC2 c1(CC)c(C(=O)NC(C)CN(C(=O)CC2CCCN2C)CC)cnn1C C1(C2(C)CC2)CCCC1(C)O.N1(C2CCNC2=O)CCN(c2cccnn2)CC1 C(=O)(CCCCCN(C)C(C1CC2(C1)CC21CC1)=O)N1CCC(CN(C)C)C1 C#CCCC(C(=O)NCCC1COCCO1)NC(c1ccn(C)c1C)=O c1(NC(=O)NC2CC2CC2CC2)ccc2nccn2c1 Cc1cc(=O)oc2cc(NC(=O)CC3CN(C(c4cnc[nH]4)=O)C3)ccc12 Cc1cc(C)c(C(=O)NC2CC2NC(c2c[nH]c3ncccc23)=O)cc1Br Cc1cc(C(=O)NCC(CO)C(C)C)c(C)n1CC1CC1 c1(C(N2CC(CNC(Cc3cccc(OC)c3)=O)C2)=O)cnn2c1CCCC2C Cc1c(C(=O)N)ccn1C(C)C.C1C2CN(C(=O)C)CC12.c1cnn(C)c1.C C1(NC(c2c(C)c[nH]n2)=O)CCC12CCN(C(=O)CCC1CCC(C(N)=O)O1)CC2 n1(CC(N2CCC(C)C2)=O)ncn2nccc2c1=O.CC(C)COCC(=O)N.C C1(OC)CC(C(=O)NC2C=CCCCC2)N(C(c2ccc(C(N)=O)o2)=O)C1 c1(C(=O)NC2C(NC(CC(=C)C)=O)CCCC2)cc(C(F)(F)F)ncc1Cl n1(CCC=C)c(N2CCOC(COC(C)(C)C)C2)nnc1-c1nnc(C)s1 C1(C(=O)NC(C#C)CC2CCCC2)CN(C(C)=O)CC12CC2 C1(CNC(CC(CCC)C)=O)CC2(CCC2)CN1C(c1cnc(C(F)F)nc1)=O N1(C(C(C(C)C)NC(=O)CC(C)F)=O)CC2CC(O)CC1C2 C1(OC)(C)CCN(C(C2CCNC(=O)C2)=O)C1.c1(C=O)ccoc1C1CC1.N c1(C=O)cc(C(=O)NC(C)C)[nH]c1C.C(=O)CC=C(C)C.C1CC1.C C(C(CCCC)NC(C1CCCN1C1CCCC1)=O)NC(C(CC)=CC)=O CCC(O)C(F)(F)C(=O)NCC1CCCC(CNC(=O)C)C1.c1ccncc1 C1(C(N2CCC(C)(NC(c3cc(C)c(O)nn3)=O)CC2)=O)CCCC12OCCO2 c1(CCC(=O)NC2(C)CCC2)ccc(F)c(F)c1.c1(C=O)cc(O)nc(Cl)c1.N C(C(COC)C(=O)NOC1CC1)NC(c1ccc(CC)[nH]1)=O n1(CCN(C)C(c2sccc2CC#N)=O)cc(CCC2COC(=O)O2)nn1 c1(C(C)(C)C)cnc(C(C(=O)NCC2CC2)N2CCC2c2cccc(F)c2)cn1 C1(CN(CCN(C(=O)Cc2ccccc2F)C(C)C)C)CNC(=O)C(C)(C)C1 C(=O)(CCC(C(=O)OCC1C(C)CCC1)NC(N)=O)OC(C)(C)C c1(CCC=O)c(C)n[nH]c1C.C1(C(N(C(C)C)CC)=O)CC1(C)C(=O)O c1(C(N2C(CNC(C(CC)CO)=O)CC(F)(F)C2)=O)ccc2c(c1)NC(=O)C2 C1(C(=O)NCCCN(c2nnc(CC)c(CC)n2)CC)CN2CCN1C(C)C2 N1(C(c2nc(C(C)C)sc2)=O)CC2(CCN(C(=O)C=CC3CCC3)CC2)CC1C Cc1ccc(N)cc1C(N1CCCC(C(C)NC(c2cnc(C)nc2)=O)C1)=O N1(C(=O)OCC)CCC(NC(=NCc2cccc(C)c2)NC2COC(C)C2)CC1 C(=O)(C(C)C(O)C(C)C)NC(CC)CNC(c1cccc(C2CC2)c1Cl)=O C1(NC(C(c2cn(C)nc2)(C)C)=O)CC(F)(F)CC1NC(c1cncs1)=O C(=O)(CCCCC(C)CC)N1C(CNC(c2c(CCC)n[nH]c2)=O)CCCC1 C(=O)(C1=CCN(C(=O)Cc2cccc(O)c2)CC1)N1C(CSC)CCC1 C1(NC(C(n2ccc(C)n2)C)=O)CCC12CN(C(C1(c3cc(C)no3)CC1)=O)C2 c1(CN2CC(C(=O)Nc3ccc(C)cn3)OCC2)ccc(F)c2ccoc12 Cc1nc2c([nH]1)CC(C(=O)NCCCNC(=O)C(C)Cc1cccc(F)c1)CC2 CCCCCC(O)CC(=O)N1CCC=C(C(=O)NC(C)C(C)C(=O)OC)C1 c1(C(C)(C)C)cc(C(=O)O)on1.c12ocnc1CNC2 O=C1NC(C(N2CC3C(C)C3C2)=O)CC1F.c1(C(=O)N)c[nH]nc1C(F)(F)F c1(CN2C(C)(C(=O)NCc3c(C)cccn3)CC2)cccc(O)c1C Cc1cc(=NC(=O)C=CCN(C)C)[nH]n1CCC#N C12(C(=O)NCC(CCNC(c3ccc(O)nc3)=O)O)CCC(CF)(CC1)CC2 C1(C(N2CCC(NC(CNS(N(C)C)(=O)=O)=O)CC2)=O)CC2OC1C1CC21 C(=O)(C(O)P(C)(C)=O)N(C1CN(C(=O)C=CC2CCCC2)CC12CC2)C c1(C(N2C(CC)CN(C(=O)CC3COCCO3)CC2)=O)nccc2ccccc12 CC12CCC(C)(O1)C(C(N1CCCC1CCC(=O)O)=O)C2 c1(C(=O)OC)cc(CNc2cccc(CN3CCOCC3C(N)=O)n2)ccc1O C(CNC(=O)C1=NOCC1)(C(C)(C)C)NC(Cc1nnc(C)s1)=O C(=O)(CCCCC(C)CC)NC(CCC)C(N1CCn2cncc2C1)=O C1(C(=O)NC2(CC)CCCCC2)CCCCC1(C)NC(C1CC(CC)(C)C1)=O C1(C(N(CC(N2CC(CC(C#C)C)C2)=O)C(C)C)=O)CC=CCC1 c1(C(N2CC(OC)(CNC(c3c[nH]nc3C3CCOC3)=O)C2)=O)nccnc1C N1(C(COc2cn(C)nc2)=O)CCCC(O)C1.C1(C(=O)N)(CCN(C)C)CC1 c1(NC(C2C=CC(NC(C(CC)C)=O)C2)=O)cc(C)ccc1C N1(C(C(C)NC=O)=O)CC(N=[N+]=[N-])CC1C(N1CCC2CCC(C2)C1)=O c1(C(=O)NCC(CNC(C(=Cc2cccs2)C)=O)O)ccc(C)c(O)n1 Cc1nc(NCC2CCC(=O)NC2C)cc(NCC2CCN(C3CCC3)CC2)n1 N1(C(C(CC)c2ccccc2)=O)CCN(C(c2cscc2C#N)=O)CC1CF c1(C=O)ccnc(Cl)c1N.C1(C)(C=O)CCC1.C(CC)N(C(=O)C)C(C)C.N N1(C(CCC(=O)NCCC)=O)C2CC=C(C(=O)N3C4CCC(C4)C3CO)C1CC2 Cc1cccc2c(C(=O)NC3CN(C(C4CC=CC4)=O)CC3C)c[nH]c12 N#Cc1c(NC(C2CC(F)CN(C(c3cscn3)=O)C2)=O)cc(F)cc1F N=C(NOCC(C1CCOCC1)N1CCCC1)c1ccccn1 C1(C(=O)NCCSC)(CC)CCCN1C(c1ncsc1C)=O C(=O)(CCCCCC#N)N(CCNC(c1cc(OC)cc(CO)c1)=O)CC C(=O)(C#Cc1ccc(Cl)cc1)NC1C2CN(C(Cc3c(C)ccc(Br)c3)=O)CC21 CCCCC(CCC)N=c1nc(N(CC(C(C)C)OC)C)c2c(ncn2CC)[nH]1 O=S(=O)(CCN=c1[nH]c(=NCC2CCC(F)C2)c2ncccc2[nH]1)CC(F)(F)F c1(C(=O)NCC2(CNC(C(CC)(C)O)=O)CCCC2)ccc(Br)cc1N C(=O)(C1(C)CCOc2ccccc21)N1CC(N(C(=O)CCC2CCOC2)C)C1 c1(C(N(CC(CN(C(C(C(C)C)SC)=O)C)O)C)=O)cc(C(C)C)nc(O)c1 C1(C(=O)NC(C2(C(=O)NCCC3C=CCC3)CC2)C)CCCC(=O)C1 N1(C(c2cc(C)cc(Cl)n2)=O)CCCC2CN(C(C3COC(=O)O3)=O)CCC12 C(=O)(CCS(N)(=O)=O)N.CC(C)CCNC(C1C(c2ccccc2)C1(C)C)=O c1(N)cccc(N)c1C.c1(C(=O)NC(CC)(C)C)csc(CNC(C)C)c1 CCCCCC(C(=O)NC1CC1C)C(C)C.n1(CC(=O)N)c(C)cc(C)nc1=O Cc1cc(C)cc(S(=O)(=O)NC2CCC3(CC2)CN(N2CC4(CCC4)C2CO)C3)c1 C1(C(=O)NC(CNC(C2(CC=C)CCOC2)=O)CC)CC(F)(F)C1(C)C C1(C(N(CC(C)C)C)=O)CC(NC(=O)CSCC(F)F)C1(C)C c1(C(N2C(C(=O)NCCOCC)C3CC3C2)=O)cc(O)cc(=O)o1 c1(CC(N2C(C)CC(NC(C(C(C)C)N(C)C)=O)C2)=O)cnc2n1CCCC2C C12(NC(C=CC(C)C)=O)CC(C)(C1)OC2C.c1(CC=O)cc(Cl)no1.N C1(CC(N2C(C)CC(CNC(C3(CF)CCC3)=O)C2)=O)CC2CCC1CC2 N1(C(C2COC2)=O)CC2(C1)CN(C(=O)C(C)(O)C1CCC1)CC2C(=O)O.C N1(C(C2(OC)CCSC2)=O)CC2CCS(=O)(=O)C2C1.C1(C=O)CC2(CCC2)C1 Cc1cc(N2CCC(C(C)(C)NC(=O)C(O)C3CC3)CC2)c([N+](=O)[O-])c(C)n1 C(CCCC(=O)N(C)Cc1nncs1)N(C(C(CSC)O)=O)C c1(C(N(CCN(C(c2cnn(C)c2)=O)C(C)C)C)=O)c(C#N)cnn1C.C CCC(C)(C)C(O)C(=O)NC(CNC(=O)C(F)OC(F)(F)F)CC(C)C C=CCCCCC(C(=O)NC(C)CC)N(C(C)CCCCO)C Cc1nnc2n1CCN(C(C1CC(F)CN(C(=O)C(F)F)C1)=O)C2 CC1(C)CN(C(c2n[nH]cc2[N+](=O)[O-])=O)CCN(C(C2CN3CCCC2C3)=O)C1 C=C(F)C1(CC(=O)NCCC)CCC1.C1(=O)CCC(=O)NC(C)C2CCN1C2 CCCCCC(O)C(=O)NCCOCCC(=O)NC(C)CCc1cn[nH]c1 C1(CNC(c2c(C)cc(F)cc2)=O)C2CCCC1N(C(c1cccn1C)=O)C2 C(=O)(C(F)C(F)(F)C(F)(F)F)N1CCC1.c12cnn(c1)Cc1cn-2nn1.CCC C1OCCC1(C)C.C(C)(C)(C(c1nnn[nH]1)NC)N(CC)CC.c1ccco1 C(CCC(C)C)(C(=O)NCC(C)(C)CC)NC(c1n(CCC)ncc1)=O C1(NC(c2c(CC)c[nH]c2)=O)CC2CC1N(C(=O)CCc1cocn1)C2 CC#CCCCC(=O)N1CC(N(C(=O)C(CC)n2nccc2C)C)C(C)(C)C1 c1(CCC(=O)N(CC(C)(C)NC(C2(Cl)CC2(F)F)=O)C)nc2cnccc2[nH]1 C1(N(C(C23CCC(OC)C2C3)=O)C)CN(C(=O)Cc2ccoc2)CCC1O N(C(=NCCOC)NCc1ccccc1Cl)C(C1CC1)C.C=CCOCC=C N1(C(CSC2CC(=O)C2)=O)CCC(n2cc(-c3cscn3)nn2)C1 c1(C(N(CC(C)NC(C(CC)COC)=O)C)=O)ccc2c(c1)NC(=O)CS2 C12(CNC(C(C)=CC3CC3)=O)CC(CO1)N(C(=O)Cn1ncc(Cl)c1C)C2 N1(C(C2(C)CC(C)C2)=O)CCCOC(CNC(=O)Cn2cc(Cl)cn2)C1 C1(C(=O)NCCC2CC(NC(C3(N(C)C)CC3)=O)C2)CCc2ccccc2O1 CCCC(CC(C)C)C(=O)NCC1CCC1NC(c1nnn2ccccc12)=O N1(C(C2(C)CSC2)=O)CC2(CCOCC2)CC1CNC(c1cncs1)=O CC1(C)COc2c(C(=O)OCCC)cnn2C1.C(C)(C)(C)NC=O.C1CO1 CS(=O)(=O)C1CC(C(N2CCCC(CNC(C3C=CCC3)=O)C2)=O)C1 C(=O)(CC(O)C(C)CC)NCCCCNC(c1cncc(COC)c1)=O N1(C(COC)=O)CCN(C(C2(c3ccc(OC)cc3)CCCC2C)=O)CC1 Cc1nn(C(C)(C)C)cc1C(=O)NC1CC(C)N(C(c2cnc(Cl)s2)=O)C1 c1(C=O)cc(=O)cc(Cl)[nH]1.C1(CNC(=O)CC2CC(F)C2)CC12CCC2.C c1(N(C)Cc2cccnc2)nc2ccccc2nc1N1CC2C(C(N)=O)C2C1 N1(C(C(CC)N(C)C)=O)CC2CC3CC2C1C3NC(=O)COC Cc1cncnc1N1CCCN(CCS(C)(=O)=O)CC1.C(C)(C)C(C)C.CCN.N N1(C(c2cccs2)=O)CC(C(N2CCC(C)(C(N)=O)C2)=O)C(C(C)C)C1.CC N1(C(C2C(C)N(C(c3cnc(=N)[nH]c3)=O)CC2)=O)CCC2CCCC2CC1 C(=O)(CC(C)P(C)(C)=O)NC1CCN(C(c2c(C)cccc2)=O)C1(C)C CC1(C)COCC(CC(=O)N)O1.C1CC2(C1)CCC2.C1(C(C)(C)O)(C=O)CC1 C1(C(=O)NC2(C(=O)NC3CC(=O)NC3=O)CCC2)CC2(CCCO2)C1 C(CCC(CCC)NC(c1ccc(-c2cnn(C)c2)o1)=O)NC(C(CC#C)O)=O C(CCCCNC(C1CCCSC1)=O)NC(C1(CC=C)CC1)=O c1(NC(C2(C)NC(=O)NC2=O)CC)ccc(S(=O)(=O)N2CCCC(F)C2)c(Br)c1 C(=O)(CC(O)CNC(c1ccc(CO)cc1)=O)NCC(C1CCCC1)OC N1(C(CSC(C)(C)C)=O)CC2CCC1CN2C(=O)C(=O)Cc1ccc(F)cc1 S(=O)(=O)(c1cnn2c1OCC(C)(C)C2)NC(c1nnc(C)s1)C c1(CC)[nH]nc(Cl)c1C(=O)NCC1CCCCC1NC(c1csnc1Cl)=O Nc1ccc(C2CC2)cc1C(N1CC(O)C(O)C1CNC(c1ccsc1)=O)=O c1(C(N2CCC(CNC(c3cccnn3)=O)C23CC3)=O)ncnc2sccc12 C1(CC(=O)N(C)CCNC(=O)C=Cc2cccs2)C(C)(C)C1(C)C c1(C(N2CC3CN(Cc4ccc(F)nc4)C3C2)=O)ncnc2ccsc12 N1(C(c2cc(C)cc(N)c2)=O)CCCC2(C1)CN(C(C1CC=CCC1)=O)CCO2 C1(C(=O)OCC)OCCNCC1N(C1CCNC1=O)C1CCSCC1 c1(C(N2CCN(C(C3C=CCCC3)=O)CC2CCO)=O)n[nH]c2c1CCCC2 C(=O)(CC1COc2cc(O)ccc21)NC(CNC(CC12CC(C)(OC1)C2)=O)(C)C N1(C(CCC(CC)NC(C2CC(SC)C2)=O)=O)CCC2CN(C)CCC12 c1(NC(CSCC(=O)Nc2ccc(F)cc2Br)=O)cccc([N+](=O)[O-])c1 c1(C(=O)NCc2cn(CC(=O)NC3COC(=O)C3)nn2)cc(F)cnc1O Cc1cc(N)cc(C(=O)NCC(CNC(c2cnc3[nH]ncc3c2)=O)CO)c1F C(=O)(C1CCc2c[nH]nc21)NC1C(C)CN(C(=O)CS(=O)(=O)CCO)CC1C O=C(CCS(=O)(=O)C1CCCC1)NC1CC(F)(C)C1.C1(C=O)CCC2(CC2)C1 c1(CC(=O)NC2CN(C(C=CC=CCC)=O)CC2C)cc(F)ccc1Br C(=O)(C1=CC(O)C(NC(C2CCCC(C#N)C2)=O)C1)NC(CCC=C)C(=O)OC C1(C(N(C)Cc2ccccc2Cl)=O)CCCN(c2ccc(Cl)cc2)C1=O c1(C(=O)NCC(C)N(C(C(C)C2CCC2)=O)C)sc(N(C)C)nc1Cl n1(CC)nc(C)c(C(N2CC(C)C(O)C2)=O)c1Cl.O(C(F)(F)F)CC(=O)N C(=O)(C1=Cc2cc(F)ccc2OC1)NC(CNC(CCCCCCCC)=O)CC c1(CN2CC3(CC(C(=O)NCc4cscn4)C3)C2)cccc2c1CCC2 C1(CNC(c2cnc(CCCC)s2)=O)CN(C(C2CC(O)C2)=O)CC1O C(=O)(C1=CS(=O)(=O)CCC1)NC1C(CC)COC1 c1(C(=O)N)cccc2c(C)cccc12.C1(C(=O)NC(C)C2CC2)(OC)CCC1 C#Cc1cc(C#N)cc(C)c1NC(C1COCCC1c1ccccc1)=O N1(CC(=O)N(CC(C)N(C(=O)Cc2cnc[nH]2)C)C)CC(=O)NC1=O C(=O)(C(CCC)OC)NCC1(C(=O)NC2CCCC2O)CC(=C)C1 N1C(N2CCC(c3cccnc3C(=O)OC(C)(C)C)C2)=NCC2CC12.CCC c1(CC)noc(C)c1NC(C1CC(=O)CN1C(c1cn[nH]c1)=O)=O C1(c2ccccc2)(NC(CC(CC)SC)=O)CCN(C(=O)CN(C)CCO)CC1 C1(OC)CCN(Cc2cn(C3CCCN(C(c4cnc(Cl)[nH]4)=O)C3)nn2)CC1 CC1(C)CCN(C(c2cnsc2)=O)C(C(=O)NC23CCC(CC2)CC3)C1 CCCCCCCCNC(=O)C(C1CC1)NC(=O)Cc1cncn1C CC(C)CC(c1nnnn1CC1CCCO1)NCCc1ccno1 C1(CC)COCCN1C(=O)C(c1ccco1)NC(=O)COCCN(C)C N1(C(c2ccc(C)n2C)=O)CCN(C(c2ccnn2CC2CCC2)=O)C(C)C1 C=CC(CC)CC(=O)NC1(C)CCN(C(=O)C(C)=CC)C1 CC1CC(NC(C2CC(CC3CC3)C2)=O)CN1C(c1ccn(C2CC2)n1)=O CC1(C)COC(CC(=O)NCCC2CC2)C1.c1(C=O)ccccc1C(F)(F)F N1(C(C(N2C(CC)CCC2)=O)=O)CCN(C(=O)CCN(C)CC)CC(C)(C)C1 CC1CN(C)CCC1NC(c1occc1-c1cccc(Br)c1)=O c1(CC(C(=O)NCC(n2cc(C3CC3C)nn2)C)NC=O)ccc(Cl)c(Cl)c1 N1(C(CCC(=O)NC)=O)CCC(CNC(C23CC(C2)C(C)O3)=O)CC1C N1(C(C2C(CCC)C2)=O)CCC2(CC1)CCN(C(C1(OC)CCSCC1)=O)C2 N1(C(c2cc(O)nc(C3CCOCC3)n2)=O)CC2CCN(C(C3CCO3)=O)C2C1 c1(CC=C)cccc(C(N2CCC(N(CCO)C(c3cccc(O)n3)=O)C2)=O)c1 C(=O)(C1=NOC(C)(C)C1)N(C1CN(C(C2CC(C)(F)C2)=O)CCC1O)C c1(CC)ncc(Cl)c(C(=O)NCC(C)N(C(c2scnc2Cl)=O)CC)n1 CS(=O)(=O)c1csc(C(=O)NC2CCN(CC)CC2)c1.C1(C(=O)N)CCCC1O C1(C(N(C2CCN(C(=O)C3=NOCC3)C2)CC)=O)CC(C)C(C(=O)OC)O1 N1(C(c2c(N)ccc(C)c2)=O)CC2CCC(C)(C2)C1.C(=O)(C(C)P(C)(C)=O)N C1(C(N2CCC(NC(C(C)(C)c3cccs3)=O)C2)=O)CCOC2(CCC2)C1 c1(C(=O)NCC(C)CNC(C2CC3(CCC3)CO2)=O)c(O)nnc2c1CCCC2 C1(NC(C2(C)N(C(CSCC=C)=O)CCC2)=O)CCN(C)C(=O)C1 C(CCC(C)C(=O)NCCC1CCN(C(=O)CCSC)C1)OC c1(C(=O)OC)cc(C(N2CCC(C)C2)=O)cc(O)c1.c1(C=O)ncn(C)c1C.N C(=O)(CC(C)(C)NC(C1CC12CC2)=O)NCC(CCC)C c1(OC)c(Br)cc(F)c(F)c1NC(=O)NCc1cccc(CC(F)(F)F)c1 N1(C(C)=O)CCOC2(CCCN(C(=O)C3CCc4ccc(O)nc43)C2)C1 C(=O)(CC(C)(C)N(C(=O)C(O)C1CCC1)C)N(C(CC)CSC)C C1(CCC(=O)OC)CCN(CC(C(F)(F)F)C2CC2)CC1 C(=O)(C1CNC(=O)c2ccnn21)NC(CNC(CCC1(C)CC1)=O)(C)C1CC1 c1(C(N(CCCNC(C2CCC(OC)C2)=O)C)=O)cnc2onc(C3CC3)c2c1 N1(C(CN2C(C)CC2)=O)CCCN(C(C23COC(CCO2)C3)=O)C(C)C1 C(=O)(CCC(N)C(N)=O)N1CC(F)CC(NC(C2(c3ccc(C)cc3)CC2)=O)C1 CC1CN(C(=O)CC2CCCSC2)CC1(C)C(=O)NCC1CCCN1C C(=O)(C(CCC)C(=O)OC)N1C2CC(NC(CCCC)=O)C2CC1 CC1(NC(c2csnc2Br)=O)CC(NC(=O)CNC(c2ccccc2)=O)C1 c1(C(=O)NC2C(NC(C(=Cc3ccco3)C)=O)CCC2)cncc(C)c1 C(=O)(C1=CCc2ccccc21)NCCCCN(C(=O)C(O)C(C)(C)C)C C(C(CC(C)C)C(=O)NC1CC1(C)C(C)C)NC(C(COC)(C)OC)=O c1(C(N2CCC(C(=O)NCCC(CC)(F)F)(CO)C2)=O)ccc(C)c(F)c1 c1(CC(=O)N(CC(C)NC(C2CC3(C2)CC3(F)F)=O)C)ccc(F)c(Cl)c1 c1(C(=O)NCCCC(C)(C)NC(C(CC)C#N)=O)ccc(S(=O)(=O)NC)o1 C1(CC)CCCCCN1C(c1cc2sccc2s1)C(=O)NC1CCC1 C#CCCCCC(C(=O)NCC1CCCO1)N(C)Cc1cc(Br)cs1 Cc1ccc(C(N2C(C(=O)N(CCCO)C(C)C)CCC23CC3)=O)c(C)c1 c1(C(=O)OC)oc(C(=O)NC(C)C2CC2)cc1C.N1(C(C=O)C)CCOCC1 C1(C(=O)NC2CC(CCNC(C(c3cnn(C)c3)C)=O)C2)COCC(C)(C)O1 N1(C(c2ccc(C)c(O)c2)=O)CC2CCC1CN2C(C1CCc2nncn2C1)=O C1(NC(CC2(OC)CCC2)=O)C2CC3C1C3C2C(=O)NC1CCOC1 Cc1nc(C=CC(=O)NC(C)CN(C(=O)Cc2ccccc2C)C)cs1 C1(C2C(c3nc(-c4cn(C)nc4)on3)CCO2)CCN(C2CCCC2)CC1 C1(CC#C)(C(=O)NCC(O)CN(C(=O)CCn2ccnc2C)C)CC=CCC1 c1(OC)ccc(S(=O)(=O)NOC2CCS(=O)(=O)C2)cc1[N+](=O)[O-] N1(C(C(C=C)(C)O)=O)CCCC(N(C(=O)Cc2cc(C(F)(F)F)nn2C)C)CC1 c1(C(=O)NC2(CNC(C=CC)=O)COC2)ccc(-c2ccccc2)nc1C c1(C(N2C(C(=O)NCc3n(CC)ccn3)C(C)OCC2)=O)cc2ncccc2[nH]1 N1(C(C=CC(=O)N(C)C)=O)CC2CC(NC(C3CCCCO3)=O)CC2C1 CC1(C2CCN(C(=O)CC3CC(C)(C)CN3C(c3ccc(Cl)cn3)=O)C2)CC1 c1(CC(C(=O)N(CCC)C2CC2)O)ccc(Cl)cc1.CCC=O.C(C)(C)C.N C1(C(N2CCN(CCN(C(Cc3nc(C)[nH]n3)=O)C)CC2)=O)CC(=O)NC(C)C1 c1(C(N(CCCCNC(=O)C(F)(F)C(F)F)C)=O)n[nH]c2ccc([N+](=O)[O-])cc12 c1(C(=O)NCC(C)CNC(=O)CCCCc2ccccc2)cc(Cl)c(F)c(Cl)c1 C(C(C(=O)NCCC(=O)N)C(C)(C)C)NC(C1(CC)CCCO1)=O.C(C)C C1(C)(OC)CC(NC(=O)CCOCCCNC(C2CCCOC2)=O)C1(C)C C(CCCCC(=O)N1CCC(NC(C2(c3ccc(F)cc3)CC2)=O)C1C)SC N12CCc3c(n[nH]c3C1)C2.c12ccc(-c3cccc(Cl)c3Cl)c-1c2.CO N1(C(C(C)c2cccs2)=O)CC(NC(C2CCC(F)(F)C2)=O)C(C)(C)C1 N1(C(C2N(C(CN(C(COC)=O)C)=O)CCC2)=O)CCCC(C)(F)C1 Cc1cc(C)c(NC(=O)OC(C)(C)C)cc1C.C123CC1CCCN2C3 c1(-c2ccc(CN(C3CCOC3)C)s2)n[nH]c2ccccc12 N1(C(CC(=O)OC)=O)CCCC2(CCCN2C(c2ccc(O)nc2)=O)C1 N1(C(C(C)NC(C)=O)=O)CC2CC1C2.c1(C(C=O)(C)C)ccc(C(C)C)cc1 Cc1cc(C(=O)N(C(C)CNC(C2(C)CCCNC2=O)=O)C)c2ncccc2c1 C1(N(C(c2cc(C(N)=O)no2)=O)CC)CCCNC1.c1cccc(N(C)C)n1.C c1(C(C)C)c[nH]nc1CNCC(C)(CO)NC(=O)OC(C)(C)C CC(C(C)C(=O)N1CCCc2nccn21)NC(=O)CCNC(=O)CO c1(C(N2CC(NC(c3cc(C)sc3C)=O)C3C2C3)=O)ccc(OC(F)F)cc1Cl C1(C(N2CC(CCNC(C(C)NS(CC)(=O)=O)=O)C2)=O)CCOCC12CCC2 CC1CCN(C(C2OCC2(C)C)=O)CC1NC(=O)Cc1sc(O)nc1O C1(COC)CN(C(=O)C(=O)NCCCCCCN(C)C)CCO1 C(=O)(CC(C)(C)C(F)F)N1CCC(NC(C(Br)=C(C)C)=O)C1C(C)C C=CCC(C)C(=O)NCC#CCNC(=O)Cc1cccc(OCC2CC2)c1 C1(CC(=O)NCc2nc(C)sc2)C2CCC1CN(C(C1CCC(=O)NC1)=O)C2 C1(CC=C)(C(=O)NC(C)C(C)CCC)CCN(C(=O)C(c2ccccc2)F)CC1 CN=C(NC1CCN(Cc2ccccc2NC)C1)N1CCC(C(F)F)C1 C1(C(=O)OC)CN(C)C(=O)CN1C(C12COCC1C2(F)F)=O c1(CNC(=O)NC(C2CCCCO2)C(C)C)ccnn1CC(F)F C(C1CN(C(=O)CSSC)Cc2ccccc21)NC(c1ccc(OC)cn1)=O N#CC1(C(N2CCCCC2CNC(=O)Cc2ccc(F)cc2)=O)CCCOC1 CN1CC(=O)N2CC(NC(N3CCCC(C)(C)CC3)=O)CC2C1=O c1(CNc2ccc(C(=O)Nc3cn(C)nc3)nc2)cc2ccccc2cn1 C1(C(=O)NCCc2c(C)ocn2)C=CCCN1C(=O)CCC(N)=O c1(C(N(CC)CC)=O)ccc2c[nH]nc2n1.c1(C(C=O)N(C)C)ccccc1.N N1(C(c2c(C)cccn2)=O)CCN(C(C2(C)CCCCO2)=O)CC1C N1(C(C2C(OC)CNC2)=O)CCn2c(C3CCCC3)nnc2C1 C(=O)(NNc1cccc(N(C)C)n1)Nc1nc(C)cc(C(=O)OCC)n1 Cc1nn(C2CCOC2)cc1C(N1CC2CC2(NC(c2cc(CO)[nH]n2)=O)C1)=O c1(C(=O)N)cnc2cc(C)ccn12.N1(C(c2c(CC)onc2)=O)CC2C(C)C2C1 c1(C=O)ccc(Cl)c2c1OCCO2.c1(CC)nc[nH]c1C(=O)NC1CCC1C.N c1(C=O)cc(C(C)(C)C)n(C)n1.c1ccc(C(=O)N(C(C)C)C)s1.CO.C C(CC(C)(C)C(c1nnnn1-c1ccccc1C)NCC1SCCS1)OC C1(C(N2CC(C)N(c3cc(F)cc(F)c3)CC2)=O)C2CCC1(C)C2(C)C C1(C(N2CC(CC)(NC(C3C(C(=O)O)C3(C)C)=O)C2)=O)CC(C)CCO1 c1(C(N2CCC(NC(C(CC=CC)CC)=O)C2C)=O)cccc(C)c1C#N C1(NC(CCSCC)=O)CN(C(=O)CC2(C3CC3)CC2)CCC1C C=CCC(CNC(=O)C=Cc1cnn(C)c1)C(=O)N(CC(C)(C)N(C)C)C C1(C(=O)NCC23CC2CN(C(=O)CCc2ncc[nH]2)C3)CC2CCC(C1)C2O Cc1cncc(C(N2CCC(O)(CNC(=O)CC3CC(O)C3(C)C)C2)=O)n1 N1(C(CCOCC)=O)CC(CC(=O)N(C)CC2(C)CC2)CC1C N1(C(CCc2n(C)ccc2)=O)C2CC1CN(C(c1cnc(N)cn1)=O)C2 C(CN=C(NCc1cc(C(F)(F)F)cs1)NC(c1ccc(C)cc1C)C)OCC c1(C(=O)NCC(CC=C)NC(c2ccc(F)cn2)=O)ccc(C(C)F)cc1 CC1CC(C(C)(C)C)CCN1C(CC1CCOC1)C(=O)NC1CCCC1 c1(N2C(CC)CN(C(=O)CC3CCC(O)C3)CC2)nc(C)nc2c1cnn2C Cc1ccc(C)c(C(=O)NC2CC3C(NC(c4c(C)coc4C)=O)C3C2)n1 N1(C(c2c(COC)cco2)=O)CCC2(CCCC2CNC(=O)CCC)CC1.O C1(NC(c2cnc(Br)o2)=O)C2CCC1CN(Cc1ccc3ccsc3c1)C2 C1(C)(CC)NC(=O)N(CC(=O)NCCC(C)NC(=O)C(F)(F)CO)C1=O CCC(C(C)C)C(C(=O)NCc1cccs1)N1CC(F)(F)CC1C(=O)N(C)C c1(C(N(C2CCN(C(CC=C(C)C)=O)C2)CCO)=O)cc2ccccc2c(O)n1 C(=O)(C1CCCc2n[nH]cc21)N1C2CCN(C(=O)CCC3CCCC3)CC2C1 C1(=CCNC(C(N2CCCCCC2)C)=O)CCN(C(=O)CCc2ncc[nH]2)CC1 O(NC(=O)C(CCSC)NC(C1(c2ccncc2)CC1)=O)CC=C Cn1cc(C(C(N2CC3(CC3)C2)=O)NC(C2CCC3CC23)=O)nn1 O=C(C1=NN(C2CC2)C(=O)CC1)N1CCOC2CN(C(=O)C(F)(F)CCCC)CC12 C(c1cnc(O)nc1O)=CC=O.N1(C(C2C(COC)C2)=O)CCCC(C)C1.N C12(NC(CCC(=C)C)=O)CCCC1N(C(=O)CC(C)COC)CC2 c1(C(=O)NCC(CC(C)C)(C)NC(c2csc(Cl)n2)=O)ccc2c(c1)CCCC2 c1(C(=O)NC(CC(C)C)CNC(c2cnc[nH]2)=O)cncc(S(N)(=O)=O)c1 CCC(C)CCCC(=O)NC(C)(C)C=CC(=O)NC(C)CCF C#CC(CC)(CC)NC1CC(CC(=O)NCC2CCOC2)C1 N1(C(C2(SC)CCC2)=O)CCOC2(CCN(C(C3COCCC3(F)F)=O)CC2)C1 Cc1cc(=NC(=O)C(=O)NCC(CNC(c2[nH]ncc2C#N)=O)CO)[nH]o1 c1(NCCNC(CN2CCCC(N(C)C)C2)=O)nc2c(cc1C#N)CCOC2 C1(C)(NC(CCCSC(C)(C)C)=O)CCCN(C(=O)CC2CCCCC2(C)C)C1 Cc1cc(C(=O)NCC(C)N(C)C(c2nc(Br)c[nH]2)=O)sc1Cl N1(C(C(C)=O)=O)CCC2CC(CNC(c3ccno3)=O)CCC2C1 Cn1cc(Cl)c(C(N2CC(O)(CCNC(=O)C=CC3CCCCC3)C2)=O)n1 c1(NC(C2CCN(C(C3CCS3(=O)=O)=O)CC2)C)ncc(Br)cc1[N+](=O)[O-] C(CCC(C)CC(=O)NCCN(C(=O)CF)CC)=C(C)C.CCO.C(C)C.O N1(C(c2cc(COC)oc2C)=O)CCC(NC(=O)C#CC2CC2)C(O)C1 C1(C(N2CC(CCC)N(C(C3CC(O)CN3C)=O)CC2)=O)CCC2(CCC2)CC1 Cc1cncc(C)c1NC(=O)Nc1nc(COc2ccc(Br)cc2Cl)cs1 C(CC(C(=O)NCc1cnn(C)c1)NC(=O)CCC1CC1(F)F)OC C1(C)(NC(c2c(C)oc(-c3ccco3)n2)=O)C2CCNCC12 C1(CC(=O)OC)CNCC(C)(C)O1.c12ccc(cc1)-c1cn(nn1)C1CCCC21 C(=O)(C(c1ccccc1)=C(C)C)NC1C2N(C(C(CC=C)(F)F)=O)C(CC2)C1 CCCC(C(=O)N(CCCN(CC)CC)C)NC(=O)C(C)CO c1(C(COC(=O)Cc2ccc(Cl)s2)OC)cc(Cl)cc(Cl)c1 C(Cc1cn[nH]c1)(C(=O)N)NC(C(C)OCC=C)=O.c1(C2CC2)cncs1 N1(S(CC)(=O)=O)CCN(C(=NCCc2cc(Cl)ccc2Br)NCC(C)C)CC1 S(=O)(=O)(c1ccc(NCC23CCC(CC2)C3(C)C)c(F)c1)NCC(=C)C c1(C(c2nnnn2C2CCCC2)NC(c2nccs2)C)cnc2c(c1)CCC2 c1(CCCC(=O)N)cc(F)ccc1F.c1(SC)ccsc1C(=O)NC1CC1C C1(CNC(C2C(C)OCC2)=O)CCCCN(C(c2cc3occc3n2C)=O)CC1 Cn1nccc(C(=O)NC2(C)CCN(C(C3(C)C=CCC3)=O)CC2)c1=O N(C(=NCCCc1c(C)nn(C)c1C)NCc1ccc(N(C)C)cc1)CC(=C)Br C12(C(N3CCC(C=C)C3)=O)CCC(CC1)N(C(c1cc3occc3[nH]1)=O)C2 C(CC)(CCCC(=O)NCC1(OC)CCCC1)NC(CCC(=C)Cl)=O C(CC(=O)NC1CCN(CCCO)C1)(C(F)(F)F)NC(C1(C)CC2C=CC1C2)=O c12ccc([N+](=O)[O-])c(n1)NC13CCCN(CC1C3)C2=O.C1(CC=C)(CO)CC1 Cc1ccc(C(CF)NC(=O)CCNC(=O)C(F)(F)CN)cc1 C1(CC)CCN(C(c2cnn(C)n2)=O)C1CNC(=O)CCCc1ccncc1 N1(C(C(C)(C)CCCNC(C2CCCS2)=O)=O)C2CCC1CC1(C2)N=N1 O=C(CC(C(F)(F)F)c1ccccc1)NC1CC(C)(NC(=O)C2=COCCC2)C1 C1(NC(c2n(CC)nnc2)=O)CCCC(C(N2CCCCC(C)C2)=O)CC1 Cc1ccc(C(=O)NCC2C=CCN2C(=O)Cc2cn(C(C)C)nn2)cc1C C(=O)(C(CNC(=O)CS(=O)CC)C(C)C)NC(C(CC)C)CO n1(CCCCC)[nH]nnc1=NC(=O)N1CCC(C2CNC2)C1 C1(CC(=O)NCC(c2ccccc2F)NC(C2C(C)CC2)=O)CC(C)(C)CO1 C12CC1CN(C(=O)C(c1cccc(Cl)c1)(F)F)C2.C1(N(C)C)(C(=O)N)CC1.C C#Cc1cncc(C(=O)NC2COCC2NC(c2c(C)n[nH]c2C)=O)c1 CC1(C)CC(CNC(=O)CSc2cn[nH]c2)N(C(=O)C(O)C(F)F)C1 N1(C(CCC(=O)OC)=O)CCC2C(CCN2C(c2cccnc2CO)=O)C1 N1(C(C2CCC(NC(=O)C(CO)C(F)(F)F)CC2)=O)CCC(O)CC12CC2 c1(C(=O)NC2C(CNC(=O)CCC3CC3)CCC2)cnc2ccccn2c1=O C1(C(=O)NCCNC(c2ccc(C(CC)(C)C)cc2)=O)SC2C=CC1CC2 c1(C(=O)NC2CC(NC(C3CC34CC4)=O)C(O)C2)ccc2ccnn2c1 C1(C(N2CCC(CC(C)C)C2)=O)CC(O)CN1C(C1C(C)C1C)=O c1(CC)cc(C(=O)N(CC(=O)NCC2(OC)CCC2)CC)n[nH]1 C1(CC(=O)NCC2(C)N(C(C(C)OCC)=O)CCC2)CCCC2(CCC2)O1 N1(C(c2nc(C)nn2C)=O)CC2(CCC2)CC1C.c1(CCC=O)ccn(C)n1.N C1(C)(CNC(c2c(CC)nc[nH]2)=O)CCN(C(c2snnc2C(C)C)=O)C1 c1(C(C)=O)cccc(C(=O)NC2CCCC2NC(=O)COC2CC2)c1 N1(C(c2c(C)nc[nH]2)=O)CCC2(C1)CN(C(=O)CN1CCC(O)CC1)CC(C)O2 C12(CNC(C(C=C)OC)=O)CC(NC(=O)C(CC)c3cccnc3)(CO1)C2 C1(NC(=O)Cc2ccoc2)CCN(C(c2c[nH]nc2-c2ccccc2)=O)C1 C1(C(N(C)CCNC(=O)COc2cccc(Cl)c2)=O)CNC(=O)CC1(C)C C(=O)(C1=C(Cl)CCC1)N1CC(CC(C)NC(=O)CC2CC3C=CC2CC3)C1 C1(S(C)(=O)=O)(NC(c2ccc(OCCC(=O)OCC)cc2)=O)CNC1 Cc1c(CC(=O)NC(CO)C(=O)NC2CC2)cnn1C Cc1csc(Cl)c1C(=O)NC(CNC(=O)C(C)Sc1ccccn1)C(C)C C1(CC)CN(C(c2cc(OC)no2)=O)CC1C(=O)NCC1CCC(CO)CC1 N1(C(C2(CC)CCN(C(C34CC(F)(C3)C4)=O)C2)=O)CC(C)C(F)(F)C1 c1(CCC)[nH]ccc1C(=O)NCC(O)C(=O)NCc1nc(C)ns1 Cc1ccc(CNC(=O)CC2CCOC2)cc1O.C1(C=O)CN(C(N)=O)C1.N c1(C=O)ccnc(F)c1.C1(OCC)CN(C(=O)CC(c2ccco2)C2CC2)C1 N1(C(COC)=O)CCCN(C(=O)C(C(C)C)C2CCC2)C(C)C1 c1(CNC(=O)NC2C(OC)C(C)(C)C2)ccc([Si](C)(C)C)cc1 c1(C(N2CC(OC)C(NC(=O)C(C)N(C)C)C2)=O)cc2ccccc2nc1O Cc1nc(C)n(O)c1C(N1C2CCC(C2)C1C)=O.C12(C=O)CCC(CC1)CC2 C1CCN(C(C23C4C5C6C4C2C6C35)=O)C(C2CC2)C1.CS(=O)(=O)CC(=O)N c1(C(=O)NCCOCCCNC(CCSC)=O)c(C)cc(Cl)nc1N N1(CC)N=C(C(=O)N2CCC2CNC(=O)C(C)n2ccnc2)CCC1=O c1(C(N2CCC(NC(CC3(C)CC(F)(F)C3)=O)C(F)C2)=O)cc2ncccc2o1 C1(NC(C(=O)NCC(F)(F)F)=O)CCCCN(C(c2cc(=O)cc[nH]2)=O)C1 C1CCn2nnnc2C1.C1(CCC)(C(N2CC(C)(OCC=O)C2)=O)CC(=O)C1.N C(=O)(C1=CCC(C)CC1)N1C(CNC(=O)C2=NOC(C)C2)CC(OC)C1 N1(C(CCCOCCC)=O)CCCC1(C(=O)NCC1CCC1(F)F)CC N1(C(CC(=O)NC2CC2)=O)CCCC2(CCCN2C(c2ncc(F)cn2)=O)C1 n1(CC(=O)NCC(CO)NC(c2cccc(F)c2)=O)cc(Br)ccc1=O CS(=O)(=O)CCC(C=O)NC(=O)NCCN1CCCOCC1.C(=O)C(F)(F)F O=C(C1=Cc2ccccc2OC=C1)N1CCOC2CN(C(C3(F)CCC3)=O)CC12 C(=O)(CCC(F)F)N1CCC(=CCNC(C2C(C(=O)OC)C2)=O)CC1 CC1CC(c2nnnn2-c2ccccc2)(NC2CCC(CO)CC2)CN1C c1(CCOC)n[nH]c(=NC2CC(O)(C)C2)s1.C(c1cccc(C)c1)=CC(=O)N C1(C=O)CC(C)(C)C1C(F)(F)F.Cc1ncc(C(=O)NCC2CCC2)s1 N#Cc1c(NCC2CCN(CCCN3CCOCC3)C2)ncc2c1CCCCC2 C1(C)(C(=O)NC2C(NC(CSCCC)=O)COC2)CCCCC1(F)F Cn1cc(C(=O)NCC2(C(N3CC(C#N)C3)=O)CCCCC2)ncc1=O C=C=CCC(C(=O)NCc1snc(C)c1N)NC(=O)OC(C)(C)C c1(C(=O)NC2C3CN(C(CCc4n[nH]c(=N)s4)=O)CC32)cc(Cl)ccc1F C1C=CCN1C(=O)CC1(C(F)(F)F)CC1.O=CCC.c1(C(=O)N)ccco1 C1(C)CN(C(=O)CC2CCC(=O)N2)CCO1.c1(CC)cc(C(=O)NC)oc1 c1(C(=O)NCC(CC)NC(=O)C(F)CC2CC2)cn(-c2ccccc2)nc1C N1(C(C2(C)COC(=O)N2)=O)CCCC(F)(C(=O)NC2CCCC2CN=[N+]=[N-])C1 c1(NC2CC3CN(C(c4cccc(SC)n4)=O)CC32)cc(C)c(C#N)cn1 c1(CN2CC(O)(CNC(=O)CC3CCOCC3)C2)cc(Cl)ccc1Cl CC(N=c1[nH]c(=NCCSC(F)F)c2ncccc2[nH]1)c1csnn1 c1(OC)ccc(C)c(OC)c1CNCc1cccc(F)c1OC(F)F Cc1cccc([N+](=O)[O-])c1C(=O)NCC(C(C)C(C)C)NC(=O)C.CC(F)F N1(C(CCCN=[N+]=[N-])=O)CCC2CCN(C(=O)CCC3CCCO3)CC2C1 C1(C(N2CCC(O)(CC)C2)=O)CN(C(=O)CCC(C)SC)CC(C)(C)C1 Cc1nn(CCO)c(C)c1C(N1CCC(N2CC(C(=O)O)CC2=O)CC1)=O C(C(O)CCNC(c1cnn(CC(F)(F)F)c1)=O)NC(=O)C=CC=C(Cl)Cl C(=O)(CC(C)(C)COC)N1CCC(C(C(=O)NCC2(CC)CCOCC2)C)C1 c1(C(=O)NCC(C)CNC(C2CCC(O)C2)=O)cc(F)cc(Cl)c1O N1(C(C(C#C)(C)C)=O)C2CCC1CC(CNC(c1cnn(C3CC3)c1Cl)=O)C2 c1nc(-c2cc3ccccc3[nH]2)c2ccccn12.c1ccnn2ccnc12 c1(OC)ccccc1CC(=O)N.C12CC1CN(C(C1(C(F)F)CCCO1)=O)C2.C CC1(C)CN(C(c2ccc(F)cn2)=O)CC(C)O1.c1(C(=O)N)cnc(C2CC2)o1 O(P(=O)(CCC1CCN1C(=O)C(C)C)OCC)CC O=C1CN(C(=O)CCC2OCCO2)C(C(=O)NCCCCC(F)(F)F)CN1 n1(CCSC)nnnc1C(C(C)(C)N1CCCC1)NCCCC1CCCCO1 c1(CCC)noc(CC(=O)NC2CCC(NC(=O)CC3CC3(C)C)C2)n1 Cc1cn2cccc(C(N3CC(CCNC(C4CC5CCC45)=O)C3)=O)c2n1 C(=O)C1=C(C#N)CCC1.C(=O)(C(O)Cn1cncn1)N(C(C1CCC1)C)C C12(CNC(c3cc(CC)on3)=O)CCC1CN(C(=O)C=Cc1ccoc1)C2 C1(C(=O)NCc2ccc(F)cc2)CCCN(C(=O)C2=CCCOC2)CC1 c1(C(CC(=O)Nc2cccc(NC(C(C)=CC)=O)c2)O)nc2ccccc2[nH]1 C12(CNC(=O)C=Cc3cnc[nH]3)CCCC(CN(C(=O)CO)C1)C2 c1(C(F)(F)F)cc2c([nH]1)C(Nc1nc(Cl)nc3sccc13)CC2 N1(c2nccc(OCC)n2)CCOC2(CCN(C(=O)C(N)=O)CC2)C1 C(=O)C(C)CS(C)(=O)=O.C1(OC)CN(C(=O)CCc2ccc(C)s2)C(C)C1.C c1(C(=O)NCC(C(C)C)NC(C2CCCCO2)=O)ccc2[nH]nc(O)c2c1 C1(C(N2CCCC2)=O)CCS(=O)CC1.c1(C(=O)NCC)conc1.C1CC1.O c1(CC)n[nH]c2c1CCCC2.Cn1cc(C(=O)C=CC(N2CC(CO)C2)=O)cn1.O Cc1c(C(=O)NC(c2nc(C(=O)NCC(C)C(F)F)co2)C)c[nH]c1C#N N1(C(c2cncc(C)n2)=O)CCC2CCC(NC(c3cc(C(N)=O)co3)=O)C1C2 C1(OC)CCCC(C(=O)NOCCn2cc(-c3c(C)cnn3C)nn2)C1 c1(C(=O)NCC(C)CNC(c2ccc(Cl)o2)=O)ccc(CN2CCCC2)o1 N1(C(c2c(C)n(CC(C)(C)O)nc2)=O)CCC2(CC1)CC(C(=O)NC1CC1)CO2 c1(C(=O)Nc2nc(CC(=O)Nc3cnn(C4COC4)c3)cs2)cnc(Cl)nc1 c1(C=O)cc2c(=O)n(C)c(=O)n(C)c2n1C.CCCCN(C(=O)CC1CC1)C C1CN(C(=O)C(c2cccc(Cl)c2)O)CC12CCC2.O=C(CSCC(F)F)NC N1(C(C(CCCC)C)=O)CC2CC(C)N(C(=O)CCCCC(=O)NC)C2C1 C(c1ccccc1Cl)=CC(=O)N.c1(C(N(CC(O)C)C)=O)cccc(C(F)F)n1 c1(CCNC(C(C)NC(COCCCC)=O)=O)cnn(C)c1C C1(NC(c2cncc(C)c2Cl)=O)COC2(CCN(C(c3ccccn3)=O)C2)C1 C1CCCN1C(=O)C=O.C(C(=O)NC1CC1)(C1CCOC1)OC.CC(F)F.C N1(C(C(C)OCC=C)=O)CC(NC(c2cnccc2Cl)=O)C(SC)C1 C1(CNC(c2csc(C(F)F)c2)=O)C2CC1N(C(c1cnsc1)=O)C2 N1(C(C(CNC(c2ccc(C)[nH]2)=O)O)=O)C(C)CCC1(C)C c1(C(N(C(C)CS)CC)=O)cc(O)nc2c1CN(C(c1cnn(C)c1)=O)CC2 C1(CC(=O)N(C(C)CNC(c2ccc(Cl)s2)=O)C)(C(=O)OC)CCCC1 C1(C(=O)NCCn2ncc(C)c2)COCCN1C(c1n[nH]c(C)c1C)=O N1(C(CC2(OC)CN(C(=O)Cc3ccnn3C)C2)=O)CC2CSCC(C2)C1 c1(C(N(CC(C)NC(C(C=C)(C)O)=O)CC)=O)ccc(OC)c2ccncc12 c1(CC(=O)NC2C(NC(Cc3ccc(C)nc3)=O)CC2)ccc(Cl)c(F)c1 C1(CNC(=O)COCC2CCCCO2)CCCCCN1C(=O)C1=CCCSC1 N1(C(C(C)CN2CCOCC2)=O)CCN(C(=O)COCC2CCCC2)CC(O)C1 c1(CC(=O)NC2C(F)CCN(C(C=C(COC)C)=O)C2)ccc2nn[nH]c2c1 Nc1cccnc1C(=O)NCCC1(O)CN(C(C2CCNC(=O)C2)=O)C1 c1(C(=O)NCC(CC)N(C(=O)C=C2CCN(C)C2)C)occc1C1CC1 CCCCCC(C)CC(=O)N(C(C)C(=O)NC1CC(O)CC1O)CCC C(=O)(N=c1ccn(C)[nH]1)C1CCCC(NC(C(CSC)C)=O)C1 c1(CCCCc2n(C)cnn2)cc(=NCCC2CCOC(C)(C)C2)[nH]cn1 N1(C(c2c(CC)nns2)=O)CC2CCCC2(NC(c2cc3sccc3n2C)=O)C1 N1(C(CNC(C)=O)=O)CC2CC(NC(=O)C[SH](=O)=O)C1C2.C1CCC(C)CC1 Cc1ccncc1C=CC(=O)NCC1CN(C(c2c(C)cnn2C)=O)CCN1C CC(C)CCCC(=O)NC1(C)CC(NC(c2cc[nH]c(=N)n2)=O)C1 C(c1ccccc1)=C(CC)C(=O)NC(C)C(C)NC(=O)Cc1cccnc1 Cc1nc(Br)sc1C(=O)NC1CN(c2cc(C(F)(F)F)ncn2)CC1C C1(C(=O)NCCC2CC(C)(C)OC2)CN(C(c2cc(=O)cc[nH]2)=O)CC1(F)F c1(C(=O)NC2C(CNC(c3c(C)ccs3)=O)CCC2)csc2cncn12 N1(C(COCP(C)(C)=O)=O)CC2CCN(C(c3cc(Cl)c([N+](=O)[O-])[nH]3)=O)CC2C1 C1(NC(C(C)NC(C)=O)=O)CCN(C(C2CSC2)=O)CCC1c1ccccc1 C(=O)(C#CC1(CC)COC1)N(CCC(=O)NCCCCC)CC CC(C)(O)C(F)C(=O)NCC1(CO)CCN(C(c2nonc2N)=O)C1 c1(C(N2CC(Nc3ncc4cn[nH]c4n3)C3(CC3)C2)=O)cnc2c(Cl)cccn12 C1(NC(CSCC)=O)C2CCC1CN(C(c1ccc(CC)cc1)=O)C2 c1(C2(C(N3CC(C)(NC(c4sccc4OC)=O)C3)=O)CC(C)C2)ccccc1F C1(C(=O)NC(C2(O)CN(C(C(C)N(CC)CC)=O)C2)C)CCC(C)CC1 c1(NC(C)=O)cccc(C(N2CCSCC2CCNC(=O)CC(C)F)=O)c1 C1(C)(C(N2CC(CC=C)(NC(c3ncccc3)=O)C2)=O)CCCNS1(=O)=O.O c1(C(N2CC3C(NC(C(CC=C)C(C)C)=O)(C3)C2)=O)ccc2[nH]ccc(=O)c2c1 C(c1ccccc1OC(F)F)=CCNC(CN1CC(C(C)C)OCC1)=O C=CCCCC(C(=O)N1CC2CC2C2CC12)NC(c1cc[nH]n1)=O C1(C(C)=O)CCC(CC(=O)NCC(O)CN(C(=O)CCc2nccn2C)C)CC1 c1(CC(=O)NCC2CCCN(C(C3(C(=O)OC)CC3)=O)C2)ccccc1F N1(C(CCc2n(C)cnc2)=O)CCN(C(C2CCCCC2)=O)C2CCCCC12 CCC(C)C(=O)C(=O)NCC=CCNC(c1ccns1)=O c1(N(CCC)C(N2CC(C)C2C)=O)cn(C2CCCCC2)nc1C N1(C(c2ccncc2Br)C(=O)NCCOC)CCC(C#N)(CN(C)C)CC1 N1(C(c2cn(C)c(=O)cn2)=O)CC2CCN(C(C3(C)CCCO3)=O)CC(C2)C1 c1(CC)ccc(NC(C2CSCCN2Cc2ccc(Br)cc2Br)=O)cc1[N+](=O)[O-] N1(C(C(CC#C)O)=O)CC(C(=O)NCc2ncsn2)C(F)(F)C1 C(=O)(N=c1ccn(CCF)[nH]1)C1C(NC(C(C)c2ccsc2)=O)COC1 N1(C(COCC(C)C)=O)CCCC2(CCN(C(c3ccc4c(c3)COC4)=O)C2)C1 c1(CN2CCC(NC(CC(=O)OCC)=O)C2)cccc(I)c1O c1(C(=O)NC2C(C)CN(C(c3cccc(O)n3)=O)C2)cc(C(F)F)ccc1F C1(N(C(C2C(C)CCO2)=O)C)CN(C(c2ccc(C(N)=O)nc2)=O)CC1(C)C c1(C(N2CCC(C(F)(F)F)(CNC(C)=O)CC2)=O)ccc(C#N)c(O)c1 CN1CCC(C(=O)NC2(CO)CN(C(C3CCCCC3C(N)=O)=O)C2)CC1 Cc1cc(C(=O)NC2CCCC(NC(C3CCCCC3O)=O)C2)c(N)c(Cl)c1 c12ccc(cc1)Cn1cc(nn1)C(=O)NC(=O)C2.C1(CC)CCCCO1.CCO.N CCC(CC(=O)NC1(C)CCCN(C(c2cc(C)cc(O)c2)=O)C1)C(F)F c1(CN(C)C(C2(F)CCCOC2)=O)ccccc1CNC(C1CCCCS1)=O C1(C(=O)NC(C(=O)OC)(C)CO)CCN(C(=O)CCC(N)=O)C(C)(C)C1 C=CCCCC(=O)N(CCCCCNC(c1cc(-c2ccco2)[nH]n1)=O)C C1(C)(OC)CCCN(C(=O)CC2CCCCC2NC(=O)CNC(C)=O)C1 N1(C(CC=CC)=O)CCCC2C1CCCN2C(c1cccc(C(F)F)n1)=O Cn1cncc1C=CC(=O)NCC1C2CN(C(=O)Cn3cc[n+](C)c3)CC12 N1(C(C(C)Cc2ccncc2)=O)CCCC(N(C)C(C2CC(C)(C)C2)=O)C1 CCCC(C(=O)OC)C(=O)N1CCC(NC(=O)C(CC2CCC2)OC)C(O)C1 Cc1cnc(C(C2CC2)NC(=O)NC2COCC2N(C)C)s1 C(=O)C(C)(C)CC(F)(F)F.C1(C(NCC)=O)C2CCC1(c1cnco1)C2.CC C(=O)(C1Cc2ccccc21)N1C2(CNC(C(C)CN3CCOCC3)=O)CC(C1)C2 C1(C(N(CC(C)N(C(c2ccc(C)nc2O)=O)C)C)=O)CC2CCCCCC12 c1(C(N2CCC(O)(c3cn(CCCF)nn3)CC2)=O)ccc2ncc(Br)n2c1 C12(C(N(C(CC)CC)C)=O)C(NC(=O)Cn3ccc(C)n3)C3CC1C2C3 CC1CCNCCC1N(C1CC=CC1)C(C1(C2CC2)CC1)=O Cc1cc(Cl)cc(C(N2CC(CNC(c3ccc(O)nn3)=O)C3(CC3)C2)=O)c1N C1(CC#C)(C(=O)N(CCCO)Cc2ccccc2)CCN(C(c2cnsn2)=O)C1 C(=O)(C1c2ccoc2CCN1C(=O)OC(C)(C)C)NCC(CNC)OC C1(NC(C2C3(CCN(C(C(C(C)C)=O)=O)C3)C2)=O)Cc2ccc(Br)cc2C1 C(C(C)N=c1cc2n([nH]1)CCN(C(=O)OC(C)(C)C)C2)N1C(C)COCC1 C=CCCCCCCC(=O)N1CCCC(NC(=O)Cc2cnc(C)s2)CC1 C1CC2(CCN(C(C34C=CC(CC3)C4)=O)CC2)C1.C#CC1(C(=O)N)CCCC1.C c1(C=O)cc(F)ccc1-n1ccnc1.c1(C(N(C(C)C)CC)=O)csc(Cl)n1 C12(CNC(C3(C=C)CCC3)=O)CC(NC(=O)CC3CCCC3)(CO1)C2 C1(C)(CC)CCN(C(=O)C(C)N(C)C(c2cnc[nH]c2=N)=O)CC1 C1(NC(NCCn2nccn2)=NC)CCC12CCCC2.c12ccccc1C2OC N1(C(c2ccc(CSC)cc2)=O)CCC(C)C(C)C1.C1(O)(C=O)CCOCC1.N Cc1ccc(N)c(C)c1C(=O)N(C1CCCN(C(C23COC(CF)(C2)C3)=O)C1)C c1(C(N(CCNC(=O)C2=NOCC2)CC)=O)nccc(Br)c1O N=c1[nH]c(CC(=O)NCCOCC)cs1.c1(CC=O)ccc(Cl)s1.CC.O N1(c2snc(SC)n2)CC2CCCC(NC(c3ccc4cnnn4c3)=O)C2C1 C=CCN=C(NCCS(=O)(=O)CC1CCC1)NC1CC(C)C1 Cc1cc(C(=O)NC2(CNC(=O)Cc3ccsc3Cl)CCCC2)c2n[nH]cc2c1 c1(C(N2C(C(=O)Nc3c(Br)ccc(C)n3)CC(C)C2)=O)cc(Cl)nc(Cl)c1F c1(C(=O)NC23C(CN(C(CCCCC(N)=O)=O)C2)C3)ccc2c(c1N)CCCC2 C1(C(N2CC(C(C)NC(c3ccnc(Cl)c3)=O)C2)=O)CC(=O)NC(=O)N1 Cc1nn(C)c2ncc(C(=O)N)cc12.C1(C)CCN(C(=O)C=C2CCC2)CC1.C CC(CNC(C1(Cl)CC1)=O)(CO)NC(C1CC(=C2CC2)C1)=O C1(C)CCCCC1.c1(CC=O)c(Cl)cnn1C.CCS(=O)(=O)NCC(=O)N.C CCC(COC)C(=O)NC(C)C(C)(C)NC(C1CCC(C)(C)C1)=O C1(C(=O)NCC2C(C(=O)Nc3cccc(C)c3)CCCC2)CC2CC(=O)C1C2 CCCC(CC)(c1ccccc1)NCC1CCN(S(C)(=O)=O)C1 N1(C(CCSC)=O)CCCC(C2CN(C(=O)COCc3cccnc3)C2)C1 CC(C(=O)N1CC(O)CC1CNC(c1cncnc1C1CC1)=O)C(F)(F)F C1CCOCC1.c1(C(N(C(C)C)CCNC(=O)C)=O)ncn(C(C)(C)C)n1 N1(C(c2ncc(C)nc2)=O)CC2(CCC(NC(=O)C(Cl)=CCl)CC2)C1 c1(CNC(C2CCC(C)S2)=O)ccc(CNC(=O)CCC=CC(C)C)cc1 C1(NC(c2c(C)nc(-c3ccsc3)s2)=O)CCCC2(C1)OCCO2 N1(C(C(C)(C)CF)=O)CC(NC(c2cccc(Cl)c2N)=O)C2CCCC2C1 Cc1ccc(CC(C(=O)N2CCCC2)Nc2ncc(F)cn2)cc1.N1CCOC(C)C1 CC1(C)CCN(C(C2CCCC(O)C2)=O)CC1C.C1(C=O)CC2C(C1)C2(F)F.N c1(-c2cncc(C)c2)nc2ccc(C(=O)NCCc3cccc(Br)c3)cc2s1 C=CCCCCCC(=O)N(CC(O)CN(C(=O)C(CN(C)C)C(C)C)C)C C(N=c1[nH]c(=N)[nH]cc1Cl)c1cc(N2CC3OCCN(C)C3C2)ncn1 C1(C=O)CCC(C2CC2)C1.C1(C(=O)OC)(C(=O)NCC2CCC2)CC1C CCCC(C(=O)NC1C(C)CCN(C(C2CSC(C)=N2)=O)C1C)C(C)C c1(C(N(CCC(=O)NCCCN2CCCC2)CCO)=O)csc(O)n1 Cc1ccc(C=CC(=O)NCCC2CN(C(=O)C(C)c3ccsc3)C2)nc1 C(=O)(C1CCCc2scnc21)N1CC(CNC(c2c(C)snc2)=O)C(F)(F)CC1 c1(N(CCOCC)C)nc(N2CCc3[nH]nc(O)c3C2)c2cnn(C(C)C)c2n1 C1(C=O)CCn2cc(C)nc2C1.C(C)(CCC(=O)NCC1CCC1)OCC.C c1(OC)ccc(CC(N2CCCC(c3cc(C(N)=O)n[nH]3)C2)=O)c(Cl)n1 CCC(C(=O)N1CCC(C(=O)NC2C3CCC(F)(F)C23)O1)OC C1(C(=O)NC2(CCF)CC2)C2CCC(C2)N1C(=O)C(C1CC1)C1CC1 CC1CCCn2c(CC(N3CCC(CN(C(=O)CC=C(Cl)Cl)C)C3)=O)cnc21 c1(CC)cc(C(N2CCC(O)(C(C)NC(C3CCCN3C)=O)C2)=O)ncn1 Cn1ncc(C(N2CCN(C(=O)CS(C)(=O)=O)C(C(F)F)C2)=O)c1S(C)(=O)=O c1(NC(C2C3CN(C(C(c4ccccc4)C)=O)CC32)=O)cnc(C#N)cn1 N1(C(c2c(C)sc(Cl)n2)=O)CCC(NC(C2CC(OC(C)C)C2)=O)C12CC2 c1(C=O)c(C)nsc1.C1(CCC)CCCC1C(=O)NCCC1CC1.C1CC1 Cc1cc(C(=O)N(C2CCCN(C(C3CC3F)=O)C2)CCO)cc(Br)c1C c1(C(N2CC3(N(C(C(C)C#N)=O)CC3)C2)=O)ccc2c[nH]nc2c1 c1(C=O)nc(N)cc2ccccc12.C1(CC(=O)NCCCC)CCS(=O)(=O)C1.N [N-]=[N+]=NCCCC(=O)N1CC2CC(NC(=O)C(F)(F)c3cnccn3)C2C1 N1(C(C(C)(C)OCC)=O)CCC(NC(=O)Cn2cncn2)C(C)C1 Cc1cc[nH]c1C(=O)NCC(C1CCCN1C(=O)CO)(C)C.c1ccncc1.C c1(OC)cccc(C(C)(C)C(=O)N2CCC(NC(=O)C(C3(O)CCCC3)F)C2)c1 C1(C(N(CCCCCNC(CCC)=O)C)=O)C2CCC1(c1ccco1)C2 C1(CNC(C(C2CC2)SC)=O)CC2CCC1N2C(=O)CC1CC=CC1 C1CN(C(=O)C=Cc2ccsc2)CC12CCOCC2.C1(C(=O)OC)CC1C=O.N c1(C(N2CCC(C)(CCOC)C2)C(=O)NCC=C)cn(C(C)C)nc1Br C1(NC(C2(NC(C)=O)CCCC2)=O)CC(C(N2CC(CC(F)F)C2)=O)CC1O c1(CNCc2nccc(C(=O)NC(C(CC)C)CO)c2)cc(Cl)cnc1F N1(C(C(COC)O)=O)CCCCC1C(C)(C)CNC(=O)C1=COCC1 C(CCCc1ncc[nH]1)NC(C=C(C)CNC(C1(CO)CC1)=O)=O c1(CN2C(C(N(C)Cc3cccc(Br)c3)=O)CCCC2)ccccc1S(C)(=O)=O C(C(CC)(CC)C(=O)NCC(COC)C(C)C)NC(c1c(CC)nns1)=O N1(C(C(c2ccccc2)NC(C)=O)=O)CC2CN(Cc3cc(Cl)cs3)CC2(C)C1 CC1CN(C(=O)CC2CCCN(C(C3(O)CCCCCC3)=O)CC2)CC(C)(C)O1 Cc1nc2ccc(NC(c3ccc(C4CC4)nc3C)=O)cc2s1 c1(C(=O)NC2(C(=O)Nc3c(OC)ccc(O)c3)CCCC2)cccc2ccnn12 c1(C(N2CCC(CN(C)C(c3cccn3C)=O)C2)=O)cc(F)c(O)c(F)c1 N1(C(c2cc(C)c(C)[nH]2)=O)CCC2CN(C(C3CCC(C(N)=O)O3)=O)CC12 CC1(C#CC(=O)NCC(CO)NC(C2CCCC2F)=O)COC1 C1(CNC(=O)C2=CCOCC2)CN(C(C2CCC(=O)N2)=O)CCC1(F)F C12(CNC(c3c(C)cco3)=O)CCC(CC1)N2C(C1C2CCCOC12)=O Cc1c(C(=O)N)cnn1CC(C)(C)O.C1(O)(CC)CCN(C(c2cscn2)=O)C1 n1(CC(=O)N(C2CCCCC2N(C)C(=O)O)C)ncc(C#N)c1N.C(C)(C)C CC1(C)CCCN1C(=O)C=Cc1ccc(C(N)=O)o1.c1(CC=O)cnsc1.C c1(C(N2CCC(NC(=O)CC3CC3(Cl)Cl)C2)=O)cc[n+]([O-])cc1 c1(C(=O)NCCCCC2CN(C(c3cc(C)sc3)=O)C2)csc2cc(Cl)cnc12 c1(NC(CSCc2c(C)cc(C)s2)=O)noc2c1CC(F)(F)CC2 C1(NC(CC=CC=C)=O)CC(C(N2CCC(CC(C)C)CC2)=O)C12CCC2 C1(C(=O)NCC)C2CN(C(=O)CNc3ccccc3F)CC12.C[SH](=O)=O.N c1(C(=O)NCCCN(C(C)C)CC)cnn2c(OC)cccc12 N1(C(c2c(CC)c[nH]n2)=O)CCC2CN(C(C3C4(CC4)C34CC4)=O)CCC2C1 c1(NCC(=O)NC(C)CCNC(C2CCCC(=O)N2)=O)ccc(C#N)cc1 C1(C(N(CC(C)C)CC#C)=O)C2CCC(C2)N1C(=O)C(F)CC1CCOC1 c1(C(=O)NC2CCC(N(C(C(CC#C)O)=O)C)CC2)cc2n(n1)CCCC2=O C1(C(=O)Nc2cc(C)cc(F)c2)CN(C(=O)C(O)CN(C)C)CC(C)(C)C1 Cc1cc(N2CCN(CCNC(c3cccc4cc[nH]c34)=O)CC2)c(C#N)cn1 C1(O)(CNC(=O)CCCn2cccn2)CCCN(C(C2CC23CC(F)(F)C3)=O)C1 c1(OC)ccc(C)cc1NC(C1CC1C(N1CC2CCC1CC2)=O)=O CN1CCCC1C=CC(=O)NCCC(C)(C)NC(=O)CCC1CCCO1 c1(CCNC(c2ccc(C)cn2)=O)cc(F)cc(Cl)c1.C1(C#N)(C=O)CCC1.N c1(OC)cc(C(=O)NCC(CNC(C2CC=CCO2)=O)CO)cc(OC)c1.O c1(CNCC2(NC(=O)OC(C)(C)C)C(C)CCCC2)cnc2ccccn12 C1(C(N2CCC2)=O)C(C)(C)C1(C)C.N1(C(C(C)C)=O)CCCC1C(=O)N.C O=C1CCc2cc(C(=O)OCC(=O)NC3CCC3c3ccc(Br)cc3)ccc21 Cc1cc(F)c([N+](=O)[O-])cc1C(=O)NC1CCCN(Cc2nn(C)cc2Br)CC1 CCC(CNC(c1cnc(C2(C)OCCO2)s1)=O)CC.C(=O)C=CC(C)C.N Cc1[nH]c(C(=O)NC2C=CCN(C(=O)C=CBr)C2)c(C)c1C c1(C(COC)(C)NC(C2CCCCC2)C(C)C)nnnn1C1CC(F)(F)C1 c1(OC)cc(CO)ccc1C(=O)NC1(CNc2ncnc(O)c2Br)CCCCC1 c1(C(N2CCC(C)(CC(=O)NCc3cccc(Cl)c3)C2)=O)ccn2cncc2c1 N1(c2cccc(OC)c2)CCCC(NC(C2CC3CCC(C2)O3)=O)C1=O N1(C(c2c(CC)nc[nH]2)=O)CCOC2CN(C(c3ccoc3Br)=O)CC12 CC1CN(C(c2cccc3ccoc23)=O)CC(C)C1NC(C1CC(O)C1)=O N1(C(CC(C)N(C)C)=O)CCCC2(CCCN2C(C2CCN(C)CC2)=O)C1 N1(C(C(C)(CO)OC)=O)CCC2(CCC2)C(C)C1.c1(CC(=O)N)ncc(Cl)s1 C1(C(=O)N)(C(C)C)CCN(C(=O)C=Cc2cncs2)C1.CCCCC1CCCC1 Cc1cc(C)n(C(C)CC(=O)NC2CC3(C2)CC3)n1.C1(CC=O)OCCCO1.N CC1CN(C(=O)C=C2CCCCC2)CCCN1C(c1cc(F)c[nH]1)=O N1(C(CC(CC)NC(=O)C(C)NC=O)=O)Cc2nc(C)sc2C1 C1(N(C(=O)Cc2ccsn2)C)CN(C(c2sccc2-n2cnnn2)=O)CC1F c1(C(=O)NC2C(NC(CC=CC(C)(C)C)=O)CCC2)cccc(Cl)c1Cl C1(N(C(C(F)=C(C)C)=O)C)CC2CC1N(C(C1CCC1(C)C)=O)C2 C(C(CC(C)C)C(=O)NC1CCOC2(CCC2)C1)NC(C(CCC)C#N)=O c1(NC(C2CC3(CN(C(CSC(C)=O)=O)C3)C2)=O)c(F)c(F)nc(F)c1F C1(C(=O)NC2CC(NC(Cc3cccc(C)c3Br)=O)C2)CC1C1CCOCC1 CC(CC(=O)NCc1nc(C)cs1)C(F)(F)F.c1(C(=O)N)cccc2[nH]ccc12 OC1CC(c2nc(-c3ccsc3Br)no2)C12CCC2 N1(C(CCCCOC)=O)C2CCC1CC(C(=O)NCC(O)C(F)F)C2 C=CCCCC(=O)NCCN(CCCN(C)C)C(=O)Cc1ccccc1O C#Cc1ccc(C(=O)NCC2C3CN(C(C4(C(N)=O)CC4)=O)CC23)cc1Cl C(=O)(C(F)(CNC(=O)CC(O)C(C)C)C(C)C)NCC(CCC)(C)C N1(C(Cc2n(C)ncc2)=O)CCCC1(C)C(=O)NCCCCF C(=O)(C1Cc2ccc(Cl)cc21)NC1(C2CCN(C(CC(C)C(F)F)=O)CC2)CC1 N1(C(c2c(OC)nccc2)=O)CC(NC(=O)C2=CCCC2C)C(C)(C)C1 c1(C(=O)NC(C(C(=O)NC2(CCC)CCNC2=O)C)C)nnc(O)nc1O c1(CC(=O)NC2CN(Cc3ccc(-n4cccc4)cc3)CC2O)cc(Cl)cnn1 C(C(O)C(=O)NC1COCC1C(=O)NCc1cc(O)ns1)=CC N1(C(C=Cc2ncc(C)[nH]2)=O)CCN(C)CC1CNC(c1csc(C)c1N)=O Cc1nc(C(=O)NCC(O)CN(C)C(c2c[nH]nc2C(F)(F)F)=O)c(C)n1C N1(C(c2cnc(C(F)(F)F)s2)C=O)CCC(CO)=C(F)C1.C(=O)(CC)OC.N N1(C(CCSCC)=O)CCC2CCN(C(c3ccc(N)c(CC(C)C)c3)=O)CC12 N1(C(c2c(C)ccnc2)=O)CC(F)(F)CC1C(=O)NCC1CC(O)CN1C c12ncc(cc1C#N)c(=O)[nH]2.c1(CC)ccccc1N1CCOCC1 C1(NC(CC(CC)O)=O)CCN(C(c2cccc(CF)c2)=O)CC12CCC2 N1(C(c2ccc(COC)cc2)C(=O)NCC2CCCO2)CC=C(C#N)CC1 C1(O)(CNC(CC(C)N(C)C)=O)CCN(C(=O)C(c2ccccc2)O)CC1 c1(C(=O)NCCCC2CCCN2C(=O)CCF)nccc2occc12 c1(CC(N2CC(NC(C3CN(C)C(=O)CC3)=O)C3C2C3)=O)n[nH]c2ccccc12 c1(CN2CC(NC(c3c(CCC)nco3)=O)(CO)C2)ccc(OC)cc1 N1(C(COC)=O)CCC2(CC1)OCCC2NC(=O)CCc1ccccc1C C=CCC(CC=C)C(=O)N1CC2(CC2)CC1C(N1CCCC(CC)(CC)C1)=O c1cnc(Cl)c(Cl)c1.c1(C(=O)OC)ncncc1NC(=O)CC1CN(C)CCO1 Cc1noc(C)c1C(=O)NC1CN(C(=O)CC2CCN(C)C2=O)C1 CCC1=C(C(=O)NC2C(C)(C)C(NC(=O)C(CCOC)O)C2(C)C)SCCO1 C1(NC(=O)NC)CCN(C(=O)CC2CCN(Cc3csc(Br)n3)C2)C1 c1(C(=O)N)cn2ccc(F)cc2n1.CC(CC(=O)N(C)CCOCC)C(F)(F)F CC(C)CC(C)C(=O)N1CCCCC1C(C)NC(=O)Cn1cnnc1O c1(C(=O)NC(C2CCCN2C(=O)C2=COCCO2)(C)C)cnc2c(c1)CCCO2 c1(NC(C2CCCO2)C)nc(N2CCN(c3cnccn3)CC2)nc2scnc12 c1(C(=O)NC2C(CC)CN(C(=O)C(C)(C)C(C)C)CC2)nccc2nn[nH]c12 Cn1nnc2cc(C(=O)NC3CCC3F)cnc12 c1(C(=O)NC(CCC)CNC(C2CCCO2)=O)nccc2n[nH]cc12 N1(CCC)CCCC1C=O.c1(CN(C(C)CCC)C)cn(C)nn1.c1ccccc1 C(=O)C1=NNC(C(F)(F)F)C1.c1(C(=O)NCCC(C)C)cccnc1C1CC1 C1(CNC(C(C)SCC)=O)COC(C)(C)CN1C(c1cc(C)n[nH]1)=O.C C1(C(=O)NC2C3CC(NC(C4C(C)(C)C4)=O)CC32)CCCCC1N=[N+]=[N-] CC(C)(O)C(F)C(=O)NC1(C)CCN(C(=O)COc2ccc(Br)cc2)C1 CC(C)CN=C(NCC1CC12CC2)NCC1COC(=O)O1 CC(C)(CCC(=O)Nc1cnc(F)nc1)NC(=O)CN1CCSCC1 CCC(CC)(CC)C(=O)NC(CNC(c1cc(F)ccc1C)=O)C(C)(C)C N1(C(C2C(COC)C2)=O)CCC(C)(C)CC1.c1(C=O)cc2n(c1)CCSC2.C c1(C(=O)NC2(CNC(=O)CCC3CCOCC3)CCOC2)cccn2ccnc12 CC1CCC(C)(C)N1C(=O)CC1CC(C=O)C1.C(C)(C)C.N(C)(C=O)C CC(C(C)C(=O)NCCCCn1cc(COC(=N)O)nn1)S(C)(=O)=O C1(NC(C#CC(=O)N(C)C)=O)CN(C(=O)C(F)Cc2ccccc2)CC2(CC2)C1 c1(OCC)ccc(C(=O)NCC(c2cccc(C(=O)OCC)c2)O)cc1 c1(CC)nc(C)oc1C(=O)NOCC(N1CC(C)CC1OC)=O N1(CC(=O)NCC2(F)CN(C(c3cc(Br)sc3Cl)=O)C2)CCC(F)CC1 C1(NC(c2c(C)n(-c3cccc(Cl)c3)nn2)=O)(CO)CCN(C(=O)CC(C)O)CC1 C1(C)(C(=O)NCC(c2ccccc2)C)CCCN(CC2CCC(C)O2)C1 S(=O)(=O)(c1ccc(NCc2ccc(S(C)=O)cc2)c(F)c1)NCCCSC C1(C(N(C(C(C)C)CO)C)=O)CCCCCCN1C(c1cncnc1)=O N1(C(CSCCC)=O)CCC2(CCC(NC(C3CC4(CCCCO4)C3)=O)CC2)C1 N1(CC=C)CCN(C(C2COCC2NC(C23CC(F)(C2)C3)=O)=O)CC1 CCC(C(=O)NCC1CN(C(=O)C(C)(C)C(=O)N(C)C)CCCO1)C(C)(F)F CC(CCNC(=O)C(C)N(C)C(c1cc[nH]n1)=O)C(F)F Cc1ccc(Cl)c(C(N2CC(OCC(=O)Nc3cncc(Cl)n3)C2)=O)c1 Cc1noc(Cl)c1CCC(=O)N(C)CC1CCCCN1C(=O)CNC(N)=O CC1(C)C2CN(C(=O)C(=O)NCC=C(Cl)Cl)CC12 Cc1cc(F)cnc1CNC(=O)NCC(c1cccc(F)c1)(F)F C(CNC(c1cn(C)nc1Br)=O)(C(C)C(C)C)NC(CC(=O)OC)=O Cc1cc(NC(C2(C3CC3)CN(C(=O)CC(C)CN(C)C)C2)=O)cc(C)c1F c1ccccn1.CC(C)(C)CC1(NC(=O)C2CC2)CC1.C(=O)(C)N.CCF C(C(CC(C)C)C(=O)N1CCOC(CCF)C1)NC(C(C)SCC)=O CC1CCC(=CC(=O)NCC2OCCC2C(=O)NOC2CCOCC2)CC1 N1(C(c2c(C)cccc2)=O)CC2CCCC(CNC(=O)C(F)C(C)(C)O)(C2)C1 C1(NC(C(C)O)=O)CCN(C(c2ocnc2C(F)F)=O)CCC1CO C1(NC(Cc2nc(SC)sc2)=O)CCCCC1NC(C1CCCN(C(C)C)C1)=O c1(C(N(C(C)CNC(=O)C=CI)C)=O)cc2n(n1)CCC2 N1(C(CSCC(=O)OC)=O)CCCC1(CC(C)C)C(=O)NC1CC1 C1(NC(CN2CCN(C)CC2)=O)CN(C(c2cnc[nH]2)=O)C2CCCC12 CCCCCC=CCC(=O)NCC=CCOC.C12(CCCC1)CCC(=O)N2 C1(C(N2CC(CCNC(CCSCCC)=O)C2)=O)CC2CC1C2 N1(C(CCC(C)=O)=O)CC2CCC(C(N3CCOC(CC(C)C)C3)=O)(C2)C1 Cc1ccc(C)c(C2=NOC(C(=O)NC(CNC(c3cscn3)=O)CO)C2)c1 N1(C(c2c(C)cc(C(F)F)nc2)=O)C2CCC1CC(CC(C)O)C2 c1(C(N2CCC(NC(C3CC(C)C3)=O)C(O)C2)=O)cc(N)c(F)c(F)c1F c1(C=O)ccc2c(c1)C=CS2(=O)=O.C1(N(C(COC(C)C)=O)C)CCCCC1.N C1(N(C(c2nc(OC)oc2)=O)C)CCN(C(C2CN(C)C(=O)N2)=O)CC1 c1(NC2CN(c3nc(C)c(Br)cn3)CC(C(F)(F)F)C2)ncnc2c(Br)csc12 c1(OCC)ccccc1C(=O)NC1CC1.C1(C)CCCN1C(=O)CCC.O N1(C(CCOCC#C)=O)C2CCC1CN(C(=O)CC1CCOC1C)C2 O=C(CCOc1cc(F)ccc1F)N=c1nc(CC(=O)O)[nH]s1 c1(CC(=O)NCCCNC(C(=O)N(CCC)CCC)=O)ccnn1C C1(C(=O)NOCCOCCF)CC1C1CN(C(c2coc(CO)c2)=O)C1 n1(CC(=O)NC2CC(F)(F)CC2)cc([N+](=O)[O-])ccc1=O.C1(C=O)CCCS1.N C12(NC(CCc3n(C)ncc3)=O)CCN(C(c3c(F)cccc3Cl)=O)CCC1C2 CCCC(CNC(=O)CCN(C(=O)C(CC(C)C)OC)C1CC1)CCO c1(C(=O)NC2CCN(C(C=CCN(C)C)=O)CC2(C)C)cnc2cnccc2c1 C(C(C(=O)N1CC(C(C)NC(C2CCCO2)=O)C1)N(C)C)OC C(=O)(C1=CC2(CCN(C(=O)C3=C(Cl)CCC(C)C3)C2)C1)OC c1(C(=O)NC2C(CNC(=O)CSc3ccccn3)CC2)cccc2cccnc12 C1(CCC)CN(C(=O)COc2ccc(CC(N)=O)cc2)CCN1C(=O)CCOC c1(CC(=O)NCCC(C)NC(C2C3CCC23)=O)ccc(F)cn1 Cc1nscc1C(=O)N(C)CC1(O)CN(C(=O)CC2CCC3CC23)C1 c1(OC)c(CN2CC3CC2C3C(N2CCC(F)(CO)CC2)=O)cc(F)cc1Br c1(C(=O)OC)ncc[nH]c1=NC(C)CC(C)NC(=O)C(C)OC C(=O)(CC(C)C(F)F)NC(C)CCCCNC(C1CC1(F)F)=O CCC(C(=O)Nn1cccn1)C1CCCN(C(=O)COC(c2cccn2C)=O)C1 C1(NC(c2nc(SC)sc2)=O)CC2CC(C1)N(C(=O)CCc1nccs1)C2 C(CNC(=O)CCCF)(C(C)C(C)C)NC(c1cn(CCCC)nn1)=O Cc1cc(=NC2CCN(C(c3cc(C)c(C)o3)=O)CC2C)c([N+](=O)[O-])c(C)[nH]1 Cc1ncc(Br)c(C(=O)NC2CC(CNC(=O)Cc3ccsn3)C2)n1 c1(CCCC(=O)NC2(c3cn(CC(CC)C)nn3)CCC2)ccc(Cl)cc1 C1(C(=O)NCCCN(C(=O)C(F)(F)CC2CC2)CC)COC(C)(C)C1 c1(CNCC2OCCN(C(c3n[nH]c(CC)c3F)=O)C2)nc(C)c(C)nc1C CC(C)(C#Cc1cn(C2CCCC2C(F)(F)F)nn1)NC(=O)C(F)=CC1CC1 Cc1noc(Cl)c1CCC(=O)NC(C)(C)CNC(=O)CCC1CCCCO1 C(=O)(C(C)(C)n1cnnn1)NC(C1CCCC1)CNC(C(C)OCC)=O C(=O)(C1=CC2(CCOC2)C1)N(CCCNC(C12CCC(CC1=O)C2)=O)C c1(N(C(C(CCNC(C(CC(C)C)OC)=O)O)=O)C)cccc2c1OCO2 C(=O)(C(=O)N=c1cc(-c2ccc(Cl)cc2)o[nH]1)NCC(C)(C)OC C1(SCC(=O)N(C2CCN(C(=O)Cc3c[nH]nc3O)C2)C)CCS(=O)(=O)C1 c1(C(=O)NC2CCCN(C(c3ncccc3Cl)=O)C2)ccc2nc(O)oc2c1 C(CN=c1nc(C)c(Br)c[nH]1)(C(C)(C)C)NC(C(CCC)CCc1ccccc1)=O c1(CONC(CNC(C(CC)n2ccnc2)=O)=O)ccc(CCF)cc1 CN1CCCC1C1COCCN1C(c1cnccn1)C(=O)NC1COC1 C1(N(C(=O)Cn2nnc(C(C)(C)C)n2)C)CCCN(C(=O)CCCN(C)C)CC1 c1(CCC)c(F)cccc1F.c1(OC)ccc(C(=O)N(C)CCNC(=O)N)cc1 C1(NC(=O)CCCCC2CC2)CC(O)CN(C(=O)C(F)(F)C(F)F)C1 c1(C(N2C(C)CC(NC(=O)CC3CCCC3(F)F)C2)=O)ccc2cccnc2c1 C1(NC(=O)Cc2cnco2)CCCN(C(c2cc(C(F)F)ccn2)=O)CC1 c1(C(N(C2CCN(C(CCCOC(C)C)=O)CC2)C)=O)ccc2[nH]nc(Cl)c2c1 C1(C(=O)NC(CNC(C2(C=C)CC2)=O)(C)CO)CCCC(O)C1 c1(C(=O)NC2C(C)N(C(=O)C(C)C(C)(F)F)CC2)ccc([N+](=O)[O-])s1 O=C1NC2(CO1)CC(C=O)C2.C(=O)C(C1CCC1)C1CCC1.CC=CC.N C1(C)(C(N(CC=C)Cc2cn(CCCCCC)nn2)=O)CCC(C)C1(C)C N#Cc1cc(Cl)ccc1NC(C1CC2CC2N1C(c1c(F)cc(F)cc1F)=O)=O C(=O)(C(CC)(CC)CC(=O)OC)NCCCN(C(C1(OC)CCOC1)=O)C C(N=c1cc(F)nc[nH]1)C1C(C(F)(F)F)CCN(C(C2(C)CCNC(=O)C2)=O)C1 c1(OC)ccccc1NC(=O)CC1(O)CCN(Cc2cnn(CC(C)C)c2)C1 c1(OCC)cccc(-c2nc(CC(N3CC(F)(F)CC3CCO)=O)cs2)c1OC N1(C(c2nnc(CC)s2)=O)CC2CCC1C(CNC(c1cnn(CCF)c1)=O)C2 C1(C(C)NS(=O)(=O)CCN(C)CC2CC2)Cc2ccccc2C1 Cc1nn(CC(C)C)c(Cl)c1C=CC(N1CCN(C(C23CCC2C3)=O)CC1)=O C1(CNC(C2(C=C)CCC2)=O)CCCC2CN(C(=O)Cc3sc(O)nc3O)CC12 c1(OC)ccc(C(=O)NC2CN(C(c3ccccc3CC#N)=O)C3CC23)c(C)n1 C#CCC(CC(=O)NC1(C2CC2)CC1)NC(c1ccnc(C)c1C)=O c1(-c2ccc(OC)nc2)ccc2[nH]c(C(=O)NCCc3ccc(C)cc3)nc2c1 CC1(C)CCCC(CC(N2CC(O)(CNC(=O)C(c3ccccc3F)O)C2)=O)C1 c1(C(N(C2CCN(C(C3CCNC3=O)=O)C2)C)=O)ccc(Cl)c(F)c1N c1(C(N(C2CN(C(CN(S(CC)(=O)=O)C)=O)C2)C)=O)ccc2nn[nH]c2n1 N1(C(C2CCC(=C)CC2)=O)CCN(C(c2ccc(Cl)s2)=O)CC(CO)C1 Cc1cccc(C(=O)NCCOC(C)(C)C)c1F.C1(O)(CC=O)CCC1.N C1(NC(COC(CC)C)=O)CCCN(C(=O)C=Cc2ccccc2)C1 c1ccc(Cl)cc1F.C(CC(C(C)C)NC(C1CC1)=O)N(C(C(C)SC)=O)C.O c1(CNC(C(C2CCCNC2)C)=O)cc(-c2ccncc2)ccc1Cl Cc1nc(C(=O)NC2CCOC(C)C2)c(C)o1.C(C1C(C)C1(Cl)Cl)=CC=O c1(OC)cncc(C(=O)NCCC(C)(C)NC(C2CC(=O)OC2(C)C)=O)c1C CC1=NOC(C)(C(=O)NCC(c2ccccc2)NC(=O)CC2(C)CC2)C1 N1(C(=O)Cn2cc(CO)nn2)CC2(CCC2)CC1C(N1CC2(CC(O)C2)C1)=O c1(C(=O)OCC)cccnc1N(C1CNCCC1O)C(=O)C(=O)O C1(CC)OCCCC1C(=O)N(C)CC1C2CN(C(=O)CC(=O)N(C)C)CC12 C(C(CNC(=O)C=CCC)C1CCC1)OC.C1(C=O)CCC1.C1CC1.N C1(C(N(C(C)C(=O)OC)CC)=O)CN(C(=O)CCc2ccncn2)CCN1C Cc1ncoc1CNCC1CCCN1S(C)(=O)=O c1(SC)cc(C)nc(N2CC3CC2CN3C(c2ccc(C)cc2I)=O)n1 c1(C(=O)N)ncc2n1CCCC2.N1(C(C2(C(=O)NC)CCC2)=O)CCC(CC)C1 Cc1cnc(N2CCCC(C(=O)NCCCN3CCNC3=O)CC2)nc1C c1(C(N(CC(CC)NC(=O)C=CC2CC2)C)=O)ccc(CO)cc1OC c1(C(=O)OC)ccc(CNc2cn(C)c(C=O)n2)cc1.c1ccc(C#N)s1.N C(C(=O)NCCC1CC1)(C(C)C)N(CC)CC.C(=O)CC.C1COC1.N N1(C(C(C)=C2CCC2)=O)CCC(O)(CNC(c2cn[nH]c2C)=O)CC1.C1CC1 C(CCCC(C)(C)C)NC(C(CCC1CC1)NC(C(C)C)=O)=O C12(CNC(C(CSC)C)=O)CCC(CC1)N2C(=O)C(n1ccc(Br)n1)C N1(C(C(C)OCC#C)=O)CC2C(C(=O)NCCCN3CCCC3)C2C1 CCC(C)C(O)CC(=O)NCCCCN(C)CC.C1(=O)CCCCOCCCN1 C1(C(N2CC(OCC)C2)=O)(OC)CCC(C)C1.c1(C=O)cnn(C2CC2)c1 N1(C(CCN2CCC(C)CC2)=O)CCN(C(=O)CN2CCC(C)(C)C2)CC1C C(=O)(CCC(C)(F)F)N1CC(F)(CNC(c2nc(C)c(C)s2)=O)C1 C(=O)(C1OCCn2ccnc21)N1CC(COC)(CNC(c2cc(C)sn2)=O)C1 Cc1cc(O)ncc1C(N1CC(NC(C2(O)CC(C)(C)C2)=O)CC(C)C1)=O c1(C(=O)NCC(C(CC)C)(C)O)coc2c1CN(C(=O)CC1CC1)C2 C1(C(C)(C)C)(C)CCN(C(=O)CC2CCCS2(=O)=O)C1.c1(C=O)ccon1.N c1(C(=O)NCCCCN(C(C23CC(CC)(OC2)C3)=O)C)cc2n(c1)CCSC2 c1(OC)ccc(F)c(C(=O)N(CCC(C(C)C)NC(C2CC2C=O)=O)C)n1 C1(OCC)CC2CN(C(C3CCCN3C(C3C(C(C)=O)C3(C)C)=O)=O)CC12 N1(C(COCC#C)=O)CC2CC(NC(c3ccccc3)=O)C1C2.CCN(C)C c1(CNC(c2n(CCOC)nnn2)C2CC2(C)C)ccc(OC)c(OC)c1 C1(NC(c2cc(CCC)[nH]n2)=O)C=CCC(C(=O)NC(C=O)C2CC2)C1.O O=C(O)CC(CNCC1CC(c2ccccc2)CO1)CO CCC(CC(=O)NCC1CCC1)c1ccco1.c1(C=O)sc(C)nc1C1CC1.N N1(C(c2csc(O)n2)=O)CCN(C(=O)Cc2cccc(O)c2F)C(C2CC2)C1 C12(CNC(c3cc(C(C)C)[nH]n3)=O)CC1CN(C(C1CSCCS1)=O)C2 N1(C(=O)CC2OCCCO2)CCC2(CCCN2C(=O)Cc2c[nH]nc2O)C1 C1(CNC(c2scc(C(N)=O)c2)=O)CN(C(=O)CS)CCO1.C1CCOC1=O C1(C=O)(COC)CCCCC1.C1CC(=O)N(C2CN(C(=O)C)C2)C1.CCF.N C1(OC)CC2(CCN(C(=O)C(C3(O)CN(C(=O)CS(C)(=O)=O)C3)F)C2)C1 N1(C(C(N2C(=O)CCC2=O)C)=O)CC2C(CNC(=O)C(C)(C)CO)C2C1 c1(OCC)cccnc1C(N1CCC(F)(CNC(=O)C(C)(C)C)C1)=O.S N1(C(C(C)(O)C2CCCCC2)=O)CCC(C)(NC(c2cccc(C(N)=O)n2)=O)C1 c1(CC)ccc(C(N2CCCC2CCCO)C(=O)NCC2CCOC2)nc1 c1(SCC(=O)N(c2ccnn2CC)CC)ccc(OC)c(OC)c1 CCCCC(O)C(C)C(=O)N1CCN(C(=O)C(C)NC(=O)C2CC2)CC(C)C1 C1(C=O)CCCC12CC2.c1(CN(CC)CC)ccc(C(=O)N)o1.C1CCC1 C1(NC(C2(N(C)C)CC2)=O)CCC(C)(C)CC1CN=c1ccnc(Cl)[nH]1 N1(C(=O)NCc2c(CNC(C)=O)cccc2)CCC2(CC1)OCCc1sccc12 c1(C(=O)NC2C(NC(C(CC)F)=O)CC2)cccc(Cl)c1C(F)(F)F CCC(CCCC(=O)N1CCC(C2CCC2)C1)NC(C1(Cl)CC1)=O C1CC2(CC2)C(=O)O1.C1(CC(=O)N(C(C)C=O)CC)CC2(CCC2)C1.N c1(NC(C)=O)cccc(C(N2CCC(C)C2)=O)c1.c1cc(C)on1.C(=O)(C)N N1(C(c2cc(C)n(C)c2)=O)CCC(C2CCN(C(c3cc(Cl)ncc3N)=O)C2)C1 N1(C(c2ccn(C(C)C)n2)=O)CC2CCN(C(c3ccc(Cl)cn3)=O)CC2C1 N1(C(C(C)CBr)=O)CC2(CCCCN2C(c2ccc3c(c2)CCCO3)=O)C1 n1(CC2CN(C(C3CCN(c4ccncn4)C3)=O)C2)cc(-c2cnccn2)nn1 C1(OC)CC2CC(Nc3cc(Cl)nc(C4(CO)CCC4)n3)CC12 Cc1nc(O)ccc1C(=O)NC1CC(NC(c2nc(Br)c[nH]2)=O)C12CCC2 C12(CNC(CSC(C)C)=O)CCC(CN(C(c3ccc4sncc4c3)=O)C1)C2 c1(C(=O)OCC)cc(C#N)ccc1NC.c12ncc(C)c(n1)NC1CSCCN21 N1(C(C(C)OCCC#C)=O)CC2CCC1CN2C(c1cc(C(F)(F)F)cn1C)=O C(=O)(CC(C(=C)C)OCC)NC1CCC(NC(c2nc(CCC)oc2)=O)C1 C1(C(=O)OCC(=O)Nc2cccc(C#N)c2)CCc2n[nH]cc2C1 CCCC(C)CC(=O)NC1CN(C(c2cn(-c3cnn(C)c3)cn2)=O)CC12CC2 C(CCC(=O)NC(c1nocc1C(=O)NC(C)C)C)OC(C)C.C1CCCO1 c1(C=O)csc(=NC2CC2)[nH]1.C1(CNC(=O)Cc2cscn2)CC2(CCC2)C1 C(CN=c1ncc(I)c[nH]1)N(C(c1conc1C(F)(F)F)=O)CC Cc1noc(Cl)c1CC(N1CCCC1C1CCN(C(=O)C#CC(=O)N(C)C)C1)=O C(C(C(=O)N1CC(C(C)(C)O)C1)NC(c1ccsc1)=O)OC(C)C N1(C(CCCC(C)C)=O)C2CCC(C(=O)NCCCCCCCO)C1CC2 C1(C=O)(C(C)C)CNC(=O)C1.c1cccc(F)c1.C(CC)N(C(=O)C)CC Nc1ccc(F)cc1C(=O)NCC1CCCC(NC(c2cc(O)cs2)=O)C1 C12(C(=O)NCCC3(NC(Cc4cnc(C)[nH]4)=O)CCC3)CCCC(CO1)C2 c1(C(N2CC(CC=C)(NC(=O)CC(C)O)C2)=O)ccc(C2CCC2(C)C)cc1 CCC1=NOC(C(=O)NCCCCCNC(=O)CS(=O)CC)C1 N1(C(C2CN(C(=O)NC)C2)=O)CC(C2(NC(=O)CCC(C)OC)CC2)C1 C1(NC(CNC(N)=O)=O)CCCC12CN(C(c1cccc(N)c1C(F)F)=O)C2 N1(C(c2c(C(C)C)noc2)=O)CCOCC(C(=O)NC(C)CN2CCOCC2)C1 c1(C(N2CCC(CCNC(=O)C(O)CC(F)F)C2)=O)c[nH]c2ncccc12 CC1CN(C(=O)C(=O)NCC(C2CCCCO2)(C)C)CCN1C1CCCC1 C1(NC(=O)NCC(C2CCCOC2)OC)CC(C(=O)O)C2CC12 c1(C(N2CCOCC(NC(C3(CC=C)CC=CC3)=O)C2)=O)n[nH]c2c1CCSC2 C1(CNC(C2(CC)CC2(F)F)=O)CCN(C(=O)Cc2cccc(O)n2)CC1 c1(C(=O)NC2CCCCN(C(COC(C)=O)=O)C2)cnc2c(c1)NC(=O)CN2C c1(OC(C(N2C(c3ccc(OCC)cc3)CCC2)=O)N)cc(Cl)c(Cl)cc1Cl c1(C(=O)NC2C(C)N(C(=O)Cn3cnnn3)CCC2)ccc(=O)n2c1CCC2 C(=O)(C1CCCCn2ccnc21)N1CC(NC(=O)OC(C)(C)C)CC(OC)C1 C(=O)(CCCC(F)F)NCC1C(OCC)CN(C(C2C3CCCCC23)=O)C1 N1(C(C2N(C)CC3(CC3)C2)=O)CCC2(CC1)CC2C(N1C2C=CCC1CC2)=O c1(C(C)O)cn(CC(=O)NCC2CC2(Cl)Cl)nn1.C12(CCC1)CC2 CC(C)CCC(O)C(=O)NC12CCCC1N(C(=O)Cc1cncnc1)CC2 c1(C(=O)NCC(CC=C)NC(C2C=CCCC2)=O)ccc(NC)c([N+](=O)[O-])c1 c1(C(=O)NC2CCC(CNC(C3C4COCC34)=O)C2)cccc(F)c1Cl c1(C(=O)NCC(C)OC)cccc(S(C)=O)c1.c1(C(=O)N)nccc(C)c1F C1(C(=O)NC2C(CN(C(C(CC)n3cccn3)=O)C)CCC2)CC2C=CC1C2 CCCCCCC(C)CC(=O)NC1CC2CC1N(C(=O)CN=c1cc[nH]cc1)C2 c1(NC2C(C#N)CN(Cc3cc(OC(F)F)cc(Cl)c3)C2)ncnc2c1CCCC2 c1(CNC(CCC=CCC=C)=O)cncc(C(=O)N(C2CC2(C)C)C)c1 c1ccc(C)c(S(N)(=O)=O)c1.Cc1cc(C#N)c(F)cc1.C1(C=O)CC1C=O C1(NC(C(CC(N)=O)NC(C2CCN(C)C(=O)C2)=O)=O)CCC(C2CC2)CC1 Cc1cc(C(C)C(=O)NC2C3CC2N(C(=O)C(C)(C)CC2CC2)C3)cc(C)c1 c1(OC)ccc2c(c1)OCC2CC(=O)Nc1cc(F)ncc1C N1(C(CN(C(c2sccc2Cl)=O)CC2CC2)=O)CC2(CCC1CO)CC2 N1(C(c2cnc(OC)s2)=O)CC(C(=O)NC2(C)CCCC2C)OC(C)C1 C1(C(N(CC(C)O)C)=O)CCC(O)CN1C(C1CC=CC(O)C1)=O C1(n2cc(-c3c(OC)cccc3)nn2)CCN(C(c2cc(OC)cs2)=O)CC1 Cc1cccc(C(=O)NC2CC(CCNC(C3CC3Cl)=O)C2)c1C(F)(F)F C#CCC(CC(F)F)C(=O)NCC(C)NC(=O)CN1CC(C)C1 c1(C(=O)Nc2c(C)cc(NC(C3CCC3(F)F)=O)cc2)cnc([N+](=O)[O-])cc1C C=C(C)CCCC(=O)NC(C)C=CC(=O)NCCc1ccnc(C)c1 N1(C(C(C2CCC2)NC(c2c(C)n(C)cn2)=O)=O)CCNC(=O)C1CCO C1(C2CCCN(C(c3cc(F)c(O)c(Cl)c3)=O)C2)(NC(C(C(C)O)(F)F)=O)CC1 c1(C(N(CC(C)(C)CNC(c2cc(C)cs2)=O)CC)=O)nn(C)cc1C c1(OC)cc(F)cc(C=CC=O)c1.C(=O)(C(F)C(F)(F)F)N(CCCCC)C.N N1(C(CC2CCN(C)C2)=O)CCCC(C2CCN(C(=O)C(C)(F)F)CC2)C1 C(=O)(C1c2ccccc2C2CC1C2)NC1CCN(C(C(CC(C)C)OC)=O)C1 C1(C(=O)NCC(C)(F)CNC(c2ccncc2N)=O)CC2(C1)CC21CC1 Cc1nn(C)c(C)c1C(=O)NCCC(C)NC(c1ccc(-c2cc[nH]n2)cc1)=O C1(F)(C(=O)NC2CN(C(C=CC(=O)OCC)=O)C2)CC=CCC1 N1(C(C(CCCC#C)C)=O)CCC2(CC1)OCCCC2NC(=O)C1=CC(C)(C)C1 CC(CNC(=O)C(O)C1CN(C(C2CNC(=O)N2)=O)C1)C(C)(F)F N1(C(c2cccc(OC)n2)=O)CC(C2CCN(C(C3C=CC=CC=C3)=O)CC2)C1 CC1=C(C)CC(C)(C(N2CC(O)(C)C2)=O)CC1.C(=O)C(O)Cc1cnc[nH]1.N c1(C(=O)NCC(CNC(c2ccc(CC)cn2)=O)O)c(C(F)F)cccc1Cl C(c1ccccn1)=C(C)C(=O)N1CC(CNC(=O)CC(C)CF)C1 Cc1nc(=NCC(C)NC(C2CC(C)C2)=O)s[nH]1 c1ccc2sccc2c1.N1(Cc2ccc(CC(=O)OC)s2)CC(O)CC1C(=O)N Cc1cc(-c2nc(-c3ccnc(C(C)(F)F)c3)n(CC3CCCO3)n2)ccc1F Cc1cc(F)ncc1NC(C1CC(O)CCN1C(c1ccc(C(C)C)o1)=O)=O C12=CC=C(C(F)=C1)C2.C1(O)(C(N)=O)CCN(C(C2(CN)CC3CCC2C3)=O)CC1 N1(CC(N2CC(N(C(C3C(C=O)CC3)=O)C)C2)=O)CCN(C)C(=O)C1.CO C1(C(N2CCC(NC(C)=O)C2)=O)CC(=O)CC(=O)C1.CC(C)CC.C1CC1.O c1(OC)c(Br)ccc(CC(=O)NCC2CN(C(C)=O)C2)c1F C1(C(=O)NC2CCC(NC(C3CC3c3ccncc3)=O)CC2)CC2CC1CC2O CC(C)CC(C(=O)NC1(C(F)F)CCC1)ONC(C1CC(=O)NC1(C)C)=O N1(C(C(COC)C)=O)Cc2n[nH]cc2C1C(=O)N1CC(C2(C)CC2)C1 C=CCCC(C(=O)N1CCCC(NC(C)=O)CC1)NC(=O)Cc1cnc(C)s1 c1(OC)cccc(C(N2CCC(C(C)(C)NC(=O)C(C)C(F)F)C2)=O)c1C C(CCCCCO)NC(c1ccc(C(F)(F)F)s1)=O.C12(C=O)CC(F)(C1)C2.N C=C=C(C)CC(=O)NCC(C)(O)C(=O)NCC(=O)N(C1CC1)CC N1(C(CSc2cccc(C)c2)=O)CCC(C)(NC(c2cncc(O)c2)=O)CC1 C1(C(=O)N)C2CCC(C2)C1(C)C.c1(OC)cc(C(N2CC(CF)C2)=O)ccc1C N1(C(COCCC=C)=O)C2CCCC1CCC2.c1(C(=O)N)cc(S(C)(=O)=O)cs1 CCCC(CCC)=CC(=O)NCCC1(OC)CN(C(=O)C(C)(C)c2ccno2)C1 C1(C(C)C)CN(C(C2(CC(F)F)CCC2)=O)CCN1C(=O)C(C)CC1CCC1 c1(C(=O)NC2C(NC(CCCOCCC)=O)COC2)c(Cl)ccc2ccncc12 C=CC(C)(C)CC(=O)NC1CC(C)C1.C1(CCC=O)CCC(C(F)(F)F)O1.N CC1(NC(=NCC2CC2CF)NC2CC2)CCCCO1 C(CCF)(C(=O)Nc1ccc(C2CC2)cc1)NC(=O)CC1(O)CCOC1 C1(OC)CN(C(C2CCc3c(ncn3C)C2)=O)CC12CCOCC2 c1nc2ccccc2o1.N1(C(C2(C=C)CC2)=O)CCC(=CCNC(=O)C)CC1.S CC(C)(C#N)CCC(=O)NCC1CCOC1C(N1CCC1CC1CC1)=O c1(NC(c2n(CCSC)nnn2)C2CC2)cc(OC)cc(Br)c1 CC(C)C(O)CC(=O)NC(c1ccc(F)cc1F)CNC(C1CCCC1C)=O N1(Cc2c(C)[nH]cc2)CCCCC(C(=O)NC2CC(F)(F)C2)C1 c1(C(N2CCCCC2CNC(C2(CO)CC2(F)F)=O)=O)ccc(Br)cc1F Cc1ccc2c(C(=O)NC(CNC(C3OCCC3C)=O)CC(C)C)n[nH]c2c1 c1(C(N2C(C)(COC)CC(NC(c3occc3C)=O)C2)=O)nc[nH]c2nccc1-2 C(=O)(C(C)(CO)OC)N(CCCNC(c1coc(C)c1)=O)CC Cc1ccc(N2CCN(C(=O)CCNCC3CC3)CC2)nc1 Cc1ccc(C(N2CC3CCC3(CC(=O)NCc3nncn3C)C2)=O)nc1O CC1CN(C(=O)CCCc2ncco2)CC(C)C1NC(c1cc(O)cs1)=O c1(C(N2CC3N(C(c4c(C)ncnc4)=O)C3C2)=O)c(F)cc(C#N)cc1Cl c1(NC)ccc(C(=O)OCc2ccccc2NCc2ccn(C)n2)cc1 CCC(CC(C)C)C(=O)NCC1CN(C(=O)CC2CC2C)C1 Cn1cc(C(N2CCCC2(C)CNC(=O)CCc2ccc(Cl)nc2)=O)n(C)c1=O C(C)(CNC(=O)CNC(=O)C(C)CSC)(CO)OC c1(SC)ccc(N)cc1C(N1CC(NC(c2cnns2)=O)CCC1C)=O c1(CNC(CC2(CC)CCC2)=O)cccc(C(=O)NCC(C)C(C)(C)C)c1 C(c1ccc2c(c1)OCCO2)=CC(N1CCC2(CCC2)C1)=O.C(C(=O)N)=CC c1(-c2cn(C(C(=O)N(CCCCC=C)CC)C)nn2)c(F)cccc1Cl N1(C(COC)=O)CCOC(C)C1C(=O)NCCC(C)C(F)F c1(C(=O)NC(CC)(C)CNC(=O)COc2ccsn2)ccc(C#N)c(Cl)c1 Cc1cc(=NCc2cc(F)cc(Cl)c2)[nH]c(N2CCOC(COCC3CC3)C2)n1 C=C(C)CC(C(=O)N1CC2(C1)CN(C(=O)Cc1c(F)cncc1Cl)C2)OC C1(C(N2CCOCC(CNC(C(NOC)=O)=O)C2)=O)CC2(C1)CC1(CC1)C2 CS(=O)(=O)C(C)C.C1(CC(=O)N)CC2C=CC1CC2.C(=O)CCn1cncn1 C1(C#N)(C(N2C(C(C)NC(=O)Cn3ccnn3)CCC2)=O)CCCO1 c1(C(=O)NC(C)CC2CN(C(=O)C(C)n3ccnc3)C2)ccccc1Cl N1(C(C(C)Oc2cccnc2)=O)CCC(N)CC12CCC2 Cc1ccc(C(=O)NCC(O)CNC(=O)CSc2cccc(F)c2)c(N)c1Cl N1(CC(=O)OCC)CC2CCC1CN2C(C1CCCC(OS(C)(=O)=O)C1)=O Cc1ncc2n1CCC(C(=O)NC1CCC(CCN=c3[nH]nco3)C1)C2 C1(CNC(=O)CCF)CC(C(F)(F)F)CN1C(c1ccsc1Cl)=O Cc1cccc([N+](=O)[O-])c1NC(N1CC=CC1CNC=O)=O.C(C)(C)C C(=O)(C1CCc2nccn21)NC(CN(C(=O)C=Cc1cccc(Cl)c1)C)(C)C C1(NC(C(CNC(C(=O)N(C)C)=O)CC2CC2)=O)CCCC(C)(C)C1 C1(NC(C(c2n(C)ncc2)O)=O)CC1C1CCCN(c2ncc(F)cn2)C1 C(CC(C)(C)C#N)(c1nnnn1CCOCC)NCc1cc(CC)nn1C C1(C=O)CCS(=O)(=O)C1(C)C.Cc1nn(CCO)c(C)c1C(=O)N.C1CC1 C(=O)(C1Cc2ccccc21)NC1C2N(C(c3c(N)c(F)ccc3Cl)=O)C(CC2)C1 c1(CC(=O)N)cn2cc(F)ccc2n1.N1(C(C2CC(C#C)(O)C2)=O)CCCC(O)C1 c1(C(C=O)C)cc(C)cc(C)c1.N1(C(CNC(=O)OC)=O)CCCCC1C.N C1(NC(C2(N(C)C)CC2)=O)CC2CCCC(C1)C2NC(c1ncccc1F)=O C1(NC(c2cc(C)oc2)=O)CC2CCC(C1C)N2C(=O)Cn1cc(Cl)cn1 c1(-c2[nH]ccc(=NCc3cnc(SC)nc3)c2)cccc2c1COC2=O c1(CC(=O)NC2CN(C(=O)CCc3ccc[nH]3)CC2F)cc(Cl)ccc1Br c1(NC(C(C2CCC(CO)CC2)N(C(C)C)C)=O)ccc2c(c1)OCO2 c1(OC)c(C(=O)NCC2CN(C(=O)CCCC)C2)c(C)nn1C.C(C)=O.O C1(NC(C2CCN2C2CCCC2)=O)CCN(c2ncncc2I)CCC1CO C(=O)(CCP(C)(C)=O)NC1CCCC(CN(C(C2CCCN(CCC)C2)=O)C)C1 C(=O)(C(C)(C)CC#N)NC(C1CCOC1)CNC(c1n(CC)nnc1)=O C(C(C(=O)N1CCC2CC12)C(C)(C)C)NC(c1nccc(C#C)c1)=O C12(NC(c3n(CC)ccc3)=O)CCOC(C)(C1)C2.c1(C=O)cc2scnc2[nH]1 N1(CC2([Si](C)(C)C)CC2)CCC(F)C(NCc2ccccc2)C1 c1(C(=O)NCC2CC3(CN(C(CCCCC)=O)C3)C2)cc(Cl)cc(C)c1N C(C(O)CN=c1[nH]c2c(cc1C#N)C(=O)CCC2)N.CCC(C=O)C(C)(C)CC N1(C(CCC(=O)c2c(C)ccs2)=O)CCC2CCN(C(=O)C3=NOCC3)C2C1 c1(C(=O)NC(C(C)OC)C(F)(F)F)ccc(CO)cc1F c1(CC(=O)OC)ccc(Br)c(NC(=O)C(=O)N)c1.C1(C)NC(=O)NC1=O CC1CN(C(=O)CC2CC=CC2)CC1NC(=O)C(c1ccccc1)C1CC1 c1(OC)cc(CC2CCOC(C)C2)nn1C.C12CCCN(C1)CC(=O)NC2C CCCC(CCCO)C(=O)N(C1CCN(C(=O)CS(=O)(=O)C2CC2)CC1)CCC c1(-n2ccc(C(=O)NC(CC)CN(C)C=O)n2)ccc(Cl)cc1.c1(C)cncn1C N1(C(C2CCC(=O)O2)=O)CCC(=CCNC(C2CCOC2)=O)CC1 C1CN(C(C2CCN(C)C2=O)=O)CC(C)(C)C1.c1(CC)cc(C(=O)N)nn1C.C c1(OC)ccc(C)c(C=O)c1N.C1(C(N(CC(C)O)CC)=O)COCC1(C)C.N C1(NC(C(C)=C2CCCC2)=O)C2CC1CN(C(=O)COc1cccc(C)c1)C2 C1(CNC(=O)CSc2cccnc2)CCCC(NC(c2ccccc2S)=O)C1 c1(C(=O)NCCC(C)NC(CCCCSC)=O)cc(C)c(Cl)c(N)c1 C1(NC(CC(CC)OC)=O)CC(O)CN(C(=O)CCCCCc2cccs2)C1 C1(C(C=O)O)CCS(=O)(=O)CC1.CC(C)(C)C=CC(=O)N.C1(CC)CC1 N1(C(C(F)=CCC)=O)CCN(C(C2CCC2C)=O)CC1CS(C)(=O)=O C(=O)(C(O)C(C)C)N.C1CCCO1.C(C(=O)N(CC)CC)N(CC)CC C1(C(=O)NC(C(=O)N(CC)CC)C)CN(C2CCOC2)CCC1O C1(NC(=O)CCc2cccnc2F)CS(=O)(=O)CC1NC(c1cc(Cl)c[nH]1)=O C1(CC)CN(C(C23CC(C#N)(C2)C3)=O)CCC1NC(=O)CCCCCOC c1(N(C(c2nc(C)c(F)cc2)=O)CC2CCCNC2)ncc2cc(Br)ccc2n1 c1(OCCCOC)ccc(NC(=O)NC(CO)CC(O)c2ccccc2)cc1C C1(O)(CC(N2CC(CNC(C(CC)C)=O)C(C)C2)=O)COC(C)(C)C1 Cc1cc(F)c(C(=O)NC(CNC(c2cocn2)=O)CC(C)C)cc1Br CC1Oc2ccccc2OC1C(=O)NCCC(=O)NCc1ccc(O)cc1 c1(C(=O)NCCOC2CN(C(CC(C=C)C)=O)C2)cccc2ccnn12 c1(CN(C)C)cc(C(=O)NC2CCC(NC(=O)C(F)n3cccn3)C2)no1 C1(C(=O)OC)CCCC(C)N1Cc1nc(C(C)(C)C)cs1 C#CCCCC(C)C(=O)N1CCC(C)(C)C1CNC(C1CCC(C=O)CC1)=O.N C=CCCC(O)CNC(=O)CN(CCC)C(C1CC(=O)CS1)=O Cc1nc(NC(C2C3CN(C(c4ncccc4Br)=O)CC23)=O)ncc1Br c1(C2C(C(=O)NC(CC=C)CNC(c3[nH]nnc3C)=O)C2)ccc(F)cc1 C1(CCNC(C(c2ccc(Cl)cc2)(C)O)=O)CCCN(C(C2CCC(=O)O2)=O)C1 C1(C(=O)NC2(CC)CC2)(CCNC(=O)OC(C)(C)C)CCOCC1 c1(CC)ccc(C(=O)NC)c(C)n1.C12CCC1CCN2C(=O)CC.C(=O)CO C#Cc1ccc(CC(N2CC(NC(=O)COC(F)(F)F)C(C)C2)=O)cc1 C1COC2(CCN(C(c3cc(N)nc(Cl)c3)=O)C2)C1.C(C=O)N(S(C)(=O)=O)C c1(C(N2CCCC2c2ccc(F)cc2)C(=O)NCCSC)ccc(C#N)nc1 N1(C(C(CC)n2cccn2)=O)CC(CNC(c2ncccc2C)=O)C(C)(C)C1 c1(C(=O)NCC(C)(CO)NC(Cn2c(=O)ccc(C)n2)=O)nccn2nccc12 Cc1cc([N+](=O)[O-])cc(C(=O)NC(C)CNC(C2CCC(C)C2)=O)n1 c1(C(=O)Oc2cnc(OC)nc2)cc(F)cc2ccccc12 C1(NC(c2n(CC)cnn2)=O)CN(C(c2cc(F)n(C)n2)=O)CC2(CCC2)C1 CC(C)CC(C)CC(=O)NCC1(C2CCN(C(=O)C(C)(C)CCC#N)C2)CC1 Cc1c(CN(C)C(C2CC2C(C)NC(c2cnsc2)=O)=O)cnn1C n1(C2CC(C(N(CC(F)F)CC)=O)C2)cc(-c2csc(C)n2)nn1 N1(C(C(=O)NC(CC)(C)C)C)CCC(NC(C23CCCC(CO2)C3)=O)C(C)C1 CCCC(C)(C)C(=O)NC1CC(C(F)C(=O)NCCC(O)(CC)CC)C1 N1(C(c2cccn(C)c2=O)=O)CCC2CCN(C(c3cc(F)ccc3O)=O)C2C1 Cc1c([N+](=O)[O-])cc(N2CCC(C(F)(F)F)CC2)c([N+](=O)[O-])c1C C1COC2(CCN(C(=O)C(=O)N(C)C)C2)C1.Cc1ccc(C(=O)N)c(C2CC2)c1 Cc1[nH]nc(Br)c1C(=O)NCC1CC(NC(c2c[nH]c(C#N)c2)=O)C1 C1(NC(C(C)OCCOC)=O)CCN(c2ncnc(CC)c2F)CC1O C1(NC(C2(CC#C)CCOC2)=O)CCCN(C(=O)C=Cc2nnn(C)n2)C1 C1(N(C(=O)C2=CCCC2)C)CCN(C(=O)CC(C)C(C)(C)C)CC12CC2 C(=O)(C1CSc2ccccc21)NCCN(C(C)C)C(C1CCN1C1CC1)=O C1(C(=O)OC)CCCN(CC(N2CCCCC2CCNC(=O)C)=O)C1.C1CC1 C1(C(N(C)Cc2ccncc2)=O)CN(C(c2ccoc2C2CC2)=O)CCC1(C)C N1(C(CCN(C)CC)=O)CC(CNC(=O)CCSc2ccccc2Cl)CC1C CC1CN(C(=O)C(C)(C)CN(C)C(C2CC2(C)C(F)F)=O)CC1(F)F C(=O)(C1Cc2ccccc21)NCC1C2N(C(CC(C)n3cccn3)=O)C(CC2)C1 Cc1c(C(=O)NC2CCCC(NC(c3cc(-c4cccs4)[nH]n3)=O)C2)cnn1C C1(NC(c2c(SC)c(F)ccc2)=O)CCC2CCN(C(=O)C(F)(F)C(F)F)C1C2 C1(CN(C2C(SC)CCC2)C)CC(N)C12CCC2 C1(NC(c2c(Cl)cnc(OC)c2Cl)=O)CCC12CCN(C(c1cc[nH]c1)=O)CC2 N(C(=NCCCCl)NCC1CC(=C2CC2)C1)Cc1nnn(CC)n1 Cc1c(C(=O)NC(C)CC(C)NC(=O)COC2CCCCC2)nn(C)c1Br c1(C(=O)NC2CC(NC(c3cncs3)=O)C23CCC3)coc2cc(F)cc(F)c12 C(=O)(C1CCCc2sc(=N)[nH]c21)NCC(CNC(C1(CCC=C)CC1)=O)C c1(C(N2CCN(C(C(C)O)=O)C3C2COC3)=O)cc(F)c(Cl)c([N+](=O)[O-])c1 C#Cc1cccc(C(=O)NC2CCN(C(=O)C(C)(C)CCC)CC2C)c1F N1(CC(=O)NC(C)C)CC(NC(=O)CC(C)O)C(O)C1 Cc1cnc(C=O)cc1C.C1(CC(=O)N(C2CC2)C)CC2(CC2)C1.C1CC1 c1(CN(CCNC(=O)CCc2cc(C)n(C)n2)CC)c[nH]c2ncccc12 Cc1cnc(Cl)[nH]c1=NCC1CN(C(c2ccn(C(F)F)n2)=O)CC1(C)C C1(C(N2CCN(CC(=O)NCc3ncc(C)s3)CC2)=O)(OC)CCCOC1 N1(C(Cc2c(C)oc(C3CC3)n2)=O)CCCC(N2CCOC2=O)CC1 c1(CC)nnc(C)cc1C(=O)NCCCN(C(=O)C(C)C)C1CC1 CCCCC#CC(C)(C)NC(C12CCCC1CCN2C(=O)CCCC(=O)NC)=O c1(C(=O)NCC2C3CN(C(CC4C(C)(C)C(O)C4)=O)C2C3)cc2n(n1)CCCO2 c1(CC)nc(Cl)c(F)c(=NCC2CCN(C(c3ccnc(Cl)c3F)=O)C2)[nH]1 c1(SC)ccc(CCCC(=O)NCC2CC(NC(c3csc(C)n3)=O)C2)cc1 N1(C(c2c(C)[nH]c(=N)s2)=O)CC2CCN(S(=O)(=O)Cc3ccc(F)cc3)CC2C1 CC1(C(=O)NCCC2CC(NC(C3(O)CCOC3)=O)C2)CCNC1=O C1(CNC(CC)=O)CN(C(C2(CF)COC2)=O)CCN1C c1(NC(CCCNC(C=C=C(C)C)=O)=O)c(C)cccc1O N(C1CCOc2ccc(Br)cc21)C(=O)C(N1CC2CC(F)(F)C2C1)=O C12(C(=O)NC(CC#CC)CO)CCCC1CCN2C(C1SCC=C1C)=O C1(CCC)CN(C(=O)CC2(C(F)(F)F)CC2)C1.CCCCOCC(=O)N N1(C(C2CCC(C)O2)=O)CCC(C(=O)NC(C2CC(=C)C2)C2CCCC2)C1C CC1(CNC(=O)CC2CC(=O)C2)CCN(C(=O)C(O)C2CC2)C1 C1(c2cn(C)nc2)CS(=O)CCN1C(=O)CCc1ncc(-c2ccc(F)cc2)o1 c1cc(C(=O)NC)n(C)n1.C1(CCC)(C=O)CCCC1.C1CN(C(N)=O)C1 CCC(Cc1ccccc1)C(=O)NC1CN(C(C2CCCO2)=O)CC1C(F)F c1(C(=O)NC2COCCN(C(C=C(CC)C)=O)C2)cc(OC)cc(Cl)c1F c1(C(N(C2CCC(NC(CN(C)CCO)=O)CC2)C)=O)ccc([N+](=O)[O-])s1 C(C)(CCC(=O)N(C)CCOCC)NC(C(C)OCC=C)=O c1(C(=O)N)cocn1.c1ccccc1.CC(C(=O)NC1CCC1)OC(C)(C)C C1(C(=O)N)CC2CCC(C1)C2O.C1(CNC(CCNC(=O)CO)=O)CCCCC1 CCC(C)CCCCC(=O)NC(CNC(=O)Cc1ccc(C)c(C)c1)CCOC CC1CCCN(C(=O)CCCNC(=O)CN2CCSCC2)CC1 C12(NC(c3n[nH]c4c3COCC4)=O)CCCC1N(C(C1CC3(CC3)CO1)=O)CC2 c1(CNCC2CCC(C(=O)NCCNCCO)C2)ccc(Br)c(Cl)n1 c1(OC)ccc(C(=O)NCC2CCCC2NC(=O)CC(O)C(C)C)cc1O Cc1onc(CC(N2CC(NC(c3cc(Cl)on3)=O)C(C)C2)=O)c1C#N N1(C(C)=O)CCOCC1C(=O)NCC1CC1NC(=O)C(C1CCCCC1)F C1(C#N)(C(=O)NCC(CCNC(c2ccc(CC)[nH]2)=O)OC)CC(C)C1 Cc1cncc2cc(C(=O)NC3CCN(C(C4CC(O)C4)=O)C(C)C3)sc12 C1(CNC(c2c(C)cco2)=O)CN(C(=O)C(C)P(C)(C)=O)CC2(CCC2)O1 C(=O)(C1CNC(=O)c2ccnn21)NCCCNC(C(c1cccnc1F)(C)C)=O N1(C(c2n(CCC)ncc2)=O)CC=CCC1C(=O)NCc1nc(C(C)C)n[nH]1 N1(C(C2C(CC)CCN2C(=O)COC(C)(C)C)=O)CC2CC(C1)C2(C)C C(=O)(C(CCN(C)C)NC(=O)CC1(O)CCCC1)N(C)Cc1cncn1C C(=O)(CCCC(C)=O)NCC(CC)N(C(c1c(CC)nns1)=O)C CC1=C(C(=O)NC(C)C2CCC2)CCS1(=O)=O.c1(C=O)ccn(CCO)c1C.N C(=O)(N=c1cc[nH]cc1[N+](=O)[O-])Nc1cc(C(C)C)cc(Cl)c1 C(=O)(CCS(=O)(=O)CC(C)C)N(C1CCC1)C.Cc1n[nH]c(C)c1C(C)C(=O)N CC1CCCc2cc(C(=O)NCCCCn3cc(CCCO)nn3)nn21 C(=O)(C1CCc2ccccc21)NCC(C(=O)NCc1cnco1)N(C)C c1(CC(C)C(=O)NC(C2CCN(C(C3(F)CCC3)=O)C2)(C)C)ccccc1F C1(CNC(c2ccc(CC)cc2)=O)CC2CCC1C2.c1(C=O)cnc(S)n1C.N c1(SC)cc(C(=O)NC2CC2CNC(C2CCSCC2)=O)cc(SC)c1 C12(C(N(c3c(C)cccc3)C)=O)CCN(C(=O)CC(=O)N(C)C)CCC1C2 C(=O)(C(O)CC(C)(C)C)N(CCCCC(=O)NCCNC(=O)C(C)(C)C)C C1(NC(COc2cncc(C)c2)=O)CN(C(=O)CSc2ccccc2)CC2CC12 N1(C(C(n2ncc(C)c2)C)=O)CC2CC1CN2C(c1cc(N)ccc1F)=O C(=O)(C(C(C)(C)C)N(C)C)NC(COC)CNC(=O)C(O)C1CCC1 C1CCCCN1C(=O)CC1CCCC(=O)C1.C1(C(N(C)C)=O)CCC1.C1CC1 C1(NC(C(CNC(CCC(=C)Cl)=O)N(C)C)=O)CC(C)(C)OC1(C)C CC1(C)CC(NC(C2CCCN(c3ccc(Cl)cc3Cl)C2=O)=O)CN1C(=O)CN C1CN(C(=O)CS(=O)(=O)N(C)C)CCC1C.Cc1csc(C=CC(=O)NC)n1 C=CCC(C)(O)C(=O)NCCCC(O)C(=O)N1CCC(C(C)C)(CO)C1 Cc1ccccc1SCC(=O)NCC1CC(NC(c2cocn2)=O)C1(C)C Cc1ccc(C(=O)NC(C(=O)NCCc2ccccc2C)C2CC2)cc1 c1(Cn2nnc(-c3c(C)ccc(Cl)c3)n2)c[nH]c2ccccc12 N1(C(C(F)=C)=O)CC2(CCCO2)C1.c1ccccc1.C1(C=O)CCC1C(N)=O.CC c1(C(=O)NCC(CN(C)C(c2cc(Cl)n[nH]2)=O)(C)C)cc2occc2n1C C1(CC)CC(F)(F)CN1C(=O)CCC1CC1(C)C.C(C=O)SCCOC.N N=c1[nH]c(C(=O)NC2CN(C(=O)CC3CCCOC3)C2)c(C(F)(F)F)s1 c1(C(N2CC(NC(C3CCC(=O)N3)=O)CC(C)C2)=O)cc2ncccc2[nH]1 N1(C(C2CCC(CC)C2)=O)CCc2[nH]nc(CNC(=O)CC(F)(F)F)c2C1 c1(CN(CCNC(C=CC)=O)C(C2(C)COC2)=O)ccccc1 C(N=C(NCc1cn(C2CC2)nn1)NC1CCOCC1)C1C(CCC)CCC1 C1(NC(c2nn(C)c(C3CC3)c2)=O)CS(=O)(=O)CC1.c1(CC=O)ccno1 N1(C(c2c(F)ncc(-c3c(OCC)ccc(Cl)c3)c2)=O)CCc2oc(C)nc2C1 C1(C(N2C(CN(C)C(c3cn(C)nc3O)=O)CCC2)=O)CCC(C)(C)OC1 Cc1ncc(CC(N2CCCC2CCNC(=O)Cc2cnns2)=O)s1 c1(CN(C(C)Cc2cccc3ccsc23)C2CC2)ccc(C#CC2CC2)cc1 N#Cc1ccc(Cl)c(NC(C2CC3(CC3)CN2C(c2cnccc2Br)=O)=O)c1 CC(C)C(O)(C(=O)N1CCCC(CNC(=O)CCc2cn[nH]c2)C1)C(F)(F)F C1(C(=O)NC2CCN(C(=O)Cc3cc(F)cc(Cl)c3)C2)CC2(C1)CC21CC1 C1(C(=O)NCCOCCC)N(C(C2CCCOC2)=O)CCC1(C)C n1(CC(=O)NC2CCCC2NC(=O)C(=Cc2c[nH]cn2)F)cc([N+](=O)[O-])cn1 CCCC(F)(F)F.c1(C=O)ccc([N+](=O)[O-])s1.c1(COC)ncc(C(=O)N)s1 N(C(=NCC1CCC1)NC1CCC1)C1CC(C)SC1.c1cscc1Br N1(C(C2CCN(C(c3n(C)nc(Cl)c3)=O)C2)=O)C2CCC1CC(CO)C2 c1(NCC(CNC(=O)NCC=C)C)ccc(C)cc1OCCN(C)C C1(NC(C2CC2[N+](=O)[O-])=O)CCN(C(=O)CC2CN3CCN2CC3)CC1F c1(C(N2C(C)(CC)CC(NC(C3(CF)COC3)=O)C2)=O)ccc2cnnn2c1 N1(C(c2nccc(OC)c2F)=O)CCN(C(=O)Cc2cn(C)nn2)CC(C)(F)C1 Cc1cncc(C(=O)NC2CCC2NC(C2CCOC(=O)N2)=O)c1Cl c1(CN2CC3(C(C(=O)Nc4cccc(C5CC5)c4)C3)C2)ccc2c(c1)CCCC2 C12(C(=O)Nc3cc([N+](=O)[O-])c[nH]3)CCC1CN(C(=O)C)C2.C1CC2CC2C1.O N1(C(C2C(CC)CCC2)=O)CC2CCC(NC(c3cc4c([nH]3)CCC4)=O)CC2C1 C(=O)(NNC(=O)C(C)Cc1ccc(Cl)cc1)c1ccc(C)c(C)c1 c1(CSC)c(C(N2CCC(NC(c3ccccc3)=O)C2C)=O)oc2ccccc12 N1(C(C(COC)C)=O)CCC(NC(=O)Cc2ccnnc2O)C12CC2 C12(NC(C3(NC(CC4CC(SC)C4)=O)CC3)=O)CCCCC1OCC2 c1(C=O)cn(C)c(=O)n(C)c1=O.c1(CC)cnccc1C(=O)NC1CCC1.C C(=O)(C(C)(C)c1ccc(Cl)s1)N(CCC(C)NC(=O)CN1CCCC1=O)C C1(CC(=O)NCCCC(C)O)N(C(=O)C(c2ccn(C)n2)C)CCC1(C)C C(=O)(C(Cc1ccccc1)C(F)(F)F)NCCCOC(C(=C)C)=O c1(C(C(=O)N(CCCC)C)F)ccc(C(F)(F)F)cc1.C(=O)C(F)=C(C)C.N CCCC(CC)C(=O)NCCCOC1(COCCC(=O)O)CCOC1 c1(CC(N2CC(CC=C)C2)=O)nc([N+](=O)[O-])n[nH]1.C1(C=O)CC(N(C)C)C1 c1(C(C(=O)NCCCC2CC2)N(CC=C)C(C)C)nc(F)ccc1Br C1(NC(C2CC=CCC2)=O)CCCCC1NC(C1(C2CCCO2)CCCC1)=O C#CC(C)(CC)NC(=O)CC1(C)CN(C(=O)C(C)OCCOC)C1 CC1(C(N2CCOC(C(F)F)C2)=O)CCC12CCC2 Cn1nccc(C(=O)NCC2CC3CCC2N3C(=O)CN2CC3CCC2C3)c1=O C12(CNC(=O)CCCC(F)F)CC3CC(CC(C3)C1)C2.c1(CC=O)ccco1.N N1(C(c2ccc(C)s2)=O)CC2CCC(C1)C(NC(=O)C1=CCC(C)CC1)C2 c1(C(N2C(CCNC(CC(CCC)O)=O)CSCC2)=O)cc(C)[nH]c2ncnc1-2 C1(NC(C2CCC(CC)CC2)=O)CC(F)CN(C(=O)C(c2ccc(C)cc2)O)C1 N#Cc1c[nH]c(C(N2CC3C(C(=O)NCc4cccc(I)c4)C3C2)=O)c1 C1(C(=O)NCC(CC)NC(=O)CSCCOC)CC(=O)NC(=O)C1 C1(CC)(OC)CN(C(c2cn(CCNC(=O)C(=O)N)nn2)=O)C1.C1CC1 C1(c2n(CCOC)cnn2)CCCN(C(=O)N(c2ncncc2Br)C(C)C)C1 N1(C(Cc2c(C)non2)=O)CCC(NC(c2cc(CF)on2)=O)C1(C)C N1(C(C(CC)CC)=O)CCN(C(c2ccc3c(c2)OCCO3)=O)C2CCCC12 Nc1cccc(-c2cn(CC3CCCN3C(=O)CC3CC3C3CC3)nn2)c1 C(=O)(C1=NOC(C)C1C)N(C)CC1CCCN(C(Cn2ncc(C)c2)=O)C1 CCC(CCCC(=O)N(c1cccc(C)c1C)C)NC(=O)CSC(F)(F)F Cc1nccc(C(=O)NC(CNC(=O)Cc2c[nH]ccc2=O)C2CC2)c1Cl C1(NC(N2CCOC(c3nn[nH]n3)C2)=O)CCC(Oc2ccccc2)CC1 CC(C)(O)C#CC(=O)NCC1(NC(c2cncc(-c3ccncc3)c2)=O)CCC1 Cc1cc(C)c(C(N2CCC(C(=O)NOC3CC3)C23CC3)=O)cn1 c1(C(=O)NC(CNC(c2[nH]n(C)c(=O)n2)=O)CO)cccc2nn[nH]c12 C1(NC(CC=C=C)=O)CN(C(=O)CC(C(F)F)c2ccccc2F)CC1C1CC1 N1(C(COCC)=O)Cc2ccccc2C(CNC(=O)CCO)C1.C(=O)C(C)C.N N1(C(CC2(O)CCCN(C)C2)=O)CC2(CCN(C(=O)C3=NNC(=O)C3)CC2)C1 N1(C(c2cccc(CCC)c2)=O)CCC2CN(C(=O)Cc3cccn3C)CC2C1 c1(CC)nc(NC(=O)Nc2ccc(-n3cc(Cl)cn3)cc2)cc(Br)n1 N1(C(C2C(C(=O)OC)C2)=O)CC2CCN(C(c3cnc(OC)cc3C)=O)CC2C1 CC(CNC(C1(CCF)CC1)=O)(Cn1cccn1)NC(c1cnsc1)=O c1(NC(CC2CCCN(C(C(C3CCC(=O)N3)C)=O)C2)=O)ccc2c(c1)CCO2 CCCCCCCCC(=O)NC(c1cn(C)nn1)C(=O)N1CCC1CC(C)(C)C CC1(NC(C2C3CCN2CC3)=O)CCN(C(c2cccc(C(F)F)c2)=O)C1 C=CC(C)CC(=O)NCc1cn(C2CCCN(C(C3(CO)CCC3)=O)C2)nn1 N1(CC=CC(C)C)C2CN(C(=O)Cc3sccc3C)CC12.CC1=CCC=CC1 c1cc(F)cc(Cl)c1.C1(C(=O)NCC2CCN(C(=O)C)C2)CC2(CCO2)C1 C12(C(=O)NCC3(C)CCC(O)CC3)CCCC1CN(C(=O)C1=CCCSC1)C2 C1(CC(=C)Cl)NC(=O)N(C(C)Cc2ccc(F)cc2)C1=O C(=O)(CC(C)n1ccnc1)N(C1CN(C(C(=O)NCCOC)=O)C1)C C12(C(=O)NCC3(C)CC(C)(C)C3)CCCC1CN(C(=O)Cn1cnnc1)C2 C(=O)(C=CS(C)=O)NCCCCN(C(C(C)N(C(C)=O)C)=O)C CC1CCCN1CCNC(c1nnc(-c2ccns2)o1)=O C1(C(=O)N)CCCC12OCCO2.c1(C(N(C(C)C)CC)=O)cc2n(n1)CC(F)C2 CC1CCN(C(=O)C(C2(O)CCCC2)F)C(C)C1NC(c1ccc(CO)s1)=O C1(C(=O)NC2C(C)CN(C(C3CCCN3C)=O)C2)CN=C2N=CNN2C1 N1(C(C(c2cn(CC)nc2)=O)=O)CCN(C(=O)CC2CCCCC23CC3)CC1C c1(C(=O)OC)nnc(NC(=O)NC(C)Cn2ccnn2)s1.c1cnn(C)c1 C1(C(C)C)(C(=O)N(C)CC2CC2(F)F)CCN(C(=O)CC2(O)CCCC2)C1 C12(C(=O)NCc3[nH]nc(C(C)=O)n3)CCCC1CCN2C(=O)Cn1ccnc1C CC(CC(=O)N1CC2C(CNC(c3ccc(C4CCC4)nc3)=O)C2C1)C(F)(F)F C1(NC(c2c(CCC)n[nH]c2)=O)CC(CC(=O)NCc2ocnc2C)C1(C)C CC(C(=O)N(C)CC=CC(=O)NCC(N1CCOCC1)C)S(N)(=O)=O c1(OC(C)C(N2CC3CC2CN3C(=O)CNC=O)=O)ccc(Br)cc1F N1(C(C2C(C)(C(C)C)C2)=O)CC2(CCCO2)C1.C1(CC=O)CN2CCC1CC2.N c1(CC)cc(OC)cc(OC)c1C(=O)N.C(=O)C(C)(CC)C(N)=O.C(C)CC c1(C(N2CCC(COC)(NC(C3CC34CC4)=O)C2)=O)ncc2ccccc2c1N CN=c1nc(N(CC(C)C)C)[nH]c(N2CCC(c3nc4ccccc4[nH]3)CC2)n1 c1(C(N2CCC(C(C)NC(C(C)P(C)(C)=O)=O)CC2)=O)cc(F)c(F)c(F)c1N c1(C(C)NC(c2c(C(C)C)cnn2C)=O)nnc2n1CCCC2 C(=O)(CS(=O)(=O)C1CC1)N(CCCN(C(=O)CCc1ccc(C#N)cc1F)C)C c1(C(c2nnnn2CC(F)F)NC2(C)CCCC2)ccc2ncsc2c1 c1(CC)c(C(=O)NC(CNC(C2CCOC2C)=O)C(C)C)sc2ccccc12 c1(C(=O)NC2C(C(C)(C)O)C2)cncc(CNC(=O)CO)c1.C1CC1 C1(C(=O)NCc2cc(C)nn2C)CCC(O)CN1C(=O)Cc1ccc[nH]1 C(CCC(C)(C)C(=O)N1CCC1(C)CCO)NC(C(C)=CC=C)=O C(=O)(C(CC(C)(C)F)NC(=O)CC1CCC1)OC.c1(C=O)nc(Br)ccc1C c1(CNc2c(C(=O)OC)sc(I)c2)cc(Br)ccc1[N+](=O)[O-] Cc1cccc(=O)n1CC(C)(O)C(=O)NC1CCC1C.c1(C=O)ccc(Cl)o1 N1(C(=O)Cc2cn[nH]c2)CCN(C(c2ccc(C3CCCCC3)s2)=O)CC1 C#CC12CCC(C(N3CCC(O)C3)=O)(CC1)CC2.c1(C(=O)N)ccc([N+](=O)[O-])[nH]1 c1(C(=O)NC(CCNC(C2N(CC)CC2)=O)(C)C)cnc2c(c1)nnn2C CC(CC(N)=O)C(=O)N1CCC(C(C)NC(=O)Cn2ccc(C3CC3)n2)CC1 c1(CC(=O)NC2CC(NC(C(C=CC)O)=O)C2)ccc(-n2cnnn2)cc1Cl CN1CC(C(N2CC3C(CNC(c4cc(Br)no4)=O)C3C2)=O)NC1=O C1(C2CCCCC2)(C(=O)NC2CCN(C(C3C(C)(CC)C3)=O)C(C)C2)CC1 C1(C(C)C)C(C(=O)NCC2C=CCOC2)CCN1C(=O)CC1CCC1 Cc1noc(NC(C2CN(C(c3cc(Br)ncc3Br)=O)CCC2O)=O)c1C#N N1(C(C2(c3onc(C)n3)CC2)=O)CC2CNCC1COC2 CCC(C)(CN(C)C(C1C=CC(NC(c2cc(Cl)ns2)=O)C1)=O)OC C#CCCCC(C)C(=O)N1CCC(CO)(CC)C1.N1(C(=O)C2CC2)CCOCC1C C1(NC(C(C)CF)=O)CN(C(c2cn(C)nc2C(C)(C)C)=O)CC1C C1(C(N2CC(NC(C=C(C)Cl)=O)C(c3ccc(F)cc3)C2)=O)CCC2(CCC2)C1 c1(OC)ccc(C2CC2C(=O)NC2CCCC2n2nc(C)cc2C)c(Cl)c1 C#CCN(OC)C(=O)C1CN(C(=O)CC2CCC=CCC2)CCN1C c1(C(=O)NCC(C)CN(C)C(C2CC3CC3C2)=O)cnc(S)[nH]1 CCCC(CC)CC(=O)N(C1CCCN(C(=O)CC(C)(C)C2CC2)C1)C c1(C(N2CC(C)C(F)(F)C2)=O)ccc(C(F)(F)F)c(F)c1Br.c1nn[nH]n1 C1(CNC(C2(C)CCC2)=O)CC(C(N)=O)=NO1.c1(C(=O)N)ccc(O)nn1 C(CCC(=O)N(CC(CC)NC(c1ccc(Br)s1)=O)C)OCC=C N1(C(c2cc(C)cc(C)n2)=O)CC(C(=O)N(C2CCCC(O)C2)C)CCC1(C)C C1(C(=O)NCC(C)(C)NC(C(C)NC2CCCCC2)=O)CCC2CC2CC1 N1(C(CCC2CCC(NC(Cn3c(C)ncc3)=O)C2)=O)CCOCC1CC(N)=O C1(C(=O)NCCc2onc(CC)n2)CC(F)(F)CN1C(=O)C(C)C1CC1 C1(NC(=O)CC2(O)CCC2)CN(C(=O)CN2CCCS2(=O)=O)Cc2nccn2C1 C(=O)(C1=CCCCCC1)N1C2CC(C(=O)NCC(CCC)O)C1CC2 C1(C(N(C)CCN2CCN(C(c3cc(N)ccn3)=O)CC2)=O)CCC2CC1CO2 c1(CC=O)csc2sc(C)cc12.C1(NC(C2(OC)CCC2)=O)CCC(C)C1.C C=CC(C)(C)CC(=O)NCC1CC1CC(=O)Nc1cc(N(C)C)cc(F)c1 C12(NC(C3CC(OC)CN3C(=O)CN(C)C)=O)CCC(CC1)C2(C)C C1(CN(C(=O)CC(F)(F)F)C)CN(C(=O)CO)CC12CC2.C1CCCOC1.C C1(C(=O)NC2CC2C(F)F)CCCN(C(=O)CC(=O)NCCCO)CC1 c1(C(N2CC3N(C(c4n(CCOC)ncc4)=O)C3C2)=O)ccc(Cl)c(F)c1 C1(NC(Cn2c(C)cc(C(F)F)n2)=O)C2CC1CN(C(C1CCCN1C)=O)C2 C1(N(C(=O)CC2CCOCC2)C)CC2CCC(C1)N2C(C1(C#N)CC(=O)C1)=O C(CCCCC(=O)N1CCC(NC(=O)C=C2CCC(C)CC2)C1C1CC1)SC C(C(=O)N1CCC(CN(C)C)C1)(C(C)(C)C)NC(CCC(C)N(C)C)=O C(=O)(CCC(=O)N1CCC(C)(NC(=O)CNS(N)(=O)=O)C1)OCC C(=O)(C1Cc2ccc(F)cc21)N1CCC(OCCNC(C(C)(C)CF)=O)C1 N12CCC(C(C)C1)NC(=O)NCCC2.C1(OC)(CO)CCCOC1 c1(C(N2C(CCNC(C3(C)C(C)C3)=O)CCC2)=O)ncc2[nH]ncc2n1 c1(C(=O)NCCC(C)C)cnc2c([N+](=O)[O-])cnn2c1.C1(C(=O)N)CCN(C)C1 CCC(C)(CC)C(=O)NC1CC(c2cn(-c3cc(C)cc(Br)c3)nn2)C1 c1(C(C(=O)NC2CCCC2)N(C2CC2)Cc2cccs2)c[nH]ccc1=O Cc1sc2ccccc2c1C(=O)NC1CCCN(C(=O)C(CO)C(C)(C)C)C1 C1CCCCC1.c1(C=O)cc(C(C)(F)F)on1.C1(C(=O)O)(C=O)CC1.CC Cc1ccc(C(N2CCS(=O)CC2c2ccccc2)C(=O)NC2CC2)c(F)c1F C#CCCCCCC(=O)N1CCOCC(C(N2CCC(OC)C2C2CC2)=O)C1 C(=O)(C(F)CC(C)(C)C)N1C(C(C)C)CN(C(=O)C(O)CN(C)C)CC1 C(=O)(C1=NOC2(CCN(Cc3cc[nH]c3)C2)C1)Nc1ccc(OC)cc1O c1(C(=O)NS(=O)(=O)c2[nH]ccc2Cl)cc([N+](=O)[O-])ccc1N1CCCCC1 C(CN=C(NC1CC1)N1CCC=C(C)C1)(C(C)(C)C)OC c1(NC(c2n(CCSC)nnn2)c2ccsc2)ccc2c(c1)CCS2(=O)=O C1(CC(=O)NCCOCCC(C)C)CCC(NC(=O)Cc2ccsn2)CC1 C1(O)(C(=O)NCCCCC(C)NC(=O)CCCN2CCCC2)CN2CCC1CC2 C(=O)(C(CC)(CC)CC)NCC1CCC(NC(CCCOCCC)=O)CC1 N1(Cc2c(CC)ncs2)CCC(C(N2CCC(C)(C(=O)OC)C2)=O)C(C)C1 N1(C(C(F)=CCC)=O)CC2CC2C1.N1(C2(CC(=O)NC)CC2)CCCC1 c1(NC2C(C(=O)OC)CCCC2)ccc(F)c(NS(=O)(=O)C2CC2)c1 N1(C(COC(C)=O)=O)CCC(NC(=O)C(C)CCO)C(C)(C)C1 CC(O)C(C(=O)N1CCCCC1CC(N)=O)NC(=O)CN1CCOC1=O C1(c2n(CCOC)nnn2)(NC2CCCN(C)CC2)CCN(C2CCOC2)CC1 N1(C(CCSCC)=O)CC2(C1)CN(C(=O)CC1CC(O)C1(C)C)CCO2 C(C)(C)(CC(C)C)NC(=O)NC1CCN(C(=O)OC)C1.C1C2CCCC12.N N1(C(C2(CC)CCOC2)=O)CC2CC(C)N(C(c3cc(F)ccc3C)=O)C2C1 c1(C(C)C)nocc1C(=O)NCC1CCCC1C(=O)NCCCOC(=N)O C1(Cc2nnnn2C2CCCCC2)CC2C(C1)C2(F)F.C(=O)(CN)OC(C)C CC1CN(C(C2CNC(=O)O2)=O)CCN1C(C1CCC(=C)CC1)=O CCCCCCC(CC)CN=c1ccnc(NCC(C)C(F)(F)F)[nH]1 C1(C(CC)(C)C)CCC(C(=O)N(CCC(C(C)C)NC(=O)C=CI)C)CC1 C1(C(N2CC(NC(c3ncc(N(C)C)nc3)=O)C(O)C2)=O)CN2CCCC2CO1 c1(C(N2CCC(CNC(CS(=O)(=O)N(C)C)=O)C2)=O)nnc2ccccc2c1N C(C(C(C)(C)C)NC(=O)NC1(CO)CCCC1)SC c1(CNC(C(CC)(C)CO)=O)ccc2c(c1)CCCC2NC(=O)Cc1cc[nH]n1 c1(C(=O)NC2C(OC)CN(C(CCCCCC)=O)C2)ccc2nc(S)[nH]c2c1 C1(NC(C(CC)CO)=O)CCCCN(C(=O)CCc2nnc(O)nc2O)C1 C1(NC(CSC)=O)CCC2(CC1)CC2NC(=O)CC1CC2CCC(C1)N2C C1(O)(C(C)NC(C(C)C2CC2)=O)CCN(C(=O)C=O)CC1.c1ccc(Cl)cc1.N c1(OCC)cccc(F)c1N1CCN(C(=O)C(C(C)C)NC(C)C)CC1 CN1C(=O)CCCC1C(N1CC(F)CC1C)=O.C1(C(=O)N)(C(N)=O)CCC1 C(=O)(C(F)C(=O)NC(CSCC)C(=O)N(CC(C)C#N)C)OCC N1(C(C(C)=C(CC)C)=O)CCC(CNC(=O)C(CO)OC)C(F)(F)CC1 C1(CCC)CCCN(C(c2ccc(CNC(C34CCC(OC)C3C4)=O)o2)=O)C1 Cc1nc(N2CCC(CCNC(=O)CN3C(=O)CNC3=O)C2)c(C)c(O)n1 CCCC(C(=O)OC)C(=O)N1CC=CC1CNC(c1cnn(CC)c1Cl)=O N1(C(c2ccc(CC)cn2)=O)CC(C)(C)CC1C(=O)NC1CCN(CC)CC1 N1(C(C=CC(C)C)=O)CCC2(C=C(C(=O)N(C34CC(C3)C4)C)C2)C1.CS O=C1CCN(CC(=O)NC2(C(=O)NCCc3cccc(O)n3)CC2)CC1 CC1CC=C(C(=O)NC2(C(N3CC(C(=O)N(C)C)C3)=O)CC(O)C2)CC1 c1(C(N2CCN(C(CCC=C(C)C)=O)C(C(C)C)C2)=O)nnn2c1CCCC2 c1(CC)ccsc1C(N1CC=CC1C(=O)NCC(N1CCCCC1)C)=O C(=O)(C#CC1(C)CCCO1)NC(C1(C(N2CCCCC(C)(C)C2)=O)CC1)C C(=O)(C(C)NC(=O)CNC(=O)C(C)C1CCOC1)NC(CC)C C1(CNC(CC(CC)C)=O)CCC12CN(C(c1scc(C)c1Br)=O)C2 C1(C(=O)OC)CN(C(=NCCOCc2ccccc2)NCC(C)(C)C)CCO1 N1(CC(=O)OC)CCCC(C(F)(F)F)C1=O.c12nnc([nH]1)SC2 N1(CC)CCC(C(=O)NC2CCCC2C)C1.c1(C=O)ccc(C(F)(F)F)[nH]1 CC1(C(=O)NC2CC3CCCC2N3)Cc2cc(Cl)ccc2C(=O)O1 c1(OC)ccccc1.C(=O)(CCCN(C)C(C)C)N(CCCCN(C(C)=O)C)C.O c1(C(N2C(C)(COC)CC(NC(=O)CO)C2)=O)ccnc2ccnn12.CC Cc1cccc(-n2ncc(C(=O)NCC(C(C)C)NC(=O)Cn3cccc3)n2)c1 C=C=C(C)CC(=O)NC(CCNC(c1ccnc(-c2ccccc2)n1)=O)C(C)C C1(NC(CCSC)=O)CN(C(C2CC(C)CO2)=O)CC(C)(C)C1 CCC(CC)CC(=O)N1CC(O)CC1(C)C(=O)NCCCOC(F)(F)F N1(C(c2snc(OC(C)C)c2Br)=O)CC(Cc2ccccc2)CC(C)C1 c1(C(=O)N)oc(C)nc1C.c1(C(C)(C)OC)cn(CC2C(C)C2(F)F)nn1 C(=O)(C(CC(C)(C)C)NC(=O)CC(C)C1CC1)NC1(CC=C)CCC1 N1(C(C)=O)CC(O)CC1C(=O)NCC1CC(O)CN1C(c1ccon1)=O.C c1(OC)cc(Cl)ncc1C(N1C2CC1CN(Cc1ccc(C(F)(F)F)cn1)C2)=O N1(C(c2c(OC)c(C)sc2)=O)CCN(C(=O)CCC(C)c2ccccc2)C(C)C1 C1(C(=O)NCC2CC3CC3N2C(=O)C#CC2CC2)CCn2c(cnc2Br)C1 C(=O)(C(C)(C)CS(N)(=O)=O)OCC1=CCCC1C C1(O)(C(=O)NC2CCN(C(C(C=C)(F)F)=O)CC2C)CCC(C)(C)CC1 Cc1cc(NC2CCCC2C(=O)NCc2cc(F)ccc2Cl)nc(C)n1 N1(C(C2C(CC)C2)=O)CCCC2(CCN(C(=O)Cc3cncs3)C2)C1 C(CC(F)F)(C(=O)N1CC(N(C)C)C1)N(C)C(C1C=CCCCC1)=O N1(C(C2N(C)CCC2)=O)CC(CNC(=O)CC2(C)CC2(F)F)C2(CC2)C1 c1(C(N2C(C3(NC(c4ccc(C)s4)=O)CC3)CCCC2)=O)cccc(CO)c1C C1(SCC(C)C)CCCC1C(=O)NCC1CC1.c1ncc[nH]1.C(=O)C.N C(=O)(CCN=C1NS(=O)(=O)c2ccccc21)N(CC(c1ccccc1)O)C C1(NC(CC2CCC(=O)N2)=O)CCCC2CN(C(C3(C(F)(F)F)CCC3)=O)CC12 C(C)(C)(CCC(=O)N1CCNC(=O)CC1)NC(C1OCCC(C)C1)=O N1(CCSC)CCC2(CC1)OCCc1cc(C(=O)NCCC3CCCOC3)sc12 c1(NC2CCN(C(C(CCC)(C)O)=O)C2)cc(C)nc2cc(C)nn12 O=C(O)C#CC(=O)NCC1(O)CN(C(c2cccc(O)n2)=O)C1 N1(C(C2N(C(c3c(C)nccn3)=O)C(C)C2)=O)CCN(C)C2(CC2)C1 C1(c2cn(C(COC(c3c(OC)cccc3Br)=O)C)nn2)CCn2ccnc2C1 C1(CNC(CCc2c(C)n(C)nc2)=O)CC(C)CN(C(=O)CC2(O)CCCC2)C1 C1(NCC(CO)NC(=O)NCCCOCC#C)CCCCC1C(C)(C)C C12(CNC(C3C(=O)NCCC3)=O)CCC(CC1)CN2C(=O)COCCF c1(SCC)ccc(-n2nc(CCO)nc2Cc2cccc(Br)c2)cc1 CC(C(C)C(=O)NCc1cn[nH]c1)NC(=O)CC1CC2(CC2)CO1 c1(OC(C)C)ccc(COC(c2cccc(F)c2N)=O)nc1Cl c1(C(N2CCC3CN(C(=O)CCN4CCCC4)C3C2)=O)cc2sc(Cl)cc2[nH]1 C=Cn1nccc1C(=O)NC(c1cn(C)nn1)C(N1CCC(CCN(C)C)C1)=O CC1CCC(C)(C(=O)NCC2CCC2)C1(C)C.c1(C(=O)N)cc(O)n(C)n1 c1(C(N2CC(CNC(C3CC(OC)C(OC)C3)=O)C(C)C2)=O)nc(C)ccc1C CC1CC(C(=O)NCC2CCN(C(C3CC=CC(O)C3)=O)C2(C)C)=NO1 C1(C2(O)CCOCC2)(C(=O)NC2CN(C(C(CCCC)C)=O)CC2(C)C)CC1 C1(C(N2C(CNC(c3cnn(C4CC4)c3)=O)CC2)=O)CCc2ccccc2O1 CCC(CNC(=O)C1=CCC1)NC(=O)C(C)OC(C)(C)C C1(C(N(C)C)=O)CCN(CCC(=O)Nc2ccccc2C2CCOC2)CC1 c1(CC)ncc(C(=O)NCC(C)CN(C(=O)COc2cn[nH]c2)C)[nH]1 C(=O)C(C(F)(F)F)C(F)(F)F.CC1(C(N2CCC2C)=O)CCCNS1(=O)=O.N N1(C(c2n(C)ncc2Cl)=O)CC2CC1CCN2C(=O)CCC1CCCO1 c1(C(=O)NCCCCC(C)NC(C2CCCC2O)=O)ccc2n[nH]cc2c1 C#Cc1cn(C)nc1C(=O)N(C(C)CC(=O)NC1C2CCCC1CC2)C N1(C(c2c(C)sc(O)n2)=O)CC(C(N2CCOC(C3CC3)C2)=O)CC1(C)C CC(C)CC(CNC(C1CC12CCC2)=O)C(=O)N1CCC12CC(CO)C2 O=C(C1=COCC1)NC1CC(NC(C2(Oc3ccc(Cl)cc3)CCCCC2)=O)C1 c1(NC(N2CCCC(S(=O)(=O)N3CCOCC3)C2)=O)cc2ccc(Cl)cc2nn1 CN1C(=O)CCCC1C(=O)NCCC1(C)CCN(C(=O)C=CS(C)=O)C1 c1(CN(CCOCCNC)C)nn(C)c2c1COCC2 C1(CNC(CCOC)=O)CCN(C(c2cnc(C(F)(F)F)s2)=O)C1C1CC1 C1(NC(c2cc(C)c(-c3ccc4scnc4c3)cc2)=O)CC2CCC1(C)C2(C)C c1(C(=O)NC(C)CC2CN(C(=O)C=CBr)C2)csc(Br)n1 c1(C(=O)NCC(CC=C)NC(c2ncccc2OC)=O)c(SC)cccc1F c1(CCC(=O)NC(CCC)CNC(=O)CC2CC2)cccc(Br)c1 c1(CN(C(=O)C(F)(F)c2cscn2)C)ccccc1C.C1(C=O)CCCN1C.N CCCCC(C)C(=O)N(CCC(C(C)C)NC(c1c(Br)cnn1C)=O)C C(=O)(CC(C)CC(=O)N1CCN(C(c2ccc([N+](=O)[O-])nc2)=O)C(CO)C1)OC C1(NC(C=CC)=O)CN(C(=O)C(c2cccc(CC)c2)N(C)C)CC12CC2 c1(C=O)cccc([N+](=O)[O-])c1N.CC1C(CC(=O)NCC2CCOC2)C1(F)F.N N1(C(Cc2cc(C)cc(F)c2)=O)CC(C)N(C(=O)C(C)(C)F)CC1C c1(C(=O)NCC(C)NC(C2(N(C)C)CC2(F)F)=O)csc(-c2cnc[nH]2)n1 C1(CC(=O)NCC2CC(SC)C2)CC(F)CN1C(C1COCCC1C)=O CC1(CNC(=O)NCCCOc2ccccc2)COc2ccccc2O1 N1(C(c2c(C)occ2)=O)CCCC1C1CCCN1C(=O)COCCCF C1(C(=O)NCCSC(C)C)CCN(C(C2(C)CCOCC2)=O)CC1C c1(CNCc2c(C)n(C(C)C)nc2)cnc2cc(Cl)ccn12 c1(CC(=O)NC2C(C)(C)CN(C(=O)CC3COCCO3)C2)ccc2ccoc2c1 c1(C(N2CC(NC(c3ccc(-n4nnnc4O)cc3)=O)C2)=O)ccc(O)c(Cl)c1 c1(CNC(=O)CN(C(c2ccoc2)=O)CC2CC2)cncc(O)c1 CC(C)(O)C(F)C(=O)NCC1C2CCC(C2)N1C(c1cocn1)=O.C1CC1 N1(C(C2CCCC(C)C2)=O)CCOCC(NC(c2cc(C3CC3C)on2)=O)C1 N1(C(c2c(C)ncnc2C)=O)CCS(=O)(=O)C(CCNC(=O)CCC(C)C)C1 Cc1nnc(C(C)NC(C2CCC(NC(=O)C(C)NC(N)=O)C2)=O)s1 C(=O)(CC1=CCN(C(=O)C(C)CC2CC2)CC1)Nc1c(CC)csc1 c1(CC(C(=O)N(CCC(C)NC(c2ccc(C)cc2)=O)C)C)ccc(F)cc1F Cc1ccc(CCCC(=O)N2CC(C)(NC(=O)CC3CCCCN3C)C2)cc1C C1(O)CC2CCC(C1)N2C(C1CC(C)N(C)C1)=O.Cc1scc(C(=O)N)c1C.C CCCCC(O)C(C)C(=O)NCC(CCC)C(=O)NC1CC(=O)N(CC)C1 C(c1cccc(F)c1)=CCC(=O)NC(CN(C(c1occc1F)=O)CC)C CC(C)(C(=O)N=c1[nH]n(CC(F)(F)F)cc1Br)c1cccc(F)n1 c1(C=O)coc(S(C)(=O)=O)c1.C1(NC(C(C)SC(C)C)=O)CCC(C)CC1 N1(C(CC(C)c2cccnc2)=O)CCOC2CN(C(=O)C3=CCOC3)CC12 c1(C(F)(F)F)csc(C(c2nnnn2C2CCCCC2)NCCSC(F)F)c1 C=CC(C)(C)C(=O)N1CC=CC(C(=O)N(C)CC2CCN(C)CC2)C1 C1(NC(CCOCC)=O)CCN(C(c2cccc(O)c2Cl)=O)C12CC2 c1(SC)cc(C(=O)NC(C)(C)C(C)NC(c2ccn(C)n2)=O)c(Cl)cc1Cl CC1CNC2(CCN(C(=O)NNc3cccnc3)CC2)CO1 c1(C(C=O)C)ccc(S(C)(=O)=O)cc1.C1(CC)CCN(C(=O)C(C)(F)F)C1.N c1(C(C(=O)NC(C2(C(=O)OCC)CC2)C)N)c(C)cccc1Br C12(C(=O)NCC(C)C)CCC(NC(c3cc(Cl)cnc3Cl)=O)(CC1)CC2 CC1CN(C(=O)C=C(Cl)Cl)CCN(C(=O)Cc2ccn(C)c2)C1 C1(CCNC(=O)C(c2ccccc2)O)(NC(C2C(C)C2(F)F)=O)CCOCC1 N1(C(C(C=C)O)=O)CCC(c2nnc(CNC(C3CC(CC)=NO3)=O)s2)CC1 Cc1nccn1CC(N1CCC(C2CCCN2C(=O)CCc2nncn2C)C1)=O N#CC1CN(Cc2ccc([N+](=O)[O-])s2)CC1NC(=O)CCCCn1cccc1 O=C(CCC(F)F)NCC(c1ccc(F)cc1)NC(=O)C(F)(F)c1ccccc1 N1(C(CCC(C)(C)OC)=O)CCCC(C)(C)C1C(=O)NCC1CNC(=O)CO1 c1(C(N2CC(CC(=O)Nc3cccc(SC)c3)C(C)C2)=O)cccc2ccoc12 C1(CNC(C(C)(C2CC2)OC)=O)C(C)CCN1C(=O)C(CC)N(C)C.S C12(NC(c3ncc(NC)nc3)=O)CCC(C)(C1)OC2.c1(C(=O)N)ncoc1C c1(C=O)n[nH]cc1[N+](=O)[O-].C(CCC(=O)NC(C)(C)C)N(C(=O)OCC)C CS(C)(=O)=NCC(=O)N1CCCCC1CCCNC(c1scnc1Cl)=O c1(C(=O)Nc2c(C(=O)Nc3cn(CC)nc3C)cccc2)ccccc1C#N N1(C(c2ccc(C(=O)OC)o2)=O)CCCN(C(c2[nH]ccc2C2CC2)=O)CC1 C1(C(=O)O)(C(=O)O)CC(F)(F)C1.c12cn(nn1)CCCC(=O)NC2C c1(C(N(C2CCN(C(=O)C(C(C)CC)OC)CC2)CCC)=O)cccc(F)c1N C(=O)(C1=CC2(CCN(C(=O)CN3CC(C)C3)C2)C1)N1C(CC)CC(C)CC1.O C(C(O)CC(=O)N1CCC(C(=O)NOC2CCCCC2)CC1)N(C)C.C(N)(=O)N CC1C(=O)NC(=O)CN1C(=O)CCC1CCN(C(=O)CCCNC(N)=O)C1 c1(C(=O)NCCCN(C(c2cccnn2)=O)C2CC2)ccccc1-n1ccnn1 C(C1CCCO1)=CC(=O)NCC(CC)NC(C1CCC(=O)N1)=O N1(C(C(CC=C)C)=O)CC2CC(NC(=O)CN3CCOCC3=O)CC(C2)C1 C1(NC(c2c(C)csn2)=O)CCC2CCN(C(C3(N4CCCC4)CC3)=O)C1C2 CCC(C)C(O)C(=O)N1CC(CNC(c2cnn(-c3ccccn3)c2)=O)C(C)C1 C(=O)(C(C)(C)CC(C)C)NC1CCN(C(COCc2c(C)ncs2)=O)C1C N1(C(C(C)NC(C23CC2C3)=O)=O)CCC(C(=O)N)C1.n1(C2CC2)cccn1 CC1(C)CCCC(C(=O)N(CCNC(C2(F)CCCOC2)=O)CC2CC2)C1 C(c1cccnc1)=C(C(=O)N(CC(CN(C(c1cccs1)=O)C)O)C)C.CC.O c1(CC)noc(C)c1C(c1nnnn1C(C)C)NC1CC1.C1(C)CC1.C N1(C(COCCOC)=O)CCC2(CCC2)CC1.c1(CCC(=O)N)c(C)noc1C c1(OC)cc(S(=O)(=O)N)ccc1NC(c1ccc(F)cc1)=O.CC(F)(F)F C1(CNC(c2[nH]cc(CC)c2)=O)CCCCC1NC(c1ccnn1CC)=O C1(OC)CN(C(=O)CCC2CC2(F)F)CC1NC(=O)C(F)n1cccn1 N(C(=NCc1ccc(C(C)(C)C)s1)N1CCC(CN2CCOCC2)C1)C(CC)CC CN1C(=O)CCCC1C(N1CCC1C(=O)NCC1CC(C#N)C1)=O N1(C(c2cc(Cl)c[nH]2)=O)CCC(F)(C(=O)NCC2(CO)CC=CC2)C1 Cc1cc(C(N2CCC3CC23C(N2CCCC(C)(CO)C2)=O)=O)nnc1O C1(NC(c2c(=O)ccn(C)c2)=O)CCN(C(=O)CC2C=CCCC2)CCC1(F)F C1(NC(C2OCCN(C(C)C)C2)=O)CN(C(C2CC2C)=O)CC2(CC2)C1 N1(C(C(C)N(CC)CC)=O)CCCOC(CCNC(=O)Cc2ccccc2Cl)C1 Cc1noc(C)c1C(=O)NCCCCCNC(=O)CC1CCCC(C)O1 CCCCCCC(=O)NC1C2CC1N(C(=O)COCc1ccc(C#N)cc1)C2 c1(NC2C(NC(=O)C(=Cc3c[nH]cn3)F)CCCC2)ncnc2c1CCO2 C(N=c1[nH]c(=NCc2cccc(Cl)c2Br)[nH]c2c1CSC2)c1nc(C)sc1 c1(C(=O)NC2(CO)CCCN(C(c3ccns3)=O)C2)nncc2c1CCCC2 c1(CN2CC3(C(C(=O)NCc4cnccn4)C3)C2)ccc(I)c(Cl)c1 C(=O)(C1Cc2c(Cl)cccc21)NCC1CN(C(CCc2n(C)nnn2)=O)C1 CC(CC(=O)N1CC2CN(C(c3cc(F)ccc3F)=O)CC2C1)CC(F)(F)F c1(C(=O)OC)ccc(C(N2CCCN(C(C3CCC3C)=O)CC2)=O)c(C#N)c1 Cc1c(Br)c(C(N2CCNC(C(N3CCC(F)CC3)=O)C2)=O)nn1C Cc1cc[nH]c(=N)c1C(N1CC(NC(c2cc(O)n(C)n2)=O)CC(O)C1)=O C(CCC(C)C(C(=O)NCC1(CC(C)C)CC1)N(C1CCC1)C)=C(C)C Cc1cnc(C)c(NC(=O)CC2CN(C(c3cccc(Cl)c3F)=O)CCO2)n1 Nc1cc2ccccc2cc1C(N1CCCCC1CCNC(=O)C#CC1CC1)=O c1(C(=O)N)cnc2cc(O)ccc2c1.CC(C)CC(C)(C)C(=O)NCCOCC C1(NC(c2c(C)c[nH]c2)=O)CC2CCC(C1)N2C(C1CCCCC1(F)F)=O CCCC(CCC)=CC(=O)N(CC(C)N(C)C(c1csc(C)c1CC)=O)C N1(C(c2c(CC)cno2)=O)CCC2(CCCN2C(=O)CC(C)CN(C)C)C1 c1(C(N2C(CN(C(CCOC(C)C)=O)C)CCC2)=O)ccc(Br)c(N)n1 c1(C(=O)NCC(c2ccccc2)NC(CC(C=C)CC)=O)cnc2n1CCCC2 C#CCCC(O)C(=O)NC1CN(C(=O)CCC(=O)N(C)C)CC1OC c1(C(=O)NC2C(CNC(c3csnn3)=O)CCC2)cccc(Br)c1[N+](=O)[O-] c1(CNC(c2n[nH]c3ccccc23)=O)nc2c(s1)CCN(C(c1cnco1)=O)C2 C(=O)(C(C)CC(N)=O)NCC1C(N(C)C)CN(C(C(C)=CC2CC2)=O)C1 C(=O)(CCC(=O)NC)N(CCC)CCC.C1CCN(C(=O)CCCC2CCC2)C1 N1(C(C)=O)CCCC1C(N1CC(C)C1)=O.n1(CC(=O)N)cc(C(F)F)cn1 Cc1c(C(N2CCC(NC(=O)CC(F)F)C2Cc2ccccc2)=O)cccc1N c1(C(C)NC(Cc2nccn2C)C(N)=O)ccc(C(C)C(F)(F)F)cc1 C(CCC(C)(C)C(=O)N(CCCOCCNC(c1cc(C)sn1)=O)C)OC C1(NC(c2cnn3c2CCC3)=O)C2CC1CN(C(C1CCCS1(=O)=O)=O)C2 N1(C(CCNC(=O)NC)=O)CCC2(CC1)CN(C(=O)CN1CCCS1(=O)=O)C2 c1(C(N(C)CCF)=O)ccn(C2CCCC2)n1 c1(CN(C(CCCCN(CCC)CCN(C)C)=O)C)nncn1C(C)C Cc1cc(C)c(C(=O)NC2(CCC(=O)N(C)Cc3ccc(F)cc3)CCC2)o1 Cc1cc(C(N2CCCC3CCN(C(=O)CC(F)F)CC23)=O)cc2ccncc12 CCC(CCC(=O)N1CCCC1C1(O)CN(C(c2[nH]nc(Cl)c2C)=O)C1)OC CC1(C)CC(CNC(=O)C(F)OC(F)(F)F)N(C(c2cnc(O)o2)=O)C1 C1(NC(c2ccc(Cl)o2)=O)CC2CCC(C1)N2C(C1CC2C=CC1C21CC1)=O Cc1nc(C=CC(=O)N)[nH]c1C.C1CCN(C(=O)C=Cc2cnn(C)c2)C(C)C1 c1(NC(CC2N(C(C3(CC)CC3)=O)CCOC2)=O)c(O)cccc1[N+](=O)[O-] C1(C)(C(N2CCCC(CN(C)C(C3(C)CC(C#N)C3)=O)C2)=O)CC2CCC1O2 CN1CCC(F)(C(=O)NC2CCCCC2NC(=O)C(C)(C)C2CCC2)CC1 c1(NC(C)=O)ccc(Cl)cc1Oc1ccn(Cc2ccccc2)c1 Cc1n[nH]c(C)c1CC(N1CC(CC(C)NC(C2C=CCC2)=O)C1)=O c1(C(N(C2CC(NC(CN(CCC)C)=O)C2)C)=O)c(C)cccc1Cl c1(C(N2CCC(O)(C(CNC(C=NOC)=O)C)C2)=O)cnc(C)cc1Cl C(=O)(C(Cc1ccccc1)NC1CNC(=O)C1)N(C)CC c1(C(=O)NC2CCN(C(C3(C)CCCC3(F)F)=O)C2)n[nH]c2c1CCCC2 CC1(C)CN(C(=O)C(O)C2(c3ccccc3)CC2)CC(CC(=O)O)O1 c1(CN2CCC(CC(=O)NC3CCC(CC)CC3)CC2)cnccc1C#N C12(C(N3C(CC)CCC(C)C3)=O)CC(CN(C(c3ccn(CC)c3C)=O)C1)C2 c1(C(=O)NC2C(NC(c3nc(OC)oc3)=O)CC2)c[nH]c2ccc(F)cc12 c1(C(N(C)C)=O)cc(Cl)cn1C.c1(C(N2CCC2)=O)ccnn1CCN(C)C Cc1ccc(Br)c(C(=O)NC2CCC(CNC(C3(CO)COC3)=O)C2)n1 c1(C(N2CC(CNC(c3c(OC)scc3)=O)C(C)CC2)=O)ccc(Cl)c(C)c1N C1(C(=O)NCC(C(=O)OC)(F)F)CC(C)CN(C(c2cnncc2O)=O)C1 C(CCCCCN(C(=O)C(C)COCc1ccccc1)C)NC(CC=C)=O C1(CC)CCC(O)(C(=O)N(C)CCOCC)C1.c1(C(=O)N)c(C)csc1Cl O=C(C1=CC2CCC(C1)C2)NCc1nc(C)cs1.C1(C=O)CCCC(F)(F)C1 c1(C=O)cc(C(F)(F)F)ccc1C.C(=O)(C(C(=O)N)OC)OC.C1(C)CCC1 C(C(C(=O)NC(C1CN(C(=O)Cc2ccccc2)C1)C)c1ccccc1)SC C=CC1(C)CCOCC1.C1(C)(C(N2CCCC(CC(=O)N)C2)=O)CC2(CCC2)C1 N1(C(C(=O)NCCOCC)CCc2cnccc2C)CCc2c[nH]nc2C1 C1(C(N(C2C3CN(C(CCC=CC(C)C)=O)CC32)C)=O)CCc2nc[nH]c2C1 C=CCC(C)(C)C(=O)N1CCCC1C(=O)NCc1ccc(Cl)nc1F C1(CC(=O)NCCC(=O)OC)CN(C(=O)CC(C)N(C)C)C(C)(C)C1.O c1(C(N2C(C)CC(NC(c3ccnn3CCF)=O)C2)=O)nccn2cnnc12 c1(OC)c(C)csc1C(N1CCCC(C2CCCN2C(=O)C=C(Cl)Cl)C1)=O c1(CC(N2CC(CNC(Cc3ccn(C)n3)=O)C3C2C3)=O)ccc2c(c1)OCO2 NC1CCN(C(c2nn(-c3ccc(F)cc3)ccc2=O)=O)CC1C(=O)O c1(C(=O)N)cccc(F)c1C(F)(F)F.CC(CN(C)C)C(=O)NC1CCC1 C12(NC(COC3CCN(C(C4CC(SC)C4)=O)C3)=O)CCC(CC1)OC2 c1(C(=O)NC23CCCN(C(c4ccc[nH]4)=O)CC2C3)cc(=O)n2nccc2[nH]1 Cc1ccc2c(CC(=O)NC3CCN(C(C4C=CCC4)=O)CC3C)c[nH]c2c1 C(CCS(C)(=O)=O)(C(=O)N(C1CN(C(=O)C(C)n2ccnn2)C1)C)OC C(=O)(C(CCC1CCC1)NC(C1CC1OC(C)(C)C)=O)NCCCC#C c1(C(N2CC(C)(C(N(CCOCC=C)C)=O)C2)=O)cccnc1CC C1(OC)(OC)CC(C)(C(=O)NC2CC2)C1.C1(C=O)CCCN1C(C)C.C c1(OC)ccc(Cl)cc1NC(c1sccc1NC(c1cc(C)n(C)c1C)=O)=O CCCC(CC)C(=O)NCC(C(C)C)NC(=O)C(CCO)N(C)C Cc1ccc(C)c(NC(c2nc(NC(c3ccccc3C#N)=O)cn2C)=O)c1 N1(C(C(CC)(C)C)C)CCC(c2nnnn2C2COC2)(NC(C)C(C)C)CC1 CCN=c1ccc(C(=O)NCC2CCCC2)c[nH]1.C(=O)CCCN(C)C(C)=O.N c1(C(=O)NCC2CCCN(C(C(C)SCCCC)=O)CC2)cc2cnccc2o1 N1(C(CC2(C(=C)F)CCC2)=O)CCC2CCC(C1)N2C(=O)CCCOC(C)(C)C c1(CN(C(C(N2CCC(C(=O)OC)C2)=O)=O)C)cccc(N(C)C)c1C C(=O)(C(F)(CNC(=O)C(C)C(O)C(C)C)C(C)C)N1CCC(CSC)CC1 CCS(=O)(=O)CC(=O)N1CCOCC1C(=O)NCc1nc(Cl)ccc1F Cc1cc(C=O)ncc1C(F)F.C(C)C(C)C.C(=O)CC1(C(F)(F)F)CC1 c1(CN2CC3CN(C(c4ccc(C)s4)=O)CC32)ccccc1[N+](=O)[O-] c1(CNC(COC)CC2CCCCC2)cccc(F)c1 C(=O)(C1=Cc2ccccc2C1O)NC1C(NC(=O)CC2(N3CCCC3)CC2)CC1 N1(C(C)C(=O)NCCN(C(=O)C)CC2CC2)CCCCC1.c1nnnn1C.S Nc1cc2[nH]cnc2cc1C(=O)NCCCNC(C1Cc2ccccc2O1)=O N1(C(C2(C(C)C)COC2)=O)CCC2(CC2NC(c2ccc(CN=[N+]=[N-])o2)=O)C1 N1(C(C2CC(OC)C2)=O)CCCC(O)(CN(C(=O)C(=CC2CCCC2)C)C)C1 N1(C(c2c(OC)csc2)=O)CCN(C(c2cc(C)cc(O)n2)=O)C(C(C)C)C1 C1(NC(Cn2c(C)ccn2)=O)CCC(NC(=O)CN2CCC2CO)CC1 C12(COC)CC(CN1C(c1cc(C)ccn1)=O)C2.c1(C=O)cnnc(O)c1.C C1(C)(C(=O)NCCC(CCC#C)O)CN(C(C2CC3CCC(C2)O3)=O)C(C)(C)C1 c1(OC)cc(C#N)ccc1C(=O)NC(C)C(C)NC(=O)CCOCC.O C(=O)(C(COCc1ccccc1)N1CCCC1c1ccnn1C)NC C12CCC(CC1)N2C(=O)C(C)CNC.n1(CC=O)nnnc1C(C)(C)C N1(C(c2cn(C=C)nc2)C(=O)NCC2CCOC2)CCc2c(Cl)cc(Cl)cc2C1 C1(NC(C(CSC)C)=O)CCCCC1NC(=O)Cn1cnnc1 C1(CNC(c2c(C)nc[nH]2)=O)CCCCN1C(c1cc(C2CCCO2)n(C)n1)=O C1(O)(CSC)CCCN(C(C2(C(=O)NC)CNC(=O)C2)=O)C1.c1cn[nH]c1.C C1(C(=O)NCCN(C(=O)CCc2ccoc2)C)CCC(N(C)C)CC1 c1(C(=O)NCCCC)cc2c(o1)CCCC2.c1(C2(C(=O)N)CC2)ccnc(Cl)c1 C1(C(=O)NC2CN(c3nccc(C(=O)OC)c3)C2)CCC([N+](=O)[O-])CC1 N1(C(COC(CC)C)=O)CC2(CCCC2NC(c2cc3cn[nH]c3cn2)=O)C1 c1(C(NC(C)C)=O)cnc(S)n1-c1ccccc1.C1(C)(CC=O)CCC1.C C(C)(C)(C(C)CC(=O)N1CCOC(C)CC1)NC(c1n[nH]c(C)c1C)=O C12(C(N3CCC(CNC(=O)C4=CCCS4)C3)=O)COC(CCO1)C2 c1ccc(C)cc1C.C(C)(C)(C(=O)NC(C)CCN(C(=O)C)C)OCC.S N1(C(C(C)=CC)=O)CCC(C2CCCN(C(=O)C(C3CCOCC3)=O)C2)C1 C=CCC(C(=O)N1CCC(N(C(=O)CC(C)(F)F)C)C1)c1ccccc1 CC1CC(O)CCN(C(C2C=CCN(C(=O)C(c3ccn(C)n3)C)C2)=O)C1 C(CC(CC)C(=O)NCC1CC(F)CN1C(=O)C=Cc1cccn1C)=CC C12(NC(COc3ccc(C)cc3)=O)CCC1CN(C(=O)CC1CC3(CC3)C1)C2 N#Cc1cc2c(nc1Nc1ccc(C#N)c(Br)c1)COCC2 n1(CCC(N2CCCC(NC(C(C(CC)C)O)=O)CC2)=O)ccc2ccccc12 C1(C=O)CCC2(CC2)C1.c1(C(N(C(C)C)CC)=O)ccnn1C(C)(C)C.N C(=O)(C1=CCN(C(c2cc(O)cs2)=O)C1)NCC(CC)C(C)C C1(NC(C2(CCNC(CSC(C)C)=O)CCCC2)=O)CCOCC1(C)C C1(CC)CC(C(N2CC(CNC(C3(C)CC3Br)=O)(C)C2)=O)CCC1=O.O C(=O)(C(C)(C)CC(C)(C)C)N.N1(C(C(C2CCCC2)OC)=O)CC(C)C(C)C1 c1(C(C(=O)N)C)ccc(F)c(Cl)c1.N1(C(c2cc(OC)n[nH]2)=O)CCC(CO)C1 C1(C(=O)NC(CNC(c2cc(C)c(C(F)(F)F)nc2)=O)C)CCc2n[nH]cc2C1 Cc1cc(N)cnc1OCc1cncc(-c2cnn(C)c2)c1.CCCCS(C)(=O)=O N1(CCC(=O)OC(C)CN2CC(C)S(=O)C(C)C2)C(=O)C2CC=CCC2C1=O N1(C(c2c(CC(C)C)nc(C)s2)=O)CC2(CCN(C(C3CNC(=O)N3C)=O)C2)C1 C1(C)(OC)CCCN(C(=O)NCc2cc(C(C)(F)F)ccn2)C1 C1(C(N(C(CSC)C)C)=O)N(C(c2cccc(F)c2)=O)CC12CCCC2 C1(NC(c2cccc(CC)c2O)=O)CCN(C(=O)C#CC2CC2)C12CCCC2 C1(N(CCCC=CC)C(C(=O)NCC(F)F)C2CCSC2)CC(F)(F)C1 C1(COCC)C2CCC1CN(C(c1cc(F)cc(F)c1)=O)C2.c12ccoc1N2 C(C(C)(C(=O)NC1CC1c1cnnn1C)NC(=O)CC1C=CCC1)SC N1(C(c2ccc(CC)o2)=O)CC2CCCC2(CNC(=O)C)C1.c1ncccn1.N C12(C=O)COC(C1)C2.C1(C)CN(C(C)=O)C1.c1csc(C=O)n1.NC.C Fc1cncc(Cn2cc(-c3nnnn3Cc3cccs3)nn2)c1 CC(C)C(CNC(c1ccsc1Cl)=O)C(=O)NCC(C)Cn1ccnc1 C1(C(N2CCC(NC(C(C)c3cncs3)=O)C2C)=O)Cc2cscc2C1 C(=O)(CC(C(F)F)C(C)(C)C)NCCCCCNC(C(CO)N(C)C)=O c1(-c2cc(OC)ncc2F)ccc(S(=O)(=O)NCC2CCS(=O)(=O)CC2)cc1 Cc1sc(C(=O)NCCC2COCCN2C(c2ccc(N)cn2)=O)c(C)c1C CCCCCCCc1csc(NC(=O)CC2CC(C)C2)n1.C(C)(C)C.C(=O)N n1(CC(=O)N(CC(CC)NC(c2nc(C)ccc2C)=O)C)c(C)cc(C)nc1=O C(=O)(C(F)C(C)(F)F)NCC(C(C)(C)C)NC(=O)C=CSc1nc[nH]n1 c1(OC)ccc(CCC(=O)NCC23CC2CN(C(=O)Cc2ccoc2)C3)cc1 c1(OC)ccc(NCc2cc(-c3ccccc3I)no2)c(C(F)(F)F)c1 C1(OCCNC(c2cocn2)=O)CCN(C(c2coc(-c3ccsc3)c2)=O)C1 C1(C(=O)NCC=C=C)CN(C(=O)C(c2ccnn2C)C)CCN1C n1(CC)ccc(C(=O)NC2CCC(CC(=O)NC)C2)c1C.C1NC(=O)NC1=O c1(CN2CCN(C(c3c(C)cc(O)cc3)=O)C3C2C3)cnc2ccccc2c1Cl C12CCN(C1)C(=O)CCC1(CCC1)NC2=O.c1(C(=O)N)cnn[nH]1.C1CC1 CN=C(NCC1CC1Cl)NCC(C)(C)C1CC1 O=C(C#CC1CCCO1)N1CCN(C(c2ccn3c2CSCC3)=O)CC1 C1(NC(C2CC3(CC3)CO2)=O)CC12CCN(C(c1cccc(O)n1)=O)C2 O=C1CC(C(=O)NCC(O)CNC(=O)Cn2nnc(C3CC3)n2)CCN1 c1(SC)cc(C(N2CCOCC2c2ccc(F)cc2)=O)c(C)o1 c1(C(COC(C2(C)C(C)CCC2)=O)=O)ccc2c(c1)CC(=O)N2C Cc1cccc(Br)c1NC(N1CCC(C(N2CCCC(Br)C2)=O)CC1)=O n1(CC)nc(C)cc1C(=O)NC(C(C)C)c1cnn[nH]1 C(=O)(C(C)(C)CC(=O)NC(C)C(C)NC(c1csc2nnsc12)=O)OC CN1CCC(C(=O)Nc2ccc(-n3cccc3)cc2F)CC1C(=O)OC(C)(C)C Cc1ccc(F)cc1CC(=O)NCC.C(=O)(COC(C)(C)C)NCC.O C(=O)(C1CCc2nccn21)N1C(CCNC(c2csnn2)=O)CCC1 CCC(CC)C(=O)N1C(C(=O)N(CCO)CCOC)CC1C N1(C(C(C)(C)C(N)=O)=O)CCC2(C1)CN(C(c1cc[nH]c(=N)c1)=O)C2 C(=O)(C(=O)N(CCC(=O)Nc1cnsc1)C1CC1)NCC C1(C(N(C)CC2CCN(C(c3ccnc(C)n3)=O)CC2)=O)CCc2nccn2C1 C1(C(N2CC(OC)(CNC(=O)CC3CCSC3)C2)=O)CCOCC12CCC2 Cn1c(C(=O)NC2CC3CC(NC(=O)CCC4CCC4)C2C3)cc2occc12 C(=O)(CCC(C)S(C)(=O)=O)NC(C1CN(C(=O)C=Cc2ccsc2)CCO1)C C(=O)(C#CC1CCOC1)N(CC(N1CCCC(CSC)CC1)=O)CCOCC C1(C)(C(=O)NCC=CCNC(C2C(OC)C2)=O)CC1(F)F c1(C(=O)NC(CCN(C(C=C(C)Cl)=O)C)C)cnn(-c2ccccc2)n1 C12(CC=O)CCC(CC1)C2.C1(CCNC(C=C(C)C(F)F)=O)CCCC1O.N N1(C(C2CC(=C)C2)=O)CCC2(CC1)CC(C(=O)Nc1cc(OC)n[nH]1)CO2 N1(C(C(CC)n2ccnc2)=O)CCC(NC(c2nocc2Cl)=O)C(C)C1 CC1=C(C(=O)NCCC(O)CNC(=O)CC2C=CS(=O)(=O)C2)CCO1 C(CCCCC(=O)NCc1cc(C)c(C=O)o1)=CC.C1CCOC(C(C)C)C1.N c1(CC)nc(C)c(C(=O)N(C(C)C)CC)s1.c1(C(C(=O)N)C)ccccc1C c1(C(=O)NC(C=CCC(=O)NCC(O)CCC2CC2)=O)csc(S)n1 c1(OCCC)cc(CNC(c2ccc(-c3csc(C)n3)cc2)C)ccn1 C(=O)(CC(C)CC(=O)N1CCCC(C(=O)NCC2CSC2)CC1)OC C1(N(C(=O)CCC2CCOC2)CC)CCCN(C(c2[nH]c(O)nc2C)=O)C1 C(=O)(C1=CCC(C)CC1)NC1CCCC1NC(c1c(CC)c(OC)ccc1)=O c1(C(=O)NC2CCN(C(C(C(C)O)C)=O)C(C3CC3)C2)nccc2ccccc12 C1(NC(COCC(C)C)=O)CC(NC(=O)COCC(F)(F)F)C1 Cc1nn(CC(=O)N(C(C)Cc2ccccc2C)C)cc1Br C1(NC(Cn2c(C)nnn2)=O)C2CCC(C2)C1C(N1CCOCC12CC2)=O C1(OC)CCCCN(CC(N2CC(C)C2)=O)C1=O.c1(CC(=O)N)ccc(C#N)s1 c1(C(N2C(C)C(NC(C3CC3CN(C)C)=O)CC2)=O)c(F)cncc1Cl N1(C(c2c(C)nco2)=O)CCN(C(=O)C(Cl)=CCl)C(C)C1C CCCC(C(=O)NCC(Cl)Cl)c1cccc(Cl)c1 C1(C(=O)NCC=C(C)C)CN(C(c2nccc(C)c2N)=O)CCC1(C)C c1(C=O)c(C)ncn(C)c1=O.C12(CSC)CC(C(N3CCCCC3)=O)(CO1)C2 C1(NC(c2cc[n+]([O-])cc2)=O)CCN(C(C23CC4CC2C3C4)=O)CC1 CC1(C(=O)NC2CC2(F)F)CCCN1C(c1ncccc1Br)=O c1(C(N2CC(C(C)NC(=O)CC(C)CF)C2)=O)cc2ccc(Cl)c(F)c2o1 C1(NC(CCOCC#C)=O)CCC(C)C1.c1(C=O)cnn(C(C)(C)C)c1C.C C(=O)(C#CC1CCOC1)N(CC(CNC(c1c(OCC)cccc1)=O)O)C C(=O)(C(=O)C(C)C)ONC(CNCCCCC)=O C(C(C)(C)Cc1ccccc1Br)(c1cn(CC)nn1)Nc1cccc(NC)c1 C1(O)(CNC(C=C(C)C)=O)CCN(C(C2CCC2C(F)F)=O)C1 c1(C(N(CC(=C)C)Cc2cccc(C(=O)OC)c2)=O)cc2c(o1)CCCC2 C=CC1(CC(=O)N(CC(C)CNC(=O)Cn2ccnc2C(C)C)C)CCC1 c1(CC(N2CC(C(=O)NCC(CC)CO)C2)=O)cccc(C)c1 C1(C(C)(C)NC(Cc2scc(CC)n2)=O)CCN(C(C2CCCOC2)=O)CC1 C1(C)(C(N2CC(CCOC)C2)=O)CC(O)CN1C(c1c[nH]c(=O)cn1)=O c1(C(=O)NCCC(C)NC(CC2ON=C(CC)C2)=O)cc(C#N)ccc1C CCCC(CCCO)C(=O)NC1CCN(C(=O)CC2CC=CCN2C)C1(C)C N1(C(=O)Cc2cc(Cl)cs2)CC2(C1)CN(C(C1CC3C=CC1C3)=O)CCO2 C12(C(N3C(CC(C)(C)C)CC3)=O)CCCC1CN(C(C1CCCCCC1)=O)C2 N1(C(c2c(C)ccnc2O)=O)CCN(C(=O)C(=Cc2cn(C)nn2)F)CC12CC2 Cc1nccnc1C(N1C(C(=O)NC2(C)CC(O)C2)CCC1C(C)C)=O CCC(CC)C(=O)NCC(C)(C)NC(=O)CC1C=CCCC1 c1(C(=O)NCC(CNC(CC(CCC)C)=O)(C)C)ccc2c(c1)OC(C)(C)OC2 C1(NC(c2sccc2F)=O)CC(F)(CNC(C2(n3cccn3)CCC2)=O)C1 CCC(C)C(C)CN=c1[nH]c(=NCc2cc(C)oc2C)[nH]c2cc[nH]c12 C(CN(C(=O)C(C)n1ccnc1)C)(CO)(CO)NC(c1c(C)ncs1)=O N1(C(C)C)N=C(C(=O)N2CC(NC(C34CCCC(C3)OC4)=O)C(O)C2)CCC1=O C1(C(N2CCC(CC)C2CNC(c2coc(CO)c2)=O)=O)CCc2nnnn2C1 c1(NC(C(N2CCC(C(C)(C)CN)CC2)=O)=O)cc(I)ccc1F Cc1cc(C)c(C(=O)NCC2(O)CCN(C(C3(C)COCCO3)=O)C2)c(=O)o1 Cc1nn(C2CCC2)cc1C(=O)NCC1CC(O)CN1C(c1ccc(F)o1)=O c1(OC(C(C)(C)C)=O)ccc(NC(c2ccc(C(C)(C)C)cc2)=O)cc1 N1(C(CC2(OC)CC2)=O)CCCN(C(c2ccc(N3CCCC3)nc2)=O)C(C)C1 C(=O)(C(CC(C)C)OC)NC1(CF)CCN(C(c2c(CC)ccs2)=O)C1 CCC(C)(C)C(O)C(=O)NCC1(F)CCC(NC(=O)CC2(O)CCC2)C1 N1(C(=O)COc2cccnc2)CCN(C(C2(C(F)F)CC2)=O)CC1CO CCCC(C(=O)N1CC(c2nncn2C)C1)NC(=O)CC1CCCOC1 C1(C(=O)NCCC(C)NC(C2(CCOC)CCCC2)=O)CCOC1(C)C Cc1cc(C)n2ncc(C(=O)NC3CC(O)CN(C(C4CN(C)C4)=O)C3)c2n1 C(=O)(C(C)Cc1cnc[nH]1)N(CC(CN(C(CC1CC(C(C)=O)C1)=O)C)O)C C=CCC(C(=O)NCC1(NC(C2CCCSC2)=O)CC(OC)C1)C(C)C N1(C(C2CC(=C)C2)=O)CCC(C)N(C(=O)CCCC(C)c2ccccc2)CC1 C1(C(C)C(=O)NC2(C)CSC2)CCN(C(C2CC3CC3C2)=O)C1 N1(C(C(C)NC(N)=O)=O)CCC(C2CCCN(c3ncnc4c3CCO4)C2)C1 C(=O)(CC(C(F)(F)F)NC(c1cc(C)cc(O)n1)=O)Nc1c(OC)c(F)ccc1 c1(C(=O)NCCC(=O)NCC(COC)OC)cc(C)cc(C#N)c1 Cc1cc(C(=O)NC2CC2CNC(C2CCC(C)(C)OC2)=O)nc(O)n1 c1(C(=O)NC2C(NC(C3=C(C)OCCC3)=O)CCC2)ccc2nc(CO)[nH]c2c1 Cc1ccc(C(=O)N)c(N)n1.C1CCN(C(C2CN(S(C)(=O)=O)C2)=O)C(C)C1 N1(C(c2scc(C)c2)=O)CCCC(C)C1CNC(c1cc(Br)ccn1)=O Cc1ccc(C(=O)NC2CCN(C(c3nnn(C4CC4)c3C)=O)C(C)C2)nc1C C(=O)(CCC(C)(C)C(=O)NC)OC.C12(C(N3CCC(C)C3)=O)CCCC1OCC2 C1(NC(c2ncc(OC)cn2)=O)CN(C(c2cc(Br)cnc2C)=O)CCC1O C(=O)(CC(C)(C)C)NCC#CC(=O)NCC1OCC(C)C1 c1(NC(C(OCC)OC)C)nccc(=NCCSC(C)(C)C)[nH]1 c1(CC(=O)N(CCNC(c2c(CCC)[nH]cc2)=O)CCOC)ccnnc1O C1(C(N2CCCC(N(C(C(C)(C)OC)=O)CCF)C2)=O)CCc2nnn(C)c2C1 N1(C(c2cc(OC)cc(C)c2)C(=O)NC2CC(F)(F)C2)CCCc2[nH]ccc2C1 Cc1[nH]nc2cc(C(=O)NC(C)(CNC(=O)CN3CCC(C)CC3)CO)ccc12 C1(N(C(=O)C(C)(C)NC(=O)CC2CCCC3CC23)C)CCCCC1(C)C Cc1ccn2c(-c3ccc(CN4CC5CCC(C4)N5C)c(F)c3)nnc2n1 CC(CNC(=O)COC1(C)CCCC1)C(=O)NCCC1CC=CCC1 CCC(CCC(=O)N1CCCC1C1CCN(C(C2CCCCCCC2)=O)C1)OC C1(NC(c2cccc(C(C)C)c2)=O)CC2CN(C(=O)C=C3CC3)CC12 N1(C(CN(CC)CC)=O)CCCC1C(C)NC(=O)CCN1CCC(F)C1 N1(C(c2ccc(C)nn2)=O)CC2CCN(C(c3ccnc(S)c3)=O)CC(C2)C1 c1(C=O)cc2[nH]nc(C)c2cn1.CCC(C)OCC(=O)NCCC1(C)CC1.N c1(C(N2CC(NC(C3(COCC)CC3)=O)C2)=O)noc2cc(Cl)ccc12 c1(N2CCN(C(c3c(OC(C)C)cccc3)=O)CC2)ncnc2[nH]c(Br)cc12 N1(Cc2scc(C)c2)CC2CN(C(=O)NCCCc3ccccc3)CC2C1 CCC(CC)C(C(=O)N1CCC(C)CC1C(C)O)N1CCOCC1 C1(C(=O)NCC(CC)CO)COC2(C1)CN(C(=O)C=Cc1ccnn1C)C2 c1(C(=O)NCCC2(O)CN(C(c3c(CC)noc3)=O)C2)c[nH]c(C)cc1=O C1(NC(=O)C=CC2CCOCC2)CN(C(C2CCC2)=O)CC12CCC2 c1(OC)cccnc1CNC(C1CCCC1NC(c1ccnc(O)c1)=O)=O C1(CC(C)O)CCCN1C(=O)CNC(c1scnc1Cl)=O Cc1n[nH]c(C)c1SCC(=O)N(CCCNC(C1CCCCC1O)=O)C c1(C(N2CCC(CN(C(=O)CCN3CCC3)C)C2)=O)cnn2ccnc(N)c12 Cc1nn(C)cc1-c1cn(C(C)C(=O)NCC2(OCCO)CCC2)nn1 c1(OCCC(=O)NCC23CC(NC(C4CC4Cl)=O)(CO2)C3)ccccc1F c1(OC)ccccc1C(C)C(=O)NC(C)CC(C)NC(c1ccn(C)n1)=O c1(C(C(=O)Nc2ccccc2O)N(CC=C)CC2CC2)ccc(Br)c(Cl)c1 Cc1cc(C(=O)NCC2(NC(c3cc(O)nn3C)=O)CCOC2)cc(C)c1N Cc1cnc(NCC2CC(O)C2)c(S(=O)(=O)N(C2CCCC2S(C)(=O)=O)C)c1 C(=O)(CC(CNC(=O)C=O)C(F)(F)F)Nc1cccc(OC)c1.c1nccs1 C1(CNC(C(COC)C)=O)CCN(C(=O)CC(C)(C)C(F)F)CC1(F)F c1(OC(C)C(=O)NC2CCCC2CNC(C2CCOCC2)=O)ccccc1 N1(C(C(C)(C)NC(C)=O)=O)CC2(C(N3CC4(CC4)C3)=O)CC1CO2 c1(N2CC(NC(C(C)SCCCC)=O)(CO)C2)ccc([N+](=O)[O-])cc1C c1(OCC(N2CCCC2C2(NC(=O)C)CC2)=O)ccc(F)cc1.c1ccsn1 c1(C(=O)NC(CC)CN(C(=O)C(O)CC)CC)nn2c(c1C)OCCC2 C(=O)(C(C)(C)CCC#N)N1CCN(C(C2C(C)C2C)=O)C(c2nccn2C)C1 N1(CC(=O)Nc2n(C)ccn2)CCCC(C(F)(F)F)CC1 C1(NC(c2nc(OCC)sn2)=O)(CO)CCN(C(C2(OC)CCCSC2)=O)C1 N1(C(C(=O)OCC)=O)CCC(CNC(C2CC2(C)CC)=O)C(O)C1 CC(C)(C)CC(O)CC(=O)N1CCCC1(C)C(N1CC(C)(C)C12CCC2)=O c1(C(C(=O)NCCNC(Cc2c(C)cccc2)=O)=O)ccc(Cl)cc1O C(=O)(C1=CCCCO1)NC(c1cccc(C)c1)CNC(=O)CN1CCOCC1 c1(OC)cc(N)ccc1C(N1CCCC(N(C)C(C2CC2(F)F)=O)CC1)=O N1(C(c2c(CC)cns2)=O)CCOC(CCNC(c2cccn2C(C)C)=O)C1 c1(C(N(C2CCCN(C(CSCC=C)=O)C2)C)=O)cnc2sc(C)cn2c1=O CC1CC2(C(=O)N(C)CCN(C(=O)Cc3ccccc3)C)CC12.C(=O)CC N1(C(Cc2cc(C)nn2C)=O)CCCC12CCN(C(C1(CO)CC1)=O)C2.C(C)C N1(C(c2cc(I)cc(I)c2I)=O)CCC2(CC1)CC(O)CO2 CN1C(=O)CCCC1C(=O)NC1CCC(NC(C2CNC(=O)N2C)=O)CC1 CC(C)C(C(=O)NCCCN1CCCC1)C(C)NC(=O)CCCC(=O)C1CC1 C1(NC(c2c(C)con2)=O)CN(C(c2cc(=O)cc[nH]2)=O)C2CCCCC12 CN1CCC(O)(CNC(=O)CC2CCCC(NC(c3cn[nH]c3)=O)C2)CC1.C N1(C(C(F)(F)Sc2cn(C)nc2)=O)CCOC(C)C1.C1(C)(C=O)COC(=O)C1 c1(C(=O)NC2CC(NC(C(CCC)O)=O)C2)n[nH]c2c1CCSC2 N1(C(C2CCC(CC)O2)=O)CC(CNC(=O)CC(=O)N)CC1(C)C.C1CC1 N1(C(C(CC)CN(C)C)=O)CCC(CNC(=O)CN=S(C)(C)=O)C(F)(F)C1 C(C(C(=O)NC1CCCOC12CCC2)C(C)(C)C)NC(c1c(C)cn(C)n1)=O CC(C(=O)NCC1CCN(C(C2CCCCC2C)=O)CC1C)S(N)(=O)=O C(=O)(C(C)(C)C1CCCN1C(=O)CCOCC(C)C)N1CC(SC)C1 C=C=CCCC(=O)N1CC(CNC(c2csc(C(C)=O)n2)=O)C1 C1(NC(C(C(CC)C)O)=O)CC2CCC1CC2NC(c1cn(C)nc1CO)=O c1(CC(N2C(C)CC(CNC(=O)Cc3ccco3)C2)=O)ccc(Cl)nc1F Cc1nc(CNC(=O)C(C2CCCC2)NC(=O)CC2COCCO2)co1 C(=O)(CC(C)(C)C(F)F)NC1CN(C(c2cc(C(C)C)[nH]n2)=O)CC(C)C1 C1(C(=O)NC2CC(SC)C2)CC2(CCN1C(c1cc(CO)ccn1)=O)CC2 N1(CC2CC(C)(C)OCC2)CC2CCCC1C2c1cn(CCCCCCO)nn1 c1(C(=O)NC(CNC(CCOC)=O)C)ccc(Cn2ccnn2)cc1 N1(C(Cc2c(C)cccn2)=O)CCCC12CCN(C(c1ccccc1Cl)=O)CC2 C(=O)(C(CC(C)CC)NC(C1CCC1)=O)NCC1(CCOC)CCC1.O CCCCCNC(c1cn(CC2CC2)nn1)=O.C(=O)(C)N.CCCN(C)C Cc1cnc(S(C)(=O)=O)nc1N1C(C(N2CCCC(C)(O)C2)=O)CC2CC12 N1(CCn2cc(C3(OC)CCOC3)nn2)CCC(F)(F)C(C(=O)N=S(C)(C)=O)C1 c1(C(=O)NC(C(N2C(C#C)CCC2)=O)CC2CC2)cc(CC)ccc1F C(CN=C(NCc1ccnc(N2CCCC2)c1)N1CCCC(C)(C#N)C1)OC c1nc(Cl)c(C)c(=NCC2(C)CCCN(C(=O)C=CC=O)C2)[nH]1.C(C)(C)C c1(N(C)C)ncc(C(=O)NC2CC(n3cc(C4CCCO4)nn3)C2)s1 CCC(CC(=O)NC1C2CCC1CN(C(c1c(C)oc(C)c1C)=O)C2)C(F)F C12(C(=O)NCC(CN(C(=O)CC3C=CCCC3)C)O)CCC(CC1)CO2 C1(F)(CNC(CCCC=C)=O)COCCN(C(c2cc(CCC)on2)=O)C1 C1(CNC(C(C2CCC(=O)N2)C)=O)CCCCN1C(=O)Cn1cnnn1 O=C(C1=NOC2(CCC2)C1)NCC1CC1C(=O)Nc1ccc(C2CC2)cc1 N1(C(C(CC)n2cncn2)=O)CC(NC(c2cnn(C)c2)=O)C(C)(C)C1 c1(NC2CCCC(SCC)C2)ccc(S(=O)(=O)NCC(Cl)(Cl)Cl)cc1Br c1(C(N2CC(O)(C(CNC(c3c(C)cno3)=O)(C)C)C2)=O)ccc(CO)cc1F c1(C(N2CC(CN(C(C(C=CCCC)O)=O)C)OCC2)=O)nc(C)ccc1F CCCC(C(=O)OC)C(=O)NCC(C(N1CC2(CC2)CC1C)=O)N(C)C c1(C(=O)NCC2CC3CN(C(c4ccc(C)o4)=O)CC32)nc2cc(O)ccc2[nH]1 c1(C(=O)NC(CC)C)ccc(C)cc1OC.N12CCC(C1)CCNC(=O)C2C c1(C(N(C(CNC(C=CCCC)=O)C)C)=O)nc(C2CC2)sc1Br c1(CCNC(c2n(CCCSCC)nnn2)C2(CC)CC=CC2)cccnc1 c1(C(=O)OCC)cscc1.C12(C)CC(C1)C(=O)N2.C1(C=O)CCCC1.N N1(C(COCC=C)=O)CC2CS(=O)(=O)CC2C1.C1(C=O)CCC(=C(F)F)CC1 N1(C(=O)CC2C=CCC2)CC2(CCN(C(C3(c4cccs4)CC4(CC4)C3)=O)C2)C1 N1(C(C(CC)C2CCOCC2)=O)CCN(CC2(NC(=O)C(C)(C)CO)CC2)CC1 CCCC(C(O)C(=O)Nc1cccc(C(F)F)c1)NC(=O)CCC1CCC(=O)C1 c1(CC)ncnc(N2CC(C(C)NC(C3COCCN3CC(F)F)=O)C2)c1F N1(C(C(C(C)(C)O)F)=O)CCC2(CC1)CC(CNC(=O)C(O)c1ccco1)C2 CP(C)(=O)C(CC(=O)N1CCCC1C(=O)NC)c1ccccc1.C1(C2CC2)CC1 CCCC(CNC(c1nnnn1CCCF)c1ncc[nH]1)OC CC(C)CCCC(C)C(=O)NC1(C)CC(NC(c2ccc([N+](=O)[O-])o2)=O)C1 O=S(=O)(c1ccc(O)cc1)Nc1ccn(C(c2ccccc2S)C(=O)O)n1 CCC(C)C(=O)NC(c1nocc1C(=O)N(C1(C2CC2)CC1)C)C C1(C(F)F)CCN(C(c2ccnn2C2CC2)=O)C1.CC=O.NC=O.C(N)=O.N c1(C=O)ccc(P(C)(C)=O)o1.C(CCC(=O)NC1CCCC1C)OCCC.N c1(C(N(C2CCN(C(=O)C(C)C3CC3)C2)CC)=O)ccc(-n2nnnc2O)cc1 c1(C=O)cc([N+](=O)[O-])cnc1N.C1(NC(C(=C(C)C2CC2)F)=O)CCC(C)C1 c1(C(=O)NCC(CC)N(C(=O)C(c2ccccc2C)C)C)cnn(C)c1C#N CC(CN=c1ccc(S(C)(=O)=O)c[nH]1)C(C)(C)NC(=O)CC12CCCC1C2 C1(CNC(C(c2ccn(C)c2)C)=O)CCN(C(C2CC23CCCC3)=O)C12CC2 c1(C(=O)NCCCCC(C)NC(C(C)SCC)=O)cc(=O)c(OC)co1 CCC(CN(C(=O)CCc1ccoc1)C)NC(=O)CSCC(=O)OC c1(NC(CNC(CCc2cn(C)nn2)=O)CO)ccc([N+](=O)[O-])cc1[N+](=O)[O-] Cc1cc(C(N2CCC2CO)=O)ncc1-c1cc(OC(F)(F)F)cc(F)c1 C(=O)(NNc1ccc(F)cc1OC)NC(C(COCC)n1cc(CNC)nn1)=O c1(C(N2C(COC)CN(C(=O)CC(C)COC)CC2)=O)cc(F)cc2nc[nH]c12 C1(NC(CC(C)(C)OC)=O)CCC2CN(C(c3ccc(Cl)c(C)c3O)=O)CC12 Cn1cc(S(=O)(=O)NCCc2nnc(-c3cccc(Cl)c3)s2)c2ccc(Br)cc12 CCCCC(C(=O)NC(CC(C)C)C(=O)N(CC1=CCSC1)C)C(C)C N1(C(CCC)=O)CCCCC1C(=O)NCCNC(C1(OC)CCOCC1)=O C1(C)(C(=O)NCC(C)(O)C2CC2)CC(NC(=O)Cc2cc[nH]c2)C1 C(=O)(C(C)(O)C1CCC1)N(CCNC(=O)CC1C=CCC1)CC C1(O)(C(C(=O)NC2C(NC(c3cn(C4CC4)cn3)=O)C2)F)CCCC1 c1cc(C)c(OCOC)c(C)c1.C(=O)(C(C(C)O)NC(C1CC2CC2N1)=O)OC c1(-c2c(NC(CONC(=O)C3CC3(F)F)=O)nco2)c(Cl)cccc1Cl C=C=CCCC(=O)NCC(CC(C)C)NC(=O)CCN1CCCC(C(N)=O)C1 c1(C(N2CCC(C)CC2CNC(=O)Cc2cnc[nH]2)=O)cc2ccccc2[nH]1 c1(CC=O)ccc(C(=O)N(CC)C2CC2)cc1.C(=O)C(C)=C1CC1.C N1(C(=O)C2CC2)CCCC1.c1ccon1.C(C(F)(F)F)NC(C1CC1)=O.O C(=O)(C(CC(F)F)N(C)C(c1cnsc1C)=O)N1C(CC(=O)OC)CCC1 Cn1nnc(C(F)(F)F)c1CNC(=S)NC1CC(C)(C)C1 N1(C(C=CCC)=O)CC(CCNC(=O)C(C2CCOCC2)O)(OC)C1 CN1CCC2(CCN(C(C3CCCCN(C(c4cn(C5CC5)nn4)=O)C3)=O)C2)C1 C#CCC(C(=O)NCC(CC)NC(c1cnc(C(C)C)s1)=O)C1CC1 c1(C(=O)NCCCC=C)cc(Cl)c(N)cc1F.C1(CC(=O)N)CCCC(C)(C)O1 N1(C(CC(C(=O)OC)C)=O)CCCC12CCN(C(c1ccc(S(C)=O)cc1)=O)C2 C1(NC(C(=O)OCC)=O)CCc2onc(NCC(C)Oc3ccccc3)c2C1 C1(C(=O)NCCN(C(c2cn(CC)nn2)=O)C)CCCCC1(F)F Cc1cc(=O)ccn1CC(N1CCC(NC(c2cccc(=O)o2)=O)C1)=O n1(CC)cc(C(=O)NCC(C)CNC(c2cn(C)nc2)=O)c(C(C)C)n1 C(=O)(CC(O)(C(F)(F)F)c1ncc[nH]1)N(CCC)CC.C(=O)CC.C(C)C.N C1(NC(CNS(N(C)C)(=O)=O)=O)CC2CCC1CN(C(c1sccc1C#N)=O)C2 c1(NCC(C)N(C(C(COC)C)=O)C)cc(C#N)ccc1[N+](=O)[O-] C1(NC(c2sc(CC)c(C)c2)=O)CCC2(CCCN(C(=O)OC(C)(C)C)C2)C1 C1(CC(=O)NC(C)C(CO)NC(=O)CSC(C)(C)C)CC(=O)NC1=O CCCC(C(=O)OC)C(=O)N1CCC1(C)CC(=O)NC(CC(F)(F)F)C1CC1 N1(C(C(C)NC(CC(CC)C)=O)=O)CCc2ccsc2C1 C1(NC(c2cccc(-n3ccnc3)c2)=O)CC2CC1N(C(c1ccon1)=O)C2 Cc1cc(Cl)ccc1C(=O)NCC(F)CNC(=O)Cc1cc(C2CC2)nn1C c1(C(N(C2CCCN(C(C3CC=CCC3)=O)CC2)C)=O)n[nH]c2c1CC1CC21 O=S1(=O)CCC2(CC1)CC(N=c1[nH]c(=NCC3CC(F)C3)[nH]c3cccnc13)C2 c1(C(=O)NC2C(N(C(c3cc(CC)ncn3)=O)C)CCCC2)cnc(O)c(C)c1 C1(C(C)NCc2ccccc2)CCC12CCC2.c1(N2CCCN2)c[nH]c(=N)s1 C1(CNC(c2c(C)c[nH]n2)=O)CN(C(C2C3CCCC23)=O)C2CCCC2O1 C(=O)(C1=CCCOCC1)NCC1CCCN(C(C(c2ccccc2F)C)=O)CC1 n1(CC(=O)NC(C(C)NC(C2CC(F)C2)=O)(C)C)ncc(O)nc1=O C1(C(=O)NC2(C(N)=O)CC2)CCN(C(=O)C(F)CC2CCOC2)CCO1 n1(CC#C)c(C)cc(C(=O)N(CC(C)C)C(C)CO)c1C c1(C(=O)N)cc(Cl)ccc1-n1ccnc1.C1(NC(C=CC)=O)(C)CCCCC1 C1(CCNC(C(C)=C(C)C)=O)CCN(C(=O)CC(C)O)CC1.C(=O)C1CC1 C(=O)(C(C)CC(C)C(C)=O)N1CCCC(C)(CNC(c2cn(CC)nn2)=O)C1 C1(OC)CN(C(c2cccc(=O)o2)=O)CC1NC(=O)C(c1cccnc1)C N1(C(c2c(CC)cccn2)=O)CCc2ccc(-c3cccc4nccn34)cc2C1 c1(C(C(N2CC(NC(c3cscn3)=O)C3(C2)CC3)=O)(F)F)ccc([N+](=O)[O-])cc1 C1(C=O)CN(S(N)(=O)=O)C1.C1(C(N)=O)(C(=O)NCC2CC2)CC1.C C1(C(N2CC(N(C)CCO)C2)=O)CC12CCN(C(=O)C1=CCCC1)CC2 N1(C(C2N(C(CCC(=O)NCC)=O)CCC2(C)C)=O)CC(C)(C)C12CCC2 CCC(CC)(C(=O)N(CC(C)NC(c1cnn(C(C)(C)C)c1C)=O)C)OC C(=O)(CC(F)(F)CS(C)(=O)=O)NC1C(F)CCN(C(CC(CC)C(C)C)=O)C1 C1(c2c(C(C)(C)C)noc2)NC(=S)N(C2CC2)C2=C1C(=O)NC21CCCCC1 C(=O)(C(C)(CO)NC(=O)CNC(=O)C(C)(C)C)N(CCOCC)C C1CC(C(=O)N2CCC(F)(C(N)=O)C2)=NO1.c1(OC)cscc1C(=O)NC CC(CCCN=c1[nH]cnc(Cl)c1[N+](=O)[O-])NC(c1cc(C2CC2)on1)=O C1(CNC(Cc2cn(C)nc2)=O)CC(F)CN1C(c1csc(-c2cn[nH]c2)c1)=O N1(C(C=CCOC)=O)CCN(C(c2coc(C)c2)=O)CC1c1ccccc1 C(=O)(CCCCCN(C(=O)C(C)(C)Oc1ccc(Br)cc1)C)NCC C(=O)(C1=CCCSC1)NC1CCC(C)(CNC(C(CSC)(C)C)=O)C1 C1(C(N(CC(CNC(C2(C(C)C)CCC2)=O)C)C)=O)CCCN1C1CC1 C(CC(=O)NOCC=CCl)(N(C(C1C(C(C)C)C1)=O)C)C1CC1 C1(C(=O)NC(CCNC(c2c(SC)csc2)=O)C)CC2(CCOCC2)C1 C12(NC(C3CC34CC4)=O)CCCC(CN(C(=O)C=Cc3cccs3)C1)C2 C#CC1(C(=O)NCC2CCOC(C)C2)CN(C(c2ccn(C)n2)=O)C1 C1(NC(C2C(C=C)CC2)=O)C2CCC1N(C(=O)C=C1CCN(C)C1)C2 CCCCCCC(=O)NCC(C(C)(C)C)NC(c1cccc(-n2cncn2)n1)=O C=C=C(C)CC(=O)NCC1(C)CC(NC(c2cccc(-n3cnnn3)c2)=O)C1 C1CC(O)CN(C(=O)Cc2nc(C(C)(C)C)cs2)C1.CC(C(=O)N)=CC1CC1 N1(C(c2c(CC)c[nH]n2)=O)CC(C(=O)NCC2(C#N)CCCCC2)CC(C)C1 C(=O)(C1=C(C)CCCC1)N1CCC(C)(NC(C(C)=CC)=O)CC1 c1(C(C(=O)NC(C)CC)N(CCC)CCOC)ccc(Br)c(C(=O)OC)c1 C1(C(=O)NC(c2nn[nH]n2)CC)CC2(CC(NC(=O)CCn3cnnn3)C2)C1 N1(C(CN(CCC)C(c2csnc2Cl)=O)=O)CCCC(C)(O)CC1 C1(C(N2CC(CCNC(C(C)OCC)=O)C2)=O)COC2(CO)CC1C2 C1(CCOC)CCN(C(=O)CC2CC2C(F)(F)F)C1.c1(C=O)cscn1.N c1(OC)ccccc1-c1cc(C(N2CC(C)C2)=O)n[nH]1.C(=O)(C(CO)N(C)C)N N1(C(C(CCC)NC(C2CCCN2CCC)=O)=O)CCN(CCO)C(=O)C1 c1(OC(C)C)cccc(C(=O)NCC(F)CNC(=O)Cn2cncn2)c1 C(CC(C)(O)C(=O)N1CCCC1CC(=O)NCCCc1nccs1)N(C)C CC(CC(=O)NCc1cnc(O)nc1O)C(C)(C)NC(c1n[nH]c(=N)[nH]1)=O N(C1CN(Cc2ccccc2)Cc2ccccc21)C(N(CC(C)OC)CC)=O O(C=C(C#N)C(=O)NCCN(C(=O)C(C)NC(=O)COC)C)CC C1(NC(C2(C)N(C)CC(O)C2)=O)CCC2CN(C(c3cscc3C#N)=O)CC2C1 CC(C)C(Cc1ccccc1)C(=O)NC(C)CC1CCCN1 c1(N2C(C)CN(C(=O)C(=O)NC3CC4CC4C3)CC2)nc2ccccc2s1 C1(NC(c2n(CCC)ccc2)=O)CCN(C(=O)CCc2ccc(C)s2)CC1O c1(C(=O)Nc2c(-c3ccc(OC)cc3)nn(-c3ccccc3)c2)nnn2c1N(C)CCC2 C(C(CC(C)C)NC(c1cnoc1C1CCC1)=O)NC(CCC1CC(OC)C1)=O c1(C=O)c(N)cc(C)cc1F.C12COC(C1)C2.C1(SC)CC(C(=O)NC)C1 C1(CN(C(c2c(C)scc2)=O)C)C2CN(C(=O)CC3CCCCN3C)CC12 c1(C(=O)NCC2(F)CCCN(C(CC(CC)(C)C)=O)C2)cnn2c(C)cccc12 CC1CC(CO)CN(C(C23CC(NC(c4cccc(CO)n4)=O)(C2)C3)=O)C1 c1ncc([N+](=O)[O-])cc1F.c1(C(=O)NC2CC(CN)C2)cccn1C1CCCC1 N1(C(CC(C)F)=O)CCN(CC(C)NC(=O)C=CBr)CC1 Cn1cc2c(n1)CC(C(=O)NCC1CCN1C(c1noc3c1CCCC3)=O)CC2 CCCCC(C)C(=O)NCCC1(O)CCN(C(C2NC(=O)CC2C)=O)CC1 C(CN=c1[nH]nc(C2CC2)s1)(CC(C)C)NC(C1(OC)CC1)=O c1(CC)n[nH]cc1CNC(=O)N(C)CCOCCO CCC(CC)C(F)C(=O)N1CCN(C(=O)CC(O)CC(C)C)CC(O)C1 c1(NC(C2OCC2(C)C)=O)ccc(C2(C)CNC2)cc1 C1(CNC(c2c(CC)[nH]nn2)=O)CCC(C)CN1C(=O)CCc1csnn1.C c1(OC)cc(O)ncc1C(=O)N.C1(C)CCN(C(C2CCN2C2CCCC2)=O)C1 C12CC3CC(CC(C3)C1)C2.CC(C(=O)N)C(F)(F)F.C1(C=O)CCN(C)C1.C N1(c2snc(COC)n2)CCC(C)C1CNC(c1cccc(F)n1)=O Cc1cccc2cccc(C(N3CC(NC(=O)CCCN=[N+]=[N-])CC(O)C3)=O)c12 C(CCC(O)C(=O)OC)NC(C(N1CCC2CCCC12)c1ccn(CCC)n1)=O N1(C(c2c(C)nn[nH]2)=O)CCCCC1C1(CNC(c2cncs2)=O)CCOCC1 c1(-n2ncc(C(N(CC(C3CCC3)OC)C)=O)c2)cccc(Cl)c1 n1(CC)nc(C(N2CCOC(CC(N3CC(OC)CC3CF)=O)C2)=O)cc1O c1(C(=O)NC2CC2C(N2CCOC3CC23)=O)ccnc2ncccc12 C1(C)(C(N(CC(C)NC(=O)CC2CC2)C)=O)CC2CCC(C1)S2 N1(C(CCCC(=C)C)=O)CC2CN(C(C3CC34CCOCC4)=O)CC2(C)C1 C1(C(=O)NC2(C(=O)NC(CCN(CC)CC)C)CC2(C)C)COCCC1C C1(CC)CN(C(C2CC(C)CO2)=O)CCC1NC(c1cc(F)ccc1O)=O Cc1ccc(C)c(C(=O)NCC(=O)NCC(N2CCSCC2CO)=O)c1 C(=O)(C1=NOC(C)(C)C1)N1CCC(C)C1C.c1(C2(C=O)CC2)ccn(C)n1.N c1(C(=O)NCC23C(CN(C(C(CCOC)C)=O)C2)C3)cc(C2CC2)ccc1F C1(C2(NC(C3C(CC)C3)=O)CC2)CCCCN1C(c1cnc(N(C)C)o1)=O C1CC2CCC(C1)N2C(C1CC2(C1)CC2F)=O.O=C(CCOCC(F)F)N.C c1(N2CCC3(C(C(=O)NCCCCCCCC)C3)C2)ncnc2n[nH]c(I)c12 N1(C(CCOCC#C)=O)CCN(CCCNC(c2cc(CCC)n(C)n2)=O)CC1 N1(CC)CCN(C(=O)CC2CCCN(C(C3(C)CCN(C)C3)=O)C2)CC1 c1ccc(F)cc1F.N1(C(C=CC)=O)CCCC1CCCNC(C1(O)CC1)=O C(=O)(CCCCC(C)(C)C)NCC1CCC(C(=O)NC(c2nc(C)sc2)C)C1 C(=O)(C1=CCCCCC1)NC1(C(=O)NCCC2CC2C)C(C)C1 N1(CC)CCCC(Cc2nc(C)cs2)C1.C1(C)(C2CC2)C(C)NC(=O)N1 C1(CC(=O)NCC2CCN(C(c3ccn(C)n3)=O)C2)CC2(CCOCC2)CO1 C(=O)C(=O)N=c1cc(C)o[nH]1.N1(C(C(C)=CC)=O)CSCC1C=O.CCC.N CN1C(=O)CN(C(C2CCN(C3CC3)CC2)=O)CC1=O CCCCCC(C)(C)CN(C(=O)C(=O)N(C(C)CC(F)(F)F)C)CC c1(C(=O)NCC(C)NC(=O)Cc2ccn3cncc3c2)ccc2cncn2c1 Cc1cccc(C(F)C(=O)NCc2ccccc2)c1.C1(C(=O)N)C2CN(C)CC12 N1(C(CSCCC)=O)CCC(C)(C)C(NC(=O)Cc2c(C)cnn2C)C1 c1(C(CC)OC(C2CC2c2csc(Br)c2)=O)ccc(F)cc1F c1(CC)cc(=NCC2(O)CCCN(C(C3(C)CCNC(=O)C3)=O)C2)[nH]cn1 S(=O)(=O)(c1cccc(=NCC(O)c2ccco2)[nH]1)NCc1scc(C(N)=O)n1 C(=O)(C(CCNC(=O)C(C)OCC(C)C)OC1COC1)OCC N1(c2nc(C)nc(=N)[nH]2)CCC2(CC1)COC(CNC(=O)C1=NOCC1)C2 C(=O)(C(CCC(N)=O)Sc1ccncn1)NC1CN(C(C2(C)CC2)=O)C1 C1(C(=O)NC(C(C)NC(=O)C=CCN2CCCC2)CO)CCC(C2CC2)CC1 C1(NC(CCN(C(C)=O)C)=O)CC(NC(=O)CC2(O)CCC2)C(O)C1 C1(NC(=O)Cn2ncc3ncccc23)CCN(C(=O)C(O)C(F)(F)F)C12CCC2 c1(C(N(CCCNC(C(C)CC2CC2)=O)CCO)=O)cc(F)cc(Cl)c1 CC1CCOC(C(N2CCSCC2CC)=O)C1.C1(OCC(=O)NCC)CCOCC1 N1(C(C=CCN(C)CC)=O)CCCC2(NC(=O)Cc3csnn3)CCCC12 C(CC(N)=O)(C(=O)N(CC(C)(F)F)C)NC(C(N1CCCCC1)C)=O N1(C(C2(C)CC2(F)F)=O)CCCCC1C(=O)NOC1CC2CCC1C2 C1(C(=O)NC(c2nocc2C(N2C3CSCC2C3)=O)C)CCCCCCC1 C1(C(N(CC)Cc2ccc(OC)c(O)c2)=O)CCn2c(Br)cnc2C1 c1(C(N2CC3(C)CC2(C(=O)NCCC2(C)N=N2)C3)=O)cc2ccccc2[nH]1 N1(C(C(=O)NCCC)C)CCC(NC(=O)CN2CCCC2=O)C(O)C1 c1(C(=O)NC2CCCN(C(=O)C(F)(F)c3cncs3)C2)ccnc2[nH]ncc12 c1(C(N2C(CNC(CCCN(C)C)=O)CCCCC2)=O)cc(F)c(O)c(Cl)c1 N1(C(C2(C=C)CCC2)=O)CCC(O)(C2(NC(c3oc(CC)nc3C)=O)CC2)CC1 CC1CC(NC(=O)C(F)Cc2ccccc2)CCN1C(c1cc(C(N)=O)[nH]n1)=O c1(C(CNC(C(C)N(C(C2CN(C3CCC3)C2)=O)C2CC2)=O)O)cccnc1 C1(CC)CCCN1C(=O)C(=O)NCCCN1CCC(C)C1 CCC(C)(C#N)C(=O)N(c1cnn(C(C)(C)C)c1)CC(C)C.C12CCN(CC1)C2 c1(OC)ccc(CN2CCCC(CCNC(c3ccncn3)=O)C2)c(C)c1 Cc1cc(C(=O)NCCC2COCCN2C(=O)C(C)Cc2ccnn2C)cn1C Cn1cc(C=CC(=O)NCC2CC(O)CN2C(=O)C(F)C2CCCC2)nn1 C1(C)(C(=O)Nc2c(CC)nccc2)CCN(C(C2CCCC2O)=O)CC1 CCC(C)(C(=O)NCCCCC(CO)NC(C1CC1c1ccccc1)=O)C(N)=O Cc1cnc(O)n1-c1cccc(NC(C2CCN(CC(=O)O)CC2)=O)c1 N1(C(C2(CC=C)CCOCC2)=O)CCC2(C1)CN(C(C1C3CCN1CC3)=O)C2 C1(C)(CC)C=C(C(=O)N2CCCC2C(C)(C)CNC(=O)C=CCO)C1 C1(CNC(CCc2ccc(C)o2)=O)(NC(=O)CC2CCCO2)CCCCC1 c1(CC(=O)OCC)cn(CC2CC23CCC3)nn1 C(CCCC(=O)NOCc1cn(CCCC#N)nn1)N(C)Cc1ccccc1 N1(C(CSC)=O)CCCC(NC(c2nnn(C)c2C(F)F)=O)C(F)C1 N1(C(C(C)C#N)=O)CC=C(CC(=O)NC2(C)CSC2)CC1 N1(C(C(C=CCCC)O)=O)C2CCC1CC(CNC(c1cc[nH]n1)=O)C2 N1(C(C2C3(CC(OCC)C3)C2)=O)CCC(NC(=O)C(C)OC)C12CCCC2 N1(CC)CCN(c2nnc(C3CC=CC3)n2C2(C(F)F)CC2)CC1.C(CO)OC c1(NC(C2(NC(C3C(OCC)C3)=O)CC2)=O)cccc(C(C)=O)c1 c1(CC)nc(C)c(C(N2CCCC(C)(C)C2)=O)c(C)n1.C1(C(=O)N)CC1(C)C N1(C(CNC(CCCOCC=C)=O)=O)CCN(CC2CCC(=O)N2)CC1 Cc1ccc(CNC(CC(C)(C)C)C(=O)O)c(O)c1F c1(C(C=O)C)cccc2ccccc12.C1(NC(C2C(COC)C2)=O)COCC1.N C(=O)(C(F)CC(CC)CC)NC(CCC=C)C(=O)N1CCC(C)(CCO)CC1 N1(C(C(C)SC)=O)CC2=C(C1)CN(C(=O)CCC1CCC(C)O1)C2 N1(CC(=O)N(CC(C)NC(C2(C)CC2C)=O)C)CCC(C(N)=O)CC1 c1(CC=O)ccc(C)c(Cl)c1.C(=O)C=O.C(C)(C)C1CCC1.C(C)OC.N N1(C(c2n(CC#C)ccc2)=O)CC2(NC(C3CC3(Cl)Cl)=O)CC1C2 CP(C)(=O)c1cccc(C(=O)NC2CCC2NC(C2CCC2(F)F)=O)c1 C(=O)(CC(C)C(=O)NC(C)C(=O)N(C)CC1CCCC1)OC c1(SC)ncc(C(N2CCC(CCNC(=O)C(c3cccnc3)O)C2)=O)s1 Cc1ccc(CNC(c2cn(-c3ccccc3)nn2)C)c2ccccc12 c1(C(N2C(C)COCC2)=O)cn2c(n1)CN(C(c1ccc(NC=O)cc1)=O)CC2 C1(C(=O)NCC2CCC(NC(c3[nH]c(C)c(C)c3C)=O)C2)Cc2ccccc2O1 CC1CCC(CSC2C=CC2)CC1 CC1(C)C(CNC(=O)CC2CCCCC2(F)F)CCN1C(c1ccc(N)cn1)=O C1(NC(C2C(c3ccn(C)c3)C2)=O)C2CN(C(C3CC4(CC4)C3)=O)CC12 C(C)(C(CC(=O)N1CCC1CO)NC(c1ccncc1Cl)=O)OC C1(NC(C(CC2CC2)OC)=O)CC2(C1)CC2NC(c1nc(Cl)cs1)=O c1(C(=O)NCCC2(O)CN(C(c3ccc(Cl)[nH]3)=O)C2)cccc2occc12 n1(-c2ccn(COC)n2)nc(C(c2ccc(F)cc2)O)nc1CSc1cccs1 C1(NC(C(CNC(C=NOC)=O)(C)F)=O)CC12CCCCCC2 C1(C(N2CC3CCC2C3)=O)C2CCCC1CN(S(=O)(=O)c1cc(Br)c(Br)s1)C2 c1(C(=O)NC2CCC(C(=O)NC(C(=O)NCC)C)C2)c(C)oc(C)c1C N1(Cc2c(C)cc(C#N)cc2)CC(C(N2CCN(C)C(=O)C2C)=O)CC(F)(F)C1 C1(C(=O)NC2CN(C(CC3CC(=O)C3)=O)CC2CO)CC1C1CCOCC1 CCS(=O)(=O)CCCN=C(NC(C)C)N1CCC2(CCCOC2)C1 C1COCCN1C(C1(NC(c2cc(C)n[nH]2)=O)CC1C)=O.C(C)(C)(C)C=O.C N1(C(C(CC(=C)C)NC(c2cnsc2C)=O)=O)CCC2(CCOCC2)C1 C(CCC(C)(C)NC(c1ccc(-c2cnn(C)c2)o1)=O)NC(COCC)=O N1(C(CC2C3CN(C(c4snc(C)c4N)=O)CC32)=O)CCC2(CCN(C)C2)C1 c1(CC(=O)N(CCCCNC(C2(OC)CCC(C)C2)=O)C)cn2ccccc2n1 Cc1ccc(CC(=O)NC(C2CCCN(C(=O)CN3CCCC3=O)C2)C)cc1Cl c1(OC(C(c2cccc(Cl)c2)NC(COCCOC)=O)=O)cc(F)ccc1F C1(O)(CNC(c2occc2F)=O)CN(C(=O)COCC2CC2)C1 N1(C(=O)OC(C)(C)C)C2CCC1CN(Cc1cc3cccnc3[nH]1)C2 C1(C(=O)NC2C(CNC(C3CC(=C)C3)=O)CCCC2)CCCC2CCCN12 c1(C(C)NC(=O)NC2CCCC2C#N)ccccc1Cl N1(C(C(C)(C)F)=O)CC(NC(c2cc(-c3ccccc3)[nH]n2)=O)CC2(CC2)C1 CCCCCCC(=O)NCC1CCC1NC(=O)CS(=O)(=O)NCC c1(-n2c(CCCn3ncc(C)c3)nc(C3CC=CCC3)n2)cc(Cl)cc(Cl)c1 N1(C(C2(COC)CC2)=O)CCC(CNC(=O)CC2CC3CC3C2)CCC1 CCC(C=O)C(=O)NCC(C)(C(C)C)NC(c1ccnc(C(C)(C)C)n1)=O.O C1(C(=O)NC2C(C)CN(C(=O)CCC3CCCOC3)C2)CC2C=CC1CC2 c1(OC)ccc(CNC(C2(C(C)C)CCCN2C(=O)CCSC)=O)nc1.O c1(C(N(C2C3CN(Cc4nccs4)CC23)C)=O)ccc(C(F)(F)F)nn1 c1(CC(=O)Nc2ccc(N3CCCS3(=O)=O)cn2)ccc2c(c1)OC(F)(F)O2 C#CC1(C(=O)NCC(C)=CCC)CCN(C(=O)CCc2nc[nH]n2)CC1 C(=O)(C(O)C1=CCCCC1)NC(CCC)C(O)C(=O)NC1CN2CCCC1C2 C1(NC(c2nccc3cc[nH]c23)=O)CCC2(CCN(C(C3CCCO3)=O)CC2)C1 N1(C(C(C(C)C)OC)=O)CC(F)(F)CC1C.n1(C2(C(=O)N)CC2)ccnn1 N1(C(C2(COC)CCOC2)=O)CC(C)C2(C1)CN(C(=O)Cn1nccc1N)C2 c1(OC)ccc(CN(C(=O)COC(c2ccnn2-c2ccccc2)=O)C)cc1F C(C)(C)(CCC(=O)NC1CCCC12CC2)NC(CC(C)SC)=O CC1CN(C(CCCC2CC2)C(=O)N(c2ccccc2)C2CCOC2)C(C)C1C N1(C(C)=O)CCN(C(=O)CN(C(=O)CC2CCC2)C2CC2)CC1.NC=O.N c1(C(N(C2CCN(C(=O)CC3CC(O)C3(C)C)C2)CC)=O)sc2cncn2c1C CCC(CC)CC(F)C(=O)NC(C(N1CC(CC)C(F)C1)=O)c1ccco1 Cc1cc(C(=O)NCC2CCCN2C(C2CCC23CCC3)=O)cc(C)c1O N1(C(C2C(C)CCOC2)=O)CC2CCC(C1)C(NC(C1(CO)CCOCC1)=O)C2 CC1CCN(C(=O)CCc2cocn2)CC1CCNC(=O)OCc1ccccc1 C1(C(=O)NCc2ccc(OC)cn2)N(C(=O)C(SC)SC)CCCC1(C)C CCC(CO)CCNC(c1ncoc1CNC(c1ccc(F)cn1)=O)=O C(C(=O)NOCC1CCOCC1)(C1CCCO1)NC(C(C)C1(O)CCC1)=O C1(O)(C(C)(C)CN(C(=O)CC2CCN2C=O)C)CCCC1.C(C)(C)C Cc1cccc(CC(=O)NC2(CNC(=O)C(C3CCC(=O)N3)C)CC2)c1Cl C(CC(F)F)(C(=O)NC1CCC(F)(F)C1)NC(COCCC)=O Cc1cc(C(N2CCCN(C(=O)C(C)N3CC(C)C3)C(CO)C2)=O)cc(C)c1N C1(NC(CCC2(C)CCCN2C(c2cc(CO)ccn2)=O)=O)CC2CCCCC12 c1(C(N2CCC(NC(C(C)(C)CCl)=O)CC2)=O)cc(F)c(F)c(Cl)c1 C1(C(=O)NCCC2(NC(C(C)CC(N)=O)=O)CCC2)CCC([N+](=O)[O-])CC1 C1(F)(CNC(CCC)=O)CCCN(C(=O)CCc2ccc(F)c(Br)c2)C1 c1(C(=O)NCC2(NC(C=CCC)=O)CCC2)cnc2ncnn2c1CC CC(O)C(C(=O)N1CCCCC1CNC(=O)CO)N(C)C.c1ccc(F)cc1 C(C(CC(C)C)C(=O)NC1(COC)CC(C)C1)NC(CC1CC(CC)C1)=O C1(C(=O)NCC(CC(C)C)NC(=O)C(C2CCOCC2)C)CC2(C1)CC(O)C2 O=C(N1CC(n2cc(-c3cccc(CC4CC4)c3)nn2)CO1)N1CCCC1 N1(C(CN)=O)CC2(C1)CN(C(c1csc([N+](=O)[O-])c1)=O)C2.c1(OC)ccncn1 N(C1COc2cc(F)ccc21)C(=O)Nc1nnc(C(=O)OC(C)C)s1 C1(C(N2CCC(c3nc[nH]n3)C2)=O)(CC)CCN(C(=O)C(CO)N(C)C)CC1 c1(C(=O)NCC2C(NC(c3cnn(C)n3)=O)C2)c(F)cc(N)cc1F C1(CC=C)(NC(C2CCCN2N=O)=O)CCN(C(c2cccnc2)=O)C1 CCS(=O)(=O)CC(=O)NC(C)C(C)NC(=O)CCc1ccccc1.C(C)C.O CC1CN(C(C23CCC(C2)OC3)=O)CC1(C)CNC(C1CC(C2CC2)=NO1)=O CC1CC(O)CCN(C(C2CSCCN2C(=O)CCc2cncn2C)=O)C1 C(=O)(C(Cl)=CCl)NCCCCN(CCCNC(=O)CCc1cnccn1)C Cc1noc(C)c1C(N1CCN(CC(=O)NC2C(C)C2(C)C)CC1)=O C1(C(N2CCCC(CCNC(CCOCC#C)=O)CC2)=O)CCCC1S(C)(=O)=O C(=O)(C(O)CN1CCOCC1)NC(COCCOCC(=O)N)CO.C1CC1 Cn1nc(C(=O)NCC(C)(O)C)cc1C1CCCO1.C(=O)(CC1(C)CC1)N c1(OC)ccc(C(=O)NCC2(C)CCCC2)c(C)n1.C(=O)C.CC(F)F.N c1(C(=O)NCCC(C)N(C)C(C2CCOC2)=O)cccc2c1COCCN2 c1(C(N2CCCC(CC(=O)Nc3ccc(CO)cc3O)C2)=O)ncc(F)cc1F Cc1nn(CCC(=O)NC(C)(C)C(C)C)c(C)c1C.c1(C(=O)N)cc(=O)cc[nH]1 c1(OC)cc(F)ccc1C(=O)NC1CC1NC(c1ccc(C(C)C)nc1)=O c1(C(N2CCC(NC(C3(CC4CC4)CC3)=O)CC2)=O)ccn2ncnc2c1.C c1(OCC#C)c(OCC)cccc1CNC(C)(CO)CC(F)F CCC(CNC(=O)C=CC(C)NC(C1CC(C)(O)C1)=O)(CC)CO Cc1cc(OCC(=O)NCCCCC(C)NC(c2c(C)n[nH]c2C)=O)ccc1Cl N1(C(C2(CC)CCCC2O)=O)CCC2CCN(C(C3CCCCCC3)=O)C2C1 c1(CC)ccc(C(N2CCC(C(O)C(F)F)C2)C(=O)NC2(C)CC2)cc1Cl c1(C(=O)NC2CN(C(C(C)n3cncn3)=O)CC23CC3)ccc2c(c1)COC2 CC1CC(=O)NC1C(=O)NCCCCNC(=O)Cc1cnn(C)c1C(F)F C1(C(=O)NC2CCC(C(=O)NC3C(C)CN(C)C3)CC2)CCC(O)CN1C c1(C(N2C(CNC(c3nccc(CC)c3)=O)CC2)=O)cncc2c(O)nccc12 C1(CC(=O)N(C2CN(C(CN(C(C)C)C)=O)CC23CC3)C)Cc2ccccc2O1 CC(C)CC(C)C(=O)NC1CCCC1NC(c1cccn1C1CCCC1)=O N1(C(c2nc(C)sc2Br)=O)CCC2(CCCN(C(=O)CCC(N)=O)C2)C1 C1(C(=O)NC(C2CCCN2C(c2ccoc2)=O)(C)C)CCc2ccnn2C1 C1(NC(C2(C#C)CCCC2)=O)CC2(NC(=O)C(C(C)(C)C)OC)COC1C2 C=Cn1nncc1C(N1CC=CC(NC(=O)C(c2ccccc2C)C)C1)=O S(=O)(=O)(C1(Nc2ccccn2)CC1)NC(N1CC(O)CC1C(F)(F)F)=O CC(C)C(C)(F)CNC(C1(C)CCCN1C(C1CC(C)(F)C1)=O)=O C1(O)(CNC(c2c(CC)ccs2)=O)CCCN(C(c2ccc(N)c(Cl)n2)=O)C1 N1(C(Cn2ccc(C)n2)=O)CC2C(C(N3CCCC3CCO)=O)C2C1 CC(C(=O)N1CC(C(N)=O)C1)C(C)(F)F.c1(C=O)ccc(C(F)F)c(Cl)c1.C c1(C(=O)NCC2CC(OC)CN2C(c2ncoc2C)=O)ncnc2sccc12 C1(CC)CN(C(C2(N(C)C)CCC2)=O)CCO1.N1(C(C)C(=O)N)C(=O)CCC1=O N1(C(COC)=O)CCCC(F)(COC2CN(C(C3CC(C4CC4)C3)=O)C2)C1 C1(C(N2CCC(CN(C(c3n(C(C)C)ncc3)=O)C)C2)=O)CCCC(=O)N1C N1(C(Cc2c(C)cccn2)=O)CC2CCC(C1)N(C(=O)C(N1CCOC1=O)C)C2 C1(C2(O)CCN(C(c3cc(C4CC4)[nH]n3)=O)CC2)(NC(CC(=O)NC)=O)CC1 N1(C(C2C(C#N)C2)=O)CC2CCC1C(C)C2.n1(CC=O)cnc(C(F)(F)F)c1 C1(CNC(C(C)=C(CC)C)=O)CCCN1C(=O)CC.c1(C=O)ccco1.O C(CC(F)F)(C(=O)Nc1cncc(N(C)C)c1)N(C(C(C)C(F)F)=O)C N1(C(=O)CCOCC(F)F)CC2CCN(C(C3CCC(F)(F)CC3)=O)C2C1 c1(C=O)nc(CC(=O)N)cs1.CC(O)C.C1(CC)CC(C=O)C1.C(C)(C)C CC(C)CCCCC(=O)NCC(=O)N(C)C(c1ccccc1)C N1(C(CC2N(C(C=C(C)C(C)C)=O)CCOC2)=O)CC2COCC(C2)C1 c1(CC(=O)NC2CC(NC(C(C)(C)c3cscc3Cl)=O)C2)ccc2nc[nH]c2c1 C1(CC#C)(C(N2CCOC(C(C)C3CC3)C2)=O)CCOCC1.C1(=O)CC(C)(C)N1 c1(CC(N2CCC(O)C2)=O)nc(F)c(F)cc1F.C1(C(=O)N)CC1[N+](=O)[O-].C S(=O)(=O)(c1ccsc1)N(CC)CC1CCCCN1C(=O)Cc1ccccn1 C(=O)(CCS(=O)(=O)NC(c1ccc[nH]1)C)NCCC(C)N(C(CC(C)C)=O)C N1(C(C(C)NC(CC)=O)=O)CC(=O)NCC1C(N1CCC(C(=O)OC)C1C)=O c1(C(=O)NC2CN(C(c3cnc4n3CCCC4)=O)C2)c(O)nnc2c1CCCC2 c1(CCCCNC(=O)C(=O)Nc2ccc(Cl)cc2CO)cc(F)c(F)c(F)c1 CC1(C)CC(CNC(C2CC(O)CN2C(C2(CO)CCOCC2)=O)=O)CO1 CC(CC(=O)N1CC(C(C)NC(=O)C(N2CCCCC2)C)C1)C1CCCCC1 C(C1c2ccsc2CCN1C(=O)CC1CS(=O)(=O)C1)NC(C(C)CN(C)C)=O N1(C(c2ccc3c(c2)CCC3)=O)CCN(C(C2CC(Cl)(Cl)C2)=O)C2(CCC2)C1 CCCS(=O)(=O)CC(=O)NC1CCCC(NC(C2C=C(C)CS2)=O)C1 N1(CC(=O)NCc2ccns2)CCN(Cc2nnnn2Cc2cccs2)CC1 CCC(C)N(OC)C(=O)C1CCCCCC1NC(=O)CC1(C)CC1 Cc1nc(Cl)ccc1CC(N1CCN(C(C2CC(F)(CO)C2)=O)C(C(C)C)C1)=O C1(C(N2CCN(C)C(CNC(=O)CCc3nc[nH]n3)C2)=O)CCn2nccc2C1 c1(CN(C(=O)Cc2ccsc2Br)CC)cc(Cl)cc(Cl)c1 N1(C(=O)NC(c2ccccc2Cl)CC(=O)O)CCCC(C(c2ccccc2)=O)C1 N1(C(C(CCC)C#N)=O)CC2(CCC2)CC1CNC(c1cnc(C)n1C)=O C1(F)(C(=O)NCCCCCN(C(c2cnc(CC(C)C)[nH]2)=O)C)CCOC1C C1(NC(C2C(CC)C2)=O)CCC(CC(=O)NCc2cc(Br)ccn2)CC1 C1(NC(c2cc(C3(C)CC3)on2)=O)CCCCN(C(c2cc(O)nnc2O)=O)C1 Cc1nn(C(F)F)cc1NC(N1CCC(CO)(Cc2ccccc2)C1)=O c1(C(=O)NC2C(NC(C(C)=C(CC)C)=O)CC2)ccccc1.C1(O)CCCC1 C1(O)(C(C)NC(COCC)=O)CCN(C(c2cnc(C(C)C)nc2)=O)C1 N1(C(COC(CC)C)=O)CCCC(N(C(=O)C(c2cccc(Cl)c2)C)C)CC1 C1(NC(c2n(CC)ccc2)=O)CC2(NC(=O)CCc3ncno3)COC1C2.O c1(NC(=O)NCCc2scc(C)c2)cnc(O)c(C(F)F)c1 c1(C(=O)NC2CC(N(C(CCCCCC)=O)C)C2)c(C)cc(F)cc1C c1(COC)ccoc1C(=O)NC(CNC(c1csc(C)n1)=O)C1CC1 C=CCC(C)(C)C(=O)N1CCCC(C2c3nnnn3N2)C1.c1(CC)scc(C)c1C N1(C(CC(C)(C)C(F)F)=O)CCC2(CCN(C(=O)CC3CCCC3)CC2)C1 C(=O)(C(C)(C)CC(=O)NC1(C)CC(NC(C2CCn3ncnc3C2)=O)C1)OC c1(C(=O)NCC2N(C(C(C)OCOC)=O)CC(F)(F)C2)cc2cccc(C)c2[nH]1 C1(C)(C(N2CCC(OCC#C)C2)=O)CCN(C(=O)CC2(C)OCCO2)C1 N1(CC)CC(C(=O)N2CCOC(C3CC3)C2)c2ccccc21 CCC(C#N)(CC)C(=O)NC(c1ccc(C)cc1)CNC(=O)C.C(C)(=O)N C(=O)(C1=CC2CCCC12)N.C1(COC)(C)CCCN1C(C1CNC(=O)N1)=O c1(CC(=O)Nc2c(C)n(C(C)C)nc2)ccc2c(c1)CN(C)C2=O n1(CCOC)cc(C(=O)NC2CCCC2)ccc1=O.C(=O)CN(C)C(C)=O C=CCC(CNC(c1ccc(=O)n(C)n1)=O)C(=O)NCc1[nH]nnc1C c1(C(=O)NCC2(F)CC(CNC(C(CC)F)=O)C2)ccc(OC)cc1C.O C1(C(N(C2CN(C(C3CCC(F)(F)C3)=O)C2)C)=O)CCc2nccn2CC1 C1(C(=O)NCCNC(CNS(NC)(=O)=O)=O)Cc2ccc(OC)nc2N1 C1(NC(C(CC)N(C)C)=O)CCOC(C(=O)NCC2COCC(C)O2)C1 CC(C)C(C)(O)C(=O)N1CC(C(=O)NCCCOCC(F)F)C(C)(C)C1 C1(NC(CCCNC(c2ccc(C#N)cn2)=O)=O)CCn2nccc2C1 CCC(C)(CCNC(=O)Cn1cccn1)NC(=O)CCc1cncn1C C1(CNC(C(C)N(CCC)C(C2CC(C)(C)C2)=O)=O)CC(O)C(O)C1 S(=O)(=O)(c1ccccc1F)NC(C)C(=O)N(C)CC.C1(C(=O)N)CCC12CCC2 CN=c1[nH]ccc(C(N2CCCC(CNC(=O)C3=CCCC3)CC2)=O)c1N c1(OCC)ccccc1C=CC(=O)NCc1ccc(C(C)(C)C)o1 C1(NC(C(c2ccc(OC)cn2)(F)F)=O)COC2(CCOCC2)C1 C(CCN(C)C(c1cncc(N)n1)=O)C(C)(C)C.c1(C(C)C)cc(C(=O)N)n[nH]1 c1(-c2ccc(C(C)NCC3(CCOC)OCCO3)s2)ccc(Cl)cc1 C1(CC=O)CCCN(C)C1.c1(C=O)cn(C(C)(C)C)nn1.CCCC.C1CC1.N N1(C(C(=O)NCc2nc(C3CC3)n[nH]2)=O)CC2(CCC2)OCC1CO C1(C(=O)NCC(c2ccccc2)CCO)COC2(C1)CN(C(c1ccsc1)=O)C2 c1(CNC2C(C(N3C4CN(C)C(C4)C3)=O)CCC2)cc2ccccc2[nH]1 c1(CN(C)Cc2noc(C3CCC3)n2)nn(-c2ccc(Cl)c(F)c2)c2c1CCC2 N1(C(C2CC(OC)C2)=O)CCN(C)CC1C(=O)NC1CCN(C(C)(C)C)C1 N1(C(C2C3(CC3)C23CC3)=O)CCC2(CC1)CC2C(N1CCCC(CCO)C1)=O N1(C(C2(COC)CC=CC2)=O)CC(NC(C2CCC=CCC2)=O)C(C)(C)C1 c1(C(C(=O)O)NC(C(n2cc(-c3c(C)ccs3)nn2)C)=O)ccccc1C(C)C c1(C(N2CC(NC(c3ccc(C)s3)=O)CC(OC)C2)=O)cc2c(Cl)ccnc2s1 c1(C(=O)NCCC(=C)CNC(=O)C(CCC)N(C)C)cc([N+](=O)[O-])cnc1O C(=O)(C(C)CCC(C)(C)C)N1CCC(C(=O)NC2C(C)NC(=O)CC2)OCC1 c1(CN2C(C(N(C3CCOCC3)CC)=O)CCCC2)cc(Br)c([N+](=O)[O-])s1 c1(N2C(CC)CN(C(=O)Cc3c(C)nn(C)c3C)CC2)ccn2nccc2n1 c1(OC)ccccc1C(O)C(=O)N(CC(C)NC(c1cc(C(C)C)no1)=O)C N1(C(C2CC(C#C)(O)C2)=O)CCCC(C)C1CNC(c1ccsc1C)=O C(=O)(CCCCCNC(c1nc(C)ccc1F)=O)N(CC(=O)N(C)C)CC c1(CC)[nH]nc(C(=O)NCC(CC(C)C)NC(=O)C(C)=CC2CC2)c1C c1(C(=O)NC(CC2CN(C(C3C(C)N(C)CC3)=O)C2)C)[nH]nc2c1CCC2(C)C C1(CNC(C=CCOCC)=O)CCN(C(=O)Cn2cc(Cl)cn2)CC1 c1(CC(=O)N(C2CCCC2)CC)ccc2c(c1)CCO2.NC(=O)CC(O)C(=O)N CCC(CC)C(C)C(=O)NCC(N1CCN(C(=O)CCCOCCOC)CC1)=O C(=O)CC(C)(C)CC(C)=O.c1(CC)nc(N2CCC(NC(=O)C)C2)[nH]c(=N)n1 C(=O)(C1CCCn2cncc21)NCCC(C)N(C(=O)CCc1ccc(F)cc1)C C(N=c1ccn2c(Br)cnc2[nH]1)C1(O)CN(C(C(=Cc2ccc(F)cc2)C)=O)C1 CC(C)CS(=O)(=O)CCC(=O)N(C1C2CN(C(c3ccsc3C#N)=O)CC12)C C(c1nc(C)c(C)[nH]1)=CC=O.C1CCCC1.C1(CC)CC(CC(=O)NC)C1 C1(CNC(c2n(CCCCCC)nnn2)C(C)(C)C)OC(=O)CC1(C)C c1(C(N(C2CCN(C(C(C)C3CCC3)=O)C2)C)=O)ncnc2c1OCCO2 Cc1nc(C(=O)NC(CNC(c2csc(Br)c2)=O)C(C)C)sc1C C(=O)(C1=NNC(=O)C1)N(CCC(=O)Nc1c(CC)ccnc1)CCCO c1(OC)ccc(Cl)c(Cl)c1C(N1CCN(C(=O)C(C)CC(C)C)C(C)C1)=O C(=O)(C(C)CC(C)(F)F)N1C(C)CCCC1.c1(C(=O)OC)ccc(C(=O)N)[nH]1 Cc1cc(C(=O)NC2CCCC2C)n(C(F)F)n1.C(=O)C(C)(C)n1cccn1 C(=O)(CCC(=O)NC(C)CCN(C(=O)CC(C)(F)F)C)NC C1(CC(N2C(C(C)NC(c3ccc(C)cn3)=O)CCC2)=O)CCS(=O)(=O)CC1 c1(C(N2CC(O)C2)=O)ccc(C#N)c(C)n1.C(C)(C(=O)N)(c1ccccc1)OC C(CCCC(=O)NCC(C)(C1CC1)NC(c1conc1C(F)(F)F)=O)OC N1(C(c2ncc[nH]2)C(=O)NC)CCN(CCC(=O)N(C)C)CC1 c1(CS(=O)(=O)NC(c2ccc(F)cc2F)C2CCCC2)cc2cc(F)ccc2o1 N1(C(C)C)CCOC(C(=O)NC(C)CN(C(=O)Cc2cccs2)C)C1 c1(CC)cncc(C(N2CCCC(N(C(=O)Cc3c(C)cnn3C)CC)C2)=O)c1 C1(NC(=O)C(F)=C2CCC2)CCN(C(=O)CCOCC(F)(F)F)CC1F C1(C(C)(C)C)(CNC(C(CN(C)C)O)=O)CCN(C(=O)COC(F)F)C1 Cc1occc(=O)c1OCC(=O)NC.C(=O)C(C)CC1CCCC1.C1CCC1 CCCC(C)CCCC(=O)NC1(CO)CN(C(=O)CC2CCCCC2(F)F)C1 N1(C(c2cc(OCC)no2)=O)CC2CC(C)N(C(C3COCCC3C)=O)C2C1 CC1C(NC(c2cnc(Cl)s2)=O)CCN1C(=O)Cc1ccc(Cl)cc1 c1(C(N2CC(C(C)NC(c3cocn3)=O)OCC2)=O)cccc2c1NC(=O)CC2 c1(C(=O)OC)ccncc1C#CCNC(C1CCCN1C(=O)CC1C=CCC1)=O c1ccc2c(c1)CCC2.CCC(C(=O)NCCCNC(=O)C)NC(N)=O.S c1(OC)ccc(Cl)c(CC(N2CC(CC(C)NC(c3nccnc3N)=O)C2)=O)c1 c1(C(=O)NC(CC=C)CNC(c2cc(O)n(CC)n2)=O)cc2scc(Cl)c2[nH]1 C1(C(N2CCN(CC(C)C)CC2)=O)CCN(C(=O)CC2CCSC2)CCO1 c1(CNC(C(C#C)(C)C)=O)cc(O)nc(C)n1.C(=O)CC(C)c1cnn(C)c1 c1(CC(N2CCCCC(CNC(C(C)(C)C3CC3)=O)C2)=O)n[nH]c2ccccc12 C=C(C)CCCC(=O)NCCCCN(C(=O)CCn1nc(C)c(C)c1C)C C1(SC)CN(C(C2CCC(O)CC2)=O)CC1n1cc(C2CCN(C)C2)nn1 Cc1cnc(C(=O)N(CC(O)CN(C)C(c2coc(C3CCCC3)n2)=O)C)cn1 C(=O)(C1=NOC(CO)C1)N1CCN(CC=C)CC1.C1(=O)C(C)(C)CCN1 C1(OC)CCN(C(=S)Nc2c(C)cc(Br)cc2C)CC1(C)OC C12(C(N(c3c(C)nsc3)C)=O)CC1CN(C(c1cn(C3CC3)nn1)=O)C2 C(C(C)(C)CC(=O)NC(C)CCNC(c1cc2n(n1)CCO2)=O)OC(C)=O C(CC(C)(C)C)(C(=O)N1CC2(CC(C(N3CCCCC34CC4)=O)CO2)C1)OC Cc1cc(=NCC(CO)C(C)C)[nH]c(N(C)CC2CCC2)n1 C1(C(N2CC(C)(C)C2)=O)C2CN(C(c3cc(C(F)F)ncn3)=O)CC12 CC1(C)CN(C(=O)CC2(O)CCCOC2)CCC1NC(c1cc[nH]n1)=O N1(C(C(c2cnn(C)c2)C)=O)CC2CC1CN(C(c1cccc(=O)o1)=O)C2 C1(NC(CCN2CC(=O)NCC2)=O)CC2CCC1CN2C(C1C2CC3C(C2)C13)=O c1(C(=O)NCCc2ccc(OC)c(O)c2)cc2cc(C(F)(F)F)ccc2n1C C(=O)(C(C=O)c1ccccc1)OCC.c1(C(N(CC)C)=O)cc(C)c(C)s1.N N1(C(c2cc(C)nnc2)=O)CCCC2(CCN(C(=O)CC(C)NC(N)=O)C2)C1 C1(C)(OC(C)C(=O)NCC2CC=CCO2)CN(C(=O)CO)C1.C1CCCO1 Cc1cc(C(=O)NC2COCCC2NC(C2CCCC2(C)C)=O)nn1CCO C(C)(C(=O)Nn1cnc2ccccc12)(N(C)C(c1csc(=N)[nH]1)=O)C1CC1 CCCCC(CC(=O)Nc1ccc(F)cc1C)NC(c1cc(C)[nH]c1C)=O C=CCN(OC)C(=O)C(CC(C)CC)NC(c1ccnc(OC)c1)=O C1(NC(CSC)=O)CN(C(c2cnn(C)c2N)=O)CCC1c1ccccc1 N1(C(CC(CC)C)=O)CC(NC(c2ccc(OC(F)(F)F)nc2)=O)CC2(CC2)C1 CC(C)C(CC(=O)N1CCCC(OCCO)C1)NC(=O)CCC1OCCO1 CCCCN=C(NCC(C)CC(F)F)N1CCC(N2CCCS2(=O)=O)CC1 N1(C(=O)CCCC(F)F)CCC2CCN(C(c3occ4c3CCCC4)=O)CC2C1 CCC(CNCC(=O)N(C)Cc1ccco1)NC(=O)Cc1cnoc1 CC1CC=CCC1C(=O)NC(C)CN(C(=O)CC1CC2(CCC2)C1)C c1(C(N2CCC(O)(C(CNC(C(C=C)C)=O)C)C2)=O)cc(F)c(C)cc1O c1cc(C(F)(F)F)c(C#N)c(=NCC2CN(C(=O)C=CC3CC3)CC2C)[nH]1.C c1(CNC(C2(NC(CCC3C(C)C3)=O)CC2)=O)nn(C)cc1CO CCCCC(C(=O)N(CC(O)CN(C)C(c1cc(CC)cc(C)c1)=O)C)C(C)C c1(CC)cccc(CC)c1C(=O)N(C)CCN(C)C(c1c(C)noc1C)=O.S c1(CN(CCC#N)C(=O)NC(C)Cc2ccncc2)cc2ccsc2n1C C=CCC(C(=O)NCCO)NC(C)=O.C(=O)(C(CC)n1ccnc1)N1CCC1 N1(C(C(C)NS(CCCC)(=O)=O)=O)CC(NC(c2cc(C)cs2)=O)CCC(O)C1 C12(C(=O)Oc3c(C)cccc3Br)CCC(=O)N1c1ccccc1S2 CCCCC(CNC(=O)C(C)N(C(=O)CC1CCCC1O)C)CCC c1(C(=O)NCCC2(O)CN(C(c3cscn3)=O)C2)cnn2c1CCCC2 c1(C(N(C2CCCN(C(C3CC(F)C3)=O)C2)CC)=O)cc(F)ccc1OC c1(C(=O)NCCCC(CCC)NC(=O)C=CC2CC2)ccc2nc(O)oc2c1 C12(NC(=O)NCC3(C)OCCO3)CC3CC(CC1C3)C2 C1(N(C(C2=NOC(C)C2)=O)C)CCCC2CN(C(c3cn[nH]c3)=O)CC12 C(=O)(CC1=NNC(=O)C1)N1C(CC)CC(F)(F)C1.C(C(=O)N)N(CC)CC C1(CC=O)CCCC(C)(C)O1.CC1OC2(C(=O)NCC(C)C3CC3)CC1C2.N C(=O)(C1=C(F)CN(C(=O)C(C)CC#N)CC1)N(C(CCSC)C)C N1(C(CC(C(C)C)O)=O)CC2CCCC(CNC(C3(C)CC3(C)C)=O)C2C1 Cc1cc(C(=O)NC2CC(F)(C)C2)n(C2CCC2)n1.c1(C=O)cccnc1S.N C1(CCC(=O)NCC(CC)NC(c2c(C)cnn2C)=O)CC(C)(C)CO1 c1(OC)ccc(CCC(=O)N(CCCNC(=O)CCc2cccs2)CCO)cc1 C(=O)(C(O)CNC(=O)C(O)Cn1cncn1)NCC(CC)O c1(C(=O)NCC(C)NC(=O)C(C)OC(C)(C)C)ccnc(Cl)c1O c1(C(N(C(CC(F)F)C(=O)N2CCC=C(F)C2)C)=O)cccc2ccoc12 CC1CC=C(C(=O)NC2CC23CC(NC(C2(C)CCCC2)=O)C3)CC1 C(c1nc2ccccc2o1)=CC(N1CCCC(N(C(C(C)=C(CC)C)=O)C)C1)=O C1(N=[N+]=[N-])(C(=O)NC2C(CC)C2)CCN(C(=O)CN2C(=O)CNC2=O)C1 CC1CCC(CCNC(C2CC(NC(=O)C=CCF)C2)=O)O1 C(CS(=O)(=O)CC(=O)NC(C(=O)NCC(C)(F)F)C1CCCC1)OC N1(C(C2(CC)CCNC2=O)=O)CCc2c(ncn2C)C1C C1(C)(C(N(CC)C2CC2)=O)CCC(C)(C)CC1.CC1CCC(C)(C(=O)N)C1 CC1CC(C)(C(=O)NC2CC(NC(c3cn(-c4ncccn4)cn3)=O)C2)C1 c1(C(N(CCC)CCNC(C2CC(C)OC2=O)=O)=O)c(C)nc2ccnn2c1C Cc1nc(Br)ccc1NC(C1CC2CC1CN2C(=O)COCC(C)C)=O C1CCN(C(C2CC3CC2C2CC32)=O)C1(C)C.C(C(=O)N)N(C)C(=O)C1CC1 C1(C)(NC(c2n(C)nnn2)c2cc(Br)cs2)CCCOC1 C1(C(C)C)C(NC(=O)Cc2cc[nH]c2)CCN1C(=O)CC(C)n1ccnc1 C1(C(OCC)OCC)COCCN1C(=O)C(c1ccc(C(C)C)cc1)C N1(C(c2nc(CCC)sc2)=O)CCC(O)(CC)CC1.C12(CC(=O)N)CCCC1C2 C1(c2nccs2)(NCC(c2cccc(F)c2)C)CCOCC1 c1(NC(C)=O)cc(Br)ccc1CN1CCOCC1CC(N1CCCC(F)C1)=O C1(C(=O)NC(C)C(=O)Nc2ccc(-c3cnco3)cc2)CCCN(C(C)(C)C)C1 C1(C(N2CC(NC(=O)C3CC3)C(C(F)(F)F)CC2)=O)CCc2nnc(O)cc2C1 N1(C(CCCC#C)=O)CCN(C(c2cccc(CO)c2)=O)C(C#C)C1 Cn1ncnc1CCC(=O)NCCOCCOCCNC(C1CC1F)=O O=C(C1CCc2c[nH]nc21)NCC1CC(F)CN1C(=O)C1=CCS(=O)(=O)C1 C(C1(O)CCc2ccccc21)N(C1CCC(F)CC1)C c1(C(N2CCC(N(C)C)C2)=O)cc2n(n1)CCC2.C12(CCNC1)N(CCO)C2 N1(C(c2cn(CC(C)O)c(=O)cc2)=O)CCN(C(=O)OC(C)(C)C)C(C)C1C c1(C(C(=O)NC(C)C)N(C)Cc2cc(CCC)nn2C)sc2ccccc2c1Cl C1(C)(CNC(C2(OC)CCC2)=O)CCCN1C(=O)C(C(C)C)c1ccccc1 c1ccc(C)cc1Cl.C(=O)(CC#N)NCC(C1CC1)NC(COC)=O.CC.O N1(C(C(C=C=C)C)=O)CCC(C2(O)CN(C(c3cccc(=S)n3O)=O)C2)CC1 c1(C(=O)NC2C3CN(C(c4cnc(CC)[nH]4)=O)C2C3)cc(OC)cc(F)c1 N1(C(CC2(NC(CCCCSC)=O)CCCCC2)=O)CCn2cncc2C1 C12(NC(C3CCS(=O)(=O)C3)=O)CCC1CN(C(C1(CO)COC1)=O)C2 Cc1sc(CN2CCCC2CCC(=O)NC2CCCCCC2)c(C)c1C C1(C(=O)N)CCC(C)N(C(c2ccc(C(N)=O)s2)=O)C1.C(CC(C)(C)C)OC CCCCCCC(C)(C(=O)O)NCC1(N)CC1(C)C Cc1cc(CNC(c2ccc(F)cc2)C2CCCCC2)c(C)o1 N1(C(Cc2onc(C)n2)=O)CCC(C(=O)Nc2cccc3c2OCC3)CC1(C)C N1(C(C=Cc2ccc(C)s2)=O)CCC2CN(Cc3ccnnc3)CC12 C1(C=O)CNC(=O)CC1(C)C.c1(C(OC)OC)ccc(C=O)o1.C1CCC1.N Cc1ccc(C)c(C(=O)NCC(C)NC(c2cc(N)c(Cl)c(O)c2)=O)c1C N1(C(c2cc(C)nc(O)c2)=O)CCN(C(=O)CCCS(N)(=O)=O)C2CCCC12 N=c1nnn(CC(=O)NCC2(CCNC(=O)Cc3ccccc3)CC2)[nH]1 C1(N(C(C=CSC)=O)CC)CCCN(C(c2cccnc2-n2cncn2)=O)CC1 c1(COC)cc(N2CCCCC2CNC(C2(O)COC2)=O)ncn1 c1(C(N2CC(C)C(NC(=O)CCCC(C)(C)C)C2)=O)cc2c(F)cccc2s1 C(CC(C)(C)CC(=O)NC1CC=C(C(=O)N2CC3C(C(N)=O)C3C2)C1)OC C12CCCC(C1)NC2=O.C(=O)(CN(C)CCO)N(CC)CC N1(C(CCCCCSC)=O)CC(NC(c2cn[nH]c2)=O)CC12CCOCC2 C(=O)(C(C)(C)C1CCN(C(=O)Cc2cncn2C)C1)N(C1C(C)CC1)C C(=O)(C(F)C(=O)N1CCCC(CC)C1)OCC.c1ccc(C)cc1.C(=O)(C)N C#CCCC(C(=O)N(CCS(N)(=O)=O)C)NC(=O)C(N)=O C(=O)(C1=CN=C2N=CNN2C1)N1C(CNC(CCCCOC)=O)CC(F)(F)C1 c1(OC)cc(N)c(C(=O)NC(C)CNC(=O)C(c2ccccc2Cl)C)cc1.O N1(C(CSCC#C)=O)CC(CNC(=O)CSCC)C(c2cncn2C)C1 Cc1ccc(C(C(C)C)NC(C2C3CN(C(=O)CS)CC23)=O)cc1.c1nn[nH]n1 c1(C(N2CC(C)N(C(=O)C=CC3CCCC3)CC2)=O)ccc2[nH][nH]c(=N)c2c1 N1(C(c2cc(OC)n(C)n2)=O)CCOC2CCN(C(=O)C(C)(CC)C(N)=O)CC12 c12ccc3c(cnn3c1)CNC(=O)c1ccc(F)cc1-2.N1(CC)CC(O)C(O)C1 C1(CCC#C)CCCN(C(=O)COC(C)(C)CNC(c2ccccc2C)=O)C1 C1(CNC(CCc2cnc(C)o2)=O)CCCN(C(=O)C(C)O)C1 C(C(C)(C)C(C)C)(c1nnnn1C1CCC1)NCc1cc(C)ncn1 C(CCCC(C)NC(=O)C(O)C1CC1)NC(C1(C=C)CC1)=O N1(C(c2ccc(C)nc2)=O)CCC(NC(C2Cc3nncn3C2)=O)C2(CCC2)C1 N1(C(CC2C(NC(C3(CC)CCCC3O)=O)CCCC2)=O)CCC(C)(C2CC2)C1 C(N=c1cc[nH]cc1S(=O)(=O)NC12CCC(CC1)C2)c1c(C)ccc(Cl)c1 C1(N(C(=O)C(O)COCc2ccccc2)C)CCCCN(C(c2cnn[nH]2)=O)C1 CC(C(=O)N(CC(O)CNC(=O)CC1CSC1)C)SC(F)(F)F.C(C)(C)C C1(C(=O)NCCn2c(CC)ncc2)CN(C(C2CC(N(C)C)C2)=O)CCO1 C1(C(=O)NC2C(CNC(COC3(C)CCC3)=O)C2)CNC(=O)CC1(C)C C1(c2n(CC)cnn2)CN(C(c2ccc(C(F)(F)F)cc2)=O)CCO1 C(C(C(=O)NOCC1CC1)NC(=O)CCc1ccn(C)c1)OCC c1(C(=O)NC2CC(C)N(C(=O)Cc3ccc(N)cc3)C2)cnc(Cl)cc1Cl C1(C(=O)NCC2(NC(C3C(=O)NCC3)=O)CCOCC2)Cc2ccccc2N1 C=CCC(CNC(c1c(C)nn(C)c1N)=O)C(=O)NCC1(C)C=CCCC1 C1(C)CCN(C(=O)CC2(C=C)CCC2)CC1.c1(C)ccc(C)s1.C(=O)C=O CC(C)C(C)C(=O)NC1CN(C(C2(C)CCC(=O)C2)=O)CC1CO CC(C)CC(O)C(=O)NCC(c1ccc(F)c(F)c1)N1CCOCC1 C12(C(N3CC(C)C(CNC(=O)C4=CCCOC4)C3)=O)CCC(CC1)C2(C)C c1(OCC)cc(NC(CNC(=O)Cc2c(C)noc2Cl)C(C)C)ncn1 C1(CN2CCCCC2)C2CCC(C2)N1C(=O)C=C(C)S(C)(=O)=O.CC=O c1(OC)ncnc(C(=O)NCC(C(C)(C)C)NC(C2CCCCN2C)=O)c1F N1(C(C(CC)N(CC)CC)=O)CCN(C(c2ccccn2)=O)CC(O)C1 C1(NC(CCOC(C)=O)=O)COCC1NC(=O)COC(F)F C(=O)(C(C)(C)C(=O)N1CCC(CNC(=O)C2=C(Cl)CCC2)C(O)C1)NC CC(CCCCN=c1cc(Cl)c(O)n[nH]1)NC(=O)C(N1CCOCC1)C N1(C(CC2CC(C)OC2C)=O)CCC2(CC1)CCN(C(=O)CCc1cc[nH]n1)C2 C12(CNC(CC3N(C)CCCC3)=O)CN(C(c3ccc(Cl)cc3)=O)CC(F)(C1)C2 N1(C(C2C(CC)CN(C(=O)CSC)C2)=O)CCN(C)CC(C)C1 N1(CCNC(C)=O)CCC(NC(c2cnn(-c3ccc(C)cc3)c2C)=O)CC1 C(=O)(CC(O)CCCC)NC1(C(N(CC(=C)C)CC(=C)C)=O)COC1 c1(C(=O)OCCCC(=O)N2CC(C(=O)Nc3ccccc3)C2)snc(Cl)c1Cl c1(C(=O)NCCN(CCC)C(c2nnsc2C(F)F)=O)ccc(CC)[nH]1 C1(NC(C2C=CC(C)(C)CC2)=O)CCC2CN(C(=O)OC(C)(C)C)CCC2C1 CC1(C)CC(C(=O)NCC2CCCN2C(C2(C)CC=CC2)=O)CCO1 CC1(CNC(C2CCN(C3COC3)C2)=O)CN(C(=O)C2=CCCSC2)CCO1 C(C)(CNC(c1ccnc(OC)n1)=O)(C(C)C)NC(CCCOCC=C)=O C1(C)(C(=O)NCCCSC)CCCN1C(C1CCSC1)=O CCCC(C#N)C(=O)NC1(CCc2c(C)cccc2C)CCCSC1 CC1C(NC(c2ccn(C(C)(C)C)n2)=O)CC2CCC1N2C(=O)CC1CCCC1 c1(C(=O)NC2(C)CCN(C(CCOCCN(C)C)=O)C2)ccc(N)c(O)c1 CCCC(CC)CCC(=O)NC1CC2CC(C1)N(C(=O)CCCN(C)C)C2 C1(C(N2CCC(C(C)O)CC2)=O)CCN(C(c2cc(O)nc(O)n2)=O)CCO1 C1(C(N2CCC(C)(NC(CCC3(C)CC3)=O)C2)=O)CCC2CCCCC2C1 C(=O)(C(C)CC(C)(F)F)NC1CCN(C(Cc2cc(C)no2)=O)CC1CO Cc1coc(C=CC(=O)N(C)CC2CCCN2C(c2oncc2C)=O)n1 C1(N(C(C(C)N(C(c2c(C)nns2)=O)C)=O)C)CCOC(C)(C)C1 CC(C)C(C)CC(=O)NCC(C)(O)CNC(=O)CC(C)C.c1(C=O)ccco1 N1(CC)CC(C(N2CCSCC2CCNC(=O)C(C)CF)=O)CC1=O Cc1nc(C(=O)N(CC(=O)NC(C)Cn2cnnc2)C2CCC2)ccc1C#N n1(CC(=O)NCC2N(C(C(CC)N(C)C)=O)CCSC2)ncc(O)nc1=O N1(C(CN(C(c2cc(C#N)n(C)n2)=O)CC)=O)CCC2(CNC(=O)O2)C1 CC1(C)COC(C(=O)NCC2CC(C(N3CCC(c4ccon4)C3)=O)CO2)C1 C12(C(=O)N)CC1COC2(C)C.c1(C(=O)NCC(C)C)cc(C(F)(F)F)ns1 c1(C(N2CC=CC(NC(C(C)OC)=O)C2)=O)ccc2c(c1)CCC2(F)F C1(C#N)(C(N2CCN(C(c3cc(C(C)C)no3)=O)CC2)=O)CCS(=O)(=O)CC1 C12(CNC(c3cc(CC)[nH]n3)=O)CC(CO1)C2.C(=O)CCC.C(N)=O.N C(=O)(C(C#N)(CC)CC)NC(CNC(c1cc(CCC)[nH]n1)=O)C c1(CCS(=O)(=O)NC(=O)CN2CC(NSC(F)(F)F)C2)c(F)cccc1Cl N1(C(C2(C#N)CC(C)C2)=O)CCCC(N(C)C(C2CN3CCC2CC3)=O)CC1 N1(C(c2cc(C)no2)=O)CCN(C(C2CCCN2C=O)=O)CC1c1ccnn1C c1(C(=O)NC2CCC(C)(CNC(C(C)O)=O)CC2)ccc2sccc2c1 c1(C(N2C(CNC(=O)CC(O)C3CC3)CC3(CC3)C2)=O)cnc(O)c2ccsc12 C1(CC(=O)N(CCNC(=O)C(F)=C2CCC2)C2CC2)CCCOC1 C1(NC(c2ccc(N(C)C)cn2)=O)CCCCCC1.C1(C=O)CCCN1C(N)=O.N Cc1cc(N)c(C(=O)NC2CCC2NC(=O)CN2Cc3ccccc3C2)cc1C Cc1nc(C(=O)NC2CCN(C(c3cnc(S)n3C)=O)CC2C)ccc1[N+](=O)[O-] c1(C(N2C3C(CNC(CN(C(C)=O)C)=O)C(C3)C2)=O)n[nH]c2ccc(Br)cc12 c1(C(N2CCC(Sc3cccc(Cl)c3)CC2)=O)onc2c1CCCC2 c1(OC)cccc(CC(=O)NC2CC(NC(=O)CO)C(O)C2)c1.C1CCC1 c1(C(=O)NC(C)CN(C(=O)CCc2nncn2C)C)cc2cccnc2cc1F c1(C(C)C(=O)NC2(C)CN(C(=O)CSc3cccc(F)c3)C2)c(F)cccc1F c1(C(C)NC(=O)CC2CN(C(=O)CN)CCO2)cc(F)cc(Cl)c1 N1(C(COC)=O)CC2CC1(C)C2.c1(C=O)ccc(-c2nc(C(C)C)no2)cc1.N CCCC(C(=O)N1CC(CNC(=O)CCCc2cccnc2)C2(CC2)C1)C(C)C C(=O)(CC(F)(F)Br)N1C(C)(c2cn(C3(C(=O)O)CC3)nn2)CC1 c1(C(=O)NC2CC(C(=O)NC(C3CCOC3)C)C2)cc[n+]([O-])cc1 c1(CNC(CN(C)CC)=O)ccc(C(=O)N)cc1.c1cncn1C1CC1.C CC(CC(=O)NC1CC(F)CN(C(=O)C(O)C2CCC2)C1)C(C)(C)C C1(CNC(COCCC(C)C)=O)CC(O)(CO)C1.c1(C=O)cccnc1 C(CN=[N+]=[N-])(C(=O)NC1CCC1)NC(Cn1c(C)nnn1)=O.c1(C)ccco1.S C1(C(N2CCCC(n3cc(CSC)nn3)C2)=O)CS(=O)(=O)CC12CCNCC2 c1(C(=O)NC2C3CN(C(c4c(C)cccn4)=O)C2CC3)n[nH]c2c1COCC2 c1(SCC2CCC(C(=O)O)CC2)ccc(OC(F)F)c(O)c1 c1(C(CN)=O)ccc(OC)cc1F.C(CC)(C1CC1)OC c1(C(N2C(CN(C(CCCCC)=O)C)CCC2)=O)cc(OC)cc(Br)c1 c1(C(=O)NC(C2CN(C(CN(CCOC)C)=O)C2)C)cc(Cl)c[nH]1 C12(CNC(c3cc(F)cc(Cl)c3)=O)CN(C(c3csnn3)=O)CC1CCO2 c1(OCC)ccc(C(=O)NCC2(C)CCCN2C(=O)C(OC)O)cc1F c1(C(N(C2CCNCCC2C)C(C)C2CC2)=O)cnc2ccccc2n1 c1(C(N2CCC(OC)(C)C2)=O)cc(C)c(N)cc1F.c1(C(=O)N)ccc(O)nn1 c1(CC(=O)N(C)CC2(NC(c3c(C)nsc3)=O)CC2)ccc(F)cc1 CC1(NC(C2C3CC2N(C(c2cc(=O)cc[nH]2)=O)C3)=O)CCCCC1C(=O)O N1(C(C(=O)NC(CN(C(C2CCCC2O)=O)CC)C)C)CCOCC1 C=CCCC(CC(C)C)C(=O)NC1CN(C(=O)Cn2nc(C)nc2C)C(C)(C)C1 c1(C=O)cc(S(=O)(=O)N2CCCC2)c(C)s1.c12cnccc1N2CC(F)F.CO C1(C)(CNC(C(COC)NC(C)=O)=O)CCN(C(c2cnco2)=O)C1 C1(COC)CCN(C(c2ccon2)=O)C12CCC2.C1(C(=O)N)CC1.C1CC1 CCCC(C)(O)CC(=O)NC1CCC(C(=O)NCC2OC(=O)CC2(C)C)C1 N1(C(c2c(CC)scc2)=O)CC2CC(CNC(c3cc(N)nc(Cl)c3)=O)C2C1 N1(C(C2CC(=C)C2)=O)CC2CN(C(c3cccn(C)c3=O)=O)CC2C1 Cc1ccc(C#N)c(NC2CCCCN(C(C3CCCOC3C)=O)C2)n1 Cc1cc(C(F)(F)F)nc(N2CCN(C(c3c(C)nn(C(C)C)c3C)=O)CC2)n1 N#Cc1nc(=NC(c2ccccn2)C2CCCCC2)cc[nH]1 C=CC1OCCC1C(=O)N(C(CNC(=O)C(=Cc1ccccc1)OC)C1CC1)C Cc1ncc(CC(=O)N)c(O)n1.c1(CC(=O)N(C(C)C2CC2)C)cccc(F)c1 c1(N2CCC(C)C(NC(C3C4COCC34)=O)C2)c([N+](=O)[O-])cccc1[N+](=O)[O-] C1(C)(CC=C)CN(C(=O)C(CC2CCC2)NC(=O)C(N2CCCCC2)C)C1 c1(C(=O)OC2CC(OCCCC)C2(C)C)c(F)cnc(Br)c1C N1(C(C=COCC)=O)CC2CC1CN(C(C1CCC(CC)CC1)=O)C2 c1(C(=O)NC2C(OC)CN(C(c3ccc(C)cn3)=O)C2)cc2c(C)nn(C)c2s1 c1(OC(C)C)ccccc1CC(=O)Nc1ccc(CC(=O)O)cc1 CC(CCCCNC(=O)C=C1CCC1)NC(C1CC1c1ccccn1)=O C1(OC)CC(C(=O)NC2(n3cccn3)CC2)N(C(=O)CCC2CCCC2)C1 c1(C(C)C)cccc(NC(c2csc(C(N3C(C)CCC3C)=O)n2)=O)c1Cl O=C1CCN(Cc2ccc(F)cc2)C(=O)N1CCCCCC1CCCC1 CN1CCCC(C(N2CCC(C)(CNC(C3CC3c3ccccc3)=O)C2)=O)C1 C1CC(S(C)(=O)=O)CN1C(=O)NC1CC1.c1cc2ccccc2o1.CC(=O)N N1(C(c2ncc(Cl)cc2Cl)=O)CCN(C(C2CC2F)=O)CC(O)C1 C(C(C)(C)C(=O)N(CCC(C)NC(=O)Cn1cccc1)C)OCC C(=O)(CCCCCCNC(C1C(C)(C)C1(F)F)=O)N(c1ccc(F)cc1)CC C1(NC(c2c(C)n3c(s2)cnc3)=O)CN(C(=O)C2=CCC2)CCC12CCOCC2 N1(C(c2ccn(C)n2)=O)CC2CCCC1C2CNC(=O)C(F)(F)c1cccnc1 Cc1nn(C)nc1C(=O)NC(C1CCOC1)CNC(C1(C)CCCCC1)=O C1(C(C)(C)C)CCCN1C(=O)C=CC=O.C(C)(C(=O)N)=C(C)C.C1CC1 C1(C(=O)NC2CCC(CCC(=O)Nc3c(C)scc3)C2)CCC(C)(C)CC1 c1c(C)nn(C)c1C.C1(CC(=O)NCCCC=C)CCCC(=O)N1.C(=O)(C)N C(=O)(C(C)(CNC(c1nscc1C)=O)CC)N(C(CSC)C)C C12(C(=O)NC3CC(CNC(c4nc(CC)oc4)=O)C3)CCN(CC1)C2 N1(CCNC(CC2CC(=O)NC2)=O)CCCN(C(=O)CC2CCCOC2)CC1 C1(C)(C(N2CC(C(C(NOCCC#C)=O)O)C2)=O)CC(=O)N(C)C1 N1(C(c2c(C)c3c([nH]2)c(C)ccc3)=O)CCCC12CCCN(C(=O)CC(C)F)C2 C1(CC)CCOCCN1C(=O)CCN(C)C(C1(C)CC=CCC1)=O c1(NCC(C(C)C)NC(c2cnn(CC3CC3)c2)=O)ncc(Br)cc1[N+](=O)[O-] C(=O)(CCCC(C)(C)CC)N(CC(C)(C)NC(c1ccc(=NCC)[nH]c1)=O)C C12(NC(c3ccc(CCC)s3)=O)CC(C1)N(C(c1sncc1CC)=O)C2 c1(C(=O)NCC(C)(CNC(c2cnns2)=O)OC)cccc(C)n1 CC(C)CCC(CO)NC(=O)CCN1CCN(c2cnsn2)CC1 CCCCC(C)CCC(=O)NC12CCC(CN(C(c3cnn(C)c3F)=O)C1)C2 C1(C(=O)NC23CC(CNC(c4c(C)[nH]cc4)=O)(C2)C3)CC2CCCCN2C1 CC1(C)OC(C(N2CCC2C)=O)C(C)(C)O1.C1(C)(C(=O)N)CC(C)(C)C1 C1(NC(C2C(=C)CC2)=O)COCCN(C(=O)C(CCCC)N(C)C)C1 CS(=O)(=O)CC(=O)NC(CNC(=O)CCc1cn[nH]c1)CO C(=O)CS(=O)(=O)CCO.c1(CC)nc[nH]c1C(=O)NCC12CC(C1)C2.N CCC(C)C(C)C(=O)N(CC(C)(C)CNC(C1C(C)(C)C1(C)C)=O)CC C12(CCNC(c3cc(OC)ns3)=O)CCC(CC1)C2.c1(CC=O)cncnc1 C1(C(n2cc(COCCC#N)nn2)C)CCCCN1C(=O)CC1CCCO1 N1(C(c2c(CC)csc2)=O)CCCC(N(C(=O)C(C)c2ccsc2)C)CC1 CC(C)(C)CC(=O)N1CCC(C(=O)NCCC2CC2)(CO)C1 c1(N2C(C(N3C(c4scc(C(=O)OC)n4)CCC3)=O)CC2)ncnc2c1cnn2C C1(C(N(C)Cc2ccsc2)=O)CC(=O)CN1C(C1OCCC1(C)C)=O c1(OC)ccc(Br)c(CN2CC(O)(CNC(=O)Cc3ccccc3)C2)n1.O N1(C(c2ccc(C(F)F)o2)C(=O)NC2CCCC2)CC(CO)C(S)C1.C1CC1 C(=O)(CCCCCS(N)(=O)=O)NC(CN(C(C1CCCCN1C)=O)CC)C N1(C(C2CCC(C)C2)=O)CC(NC(C2CCC(=O)NC2)=O)CC12CCOCC2 c1(OCC)nccc(C(N2CC(O)(C)C2)=O)c1F.C(=O)(C(F)(F)C(C)O)N C(=O)(CC1=CCN(C)CC1)NCCCCCC(=O)Nc1c(SC)cccc1 c1(C(=O)NC2CCN(C(C3N(C)C(=O)NC3)=O)C2)cc2cc(F)ccc2[nH]1 C(=O)(C(F)C(F)(F)F)NC1CCN(C(C=CC(=O)OCCCC)=O)C1 C(=O)(CC(C)(C)NC(c1cc(O)cs1)=O)NCCc1cn(CC)nn1 C(CC(C)CCNC(c1ccoc1Br)=O)NC(CN(C(C)=O)C)=O CC1(C)CCCC(CN=c2[nH]c(C(=O)C3CC3)ns2)O1 c1(NCc2n[nH]c(C)c2C)nccc(=NC(C)Cc2cnccn2)[nH]1 c1(OC)cccc2c(C(=O)NCC(CO)NC(c3cnc(N)cn3)=O)c(C)[nH]c12 CC1Nc2cc(C(=O)NC(CF)C(C)(C)C(=O)O)ccc2NC1=O c1(CC=CC(=O)NOC2COCC2O)c(F)cccc1F c1(C(N2CC(CCO)(NC(C3CC(CCC)C3)=O)C2)=O)ccc(F)cc1F C12(CNC(C(C(C)(F)F)F)=O)CCCC1CCN2C(c1ccc2c(c1)CC2)=O c1(NC(C2N(C(c3cccn(C)c3=O)=O)CC(F)C2)=O)cnn2ccc(Cl)nc12 N1(CCN(C(=O)C(F)=C2CCC2)C)CCN(C(c2cncnc2CCC)=O)CC1 c1(C(N2CC(C)N(C(C3CC34CCCC4)=O)CC2)=O)cc(N)c(Cl)c(O)n1 CC1C(NC(=O)CC(C(F)F)NC(=O)CN2CCCCCC2)C2CCN1CC2 CN=c1[nH]cc(CN=c2cc(C(C)(C)C)nc(Cl)[nH]2)cc1C#N c1(CC(=O)NC2CN(C(=O)C(F)CC3CCCC3)C2)cccc2c1OCO2 C1(CNC(C(CC)O)=O)C2CC1N(C(C1(OC(C)=O)CCCCC1)=O)C2 C(=O)(C(F)CCC(C)C)NCC1C(NC(c2c(C)c(F)ccc2)=O)C1 c1(OC)cccc(CCC(=O)NCC23CC2CN(C(C2(C)CC2C)=O)C3)c1F N1(C(CN(C)C2CC2)=O)C2CCC1C(NC(=O)C(C)(C)c1cccs1)C2 C#Cc1cccc(C(=O)N(CC(=O)N(CCC)CC)CC)c1C.OC(F)F N1(C(=O)C=CC2CCCC2)CCC2(C1)CN(C(C1CCO1)=O)C2 CC(C(=O)N(C1CCCN(C(c2nnn(C)n2)=O)C1)CCO)C(F)F C=CC(CC)CC(=O)NC(C)CCNC(C12CCC(C(F)F)(CC1)C2)=O c1(NC(C2C3CC2N(C(c2c(I)ccnc2F)=O)C3)=O)cc(Cl)c(F)c(Cl)c1 C1(C(=O)NC2C=CC(CNC(c3cccc(C)c3)=O)C2)CN2CCN1CC2C c1(CN2CC3C(NC(c4ccc(OC)c(F)c4)=O)C3C2)cc(Br)cc(Cl)c1O c1(NCC(CNC(C(C)CN(C)C)=O)C)cc(C2CC2)ncn1 c1(C(=O)NC(C2CCN(C(C3C(C)(C)C3)=O)C2)(C)C)cc(C2CC2)ccn1 c1(N2CC(c3c(CNC(CC(CC)C)=O)nco3)C2)ncnc2c1cnn2C Cc1cc(=O)n(C)nc1C(=O)NC1CC(NC(C2CC(F)C2)=O)C12CCC2 N1(C(C(CC)O)=O)CCCN(C(=O)C(F)C2CC2)CC1 C1(C)(C(=O)NC2CCC(NC(C3CCC(C)CC3)=O)CC2)COCC1(F)F Cc1cc(C(=O)NCCCNC(C2CCCC(OC(F)(F)F)C2)=O)nc(C)n1 C1(CNC(CN(C(=O)CCC2(O)CCC2)CCC)=O)CCC=CO1 C1(C(=O)Nc2c(C)nc[nH]2)CN(S(=O)(=O)Cc2ccc(C#N)cc2)CCC1O c1(N(C(C)CNC(=O)CO)C)ncnc(O)c1Br c1(C(N(CC(C)O)CC)=O)ccnn1CC.CCS(=O)(=O)NCC(=O)N N1(C(C#C)C)CCCN(C(c2ccc(F)c(Br)c2)C(=O)NCCCOCC)CC1 N1(C(Cc2ccc(OC)cc2)=O)CCN(C(c2cnn(C)c2)=O)C(C(F)F)C1 C(C(F)(F)CCC(=O)NC1(C)CC(F)(F)C1)n1cc(C2(OC)CCCCC2)nn1 c1(CC)ccc(F)c(C(=O)NC2CCCCC2)c1.C1(C)(C=O)CCN(C)C1=O.N N1(C(CC(C)F)=O)CCCC2(CCN(C(c3cnc(N)cn3)=O)C2)C1 CC1(C(=O)NCCN2CCNC2=O)CCCN1C(=O)CC1CC=CC1 c1(C(=O)NC(CN(C(c2coc(C(C)OC)n2)=O)CC)C)cccc(N)c1C c1(C(=O)NC2(CNC(CC)=O)COC2)cc(N)cc(C)c1F C1(CC(=O)N(C(C)C)C)CCC1.n1(CC=O)cccc1.C(=O)(OCC)N c1(C(=O)NC2CC(C)CN(C(c3ccnc(Cl)c3O)=O)C2)nccc2cc[nH]c12 n1(C(C(=O)N(CCCNC(CCCCC=C)=O)CC)C)c(=O)oc2ccccc12 Cc1cccc(CNC(C2(NC(C3C=CCS3)=O)CCCCC2)=O)c1O N1(C(CCNC(=O)NC)=O)CCCC1C(N1CC(O)(COC)C1)=O N1(C(C2CC=C(C)CC2)=O)CCCC(NC(=O)C=CC(C)(C)C)CC1 C(=O)C(C)C(=O)N1CC(O)(CC)C1.c1(C=O)cccnc1.[SH](C)(=O)=O.CO C1(C(C)NC(=O)CSCc2ccncc2)CN(C(c2nncs2)=O)CCO1 C1(C(=O)NCC(C#C)CC)C2CCC1(C1CCN(C(=O)O)CC1)C2.C(C)(C)C c1(C(=O)NC(C(C)NC(=O)CC2(C)CCCCC2)CO)cnc(O)n(C)c1=O c1(C(C)C)[nH]nc(C(=O)NC2CC(F)C2)c1[N+](=O)[O-].C(=O)C=CC1CC1.C N1(C(CC2C=CC(NC(c3cc(OC)ncc3)=O)C2)=O)CC(C2=NOCC2)C1 c1(N2C(CCNC(c3cnn4c3CCC4)=O)CCCC2)nc2ccc(Br)cc2o1 CCCC(CC(C)C)C(=O)NC1CN(C(C23CCC(C2)C3)=O)C2(CCCC2)C1 C1(C2(O)CN(C(=O)Cc3cc[nH]n3)C2)CC1.Cn1cccc1C=CC(=O)NC C1(NC(c2c(OC)n[nH]c2)=O)CC2CCC1CN2C(C1CCCC(F)(F)C1)=O CCC(C)(CN=c1[nH]c2c(c(=NC3CC3C(C)C)[nH]1)SCC2)c1cnccn1 c1(CCC)ccc(Cc2ccc(OC(C3CCN(C)C3)=O)cc2)cc1 c1(C(N2C(CN(C(CC3C(C)C3)=O)C)CCC2)=O)c(Br)c2ccccc2n1C N1(C(CC(C)C2CC2)=O)CCC(NC(=O)C(c2ccc(Cl)cc2)(C)C)C(C)(C)C1 c1(NC(C2C(NC(=O)CC3CCC3)CCC2)=O)ccc2nc[nH]c2c1 C1(NC(CC(CCCCC)O)=O)CCC2(CCCN2C(=O)Cc2cscn2)CC1 N1(C(CC(CCC)O)=O)CCN(C(=O)CCCOC(C)C)CC2(CC2)C1 C(c1cn(C)nn1)=CC(NOCC(N1CCC(COCC)C1)=O)=O C1N=C2NC=NC(=C2C)NC12CCSCC2.c1(COC)ccnn1C(C)(C)C c1(C(=O)NC(C)CNC(C2CC(C)CO2)=O)ncc2c(F)cccn12 c1(N(C)CC2CCCN(C(=O)C=CCF)C2)nc2cc(Cl)ccc2s1 c1(CC)cc(CC(=O)NCC(C)CN(C(=O)C=CCO)C)n(C)n1 c1(C(=O)NC2(CC=C)CCN(C(c3coc(CC)n3)=O)C2)cnc2n1CCCC2 N1(C(c2cc(CC)on2)=O)CC(=O)NCC1C(=O)NC(COC)CO C1(C(=O)NC2C(C)CN(C(C3(c4cccs4)CC3)=O)C2)CCc2ccc(F)cc2O1 N1(C(C(C)OCC2CC2)=O)CC(NC(=O)C=C2CCCCC2)CC(F)C1 CC1=C(C(=O)N(C2CCN(C(=O)CCC3CC3)C2)CCO)S(=O)(=O)CCO1 N1(C(c2onc(COC)n2)=O)CC(NC(C2(C)CCCOC2)=O)CCC1C c1(C(=O)N)ccc(C(F)(F)F)c(N)c1.C12(C(N(CCC)C)=O)CC(C)C1C2 CN1C2CCC1CC(C(=O)Nc1ccc(=O)n(-c3ccc(I)cc3)c1)C2 c1(OC)cc(C(=O)NC2CC(O)(CNC(=O)C(C)C(C)C)C2)ccc1O N1(C(CN(C)CC2CC2)=O)CCN(C(=O)COC2CCOCC2)CC1CF c1(SC(c2nnnn2C)C(C)OCC2CN(CCC)C2)ccccc1 c1(C(N2C(CC)CCC2)=O)ccc2c(c1)C(=O)CCC2.C(C=C(Cl)Cl)=CC=O.N N1(C(C2CN(C(C)C)C2)=O)CCN2CCN(C(c3cc(C#N)oc3C)=O)CC2C1 N1(C(c2c(C)cc[nH]2)=O)CCC(O)(C(C)CNC(C2(C)CCC2)=O)C1 c1(NC2CCC(N(C(=O)C3=CCCCC3)C)C2)ncc(Cl)c(O)n1 N1(C(=O)CC2COC(=O)C2)CCC2CCCC12C(=O)NC1CCC2(CCC2)C1 C(C1C(C)C1(Cl)Cl)=CC(=O)N(CCCCN(C(C1CC1)=O)C)C.COC c1(C(N2CCN(c3nccc(C)c3)CC2)=O)cc(I)cc2ccccc12 CC(C(=O)NC(C)CCC(=O)Nc1ccccc1O)C(F)F C(=O)(CC(C)(C)C1CCCCC1)NCC1C(NC(C2(N(C)C)CC2)=O)C1 c1(C(=O)NC(CCCNC(C(CC#C)C2CC2)=O)CCC)cc(F)c(N)cc1OC C(C)(C)C(O)C(F)F.Cc1cc(CNC(c2cc(O)ncn2)=O)oc1C=O.N N1(C(c2n(CCC)ncc2)=O)CCOC(C(C)NC(=O)Cc2cccnc2Cl)C1 C1(N=[N+]=[N-])(C(=O)NCCCCCCCC)CCN(C(c2coc(CO)c2)=O)C1 C1(NC(=O)CCc2cnc(O)[nH]2)CCCN(C(C2CC3C=CC2O3)=O)C1 C1(C(N2CC(O)(C(C)NC(=O)CCC=O)C2)=O)CCC(F)(F)C1.C1CCCC1 CC(C)S(C)(=O)=O.c1(OC)noc(C)c1C=O.C1(CC=O)CC(=O)C1.N CC1CC2(CO1)CN(C(C1C(C)CCN1C(=O)C=Cc1cocn1)=O)C2 C(=O)(C1=CCN(C(=O)CCCCC=CC)CC1)N(CC=C)CCC Cc1ccc(CC(N2CCC(NC(=O)CCc3nccn3C)CC2)=O)cc1C C(=O)(C(C)C(C)(C)C)Nc1cc(OC)c(C)cc1.C(=O)C(O)Cn1cncn1.N C(=O)(C(CNC(C1(CO)COC1)=O)C(C)(C)C)NC(c1nc[nH]n1)C c1(NC(CC(C)C)=O)ccc2c(c1)CN(C(c1cccc(F)c1Br)=O)CC2 S(=O)(=O)(c1c[nH]ccc1=NC(CN(C)C)CO)NCC(C1CC1)OC c1(NC(C2CC3CC3N2C(c2ncc[nH]2)=O)=O)cnc2c(c1)CCCC2 c1(OC)cccc2c1nc(NC(=O)Nc1cnn(C3CCS(=O)(=O)C3)c1)n2C C1(NCC(CNC(CNC(c2c(C)occ2)=O)=O)C)CCC2(CCC2)C1 C1(F)(C(N(CC(CC2CC2)CO)C)=O)CCN(C(c2ncccc2N)=O)CC1 C(CCCNC(C1(CNC(=O)Cc2cnsc2)CC1)=O)C1C(C)C1.CC c1(N2CC(C(C)NC(C3CCN(CC#C)CC3)=O)OCC2)ccnc2ncnn12 c1(C(=O)NCC(C2CCOC2)NC(CCCOC)=O)ccc2c(c1)CCCO2 N1(C(COCC=C)=O)CCCC(C2CCN(C(=O)Cc3cc(C)no3)CC2)C1 Cc1ncc(Cl)c(C(=O)NCC(C(C)C)NC(c2ccc(CC(C)C)cc2)=O)n1 c1(CC)cc(OC)cc(C(=O)NCCNC(=O)Cn2cc(F)ccc2=O)c1 c1(C(=O)N)cnn(C(C)(C)C)c1Cl.Cc1csc(CC(=O)NCC2CCC2)n1 C1(C(NOCCOCC#C)=O)CCN(C(=O)C2(CC3CCC3)CC2)O1 CN1CCC(F)(C(N2CC(NC(C3(C#N)CC3)=O)CC(O)C2)=O)CC1 c1(NC(=O)CCNC(=O)C(=O)Nc2cccc(Br)c2)ccc2nc(O)sc2c1 c1(OC)ccc(CC(=O)NC(C)(C)CO)cc1.c1(C=O)ccn(CC(C)C)n1.N Cc1ccc(C(=O)C2CC2)cc1OC(F)F.C1CCCC1.C1(C=O)CC1.NC N1(C(COC)=O)CCC(F)C(C(=O)NC2CCN(C3CCN(C)CC3)CC2)C1 c1(C(c2nnnn2C)NC(c2c(OC)cccc2)C(C)C)ccc(F)cc1F c1(C(=O)NCC(CNC(CCC(C)(C)F)=O)C(F)(F)F)ccc2ocnc2n1 c1(COC(c2ccnc(Oc3ccccc3F)c2)=O)nc2ccncc2[nH]1 C1(OCC(=O)NC2C(C)C2C)CCN(C(C2(C)CCCC2)=O)C1 C12(C(=O)NCC3N(C(c4c(CC)cccc4)=O)CC3)CCC(C)(CC1)CC2 C1(OC(C2CCC(C(N(C(=O)CC(C)C)CCC)=O)C2)=O)CCCC(C)C1 c1(OC)ccc(C(=O)NC2CC(C)(NC(=O)C(C)CC(N)=O)C2)cc1Cl CCC(CCC(=O)NOCC(F)F)NC(C1CCC1(F)F)=O C(C(C)S(C)(=O)=O)NC(CC1(CSC)CC1)=O.C1CCCOC1.C(=O)C N1(C(C(CCSC)O)=O)CC=C(C(=O)N2CCC(C)(C(N)=O)C2)CC1 C1(NC(C2N(CC)CCC2)=O)CCCCN(C(c2sccc2C(C)(C)C)=O)CC1 c1(C(=O)NC(CNC(C(C)SCC)=O)CC)csc(-c2ccncc2)n1 CCCC(C)(C)CC(=O)NC1(C)CN(C(c2cnn(C(C)C)c2F)=O)C1 CCC(C(=O)N(CC(C)N(C(=O)CCc1nccn1CC)C)C)N(C)C C(=O)(C1=Cc2ccccc2C1C)N1CC(O)C(O)C1.C(C(C)=CC(=O)NC)OC C(C)(C)(CC(=O)NCCC1(O)CCN(C(=O)C(c2ccc(O)cc2)=O)C1)SC c1(C(N2CC(CNC(c3cnc4ccsc4c3)=O)C2)=O)cnc2ccnn2c1O N1(C(CCCOCC=C)=O)CC2CC1CCC2NC(c1cscc1F)=O CC1CCC(C)N(C(C2CC3(CSC3)C2)=O)C1.c1(C(=O)N)cc(C(F)F)nn1C c1(CNC(c2coc(-c3ccc(F)cc3)n2)C)cc(F)cc(C#N)c1 C(=O)(C(C)C(C)(C)c1ccccc1)NC(C)C(c1ccccc1)=O C1(O)(CN(C(c2c(SCC)cccn2)=O)C)CCN(C(C2CC2C)=O)CC1 C1(NC(c2occ(C)c2)=O)C2CC3CN(C(c4cc(Br)no4)=O)C1C3C2 N1(C(C2(COC)CC=CC2)=O)CC2CC(NC(c3nc(C)ccc3O)=O)CC1C2 N1(C(C(NOC)=O)=O)CCCC(C)(c2ccccc2)C1 C1(C(=O)NCC2(O)CCSC2)(CC)CN(C(=O)CC=O)C1.C(C)(C)C.O c1(C(N2C(C(N(C(C)C)C)=O)CCC2)=O)ccc2c(c1)CCO2 Cc1ccc(C)n1CCC(=O)NC1(CNC(C2(F)CCCOC2)=O)CCOC1 N1(C(c2cc(C)nnc2)=O)CCC(F)(CNC(=O)CC2CCC2C)CC1 c1(CC)cc(C(N2CCC(c3cccc(Cl)c3)CC2)C(=O)NCC(C)C)n(C)n1 C1(C(N2CCC23CC3)=O)CC2CCCC(C1)C2=O.c1ncccc1CC=O.CO C1CC2(C1)CN(C(C1CC1c1ccccc1C)=O)C2.CCCC(C)=CC(=O)NC c1(C(N(C(CNC(C(=COCC)C#N)=O)C2CC2)C)=O)ncnc2sccc12 c1(C(C)=O)ccc(N=c2scc(-c3cnn(C)c3)n2CC(C)C(C)C)cc1F C1(CC=C)(C(=O)N(C2CCN(CC)C2)C)CCN(C(=O)Cc2csc(C)c2)C1 c1(C(=O)NCCN(CC(CC)C)CC)cc(C)nc(C)c1 c1(CCCCC(=O)N)nc2ccccc2s1.CN1CC(C(=O)NCC=CC)NC1=O C1(NC(=O)Cc2cccs2)CC(F)CN(C(=O)CCn2cnnn2)C1 C1CCN(C(=O)C)C12CC2.C#CC1(C(=O)NC)CCC1.C1CN(C(C)=O)C1 C1(C(=O)NCCC(=O)N(C)C)CC=CC(n2cc(C(C)(C)C(N)=O)nn2)C1 N1(C(C(C)S(C)(=O)=O)=O)CCC2CCCC12C(=O)NC(C(O)CO)C1CC1 c1(N(C)C)cnc(NC(=O)NCCC2(C)CCOCC2)nc1C(F)(F)F CC1CC(NC(=O)C(C)C(F)(F)F)CCN1C(c1cccc(Cl)c1N)=O c1(SC)cccc(F)c1C=O.C(=O)(C1=CC(C)(C)C1)N1CCC(C)(CC)C1.N C1(C(=O)OCC)CCN(C(C2(N(C(=O)C(C)(F)F)C)CC2)=O)C1 c1(C(N2CC3C(CNC(C(N)=O)=O)(C3)C2)=O)cc(Br)ccc1OC(F)(F)F S(=O)(=O)(c1cc(F)cc(F)c1)N1C2CCN(C(CCN(C)C)=O)CC2CC1 c1(C(=O)NCCCCNC(c2cncc(OCC)c2)=O)cc(C)c2[nH]nnc2c1 C(=O)(CCC(C)(C)OC)N(C1CCN(C(=O)Cc2ccc(F)cc2Cl)C1)CC c1(C(N(C2CCN(C(c3cc(F)n(C)n3)=O)C2)C)=O)csc(Cl)c1Cl C(=O)(C(C)CCCC(C)C)NCc1c(NC(c2c(C)cnn2C)=O)nccc1 N1(C(c2c(C(C)(F)F)n[nH]c2)=O)CC2CCC1C1CN(C(=O)COC3CC3)CC21 CCCC(C)(CCC)C(=O)N1CC(NC(C2CCC2C#N)=O)C2(CC2)C1 N1(C(=O)C2CC2)CCCC(C2CCN(c3nc(C4CCCCC4)ns3)C2)C1 CC1(C)OCC(NC(=O)NCc2ncc(C(F)(F)F)cn2)C1O CCCC(C(=O)NC1CCOC(CO)C1)C(C)C c1(C=O)cncc2ncn(C)c12.C(C)(CC)NC(C1(C(=O)NC)CC1)=O.O Nc1c(F)c(F)cc(C(N2CC3CC2C3NC(C2CCS(=O)(=O)N2)=O)=O)c1Cl CCC(C)C(C(=O)N(CC(F)(F)CO)C)N(C)C(c1cccnc1)=O C1(N(C(=O)COc2ccsn2)C)CN(C(=O)COC2CCC2)C1 c1(NC(C(C(C)C)OC)c2n(CC=C)nnn2)ccc(F)cc1SC C(=O)(CCC(C)C)N1C(CC(=O)N(C)Cc2c(C)n[nH]c2)CCC1 N1(C(CCSCC)=O)CCN(C(C2COC(=O)N2)=O)C(CC)C1 CCC(CCCC(=O)NC1CNC(=O)C1(C)C)NC(c1ccc(Cl)cn1)=O c1(C(=O)NCC2(C)CCN(C(C3CCC(C)(C)CO3)=O)C2)ccc(F)c(N)c1F c1(C(=O)NCCC2CSCCN2C(=O)C=CC2CCOCC2)n[nH]c2c1COC2 CC(CC(C)(F)F)C(=O)NCCCCCNC(C1(Cl)CC1(C)C)=O C1(C=O)CNC(=O)CC1C.n1(CC(=O)OCC)cc(-c2ncoc2C)nn1.N C#Cc1cc(C(=O)NC2CCN(C(=O)C(F)(F)CC(C)C)CC2C)cc(Cl)c1 c1(C(=O)NC(C(C)NC(C2CCCS2)=O)C)ccc(-n2ccnc2)cn1 N1(CCNC(=O)NCC(c2cccc(C)c2)OC)CCC2(C1)OCCO2 C=CCCC(C(=O)N1CC2CC=CC1C2)NC(C1CC=CCO1)=O C(CCCCCO)(C(=O)NC)NC(CN(C(CC)CC)CC(C)C)=O N1(C(C(C)OCC#C)=O)CCC(C)C12CC2.c1(CC(=O)N)cnc(Cl)cc1C C1(C(=O)NCc2cccc(SC)c2)CC12CCN(C(c1ccccc1SC)=O)C2 c1(OCC(N2CC3(C(CNC=O)C3)C2)=O)ccc(F)cc1F.C1CCOCC1 c1(C(N2CC(NC(CC(C)(C)OC)=O)C(O)C2)=O)cc(=O)c2ccccc2[nH]1 Cc1cc(Br)ncc1NC(=O)C(=O)Nc1ccc(N2CCOCC2)c(Cl)c1 CC(C)C(C)C(C)CC(=O)N1CCCC(N(C(=O)CC(C)(C)C(F)F)C)CC1 C1(N(C(CN(C(CCOCCOCC)=O)CC(C)C)=O)C)CCCC(C)C1C C1(OC)CCC(C)C1.c1(Cc2nnnn2C(C)C)cn(CC)nn1.C(C)C.N c1(C(=O)NC2(CNC(COCCCC(C)C)=O)CCOC2)cc(O)ccc1F N1(C(C=CC(=O)OCC)=O)CCN(c2cc(-c3cc(C)nn3C)ccn2)CC1 C1(CNC(C(=O)NC(c2ccc(Cl)s2)C)=O)CCC2(CCCC2)O1 C(=O)(CCCC(C)=O)NC(CC)CNC(c1n[nH]c(=N)s1)=O c1(C(=O)Nc2nc(C)c(C)s2)cc(F)ncc1NC(c1ccc(F)cn1)=O C1(C(N2CC(C(C)(C)O)C2)=O)CNC(=O)CC1C.C1(C=O)(CC)CC=CC1.N C(=O)(CCC(C)C1CC1)N1CC(OCCNC(C2OCC(C)C2)=O)C1 c1(C(=O)OC)c(NC(C)=O)cccc1NC(N1CCC(C(=O)O)CC1)=O C(=O)CP(=O)(C(C)C)C(C)C.N1(C(c2n(CC)nnc2C)=O)CCCC(C)C1.N S(=O)(=O)(c1ccc(Cl)c2c(Cl)cccc12)N(C1CC[Si](C)(C)C1)CC=C N1(CCCCOCC)CC(F)(c2nc[nH]n2)C1 C1CCCN(C(=O)Cc2ccccc2N2CCOCC2)CC1.C=C1CC1C(=O)NC N1(C(c2n[nH]c(C)c2O)=O)CCCC(O)(CNC(=O)C(O)CC(C)C)C1 c1(C(N2CC(O)C2)=O)ccc2nc(S)[nH]c2c1.C1(CCC(=O)N)CC(F)(F)C1.C C12(NC(c3c(CCC)occ3)=O)CCC(CC1)N(C(=O)C(C(C)C)OCC)C2 c1cc(F)cc(F)c1.C1(CCC(=O)NCC2CC2)CCCC(O)C1.C(=O)C.C C1(NC(c2cc(C(=O)OCC)sc2)=O)CN(C(=O)C)CC1C1CC1.C=O N1(C(c2c(C)cccc2C)=O)CCN(C(=O)CC2CCCOC2C)C2(CCC2)C1 C1(NC(=O)CC(O)c2ccccc2)CN(Cc2ccnc(Cl)c2)CC1O CC1CN(c2cc(Cl)nc(C3CC3)n2)CCC1CNC(c1ccnn1CCF)=O C(=O)(C1=CCC(F)(F)CC1)NCCC(C)N(C)C(c1cccc2c1CCCC2)=O C1(N(C(CC(C)C)=O)C)CCCC(NC(=O)C(C)(C)c2ccnn2C)C1 C1(C)(NC(C(CC)n2cncn2)=O)CCCN(C(=O)Cc2cc(O)nnc2O)C1 c1(C(N2CC(CC=C)(NC(C34CCOCC3C4)=O)C2)=O)cccc(F)c1Cl C1(CN(C)C(C2(C#N)CC2)=O)CCN(C(C2CCC(C(N)=O)C2)=O)C1 N1(C(CC2C(=O)NC(=O)N2)=O)CCCC(C(=O)NCCn2cncn2)CC1 c1(C(F)(F)F)[nH]c(=NC2CCC=CCC2)sc1-c1ccccc1 N1(C(CCC(=C)Cl)=O)CCOCC(C)(CNC(c2cc(SC)c(C)o2)=O)C1 c1(N2CC(NC(c3c(OC)c(C)ccc3)=O)C(O)C2)cc(C)nc2cc(C)nn12 c1(C(=O)NCC2(O)CCN(C(C(C)C3(O)CCC3)=O)C2)nccc2ccn(C)c12 c1(-c2c(C)occ2)nc(CCC(=O)OC(C)(C)C)n(Cc2ccccn2)n1 C1CN(C(C2(C(N)=O)CC2)=O)CC(C)(C)C1.Cc1ncnc(C)c1CC(=O)N C(c1cncs1)=CC(=O)N(CC(=O)NC1CC(OC)C1)CC(C)C C(=O)(C(C)(C)c1ccns1)NCC(n1cc(CNC2CCC2)nn1)C CS(=O)(=O)C1CC(C(=O)NCC2CCN(C(c3ccnnc3S)=O)C2)C1 C(CO)(CCC)NC(c1cc(CC(C)C)[nH]n1)=O.C(=O)(C)N.C(=O)C1CC1 Cn1nc2c(c1C(N1CCC3(NC(c4ccc(=N)[nH]c4Cl)=O)CC3C1)=O)CCC2 CC(C)(CO)C(C)(O)CC(=O)NCc1ccc(Br)cc1Cl N1(C(C2(C)CCN(C(CCC(CC)OC)=O)C2)=O)CC(C)C(N=[N+]=[N-])C1 N1(C(C(CC=CC)C)=O)CCC(C(=O)NCC(C(C)(C)C)OC)C(C)(C)C1 C1(C(=O)OC)CC(n2cc(CCOC)nn2)CN1C(=O)CCCCN(C)C C(=O)(C(C(C)C)OCC(C)C)N1CC(O)(C(C)NC(Cn2c(C)nnn2)=O)C1 c1(C(NCC)=O)nn2c(c1C)CCCC2.C1CCCN1C(C1CCC(=O)N1)=O.C Cc1nsc(C(=O)NCC(C2CCN(C(C3(F)CC3)=O)CC2)(C)C)c1N N1(Cc2c(C)nc(C)o2)CC(C(=O)NCCC2CCOCC2)CC(C)C1 N1(CC=C)C2CCC1CN(C(=O)Nc1ncc(C(C)(C)C)cn1)C2 C1(C(C)C)CN(C(=O)CCCc2cc[nH]c(=N)c2)c2ccccc2N1 N1(C(C(CC(C)C)O)=O)CCC2(CC1)CCN(C(=O)CC(C)C1CCCC1)CC2 N1(C(COC(CNC(COCCOCC#C)=O)(C)C)=O)CCCCCCCC1 c1ccccc1.C(C)(C(=O)NC(C)(C)CNC(=O)CNC)NC(CC)=O C(c1cccnc1)=C(C)C(=O)NC(CNC(c1nn(C)cc1Br)=O)C(C)(C)C C(CN=c1[nH]c(=NCC2CCCO2)[nH]c2c(F)cc(F)cc12)c1cn(CC)nc1 Cc1nn2c(C(=O)NC3CC(O)(CNC(=O)CCF)C3)c(C)nc2s1 N1(Cc2n(CC)ncn2)CCC(=O)N(Cc2ccn(C(C)C)n2)C1=O c1(CC(N2CCC3(NC(CC(CC)CC)=O)C(C2)C3)=O)c[nH]c2c(C)cccc12 C1(C2CCN(C(c3ccccc3CO)=O)C2)(NC(c2c(C)cc(F)nc2)=O)CC1 S(=O)(=O)(c1ccc(Cl)s1)N1CCN(C(Cc2ccc(C(=O)OC)cc2)=O)C2C1C2 C1(C(N2CCCCC(N(C)C(c3ccc(Cl)s3)=O)C2)=O)CCc2nc(O)[nH]c2C1 C(c1ccccn1)=CC(=O)N(C)CCOCCCN(C)C(c1cnc[nH]1)=O N1(CCN(Cc2ccccc2)Cc2cnc(-c3cn[nH]n3)s2)C(C)CCC1C C1(NC(C2(OC)CC2)=O)CN(C(=O)Nc2cccc(C#N)c2)CCC1C CN1CNC(=O)C12CCN(C(=O)NCCn1cc(Cl)cn1)CC2 C1(CNC(c2ccc(C3CC3)cc2)=O)CCN(C(C23COC(C2)C3)=O)CC1 C=CC(CC)CC(=O)NC1CCCN(C(=O)CCc2cnn(C)c2)CC1 c1(CC(=O)NCCCN(C(c2cc(C)c(O)nc2)=O)C)cc(S(N)(=O)=O)cn1C CC1=NS(=O)(=O)NC(C)=C1CC(=O)N1CCC(NC(c2cn(C)nc2O)=O)C1 c1(C(C(=O)NCC(F)F)N(C(C(=O)OC)C)C)cc(C(F)(F)F)n(C)n1 N1(Cc2c(F)ccc(C)c2)CCC2(CCCC2C(=O)NCc2cncn2C)C1 N1(C(Cc2ncc(CC)[nH]2)=O)CC(CNC(=O)Cc2ccc(C)cc2)CCC1C C1(S(C)(=O)=O)(C(N2C(CNC(C3CCN(C)C3)=O)CCC2)=O)CCCC1 c1(C(=O)NC2(CCCC(=O)N(C3CCN(CC)C3)C)CCC2)nc(O)sc1C CC1(CNC(=O)CSCC(F)(F)F)CCCN1C(=O)C=Cc1cnc[nH]1 O=C(CC(F)(F)C(F)F)NCCNC(C1(CS(C)(=O)=O)CCC1)=O c1(CN2C(C(N3CCC(F)C3)=O)CC(F)C2)cccc2nonc12 CC(CCNC(=O)CN(C(=O)CC12CC(C1)C2)C)NC(N)=O Brc1ccc2nc(C3CCCN(Cc4nnnn4Cc4ccccc4)C3)[nH]c2c1 [SH](=O)(=O)CCC.C(C(C)N)N(CC)CC.C(C)(C)C.C(C)(C)C.C=O N1(C(C(CCC2CC2)NC(c2cc(C)oc2)=O)=O)CCN2C(=O)NCC2C1 CC1c2cc(Br)ccc2CCN1Cc1ccc(-c2ccc(OC(F)(F)F)cc2)s1 c1(CC)cc(NC)cc(C(N2CCC(CCNC(=O)C)CC2C)=O)c1.C(N)=O N1(CC)CCc2cc(Nc3c(Cl)ncnc3Cl)ccc2C1.c12ccsc1C(=O)N2 N1(C(C2(C#C)CC2)=O)CCC(C(CO)NC(=O)C(C)OCCN(C)C)CC1 C(=O)(N1CCCc2nccn21)C1(NC(=O)CNC=O)C(C)CCC1 N1(C(COCCC)=O)CCC(CNCc2nnc(C(C)(C)C)o2)C(C)C1 N1(C(CN2CCC(C)(C#N)C2)=O)CCC2C(F)(F)C2(C)C1 Cc1cc(CCC(N2CCCC(NC(c3cccc(CO)n3)=O)C2)=O)cc(C)c1 Cc1cc(C(=O)NC(CNC(=O)C(C)(C)F)C(C)C(C)C)cc(C)c1Br N1(C(CCCOC(CCC)=O)=O)CCOCC1CCNC(C1(C(N)=O)CCC1)=O C(N=C(NC1CCS(=O)(=O)C1)NC1CCc2sc(Cl)cc21)c1ccc(F)s1 C1(NC(c2c(C)scn2)=O)COCCN(C(c2ccc(-c3cccs3)cn2)=O)C1 C1(CN(C(C2CC2C)=O)CC)CCN(C(=O)COc2ccc(Cl)nc2)CC1 c1(C(N2C(C(=O)NCCC3CC4C=CC3C4)C=CC2)=O)nc2ccc(F)cn2n1 C1(C(C)NC(C2CN(C(C)C)C2)=O)CN(C(=O)CN2CC=CC2)CCO1 C12(C(=O)NC3(CC=C)CN(C(=O)Cc4cccnc4)C3)OCCCC1C2(F)F c1(C(=O)NC(CN(C)C(C2CC2Cl)=O)(C)C)cnc2c(c1)CCC(=O)N2 CC1CN(C(c2ccnc(N3CCC(C)C3)c2)=O)CCCN1C(=O)C(F)F c1ccncn1.C(=O)(C(C)N(C(C1(C=O)CC1)=O)C1CC1)OCCC.N C1(NC(C(c2cccc(C)c2)=O)=O)CCN(C(c2cnc[nH]2)=O)CC1C(C)C c1(C(N2CC(C(=O)NCc3cc(C)nn3C)SCC2)=O)ccc2nc(O)[nH]c2c1 c1(C(C(=O)NCC(CNC(c2c(CC)c[nH]n2)=O)O)C)ccncc1C N1(C(COC2(C)CN(C(c3nn(C)c(O)c3)=O)C2)=O)CC2CCCC2C1 C(=O)(C1CCc2ccccc21)NC1(C)CCN(C(C2(F)C(C)(C)C2(C)C)=O)CC1 c1(C(=O)NCC(CO)NC(c2cc(CCC)[nH]n2)=O)cccc(OC)c1OC N#Cc1ccc(C(=O)NCC2CCCCN2C(=O)Cn2ccsc2=N)[nH]1 CCCCC(C)C(=O)NC(C)(C)CN(C)C(c1ncnn1CC)=O c1(C(=O)NC(C(C)NC(c2cccc(CC)n2)=O)C)ccc(F)c2ccncc12 c1(C(N(C2CN(C(C(c3ccc(C)cc3)C)=O)C2)C)=O)cc(C)nc(Cl)c1N Cc1cccc(C(N2C(C(=O)NC3(C)CC3(C)C)CC3CCCC23)=O)c1C#N N1(C(c2cc(CC)ncn2)=O)CCC2(CCCC2NC(=O)CC(C)OC)CC1 C1(F)(CNC(c2cc(SC)oc2)=O)CCN(C(C2NC(=O)OC2C)=O)C1 CC(C)(O)C(CCO)NC(C12CC(CO1)N(C(C1(C)CC(C#N)C1)=O)C2)=O N1(C(c2c(SCC)nccn2)=O)CC(NC(=O)CS)C(C)C1.C1CCCO1 c1ccc(C(=O)N(CC(C)C)C2CCC2)cn1.C(CC(=O)N)OCCCOC N12CCc3ccc(cc31)CN(CC)C2=O.c1(OCC)nc(C2CCCCC2)cs1 c1(C=O)ccc(C)c([N+](=O)[O-])c1.C1(NC(C2(C)CC(=C)C2)=O)CCCCC1.C C1(C(=O)NC2CN(C(C(C(CC)C)O)=O)C2)COc2cccc(OC(C)C)c2C1 c1(C(N2C(C)CC2CO)=O)cccc(O)c1Cl.c12csc(n1)CNC2=O c1(CNC(C2N(C(CCCSC)=O)C(C)CC2)=O)ccc(F)cc1O N1(C(c2n[nH]cc2I)=O)CCc2sc(-c3ccc(CO)c(Cl)c3)cc2C1 c1(CN2C(C(N3CCCC3C(F)(F)F)=O)C3CCC2C3)ccc([N+](=O)[O-])cc1 Cn1ccc(C(N2CCCN(C(=O)CC3(C)CC3(F)F)CC2)=O)cc1=O C(N=c1[nH]c(C)c(C(N2CCC(Br)CC2)=O)s1)C1(C(=O)OCC)CC1 N1(C(C=CC(=O)OC)=O)CCC2(CC1)CCN(C(=O)C(C)(C)C(F)F)CC2C C1(N(C)C)CCCCC1C(=O)Nc1cnc(C(C)(C)C)s1 C1(CNC(CCCC)=O)CN(C(c2ccc(-n3cnnc3)cc2)=O)CCC1C C(=O)(CC(C)(C)C#N)N(CC(CO)(CO)NC(c1c(CCC)[nH]nn1)=O)C.C c1(CN2C(CC)CN(C(=O)CCC(F)(F)F)CC2)nccc2occc12 N1(C(c2cn(CC)nc2)=O)CC2(C1)CC1(CCC1)C2.C1(C=O)CC12CCCC2.N N1(CC(CC)OC)CCC2(CC1)CC(C)N(C(c1ccncc1C)=O)C2 c1(C(=O)NC(C(=O)OC)CC2CNC2)nn(-c2ccccc2F)ccc1=O C1(C(=O)NC2(CF)CCN(C(C3(n4nccn4)CC3)=O)C2)CC2C=CC1CC2 Cc1cc(NC(C2(NC(=O)Cn3cnnn3)CC(O)C2)=O)c(O)c(C)c1 N1(C(CC2CC(=C)C2)=O)CC2CCC1C1CN(C(=O)CN(C)C(C)C)CC21 CC1(CNC(c2csnc2C2CC2)=O)CCCN1C(=O)CN1CC2CC2C1 C(=O)(CCC(=O)NC(c1ccccc1)C(C)NC(=O)C1CC1)NCC c1(OC)cccc(CNc2cnn(C3CC(NC(C)(C)C)C3)c2C)c1F CCCCC(O)CC(=O)N1CCN(CCN(C)C(C2(CO)CCCC2)=O)CC1 N1(C(CC2CC(=C)C2)=O)CC(NC(=O)CC(=O)NC2CC2)CC12CCOCC2 c1(OC)ccc(C(N2CC(CC(C)NC(=O)C(C3CCCCC3)O)C2)=O)cc1N N1(C(c2c(C)cc(C)o2)=O)CCC(NC(C2CC(=O)NC(CCO)C2)=O)C(F)C1 n1(CC(C)C(=O)Nc2cnc(N(C)C)c(Cl)n2)ncc2c1CCCC2 N1(C(Cn2nnc(C)n2)=O)CCC(C)C1CNC(C1(N2CCOCC2=O)CC1)=O c1(C(N(CCNC(=O)CCC2CC2)CC)=O)ccc(N2CCOCC2)cn1 Cc1ccc2c(C(=O)NC3CC3NC(C3CC(F)C3)=O)cnn2c1C N1(C(C(N2CCC(C)C2)=O)=O)CC2CCN(C(=O)COC3CCCC3)CC12 c1(NC(CC2(CCC#C)N=N2)=O)cc2ccc(Br)cc2n1C N1(C(c2c3cccc(C)c3[nH]n2)=O)CCC2CC(CNC(=O)C(C)C)CCC2C1 C1(CC(=O)NCC(CC)NC(c2cc(O)cc(F)c2)=O)CSc2ccccc2O1 c1(C(C(=O)NCC=C)N2CCC2C(=O)NC)ccc(F)c(C2CC2)c1 N1(C(CSCCCC)=O)CCN(C(c2ccc(CO)cc2F)=O)C(CO)C1 C1(C=O)CC(=O)NC(c2ccccc2)C1.C(C)CC.C1(CSC)CC1C=O.N C1(CNC(CC)=O)CCCC(CNC(=O)C=O)C1.c1ccccc1SC(F)F C(=O)(CCCCCCCC1CC1)NC1CCN(C(CCOC)=O)C1 c1(C(N2CC(CNC(c3coc(Cl)c3)=O)C3(C2)CC3)=O)ccc2cc[nH]c2n1 c1(C(=O)NCC2C3CN(C(c4c(CCC)[nH]cc4)=O)CC32)cn2ccccc2n1 C(C(CC(=O)NC(COC)C(C)C)OC)NC(C(C1CCC1)OCC)=O C1(NC(C(C(CC)O)C)=O)CC2CCC(C1)N2C(=O)Cc1ccc(C(C)=O)cc1 C(CC(C)(C(=O)O)NCCNC(=O)COC1CCCCC1)SCC C1(NC(C(CC(C)C)N(C)C)=O)CCC2(CC1)CN(C(=O)Cc1ccn(C)c1)C2 CC1(NC(=O)C2=NOC(CNC(c3cncs3)=O)C2)CCCC1(F)F N1(C(C2C(C)C2)=O)C2CCC1CC(CNC(c1ccc(C(C)(C)C)s1)=O)C2 c1(CC)cc(C(N2CCC(N3CCN(C(=O)C(C)C4CC4)CC3)C2)=O)ncn1 c1(C(=O)N)ccc(F)cc1C.C1(CNC(CC=C)=O)CCCCC1NC(=O)C C(=O)(C1CCc2nccn21)N1Cc2c(C(N3CCC(C(C)(C)C)C3)=O)coc2C1 N1(C(C(CCC)C)=O)CCC(C2(O)CN(C(c3cnn(C(C)C)c3)=O)C2)CC1 S(=O)(=O)(CCC(F)(F)F)N1CC(CN(CC(C)(C)C)CC(C)(C)O)C(O)CC1 N1(C(CN(C)C(N)=O)=O)CCCC(C2CCCN2C(c2ccncc2O)=O)C1 c1(C(C)OC(C2CCC(=O)C2)=O)ccc(Br)cc1F C12(C=O)CCC(CC1)CC2.C1CCC1.C1(COC)CC1C=O.C(C)=O.N N1(C(=O)NC(c2ccccc2Cl)C(N)=O)CC(c2ccccc2)C(O)C1 c1(C(=O)OC(c2ncccn2)C2CCCC2)c(F)ccc(F)c1Br C1(c2cccc(F)c2)(C(=O)NC(c2nnc(C3CC3)n2C)C)CCCCC1 C(=O)(CC(F)(F)F)NCc1scc(CNC(C(N2CCNC2=O)C)=O)n1 C12(CNC(c3scc(C)c3)=O)CCC(CN(C(C3CCCN3N=O)=O)C1)C2 c1(C(=O)NCCC(CC)N2CCCC2=O)ccc2c(n1)NCCO2 N1(C(C(C)OC)=O)CCCCC1CNC(c1cnn(C2CCOC2)n1)=O C=CCC(C(=O)N1CCC(C)C(NC(=O)CCc2ccc(Cl)c(Cl)c2)C1)C(C)C N1(C(c2c(C)cc(C)s2)=O)CCC(C(=O)NCCCc2ccco2)CC1C CCCCCC(C)(C)CNC(CSC1CC1)(C(C)C)c1nnnn1C CN1CCC(C(=O)N(C2CCN(C(C3CCOC3c3ccccc3)=O)C2)C)C1 C1(NC(c2cncc(OC)n2)=O)CCC12CCCN(C(=O)C(O)CC(C)(C)C)C2 S(=O)(=O)(c1cccc2scnc12)NC(c1ccnc2c1CNCC2)=O c1(OC)ccc(NC(=O)C(O)CCCNC(=O)CCC2OCCO2)cc1F C1(C#N)(C(N2CC(C)(NC(=O)C)C2)=O)CC12CCOCC2.C1(CC)CCCC1.O N1(C(CSCC(C)C)=O)CCC(C(=O)NCC2(Cl)CCC2)C(C)(C)C1 Cc1cccc(C(=O)C(C)N(C(=O)CCc2cncc(C(=O)O)c2)C)n1 C(=O)(C(C)(O)CC(F)F)N1CCC(CN(C)C(C2CCSCC2)=O)C1 c1(C(N2CCC(O)(CCNC(C3(OC)CC3)=O)C2)=O)c(F)cc(C)cc1Cl C1(c2n(C)ncn2)CCCCC1C(=O)O.c1(CC=O)cccc(C(F)(F)F)n1.CC c1(OC)ncc(C(=O)NC2CCCCC2NC(=O)C=Cc2ncc[nH]2)cc1Cl c1(C(=O)NCC2C(C)CCN2C(=O)CN2CCOCC2)cnc2cnccc2c1 CC(CC(F)F)C(=O)NCCC1CCCN(C(c2c[nH]nc2F)=O)CC1 c1(OCCC)ccc(C(=O)N(C2CCC(NC(c3cc[nH]c3)=O)C2)C)cc1O C(=O)(C(C)(C)C1=CCN(C(=O)CCCCSC)C1)NC1(CC=C)CCOCC1 CC(COC(C)(C)C)N=c1nc2c(cnn2C)c(NCC2CCCOC2(C)C)[nH]1 c1(SCC(=O)NCC2N(C(c3ncc(C)nc3)=O)CC=C2)nc2ccccc2o1 C1(NC(COC)=O)CCN(Cc2ccc(Cn3cccn3)o2)CC1(C)C c1(OC)ccc(Br)c(C(=O)NCCC2COCCN2C(=O)CNC=O)c1 CC(CC(C)(F)F)C(=O)N1CCCN(C(c2cn(C)ccc2=O)=O)CC1C C#Cc1ccc(CC(N2CCCC(NC(C3CSC3)=O)C2)=O)cc1 C1(C(N2CC(OC)C2)=O)(NC(C2CC(N=[N+]=[N-])C2)=O)CCN(C)C1 N1(C(C(C)Sc2ccccn2)=O)CCOC2(CCN(C(C34CC(C3)C4)=O)C2)C1 C1(CC)CN(C(=O)CNS(=O)(=O)NC)CCN1C(=O)C(c1ccncc1C)C CCCCCC(C)NC(C1CC1CNC(=O)CCC=CC(C)C)=O N1(C(=O)C2COc3ccccc32)CC2CC(C1)C2N=c1[nH]nco1 Cc1cccn2ncc(C(=O)NC3CC(n4cc(-c5cc(F)ncc5F)nn4)C3)c12 CCCC(CCCNC(c1cc(C)n(C)c1C)=O)NC(=O)CC(C)OC N1(C(C2CC(OC)C2)=O)CCC(C2CC2)C1CNC(c1ccnc(Cl)c1Cl)=O C(=O)(C#CC1CCCOC1)NCC1(CNC(Cc2ccc(C)s2)=O)CCCC1 N1(C(c2ccccn2)=O)CCC2(CCCO2)C1.c1(CC(=O)O)cccc(CN)c1.C CCCCC(CC)CC(=O)NCCn1cc(C(=O)N(CCC(F)(F)F)C)nn1 c1(-n2ncc(C)c2)cccc(C(=O)NCc2ccc(CO)o2)c1 C1(N(C(=O)CCc2cscn2)C)CN(C(c2nocc2Cl)=O)CC1F c1(N2CCC(O)C2)nccc(N2CCN(c3ccc(-c4cscn4)nc3)CC2)n1 C(C(CNC(c1cccc(CO)n1)=O)C(F)(F)F)NC(c1nnc(C)s1)=O c1(C(=O)NCC(CCC)NC(c2cccc(CC)n2)=O)cncc(N)n1 C1(C(=O)NCCCn2c(C)ncc2)CCCCCN1C(c1cnccn1)=O N1(C(c2c(C)cc(F)cc2)=O)CC(NC(=O)C(C)C(C)(F)F)Cc2ccccc21 N1(c2cn(C)nc2)CCC(C(=O)OCc2nc(CS(C)(=O)=O)no2)C1=O O=C(NNS(=O)(=O)Cc1ccc(Br)cn1)c1ccc(F)c(Cl)c1 N1(C(C2C(SCCCC)C2)=O)CC2CC(C(=O)NC(CCC)CCO)C(C2)C1 c1(C(=O)NC2C(NC(c3cnc(C)s3)=O)CCCC2)ccc2[nH]c(C)c(C)c2c1 CC(F)CC(=O)NCC1(C(N)=O)CN(C(=O)CC2C=CCC2)C1 N1(c2snc(CCC)n2)CCC(C2CC2)C1CNC(=O)C(C1CCOCC1)F N1(C(C=C(CCC)C)=O)CCCC(CCC(N2CC=CC2CF)=O)C1 C(=O)(CCCCCCC(=O)NC12CCCC1CN(C(c1n[nH]cc1C)=O)C2)OC C(=O)(CC(C)(C)CCC)N1CCC(CC=C)(NC(c2ccc(N)cc2F)=O)CC1 Cc1ccc(C=CC(=O)NC2CCC(N(C)C(C3CS(=O)C3)=O)C2)cc1C c1(OCC)cnc(C(N2CCCC(C)C2)=O)c(Cl)c1.C(=O)(CC(C)N(C)C)N c1(C(N(C(=O)CCN(C(=O)CN=[N+]=[N-])CC2CC2)CC)C)ccccn1 C1(C(=O)Nc2cncnc2Br)CC2(CC2)CN1C(c1cnc(O)c(Br)c1)=O C12(C(=O)NCC(CSC)(C)O)COC(C1)CC2.c1(C=O)cc(N)cc(F)c1 C#CCCCCCCCC(=O)NC(C)CCNC(=O)CC(C)(C)COC CCC(CC)CC(=O)NC1COCCC1C(=O)N(C(C)(C)COC)C Cc1cc(C)n(CC(=O)NC2CCCCC2N(C(=O)C2=CCCSC2)C)c(=O)n1 CCCC(O)(CCC)CC(=O)NCC(O)CN(C(=O)CC1CCS(=O)(=O)CC1)C C1(C(=O)NC2C=CCN(C(c3cnc(Cl)[nH]3)=O)C2)CC2(CCCO2)C1 S(=O)(=O)(c1cccc(=NC2CCN(CC3CC3)CC2)[nH]1)N(C(C)(C)CCO)C C#Cc1ccc(OCC(=O)NCC(C)NC(=O)Cc2ccc(O)cn2)c(O)c1 c1(C(N(C2CCCN(C(C34CC(F)C3C4)=O)CC2)CC)=O)cc2occc2n1C Cc1nn(C)c(C(=O)NC2CC3(C2)CC(NC(=O)CC)C3)c1Cl.C(C)(C)C C12(NC(c3cnn[nH]3)=O)CC1CN(C(c1cc(-c3cccc(Br)c3)on1)=O)C2 Cc1nn2ccccc2c1C(N1CC2C(C1)C2(F)F)=O C(=O)(CC1=CCOCC1)NC1(CC(c2ccc(C)cc2)=O)CC1.Cn1cncc1 CON(CCC(=O)NC(C)CCF)C(=O)C1(OC)CCOC1 C1(NC(C(C)NC(=O)NC)=O)CCN(C(=O)C(N2CSCCSC2)C)C(C)C1 C1(C(=O)NCC(CCC)NC(=O)Cc2cc(C)on2)CC12CCOCC2 Cc1ccnc2c(C(=O)NCCCC3CCCN3C(=O)C(C)CC3CC3)cnn12 N1(C(C2(OC)CC2)=O)CCC(CCC)CC1.c1(C(=O)N)c(C)noc1C(F)F C1(C(=O)NC2CCN(C(c3c(C)onc3)=O)C2(C)C)CCCCN1S(N)(=O)=O c1(C(=O)NCCC(=O)NC2CCCC(C(=O)NCCCO)C2)cccnc1O.CC c1(CN2CCC(F)(C(=O)NCC3(O)COC3)C2)cc(F)ccc1Cl c1(CN2CC(C(N3CCC(F)(CO)C3)=O)C2)ccc(C(F)(F)F)c(Cl)c1 S(=O)(=O)(c1ccc(NC2CCCCC2N(C)C)cc1Cl)N1CC=C(C)C1 CC1=C(C(=O)N2CCCC2CCC(=O)N(C)Cc2cnc[nH]2)CCCO1 c1(C(N2CC(C(C)NC(C(C)CO)=O)C2)=O)cnc2[nH]nc(O)c2c1 N1(C(CC(=O)OC)=O)CCCC1C1CCCCN1C(=O)Cc1csnn1 C1(N(CCCNC(=O)CCOC2CCCOC2)C(C)C)CCN(C2CC2)C1=O CCCCC(O)C(=O)NCC1CCC(NC(c2coc(-c3cnn(C)c3)n2)=O)C1 C=C(C)CC(C)C(=O)NCC1CN(C(=O)CCc2cnoc2)CCCO1 c1(C(N2CC(CCC)C2)=O)ncoc1C.C1(OC)CCCC1C(=O)N.C1CC1 N1(C(CSCCC(C)C)=O)CCC(NC(=O)CS)C(F)C1.c1cccc(Cl)c1 c1(C(=O)NCCCNC(C2(C#N)C(C)(C)C2)=O)nc2ncc(Br)cc2[nH]1 CCCCCC(=O)NCC(=O)N.c1(C(N(CC)C)=O)ccc(CS(C)(=O)=O)cc1 C(=O)(CCC(C)CC)N.N1(C(c2n(CCC)ccc2)=O)CC(C(F)(F)F)CC1C N1(C(C2(OC)CC2)=O)C2CCCC1CN(C(=O)CC(C(F)F)c1ccccc1)C2 C(=O)(CCCCNC(=O)Cn1cnc(C#N)n1)Nc1cn(CCOC)nc1 C1(NC(c2cnc(C)[nH]2)=O)C2CN(C(c3csc(C4CC4)n3)=O)CC12 Cc1cccn2ncc(C(=O)NCC#CCNC(=O)CC(C(C)C)C(C)C)c12 N1(C(CCc2cc(C)[nH]n2)=O)CC2(C(N3CC(O)(C(=O)OC)C3)=O)CC1CO2 c1(C=O)cnc(C)cc1C.N1(C(C=CCN(CC#C)C)=O)CCC(C)C1C.N CC1CCCc2ncc(C(=O)NCC(O)CCNC(=O)CC3CC=CC3)n21 Cc1nc2sc(C(=O)NCC3(NC(=O)CN(C)C)CCC3)cn2c1Br c1(NC(C(CCF)NC(C2CCCC2O)=O)=O)ccc2cccnc2c1 C1(C(=O)NCCNC(c2cccc(CC)n2)=O)CCC(=O)N(C)C1 CS(=O)(=O)C1CCN(Cc2cc(Cl)ccc2OCc2ccccc2)C1 CC1=C(C(=O)NC(C(=O)NCCCC(F)(F)F)C2CCOC2)CCO1 N1(C(Cc2ncc(C)s2)=O)CCC(CNC(=O)C=Cc2ncc(C)[nH]2)C(C)C1 CCC(C)(O)C(=O)NC1CCCCC1CC(=O)NCCc1cc(C)no1 c1(OC)ccc(C(=O)NC2CC23CC(NC(c2c[nH]nc2F)=O)C3)c(N)c1 n1(CC)cccc1C(=O)NCC(O)CNC(C1(C2CCCCO2)CC1)=O C12(NC(C3CC(F)(F)C3)=O)CCCN(c3ncc(Cl)cn3)CC1C2 c1(NCC(CC)C)ccc(S(=O)(=O)N2CCCC(c3ccn(C)n3)C2)c(Cl)c1 C1(CCC)(NC(=O)CC(C)(C)C)CCCN(C(c2cnc(N(C)C)cn2)=O)C1 c1(C(N)=O)ccc(C(N2CCN(C(C3CC3C#N)=O)C(CF)C2)=O)cc1Cl C1(n2cc(-c3cn(CC)nc3)nn2)CON(C(=O)CCc2ccccc2F)C1 CC1CCc2[nH]c(=NCc3ncc[nH]3)[nH]c(=NCC3CC3(Cl)Cl)c2C1 CC1(C)CC(C(=O)NCCc2ccoc2)(CNC(=O)CC2CCSC2)C1 C1(C(=O)NCc2ccc(CC)s2)CC12CC(NC(=O)C=C(C)C)C2 c1(C(=O)NC2CN(C(C(CC(C)C)N(C)C)=O)C2)cccc2ccncc12 CC1CC(NC(C2CCCC2NC(=O)CC2CC(=O)C2)=O)CC(C)(C)C1 N1(C(Cn2c(C)ncc2)=O)CC(CNC(C2CC(C)CC(C)C2)=O)C(F)(C)C1 c1(C=O)ccc(N(C)C)cc1.C(C(C)C(=O)NCC)OC.CCC.C1CC1.N C1(C(=O)NC(CC)CNC(c2ccc(Br)o2)=O)CCC(F)CC1 C(C(=O)NC1CCN(C(C2CC2CF)=O)CC1)(C(C)C)OCC C1(NC(=O)Cc2ccnc(O)c2)CC2CCC1N2C(C1(F)CCCC1)=O c1(OC)cc(C(N2CCCC2CCC(=O)NC(c2ncc(C)[nH]2)CC)=O)[nH]n1 CC1(C(=O)NCc2ocnc2C(=O)NCCn2cccn2)CCC2CC2C1 c1(OC)ccc(CCNC(=O)NCC23COCC(COC2)O3)cc1OC C(S(=O)(=O)CCC(=O)NC1CN2CCC1CC2)c1ccc(C)cc1C Cc1cnc(C)c(NC(=O)C(=O)Nc2cncc(Cl)c2)c1 Cc1cc(=O)oc(C)c1C(=O)NCC1CCCC1.C(=O)CCCn1ccnn1.N C1(NC(CCc2cc(OC)no2)=O)COCCC1NC(c1cnns1)=O N1(C(C2CCC(C)O2)=O)CC2(CCOCC2C(N2CCCC(O)CC2)=O)C1 c1(CC)cn2c(n1)CCC(C(=O)NCc1ncc(CC)cc1C)C2 c1(C(=O)NC(C2OCCN(C(Cn3c(C)cc(C)n3)=O)C2)C)cc(F)ncc1C C1(NC(c2cnc(C(C)C)s2)=O)CCN(C(C23CC2C3)=O)CC1C Cc1cc(C(N2CC(O)(C)C2)=O)cc(C)c1N.C1(CC(=O)N)COC(C)(C)C1 C(=O)(C1CCCn2c(C)nnc21)N1CCN(C(C=COCC)=O)CC(CO)C1 C1(NC(C2CCCCCC2)=O)CC12CCN(C(C1Cc3ccccc3S1)=O)CC2 c1(C(=O)NC(CC)CNC(c2ccccc2C(F)(F)F)=O)cc(C)c(C)cn1 CCC(CCCC(=O)NCC1CC2CCC(C1)C2)NC(=O)CCC1CCOCC1 c1(C(N2CCC(C(C)C(=O)NCC(CC3CC3)CO)C2)=O)cc[n+]([O-])cc1 C=C(C)C(C)(C)C(=O)NCC(CC)N(C)C.N12CCCC(C)(C1)C2=O c1(C(N(C)CC2CCN(C(=O)CCC3CCOCC3)C2)=O)cccn2ccnc12 C1(C(N(CCN(C(=O)C(CCO)N(C)C)C)C)=O)CC2OC(=O)OC2C1 C1(C)CCN(C(C2CC(=O)N(C)C2)=O)CC1.C1(C(=O)N)(OC(C)=O)CC1 Cc1nc2nccc(C(=O)NCC(C)N(C(=O)CCC(C)N(C)C)C)n2n1 c1(OCC)ccc(C(C)NC2CCN(C)C2)c(Cl)c1 N1(C(c2ccn(CCC)n2)=O)CCC(NC(=O)CC2(C)CCC2)C(C)C1 c1(CC)c(OC)cccc1C(N1CCN(CCNC(=O)CCCCCO)CC1)=O N1(C(CSSC)=O)CCCC(C2CN(C(=O)CC3CCCCC3(F)F)C2)C1 C(=O)(C1=C(C)NC2=NCCCC2=C1)N1CC(CNC(C(CC)(C)CO)=O)C(O)C1 C(=O)(C1CCCc2sccc21)NC1CC(C)(NC(Cn2c(CCC)ncc2)=O)C1 c1(CCC)onc(C)c1C(=O)NCCC(C(C)C)NC(c1ccc(CC)cc1)=O Cc1csc(C(=O)NCCOC2CCN(C(=O)C(O)C(C)C)C2)c1Br C1(NC(COCC)=O)CC(NC(=O)CNC(=O)C2CC2)CC1O c1(N2CC(CC)SCC2)[nH]c(=NC2CCOC2)nc2c1ncn2C(C)C Cn1c(C(=O)NCCOCC(N2CCC(CSC)C2)=O)cnc1Cl c1(-c2cn(C(C(=O)NC(CC(=O)NC(C)C)C)C)nn2)cccc(OC(F)F)c1 c1(N2CC(C)CC(OC)C2)nc(=NCC2(n3nccn3)CC2)[nH]c2c1CCC2 CC(C)C(F)C(=O)NC1(C2CCCN2C(c2cccc(CN=[N+]=[N-])c2)=O)CC1 c1(C(=O)NC2C(NC(COCCCOC)=O)C2)cnc(-c2ncccn2)s1 N1(C(CC2(C=C)CN(C(c3cnn(C(C)C)n3)=O)C2)=O)CCC(OC)C(C)C1 N1(C(c2cc(C)c(Cl)s2)=O)CCOC(C)(CNC(c2ccnc(C)c2C)=O)C1 C1(C(=O)NCC2CCC=CO2)(CC)CCN(C(=O)CCCCSC)C1 C1(NC(c2c(OC)ccs2)=O)CCCN(C(c2cc(Cl)c(Cl)cc2N)=O)CCC1 C1(CCC)CN(C(=O)Cn2nnc(C)n2)CCN1C(=O)C(=O)NC(C)C N1(C(c2cc(C)nc(Cl)c2)=O)C2CCCC1CC(NC(C1CCCN1C)=O)C2 Cc1cc(=N)[nH]cc1C(=O)N(C1CCN(C(=O)CC(C)n2ccnc2)CC1)C C1(c2n(C)ncc2)CN(C(C(=O)NCCC2CC2)C2CC2(C)Br)CCN1 c1(CNC(C2(NC(c3cnc(C)[nH]3)=O)CCSC2)=O)ccc(C)c(C)c1 c1(OC)cc2cc(NC(N3CCSC(C)C3C)=O)[nH]c2cc1C(C)=O C1(CC(=O)NC2CC(NC(C3CC(O)(CC#C)C3)=O)C2)(O)CCOCC1 c1(C=O)ccc(N)c(F)c1.CC(C)(C)CCNC(c1cn[nH]c1)=O.C1CC1.C C1(CCC)CN(C(=O)C(C)OC)CCN1C(=O)CCc1cccc(OC)n1 C1(NC(CCc2ccc(C)c(Cl)c2)=O)CN(C(C2(CF)CCC2)=O)CCC1(C)C C1(C(N2CCC(CC(C)C)CC2)=O)CN(C(c2cnn(C)n2)=O)C(C)(C)C1 c1(SCC(=O)NC(CC=C)CNC(=O)Cc2cc(C)cs2)ccccc1.C C(=O)(C1=CC2C=CC1C2)N.CC1(CCNC(c2cc(C)cs2)=O)CC1(F)F C1(C(N2CCC(N(C(c3c(C)nns3)=O)C)C2)=O)CC2(COC(=O)N2)C1 c1(C(=O)OCC)ccccc1C(=O)NCc1ccnc(O)c1.c1cccnc1 N1(C(COCCCC#C)=O)CC(N(C(=O)C(F)=C2CCCC2)C)CC12CCOC2 CCC(C(=O)NCc1nocc1C(N1CCCC1CC(N)=O)=O)N(C)CC CC(C)CC(C(=O)NC(C)(C)C(=O)NCC1CN(C2CC2)C1)C(C)C c1(NC(C)=O)cc(C(N2CCC(CCNC(c3ccns3)=O)C2)=O)ccn1 CC(C)(CO)CCNC(C1COC(CNC(=O)CC2CC(F)C2)C1)=O c1ccccc1OC1CC1.c1(C(C(=O)NC)N(C)CC)ccn(C2CCC2)c1 c1(OC)ccc(F)cc1C(=O)N(C(C)CNC(C1CCC(=O)N1)=O)C C(C1CC1)(C1CC1)=CC(=O)NCc1ncccc1C=O.c1(CC)ccccc1 c1(C(=O)NC2CN(C(Cc3cc(C)no3)=O)CC2O)c(F)cncc1F C#CCC(C)(C)C(=O)NCCCNC(C1CC1)=O.c1(C2CC2)ccccc1.N Cc1ccoc1C(=O)NCC1CCCC1NC(=O)CSC(=N)N Cc1cnc(CNCC(c2ccccc2F)N2CCOCC2)c(O)c1 C(CC(=O)NCCCN(C(c1cnsn1)=O)Cc1ccsc1)OC(C)C c1(CC(c2n(C)ccn2)NC(c2cnc(-c3ccc(Cl)s3)s2)=O)ccc(F)cc1 C(=O)(C(F)C(C)(C)O)N.c1(C(=O)NC)ccc(C(=O)NC(C)CCCC)cn1 CC1CCCC(C(=O)NCc2ccccc2CNC(c2ccncc2)=O)C1 N1(C(CC2(OCC)CC2)=O)CCOC(C(=O)NC2C(C)CCC2C)C1 c1(NC(C2CCN2Cc2ccc(Br)cc2CO)=O)c2c(cc3c1CCC3)CCC2 N1(C2CCN(C(c3c(C(C)(C)C)ncs3)=O)C2)CCN(C(C2CC(F)C2)=O)CC1 C1(NC(=O)NC2(C)CCSC2)CCCCC1C(=O)NCC1CC1 C1(NC(C2(C)C(C)(C)C2)=O)C2CC(NC(=O)CC3CCSC3)CC12 N1(C(COCC)=O)CCC2(CO)CN(C(c3cncc(P(C)(C)=O)c3)=O)CC2C1 CC1CC(CNCC2(OCCO)CCC2)C1(C)C c1(C(C)(C)C(=O)N(CCCNC(=O)CCc2nncs2)CCO)cccc(Cl)c1 n1(C(C)C)ccnc1CNC(C1CCN(C(C2CC=CC2)=O)C1)=O N1(C(C=CC=CC)=O)CC(NC(=O)Cc2ccc(O)nc2)C(O)C1 C(=O)(CS(F)(F)(F)(F)F)NC(CN(C(=O)CC1CCCC(O)C1)C)(C)C CCCC(C)(O)CC(=O)N1CCOCC(CNC(c2ccon2)=O)C1 O=C(CS(=O)(=O)NCC)NC(=O)Cc1csc(S)n1.C1(CC)CCCO1 C(=O)(CC(C)(C)CC(F)F)N.n1(C(C(=O)NCCC)(C)C)cc([N+](=O)[O-])cn1 N1(C(COC)=O)CCC(C)(NC(=O)CCN2CCCC2)CC1.c1cn(C)nc1O C(CN=c1cccc(S(=O)(=O)NCC2CCOC3(CCC3)C2)[nH]1)(OCC)OC c1(C(N)=O)cc(C(N2CC3C(NC(=O)C(O)C4CCC4)C3C2)=O)ccc1O CCC(CC(=O)N1CCCC1C1CCCC1)N(C(=O)CC1(OC)CC1)C C1(CCC)CN(C(=O)C(C)(C)c2ccsc2)CCN1C(c1ccc(COC)s1)=O c1(C(=O)NCC(C2CCC2)NC(=O)C(F)=C2CCCC2)csc(O)n1 C1(C(N2CCC(c3ccccc3)(NC(C3CCC3)=O)C2)=O)CCC(F)(F)CC1 C=C(C)C(C)(C)C(=O)NCC(C)N(C(c1cnc(C(F)F)s1)=O)CC C1(NC(CCN2CCN(C)CC2)=O)CC2(CO1)CN(C(=O)COCC(F)F)C2 C1(CC)COCCN(C(=O)CN(C(=O)CC2CCCC3CC23)C2CC2)C1 C1CC2CCC1N2C(c1cc[nH]n1)=O.c1(OCC)cc(C(=O)N)on1.N(C)C c1(C(=O)NCC2CC3CN(C(C4C(CC)C4)=O)CC32)nc2ccccc2s1 N12CCC(C1)CSC1CC1C2=O.CC(C)(C)SC(C)(C)C c1(NC(CNC(CC(=C)C)=O)(C)CC)ccc(OCCCOC)c(OCC)c1 c1(C(c2nnnn2C(C)C)NC(CC)CC)c(C)nn2cc(Br)cnc12 N1(CC(N2CCN(C(C)=O)CC2)=O)C(=O)CN(C)C1=O.C(C=O)(C1CC1)OC N1(C(c2ccc(CC)c(Cl)c2)=O)CCCCCC(NC(=O)C(C)C(C)(F)F)C1 Cc1cnc(NC(=O)CCCc2cc(C)ccc2C)c(C)c1 c1(C(=O)NCC(CC)NC(C2CN(C)CCO2)=O)cc2c(F)c(F)c(F)cc2[nH]1 C(=O)(C#CC1CCCO1)NC1CC2CC(NC(c3ccc(CC)cc3O)=O)C2C1 CC1CN(C(c2cc[nH]c2C2CCC2)=O)CC1CNC(c1csnc1Cl)=O Cc1c(NC(C2CC(O)CN2C(c2cc(Cl)ccc2F)=O)=O)cncc1Br C(=O)(C1CCc2nccn21)N1CCCC(C(=O)NCCC2C(=O)NC(=O)N2)C1 c1(NC2CC(NC(CNS(N(C)C)(=O)=O)=O)C23CCC3)nc(Cl)nc2sccc12 C1(NC(c2cc3n(c2)CCSC3)=O)CCCCCN(C(c2cc(O)cs2)=O)C1 C1(CC(=O)N(CC#C)CCOC)CN(C(=O)C(C)(C)CC#N)CC12CC2 N1(C(C2C(OC)C2)=O)CCN(C(c2cnn3cc(C)cnc23)=O)CC2(CC2)C1 CC(C)C(C)(CNC(c1cc(CO)[nH]n1)=O)NC(C1CC(=O)N(C)C1)=O Cn1c(CN2CC3(CC(C(N4CCC5(CCOC5)C4)=O)C3)C2)cc2ccccc12 c1(C(=O)NC2CC(NC(CCCOCCC)=O)C2)cc(C(N)=O)ccn1 c1(C(N2CCC(NC(=O)CC3C=CCC3)C2C2CC2)=O)cc([N+](=O)[O-])ccc1O CC(CO)C(=O)N1CCCC1CCNC(c1ccc(C(N)=O)s1)=O N1(C(c2cnc(COC)[nH]2)C(=O)NC(C)(C)C)CCC(CC2CCC2)CC1 c1(N(CCCNC(C(C(=O)OC)C)=O)C(C)C)cc(OC)nc(C(C)C)n1 C(=O)(CC(C)CC(=O)NCC1(F)CC(NC(c2sccc2F)=O)C1)OC C(N(CC(C)O)N1CCCC(CO)C1)c1ccc(OC)cc1 C1CN(C(C2CN(C(=O)N(C)C)C2)=O)CCC1(F)F.CC(C(=O)NC)C(F)F C(=O)(C1=CC2(CCOC2)C1)NCC(C1CCCC1)NC(CN1CCC(C)CC1)=O c1(C(=O)NC(C2CCCN(C(=O)C(N)=O)C2)C)cccc(F)c1C(F)(F)F Cc1cnc2n1CCN(C(=O)NCCSCc1cccc(C#N)c1)CC2 C#CCCCC(C)C(=O)NC1(CNC(=O)C=Cc2cc[nH]c2)CCOC1 c1(C(=O)NC2C(NC(C(COC)(F)F)=O)COC2)cc(OC)c(OC)cc1O Cc1cc(C(=O)NCC(F)CNC(=O)C(C)Cc2cccc(F)c2)cc(Cl)c1 N1(C(=O)C(C2(O)CCOCC2)(F)F)CCCC(n2cc(COCCO)nn2)CC1 Cc1ccc(F)cc1CC(=O)NCC(CNC(C1CC(=O)CCO1)=O)CO c1(NC(C2CCC(N(C)C(c3cccc(C#N)c3F)=O)C2)=O)ccc2c(c1)OCO2 C12(NC(C3CC4(CCC4)C3)=O)CCN(C(=O)CCN3CCNC(=O)C3)CC1C2 CCC(CC(=O)NC(C)(C)CCNC(C1CCn2c(C)cnc2C1)=O)C(C)(C)C Cc1ccncc1CC(=O)NCCn1cnc(C(=O)NCCCC(=O)N(C)C)c1 C1(C(=O)NCCNC(c2cc(C)no2)=O)CC12CCCCCC2 c1(C(N2C(C)C(NC(C3CC3C)=O)CCC2)=O)ccc2ncn(C)c2n1 C(=O)(CCCN=[N+]=[N-])NCC=CCC(=O)NCCCc1n(C)nnn1 N1(C(C(CC#C)(C)C)=O)CCC(C)(C)C(C(=O)NCCN=[N+]=[N-])C1 C1(C(=O)NC2CN(C(c3ccc(NC)cc3Cl)=O)CC2C)CC2CCC1C21CC1 c1(NC2CCC3CN(C(c4c(C)cccc4Cl)=O)CC32)ncc(Cl)c(C)c1C#N N1(C(Cc2cncc(C)c2)=O)CCC(C2CCN(C(=O)CCCC3CCC3)C2)C1 c1(N2C(CNC(c3c(=O)cc(C)[nH]c3)=O)CCC2)ncnc2cnccc12 c1(CCC(=O)NCC#CCNC(C2CC2c2ccsc2)=O)ccccc1F N1(C(C2(NC(=O)CC3CCCC(O)C3)CC(O)C2)=O)CCC2(CC2)C1 N1(C(C2CC23CCC3)=O)CC2CC(C1)N(C(=O)CC(F)(F)Cl)C2 c1(C(=O)NCC(C2CC2)NC(c2ccc(C#N)o2)=O)ccc([N+](=O)[O-])o1 c1(C(=O)NC2C(NC(C(CCC)C(C)C)=O)CCCC2)c(Cl)c([N+](=O)[O-])nn1C CC(=O)CCCCC(=O)NC1C=CC(CC(=O)NCC(O)CNC(N)=O)C1 c1(NC(C2CN(C(c3cc(Cl)c(Br)cc3F)=O)CCO2)=O)ccc2cnoc2c1 c1(C(C)NC(=O)N(CCc2ccccn2)C(C)C)ccccc1.c1ncon1.C C1(C(=O)O)CCCCC1N(C1(c2ccon2)CC1)Cc1ccccc1 C1(CCOC)CN(C(C2(C)CCCC2)=O)CCN1C(=O)C(CO)OC N1(C(Cn2nnc(C)n2)=O)CCC2CCCN(C(=O)Cc3ncc(F)cn3)C2C1 c1(C(N2CC(N(C(CCOCCOC)=O)C)C(F)C2)=O)ncnc2c(C)csc12 c1(CC(=O)OC)ccccc1C=O.C1CCCC1C(=O)N(CC(F)(F)Cl)C.N C=CCC(C(=O)N1C2CCC1C(C(=O)NC1(CSC)CC1)C2)C(C)C c1(C(=O)NCC(CC)NC(C2CCC(N(C)C)C2)=O)c(F)ccc(F)c1F N1(C(Cc2cnc(C)o2)=O)CCC(NC(C2CC(C)CC(C)C2)=O)C(C)C1 c1(NC(C(N2CC(C)C2)C)=O)ccc2ncccc2c1.C1(C)(C)C(=O)N1 c1(OCCNC(Cc2nc(-c3cn(C)nc3)sc2)=O)cc(C(F)(F)F)cc(Br)c1 C(CCC(C)(C)C(=O)NC(C)C(C)(C)C)OC.c1(C=O)ccc(=O)n(C)n1.N C1(CC(=O)NCCC2(C)CC2)Cc2cc(F)ccc2O1.C1(C=O)CCC(O)C1 C(=O)(CC1=CCN(C(C2CC2(F)Cl)=O)CC1)N(CC(=C)C)C C1(NC(c2cc(C)ns2)=O)CN(C(=O)Cc2ccc(Cl)nc2F)CC2(CCC2)C1 C(C)(CC1CCC1)(C(=O)NCC1CC(C)C1)OC.C(=O)C(C)(C)C.N CN1CCOC(C(=O)NCc2ccccc2Cn2cc(CN)nn2)C1 N1(C(CCCC=C)=O)CCN(C(=O)C(F)=C(C)C2CC2)CC12CC2 C#Cc1ccc(OCC(=O)NC(C)(C)C(C)NC(c2ccnc(C)c2)=O)cc1 C=CC1CN(C(C23CC(CN(C(=O)C=Cc4ccccc4)C2)C3)=O)CCO1 c1(CCC)n[nH]cc1C(=O)NC1CCCC1C(N1CCC1C(C)O)=O C1(CNC(CSCC#C)=O)C(C)CCCN1C(c1cc(F)ncc1C)=O N1(C(=O)CCCn2ccnc2)CCC(NCc2c(C(F)(F)F)cccc2Cl)C(F)C1 C1(C(NOCC(C)(C)C)=O)CCCC(NC(c2cc(=N)[nH][nH]2)=O)CC1 C12(C(=O)NC3CC(C)(C)OCC3)CCCC1CCN2C(c1cscc1Cl)=O C1(OC)CC2(C1)CN(C(c1ccnc(CNC(=O)CC3CCCO3)c1)=O)C2 c1(C(N(C(CNC(CCOC)=O)C2CC2)C)=O)cc(Br)c([N+](=O)[O-])s1 c1(C(=O)NC2CN(Cc3cc(OC)c(O)cc3)CC2C#N)cc(C)c(Br)cc1C C(=O)(C1=CCCCC1C)N1CCC(O)(CNC(CS(=O)(=O)NCC)=O)CC1 CC(C)CCC(O)C(=O)N(C)CCOCCNC(=O)CC1CC(F)(F)C1 C1(C(=O)NCC2CCCN(C(=O)C3=CCCSC3)C2)CS(=O)(=O)CCO1 C1(NC(c2cc(CC)cn2C)=O)CCCCCN(C(=O)C(C)OC2CCOC2)C1 Cc1nc(N(CCCNC(c2nccnc2C(N)=O)=O)C)cc(C#N)n1 CCC(c1ccc(C)cc1)=CC(=O)NCC1CCCCN1C(C12CCC1CC2)=O c1(C(N2C3CC(C3)C2)=O)c(F)ccc(OC(F)F)c1F.C1(COC)CC1C=O C(=O)(C(O)C(C(C)C)O)N1CC(C)CC(C(=O)NC(C(=O)NCCC)C)C1 CC1(C)CCC(=CC(=O)NCC2CN(C(=O)CN3CCCOC3=O)CCO2)CC1 C(=O)(C(C)CCCC(C)=O)NCC1(COC)CCN(C(=O)C2=CCCOC2)C1 N1(C(C)=O)CCC(O)C1.C1(C)(N(C(COC(C)=O)=O)C2CC2)CCC1 CC(C)C(CC(=O)N(C1CCC(CO)CC1)C)NC(=O)C(N)=O N1(C(=O)NCC2CC(C)(C)OCC2)CCCc2occc2C1 c1(NC(c2ccc(-c3cncc(NC(C)=O)c3)cn2)=O)ccc(C#N)c(Cl)c1Cl c1(C(=O)NC2C(CC)CN(C(=O)C=CCOC)CC2)cc(C#N)ccc1F CC1CC(NC(=O)C=Cc2cn(C)nn2)CCN1C(=O)CC1CCC(O)C1 c1(CNC(c2c(C)nsc2)=O)cc(C)c(C(N2CCN(C3CCC3)CC2)=O)o1 C(=O)(N=c1cc(C)n(-c2nc(C3CCOCC3)ns2)[nH]1)c1nccc(C)c1 C(CCCCCO)(C(=O)NCCSC1CCOC1)N(C1C(OC)COC1)C N1(C(=O)Cc2nncs2)CC23CCCC2(C1)CN(C(C1CCCC1)=O)C3 CCC(C)C(O)C(=O)N1CC(O)CC1CNC(=O)CC(C)c1cnn(C)c1 CC1CCC(NC(=O)Cc2ccco2)CN1C(=O)C(O)CC1CCOCC1 N1(S(CCCC(=O)OCC)(=O)=O)CCc2[nH]c3c(C(=O)OC)cccc3c2C1 C(CCN=C(NCc1ccc(C)c(C)n1)N1CCC(C)C(C)C1)N(CC)CC CCCC(C)CO.C1(CC(=O)N)CCCN(C(C2CC2C=O)=O)C1.C(C)(C)C Cc1cc(C#N)cc(C(N2CC3(CCCC3NC(=O)CN3CCC3)C2)=O)n1 S(=O)(=O)(c1cccc([N+](=O)[O-])c1)N1CCN(C(c2ccnc(C)c2C)=O)CC1 C(C)(C)(CC(=O)N1CC(O)(CNC(C2(C)CCCC2C)=O)C1)OC CCC(O)(CC(=O)NC1(CN(C(=O)CC2CN(C)C2)C)CC1)c1ccccc1 c1(CC)cnc2c(c1)C(NCC(C1CCCN(C=O)C1)=O)CCC2 N1(C(c2cncc(OC)c2)=O)CCC2(CNC(=O)CC3CC3C)CCCCC12 c1(C(N2CCN(C(C(CCC)C)=O)CC2CC)=O)ccc2c(n1)OCC(=O)N2 C1(CNC(C(C(C)C)n2ncc(C)c2)=O)N(C(=O)CS(N)(=O)=O)CCC1(C)C CCCCC1CN=C2C=C(C)N=C(N2)O1.C(=O)(C(C)CC(C)C)NCCCC c1(C(N(CCCN(C(=O)COCP(C)(C)=O)C)C)=O)ccc2ccncc2c1 N1(C(C(C)C)=O)CCCN(C(=O)CC2COC3(CCC3)CO2)CC1C CC1CCC(CO)(NC(c2cc(CNC(=O)CSC3CC3)on2)=O)C1 C1(C(=O)OC)CC(NC(c2ccc(C)s2)=O)C(O)C1 c1(C(N2CCC3(C(C(=O)Nc4nn(CC)c(C)c4)C3)C2)=O)cc(C)cc(F)c1F c1(C=O)cc2c(C)cccc2o1.Cc1nn(C)cc1C(=O)NC1C=CC(C)C1.N C1(CC(=O)N(C2CCN(C(=O)Cc3nnc(C)s3)C2)CC)CC(C)(C)CO1 c1(C(=O)NCC(C)NC(C2CCCN(C(CCC)=O)C2)=O)cccc(F)c1C CC1CCC(NC(=O)CC23CCCN2CCC3)CN1C(c1cnoc1)=O C=CCC(C)N=c1nc(N2CCN(c3nc(O)cs3)CC2)c2[nH]ccc2[nH]1 Cc1ccc(C(N2CC3CCC2C3NC(C2CC(=O)NC2(C)C)=O)=O)cc1C CC1(C)CCCC(C(=O)NC(C)(CNC(C2CCCOC2)=O)C2CC2)O1 C1(C(N2CC(CC)OCC2)=O)CC1C1CN(C(c2cc(C)c(CO)cn2)=O)C1 C(=O)(C(C)(C)CC(F)(F)F)N(C)CC1N(C(c2occ(C)c2)=O)CCOC1 C1(OCC)CC2CC(C(N3CCCC(NC(=O)CC4(O)CCC4)C3)=O)CC12 c1(C(=O)N)ccc([N+](=O)[O-])c(O)c1.C(=O)(CCP(C)(C)=O)N1CCCC(OC)C1 C=CCC(C)(C)CC(=O)NCC1COCCN1C(C1CCCC2(CC2)C1)=O C=CCCCCC(=O)N1CCC(C)(CNC(C2NC(=O)CC2C)=O)CC1 CCCC(O)CC(=O)NC1CCC(N2CCN(C(=O)COC(F)F)CC2)CC1 C1(C(=O)NCCCCOC)CC(c2cc(F)ccc2F)=NO1.C(=O)(CNC=O)N Cc1cc(CCC(=O)NCCCN(C(c2cnc(O)s2)=O)C(C)C)no1 N1(C(C(C(C)C)F)=O)CCOC2(CCC(NC(=O)C(N)=O)CC2)C1 c1(C(N2CCN(C(C(C(=C)C)(C)C)=O)CC2C)=O)cccc(S(C)(=O)=O)c1 c1(CC)nc(C)c(C(N2CCC(CCNC(c3c(C)ncn3O)=O)C2)=O)s1 C1(CC)CN(C(c2csc(CO)n2)=O)CCC1NC(c1cccn1C)=O c1(-c2cc(C(F)(F)F)cc(OC(C)C)c2)ccc2c(c1)OC(C)C2 CN1CCC(C(=O)N)S1(=O)=O.C1(CC)COCCN1C(C1CN(C2COC2)C1)=O N1(C(CCCC)=O)CCN(C(=O)Cc2ccc(O)nc2)CC1CCOC CC1=C(C(=O)NC(C2(CNC(=O)C)CC2)C)CCO1.c1cc(F)ccc1F C1(N(C(CS(CC)=O)=O)C)CN(C(=O)C(=O)NCC2CC2)CC1(C)C CC(C)C(C)C(=O)NC(CNC(c1ccc(-c2nncn2C)cc1)=O)C1CC1 C1(NC(c2c(CC)nco2)=O)(C)CCCCC1C.c1(CC=O)nn(C)cc1Cl.N c1(CC)ccc2occ(C(N3CCCCC3C(=O)NCc3ccccn3)=O)c2c1 c1(NC(=O)NC2(c3ccc(C(=O)OC)cc3)COC2)ncnc2c(Br)cccc12 c1(C(N2CCC(NC(COCCC=C)=O)(CO)CC2)=O)c(F)cc(F)c(F)c1F Cc1c(Cl)ccc(C(C)NS(=O)(=O)CC2CCCS(=O)(=O)C2)c1Cl C12CCN(C1)C2.c1(C(C(=O)NCCCF)N(C)CC)nnc(C2CC2)s1 N1(C(Cc2nc(C)[nH]n2)=O)CCC2(CCC2NC(c2cc(C#N)cn2C)=O)CC1 C(C)(CCC#N)(c1n(CC(=C)C)nnn1)NCC(C)Oc1cccc(Cl)c1 C1(NC(CS(C)(=O)=O)=O)CN(C(c2cc(F)c(N)cc2F)=O)CCC12CCC2 c1(CC(=O)OCC)ncc(C(F)(F)F)s1.c1cnc(CNC(C)CC)s1 C1(C(N2CC3C(C(N(CCO)CC)=O)C3C2)=O)CCC2CCC(=O)N2C1 C1CN(C(=O)C#CC(=O)N(C)C)CCN1C(c1cc(C(C)C)oc1C)=O.COC c1(C(=O)NCC(CC(C)C)(C)NC(=O)Cn2cccn2)cccc2cc[nH]c12 Cc1cc(NC(=O)C(O)Cc2cnc[nH]2)ccc1NC(=O)Cc1csc(=N)[nH]1 c1(CNC2CCC(C(N3CCN4CCOCC4C3)=O)C2)ccc(Br)c([N+](=O)[O-])c1 N1(CCOC)CCCC(C(C)NC(C2CC(CNC(=O)CO)C2)=O)C1 C(=O)(C1=Cc2cc(Br)ccc2OC1)N(CCNC(C=C(CCC)C)=O)C1CC1 c1(C(=O)NC2(C)CCN(Cc3ccccc3C#N)C2)ccc2c(c1)CCC2 c1cnc2cc(F)c(F)cc2n1.CCCC(C(=O)NCC1(N)COC1)NC(N)=O Cc1c(C(=O)NC(C)CCNC(=O)CCc2cscn2)cccc1[N+](=O)[O-] C1(NC(c2ccc(Cc3n(C)ncc3)cc2)=O)C2Cc3ccc(Br)cc3C12 N1(C(C2(CC)CCOC2)=O)CCC(C)(NC(c2ccc(C)cc2)=O)C1 CCC1=CCN(C(C23CC(CO2)C3)=O)CC1.c1(NC(C)=O)cc(C(=O)N)ccn1 C1(CC(=O)NC2(CCOC)CC2)CC=CCC1.S(C(F)(F)F)CC=O.N N1(C(CC(CC)C)=O)CCC(C(=O)Nc2ccc(OC)c(O)c2)C(C)(C)C1 C12(NC(=O)CCC3CC3(F)F)CCC(CC1)C2.c1(C(=O)N)ccc(Cl)c(F)c1 C12(CNC(C3CNC(=O)N3)=O)CCCC1N(C(c1cncc(F)n1)=O)CCC2 C(=O)(CN=c1[nH]c(C)cs1)NCC1N(C(c2cncc(C#C)c2)=O)CC1 CC(C)C(C(=O)N1CC(NC(C2CNC(=O)N2)=O)C1)NC(N)=O c1(C(=O)NCC(CC(=O)NCC(CCCC)CC)O)n[nH]c2ccccc12 c1(C(N(CC(C)NC(C2CC2C2CCOCC2)=O)C)=O)cc(O)c2sccc2c1 CCC(O)C(F)(F)C(=O)NC(C)CCN(C)C(c1cnc2n1CCS2)=O N1(C(c2cc(C)ncc2)=O)CCCC2(CNC(C3CCC(=O)N3)=O)CCCCC12 CC(CF)CC(=O)NCC(C1CCCN1C(c1ccnc(S)c1)=O)(C)C c1(CNC(=O)NC(C#C)CC2CC2)ccc(O)cc1F Cc1ccc(C)c(S(=O)(=O)NC(=O)CC(C(=O)C(C)(C)C)c2ccccc2)c1 C1(CC(=O)OC)(NCc2ccc(O)cc2Br)CC2CCC1C2 c1(C(=O)NC2CCCCN(C(CC(CC)C3CCC3)=O)C2)ccc(S(C)=O)cc1 N1(C(C(C)(Cl)Cl)=O)C2CCC1CN(C(=O)Cn1nnc(C(C)(C)C)n1)CC2 c1(CN(C(=O)C(C)(F)F)C)cnn2c1CN(C(=O)CC(O)Cc1ccccc1)CC2 Cc1cc(C(N2CCC(C3CCCN3C(C3CCC(CO)CC3)=O)C2)=O)nnc1O N1(CCC(=O)NC2(C(F)F)CCOCC2)CCC(O)CC1 c1(NC(CC(C)N(C(CCCOC(C)=O)=O)C)=O)ccc(Cl)nc1 N1(C(C2C(C(C)C)C2)=O)CCC(OCCNC(C2(F)CC2(F)F)=O)CC1 c1(C(=O)NC2CC(NC(C=CC(CC)C)=O)C2)cc(Cl)sc1.C(C)=O.N Cc1cc2n[nH]cc2cc1C(=O)NCC=CC.C1(CC=O)COC(C)(C)C1.N C1(CCNC(CC(C)SC)=O)CCCCN1C(C12CC(C(C)C)(CO1)C2)=O C(CCCNC(C1CC(SC)C1)=O)OC.C1(CC(=O)N)(N(C)C)CCCC1 C(=O)(CCCCCO)N1CCCC(NC(C2(c3ccc(Br)cc3)CCCC2)=O)C1 C1(OC(N(C2CCNCC2)C)=O)CCCC(CNC(=O)C(F)(F)F)CC1 CCCCCCCCCC(=O)N1CC(OCCNC(C2CC(CC)C2(C)C)=O)C1 Cc1csc(C=CC(N2CC(NC(=O)C(F)C3CC3)C(c3ccccc3)C2)=O)n1 c1(C(=O)NC2CCN(C(C(C)C3CCOC3)=O)C2(C)C)ccc2nc(O)oc2c1 C1(C(N(C2CCC(NC(c3ccc(C4CC4)cc3)=O)CC2)C)=O)CC2CC1CO2 C1(C(=O)N)CCCC2(CC2)C1.C(CC)(C(=O)NCCCN(CCCC)C)=CC C1(NC(N)=O)CCCN(C(c2occc2C2CC2)C(=O)NC2CCCC2)C1 N1(C(C(=O)NC2CC2)=O)CC2C1CCCN2C(c1ccccn1)=O CN1CC=C(CCN=C(NCC2CNC(=O)O2)NC(C2CC2)C2CC2)CC1 c1(C(C(=O)NCCNCC)N(C)CCOC)cc(F)cc([N+](=O)[O-])c1C c1(OC)cc(OC)cc(CC(CNCC2CNCCO2)CO)c1 Cc1c(C(N2CC(CC(C)NC(C3CCOC3)=O)C2)=O)cnc2ccccc12 N1(C(c2cc(OC)ns2)=O)CC2CN(C(=O)C(C)N(C)C)CC2(C)C1 n1(C(CC(=O)N(CC=C)Cc2cccc(OC)c2)C)cnc2ccccc12 c1(-c2c(C)occ2)cc(=NC(=O)C(=O)Nc2cc(Br)cc(I)c2)[nH][nH]1 Cn1ncc(C(=O)NCC(C2CC(F)(F)C2)O)c1-c1ccccn1 N1(C(COCCCCC)=O)CCC(C(C)(C)NC(c2sncc2CC)=O)CC1 c1(-c2nn(CC(C)C)c(Cc3ccccc3)n2)cc(N2CCCCC2)cc(F)c1 C(=O)(CCC(c1nnnn1CC1CC1)NC(C)(C)CCO)OC C1(C(=O)NC(C)Cn2cncn2)C(C)OCCN1C(=O)CCCC1CC1 c1(OC)cnc(F)c(C(=O)N(CC(O)CNC(C2(C#N)CCCOC2)=O)C)c1 Cc1cc(=O)n(CC(N2CC(C(=O)O)CC2(C)C)=O)c(=O)n1-c1ccccc1 C(C(CO)C(F)(F)F)NC(C(CNC(c1cnn(C)c1Cl)=O)CC1CCCC1)=O Cc1nc2ccc(C(N3CC(CCCCNC(=O)C(C)SC(C)C)C3)=O)cc2[nH]1 Cc1ncnc(NC=O)c1C.c1cccnc1.C12CN(C1)C(=O)C(C)OC(=O)C2 N1(C(C(CC)C(C)(F)F)=O)CCCC2CN(C(C3CCN3CC)=O)CC12 c1(NC2C(C)CN(C)C2)ncc(S(=O)(=O)NCc2ccc(Br)o2)cc1Cl C1(C(=O)NC(CCOCC)CO)CCCN(CC(F)(F)F)C1=O C1(NC(=O)Cc2ccnc(O)c2)CCCCC12CCN(C(C1(C(F)F)CC1)=O)C2 c1(C(=O)NCCC(C)NC(=O)CCCC(C)(C)C#N)c(Cl)oc2ccccc12 Cc1cc(C)c(C(N2CC(C)N(C(=O)C(O)CF)CC2C)=O)cc1Br c1(CC(=O)NCCN(C(C)C)C(C2CC2C2CC2)=O)ccccc1Cl c1(C(=O)NC2CC(NC(=O)CCCc3ccccn3)C2)snc(O)c1Cl N1(C(COCCCCC)=O)CCCCC(CNC(=O)C(O)C(C)(C)C)C1 C1(OC)(CNC(C2CC2F)=O)CCN(C(=O)CCN2CCC(O)CC2)C1 C(=O)CC(C)C(C)(C)C.c1(C(CC)=O)ccc(C(=O)NC2(C)CCOC2)cc1.N Cc1ncc(CNC(=O)CC(C2CC2)NC(c2ccnn2CCF)=O)[nH]1 C1(NC(CCC#C)=O)CCN(C(=O)C(C)Sc2ccccc2)C12CC2 C1(C(N2CCCCC(NC(c3ccc(C)s3)=O)C2)=O)Cc2ccc(F)cc2O1 N1(C(c2cccc(C)c2O)=O)CCCC2C(CCCN2C(c2cnnn2C)=O)C1 N1(C(c2nc(COC)sc2)=O)CCC(C(F)F)C1.C(=O)C=O.CC(F)(F)F c1(CC)cncc(NC(c2ccc(CC)s2)c2nnnn2CC2CCOCC2)c1 CN1CCOCC1C(=O)NCCCN(C(=O)C(O)C1CC1)Cc1cccnc1 C(=O)(CC(F)(F)C(F)F)N1C(CC(N2C(C)CN(C3CC3)CC2)=O)CC1 C12(CC=O)CC3CC(CC(C3)C1)C2.C(CC(=O)NCC#CC)OC.C(=O)C c1(C(=O)NC2CCCN(C(c3cc(C(N)=O)co3)=O)C2)ccc2nccnc2n1 N1(C(C2(C(N)=O)CC2)=O)CC(C2CCN(C(=O)Cc3cc(O)nc(O)n3)CC2)C1 c1(C(N(CCC(OC)OC)C)=O)ccc(-n2cc(Br)cn2)c(F)c1 C1(CNC(c2c(OC)nsc2)=O)CN(C(=O)CC(C)C(C)(C)C)CC12CCC2 CC1C(NC(C2C3CCC2(c2ccco2)C3)=O)CCCN1C(=O)C1=CCCC1C N1(C(C2CCN(C(c3nn(C)c(F)c3)=O)CC2O)=O)CCn2nncc2C1 C(CN=c1cc(C(N)=O)nc(Cl)[nH]1)(C1CC1)NC(C1(C)CCC(F)(F)CC1)=O CCCC(C(O)C(=O)NCC1CC(C)(O)C1)NC(=O)C(CC)(CC)CC c1(C=O)c(C)[nH]c2ccc(O)cc12.C1(CNC(C=CCOC)=O)CCCCC1 CC(C)C(CCNC(C1CCS1(=O)=O)=O)NC(=O)C=Cc1ncc[nH]1 c1(SCCOC)nccnc1NC(=O)CCCC1CN(C=O)C1.C(C)(C)C CN(CC(F)(F)F)NC(=O)COc1ccc(S(C)(=O)=O)cc1 c1(C(N2CCC(N(C)C)CC2)C(=O)NC(CC)C)cccc(OC)c1F C1(C(=O)NCCCC(C)NC(c2ccc(C(N)=O)[nH]2)=O)CCC(=O)N1C N1(CC(C)(C)NC(C=C(C)C(C)(C)C)=O)CCN(C(C2CCC2)=O)CC1.C c1(C(N2C(CNC(C(C)(C)C3CCC3)=O)CC2)=O)ncc(Cl)cc1Cl C1(CN(C(=O)C(C)(C)C2CCOCC2)C)CCN(C(=O)Cc2ncc(Cl)s2)C1 c1(C(N(C(C)C(=O)N(CC(C)(C)C)C)C2CC2)=O)cncn1C1CC1 c1(NC(C2N(C(CC(CC)C)=O)CSC2)=O)ccc(C)c(OC)c1 c1(NC2(C)CCC2)ccc([N+](=O)[O-])cc1C(F)F.C1(CC=O)COC(C)(C)C1 N1(NC(C=C2CCC(C)C2)=O)CCC(CC2CCCN2C(=O)C2=CCSC2)CC1 C(=O)(C(C(=O)NCC(C)(C(C)C)NC(=O)Cc1c(C)noc1C)OC)OC Cc1ccc(C(N2CC3CC2(CNC(C2CCCC(F)C2)=O)C3)=O)nc1C Cc1nn(C)c(C)c1C(C)C(=O)NC1CCCCN(C(c2cccc(=O)o2)=O)C1 c1(C(=O)NC2CCN(C(C3C(=C)CC3)=O)C2C)cc(Br)cc2nc[nH]c12 C1(O)(C(C(=O)NCc2cc(O)cs2)F)CN(C(C23CSCC2C3)=O)C1 CC1CCCC(CC(=O)NC2C=CCN(C(=O)C(F)=CC3CC3)C2)O1 N1(C(CCC#CC)=O)CCCC(C)(CNC(C2CCCN2C=O)=O)C1 Cc1ncnc(N2CCC(CNC(=O)Cc3cnn(C(C)(C)C)c3)C(C)C2)c1F CCC(C)CCC(=O)N1CCC(NC(c2n[nH]cc2Cl)=O)C1C(C)C C1(NC(=O)C=CBr)CCN(C(C2Cc3nncn3C2)=O)CC12CCC2 CON1CCC(CC(=O)NC(C)(C)CCCNC(c2cc(C3CC3)ns2)=O)CC1 C(=O)(CCCC1CCOCC1)N(C(c1ccccc1)CNC(C1(CO)CC1)=O)C O=C1NCCC2CCCN(Cc3c[nH]nc3-c3ccccc3F)C12 c1(OCC(CNC(=O)NC(C(C)C)C2(C)CC2)O)ccc(Cl)cc1 C1(C#N)(CN(C(C=CC(C)NC(c2cc(Cl)ns2)=O)=O)C)CCC1 N1(C(C(CCC)Cl)=O)CCC2(CC(C(=O)Nc3ccc4nccn4c3)=NO2)C1 O=C(C1CCOc2ccc(Cl)cc21)N1CCCCC1C1CCN(C(C2(F)CC2)=O)C1 c1(C(=O)NC2CN(C(C3=NOC(C)C3)=O)C(C)CC2)cc2ccc(Cl)nc2s1 c1(C(=O)OC)nc(Cl)c(NCC(CO)C(C)(C)C)nc1N C1(NCCS(CCC)(=O)=O)CCC(O)CN(Cc2ccccc2)C1 C#CC1(C)CCCN(C(C2CN(C(=O)CN(C3CCC3)C)CC2OC)=O)C1 N1(C(c2cc(C)c(Cl)s2)=O)CC2CCC1CN(C(c1cc(CO)[nH]n1)=O)C2 C(=O)(N=c1[nH]c(Cl)ncc1C(=O)OC)C1CCCC(OC)C1 C1(F)(C(=O)O)CCCCC1.CC1C(NC(=O)C2CC2)C1C Cc1csnc1C(=O)N(C)CCOCCC(=O)N1CCC1C(N)=O C1(CC)(CN(C(=O)CC2CCC2)C)CCCC1.c1(C=O)ccn(CCF)n1.N c1(C(N2C(C)(C(=O)NCC3CCC(F)C3)CCC2)=O)cccc(Cl)c1[N+](=O)[O-] c1(CN2C(C(=O)Nc3cccc(OC)n3)CC(O)C2)c(O)cc(O)cc1O CCC(CNC(=O)C(F)C1CC1)(CC)NC(=O)CC1CCN(C)C1=O Cc1cc(O)cc(O)c1C(=O)NC1CC(C(=O)NC(C)C)C1 C(CCC(C)C)NC(C(n1cc(C)nc1)(C)C)=O.C(=O)(C(F)(F)CC1CC1)N c1(C(N2CCN(C(c3c(CC)ccs3)=O)C3C2C3)=O)ccc2c(c1)COC2(C)C C12(CNC(C(CSC)O)=O)CC1CN(C(=O)C)C2.c1(C=O)cc(Cl)ccn1 C12(C(=O)NCC3(C)CCCC3O)CC(CO)(CN1C(=O)CCc1ccoc1)C2 C=CCC(C)(C)CC(=O)NC12CCCN(c3nnc(C4CC4)o3)CC1C2 C1(C(C)C)CCC(C(N2CCOC(CN(C(=O)C(C)(C)F)C)C2)=O)C(=O)N1 Cc1cc(F)c(C(N2CCC(C(=O)NC(C)C)C2)=O)cc1S(C)(=O)=O C(CC)(CC(=O)N(C)C)NC(CCN(C(C(C=C)O)=O)CCO)=O N1(C(CCC(C)SC)=O)CCC2CCCC12C(N1CCCC(C)(C(N)=O)C1)=O C1(NC(CSC)=O)CCN(Cc2nn(C)cc2Br)C(C)C1 C1CN(C(C23CC(C)(C2)OC3(C)C)=O)CC(C)(C)O1.C(C(=O)N)=C(C)C.C C1(C(=O)NCCCN(C(C(CC)C)=O)CCO)CCC(=O)N(C2CC2)C1 C1(CNC(C2C(NC(COCCCOC)=O)C2)=O)CC12CC2 c1(OC)cccc(C(=O)NC23CC2CN(C(C24CC(C2)C(C)O4)=O)C3)c1 Cc1cc(C)c(CNC(C2(C)CCN(C(c3cnccc3C)=O)C2)=O)s1 C(=O)(CCCC(C)(C)C)N1CCCC(N(C(c2csc(F)c2)=O)CC)C1 c1(N(c2cccc(Cl)c2)CC(=O)NC(c2cccnc2)C(C)C)ccc(F)cc1 N1(C(C(CC(C)C)ONC(c2ccco2)=O)=O)CC2COCC(C2)C1 c1(C(C(=O)NC2CC(NC(CCN(CCC)C)=O)C2)OC)ccc(OC)cc1 c1(C(=O)OC)ccc2nc(NC3(C)CC3)sc2c1.CC(C)(C)C.C(=O)C.N C(C)(C(=O)NC(C)CCC1CCCC1)N(C(COCCC=C)=O)CCC c1(OC)c(CC(=O)NC2CN(c3ncnc(Cl)c3C(C)C)C2)cccc1C#N C1(CNC(CCn2c(C)ncc2)=O)C2CC1N(C(c1cnn(CCO)c1)=O)C2 c1(CN(C)Cc2cccc(OCCOC)c2)ccccc1O.C1COC(=O)N1 N1(C(C(CC2CC2)OC)=O)CC(C(=O)NC(c2cn[nH]c2)C)C2(CC2)C1 C1(C(N2C(C(C)NC(C3CCCCC3)=O)CCCC2)=O)CC(=O)CC(=O)N1 C(C)(CSC)(C(=O)N(CC(F)Cl)C)NC(CC=CC)=O C1(CC(N2C(C(=O)Nc3c(OC)noc3C)CSC2)=O)CC2(CCC2)CCO1 c1(CC)nnc2c(C(=O)NC(C)C)cccn12.C(=O)C[SH](=O)=O.C(C)(C)C N1(C(C(=O)NC(C)C)=O)CCCCC(CNC(=O)C(c2ncccc2F)(F)F)C1 CC1CN(C(c2cc(-c3cccs3)[nH]n2)=O)CC1NC(C1(C)CC1)=O c1(CC2CC2)ccccc1.C(=O)(CCC)NC(C1(COC)CCC1)=O.C c1(C(N2CCC(O)(CNC(C(C)n3ccnc3)=O)CC2)=O)nccn2ccnc12 C=C=CC(C)C(=O)NCC12CC(CN1C(=O)CCc1nc(CCC)no1)C2 CC(C)(CC(=O)NCC(=O)NC1CCOC1)n1cc(CN2CCCCC2=O)nn1 CCCCC(CNC(C)=O)NC(C1CC2(CC2)C1)=O N1(C(=O)CC2CC(OC(F)F)C2)C2CCC1CC(CNCc1ccc(Cl)cc1)C2 C1(N(C(C=NOC)=O)CCO)CCCN(C(=O)COc2ccc(F)nc2)CC1 N1(C(c2cc(COC)sc2)=O)CCCC12CCN(C(c1cc(C)ccn1)=O)C2 C#CC(C)(CC)NC(=O)C=C(C)CNC(=O)Cn1cc(C2CC2)cn1 Cn1ncc2ccc(CN=c3[nH]cc(CCNC(=O)Cc4cncnc4)s3)cc12 N1(C(C(CC#C)C)=O)CCc2nc[nH]c2C12CCN(C(=O)OC(C)(C)C)C2 O=C1CCC(CC(=O)NC2(C(N3CC4CC4C3)=O)CSC2)O1 Cc1ccc(C#N)cc1C(=O)NC1CCCCN(C(C2CCCC2O)=O)C1 C(CCCCC(=O)NC(C(=O)NCC1(C)CC(F)(F)C1)C(C)OC)=CC C(=O)(C1=NOC(C)C1C)NCCC1CCN(C(C2(CSC)CCC2)=O)C1 c1(C(N2CCC(F)(CNC(C(COC)O)=O)C2)=O)cc(C(C)C)nc(O)c1 CC1CCC(NC(=O)NCc2cccn2Cc2ccccc2)CN1 C1(C(N(CC(N2CCC(CC(C)(C)C)C2)=O)CC)=O)CC(=O)C12CCC2.CO C1(C(N(CC(C)C)CCC)=O)CCCN1C(=O)C(C)c1cc[nH]n1 C1(C(=O)NC2(C)CCN(C(Cc3cc(OC)no3)=O)C2)CCC12CCOCC2 c1(C(N)=O)ccccc1OCC(=O)N.C1CC2(C1)CC2.n1(CC=O)nccn1 C1(NC(=O)C(F)=C2CCC2)CCN(C(=O)CS(=O)(=O)CC2CCCO2)CC1.C C(=O)(C1CNc2ccccc21)N1C(CNC(C(C=CC)O)=O)C(C)(C)CCC1 C1(Nc2cc(NCC(c3ccc(F)cc3)(C)C)nc(C)n2)CCC(=O)N(C)C1=O Cc1cc(F)c(C(=O)NC)c(F)c1.C1CN(C(=O)C(C)C(C)(F)F)CCC1(F)F C#Cc1cncc(C(=O)NCC(C)(C)CNC(=O)C(C)C(F)F)c1 N1(C(c2ccc(C)s2)=O)CCC2(CC1)CCN(C(=O)CCC1(C)CCC(=O)N1)C2 C1(C)(CNC(C)=O)CCN(C(C2CN(C(c3cc[nH]c3C)=O)CCO2)=O)C1 Cc1cc(CC(=O)NC2CCCC(C(=O)NCC(C)(C)n3cccn3)C2)n(C)n1 CC(O)C(C)(C)C(=O)N1CCC1(C)CC(=O)N(C)CCc1nccs1 C1(NC(CNS(N)(=O)=O)=O)CCC2CCN(C(=O)COc3ccccc3F)C1C2 C1(NC(c2n(C)ccc(=O)c2)=O)CC12CCN(Cc1cc(Br)ccc1F)CC2 c1ncccc1.n1(C(C=O)C)ccc(C(F)(F)F)n1.C(C(=O)N)NC(C)=O.C C(CN=c1[nH]c2c(c(=NCC3(C4CC4)CCCCC3)[nH]1)CCC2)C1CCCCC1 C1(NC(C(C)n2cncn2)=O)C2CN(C(c3cccc(C4CC4)n3)=O)CC12 Cc1cc(O)c(C(=O)NC2C3CN(C(c4ccc(F)cc4O)=O)CC23)nn1 CC1(C)CN(Cc2csc(-c3cccs3)n2)CCC1NC(=O)Cn1cnnc1 N1(CCCC=CCC=C)CCC(C(=O)NCc2cccc(N)c2)CC1 C1(NC(c2cc(C(C)NC(C3C=CCS3)=O)on2)=O)COCC(C)(C)C1 C1(CN(C(=O)CCCc2cncs2)C)CCCN(C(=O)COC(C)(C)C)C1 c1(C(=O)NC2CN(Cc3cnc(C)s3)C(C)CC2)cc2cc(C)c(C)cc2o1 c1(C(=O)NCC2(NC(C(C(=O)OC)C)=O)CCOC2)ccc2cnoc2c1 C(=O)(C(CC(C)C)C(C)C)NCC(C(=O)Nc1c(C)ncc(C)c1)C(C)(C)C c1(-n2c(CCCOC)nc(CN3CCCCC3)n2)cc(F)cc(F)c1 C1(C2CCOCC2)(C(N2CC3CCC(C2)N3C(c2cn3c(n2)COCC3)=O)=O)CC1 c1(OC)cccc(C(C2COCCO2)NC(=O)C(=O)NC)c1.c1ncc[nH]c1=O C1(CC(=O)N(C(C)C(F)F)C)CC(NC(=O)CN(C2CCC2)C)C1(C)C CC1CCCCC1C(=O)NC1CCC1NC(c1ccc(COCC)cc1)=O C1(C(=O)NC(CC)CNC(=O)C=Cc2ccccc2)C(O)C(=O)N(C)C1C n1(C(C(=O)OC)C)nnnc1C(COC)NCc1cnoc1 c1(CN2C(C(N3CCCC3(C)C)=O)CC(=C)C2)cc(Br)cnc1OC CC(C)C(CO)C(=O)NCCC1CCCCN1C(c1cn(C2CC2)cn1)=O CCC(CC(F)(F)F)C(=O)N1CC2(C1)CN(C(=O)CCS(C)(=O)=O)C2 N1(C(C(CCCNC(CCN(C)CC)=O)O)=O)C2CCC1CC1(C2)N=N1 C1(C(N2CCCC(NC(C3CC(C)SCC3)=O)CC2)=O)C2CC3CC(C2)CC1C3 C1(NC(C2C(NC(=O)Cn3ncnn3)COC2)=O)CC2CC2C1 CC(O)(C(=O)N1CCN(Cc2cscc2Br)CC1Cc1ccccc1)C(F)(F)F c1(C(=O)NC(CCCNC(C(CC)CC)=O)C)cc2ccoc2cc1F Cc1cc(Cl)ccc1S(=O)(=O)NCCOCCN=[N+]=[N-] C=CC(CC)CC(=O)N1CCC=CC1C(=O)NCc1cc(C)c(C)s1 N1(C(C(C(C)C)C)=O)CC=C(C(=O)NCCC2C=CCC2)CC1 C1CCCN(C(c2cn(CC(=O)OC)nn2)=O)C1.c1(N)scnc1C(C)(C)C N1(C(Cn2ncc(C)c2)=O)CCC(C2CN(C(=O)CC3C=CCC3)C2)CC1 C1(NC(CC)=O)CCN(C(=O)CCS(N)(=O)=O)CCC1c1ccccc1 C(=O)(C1CCCc2ncccc21)NCCN(C(=O)C(C)(C)N1CCCC1)CCC N1(C(C2C(C)(C)CCC2)=O)CCCC(C)(NC(=O)Cc2csc(NC=O)n2)C1 Cc1nc2cc(CN3CC(O)CC3C(=O)NCc3cc(C#N)cs3)ccc2s1 N1(C(C2C(C)(CC)C2)=O)CCN(C(=O)Cn2nc(C)oc2=O)C(C(C)C)C1 N1(CC=O)C(=O)c2ccc([N+](=O)[O-])cc2C1=O.C1(CC=O)(OC)CC1.CC.N N1(C(C2C(C)(C)C2(C)C)=O)CCc2sc(C)nc2C1.C(c1nccs1)=CC=O.N c1(NC(C)=O)sc(Cl)cc1C(N1CCC1)=O.C(=O)C(C(C)C)c1cccnc1.N c1(CC)n[nH]cc1C(=O)NCC(C(=O)NC1CC(O)C1OC)N(C)C C1(OC)CC(NC(=O)N(CCn2cc(CO)nn2)CC)C1(C)C Cc1cc(N2CCC(C)C2C(=O)NCc2ccn(C)c(=O)c2)n2nc(C)nc2n1 C=C(Cl)CCC(=O)N1CCC(CNC(c2n[nH]c(C3CC3)c2Cl)=O)C1 c1(C(NOC(C)C)=O)nn(-c2cccnc2)c2c1CCCCC2 C1(NC(=O)Cc2nc[nH]n2)CCCN(C(c2cccc(C(C)(F)F)c2)=O)C1.CC C1(C(N2C(C)CC2CO)=O)C2CCCC2CN1C(=O)C=Cc1ccnn1C CCC(CNC(=O)COC1CC(NC(=O)C(CCOC)OC)C1)C(C)C N1(C(C(=O)NC(c2ncc(F)cn2)C)=O)CCN(C(=O)O)CC1C.C(C)(C)C C1(CCOC)(C(=O)N)CCN(C(=O)CC(F)(F)Cl)CC1.c1(CC)nc(C)oc1C Cc1nn2cc(C(=O)NC(C)C(C)NC(=O)CCC(=O)O)nc2s1.C(C)(C)C C1(CC=O)OCCC1(C)C.c1(COC)noc(C(C)NCCC)n1.C(C)=O c1(-c2c(C(N3CCN(C4CCCC4)CC3)=O)scn2)ccnc(N2CCCC2)n1 Cc1nc2n(n1)CC(Nc1ncc(-c3ccc(F)cc3)s1)CC2 C#CCC(C)(CC)C(=O)NCCCC1(NC(=O)Cc2ncc(CC)[nH]2)CC1 Cc1nc(CNC(=O)CCN(C)C(c2cocc2C(N)=O)=O)c(C)s1 N1(C(CC(c2c(C)noc2C)C)=O)CCCC(CNC(N)=O)CC1 C1(C(=O)NC2C3(CC(NC(c4cnc(C)nc4)=O)C3)C2)CN=C2N=CNN2C1 c1(C(=O)NC2CC(C)(CNC(C3CC34CC4)=O)C2)c(F)cccc1Br C1(C(N(C(C2CCOCC2)C)C)=O)CCN(C(C2CC(=O)N(CCC)C2)=O)CC1C [nH]1cc(C(=O)N)c(C(C)(C)C)n1.C(C)(C(C)C)NC(C1C(CC)C1)=O C(=O)(C1=NNC(=O)CC1)N(CCC1CCN(C(c2cc(CC)ncn2)=O)CC1)C CC1Cc2cccc(C(N3CCC(NC(=O)CC4=CCCC4)C3C3CC3)=O)c2O1 Cc1ccc(OCC(N2CC(CC(C)NC(C3(C)CC3(Cl)Cl)=O)C2)=O)cc1 C1(OCC#C)CCN(C(C2CC(NC(=O)CCCC3CCCO3)CCO2)=O)CC1 N1(C(CCC(=O)c2cn(C)nc2)=O)CC2(CCN(C(C34CC(C3)C4)=O)C2)C1 c1(OC)ccc(CC2(C(=O)OCCC(O)CO)CCCCO2)cc1 C12(NC(C=Cc3cncc(C)c3)=O)CCCC1N(C(=O)Cc1cccs1)CC2 N1(C(c2ccc(I)s2)C(=O)NC)CCC(CCF)CC1 c1(SCC)cc(C(N2CC(CO)(NC(=O)COC(F)(F)F)C2)=O)ccn1 N1(CC(N2CCC(CCNC(C3(C)C=CCCC3)=O)C2)=O)CCC(=O)NC1=O c1(C(=O)NCC(CC)NC(c2c(Cl)nsc2Cl)=O)cnc2c(c1)CCCC2 C(=O)(CN=C1NS(=O)(=O)c2ccccc21)N1CC=CC1.C(C(O)C(=O)NC)OC C=CC1(C(=O)NCC2CN(C3CC3)C2)CCN(C(=O)CCc2cccn2C)C1 CCCC(C)(CC)NC(C1(C(C)C)CCN(C(c2cc[nH]c2C)=O)C1)=O C(=O)(CC(C)(C)C(C)(F)F)N1CC(NC(C2N(C(CC(C)C)=O)CCCC2)=O)C1 c1(CNC(C(C2CCN(C(=O)CN3CCOCC3)C2)C)=O)cc2n(n1)CCO2 C1(NC(CC2CCCC(C)C2)=O)CCC(C)(N=c2ccnc(C3CCC3)[nH]2)CC1 N1(C(CC2(N(C(=O)CCC3CCC(=O)C3)C)CC2)=O)C2CSCC1C2 c1(C(=O)Nc2c(OC)nn(C)c2)nnn2cc(-c3ccccc3)nc(O)c12 N1(C(C2N(C(c3c(C)non3)=O)CCC2O)=O)CCC(F)(F)CC1 C1(C)(CNC(C(C)(C)OC)=O)CCN(C(=O)C(C)SC)C1 N1(C(c2cc(OCC)ns2)=O)CC(NC(c2csnc2C)=O)CCC1C c1(NC(CC)CNC(C2C3CCCCCCC23)=O)nnc(C)c(C)c1C#N C1(NC(c2cn[nH]c2)=O)CC(F)(CNC(C2CCCSC2)=O)C1 CC(CCC(=O)N(CC(C)(C)C)C)S(C)(=O)=O.c1(C(=O)N)nc(O)nc(O)c1N c1(CC(N2CCC(CC(=O)NC(C)Cc3nn[nH]n3)C2)=O)nccn1C c1(C(=O)NC2(C)CN(C(=O)Cn3nccn3)C2)cc(Br)c(=O)n(O)c1 C1(CCNC(C(C)SCCCC)=O)CN(C(c2cccnc2NC)=O)CC1C N1(C(c2cc(C)on2)=O)CCC2CCCC12CNC(=O)Cc1nonc1C Cc1cc(N(C)CCNC(=O)CC2CCC=CCC2)c(C(F)(F)F)cc1[N+](=O)[O-] Cc1nc(C)c(CC(=O)NC23CC(C2)N(C(c2ccc(NC=O)cc2)=O)C3)s1 N1(C(CN2CCCC(F)(N(C)C)C2)=O)CCC2(CCSCC2)CC1 c1(CNC(CC)=O)cn(CC2C(C)C2(F)F)nn1.c1(C(=O)N)ccncc1 Nc1ncnc2c1ncn2CC(=O)Nc1cnn2ccncc12 N1(C(C(N2C(=O)CCC2=O)C)=O)CCCC(CNC(c2cccnc2S)=O)C1 C1(NC(C2CC2)=O)CC12CCOCC2.C12CC(C1)CN(CC(C)C)C2=O CCCCC(C(=O)NCC(C1CC(C)(C)C1)O)NC(=O)C(C)S(N)(=O)=O c1(NC2CCC(OC)CC2)ncc(C)cc1S(=O)(=O)NCC(=O)NC(C)C N1(C(C(CCC)(C)C)=O)CCCCC12CC(NC(=O)C(C)COC)C2.C(C)(=O)N CCC(C)(C)C(C)CC(=O)NCCC1CN(C(C2CC(C)(F)C2)=O)C1 N1(C(C(CCC)n2cccc2)=O)CCc2cc(OCC)c(Cl)cc2C1 C(=O)(N=c1cc(C)[nH][nH]1)c1ccc(-c2cccc(OCCC)c2)nc1 N1(C(CCCCOC)=O)CCC2(CCCN2C(c2ncc(Br)cn2)=O)C1 CCCN(OC)C(=O)C1(CNC(=O)C(C)CC2CCCO2)CCC1 N1(CC#C)CCN(C(=O)CCN(C(=O)C(F)C(C)(C)O)CCCO)CC1=O S(=O)(=O)(CCC(=O)NCCC1CCC1)NC.c1(C=O)cccc(C=O)c1.N C(=O)(CCCCCC=C)NC1CCN(C(Cn2ncc(C#C)c2)=O)C12CC2 CN1CCn2ncc(C(N3CC4CC(NC(=O)Cc5cnc[nH]5)C3C4)=O)c21 C1(NC(C2C(C)=C2)=O)CN(c2ncccn2)CC12CCOCC2 c1(CC)ccc(C(=O)NC2CC2C=O)cc1.C(=O)C(O)Cc1cnc[nH]1.N CC1=C(C(=O)N2CC3(COC(CNC(c4cc(Cl)no4)=O)C3)C2)CCCC1 c1(COC)ncc(C(=O)NCC(CO)NC(c2n[nH]cc2C)=O)s1 Cc1ncc(C=CC(=O)N(CCC)C)c(O)n1.C(=O)(C(C)(C)C1(O)CCC1)N N1(C(C=C(C)CNC(C2CCCCC(=O)C2)=O)=O)CC(C)C(C)C1C C(C(O)CC(=O)N1CC=CCC1C(=O)NCC1CC(F)(F)CO1)N(C)C C1(C)(C(=O)NC2(C)CCN(C(c3cnc(C4CC4)nc3O)=O)C2)CCCNC1=O C1(N(C)C(c2cc[nH]n2)=O)CN(C(=O)C(C2CCCCC2)O)CCC1O N1(C(c2c(C)cn(C)c2)=O)CCC(C)(C)C1C(N1CCCCC1CC(N)=O)=O N1(C(c2c(C)noc2C)=O)CCC(NC(C2CC(N=[N+]=[N-])C2)=O)C(C)(C)C1 N1(C(c2n3c(nn2)SC(=C)C3)=O)CC2CCC1C1CN(C(=O)C(F)F)CC21 c1(C(C)N(C(c2cccc(I)c2)C(=O)NCC(F)F)C)ccccc1Cl.C1CC1 C1(CC)CN(C(=O)COc2ccccc2O)CCN1C(=O)C(C)(C)c1cc[nH]n1 C1(C)(CNC(Cc2c(C)nccc2)=O)CC(F)(F)CN1C(C1CC1F)=O c1(C(=O)NCCC(C)N(C(=O)CC2CCC(=O)N2)C)cc(C(F)(F)F)c[nH]1 c1(CNC(C(c2cnn(C)c2)NC(C(CC)O)=O)=O)ncc(C)cn1 C1(C(NOC(C(=O)OC)(C)C)=O)N(C(=O)C(F)C(C)C)CCC1(C)C c1(C(=O)NC2(CC)CN(C(c3cnc(S)n3C3CC3)=O)C2)cncnc1O.S C(c1ccc(F)cc1F)=CC(N1C2CN(S(=O)(=O)CC3CCC3)CC12)=O C1(CC)CCN(C(C2(C3CC3)CC2)=O)C1.C(=O)(CN(S(C)(=O)=O)C)N c1(N2C(CCNC(c3ccc(O)nc3Cl)=O)CCCC2)cnc2ccccc2n1 CC1CCN(C(=O)Nc2ccco2)CC1.C(=O)C1=NOC(C)C1.C(=O)(C)N.C O=C1CN(C(C2CC(F)CN2Cc2ccc(OC(F)F)cn2)=O)CCO1 C(c1cccc(F)c1)=C(C=O)F.n1(CC)nc(C(=O)NC2CC2)c(C)n1.C C1(C(N2CC(N(C(=O)CCCN=[N+]=[N-])C)C2)=O)CCCN1S(=N)(=O)N(C)C c1(C(N(C2CCN(C(c3c(C)nc(COC)s3)=O)CC2)C)=O)cc(O)cnc1N c1(C2CC(SCC(=O)OC)C2)nc(CNC2(c3ccccc3)CC2)co1 N1(C(C(CCOC)NC(c2cc(CO)n(C)n2)=O)=O)CCC2=C(CCCC2)C1 C(C)(C)(CCC)N1CCC(CC(=O)N)C1.N1(C(C)C2CC2)CCN(C)CC1.C C=CC(C)(O)C(=O)NCCCCCCNC(=O)Cc1cncn1C1CC1 C(C(C)(C)CNC(c1ccoc1C1CC1)=O)N(C(=O)Cn1cnnn1)C Cc1ccccc1CC(=O)N(C1CCN(C(=O)Cc2cc[nH]c2)CC1)CCO N1(C(C2(C#N)CC2)=O)CCN(C(=O)Cc2ccc(Cl)c(Br)c2)CC12CC2 C1(NC(C(C(C)(C)C)OC)=O)CC2(CCN(C(=O)C=Cc3ccc[nH]3)C2)C1 Cc1cnsc1C(=O)NC1(CN(C(=O)C=CC2CC2)C)CC1 O(N1CCC(c2ccccc2)CC1)CC.C(=O)(CC(C)(C)S)NC(CNC(C)=O)C CC1CN(C(c2ccc(CCF)cc2)=O)CC1NC(C1(C)CCCCC1)=O Cc1cc(C(=O)NC2CC(CNC(c3cnc(C4CC4)o3)=O)C2)nc(C)n1 CCC(CNC(C1CC(OC)C1)=O)N=c1[nH]nc(C2CCCC2)s1 N1(CCO)CCCCC1=O.C(C=O)=CCN(C)C(=O)OC(C)(C)C c1(NC(C2(F)CCN(Cc3cnc(O)nc3O)C2)=O)nc2cc(F)ccc2s1 c1(C(=O)NCC(CC)NC(=O)CC(O)(CC)c2ccccc2)csc2cccnc12 Cc1c(C(N2CCCC2CCCNC(c2ccc(Cl)o2)=O)=O)cnn1C N1(C(c2c(C)nns2)=O)CCCC(C(=O)NC2CC(n3cncn3)C2)C1C C1(CC(=O)NC2(C)CCN(C(CCCCC=C)=O)CC2)CCc2sccc2C1=O N1(C(C2C(OCC)C2)=O)CCC(c2ccccc2)C1.C(=O)C(C)n1cccn1.N CC(C)CN=C1NC2=CC=CC=CC(CN1)COC2.C1(N(C)C=O)CCC1 n1(CC)nnc(C)c1C(=O)NC1CN(C(c2cc(OC)cnn2)=O)C1 C1(CC)(CC)CC(C(=O)NCCOCC(=O)N)C1.C1(O)(CC)CCOC1 C1(CC(=O)N)CCN(C(C)=O)CC1.CCC(C)CNC(C1CC(C)=NO1)=O CC1CCCCC1(CNC(=O)C(C)(C)n1cccn1)NC(=O)C#CC1CC1 c1(N2CCCC(CNC(=N)N)C2)c(-c2ccc(F)cc2)nc2ccccn12 CC(C)C(C)C(=O)N1CCC(c2n[nH]c(C)n2)CC1.C1(C(=O)N)(C(C)C)CCC1 N1(C(CC(=O)N2CC(C(C)NC(CCC=C)=O)C2)C)CCCCC1=O CC(C)C(O)CC(=O)N(CCNC(=O)C(c1cc(Cl)ccc1F)(C)C)C1CC1 CCCCCCC(C)C(=O)NC1(C2CC2)CCN(C(c2csc(C(F)F)c2)=O)C1 C(=O)(CCCCC(F)F)N1CCN(C(C(C)c2cccs2)=O)C(CC(C)(C)C)C1 c1(SCCC)ccc(C(=O)NCC2C=CC(NC(=O)COC)C2)cc1 N1(C(c2c(OCC)cccc2)=O)CCC(F)CC1C(=O)NC(C)C(C)(C)CC C1(OC)(CNC(C2CC2CF)=O)CCN(C(c2cnc(Br)s2)=O)C1 c1(C(C)C)ccc(C(=O)NC(C)(C)CO)c(F)c1.n1(CC=O)ccccc1=O.N Cn1cc(CC(O)C(=O)NCC2CCC2NC(=O)Cc2cscn2)cn1 Cc1ccsc1CC(N1CCC(N(C)C(c2ocnc2C(C)C)=O)C1)=O C(CC(C(=O)N1CC2CC2(CSC)C1)NC(c1ccns1)=O)SC c1(OCC)ccc(C(=O)O)cc1S(=O)(=O)NC(c1cccnc1F)C c1(CCC)nccn1CCC(=O)NC(C1CCCO1)C N1(C(C(=C)F)=O)CCCC2(CCN(C(=O)CN3CCCC3)C2)C1 CC12CCC(C(N3CCCC(NC(C4CC(=O)N4)=O)CC3)=O)(CC1)CO2 C=C1CC(C)(C(=O)NCC2CCC2NC(=O)C=Cc2ncc[nH]2)C1 c1(CC(=O)NC2CN(C(C(CSC)C)=O)CC2C)n[nH]c2ccccc12.C1CC1 C(=O)(C(C)(C)CCCO)N(CCCCN(C(C1CCN(C(=O)NC)C1)=O)C)C c1(C(N2CCC(F)(CNC(c3cc[nH]c3)=O)CC2)=O)cnn2c1OCC(F)C2 C1(c2cn(C(C)C(=O)N(C)C)nn2)C2CCCC1N(C(c1nnc(C(=O)O)s1)=O)C2 CCC(CC)CCCC(=O)NC1CCCCC1NC(c1cn(C(C)(C)C)cn1)=O N1(C(C(C=C)OC)=O)CC=C(CC(=O)N2C3CCCC2COC3)CC1 c1(C(N2CC(N(C)C(C3CC3c3ccccc3)=O)C2)=O)ccc2nnn(O)c2c1 N1(C(C=C(CCC)CCC)=O)CCC(C)S(=O)(=O)CC1 Cc1cc(O)c(C(=O)N)nn1.C1CN(C(C2CC(CC=O)C2)=O)C1.C(C)(C)C C(C(CC(F)F)NC=O)NC(N(c1cncc(C)c1)CCC)=O.C(C)(C)C C(=O)(C(CNC(=O)C(C)S(N)(=O)=O)C(C)(C)C)Nc1c(C)nc(F)cc1 C1(CC=O)N(C(=O)CC2C(=O)NN=C2C)CCC1(C)C.C(=O)C(C)CC.CC CCCCCCC(C)C(=O)NCCOCC(N1CCCC1(C)C1CC1)=O c1(NC)cncc(C(=O)NC2CCC(N(C)C)C2)n1.C(C)(C)C=CC=O.N c1(NC2(C(=O)OC)CC2)ccccc1C(C)(C)C.C(=O)C(=O)N(C)C.N C#CCC(CC#C)C(=O)N1CCC(CNC(=O)Cc2ccc(Cl)cn2)CC1 c1(N2CC(O)(CCNC(C3CCC(C)(CC)O3)=O)C2)ncc([N+](=O)[O-])cc1F C1(CC)CN(C(c2csnc2C)=O)CCN1c1ncc(I)cn1 C=CC1(CC(=O)NCC(CC)NC(c2sc(C3CC3)nc2C)=O)CCOCC1 N1(C(C(CCC=C)CC(C)C)=O)CC(=O)NC2CCCC2(C)C1 c1(C(=O)NCC2CCC(NC(C(CC)OC)=O)CC2)coc(S(C)(=O)=O)c1 c1(C(=O)NC2(C#N)CCN(c3ncc(NC4CC4)cn3)C2)ccc2[nH]ccc2c1 c1(OCC)cnc(C(=O)N)c(Cl)c1.c1(C=O)cc(C(N)=O)[nH]n1.C1CCC1 N1(C(C2(C(F)(F)F)CC(=C)C2)=O)CCC2CN(C(C3CC3(F)F)=O)CC2CC1.O CCC(CC)C(C)C(=O)N1CCCC(C)(NC(=O)Cc2ccc(C(N)=O)cc2)C1 C(=O)(C1=C(NC2CCCC2c2ccc(F)cc2)CCCC1)OC C1(C(N(C(C(=O)N(C2CCCC2)CC(C)C)C)C)=O)C=CCCC1 CC1CN(C(=O)CN(C)C(=O)C2CC2)CCC1NC(=O)C(C)(C)C(N)=O N1(C(C2CC3(CCC3O)C2)=O)CC2CCC1CN2C1CCCCC1NC1CC1 S(=O)(=O)(c1ccc2c(c1)CCO2)N1CC(NC(=O)CCc2ccsc2)C(O)C1 CC(CNC(=O)C=Cc1cncn1C)CC(=O)NCC1C=CCC1 N1(C(c2ccc(C)n2C)=O)CCN(C(C2(C)CCCC2C)=O)CC(C)(F)C1 C12(NC(C3C(C)OCC3)=O)CC1CN(C(c1cccc(OCC(F)F)n1)=O)C2 CCCCC(CNC(c1cnns1)=O)NC(=O)C(F)(F)C1CCCC1 c1(NC(C)=O)cccc(C=O)n1.CCC(C)(C)C.C1(O)(CC=O)CCCOC1.N N1(C(c2c(C)cno2)=O)CCC(NC(c2cccc(N(C)C)n2)=O)C(CO)CC1 C(Cc1ccccc1)(CCN=c1nc(C2CC2)[nH]s1)N(C(CC(C)C1CC1)=O)C N1(C(CCC(C)NC(Cc2ccc(C)cc2)=O)=O)CCC(F)(F)CC1C C(=O)CC(C)(O)C(F)(F)F.N1(C(c2c(NC)nc(C)cc2)=O)CCC2(CCC2)C1 CCCC(C(=O)NCC1CC(C)N(C(c2ccc(C3CC3)nc2)=O)C1)OC c1(C(=O)NC2C(C)(C)CN(c3ncccc3[N+](=O)[O-])C2)ccn2c1CCCC2 N1(C(Cn2c(C)nc(C)n2)=O)C2CCC1C(NC(C1CC13CCCC3)=O)C2 c1(N(CCOCCNC(CCn2ncc(C)c2)=O)C)c[n+]([O-])ccc1[N+](=O)[O-] C1(CNC(CC=C)=O)CCN(C(=O)C(O)C(F)(F)c2ccccc2)C12CCC2 C1(NC(C2(C)CC2(F)F)=O)CC2CC1N(C(=O)Cc1cccc(F)c1Cl)C2 C1(C2(O)CCOCC2)(C(=O)N)CC1.N1(C(C2C(C)(C)C2(C)C)=O)C2CCC1CC2 CCC(CN(C)C)CC(=O)NC(C)CCCCNC(=O)COc1ccccc1O C1(NC(C(CC#C)O)=O)CCCCCC1NC(=O)CN(C)CCO c1(N2CCCC(CN(C)C(c3cc(C4CC4)no3)=O)C2)ncc(C#N)cc1F C(=O)(CC(O)C(C)C)NC(CNC(c1c(C)cc(CC)o1)=O)(C)CO N1(C(C2CCN(C(C3(CC)CCCO3)=O)C(C)(C)C2)=O)CCC2(COC(=O)N2)C1 Cc1cc([N+](=O)[O-])c(S(=O)(=O)NCC2(C)CCCOC2)cc1C c1(C(=O)NCCN(C(=O)C(C)N=[N+]=[N-])CCOC)cnc(O)c(F)c1 c1(C(=O)N)cn2ccccc2n1.CC(C(C)(C)CN(C)C)NC(=O)C=CC Cc1ccc(C(=O)N(C2CN(C(c3ccn(-c4ccncc4)n3)=O)C2)C)cc1F C(C)(CCCCC#N)(c1nnnn1CC1CC1)NCC1(COCC)CC1 [SH](=O)(=O)c1cnc(N2CC(C(F)(F)F)C(F)C2)c(Cl)c1.Cc1cccc(CN)n1 c1(C(N2CC(CNC(C3CCCC3n3cccn3)=O)C2)=O)cnc(Cl)cc1Cl N1(C(C(c2[nH]c(=N)sc2)(F)F)=O)C2CCC1CC(NC(=O)C(F)C(F)(F)F)C2 c1(C(=O)NCC(CC)NC(=O)C(C)Oc2ccc(C)cc2)ncn2c1CCC2 CC(C)C(C(=O)NCCCC1CCCN1C(c1ccccn1)=O)n1ccnc1 CCC(CC)C(=O)NCC1CCC(NC(C2(C)CC(C#N)C2)=O)CC1 C1(O)(CNC(CCC#CC)=O)CCCN(C(=O)CC2CCC3(CCC3)O2)C1 C1(C(N2C3CN(C(c4cccc(CC)c4N)=O)C(C3)C2)=O)CCc2nc(C)nn2C1 c1(C(=O)NCC2C3CN(C(C4CC(C)CC(C)C4)=O)C2C3)nccc2ccsc12 C(=O)(C(C)(C)CC(F)F)N1CCC(C)(Cn2cc(-c3c(C)cccc3F)nn2)CC1 C1C2CC1N(C(=O)C)C2C.c1ccc(F)cc1.CCS(=O)(=O)N1CC(C=O)C1.N CCCC(F)(F)C(=O)NCC(C)(C)CC(=O)NCC1CC=CCC1 C1(CNC(=O)NCc2scc(C(=O)OC)c2)CNC(=O)N1C c1(C(N2C(CNC(C(C=C=C)C)=O)CCC2)=O)ccc(F)c(O)c1F Cc1sc(C(=O)NCC2CC2)cc1S(N)(=O)=O.C(=O)C(C)(C)n1ccnn1 N1(C(CC2CC(SC)C2)=O)CCN(C(=O)CC(F)(F)Cl)C(C)C1 C(CCCCCO)N1CCC(CC=O)C1.C1(CCC(=O)C)NC(=O)NC1=O.CCCO c1(CC)ccccc1C(=O)NC1(C(=O)NC(CN(C)C)CC)CCSC1 C1(C(C(=O)NCCCSC)F)CCN(C(c2cc(C3CC3)on2)=O)C1 N1(S(=O)(=O)c2sc(Br)cc2Br)CCc2cc3c(cc2C1)CCCC3.C1(CC#N)CCCC1 CC1CC(NC(=O)CN2C(=O)CNC2=O)CN1C(=O)C=Cc1cn[nH]c1 C(=O)(C1c2cnn(C)c2CCN1Cc1ncc(Br)cc1Cl)N(C)C CN1CC(CCNC(=O)CN(C(=O)C(O)C2CCC2)C2CC2)CC1=O n1(C(CC)CC)nc(-c2ccoc2C)nc1CC1CCSC1 N(C(=NCCS(=O)(=O)C1CC1)NCc1cccc(CO)c1)C(C)C1CC1 Cc1nnc2ccc(C(=O)NC(C3CCN(C(C4(CO)CCCO4)=O)C3)C)cn12 CC1=CCN(c2nnc(-c3ccc(C)o3)n2CC(=O)NCC2CCOC2)CC1 c1(N2CCC(CC)C2)ccc(S(=O)(=O)N2CCCC(C)(F)C2)c(Br)c1 C1(NC(C2CCS(=O)(=O)CC2)=O)CC2C1CCN2C(c1cc2ccsc2s1)=O N1(C(C2N(C)CCC2)=O)CC(S(=O)(=O)N2CCN(C(c3cccn3C)=O)CC2)C1 C1(C(N(C(C(C)C)C)C)=O)CCCCN1C(c1cscc1Cl)=O N1(C(C=Cc2ccn(C)c2)=O)CCOCC(C)(CNC(C2(C)CCCC2)=O)C1 C#CCC(CC(=O)N(CC(C)O)C)NC(=O)CC1(OC)CCC1 C(=O)(C(C)(C)C(=O)N1CCOC(C(N2CCC(n3ccnn3)C2)=O)C1)OCC c1(C(N(CCNC(c2ccc(C#C)nc2)=O)CCC)=O)ccc2nc(O)oc2c1 CN1CC=C(C(=O)NC2(CNC(=O)Cc3cncc(F)c3)CCC2)C1 c1(C2C(OC)C2)nc(-c2cnn(C)c2)nn1CC1CCCO1 c1(NC(C2CN(C(C3(C(F)(F)F)CC3)=O)C2)=O)c(-n2cccn2)cccc1F CC1(C(=O)NC2CN(C(c3cnc(Cl)s3)=O)CC2O)COc2ccccc21 c1(C(N2CC(O)(C(=O)O)C(O)C2)=O)n[nH]c2c(Br)cccc12 Cc1cc(Cl)ncc1NC(=O)C(F)C(C)CNC(=O)CCCC(C)C N1(C(CN2C(C)CCC2)=O)CC(NC(=O)C(C)(C)N(C)C)CC(F)(F)C1 c1(CCNC(C2(CC=C)CC2)=O)cc(C(=O)NC(C)(C)C#C)no1.C C=CCC(CC=C)C(=O)N1CC(C)(C)CC1CNC(c1cc2ccccc2[nH]1)=O C(C)(C)(CC(=O)N1CCCC(CC2(O)CC2)C1)OC C1(C(=O)NCCCC(C)C)CCCCC1(C)NC(=O)CNc1ncccn1 CN(C(=NCCc1cc(Br)ccc1F)NC(C1CC1)C1CC1)CC1CC1 C1(NC(=O)C2=CCCC2)CCN(C(=O)C(F)(F)c2ncc[nH]2)CC1O c1(NC(N2CC3N(C(c4cc(CC)ncc4)=O)C(C3)C2)=O)c(F)cc(F)cc1F Cc1cc(NC(c2ccncn2)=O)ccc1NC(=O)CC1COCC(C)(C)O1 Cc1nccn1C(C)C(=O)N(CCCNC(=O)C(C)c1ccsc1)CCO C=CCC(C(=O)NC(CO)C(=O)NCCc1ccccc1)NC(C)=O c1(C(=O)NCC(CC)NC(C2CC(CF)C2)=O)ncc2ccccc2c1N C1(C(C)(C)NC(C(C)(F)F)=O)CCN(C(=O)C(c2ccc(C(F)F)cc2)O)CC1 C(CCCCNC(=O)CCc1cc(Cl)no1)NC(CSC)=O c1cccc(Cl)c1Br.C(=O)(CC(C)NC(=O)CN(C1CCCN1)C)NC(C)C.C CCC(CC)(CO)C(=O)NCC(CNC(c1cc(F)n(C)n1)=O)OC C1CCCCCC(=O)N2CCC(C2)C(F)C(=O)N1.C(C1=CCN(C)CC1)SC N1(C(C(C(=O)OC)OC)=O)Cc2[nH]nc(C(=O)NC)c2C1.C1(C)CC2CC2C1 C1(C(=O)NCC(CNC(c2cccc(CC)c2)=O)C)CCCCC(=O)C1 N1(C(=O)COC2CCCC2)C2CCC(C(N3CC4C=CCC(C4)C3)=O)C1CC2 N1(C(c2c(CC)noc2)=O)CCCC2(C)CC12.c1(C=O)ccc(C(C)C)cc1.N c1(NCCS(=O)(=O)NC)ccc(Br)c(S(=O)(=O)N)n1.C1COC2(CCC2)C1 N1(C(COCCC#C)=O)CC2CC1(CNC(=O)C(CCSC)OC)C2 c1(C(=O)OCCC(=O)N(CC(C)O)C(C)C)cn2c(n1)COCC2.C1CO1 c1(OC)cc(C=O)c(Cl)cc1Cl.c1(C(N2CC(CCC)C2)=O)cnc(=N)[nH]c1.N c1(C(N2C(C(=O)Nc3ccc(OC)cc3Cl)CC3CC32)=O)cccc2nc[nH]c12 N1(C(c2cn(CCNC(C3CCN(C)CC3)=O)nn2)=O)C(CO)CC2CCCC12 c1(NCC2CN(C(CC(=O)OCC)=O)C2)cc(-n2nnnc2C)cc(F)c1.O CC1CN(C(C2(C#N)CC=CC2)=O)CCCN1C(=O)C1=CCC1 c1(OC)cc(C(N2CC3CC(CNC(=O)C4=CCC4)C3C2)=O)cc(F)c1C#N N1(C(CN(C(c2c(CC)nn(C)c2)=O)CC)=O)CC(=O)N2CCCC2C1 N1(C(COc2cccc(OCC)c2)=O)CCN(C(=O)CC)CCC1C.C(N)(=O)N C=CCC(CNC(c1ccon1)=O)NC(=O)Cn1cc(C2CC2)nn1 C(C)(C)C(C)C.C(CCC(=O)N)N(C(C)=O)C.N1(CC=CC=O)CCOCC1 c1(CC(=O)N(CCNC(c2cccc(F)c2)=O)C2CC2)cccc2sccc12 c1(C=O)oc2c(c1C)C(=O)CCC2.C1(NC(CCOCC#C)=O)CC(F)C1.C N1(C(=O)NC2C(SCC)CCCC2)CCOC2CCN(C)CC12 Cc1cc(Cl)ccc1C(=O)NCCCCNC(=O)C(C)Cn1cccn1 CCC(CCC(=O)N1CCC(O)(C(C)NC(=O)Cc2cccs2)C1)OC C12(C(N3CC(CC)OC(C)C3)=O)CCC(CC1)N(C(C1(O)CC1)=O)C2 c1(C(N2CCC(N(C(C)=O)C)C2)=O)cc(Cl)ncc1NCc1cccc(O)c1C CC(CCNC(c1csc(O)n1)=O)C(=O)Nc1cccc(OCF)c1 N1(C(c2cc(COC)[nH]n2)=O)CCOC2CN(C(c3ccn(C)c3)=O)CC12 C(=O)(C1=NOC(C)(C)C1)N1CCCC(C)(CNC(CC(C)(F)F)=O)C1 c1(C(=O)N)n[nH]c2cccnc12.C1(CC)CCCCN1C(C1CC1C(C)(F)F)=O C12(CNC(Cc3c(C)ccs3)=O)CCCCC1N(C(=O)CC(C)F)CCC2 C1(NC(c2nc(COC)oc2)=O)CN(C(=O)C(c2cncnc2)C)CC1SC O=C1COc2cc(C(N3CCC4C(C3)CN4C(c3cccnc3)=O)=O)cnc2N1 c1(C(N(CC=C)C2CC2)=O)ccc(CNC(=O)CCC2CCCO2)s1 C1(CSC)CN(C(=O)OCCOc2ccc(NCCCC=C)cn2)CCO1 c1(C(N(C2CCN(C(C3(C)C=CCCC3)=O)C2)CCC)=O)cc2ccsc2n1C C1(C(N2CC(C)(NC(c3cc(OC)ns3)=O)C2)=O)CSCC(=O)N1 c1(CC)cc(=NCC2CCN(C(c3nonc3COC)=O)CC2C)[nH]cn1 N1(Cc2ccc(C)cc2Br)CC2CN(C(=O)C(C)NC=O)CC2C1 c1(CN(CCC)Cc2cccc(-c3ccsc3)c2)ccccc1F c12csc(n1)C(C)NC(=O)C2.C(C(=O)O)(C1CC1)SCC c1(C(=O)OCC)cc(O)nc(NC23CCN(C(C)C)CC2C3)n1 C1CC2CCC(C1F)N2C(c1cccn1C(C)C)=O.n1(CC)cc(C(=O)N)cn1 c1(CNc2ccc(C(=O)Nc3ccnc(O)c3)nc2)ccc(Cl)cc1O C(C(CC(C)C)C(=O)N1C2CCC1CC(CO)C2)NC(C(C=C)OC)=O N1(C(C(CCC)C)=O)CCCCCC1C(=O)NCc1cnnn1C N1(OC)CCN(C)CC1.C(C)(CO)(C(=O)N)NC(C1CCC1)=O.C1CC1.C N1(c2c(Br)cnc(C)n2)CCc2nc(-c3ccc(Cn4ccnc4)cc3)sc2C1 n1(CC(N2CCC(CNC(C3CC(F)C3)=O)C2)=O)nc2ccccn2c1=O C1(CC(=O)N(CCCC)C)COC(C)(C)CO1.c1(C(C)OC)nc(C=O)cs1.N C1(C2CCCNC2)(NC(c2cccnc2Oc2ccccc2F)=O)CCC1 c1(C(=O)NCC2(NC(CCNC(C)=O)=O)CCOC2)cnc2scc(C)n12 c1(NC(C2CC2NCc2ccc(C(F)(F)F)cc2)=O)cnc2ccccc2c1Cl CC(C)CC(C)(C)C(=O)NC(C)C(C)NC(=O)CC1CC1 C(CN=c1nc(N2CCC(CC#N)C2)c2cccc(F)c2[nH]1)=CCCC CC(C)(C(=O)NC1CCCCC1C(F)(F)F)C(O)c1ccccc1 C#Cc1cnc(C(=O)NCC(C)=CC(=O)NCC2NC(=O)NC2=O)c(C)c1 c1(C(N2CCCC(NC(CC(C)C)=O)C2)=O)cc(C(F)(F)F)cc(Cl)c1 CCC(C)CC(=O)NC1CCN(CC(=O)NCc2ccc(-c3cnn(C)c3)o2)C1 C1(CNC(C(C=C)O)=O)CN(C(=O)CCc2ccc(C)nc2)C2(CCC2)C1 CC1(C)CCCC(C(N2CC(O)CC2C(N2CC(CN=[N+]=[N-])C2)=O)=O)C1 Cn1cc2c(n1)C(C(=O)NNc1ncc(C(=O)OC(C)(C)C)s1)CCC2 c1(C(=O)NCC(CNC(c2cccc(Cl)c2O)=O)F)ncnc2c1CCCC2 C(C)(C)(C#Cc1cn(CCCCF)nn1)NC(CCCCC(CC)C)=O N1(C(COC)=O)CCCCC(NC(=O)C(C(C)C)c2ccccc2)C1 C1(n2cc(-c3ccc(C4CC4)cc3)nn2)(C(=O)NCc2ncsn2)CCOCC1 c1(CC=O)cncc(C#N)c1.C(C=O)(C1CCCC1)OCC.CCC1CC1.N N1(C(c2c(COC)ncs2)=O)CCN(C(c2cc(C(F)(F)F)no2)=O)C2CC12 c1(C(N2C(C)CC(CNC(Cn3nnc(C)n3)=O)C2)=O)cc(F)c(N)cc1F C1(C(=O)NCC(C=C)O)CN(C(C2(O)CCC2)=O)CCC1(C)C c1(C(N2CC(C)C(CNC(c3ccnc(F)c3)=O)CC2)=O)ccc2nncn2c1 CC1CC(N(C(=O)CSCCNC(=O)C2=CCSC2)C)CC(C)C1 N1(C(c2c(C)c(Br)c(C)o2)=O)CCCN(C(c2cc(O)nn2C)=O)C(C)C1 C(=O)(C1CCCc2nn(C)cc21)NCC1(C)CCCN(C(C=COCC)=O)C1 c1(C(N2C(CC)CN(C)C(=O)C2)C(=O)NC(C)(C)CC)cc(Br)ccc1[N+](=O)[O-] c1(CN)cccc2c1CCCN2C(C1CC(c2ccc(C(F)(F)F)cc2)C1)=O N1(C(c2c(OC)ccc(CO)c2)=O)CC(NC(=O)CS)CCC(O)C1.C1CC1 C(C(C)(C)O)(C1CC1)NC(CN(C(=O)CCc1nccs1)CCC)=O N1(C(C2C3CN(C(c4ccc(CN)cc4)=O)CC32)=O)CC(CO)CC(CO)C1 c1cc(Cl)ccc1C(OC)OC.c1(CC(=O)NCC)cnc(NC)s1 CCC(C(=O)NCC1CCN1C(=O)CCCN(C)C(C)=O)C(C)(F)F C12(CNC(c3c(OCC)scc3)=O)COC(C1)C2.c1(C=O)ccco1.C c1(CCC)c(C(=O)OC2CCCCC2C)cnn1-c1cccc(C)c1 C1(C(C)CNC(=O)Cc2cscn2)CCN(C(C2(C)CCCCO2)=O)CC1 C1(NC(C(C)CN2CCCCC2)=O)CCN(C(=O)CCc2ccccn2)CC1 C1(NC(CC(C=C)C)=O)CCCCCC1NC(=O)CCc1ccccc1O c1(C(N2CCC(CCNC(c3n[nH]c4c3CCC4)=O)C2)=O)cn2c(n1)SCC2 c1(CCOC)nc(=NC2(CNC(=O)C=Cc3cncnc3O)COC2)s[nH]1 c1(NC2CC(NC(Cn3c(C(=O)OCC)cnc3)=O)C2)cc(Cl)cc(Cl)c1 c1(C(=O)Nc2cc(F)c(O)c(Cl)c2)[nH]nc2ncc(-c3nn[nH]n3)cc12 CCCCC(C)C(=O)N1CC(CNC(=O)C(C2CC(F)(F)C2)O)C1 C(N=c1nc[nH]cc1C#N)C1CCN(C(C2C(C)CC3CC3C2)=O)CC1C Cc1cc(C(N2CCC(N(CCO)C(c3cc[nH]n3)=O)C2)=O)c2nc(C)n(C)c2n1 C1C(O)C(O)CN1C(=O)Cc1ccc(C)cc1Cl.C(C)(C(=O)N)NC(CC)=O N1(C(c2nc(OC)oc2)=O)CCCC(C(=O)NC2CC2C(=O)O)CC1 C1(O)(C(C)NC(C2C(=C)C2)=O)CCN(c2nccc(CO)n2)CC1 N1(C(=O)C(O)CF)CCC2(CCC(CNC(C34CCC(CO)(CC3)C4)=O)O2)CC1 C1CC(C)CN(C(=O)C(CN(C)C)N(C)C)C1.C(CC1CC1)(C(=O)N)OC Cc1ccc(C(C2CC2)NC(C2CC(N=[N+]=[N-])C2)=O)nc1 C1(CNC(CC(C)c2ccco2)=O)CN(C(=O)CN2CC(C)(C)C2)CC12CC2 N1(C(CSCCCC)=O)CC(C)C2(CC2)C1.c1(C=O)[nH]ccc1-c1cccs1.N Nc1ccccc1NC(=O)C(=O)NCc1ccc(-n2cnnn2)cc1 CCC(CC)C(C(=O)NC1CCC(F)CC1)N1CCOCC1 N12CCN(CC1)c1cccc(c1)OC=CC2=O.c1(C(=O)NCC)cnncc1C c1(C(N2CCN(CC(=O)NC(CC#C)CO)CC2)=O)ccc(C)c(C)n1 CC1CN(C(=O)C=CCF)CC1(C)C(=O)NCC(C)C(C)(F)F N1(C(CC)=O)CCN(C(=O)C(CN=[N+]=[N-])NC(c2cc(F)ccc2F)=O)CC1 N1(C(CC)=O)CCCC(C)(C)C1.C(CC(=O)N)NC(CN(C(C)=O)C(C)C)=O CCCCCC(O)CC(=O)NCC(C)(CO)NC(c1conc1COC)=O C1(C(=O)NC2C(C)N(C(c3ccc(Cl)nc3N)=O)CC2)CC2CS(=O)(=O)CC2C1 C(=O)(C(C)(C)C(O)C(C)C)N1CCC(CN(C(c2c(C)cc(C#N)s2)=O)C)CC1 C1(OCCNC(=O)Cn2cc(C(F)(F)F)nn2)CCCCC1.C(CC(O)CO)S CC1CCC(CN)N(S(=O)(=O)c2sccc2Cl)C1 C(=O)(C1COc2ccccc21)N1CC(C(C)NC(C2C=CCC2)=O)OCC1 CCC(O)C(C)C(=O)N1CCC1(C)CC(=O)NCCc1ccc(O)nc1 CC1(CC(=O)NC2(C)CCOCC2)CC(F)(F)C1.C1(C(=O)N)CCN(CC)CC1 CC(C#N)C(=O)N1CCC1CNC(c1cc(C2CCCN2C)[nH]n1)=O CC(C)CC(C)C(=O)N(CCCOCCNC(=O)CCC1CC(F)(F)C1)C C=CCCC(C)(C)C(=O)NCCCC(CCC)NC(c1cc([N+](=O)[O-])cn1C)=O C1(C)CCC(O)CC1.N1(C(C2C(CCOC)C2)=O)CC2C(C(=O)N)C2C1.C C1(NC(CC2(C)CC2)=O)CN(C(=O)CC2CC2c2ccc(F)cc2Cl)CC12CC2 CCC(C)C(O)C(=O)N1CCC(O)(CNC(C2CCC(C)(O)CC2)=O)C1 N1(C(c2cc(C)n(C3CC3)n2)=O)C(C)CC2CN(C(C3(C)CCCOC3)=O)CC12 CCCC(CC)C(=O)NC1CCCCC1C(=O)N(C)CC1CCCCC1 C(=O)(C1=CCCN(C(c2ccc(Br)c(Cl)n2)=O)C1)NC(C=C)CO Cn1c(CC(=O)OCC2=CC(=O)OC2)nc2ccccc12 c1(NC2CC3CN(C(c4cnc(C(C)O)s4)=O)CC32)cc(O)nc(=O)n1C C1(NC(CC(=C=C)C)=O)CC2(C1)CN(C(c1cc(C3CC3)nn1CC=C)=O)C2 C1(C)(CNC(C(C=C)(C)O)=O)CN(C(=O)C(F)(F)COC)CC1C c1(OCCOC)ccccc1.C1(C(=O)N)CN(C(C2(C(N)=O)CC2)=O)C1 c1(C(C)C)cncc(C(N2CC=CC(NC(C3CC(C)(C)CO3)=O)C2)=O)c1 N1(S(=O)(=O)C2CC2)CCN(N2CCC(F)(F)C2)CC1 CS(=O)(=O)c1sccc1C(=O)NC1CC1.C1(C=O)CC(n2cccn2)C1.C N1(C(=O)Cc2cnccn2)CC2CCC(C1CO)N2C(c1ccc(F)c(F)c1)=O C(=O)(C1CCCc2n[nH]cc21)NCC(C1CCC1)NC(c1c(Cl)ccc(C)c1)=O N1(C(C(C)OC2CCCC2)=O)CCOCC(NC(c2ccc(N)cc2F)=O)C1 c1(SC)cc2ccccc2c(CC2COCCN(CCOc3ccccc3)C2)n1 C(=O)(C(CC1CC1)CC1CC1)NCCCCNC(C1CCCS1)=O CC(C#N)CCC(=O)N1CCOC(CNC(c2cc(-n3cccn3)ccn2)=O)C1 c12nnc(n1-c1ccccc1Cl)NC(=O)C(C)S2.C1(N(C)C)(CN)CCCCC1 C(C)(CN=c1[nH]cnc(Cl)c1F)(C1CC1)NC(C1CC(C)SCC1)=O c1(C(N(C2CC(NC(c3c(COC)noc3)=O)C2)C)=O)cc(OC)cnc1 c1(C(N2CCCC(NC(C(CC=C)NC(C)=O)=O)C2)=O)cc([N+](=O)[O-])c[nH]1 c1(CC)cc(OC)ccc1C(=O)NC1CC(NC(=O)C(C)CSC)CC1O Cc1ccc(F)cc1-n1nc(-c2cnn(CCO)c2)nc1-c1cc(Cl)cn1C Cc1cc(C#N)sc1C(N1CCOCC(CNC(=O)C=CC(F)(F)F)C1)=O c1(C(=O)NCC(CNC(Cc2nnc(C)s2)=O)O)cc(F)cc2nc[nH]c12 C1(CC(=O)NCCC)CCN(OC)CC1.CCC1C(=O)N(CCO)CCC1.SC.S c1(C(N2C(CCNC(C=C(C)C)=O)CCCC2)=O)ccc(C2CC2)c(C)c1 C1(C(=O)NCCC2CC(C)C2)CC2CCC(C1)N2C(c1nc(Cl)cs1)=O c1(C(=O)NCC(C)N(C(c2c(CC)nns2)=O)C)cc(Cl)ccc1F c1ccc(Cl)cc1.c1(C2C(C(N(CCN(C(=O)CS)C)C)=O)C2)ccncc1 C1(CNC(Cc2n(C)cnc2)=O)CC(C)(C)CCC1.c1(C(=O)N)ccnc(O)c1 C(=O)(CS(=O)(=O)CC(=O)OC)N1C(CC)C(NC(=O)CC(F)(F)CC)CC1 c1(C(=O)NCC2(C)CCCN(C(C3=C(C)OCC3)=O)C2)nn(C)c2c1COCC2 N1(C(C(C)(O)C2CCC2)=O)CC2(CCCCN(C(c3cccc(Cl)c3)=O)C2)C1 C=CC1CN(C(=O)CCC#CC)CC1NC(=O)C=CCN(C)CC C1(C(N2CC(C)N(C(c3ccc4nonc4c3)=O)CC2)=O)CC2CCC(C1)N2C CCC(CNC(=O)C(C(C)C)NC(c1ccc(C)o1)=O)(CC)C(N)=O c1(C(=O)NC2CCC(NC(C3CC3C3CC3)=O)C2)cc2ccccc2cn1 Cc1cc(C(=O)NCC(O)CCNC(c2cccc(C)c2N)=O)cc2nn[nH]c12 C1(CNC(C=C(CC)C)=O)CCCC1NC(c1nn[nH]c1C(F)(F)F)=O C1(CC)CC(C)CN(C(=O)CNC(C2CC3CC(=O)C2O3)=O)C1 N1(C(CC(C)C2CC2)=O)CC(CNC(=O)Cc2cc[nH]n2)C(F)(F)C1 N1(CC(=O)NCC(CN(C(=O)CCC2CCCC2)CC)(C)C)CCCCC1 C1(NC(C(CCC)OC)=O)CN(C(c2ncccc2O)=O)CC(F)(F)C1 C1(C(=O)NCC=CC)CCC(C)(C)N(C(=O)CC(C)C(C)(C)C)C1 CCCC(CNC(c1ccnn1COC)=O)C(=O)N(C1(C)CCCC1)C C1(C(=O)NCC(C)(C)O)CN(C(=O)CN2CCOC2=O)CCO1 c1(C(=O)NCC(CO)NC(C(CC)CC)=O)c(C)oc(C)c1Br c1(OC)ccc(Cl)c(CCNC(c2cc(Cl)ncc2N)c2nnnn2C2CC2)c1 Cc1cn2c(CC(=O)N(C)CCOCCCNC(=O)C(O)C(C)C)csc2n1 N1(C(COC)=O)C(CNC(=O)CNC(=O)CN(C)C)CC2COCC12 COn1cnc(C)c1C(=O)NCC1CN(C(C2(Br)CC2)=O)CCC1C c1(CC(=O)NCC(C)CNC(c2ncc(F)cc2F)=O)cccc2cccnc12 N1(C(C2(NC(c3c(C)ccc(F)c3)=O)CC2(C)C)=O)CCCC(C2CCC2)C1 CCCCC(CC(=O)N1CCC(C2CC2)CC1)NC(C1(O)CCOC1)=O C1(C(N2CCC(c3nc(-c4cccc(F)c4)no3)CC2)=O)CCc2[nH]nc(O)c2C1 c1(NC(=O)NCCC(N2CCN(C)CC2)C)cccc(F)c1 C1(CC(=O)NCC=CC(=O)NCCCSC)CCCCO1 CC12CN(C(=O)CN)CC1(C)C(=O)N(Cc1cn(C3CCNC3)nn1)O2 Cc1cc(C(N2CCC(NC(c3sccc3C)=O)C(C)C2)=O)c(N)c(Cl)c1 C(C)(C)(C(C)CC(=O)NC1CC(C)(C)C1)NC(C1=NOC(C)C1)=O N1(C(C(=O)NC(c2nnc(C)o2)C)=O)CC2CCC2(C)C1 N1(C(C=C(CC)CC)=O)CCCN(C(=O)CC(C)CC)CC1CO N1(C(C(C)N(C(C)=O)C)=O)CC(NC(c2ncoc2C)=O)C(C)C1 c1(C(=O)NC(C2CCCCC2)C2CCCCC2)ccnc2ccncc12 c1(C(=O)NCC2CCN(C(=O)CC3C=CCC3)CC2)nsc2c(Cl)cccc12 C(CC(C(=O)NCC1C=CCC1)NC(c1cscn1)=O)SC O=C(CCCCCn1cc(CC2(CC3CCCCC3(F)F)OCCO2)nn1)NO Cn1cc(NCC(C)(C)C#N)c(OC2CCNCC2)n1 N1(C(c2ccc(N(C)C)cn2)=O)CC(C2CN(C(c3cc(F)cc(Cl)c3)=O)C2)C1 Cc1cc2[nH]c(C(=O)NC3CCN(C(=O)COC)C34CC4)cc2o1.C1CCCO1 N1(C(CCc2ccc(C)nc2)=O)CC(C)(CNC(C2CNC(=O)C2)=O)CC1(C)C Cc1cc(C(N2CCC(NC(c3nnn(C)c3N)=O)C(C)C2)=O)c2n[nH]cc2c1 N#CC1(C(=O)NNC(C2CCC(=O)NC2=O)=O)CC12CCN(CCF)CC2 c1(C(=O)NC(CC=C)CNC(=O)C(O)CC(C)C)cccc2c1COC2 N1(C(CC2CCCC(C)C2)=O)CCCCC(NC(=O)Cc2csc3nccn23)C1 n1(C(C)CNC(=O)N(CC(C)(C)C)CCCO)cc(Br)cn1 c1(CNC(C(C2CCN(C(=O)C(O)C3CCC3)C2)C)=O)ccc(F)cn1 c1(CNC(C(=O)NCC)=O)cccc(C(=O)N(C)CC2CCCO2)n1 c1(C(=O)NC2CCC(CNC(C(C)N(C)C)=O)C2)ccc(F)c(O)c1F C#Cc1ccc(C(N2CC(CC(=O)NC3(c4nccs4)CC3)(OC)C2)=O)cn1 c1(C(N2CCCCC(NC(=O)COC3CCCOC3)C2)=O)c(F)ccc(F)c1Cl N1(C(C2(CCOC)CCCC2)=O)CCCCC(NC(=O)Cn2cnc(C#N)n2)C1 c1(CCC(=O)NCC(=O)NC(c2cnn(C)c2)CC)ccc(Cl)c(C)c1 CC1CCCC1CC(=O)N(CCCNC(c1cnco1)=O)C1CC1 C(=O)(C1=CCCC1C)NC1C(C(=O)NCC(C)(C)OC)COC1 CCC(C)(C)C(C)CC(=O)NC1CCCC1CNC(=O)C1=CCOCC1 c1(C(=O)NC2CN(Cc3c(F)ccc(C(=O)O)c3)CC2O)cc(F)c(F)cc1I c1(CC)cccc(CC)c1C(=O)NC(C1CCCC1)C.C(=O)CC(O)C(C)C.N c1(CC)ccccc1CCOC(c1cnc(C2CCC2)s1)=O C1(CNC(C(CC)(C)C)=O)CN(C(C2CCC(=O)O2)=O)CC(C)(C)O1 N1(C(CCCCC)=O)CC2(CCCC2NC(C2CCN(CC)C2)=O)C1 C1(NC(c2ccncc2)=O)CC2CCC(C1)N2C(C1COCCO1)=O C1(NC(C(C(=O)OC)C)=O)CC2(C1)CN(C(c1csc(=N)[nH]1)=O)C2 C(=O)(CCCCSC)NC(CN(C(=O)C(=O)NC(C)C)CC)C CC1(C)CC(C)(C(=O)NC(CF)C(F)F)CN1C(=O)CC1CCCC12CC2 c1(C(=O)NCCCCNC(CSCCOC)=O)ccc(CC(C)C)nc1 C1(C(=O)NCC2(F)CN(C(CCCSC)=O)C2)CN2CCN1CC2C c1(C(=O)NCC(CC)NC(=O)C(F)C2CCOC2)cnc2ccccc2c1OC C12(O)CCN(CC1)Cc1ccc(cc1O)NC(=O)C2.C1(CC#N)CCC1 N1(C(C(CC)C)=O)C2CCC1CN(C(C1(C3CC3)CC=CC1)=O)C2 CC1CC(C(=O)N2CCCCC2C2(NC(=O)C=CC3CC3)CC2)=NO1 c1(N2CCC(N(C(=O)C(=O)N=S(C)(C)=O)C)C2)ncccc1[N+](=O)[O-] CON=C(C(=O)N(C)CC1CN(C(c2cc3sccc3[nH]2)=O)C1)c1ccco1 N1(C(c2n[nH]c(C(C)C)c2Br)=O)CCN(C(=O)C=C2CC2)CC1CF N1(C(C(=O)NCC2(C(C)(C)C)CCNC2)=O)CCCC(c2ccncn2)C1 c1(C(=O)NC2CCCN(Cc3cccc(Br)c3Cl)CC2)cc(Br)cc2cc[nH]c12 Cc1cc(C(N)=O)cc(C(=O)N)c1.c1(C(N2CCCC2)=O)cc(C)c(C)nn1.C C(=O)(CN=c1cc[nH]cc1)N1CC(O)(CCNC(c2nc(COC)sc2)=O)C1 CC1(CNC(C2CCCCCN2C(=O)CNC=O)=O)NC(=O)NC1=O c1cc(C)ccc1[N+](=O)[O-].c1(CC)nn(C)c(C(C(=O)NC(C)C)N(C)C)c1Br O=C1CN(C(C2C3CC4C(C3)C24)=O)C(C(N2CC3CCCC3C2)=O)CN1 C1(C)(C(=O)OC)CC(C(=O)N(CC(C)C)C)C1.C1(C)(CC=O)CCC1.N C(=O)(C(C)CC(C)(C)C)N1C(C(C)C)CN(C(=O)CC2CCC(F)(F)CC2)CC1 c1(CC)cc(CC(=O)NC(C)CCNC(=O)C(n2nccc2C)C)n(C)n1 C(CNC(C1(NC(C2COCCO2)=O)CC1(C)C)=O)(C(F)(F)F)OC C(=O)(Nn1cccn1)C1CCCN(C(C2(C)CC(=O)C2)=O)C1 C1(CCC)CCCN(C(=NC)NCC2c3ccccc3CN2C)C1 C(CCC(F)(F)F)NC(c1c(CC=C)cccc1)=O.C1(=CC=O)CCC(C)C1 c1(OC)cccc(N2CCC(OC)C2)n1.C1C(F)C(=O)NCc2nc1no2 C(=O)(C1CCC(=O)c2ccccc21)N(C)Cc1cn(CC2CCOC2)nn1 C1(CCC=C)(CNC(c2csc(C(C)C)n2)=O)CCNCC1 Cc1cccc(C(O)C=O)c1.c1(C(N(CC)C2CC2)=O)c(C)noc1C(F)F C1(C(=O)NCCn2cc(CO)nn2)CCCC(C(F)(F)F)O1.N1(C)CCOCC1 c1(C(=O)NC2(CCC)CCCN(C(c3ccoc3)=O)C2)cnc2n1CCCCC2 CCCCC(CNC(=O)CSCc1cccnc1)NC(c1cnc(O)o1)=O c1(CNCCNC(C)=O)cc(=NCc2cccc(C)n2)[nH]c(C(C)C)n1 CC(C1CCCCC1)=CC(N1CCCC(CCNC(=O)C(F)C(F)(F)F)C1)=O C12CCC(CC1)N2C(c1cccc(C(N)=O)n1)=O.c1(SC)cscc1C(=O)N C1(CNC(C=C(C)c2ccco2)=O)N(C(=O)CCn2cncn2)CCC1(C)C c1(C(N2CCN(CCCNC(C=C(C)Cl)=O)CC2)=O)ccc2ccccc2c1C C(CN=C(NC(C)C)N1CC(F)(F)C(F)(F)C1)N1CCc2c(C)cccc2C1 C=Cc1ccc(CNC(Cc2ccco2)C(N2CCC(C(=O)OC)C2C)=O)cc1 C1(CNC(c2n(CC)ncn2)=O)CCC12CCN(C(C1COC(=O)C1)=O)CC2 N1(C(CCCC#CC)=O)CCC2CCCC12C(=O)N(C1CC(F)(F)C1)C C12(C(=O)N)CC(CN(C(=O)C=Cc3ccoc3)C1)C2.c1(CC)cccc(O)c1 Cc1ccc(C(C)CC(=O)NCCN(C)C(c2cnccc2Cl)=O)cc1 C1(OC)CCC(C(N2CCC(C(C)NC(C3CC4CC4C3)=O)CC2)=O)CC1 c1(CN(C(c2ncccc2F)=O)C2CC2)cccc2nccn12 c1(C(=O)NCC2(C(=O)Nc3cn(CC=C)nc3)CC=CC2)ccccc1Cl C1(CNC2(c3n(CS(=O)Cc4ccccc4)nnn3)CSC2)CC2(CCOCC2)O1 N1(C(CC2(OC)CCOCC2)=O)CC(NC(c2c(C)ncn2O)=O)CC(O)C1 n1(CCCC)cc(S(=O)(=O)N2CCN(C(=O)C(=O)N(CCC)CC)CC2)cn1 C1(CC)CN(C(=O)CNC(=O)CNC(=O)CC2CCCSC2)CC1O C1(C(C)C)(C(=O)NCC2C=CCOC2)CCN(C(=O)CCCC2CCC2)C1 N1(C(=O)CC2CC(CF)C2)CCC(O)C1C(=O)N(CCCO)CCCO N1(C(c2c(C)cc(C)o2)=O)CCCC2(CC2)C1.C1(CC(=O)N)CCC(C)(C)CO1 c1(C(N(C2CCN(C(CC(C)F)=O)C2)CC2CC2)=O)ccc(N2CCCC2)nc1 CCCCCC(O)CC(=O)N1CCN(C(=O)C=Cc2c(C)nn(C)c2Cl)C(C)C1 C1(NC(C=NOC)=O)CN(C(=O)COCc2ccnn2C)CC2(CC2)C1 N1(C(C(=O)Nc2ccc(S(C)=O)cc2)=O)CCOc2cc(N)ccc2C1 C(=O)(CCCC(F)(F)CO)N(c1nnc(C2C(C)NC(=O)CC2)n1C1CC1)C c1ccc2c(c1)CCC2.C(CC(=O)NC(CN(C(=O)CC)C)CC)OCCC.O N#Cc1ccc(C2C(NC(=O)NC(C3CCC(c4ccccc4)CC3)=O)C2)s1 c1(C(=O)NC2CCC(NC)CC2)ccc2nc(COC)[nH]c2c1 Cc1cccn2ncc(C(N3CC4CC(C3)N4C(=O)CC3CC=CC3)=O)c12 c1(C(N2CC(NC(C3CCC(=O)NC3)=O)C(F)CC2)=O)noc2c1CCCCC2 C(=O)(C1CCCc2cccnc21)NCC(CNC(CCCOC(C)(C)C)=O)O N1(C(Cc2c(C)n[nH]c2C)=O)CC2CCC(C1)N2C(=O)C#CC(=O)N(C)C C1(CC(=O)NCC=CCNC(CC(C)CF)=O)Oc2ccccc2NC1=O c1(C(c2nnnn2CCCF)NCC(CC)CO)cc(C(F)(F)F)ccc1Cl C1(C)(CNC(C=CC(CC)C)=O)CCN(C(c2cnn(C3CC3)c2Cl)=O)C1 N1(C(C(CC#C)O)=O)CC(CNC(c2sccc2C)=O)CC(C)(C)C1 S(=O)(=O)(c1c(OC(C)C)c(Cl)ccc1Cl)NC(CCCCOC)=O C1(O)(CNC(=O)CCC2CCCC2)CCCN(C(c2cncc(Cl)c2Cl)=O)CC1 Cc1ccc(OC(=O)CC2(O)CCC2)c(-n2cc(C)nn2)c1.C1(C=O)CC1C C1(CC)CC(C(=O)NCC(C)CNC(c2c(Cl)nn(C)c2Cl)=O)CC(=O)N1 C12(C(=O)OC)CCCC1(C(=O)NCCCNC(=O)CCc1cnccc1)C2 Cc1cc(C)c(C(=O)NC23CC2CN(C(c2ccc(-c4ccccc4)n2C)=O)C3)o1 C=C1COCCN(C(C2CN(C(c3ccnc(CC)c3)=O)CCN2C)=O)C1 C12(CNC(c3scc(C)c3)=O)CCC1CCN2C(c1cc(C(C)C)nn1C)=O c1(C(=O)NCC=CCNC(c2cnn[nH]2)=O)csc2c(Br)cccc12 C1(C(=O)NC(c2ccoc2)C)(CNC(C23CCCC2C3)=O)CC=CC1 C1(C(N2CCCC(C)(NC(c3n(C=C)ncc3)=O)C2)=O)CCc2nn(C)cc2C1 c1ccc(F)cc1.Cc1oncc1C(=O)N(C)CC1CCCN1C(=O)C(C)O.C c1(C(COC)NCc2cnn(C3CC3(F)F)c2)ccc(C#N)cc1 c1(C(=O)NCC(CNC(C2CC(C)C2)=O)O)cccn2nncc12 C1(NC(C(=O)N(CCNC(CNC(CCC)=O)=O)CC)C)CCC(C)CC1 Cc1ccnnc1C(=O)NCC=CC(=O)N(C1CC1)CC1CCCC(O)C1 S(=O)(=O)(c1ccc(Cl)s1)N1C(C)C(=O)N(C(C2OCCCC2(C)C)=O)CC1 c1(C(=O)N)cc(F)cc(F)c1.C(CC(=O)NC(C)CC)SC.C=O.C(C)C Cc1cccc(F)c1NC(C1(c2ccnn2C)CC1)=O CC1(C)CC(NC(=O)C(O)C2CC2)CCN(C(c2[nH]nnc2C2CC2)=O)C1 N1(C(Cc2nc(C)oc2)=O)CCCC(N(C)C(c2oc(C(F)(F)F)nc2C)=O)C1 Cc1ccc(CC(=O)NC23CC(C2)N(C(=O)CC2OCCC2C)C3)cc1 C12(C(C)NC(CCCCSC)=O)CCC1CN(C(=O)CSc1ccncc1)C2 CC(C(=O)NC1C2CN(C(=O)C(C)(C)Oc3ccccc3)CC12)C(F)F c1(N(C(COC(C2C(C)CCS2)=O)=O)C)cc(C(N)=O)ccc1[N+](=O)[O-] n1(CC(N2CC3CC(NC(c4cncc(F)n4)=O)C3C2)=O)cc2ccccc2n1 c1ccc(Cl)c(Cl)c1.c1(C(N2CCN(C3CC3)CC2)C(=O)NC)cc(Cl)c(Cl)s1 C1(NC(=O)Cc2nnc3n2CCOC3)CN(C(C2CC2(F)F)=O)Cc2nccn2C1 CCC(C(=O)N1CC(F)(C)C1)Oc1ccccc1.C1(C(=O)N)CCC1.C1CC1 C1(C(=O)NC(CCC)CC)(CC)CCCN1C(C1CC(N(C)C)C1)=O C(=O)(C1=CCN(C(C23CCC(CC2F)C3)=O)CC1)N1C(C)CC1C(=O)O CC1=C(C(=O)NCC(O)CC(=O)NC(C)C2=CCN(C)CC2)SCCO1 c1(C(=O)NC(CC(=O)NCC(C(C)C)CO)(C)C)ccccc1C#N N1(C(c2nc(C(C)(C)C)[nH]n2)=O)CCCC(NC(C2(C(F)F)CCCO2)=O)C1 C1(NC(c2n(C)cc(Cl)c2)=O)CCC2CC1CN2C(=O)CCN1CCOCC1 c1(CC(=O)NCC(CC)(C)NC(=O)CCO)ccc(Cl)nc1C.C1CCCOC1 C1(C(=O)NC2C(CC)N(C(=O)CC3CCC(=O)O3)CC2)CN2CCN1CC2C c1(C(=O)NCCCC2OCCN(C(C=CCOC)=O)C2)cccc(C#CCO)c1 Cc1cn2c(n1)CC(c1nc(-c3cc(Cl)ccc3Cl)nn1CCO)C2 C(C(COC)C(=O)NC1CCC(CNC(C2(F)CC2C)=O)CC1)OC N1(C(CN(C)CCO)=O)CCCC1C1CCCCN1C(=O)Cc1ccnn1C N1(C(C(c2ccc(F)cc2)(C)C)=O)CC2(CCC(NC(c3nc[nH]n3)=O)CC2)C1 CCCC(C)C(=O)N1CCCC1C=CC(=O)N(CCOC)CCOC Cc1cn[nH]c(=NC(=O)C2(C)CCN2C(c2cc3c(s2)CSC3)=O)c1 Cc1cc(C(=O)NCCOC2CCN(C(=O)Cn3cnc(C#N)n3)C2)ccc1F n1(CC=C)cccc1C(=O)NCCN(CC(C)C)Cc1ccc(Br)s1 C(=O)(C(C)(C)C(C)NC(=O)C1CC1)NC(CCCC)CO c1(NC(CN2CC(NC(=O)Cc3csc(Cl)n3)C2)=O)nnc2n1CCCCC2 c1(C(N(C2C(N(C(CC3CC(C)C3)=O)C)CCCC2)C)=O)ccc(N)cc1Cl c1(OCC)ccc(NC(C2CC(F)CN(c3cc(C)ncn3)C2)=O)cc1I C1(C(=O)N)C(C2CC2)C1(F)F.S(=O)(=O)(CC(=O)NCC(C)(O)C)N(C)C c1(NC(C2CN(C(c3cc(C)cc(F)c3)=O)C2)=O)c(F)c(F)nc(F)c1F N1(C(CN(S(C)(=O)=O)C)=O)CCCC2(CCN(C(=O)CN3CCC(F)C3)C2)C1 N1(C(c2ccc(OC)c(Cl)n2)=O)CCC2CC1CN(C(c1ccc(Cl)o1)=O)C2 C1(CNC(c2n(CCC)cnc2)=O)CCCN(C(c2ncc(C)cc2C)=O)CC1 Cc1ccc(C)c(CC(N2CC3CC2C3NC(C23CSC(C2)C3)=O)=O)c1 N(C(=NCCCCl)N1CN(C)C(=O)C1C)Cc1c2cc(C)[nH]c2c(F)cc1 c1(CC(C)NC(=O)C(C)CN(C)C(c2c(Cl)cnn2C)=O)cnn(C)c1O C1(C(N2C(C)CC(Nc3cc(COC)nc(C)n3)C2)=O)Cc2cc(Cl)ccc2O1 C(=O)(C1=CS(=O)(=O)CCC1)NC1C(NC(C(CC(N)=O)O)=O)CCC1 C=C(C)CN=C(NCc1ccc(C(C)(C)C)s1)N(C)CC1CCC2(CC1)OCCO2 C(=O)(CCC(C)(C)C(=O)NCCC1CC1)OC.c1(C=O)ccc(=O)n(C)n1 C1(C(N(CC(C)NC(CC2(C=C)CC2)=O)C)=O)OCCN(C)C1=O c1(C(=O)N)cc2ccc(Cl)cc2[nH]1.C(F)(F)(C(F)(F)F)OCC(=O)NCC C1(NC(C(C)n2cccn2)=O)CC2CCC1N2C(C1CN(S(N)(=O)=O)C1)=O N1(CC)CC(CNC(c2cn(CC(O)CSC)nc2C)=O)(CC)CC1C c1(CC)ccc(C)c(C(=O)NCC(C(=O)N)N(C)C)c1.C12CCCC1CCO2.C n1(CC)nccc1C=CC(=O)NCCCCC(C)NC(=O)CCN1CCC(F)C1 c1(C(=O)NC2CN(C(CC=C(C)C)=O)CC2O)ccc(F)c(OC(F)(F)F)c1 Cn1nc(Br)c2c(N3CCCCC(NC(c4ccnc(F)c4Cl)=O)C3)ncnc12 c1(C(=O)OC)ccc(C)nc1N1CC(NC(C2CCCOCC2)=O)CCC1C OC1(CNC(c2cnc(-c3ccoc3)[nH]c2=N)=O)CCCC(O)C1O c1(C(N(CCC#C)CC)=O)n[nH]cc1CNC(c1ccco1)=O Cn1cnnc1COCC(=O)NCCc1cc[nH]c1 c1(C(=O)NCCOCCCNC(CC(CC)C)=O)cc(=O)c(O)c[nH]1 c1(N2CCC(c3sc(C(=O)OC)c(C)n3)C2)ccc([N+](=O)[O-])c(C(C)=O)c1 N1(C(c2cn(CCCC)nn2)=O)CC2CC2(CNC(=O)C(F)CC)C1 Cc1cc(N(CCCF)C)ncc1S(=O)(=O)NC(C(C)C)C(CO)C(C)C C(=O)(C(C)CC1CCCC1)N(C1CN(C2CC2)C1)C.C1(C(=O)N)CC(O)C1 CCC(O)CC(=O)N(CC(C)(C)C(=O)N1CCCC(CCCO)C1)C c1(C(=O)OCC)n[nH]c2c1CN(c1ncc3ccsc3n1)CC2.Cc1cnc(N)s1 c1(C(=O)NCc2ccc(Cl)cn2)c(OC(F)F)cccc1F c1(OC(C)C)cnccc1C(N1CCC(F)(CNC(=O)C(C)NC=O)C1)=O C(CC)(CC(=O)N(C(C)C)C1CC1)NC(c1cn(CCC)nc1)=O C1(C(=O)NCC(C2CCOC2)NC(C(CSC)C)=O)C2CCC1(C)C2(C)C Cc1cc(C(=O)NCC2CC(F)CN2C(=O)CC(C)C(C)C)nc(O)c1 C1(CC(=O)NCc2cnsc2)CC2(CC2)CN1C(=O)CC1CCSC1 c1(OC)cc(Cl)ccc1C(N1CC(OCCNC(=O)CCC(C)SC)C1)=O N1(C(C(C)C2CCCC2)=O)CCC(C2CCCN2C(c2cncn2C)=O)CC1 N1(C(C(CCCC)F)=O)CCCC(O)(CNC(c2ncsc2C)=O)CC1 N1(C(CSc2cccc(OC)c2)=O)CC(C(=O)NCCn2ccnc2)CC(C)C1 N1(CC(=O)NCC2(C)CCCC2)Cc2ccccc2C1.C12(C=O)CC(C1)C2.N c1(NC(=O)NCc2ccc3occc3c2)nccc2ccc(Br)cc12 N1(C(C(C)N(C(CSCC=C)=O)C)=O)CC2CCC(O)CC2C1 c1cc(F)c(Cl)cc1F.N1(CC(=O)NC)C(=O)CNC1=O.C1(CC=O)CCC1 c1(CC(=O)NC(C2CCCN2c2ncncc2I)(C)C)ccccc1Br c1(OC)c(Cl)cc(CN2CCCC(C(=O)NCCc3ccsc3)CC2)cc1Cl c1(CC(=O)NC2C(NC(Cc3cc(C)[nH]n3)=O)CCCC2)ccc2c[nH]nc2c1 C1(C(=O)NC(CC(=O)NC(CC)C)C)(CC)CCOCC1 c1(NC(CNC(=O)NC(CC)C)=O)ccc2cc(CO)ccc2c1 C=CCCC(C1CC1)NC(C1C=CCN1C(=O)CCc1ccsc1)=O C1(C(N2CC(C)C(NC(=O)CCC(F)F)C2)=O)Cc2ccccc2C(=O)O1 N1(C(CC(CNC(CN(C(COC)=O)C)=O)O)=O)CCN(C)CC1CCO C(c1cncn1C)=CC=O.C1(CC=C)(CNC(C2CC2C)=O)CCCC1 c1(C(N(CCN(C(=O)C=CCO)C)C)=O)cnc(C(C)(F)F)s1 C1(OC)CCN(CC(=O)NC2(NC(=O)CCc3cnccn3)CC2(C)C)C1 C(c1ccc(Br)c(Cl)c1)=CC(=O)N(CCNC(C(CCC)(C)C)=O)C c1(C(=O)NC23CC(CNC(C4CCCCC4F)=O)(C2)C3)cncc2nc[nH]c12 C1(NC(c2cnn(CC)n2)=O)COCCC1NC(c1ccccc1)=O.C(N)=O Cc1cc(F)cc(C)c1C(=O)NC1COC2(C1)CN(C(C1CCC(C)C1)=O)C2 C#CC(CC(C)(C)C)NC(C1CN(C(=O)C(C#N)CC)CC12CC2)=O C(C)(C)(CCN=c1[nH]nc(O)s1)NC(c1cc(C)nnc1O)=O CC(CC(=O)NC(CC(=O)N(C)CC1CC(F)(F)C1)C(F)F)C(F)F c1(CC)cc(C(=O)NCC2CCCN2C(c2cc3n(c2)CCC3)=O)cc(Cl)c1 c1(N2C(CC(=O)NCc3ccc(OCC)cc3)CCC2)ncccc1C#N n1(CC)ccc(C(=O)NC(C2CCN(C(=O)C(C)(C)F)C2)(C)C)c1C C#CCC(CC(F)(F)F)NC(=O)Nc1ccc(-c2cccc(C)c2)cc1 C1(N(C(CNC(C)=O)=O)C)CN(C(c2ncccc2Cl)=O)CC1F c1(C=O)cccc2cnsc12.C1(CC)CC(F)(F)CN1C(=O)C(F)CC1CC1.N c1(C(N2CCN(C(CC3CC(CC)C3)=O)C(CCO)C2)=O)cc(C)cc(C#N)c1 Cc1cccc(C2(C(N3CCC(C)C3C)=O)CC2)c1.C1(C)(C(=O)N)CCOCC1 C1(O)(CC)CCN(C(=O)CCc2ncc(C(C)(C)C)o2)C1.CC=O.C#CCS c1(OC)cc(C(N2CCC(C(=O)NCC3CCC(=O)O3)C(O)C2)=O)ccc1Cl C1(C(C)C)CN(C(C2CC2[N+](=O)[O-])=O)CCN1C(=O)CCSc1ccc(Cl)cc1 c1(CC)ccc(C(N2CC(CO)(NC(=O)CC3COCCO3)C2)=O)[nH]1 Cc1nc[nH]c1CNC(N1CC(N2CC(C)(C)C2)C1)=O c1(C(=O)NCC2CC3CC3N2C(=O)Cc2ncc(Cl)s2)n[nH]c2c1COCC2 Cc1cc(=O)n(C)nc1C(N1CCN(C(=O)Cc2cc(Cl)cnc2C)CC1C)=O CC(C)C(CNC(C1(C)CC(=O)N(C)C1)=O)C(=O)N1CCOC(C)C1CO Cc1cc2sc(C(=O)NC3(CNC(C45CCC4C5)=O)CCOCC3)cc2s1 c1(C(N2CCC(N(C(=O)Cc3cscn3)CC#C)C2)=O)ccc(C)cc1SC Cc1cc(C(=O)NC23CCC(C2)N(C(C2CC4CCC2O4)=O)C3)c(C)cc1Cl C1(NC(=O)CN2CCCCC2=O)CC2CN(C(c3ccc(Cl)c(Cl)c3)=O)CC12 C1(C(C(=O)O)O)CCCCN1CCCc1ccc(F)cc1 CC(C)(C(=O)NCC(CO)NC(=O)CN1CCNC1=O)n1ccnn1 c1(C=O)cc(Cl)c(O)c(Cl)c1.c1(OC)cccc(C(=O)NCC2CCCC2)n1 N1(C(C(C)N(C(C2CC(=O)C2(C)C)=O)C2CC2)=O)CCC(C)(CCO)CC1 c1(C(=O)NC(C(C)NC(CCSC)=O)C)ccc(C)c(Cl)c1Cl C12(C=O)CCCCC1CS(=O)(=O)C2.C1(C)(CC(=O)NCC)CCCCC1.CC C(C(=O)N1CCCC(C(N2CC(C)=C(C)C2)=O)C1)(C(C)C)OC c1(C(=O)NCC(CC)NC(c2sccc2F)=O)nnn(C(C)C)c1C C(CC1=CCN(Cc2ccccc2C(C)C)CC1)NC(CN(CCC)C)=O N=c1[nH]c(C(=O)N(C2CCNCC2)C2COC2)cs1 CC1(C)CCN(C(c2cnco2)=O)CC1CNC(=O)CC1=CCOCC1 c1(SCC(=O)CC2CCCCC2)ccc(F)c(F)c1.c1(CC)ccc(SC)cc1 C1(NC(=O)C=CBr)CCCC12CN(C(c1cncc(C(F)F)c1)=O)C2 C1(C(=O)NC(CN2CCN(C(c3cnc(C)[nH]3)=O)CC2)C)CCn2nncc2C1 CCCCCC(=O)NCC(=O)N(C)CC1COCCN1C(c1cc(Cl)ns1)=O CN=c1[nH]c(C(N2CCCC(CCC(=O)N)C2)=O)cs1.CCN(C1CC1)C(C)C C(=O)(C(O)CC(C)C)NCCN(C(C(COCC)C)=O)CCCN(C)C C1(C(=O)NCC2(NC(CC(C)(C)O)=O)CCOCC2)C(C)(C)CCCC1(C)C N1(C(CCCCCSC)=O)CC(C)N(C(=O)C(O)C(C)(C)C)CC1C N1(C(c2cc(C)c(C)o2)=O)CC2CCN(C(C3CCC(N(C)C)C3)=O)C(C2)C1 CCC(CC(F)(F)F)C(=O)N1CC(CNC(c2cnc(C)nc2OC)=O)C(C)C1 c1(CC)c(OC)cccc1C(=O)NC(C)(CNC(=O)CC1CCC1)CO C(=O)(CCC(C)(C)OC)NC(C(=O)NC1CC(=C)C1)CC N1(C(C(C)=C2CCC2)=O)CCN(C(c2cnn(C3CC3)c2C)=O)C2(CC2)C1 CCC(CNC(=O)C(c1cccs1)NC(=O)CC1CCN(C)C1=O)CCO C(=O)(C1Cc2ccc(Cl)cc21)N1CCCCC(NC(c2c(C)nc(C)s2)=O)C1 Cn1nccc1C1CC1C(=O)NC1CCC1NC(C1(CO)COC1)=O c1(N2CC3CN(C(C#C)=O)CC3C2)ncnc2cc(Br)ccc12 C=CCC(CC(=O)NC(C)C(C)(C)CN(C)C)NC(=O)C(C)(C)C(C)C C12CCC(CC1)NC(=O)C2.C(C(O)CO)N(C(=O)CSCC#N)C(C)C Cn1nc([N+](=O)[O-])cc1C(=O)NCC(CNC(c1cccc2[nH]ncc12)=O)CO C(CC(F)F)(C(=O)NCCC1CCCCC1)N(C(CCN(C)CC)=O)C Cc1noc(C2CC2)c1C(=O)NC1CCC1.c1(C=O)cn(CC(F)F)cn1.C C(=O)(C#CC1CCCC1)N1C(C(=O)NCc2c(C)nsc2)CNC(=O)C1 c1(COC)nc(C)ncc1C(N1CCC(O)(C(C)C)C1)=O.c1(C=O)cscn1 C(=O)(C(=O)N=c1ccn(CCCCC#N)[nH]1)OCc1cc(OC(CC)C)ncc1 c1(C(=O)NC(CNC(c2c(C)nc[nH]2)=O)CC(C)C)cc(F)cc(Cl)c1O N1(C(C2(CC)CC2)=O)CCCCC(CNC(c2ccc(-n3cncn3)cc2)=O)C1 c1nc(C)c(S(=O)(=O)N2CC(C)(CC(N3CCNC(=O)C3)=O)C2)s1.CC(=O)N C1(CCNC(C=CSC)=O)CN(C(c2ccc(CSC(F)F)o2)=O)CC1C Cc1cc(C(=O)NC(C2CCN(C(c3nn[nH]c3Cl)=O)C2)C)cs1 N1(C(C2C(CNC(c3cccc(C)c3N)=O)C2(C)C)=O)CCC(C)(C2CC2)C1 c1(OC)cccc(CCC(=O)NC(C2CCN(C(=O)C3=CCC3)C2)C)c1 N=c1ccc(C(N2CCCC2C2CCN(C(C3(C(F)(F)F)CC3)=O)C2)=O)c[nH]1 C1(NC(C(CC2CN(C(C(CSC)C)=O)C2)F)=O)CCCC1(C)CO c1(N2CC3C(NC(c4cnc(SC)nc4)=O)C3C2)ncnc(C)c1Br N1(C(C(CCC2CC2)NC(CCCOC(CCC)=O)=O)=O)CCC(O)C(C)C1 C(=O)(CCC(C)(C)C)NC(C)CCNC(c1[nH]ccc1-c1ccc(Br)cc1)=O C1(Nc2cc(C(=O)OC)sc2[N+](=O)[O-])CCC2(CC1)CCN(C)CC2 C12(CNC(COC3CCN(C(c4cn(C)nc4)=O)C3)=O)CCCN(CC1)C2 C#Cc1cncc(NC(=O)CC2CCCN(C(=O)C(C(C)C)SC)CC2)c1 C(=O)CCC(C)C.c1(OC)c[nH]nc1C(=O)NC1CC(OC(C)(C)C)C1.N c1(CC(=O)N(C(C)CN(C)C(C2CC(O)C2)=O)C)ccc(Cl)c2cccnc12 N1(Cc2c(C)ncs2)CCC2(CN(C(=O)COCc3ccns3)CC(C)O2)C1 C1(C(=O)NC2CCN(CCC)C2)C2CC1N(C(=O)Cc1cccnc1F)C2 Cc1[nH]nc2ccc(C(=O)NC3CN(C(C4C=CC=CC=C4)=O)CCC3C)cc12 N1(C(Cc2cc(C)sc2)=O)CCC(CNC(c2c[nH]c(=N)s2)=O)C(O)C1 C(C)(CNC(=O)CCC(F)F)(CC(C)C)NC(c1c(CC)nn[nH]1)=O C1(N)(C(=O)NC(C)CCc2ccncc2)CCS(=O)(=O)C1 C1(NC(C=CC)=O)(CNC(C2COCCO2)=O)CCC(F)(F)CC1 c1(CNC(=O)NC(C)Cc2nc[nH]n2)ccc(C2(O)COC2)cc1 c1(CCNC(c2c(Cl)ccc(C)c2)c2nnnn2C)ccc2c(=O)n(C)ccc2c1 c1(NC(c2n(C(CC)C)nnn2)c2csc(Br)n2)cnc2n1CCC2 C1(C(=O)NC(c2ccc(C)cc2)CNC(CCCC)=O)CC(O)CN1C C1(NC(=O)COc2ccon2)CCN(C(C2(O)CCSCC2)=O)CC12CCC2 C(=O)C(=O)N(O)C(C)C.C(C(C)Cn1cccn1)NC(C1CC(C(C)C)C1)=O C(CC(C)C)(C(=O)N1CCC1C(=O)N(C)C)NC(CCc1n(C)cnn1)=O c1(C(N2CCN(C(CC(CCC)O)=O)CC2)=O)sc2ccc(Cl)cc2c1C C12(NC(c3ccc(C(C)C)cc3)=O)CCC(CN(C(=O)CC3(C)CCCO3)C1)C2 Cc1cc(NC(=O)C(CC2CCCC2)NC(=O)OC(C)(C)C)cc(C)c1O N1(C(c2c(CNC(c3c(OC)ccnc3)=O)cc[nH]2)=O)CC(C)N(C)C(C)C1 Cn1c(NCc2nc(-c3c(Cl)cccc3Cl)no2)nc2c(Br)cccc12 C1(NC(CC2C(C)(C)C2)=O)CN(C(c2ccnc(C(F)(F)F)c2N)=O)CCC1F C1(CNC(C(Cc2ncn(C)c2)O)=O)C2CC1N(C(C1CCCCC1)=O)C2 C1(C(=O)NC(c2ccnn2C)C(=O)N(C2CC(C)OCC2)C)CC2(CCC2)CO1 N1(C(C=CC(=O)N(C)C)=O)CCC2CC1CN2C(c1cnc(S)n1C)=O N1(C(C(C)OC)=O)CC(C)(C)OCC1CNC(=O)CCc1scnc1C N1(C(C2C(CC)CCC2)=O)CCC(C2CCN(c3ccnc(COC)n3)C2)CC1 N1(C(CN2C(=O)CCCC2)=O)CCN(C(=O)C(F)(F)CO)CC1c1ccncc1 c1(C(N2CC(COC)N(C(=O)CO)CC2)=O)ccc(F)c2cccnc12 C#Cc1ccc(C(=O)NCCC(CNC(=O)C(C)=CC)OC)o1 C1CCN(C(=O)C=C(C)c2cccs2)CC1C.N1(CC)CCC(C(=O)NC)CC1 CC(C)CC(C(=O)NCCC)C(N)=O.c1(C(C(=O)N)(C)C)cc(F)cc(C#N)c1 C(=O)(C(CC(C)C)C(N)=O)NCC(CNC(c1ccc(C)c(Cl)c1)=O)O C(C(CC=C)C(=O)NOC1CCN(C)CC1)NC(Cc1c(C#C)cccc1)=O CCCCC(C(=O)NC1CN(C(C23CC(CO2)C3)=O)CC1O)C(C)C C1(NC(C(F)=CCC)=O)CCC(C(=O)NCCc2nnc(C)n2C)CC1 Cc1c(Br)ccc(F)c1C(N1CCN(C(=O)CC2CNC(=O)C2)CC1C)=O c1(C(=O)NC2C(NC(C(C)n3cncn3)=O)CCOC2)c[nH]cc(F)c1=O N1(C(CCC=C=C)=O)CCC(N(C(=O)CCNC(=O)COCC)C)C(C)C1 CN1C(=O)CCC1C(=O)NCCNC(c1cn(C)c(O)n1)=O C12(CNc3ccc(OCCOCC)nc3)CCC1CCN2C(=O)CC=O.O C1(C(N(CC(CN(C)C(C2CN3CCN2CC3)=O)O)C)=O)CCOCC12CCC2 CN1CCN(C(C23CCC(C)(C2)OC3)=O)C(CNC(C2CCCC(O)C2)=O)C1 C1(NC(CCC=C)=O)CN(C(=O)C(C)NC(c2ccco2)=O)CC2CC12 C1(CC)OCCC1NC(=O)CC(C)NC(=O)CC1CCOC1 c1(C(C)(C)C)ccc(C(N2CCC(C)(C(=O)NC(COC)CO)CC2)=O)cc1I C(=O)(C1=CC(O)C(NC(=O)C(CC)C(=O)OC)C1)NC(c1nccn1C)CC N1(C(C(CC)(C)O)=O)CC2CCC(C1)N2C(c1snc(O)c1Cl)=O C(=O)(CCCC(C)C)NCC(C(C)C)NC(C=COC)=O.C(C)(C)C.C=O.N c1(C(N2C(C(=O)OC)CCC2)=O)ccc(NCC(C)(F)C(C)C)nc1 N(C(=NCCNS(C)(=O)=O)N)CC1CCC(C(C)(C)C)O1.C1OCCC1(C)C C1(NC(CCCN=[N+]=[N-])=O)CN(C(C2CCCCC2O)=O)CCC12CCOCC2 CCC(CC(C)C)C(=O)N1CC(C(C(=O)NCC2CCOC(C)(C)C2)OC)C1 C1(CC)CCC(C)CN1C(=O)CSCCNC(c1ccc(C2CC2)o1)=O Cc1cccc(CC(N2CCCOC(CNC(C3(N(C)C)CC3)=O)C2)=O)c1F C1(c2ccccc2)(C(N(CC(C)NC(C(C)C2CC2)=O)C)=O)CC(O)C1 c1(OCCC)cnc(C(C(=O)NC2CC(F)(F)C2)N(C)CCC2CC2)s1 N1(CC2C(=C)C2)CCOc2ccccc2C1C(F)F C1(C(N(C)Cc2cccs2)=O)CCC(O)CN1C(=O)Cc1nccn1C Cc1cccc(OCC(=O)NCC2CCC2(C)C)c1.c1(C=O)snc(O)c1Cl.N c1(C(c2n(C(CC)C)nnn2)NCC2CSCCO2)nccc(Cl)c1F Cn1c(C(=O)NCCC(N2CC3CC3C3CC23)=O)cccc1=O C1(NC(C2CCN(C)C2)=O)(C)CCN(C(=O)Cc2cc(C(F)(F)F)co2)CC1 N1(C(c2c(CC)scc2)=O)CC2CC(C1)CN(C(c1cscc1C#N)=O)C2 C1(C(C)OC)CCN(C(=O)CC2CCCCC2NC(=O)CCCCC2CC2)CC1 c1ccccc1.C1(C)(C=O)CN(C(C2CCC2)=O)C1.C(C(=O)N)OCC.C CCCC(CCC)C(=O)N1CC(C(=O)NCC2(CN(C)C)CC2)C(F)(F)C1 CCC(C)(COC)C(=O)N1CCCC(NC(c2cc(CF)on2)=O)C1 Cc1cnc(CNC(=O)CCC2CCN(C(C3CC3Cl)=O)C2)o1 c1(C(=O)NCC(C)NC(c2c(CC)occ2C)=O)c[nH]cc(F)c1=O [SH](=O)(=O)c1ccc(F)cc1.N1(CC)CCC(C=O)CC1.C(C)C.[SH](C)(=O)=O c1(C(N2CCC(N(C(C(C)N3CCCC3)=O)C)CC2)=O)ccc2[nH]nc(Cl)c2c1 N1(C(c2nc(C#C)sc2)=O)CCC2CCN(C(=O)CCC(=O)N(C)C(C)C)C2C1 c1(CC)[nH]nc(C(N2CC3CC2(CNC(=O)CCC)C3)=O)c1Cl.C(C)(=O)O C(=O)(CCCC(=O)NC(CN=c1nc[nH]s1)C1CCCC1)NCCC c1(C(=O)NC2CC(NC(C(COC)O)=O)C2)cc(C)c2nc(C)nn2c1 c1(C(=O)NC2CN(C(c3c(C)c(N)ccc3)=O)CC23CC3)cc2scc(C)c2[nH]1 C(=O)(C(C(C)(C)C)NC(C1CCCCN1C)=O)NC(C)Cn1cnnc1 CN1CCC(N(C(=O)CC2CCN2C(c2ccn(C)n2)=O)C)C1 C1(CC)CN(C(C2(CC)COC2)=O)CCC1NC(C1CCCC12CCC2)=O C(=O)(CC1CCCc2ccccc21)N1C(C)CC(CNC(c2n[nH]c(=N)s2)=O)C1 N1(C(=O)NC2C(C)=C2)CCOCC1c1nnc(C2CC2)o1 Nc1nccc2cc(C(=O)NC3CCCN(C(=O)CC4CCCCC4)C3)ccc12 C#CCC(O)C(=O)N1CC(OCC(=O)NCCCC(C)O)C1 Cc1cc(N2CC3CC(NC(c4n[nH]c(O)n4)=O)C3C2)c(C#N)cc1[N+](=O)[O-] c1(C(N2CCN(C(CCCC#CC)=O)C(CO)C2)=O)ccc2nncn2c1 CC(C)C(C)C(CNC(c1ncccc1O)=O)NC(=O)CCc1ccncn1 C1(NC(Cc2cccc(COC)c2)=O)CCC(C)N(C(c2ccccn2)=O)C1 CN1CCN(C(c2cn(CCO)nn2)=O)CC1C(=O)NC(CC1CCC1)CO c1(C(=O)N)ccc2cnsc2c1.N1(C(C2C(CC(C)C)C2)=O)CCC(C)(CC)C1 C(=O)(C1=CCCOC1)N1CCC(CC)C1CNC(=O)C(O)CC1CCCCC1 c1(C(=O)NCCNC(c2c(OC)cc(F)cc2)=O)cccn2cnnc12 c1(OCCN2CCC(C(=O)NC3CCCC3CCCO)C2)ccc(F)cc1Cl CCCCCCC(C)C(=O)NCC(C(=O)N(CC(O)C(F)(F)F)C)N(C)C C=CC(C)(CCOC)C(=O)N.c1(C=O)cc(C)nn1C(F)F.C1CC(CC)C1 N1(C(C(C)(C)N(C)C)=O)CCOC(C)(CNC(C2(CO)CCOC2)=O)C1 C1(NC(=O)CC(F)(F)Cl)CC2CCCC12.c1(CC(=O)N)nnn(C(C)(C)C)n1 c1(C(N2CCC(CCOC)(NC(c3cncc(Cl)n3)=O)C2)=O)ccc(Cl)cc1F N1(C(C(COC)C)=O)CCC2(CC1)CC2NC(=O)CC1(CSC)CC1 C12(C(=O)NCCCC(=C)Cl)CCN(C(c3c[nH]c(=O)cn3)=O)CCC1C2 CCC(CC)CCC(=O)N1CCC(F)(C(=O)NCC(F)Br)C1 CC1(C)Cc2c(C(=O)NCC3CC(O)CCO3)cccc2O1 S(=O)(=O)(c1ccc(OC(F)(F)F)cc1)Nc1ccc(C)cn1 c1(C(=O)NCC2N(C(CC=CCCCCC)=O)CC=C2)cccc([N+](=O)[O-])c1Cl N1(C(C2(OC)CCCC2)=O)CCC(O)(C(C)NC(c2ccnc(C)n2)=O)C1 C1(N(C(Cn2c(C)ccn2)=O)C)CN(C(=O)C(c2cccnc2)O)CC1(C)C c1(C(=O)NC2C(NC(CC(C)N(C)C)=O)CCC2)csc(S(N)(=O)=O)c1 C1(C(N2C(C)COC(C(F)(F)F)C2)=O)CCC2S(=O)(=O)CCC12 Cc1c(C(N2CCC(N(C3CCN(C)CC3)C)CC2)=O)ccc(Br)c1Cl CC1OCCN(C(=O)CCCNC(C2CCS(=O)CC2)=O)C1CO N1(C(CC(=C)C)=O)CCC2(CC1)CC(NC(=O)C(CCSC)N(C)C)CCO2 CCCCC(CC(=O)NCC12CC(F)(C1)C2)NC(c1c[nH]nc1CC)=O Cc1cccc(C(N2CC(O)CC2C(=O)NCC2CN(C)C2)=O)c1Br C1(C(=O)NC(COC)CNC(=O)CCC2CC2C)CC12CCC(=O)CC2 Cc1ncc(C(N2CCC(NC(=O)CSCCN(C)C)C2C)=O)n1C C(C)(N=c1[nH]c(=NCC2(N(C)C)CC2)c2c(F)cccc2[nH]1)c1c(C)cccc1 C#CCCCCC(=O)N(C)CCOCCNC(=O)CCNC(=O)OCC CC1(C)CCCCN(C(C2CN(C(=O)C3=CC4C=CC3C4)CC23CC3)=O)C1 C1(NC(=O)C2CC2)CCC2(CC1)CN(C(C1CCC3CC3CC1)=O)CCO2 C(=O)(C1=CCCC(C)(C)C1)NCC1C(NC(c2ccc(C=C)cc2)=O)CCC1 C1(NC(C(C)OCCOC)=O)CCCCCN(C(=O)C(C)(C)CC(F)F)C1 N1(C(c2c(C)cncc2)=O)CCC2CN(C(=O)C=CC3CCCN3C)C2C1 c1(C(N2CC(NC(CCNC(C(C)(C)C)=O)=O)C3C2C3)=O)ccc2nc[nH]c2n1 c1(C(=O)NCC(CCOC)NC(CSCC=C)=O)nccn2c(C)nnc12 C1(OC)CCCC(CNC(=O)CN(C(=O)Cc2conc2C)C2CC2)C1 c1(CNC(=O)C=CC2CCC2)ccc(C)cc1F.C1(C=O)CC2(CCC2)CO1 c1(C(=O)NCC(CC=C)C(=O)N2CC3CCCC3C2)ccc2c[nH]nc2c1 C12(CNC(c3[nH]cc(CC)c3)=O)CCCC1CCN2C(c1cnncc1O)=O C1(NC(CCN(C(=O)Cc2ccccc2Br)CC)=O)CCCC(CO)C1 C1(NC(c2c(C)nc(C(C)(C)C)s2)=O)CCCCN(C(c2cnnn2C)=O)C1 N1(C(CCOCCC)=O)CC2(CC(C(=O)N(CC(F)(F)Cl)C)CO2)C1 C#Cc1ccc(C(=O)NC2CCN(C(C3C(C)(C)C3(F)F)=O)C2(C)C)c(F)c1Cl CC1CCN(C(c2ccc3c(c2)COC3)=O)CCN1C(C1OCC1(C)C)=O C1(C)(CC(=O)NCCN(CC(F)F)C)CCN(C(c2cc(Cl)cn2C)=O)C1 N1(C(c2c(C)n(C)cn2)=O)CC2CCC2(CNC(=O)C=C2CCSCC2)C1 C(c1ccc(Cl)c(F)c1)=CC(=O)NC(c1cncc(Br)c1)C c1(C(N2CC(C(C)NC(COC3C(C)CCCC3)=O)C2)=O)ccc(O)c(F)c1F N1(C(C(c2cc(C)oc2C)C)=O)CC2OCCN(C(c3cccc(O)c3)=O)C2C1 Cn1nnnc1C(C)(CC1CCC1)NCCC1(C)CCCO1 C12CC(CCO1)N(C(C1CC13CC(F)(F)C3)=O)C2.C1(C(=O)N)CC1(F)F.C O(NC(=O)C(C1CCC1)NC(=O)CCCC1CCCO1)CC(=O)OC N1(C(c2nc(OC)c(C)s2)=O)CCC(NC(=O)CCC2CCCOC2)C(O)C1 C1(NC(C(CC)N2CCCC2=O)=O)(CF)CCN(C(c2cc(Cl)no2)=O)C1 N1(C(CC2CCN(C)C2)=O)CCSCC1CCNC(=O)CCc1cccnc1 C12(C(=O)NCC(C3CCOC3)NC(Cc3ccn(C)n3)=O)COCC(C1)C2 C(=O)(CCCCCN(C)C)NC(C1CCN(C(c2cc(OC)n(C)n2)=O)C1)(C)C CC(C)S(=O)(=O)C(C)C(=O)NCCCNC.c1cn(C)nc1C(=O)N(C)C C1(C(N(CCC)C)=O)CCN(C(=O)C(C(=O)OC)OC)C1C(C)C CC#CC1CCN(C(=O)C(C2(O)CN(C(c3ccnn3C(C)C)=O)C2)F)C1 c1(C(=O)N)ccc(S(=O)(=O)N(C)C)cc1.C1CCCC1.C1(C=O)CC1C1CC1 C1(NC(Cc2cc(C)[nH]n2)=O)CCN(C(C2CCC=CO2)=O)CC1 c1(C(=O)NC(CCNC(c2c(CC)nn(C)c2)=O)C)cccc(C(C)C)c1N CC(C(=O)N(C1CC(NC(=O)CCC(=O)N(C)C)C1)C)C(F)(F)C(F)F N1(C(CN(CCOC)C)=O)CCC2CC2CC1.c1(C(=O)N)cnc(C(N)=O)cn1 N1(C(C23C(CN(C(=O)Cc4cccnc4O)C2)C3)=O)Cc2cccc(F)c2C1 CC1(C)CN(C(=O)C(C2CC2)C2CC2)CC2(CN(C)C2)O1.C12CC3CC1C2C3 C(CC(C)(C)C(=O)N1CC(O)(C2CC2)C1)NC(CCSCCC)=O C(=O)C(F)C(F)(F)F.C(CC(C(=O)NCC1(C)CCCCC1)N(C)C)N(C)C C12(C(=O)NCCC(C)NC(CSCC=C)=O)CC(C(C)C)(C1)C2 CC1CN(C(C2SCCS2)=O)CC1C(=O)N(C1CC=CC1)C C(C1=NOC2CN(C(c3ncc(Cl)cc3F)=O)CC12)NC(C(=O)NC1CC1)=O C(=O)(C1=CCCCO1)NCCN(C(CC(C)C1CCCO1)=O)CC1CC1 N1(C(C(CCF)NC(Cc2cc(C)[nH]n2)=O)=O)CC(C)(C)CCC1CO CC1CN(C(C2(c3ccccc3)CC2(C)C)=O)CCN1C(=O)C1=CC(C)(C)C1 Cc1ccc([SH](=O)=O)cc1.C1(C(N(CC)C(C)C)=O)C2CCC12.C(C=O)N c1(OC)cc(C)ccc1CNC(=O)NCCC1(CO)CC1(F)F Cc1nc(C)n(CCC(=O)NC2C3CN(C(C4CCC(C(F)(F)F)O4)=O)CC23)n1 c1(N2CC(CC(C)NC(c3cccn3C)=O)C2)ncc(C#N)cc1F c1(C(C(=O)NCC)N(CC=C)CCOC)cc(Br)c(O)cc1.C(C)(C)C c1(C(=O)NC2CCC(NC(C3C(C)C3)=O)CC2)cc(Br)cnc1N c1(OCC)cc(Br)cc(C(=O)N(c2cccc(F)c2C#N)CC)c1N CC1CC(CC(=O)NCC2=NOCC2)CN1C(=O)CCCn1cccc1 c1(C(c2cn(CC(=O)NC(CC)CC3CC3)nn2)O)ccccc1F N1(C(C2(CC)CN(C(=O)CC3CCN(C)C3=O)C2)=O)CCOC2CC12 C(=O)(CC1=NNC(=O)C1)N(C)CC1C(CO)CN(C(C(SC)SC)=O)C1 C(=O)(C(F)C(C)(C)O)NC(C)C=CC(=O)NCCCC1CCOCC1 CN=c1ccc(C(=O)NC(C2CN(C(c3n[nH]cc3OC)=O)CCO2)C)c[nH]1 N1(C(C(C)OCC)=O)CCC(O)(CNC(C2(CCF)CCC2)=O)C1 c1(C(N2CCC(C)(CCNC(CC(CC)(C)C)=O)C2)=O)cnc2n1CCC(C)C2 C1(C(N(CC)Cc2cncn2C)=O)CCN(C(=O)CS(=O)CC)C1C Cc1cc(C(=O)NC2CC3CCC(C2)N3C(=O)C=CC2CCC2)c(N)c(C)c1 C=CCCCCCC(=O)N(CCCNC(c1cncc(N)c1)=O)CCO C(C(C(=O)NCCN1CCC(CO)C1)C(C)(C)C)NC(CN1C(C)CCC1)=O C(=O)(CC(C)(C)C(=O)N1CCCC(O)C1)OCC.C(=O)C(CN(C)C)CC.C C(=O)C1=NOCC1.c1(C(=O)Nc2c(OCC)cccc2)ccc([N+](=O)[O-])o1.C C12(OC)CCC(C(=O)NCCCNC(c3cnc(C)cc3Cl)=O)(CC1)CC2 C1(CC)CN(C)CCCN1C(c1ccc(CNC(=O)C(O)CCC(C)C)s1)=O c1(C(N2CC(N(C(C3(CCCC)CC3)=O)CC)C2)=O)sc(N2CCCC2)nc1Cl c1(CCC(=O)NC2(C)CC(NC(C(c3ccccc3)OC)=O)C2)ccncc1Br CCC(CC)C(C(=O)N(C)CCNC(c1cnn(C(F)F)c1)=O)OC C1(CN2CCCC(c3ccc(OC)cc3OC)C2)CCn2ccnc2C1 N1(C(c2nc(COC)sc2)=O)CC(F)(F)CC1C.C1(C=O)CC(C)(C)C1 n1(C(CC)C)ncc(C(=O)NC(C)CC)c1C1CC1.c1(C(=O)N)cc(C)on1 c1(C(C)C)c[nH]nc1C(=O)NCC(O)CN(C)C(C1(CO)CC1)=O C(CCCCC(=O)NC(CC(N)=O)C(=O)NCC(O)(CO)CO)OCC N1(C(CN(CC)CC)=O)CC2(CCC2NC(=O)CSc2ccccc2Cl)C1 C1(NC(Cc2ccc(CC)cn2)=O)CC(C)CN(Cc2cccc(O)c2Br)C1 C=CCC(CC(C)C)C(=O)NC1(CNC(c2c(N)cccc2Cl)=O)CCC1 N1(C(c2c(C)cn(C)n2)=O)CCCN(C(c2ccn3nccc3n2)=O)C(C)C1 N1(C(C(C)C)=O)CCOC2(CCN(C(C3(CC(C)C)COC3)=O)C2)C1 C1(NC(C2(C(C)(C)C)CCC2)=O)CCCCC1.c1(C(=O)N)ccc(CC#N)cc1 c1(CC(=O)OCCCN(C)C)ccc(S(=O)(=O)CN2CCOC2=O)cc1 C12(C(N(CCC(C)NC(c3cnc(CCC)s3)=O)C)=O)CCC(C)(CC1)OC2 N1(C(c2cc(CCC)[nH]n2)=O)CCCC1C.c1(C(=O)N)nc(C)c(C(F)(F)F)s1 Cc1cccc(CN2C3CCC(C3)C2C(=O)Oc2ccc(CN(C)C)cc2)c1C C1CCCC2CN(C(C3(S(N)(=O)=O)CC3)=O)CC12.Nc1cc(=O)nc(C=O)[nH]1.N c1(C(=O)N)ccc2ncccc2c1.CC1CCC(C)(C(=O)NCC2CC2)C1(C)C N12CCCCC1C2=O.O=C1CN(Cc2ccncc2)C(=O)N1C1CC1 N1(C(CCCC)=O)CCCN(CCNC(=O)C(c2c(F)cccc2F)(C)C)CC1 C1CCCCC1.C1(N(C(=O)CS)CCC)CCN(C(=O)C(C)c2ccsn2)C1.C C=C(C)CCCC(=O)NCC1CCN1C(C1CC2(CCC2)CO1)=O c1(C(=O)N)cccc(O)c1.c1(C(C)=O)cc(C(=O)NC(c2ccccc2)C)cs1 c1(CC)ccc(F)cc1C(N1CCCC1C)=O.C(=O)C(C1CC1)N(C)C.N C1(C(N(C2CCN(C(c3c[nH]c(Br)c3)=O)CC2)C)=O)CC(C2CC2)=NO1 C(=O)(C(C)C(O)CCCC)NC(C(=O)NC1(C#C)CCOC1)Cc1ccoc1 Cc1ccc(C(=O)NCCC2CCC2)c([N+](=O)[O-])c1.C1(C=O)CNC(=O)C1.N c1(OC)c(NC(C2C=CCN2C(c2cc(C)ccc2OC)=O)=O)cc(Br)cc1F c1(C(N2CCC(CCNC(COCc3n(C)ncc3)=O)C2)=O)c[nH]c(=O)cn1 N1(C(=O)Nc2cccc(C(=O)NC)c2)C2C=CC1c1ccccc12 c1(OC)ccc(CC(N2CCCCC2C2CNC(=O)C2)=O)c(C(F)(F)F)c1 C1(C(N2C3CN(Cc4n(C)ncc4)C(C3)C2)=O)COc2ccccc2O1 N1(C(C2OCC(C)(C)OC2)=O)CCC2(CC1)CC2NC(C1CC(N(C)C)C1)=O c1(C(=O)NCC2N(C(c3ccc(CN=[N+]=[N-])o3)=O)CCCC2)cc(N)ccc1O C(=O)(CC(C)NC(=O)C(F)(F)C1CCOCC1)NCC(C)=O CC1(O)CN(C(=O)CC2CCC(NC(c3cc(C(N)=O)co3)=O)C2)C1 Cc1coc(C=CC(=O)NC2CCOCC2NC(=O)CC2CCCC2O)n1 S(=O)(=O)(c1cc(C(=O)O)cc(Cl)c1)NC(CC)C(c1c(F)cccc1Cl)O c1(C(=O)NC2C(C)CN(C(=O)CN3CC=CC3)CC2)cc2occc2n1C C(=O)(C1=CCCC1C)NC(COC)C(=O)NCC1C2COCC12 c1(C(N2CC(NC(c3nc(C)sc3)=O)C(CO)CC2)=O)cc(O)ccc1[N+](=O)[O-] Cc1nnnn1CC(=O)NC(c1cccnc1)C(=O)NCC(C)O Cc1cc(Br)cc(C)c1CC(=O)NCC(CO)NC(=O)Cc1cnn(C)c1 C12(C(=O)N)CCC(CC1)CO2.c1(CC)ncccc1C(=O)NC1CCC(C)C1 C1(C(N2CC(N(C(=O)C=Cc3cc[nH]c3)C)C2)=O)CCOC(C)(C)C1 C1(OC)CC2CC(NC(C3CC4CCC3N4C(c3cnccc3C)=O)=O)CC12 N1(CC)CCCCC1C(N1CCCC1(C)CNC(=O)CCCCSC)=O CC1(C(N2CC(O)C2)=O)CCN1C(=O)Cc1nc(Cl)cs1 c1(OC)ccc2c(c1)OCC(NC1CC1c1cccc(C)c1F)C2 c1(C(=O)NC(C(C)NC(c2coc(N(C)C)n2)=O)CO)cc(N)c(O)c(F)c1 c1(N(C2CC3CC2CN3)C(C2N(C)CCOC2)=O)nc(O)ncc1I c1(CNC(c2n(CCC3(C)CC3)nnn2)C2CCSC2)ccnc(F)c1F Cc1nc(N2CC(C)(NC(C3CCS(=O)(=O)N3)=O)C2)ncc1[N+](=O)[O-] CCCCC(CC)CC(=O)N1CCC(C)(C(N2CCCC(OC)CC2)=O)C1 N1(C(=O)C=CCF)CCN(C(=O)CC2CCCN2C(c2cc(Cl)ns2)=O)CC1 N1(C(C(CO)NC(CCn2ncc(C)c2)=O)=O)Cc2ccnn2CC1C c1(CC(N2C(CNC(C(CC)C(C)C)=O)CC2)=O)ccc(C)c([N+](=O)[O-])c1 c1(C(N(CCCCN(C(=O)CCc2cn[nH]c2)C)C)=O)nccc2c[nH]nc12 c1(OC)ccc2c(CC(N3CCCC(NC(C4CC4C(F)F)=O)C3)=O)c[nH]c2c1 C1(NC(c2c(C)cnn2C)=O)CC(C)CN(C(=O)C)C1.c1cc(Cl)cc(Cl)c1.S c1(CNC(CC(C=C)C)=O)nnc2n1CCN(C(=O)C(F)(F)C(O)CC)C2 N1(C(c2ccc(OC)cn2)=O)CC(NC(c2cnn(C)n2)=O)CC12CCCOC2 n1(CC(=O)OCC)cc(C2CCN(C(=O)C(c3cnn(C)c3)OC)C2)nn1 c1(-n2ncc(SCCNC(C3CC3)=O)c2)ccc(F)cc1F.c1(N)ccccn1 C(=O)(CS(=O)CCC(F)(F)F)NC(CNC(c1ccc(C)c(C)n1)=O)C C(C)(N=c1[nH]c(=NCCC2CC(F)C2)[nH]c2ccsc12)c1c(C)nc(C)s1 c1(C(=O)NCC2N(C(C=CC=CC)=O)CCC2)cccc2c1OCC2 N1(C(CCCC=C)=O)CCC2CN(C(C34CC3COC4(C)C)=O)CC12 Cc1ncc([N+](=O)[O-])cc1C(=O)NC1(C)CCN(c2nc3ccc(F)cc3s2)C1 C1(COC)CCC(NC(=O)C(C2CCC2)NC(=O)CSC(F)(F)F)C1 C12(CCCCC1)CC(=O)NCCCS2.N1(CC)CCC1C(=O)O.C(C)(C)C N1(C(Cc2cc(OC)no2)=O)CCCC(C(C)NC(=O)CC(F)(F)Cl)C1 C=C=CC(C)C(=O)NC1COCCC1C(=O)Nc1cccc(CCC)c1 N1(C(Cn2c(C)ncc2)=O)CCCN(C(C2(C)CCCCO2)=O)CCC1 Cc1ccc(C=CCC(=O)NC(C)C(CO)NC(=O)CCc2cccnc2)cc1 CC12CCN(CC(CO)Oc3ccccc3)C1CNC2 N1(C(CCOCCOC)=O)CCC(C)(C(=O)NC(C2CCCC2)C)CC1 c1(C(=O)N)c(N)cc(F)cc1F.C(C(=O)NC(C)CC)(C1CCCC1)OCC C1(C(N2CC(C)C(NC(c3cc(Cl)nnc3O)=O)C2)=O)CN(S(N)(=O)=O)C1 C1(NC(=O)C=O)CC(C(=O)NCC2CC2)C12CCC2.c1(CC)ccc[nH]1.N N1(C(COCCC)=O)CC(OC)CC1C(=O)NCCC1CC(C)(C)CO1 C1(C(N2CC(CCNC(C=CSC)=O)OCCC2)=O)Cc2cccc(C)c2O1 C#CC1(C(=O)NCCCOCC=C)CN(C(=O)CC(C)C2CC2)C1 C1CN(C(C2CC23CC(C)(C)C3)=O)CCC1(C)C.C(=O)(CCCC(=O)NC)NC c1(C=O)csc([N+](=O)[O-])c1.c1(C(C(N2CC(=C(C)F)C2)=O)=O)ccc(F)cc1 CCCCCCCCC(=O)NCC1CC1NC(=O)C(CO)OC C1(C)(C(N2CC(COC)C2)=O)CCCCC1C.c1(C=O)ccc(C(C)C)o1.C C=CC1(C(=O)NCC2CCCN(C(=O)CCc3ccco3)C2)CCCC1 Cn1cnc(C=CC(=O)NC2CC2NC(=O)CC2CC3CCC2O3)c1 CC(C)(F)C(C)(F)C(=O)NC1CC1NC(=O)CCc1ccncn1 c1(C2(C(N3CC(OC)(C)C3)=O)CC2)ccccc1C#N.C(=O)(C1=CCCSC1)N C1(C(N(CCC(=O)NC2CCOCC2C)C(C)C)=O)CC2CCCC2C1 CCCC(CCC)C(=O)NCC(C1CCCCC1)NC(C1CCOC1(C)C)=O Cc1cc(C(=O)N(C)Cc2ccccc2CNC(C2C3COCC23)=O)cn1C C(=O)(C1=CCc2ccccc21)NC1(CNC(C=C(C)c2ccsc2)=O)CCOC1 C1(C(=O)NCC(C)NC(c2cc3ccccn3n2)=O)CCCC2(C1)CC2(F)F c1(OC)ccc(CNC(=O)C(CCF)NC(=O)CC2CCOC2(C)C)nc1 c1(C(C(N2CC(NC(CCN(C)CC)=O)C(C)C2)=O)O)cc(Cl)cc(Cl)c1 Cn1ccc(C(=O)NCCNC(C2(c3ccc(Cl)c(F)c3)CC2)=O)cc1=O c1(C(N2C(C)CC2C(=O)NOCCSc2ccccn2)=O)cccc(F)c1F CCC(CC(=O)N1CCC(F)(C(N2CC(C)=C(C)C2)=O)C1)C(C)C Cc1ncnc(C(N2CCC(F)(C(=O)Nc3ccc(F)cc3O)C2)=O)c1C C1CN(C(=O)CCc2cncn2C)CC(C)(C)O1.C(C(=O)N)(C(C)(C)C)OC.C N1(C(C2NC(=O)OC2)=O)CCC(C(c2csc(Cl)n2)=O)CC1.C12CCCN1C2 c1(OC)ccccc1C(CNC(=O)C=CCF)NC(C1CC1F)=O c1(CC)occc1C(=O)NC1(CC)CN(C(=O)C(O)CC2CCOCC2)C1 CC1CN(C(C2C3COCC23)=O)CCC1CNC(=O)CS(C)(=O)=O c1(NC(CC(COC)C)=O)ccc(-c2cn(CCCCC(=O)NC)nn2)c(C)c1 C(=O)(C1=NOC(c2ccccc2)C1)C(C=C(CC)CC)=O.C1(N)(CO)CCNC1 C=CC(CC)C(=O)NCC(C)NC(=O)CCNC(=O)CC(C)C C1(C(=O)NCC2OCCN(CC)C2)CC(F)CCN1C(c1ccnnc1O)=O C1(O)(CN(C(C2ON=C(C)C2)=O)C)CCN(C(c2cnn(C(C)C)c2)=O)C1 N1(C(CCC2CC(C)C2)=O)CC(O)(c2cc[nH]n2)C1.c12cn(nn1)C2C n1(CC(=O)NC(CN(C)C(C2CCCOC2)=O)(C)C)cc(Br)cn1 c1(C=O)ccc(C2CC2)cn1.C(=O)(C(C)(O)Cc1ccccc1)N(CC)CC S(=O)(=O)(c1ccc(NCCN(C)C)cc1)SC(CC1C(C)C1)C(=O)O CC1CN(C(c2ccc(C(F)F)o2)=O)CC(C)N(C(c2cnc(C#N)s2)=O)C1 c1(C(=O)NC2CCN(C(c3cc(C)[nH]c3C)=O)C23CC3)ccc2c(C)noc2n1 c1(OC)ccccc1C(=O)NCCC(O)CNC(C1CCCOCC1)=O Cc1cccc(C(=O)NCCSCC(C)(C)N(C)C)c1C.C1CC(=O)N1C c1(N2C(C(=O)Nc3ncc(Br)nc3Br)CC(O)C2)ncnc2sc(Br)cc12 c1(C(N)=O)cccc(CC(N2CCN(C(C3(F)CCCC3)=O)CC2CO)=O)c1Cl CN1CCN(C(C2CC(=O)N2)=O)C(CNC(=O)CCN2CCCC2=O)C1 N1(C(C(COCC)C)=O)CCC(O)(CN(C)C(c2[nH]c(O)nc2C)=O)C1 C1(C(=O)NCC(C)NC(=O)CC2CC2(C)C)CCCCN1N=O Cc1ccc(C(C)C)c(C(=O)NC2CCCC2NC(C2(C3CCC3)CC2)=O)c1 N1(CC(C)N(C)C(C2(C(F)F)CCCC2)=O)CCc2ccccc2C1 CN1CCN(Cc2ccc(C(=O)O)nc2F)C(CCO)C1 c1(C(=O)OCC)cccc(C(N2CC(O)CC2C)=O)n1.C(=O)C=CC C(CCCNC(=O)C(C)O)OC.CC(F)(F)F.C1(C=O)CC(=C2CC2)C1 C[Si]1(C)CCC(CNC(=O)CC2CCN2C(=O)Cc2cnoc2)C1 c1(C(=O)NC(CCN(C(c2ccc(C)nc2)=O)C)C)ccc(=O)n(CCF)n1 N1(C(C(C)OCCC(C)C)=O)CC2CN(C(C3CCCC(=O)N3C)=O)CC2C1 CC1C(C)N(C(=O)CC2(C(F)F)CC2)CCN1C(=O)C1=C(Cl)CCOC1 N1(C(=O)NCC2N(CC)C(=O)CC2)CCCn2nccc21 C1(C2(O)CN(C(=O)Cc3nccn3C)C2)(CNC(CC(CC)C2CCC2)=O)CC1 C12(NC(C(C)SC)=O)CCCC1N(C(=O)C=Cc1ncccc1C)CCC2 c1(C(=O)NCC(C)(O)C)ccc(=N)[nH]c1Cl.c1(C(C(=O)N)(C)F)ccccc1F C1(NC(COCCCCC)=O)CCN(C(c2cc3scnc3[nH]2)=O)CC1C(C)C C1(F)(C(=O)NC(CC)CNC(=O)C(C)(C)c2ccn(C)n2)CC12CCCCC2 CC1(C)C(C(=O)NC)CC1O.N1(CCC=O)C(=O)CCC1=O.C1(CC)CC1 CC(O)C(C(=O)NCC=CC(C)(C)C)NC(=O)Cc1ccccc1 c1(C(C(=O)NC(C2CCN(C(c3cncc(Cl)c3)=O)C2)C)C)c(F)cccc1F C1(CCOc2ccc(CC)cc2)CCN(C(C2CCCCS2(=O)=O)=O)C12CC2 CC1=CCC(C)(C(N2CC3(C2)CN(C(c2snc(O)c2Cl)=O)C3)=O)CC1 N1(C(C(C2CCOC2)OCC)=O)CCC(C)C1CNC(c1cccnc1)=O n1(CCC)nc(C)cc1C(=O)NC1CC(N(C)C(c2nonc2N)=O)C1 Cc1cn2c(n1)CC(C(=O)NCCCO)C2.C1(C=O)CCOC1C1CC1.CC N(C(=NCC(C)(C)C(O)(CC)CC)NCC1CCS(=O)(=O)C(C)C1)C(CC)CC C(=O)(C(C)(F)C(C)(C)F)N1CC(C)C(CNC(c2ccc(C#N)[nH]2)=O)C1 c1(C(=O)NC2CCN(C(c3nc(C(C)C)sc3)=O)C2)cc(O)c2ccsc2c1 C1(NC(C(=O)NC(C)C)=O)CCC2CN(C(C3CCCCC3(C)C)=O)CC2C1 N1(C(c2ccc(N=[N+]=[N-])cn2)=O)CC2(CCC(N3CC4C(C3)C4(F)F)CC2)C1 C=CCC(C(=O)NC1CN(C(=O)C(C(C)C)NC(C)=O)C1)c1ccccc1 C1(C(=O)NCC(C)C2CCC2)CCCN(C(=O)C2=CCCCC2)C1C c1(C(=O)NC2(CC(=O)NCCC3CCCN(C)C3)CCC2)ccc(F)c(O)c1 C=C=C(C)CC(=O)NC(C1CCOC1)CNC(c1cnccc1OC)=O N1(C(C2N(C)CC(O)C2)=O)CC=C(CNC(=O)CN2CCOCC2=O)CC1 CC1CN(C(C2(Cl)CC2)=O)CCC1CNC(=O)CN1C(C)CCC1C C1CC(F)(F)C1.c1(C(=O)NC2CCC2)csc(C(F)(F)F)c1.C(=O)C.N CCCC(CNC(C1CCOC1)=O)C(=O)NCC1(CCCO)CC1 C(=O)(C(C#N)C(C)C)NCC(CC(=O)NCC(CC)N(C)C)C1CCC1 Cc1cc(C)c(CNC2(c3nnnn3C3CCOC3)CCC(=O)NC2)cc1Cl c1(C(=O)NCC(C)CN(C(=O)CC)C)occc1F.n1(CC=O)cnnn1.N O=C(C(C1CCCC1)C(=O)NC1(c2cncs2)CC1)N1CC(N2CCC2)C1 C1(NC(COCCCC)=O)CCC(CNC(=O)CCCN(C)C(C)C)C1 C12(C3(NC(NOC(C(=O)OC(C)(C)C)C)=O)CC3)CC(CO1)C2 Cn1cc([N+](=O)[O-])cc1C(N1CCCC1C)=O.c1(C2(C=O)CC2)ccncc1.N CCC(C)CCCC(=O)NC1(CCCNC(c2cc(C)c(C(N)=O)cn2)=O)CC1 C#CCCCCC(=O)N1CC(C)(NC(=O)CC23COC(CF)(C2)C3)C1 Cc1cc(C)c(NC(=O)N(CC(C)(C)O)C2CCCC2)c(F)c1 C(CN=c1[nH]ccc2ccccc12)NC1(CC(N)=O)CCC1 C1(C(C)NC(C2(n3cccn3)CCCC2)=O)COCCN1C(=O)CCCC#N C1(O)(CN(C(c2c(CC)scc2)=O)C)CCN(C(C2CCC(C)(C)C2)=O)CC1 C(=O)(C(C)C(O)CC(C)C)NC1CCN(C(c2csc(C)c2C)=O)CC1 C12(NC(COCCC(C)C)=O)CCN(C(=O)C=Cc3cc[nH]n3)CCC1C2 C(=O)(C1=C(C)N(C)c2nnnn2C1C)NC(CCNC(C(CSC)C)=O)C(C)C c1(C(=O)OC)ccc(CNc2cc(Cl)ccc2-n2cncn2)c(F)n1 c1(C(=O)NCC(CNC(C(CC2CC2)OC)=O)O)sc2ncccc2c1Cl c1(NC(C2CCCN(Cc3cccnc3)C2)=O)ccc(I)cc1 Cc1cc(C)n(Cc2ccc(CNC(C3CCCCN3C(C)C)=O)o2)n1 N1(C(c2cc(C)[nH]c2C)=O)CCCN(C(c2cnsn2)=O)C(C(C)C)C1 C1(C(N(CC(CC)C)C)=O)CSCN1C(C1(n2cnnn2)CC1)=O C1(CC(C)(C)C)CCN(C(=O)CCOC2CN(C(=O)CC3(C)CC3)C2)C1 N1(CCc2ncc(C)o2)C(=O)C(C2CC2(C)C)N(C)C1=O c1(CC(C(N2CC(C)C(NC(=O)CN3CCCC3=O)C2)=O)C)ccc(C#N)cc1 C(=O)(CC1=CCN(C(C2CCC3(CC3)C2)=O)CC1)N1C(CSC)CCC1 C1(NC(C2(C)CCC(C)C2)=O)CCCCN(C(=O)Cn2ccsc2=N)C1 CC1CN(C(=O)CC2OCCO2)CCCN1C(=O)CCSCc1ccccn1 c1(C(N2C(CCNC(CC3(C=C)CCC3)=O)CC(OC)C2)=O)ccc(O)c(F)c1 c1(CC)ncc(C(=O)NC2CCC(CCNC(=O)C3=CCC3)C2)cn1 c1(NC2C(NC(CCc3ccc(C)cc3)=O)CCCC2)nnc(C)c(C)c1C#N c1(NC(=O)OC(C)(C)C)ccc(OCCCNC=O)s1.c1cccnc1.N C1(C(=O)NC2(C(=O)NCCC3CCCC(C)C3)CSC2)CC2(C1)CC(O)C2 C1(C(CNC(CN(CCC#C)C)=O)NC(=O)C(C)N2CC(C)C2)CCOCC1 C=C(CNC(=O)Nc1cccc(Cc2ccc(Br)cn2)c1)c1ccccc1F C1(CC#C)(C(=O)NC(C)CCC2CC2)CCN(C(=O)CCOC)C1 C1(CC(=O)NCCC(C)NC(=O)CC2CN(C)C2)CCCC2(CCC2)O1 CC(C)(C)C#CCCNC(c1cc(CNC(c2ccnnc2)=O)ccn1)=O c1(C(=O)NC2CN(C(c3c(C)[nH]nc3C(F)(F)F)=O)C2)cc2cncn2c(O)n1 c1(OCCC)cccc(-c2cn(CC(=O)NCCc3cccc(Cl)c3)nn2)c1 c1(C(N(C(C)C(=O)N(C(C)C(C)C)C)CC)=O)cc(C)cc(C#N)c1 c1(C(=O)NCC2(CNC(C(C)(F)F)=O)CCC2)nccc2ccccc12 c1(C(N2CCC(NC(C(CC)N(C)C)=O)CC2C)=O)ccc2c(n1)CCCC2 Cc1cc(C)c(OCC(=O)NC2CC2)c(C)c1.C1(CC=O)OCCC1(C)C.C N1(C(C(C)OCC#C)=O)CCCOC(CNC(=O)CCCCCO)C1 N1(C(c2c(OC)ccs2)=O)CC(F)(F)CC1C(=O)Nc1cc(F)nc(F)c1 C1(CCOC)CN(C(=O)CS)CCN1C(=O)CC1CCC1(C)C.c1ccccc1 c1(C(=O)NCC2(C)CN(C(=O)C3=CSCS3)CCO2)ccc2n[nH]cc2c1 CCCC(C)(C)CC(=O)NC1CCN(C(c2cnn3ccccc23)=O)C1C1CC1 Cc1nn2c(c1C(=O)NC(CNC(c1ccon1)=O)CC(F)(F)F)CCCC2C C(=O)(C1CCCc2cccnc21)NC1C2(CC(NC(=O)COC3CCCC3)C2)C1 CC1=NOC(CCNC(C2(c3nccs3)COC2)=O)C1 c1(OC)c(C(=O)NCC(C)NC(c2nocc2C)=O)sc(C)c1Br C1(CNC(N(CCNC(N(C)C)=O)C)=O)CCN(C)C(=O)C1 C1(CNC(C(C)NC(CC)=O)=O)CCCN(C(C2(Cl)CCCCC2)=O)CC1 C(C(C)(C)CC(=O)N1CCCC(N(CCO)C(C2CCSC2)=O)C1)OC c1(CC)ncc(C(N2CCC(CO)C(NC(C3CC(F)CN3C)=O)C2)=O)c(C)n1 C1(CNC(CCN(C(CCC)C)C)=O)CCCN1C(c1coc(C2CC2)c1)=O S(=O)(=O)(c1ccc(NCC2(C)CC2(F)F)c(Cl)c1)N1CCCC(CCC=C)C1 c1(CC(N2C(CNC(CSCC)=O)CCCCC2)=O)ccc(F)cc1[N+](=O)[O-] C1(NC(C2CCc3cncn3C2)=O)CC2CCC(C1)N2C(=O)C#CC1CC1 c1(C(N2C(C(N(c3ccnn3C(C)(C)C)C)=O)CC2)=O)cc(F)cc(F)c1 CC(CC(=O)N1CCC(C(N2CCC(c3nn[nH]n3)C2)=O)C1C)C(F)(F)F c1(C(C)C(N2CCC(NC(=O)C=Cc3ccsc3)C2CO)=O)ccc(C#N)cc1 C1(CNC(=O)CCn2ccnc2)CCCCC1NC(=O)CC1CSCCS1 C1(CNC(Cc2c(C)ocn2)=O)CCN(C(=O)C)CC1(F)F.CCCN(C)C.O C(CCC(C)C(=O)NC(CC(=O)Nc1ccc(CO)cc1O)C(C)OC)OC c1nc(C)[nH]c2nccc1-2.C(=O)(C(CC=O)NC(=O)O)OCC.C(C)(C)C CC1(C)CC(CNC(=O)CSc2ccccc2)N(C(C2CCCCS2)=O)C1 C1(NC(C(CC=C)(C)CC)=O)CC2CCCC(C1)N2C(=O)C(CC)(CC)CC C1(CCCC)CN(C(C2(C)CC(C)(C)C2)=O)CCN1C(c1cc(C(C)C)[nH]n1)=O CC1CC(C(N2CCCC(O)C2)=O)N(C(c2cc(Br)cs2)=O)C1 c1(C(C(=O)NC)N(C)Cc2cnc(C3CC3)s2)cccc(OC)c1 N1(C(CN(CCC)CCN(C)C)=O)CCCC(c2noc(C(C)C)n2)C1 CCC(CC(C)C)C(=O)NC1CC(NC(=O)C(C)COc2ccccc2)C1 c1(NC(C(CCNC(C(CC)CCOC)=O)OC)=O)cccc(C#N)c1F N1(CCC(=O)N(CCOC)CC)CCOC1=O.C1(C(=O)N)CC1.C(C)C c1(N2CCC(Br)=C(C)C2)nc(=NCc2cn(C(C)(C)C)nn2)[nH]c2ccsc12 C1(NC(C(C)N(C)C)=O)CC2CN(C(c3cc(Cl)ccc3Cl)=O)CC2C1 C(c1cccc(F)c1C(F)(F)F)=CC(N1CCCC(C)(F)C1)=O C1(CCN(C(C(C=C)O)=O)C)CCCCN1C(c1ccnc(C2CC2)n1)=O C1(c2ccc(CC)cc2)CSCCCN1C(c1cnc(O)n1C)=O c1(C(=O)OCC)ccnnc1NC(c1cscn1)=O.N1(CC=O)CCCCC1 C(=O)(CCCCC#N)N1CCCC(N(C(Cc2c(SC)cccc2)=O)CCF)C1 N1(C(c2nn(C)c(O)c2)=O)CC2CC(CNC(c3cnns3)=O)CC1C2 CC1(C)CN(C(=O)CC2CCN(C(c3cnn(C(F)F)c3)=O)C2)C2COCC12 c1(OC)ccc(C(=O)NC2CCN(C(C3(S(C)(=O)=O)CC3)=O)C2)c(F)c1Cl N1(C(c2c(CC)ncnc2)=O)C2CCC1C(C(=O)NCc1[nH]cnc1C)C2 Cc1cc(C(=O)N(CC(C)C)C(C)C)nnc1O.C1(C)CCC(C)C1.CC(=O)N CCCS(=O)(=O)CC(=O)N1CCC(O)(CNC(C2CCCC2OC)=O)CC1 c1c(C)nn(C)c1C.c1(C(=O)OCC)cc(NC(C2(C)CCNC2)=O)ncn1 C1(C(CO)NC(CC=C)=O)CCN(C(=O)CCN2CCC(F)C2)CC1 N1(C(c2ccc(CNC(C3(O)CCC3)=O)s2)=O)CCOC(CO)C1 C(N=c1ccnc(CCC2CC2)[nH]1)C1(CNC(C2(C=C)CCC2)=O)CC1 N1(C(COCC)=O)CC(NC(=O)C(C(C)C)SC)CC12CCC2 N1(C(c2c(C)[nH]c(=N)s2)=O)CCC(C(N2CCC(N3CCCC3)CC2)=O)C(O)C1 C(CC(=O)NC(c1ccnc(F)c1)C)(C(C)(C)C)NC(CC=CC)=O c1(C(N(C(CNC(c2cc(CC)no2)=O)C)C)=O)ccc2c(c1)SCC(=O)N2 CC1(C)CN(C(C2CC3(C2)C(F)(F)C32CC2)=O)C(C)(C)C1O C12(C(=O)NCC3(CC)CCCC3)CC1CCN2C(=O)C(N1CCNC1=O)C c1(C(CC(=O)NCCC2(COC)CCC2)C)ccc(C2CC2)cc1 CCCCCC(F)C(=O)N1CCCC1CC(=O)NC1CCN(C)C1 c1(CN(c2n(CC=C)c(C(C)(C)O)nn2)C)c(Cl)cccc1Cl n1(CC(F)F)nc(C2CCCO2)nc1-c1ccc(Oc2ccccc2)cc1 C(=O)(C(C(C)C)NC(c1nn(C)cc1C)=O)NC(CC)Cn1cncn1 C1(C(=O)NC(c2nncs2)C)(NC(=O)CCc2nccn2C)CCSC1 c1(CC)cccc(C)c1CC(N1CC(N(C(=O)C=C2CCCC2)C)C(O)C1)=O c1(C(=O)NC2CCCC(C(=O)NC(CO)CC(F)(F)F)CC2)ccc2cccnn12 c1(C(N2CC(C)C(NC(C3CCCCO3)=O)C2)=O)c(Br)ccc2c1OCO2 N1(C(C2(NC(=O)CCC3CCOCC3)CC(O)C2)=O)CCn2ncnc2C1 C1(C(=O)NCC(COC)(C)C)CCC(C)(C)N(C(=O)C)C1.C(C)(C)C.O C(=O)(C1CCCc2cc(OC)ccc21)N1C(CNC(CCC#C)=O)C(O)C(O)C1 N1(C(C(CC2CCC2)NC(c2c(OC)nn(C)c2)=O)=O)CCOC(C)C1CO c1(C(N(CCNC)C(C)C)=O)nnsc1-c1ccccc1 N12CCCC3(C1)C(CCN3C)CNC(=O)CCSCC2=O.C(C(C)C)CC=C c1(C(N2CC(F)CC(NC(c3cccc(C)c3O)=O)C2)=O)cnc2ccoc2c1 N1(C(c2c(C)c(=O)cc[nH]2)=O)CC(C2CN(C(c3ccc(F)c(F)c3)=O)C2)C1 CC(C)CC(O)C(C)C(=O)N1CCCCC1CCC(=O)NC1C=CCCC1CO Cc1c(F)ccc(C(=O)N(C2CN(C(=O)CC34CC(C3)C4)C2)C)c1N C1(N(C)C(c2cn(C3CCC3)nn2)=O)CN(C(c2ccccc2O)=O)CC1F C(=O)(C1=CNC2=NCCCC2=C1)NC(CCCNC(c1nc(C)sc1C)=O)C C1(CC)CCC(C(N2CCC(N(CCO)C(c3csc(Cl)n3)=O)C2)=O)O1 C1CCCN1C(=O)C.C(C)(C)(C(=O)NC)NC(=O)NCCC.C(C)C n1(C(CC)C)ncc2cc(C(=O)NCC(C)(C)NC(=O)CCC#N)cnc12 N1(C(c2c(C)n(C)cn2)=O)CC(C2CN(C(c3cnccn3)=O)C2)C1 C(C1(C)CCC(C)C1(C)C)=CC=O.CC(C)C.CCC(=O)C1(C(=O)N)CC1 S(=O)(=O)(c1cc(F)c(F)c(F)c1)N1CCC(CNC(CN(C)C)=O)C(F)(F)C1 c1(CC)ccc(O)c(C(N2CCCC2CNC(=O)Cc2cnnn2C)=O)c1.C C1(C(N2CCCC(CN(C)C(c3cc(C#N)on3)=O)C2)=O)CC2CCC(C1)S2 C1(C(=O)OC)C2CN(N(CC3CCCCC3)Cc3ccc(F)c(F)c3)CC12 c1(C=O)cccc2c[nH]nc12.C(C(=O)NCCC1CCOC1)(C(C)O)NC(C)=O c1(C(=O)OCC)ccc(OC)c(S(=O)(=O)NC(CO)C2CCc3ccccc32)c1 C1(O)(CNC(CCC=CCC=C)=O)CCCN(C(=O)C(O)CSC)CC1 c1(C(N(CCCC(C)C)C)=O)nn2c(c1C)OCCC2.C(C)(C=O)OCC#C.N C1(C)(OC)CCN(C(=O)C(=O)N(C(C)C)CC2(C)CC2)CC1 c1(CC(=O)NC2(CO)CN(C(C=CCCC(C)C)=O)C2)cc2ccccc2s1 c1(C(=O)NC2CCN(C(CSC)=O)CC2C)ccn2c(O)nnc2c1 C(=O)(CC(CC(C)C)NC(c1csc(Cl)n1)=O)NCc1cc(CC)no1 C#Cc1ccc(C(=O)NCCC2CSCCN2C(C2CCCC2OC)=O)c(C)c1 c1(C(N2C(C)CC(O)C2)=O)n[nH]c2c1CCN(Cc1ccc([N+](=O)[O-])o1)C2 CCCCCCCCC(F)C(=O)NCCC(O)CNC(=O)C(C)=CC(C)(C)C N1(C(C=C(COC)C)=O)CCCC2(CCCN2C(c2ccc(NCCO)cc2)=O)C1 CCCCCCN(C(C1CCN1C1CCCC1)=O)Cc1cc(Br)no1.OCC c1(C(=O)NC2CCCC(CN(C(CCSCC)=O)C)C2)cc2cccn2c(O)n1 Cc1cc(OCC(=O)NCC2CCN(C(C3CC=CCO3)=O)C2)cc(C)c1Cl c1(C(=O)N)ccc(Cl)c(Cl)c1N.C(CCC(C)(C)C)N(C(C1(CC)CCC1)=O)C c1(C(=O)NCCCN(C(C(CC)OC)=O)C)ccc([N+](=O)[O-])cc1Br N1(C(c2c(C)c(C3CC3)ccc2)=O)CCC2C1CCCN2C(=O)CSCC(N)=O C12(CC)CC3CC1C2C3NCC(=O)Nc1cc(-c2ccc(C)cc2)nn1C C(=O)(CS(=O)C(F)(F)F)NC(CCNC(c1c(CC)n[nH]c1)=O)C(C)C C1(N(C(C=CC(C)C)=O)CCO)CCN(C(=O)CC)CC1.C(=O)(N(C)C)N N1(C(C2(COC)CCCC2)=O)CCC(F)(CNC(C2C3COCC23)=O)C1 C12(OC)CCC(NC(c3cccc(CN4CCCC4)c3)=O)(CC1)C2 C1(NC(C(CC=C)CC=C)=O)CN(C(c2ccc(OC)cn2)=O)CC2CCCC12 Cn1cnc(CN(CCC(=O)N2CCCC2)CCN2CC3CC3C2)c1 C(=O)(C(C)C(F)(F)F)NC1CC(Cn2cc(COCC(C)O)nn2)C1 C1(NC(c2cnoc2C2CCC2)=O)CCCC2CN(C(=O)C=CC3CC3)CC12 C1(C2CC2)(NC(CC2OCCN(C(CC(CC)OC)=O)C2)=O)CCOCC1 N1(C(C2N(C(C)=O)CCC2)=O)CCCC(C)(CNC(c2ccc(O)nc2C)=O)C1 c1(N2CCCC(c3nc(C)[nH]n3)C2)nccc2ccc(Br)cc12 C=CC(CCC)CC(=O)NCC1CN(C(=O)C(CC)CC)CC1C(F)(F)F c1(C(N2C(CCCNC(CN(CCC)C)=O)CCC2)=O)cc(F)c2[nH]nnc2c1 O=C1CCC(C(=O)N2CCC(NC(C3(C4CCCCO4)CC3)=O)C(F)C2)=NN1 c1(OC)nccc(C(N2CCC(N(CC(F)F)CCO)CC2)=O)n1 C1(CNC(c2ccc(C#N)s2)=O)CN(C(C2CC2C(F)F)=O)CC12CCC2 C1(C(=O)NC(CC=C)CO)CC2(CC2)CN1C(=O)C(Cl)=CCl CN1CCn2nc(C(=O)NCC3(O)CCN(C(c4cc(C#N)c[nH]4)=O)C3)cc2C1 Nc1cc(Cl)nc(Cl)c1C(N1CCCC(NC(c2n[nH]c(C3CC3)n2)=O)CC1)=O N1(C(c2c(C)nns2)=O)CCC2(CC1)C(NC(=O)C(C)(C)C(N)=O)CS2(=O)=O Cc1nc(=NC(=O)C2CC3(CC3)CN2C(c2ccc(Cl)cc2C(N)=O)=O)s[nH]1 CC1OC2CCC1(C(=O)NCC1CC(F)CN1C(=O)C=CCO)C2 C(CC1c2ccccc2CCN1C(=O)Cc1cnc(C)s1)NC(CC=C(C)C)=O C(=O)(C(CNC(C1C2CCC(C2)C1C)=O)CC(C)C)NC(CC=C)CO C(=O)(CN=c1ccc(Cl)n[nH]1)NC1CC(NC(C(CCCOC)C)=O)C1 c1(CC)cnc(C)c(O)c1COC.c12c(cccc1O)C(=O)CN(C)CC2 c1(C(=O)NCC2C(NC(=O)C=CC3CCCO3)CCC2)ccc(CO)nc1 C1(C=O)CNC(=O)C(C)(C)C1.CC(C)(C)OC(=O)NC(C)C1CCC1.N Cc1cccc(C(CNC(=O)CS(C)(=O)=O)NC(=O)C(N2CCCCCC2)C)c1 c1(C(N2CC3CC3(C(=O)Nc3ccc(C(F)F)nc3)C2)=O)ccc(O)c(O)c1O N1(Cc2cn(C)nn2)CCN(Cc2cccc(C3CCC3)c2)CC1 CC1(C(N2CCC(O)C(NC(=O)C=Cc3ccncc3)C2)=O)CCC12CCC2 C(=O)(CCCCC(C)(C)C)N(C)CC1CCCCN1C(=O)C(O)Cc1cnc[nH]1 c1(C(=O)NC(CC)CNC(c2occc2F)=O)c(F)cccc1[N+](=O)[O-] C(CC(CO)C(C)C)NC(c1nc(C)[nH]n1)c1nnnn1CCN1CCOCC1 c1(C(=O)NCC(=O)NC(CC#C)CO)cccc[n+]1[O-] c1(C(N(C(C)C)CC)=O)c[nH]nc1[N+](=O)[O-].c1(C=O)csc(C)c1C1CC1 c1(C(N2C3CCN(C(C4(C)CC4)=O)C3CC2)=O)cc(F)c(Br)cc1[N+](=O)[O-] CCC(C(=O)N1CCC(CN(C(=O)CCc2cnc[nH]2)C)C1)C(C)C C1(C(N2CCCC(CN(C(c3ccc(CC)s3)=O)C)C2)=O)CC2(CCC2)C1.O Cc1cnc(C#N)c(NC(C2CCCC2NC(c2cccn3nccc23)=O)=O)c1 N1(Cc2ccc(CCC)cc2)CCC2(CCN(c3ncnc4ccsc34)CC2)C1 c1(OC)ccc(CCC(=O)NCC(C)(C)OCC)c(F)c1.C(=O)C.C1CC1 c1(CN2CC3(CC(CC(=O)Nc4cc(Cl)cnc4Cl)C3)C2)ccc2cc[nH]c2c1 N1(CCCNC(CC2(C(=O)OC)CC2)=O)CCN(C(C2CCSC2)=O)CC1 C1(C(C)(C)NC(=O)NCC2(C)CCN2)COc2ccccc2C1 N1(C(C2CC(C#C)(O)C2)=O)CCN(C(C2(N(C)C)CC2)=O)CC1CCO Cc1c(C(=O)NC2CC2NC(=O)C(C(C)C)n2cccc2)cc(F)cc1Br C1(CC(=O)NC2(C)CN(C(=O)CCc3cncc(O)c3)C2)CCCCCCC1 C1(OC)CCN(C(=O)CCCC(CC)NC(=O)C(F)C(F)(F)F)C12CCC2 Cc1noc(Cl)c1CC(=O)NC1CCCC1CNC(=O)Cc1nncs1 N1(CC(=O)NCC=C(C(=O)N(CCOC)C)C)CCNC1=O CCCCC(C)C(=O)NC(CC1CC1)CC(=O)N(CCCC(O)CO)C c1(NC(Cn2cc(CNC(C(CC=CC)C)=O)nn2)=O)cc(C)cnc1C C(CCSC)(C(=O)NC(C1CCCC1)CNC(=O)CC(C)(C)O)OC CCC(C)CCCC(=O)N1CCCC1(C(=O)N(CC(C1CC1)OC)C)CC C(CCCCC(=O)NC(C(N1CC(O)(c2nn[nH]n2)C1)=O)C1CCCC1)N(C)C C=C=CCCC(=O)NC1CC(F)(CNC(C2(c3cccnc3)CCC2)=O)C1 N1(C(C(C)CC2CCC2)=O)CCC(NC(=O)C=CC2CCOC2)C12CCCC2 CC1(C)CC(C(=O)O)CN1C(c1nn(-c2ncc(Cl)cc2Cl)cc1O)=O c1(N(C)CC2CCN(N3CCCCC3CO)C2)nc(Cl)nc2c1oc1ccccc21 n1(CC(=O)NC(CCNC(c2c(C)nn(C)c2)=O)(C)C)nc2ccccn2c1=O c1(CC)cc(NC(C2CCC(NC(=O)CCN3CCOC3=O)CC2)=O)cc(Br)c1 C(=O)(C(CC(C)C)NC(=O)CCCNC(=O)CC(C)(C)C1CC1)NC c1(C(=O)NC(C(=O)N(C2(CSC)CCC2)C)CO)cc(CO)oc1C c1(C(=O)NCC(CN(C)C(c2cnnn2C)=O)O)sc2cc(F)ccc2c1Cl c1(OCOC)cccc(-c2cnc(Cl)c(C(=O)Nc3cccc(I)c3)c2)c1F C1(NC(c2n[nH]c(C)c2C)=O)CCCCN(C(=O)C(C)(C)C(F)(F)F)CC1 C1(C(=O)Nc2ncc(C)s2)CN(c2ncc(Br)c(C)n2)CCC1O c1(NC(CC(C)(C)OC)c2nnnn2CCSC)cccc([N+](=O)[O-])c1 C(Cc1ccccc1)(CC)NC(C1C(OC)CC1)=O.c1(C(=O)N)cn(C)nn1 C1(NC(Cc2ncc(C)s2)=O)CCC2(CC1)CCN(C(=O)C(F)OC(F)(F)F)C2 C(=O)(CCCCCC#N)NC1CCCC(NC(C23CC(CC(C)C)(C2)C3)=O)C1 CCCCCCCCCOC(=O)CCOC(c1cnc(=N)[nH]c1)=O C(=O)(C(O)CCC(C)C)NCCCCCCN(C(C(F)OC)=O)C c1(OC)cc(C(=O)NC(C2CCN(C(c3c[nH]nc3F)=O)C2)(C)C)cc(F)c1 CC(C)CC(CC(C)C)C(=O)NC1CN(C(C23CCC2CC3)=O)C1 N1(C(C2CCC(C)C2)=O)CCC(N2CCN(C(C3(C#N)CC3)=O)CC2)CC1 N1(C(c2c(COC)cc[nH]2)=O)CCCCC(C)(C)C1.C(=O)(C(F)C(F)(F)F)N C(=O)(C(O)C1=CCCCC1)NC1C(NC(c2cocn2)=O)CCCC1 S(=O)(=O)(C1CCN(C(c2ccc(C(F)(F)F)cc2Cl)=O)C1)NC(C)C c1(C(N2CC(C(C)NC(CCCOCCOC)=O)C2)=O)cc(N)c(Cl)cn1 C1CCCC(C=O)C1.C1CC1.C(=O)(CC1(C(F)(F)F)CC1)NC1CC1 C12(C(N(C)C)=O)CC(C(=O)NCCCOCC(C)(C)O)(C1)C2 C(C(O)C(=O)NC1(C(=O)NC2(C)CC(N(C)C)C2)CC1(C)C)SC c1(C(N2CC(Cc3cncc(C)n3)C2)=O)cc(-n2cc(C(=O)OC)nn2)ccn1 CCC(C)(C)C(O)C(=O)N1CCCC1CNC(=O)CCCc1ccc(SC)cc1 c1(C(=O)NC(CCCCNC(C(C)(C)OCC)=O)C)cnc(O)c2cccnc12 CC1=C(C(=O)N2CCCC(N(C(=O)CCC3CC3)CCO)C2)CCC1 C12(C(C=Cc3cnc(C)s3)=O)CCCC1C2(F)F c1(CN2CCC(C3N(C(C=CC)=O)CCC3)C2)ccc(OC)nc1C c1(C(N(C)CC)=O)cccc(C(N2CC(C)C3CC23)=O)c1.C(=O)(C=NOC)N c1(C(=O)NCC(C(C)C)NC(c2nc(Cl)ccc2F)=O)coc2c1C(O)CCC2 Cc1cc(NC(c2cnc3n2CCCC3)C)ncc1S(=O)(=O)NCCCC(C)O Cn1cnc(S(=O)(=O)N2CCN(C(=O)NCCC(C)(C)O)CC2)c1 C1(S(N)(=O)=O)(C(=O)N)CCCC1.C(CC(C)C(C)C)NC(C(F)=CC)=O C1(CN(C(=O)C(C2CC2)SC)CC)CCCN1C(c1cocn1)=O N#Cc1cccc(CCC(N2CCCCC(NC(C3CCC3)=O)C2)=O)c1 n1(CC(C)C)ccc(=NC(=O)C(=O)N2CCN(C(=O)N(C)C)CC2)[nH]1 C1(NC(C2CC3(CCC3)C2)=O)CC(O)CN(C(c2ccsc2Br)=O)C1 c1(C2(C(=O)NCC=CCNC(C3(C)CC3)=O)CCCO2)ccc(Br)cc1 c1(CNC2CCCC(C(=O)Nc3cccc(F)n3)C2)ccc2c(c1)OCCCO2 C=CCC(Cc1ccccc1)C(=O)NC1CN(C(C2(CF)COC2)=O)CCC1O N1(C(c2ccn(C)c2)=O)CCC(C(F)CNC(=O)CC2CCCOCC2)CC1 c1(C(=O)NCCCC(C)(C)NC(c2cnccn2)=O)cc2c(cn1)NC(=O)CO2 c1(-n2ccc(CN(C(CCSCC)C)CC3CC3)n2)ccccc1F Cc1cc(CNC(c2cnn(-c3ccncc3)c2C)=O)nn1-c1ccccc1 c1(C(=O)NC2C(OC)CN(C(c3cnns3)=O)C2)c2c(c[nH]c1=N)CCC2 C1(COC)CN(C(c2sccc2Cl)=O)CCN1C(=O)Cc1cnn(C(C)C)c1 C(CC(C)(C)C)(C(=O)N)NC(C(C)OCC(C)C)=O.C1CC2(CCCCC2)C1 C(CC(C)C)(C(=O)NCCOCCNC(=O)Cc1cc(C)ccc1O)OC C1(C(N2CCC(CNC(C3CCC(=O)C3)=O)C2)=O)CCCCC1C1CC1 Cc1sc2ncc(C(=O)NCCCCCCNC(=O)CC(C)F)n2c1C C(=O)(C(O)C(F)(F)c1ccccc1)N1CCCC(NC(Cc2cc(C)sc2)=O)C1 c1(C(N(CCC)CC)=O)cc(C)n(C(C)(C)C)n1.c1(C(C=O)O)ccnn1C C#CCC(CC#C)C(=O)N1CCN(C(=O)CC2CCC(=O)N2)C(CO)C1 C1(N(C(=O)CC2CNC(=O)O2)C)CCCN(C(=O)C=CCO)C1 c1(C(=O)NCCC2(O)CCN(C(COCC=C)=O)CC2)cn2cc(Cl)cnc2n1 c1(C(=O)NCC2(CNC(=O)Cc3ccoc3)CC2)cc2cccnc2cc1F Cc1nc(C2CC2)[nH]c1C(N1CCC(C2CCCN2C(=O)CSC(F)F)C1)=O c1(C(=O)NC2C(NC(C3(C(C)C)CCC3)=O)CCC2)ccc(N)c(O)c1 c1(CC)cnc(C(=O)N(C)CC2(O)CCN(C(c3coc(O)n3)=O)C2)nc1 C(c1cccc(F)c1)=CC(N1CCC(NC(C(=O)NCC2CC2)=O)C1)=O c1(C(N2CC(C)(C(=O)NC(C(=O)NC)C)C2)=O)cc(OC)c(O)c(I)c1 C1(CNC(C(CC)NC)=O)CN(C(=O)CS)CC(C)(C)O1.c1ccccc1.C C1(O)(CCNC(C2(C)CCCS2)=O)CCCN(C(=O)CC2(NS)COC2)C1 C(c1ccc(F)cc1)=CC(=O)NCC=C1CCN(C(=O)CC2CCCCO2)CC1 C#CCC(C(=O)N1CCC(O)(CC(=O)O)C1)NC(=O)COCC1CCCO1 C=C(C)CCCC(=O)NCC(C)N(C(c1cnc(C(F)(F)F)c(C)c1)=O)CC Cc1ccc(C(=O)NC2CC2)cc1.c1(N(C(=O)N)C(C)C)c(Cl)cccc1Cl c1cc2c(cc1C1(NC3C4CCCC3NCC4)COC1)OCO2 C1(CCOC)CCN(C(=O)CCc2ccccn2)C1.c1(CC(=O)N)ccc(Cl)s1 C(=O)(C1SCc2cccnc21)N1CCN(CC(=O)OCc2cccnn2)CC1 Cc1cc(CNC(=O)CN2CCN(C(C3COC(=O)N3)=O)CC2)cnc1C C1(C(=O)OC)CCN(C(C2(N(c3cc(C)sn3)C(=O)CC)CCCC2)=O)CC1 C(C1CCc2cccnc21)NC(=NC)NCc1ccc(Cl)c(Cl)c1 C1(C(=O)N(CC(O)CNC(=O)C=O)C)(OC)CCS(=O)(=O)C1.C1CC1 C(c1cccc(F)c1)=C(C(=O)NCC(CC)NC(C1(CO)CCOC1)=O)F c1(C(N2CC3(CN(Cc4c(C)n[nH]c4C)C3)C2)=O)c[nH]c2cc(C#N)ccc12 c1(C(N2CCC(C(NOCC=C)=O)(Sc3cnn(C)c3)C2)=O)cc(O)nc(C)n1 C1(NC(c2n(C(CC)C)ncc2)=O)C2CC1N(C(=O)CC1(O)CCOCC1)C2 C#CC1(C(N2CC(C(C)(C)C)C2)=O)CN(C(C2CC2CC)=O)C1 c1(CC)nccnc1C(=O)NCCC(O)CNC(=O)CC(C)C.C(C)(=O)N c1(C(=O)NC2C3CCCC23)ccc2c(n1)CN(C(=O)CSC(F)(F)F)CC2 N(C1COc2c(OC)cccc21)C(C1Cc2c(ccc(OC)c2)OC1)=O C1(C(N2CC(O)(C(C)(C)CNC(=O)CC3CC3)C2)=O)CCC(CCO)CC1 C1(CC#C)(C(=O)NC(c2nn[nH]n2)CC)CCN(C(c2sc(C)cc2C)=O)C1 c1(C(N2CC3(C2)CN(Cc2cc4cnccc4[nH]2)C3)=O)cccc2cccnc12 c1(C(NOCCCC)=O)oc(CNC(c2cn(C)c(C)n2)=O)cc1C C1(C(N2CCC2)=O)CNC(=O)C(C)(C)C1.c1(C(N(C)C)=O)ccc2c[nH]nc2c1 Cc1c(C(=O)NCC2(C(=O)O)CC(C)C2)nnn1C(C)C Cc1c(C(=O)N)c(C(F)F)nn1C.c1(CC(N2CC3C(C3)C2)=O)cccc(F)c1F c1(C(=O)NC(CNC(c2n(CC)nnc2)=O)(CC)CC)[nH]c2ccccc2c1Cl c1(CC(=O)NCC2(OC)CN(C(c3cccc(O)n3)=O)C2)cccc(O)n1 C1(O)(C(=O)NCC=CC(=O)NCC2C(C)(C)C(O)C2)CC2CCC1C2 N1(C(=O)C#CC2CCOCC2)CCCC2(CCN(C(C3CCCCC3)=O)C2)C1 C1(C(NCC#C)=O)CC12CCN(C(=O)C=C1CCOCC1)C2.c1ccccc1.C N1(C(C2(C#C)CC2)=O)CCOCC(C(=O)NC(C2CCOC2)CO)C1 C1(NC(CCCC#C)=O)CCN(C(c2ccc(SCC)nc2C)=O)C1(C)C N1(C(C2C3CN(C(CCC(=O)N(C)C)=O)CC32)=O)CCOCC(C2CC2)C1 C1C(O)C(O)CN1C(=O)C(CCO)N(C)C.c1(N(C)C)cnc(C(=O)NC)cn1 c1(C=O)ccc2c(c1)ncn2C(C)C.c1(CC)nonc1C(=O)NCC(F)C S(=O)(=O)(CC1CCCc2ccccc21)Nc1cccc(CN(C(C)=O)C)c1 C1(C(N2CC(O)(CNC(=O)C=Cc3cn[nH]c3)C2)=O)CC12CCCCCC2 N1(C(c2ccn(C)c2)=O)CCCCC(CNC(=O)CC2COCC(C)(C)O2)C1 c1(C(N2C3CCN(C(C(CC=CC)C)=O)CC3C2)=O)cccc2ccncc12 C(=O)(CCC(=O)N(C)C1CC1)NC(C)CC1CN(c2nc(C(C)(C)C)ns2)C1 c1(OC)ncc(F)cc1C(=O)N.C1(CC)C(C)CCCN1C(=O)CC1CCCC1 C12(C(=O)NC(C3OCCN(C(CN(CCC#C)C)=O)C3)C)CCC(F)(CC1)CC2 N1(C(c2ccc(C(=O)OC)o2)C(=O)NC(C)C)CC2(CCC(C)(C)CC2)C1 c1(C(N2CCN(CC=O)C(=O)C2)=O)cc(C(F)F)nc(Cl)c1.c1ccccc1CO.N N1(C(COCCCOC)=O)CCN(C(c2cc(C#N)cs2)=O)C(C)C1C CCCCC(C(=O)NCCCC1CCCN1C(=O)C(C1CCC1)OC)N(C)C c1(OC)cccc2c1OCC(C(=O)NCC1CCN1C(c1cc(C)sc1C)=O)C2 c1(CN(C(=O)CCc2csc(C(=O)O)n2)C)ccc2c(c1)OCO2 c1(N2CC(NC(C(C)Oc3ccc(C)cc3)=O)C2)ncnc(Cl)c1Br C1(NC(C(C)Cc2cnc[nH]2)=O)CN(C(C2CC(O)C2)=O)CC1F C1(NC(CNC(=O)NC)=O)CN(C(=O)C(C)(C)c2cncs2)CCC1C C1(C)(c2cn(-c3cn(C)nc3)nn2)CN(C(=O)C(F)(F)CO)CCO1 c1(C(=O)OC)ccc(OC)c(NC(=O)C(=O)NC)c1F.c1nc2ccccc2s1 C1(F)(CNC(C2OCCN(C)C2)=O)CCCN(C(C2COC2)=O)C1 c1(C(=O)NCC(CCCC)NC(c2ocnc2CC)=O)cccc2nc(C)nn12 C1(C)(CNC(C(CC)C2CCOC2)=O)CCCN1C(c1ccc[nH]1)=O C(C(C(C)(C)C)NC(C1CCO1)=O)N(C)C.C1=CC(=O)NC1(C)C N1(CC(N2CCC3(NC(CCN(C)CC)=O)C(C2)C3)=O)CCc2sccc2C1 C(CC(C)C(C)=O)OCCC(C=C)C c1ccc(C(=O)N(CC(O)CN(C)C(c2cn(CCO)nn2)=O)C)cn1.CCS N1(C(C=C(C)C(C)C)=O)CCC(N(C(c2cc(F)n[nH]2)=O)CC2CC2)CC1 C1(C(=O)OC(C)(C)C)C2CCC(C2)C1C=O.N1(C(CC)=O)CCC(O)C1 N1(C(C2CCCN(C(C)=O)C2)=O)CC(NC(=O)Cc2cccnc2)CC2(CC2)C1 CCCC(C)CC(=O)N1CCC(C(O)CNC(C2OCCCC2(C)C)=O)CC1 C1(C(=O)NCCC2COCCN2C(c2ns[nH]c2=O)=O)CCc2cncn2C1 Cc1cc(C)n2ncc(C(N3CC4(CC4)CC3C#C)=O)c2n1 CCN(OC)C(=O)CNC(C1CCC(C)CN1C(=O)C=Cc1ccccc1)=O c1(N(C)CC)ccc(CNC(C2CCCN2S(C)(=O)=O)=O)cc1 C1(F)(C(N(CCCN(C)C(c2ccc(C3CC3)s2)=O)C)=O)CC2(CCC2)C1 Cc1cccc(N2CCC(CN3CCCC3CC(F)F)C2=O)c1 C1(CC)CN(C(=O)C(c2ccncc2C)C)CCN1C(=O)CCOCC(F)(F)F c1(C(C)C)ccc(CNC(=O)CNC(=O)CC(C)CN(C)C)cn1 N1(C(c2n(C)nc(C)c2Cl)=O)CC2ON=C(CNC(c3cccc(O)n3)=O)C2C1 C(C1CC1)(C1CC1)=CC(N1C(CCCNC(C(C)=CC2CC2)=O)CCC1)=O Cc1sc(O)nc1C(N1CCC(O)(CNC(C2(C)CCC(C)C2)=O)C1)=O c1(CC)c(C(=O)Nc2nc(C(=O)NC3CC3(F)F)cs2)nnn1CC CCCC(C(=O)NC(CC(F)F)C(=O)NC(C)CCCCCO)C(C)C N1(C(C(C=C)O)=O)CCCN(C(c2ccn(C3CCCCC3)n2)=O)CC1 C=CC1(CC(=O)N(C)CC2CCCO2)CN(C(c2cnn(C)c2C)=O)C1 c1(CNc2c(OC)nc(C)nc2Cl)cc2nc(Cl)ccc2[nH]1 CCCC(F)C(=O)NC=O.C1(CNC(C2CC2)=O)CC1N.C1CCC1 c1(C(=O)NCC2C=CC(NC(CC)=O)C2)cc(C)cc([N+](=O)[O-])c1 c1(C(CC)(C)C)ccc(C(=O)N(C2CCCC2)CCNC)cc1.c1cnc(C)o1 C(C(O)CC(F)(F)F)NC(C(CNC(c1ccn(C)c1)=O)O)=O c1(C(N2CC(=C(C)F)C2)=O)csc([N+](=O)[O-])c1.C1(CC=O)NC(=O)NC1=O.N CN1CCc2[nH]nc(C(N3CCCC4CC34C(=O)NCCO)=O)c2C1.C(C)(C)C C1(CNC(CCC=CCC=C)=O)CCN(C(=O)C)C1(C)C.c1cccc(Cl)c1.S C(=O)(CC(C(C)(C)C)NC(=O)C(=O)NC(C)C)NC(CC)CSC Cc1coc(C(C)(C)C)c1C(N1CCC(C)C1)=O.C1(CC=O)CCN(C)C1=O N1(C(C23CC(C=O)(C2)C3)=O)CCC2CC2C1.c1(CC=O)ccon1.CC.O c1(C=O)ccc(S(C)(=O)=O)o1.N1(C(C=CC=CC)=O)CCOC(C)C1.N CC1(C(=O)NC2CC3(C2)CC3C(=O)N)CC(F)(F)C1.C1(O)CCOC1.C Cc1ccc(CCC(=O)N(CCCNC(C2CCOC2)=O)C)o1 c1(C(=O)NC2CC3(CN(C(Cc4c(C)c(Cl)ccc4)=O)C3)C2)ccc2n[nH]cc2c1 C1(C(=O)NCCc2ccn(CC)n2)C2CN(C(=O)C(F)CC3CCOC3)CC12 C1(C(N2CC(CCC)C2)=O)(N(C)C)CCOCC1.c1(C2C(C=O)C2)cn[nH]c1.N C(C(=O)NC(C)(C)CC(N)=O)(C(C)CC)NC(CNC(=O)OCC)=O c1(C=O)ccc(Cl)c(N)c1Cl.C1(N(S(C(C)O)(=O)=O)C(=O)C)CCN(C)CC1 Cc1cccc(C(C)C(N2CC(NC(=O)Cc3cc(C)no3)C(O)C2)=O)c1 C(CCN=c1nc2scnc2c(NCc2cccc(Cl)c2Cl)[nH]1)OC Cc1nc2c(o1)CCN(C(C1CC1NC(=O)CC1CCC1)=O)C2 N1(C(C2C(NC(=O)OC(C)(C)C)CCC2)=O)CCOC2COCCC12 C(=O)(CC(C)(C)C(C)(F)F)NC1(CNC(Cc2n[nH]c(=NC)s2)=O)CCC1 c1(-c2nc(CC(C)C)nn2C(C)C(C)C)cc2sccc2cn1 c1(C(C)NC(C2(CN)CC(C)C2)=O)ccc(N2CCN(C)CC2)cc1 C1(O)(CC(=O)NCc2ccc(C)cc2)CCN(c2nccc(C)n2)CC1 C(CNC(=O)CC=Cc1ccccc1)(CC(=O)N1CC(CS(C)=O)C1)OC C(=O)(CC(=O)N(C1CC(C(=O)N(C(C)C(=O)OC)C)C1)C)NCC#C CC(CCC(=O)NCC1CCC(F)(F)C1)NC(=O)C(C)(C)N1CCCC1 N1(C(c2cnn(C)c2Cl)=O)CCC2CN(C(c3cccc4scnc34)=O)CC2C1 N1(C(C2CN3CCN2CC3)=O)CCCN(C(=O)CN2CCCCC2)C(CO)C1 Cc1cc(C(=O)NC23CC2CN(C(C2CCS(=O)(=O)CC2)=O)C3)ccc1Cl C1(CN(C)C(c2ccc(-c3ncc[nH]3)cc2)=O)CCCCCN1 c1(CN2CC(CC(=O)Nc3cc(C)ncc3)OCC2)cccc2c1OC(F)(F)O2 C=CC1CCCN1C(=O)C(c1ccnn1C)NC(=O)Cc1csnc1C c1(OC)cc(F)c(C(N2CCC3(CC3)C2)=O)c(F)c1.c1(C=O)ncc(C)cn1.N c1(C2N(C(C(=O)NCC=C)c3ccsc3)CCC2)ncc(Br)cn1 N1(C(CC2=CCN(C)CC2)=O)CCC2CN(C(C34CC(F)(C3)C4)=O)CCC2C1 Cc1scc(C(=O)NC23CC(NC(=O)C(C)Sc4nncn4C)(C2)C3)c1C c1(C(=O)NC(C(C)NC(=O)C(C)(C)CF)CO)nnc2ccccc2n1 Cc1ccc(C(C)NC(=O)C(C)N(C(=O)CCCC2CCCO2)C2CC2)cn1 C(=O)(C1=CC2C=CC(C1)C2)N1C(C)CC(NC(=O)CN2CCCCC2)C1 c1(C(=O)N)cc(F)cc2nn(C)cc12.C(=O)(CC(=O)NC1CC1)NCCCC O=C1CC2(CCOC2)C(C(N2CCCC23CCOC3)=O)CN1 N1(C(C2CN(CCC)C(=O)C2)=O)CCC2(CCN(C(c3cnc(C)n3C)=O)C2)C1 c1(C(N2CC(NC(c3c(C)cc(C)nc3)=O)(CO)C2)=O)cnc(O)c2cncn12 CC1(C)CN(C(=O)Cc2ccccc2)CC1NC(=O)CC1CCC(C)(O)CC1 c1(CN2CCC(NC(c3cccc(C)c3I)=O)(CO)CC2)ccc(F)c(F)c1Br c1(C=O)cccc([N+](=O)[O-])c1.C1(C)(C(N2CCC(CC)C2)=O)COC(=O)OC1.N C(=O)(C(O)C(C)(C)C)N1CCCCC1.c1(C(C)C)c(C(F)(F)F)n[nH]c1C=O.N CCCC(O)CC(=O)NC(C)CCCNC(c1ccc(C)nc1OC)=O c1(C(=O)N)ccc(S(N)(=O)=O)cn1.CC(C)C(C)CC(=O)N1CCCC1C1CC1 C(C(C(=O)NC(c1cccc(C)n1)C)C(C)C)NC(C(CC)=CC)=O S(=O)(=O)(c1cccc(C(=O)N(C(C)Cc2nn[nH]n2)C)c1)NCC(CC)=O Cc1cc(N(CC(Cl)Cl)C)nc(N(CC(N)=O)C)n1 N1(C(Cn2c(C)ccn2)=O)CCC(Nc2cccnc2)CC1 C1(CN(C(=O)C(C)C)CC)CCCCN1C(c1cc(Cl)ccn1)=O N1(C(c2cnc(C)nc2)=O)CC(N(C(=O)COc2cccc(Cl)c2)C)C(C)(C)C1 c1(OCC)cc(N(CC(C)CNC(=O)C(C)c2cncs2)C)ncn1 c1(C(=O)NCCCC)ccccc1.n1(CC=CCC=O)cnnn1.C(N)=O.N c1(CN(C2CC3CNC2C3)CC2CC(=O)NCC2)ccc(I)cc1F N1(C(=O)CC23CCCC2C3)CC2(C1)CN(C(C1COCCO1)=O)C2 CC1CCCN(C(=O)C2=CCN(C(=O)CCCNC(N)=O)C2)C1CCO C(C(CC(C)C)NC(=O)CCC(C)N(C)C)NC(C(CC)N(C)C)=O Cc1cc(CNC(=O)CCC2CCN(C(C3CCN3C)=O)C2)n[nH]1 C1(C(N2C3CN(Cc4n(C)ncc4)C(C3)C2)=O)CCC2CCC(=O)N2C1 Cc1sc2ncnc(NC3CCCN(C(=O)C(C)OCCN(C)C)C3)c2c1C N(C1CCOc2ccc(Br)cc21)C(C1CCN1C(c1cn2cccnc2n1)=O)=O Cc1ccc(C(N2CCN(C(=O)C(O)C(F)(F)F)CC2CF)=O)c(F)c1Cl c1(C(=O)NCc2cn(C3CN(C(c4n(C)cnc4)=O)C3)nn2)ccnc(Cl)c1N N1(C(C2(CC=C)CCCC2)=O)C(CC(=O)NC(C)CC(=O)NC)C2CCCC12 N1(C(C(CC=CC)C)=O)CCN(C(c2cc(O)nc(O)n2)=O)C(C)C1 C1(NC(COC)=O)C(C)OCC12CCN(C(c1cccc(=O)n1O)=O)CC2 c1(C(N2CC(S(CC)(=O)=O)C2)=O)[nH]nc2ncc(C)cc12 N(C1CC2(CN(C(=O)CN3CC(=O)NC3=O)C2)n2ccnc21)C(C1C(C)C1)=O Cc1ccc(-n2[nH]c(C(=O)N(CC)C3CC3)cc2=O)cc1.C(=O)(CNC=O)N Cc1ncnc(C)c1CC(=O)NCCCC(C)NC(C1(C(F)F)CCCCC1)=O N1(C(CCOCC)=O)CCN(C(=O)Cc2sc(O)nc2O)CC1c1ccnn1C C(=O)C(C(F)(F)F)C(F)(F)F.C(=O)(C(F)OC(F)(F)F)N(C)CC1CC1 N1(C(C(C2CCN(C(=O)C=CCN3CCC3)C2)C)=O)CCC2(C1)CC2(F)F Cc1cn(C(C)C)cc1C(=O)NC(C)(C)CC.C(=O)(CN(C)C(C)C)N N1(C(c2n[nH]c(CC)c2C)=O)CC2(CC2)CC1C(=O)NC(CCF)C(=O)O C(=O)(CCC(F)(F)C(F)F)N1C(CNC(c2c(OC)ccs2)=O)C(C)(C)CC1 Cc1cc(=NC(=O)C(=O)NC2CCCC2c2ccccc2)[nH]o1 C(=O)(C(F)CCC(C)(C)C)NC1C(Cn2cc(CC(C=C)O)nn2)CCC1 C1(C(C)C)CN(C(C2CCC2CF)=O)CCN1C(=O)CCc1cnccn1 N1(C(CC(C(C)(C)NC(C#CC(C)C)=O)C)=O)CCOC(C2(C)N=N2)C1 C1CN(C(=O)CCc2ccoc2)CC1C(F)F.c1(CCOC)cc(C=O)no1.N c1(C(N(Cc2cn(-c3ccc(C)cc3F)nn2)O)=O)c[nH]c2nccc-2c1 c1(NCC2OCCN(C(C(CC(C)C)NC(C)=O)=O)C2)ccnc2ncnn12.OC O=C1CCC(CO)(CNC(=O)C#CCNC(C2CCC3CC23)=O)N1 CC1(C)CCC(CNC(C2(C)CCCN2C(=O)C(C)(C)F)=O)OC1 N1(C(CC)=O)c2ccccc2C(n2cc(CCCCO)nn2)C1(C)C C1CCC(N(C(=O)CNC=O)C)CC1.C(=O)(CCC1CCC1)N.CC[SH](=O)=O C(=O)(C1CCCn2nccc21)N1CC(N(C)C(C2CCn3nccc3C2)=O)C1 N1(C(C(C=C)OC)=O)CCN(C(C2CCCCC2N=[N+]=[N-])=O)CC(O)C1 C(CCF)(C(=O)NCCCC1CCCCO1)NC(Cn1nnc(C)n1)=O c1(OCC)ccc(CNC2CCC(C)N2Cc2ccc(Br)nc2Br)cc1[N+](=O)[O-] C1(CC=O)COCCN1C(C)C.C1(C(N2CC(OC)(C)C2)=O)CCC(C)CC1 C(=O)(CS(=O)(=O)c1ccccc1Cl)N1CC(N(C(C(C)O)=O)C)C1 c1(N2CCOCC(C(N3CCC(C(CC)O)CC3)=O)C2)ncnc2n[nH]cc12 CC1(C(N2CCC(C)CC2)=O)CCC(=O)C1.c1(C2C(C=O)C2)ccc(F)nc1.N c1(C(C)C)cccc(C(=O)N(CC(C)(C)CNC(=O)CC(C)C2CC2)C)c1F CCC(CCC(=O)NC(C1CCN(C(c2csc(C(F)(F)F)c2)=O)C1)(C)C)OC CCC(C(=O)N1CC(NC(c2cc(F)ccc2OC)=O)CCC1C)C(C)(F)F N1(C(c2c(N)cc(F)cn2)=O)CCCC(O)(CNC(c2ccc(=O)oc2)=O)CC1 Cc1cn2cc(CC(=O)NCC(N3CCC(C)CC3)C(C)C)nc2s1 N1(C(C(C)C)=O)CCC2(CC2)C1.c1(COC(C)=O)cccc(C(F)(F)F)n1 C1(CC)CN(C(=O)CCOC)CCN1C(C1CC=CC1)=O C1(C)(C=O)CCNC(=O)C1.c1(C(=O)NCC(C)C)c[nH]cc1-c1ccc(Cl)s1 Cc1cnc2cccc(C(=O)NC3CC(CNC(c4sc(F)cc4C)=O)C3)c2c1 N1(C(C(CC=C)(C)NC)=O)CC2(C1)CN(C(=O)CSCC)CC(C)(C)O2 c1(N2CCCC(CC=C)(NC(C3CC3(F)F)=O)C2)ccc(C(C)=O)cc1[N+](=O)[O-] C1(C(C)NC(Cc2c(C)non2)=O)CCCN(C(=O)CCSc2nnnn2C)C1 C1(C)(C(N2CC(NC(c3cc(C)oc3C(F)(F)F)=O)C(C)C2)=O)CCN(C)CC1 c1(OC(C(=O)N(C2CCCCCC2)CC)COC)ccc2c(c1)CCCO2 C#CCCCCCCC(=O)NC(CC(=O)NC12CCC(C1)OC2C)C(F)F c1(C(=O)NC2CC(NC(CCOCCC)=O)C23CCC3)ccc(F)c(Cl)c1N N1(C(C2CCCN(C(C)=O)C2)=O)CCCN(C(=O)Cc2cc(Cl)n(C)n2)CC1C CC(CC(N)=O)N(C(=O)CC(C1CC1)NC(=O)CNC(N)=O)C C(=O)(C(CC1CCCC1)NC(=O)CCC1CCOCC1)NC(CCC)C1CC1 C1(NC(C(CNC(C2(OC)CCOC2)=O)O)=O)CCCC1(C)C C(=O)(CC(C)(C)C#N)N1C(C(=O)NC(CC=C)C2CC2)CC(O)C1 Cc1nc2cc(C(N3CCN(C(C4CC(O)CN4C)=O)CC3CO)=O)ccc2s1 Cn1ccc2sc(C(=O)NCCCN3CCN(C(C45CCC4C5)=O)CC3)cc12 C(=O)(C(O)CC(F)F)NCC1CC(OC)CN1C(=O)Cc1nc[nH]n1 O=C(NOC1CCCCC1)C(O)CCCNC(C1CC2(CC2)C1)=O CC1CC(c2nnnn2-c2ccccc2)(NCCC(=O)N(C)C2CC2)CC(C)S1 CC(C)C(C(=O)N1CCC(NC(=O)Cn2ccnn2)C1C(C)(C)C)C(C)C.C c1(C(=O)NC2C(CNC(c3ccccc3)=O)CCCC2)cc(Cl)cc(Cl)c1O C1(C=O)CC1(C)Br.C(=O)(C(C1CCCO1)C1CC1)N(C)CCOCC.N N1(C(CC2(C)N(C(C34CCC(OC)C3C4)=O)CC2)=O)C(CO)CC2OCCC12 C(=O)(CC(C)C(C)(C)NC(=O)C(C)SC(C)C)NCC1CCC(=C)CC1 C1(C(=O)NC(Cc2ccco2)CO)CCOCCN1C(=O)CC1CCCSC1 C1(NC(c2ccc(Cl)cc2O)=O)CC2CC(C1)N(C(c1ccc(CF)cc1)=O)C2 N1(C(COCCCOC)=O)CC(C)C(O)C1.C(=O)(C(F)Cc1ccccc1)N Cc1cccc(N2CCN(C(CC3CCOC3)C(=O)NC3CC3)CC2)c1C CCC1=C(C(=O)N2CCN(C(C3CC(F)C3)=O)C(CCOC)C2)SCCO1 C1(C2CN(C(=O)C(CO)N(C)C)C2)(NC(CCSC)=O)CC1 CC1=C(C(=O)N2CCC(C(F)C(=O)NCC3(CO)CC3)C2)CCO1 C1(CNC(c2cnsc2)=O)CCCN(C(=O)CNC(c2nccs2)=O)C1 C1(O)(C(=O)NCCCN2CCOCC2)CCN(Cc2ccccc2)C1.C1(C)CC1 CC1(C(=O)N(CC#N)CC#N)CC12CCN(C(c1ccco1)=O)CC2 c1(C(ONC(c2ccccc2)=O)=O)cccc(OC(F)F)c1F.[nH]1ccccc1=O N1(c2cc(NCCC(C)CCO)nc(C)n2)CCC(C2=NOCC2)C1 Cc1cc(C(=O)NCC(C)NC(c2occc2-c2ccc(F)cc2)=O)oc1Br c1(OC)ccc(CC(=O)N(CCCNC(c2c(C)noc2C)=O)C2CC2)cc1Cl Cc1cc(OCc2cc(-c3ccc(C)c(F)c3)n[nH]2)n2nc(C(F)(F)F)nc2n1 C1(NC(C2C(NC(CC)=O)CCO2)=O)CCC=CCC1 c1(N2C(CN(C(C(C)CS(C)(=O)=O)=O)C)COCC2)cnc2ccccc2n1 C(C(CNC(C1COCCN1C)=O)S(C)(=O)=O)NC(Cc1c(C)scc1)=O c1(C(=O)N)cc2c(F)cc(F)cc2o1.C1(C(=O)NCCCC)CCCN1C(C)C Cc1cc(C(=O)NC(c2nocc2C(=O)NC(c2ccccn2)C)C)c(C)cn1 CC1CCC(C)(CNC(=O)CCCCN(C)C(C2(N(C)C)CC2)=O)CC1 N1(C(C2C(C(N(CCOC)C)=O)C2)=O)CCCC(C)CC1 c1(NCC2CCC(=C)CC2)ncccc1S(=O)(=O)NC1(C)CC(C)(C)C1 C1(NC(=O)CO)CCCCCN(C(c2sccc2-c2ccccc2)=O)C1 CCCC(O)CCNC(c1cccnc1CNC(c1cc(C)co1)=O)=O C(=O)(C(C)(F)C(C)(C)F)N(CCCCC(=O)N1CCC1)C.C(=O)(CO)NC Cc1ccccc1OCC(=O)NCC1(CC)CC1.C(=O)C(C)c1ccco1.N c1(CC(N2C(Cc3cn(CC(=O)O)nn3)CCC2)=O)cccc(Cl)c1F N1(C(C(C)Sc2cc(NC(C)=O)c(Cl)cc2)=O)CCn2cccc2C1C c1(C(N2CCC(c3ccccc3F)C2)C(=O)NCCOC)cc2c(o1)CCCC2 c1(NC(C2(C)CC23CCC3)C)cc(Br)ccn1 C1(CNC(CCc2nc(=N)[nH][nH]2)=O)CCC(NC(=O)CC2CNC(=O)C2)CC1 C1(C)(CNC(C2N=C(C)SC2)=O)CCN(C(C2CCSC(C)C2)=O)CC1 N(C1CCc2cc(Cl)ccc21)C(C(N1CC(OC)C(OC)C1)=O)=O c1(CC=O)cn2c(n1)CCCC2.C=C1CC(C(=O)N)(C(F)F)C1.C1CC1.C c1(OCC)cnc(C(=O)N)cn1.CC(C)(C)CN(C)C(C1CNC(=O)N1)=O N1(C(COC(C)=O)=O)CCC(F)(F)C(CNC(c2cnc(Cl)c(F)c2)=O)C1 c1(NC(c2c(C)c(Br)cc(F)c2)=O)ccc([N+](=O)[O-])cc1Cl C(=O)(CC(CN(C)C)CC)N1CCC(NC(CCC(=C)C)=O)C1c1ccccc1 C(=O)(C(C)(O)C(F)(F)F)NC1C(NC(C2C(C)(C)CCC2)=O)CCCCC1 C1(C(C(=O)NCCCN(CC(CC)CC)CCOC)C)CCCCCC1 C=Cn1nccc1C(N1CCC(CCC(=O)NC2CCCN(CCO)C2)C1)=O N1(C(c2cc(COC)on2)=O)CCC(=CC)CC1.n1(CC=O)nc(C)cc1C C(=O)(CC(CC)C1CC1)NC1(C(=O)NC(C(=O)NCCC)C)CC1(C)C N1(C(CN(C)C2CC2)=O)CC2CCC2(CNC(c2cncc(Cl)c2)=O)C1 N1(C(C2CC(C#C)(O)C2)=O)CCC(=C)CC1C(=O)NC(C(=O)OC)C1CC1 N1(C(C(CC)OC)=O)CCc2ccccc2C1CNC(c1ccc(F)cc1Cl)=O c1(C(N2CCC3(C2)CC3)=O)cc(S(N)(=O)=O)c[nH]1.CCC=O.C(C)OCC.O N1(C(C(C)c2cccs2)=O)CC(NC(=O)Cc2ccccc2F)CCC(O)C1 C1(C(=O)Nc2ncccn2)CC2CCCCC2N1C(C1CCCS1)=O C(C)(CCC(=O)NCCC1CCCCN1C(=O)COCCCC(C)C)OC CC(CCCCCO)NC(=O)C(C1CCOC1)NC(c1ccc(F)cc1)=O CC1(CNC(C2(C(F)F)CCOCC2)=O)CCN(C(=O)C(c2ccccc2)F)C1 c1(-c2cccc(CC(N3CCC(c4ncccn4)CC3)=O)n2)cc(F)ncc1Cl C1(C(=O)NCC#CC(F)(F)F)(CC)CCN(C(=O)C(C)CCOC)C1 N1(C(CNC(C)=O)=O)CCC2(CCC2NC(=O)CCC(=O)c2ccc(C)s2)CC1 c1(C(=O)NC2CCOCC2NC(c2ncncc2Cl)=O)c(O)cccc1Cl c1(C(=O)NC2CC(C(N3CC4CC4C3)=O)C2)ccc2c(c1)Cc1ccccc1-2 N1(C(c2ccc(NC(C)=O)cc2)=O)CCC2C(NC(=O)C)CC12.CC(C)C.O CC1CN(C(=O)CC2CC2C(F)(F)F)CC(C)N1C(c1ccn(C)n1)=O N1(C(C2C(CC)C2)=O)CCCCCC1C(=O)N(C)Cc1nnnn1C C1(C(=O)NC(c2nn[nH]n2)CC)CCN(C(=O)CCSC)C1C(C)C CC1(C)COc2ccc(S(=O)(=O)NC(C34CC(F)(C3)C4)=O)cc21 C1(C=O)CCS(=O)(=O)N1.N1(C(c2ccoc2C(F)(F)F)=O)CCCC1.CC N1(C(c2cccc(C)c2N)=O)CC2ON=C(CNC(c3coc(Cl)n3)=O)C2C1 C(=O)(C(C)CC(C)(F)F)N(CC(CN(C(Cc1ccccc1)=O)C)O)C.CCS CC(C)C(F)C(=O)NC(C)CCCNC(=O)CC1CCCCO1 C(=O)(C1=C(C)S(=O)(=O)CC1)N1CCC(F)C1.C1(C(=O)OC)CC1C(=O)N c1(C(N2C(C)(CNC(C(C3CCCC3)OC)=O)CCC2)=O)ccc(F)c(Cl)n1 N1(C(CCc2onc(CC)n2)=O)CC(NC(c2ccnn2C)=O)CC12CCOCC2 N1(C(C(=O)Nc2cccc(OC)c2)C(C2CC2)OC)CCOc2ccccc2C1 N1(C(C2(CSC)CCC2)=O)CCC2(C=C(C(=O)N3CCCCC(CO)C3)C2)C1 c1(N2CCC(CC(=O)N(C)Cc3ccc(C(=O)O)cn3)C2)ncnc2c1CCCC2 CC1CC(CNC(=O)CCOC2CC2)CN1C(=O)CCc1c(N)cnn1C CC(C)CC(C)CC(=O)NC(C1(CNC(c2cc(Br)n[nH]2)=O)CC1)C N1(C(CC=C)=O)CC(CNC(c2ncoc2CCC(F)(F)F)=O)CC1C CN1CCCC(C(=O)NCCn2cc(C=O)cn2)C1.C1CCN(C(C)(C)C)C1.N C1(N(C(=O)CC2CC(C)(C)C2)CCC)CCN(C(C2(Br)CC2)=O)CC1 c1(OC)c(Cl)ccc(C(=O)NCC2CN(C(c3ccoc3)=O)CCCO2)c1N C#Cc1nc(C(=O)NCC(C2CCN(C(=O)C=C(C)C(C)C)CC2)(C)O)cs1 C1(C(=O)N)CCc2n[nH]cc2C1.C1(NC(C=CC(=O)OCC)=O)CCCC1 c1(SC)cnn(C)c1C(=O)NC1(C2CCCN2C(=O)CC2CCOCC2)CC1 N1(C(C)=O)CCN(C(C2CN(Cc3ccc(C)cc3O)C2)=O)C(C)C1 N1(C(c2cccc(C(=O)NC)n2)=O)CC2CC(C1)C2.C(=O)CCC1CC1(F)F C1(NC(C2CC(F)(F)CS2)=O)COC2(C1)CN(C(c1cc(O)ncn1)=O)C2 C(C(=O)N1CCSCC1)(C(C)(C)O)NC(CN(CC(C)(C)C)C)=O CC1CC(C)(C)CN1C(=O)C(Cn1cncn1)NC(c1coc(CO)c1)=O c1(C=O)ccc2c(c1)C(=O)NC2=O.C(C(C)(C)C)N(C(=O)Cc1ccon1)C N1(C(c2ccc(CO)o2)=O)CCC2(CCN(C(c3ccc(Cl)cc3Br)=O)C2)C1 c1(NC(c2cccc(NC(C(C)OC)=O)n2)=O)nc(Br)c(Br)cc1Br C(=O)(C(CC(C)(C)C)OC)NC1(CCCNC(CC(=C)Br)=O)CC1 N1(C(C2(C3CCOCC3)CC2)=O)C2CCC1CN(CCn1cnnn1)CC2 C(=O)(CCCC(=O)N(C)C)NC(C)C=CC(=O)NCCC1CCC(C)(C)O1 N1(C(C2(COC)CC2)=O)CC(C)C2(CC2)C1.C1(C(C=O)O)CCCCC1.N Cc1cc(C)n2nc(C(C)(C)O)nc2n1.n12c(N3CCOCC3)nnc1C2 c1(N2CC3CC(C)(C)C3C2)nc(=NCc2ccc(Br)s2)[nH]c2cc[nH]c12 n1(CC#C)c(C)cc(C(=O)N(C2CN(C(c3n[nH]c(C)n3)=O)CCC2C)C)c1C C=C=C(C)CC(=O)NCC1CC1C(=O)NC(C)CCNC(=O)OC C(=O)(C1CC=Cc2ccccc21)N1CCCCC(CNC(CCCCOC)=O)C1 c1(C(N2CCC2)=O)cc2n(n1)CCCC2.c1(C(C(=O)NC)OC)ccc(F)cc1 N1(CCC)CC(C(=O)NC2C3CN(C(C)CCOCC)CC23)CC1=O C12(OC)CCCC1(C(=O)NCC(O)CN(C)C(c1[nH]c(C)nc1C)=O)CCO2 C(CCCC(C)(C)C(=O)NNC(=O)C1(Cl)CC1(C)C)NC(C1CCN(C)CC1)=O N1(C(c2ccnn2C)CC)CCCC(C)(C(N2CCC(CC)CC2)=O)C1 C1(NC(COC(C)C)=O)CC2(CCC(NC(C3CC(=O)C3C)=O)CC2)C1 C1(OC)CCCCC1C(=O)NCCCCCN(C)C(c1ccc(C(C)=O)s1)=O c1(CC)c(C)[nH]c(C(=O)C(N2CC(F)(F)CC2C(N)=O)C)c1C Cc1cc(C(N2CCOC(C(C)NC(c3n[nH]cc3Br)=O)C2)=O)nc(C)n1 c1(C(N2CCOCC(C(=O)NC(c3ccno3)C)C2)=O)cn2cccnc2n1 n1(CC)cnc2c(N3CCC(C(C)C)C3)nc(N3CCC4(CC=CCO4)C3)nc12 Cn1cc(C(=O)NCc2nocc2C(=O)NC(CCO)C2CCCC2)nn1 N1(C(C(CCC)C)=O)CCC(O)C(C(=O)N(c2cccnc2C)C(C)C)C1 n1(CC(N2CC(CC(C(=O)NC(C)CC3CCC3)F)C2)=O)ccccc1=O N1(C(CCCCCC)=O)CCCC(C)(C)C1CNC(=O)C=CS(C)=O c1(CN(C(CC2CCN(C(C(C)OCCC=C)=O)C2)=O)C)cccc(C)c1 C=C=CC(C)C(=O)NCCC1(C)CCN(C(=O)Cc2cnc(C3CC3)[nH]2)C1 CC1(C(=O)NCC2(F)CN(C(=O)C(Cl)=CCl)C2)CC1(Cl)Cl c1(NC(=O)NCCC2(C(=O)OC)CCCC2=O)ccc(F)nc1 C(CC(=O)NC(CO)CO)(c1ccccc1)NC1CC(N)C1 CON1CC(C(=O)NC23CCC(CC2)C3)CC1=O.C1(C(=O)N)CC1C(N)=O N1(C(C2CC(C)CN(C(c3cncn3C)=O)C2)=O)CCc2ccc(F)cc21 CC1CC(C(=O)NCC23CC(CO2)C3)CC(C)O1.C1(=CC=O)CCCCC1 Cc1cnnc(O)c1C(=O)NCC1C2CN(C(C3Cc4nccn4C3)=O)CC12 c1(N2CCC(NC(=O)CCCCCOCCO)(CF)C2)c[n+]([O-])ccc1[N+](=O)[O-] CC1CN(C(c2ccccc2N(C)C(C)C)=O)CC(C)N(C(=O)CN(C)C)C1 C=C(C)CN=C(NCCOC)NCC1(C)CCC(=O)N1.C1CCC(C(F)F)CC1 Cn1cnc2cccc(C(N3C4CCC(C4)C3C)=O)c12.N(S(N)(=O)=O)CC=O C(=O)(CCCC(C)(C)C)NC(C(C)(C)NC(C=C(C)c1cccnc1)=O)C N1(C(c2cncc(OC)n2)=O)CC(=O)NCC1C(=O)NCC1CCCC1(C)C N1(CC)CCOCC1C(=O)NC(C)(C)C=CC(=O)Nc1ccc(Cl)cc1 CC(C)(CC1CC1)C(=O)N1CCC(CF)(NC(=O)CCF)C1 C1(C(=O)N)CC2CC(=O)C1C2.c1(C(=O)NC(C)CC2CC2)cn(CC)cn1 N1(C(C2(C(=O)OC)COC2)=O)CCC(CCC(=O)NCCSC(C)C)CC1 c1cc(Cl)c2c(c1)OCCO2.c1(C(=O)OCCC)ccc(NC(=O)NC)cc1 C1(S(N)(=O)=O)(C=O)CCCC1.CC(CC(F)F)C(=O)NCc1nc(C)cs1 C(=O)(CCS(C)(=O)=O)NC1(CO)CCN(C(C(c2ccn(C)c2)C)=O)C1 C1(C(=O)NCC(CN(C(C(C2CC2)OCC)=O)C)(C)C)CCCC(O)C1 c1(C(n2cc(C(C)C(=O)O)nn2)OC2CCOC2)cc(N2CCOCC2)cnn1 c1(C(N2CC3C(CNCc4cccc(OCC)c4)(C3)C2)=O)cc(Cl)ncc1F c1(CC)cccc(C(=O)NC2CC3C(NC(=O)C(C(C)C)N(C)C)C3C2)c1C c1(C(=O)NCC(C)N(C(C(C=CC)O)=O)CC)cc(C)cc(O)n1 c1(OC)cc(C)nc(NC23CC(C(=O)NC(CO)C(C)C)(C2)C3)n1 S(=O)(=O)(c1ccc(OC(F)F)c(F)c1)NC1CCN(C(=O)NCC)C1 C1(CNC(C2(NC(C)=O)CCC2)=O)COCC1.C(c1ccsc1)=CC=O CC1CC(C(=O)NC2CCCN(S(=O)(=O)C3CC3)C2)CC(C)N1 C1(C(N)=O)COCC1NC(C1CCC(CNC)O1)=O.c1c[nH]nc1C(=O)NO N#Cc1cccc(C(=O)NC2CN(C(c3conc3C3CCC3)=O)CC2O)c1F C(C)(CO)(CCF)NC(CC1C(NC(C2C(C)=CCS2)=O)CC1O)=O n1(CC)nc(C)cc1C(=O)NCC1COCC1.n1(CC=O)ncn(C)c1=O CCC(C(=O)OCCCCCSc1noc(C)n1)N1CCCC1=O N1(C(C(=O)NC(C)C)=O)CCCC(CCNC(C2CC2C2CCC2)=O)CC1 C1(CCC)CN(C(C2CC23CCOCC3)=O)CCN1C(=O)C1=CC(C)(C)C1 Cc1nc(C)c(CC(=O)NCC2(C(C)(C)O)CC2)s1 C1(C(=O)NCC(C)CNC(c2cnc(Br)s2)=O)CC(=O)N(C(C)C)C1 CCCC(CN1CCCC(COc2ccccc2)C1)CC C1(NC(c2c(C)ocn2)=O)CN(C(=O)CCCC2CCC2)CC1(C)C C1(NC(c2cnco2)=O)C2CC3C(C2)C13C(N1CCOCC1CO)=O N1(C(C(C(C)C)(F)C)=O)CC2(COC(C)(C)C2)C1.C1(=CC(=O)N)CCCCC1 C1(O)(CN(C(CCC(=C)C)=O)C)CCN(C(C2(C)CC2C(F)(F)F)=O)CC1 CCC(C#N)C(=O)NCCN(C(=O)CCc1nnc(-c2ccsc2)o1)CC(C)O c1(C(=O)NCCC(C)(C)NC(c2ccco2)=O)cnn2c1C(=O)NCC2 N1(C(C=Cc2nc(C)c(C)[nH]2)=O)CCCC(C2CC2NC(=O)CCC(C)(F)F)C1 CC1(C)CC2(CC2C(N2CCC(C)(C)C2)=O)C1.c1(C=O)cnc(N)c(N)c1.C C1(c2n(CC(=C)C)c(N3CCC(C(=O)OCC)CC3)nn2)CN(C)CC(C)O1 C(c1cccc(F)c1)=CC(N1CCC(CC)C1)=O.c1(OC)cncc(C(=O)N)c1 c1(C(=O)NCc2cnc(OCCO)nc2)nc(O)c2c(-c3cccs3)csc2n1 C1(NC(c2cc(C)nc(C)c2)=O)CCC2CCN(C(c3oncc3C)=O)C12 CC1CC(NC(c2ccon2)=O)CN(C(C2CS(=O)(=O)C2)=O)C1.N(C)(C)C CC(C)C(C)C.C1(C(=O)N)CC(O)(C(F)F)C1.c1(C=O)cc(C2CC2)on1 c1(C=O)cc2[nH]nc(C)c2cn1.C(=O)(CC(C(=O)NC1CCC1)N(C)C)OC.N CC(C(=O)NCCCNC(C1(C(C)(F)F)CC1)=O)C1CCC1 C1(CC(=O)NCC2CN(C)C(=O)C2)CCN(C(c2cncc(N)c2)=O)C1(C)C C(C(=O)NOCCCN(C)C)(c1cccs1)NC(C(COC)C)=O Cc1ccc(C(=O)NC(C2CCCCO2)C(=O)O)c(N)c1Cl n1(CC(=O)NC(CNC(C2(C)CCCCO2)=O)C2CC2)ccc2ccccc12 C(=O)(C(C(C)C)c1ccc(F)cc1)NCC(CNC(c1ccn(CC)n1)=O)O c1(C(=O)NC(C)C(C)C(=O)NCCc2ccccc2F)ncc2ccccn12 c1(N(C)CC2N(C(C(n3cc(C)nc3)(C)C)=O)CCC2)nc2cc(Cl)cc(Cl)c2o1 c1(C(=O)NCC2N(C(c3nc(C)sc3C)=O)CCC2)ccc(P(C)(C)=O)cc1 c1(C(N2C(C(N3CCC(O)C(F)C3)=O)CC3CC32)=O)cc(O)nc2ccccc12 C=CC(CC)CC(=O)N1CCN(C(=O)CN(C(=O)CCC2CCCOC2)C)CC1 c1(CNC(CCN(C)CCO)=O)ncc(C(=O)N)cn1.C1([Si](C)(C)C)CC1 C1(C(=O)NC(C)C(C)O)(CNC(c2cnc(C(C)C)o2)=O)CCCCC1 C1CC2(CCN(C(=O)C)CC2)C1.Cc1nn(C)cc1C(O)C(=O)N.C(N)=O.C N1(C(C(CC)OC)=O)CCN(C(C2CC3(C2)CC3F)=O)C(CC)C1 C1(CC(=O)Nc2cccc(NC=O)c2)CC2(CC2)CO1.C12(CC)CCCC1C2 c1(NC)ccc(C(N2CCC(C(C)C(=O)NC3CC4CCC3O4)C2)=O)cc1 N1(C(CC=C=C)=O)CCC2(C1)CN(C(c1cc(-c3ccc(Cl)cc3)no1)=O)CCO2 c1(OC)cc(C(N2CCCC(NC(=O)C3=CCCOC3)CC2)=O)cc(Cl)n1 c1(C(=O)NCCc2cc(C(=O)NCc3c(C)ncs3)no2)cncc(Cl)c1 N1(C(C(C2CCC(=O)N2)C)=O)CCC(F)(C)CC1.C1(C=O)CCN(C)C(=O)C1.N C(CC(F)(F)F)(c1ccc(C(F)(F)F)cc1)OC(CC(C)C1CC1)=O C(=O)(CC(C)(C(F)F)N(C)C)N1C2C(NC(Cc3cncc(C)c3)=O)CC(C2)C1 N1(C(CN(C)CC)=O)CCCCC(N(C)C(c2cnc(C)nc2NC)=O)C1 c1(NC(c2ccc(CCC(=O)Nc3ncco3)[nH]2)=O)cccc2c1OCC2 Cc1cccc(NNC(=O)NC(c2nc(-c3cccs3)n[nH]2)C)c1Cl C1(COC)CCN(C(=O)C(C)(C)c2sccc2Cl)C1.C(=O)(CCc1ccco1)N CC(C)CC(CCO)NC(=O)CC(O)CNC(=O)Cc1cccnc1O c1(C(N2CCC(C)(CNC(CCCCCC)=O)C2)=O)ccc2nc(C)cn2c1 c1(C(C#C)NC(=O)N(CCN(C)C)Cc2cccc(Br)c2)ccccc1.O N1(C(Cc2nc(C(=O)Nc3ccnc(F)c3F)sc2)=O)CCC(S(N)(=O)=O)CC1 c1(C(=O)NCC(C)C2CC2)n[nH]c(C2CC2)n1.c1(C=O)cscn1.C1CC1 c1(CC)cccc2c(C(=O)N(CCCCC)C)c[nH]c12.C1(C(=O)N)(C(N)=O)CC1 Cc1[nH]nc(C(F)(F)F)c1C(=O)NCCC(C)NC(=O)C.c1ccccc1O.O Cc1ccc(CC(CO)NC(C2CCN(C(c3ccc(C)nc3)=O)CC2)=O)cc1 c1(NC2C(NC(CCC(C)OC)=O)CS(=O)(=O)C2)nc(Cl)[nH]c2ncnc1-2 C1(CNC(CCN(C(=O)C(C(C)C)SC)CC)=O)CCC2(CCC2)O1 N1(C(C(C(C)C)NC(=O)CC2CCOC2=O)=O)CCCNC(=O)C12CC2 CC1(C)OC(C(=O)NC(C)C(C)(C)C)C(C)(C)O1.c1nc[nH]n1.C(=O)C.N C1(C(=O)NCC2N(C(C=C(C)Cl)=O)C3C(C2)C3)(N(C)C)Cc2ccccc2C1 CC1(C)CCC(C(N2CC3C(CNC(C4CC45CCCC5)=O)C3C2)=O)CC1 C(c1nc2ccccc2s1)=CC(=O)NCCS(CC(C)C)(=O)=O C=CCCC(=O)N(CC)C1CC1.C1(C2(C=O)CCC2)CCCCO1.C(C)(=O)N c1(OC)ccc(CN(C)C)c(OC)c1.c12ccc(cc1)C1(CCOCC1)N(C)C2 c1(C(=O)NC(C2CCCN2C(C2C=CCCC2)=O)C)cc2c[nH]cnc-2n1 c1(C(C)NC(=O)CC2CCCN2C(c2ccccc2)=O)cnc(N(C)C)nc1 c1(SCCC(N2CC(CCc3ccc(C)cc3)C2)=O)nc2ccccc2s1 c1(C(N(CCNC(C(C)OCC)=O)C)=O)ccc2occc2n1 C(=O)(CN1C(=O)Cc2cc(F)ccc21)N1CC(c2ccc(OC)cc2)(O)C1 Cc1cc(C)n(C(C)C(=O)N(CC(O)CNC(C2(Cl)CC2)=O)C)n1 N1(C(C=CCN(C)CC)=O)CC2COCC2(C(=O)NOCC2CCOC2)C1 c1(OC)ccnc(O)c1C(=O)N.C(CCN(C)C(C1CC(C)=NO1)=O)C(C)C c1(OC)cccc(C2(NC(=O)CCCn3ccnc3C)CC2)c1 c1(CC)nc[nH]c1C(=O)NC1CN(C(=O)CCOC)C1 CCCCC(F)(F)C(=O)N1CC=CC(C(=O)Nc2cccc(C)c2)C1 C1(c2cnc(CC)nc2)NC(=S)N(CC2CCCO2)C2=C1C(=O)NCC(C)C2 C(=O)(C(CC1CCC1)NC(=O)O)NCC1CC(N(C)C)C1.C(C)(C)C C(=O)(CC(O)C)NCCOCCOCC.C1(C=O)CC(=O)N(C)C1.N c1(C(=O)NCC2C(C)(C)N(C(C3CC3CF)=O)CC2)c(F)ccc(Br)c1Cl N1(C(c2nc(COC)n[nH]2)C(=O)NCCOC)CCCC2CCNC(=O)C12 c1(C(=O)NC2CCCC(NC(c3cc(OC)n[nH]3)=O)C2)cccc(C)c1C C1(N(C(CNC(c2ccc(C)s2)=O)C)C)CCCNC1=O C1(NC(C(CC)NC(C)=O)=O)CN(C(c2cnn(C)c2SC)=O)CC1F c1(C(=O)NC2C(NC(c3c(C)nc(CC)s3)=O)CCCC2)cnc(C)nc1C C(=O)(C(C)(C)C(C)O)NCCCOCCNC(C=Cc1c(C)nsc1)=O C(C(C)(O)CN=[N+]=[N-])NC(CN(c1ccc(-n2cccn2)nc1)C)=O CC1COc2ccccc2C1NS(=O)(=O)c1cnc(NC2CC(F)C2)c(Cl)c1 N1(C(c2c(F)ccc(C)c2)=O)CC(NC(c2cnc(O)o2)=O)C(C2CC2)C1 c1(N2CCC(OCCNC(C3N(C)CC(C)(C)C3)=O)C2)ncc(C#N)cc1Cl c1(CN2C(C(N3CCCC(C#C)C3)=O)CC3CC32)cc(Cl)cc(Br)c1F C1(C(=O)NCCCCN(C)C)CCCCN(C(=O)CCc2ccc(=N)[nH]c2)C1 N1(C(c2c(CCC)n(C)nn2)=O)CC(C)CC1(C)C.C(=O)(C(F)=C1CCCC1)N Cc1c(F)ccc(C(=O)NC2C3CN(Cc4cccc(F)n4)CC23)c1F C12(CNC(c3ccccc3Cl)=O)CC(CO1)N(C(c1cc(O)cc(O)n1)=O)C2 N1(C(=O)C=CCBr)CCN(C(c2ccc(O)c(CO)c2)=O)C2CC12 Cc1ccc(S(N)(=O)=O)cc1C(=O)NC1CC1C.c1(C=O)ccccc1.N C1(C(=O)NCC(C(C)(C)C)NC(=O)CC(Cl)Cl)CC(=O)C12CCC2 C12(C(=O)NCC3C(NC(CCC(=O)NC)=O)CC3)CCCC(C)(C1)OC2 NC(CNC(C1(c2cccnc2O)CC1)=O)CC(F)(F)F C=CC(C)(C)C(=O)NCCC1CCC(NC(=O)C(c2ccnn2C)O)C1 C1(CNC(C2C(C(=O)OC)CC2)=O)CCCN1C(c1ncsc1C)=O Cc1nc(O)[nH]c1C(=O)N(C1CCN(C(=O)C(C)(C)COCC(F)F)C1)C CC(C)C(C)(O)C(=O)N(C)CC1CN(C(=O)CSCc2ccccc2Cl)C1 c1(C(=O)NCCC(=C)CNC(=O)C=CC2CCCO2)cc(C)ccc1OC c1(C(N(C)CC2CN(C(C3CCC4CC4C3)=O)C2)=O)cc(F)c2ncccc2c1 N1(C(COC(C)=O)=O)CC(NC(c2nn(C)cc2[N+](=O)[O-])=O)C2(CCCC2)C1 C1(C(C)O)CCC(NC(=O)C(C2CCCC2)NC(=O)C(O)C2CC2)CC1 C1(C(=O)N)CC(=O)C1(C)C.C(=O)(C(C)N(C)C)N(CC)CC1CCC1 N1(C(C2CCCC2)=O)CCCC1(C)C.C(=O)C(C)CC(F)F.C(=O)(NCC)N C1(C(=O)OCC2CC(NC(=O)OC(C)(C)C)C2)CCC2COCC2O1 CC#CCCCC(=O)NCC#CCNC(=O)CCOC1CCCOC1 CN1CCCC1C=CC(=O)OCCC1CCC(F)(F)C1 CC(CNC(=O)CC(C)c1ccco1)CC(=O)N(CC(C)C#N)C1CC1 N1(C(CCCC=C)=O)CCCC(C2CCN(C(=O)CC3CCCOC3)CC2)C1 C1(C(CNC(CC(=O)OC)=O)(C)O)CCCN(C(=O)CCC2CCC2)C1 CC1(C)OCCC1CC(=O)NCC1CCCC1NC(c1cnc(S)[nH]1)=O c1(CC)ncccc1NC(c1occc1C)=O.C1(Cl)(C=O)CC1C(C)=O C1(C(=O)NC(C)CNC(=O)C(C)(C)C(N)=O)CC2(C1)C(F)(F)C21CC1 C1(C(=O)OC)C2CCC(CC2)N1CC1CCN(C(c2ccccc2OC)=O)CC1 c1(C(N2CCC(C(C)NC(c3cn(C)nc3O)=O)C2)=O)ccc2nc[nH]c2c1 C(=O)(C(CC)CC(C)C)N1C(CC=C)(C(=O)NCCN2CCNC(=O)C2)CCC1 C(=O)(C(CC(F)F)NC(C1CC(C)=NO1)=O)NCCCOCC=C N1(C(CCc2ncc(C)[nH]2)=O)CCCC(C2CCN(c3ncc(Cl)cn3)C2)C1 C1(C(=O)NCc2ncnn2C)(NC(c2c(C)noc2)=O)CC(F)(F)C1 N1(C(c2c(C)nco2)=O)CCCC(NC(C2(CN(C)C)CC2)=O)CCC1 c1(C(N2C(CNC(CCC(C)C)=O)CN(C)CC2)=O)ccc2ncncc2c1 C12(COC)CC(CN1C(c1sccc1C)=O)C2.C(=O)C(C)Cc1cnc[nH]1.N C(=O)(NNc1ccc(Br)c(F)c1)Nc1c(C(=O)OC)nsc1 N1(C(=O)Cc2cc(Cl)ccc2Cl)CCC2(CCN(Cc3ccc(Cl)nn3)C2)C1 Cc1nc(NCCC2CCCCC2O)cc(N(CCCc2ccc(Cl)cc2)C)n1 O=S1(=O)CCC(NC(c2nc(C3CC3)cs2)c2nnnn2CC(F)F)CC1 C1(CN(c2nnco2)C)COCCN1C(=O)Cn1cnc(C(N)=O)n1 Cc1cc(C(N2CCC(=CCNC(=O)C(C)CN(C)C)CC2)=O)cc(Cl)c1 C1(C(N(CC(C)NC(c2ccc3c(c2)NCC3)=O)C)=O)CC2(COCCO2)C1 C1(O)(CC)CCCN(C(=O)C(CCC2CCC2)NC(c2ccnc(O)c2F)=O)C1 C1(CNC(C(N2CCOCC2)C)=O)CCC(NC(C2(N(C)C)CC2)=O)CC1 c1(C=O)cc(O)n(C)n1.C1(NC(CN(C)C(=O)C2CC2)=O)CC(C)C1.N c1(C(=O)OC)nnc2n1CCN(C(C1(O)CCN(C(c3ccncn3)=O)C1)=O)C2 C1(CN(C(C(C)SC(F)(F)F)=O)C)CCN(C(=O)CN2CC(C)(C)C2)C1 C(N=c1cc(F)nc[nH]1)C1OCC(CNC(c2c(CC)csc2)=O)C1 c1(C(=O)NC(C2CCCCN2C(C2CCC3(CC3)C2)=O)C)ccc(N)c(F)n1 N1(C(CC)=O)CCCC(C(=O)NC2CC(Oc3ccccc3)C2)C1 CC(C)(CCCCNC(c1coc(N(C)C)n1)=O)NC(=O)CCc1cnco1 N(C1c2ccccc2CC1F)C(=O)NC1CCN(S(=O)(=O)c2cccs2)CC1 N1(C(c2c(C)nc3ncccc3c2)=O)CCCC2(C1)OCC1CC21 N1(C(CCSC)=O)CCCC(CCNC(=O)Cc2csc(Cl)n2)CC1 c1(OC)ncc(Br)[nH]c1=NNC(=O)Cc1cc(Br)c(F)cc1[N+](=O)[O-] Cc1[nH]nc2ncc(C(N3CCC(NC(C4(O)CCCCC4)=O)CC3C)=O)cc12 CC(C)C(C(=O)N1CCC1)NC(N)=O.c1(C(=O)N)cnc(-c2ccc(Cl)s2)s1 C(=O)(CCCC(C)=O)NCC1CC(NC(c2c(OCC=C)cccn2)=O)C1 C(C)(C(C(=O)N1CCCC1(CO)CNC(=O)CC)N(C)C)OC.C1CCC1 c1(NC(C)=O)nc(C)c(S(=O)(=O)N2CC3CC2CN3C=O)s1.C1CCCCC1.N CC(CC(C)(C)C)C(=O)N1CCC(CO)C(NC(c2ccc(=N)[nH]n2)=O)C1 C1(N(C(=O)C(C)SC)CC)CCN(C(=O)COCCC)C1.c1[nH]nnc1C.O CN1CCC(C)(CNC(C2CCOCC2NC(=O)C(F)CC2CCOC2)=O)C1 Cc1ccc(CCC(=O)NC2(C)CC(NC(=O)CSCc3ncc[nH]3)C2)s1 c1(C(=O)NCC(CC)NC(c2ncccc2S)=O)cccc(OC2CCC2)c1 N#Cc1ccc(C(N2CC3CC2CN3C(c2c(Cl)cccc2Cl)=O)=O)c(F)c1 Cc1cc(CCC2(CNC(=O)NC(=O)CCc3cnco3)CCC2)n[nH]1 C1(C)(NC(CSC)=O)CCN(C(=O)C=Cc2sccc2Br)CC1 N1(C(C2C(NC(=O)CN3CCSCC3)C3CCC2C3)=O)CC2CCCC(C2)C1 Cc1n[nH]c2cc(C(=O)NC(C)CNC(c3c(F)ccc4c3OCO4)=O)ncc12 C1(CC(=O)NC2C(OC)CC2O)CCCN(C(=O)CC2(O)CCOCC2)CC1 c1(OC(C)C)cccnc1C(N1CC(N(C(=O)C(F)=CC2CC2)C)C(F)C1)=O c1cc(Cl)ccc1Cl.c1(C(CNC(c2csc(O)n2)=O)OC=O)ccccc1.N c1(N2C(CC#N)CN(Cc3ccccc3CO)CC2)ncc2c(Cl)cccc2n1 N1(C(CCSCCCC)=O)CCSCC1CCNC(=O)CP(C)(C)=O C1(NC(c2cnsn2)=O)CCC(NC(C2(C3CCCCO3)CCC2)=O)CC1 C1(CNC(c2ccc(CC)cn2)=O)CC(F)(F)CN1C(=O)C#CC1(C)CC1 CC1(CNC(=O)CC2CC(C)(C)CO2)CCN(C2CCc3c(Cl)cccc32)CC1 C1(F)(C(=O)NC2CCN(C(C)=O)CC2)CCN(C(=O)CC2CC=CC2)CC1 C(=O)(C1CCc2cc(OC)ccc21)NCCN(C(=O)C(C)C)CCOC C(CC(=O)N1CCC1(C)C(=O)NC)(C(F)F)NC(c1c(CCC)nco1)=O N1(c2ncc(=O)[nH]c2)CCC2(CCCC(CO)O2)C1 CC1OC2(CNC(C3CCCN3C=O)=O)CC1(NC(c1cccc(Cl)c1)=O)C2 C1(NC(COCCC)=O)CN(C(=O)CC(C)CC)C(C)(C)C1 c1(-c2c[nH]nn2)ccc(C)cc1[N+](=O)[O-].N1C(=O)CCC1C(N1CCCC1CC)=O C1CCCN(C(C2(C#N)CC2(C)C)=O)C1.n1(CC(=O)NC)cc(C=O)cn1.N c1(C(C(=O)NCCN(C(c2cccnc2COC)=O)CC)C)ccncc1C N1(C(C(C)(C)OC)=O)CCC2CCC(C1)N2C(c1ccsc1S(N)(=O)=O)=O N1(C(c2c(CC)ncs2)=O)CCC(CNC(c2ccnc(F)c2N)=O)C1(C)C N1(C(c2ccc(CCC)[nH]2)=O)CCC(C)(NC(c2cc(Br)n[nH]2)=O)CC1 C1(C(NOCCOC(C)C)=O)(NC(=O)CCCCC2CC2)CCCC1C C1(NC(c2c(C)coc2)=O)CCOC(CNC(=O)CCCc2ccccc2)C1 N1(C(C(c2ccc(Cl)s2)C)=O)CC(C)CN(C(c2cn(C3CC3)cn2)=O)CC1C C1(O)(C(CNC(CCOCCOC)=O)C)CCCN(C(C2(SC)CC2)=O)C1 N1(C(CCc2ccc(C(=O)OC)cc2)=O)CCC2CN(C(=O)C(C)(F)F)CC12 c1(C(=O)NCC2(C)CCCN(C(Cc3c(C)ncs3)=O)C2)c(O)cc(F)cc1F C1(C)(NC(C(F)=CC)=O)CCC(NC(=O)CC2(CO)CCCC2)CC1 C(=O)(C1=CCN(C(c2ccc(O)cc2)=O)C1)NC(CC#C)CC#C Cn1nc(C(N2CCC2CNC(=O)C(C)(C)c2cncs2)=O)cc1F N1(C(c2c(CC(N)=O)occ2)=O)CCCC(NC(=O)CCC2CC2(F)F)C1 C12(C(=O)NC3(C)C(NC(Cc4nc(C)c(C)[nH]4)=O)CCC3)CC=CC(C1)OC2 c1(NC)ccc(C(=O)N(C(C)C(=O)NCCN2CCC(C)(C)C2)C)nc1 C1(C(=O)NCC(c2ccc(C)s2)NC(=O)C(C)C2CCCC2)CCC(CO)CC1 N1(C(CC(C(=O)OC)(C)C)=O)CC(CNC(C2CC2C)=O)C2(CCOCC2)C1 CCCC(CC)C(=O)NCc1ccnc(C(=O)NOCc2ccccc2F)c1 C1(C(=O)NC2C(NC(C3CCC(=O)NC3)=O)COCC2)CCc2ncsc2C1 C#CCC(C(=O)N)C1CC1.C1(C(C)(C)C)CCCCN1C(=O)CC1CC(F)(F)C1 C1(N(C(C2(COC)CCCN2)=O)C)CCC2(CC1)CC2 O=C(C=C(Cl)Cl)NCCN(C(=O)CC1C=CCC1)CCOCCO c1(NC(=O)NCC(c2ccc(F)cc2)(F)F)cc(F)c(F)cc1C(F)F C1(C(N(CC#C)CCO)=O)CC1C1CN(C(c2cc(C)n(C)n2)=O)C1 c1(C(=O)NC2C(NC(CSCCCC)=O)COCC2)nnc2n1CCCCC2 Cc1cccc2cc(C(=O)NCCCCN(C(=O)CC3C=NN(C)C3=O)C)oc12 c1(C=O)cc2c(c(S(N)(=O)=O)c1)CCC2.N#CC1(C(=O)NCCCO)CC1.N C(=O)N=c1ccn(C)[nH]1.C1(CNC(CNC(=O)NC)=O)(C)CC12CCC2 c1(C(N2C(C(N(C3CCOC3)CC)=O)CC(C)C2)=O)ccc(F)c(F)c1 C1(CC(=O)NC)CCC(=O)NC1=O.C1(O)CN(C(=O)CCCc2nccs2)C1.C c1(C(=O)NC2C=CC(CC(N3CCC(CC(F)F)C3)=O)C2)cc([N+](=O)[O-])c[nH]1 C1(CNC(CNc2c(OCC)cccc2)=O)CCCC1N=c1[nH]cnc2ccsc12 c1(CN2CCCC(CNC(c3cc(C)cc(O)c3)=O)C2)ncc(Br)cc1[N+](=O)[O-] C1(C(=O)NC2CC3C(NC(CSCC#C)=O)C3C2)CNC(=O)CC1C C1(O)CCCCCC1.Cn1cc(C(O)C(=O)NCc2ccc(C(=O)N)o2)cn1.C C1(CN(C(CC(C)C2CC2)=O)C)CCCC(NC(=O)C(F)=CCCF)C1 n1(CC(=O)NCC2CN(C(c3c(C(C)C)ncs3)=O)C2)ncc(O)nc1=O c1(OC)ccc(SCC(=O)NCC2CCCCC2)cc1.C1(C(=O)N)C=CCC1 C1(CC(N2CCCC(NC(=O)C=Cc3ccsc3)C2)=O)CC2(CCO1)CC2.C c1(C(N2CC(CC(N3C(CCCC)CCC3)=O)C(C)C2)=O)ccc(C)c(O)n1 N1(COCC)CCC(OC2(NC=O)CC2)CC1.c1ccccn1.C1CC1C c1(N(C2CCCN(C(c3ncc(Cl)cc3Cl)=O)C2)CCO)ncc([N+](=O)[O-])cc1Cl CCCCC(C(=O)N1CC2(CCN2C(=O)C(C)(C)c2ccccc2)C1)C(C)C C1(SC)CN(C(=O)CN(C)C2CC2)CC1NC(c1c(C)nsc1C)=O c1(C(C)C)ccc(C(=O)NCC2CC(C)N(C(c3ncncc3F)=O)C2)nc1 C1(c2ccc(OC)cc2)CCCCC1N=c1[nH]c(N(C)CC=C(C)C)nc(=N)[nH]1 Cc1nccnc1CNC(=O)C(C)CNC(=O)C(C(C)C)NC=O N1(C(C2N(CC)CC2)=O)CC2CC(C1)N(c1nc(Cl)ncc1F)C2 c1(OC)cc(C(=O)NC(Cc2ccco2)C(=O)N(C2(C)CC2)C)on1 C12(NC(C(=O)NCCC(N)=O)=O)CCCC1N(C(c1cc(F)ccc1Cl)=O)CC2 N1(Cc2cc(C)on2)CC2CCN(C(=O)CCCCSC)CCC2C1 C1(C(=O)NCC(CN(C(C2(C(=O)NC)CCC2)=O)C)C)CC12CC(O)C2 C1(CNC(C23C(C)(C)OCC2C3)=O)C(C2CC2)CCN1c1cc(F)ncn1 C(C)(CC(C)(C)OC)(c1n(C(CC)(C)C)nnn1)NC.c1(C2CC2)ccc(C)o1 c1(-c2cc(C)n(C(F)F)n2)cc(S(=O)(=O)C(C)C)ccc1F CC(C)C(CCNC(=O)CC1COCCO1)NC(c1cc(C#N)cs1)=O c1(COC)cccc(C(N2CC(O)(C(C)NC(=O)CC(=O)OC)C2)=O)c1 CCCCCCC(C)C(=O)N1CCN(C)CC1C(=O)NCCCC(C)C N1(C(CCOCC#C)=O)CC(C=C)(CC(=O)N(C)CC2CCOC2C)C1 Cc1cc(C(=O)NC(C)C(C)NC(=O)Cc2ccco2)c(O)nc1C CCCC(CCC)C(=O)N(CC(C)(C)NC(c1cc(C(C)C)[nH]n1)=O)C C12(C(N(C(CC)C)CC)=O)CC(C(=O)N(CC(c3ccccc3)O)C)(C1)C2 c1(C(C)=O)ncc(C(=O)NCCC(C)NC(C2C=CCS2)=O)s1 CC(C)(C)S(=O)CCc1noc(-c2ccc(OCC(N)=O)cc2)n1 c1(C(=O)NCC=CCC(=O)NCC2(F)CCOC2)cnn2c1OCC2 c1(Cn2cc(C3CCN(C(Cn4c(C)cc(C)n4)=O)C3)nn2)nccc(Cl)c1F c1(C(=O)Nc2cccc(NC(CC(C)F)=O)c2)noc2c1CCc1sccc1-2 c1(C(=O)NC(c2ccccc2)CNC(C(N2CCC(C)C2)=O)=O)cccc(O)n1 C1(CC)CC(C(N2CCC(C3CCCO3)C2)=O)CCN1 Cc1sc(C(=O)NCC(CC(C)C)NC(=O)CN2CSCCSC2)nc1O C1(C(N(CCCc2ccco2)C)=O)CC12CCN(C(=O)C=Cc1ccncn1)C2 CCCCC(O)C(C)C(=O)NCC1CC2(CCN(C(C3(C4CC4)CC3)=O)C2)CO1 Cc1cc(S(=O)(=O)N2CC(OC(=O)C(N)=O)CO2)c(C)cc1F CN1CCC(F)(CNC(=O)C(=O)Nc2cccc(-c3nccs3)c2)C1 c1(C(=O)NCC2C(NC(=O)CSc3ccncc3)CCC2)nnn2c1CCCC2 n1(CCOC)nnc2c(NC(=O)CCc3cccc(C(F)(F)F)c3)ncnc12 C1(CCN(C(c2n(CCC)ncc2)=O)C)CCN(C(=O)Cc2c[nH]nc2O)CC1 N1(C(c2cc(COC)sc2)=O)CC2CCCCC2(NC(c2sc(C)cc2C)=O)C1 N1(C(C2(OC)CCN(C(C(C)=CC=C)=O)C2)=O)CCCC(C2CC2)CC1 C1(CNC(Cn2ccc(C)n2)=O)CCCN(C(C23COC(CF)(C2)C3)=O)C1 N1(C(C(C=C)O)=O)CC(NC(C2(C)C=CCC2)=O)CC(C)(C)C1 CCCCC(CC)C(=O)NCC1CC2(CC(NC(=O)C(C)CC3CCC3)C2)C1 CC(C)(CC(F)C(=O)N1CC(CS(C)=O)C1)NC(C1CC2(CCC2=O)C1)=O CC1CN(C(c2ccccc2CO)=O)CC(C)C1Nc1ncc(C#N)cc1Br c1(C(N(C2CCN(C(=O)C(F)C(C)C)C2)CC)=O)ccc(S(C)(=O)=O)[nH]1 Cn1nc(I)cc1C(N1CC(O)CC1Cn1cc(Cn2cccn2)nn1)=O C(C)(CC(C)N=c1[nH]c(Cl)nc2c1SCC2)NC(c1c(C)ccnc1O)=O c1(C(N(C2CCN(C(=O)C(C#N)C3CC3)C2)CC)=O)cc(C)c(C)c(C)c1 N1(C(C(CC)OC)=O)CCN(C)C(CNC(C2CCC(C(C)C)CC2)=O)C1 C(=O)(C1=CCCOCC1)NCC1(O)CCCN(C(CC2CC(CC)C2)=O)C1 C1(C(=O)N)CCC(C2CC2)N1C(=O)Cc1ccc(C)s1.C1(SC)(C)CC1 O=C(C1=C(Cl)CCOC1)NC1CC(C(=O)NC23CCN(CC2)C3)C1 N1(CC)C(=O)NC(c2cncc(Br)c2C)C(C(=O)OC)=C1CC(C)C N1(CCNC(CCC2CC(NC(CCC#C)=O)C2)=O)CCCC(C)C1 C1(NC(c2ccc(O)cn2)=O)CCCN(C(C2CCC3(CC3)C2)=O)C1 Cc1ccc(=NCCC(=O)N(C(C)CNC(c2cccc3ccnn23)=O)C)[nH]c1 N1(CCCNC(c2ccccn2)CN)CCN(C(=O)Oc2ccccc2)CC1 C#CC1(C)CCCN(C(=O)CCN(C(=O)C(C)CN(C)C)CC2CC2)C1 c1(NC(=O)Nc2cn(CCOC)nc2)c(-c2ccccc2)nn(C)c1Cl C1(OC(=O)CCOC2CCCC2)CCOCC1.C1(=O)C(=O)CCN1 C(CCN(C)C)(C(=O)NCc1ccco1)NC(C(CC)N(CC)CC)=O.O N1(C(c2cnn3cccc(C)c32)=O)CC(CO)C2(CCN(C(=O)C(F)F)CC2)C1 C(=O)(C(F)(F)CC(C)C)NC(CCN(C(C(F)=C(C)C)=O)C)C(C)C N1(CC2(NC(C=NOC)=O)CC2)CCN(C(C23CCC(OC)C2C3)=O)CC1 c1(C(=O)NC2CC(c3c(OCC)cccc3)C2)ccc2c(c1)CCC(OC)C2 C1(CC(=O)N(CCCC(=O)NC(COC)C(C)C)C)CCCOCC1 c1(C(=O)NCCCCCNC(=O)CCOCC2CCC2)c[nH]c(=S)cn1 N1(C(C(CC)CCOC)=O)CC2(COC(C)C2)C1.C1(C(=O)N)CCCC(C)C(C)C1 N1(C(C(C)(C)c2ccno2)=O)CCC(O)(CNC(C2CC2Cl)=O)CC1 c1(C(=O)NC2(C)CN(C(=O)COCC3CCOC3)C2)cc2cnccc2[nH]1 Cc1ccc(CNC(=O)C(Cc2ccco2)NC(c2cncs2)=O)cn1 N1(C(c2cnc(OC)s2)=O)CC(C)C2(C1)CN(C(c1cnc(N(C)C)s1)=O)C2 N1(c2nccc(OC)n2)CC2CCN(C(c3ccc(C)c(F)n3)=O)CCC2C1 Cc1nc(Cl)ccc1OCC(=O)NC1CCNC1.c1(-c2ncon2)ccc(Cl)cc1.C C1(C(=O)NCC(CN(C(C(c2ccc(Cl)s2)C)=O)C)O)CC2(CC2)C1 CCCCC(O)C(=O)N1CCC(NC(=O)CSC2CCS(=O)(=O)C2)CC1 Cc1ccn(C)c(=O)c1NC(C1CC2CC2N1C(C1CCCN1C(C)C)=O)=O C(=O)(C(C)(F)C(=O)NC(C)CCNC(=O)Cc1ccnc(O)c1)OC N1(C(C2CN(C(c3cccc(OC)n3)=O)C(C)(C)C2)=O)CCCN(C)CC1C C1(c2n(C(CC)(C)C)nnn2)(NCCSc2ccc(Cl)nc2)CCC(C2CC2)C1 C(=O)(C1=CCCOCC1)NC1C(NC(CCc2ccc(=N)[nH]c2)=O)CCC1 C=C(Cl)CCC(=O)NC(CNC(c1nn(C)cc1C(C)=O)=O)CO Cc1ccc(C(=O)NC2CC3CC2N(C(C2CCC(C)(C)C2)=O)C3)c(Br)c1 C1(C(=O)OC)C2COCC1CN(C(=O)CCC(F)(F)F)C2 Cc1ccc(S(=O)(=O)N2CCN(S(=O)(=O)c3ccc(Cl)cc3)CC2)c(C)c1 N1(C(=O)NCC(c2ccccc2)OC)CC(C)Sc2cc(F)c(F)cc21 C1(C(=O)NC(CCC)C(=O)N2CCC(CC(C)C)C2)CCCCCCC1 N1(C(c2cccc(C(C)(C)O)c2)C(=O)NCC(F)F)CCCC(CO)CC1 N1(C(CCSCCCC)=O)CC2CCC(NC(C3CC4CCC3C4)=O)CC2C1 c1(CC(N2CC(CC(C)NC(=O)CCC3OCCO3)C2)=O)c(Cl)cnn1C Cc1cc(OCC(N2CC=CC(C(=O)NC3(CO)CC3)C2)=O)cc(C)c1 C1(c2nnnn2C2COC2)(NCC2(C(=O)NCC)CCC2)CCCOCC1 c1(C(=O)NCC2C(NC(C3N(CC)CCC3)=O)C2)cccc2c(C)coc12 c1(C(=O)NC2C(NC(C(CC)(CC)CO)=O)C2)c([N+](=O)[O-])ccc(C)c1C C1(C(=O)NC2(C)CC(NC(C=NOC)=O)C2)CC12CCOc1ccc(Cl)cc12 c1(C(N2CC(SC)C(NC(c3ccncc3Br)=O)C2)=O)ccc(F)cc1F N1(c2nc(C)c(Br)cn2)CC(C2CCCN(C(=O)C=Cc3cccc(Cl)c3)C2)C1 c1(C(=O)OC)cc(N2CCC(N(C(=O)C(C)Oc3ccccc3)C)C2)ncn1 c1(C(=O)NCC(CNC(CSCCN(C)C)=O)O)cnc(O)c2ccccc12 c1(C(N2CC3C(NC(=O)NCc4ccc(C)cc4)C3C2)=O)cccc(=O)n1C C(=O)CCC(C)S(C)(=O)=O.n1(CC(=O)N(C(C)C)CC)cnc([N+](=O)[O-])n1 CC1CCN(C(=O)CC(=O)Nc2nccs2)CC1CNC(=O)Cn1cccc1 CCCCC(O)C(C)C(=O)N1CCC(NC(c2cncn2C(C)C)=O)C(F)C1 c1(C(=O)O)cccc2ccc(CN3CCCC(CN4CCCOCC4)C3)nc12 c1(C2(COC)CCC2)cn(CCCCCNC(C2C3COCC23)=O)nn1 C1(C)(CC)CC(NC(=O)C2=CCN(C(=O)Cc3cn(CC)nn3)C2)CCO1 N1(C(CCC2CCC(=O)N2)=O)CCCC2CN(c3ncnc4cccnc34)CC12 C1(CC(N2CCC(C(C#C)C)C2)=O)NC(=O)CN(C)C1=O Cc1cnc2c(c1)S(=O)(=O)NC1(CCOCC1)CN2.C1CC(CC(N)=O)C1.C c1c(C)nc2cc(Cl)ccn12.CCS(=O)(=O)c1ccc(NC(=O)C(=O)NC)cc1 C1(C(=O)NC(c2ncccn2)CC)CC(F)CN(C(c2ccnc(C)c2C)=O)C1 Cc1cc(=NCc2ccc(C3CC3)cc2)[nH]c(N2CC(C)CC(C)C2)n1 C(=O)(C(C1=C(C)C=CCC1(C)C)N(C(C)CC1CC1)C)NC(CC)(C)C N1(C(C2(SCC)CC2)=O)CCCCC1CCNC(=O)CCCN1CCOC1=O n1(CC(N2CCCCC(NC(C(C)(C)C3CC3)=O)C2)=O)nc2c(n1)CCCC2 C12(CNC(CNC(CC)=O)=O)CCCC1CCN2C(=O)CC(C)CC(C)C N1(C(=O)COC2CC2)CCCCC1CCC(=O)NC(CN1CCCC1)CO C1(NC(C(CC)CC)=O)CCCCC12CCN(C(C1CC(C(F)(F)F)C1)=O)C2 S(=O)(=O)(c1cc2c(cc1F)NC(=O)CC2)NCc1ncn(C(C)C)n1 c1(C(N2CCC(F)(CNC(C(C)OCC)=O)C2)=O)nccc2c1CNC2=O CCC(C#N)(CC)C(=O)NCc1cc(C(=O)NC2CCC(C)(C)C(C)C2)co1 C1(CC)C(C(N2CCCCCC2)=O)CCN1C(c1ncn(C)n1)=O N1(C(Cc2cccc(C)c2)=O)CCCOC(CNC(=O)CC2CC3CCC2C3)C1 C1(C=O)CCC2(CCC2)C1.C(CC(O)C)NC(c1cnn(C(F)(F)F)c1)=O.N C(CCCC(=O)NC(C)CNC(c1cc(C)n(-c2ccccc2F)n1)=O)OCC C(CCCCCC(=O)NCc1ccc(I)s1)NC(CC1(C)CCC1)=O c1(SC(C(CCC(=O)OC)=O)C)nc2c(s1)CCCCC2 C1(C(N2C(COC)CC2)=O)C2CCN(C(=O)CC3CCCC4CC34)CC12 CC1(C)CC2(CC2C(=O)NC2CCCN(C(=O)C(=O)C3CCCC3)CC2)C1 CC1CCN(C(=O)COc2cccc(O)c2)CC1.c1(C(=O)N)cn(C(F)F)cn1 c1(C2(C(=O)NCC(CC)NC(=O)C(C)(O)c3ccccc3)CCC2)cccnc1 C12(C(=O)NCC(C(C)(C)F)(C)F)CCN(C(=O)CCn3cccc3)CCC1C2 c1(C(=O)NCC(CC)NC(=O)COCC2CCCO2)cc(C)cc(C)c1N C1(C(=O)OC)CCC12CN(S(=O)(=O)Cc1ccncc1C(F)(F)F)C2 c1(C(=O)N)ncnc2ccsc12.C1(CCC)CC(C(=O)NCC2CC2C)C1 C1(C(C)C)CCOCCN1C(=O)C(O)CNC(=O)CC1=CCCC1 N1(CC(=O)NCC(CN(C(CC(C)N(C)C)=O)C)C)CCCCCCC1=O CC1(C)CC(C(N2CCC3CCCC23)=O)CN(C(=O)CC2CCCC2)C1 C1(CCCC)CCCCN1C(=O)C(=O)NC(n1nc(C)cc1C)c1ccccc1 CCC(C)(CNC(=O)CC1CC1(Cl)Cl)NC(=O)Cc1c[nH]nc1C S(=O)(=O)(c1ccc(NCC(Br)=C(C)C)c(Br)c1)NCC(CO)OCC N1(C(Cc2c(C)nn(C)c2C)=O)CCCC2(CCN(C(C3CCSC3)=O)CC2)C1 C=CCCCCCCCCC(=O)NC1(C2CCN(C(C3CCCCC3)=O)C2)CC1 C(=O)(C(C)(C)C(C)NC(=O)Cc1ccccc1O)NCCOCC(=C)C C(=O)(CCC(C)(C)C)N1CCC(COC)(CNC(=O)C(C)C(C)(C)C)C1 C(C1CCc2nccn21)NC(c1ccccc1-c1nc(=O)o[nH]1)=O C(C)(CN=c1nc(O)c(Br)c[nH]1)N(C(Cn1c(C)c(Cl)cn1)=O)C C1(CC)C(=O)N(C)CCN1C(=O)CC1(NC(=O)Cc2cocn2)CC1 c1(-c2cn(C3CN(C(C4CC4[N+](=O)[O-])=O)C3)nn2)cc(F)cc([N+](=O)[O-])c1 C(=O)(C(C)P(C)(C)=O)NC1CC(F)(CNC(c2c(C)nccc2)=O)C1 C12(C(N(CC)CC3CCNC3)=O)CC1CN(C(c1cccc(F)c1)=O)C2 CC(C)CCC(N)C(=O)N1CCN(c2ccsc2C#N)CC1 C(C(C)(CC(C)C)NC(=O)CCC(N)=O)NC(CCOCC(C)C)=O N1(CC(=O)NC(C2CCN(C(C(C(C)C)O)=O)C2)C)CCCCS1(=O)=O c1(-n2c(C(CCC)NC(CSCCCC)C(=O)O)nnn2)ccc(OC)cc1 c1(CC(=O)NC2CCC(NC(C(c3ccc(C)o3)C)=O)C2)ccccc1F C1(OC)CC(O)C(N=c2cc(Sc3ccccc3)n3ncc(I)c3[nH]2)C1 CC1(C)NC(=O)CC1C(N1CC=CC(NC(=O)CC2CCCS2(=O)=O)C1)=O c1(N2CCC(CCCO)C2)nc2c(c(=NCC3CCCO3)[nH]1)CCCC2 C(c1cnc(O)nc1O)=CC=O.CC(C)CO.CS(=O)(=O)CC1(CC=O)CC1 N1(C(C=CC=CCC)=O)CCC(O)(CCNC(C2(CO)CCCCO2)=O)C1 Cc1ccc2oc(C(=O)NC3CN(C(=O)Cc4cccc(O)c4)CC3C)cc2n1 c1cc2ccc(-c3noc(CC45CC(C4)C5)n3)nc2[nH]1 C1(N=[N+]=[N-])(C(=O)NC2(C)CC(=C)C2)CCN(C(c2ccc(C#N)cc2C)=O)C1 C(=O)(CC(C)C(F)(F)F)NC(CC(=O)NCc1c(C)cco1)CC1CC1 Cc1ccc(-n2nc(CS(C)(=O)=O)nc2C23CC(C)(C2)OC3C)cc1C C12(CNC(CSC)=O)CCC(CNC(c3cn4ccnc4s3)=O)(CC1)CO2 N1(C(CNC(=O)NC)=O)C2CCC1C(F)C(NC(=O)CC)C2.C(C)=O.S CC(C)C(C(=O)N(C)CC1CN(C(=O)CC2CC2(Cl)Cl)C1)N(C)C C(=O)(C(C#N)C(C)(C)C)N(C(C)C)CC.c1(C=O)csc(C(F)(F)F)c1 C(CCC(=O)N(C(C)C(=O)NC)C)(C(C)C)NC(COCC)=O c1(NC(C(N)Cc2ccc3ccccc3c2)=O)nccc2c(F)cccc12 Cc1nc2cc(C(N3CCC(NC(C45CCC(C4)OC5C)=O)C3)=O)c(F)cc2[nH]1 C(C(C)(C)CC(=O)NCC(C1CCCCC1)NC(=O)CC=C(Cl)Cl)OC(C)=O c1(C2N(CC3CC(C(=O)O)(C(=O)O)C3)CCC2)ccc(I)cc1 c1(NC(C2CCCN(C(C(CC=C)(C)C)=O)C2)C)ncc2ccnc-2[nH]1 C12CCC1CCN2C(c1ccccc1)=O.C1(C(=O)N)CC(F)(F)C1.C1CC1.C c1(C(N2C(C)(C)C(CNC(=O)CC3CCCCO3)CC2)=O)cc2n(n1)CCOC2 N1(C(CN(C2CC2)CC)=O)CC2CCCCC2(CNC(=O)CCCCC(C)C)C1 Cc1cnc(C(=O)NC2CCCC2CNC(=O)C(C)O)nc1 N1(C(c2n[nH]cc2F)=O)CCn2nc(CNC(C3(C(F)(F)F)CC3)=O)cc2C1 CCCCC(O)C(=O)NC1CC(CNC(=O)Cn2cc(C)ccc2=O)C1 N1(C(c2cn(CCN(C)C)nc2)=O)CCN(C(=O)CC=C(Cl)Cl)C(CF)C1 CC1(C)CC(C(N2CCCC(Cn3cc(C(O)C(C)(C)C)nn3)C2)=O)C(C)(C)O1 C1(NC(CC(CCC)(C)O)=O)CN(C(c2cc(C(F)F)no2)=O)C2(CCCC2)C1 C(CCCCCN=[N+]=[N-])NC(C1N(C(c2cccc(Cl)c2)=O)CCC(C)C1)=O C1(C(N2C(C(=O)NCc3c(C)n[nH]c3C)CC2)=O)CCCCC(=O)C1 c1(C(N2CCC2)=O)ccc(Br)c(F)c1.CC(C)(C)C(=O)NCCCC(=O)NC c1(CC(=O)OCC)csc(NC(=O)CC2(O)CNC2)n1.c1ccsc1Br.C Cc1cc(C)c([N+](=O)[O-])c(C)c1C(=O)N.C(=O)CC(C)(C)N(C)C.C1CC1 [SH](=O)(=O)c1ccc(C=O)cc1.C1(C=O)CC2CC1C2.CC=O.CC=CC.N C(=O)(C(C(=O)N)OC)OC.CC(C)S(N)(=O)=O.c1csc(C=O)c1.C1CC1 Cc1cc(C(C)(C)C(=O)N)cs1.C1(F)CN(C(=O)CC2CC3(CC3)C2)C1.C c1(C(N2C(CNC(c3nc(C)c(C)s3)=O)CC2)=O)ccc(N=S(C)(C)=O)cc1 C(=O)(CCC1CC1)OC.C1(C=O)CC(C)N1C(C1(C(C)=O)CC1)=O.N C1(NC(c2scc(C)c2)=O)CC(NC(c2ccc(O)c(Cl)n2)=O)C12CCC2 c1(C(=O)NC2CC(CNC(c3ccc4[nH]ccc4c3)=O)C2)cnc2sccc2c1 C1(NC(C2(O)C(C)(C)C2)=O)CCCN(Cc2cc(C3CCCC3)no2)C1 CN1CC(C)(C(=O)NC2CCN(C(=O)Cc3nc(=N)[nH][nH]3)C2)CC1=O N1(C(COC(CNC(c2c(C)cc(C)o2)=O)(C)C)=O)CC2CC(C1)C2(C)C C1(C(C)C)N(C(=O)C(C)c2cccs2)CC12CCN(C(=O)C(O)C(C)(C)C)CC2 C(c1c(F)cccc1F)=CC(=O)NCC1(O)CN(C(c2cncnc2)=O)C1 C1(C(=O)N(C)Cc2cc(C)on2)(NC(COCCCC)=O)CCCC1C CCC(C(=O)NC1CC(CNC(C2CC2c2ccccc2F)=O)C1)C(C)O N1(C(c2cccc(C)c2N)=O)CCN(C(c2cc([N+](=O)[O-])nn2C)=O)CC(C)C1 c1(C=O)ccc([N+](=O)[O-])[nH]1.C(C)(CC1CCC1)(C(=O)NC1CCC1)OC.C C1(C)(CNC(C2(CCCC)CC2)=O)CCN(C(=O)C(C)(C)N(C)C)CC1 C(=O)(CC(O)CN(C)C)N1CC(CC)C1.c1(NC(C)=O)ccc(C(=O)N)o1 C(C)(C)(CCC(=O)NCCCC(C)(C)NC(C1C2CC3C(C2)C13)=O)N(C)C C(=O)(CCCCC(C)(C)C)N(C(CNC(c1c(C)nc(C(C)(F)F)cc1)=O)C)C CC1(C)CCC(CNC(C2CCC(C)CC2)=O)(NC(c2cnc(O)s2)=O)CC1 N1(C(CCC#C)=O)CCC2(CCCN2C(=O)C=CC(C)(C)SC)C1 c1(NC(c2c(C)nc(CC3CCNC3)s2)=O)ccc2[nH]c(=O)cc(C)c2c1 Cn1cc(C(=O)NCCNC(c2cncc(N)c2)=O)nc1O N1(C(CC2(OCC)CCC2)=O)CC2C(CC(=O)NCC(C)(C)C(C)O)C2C1 c1(CNc2nc(C)[nH]n2)ccc(C)nc1-c1ccn(CC(=O)O)c1 c1(C(N2C(C)CC(NC(c3nnc(C)s3)=O)C2)=O)cc2c(cn1)OCCO2 CC(CNC(c1ccc(F)cc1F)=O)C(F)C(=O)Nc1cccc(C(N)=O)c1 c1(C(N2CC(C(N)=O)(CNC(COC)=O)C2)=O)ccc2ncccc2c1Cl O=[N+]([O-])c1ccc(-c2ccc(CNC3(C(F)(F)F)CC(F)(F)C3)o2)c(F)c1 c1(SC)ccc(-c2nc(-c3ccc(C)cc3)nn2CC(C)(C)C)cn1 c1(CN2CCC(N(c3ncncc3Br)C)C2)cc2cccnc2[nH]1 C(C)(C)(CC(=O)N1CCC1CC(=O)NC)NC(CCNC(CCC)=O)=O CCC(C(C)(C)O)NC(C1OCCC1CNC(=O)CC1CCSC1)=O c1(CC)ccc(N)c(C(N2CCC(CN(C)C(c3csc(C)c3C)=O)CC2)=O)c1 c1(OC)ccn2ncc(C(=O)NC3CC34CCN(C(C3C(C)C3C)=O)CC4)c2c1 c1(C(=O)NC2C(F)(F)CCN(C(CCC(N)=O)=O)C2)ccc2cc[nH]c2c1Br c1(OC)ccc(NC(c2ccccc2NC(=O)CC(C)N)=O)cc1-c1ncon1 C1(C(N2CCCC(=C)C2)=O)CC2CC1CC2NC(C1CCC(C)(C)C1)=O N(C1CCc2ccccc21)C(C1CC2(CC2)CN1C(=O)Cc1cnsc1)=O C1(NC(c2nc(CCCC)sc2)=O)CC(=O)N(C2CN(C(c3ccco3)=O)C2)C1 c1(C(C(=O)NC2(CNC(CCOCC(C)C)=O)CC2)=O)ccc(Cl)cc1 C12CC1CN(C(C1CCCN1S(=O)(=O)CC)=O)C2.C(CC(=O)N)OCC.C C1(NC(c2csc(C(F)F)n2)=O)C=CCN(C(c2c[nH]c(-c3cccs3)n2)=O)C1 c1(CN2C(C(=O)NCc3c(C)c(F)ccc3)CSCC2)cc(Br)c(F)cc1O N1(C(CN(C(C)C)C)=O)CC(N(C(=O)Cc2ncnn2C)C)C(C)(C)C1 C1(NC(CCC=C)=O)CCC12CN(C(=O)CCc1ccc(C)cc1C)C2 N1(CCOC)CCC(NC(c2ccc(Nc3ccccc3OC)s2)=O)CC1 c1(C(=O)NCCCCC2CN(C(c3c(C)nsc3)=O)C2)scc(Cl)c1Cl c1(N(C)Cc2csnn2)nc2c(c(=NC3CCS(=O)(=O)C(C)C3)[nH]1)SCC2 CC1(C)COC(CC(N2CC=CC(NC(=O)CC3=CCCC3)C2)=O)CO1 N1(C(=O)Nc2c(C)nn(Cc3ccc(Cl)cc3)c2C)CCc2c(nnn2C)C1 N1(Cc2c(C)nccc2)CCc2cc(C(=O)N(CCO)CCO)ccc2C1 Cc1cc(C)c(C#N)c(N2CC=CC(NC(C3(CO)CCOCC3)=O)C2)n1 N1(C(C2CC3(CN(C(COC(C)=O)=O)C3)OC2)=O)CC2(COC(=O)N2C)C1 CC1=C(C(=O)N(C2CC2)CC2CCN(C(C3(C#N)CCCC3)=O)CC2)CCCC1 CC(C)(C)C(O)CC(=O)NCC(C)(CO)NC(c1cnc(-c2ccncc2)s1)=O c1(CC(c2ccncc2F)N(C)Cc2nc(CC)on2)cccc(Br)c1 O=C1CCC(CC(=O)NOCC(=O)Nc2ccnn2CCF)N1 Cc1nc(NC(=O)NCCn2ccc(Br)n2)sc1C(=O)O c1(OC)ccc2c(c1)CCCC2CNC(=O)CNc1ccccc1C(C)(C)C C1(NCc2ncc(C)s2)COC2(CCN(C(=O)CSC(C)C)CC2)C1 c1(SC(C)C)ccccc1CC(=O)NC1CC1.c1(C=O)cc(C(F)F)on1.C c1(C2(C(=O)NC(CNC(C(F)=CCC)=O)C)CCC2)ccc(C(C)C)cc1 CCC(C)CC(=O)C(=O)N1CC(O)CC1CNC(=O)CC1CCOC1 C(=O)(C(C)(C)CC(=O)N1CCC(C)C1C(N1CCC(C(N)=O)CC1)=O)OC C1(C(N2C(C=C)CC2)=O)(NC(=O)C(C)NC(=O)C2CC2)CCN(C)C1 N1(CC2CCN(C(C)=O)CC2)CCN(c2ncc(C(F)F)cn2)CC1 c1(NC(C=CC(C)(C)NC(=O)CC2CSCCO2)=O)ccc2nncn2c1 C(CC(C)C)(C(=O)NCCCN(C)C(C1CCOC(C)(C)C1)=O)OC CC1CC(CNC(C23CCC(C2)OC3)=O)CN1C(=O)COC1CCOCC1 C1(C(=O)NCc2cccnc2F)(COC)CCN(C(=O)CCCC(=O)OC)CC1 c1(CN2C(C(N3CC4CCN(C)CC4C3)=O)CC2)ccc(S(C)(=O)=O)cc1F C1(NC(c2cc(C)sc2C)=O)CC2CCC1C(NC(=O)CCC1CC1)C2 C(CCN(C)C(c1sc(C)cc1Cl)=O)(C(C)C)NC(C(C)(C)OC)=O Cc1cnn(CC(=O)OC(C)(C)C)c(=O)c1C(=O)NC1CCC1O C12(NC(C3CCC(CC)C3)=O)COC(C)(C1)C2.c1(C=O)ccnc(S)c1.N c1(C(=O)N)ccccc1CS(C)(=O)=O.Cc1cc(CCC(=O)NC2CCC2)no1 c1(C(C(=O)NCC)N(C)Cc2cc[nH]n2)cc(-c2ccccc2)cs1 C1(NC(C2(C)C(C)C2)=O)CN(C(=O)Cc2ccc(OC(F)F)cc2)CC2(CC2)C1 N1(C(C=C=C(C)C)=O)CCC(N=[N+]=[N-])(C(=O)NCC2CC3C=CC2CC3)C1 N1(C(CC(CC)OC)=O)CCN(C(c2ccc(CO)cc2F)=O)C(C)C1 CCC(C)(C)CCCC(=O)N1CCOC(C)C1C(=O)NCCCC(C)(C)CO n1(Cc2n(C)ncc2)ncc(C(=O)NC2CCN(C(=O)C(C)(C)O)C2)c1Cl C(CC(C)C)(C(=O)N1CCC(NC(=O)C(C)S(C)(=O)=O)C(F)C1)OC C1(C2CCOCC2)(CNC(CCC=CC)=O)CCN(C(=O)C=C(C)Cl)C1 C12(CNC(C3CC3c3ccsc3)=O)CC(CN1CC(O)C)C2.c1ccco1 C12(CNC(c3c(C#N)cccc3)=O)CNCCN1CCOC2 C1(C(N2CCCC(CCC)C2)=O)C2CCN(C(=O)CC3CC(=O)C3)CC12 CCCC(C(=O)N1CCOCC1CNC(=O)CN1CCc2sccc2C1)C(C)C C1(NC(c2c(C)onc2C2CC2)=O)CC2CCC1C2.C(=O)C(C(C)C)NC=O.N N1(C(c2ccc(C)cc2F)=O)CCN(C(=O)C(C2CCCC2)N(C)C)CCC1C C1(C=O)COCCN1CC(F)F.n1(C(C)C(=O)NCC)ccc(C(F)(F)F)n1.N C1CCCCN(C(=O)CC2CCOC2=O)C1.C1(OCC)CC2(C1)CC2C(=O)N c1(C(=O)NCCCN(C)C(c2sccc2C2CC2)=O)cc(F)cc(F)c1N c1(C=O)cncc(C(F)(F)F)c1.CC1(CC(=O)NCCC2CCC2)CC1(F)Cl c1(NC(c2cccc(CC(=O)NC(C)C)c2)=O)cc(Br)c(Br)c(Br)c1 Cc1cc(N2CC(C(C)NC(c3cc(=O)n(C)cn3)=O)C2)n2nc(C)cc2n1 C(=O)(CCCCC(=O)NC(CCC1CCC1)C=O)OC.C1(C#N)CC(C)(C)C1.N N1(C(C)=O)CCN(C(=O)Cc2ccc(C(C)=O)c(N)n2)CC1C1CCCC1 O=C1CCC(Nc2ccc(CCC3CC3)cc2O)CCN1 CC(C)C(C)C(=O)NCC(C)NC(=O)CCc1cnn(-c2ccccc2)c1 CCC(CCCC(=O)NCc1c(C)cccc1F)NC(=O)C(C)c1ccsc1 C1(CC=C)(NC(=O)C=CCNC(=O)CCCOC(C)C)CCCC1 CC(C)C(C(=O)NC1(CC)CC1)n1cnnn1.C1(C)(CC(=O)N)CC1(F)F N1(C(c2c(C#C)cn(C)n2)=O)CCCC1C1CCCN1C(=O)C=C(C)Cl N1(C(C=Cc2n(C)cnc2)=O)CCC(C)(C)C1C(=O)NCc1cc[nH]n1 Cc1cnc(C(=O)NCC2(C)CC2)c(F)c1.C1(c2ccccc2)(C=O)CCC1 N1(C=O)CCn2c(cnc2C)C1.C1(N(CCN(CCC)C=O)C)CCN(C)C1.N C1(C(C)NC(C(C)C2CCC2)=O)CCCN1C(=O)CC1(O)CCC1 C12(NC(c3c(Cl)cccc3[N+](=O)[O-])=O)CCN(C(c3ccc(Cl)o3)=O)CCC1C2 C1(C)(CC)C=C(C(=O)NCc2cccnc2C)C1.c1(C(=O)N)cccnc1 c1(OCC(=O)NC2(C3CN(C(=O)C(O)C(F)F)C3)CC2)cccc(F)c1F n1(CC#C)c(C(=O)NCCC(C)N(C(=O)C=COCC)C)cc2ccccc12 C(=O)(CCCCCNC(N)=O)N1CCC(C(C)C(=O)NCC(F)(F)CO)CC1 c1(-c2c(C)cc(F)cc2)cc(C(=O)NCCCN2CCCCC2)c2cc[nH]c2c1 c1(C(N2C3CC(NC(C4CCC5CC45)=O)C2CC3)=O)ccc2cc[nH]c2c1F N1(C(C=CC)=O)CC2CN(C(=O)CC3(c4ccccc4)CCCC3)C2C1 CN(C(=NCCC1CCCO1)NCc1ccoc1)Cc1cc(Cl)c(Cl)s1 C1(CNC(C(C)=C2CC2)=O)CN(C(c2ccco2)=O)CC12CCC2 C1(C(N(CCCCCC)CCNC(c2cn(C)nn2)=O)=O)CC1C1CCCCC1 n1(C(C)C)cc(C2CC2)nn1.C(=O)(CC)N(CCOC)CS(C)(=O)=O Cc1ccc(C(=O)NC2(CO)CN(C(C3CCCCC3(F)F)=O)C2)c(C)n1 N1(C(C2CCC(CNC(=O)CC34CCCN3CCC4)CC2)=O)CC2CC1CC2O N1(c2nc(N(CC(C3CC3)OC)C)nc(C)c2)CC2C=CCC(C2)C1 N1(C(C(C=C=C)C)=O)CCCCC(NC(c2cc(Br)c(F)cc2C)=O)CC1 N1(C(C)=O)Cc2ccccc2CC1CNC1(C2CCN(C(=O)C(N)=O)CC2)CC1 C1(C(N(C2CCCN(C(C3(C4CC4)CC3)=O)CC2)CC)=O)CCC(N=[N+]=[N-])CC1 C(C(C)(O)CC(=O)NC(CC1CCOCC1)C(=O)Nc1cccc(Cl)c1C)OC C=CC1CN(C(C23CC(F)(C2)C3)=O)CC1NC(c1cc(C)nnc1CC)=O N1(C(CCNC(C)=O)=O)CC2CC1C2NC(C1C2(CC2)C12CC2)=O CCCC(O)CC(=O)NC(C)C(CO)NC(=O)C(CC(C)C)c1ccccc1 c1(C(=O)NCC(C(=O)NC2C(OC)CCOC2)C)cc2cnccc2[nH]1 CC(C)CC(C)(O)c1cn(CC(C2CCN(C(C3CCOC3=O)=O)CC2)F)nn1 c1(C(=O)NC(CC(C)NC(c2cc(C)oc2)=O)C)ccc(C(C)C)cc1O c1(OC)ncc(C)cc1-c1ccc(NCc2cccc(CO)c2)cn1 N1(c2c(-c3ccc(COCC)s3)cc(C3CC3)cc2C)C2COCC1CC(F)C2 C1(CNC(CC2N(C)CC=CC2)=O)CN(C(=O)CCc2cncs2)CCN1C c1(C(N2C3C(NC(C(C)OCCC=C)=O)C(C3)C2)=O)ccc(C)c(C)c1O C1(C)(C(N(CC(CC)C)C)=O)CCCN1C(=O)CC1CCCOC1 C12(CNC(=O)COCCCF)CCCC1CCN2C(=O)C(=O)NC1CC1 C1(CC(=O)NCCC2CC2C2CC2)CCN(C(c2cnc(O)o2)=O)CC1 C(C(CC(F)(F)F)NC(=O)CCc1ccc(C(F)F)cc1)NC(C=CCC)=O Nc1cnc(C(N2CC3CC2CN3C(=O)Cc2cccnc2O)=O)c(Cl)c1 Cc1nn(C(C)C)c(C)c1C(=O)NC(C1CN(C(c2cc(C)on2)=O)C1)C C(=O)(C1=NN(C)C(=O)CC1)N1CC(C(=O)NCCC(C)SC)C(C)(C)C1 N1(C(CCCC(=O)NC(C)C)=O)CC(C)N(C(=O)CCCC2CC2)CC1C c1(C(=O)NC(CCNC(CC(CC)C)=O)C)ccc(OC(F)(F)F)cc1F Cc1c(F)cc(CNc2ccsc2C(=O)Nc2ccnc(C3CC3)n2)cc1F c1(C(C(=O)NCC(C2CCCC2)NC(COC)=O)C)ccc(F)cc1 C(CCC(=O)N1CCCC1C(C)(C)NC(C1COCCO1)=O)NC(=O)OC C(CC(C(C)(C)C)NC(=O)C(C(C)C)OC)NC(c1ccc(CC)nc1)=O C1(OC)CCC2(C(=O)NCCC3CC(NC(=O)CS(N)(=O)=O)C3)CCC12 c1(C(=O)NCCC(=O)NC)ncnc2c1ncn2C1CCS(=O)(=O)C1 N1(C(C(c2ccc(Cl)cc2F)OC)=O)CC2(CCOCC2)C1c1cnn(C)c1 c1(C(N2CCC(O)(CCNC(=O)CC3(CO)CC3)C2)=O)ccc2cc[nH]c2c1 C(C(COC)C(=O)N1CC(C)CC1C(=O)N(C(C)CC1CC1)C)OC c1(C(C(=O)NC2N(CC)CCC2)N(c2ccccc2C)C)cc(Cl)cc(C#N)c1 N1(C(CSC)=O)CCCC12CCN(C(C1CC13CCC1(CC1)CC3)=O)C2 C(=O)(C1CN(C(C2CNC(=O)N2C)=O)Cc2ccc(OC)cc21)OC c1(N2CC3N(C(c4c(C)cc(C)nc4Cl)=O)C3C2)[nH]cnc2nc(Br)cc1-2 c1(C(=O)N)cc2cc(Cl)sc2[nH]1.C1(NC(C(C2CC2)SC)=O)CC(C)CC1O c1(C(=O)NC2(CO)CCN(C(C(C)NC(CC)=O)=O)C2)ccc(F)c(SC)c1 C1(CCNC(CCc2n(C)cnc2)=O)CCCCN1C(C1CC1(C)C)=O N1(C(C(C)CN(C)C)=O)CC2CC(C1)C2NC(C1(F)CCCCC1)=O c1(CCC)csc(N(C)C)n1.c12cccn1NC2c1nnnn1-c1ccccc1 C#Cc1cccc(N(C)C(C2(C=O)COC2)=O)c1.C(=O)CCCC(=O)C(C)C.O C1(c2n(-c3c(CC)cccc3)nnn2)(NCC23CC(C2)C3)CCOCCC1C C1(C(N2CC(CNC(c3c(Br)cc(C)s3)=O)C2)=O)CCCCC1(C)C N1(CC2CCc3c(cn(C)n3)C2)CCOCC2(CCS(=O)(=O)CC2)C1 N1(C(CNC(C)=O)=O)CCCC2C1CCCN2C(=O)C=C1CCCC1 c1(CN(CC(=O)N(C(CN(C(C=CC(C)C)=O)C)C)C)C)ccc(Cl)s1 N1(C(c2cccc(N)c2)=O)CC2CCC(C1)N2C(=O)C(F)=C1CCC1 C1(NC(CC2C(CC)C2)=O)CC(C)CN(C(=O)CC(C)C(=O)c2ccccc2)C1 c1(OC)ncc(Cl)c(=NC2CN(C(=O)CCCCCSC)CCC2C(F)(F)F)[nH]1 C1(CN(C)C(C2(F)CN(C(=O)Cc3ccns3)C2)=O)CCOCC1 N1(C(CC(c2ccccc2)CC)=O)CC2CCC1CN2C(CC)C(=O)OC C=CCC(C)(CC)C(=O)N(CC(=O)NCC1(O)CCCOC1)C1CCC1 N1(C(CN(C)C(N)=O)=O)CCOCC1CC(=O)NC1(C)CCCC1 c1(CC)nc(C)c(C(=O)NC(Cc2ccccc2)C(=O)NC(C)(C)C)s1 c1(C(=O)OC)nc2c(s1)N(C(=O)Nc1cccc(-n3cnnc3)c1)CCCC2 Cc1cc(C(N2CCC(C)(N3CCOCC3)C2)C(=O)NC2CC2)cnc1C1CC1 C(c1ccc(C)cc1)=CC=O.C(C(=O)N)(C1CCC1)OC.C(C)(C)C.CC c1(C(C(N2CC(N(C(c3cnc(COC)s3)=O)C)C2)=O)C)ccc(F)cc1 c1(CC)cc(C(N2CCCC(C)(NC(c3nccnc3N)=O)C2)=O)cc(Cl)n1 n1(CC(=O)NCCCC(C)NC(C(C(CC)C)O)=O)nnc2ccccc12 CC(C)CCCCCC(=O)N1CC(CN(C)C(c2cnccc2C(C)=O)=O)C1 C(=O)(CS(=O)(=O)C1CC1)NC(CNC(CCN(C(CCC)C)C)=O)(C)C C1(C(N(CCNC(c2ccc(Br)o2)=O)CC)=O)CCC12CCOCC2 CC(C)(C)C(O)C(=O)Nc1ccc(NC(c2ccc(CO)cc2)=O)cc1F CC(C)(C)C(CC(F)(F)F)C(=O)Nc1ccccc1NC1COc2ccccc2C1 CN1CCN(C(C2CC2[N+](=O)[O-])=O)CC1CNC(=O)CN=S(C)(C)=O N1(C(c2cc(SC)nn2C)=O)CCN(C(=O)Cc2cc(Br)cs2)C(C)C1 c1(CN2C(CC=CCCC(C(=O)O)OC)CCC2)ccc2ccccc2n1 C1(C2CCN(C(=O)CS)CC2)(NC(c2cccc(OC)n2)=O)CC1.CCC(C)C c1(C(=O)O)ccc2[nH]cc(C(=O)NC3CCC4(C3)CC4(F)F)c2c1 C1(C(N(C2CCN(CC)CC2)C)=O)CC(NC(c2snnc2C)=O)C12CCC2 C=CCC(C(=O)NC(C1CCCN1C(c1cnsc1C)=O)C)NC(C)=O C1(NC(c2snc(Cl)c2Cl)=O)CN(C(C2(O)CCCCCC2)=O)CC12CC2 N1(C(c2[nH]nc(OC)c2Cl)=O)CCC=C(CNC(=O)Cn2nc(C)nc2C)C1 C1(CNC2(C)CC(F)C2)CCC(=O)N(CC(F)(F)F)C1 c1ccc(CC(N2CCCC2)=O)cc1.C1(C(C)C)(C=O)CC1.C(C)=O.CS.C c1(C(=O)Nc2ccc(-c3cc(C)[nH]n3)cn2)ccc2c(c1)C(=O)NC2 C1(CNC(c2scc(C)c2)=O)CCCC(NC(c2cncc(C(N)=O)c2)=O)C1 C1(NC(CC(CC)(C)C)=O)CN(C(=O)CC23CCCN2CCC3)C2(CCOC2)C1 c1(C(N2C(CNC(c3ccc(OC)cn3)=O)CC2)=O)nccn2c(Br)cnc12 c1(C(=O)NC(CNC(c2c(CC)cco2)=O)CC)ccc2oc(=O)oc2c1 c1(C(=O)NCC2(F)CC(NC(CN(C)C)=O)C2)cccc2nccnc12 c1(NC(C2C=CCN2C(C2(F)CC2)=O)=O)ccc(Cl)nc1 C=CCCC(F)(F)C(=O)N1CC2CCCC2(NC(C2CCCC2(C)C)=O)C1 N1(C(C(C(C)C)OCC)=O)CCC2CCC(NC(c3cn(C)nc3C)=O)C1C2 Cc1c(C(N2CCCCC2CNC(C2CCC(C)C2)=O)=O)cccc1F N1(C(CN(C(=O)C(C)=CC(C)(C)C)CCC)=O)CCC(C)(C#N)C1 C(c1ccncc1)=C(C)C(=O)N(C)CCNC(=O)Cc1sccc1Br N1(C(c2ncsc2)=O)CCN(C(C2(C(C)(C)O)CCC2)=O)CC1CC(F)F.CC C1CN(C(c2cc(C(C)(C)C)on2)=O)CC2(CC2)C1.CC1CC(C)OC1C=O.N C(c1cccc(O)c1)=CC(=O)NC(CC(C)NC(C(CC)COC)=O)C c1(-c2nc(OCC)nc(SC3CCCC3)c2)cc(C)c(N)c(C)c1 c1(CC)ccc([N+](=O)[O-])cc1C(=O)N.C1CN(C(c2cnsc2)=O)CC2(CC2)C1 C1(C(N(C(C)CN(C)C)C)=O)COCCN1C(C1CCCC(=O)N1)=O C1(C(N(C2CCC2)C)=O)CCN(C(=O)C2CC3COCC3C2)O1 N1(C(c2ccc(Nc3ccc(C#N)cn3)cc2)C)CCCN(C)CC1 CCCCCCCC(F)C(=O)NC1CN(C(=O)C=Cc2cocn2)CC1CCC C1(NC(CCOCCN(C)C(c2cc3cccnn3c2)=O)=O)CCN(C)CC1C#N c1(C(=O)NCC2CC(NC(CCCC)=O)C2(C)C)ccc2nn[nH]c2c1O C#Cc1cccc(C(N2CC=CC(NC(c3cnc(O)c(OC)c3)=O)C2)=O)c1F c1(-c2c(CC)cccc2)cc(C(=O)Nc2ccc(C#N)c(O)c2)cc2[nH]ncc12 N1(C(C2N(C(c3c(C)nc(O)s3)=O)CC(O)C2)=O)CCn2ccnc21 C(=O)(C(CC=CCc1nocc1CC)NC(=O)CCCC1CC1C)OCC C1(NC(c2c(C)nn(-c3ccc(F)cc3)c2)=O)CCCCN(C(=O)C(C)C#N)C1 CC1CC2(CC(C(=O)NCCNC(C3CN(C(N)=O)CCO3)=O)C2)C1 C1(n2cc(CCC(C)=O)nn2)(NC(c2ccncc2Cl)=O)CCOCC1 c1(C(=O)NC2CCN(C(C(C)CC(C)(F)F)=O)CC2O)cnn2c(=O)cc[nH]c12 C1(CCCNC(C=NOC)=O)CN(C(c2ccc(Cl)o2)=O)CCO1 c1(CC(=O)NC2C(NC(C(C)CN(C)C)=O)CCC2)c[nH]c2cnccc12 c1(OC)cccc(Cl)c1C(N1CCC(NC(=O)C(F)CC2CC2)C(O)C1)=O c1(NC(C(CC2CCC2)NC(C(C)NC(CC)(C)C)=O)=O)ccccc1C.C Cc1ccc([N+](=O)[O-])c(N(C(=O)CCCOC(C)C)CC2CCN(C)C2)c1 C(=O)(CS(=O)(=O)C1CC1)N1CCCC(OC)C1.c1(C(=O)N)ncoc1C1CC1 Cc1c(C(N2CC(CCNC(c3cc(C4CC4)ns3)=O)C2)=O)ccn1CCO N1(C(c2cnc(C)nc2)C)CCOCC(C(=O)NCC2CCCC2)C1 CCCC(CCC)C(=O)NCC1CCN1C(=O)Cc1ccsc1Cl S(=O)(=O)(c1cc(C(F)(F)F)cc(F)c1)NC(C1CC1N1CCOCC1)=O C=CC(C)(C)CC(=O)NC1CCC1NC(=O)C(c1c(C)cccc1C)O N1(C(CCN(CCCCC)C)=O)CC2CC(C1)N2C(C1CCCCN1C)=O C1(C(N(CCC(C)NC(=O)CN2CCCC2)C)=O)C2CCC1(c1cscn1)C2 C1(CNC(C(C2CCCC2)OCC)=O)CCCC1.n1(CC=O)cncc1C.N c1(C(=O)NC(C2OCCN(C(C3(SC)CCC3)=O)C2)C)c(Cl)nn(C)c1C Cc1noc(C)c1CNC(Cc1cccc(C(F)(F)F)c1)C1CC1 C(=O)(CCC(C)(C)F)NC(C1CCN(C(c2nccc(C)n2)=O)CC1)C CCCCC(C(C)O)NC(C)Cc1ccc(C(=O)OC)cc1 N12CCC(F)(C1)C2=O.N1(CC(=O)NCCn2ccnn2)CC(CF)C1 Cc1nc(C)c(C(C)NC(C2CCN(C(c3[nH]cc(C)c3C)=O)C2)=O)s1 c1(C(=O)NCC23C(CN(C(Cc4ccc(C)o4)=O)C2)C3)cc2sccc2[nH]1 N1(C(c2nc(CC)sc2N)=O)CCC(C)C(C)C1.c1(C=O)cc(C(F)F)cs1 c1(C(N(CCCCN(C(C(CC)C(C)O)=O)C)C)=O)c[nH]c2ncccc12 C(CCC(=O)NN1CCCC1C(N1CC=CC(OC)C1)=O)OCC Cc1ccc(S(N)(=O)=O)cc1C(=O)NC(C)CCN(C(=O)C=CBr)C c1(C=O)ccnc(C2CC2)n1.C(CO)(C(=O)NC(C)Cc1ccccc1)OC.N c1(C(N2CC(C)C(O)C2)=O)cc2c(nn1)OCCS2.C1(C2CC2)(C(=O)N)CC1 Cc1nc2c(o1)CCCC2CC(=O)N1CC2CCC(C1)N2C(c1cc(F)c[nH]1)=O C1(CCC)CN(C(C2(C(C)(F)F)CC2)=O)CCN1C(=O)CC12CC(C1)C2 C(=O)(C1CCc2nccn21)NC(C(CC)C)C(N1CC=CC12CCCC2)=O CCC(C)(CO)CN=c1cc(NCCC(C)P(C)(C)=O)nc(C)[nH]1 CC(C)(CCCN=c1nc(Cl)nc(CC2CC2)[nH]1)NC(=O)CC1CCC2CC2C1 c1(OC)ccccc1C(CCO)NC(c1nnc(C(F)(F)F)s1)=O C1(C(N2CC(OC)C(OC)C2)=O)(CC)CCCN(C(=O)CCCCCC)C1 C(CC(C)C(=O)NCC(C1CC1)NC(=O)CCc1ccon1)=CCC CCC(C)C(C(=O)NCC1(NC(c2cnc(C)[nH]c2=N)=O)CC1)OC c1(C(C(=O)NC(CC(C)NC(C2CC23CC3)=O)C)O)cccc(C(F)(F)F)c1 C1(C)(C(N2CCC(C)(NC(=O)C3=CCC3)CC2)=O)Cc2c(Cl)cccc2C(=O)O1 c1(N2C(CN(C(C3C(C)(CC)C3)=O)C)COCC2)nc(Cl)nc(C)c1Cl c1(C(=O)NCCC)ccc(C(C)(C)C(N)=O)cc1.C1(C)(C=O)CCNC1=O.N C(=O)C(C)(O)C(F)(F)F.[SH](=O)(=O)c1ccccc1.CC(CCO)NC(=O)C.N C1(CNC(C=Cc2n(CC)ncc2)=O)CC(C)(C)CN1C(c1cccs1)=O CN1CCC(C(=O)NCc2ccoc2C(=O)N(C2CC3(CC3)C2)C)CC1=O c1(C(=O)NC2CN(C(c3cccc(C)c3C)=O)CC(O)C2)cc(F)cc(C)c1C N1(C(C2=C(C)OCC2)=O)CCOC2(CCCN(C(=O)CCCCC(C)(C)C)C2)C1 C(C(=O)N1CC(O)C(O)CO1)N(C(c1cncc(OC)n1)=O)CCO CON(CCCO)C(=O)COC1CCN(C(=O)C(C)C(O)C(C)C)CC1 C(=O)(C(O)C(C)(C)C)NC(CCC)C(=O)N(c1cnn(CC)c1)C c1(C(N2CC(F)(CNC(CN3C(C)CCC3C)=O)C2)=O)cc(N)c(F)cc1F C1(NC(c2c(OC)nccc2)=O)CCOC2(CCN(C(c3ccc[nH]3)=O)CC2)C1 N1(C(CCc2cc(C)[nH]n2)=O)CCC(NC(=O)C(=O)NCCC(N)=O)C(CO)C1 CC(C)CCCCC(=O)NCC(C1CCN(C(=O)COCCN(C)C)CC1)(C)C CCC(C)CCCCC(=O)N1CC2CCC1CC2NC(C1(C)CC=CC1)=O c1(C(=O)OCC23CCC(CC2)O3)nccc2ccsc12.N12CCC(CC1)NCC2 CC1(C)CN(C(=O)CC2(O)CCOC2)CCC1NC(C1CCC(=O)N1)=O N1(C(C2(c3cc(C)no3)CC2)=O)CC2CC(NC(=O)C(C)CC(C)C)CC2C1 n1(C(C)C)nc(C2CC2)cc1CNC(=O)C(F)(F)CC1CCCO1 c1(OC)cccc(C2CCN(C(=O)C=Cc3ccc(NC(C)=O)cc3)CC2)c1F C1(CNC(C(C)N(C(=O)C(C)CN(C)C)CC)=O)OCC2CCCC12 C1(C2CCCCC2)(C(N(C)CC2(O)CCCCC2)=O)CCNC1 c1(CNC2CCC(C(=O)Nc3n(C)nc(Br)c3)OC2)c[nH]c2cc(F)ccc12 Nc1cc(F)cc(Cl)c1C(=O)NCC=CCNC(c1cccnc1)=O C=C(Cl)CCC(=O)N(CC)CC1CCCN1C(C1CCN1CC)=O C1(C(NCC(C)(C)C)=O)CN(C)CCN(C)C1.C(=O)C(C)(O)C1CCC1.CC C1(C(N2C(C)(CNC(c3c(CC)cncc3)=O)CCC2)=O)CCc2ncnn2C1 c1(CNC(C2(OC)CC2)=O)csc(C)n1.C1(=CC(=O)N)CCOCC1 c1(CC(=O)NC)cccc(F)c1F.C1CCCN1C(c1cc(C(F)(F)F)on1)=O n1(CC)cc(C(=O)NCC2(C(F)(F)F)CCC2)c(C2CCOC2)n1 C(=O)(C(CC)CC(C)C)N1CCC(C(=O)NC(CC=C)C2CC2)CC1C C(C1=NOC2CN(C(=O)Cc3ccn(CC)n3)CC12)NC(c1c(CC)nn[nH]1)=O CC1(C)CC(CC(=O)N)N(C(=O)CC(C)(C)C2CC2)C1.C12CC(C)(CCO1)C2 c1(OC)ccc(C(=O)NCCC(C)N(C(=O)C=C2CCC(C)C2)C)c(Cl)n1 c1(CNC(=O)NC(CC(=O)N(C)C)Cc2ccccc2)cc(C#N)ccn1 C(N=c1ccn(C)[nH]1)(c1c(CC)con1)c1nnnn1COC C12(NC(=O)C3=CCCOC3)CCCC1CN(C(c1cc(C(F)F)cnc1O)=O)C2 CC(C)CS(=O)(=O)N1CCC(Cn2ccnn2)C1 C1(OC(C)C(=O)NCC2CCN(C(=O)C=Cc3cn[nH]c3)CC2)CCCCCC1 CC1=NOC(=O)C1CCC(=O)NC1CCCN(C(c2c(Cl)nsc2Cl)=O)C1 c1(CC(C(=O)NC2COCC2C)O)c(F)cccc1Cl.C(=O)C1=NNC(=O)C1.N N1(C(c2ncc(C)cn2)=O)CC(C)(C)CC1C.C1(C(C)(C)C)(C=O)CCC1.N Cc1cc(C)cc(CNNC(=O)c2cnc(F)cc2C)c1 C1(OC)CCCN(C(=O)CCC2(NC(=O)CCCC#N)CCC2)C1C N1(C(c2nc(C)sc2C)=O)CCCC2(NC(c3ncccc3Cl)=O)CCCC12 CC1CC(C(=O)NC2CCN(C(c3c[nH]ccc3=O)=O)CC2)CCS1 N1(C(C(C)(C)C2CCOC2)=O)CCCC(CCNC(=O)CN2CC=CC2)C1 N#Cc1cc(Cl)c(C(N2CCCOC(CCNC(C3(C4CC4)CCC3)=O)C2)=O)s1 c1(C(N2CC(CNC(COCCOC)=O)C(C)C2)=O)c[nH]c2nc(Cl)ccc12 c1(NC(=O)NC(CNS(CC)(=O)=O)C)cccc(NC(C)=O)c1 C1(NC(C(C)C2(O)CCC2)=O)CCCC12CN(C(c1nccnc1N)=O)C2 c1(C(N2CCN(CCN(C(=O)C(O)P(C)(C)=O)C)CC2)=O)cnc2sccn12 c1(CC)ccnc(C(=O)NCC=CC(=O)NCCC2(C)CCOCC2)c1 CCCCCCCCCC(O)C(=O)N1CC2CCCCC2(CNC(=O)C2CC2)C1 CC(C)CC(C(=O)NCCCc1ncn(C)n1)NC(=O)CN1CC2CCC1C2 C1(C)(CNC(C2(NC(C)=O)CCC2)=O)CN(C(=O)CC(F)(F)Cl)CC1C CN1CC=C(CC(=O)NC(CNC(c2cc3c(s2)CCSC3)=O)C2CC2)CC1 N1(C(c2c(CC)cns2)=O)CCC=C(C(=O)NC(CSC)CC)C1 C12CC3CCC1N3C2=O.Cc1ccc(CC(=O)Nc2nccnc2N(C)C)cn1 n1(CC(=O)NCC(CNC(C(C)(C)N2CCCC2)=O)F)cc(Br)ccc1=O C1(n2cc(CN(CC)CC)nn2)CN(C(c2sc(Br)nc2C)=O)CC1(C)C C1(NC(C=COCC)=O)CCN(C(=O)CSC)C(C)C1.c1(CC)ccccc1 N1(C(c2cnc(C(C)C)[nH]2)=O)CC(NC(C2CCC(C)O2)=O)CC1CO N1(C(c2c(C)cn(C)c2)=O)CC2(CC2)CC1CNC(=O)CC1(C)CCCC1 N1(C(Cc2ccc(C(C)=O)s2)=O)CC(NC(=O)C(F)C(C)C)C(C)C1 C1(OC)CN(C(c2cnn(CC(F)F)n2)=O)CC1NC(c1snnc1C)=O c1(OC)ccc(C(CNC(=O)CCc2cccnc2)NC(C2CC2F)=O)cc1 C12(C(N3CCN(C(CC=C)=O)C(C)C3)=O)C3C4C5C3C1C5C24 CCCC(C)CC(=O)N1CC(C)(C)CC1CNC(=O)CCCSC C1(n2cc(C=CC(=O)OCC)nn2)CCN(C(C2CCCC(O)C2)=O)CC1 C(C(=O)NCC1(C)CCN(C(c2cccc(Cl)c2F)=O)CC1)(C(C)(C)C)N(C)C N1(C(C(C(CC)C)O)=O)CC(CO)C2(CCN(C(c3occ(C)c3C)=O)CC2)C1 c1(CN2CC(NC(=O)Cc3cccnc3F)C(F)C2)cnc2ccc(Br)cc2c1 c1(C(=O)NC2CC(C)(NC(c3cncs3)=O)C2)nccc(Cl)c1F C1(NC(C(c2ccccc2Cl)(C)C)=O)CS(=O)(=O)CC1NC(c1cnsc1)=O CCC(C)C(=O)NCCOC1CCN(C(c2cn(C(C)(C)C)cn2)=O)C1 CC#CCC(C(=O)N=c1ccn(CC(N)=O)[nH]1)NC(=O)C(F)CC1CCOC1 c1(C(N(CC(CNC(CC=C=C)=O)C)C)=O)cc(C)c(Br)cc1C Cc1ccc(C)n1CC(=O)NCCCNC(=O)C(C(C)C)n1cncn1 C(=O)(CCCCC)NC1(COC)CN(C(=O)CC2CCCN2C(C)=O)C1.O N1(C(CCC2CC(C)C2)=O)C2CCC1CC(NC(=O)C(c1ccnn1C)O)C2 c1(C(=O)NCC(C)NC(=O)CC2CCC2)cc2ccccc2nc1O C1(C(N2C(CNC(CCCc3ccc(C)s3)=O)CC(O)C2)=O)CC2C(C1)C2(F)F C1(O)(C(C)NC(c2scc(OC)c2)=O)CCN(C(=O)C(C)CC2CC2)CC1 CC(N=c1[nH]c(N2CCC3(CC2)CC(=O)NC(=O)C3)nc2cc[nH]c12)C1CSC1 CC(=O)CC(C)(C)CC(=O)N1CCC(NC(=O)COc2ccccc2)C(C)C1 c1(C(=O)NCC(CNC(Cc2cc(C)sc2C)=O)CO)cc(F)c(C)c(F)c1 C(=O)(C(CCOCC)NC(=O)CCc1cnn(C)c1)N(CC=C)CC=C Cc1cc(C)c(S(N)(=O)=O)cc1NC(=O)C(=O)NCCC1CCN(C)C1 C1(C(=O)NC2(C(=O)NC(c3nc(C)on3)C)CC(CO)C2)CCNC(=O)C1 CCCCCCCN(c1ccc(S)cc1)C.C1(=O)CCCn2nnnc2CO1 N1(C(c2nnn(C)n2)=O)CCCCC1C1CCN(C(=O)C(F)C2CCC2)C1 C(=O)(C(C)(F)C=O)OCC.C1CCCN(C(=O)CC2CC(N(C)C)C2)C1.N c1(OC)c[nH]c(C(N2CC3(C2)CN(C(=O)CCC2CCC(C)O2)C3)=O)cc1=O C(=O)(C(F)C(C)(C)O)N.c1(CNC(CC2(COC)CC2)=O)ccccc1 C(=O)(C1=CS(=O)(=O)CCC1)N1CCCCCC1.C(C(=O)N)(C1CCC1)OCC C(=O)(C(C)(C)CC(=O)N1CCN(C)C(C(N2CCC3CC23C)=O)C1)OCC C1CCC2(CCCN(C(=O)C=CCO)C2)C1.c1(C=O)ccc2c(c1)C(=O)NC2.N O(N=C1CCCCCC1)CC=O.C(c1ccc[nH]1)=CC(=O)NC(C1CC1)C.C C1(COC(C=C(C)C(C)(C)C)=O)CC(F)CN1C(=O)OC(C)(C)C.C c1(C(=O)NCC2N(Cc3ccc(CC)cc3)CC2)cn2c(n1)CCC(C)C2 c1(C=O)ccc2c(c1)nnn2C.C12CC(C1)C2.C1(C)(C(C)C)CC1C(=O)N N1(CC(=O)OC)CCN(C(=O)C(N2CCNCC2C(C)C)=O)CC1 N1(C(CC(CCC)(C)O)=O)C2CCC1CN(C(=O)Cc1nc(=N)[nH][nH]1)CC2 c1(CC)nonc1C(=O)NC(C(=O)NCCn1ccnc1C)C1(C)CC1 c1(C(N2CCC(C(C)NC(C3(C#C)CCC3)=O)CC2)=O)ccc(F)cc1NC N1(C(Cc2ccc(C(C)=O)s2)=O)CCCC1C1CCCN1C(C1CCCC1O)=O c1(OCCN(C)C)ccc(CN(C)C(C2CCOC(c3ccccc3)O2)=O)cc1 CCC(O)C=O.c1(C(N(CCCSC)C2CC2)=O)cccc(C2(C)CCO2)c1.N C(=O)(C(C)(C)CC(F)F)NCC(C)(C1CC1)NC(C(C)n1ccnn1)=O N1(Cc2cccc(C(C)C)n2)CC=C(CCNC(=O)C(c2ccccc2)C)CC1 N1(c2nccc(OCCC)n2)CCN(C)C(CNC(=O)C=Cc2cccnc2)C1 c1(C(=O)N)ccc(S(N)(=O)=O)cc1N.N1(C(CC(C)OC)=O)CCC2(CCC2)C1 C1(F)(CNC(c2cncc(C)n2)=O)CCN(Cc2c(Br)cncc2Br)CC1 CC(C)CCC(O)C(=O)N1CC(CNC(c2cc(N(C)C)ccn2)=O)C(C)(C)C1 c1(CCS(=O)(=O)NCC(c2occc2Br)=O)cc(F)cc(F)c1 N1(C(C2C(NC(C(C)Cc3ccccc3)=O)CC2)=O)CC2C3C=CC(C3)C2C1 C1(CN(C(C)C2CC2)C)CCCN1S(C)(=O)=O.c1(C(C)C=O)cnn(C)c1 Cc1nccc(C(=O)NC2CC(C)CN(C(c3noc(C4CC4)c3C)=O)C2)c1C c1(N2CCCC(C)C2)cc(S(=O)(=O)NCCCSC2CCCCC2)ccc1C#N c1(C(N2CCC(NC(C(=Cc3ccco3)C)=O)CC2C)=O)cnn2ncccc12 Cc1nc(C)c(C(=O)NC(C)C(C)NC(=O)CCc2cscn2)s1 N1(C(CN(C(=O)C=CCO)CC2CCCC2)=O)CCN(C(C)=O)CC1C [N-]=[N+]=NC1CC(C(=O)NCCc2cccc(F)c2)N(C(C23CCC(C2)C3)=O)C1 c1(C(=O)NCCN(CCC)C(c2cocc2C=O)=O)nc(Cl)c(Cl)s1.O C1(C#CC(=O)N2CCC2C(N2CCCC(F)(C(N)=O)C2)=O)(CC)COC1 S(=O)(=O)(c1ccc(NCCN(C)CC)c(Br)c1)NC(c1cccnc1)CC.O CCC(C)CC(=O)C(=O)N1CCC=CC1C(N1CCC(NC(N)=O)CC1)=O c1(NC(C(C)NC(C(N2CC(C)(NC(C)=O)C2)C)=O)=O)ccccc1C C(c1cnn(C)c1)=C(C(=O)NC1CCC(NC(CNS(NC)(=O)=O)=O)C1)C C1(NCC=C)CN(C(c2cccc(C(=O)OCCO)c2)=O)CCS1 c1(C(N2C(CNC(CC3C(C)(C)C3)=O)CC(F)(F)C2)=O)cnc2nccnc2c1 n1(CC)cnnc1CCNC(C1(NC(=O)CC)CCSC1)=O.C(=O)CC.N c1(C(=O)NC2CCN(C(CC(CC)C)=O)C2C2CC2)nc2c(s1)COCC2 CCCCCC(CC)C(=O)N1CC(COC)(CNC(c2cc[nH]c2)=O)C1 Cc1nnnn1CC(=O)NCCCC1(NC(=O)C(C)CC2CCCC2)CC1 c1(C(=O)NC(CCCNC(c2c(CC)cno2)=O)C)c(N)cc(F)cc1F C1(CC)CN(C(=O)C(C2CCCCCCC2)O)CCC1NC(C1CCC=CO1)=O C(CCC1CCC1)(C(=O)NOCCC(F)(F)F)NC(C(n1ccc(C)n1)C)=O C(c1ccc(C)c(Cl)c1)=CC(=O)NC1CCCC(NC(CCOCCC)=O)C1 CC1CC(C(=O)COc2ccccc2)CN(C(=O)C2CC2)C1 c1(CC(=O)NCC2N(C(C3C(COC)C3)=O)CC2)cnccc1C c1(-c2ccc(CC)nc2)ccc(O)c(S(=O)(=O)NC(c2ccncc2)(C)C)c1 c1(C(=O)NC(CNC(C2N(CCC)CCC2)=O)(C)C2CC2)cccc(C)c1Cl c1(C(=O)NCC2CCN(C(c3c(CC)occ3)=O)CC2)cc([SH](=O)=O)cs1 N1(C(=O)CC2CCCN2C(C2CCCOCC2)=O)CCC2(CC1)CC2 C(=O)(C(C(C)C)C(C)C)N1CCN(C(c2ncc(OC)cn2)=O)CC1CF c1(N2C(CNC(=O)CC3COCCO3)CC(F)(F)C2)ncnc2cccc(Br)c12 c1(NC(N2CCC(CNC3C(C(=O)OC)CCCC3)CC2)=O)ccc(C)cc1C C12(NC(C3C(CC)C3)=O)CCC(CC1)N(C(=O)C(C)OCC(F)(F)F)C2 c1(CC(=O)NCC2C(NC(c3c(C)cns3)=O)CC2)c(C)nn(C)c1C CC(C)(C)CCC(=O)NC1CN(C(C2(CCF)CC2)=O)CCC1C(F)(F)F c1(OC)cc(CNC(c2ccc(OC(F)F)c(S)c2)=O)ccc1C(C)(C)C CC1(C)CCC(CNC(=O)C2=COCCC2)N(C(=O)CNC2CC(F)C2)C1 N1(C(C(=O)Nc2ccccc2F)=O)CC2CC(C1)N(c1nc(Cl)ncc1Br)C2 CN1CCn2ncc(C(N3CC(N(C(=O)CCCCCF)C)C3)=O)c2C1 N1(C(c2c(C)n[nH]c2C)=O)CCCC2C(CCCN2C(=O)C=Cc2cc[nH]n2)C1 c1(C(N2CC(CCCCNC(C(CC)OC)=O)C2)=O)nc2ccc(Br)cn2n1 Cc1cc(F)cc2[nH]c(C(=O)N(CCCNC(=O)C(C)c3cncs3)C)cc12 C(C(C(=O)NCC#CCCO)OC)NC(C1(SC)CCC1)=O CC1COCC(CC(N2CCC(C)(CC(=O)N(C)CCN(C)CCO)C2)=O)O1 Cc1ccc(CC(=O)NC2(c3c(Cl)cccc3Cl)CCC2)c(Br)c1 c1(CN2CCC(C)C2CNC(=O)OC(C)(C)C)cccc2ccccc12 CCC(C)CCCC(=O)N(CC(=O)NCc1nnc(C)o1)CCOC C(=O)(C(F)C(C)(C)O)NC(C1(O)CN(c2cnc(F)cn2)C1)C CCS(=O)(=O)CC(=O)N(CCNC(c1occc1C(C)C)=O)C(C)C C1(NC(c2ccc(CC)c(F)c2)=O)CCN(C(=O)C=CC(C)C)CCC1(F)F CC(C)C1=NOC(C)(C(N2CC(CC)C2)=O)C1.C1(CS(N)(=O)=O)(C)COC1 c1(-c2ccc(-c3n(CC)ncc3)cc2)ccc(CNc2cncc(F)c2)cc1F C(C(CC(=O)NC1CCN(C(c2cccc3nsnc23)=O)CC1)C(F)F)N(C)C C#CCC(C)(C)C(=O)NC1CCCC1NC(=O)CC(C(F)F)c1ccc(F)cc1 C(=O)(C1=CCCSC1)N1CC(N(C(C2CCCN(CCC)C2)=O)C)C1 c1(Oc2ccc(C(=O)NCCCNC(C(C=C)(C)O)=O)cc2)ccccc1C#N C1(NC(c2ccc(C(=O)OC)cn2)c2nnnn2C(C)C)CCC(F)(F)CC1 N1(C(C2(C(C)C)CCN(C(CC(CCC)C)=O)C2)=O)CCC([N+](=O)[O-])CC1 CON1CCC(C(N2CC(NC(c3ccc(-c4ccco4)o3)=O)C(C)C2)=O)CC1 CC1(C)CCC(O)(C(=O)NC2CN(C(=O)C)CCC2F)CC1.C1CC(F)(F)C1.O c1(C(C)(C)C)nc(C(=O)NC2CC2)co1.C1CCCN1C(c1cc(O)cs1)=O C(c1ccc(Cl)cc1)=CC(=O)NC1C(OC)CN(C(C2(O)CC2(C)C)=O)C1 c1(C(=O)NCC2C(NC(=O)Cc3cc[nH]n3)CCCC2)cccc(=O)n1O Cc1cc(C(=O)N(C)CC2CC2)cc(C)c1Cl.C1(CC(=O)N)CCC(C#N)C1 CC(C)CCC(=O)NCC(N1CCOC(C(C)(C)C)C1)=O.C12(CCC1)N(C)C2 C(=O)(CC(C(F)F)C(C)(C)C)N1CC(C)CC1.CC(C)C(C(=O)N)n1cccc1.C N1(C(CCC#N)=O)CCC2(COC(CNC(=O)Cc3cnoc3)C2)C1 C(CCN(C)N1C(C)CC2(CCC2)C1C)(OC)OC C#Cc1ccc(C=O)c(C)c1.c1(N(CC(=O)N(CCC)C)C)ccc(Cl)nn1.N c1(C(N2C(C(C)C)CN(C(C3CCC(=O)N3)=O)CC2)=O)cn2cc(Cl)cnc2n1 C12(C(N3CCC(C)(CCNC(C4(CF)CCC4)=O)C3)=O)CCC(F)(CC1)CC2 CCC(CC)C(=O)NC1CC(NC(=O)CC(C)C2CCCC2)CC1O N1(c2cc(N(CC(CC)(C)OC)C)nc(C(F)(F)F)n2)CCOCC(C)(C)C1 C1(CNC(c2ncn(C)c2)=O)CN(C(c2cc(C3(C)CC3)on2)=O)CC1O C12(C(N3CCC(N(C)C(C4(c5ccccc5)CC4)=O)C3)=O)CC(CN1C)C2 N1(C(Cc2c(C)n[nH]c2)=O)CCC(C(=O)NC(C)CCC2CC2)(CO)C1 C1(C(N2C(CNC(C(CC)(C)C)=O)COCC2)=O)CCn2cnnc2C1 C1(n2cc(COCC(N)=O)nn2)CCCN(C(c2ocnc2C2CC2)=O)CC1 N1(CCC)C(=S)NC(c2cc(F)c(F)c(Cl)c2F)C(C(=O)OC)=C1C N1(C(C(CC(=C)C)C)=O)CC2CCC(C1)C(NC(=O)CN1CCCCS1(=O)=O)C2 Nc1ccc(C(=O)NC2CC(CNC(C34CCC(CC3)O4)=O)C2)c(F)c1F C=CC(C)CC(=O)NC1CCCC1CNC(=O)CCn1ncn(C)c1=O N1(C(c2c(C)nc(CC)s2)=O)CC2(C1)CN(C(=O)C(F)=C(C)C1CC1)CCO2 N1(C(c2ccccc2)=O)CC2CC(C(=O)NC3(c4ccccc4)CC3)(C2)C1 N1(C(C(CCSC)O)=O)CCC2(CCC2NC(c2cncc(N)n2)=O)CC1 c1(C(=O)NC2CCCCC2CNC(C2CC(F)(F)C2)=O)ccc2ocnc2c1 N1(CC(N2CC(CC)OCC2)=O)CCCNS1(=O)=O.c1(CC)ccoc1C(=O)N CCC(CC)C(C(=O)N1CCC(CNC(C2CC3CC(=O)C2C3)=O)C1)OC c1(C=O)cc(Cl)c(Cl)cc1O.CC1(C(F)F)CC1C(=O)NCC1CCC1.N c1(C(N2CC3C(NC(C(C)CO)=O)(C3)C2)=O)cc2sc(Br)cc2s1 C(=O)(C(F)C(C)(F)F)N1CCC(CCNC(CSCC#C)=O)C1 c1(C2(C(=O)NCC3CC(N)(CO)C3)CCC2)ccc(Br)cn1 c1(C(N(C(=O)Cc2cocn2)Sc2ccco2)=O)c(C)cccc1Br.CO c1(C(=O)OC)ccc(NC(C2CN(C(=O)C(F)F)CCN2)=O)c(Br)c1 C1(C(=O)NCC(CCC=C)O)CN(C(=O)Cc2cscn2)CC1C1CC1 C1(NC(CCCC#C)=O)(COC)CCCN(C(=O)C(C)Sc2nncn2C)C1 Cc1c(C(N2CCOC(C(C)NC(C3CCCCC3(C)C)=O)C2)=O)cccc1F C(C(=O)N(CC(C)C)C)(C(C)C)NC(C)=O.c1(C(=O)N)cnn(C(F)F)c1 Cc1nc(-c2ccccc2)sc1CC(=O)NC(C)C(C)NC(c1cnc(Cl)[nH]1)=O c1(C(N2CC(O)C2)=O)ccc(Cl)c(F)c1N.c1(CC)nc(C)n(C)c1C(=O)N c1(C(=O)N)ccc2c(c1)CCC(C)(C)O2.S(=O)(=O)(CC(=O)NCCCC)NC CS(=O)(=O)CC(=O)NCCC(O)C(=O)NC1CCOC1 C(=O)(C1=CC2CCC(C1)C2)N1C(C(N2C(C)CNC(=O)C2)=O)C(C)CC1 c1(NC(C2CCCN(Cc3cccc(-n4cncn4)c3)C2)=O)ncncc1Br CC(CC(=O)N1CCC(N(CCO)C(C2CSC2)=O)C1)n1cc(Br)cn1 c1(NCCC(c2cnn(C)c2)C)nccc(NC(c2ccccc2)CC2CC2)n1 C(=O)(C(O)CC(N)=O)NC12CC(NC(CCC3CC(OC)C3)=O)(C1)C2 C12(C(N3CC(O)(CNC(C(C(CC)C)OC)=O)C3)=O)CCCCC(=O)N1CCC2 C1(C(N2C(CNC(C=COCC)=O)CC2)=O)CCCC2(CC2)C1 N1(C(C2(C=C)CCC2)=O)CCN(CC2(NC(=O)CC3CCCOC3)CC2)CC1 N1(C(C2CCCC(O)C2)=O)CC2(CCN(C(C3(C(=O)CCC)CCC3)=O)CC2)C1 C(=O)(C1=NN(C)C(=O)CC1)N1CC(N(C(c2nc(COC)oc2)=O)C)C(F)C1 N1(C(C=C(C)c2cccs2)=O)CCC(NC(c2cccs2)=O)C(CO)C1 C(=O)(C(O)CC(C)(C)C)N(CC)C.CC(C(=O)N)N(C)C(C1CC1)=O.CC N1(C(c2cc(F)ccc2Br)C(=O)NC2CCOCC2)CCc2c(ccnc2Cl)C1 C1(C(N(CCCNC(CCNC(=O)NC)=O)C)=O)CC2C=CC1C2 c1(N2CC(CC)OCCC2)cnc2ccc([N+](=O)[O-])cc2n1 C1(CNC(c2c(C)nc(C(C)(C)C)s2)=O)CC2CN(C(c3ccsc3)=O)CC12 CC1=NC(C)(CNc2cc(N3CCC(N4CCCC4)C3)ncn2)N1C C(=O)(CC(O)C(C)C)N1C(CNC(c2cc(COC)on2)=O)CCCC1 c1(C(N2CCCN(C(C3CC(CC)C3)=O)CC2)=O)cc2scc(C)c2[nH]1 CC1CN(C(=O)C2=CCOC2)CC(C)C1NC(=O)Cc1cnc2cccnn12 C1(NC(C=C(CC)CC)=O)CN(C(C2CC2C2CCCC2)=O)CC2(CC2)C1 CC1(C)CC(NC(C2(C)CCOC2)=O)CCN(C(c2cccc(F)c2Cl)=O)C1 C#Cc1ccc(C(=O)NCC2CC2CNC(=O)CCC=CBr)c(F)c1 N1(C(CN(C2CC2)CC)=O)CCC1CC(=O)NCC(c1ccco1)O C1(C(=O)NC2CN(CC)C2)CN(C(c2ccccc2Cl)=O)CC1(C)C N#Cc1cc(C(N2Cc3[nH]nc(NS(=O)(=O)CC4CC4)c3C2)=O)ccc1Br C(C(CCC)CCCC)NC(c1ccc(CNC(CCCC)=O)cc1)=O CN1CCC(C(=O)NC2CCCCC2NC(c2ccc(N(C)C)nc2)=O)C1=O Cc1ccc(Cl)cc1C(=O)NC(C)(C)C(C)NC(C1CC1C(C)(C)C)=O C1(CNC(=O)C=CC2CCCO2)CC2CCC1N(C(C1(F)CC=CC1)=O)C2 C1CN(C(=O)C=Cc2cnc[nH]2)CCC1F.c1(C(OC)OC)ccc(C=O)o1.N c1(C(=O)NCCCCC)cc2c(s1)CC(C)(C)C2.C(=O)CC.[SH](C)(=O)=O.N C(C(CC(C)C)C(=O)N1CCC(CO)C(NC(=O)C=Cc2ncc[nH]2)C1)OC c1(C(N2CC(SC)C(NC(=O)Cc3[nH]cnc3C)C2)=O)csc([N+](=O)[O-])c1 C1CCN(S(F)(F)F)CC1.C1(SCC)CCCO1.O=C(CSCC)N.C=O CC(CC(C)NC(=O)C(C)(F)F)NC(C1(c2ccc(Cl)s2)CC1)=O C1(NC(C2(C)CC2F)=O)CC2(C1)CN(C(=O)Cn1cnc(Br)n1)C2 Cc1cc(C#N)ccc1NC(N1CCC(c2ccccc2)CC1C)=O c1(C(N2CCC(C(C)(C)NC(CC(CC)C3CC3)=O)C2)=O)cccc2nncn12 C(CCCC(=O)NCc1ncc(Cl)cn1)N(C(CCn1ncc(C)c1)=O)C C1(C(N2CCC(c3nc[nH]n3)CC2)=O)CCCN(C(C2C=CCCC2)=O)CC1 C(=O)(C(C(C)CC(C)C)N(C)CCSC)NCCCC Cc1cccc(C(=O)NC(C)(C)CNC(=O)COC)c1C#N.C1CCOC1 c1(C(=O)NCC(CNC(c2ccc(CCC)cc2)=O)(C)O)ccn2ncccc12 c1(COCC)nc(C(=O)NCCC(C)NC(c2cc(Br)c[nH]2)=O)cs1 c1(NC(C2CSCCN2Cc2cc(Br)c[nH]2)=O)nc2ccccc2nc1Cl c1(C(=O)NCC(C)C)cccc(S(=O)(=O)C2CC2)c1.c1(C=O)cccc(N)c1 c1(CC(=O)NCC2CC(NC(C3(C)CCCCC3)=O)C2)nsc2ccccc12 C(=O)(C(C)CF)N(C(C)C)CCNC(C1(CN(C)C)CC1)=O C(=O)(C(F)(F)C(C)O)N.C1(=CC(=O)NCCC(C)OC)CCN(C)CC1 C(=O)(C(C)CC(C)(C)C)N.N1(C(c2ccn(CCOC)n2)=O)CCC(C)(C)C1 C1(C(c2nnnn2C2COC2)NCc2cnc(C)[nH]2)(OCC)CCCCCC1 n1(CC)nc(C(N2CC(NC(=O)CC3(C)CCCCC3)C(O)C2)=O)c(Br)n1 N1(C(C=COCC)=O)CCC(NC(C2CCC3CC23)=O)C(C(N)=O)C1 C(Cc1ccccc1)(CCNC(C12CC(C1)C2)=O)NC(C1(Br)CC1)=O C1(C(=O)OCc2c(C)csc2)CCc2nnc(O)cc2C1 c1(CC(=O)NC2CC(O)CN(C(=O)Cn3ncnn3)C2)ccc2c(c1)COCC2 C1(NC(C2C(CNC(C(C)C3CCC3)=O)C2)=O)(CC2CC2)CCCCC1 c1(-c2c(NC(c3c(F)cccc3F)=O)ccnc2)cc(F)c(O)c(F)c1 CC(CC1CCCO1)C(=O)NC.C1CC(C(N2CC(N(CC(F)F)C)C2)=O)C1 CCCC(C(=O)NCC1CCN1C(C1(c2ccccc2)CNC(=O)C1)=O)OC CC1CC(C)(C)CN1C(C1CCCC(C)(C)C1)C(=O)NCCC1(C)CC1 C1(N(C(C23CC(CCC)(C2)C3)=O)C)CN(C(=O)C2=C(C)CCC2)CC1(C)C CC1CN(C(=O)CCc2ccc(OCC(N)=O)cc2)CCN1C(=O)CC(C)(C)F c1(OC)cc(C2(C(=O)NCC(C)(C)NC(c3cnns3)=O)CCCC2)ccc1C C1(CC(=O)N(C)CC2CCCN(C(=O)COC3CC3)C2)CC2C=CC1CC2 Cc1nc(CC(=O)N(CCCNC(C2(c3ccncc3)CC2)=O)C2CC2)n[nH]1 c1(OC)cccc(CN(C(=O)CC2CC(N)C(O)C2)CC(C)C)c1 N1(C(C(OC)OC)=O)CCc2nc(CNC(C3CC(N(C)C)C3)=O)sc2C1 c1(C(=O)NCC2CC(O)(CNC(=O)CCF)C2)cc2ccccc2cc1F c1(C(N2CCCCC2c2ncc(C)s2)C(=O)NCC)ccc(C(=O)OC)cc1 C(=O)(CCS(C)(=O)=O)N1CCCCC1.C(C)(CC)NC(=O)OC.C(=O)C.N C1(CC=C)(NC(C2CC2=C)=O)CCN(C(=O)COc2cccnc2)C1 C1(CCC(=O)N(CCNC(C(C)NC(CC)=O)=O)CC)CCCN(C)C1 Cc1nnccc1C(=O)N(CC(C)NC(=O)C(C1(O)CCCCC1)(F)F)C C(=O)(C(C)(F)C(C)(C)F)N(CCOC)CC.c1(C=O)scnc1C1CC1 C(C(C)CC(=O)N(C)CC1COCCN1C(c1c(Cl)cnn1C)=O)OC C1(NC(CC2(CSC)CC2)=O)CCN(C(c2cnc(N)cn2)=O)CC1O C1(NC(CCCCOC)=O)COC2(CCN(C(c3sc(F)cc3Cl)=O)C2)C1 Cc1cccc(C(=O)N(Cc2cccs2)CC2CCCO2)c1F C1(C(=O)NCC(CNC(C=C(CC)CC)=O)O)CC(CO)C12CCC2 C(CO)(CCCCNC(c1cccc(=O)o1)=O)NC(c1ccnc(O)c1)=O CC(C)C(C(=O)N1CCC(C)(CC)C1)NC(N)=O.C1(N=[N+]=[N-])(C=O)CC1.N C(=O)C1=NN(c2ccc(F)cc2)C(=O)CC1.C(=O)(C(C)C(F)F)N(CC)CC c1(C(=O)NC2CN(C(CC3CC(CC)OCC3)=O)C2)c(C)nn(C)c1OC c1(C(N2CC3C(NC(=O)C(O)Cn4cncn4)(CC3)C2)=O)cnc2n1CCOC2 C1(NC(CC(CC)C2CC2)=O)CN(C(=O)CN(C(=O)COC)C)CCC1O c1(C(N(CCCNC(C2(CC#C)CCCCO2)=O)CCO)=O)ccc(F)cc1Cl c1(NC(=O)OC)ccc(C(N2CCCC(C)(CO)C2)=O)c(C)c1.c1ccoc1 C12(NC(c3c(C)csc3)=O)CCOCC1CN(C(=O)C=Cc1cccc(Cl)c1)C2 c1(N2CC(N=[N+]=[N-])C(O)C2)nc2c(c(=NCC3CCOC3)[nH]1)COC2 Cc1cc(Cl)ncc1CC(=O)N(C)CC1(NC(=O)C)CC1.c1ccccc1Cl.N C1(C(N2C(C(=O)NCC(CC(=O)OC)O)CC2C)=O)CC2COCC2C1 c1(C(N2CCC(C)C(CN=c3[nH]cncc3F)C2)=O)cn2c(CN)cccc2n1 CCC(CC(=O)NCC1COCCN(C(c2cc(C)sc2N)=O)C1)C(C)(C)C c1(OC(C)C(=O)N(C)CC2CCCCN2C(=O)C(C)C(C)O)ccccc1Cl c1(NC)cccc(C(=O)NCC(C)(C)CC2CN(C(=O)CC3CCCO3)C2)n1 c1(C(=O)NCCCOC)ccc(C2COCCN2C(c2cnsn2)=O)n1C Cn1c(C(=O)NCC2CC(F)(F)CN2C(=O)C(F)F)cc2ccccc12 CCC(C)CCCCC(=O)N1CCN(C(C2CNC(=O)N2)=O)C(CCO)C1 N1(CC)CC(C(=O)NC(CNC(C23CCC(C2)C3)=O)CC(C)C)CC1=O N1(C(CCOC)=O)CCC2(CC(NC(c3n[nH]cc3C(F)(F)F)=O)CO2)C1 C1(CNC(C(N)=O)=O)CC2CC1CN2C(=O)CN1CCCCS1(=O)=O C1(C(=O)NC(CC2CN(C(C3(CC)CCC3)=O)C2)C)CCCCN1S(N)(=O)=O C1(CCC)CN(C(C2CCCC2)=O)CCN1C(c1cc(CC)no1)=O N1(C(CSc2n(C)c(S)nn2)=O)CCC(C2(NC(C3CC3)=O)CC2)C1.CCO.C C1(NC(CC(C)(C)C)=O)CC12CCN(C(c1cc(Cl)cs1)=O)C2 C1(NC(CNC(=O)NC)=O)CCCCC1NC(=O)CSC1CCOC1=O C(C1CN(C(c2cncs2)=O)CC1C(=O)NCC1(C)CC1(C)C)=CC CCC(C)CC(C(=O)NCC#CCCO)NC(C1CN(C)C(=O)N1)=O c1(CCCC)ccc(C(C)C(=O)NC2=NCC2OC)cc1 C(=O)(CC(CC)C(C)C)N1CC(c2ccccc2)C1.C=C1CC(C)(C(=O)NC)C1 C12(NC(=O)CNC(C3CCC3)=O)CCN(C(=O)Cc3cnc[nH]3)CC1C2 N1(C(C2CCC(C(=O)OC)C2)=O)CC2CC(C1)N(C(c1ccc(Br)nc1F)=O)C2 C1(CC)CN(C(=O)C=Cc2ccoc2)CCC1NC(c1ccsn1)=O O=C1C2N(CC23CCOCC3)C(=O)N1C1CCCC2(CCCC2)C1 c1(CC(=O)NC2CCC(CNC(COC(CC)(C)C)=O)C2)cccnc1N N1(C(C(C(C)C)OCC)=O)CCCC(CO)(NC(C2CCCCC2(C)C)=O)C1 N1(C(c2nn(CC)c(O)c2)=O)CC2(C=C(C(=O)N(CC(C)CO)C)CO2)C1 c1(C(=O)NC(C(C)NC(c2cn(CC)nc2)=O)(C)C)cc(C)c(C)s1 C1(C(N2CC(=C)C2)=O)CC2C=CC1N(C(=O)C(=Cc1ccccc1)C)C2 C(=O)(CCCC(F)(F)CO)NC1CCC(NC(C(C)NC(c2ccco2)=O)=O)C1 C1(C=O)CC2CCC2C1.c1(C(C)(F)F)nc(C(=O)NCCOCCC)cs1.N c1(N2CCCC(OCC)C2)[nH]c(=NC(C)CF)nc2ncn(C)c12 C1(NC(c2nccc(C)n2)=O)CCCC12CCN(C(C1(F)CC3(CCC3)C1)=O)C2 Cc1ccc2[nH]nc(C(=O)NC3(C)CC(NC(C4CCCCC45CC5)=O)C3)c2c1 C1(C)(C(=O)NCC(C)NC(C2(F)CCC(F)(F)CC2)=O)CC(C)OC(C)C1 C=CCC(C)(C(=O)NC1CCCN1C(C)C(=O)N(C)C1CC1)N(C)C N1(C(CCOCC)=O)CC(NC(=O)CC2CC23CC3)C(n2ccnn2)C1 C1(C(=O)NCC2ON=C(CC)C2)CC2(CCN1C(=O)CC(C)(C)COC)CC2 CCC(C(C)(C)O)NC(=O)C(C)NC(C1CCCCC1O)=O Cc1cccc2c(C(N3CCC(CO)C(NC(c4cnco4)=O)C3)=O)n[nH]c12 C(=O)(C1CCc2snnc21)N1CC(N(C(=O)CCn2cncn2)C)C2(C1)CC2 N1(NC2(c3nnnn3CCCC3CC3)C(C)SCC2)Cc2ccc(Cl)cc2C1 C=C(C)C1OCCC1C(=O)NCC1(F)CCC1.c1(C=O)coc(N(C)C)n1 N1(C(CC2(C=C)CN(C(=O)CC3CC(SC)C3)C2)=O)C2CCC1CC1(CC1)C2 N1(C(C(CC)C#N)=O)Cc2ccccc2CC1CNC(=O)C(C)OC C1(N(C(C2(CO)CC2)=O)C2CC2)CN(C(=O)C=CC2CCOC2)CC1.C CCC(C)(C(=O)OCC1CC(NC(c2ccsc2OCC)=O)C1)OC c1(C(=O)NCC(CC)NC(=O)CCC2CCC2)csc2ccncc12 c1(C(=O)NCCCCNC(C(C)OCC#C)=O)cc(C)cc(C)c1O C1(NC(c2n(CC)cnn2)=O)Cc2ccccc2N(C(C2CCCC2O)=O)C1 c1(C(=O)NC(C2CN(C(C3(C)CC=CCC3)=O)C2)C)ccc(Cl)c(N)c1 c1(C2C(=O)CC2)cc(-c2ccc(C3CC3)o2)[nH]n1 C(C(F)C(=O)N1CCCC1CCCNC(C1(C)C=CCC1)=O)N(CC)CC C12(CNC(c3coc(Br)c3)=O)CCC1CN(C(=O)Cc1ccnnc1O)C2 CC1CCN(C(=O)NCc2c(I)cnn2C)CC1(C)C CC(C)(C)C(CO)C(=O)NOCC(=O)NC1CC(C)(CO)C1 N1(C(C(C)CC(N)=O)=O)CCCC(C2(NC(c3cncc4c[nH]nc34)=O)CC2)C1 C1(COCC(=O)NC2CCCC2)CCS(=O)(=O)C1.n1(CC=O)cncn1 C1(CC(=O)NC(CNC(c2cc(CC)on2)=O)(C)CC)CCC(C)(C)C1 C(=O)(CS(=O)(=O)CC(F)(F)F)N1C2CN(C(Cn3nc(C)oc3=O)=O)CC1CC2 C(=O)(C1CCCc2ccccc21)NC1(C)CCN(C(c2c(C)coc2)=O)CC1 c1(NC(CC(C2CC2)NC(CCCC)=O)=O)ccc(OC)c(F)c1 C(=O)(C1=C(C)N(C)c2ncnn2C1C)NC1CC(NC(CSC)=O)C1 c1(CC(C)OC)nc(-c2ccc(CO)cc2)n(-c2ncnn2C)n1 c1(C(N(CC(C)NC(=O)C(O)Cn2cncn2)C)=O)cc(C2CC2)n(C)n1 N1(CC(=O)N)C(=O)C(=O)N(C)C1=O.C1(OC)CN(C(=O)CCC(N)=O)CC1 C1(CC)CCN(C(c2cc(CO)n(C)n2)=O)C1C(=O)NCCN1CCNC1=O C1(NC(=O)C=CC2CC2)CCN(C(c2ccn(CC(F)(F)F)n2)=O)C1.CC C1CCC2(CCN(C(=O)C(F)(F)C(O)C3CC3)CC2)O1.c1(C(=O)N)cnns1.C N1(C(CNC(C)=O)=O)CCCC(C)C1CCNC(c1ccc(C)c(C)n1)=O C1(C(=O)NCC(CNC(c2ccc(C(=O)OC)o2)=O)C)CC2(CCC2)C1 c1(CC)nocc1C(C(=O)NC1CCOC1)N(C(C)C(C)C)CC C1(NC(=O)Cn2ncnn2)CCOCC1NC(=O)C(O)Cc1ccccc1 N1(C(CC(C(C)OC)NC(=O)C(F)CC(C)(C)C)=O)CC(C2=NOC(C)C2)C1 C1(C(N2C(Cc3cccc(C)c3)CCCC2)=O)CCC(O)C1(C)C c1(C(N(CCCNC(CCCC#CC)=O)C)=O)n[nH]c2cc(Cl)ccc12 N1(C(CCc2cc(C)sc2C)=O)CC(NC(C2CC2C(C)(F)F)=O)CC12CCC2 c1(CC)n[nH]cc1C(=O)NCCN(C(=O)C(C)S)CC(C)O.C1CCCC1 C(=O)(C1CCCc2ncnn21)NCCCCNC(C1CC(F)C1)=O CON(CCC(=O)NC(c1nn(C)cc1O)C)C(=O)Cc1cncnc1O N1(C(C(c2cncc(F)c2)C)=O)CCCCC(NC(c2n[nH]cc2C2CC2)=O)C1 Cc1cccc(Cl)c1C(=O)NC1CCN(C(=O)Cc2cccc(O)c2)CC1F N1(C(C(C2CCC2)OC)=O)CCN(C)CC1CNC(C12CCCN1CCC2)=O C1(C(=O)NCC(C)NC(c2ccn(C(F)F)n2)=O)COC(=O)O1 C1(CNC(c2c(OC)scc2)=O)C2CN(C(C3(C)CCCN3C)=O)CC12 c1(C(=O)NCC2CCC(C)N(C(=O)CC3(C4CC4)CC3)C2)cc2ccncc2o1 c1(CC(=O)N(C2CCN(C(C3CC3(C)C)=O)C2)CCO)ccc(Cl)cc1F C(C(C)(C)C(C)(C)O)NC(CCC1CCN(C(CC2CCCN(C)C2)=O)C1)=O c1(N2CCC(N(C)C(C3CC34CCC4)=O)C2)cc(Cl)nc(C2CCC2)n1 c1(NC(C2CSCCN2Cc2cccc(-c3ccsc3)c2)=O)ncc(Cl)cc1O CCCCC(O)C(=O)NCC(C1CCCCN1C(c1ccc(CC)cn1)=O)(C)C c1(C(N2CCCC(N(C(=O)Cc3cscn3)CC)C2)=O)[nH]c2ccccc2c1Cl N(C(=NCC=CBr)N(C)CC12CCC(CC1)OC2)C(C)C N1(C(COCCSC)=O)CC2CC1(C(=O)NCC(O)CCO)C2 C(C(COC)CC(=O)N1CC2C(N(C(=O)C(C)S(C)(=O)=O)C)C2C1)OC C1(N(C(=O)CCC2CCOC2)CCC)CCN(C(=O)CCOC2CCOCC2)C1 C(CC(C)C)(C(=O)NCC(O)CNC(c1cnn(-c2ccccc2)c1Cl)=O)OC c1(OC)cc(C2CC2C(=O)N(C(C)CC)C)ccc1F.C(=O)(CCC(F)(F)F)N [SH](=O)(=O)c1ccc(C)cc1.C(=O)CCO.C(C)(C(=O)NCC)OCC#C.N C1(NC(C(C)(C)c2cnsc2)=O)CC2(C1)CN(C(=O)CCc1cc[nH]n1)C2 C1(C(N(CC(=O)NC)C)=O)CCN(C(c2cnn(C)c2Cl)=O)C1C c1(C(C(c2nnnn2C2CCC2)NCC)Nc2cncs2)cccc(C)c1 c1(C(N2C(C)(C(=O)NC3CC4CCC(C3)C4)CCC2)=O)nccc2cc[nH]c12 c1(CN(C(C(=O)NC(CC)C2CC2)=O)C)ccccc1C(F)(F)F c1(C(=O)N)cccc2c(C#N)c[nH]c12.CC1(C)CC1(Cl)C(=O)NCC1CCC1 Cc1cnc(N(C2CNCC(F)(F)C2)c2cc(-n3cncn3)ncn2)nc1C C1(CNC(c2cn(CC)nn2)=O)CN(C(c2ncc[nH]2)=O)CCN1C c1(C(=O)NC(CCCOC)CNC(=O)CCC2CC2C)ccc2nn[nH]c2n1 c1(C(C(=O)N)(F)F)c(F)cccc1F.C(C)(C(O)C(=O)NCC=CC)OC C1(NC(C(CC)=CC)=O)C2CN(C(C3CC3)=O)CC12.c1cccc(Cl)c1.O CCC(C)(CNCC12CCCN(CC1)C2)CN=c1[nH]cnc(CO)c1C c1(C(CN2C(c3cc(C)nn3C)CCC2)=O)c([N+](=O)[O-])c(C)nn1C C1CN(C(c2ccoc2C2CC2)=O)CCCO1.C1(C(=O)N)CCOC1C1CC1.C C1(C(=O)N)CCC([N+](=O)[O-])CC1.N1(C(c2cn(C(F)F)cn2)=O)CCC2CC2C1 N1(C(c2cc(I)c(C)c(I)c2)=O)Cc2ccccc2C1C(=O)NC1(C)CC1 c1(C(=O)N)ccc(C)c(C)c1O.N1(C(C2CC(SC)C2)=O)CCC(O)(CC)CC1 C(=O)(C(C)(C)C(N)=O)NCC(CNC(C(c1ccc(C)cc1)C)=O)F c1(C(=O)N)cc2cccnc2cn1.C(=O)(C(C)(F)C(=O)NC1CCC1C)OC c1(NC2CCN(C(c3ncn(CC)c3)=O)CC2F)cc(C)nc2cc(C)nn12 C1(O)(C(C)NC(CN2CC(CC)C2)=O)CN(C(c2ccsc2C(F)F)=O)C1 C1(C2CCCN(C(c3cnccc3C(F)F)=O)C2)CC1.C=C1CC(C)(C(=O)N)C1 Cc1ncc(C)c(N2CC(C)(C)CC2CNC(=O)CCNC(=O)C=CCl)n1 O=C(C1=CCCOC1)NC1CCN(C(c2ncc(Cl)cc2F)=O)CC1CO C1(CC(C)NC(c2cnn(CCO)c2Br)=O)CCN(C(=O)CCn2cccn2)CC1 C#CCCCCC(=O)NCC1CC2CC2N1C(=O)Cc1sccc1Br c12ccc(cc1)S(=O)(=O)NCC2.C1(CC)CC(S(=O)(=O)N(C)C)C1 C12(C(=O)NC3(CC=C)CN(C(=O)CCCCO)C3)CCCC1(C(N)=O)C2 N#CCCCC(=O)NCc1ccc(C(N2CCC(O)(CO)C2)=O)s1 C1(C(=O)NCCC2(OCC)CCC2)CCN(C(=O)C)C1.C=O.C1CC1 C(=O)(CC(C)CC(F)(F)F)N(CCC)C.c1(C(C=CC=O)=O)cnn(C)c1.N c1(CN2CC3C(CNC(Cc4ccn(C)n4)=O)C3C2)cccn2ccnc12 C1(C(=O)NC(C(=O)NCC2CCN(C)C2)C2CC2)Cc2ccccc2C1 N1(C(Cc2cc(OC)c(Cl)cc2)=O)CC2(CCCC2=O)C1 c1(C(=O)NCCCCC2CN(C(COCC=C)=O)C2)sc2cccc(F)c2c1Cl C(=O)(CCN=[N+]=[N-])NC1(C)CN(C(CSC2CC(O)C(F)C2)=O)C1 c1(CNCC(C)(OC)OC)cc(C)c(C)cc1O C1(C(=O)NC(C(=O)OC)C2CCC2)CCCCCN1C(c1cc[nH]c1C)=O C1(CC)CCCN(C(=O)C=CCF)CC1.CC(C)C(C(=O)N)NS(C)(=O)=O Cc1ncc(Cl)cc1NC(=O)CC(C)(C)CNC(=O)CC1CSC1 C1(NC(=O)CCN2CCCC2)CC2(CCN(C(=O)CC(F)(F)C(F)(F)F)CC2)C1 c1(C(=O)NCC(CNC(C2=C(C)OCCS2)=O)CO)ccc2[nH]c(=N)sc2c1 c1(CC(=O)NC2C(O)CCN(C(CC(C)CF)=O)C2)cc2ccccc2c(=O)o1 C(CCCCC(=O)N1CCC1C)OCC.c1ncn(C(C)(C)C)n1.C(=O)(C)N C1(CC)(CNC(C2CC(C(N3CC(C(=O)NC)C3)=O)C2)=O)CCOC1 N1(C(C2=CC(C)CC2)=O)CC2CCCC2(NC(=O)C=Cc2ccoc2)C1 c1(N(CCCO)C)nc(N2CCOC(C(C)(C)C)C2)c2ncn(C)c2n1 N1(C(CCCNC(C2N(CC)CC2)=O)=O)C2CCC1CC(CO)C2 C12(C(N3C(C)CCC3)=O)CCCCC1C2(F)F.C1(C(=O)N)(CC)CC1(F)F.C c1(C(N(CC(C)(C)NC(=O)C(O)Cc2ccccn2)C)=O)cccc(F)c1Cl CC(C)(C)CC(C(=O)Nc1ccc(Cl)cc1O)NC(c1ccc(O)cn1)=O c1(CC)ccc(F)cc1C(N1CCCCC1CN(C)C(c1cccc(N)c1)=O)=O Cc1ncnc(N2CCSCC2CCNC(C2(c3cccnc3)CCC2)=O)c1F C1(C(N(C2CCN(C(C3(O)CCSC3)=O)C2)CC)=O)CC2CCC2C1 CC1CN(C(C2CCCC(C(F)(F)F)C2)=O)CCN1C(=O)C1=CCCCO1 CC(C)CC(CNC(C1CC1(C)C)=O)NC(=O)C(c1ccc(F)cc1)F C1(c2ccc(C)s2)CN(Cc2ccccc2Sc2ccccc2)CCO1 C(N=c1[nH]c(=N)[nH]c(=NCCCC2CC2C)[nH]1)C1(CCOC)CCC1 c1(CC(=O)NC(CC)CN(C(=O)C(O)C(F)F)CC)ccc([N+](=O)[O-])cc1Cl C1(C)(C=O)CC(C2CC2)=NO1.Cc1c(C(=O)NCCC)cnn1C1CCCC1.N C(=O)(C(C)S(=O)(=O)C(C)C)N(C1CCCN(C(c2c(C)n(C)nn2)=O)C1)C CC1CN(C(=O)CCc2ccnn2C)CC(C)N1C(c1ccc(O)nc1)=O C1(CCOC)CCN(C(C2CCN2C(=O)CN(C2CCC2)C)=O)C1 Cc1cc(C)c(SCC=O)c(C)c1.c1(N(CC)CCO)nnc([Si](C)(C)C)s1.N Cn1cc2c(n1)CCC(C(=O)NCc1ccc(C(=O)NCC(O)CO)cc1)C2 C1CC2(C1)CCC2.C1(OC)CC(C=O)N(C(C)=O)C1.C1(C=O)CC(C#N)C1 C=C1CC(C(=O)NCCc2ccccc2)(CNC(c2cnc(Cl)s2)=O)C1 c1(SC)ccc(NC(N2CCCC2(C)C(=O)Nc2ccc(O)cn2)=O)cc1 Cc1nc(CC(C)C)oc1C(=O)NC1CC(CO)N(C(C2CC3CCC2C3)=O)C1 c1(CNC(COCCCOC)=O)nnn(C)c1C=O.C1(CCC)CCCCO1 c1(CC(C)C(=O)NCCCC2CC2)cccc(F)c1.C1(CC=O)CCOC1=O.N N1(C(C(CCCOC)C)=O)CCC(NC(=O)COc2ccc(Cl)cc2)C(C)(C)C1 C1(NC(CCOCC#C)=O)CN(C(c2nn(C)cc2[N+](=O)[O-])=O)CC(C)(C)C1 C(=O)(C(O)C(C)(C)CC)NC1C=CCN(C(c2c(CC)nccc2)=O)C1 c1(OC)cccnc1C(=O)NC1CC1NC(=O)C(C)Cc1ccccc1 Cc1cccc(C(N2CC(O)CCC2C(N2CC(NC(=O)C3CC3)C2)=O)=O)c1C C1(C(NOCC(=O)NC2(CC#C)CC2)=O)CC(C)CO1 N1(C(CCC2(C)CC2)=O)CC(CNC(C2CCCCC2(C)C)=O)C2(CC2)C1 N#Cc1cc(C(=O)NCC2CC2)ccc1[N+](=O)[O-].C(c1cc[nH]n1)=CC=O.C N(C1CCCc2occc21)C(C1CC2(CN(C(C(CC)CC)=O)C2)OC1)=O Cc1cccc(C2CCN(C(=O)NC(c3ccc(F)cc3)C(F)F)C2CO)c1 Cc1ncc(Br)c(N2CCC(C(=O)OCc3ccc(C4CCC4)cc3)C2)n1 N1(C(CCOC(CC(C)C)C)=O)CCCCC1CCN(C)C(c1cccnn1)=O C1(CN(C)C(C2(C)COC2)=O)CCC(CNC(=O)CC2CC2C)CC1 CC#CCC(CO)NC(=O)CN(CCC)C(C1CC(F)(F)C1)=O C1(C(=O)Nc2c(C)nsc2)C(C2CC2)CCN1C(=O)Cc1cncs1 N1(C(c2csc(C)n2)C(=O)NCC=C)CCC(O)(Cc2ccc(C)cc2)C1 c1(OC)cc(C(=O)NC2CCN(CC3CCC3)CC2)ncc1C C=CCC(CC)C(=O)NCCN(C)C(c1cn(C2CCOCC2)cn1)=O C#CC1(O)CC(C(N2CCCC2CNC(C2CCCCN2C2CCCC2)=O)=O)C1 C=CCC(CC)C(=O)NCC(CC(C)C)NC(=O)Cn1cc(C(=O)OC)nn1 C1(NC(Cn2[nH]c(=N)c(Br)c2)=O)CN(C(=O)Cc2csnn2)CC1C1CC1 C=CC(C)(CC)C(=O)NC1CC(NC(C2(C)COC(C)CO2)=O)C1 CC(Cn1ccnc1)C(=O)NCC(CNC(C1CC(C)(C)C1)=O)CO CC1CCN(C(=O)CCCNC(C2C3CCC(C3)C2C)=O)CC1CO N1(C(C(C#N)C2CC2)=O)CCOC2(C1)CN(C(c1cc(Cl)cnc1O)=O)C2 N1(C(CNC(C)=O)=O)CCCC(F)(F)C1.c1(C(=O)N)ccccc1C1(C)CC1 C1(OC)CCCC(C(=O)N(CC(=O)NCc2cccnc2C)CC(C)C)C1 CC1CCN(C(C2CCCC(=O)N2C)=O)CC1CNC(c1ccnnc1Cl)=O c1(C(=O)NCCOCCCN(C(=O)C)C)ccc2occc2c1.c1nccn1C Cc1nc(C)c(C(=O)N(CCCN(C(=O)C(C)(C)C(C)O)C)C)c(C)n1 CCCC(CCCO)C(=O)N1CCC2(C1)CN(C(=O)CCc1ccnc(Cl)c1)C2 C=C(C)C1OCCCC1C(=O)NCC1CCCN(C(c2coc(C(F)F)c2)=O)C1 CS(=O)(=O)c1cc(C(=O)NCC(C)CO)co1.C1(C=O)(C(N)=O)CCC1.N N1(C(CC=C=C)=O)CC2OCC(NC(c3cc(C)ncc3C)=O)C2C1 C1(NC(c2nc(C)oc2)=O)CN(c2ncc(Cl)cn2)CCC12CCOCC2 CC1Cc2cccc(CO)c2N1C(=O)NC1(C)CC(C)(C)OC1=O c1(C(=O)NCC(CNC(C2CCCN(CC)C2)=O)(C)C)ccc(C)cc1S c1(C(C(=O)NCC2CN(C(C(C)C)=O)C2)(C)C)ccc(N)cc1 C12(C(=O)Nc3ccccc3)CCN(CC1)S(=O)(=O)C2.C(=O)C(F)n1cccn1 C12(C(N3CCC(N(C(CCC(C)C)=O)C)CC3)=O)CC(CO)(C1)OC2C C(=O)(CCCC(C)(C)C)NC1C(OC)CN(C(c2ccc(OC)cc2Cl)=O)C1 c1(C(=O)NCC(C(C)C)NC(c2cnc(C)nc2O)=O)cccc2cnsc12 c1(OC)ccc(CCC(N2CCC(NC(=O)CCF)C2(C)C)=O)cc1C CCC(Cc1ccccc1)C(=O)NCC(O)CN(C(=O)Cc1ccc(F)cn1)C N1(C(c2nc(NC(C)=O)sc2)=O)CCC2(CCCCC2NC(=O)C2=CCCC2)C1 c1(C(=O)OCC2CCC(=O)O2)ccc2nc(-c3ccccc3)[nH]c2n1 Cc1cc(C(=O)NC2(C)CCN(C(=O)CCC(=O)N(C)C(C)C)CC2)cc(O)n1 Cc1cc(C=CC(N2CC3CC3(NC(C3CC(C#N)C3)=O)C2)=O)ccc1Br CC1(F)COCCN(CCCc2cn(CCCC(=O)NO)nn2)C1 N1(C(C(C2CCN(C(C3CCCN3C3COC3)=O)C2)C)=O)CCCCC1 c1(NC(c2ccc(SCCCC)o2)=O)ccnc(-n2nccn2)c1 c1(C(=O)NCC(n2cc(CCN(CC)CC)nn2)C)cc(C)cc(Br)c1 Cc1oc(CO)cc1C(=O)NCCN1CCC(NC(c2ccc(Cl)nn2)=O)CC1 C1(O)CCN(C(=O)C)C1.c1ccc(F)cc1.C1(CC(=O)N)(NC(C)=O)CC1 C12(CCCCC1)CC(=O)N2.c1(CNC(C2CC2(Cl)Cl)=O)ncsn1 CCCCCC(C)(C)C(=O)NCC(C)(O)CNC(=O)C=Cc1ccccc1 N1(C(C(C2CCOCC2)C)=O)CCCC2(NC(=O)CCc3cnc(O)[nH]3)CCCC12 Cc1ccc(C2CC(NC(c3ccn(C4CCC4)n3)c3nnnn3C)C2)s1 C1(C(=O)NC(CCNC(C(C=CC)O)=O)(C)C)CCN(S(=O)(=O)NC)CC1 S(=O)(=O)(c1ccc(Br)cc1)N(C)CCF.C1CC2CS(=O)(=O)CC2C1.C(=O)N C(N=c1[nH]c(=N)[nH]c(=NCC2CC23CCOCC3)[nH]1)c1cc(C)n(C)n1 CCC(CN(C)C)C(=O)NCCCNC(C1(OC)CCOC1)=O N1(C(C2N(C(c3c(C)ccc(C)c3)=O)CC=C2)=O)CCOCC2(CCC2)C1 N1(CCNC(C(CCSC)O)=O)CCCN(C(C2CC(F)C2)=O)CC1 C(CC)(CC)(CC)NC(C1N(CCC)CCC1)=O.c1(C2C(C=O)C2)ccco1.N C1(NC(c2c(C)nccc2)=O)CCC2(CC1)CN(C(=O)C(F)CC1CCC1)C2 C1(NC(c2ccc(C3CC3)cn2)=O)CN(C(=O)Cc2cccc(F)c2)CC12CC2 C(c1ccc(Cl)nc1)=CC(N1CCC1)=O.CC(C(=O)NC)OCC1CC1 N1(C(CSCC(=O)OC)=O)CC2CCCCC2C1.c1(C=O)cc(O)nc(Cl)c1.N C#CCC(O)C(=O)NC1CC(NC(c2ccn(C)n2)=O)C(O)C1 CC1CCc2[nH]nc(C(=O)NCC3CN(C(c4nc(Cl)cs4)=O)CCN3C)c2C1 c1(C(N2C(CNC(=O)CC3(C(F)(F)F)CC3)CCC2)=O)cccn(O)c1=O n1(CCC)cc(CNC(C2CN(CC(F)(F)F)C2)=O)nn1.C1(C=O)CC1F c1(C(=O)NCCCN(C(C(CCC)O)=O)CCO)ccc(F)cc1C(F)F C1(C(N2CCC(N(C)C)C2)=O)CC(C)(C)CCN1C(=O)C(F)C1CCC1 CC(C)CC(C(=O)NC1CCC(C)CC1)N(C)C.C1(C=O)CCS(=O)(=O)N1.N c1(C(=O)N)cc(F)c(C#N)cc1F.C1(NC(C2(C)CC2)=O)CS(=O)(=O)CC1 C1(C(=O)NCC(=O)N(C(CNC(C2C(CC)C2)=O)C)C)CCCC1 c1(C(=O)NC(CCCC)CNC(C2CC(C)=NO2)=O)ccnc2c1nnn2C c1(C(C)=O)cnccc1C(=O)NCC1CCN1C(C1CCC(O)C1)=O CC1CC(C)CN(C(=O)C(C)(C)c2ccsc2)C1.c1(C(=O)N)ccc([N+](=O)[O-])[nH]1 Cc1cn2cc(C(=O)NC(CC)C(C)C)nc2s1.C1(C(=O)N)(C(F)F)CCCC1 C1(N(C(C2CN(CC(C)C)C2)=O)C)CN(C(=O)Cc2cnn(C)c2C)CC1(C)C c1(CC)ccc(C(=O)N(c2c(C)cccc2C)C)cc1Nc1ccc(Cl)cc1 N1(C(CN(C(COC)=O)C)=O)CC2(CC(CC(N3C4CCC3CC4)=O)C2)C1 C1(O)(C(=O)NCC(C2CCN(C(=O)CNc3cccnc3)CC2)C)CCOCC1 c1(C(=O)NCC(CC)NC(=O)CCC(C)OC)c(N)cc(OC)cc1F C12(CNC(c3coc(Cl)n3)=O)CC(CO1)N(C(c1cnc(Br)s1)=O)C2 O(NC(=O)CC(C(F)(F)F)NC(=O)CC1CCC(=O)N1C)CCC C=CCC(C)(C)CC(c1nnnn1-c1ccccc1)NC1CC(CCOC)C1 C(C1CCCc2c(Br)cccc21)NC(=O)NC(c1c(C)c(Br)ccc1)C C12(NCc3cn(C)nc3)CCCC1CS(=O)(=O)C2 N1(C(C(CSC)C)=O)CCCCC(CNC(=O)Cc2cc(F)ccc2F)C1 C1(O)(CCNC(CC2CC(CC)C2)=O)CN(C(=O)CCCOC(C)C)C1 C1(C(=O)NCc2n(C)ccn2)CN(C(C2CCC(=O)C2)=O)CC1C(F)F c1(N(C2CC3CNC2C3)C(c2nccs2)=O)cnc2ccccc2c1 O=C(C1=NOC2(CCOC2)C1)NC1CCCC(NC(C2(Cl)CC23CCC3)=O)C1 Cc1cc(C(=O)NCC2CCCN(C(C34COC(CCO3)C4)=O)CC2)nc(C)n1 N1(C(C(c2ccc(C)cc2)(F)F)=O)CCC2(C1)CN(C(=O)CN(C)C)CCO2 CN1CCC2(CCN(C(=O)CC3CCN(C(C4C5CNCC45)=O)C3)CC2)CC1 C(c1ccc(F)cc1)=C(C=O)C.C(=O)(CCC(=O)NC1CCCCC1)NCC.N C1(C(N2CC(NC(c3ccc(CC)o3)=O)(CO)C2)=O)CCC(N(C)C)CC1 C1(C(=O)NCCC)CC=CC(NC(=O)CCC(=O)C2CC2)C1 N1(C(C(=O)N(CC#C)CCF)=O)CCCCC12CCCC2 CC(C)(C(=O)N1CCC(CCNC(=O)CS)C1)C1CCCO1.c1cccnc1.C c1(C(N(CCN(C(=O)C(C)(F)C(F)(F)F)C)C)=O)cc(Cl)c(O)c(Cl)c1 c1(C(=O)NCC2(NC(C(C)C3CCCO3)=O)CC2)ncc(C#N)cc1Cl N1(C(CCCCNC(C2(C#N)C(C)C2)=O)=O)CC2C(C1)C2(C)C Cc1[nH][nH]c(=NC(=O)C2CC(O)CN2C(=O)CCC(=O)OC(C)(C)C)c1Br C(=O)(C1=CCCN(C(C2CN(C)CCN2C)=O)C1)NC(CC(=O)OC)C1CC1 C1(NC(CCc2c(C)noc2Cl)=O)CCN(C(=O)Cc2nc(CN)cs2)C1(C)C C1(NC(C(N2CCC(N(C(c3n(CC)ncc3)=O)C)C2)C)=O)CCCCC1C Cc1c(C(=O)NCCNC(C2CC(O)CN2C)=O)nc2sccn12 C1(C(=O)NCCC2N(C(c3nc(C)nn3C)=O)CCC2)CCC2CC(C)CN2C1 C1(NC(CC(C)SC)=O)C2CC(O)C1N(C(c1ccncc1F)=O)C2 c1(C(NNC(=O)NCC23OCC(C)(NC2)C3)=O)ccc2c(c1)CCO2 [N-]=[N+]=NCCCCCC(=O)N1CC2CC1C2C(=O)NC1CC(O)(CO)C1 N1(C(C2(C#N)CCOC2)=O)CC(CO)C2(C1)CN(C(=O)C=CSc1nc[nH]n1)C2 C1(NC(c2c(C)n(CC(F)F)nc2)=O)CCN(C(C2CCCO2)=O)CCC1CO C=C(Cl)CC(C(=O)N1CCOC(CC(C)C)C1)NC(=O)C(CN(C)C)CC S(=O)(=O)(c1ccc(NC2CCN(CC3CC3)CC2)c(F)c1)NC1C(C)CC1 C1(CC(=O)NCCC(N)=O)C2CCCC2N1C(=O)C.C1CCOC1.C(=O)C n1(CC)ncnc1C(C)NC(C1(C)CC1)=O.C(c1nccs1)=CC=O.N N1(C(C2C(C)(C)CCN(C(C3(F)CC=CCC3)=O)C2)=O)CCC(O)(C2CC2)CC1 CCCC(C(=O)N1CC2(CCN(CC(C)OC)C2)C1)C(C)C C(C(C)C(F)C(=O)NC(C(N)=O)C(C)CC)NC(CCC#CC)=O C1(CNC(c2ccc(CC)s2)=O)CCN(C(c2ccnc(C(N)=O)c2)=O)C1 c1(C(N2CCCCC2)=O)cc(C)cc2nc[nH]c12.C(=O)(C(C)(F)C(=O)NC)OC C(CNC(C1CN(C)CCO1)=O)(C(C)(C)C)NC(COCCC#C)=O C1(NC(CC(CC)(C)C)=O)CN(C(c2ccc(O)cn2)=O)C2CCCC12 Cn1cc(S(C)(=O)=O)c(C(N2CC3C(NC(=O)C(O)C4CC4)C3C2)=O)n1 C1(C(=O)NCC2(N(C)C)CC2)CN(S(N)(=O)=O)C1 c1(C(=O)NC2CCN(C(C3C(=C)CC3)=O)CC2C)cc2c(cnn2C)nc1O C(=O)(CC(C)CC(C)(C)C)N(C1CCCN(C(CCC#CC)=O)C1)CC N1(CC(N2CCC(C)CC2)=O)C(=O)NC(C)(C)C1=O.C1(CC=O)CC1.COC N1(C(c2c(C)cc[nH]2)=O)CCN(C(=O)COCc2nc[nH]n2)C2CCCCC2C1 c1(CC(=O)OC)cn(CCCCN2CCC(N3CC=CC3)C2)nn1 C1(CCC)(Cc2ccc(C)cc2)CCCN1C(=O)NCCCSC N1(C(c2c(C)n[nH]c2)=O)CCC2(CCCN(C(c3ccc(F)c(I)c3)=O)C2)CC1 C(=O)(C(COC)N=[N+]=[N-])N1C(CCC#C)CCC1.C(=O)(CC(C)O)N(CC)CC N1(CCNC(CNC(CC)=O)=O)CCN(C(C2(OC)CCCC2)=O)CC12CCC2 CC(C)C(O)(C(=O)OCC=Cc1ccc(-c2ccccc2F)o1)C(F)(F)F N1(C(CCN(CC#C)C(C2CC(F)C(=O)N2)=O)=O)CCC(F)(F)CC1 Cc1c(C(N2CCCC(CNC(=O)C(C)S(C)(=O)=O)C2)=O)cccc1N C(c1ccco1)=C(C)C(=O)N(CCC(=O)NCC1CC(CF)C1)C C(=O)(C#CC1CCOC1)NC(C)CNC(=O)Cn1nnc(C2CC2)n1 C1(NC(=O)NCC2CCC(C(F)F)CC2)CCc2ncccc2C1 N1(C(C(C)C2CC2)=O)CCCC(N=c2nc3[nH][nH]cc-3c(O)n2)CC1 Cc1nc2n(n1)CCN(C(=O)C1=CCCN(C(=O)CN3CCC(C)C3)C1)C2 c1(C(N(CC(CO)CO)C)=O)cc(S(C)(=O)=O)oc1C.C#CCCOCC=O CC(C)CC(C(=O)N1CCOC(CF)C1)ONC(C1(C)CC(C#N)C1)=O C1(C#N)(C(N2CC(NC(C(C)OC3CCCC3)=O)C(C)(C)C2)=O)CC12CCCC2 C(=O)(C(C)CC(C)CC(C)C)NCCN(C(=O)C=Cc1cn[nH]c1)CCC C(=O)(CC(O)CC(C)(C)C)NCCN(C(=O)CC(O)CCCCC)CCCCCC C1(C=O)C2Cc3cc(Cl)ccc3C12.C(=O)(CCC1(C)CC1)N(CCC)CC.N CC1CC(NC(=O)CC2CCC2)CN1C(c1nnn(C)n1)=O c1(C(N2CCC(O)(C(C)NC(c3nccn3C)=O)C2)=O)cc2c(Cl)cccc2s1 c1(N2CC3CN(Cc4n(C)ncc4Br)C3C2)ncnc2c(Br)c[nH]c12 N1(C(c2cc(C)nc(O)c2)=O)C2CCC(C(N3CCC3(C)C)=O)C1CC2 Cc1cncnc1C(=O)NC1(C(=O)NC(c2cn[nH]c2)C)CCN(C)C1 N1(C(CCCn2c(C)nc(C)n2)=O)CC(NC(=O)CCc2nncs2)CC(O)C1 C1(C)(CC)CCC(C(N2CC(C)C2)=O)O1.c1(C(=O)N)ccc(C(F)F)nc1 c1(C(N2CCC(Cc3ncc(C)o3)CC2)C(=O)NCCCC)ccc([N+](=O)[O-])s1 C=C(C)C1OCCCC1N(C(=O)CCC(CC)OCCCOCC)CCOC C(=O)(CCCC(=O)N1CCCCC1Cn1cc(C(C2CCCCC2)C)nn1)NC N1(C(C2C(C)(C)CCO2)=O)CCCCC(NC(=O)C2=CCSC2)C1 C1(NC(CC(CC)(F)F)=O)CC(C(=O)N2CC3(C2)CN(C)C3)=CC1O c1(C(=O)NCCC(C)(C)NC(C2CCN(C)C2=O)=O)cc(O)nc2c1CCCN2 c1(-c2c(OC)ncc(OC)c2)ccc(C(=O)NCC(C)O)c2ccccc12 C(C(C(C)(C)C)NC(=O)CCc1ccc(Br)s1)NC(c1cnn(C)n1)=O Cc1[nH]c(C(C)(C)C)cc1C(=O)NC1CCN(C(C2C3CNC(=O)C23)=O)C1C N1(CC(C(C)N)(C)C)CCN(c2ncccc2F)CC1 C(CC(C)CC)(C(=O)N)NC(COC1(C#C)COC1)=O.C1(C)NC(=O)NC1=O C=CCCCCCCCCC(=O)NC(CO)CCCCNC(=O)C(F)=CC1CC1 c1(C(NNC(=O)N(CC)Cc2ccc(F)cc2F)=O)ccc(C(F)(F)F)c(O)n1 c1(C(=O)NCC2N(C)CCN(C(=O)C3=NOCC3)C2)cnc2cnc(Cl)cc2c1 C1(C)(C(=O)NC2(C(N(CC(C)O)C)=O)CCCC2)CCC(=O)NC1 CCS(=O)(=O)C=CC(=O)N1CCCC1C(C)(C)CNC(=O)C.CC(N)=O.S C1(COC)(NC(=O)C2=CCCC2C)CCCN(C(c2cnc(O)cc2O)=O)C1 C1(C(N2CCCC(CCC(C)C)C2)=O)OCC2CCCC1C2 CC1(C)CC(NC(=O)C2=COCCC2)CN1C(c1cnnc(O)c1)=O N1(C(CN(C(=O)OC)C)=O)CC(NC(=O)C(C)(C)C2CCCCC2)CC1C CC1Oc2c(C(=O)NC3CC3CNC(=O)C(F)F)cccc2NC1=O CC(CN(C)C)CCC=O.c1(CC)n[nH]cc1C(=O)N(CC(F)F)CC(C)O.N C1(NC(C(C2CCCCCC2)C)=O)CC2CCC1N2C(=O)CCCC(N)=O Cc1cc(F)ncc1C(=O)N(CC(O)CN(C)C(C1CCCCC1C)=O)C C(CCCCC(=O)NC1CC1(C)C(F)F)NC(CCc1cc(C)on1)=O CCC(CC)CC(F)C(=O)NC12CC(C1)N(C(=O)CN(C)C)C2 c1(C(N(C(C(=O)N2C(C(=O)OC)CC2)(C)C2CC2)C)=O)cc2cc[nH]c2cn1 C#CC(CC1CCCC1)NC(=O)C=C(C)C.C(=O)(C(F)OC(F)(F)F)N N1(CC)CC(C(=O)NCC2C3CC2N(C(c2sc(C)nc2C)=O)C3)CCC1=O C(=O)(C#CC1CCOC1)N1CC(NC(CCOCC(C)C)=O)C(C)(C)C1 c1(NC(=O)Nc2c(SCC)cccc2)c(I)cc(F)c(F)c1F Cn1cc(C(N2CC(CCO)(NC(=O)C(O)C(F)(F)F)C2)=O)c(O)nc1=O N1(C(c2ncn(C)c2)=O)CCCC2(CCN(C(=O)CCc3ccsc3Cl)C2)C1 N1(C(C(C)(C)OCC)=O)CCCC(NC(=O)CN2CCCCC2)C(F)C1 C1(N(C(CC(C)(C)SC)=O)C)CC2CCC(C1)N2C(c1sc(C)c(C)c1C)=O C=C=CC(C)C(=O)N1CCCC(NC(=O)Cc2c(C)cnn2C)C1 c1(C(=O)N)cn2c(n1)CCC2.C#Cc1ccc(C(=O)NC(Cn2ccnn2)C)o1 Cc1ccc(C(C)(C)C(=O)NCC(CNC(C2CC=CC(O)C2)=O)CO)cc1 c1(CCC=O)ccc(F)nc1F.Cc1cnccc1OC1CCN(CCSC)CC1 C#CCCC(C(=O)N1CC(C)C(O)C1)NC(=O)C(C)C(F)F C1(NC(CCCc2ccc(C)s2)=O)CCN(C(=O)Cc2cnc[nH]2)C(C)C1 c1(C(=O)NCCC(C)NC(c2ncc(OC)cn2)=O)ccn(C)c(=O)c1O c1(C(=O)NC2CCN(C(C3(C#C)CCC3)=O)CC2CC)cc(Cl)cc(C)c1N N1(C(C(COC)(C)C)=O)CCC(O)(CN(C)C(C2CCC(O)C2)=O)CC1 C(=O)(C=C(Cl)Cl)NC1CC(C(C)NC(C2CC(Cl)(Cl)C2)=O)C1 C(CC(C)C)(C(=O)NCCC1CCCN1C)NC(c1c(CC)nns1)=O c1(C(N(C2CCN(C(=O)CCS)C2)CCC)=O)ccc(S(N)(=O)=O)c(F)c1 CC12CC(CN1C(=O)NC1(c3ccccc3Br)CCC1)C2 C1(F)(C(=O)NCCCOCC#C)CCN(C(=O)C(N2CCOCC2)C)C1 Cc1ccc(C(=O)NC2CC3C2CCN3C(c2cnn3c2CCC3)=O)c(C)n1 C(=O)(C1=NOC(C)(C)C1)NC1CC(CC(=O)N(C(C)CS(C)=O)C)C1 c1(C(N2CCC(C(F)(F)F)C2)C(=O)N)ccc(S(N)(=O)=O)cc1.CC(C)C N1(C(C(C)(C)C)=O)CCC(C)(CNC(C2CCCC2c2ccccc2)=O)C1 c1(C(N2CCC(C)(NC(COCc3cc(C)no3)=O)C2)=O)cc2[nH]ccc2s1 C1(CNC(C2C(C)CC2)=O)C2CCCC1N(C(=O)C=Cc1nccs1)C2 C#CCCN=C(NC1CCOCC1)NCC1CC1Cl c1(C(N2CC(O)(C(C)NC(=O)CCc3nccn3C)C2)=O)onc2ccccc12 C(C1CN(C(=O)C(C)(C)C2CC2)Cc2ccccc21)NC(C(c1cnn(C)c1)C)=O C#CC1CCCN(C(C2(NC(=O)C(C)CC(C)C)CC(F)(F)C2)=O)C1 C=C(C)C1OCCC1C(=O)NCC(CCC)C(=O)NCCC1CC1 C#CCC(C)(C)C(=O)NCC1CCCC1.C(=O)(C(C(C)C)NS(N)(=O)=O)N N1(C(c2cc(OC)no2)=O)CC(N=[N+]=[N-])CC1C(=O)N.C1CC(=C2CC2)C1 C(=O)(CCS(C)=O)NCCCCCN(C)C.c1ccccc1.C1C(=O)N1.C(=O)C.N N1(C(COCC=C)=O)CCC(NC(=O)CC2CCCOC2)C(F)C1 c1(CC(=O)NC2C3CCN(C(=O)COC)C23)ccccc1O.c1cccc(Cl)c1 N1(C(C(CC)CCOC)=O)CC(C)CN(C(=O)Cc2cnsc2)CC1C C(=O)(C(C)CCCC(C)C)NCC1(NC(COC(CC)(C)C)=O)CCCCC1 C(=O)(C1=CCCCC1)NC(C1(CNC(CCc2nnc(C)n2C)=O)CC1)C N1(C(Cc2c(C)nn(C)c2)=O)CCOCC(NC(C2(C)CC(F)C2)=O)C1 c1(C(=O)N)ccc([N+](=O)[O-])c(C)c1.C(CC(=O)N(C1CCCC1)CCC)=CC c1(C2N(CCC3(C)CCOC3)CCC2)ccc(F)cc1 c1(C(=O)NCC2C(CNC(c3cc(C)c(C)nn3)=O)C2)cccc2c1CCC2 N1(C(C(CC)(CC)CC)=O)CCCCC(C2CN(C(c3cc[nH]c(=N)c3)=O)C2)C1 N1(C(c2c(C)[nH]cc2)=O)CC2(C1)CN(C(=O)COCC1CCCOC1)C2 C=CC1(CC(N2CCC(CF)C2)=O)CN(C(=O)C(C)CN(C)C)C1 N1(C(C2C(C)(C)C2)=O)CCC(C)C(F)(F)C1.c1(CC(=O)N)cccc(Cl)c1Cl C(=O)(CCS(C)(=O)=O)N1C(CCN(C(=O)C=CC2CCOC2)C)CCCC1 c1(NC(C2CCCN(CCO)C2)=O)cc(O)cc(=O)o1.C1(O)(C)CN(C=O)C1 C1CC2(CO1)CN(C(=O)C=CC(F)(F)F)C2.c1(C=O)ccc2c(n1)CCC2.N C(=O)(C(C)CC(C)(C)C)NC.C1(=O)COCC(C)N1C c1(C=O)ccc(C(F)(F)F)c(F)c1.C1(CNC(C2C(C)C2)=O)CCCC1.N C1(C(N2C(C(C)(C)NC(=O)CS)CCC2)=O)CCCNS1(=O)=O.c1cscn1 CCCCS(=O)(=O)CC(=O)N1CCCC(C)(NC(=O)C(O)CC(C)(C)C)C1 c1(OC)cccc2c1CCC2Nc1cc(NCCN2CCNC(=O)C2)nc(C)n1 c1(NC(=O)CC2CCCO2)ccccn1.C12(CC1)N(C)C(=O)CNC2=O C1(Cn2cc(C3(C)CC3)nn2)C(C2CC2)CCN1C(=O)CCn1cncn1 C1(NC(CC(COC)C)=O)CN(C(c2ccc(CO)nc2)=O)C2(CCC2)C1 c1(C(=O)NCCSCC)c[nH]c2ncc(-c3cc4cc(OC)ccc4[nH]3)cc12 c1(C(=O)NC2(CC=C)CCN(C(=O)C(CCC)OCC)C2)cnc(SC)nc1O C1(N(C)C(c2ccns2)=O)CCCC(NC(c2ccn(C(F)(F)F)n2)=O)C1 C(C)(C1OCCc2ccccc21)NC(NCCOC)=NCc1ccc2sccc2c1 C1(CC(=O)NC(C2CCCC2)C#C)(OC)CN(C(=O)CCOC)C1 C(=O)(C1CCCn2cncc21)NCC(CNC(c1cc(C)cc(C)c1C)=O)(C)O C1(CNC(CC2(C)CCCO2)=O)CC2(CCC2)CN1C(c1cccc(N)c1F)=O S(=O)(=O)(c1cccc(C(=O)NCC2CC(O)CN2C)c1)NCC=C C(CC(C(C)C)NC(c1cc(C2CCOCC2)on1)=O)N(C(CCC#C)=O)C C(=O)(CC(O)CNC(=O)C1=CCCC1)N(C1C(C)C1)C c1(OC)ccc([N+](=O)[O-])c(N2CCCC(CO)(NC(c3cccnc3Cl)=O)C2)n1 n1(CC(=O)NCCCc2onc(C)n2)nc(O)ccc1=O Cc1ccc(C(=O)N(CC(CO)CO)C)cc1C(C)(C)C.C(=O)(C(F)C1CC1)N C12(NC(c3cc(F)ccc3Br)=O)CCC(CC1)N(C(C1CC1CF)=O)C2 O=C(C1c2c[nH]nc2CN1C(C1C2CC(=O)CC12)=O)Nc1cccc(CO)c1 N#Cc1ccc(C(=O)NCc2ccsc2C(=O)Nc2cnsc2)[nH]1 C(=O)(CC(F)(F)CC(=O)NC1CC(C)N(C(c2occc2Br)=O)C1)OC CC(CC(C)NC(C1SCCS1)=O)NC(c1ccnn1CC(F)(F)F)=O C1(N(C(C2CCC(CC)O2)=O)C)CCCN(C(c2c[nH]cc(F)c2=O)=O)CC1 C1(CCNC(COC(C)=O)=O)CCN(C(C2(F)CCCCC2)=O)C(C)C1 N1(C(c2c(C)ncnc2)=O)CCCC(C2CC2NC(=O)Cn2cnccc2=O)C1 c1(C(N2CC(C)CC(NC(CC(C)O)=O)C2)=O)ccc2c(c1)NC(=O)CS2 C(=O)(CC(F)(F)C(C)(F)F)NCC(CC)CC.C(=O)(CCC(C)C)N.C(C)=O C1(NC(C(C)N2CCC2)=O)CC2CC(NC(C3CC4CC4C3)=O)CC2C1 c1(C(N(CCNC(c2ncc(C)nc2)=O)CC)=O)ccc(Cl)c(Cl)c1C.CCO N1(C(CCOCCNC(c2c(C)cncc2C)=O)=O)CCC(F)(F)C(O)C1 C1(SC)CN(C(C2CCCO2)=O)CC1NC(c1cc(C2CC2)no1)=O CC1(C)CCN(C(=O)C=CCN2CCC2)C1C(N1CC2CCOC2C1)=O CCC(CC)CC(=O)NCCN1CCC(NC(c2ccncc2OC)=O)CC1 C1(C2CCN(C(c3cc(Cl)c(Br)[nH]3)=O)CC2)(OC)CCOCC1 c1(CN2C(CNCC3CCC(C)O3)CCC2)cc(Br)c[nH]c1=N Cc1ccccc1C=CC(=O)NC(CCF)C(=O)NC1CCCC12CC2 c1(CC)ccccc1C(=O)N(CCCCN(C)C(C1CC(C)OC1=O)=O)C c1(C(=O)O)c[nH]cc1C(=O)N(CCC)C(C)C.C(=O)CCN(C)C.CC N1(C(COC(CC)(C)C)=O)CCN(C(c2cscc2C)=O)C(CF)C1 N1(C(C(C)OCCOC)=O)CCCC(CCC(N2CCCCC2CCO)=O)C1 c1(C(c2n(CCC)nnn2)NCCNC(=O)C2CC2)ccnc(CC)c1 c1(NC)c(C(=O)N(C(C)CNC(C2CCSC2)=O)C)cccc1N c1(C(=O)NCCC2(O)CN(C(c3c(Cl)ccc(C)c3)=O)C2)cnc2[nH]nnc2c1 N1(C(CCCN(C(C)C)C)=O)CCN(C(=O)CC2CS(=O)(=O)C2)C(C2CCC2)C1 N#Cc1[nH]c(=NCC2CCCCN(C(=O)CCOc3ccccc3F)C2)sc1Cl c1(CC)onc(C)c1C(=O)N(C(C)CNC(C1(O)CC(C)(C)C1)=O)C Cc1sc(C(=O)N(C2CCCN(C(=O)C(O)CC(F)(F)F)C2)C)cc1[N+](=O)[O-] N(C1CN(C(=O)CCCC2CC2)Cc2ccccc21)C(C(C(C)C)O)=O c1(C(C(=O)N(CC(C)N(C)C(C2C=CC=CC=C2)=O)C)O)cccc(N)c1 C1(C(=O)NC(C2CCCC2)CNC(Cn2nnc(C)n2)=O)OCCOC1C C12(C(=O)NCC3CCC3CO)CCC(CC1)N(C(C1CCC(O)CC1)=O)C2 Cc1cc(C2CC2)cnc1C(=O)NC(C)CC(C)C.c1(C=O)ccc(=N)[nH]c1.N Cc1cc(C(=O)NCCC(N2CCc3ccsc3C2)=O)nc(C)c1 C(=O)(CS(=O)(=O)CC(=O)NC(CNC(C1CCSCC1)=O)CC(C)C)OC C1(C(=O)NC2(CF)CCN(C(=O)CC(F)F)C2)CCC(F)(F)CO1 c1(C(=O)NCCC2CN(C(=O)CCn3cccn3)CCO2)ccc(CO)c(Cl)c1 c1(N2C(=O)CC(C=O)C2)cccc([N+](=O)[O-])c1.C1(CC(=O)OC)CCCC1.C C1(C(N2CC=CC(NC(CN(C3CC3)CC)=O)C2)=O)CCc2nc(C)[nH]c2C1 c1(CC)cc(Cl)cc(F)c1CN1CCC(O)CC1C(=O)OC c1(CC(=O)N(CCCCNC(C2(C)CCN(C)C2)=O)C)cc(F)ccc1F c1(OC)cc(-c2cscc2C(=O)Nc2cc(O)nc(C)n2)cc(F)c1CO c1(C(N2CCN(Cc3ccc(CCC)cc3)CC2C)=O)cc([N+](=O)[O-])ccc1O c1(OC)ccc(C(N2CCC(CN(C)C(C3CC4(CCC4)C3)=O)CC2)=O)nc1 C=C(C)CCCC(=O)NC1CN(C(C2C(C)(C)C2(F)F)=O)CC12CC2 N1(C(C2C(C(=O)OC)CC2)=O)CC2CCC1C(NC(C1COCCN1C)=O)C2 N1(C(C2N(CC)C(=O)CC2)=O)CCCCCC(NC(c2coc(O)n2)=O)C1 c1(C(=O)NC(CC#C)C(=O)NC(C)C(=O)N(C)CC)cccc2c1CCC2 CC1(C)Cc2cccc(CC(=O)NC3(C)CCN(C(=O)CCC(F)F)C3)c2O1 c1(C(N2CC(N(C(C3C(C#C)C3)=O)C)C3(C2)CC3)=O)nc(SC)n2ccccc12 C#CC1(C(=O)NOCCCOC)CCN(C(=O)CCC(C)CC)CC1 CC1CN(C(=O)Cc2cnn(C)c2)CC1NC(=O)C(N1CCSCC1)C Cc1c[nH]cc1C(=O)NCC1C(C(=O)NCCC2C=CCC2)C1(C)C N1(C(C2C(CC)C2)=O)CC2CCC(C)(C2)C1.C(c1cncnc1)=CC=O.N c1(OC)c(C(=O)NC2CCCC(C(=O)NCC3COCC3(C)C)C2)cnn1C c1(C(=O)NC2CCCCCN(C(=O)C3CC3)C2)nnc2ccccc2c1O C1(S(C)(=O)=O)(C=O)CC(O)C1.Cc1nn(CC(=O)NCCCCC)c(=O)o1.N CC1CCCCC1C(N1CCCC(CNC(C2CN(C3CCOC3)C2)=O)C1)=O Cc1ccc(F)c(C(=O)NC2CC(C)(NC(C3CCCC3C(C)C)=O)C2)c1Cl C(=O)(CCCCC(F)(F)F)NCC1(C)C(C)CN(C(c2ccc(=N)[nH]n2)=O)C1 c1(CCNC2(c3nnnn3C3CC(F)(F)C3)CCC(CC)C2)ccc(Br)cc1F c1(C(N2CCCC(N(C(=O)Cc3cccs3)C)CC2)=O)ccc2nnc(S)n2c1 c1(C(=O)NC(C2(O)CCN(C(=O)CC3CC3(C)C)C2)C)cccc(Cl)c1Cl N(C(=NCCCn1cnnn1)NCc1cnc(C)cn1)CC(=C)C c1(-c2cccc(CC#N)c2F)cccc2cc(C(N3CC4C(C3)C4(F)F)=O)[nH]c12 N1(C(C(C(C)C)OCC)=O)CCN(C)CC1.C(=O)C(C)(C)n1ccc(C)n1.C N1(C(C(c2ccc(C)cc2)=O)=O)CCN(C(C2CC(n3cnnc3)C2)=O)C(C)C1 Cc1cc2c(cc1C)C(C(=O)NCCC(C)N(C(=O)CCc1cc[nH]n1)C)CO2 C1(C(N2C(CNC(C(C)CC3CCC3)=O)CC2)=O)CCCC(O)C1 N1(C(C(C)C#N)=O)CCC2CN(C(=O)C(=O)Nc3ccc(Cl)cc3)CCC12 N1(C(c2c(C)con2)=O)CC2CC1CN2C(c1cccc(CC#N)c1)=O C(N=c1[nH]c(C)cc(=NC2CCC2OC(C)C)[nH]1)c1ccc(OC)cc1OC C(=O)(CCCCCNC(C1CCOC(CC)C1)=O)NC1CC(=C)C1 c1(OC)nc(C)ncc1C(=O)N.C12(C(N(CC)C3CC3)=O)CCCN1CCC2 C(=O)(C1CCc2ccccc21)N1CCC(CNC(c2cc(C3CC3)ns2)=O)C1 c1(C=O)cc(N(C)C)ccc1C.C1(NC(C2(COCC)CC2)=O)CCC1 C(=O)(C(C)CS(C)(=O)=O)NCCC.c1(C(C(=O)N)(C)C)ccc(Cl)c(Cl)c1 Cc1c(C(=O)NC2(C)CCN(C(=O)C3=COCCC3)C2)[nH]c2c1C(=O)CCC2 C1(C(N(CC(C)NC(=O)CC)C)=O)CC(S(C)(=O)=O)C1.c1ccc(F)cc1 C1(CNC(CCn2c(C)cc(C)n2)=O)CN(C(c2sncc2C)=O)CCC1C C1(CC)CC2(CCN2C(C2CC23CCN(C(C2(COC)CCC2)=O)C3)=O)C1 Cc1cc2c(C(N3CCC(NC(C4CC4CF)=O)C3)=O)cccc2o1 C1(CC(=O)NCCN(CCC)CC)(NC(C2CC2C)=O)CCCC1 C1(OC)CN(C(C2CCC=CCC2)=O)CCC1NC(c1nnsc1C)=O N1(C(c2c(OC)csc2)=O)CCN(C(=O)Cc2nnc(S)n2C)C(CF)C1 C1(C)(NC(c2c(CC)nc[nH]2)=O)CCN(Cc2cccc(COC)c2)C1 C(=O)(C(O)C1=CCCCC1)NCC1N(C)CCN(C(CCn2ncc(C)c2)=O)C1 S(=O)(=O)(c1cccc(Br)c1)N1C(C(=O)OC)CCC1.C1(=O)C(OC)CCN1 Cc1sccc1NC(=O)CCNC(=O)C(C)(C)N1CCCC1 Nc1c(C(=O)N)cc(Cl)cc1F.C12CC(C1)C2.c1(C=O)ccn(C(F)(F)F)n1 N#Cc1ccc2c(c1)C(NC(=O)NNC(=O)c1sccc1C)CCO2 n1(CCCOC)nc(C(=O)NC2CCCN(CC3CCCO3)C2)ccc1=O C(=O)(C(O)C(F)(F)F)N1C(C(=O)NC(c2ncccn2)C)C2CC2C1 C1(C(N(C(C(=O)NCCC(C)C)(C)C2CC2)C)=O)CCC(=O)C(C)C1 c1(CNC(Cn2nnc(C)n2)=O)ccccc1CNC(C1(C)CCCC1O)=O O=C1CC(C(=O)NC2CCCCCC2(F)F)c2ccccc21 c1(C(=O)Nc2c(C)c(Cl)cc(F)c2)csc2c(Br)cccc12 C12(NC(CCN(CCC)C)=O)CC3CCC(C1C2)N3C(=O)CCC1CCC1 Cc1cc(C(=O)NCC2CC2C(C)(F)F)c(C)n1C1CCCCC1 Nc1ccc(C(=O)NC2CCCC2NC(=O)C=CC(=O)N)nc1Cl.C1CC1 c1(CC=C)cc(C)c(NC(=O)C(=O)NC(C)CN(C)C)cc1C c1(C(=O)N)cc2ncc(C(C)C)cc2[nH]1.C(C)(C(=O)N(CCC)C1CC1)OC N1(C(C=O)C)C(=O)c2ccc(C)cc2C1=O.C(C(=O)NC)OCC.C1CC1 C1(C(N2CCN(c3ccc(Cl)nn3)CC2)=O)CC2CC3CC(C2)CC1C3 CN1CC2CC1(C(=O)NC1(CCNC(=O)CN3CCCC3)CC1)C2 CCCCC(O)CC(=O)N1CCC(CCC(=O)NCCOc2cccnc2)C1 CCC(C)(CCNC(=O)C(C)n1ccnn1)NC(=O)CCCc1ccsc1 n1(CC)c(SCC(=O)N(C2CN(C(=O)C(C)(C)SC)C2)C)nc2ccccc12 n1(CCNC(C2C(C(C)(C)C)CC2)=O)cc(C(=O)NCCCN=[N+]=[N-])nn1 N1(C(C(COC2CC2)NC(CCSCC)=O)=O)CC(C#N)C2(CCC2)C1 C(C(CC(=O)N)C1CCC1)NC(C1(OCC)CC1)=O.C1CCCC1.N(C)C C(C(=O)N1CCN(CC(C)C)CC1)(C(C)(C)C)NC(C)=O.C1(C=O)CC(C)C1 c1(C(N2CC3CCN(C(C(C(C)C)(C)C)=O)CC32)=O)cc2c(s1)CCC(C)C2 C12(C(=O)NCCC3(C)CCCC3)CC1CCN2C(=O)C(O)Cn1cncn1 C(=O)(C1=CCCOCC1)NCC(CN(C)C(c1cc(C2CC2)nn1C)=O)O C1(COC)CN(C(C2CC2(F)F)=O)CCN1C(c1cc(C(F)(F)F)ns1)=O N1(C(c2cccc(C(C)C)n2)=O)CC(CNC(=O)CC2CCSC2)CC(C)C1 C12(NC(c3cnc(C)[nH]3)=O)CCCC1N(C(=O)CCC1OCCO1)CCC2 C1(O)(C(=O)NCC2(CO)COC2)CCN(c2nccc(-c3cnccn3)n2)C1 CC1OC2(CO)CC1(C(=O)NCC1(C)CCCN1C)C2 c1(C(N2CC(O)CC(NC(=O)C(=C3CCCCC3)F)C2)=O)onc2ccccc12 CCCCCCN(C(=O)CC1CCN1C(=O)C(CN(C)C)N(C)C)C CCC(CC(F)(F)F)C(=O)NC1CN(C(=O)CCC2CCC(=O)N2)CC1(C)C N1(C(c2c(C)nc(C3CC3)[nH]2)=O)CC2CCN(C(=O)C3=CCC(C)CC3)C2C1 c1(C(=O)NC2(C)CCC(NC(C3CCC3)=O)CC2)nc2ncc(Br)cc2[nH]1 O=C(CN=c1[nH]c2c(c(=NCC(Cl)Cl)[nH]1)CSC2)NC1CCCC1 c1(C(=O)NCCC(=C)CNC(c2cccnc2C)=O)ncncc1C#N NC(=O)CC(C(=O)NCC(F)C1CCC1)NC(c1sccc1F)=O c1(OC)cccc2c1CC(C(N1CCNC(CF)C1)=O)CO2 C1(C)(OCC(=O)NCCN(C(=O)C(C)(C)c2cccs2)C)CCCC1 c1(C(N2CC(CC)C2)=O)ccc2cccc(Cl)c2n1.C12(CC(=O)N)CC(C1)C2 c1(CNC(Cc2c(C)occ2)=O)nc2c(s1)CCN(C(=O)C(C)(C)N(C)C)C2 N1(C(c2c(C)n[nH]c2)=O)CC(C)C(C)(C)C1.c1(CC=O)ccn(C(F)F)n1.N C=CCC(C)(C)C(=O)N1CCCC1CN(C)C(c1cnn(CCN(C)C)c1)=O C1(COC)CN(C(C2CC(=O)NC(=O)N2)=O)CCN1C(=O)Cc1ccnnc1O CC(C)C(F)C(=O)N(C1CCC(NC(=O)CCn2ccnc2)CC1)C c1(C2(C(N(CCCC)C)=O)CCC2)ccc(F)cc1.C1(C)(CC)CC1C(=O)N N1(C(C2(F)C(C)OCC2)=O)CC(C(N2CC(N3CC(O)C3)C2)=O)CC(C)C1 c1(C(C)(C)C(=O)NCC(CO)NC(=O)CC2CCC2)ccc(Cl)c(Cl)c1 C1(NC(c2cccc(C#C)c2)=O)CC2CC(C1)N(C(c1cc(COC)cs1)=O)C2 N1(C(c2cscc2OC)C(=O)NCC=C)C(C(=O)O)CCC12CC2 N1(C(=O)CCC2CCCC2)CCOCC1CC(=O)NCC1(CO)CC2CC2C1 N1(C(N)=O)CC(O)CC1C(=O)NCCC1(C=O)CC1.C1CC(F)(F)C1.N C1(NC(=O)Nc2c(N3CC4C(C)C4C3)nccc2)CC(O)C(F)C1 C1(COC)CCN(C(C2(COC)C=CCN2C(=O)C)=O)CC1.C(C)=O.N n1(CCCC)nccc1C(=O)NCC(C)CNC(C1(N(C)C)CCCC1)=O O=C(CCS(=O)(=O)Cc1cccc(Br)c1)NCC(CO)NC(=O)CO C(=O)(N1CC(O)CCO1)C1N(C)CCN(C(=O)C(=O)C2CCCC2)C1 C(C(=O)N(C1CCC(C)CC1)C)(C(C)(C)C)OC.c1(C=O)conc1C1CC1 N1(C(c2c(NC)snc2C)=O)CCC(NC(c2ccc(CO)cn2)=O)C12CC2 C1(OC)CN(C(C2(NC(=O)C(C)CN(C)C)CC(F)(F)C2)=O)CC1F C1(C(=O)NC2(CNC(C(C)=Cn3ccnn3)=O)CC2)Cc2ccccc2C(=O)O1 C(=O)(C(=O)N=S(C)(C)=O)NCC1N(C(c2cnc(CC)o2)=O)CCC1C C(C(CO)(CO)NC(C1CC(F)(F)CS1)=O)N(C(=O)C1=NOCC1)C c1(CC)cccc(C(=O)NCC2CC(OC)CN2C(c2csc(C)c2)=O)c1F C1(=CC(=O)NCC2N(C(C(CSC)C)=O)CCN(C)C2)CCCCCC1(F)F N1(C(CCC(C)NC(C2CC3COCC3C2)=O)=O)CC(=O)N(C)C(=O)C1 c1(N2CCC(CNC(C3CC(F)C3)=O)CC2)nc(C(F)F)nc2[nH]ccc12 N1(C(c2n(CC)ncc2)=O)CCC(C2(O)CCN(C(=O)Cc3cncs3)C2)CC1 C1(CC(=O)Nc2ccc(C)cc2O)C2CCC1CN(C(c1cc(C)n(C)c1C)=O)C2 C1(NC(c2cccc(C3CC3)n2)=O)CCC(O)C1.C1(C=O)CC2(CC2)CO1.N Cc1cnc(C(=O)NC2CC(O)CN(C(c3cc4c(s3)CCC4)=O)C2)cc1C c1(CNC(C(CO)NC(c2ccc(CC)nc2)=O)=O)cc(C)cnc1F c1(NC(CC2CCN(C(Cc3cc(CC)no3)=O)CC2)=O)cc(F)cc(F)c1 C1(CNC(=O)C=Cc2cc[nH]n2)CCN(C(c2cnc(O)s2)=O)CCC1(F)F c1(C(=O)NCCOCCCN(C(=O)C)C)occc1C(F)F.CC(F)F N1(C(C2N(C(c3c(OC)nccn3)=O)CCCC2)=O)CCOC(C)(C2CC2)C1 S(=O)(=O)(c1cnc(N(CCCC)C)c(Cl)c1)NC(C)CC(C)(C)C.C(C)(C)C.O c1(N2CCOCC(NC(COc3cccc(CC)c3)=O)C2)nc(C)ccc1C#N CCC(CCC(=O)N1CCCC(N(C(=O)CN(C(=O)C(C)C)C)C)C1)OC C(=O)(CC(CNC(C1(CC2CC2)COC1)=O)OC)NC(COC)C C(C(CC(C)C)C(=O)NC(C(=O)NC1CC(O)C(O)C1)C(C)(C)C)OC C1(C(=O)N)CCCCS1(=O)=O.Cc1c(C(N2CCCC2C)=O)cnn1CC(F)F c1(CC)ccc(CN2CCCC(Cn3cc(C4(N(C)C)CCOC4)nn3)C2)cc1 c1(C2C(C(NCC)=O)C2)ccco1.C(=O)N(C)CC.C1CC1.CCS C(C)(C(C)C(C)C)NC(CCc1onc(C(C)OC)n1)=O.C(=O)C(C)(Cl)Cl.N C(C)(CCC(=O)NCc1occc1C(=O)NC1CC(C)C1)OCC N1(C(c2cnc(C)c(C)c2)C(=O)NCCC)CC2(CCC2)C1C1CCCO1 Cc1ccccc1OCCC(=O)NC1CCC(CNC(c2csnn2)=O)CC1 c1(C(=O)NC(C(=O)Nc2n(C)ncc2)Cc2ccccc2)ncccc1Cl c1(C(N2CCC(N(C(c3c(C)cn(C)n3)=O)C)CC2)=O)cc(=N)[nH]cc1Br C1(C(N(CCC)C)=O)CC(C)(C)OC(C)(C)C1.Cc1ccc(Cl)c(N)c1C=O.N c1(C(=O)NCCC2N(C(c3ccc(C#N)s3)=O)CCOC2)cc(Cl)ccc1Cl N1(C(c2c(CC)ncnc2)=O)CCCC(CCO)(CC)C1.C1(C=O)CCC(C)C1 C(=O)(CC1=CCN(C(c2ccco2)=O)CC1)NC(CC#C)C C1(C=O)CCS(=O)(=O)CC1.c1(CCC(N2CC(OC)C2)=O)c(C)noc1Cl.C C1(C(=O)Oc2c(C(=O)OC)cccc2OC)CCN(CC)CC1C N1(C(=O)Cc2cc[nH]n2)CCC(CCNC(C23CCCC2CC3)=O)CC1 N1(C(c2cc(OC)cc(F)c2)=O)C2CCC1CC(NC(C1CCN(C)C1)=O)C2 Cc1nc2cncc(C(=O)NCC3CC3C)c2[nH]1.c1cccnc1.C(=O)(C)N C1(NC(C=CSC)=O)CCOC12CCN(C(C1(c3cc[nH]n3)CC1)=O)CC2 CN1CCN(C(=O)CSC2CCOC2=O)C(C)C1.C(=O)(CC(O)CC1CC1)N N1(C(=O)NCCN(C2CC2)CC)C(C)CCCC1C c1(C(N(CC(=O)OCc2ccccc2)CC)=O)cc(Br)cnc1N N1(C(C(CC=C)CC=C)=O)CCOC2CN(C(=O)C(C)NC(=O)CC)CC12 S(=O)(=O)(c1cc(Cl)ccc1OCC1CCC1)N1CC#CC(C(=O)O)CC1 N1(c2c(Br)cnc(C)n2)CC2CCC(NC(c3ccc(CN(C)C)cc3)=O)C2C1 C(=O)(CCC(C)(C)NC(c1ccncc1)=O)NC(C1CSC1)C C1(C(N2C(CN(C)C(C3(C)CCCCO3)=O)CCC2)=O)CCC(CC#N)CC1 C1(CC#C)(C(N2CCC(OCCF)C2)=O)CCN(C(=O)Cn2cc(C)nn2)C1 N1(C(c2c(C)nc[nH]2)=O)CC(CO)C2(C1)CN(C(=O)CCC1CCC(=O)C1)C2 Cc1cc(I)ccc1NNC(=O)C1(CN)CCCS1(=O)=O c1(NC(CN(C(=O)CC2(C#N)CC2)CCC)=O)cn(CC)nn1 N1(C(C2C(CC)OCC2)=O)CCCC2(CCN(C(=O)C=CCF)CC2)C1 c1(CC)c[nH]cc1C(=O)NCCCN(C(=O)C=Cc1cnc[nH]1)CC c1(OC)oc(C)nc1C(=O)NCC(C)NC(=O)C(C)Sc1ncccn1 O=C(CCCC(F)(F)F)NC(C1CCOC1)CNC(c1n[nH]cc1Br)=O C(=O)(CCCC=O)NCC.C(C)CC(F)(F)F.C1(CC=O)NC(=O)NC1=O.N C(C(O)CN=c1ccnc(CO)[nH]1)NC(c1noc(C)c1C)=O C(=O)(C(CC(C)NC(=O)OC(C)(C)C)N1CC(C)C1(C)C)NCC.O c1(C(N(CC(=C)C)CC(=C)C)=O)ccc2c(n1)CN(C(=O)CCC(=C)Cl)CC2 C(=O)(C1CCc2scnc21)NCC1N(C(C(F)=C(C)C)=O)CC(C)(C)OC1 c1(C(=O)NCCC(C)N(C(CC(=C)I)=O)C)cc(C#N)c[nH]1 C1(CC)(CO)CN(C(=O)C(C)N(C)C(C2CCC2(OC)OC)=O)C1 N1(C(c2c(C)ncnc2O)=O)CCC2(CCC(NC(C3CC3(C)C)=O)C2)C1 CC(C)(C)CCC(=O)N(CC)C1CC1.C(=O)(C(C)(C)Cc1ccc(Br)cc1)N Cc1cc(C)c(NC(=O)C(CC(C)C)ONC(C2CN(C(C)C)C2)=O)cc1O c1(C(=O)NC2C(C)N(C(=O)C3=CC(C)(C)C3)CCC2)ccc2ccccc2c1O C12(NC(c3c(C)nn[nH]3)=O)CCCC1CN(C(c1cccn3cnnc13)=O)C2 c1(C(N2CCC(c3cc(C)[nH]n3)C2)C(=O)NCC(=C)C)ccc([Si](C)(C)C)s1 C1(CCNC(Cc2nc(C)[nH]n2)=O)CN(C(=O)CC=C(Cl)Cl)CCCO1 C#CC1CN(C(c2nccc3c[nH]nc23)=O)CCN1C(C1CC(C)C1)=O C#CCC(C)(CC)C(=O)NCCO.C(=O)(C(F)F)N(CC)C.c1cnn(C)c1 C(C(C)C(C)C(=O)N1CC(N(C)C(c2cn(-c3cccc(Cl)c3)nn2)=O)C1)OC C1(CNC(C(C)C(F)F)=O)CC2(C1)CN(C(=O)C(O)Cn1cncn1)C2 c1(C(N2CCN(C(CS(CC)=O)=O)C(CC(=O)NC)C2)=O)ccc2ncnn2c1 N1(C(COCCCOC)=O)CCC(C)CC1C.c1(C=O)ccc(C(C)=O)cn1 C1(CC)C(C(=O)NCCCC(=O)OC)CCN1C(=O)Cc1ccn(CC)n1 c1(C(=O)NCC(CO)NC(C2CC3CSCC(C2)C3)=O)cccc(Cl)c1[N+](=O)[O-] C(=O)(CC(COC)NC(C1CCS(=O)CC1)=O)NC(C#C)(C)C1CC1 Cc1ncc(C(=O)NCC2(F)CCN(C(C3CCCCN3C)=O)CC2)cc1N C1(NC(c2cnn(CC)n2)=O)(CF)CCN(C(c2scnc2C2CC2)=O)C1 C1(C(N2CCC(N(C)C(C3CCS(=O)(=O)N3)=O)CC2)=O)CCOCC1.CC=O.N C1(C(=O)NCCc2cncs2)CSCCN1C(C1C=CCC1)=O C12(C(N3CC(CCCCNC(C=C(COC)C)=O)C3)=O)CCCCC1C2(F)F c1(OC)ccc(F)c2[nH]c(C(=O)NC3CN(C(c4cc(N)nc(Cl)c4)=O)C3)cc12 C1(NC(c2cc(C)sn2)=O)CC2CN(C(=O)C(C)(C)C3CCCCO3)CC12 c12ccc(c([N+](=O)[O-])c1)c(=O)[nH]2.Cc1cnn(C2CCCCO2)c1-n1cccn1 c1(C(N2CC(NC(C=CC)=O)(CO)C2)=O)cccc(-c2ccncc2)n1 C(=O)(C(CC(C)C)NC(=O)C=CC(C)CC)NCC(CCC)C c1(CC(=O)NC2C(C)N(C(=O)C(F)=C3CCC3)CC2)nsc2ccccc12 c1(C(=O)NCCCC(=C)C)cc(Cl)c(F)c([N+](=O)[O-])c1N Cc1ccc(C(=O)N(C2CCCN(C(=O)C(F)(F)CC3CC3)C2)CCO)nc1C Cn1c(C(=O)NC2CC(NC(c3ccncn3)=O)C23CCC3)ccc1C#N c1(CCNC(c2ncc(CC)[nH]2)c2nnnn2CCSC)cc(C)cc(Cl)c1 c1(C(=O)NC2(CC3CC3)CCC2)cccn(Cc2ccc(F)cc2)c1=O C(CN=c1cc(C)nc(NC(c2csc(C)n2)C)[nH]1)N1CCCC(CC)C1 C1(NC(C(C)NC(C2CCCCC2)C)=O)CCN(c2cc(Cl)ncn2)C(C)C1 C1(CNC(C2Cc3cccnc3C2)=O)CCC2(CN(C(=O)C3=CCCOC3)C2)O1 C(C(CCC)C(=O)NCCC(O)C1CCC1)NC(CC1CC(CC)C1)=O C1(C#N)(C(N2CC(C)C(NC(=O)CC=CCc3ccccc3)C2)=O)CCCOC1 C(C(C)(O)C(=O)NCC1CC(Nc2cc(CC(=O)OC)ncn2)C1)OC C1(C(N2CCC(NC(CNC(C)=O)=O)C(C)(C)C2)=O)CC12CCc1ccccc12 C=C1CCC(C(N2CC(N3CCN(C(=O)C(C)CC4CC4)CC3)C2)=O)CC1 N1(C(C=C(C)C)=O)CC(NC(=O)CCCc2ccc(C)s2)CCC(O)C1 c1(C(C)(C)C)cc(N2CC=CC(NC(=O)C(C)n3cncn3)C2)ncn1 CCCC(C(=O)N(C)C)NC(=O)CCCCN(C)C(c1cnns1)=O C1(C(=O)OCc2nc(C(C)=O)sc2)CCC(=O)NC1 C1(NC(C(CCC)NC(=O)CSc2nc[nH]n2)=O)CC(C)N(C)CC1C CC(C)(C)C(C#N)C(=O)N1CC(F)CC1CNC(=O)C(F)=CCCF c1(CNC(CC)=O)ncccc1C(=O)N(C1CCCC1)CCO CCC(C)CN=c1[nH]ccc(=NCCCN(C(=O)OC(C)(C)C)CCOC)[nH]1 Cc1c(C(=O)NC(C)C(C)C)sc2nccn12.c1(C(=O)N)cc(C(N)=O)cs1 N1(C(CC(C)C(F)F)=O)CC2(COC(CNC(c3ccc(Cl)nc3Cl)=O)C2)C1 N1(C(=O)COc2ccsn2)CC2CCCCN2CC1CNC(=O)C(F)(F)C(F)F CCC(CC)(C(C)C)NC(C1CSCN1C(=O)CCCC1CCCO1)=O c1(C(=O)NCC(CC)NC(=O)C(C)CN(C)C)coc(-c2ccccn2)n1 N1(C(C2N(C=O)CCC2)=O)CC2CC1CCN2C(C1CCCCCCC1)=O C12(CNC(CCCNC(C)=O)=O)CN(C(c3cc(O)nn3C)=O)CC1CCO2 N1(C(=O)OC(C)(C)C)CC=CC1C(=O)N.C1(C=O)CCN(C)C1.C1CC1 C1(C(=O)NCC(C)NC(CC(C=C)(C)O)=O)CC(C(C)=NO)C1(C)C c1(OC)cnc2ccccc2c1C(N1CCC1CNC(=O)CC1CCCSC1)=O CN1CC2CC1CN2C(C1CCN(C(=O)CCc2ccc(O)c(O)c2)CC1O)=O c1(OC)ccc(C(=O)N(CC(O)CN(C)C(C2(C)CCCS2)=O)C)c(O)c1 c1(C(N2C(C(N3CCC(C(F)(F)F)C3)=O)CCC2)=O)c(C(F)(F)F)cccc1F CC(C)(C)CCCC(=O)NC1CN(C(c2cc(C3CCC3)on2)=O)CC1(C)C c1(C(=O)NC2CCCN(C(C(CC)=CC)=O)CC2)ccc2c(c1)NCCC(=O)N2 c1(C(N2CC(CNC(c3cc(Cl)ns3)=O)C3(C2)CC3)=O)ccc2nc(O)[nH]c2c1 N1(C(c2ccc(C)cc2)=O)C2CC=C(C(=O)NCCC(O)C3CCCC3)C1CC2 C1(C(C)C)CCCC(NC(=O)C=CC(C)(C)NC(c2ccoc2Cl)=O)C1 c1(N(CCC(C)C)C)nc(N2CCCC(N(S(C)(=O)=O)C)C2)c2c(n1)CCOC2 C1(CC(=O)N(CC=C)C)COCCN1C(=O)CS(=O)CC C(=O)(CCCC(C)CC)N(CCCC(=O)CC(CC)C)C.C(C(C)(C)CO)NC C1(CNC(C2(C#C)CCC2)=O)CC(NC(c2n[nH]c3c2CCC3)=O)C12CCC2 c1(C(N2CCC(NC(C=C3CCC(C)CC3)=O)C2C)=O)cncc(S(N)(=O)=O)c1 C1(C=O)CC2(C1)CS(=O)(=O)C2.C(C=O)C(C)(C)C.CC(O)C.C=O.CO C(CC(F)F)(C(=O)NCC(O)C1CCC1)NC(c1c(N)non1)=O CC1CCCc2ncc(C(=O)N(C)CCNC(=O)Cc3ccc4c(c3)CCO4)n21 c1(NC(N(C(C)Cc2ccc(F)cc2)CC)=O)cc2c(cc1F)NC(=O)CO2 C1(CC(=O)NC(C2CN(C(C(C)Sc3ccccn3)=O)C2)C)OCCC1(C)C c1(OC)ccc(C(=O)NCC2CN(C(C3(C)CCC(=O)N3)=O)C2)nc1Cl.O Cc1cc(C(=O)NCC2(NC(c3cnco3)=O)CC2)sn1 Cc1ccc(C(F)(F)C(=O)NCCC(C)CCNC(=O)CC)cc1.C(N)(=O)N Cc1ccc(C(=O)NC2CC3(C2)CC3C(=O)N(CC(C)C(C)C)C)cn1 C(C)(CC1CCC1)(C(=O)NCC1COCCN1C(=O)C(SC)SC)OC C(=O)(C1=CCC(C)(C)CC1)NC(C1(O)CCN(C(C2CC(C#N)C2)=O)C1)C C1(C(N2CCC(O)(CN(C)C)C2)=O)COCCN(c2nccc(C)c2C(=O)O)C1 c1(C(=O)NC(c2ccc(C)cc2)CNC(CC(C)SC)=O)nnn2ccccc12 C12(CNC(c3cn(C)nc3)=O)CC(CO1)N(C(=O)CC1COCC1O)C2 N1(C(c2cccc(C)c2N)=O)CC2CN(C(=O)C3=CCC3)CC2(C(N)=O)C1 C1(O)(CN(C(C2C(CC)CCC2)=O)C)CCN(C(C2CCCC(C)CC2)=O)CC1 C1(C)(C(=O)NCC(COC(C)C)O)CN(C(c2nocc2Cl)=O)C(C)(C)C1 C1(NC(Cc2c(C)cnn2C)=O)CCCC(C(=O)N(C)Cc2cccs2)CC1 c1(OCC=C)ccc(Cl)c(C(=O)N)n1.C1CCC1.C1(C=O)CC1.C1CC1 N1(Cc2c(OC)cccn2)CC(NC(c2ccc(I)c(C)c2)=O)CC(C)C1 c1(C=O)ccc[nH]1.[nH]1cnnc1.C1CC(C=O)C1.CC(C)(C)OC(=O)N.C C1(CNC(=O)CSc2ccccc2)CC2CC2N1C(c1cccnc1F)=O c1(C(N2C(CC)(CC)CC2)=O)c(CNC(C23CCC(CC2)C3)=O)nnn1C c1(CC)ccc(F)c(C(=O)NC2CN(C(c3nc(O)[nH]c(=O)n3)=O)CC2C)c1 c1(C(N2CCN(C(c3cnc(OCC)s3)=O)C(CC)C2)=O)ccc2ccnn2c1 c1(C(N(C2CCC(NC(=O)C(C)(C)F)CC2)CC)=O)cnn(C)c1Br c1(CSCC(=O)NC(c2ccco2)CC)cc(OC)ncc1Cl Cc1cc(CC(N2CCCC2C2(C(=O)NOCC(O)C(C)C)CC2)=O)no1 Cc1nc(O)sc1C(=O)NCC(C)(C)OCC(=O)NC.C1(C2CC2)CC1 C1(C(N(CC(C)O)CCNC(=O)CC(C)c2ccncc2)=O)COCCOC1 C1(C(N2CC(CNC(CC3CCN(C)C3)=O)C2)=O)CCC(C)(C)O1 C1(CNC(C(c2ccccc2)SC)=O)CN(C(=O)CCS(C)=O)CC1C CC(CN(C)C)N=c1[nH]c(=NC2CC3(CNC(=O)O3)C2)c2cccc(F)c2[nH]1 c1(C(=O)NCCCCC(C)NC(=O)CO)cncc(N=[N+]=[N-])c1.c1cnn(C)c1 c1(OCC(N2CCC(CC(C)N)CC2)=O)cc(F)ccc1F C1(CCC)CN(C(=O)CCC(c2nnnn2C)C)CC1Sn1ccc(C(=O)O)n1 O=C1NC(c2ccccn2)N2CCN(c3ccc(Cl)cc3)CC12 N1(C(C(C)(C)O)=O)CCCC(C2CCCN(C(=O)CCc3ccccc3Cl)C2)C1 C(CC(C)C(C)C)NC(Cc1c(C(C)C)con1)=O.c1(CC(=O)N)cnn(C)c1 C1(CNC(NCC(C)C)=N)CCC2CC1C2(C)C c1(C=O)cc(S(N)(=O)=O)cnc1C.N1C(=O)CCC1C(=O)N(C(C)C)C.C c1(CCC(=O)N(C(=O)CCC2CCO2)CCCO)n[nH]c2ccccc12 C1(NC(c2c(C)cccn2)=O)CC2CC1CC2C(=O)N(c1ccc(F)cc1)C C1(NC(C2(C)CC2)=O)CC2CC(NC(=O)CSc3ccc(O)cc3)CC2C1 C1(CC#C)(C(=O)NC(C2CCCN2C(=O)CS(N)(=O)=O)C)CC=CCC1 c1(CNCC(C(CO)NC(=O)OC(C)(C)C)=O)cccc(Br)c1N C(CC(O)C)N(C1CCCC1)C(COCCCC#C)=O.C(=O)(CC)N.CC(C)C C(C(CC(C)C)C(=O)NCC1CCN(C(=O)CN2CCCCC2C)CC1O)OC c1(C(=O)NC2CC(CCC(=O)NCC(CCC)(C)O)C2)cc(C)cc(C#N)c1 n1(CC)cc(C(=O)NCC(C(=O)NC(C)(CO)C2CCC2)N(C)C)c(C)n1 C(=O)(CC(C)C(C)C)NCC(CCCC)NC(=O)Cn1ccc(=O)cc1C c1ccc(OC(F)(F)F)cc1.C(F)(C(=O)NCC(O)C)=CC.C(=O)(CC)N c1(N(C)C)ccc(C(=O)NCCCNC(=O)CN2CC(F)(F)C2)cn1 N1(C(c2scc(OC)c2)=O)CC2CC1(C(=O)NCC1CCCC(O)C1)C2 C1(CNC(C(C)n2ccnc2)=O)CCCCC1NC(=O)CSc1nc[nH]n1 N1(C(C(COC)C)=O)CCC(C)(C)C(C(N2CC3(C2)CN(C(C)C)C3)=O)C1 N1(C(CC2N(C)C(=O)CC2)=O)CCc2sc(CNC(C3(O)COC3)=O)nc2C1 C=CCC(C)(C)C(=O)NC(C1CC(NC(=O)C=C(C)Cl)C1)C c1(C(N(C)CC2COCCN2C(=O)C=Cc2cccs2)=O)cc(=O)cc(Cl)[nH]1 c1(CCC(N2CCN(C(=O)CSC(F)F)CC2)=O)ccc2c(c1)OCCO2 CC(C)C(C(=O)N1CCN(C(=O)COc2ccn(C)n2)CC1)c1cccnc1 c1(C(=O)NCC2(O)CCCN(C(C=CCCC)=O)C2)n[nH]c2c1CC(C)OC2C C#CC1CN(C(c2coc(CCC)n2)=O)CCN1C(=O)C(O)C(C(C)C)OC C(CNC(=O)C(C)=C1CCCC1)(C(C)(C)C)NC(C1C(=C)CC1)=O N1(C(C2CCC(=C)CC2)=O)CCC2CCN(C(C3(C4CCCCO4)CC3)=O)CC12 C(=O)(CC(C)(C)C(=O)N1CC(NC(C2(CO)CCCO2)=O)C(O)C1)OCC Cn1c(-c2ccccc2F)nn(CN2CCCC2c2ccc(Br)nc2)c1=O Cc1nc(F)ccc1NC(C1COCC1NC(C1(C(C)(C)O)CC1)=O)=O C(C1CCCN1C(=O)CC1CCCSC1)=CC(=O)NC1CC(C(C)O)C1 Cc1sc(C(=O)O)nc1CNC(N1CCCCC1CCC(C)(C)N(C)C)=O C12(CNC(C=C(CCC)C)=O)CCCC1N(c1nnc(COC)o1)CCC2 C1(C=O)CN(C(=O)CCC2CCOC2)C(C)(C)C1.C1(CC)(COC)CC1.N Cc1ccc(SCC(C(F)(F)F)OCN2CCCC2C2CC2)cc1F c1(C(N2CC=CC(NC(COCC(=O)NC)=O)C2)=O)n[nH]cc1[N+](=O)[O-] CCC(C)CCCC(=O)NC(CNC(c1ccccc1C1CC1)=O)CC(F)(F)F C(=O)(C(C)C(O)CC(C)C)N.Cc1ccc(CNC(=O)CC2(O)CCC2)nn1 c1(CN2CC3N(C(=O)CCc4ccc(Cl)nc4)C3C2)ccc(F)c(O)c1F C1(NC(c2ccn3c2CSCC3)=O)CCN(C(=O)Cc2nc[nH]n2)CCC1CO c1(NC(C2(CNC(CC3CCCC(C)(C)O3)=O)CCC2)=O)cccc2c1OCC2 CC1CCCC(CC(=O)NC2(CCCNC(=O)C(=O)N(C)C)CC2)C1 c1(C(C2CC2)NC(C2CCC(n3cc(C4CCCC4)nn3)C2)=O)nccc(O)n1 C12(C(=O)NC3CN(C(c4cn(C(C)C)nn4)=O)C3)C(=O)C3CCC1C2C3 N1(C(C(CC)F)=O)CC23CCCC2(C1)CN(C(=O)C#CC1CC1)C3 C(=O)(C(CC=C)NC(=O)C(CC)=CC)NCCSCCC=C C=CC(C)(O)CC(=O)N1CC2(CCNC(c3cccc(C)n3)=O)CCC1C2 C1(NC(=O)C(F)n2ccnc2)CCCN(C(=O)CNC(c2cccc[n+]2[O-])=O)C1 c1(C(N2CC(O)(CC)C2)=O)nc[nH]c2ncnc1-2.c1(C(=O)N)ccc(F)c(O)c1 C1(C(=O)NC)CCCCN(C(=O)C=Cc2ccc(C(F)F)o2)C1.C1CCOCC1 N1(C(C2CCC(C)(C)C2)=O)CC=C(C(C)(C)C(=O)N2CC(O)CC23CCCC3)C1 c1(Oc2ccc(NC(=O)OC)cc2C(=O)OC)c(F)c(F)cc(F)c1F c1(C(N2CCC(N)C(CO)C2)=O)cnc2c(c1)CCCC2 C1(F)(CNC(c2c(C)nco2)=O)CC2CCC(C1)N2C(=O)C(C)CC(C)(F)F CC1(C)CC(NC(=O)CN2C(=O)CCCC2=O)CCN(C(C2COC(=O)C2)=O)C1 c1ccc(O)c(NC(=O)CO)c1.C1(C(=O)OC)OCCC1NC(=O)CCO c1(OC)ccc2cc(C(=O)N(CCCNC(C3CCC(C)(C)C3)=O)C)sc2c1F CC1CCc2nc(N3CC(=O)NC(=O)C3)nc(N3CCCC4(C=CCO4)C3)c2C1 c1(CC)ccc(C(=O)NCC(O)CN(C(=O)C=CBr)C)cn1 C1(CNC(CCc2nnc(C)n2C)=O)CC(NC(C2CCSCC2)=O)C12CCC2 Cc1cccc2c1OC(C(=O)OC(c1ccccc1Cl)C)C2 N1(CC)CC(C(=O)NCC(C)(C)NC(c2cnn(CCOC)c2)=O)CC1=O Cc1cc(C(=O)NCC2CCC(NC(C3C4COCC34)=O)CC2)cn1C CC1CC(NC(=O)CC2CCN(C(c3ccc(O)cc3)=O)CC2)CC(C)(C)C1 CCCC(O)(CCC)CC(=O)N(CC(O)CNC(c1ccc(CC)[nH]1)=O)C N1(C(C(CC2CCCC2)NC(Cn2ccc(C)c2)=O)=O)CCCC(CC2CC2)C1 Cc1nn(C2CCOCC2)cc1C(=O)N(CC(=O)O)CC(F)F N1(C(C=C(CC)CC)=O)CC(NC(c2ccc(CC)cc2Cl)=O)CC1(C)COC Cc1cncc(C(=O)NCC2CCCN(C(=O)C(O)c3ccco3)C2)c1C N1(C(C(c2cnn(C)c2)OC)=O)CCC2(CC1)CC2NC(c1nnc(S)n1C)=O C1(CNC(CCC(=C)Cl)=O)CN(C(c2cn(C)cc2C)=O)CCC1C Cn1nc(Cl)c(C(=O)NCC(C)(C)NC(c2cn[nH]c2)=O)c1Cl.C1CCCO1.C CCC(C(=O)N(C1CCCCC1O)C)C(C)(C)CC C1(N(C(=O)C(=O)NCCc2ccccc2)C)CCCN(C(=O)CC(F)(F)Cl)C1 c1(C(=O)NC2CCC(N(C(c3cc(C)nc(O)n3)=O)C)C2)cc(Cl)c(O)cc1C C1(C(N2C3(CNC(C(CN(C)C)(C)C)=O)CC(C2)C3)=O)CC12CCCOC2 C(=O)(C(C)(C)Cn1ccnc1)NCC1N(C(CC2(C(C)C)OCCO2)=O)CC1 CC1CC(NC(c2cc(=O)n(C)o2)=O)CN1C(c1ncn(C(C)(C)C)n1)=O n1(CC(=O)N)sc2ccccc2c1=O.N1(C(=O)OC(C)(C)C)CCCC(C)(C)C1 c1(NC(C(C2CN(C(c3c(CC)occ3)=O)C2)O)=O)ccc(Cl)cc1O C(CCC)(CCCNC(=O)C(C)(F)F)NC(c1ccc(SCC=C)cc1)=O N1(Cc2c(OC(C)C)nccc2)CCC2(CCCN(C(C3(Cl)CC3)=O)C2)C1 n1(CC(N2CC(CCNC(CCN(C)CC)=O)C2)=O)cc2ccccc2n1 N1(Cc2n(C)cnc2)CCCC(NC(C2(C(N)=O)CC2)=O)CC1 C1CC2CC(C1)N(C(c1c[nH]nc1C(F)(F)F)=O)C2.C1(C(=O)N)CCC(F)C1 N1(C(c2ccc(O)cc2)=O)CCC2(C(=O)Nc3ccccc3F)CC2C1 c1(OC)ccnc(O)c1C(=O)NC12CC1CN(C(=O)COCCOC)C2 CC(C)(Cc1ccccc1)CC(=O)NC12CC1CN(C(C1(C)COC1)=O)C2 c1(C(C)Nc2n(C(C)C)ccn2)ccc2cccc(OC)c2n1 C(CC(C(=O)NOCCOCC)NC(C1CC2(C1)CC21CC1)=O)=CC C(=O)(C(CCCC(=O)OC)N1CCC(C)(N(C)CC)C1)NCCOCC c1(OC)cccc(-n2cc(CC3CCCN(C(c4nc(C)oc4C)=O)C3)nn2)c1 c1(C(N)=O)cccc(C(=O)NC2CCCC2C(N2CCC(CC(F)F)C2)=O)c1 N1(CCNC(c2ccc(Br)cc2F)CC(C)C)CCC2(C1)OCCO2 C1(NC(c2c(CC)ocn2)=O)CCCN(C(C2(c3ccsc3)CC2)=O)CC1 C1(CN(C(C)=O)C)CCCN(C(=O)CNC(C2CCOCC2)=O)C1 N1(C(C2(C)N(C(CC3CCC(C)(C)C3)=O)CC=C2)=O)CC=C(CO)CC1 C1(NC(C(C)Cc2ccco2)=O)CCCC12CN(C(=O)CO)C2 C1(C(=O)NCCCCNC(=O)CCc2nccs2)CCN2CCCC2C1 c1(C(=O)OC)cn2c(NC(C3(O)CCN(c4nccc(Br)n4)C3)=O)cccc2n1 N1(C(C(C)(C)C)=O)CCC(C(F)(F)F)C(NC(=O)CC2OCCO2)C1 c1(C(=O)NCCC(CNC(C(CO)NC(N)=O)=O)O)c(F)ccc2occc12 C1(NC(C(c2cc(Br)cs2)N(CCCOC(C)C)C)=O)CCCCC1 c1(C(N(C(C)C)CC)=O)cc2cccc(F)c2nc1C.C(=O)(C=O)N.C(C)C S(=O)(=O)(c1ccc(NCCS(N)(=O)=O)c(Br)c1)NC(C1CCCO1)(C)C N1(C(C(=Cc2ccccn2)C)=O)CCN(C(=O)Cc2cccc(O)c2)CC1C C1(C(N2C(C(C)NC(c3ccc(F)s3)=O)CCC2)=O)CCc2c(cnn2C)C1 C1(C(=O)NCC(COC)(C)O)CN(C(=O)CC(C)(C)C#N)CC(C)(C)C1 N1(C(Cc2cccc(C)c2)C)CCOCC(C(=O)NCCc2scnc2C)C1 N1(C(c2c(C(N(C)C)=O)cccc2)=O)CC2CC1CC2CN1CCCC1 c1(-c2nnc(-c3cn(C(C)CC(=O)N(C)C)nn3)o2)ccc(F)cc1C(=O)O C1(NC(C2N(C)CCN(C(=O)C(=O)NCC(F)F)C2)=O)CCC(=O)NC1(C)C N1(C(CC(C=C)C)=O)C2CCC1CC(NC(c1c(F)cccc1F)=O)C2 Cc1ccc(C(=O)NC(C)CNC(C23CC2COC32CCC2)=O)c(C)c1Br C1(NC(C2(CC)CC2)=O)CN(C(c2occc2C2CC2)=O)C2(CCOC2)C1 c1(C=O)cc2c(O)ncnc2cn1.C(C(C)C)N(C)C(C1CN(C(N)=O)C1)=O.N c1(C(c2n(CCCC)nnn2)NCC2CC(C(C)C)C2)cncc(SC)c1 CCC(CCC(=O)NCC(C)(C)OCCNC(=O)CSc1ccncc1)OC Cc1ccc2occ(C(N3CCN(C(C4(F)CCN(C)CC4)=O)CC3C)=O)c2c1 C1(C(N2C(C(NOCC(=O)OCC)=O)CC2)=O)CCC(O)CN1C Cc1[nH]nc2ncc(C(=O)N(CCC(C(C)C)NC(C3(C)CC3Br)=O)C)cc12 C1(NC(c2c(CC)occ2)=O)CC12CCC(NC(=O)CC=O)CC2.C1CC1.N CCC(O)CC(=O)NC(C1(O)CCN(C(c2cc(SC)c(C)o2)=O)C1)C N1(C(c2c(C)nc(C)s2)=O)CCC(NC(C2CCc3nn[nH]c3C2)=O)CC(O)C1 N1(C(C=CCCC)=O)CCC(C)C1CC(=O)C.c1ccccc1.C(=O)(CC)N N1(C(Cc2nnc(C)s2)=O)CCc2cc(CNC(C3(Br)CC3)=O)ccc2C1 C1(C)(C(=O)OCC)COCC1NC(C1(CF)COC1)=O C(=O)(CCC(=O)N1CCN(C(=O)C(C)OC)CC1)NCC C1(NC(c2cc(Cl)sc2Cl)=O)CCCN(C(=O)CC2=CCCC2)CC1F c1(C(N(CCCNC(=O)CC2CC3(CC3)CO2)C)=O)cc2cc[nH]c2cn1 N1(C(=O)OC(C)(C)C)Cc2ccccc2CC1C(N1CCOC2(CCOC2)C1)=O C(CC(N)=O)(C1CC1)NC(C=CCN(C)C(C1CCCSC1)=O)=O N1(C(C2CC(C(C)=O)C2)=O)CC2CCCC(C1)N2C(=O)CC1CCC(C)CO1 C1(C(C)C)CN(C(=O)CCS(C)=O)CC1NC(=O)CN1CCCCC1 N1(C(C2CCC2c2ccc(F)cc2)=O)CC2CN(c3ncnc(Cl)c3Br)CC2C1 c1(C(C)NC(c2ccc(C)c(N3C(=O)CCC3=O)c2)=O)ccc(S(C)(=O)=O)cc1 N1(C(COC(CC)C)=O)CCN(C2CCCN(C(c3n[nH]cc3Cl)=O)C2)C(=O)C1 CC1CC(CCNC(=O)Cn2nnc(C3CC3)n2)CCN1C(c1cc[nH]n1)=O c1(C(N2C(CN(C(c3ccc(C)c(C)c3)=O)C)CCC2)=O)cnc2scnc2c1 C#CCC(C(=O)NOC1CC1)NC(c1coc(CCC)n1)=O c1(C(=O)OC)c(OC)cncc1NC(=O)C(=O)NC1CC(C(C)O)C1 c1(C(=O)OC(C2CCCCC2)C(C)=O)cc2cccn2cn1 c1(C(C)NCC(COCC)C)[nH]c2ccc(F)cc2c1C Cn1c(C(=O)NC2(CC(=O)NCc3c[nH]nc3C3CC3)CC2)cccc1=O n12cc(nn1)C1CCCN1C(=O)C1CC2C1.c1(C2CC2)ccc(Br)o1.CO c1(NCCCN(C(=O)CC(=O)C2CCCC2)C)ccc(F)c(F)c1 N1(C(CCC2CCN(C)C2)=O)CCN(C(c2cccc(N)c2F)=O)CC(C)(C)C1 c1(C(=O)OC)c[nH]c2ccc(CNCc3c(F)ccc(Cl)c3F)cc12 Cc1cc(=NCCC2CCC(C)O2)[nH]cc1S(=O)(=O)N1CCC(=C(F)F)CC1 c1(C(N2CC(O)C2)=O)cnc2ccnn2c1O.c1(CC)occ(C)c1C(=O)NC c1(C(=O)NCC2(O)CCN(C(c3c(C)oc(Cl)n3)=O)C2)ccn2nccc2c1 C1(C(=O)NC(CSC)C)(NC(=O)C(N2CCOC2=O)C)CC(O)C1 C(c1ccccc1Br)=CC(=O)NC(CNC(c1c(C(=O)OC)cccc1)=O)C N1(C(CCc2cnc(C)o2)=O)CC2CC1(C(=O)NC1CCCN(CCO)C1)C2 CCC(CCCC(=O)N1CCC(N(C)C)CC1)NC(C1CC2(CCO1)CC2)=O C(=O)(CC1=NN(C)C(=O)C1)NC(C(=O)NCCC(CC)(C)O)C(C)(C)O c1(C(N2C3C(CNC(Cc4cc(OC)no4)=O)C(C3)C2)=O)ccc2n[nH]cc2n1 c1(CCC(N2CCC(OC)CC2)=O)c(C)nc2nc(=N)[nH]n2c1C N1(CC=C(C)C)CCS(=O)(=O)C(C)C1C.c1(C2CC2)cccc(OC(F)(F)F)c1 CC(O)(C(=O)N1CC(CO)(NC(=O)CCc2cncs2)C1)c1ccccc1 N1(C(C(C)C(=O)OC(C)(C)C)=O)C2CCC1CN(C(c1cn(C)ccc1=O)=O)C2 c1(OC)cccc(F)c1CN1CCC(F)(C=O)C1.c1cc(C(F)(F)F)nn1C.N N1(C(c2cncc(NC)c2)=O)CC=C(CNC(C2CCC3(CCC3)O2)=O)CC1 C(c1scnc1C)=CC(=O)N(C1CCN(C(=O)Cc2ccsc2C)C1)CCC C12(C=O)C3C4C1C1C2C3C41C=O.c1(CC=O)cc(C)no1.CCCC.CO N1(C(C(Cc2c(C)nc[nH]2)O)=O)CC=CC(NC(=O)C(C)N(C)C)C1 C1CCN(C(C2CN(S(=O)(=O)C(F)(F)F)C2)=O)C1C.Cc1ncc(C(=O)N)o1 C1(C(=O)NCC(CCCC)NC(=O)CC2CC(OC)C2)CCc2cnc(C)n2C1 C(=O)(C(F)(F)C(F)(F)F)N1CC(NC(c2c(CC)n(C)nc2)=O)C(CO)CC1 c1(CC(=O)N)ccc2oc(C)nc2c1.Cc1nc(CCC(=O)NCC2CC2)cs1 C1(CC(=O)N(CC(CNC(COCCCCC)=O)C)C)OCCOC1(C)C N1(C(CN(C(CS(CC)=O)=O)c2c(C)ccnc2Cl)=O)CC2(COC(=O)C2)C1 O=C(NNc1c(Cl)cccc1Cl)C12CCCC(C(=O)O)(CC1)C2 C12(C(=O)NC3CC(N(C(=O)C=Cc4cncn4C)C)C3)CCC(=O)N1CCS2 C1(CC(N2CC(N(C(C=C(C)C(F)F)=O)C)C(F)C2)=O)CCCCCCC1 C(=O)(N=S1(=O)CCC(C)(N)CC1)C1CC2(CC(C(=O)OC)C2)C1 C1(C)(CNC(C(=Cc2cccs2)C)=O)CCCC1.C(=O)C.CCN(C)C.N c1(C2CN(C(C3CC(OCC)C3)=O)C2)nc(C)c(CNc2ccccc2)o1 c1(C=O)cnc(P(C)(C)=O)cn1.CC1=NOC(C)(C(=O)NC2COCC2)C1.C Cn1ncc2c(N3CCN(C(c4cc(Cl)cnc4F)=O)CC3CO)ncnc12 N1(C(c2c(C)nc[nH]2)=O)CC(NC(=O)Cc2ccn(CC(F)(F)F)n2)CC(C)C1 CCCCCCn1cc(C(CCC)NC(=O)CC2CCSCC2)nn1 CCC(C)CC(C(=O)NC1COC(C(F)F)C1)NC(=O)CCCCC(C)=O C1(NC(CC)C(=O)OC)CCC2(CCc3ccccc32)CC1 CC1(N(C(=O)Cc2cc(O)nc(O)n2)C2CC2)CCC2(CC1)OCCO2 C1(OC)CC(C)N(C(c2cc(C)n(C)n2)=O)C1.C1(C(=O)N)CCC2(CC2)C1 N1(C(Cc2ccn(CC)n2)=O)CC2CC1CN(C(C1CC(N(C)C)C1)=O)C2 c1(C(C)C)ocnc1CNC(=O)C(C)CNC(C1CCOC1C(C)C)=O N1(C(CCC(=O)N(CC)CC)=O)CC2(CCC2)C1.C1(C=O)CCC2(CCC2)O1 c1(CC(=O)NCCCC(C)NC(c2c(CCC)n[nH]c2)=O)cnccc1C C1(c2onc(-c3cccc(C(C)N)c3)n2)CCOCC1(C)C N1(C(C)=O)CCC(N(C)C(C2CC(NC(C3CCCC(C)O3)=O)C2)=O)CC1 c1(C(=O)NC(CN(C(=O)CC(C)C(=O)OC)CC)C)ccc2ccnn2c1 C1CC(C)(C)CN1C(=O)C(=O)C(F)(F)F.c1(C(C)O)ccccc1C(=O)N.C C(N=c1[nH]c2cccc(C#N)c2s1)C1(NC(c2cc(OC)c(Cl)cc2)=O)COC1 c1(C(N2C(CNC(c3cn4c(n3)CCC4)=O)CCC2)=O)cc2ccccc2cn1 c1(C(N2C(C(C)NC(C(C)N(C)C)=O)CCC2)=O)cnnc(O)c1 c1(C(N2CCCC(CN(C(=O)C(C)C(O)CC)CC)C2)=O)cc2sccc2cn1 Cc1cc(C(=O)N(CC(C)NC(=O)C=C2CCC(C)C2)C)nn1C(C)C c1(OC)nc(C)cc(C)c1C(c1nnnn1C1COC1)NC1CC2CCC(C1)O2 CON(CCC(=O)NC1(C)CCSC1)C(=O)COCCN(C)C c1(CS(=O)(=O)N(CCC(=O)NC)C)ccsc1S(C)(=O)=O.c1ccncc1 Cc1cc(C(N2CCCC2C(C)(C)C(=O)NC(C)CCCO)=O)cnn1 c1(OC)ncc(F)cc1C(N1CCCC(CC(=O)OC(C)(C)C)C1)=O C(C(C)C)(C(C(=O)NC1CCOCC1)N(C)C(c1cccc(C#N)c1)C)OC C=C(C)CC(C(=O)NCCNC(=O)C(CO)N(C)C)OC C(=O)(CC(CN(C)C)C(F)(F)F)N1C(CCCNC(c2cc(C)sn2)=O)CCC1 C12(CCNC(C=C(CC)C)=O)CCC(C1)N(C(c1cnc(C)cc1Cl)=O)C2 N1(Cc2c(OCC)cccc2)CCC2(CC2C(N2CC(c3ccccc3)C2)=O)C1 Cc1ccc(N)c(C(=O)NC2CCN(C(C3(C)CCOC3)=O)C2)c1 C(=O)(C1=NN(C)C(=O)CC1)N1CCN(C(C(CSC)O)=O)CC1CCO S(=O)(=O)(c1ccc(NCCCC(C)CO)nc1)N1CCC(S(=O)(=O)NC(C)C)C1 C1(C=O)CC12CCCCC2.C1(C(N(CCC#C)CCOC)=O)CC(C)(C)C1.C CC1CCCC(NC(=O)CN(C2CCC2)C(c2ccnn2C)=O)C1 c1(C=O)cn(C)c(=O)cn1.N1(C(c2cc(CC(C)C)on2)=O)CCC(C)(C)C1 C1(CNC(C(F)=CC)=O)CN(C(=O)CN(C)C)C2CC12.c1ccccc1 CC(CC(=O)Nc1cn(CCC(=O)Oc2ccccc2)nn1)C(F)F c1(CN2CC(C)(N(c3cc(C(=O)O)cs3)C(CSC)=O)C2)cccc(N)n1 C(=O)(CC(C)(C)CC(F)F)N1CCC(N(C(=O)C(C)(F)C(C)(C)F)CCC)CC1 c1(C(c2nnnn2CC(F)F)NC(c2ccns2)C)cc2cccc(Br)c2o1 N1(C(C(CC)C)=O)CCC2(CCCN2C(=O)CN2CCCc3sccc3C2=O)C1 C1(C(N2CC(CCNC(c3cc(Cl)c(Cl)[nH]3)=O)C2)=O)CCCC12CCOCC2 N1(C(CN(C)CC)=O)CCCC(C(C)C(=O)Nc2cn(CC3CCC3)nn2)C1 C1(S(C)(=O)=O)(C(N2CCCC(NC(c3nc(C)n(C)n3)=O)C2)=O)CC1.C c1(C(N2CCC(c3ccc(F)c(F)c3)(C)C2)=O)cccc2c(Br)coc12 c1(C=O)ncc(F)cc1F.CC1(C)C(C(=O)NCC2(F)CC(C)C2)C1C#N c1(CCC(N2CC(N(C(COCC)=O)C)C2)=O)c[nH]c2c(C)cccc12 c1(C(N2CC(NC(=O)C(=O)NCCc3ccccc3)C2)C)cncc(F)c1 CN(C1CN(C(c2ccsn2)=O)CCc2ccccc21)C(=O)C(F)F O=C(CCCCC1CC1)NC1CN(C(c2coc(C3CCOCC3)n2)=O)CC1O CC(C(=O)NC1CC(CCC(=O)NC(C)Cc2cn[nH]c2)C1)N1CCCC1 c1(COC)nc(NCC2(Br)CC2)cc(N2CCC(c3cccs3)C2)n1 N1(c2n(C(CCCC)C)nnn2)CC(C)(C)Oc2ccccc21 C1(C(=O)NCC2CC(NC(CN3CCC(C)C3)=O)C2)Cc2nccn2C1 c1(C(N(C2CC3CN(C(C=CSC)=O)C2C3)C)=O)cc2ccnc(Cl)c2[nH]1 N1(C(=O)C=Cc2ccsc2)CCC(CNC(C2(Cl)CC2)=O)C(C2CC2)C1 c1(NC(=O)NCCS(CC)=O)ccc(F)c(F)c1OC C1(CC=C)CN(C(c2ccoc2)=O)C1.C(=O)C(C)N(C)C=O.C(C)(C)C.N N1(C(C2N(CCC)CCCC2)=O)CCC(CNC(c2ccc(F)o2)=O)C12CC2 C(=O)(C(C(=O)N1CC(CNC(=O)C(F)C(C)C)C1)c1ccccc1)OCC N1(C(CC(=O)NCC#C)=O)CCC(C)N(C(=O)CCC2OCCO2)CC1 N1(C(C=C2CCC(C)CC2)=O)CC2CCCC(CNC(C3CC3(F)Cl)=O)C2C1 c1(C(=O)NC(CNC(C2ON=C(C)C2)=O)(C)CO)[nH]nc2c1COC2(C)C Cc1cc(=N)[nH]cc1C(N1CCC(N(C(=O)C(C)C(C)O)CCO)CC1)=O C1(CNC(CCCOC)c2nnnn2C2CC2)CC(=O)N(c2ccccc2Cl)C1 c1(CC)[nH]nc(C(=O)NCCCC2CN(C(=O)CCC=C(C)C)CCO2)c1Cl C(CC(=O)NCC(CC)NC(=O)C(C)(C)c1cccs1)(OCC)OCC N1(C(C(C)(C)SC)=O)CCC2(CCC2NC(c2cccc3ncccc23)=O)CC1 C1(C(=O)NC(CC)CO)CN(C(C2(C(F)(F)F)CC2)=O)CCO1 c1(C(N2C(COC)CCCC2)=O)cn2c(n1)CCN(CC1CNC(=O)O1)CC2 C1(C)(C(N2CCC(C(N(CCCC(C)O)C)=O)C2)=O)CCN(C)CC1 C12CCC(CC1)CO2.CC1CCC(=CC(=O)N)C1.N(S(N)(=O)=O)CC=O.C N1(C(CCC(CC)NC(C2COCC2C(N)=O)=O)=O)CC2NC(=O)OC2C1 N1(C(c2c(CC)ncs2)=O)CC2(CCC2)C1.c1(CC(C=O)O)cccc(Cl)c1.N CON(C)C(=O)CNC(=O)C(CC1CC1)NC(=O)CN(C)C(N)=O C1(CC(N2CCCC(NC(Cn3c(CCC)ncc3)=O)C2)=O)CCCCC(=O)N1 Cc1sc(C)c(C(=O)N(C2CC2)Cc2cccc(N(C)C)c2)c1-c1ccccc1 C=CC(C)(C)CC(=O)NC1CCN(C(C2CCCC(=O)N2C)=O)CC1F c1(C=O)ccc(O)c([N+](=O)[O-])c1.C(CCN(CC)C(C1CC1F)=O)N(C)C.N C1(C(=O)NC2CC(C)(CNC(c3cc(C)ncn3)=O)C2)CC(C)CC(=O)N1 C1(NC(C(=O)N(C)Cc2ccnn2C)=O)CCC2(C1)OCCO2 C1(NC(c2cc(CC)nn2C)=O)CN(C(c2cc(C(F)F)no2)=O)CCC1C C1COCCN(C(=O)C=Cc2cccc(C(N)=O)c2)C1.CC1=CC1C(=O)N.C c12ccc(o1)CNC2=O.C(=O)(CC1(OC)CC1)N(CCOC)C C1(C=O)CCCCC(C)(C)C1.c1(C(=O)N)cc(C)c(Cl)c(N)c1.C(C)(C)OC C1(C(=O)NC2CN(C(N)=O)C2)CCC2CCC1N2C(=O)CCc1ncccn1 N1(C(C(C2(O)CCC2)NC(COC(CC)C)=O)=O)CCCCC1C N1(CC(=O)N(CC)CC)C2CCC1CC(NC(=O)C(C)C(C)COC)C2 Cc1ccc(NNC(=O)C(C)(C)CCCOC(C)(C)C)cc1F c1(NCc2cc(OC)ns2)cc(Br)ccc1S(=O)(=O)NCC12CCCC1C2 C1(CC)CC(O)CN1C(C1CC=CCC1NC(c1ccncc1Cl)=O)=O c1(C(N2C3CC(C(=O)NC(C(=O)NCC)C)C2CC3)=O)ccc2cc[nH]c2c1 c1(C=O)cccc([N+](=O)[O-])c1C.C1(OC)CN(C)C(C)(C(=O)N(CCC)C)C1.N CCCC(O)(CCC)CC(=O)NC(C)(C)CCCNC(=O)C(CC)(CC)OC N1(C(C(C)(F)F)=O)CC(NC(=O)CCc2ccc(Br)cc2)C(O)C1 N1(C(C2(CC#C)CCCCO2)=O)CC2CCC(NC(=O)CC3CC=CC3)CC2C1 N1(C(C(C)Cc2cccs2)=O)CCN(C(=O)Cc2cccnc2O)CC1C(F)F C(=O)(C(CO)C(C)C)N(C1CCN(C(CCCOCCOC)=O)C1)C1CC1 C1(CC)COC(C)(C)CN1C(=O)CCOC(C)C.c1(C=O)cc[n+]([O-])cc1.N C#CC1(COC)CCN(CC(=O)NC(C(C)(C)CC)c2ccccc2)C1 CC1CCCC1C(=O)N(C)CCN(C)C(c1cc(C(F)(F)F)n[nH]1)=O C(c1ccc(F)cc1)=C(C(N1C(CC)C(NC(=O)CC(C)C)CC1)=O)C c1(CC=O)ccnc(Br)c1.C(C(=O)N1CC(C)C1)(c1cscn1)NC(C)=O.N Cc1c(CN2CC3CC3(C(=O)Nc3ccnc(F)c3C)C2)cccc1Br CC(C)(CCC(=O)NCC(N1CCN(C(C2CNC(=O)C2)=O)CC1)=O)[N+](=O)[O-] c1(C(=O)NCC(CCOC)NC(=O)CCC(C)(C)C)cnc(OC)c(OC)c1 c1(C(=O)NC(CNC(c2c(C)c(Br)no2)=O)C)ccc(Cl)nc1O c1(C(=O)NCC2(O)CCN(C(Cc3cc(C)nn3C)=O)C2)cnn2c1CCCC2 c1(NC(CN(C(C(CC#C)(C)C)=O)C)C)nc(C(F)(F)F)c2ncnc-2[nH]1 C1(CC(=O)NCCCNC(CC=CC)=O)OCCCC1(C)C.c1cccnc1.C n1(CC(=O)OC)cc(CCCC(=O)NCCCCC#N)nn1 CC1=C(C)CC(C)(C(=O)NCCC2CN(C(c3cscc3C)=O)C2)CC1 C(=O)(NNC(=O)CC1CCN(C(C)=O)C1)OCCOCCOC Cc1ccc2nonc2c1C(N1CC2CCCCC2(NC(=O)COC2CC2)C1)=O C(=O)(N=c1[nH]c(OC)ncc1Br)C1(F)CN(Cc2c(OC)ncc(F)c2)C1 C1(NC(c2c(C)noc2C(C)C)=O)CCCCCCC1 c1(C(=O)NCCCC2N(C(C=CC=CC)=O)CCC2)cnc2cc[nH]c2c1 c1(CC(N2CC3(CN(C)C3)C2)=O)cc(F)cc([N+](=O)[O-])c1.C1(C(N)=O)CCC1 c1(C(=O)NC2C(NC(CC(CC)C)=O)CCC2)cc(C2CC2)nc(O)c1 C1(C(=O)NCC2(CN(C)C(c3cccnc3)=O)CC2)CCCC1(F)F C=CCC(CC(=O)N(CC(N)=O)CC(C)C)NC(=O)C(C)CCOC c1(C(=O)O)cc(Cl)ncc1NC(C1CC12CN(CC)C2)=O.c1nccn1C.N C1(C(N2C(CC=O)CC2)=O)C2CCC(C2)C1.C12(C=O)CCC(CC1F)C2.C Cc1cc(=NC(C)C2CC2)[nH]c(=NCC2CC2(C)C)[nH]1 C1(F)(CNC(C2N(CCC)CCCC2)=O)CCN(C(c2ccc(C#N)s2)=O)CC1 C(C(CC(C)C)OC)NC(C(n1cc(CNC)nn1)C)=O C1(NC(=O)NC(C)Cc2ccnn2C)C2CCCOC12 c1(CC)nc(C(=O)N)cs1.C1CC(O)C1.C1(C=O)CN(CC(F)(F)F)C1.C CC(C)CCCC(C)C(=O)NCCC(O)C(=O)N(C1(C2CC2)CC1)C C1(C(=O)NCC)CC2CCN(C(c3cc(Br)ccc3OC(N)=O)=O)CC12 N1(C(C(C(=O)OC)C)=O)CCC(C)(NC(=O)CCc2nnc(C)n2C)CC1 Cc1ccc(Cl)c(C(=O)NCC2C3CN(C(=O)Cn4ncc(Cl)c4C)CC23)c1 c1(OCC(=O)NCCC(=C)CNC(=O)C(C)CSC)ccccc1Br.O Cn1ncc(C(=O)NCC(O)CCNC(C2CCCOCC2)=O)c1C(F)(F)F C(c1ccc(Br)o1)=CC(=O)NC1CC(CNC(c2cnc[nH]2)=O)C1 C1(O)(C(C)NC(C(C=CC)O)=O)CCN(C(=O)C(O)C2CCCC2)CC1 Cc1ncc(CCNC(=O)C(C2CC2)NC(C2CCOC2)=O)o1 N1(c2ccc(C(=O)NC)nn2)CCC(O)(CC(=O)NCC(C)(O)CCC)CC1 N1(C(c2c(C)c(C3CC3)[nH]n2)=O)CCCN(C(=O)COc2ccc(O)cc2)CC1 N1(C(C(CSC)O)=O)CC2(CNC(c3sccc3CC#N)=O)CC1CCO2 N1(C(C2(OC)CC2)=O)CC(NC(C2CC(C)(C)CCO2)=O)C2(CCC2)C1 Cn1cnnc1CNC(C1CCC(NC(=O)C(O)C2CC2)C1)=O n1(CCC(=O)N(CCCNC(c2ccc(F)s2)=O)C2CC2)cnccc1=O c1(OC)cc(C(=O)N(C2CCC(NC(C3(C#N)CCC3)=O)C2)C)cc2c1OCC2 CC(C)=C=CC(=O)NCCOCCN(C(=O)CCCn1c(O)nnc1O)C N1(C(CCOC)=O)CC(CCNC(c2cccc(Br)c2)=O)OC(C)C1 C1(C(N2CC(O)(COC)C2)=O)CC12CC(NC(C1(F)CC1)=O)C2 C1(CC(=O)N(c2ccon2)C)CCN1C(=O)CCN(CCOC1CC1)C C1(C(=O)NC2CC(C)(NC(=O)Cn3cnnn3)C2)CC2(CCOC2)C1 C#CCC(C)(C(=O)NCC1CN(C)CCN1C)NC(c1cnnn1C)=O c1(C(=O)NC2CCC(N(C(C3(C(C)C)CC3)=O)C)C2)cnc(C#N)s1 C(=O)(C(O)CCc1ccccc1)N(C1CCCN(C(C2CC(O)C2)=O)C1)CC N(C1CC2(CCOCC2)Oc2ccccc21)C(c1cccnc1Cl)CC C1(F)CCC1.C(CC(=O)C(=O)OCC)N.C1(C(=O)N)CC1C=O.C c1(OCC)c(CN2CCC(N(C)C(c3ccc(C)cc3)=O)C2)cccc1O c1(C(N)=O)coc(C(N2CC(=C(F)CNC(C3CCSC3)=O)C2)=O)c1 c1(CC(N2CCN(C(C3C(C(=O)O)CC=CC3)=O)CC2)=O)c(F)cc(F)cc1F C1(C(N2C(C(=O)NCC3(C)CCC3)C=CCC2)=O)CC2OC1C1CC21 N1(C(C(C)SC(F)(F)F)=O)CCCC1.C(=O)(CCCn1cncn1)N(C1CC1)C Cc1ncc(C(=O)NC(C)CN(C)C(C23CC(CO)(C2)OC3C)=O)c(=N)[nH]1 c1(NC(C2CN(C(c3ccc(O)cc3)=O)CCC2O)=O)ncnc2sccc12 c1(OC)cc(C(=O)N)ncn1.C1(C(C)C)CCN(C(=O)CCc2ncc(C)[nH]2)C1 C=CC(C)(CCOC)C(=O)NC(CC(N1CCc2c[nH]nc2C1)=O)C1CC1 N1(C(c2c[nH]c(=NC)s2)=O)CCC2(CC1)CC(CNC(=O)C(F)(F)CC(C)C)C2 Cc1cc(C(=O)NC(C(=O)NC(CCO)C2CCCC2)C(C)C)[nH]c1C c1cc(C(F)(F)F)cc(Cl)c1.C(CC(=O)NCC1CC1CS)N(C)CC Cc1nn(CCF)cc1NC(=O)C(C)C(C)NC(=O)Cc1ccns1 CC1CC(F)(F)CCN1C(=O)CCCC(C)(C)NC(=O)CN1CCCC1 C#CCC(O)C(=O)NCC1(CNC(=O)C(c2ncccc2OC)=O)CCC1 c1(CCCC)ocnc1C(=O)NC1CCN(C(=O)CC2(C)CCCO2)C1 C(c1cn(C)c2ccccc12)=CC(=O)NC(C#C)CC CCCCCC(C1CC1)NC(c1n[nH]cc1C)=O.C(c1cccnc1)=CC=O.N Cn1nnc2cc(C(N3CC(C(=O)Nc4ccnc(O)c4)CC(F)C3)=O)ccc12 c1(C(=O)NCCC(C)NC(C2CC(SC)C2)=O)ccc(F)cc1O c1(C(N2CCC(CNC(C(CC)COC)=O)C2(C)C)=O)cc2nc[nH]c2cn1 N1(C(C(CSC)C)=O)CCCCC1CNC(C1(CN2CCCC2)CCCC1)=O Cc1cc(C(N2CCC2(C)CC(N2CCC=C(F)C2)=O)=O)nn1C c1(CO)nnn(C)c1C(=O)NCCC1(NC(C(C)C2CCC2)=O)CCC1 C1(CNC(C(CC)c2cccnc2)=O)CN(C(=O)C(c2ccc(Cl)s2)=O)CCO1 c1(C(=O)NC(C(C)C)CNC(C2(CO)CCCC2)=O)ccc(O)cc1F N1(C(c2cc(C(=O)OC)oc2C)=O)CC(NCc2ccccc2)CCC1C c1ccccc1F.c1(C(=O)NCCN(C)C(C2CC(F)(F)C2)=O)ccc(C)s1 CCCC(CC(C)C)C(=O)NCC1CCN(c2cc(CC)ncn2)CC1C CC1CCN(C(=O)Cn2cc(CO)nn2)C(C)C1.c1(C(=O)N)cc(O)cc(O)n1 C1(O)(CNC(C2C(NC(c3cc(C(C)C)no3)=O)CCO2)=O)CCOCC1 N1(C(C2CCCN(C(c3cn(C(C)C)nn3)=O)C2)=O)CCC2(CC1)CC(O)CO2 C(=O)(C1=CNC2=NCCCC2=C1)N1C(C)CN(C(c2nocc2Cl)=O)CC1 C(=O)(CCCC(N)=O)NCCCC(C)NC(C1CCC2(CCC2)C1)=O c1(C(=O)N)cc(O)nc(O)n1.N1(C(C(C)OCCCCCC)=O)CC(C)C(O)C1 C(=O)(C1=CCCSC1)N1CCC(C(CNC(C(C)NC(C)=O)=O)F)CC1 C1(CCNC(C(C)(C)c2cc[nH]n2)=O)CCCN(C(c2cnc(Cl)s2)=O)C1 CC1CC(Nc2ccc(F)cc2C(=O)N(C)C)CCN1c1nc(C(N)=O)ns1 C1(NC(=O)CCc2cncnc2)CN(C(C2(c3ccsc3)CC2)=O)CC1O c1(C(N2CC(SC)C(NC(=O)C(C)S)C2)=O)ccc(F)c(C)c1.c1ccccn1 c1(C(=O)N)ccc2c(c1)NC(=O)C2=O.CCC(C)C(C(=O)NC(C)(C)C)OC CN(C)S(C)(=O)=Nc1nc(C(N2CC(CNC(c3cncnc3)=O)C2)=O)cs1 C1(NC(c2c[nH]ccc2=O)=O)CN(C(C2CC=CCC2)=O)CC1F C1CN(C(=O)Cn2ncc(O)nc2=O)CC12CCC2.C(=O)(C(C)C(=O)N)OC.C N1(C(=O)C(F)CC2CC2)CCN(C(c2ccc(-n3ccnc3)cc2)=O)C(CF)C1 C(=O)(C1=NOC2(CCC2)C1)N(C)CC1(O)CCCN(C(Cc2cnc(C)s2)=O)C1 c1(C(N2CC(C3CN(C(CCCCC(N)=O)=O)C3)C2)=O)nccc2c1NCCC2 CC1(C)CCC2(CN(S(=O)(=O)c3ccc(N4CC=CCC4)cc3Cl)CCO2)C1 CC1c2nncn2CCN1S(=O)(=O)c1cccnc1N(C)Cc1cc(Cl)ccn1 c1(C(=O)NC2C(NC(c3c(C(C)C)nn(C)c3)=O)CC2)cc(O)cc(Cl)c1Cl C(=O)(C(O)C(F)(F)F)N1CC(C(=O)NC(CC=CC)CO)C(C(C)C)C1 C=CCCC(C)(C)C(=O)NCC(n1cc(CN(C(C)(C)C)C)nn1)C Cc1cc(=O)oc(C)c1C(=O)NCC(CO)NC(=O)CCC(F)F CCCCC(C(=O)NC1CN(C(=O)C(C)(C)CC2CCC2)CCC1C)NC(N)=O Cc1cc(C(=O)NCC2CC3(CC3)CN2C(=O)CC(O)C2CC2)ccc1F C=CCC(CSC)C(=O)[SH](C1=NC(=O)CC(C(=O)OC)C1)C c1(OCC)ccc(Cl)nc1C(=O)NCCN(C)C(C1CC1(Cl)Cl)=O C1(CC(=O)NCC2CC(OC)CN2C(c2ccn(C)c2)=O)CC2CCC1CC2 Cc1cc(Br)c2oc(C(=O)NCCCOCC)cc2c1.C1(C=O)CC(=O)N1.N CC1(C)CCC(CC(=O)NC(C)(C)CC(=O)NCC(O)Cn2cccn2)CC1 C1(NC(C2C(C)(C(C)C)C2)=O)CCC2CN(C(=O)C3=C(Cl)CC3)CC2C1 C1CC(F)CN1C(c1ccn(C2CCC2)n1)=O.C(C)(C(=O)NC)NC(C)=O.C C(=O)(C(C)CO)NC1(CNC(C(C)SCCCC)=O)CC1 C1(NC(C(C)C2CCCO2)=O)CC2(CCN(C(C3(C)CCCC3C)=O)CC2)C1 C1(C(=O)NCC2CC(NC(=O)C#CC3CC3)C2)CC12C1CC3CC(C1)CC2C3 n1(CCCSCC)nnnc1C(c1coc(Br)n1)NC(c1noc(C)n1)CC c1(CCC(=O)NC(C(=O)N(C)CC2CCSC2)C2(C)CC2)nccn1C Cn1cnc(-c2cn(CCCCCCF)nn2)c1Br Cc1nn(C)c(C)c1CC(=O)NCC1CN(C(C2CCS(=O)CC2)=O)CCCO1 CCC(C)(CCNC(=O)C(C)=C1CCC1)NC(c1cc[nH]n1)=O Cc1[nH]c(C(=O)N)c(C)c1S(N)(=O)=O.C12(C=O)CC=CC(C1)OC2.C1CCC1 C(=O)(C(CCSC)NC(c1cc(C)no1)=O)N1CC(CCC#C)C1 c1(OC)cc(C(N2CCC(O)(CCNC(C3CC3F)=O)CC2)=O)c(N)cc1F C1(C(N(C2C3CN(C(=O)C(F)(F)C(F)F)CC23)C)=O)CC(c2ccncc2)=NO1 CC1(C)NC(=O)CC1C(=O)NC1CC(C)C1.c1(C(=O)N)cc2c(s1)CCC2 C1(N(C(C(CC#C)O)=O)C)CCCN(C(c2cc(N)c(Cl)cn2)=O)CC1 CC1=C(C(=O)Oc2ccc(Cl)c(CC3CN(C)CC3O)c2)SCCO1.C1C(=O)O1 O(NC(=O)CCC1CCN(C(=O)CCC2CCCO2)C1)CCCN(C)C1CC1 N1(C(C2CCc3ccccc3C2)=O)CC2CCCC(NC(C3(CF)CC3)=O)C2C1 C(=O)(C(C)(C)CC(=O)N1CC(CNC(c2ccc3c(c2)CC3)=O)CC1C)OC C1CC2(CCN2C(C2CCC2)=O)C1.N1(CC)CCN(c2ccccn2)CC1 CCCCCCC(CC)C(=O)NC(CN(C)C(C1CC(n2ccnn2)C1)=O)CC CC1CC(NC(=O)C(C)(C)c2ncco2)CCN1C(=O)CN1CC(C)(C)C1 CCCC(C(=O)NC(C1CCN(C(C2(OC)CCCC2)=O)C1)C)NC(N)=O c1(N2C(=O)C3C(C3)C2=O)ccc([N+](=O)[O-])c(F)c1.c1nncn1C.CC=O.O c1(NC(C2C(C)(C(C)C)C2)=O)cccc(C(F)(F)F)n1 N1(C(C(C)N2CCC2)=O)CCCCC12CC(NC(c1cc3c([nH]1)CCCC3)=O)C2 c1(C(=O)OC)cc(N2CCC(NC(N3CC(CO)(CO)C3)=O)CC2)ncn1 Cc1cc(NC(=O)Nc2nccn2Cc2ccccc2)c(F)c(Br)c1 Cc1ccc(C(C)NC(=O)CCN(C(=O)CC2CCOC2C)C)cc1.C1CC1 C1(C)(C(=O)N)COC(=O)C1.C1(NC(CCOCCOC)=O)COCC1C C(c1ccc(Cl)c([N+](=O)[O-])c1)=CC=O.Cc1nc(C(=O)NC2CC2)cn1C.C c1(NC(C2CCN(C(C(CC)=O)=O)C2)=O)c(Br)cccc1Br c1(C(N2CCCN(C(CCOCCOC)=O)CC2C)=O)cc2cc(Cl)ccc2[nH]1 CC(C)(C)C(CO)N(C(c1nccc(-c2ccccc2)n1)=O)CC1CCCCC1 C1(NC(COCCC)=O)CCN(C(=O)C(C)=C(C)CC)CC1OC C(CC(F)F)(C(=O)N1CCCC(C=C)C1)NC(c1ccc(C#C)o1)=O CCC(C)CC(=O)C(=O)NC(CCF)C(=O)N1CCC1CN=[N+]=[N-] c1(C(=O)NC2CCCC(NC(CCC=C)=O)C2)ccc(Br)cc1CC#N N1(C(CCN(CC#C)C(c2ccn(CC)c2C)=O)=O)CCOCC(C)(F)C1 N1(C(C(C)OCC(F)(F)F)=O)CCCC12CCN(C(c1cc3n(c1)CCC3)=O)C2 C1(CCC)CN(C(c2cn(C)nc2O)=O)CCN1C(C1CC12CCCC2)=O CC1CC(C(=O)NC2CCN(C(c3cncc(O)c3Cl)=O)C2)=NO1 C(=O)(C(CC1CCCC1)NC(=O)CC1(C)CC1)N(CCOC)CCO C1(C(=O)NCCCCCNC(=O)Cc2ccccc2F)CCCN2CCCCC12 c1(C(CC)NC(=O)NCCCc2nnc(O)o2)nnc(C)n1C1CC1 C#Cc1cc(NC(=O)C(C)C(C)NC(=O)C(O)CC(C)C)ccc1C c1(C(=O)NC2(CC=CC(=O)NCCc3cn[nH]c3)CCC2)cnccn1 C1(C)(OC)CCC(NC(c2cc(C3CC3)on2)=O)CC1.C12COCCN(C1)C2=O C(=O)C1=NN(C)C(=O)CC1.Cc1noc(C)c1C(C)NC(c1cccs1)=O.C C1(C2CN(C(=O)CC3CCC(F)(F)C3)C2)CC1.c1(C(C)C)nc(C(=O)N)co1 C1COCCN1C(C1CC(=O)NC1)=O.CC(CC1CCC1)C(=O)NC.C1CC1 Fc1cc(CNc2ccc(-c3cccc(SC(F)(F)F)c3)cc2Cl)cnc1Cl C=C(C)CN=C(NCc1cc(Br)cs1)N1CCC(C)C1 Cc1ccc(C(=O)NC2CC(O)C2CC(=O)NCc2cn(C)nn2)[nH]1 c1(C=O)cc(N(C)C)nc(Cl)c1.c1(C(C(=O)N(C)CC)C)ccc(F)cc1 c1(NCCC(C)(C)NC(C(=O)Nc2ccc(C)c(C)c2)=O)ncccc1[N+](=O)[O-] c1(OC)cccc(-c2ccc(CNC(=O)CCCn3ccnc3C)nc2)n1 C1(C)(C(=O)NCCc2ccc(C)cc2C)CC(C)(C)OC1=O c1(OC)ncc(F)cc1C(=O)NCC1CCC1.C1(CC=O)COC(C)C1 Cc1cc(N2CCC(CCF)CC2)ncc1S(=O)(=O)NC1CC2(CCC2)C1 N1(C(C(CN(C)C)NC(COC(CC)(C)C)=O)=O)CC2(CCC1CO)CC2 C(=O)C1=CCCCO1.c1(SCC)nc(C)c(CC(=O)N(CCC)C2CC2)s1.N C1(CCC)CN(C(c2c(Br)noc2C)=O)CCN1C(=O)Cc1nc[nH]n1 C1(C(=O)NCC(CO)NC(C(c2ccc(Cl)cc2)CC)=O)C2CC3C(C2)C13 Cc1ccc(C(C)C(=O)NCC2CCN(C(=O)Cc3nc(C)no3)CC2)cc1 c1(-n2cc(C(C)NC(C3CCC3n3cnnc3)=O)nn2)ccc(CC(=O)O)cc1 c1(C(N(CCN(C(C)C)CC23CC(F)(C2)C3)C)=O)n[nH]c(C2CC2)c1Br N1(C(c2c(C)[nH]nc2Br)=O)CC2CN(C(C3(C)CSC3)=O)CC2C1 Cn1nc(O)cc1CNC(C1CCCC1)=O.C12CCCCN1C(=O)CS2 c1ccc(F)cc1.c1(C(=O)NC2CC2NC(C2CC2)=O)ccn(CCF)n1 C12(CN(C(=O)CNc3cccc(C(N)=O)c3)C)CCC(C1)NC2 N1(C(C(c2ccc(OC)cc2)O)=O)CC2CCC1CN2C(=O)C(F)(F)CO C1(NC(CC2CCCC(OC)C2)=O)CCSC12CN(C(=O)CC(C)(F)F)C2 C(=O)(C1=C(C)CCCC1)N1C(CN(C(C2CC(C#C)(O)C2)=O)C)CCC1 n1(C2(NC(c3ccn(CC4CCC4)n3)=O)CC2)cc(-c2cncs2)nn1 CCCC(CC(=O)O)NC(=O)CC1CCN(C(c2ccc(C(C)O)cc2)=O)CC1 N1(C(CCCC=C)=O)CCN(C(c2cnnn2-c2ccc(Cl)cc2F)=O)CC1C C1(C(=O)NC2CC3CC3C2)CCN(C(c2ccc(Cl)o2)=O)C12CC2 c1(NC(C)C(=O)N(C)C)[nH]c(=NCC2CC23CCOCC3)nc2c1cnn2C CCC(CC)CC(=O)NC(C)CCC.c1(C(=O)N)cnn(C(C)(C)C)c1C1CC1 CCS(=O)(=O)CCn1cc(C2CC2CNC(=O)C(C2CC2)SC)nn1 c1(C(=O)NCCNC(c2cccc(CC(F)(F)F)c2)=O)cnc2ccccn12 c1(CNC2C(C(=O)Nc3cc(OCC)ncc3)CCC2)cc(Cl)ncc1N N1(C(CCC=CC)=O)CC2CCC(N(C(=O)COC(C)(C)CC)C)C2C1 c1(OC)ccc(CC(=O)NCC2CCCN2C(=O)CC2CSCCS2)cc1F c1(C(N2CC(NC(C3CCC(=C)CC3)=O)C3C2C3)=O)coc2ccccc12 C1(C=O)CC2CCC(C1)S2.C1(C(=O)N(CC)CC)(COC)CCCCO1.N c1(C(N2CC(O)(CNC(C(C)CO)=O)C2)=O)nnc2ccccc2c1N N1(C(CC(CCC)C)=O)CCOC2CN(C(C3CCC3)=O)CC12 N1(C(CC(C(C)OC)NC(=O)Cn2cnc(C#N)n2)=O)CCc2c(cnn2C)C1 C#Cc1cccc(CC(=O)NCC2(CNC(C3CC3=C)=O)CCC2)c1 CCC(C)(C(=O)N1CCC(NC(C2(c3cc(C)no3)CCOCC2)=O)C1)C(N)=O N1(C(C(CCOC)(C)C)=O)C2CCC1C(CO)N(C(=O)C1=COCCC1)C2 C12(CNC(C(C)(C)CC#N)=O)CCC(CN(C(=O)CCc3ccccc3)C1)C2 C=C(F)C1(CC(=O)NCC(c2ccccc2)NC(C2CCCC2)=O)CCC1 c1(C(=O)NCCN(C(C2C(CC)CCCC2)=O)C)cc(N)c(O)c(F)c1 c1(NCCCC(C)NC(c2nccs2)=O)ccnc(Oc2ccccc2)c1 Nc1cc(C(=O)NC2CCN(C(=O)CCC3CCC3)CC2CO)ccc1Br O=C(C1CCc2c[nH]nc21)N1CC2(C1)CN(C(=O)Cc1cnn(C3CC3)c1)C2 C1(C(=O)NC2CN(C(C3C(=C)CC3)=O)C2)CCCN(C(=O)C2CC2)C1 N1(C(C2COCCN(Cc3c(F)cccc3I)C2)=O)CCc2c(ccc(Br)c2F)C1 N1(C(CCNC(N2CC3(CC(CC)C3)C2)=O)=O)Cc2ccccc2C1 C1(CCOC)CCN(C(=O)C(C)NC(c2n[nH]c(O)n2)=O)C1 N1(C(CCN(CC)CC)=O)CCC2CCN(C(c3cc(Br)n[nH]3)=O)CC2C1 C=Cc1cncc(C(N2CCN(C(c3ncn(CC)n3)=O)C(C(C)C)C2)=O)c1 CCC(CC)CC(=O)N1CC(C)C(C)(CNC(C2CCCC23CC3)=O)C1 C1(CNC(C2(C#N)CCC2)=O)CCCC(CNC(=O)CC2CCCCC2O)C1 c1(OC)ncc(CN2CCCC2(C)C(=O)NCc2ccccc2F)cc1Cl C1(CC(=O)NC(CN(C(c2ccc(OC)nn2)=O)C)C)CN2CCC1CC2 C(=O)(C(F)(F)C(C)(C)O)N1CC(C)C(NC(c2cccnn2)=O)C1 Cc1c(C(=O)N(C2CCCN(C(=O)C=CC3CC3)CC2)C)[nH]c2c(Cl)cccc12 N1(C(C2CCCS2)=O)CCC2CCC(C1)N2CCOCc1ccccc1 CCC(C)(C)C(O)C(=O)N(CC(N1CCC(C)(NCC)C1)=O)CCOC Cc1c(C(N2CC(NC(=O)C3=CCCC3)CC3(CCC3)C2)=O)[nH]c2ccccc12 N1(C(C(C)C)=O)CC2CCN(C(c3cn(C)c(=O)nc3O)=O)C2C1.C(=O)OC.N C1(OC)CC(CC)N(C(=O)C=CC2CC2)C1.C(=O)CCC1CC1.C1CC1 N1(C(C(CC)N2CCCC2=O)=O)CCN(C(C2(CC)COC2)=O)CC1C(F)F c1(C(=O)NCCN(C(=O)C(C(C)C)SC)CC)c(F)cccc1[N+](=O)[O-] C(c1ccc(=N)[nH]c1)=CC(N1CC(NC(c2n(C(C)C)ncc2)=O)C(C)C1)=O n1(CC)ccnc1CN(C)C(C1(C)CC(NC(C2CC(=O)C2)=O)C1)=O CCC1=C(C(=O)N2CCC(C)C(NC(=O)C=CC3CCCC3)C2C)CCCO1 C(CC(C)(C)C(=O)O)SCc1nnc(-c2c(OC(C)C)cccc2)n1N C1(C)(C(N2CCCC(CNC(C(CCC)(C)C)=O)CC2)=O)CCC(F)(F)CC1 N1(C(c2cccc(C(=O)NC)n2)=O)CC(C)CCC1C.c1(CC(=O)N)ccsc1 C(C)(C1Cc2ccccc21)N(C(C(=CC1CCC(C)CC1)C)=O)C C#Cc1cc(NC(=O)CCCNC(=O)C(C(C)C)NC(C)=O)cc(F)c1.O Cc1c(C(=O)NC2CCC2C)nn(C)c1Br.c1(C(=O)N)cccc(N(C)C)c1 C1(C(C(C)C)NC(C2(CO)CN(C(=O)C(N)=O)C2)=O)CCCCCC1 C1(C(=O)NC(C2CC(F)(F)C2)C#C)CCN(CCC(=O)OC)CC1 N1(C(C2N(C(C)=O)CC(O)C2)=O)CC(NC(c2cccs2)=O)CC(O)C1 C(=O)(C#CC1(C)CCCO1)N1CCC(CCOC)(NC(C(CCCC)C)=O)CC1 C1(CC)CC(C(=O)N(CC)Cc2ncc[nH]2)CCN1C(=O)CC(C)(F)F c1(C(N2CC(O)(CNC(CC(CC)O)=O)C2)=O)cccc2ccoc12 c1(C(N2CC(CC)N(C(=O)Cc3cccc(C)c3)CC2)=O)ccnc2c1CCO2 c1(OC)ccc(Cl)c(Cl)c1C(c1nnnn1C)NCc1ccc2nncn2c1 C1(CNC(C)=O)CCCN(C(CCC2(C#N)CC2)C=O)C1.CCC.C1CC1.N C(=O)(C(C)CCCC(C)=O)N1CC2CC2C1.C1(C(=O)NC)(C(=O)NC)CC1 CCCCC(O)C(C)C(=O)NCC(CCNC(=O)C1CCc2c[nH]nc21)OC C(=O)(C(CC)CCC)Nc1scnc1C(N1CC(O)(C(C)(C)CCC=C)C1)=O C1(C(N2CC(NC(CNC(=O)OCC)=O)C(C)(C)C2)=O)CCc2nc[nH]c2C1 C1(CNC(C(C)c2cncs2)=O)CC2CCC(C1)N2C(C1CCOCC1)=O C1(CNC(Cc2c(C)cc(F)cc2)=O)CCN(C(=O)CC(C)C2CC2)CC(O)C1 C(CN=c1[nH]c(=NCC23CCC(CO2)C3)[nH]c2cccnc12)c1sccc1 C(CCCC(C)(C)C)NC(C(CC1CN(C(CN(C(COC)=O)C)=O)C1)F)=O CC1(C)CN(C(=O)CCS(C)(=O)=O)CC1N=c1nc(-c2cc(F)cc(F)c2)[nH]s1 CCC(C)C(=O)NCC(=O)NCC(C)N(C(c1ccc(C(N)=O)s1)=O)C N1(C(CC2CCC(C)(C)C2)=O)CC(CNC(=O)C(C)(C)C(N)=O)C2(CC2)C1 C=CCC(CC(=O)NCCCCCF)NC(c1cnn(C2CC2)c1)=O c1(C(N2CCC(CNC(c3onc(C)c3C)=O)C2)=O)cccc(C)c1F c1(OC)ccc(C(=O)NCCN(C(=O)C(C)C(C)C)C(C)C)c(Cl)n1.O N1(C(C(C2CC2)OCC)=O)CCC(NC(c2n[nH]c(CC)c2Cl)=O)CC1C CC(C(C)NC(=O)Nc1ccc(-n2ccnc2)nc1)S(C)(=O)=O C1(NC(CSCCN(CC)CC)=O)CN(c2ncc(O)cn2)C2CCCCC12 CC1CCC(C)C1Cc1nnc(C2CN(C(=O)OC(C)(C)C)C2)n1N.CC.O C1(CN(C2CCN(C(C=Cc3ccc(C)s3)=O)CC2)C)CCn2ccnc2C1 c1(C(N2C(CN(C(C(CCOC)OC)=O)C)CCC2)=O)cc2[nH]ccc2s1 CN=c1nc(C(N2CC(N(C)C(c3cnc(C4CC4)s3)=O)C(O)C2)=O)cc(C)[nH]1 N1(C(=O)Cn2ccnc2)CCN(c2ccnc(-c3ccccc3)n2)CC1CCO c1(CN2C(C(=O)Nc3cnc(OC)c(C)c3)CC(=C)C2)ccc2c(c1)CCN2 C1(C)(OC)CCCN(C(=O)C(C(C)C)NC(=O)CC2(O)CCCC2)C1 c1(N2CCCC(C(=O)NC3C(OCC)CN(C)C3)CC2)ncnc2cnn(C)c12 S(=O)(=O)(c1c[nH]ccc1=NC(CC)C1CCC1)NC(C=C)C1CC1c1ccoc1 Cc1cc(O)cc(C)c1C(=O)NCC12CCCN(C(c3cocn3)=O)C1C2 CCC(C)(C)CC(=O)NCCCCCN(C)C(c1cnn(CC2CCCO2)c1)=O Cc1c(C(=O)NC2CC(CNC(C3CCCO3)=O)C2)n[nH]c1-c1ccccc1 C12(NC(C3CC(NC(c4cc(CC)c(C)s4)=O)C3)=O)CCCC1OCC2 C(=O)(C(C(=O)N)OC)OCC.c1(C(N2CC(O)C2)=O)cccnc1.C(C)C c1(C(N2CCCC(CNC(CC3(C=C)CC3)=O)C2)=O)cc2ccnc(Cl)c2s1 c1(C(=O)NC2CCC(N(C(=O)C=Cc3cc[nH]n3)C)CC2)cccc2cnnn12 C(CCC(=O)NC(C)(CNC(=O)CCCC1CCC1)CC)N(CCC)CCC CC1=C(C(=O)N2CCC(NC(C3CCCCN3N=O)=O)CC2C)CCCC1 C1(CCC(=O)NCCN(C(C)C)C(C)C)CCCN(C(C2CC23CC3)=O)C1 N1(C(C2(CC#C)CCCO2)=O)CC(NC(=O)CCCc2nncn2C)C(SC)C1 N1(CC(=O)NC2(CO)CN(C(=O)C(F)CC3CC3)C2)CCCNC1=O C1(NC(C2(OC)CCCOC2)=O)CCN(C(=O)CCn2c(C)ccc2C)C(C)C1 CC1(C)C(NC(C2(n3ccnn3)CC2)=O)CC1CC(=O)NCCF N1(C(c2cc(C)sn2)=O)CCCCC1CN(C(=O)C(C)NC=O)C1CC1 N1(C(C(C)OCCOCC)=O)CC=C(CNC(=O)CC2CC2C)CC1 c1(C(=O)NC2CN(C(c3ncc(C)c(Br)c3)=O)CC2C)cc(C)cc2[nH]ccc12 N1(C(CC(C)SC)=O)CCCCC(CNC(=O)CN(c2ccccc2)C)C1 C1(C(N2C(C(N(CC(F)F)C(C)C)=O)CC2C)=O)CCC(O)CN1C S(=O)(=O)(c1c(Cl)cccc1Br)N1CCN(CC2(CC)CCCCCCC2)CC1 C1(C2CC2)(CNCc2cc(COC3CCCCO3)ccc2)CCNC1 C1(C(NOC(COC)COC)=O)CCN(C(C2CN(C)C2)=O)C1C(C)C Nc1ccc(C(N2CCN(CCCNC(C3CC4C=CC3C4)=O)CC2)=O)nc1 Cn1cc([N+](=O)[O-])c(N2CCC(COC(=O)NC3(O)CCCCCC3)CC2)n1 N1(c2nc(C)nc(C(C)C)c2)CCC2C1CCCN2C(=O)C(C)Cc1ccco1 C(=O)(C1=CN=C2N=CNN2C1)N1CC=CC(NC(c2ccc(N(C)C)nn2)=O)C1 c1(C(=O)NC(CNC(Cc2c(C)n(C)nc2)=O)C2CCC2)ccc(O)c(CO)c1 c1(OC)ncccc1C(=O)N.C1C(C)CCN1C(c1cc(C(N)=O)[nH]n1)=O.C Cc1cc(C(=O)NCC2CCN(C(c3cnnc(Cl)c3)=O)C2)cnc1Cl CC1(C)C(O)CC1(c1ccccc1)NC(=O)C(c1cccc(Cl)c1)N Cc1cc(Cl)nc(Cl)c1C(N1CCCN(C(c2[nH]ncc2C#N)=O)CC1C)=O Cc1ccc(Nc2cc(O)nn2C)c(C#N)c1 Cc1cccc(CCC(=O)N(C)CC2CN(C(C3(C#N)CCCO3)=O)CCO2)c1 c1(OC)cccc2cc(NC(C)CNC(c3ncc(F)cn3)=O)oc12 C1(N(C(=O)CN2CCN(C(=O)CCCF)CC2)C(C)C)CCC1C1CC1 c1(CN2CC3N(C(C4(C)COC4)=O)C(C3)C2)c(Br)cc(F)c(F)c1F C1(CC(=O)N(C(C2CCCN2C(c2ccco2)=O)C)CCC)OCCCC1(C)C C1(C)(C(N2CCC(NC(c3c(C)[nH]cc3)=O)C2)=O)CCCC1(F)F c1(-c2nc(NC(=O)Nc3ccccc3CN3CCOCC3)sn2)cccc(F)c1 N1(C(C=C(C)C(F)F)=O)CC(C)(C(=O)NCCCCO)CC1(C)C CN=c1cc(C(N2CC3(CCCCN3C(C3CC3F)=O)C2)=O)c2ccccc2[nH]1 Cc1noc(C)c1CC(=O)NCC1CCCN1C(C12CC1COC2Br)=O Cc1noc(CCC(=O)NC(C)CC(C)NC(C2(NC(N)=O)CC2)=O)n1 N1(C(c2c(C)n(-c3ccc(F)cc3Br)nn2)=O)CCC2C(O)CCCC2C1 C1(CNC(C2N(CC)CC2)=O)CCCCN(C(c2csc(C(C)=O)c2)=O)C1 c1(CNC(=O)OC(C)(C)C)nc2ccccc2s1.CC1C2CCCN1C2=O C1(NC(C2(NC(CC3C(C)OCC3)=O)CC2(C)C)=O)CC2C(C1)C2(F)F n1(CC(=C)C)nc(-c2ccc(C)c(Cl)c2)nc1C1CCc2nnc(C)n21 N1(C(c2ccc(C(O)CO)cc2)=O)CC2CCN(C(c3sc(Br)cc3Br)=O)C2C1 C(=O)(C(O)CC[S+](C)C)NC1CN(C(C(c2cc(C)sc2)(C)C)=O)CC1O C(N=c1cc(Cl)c(O)n[nH]1)C12CCC(NC(CSSC)=O)(C1)CO2 N1(C(C=C(CCC)C)=O)CCC(C)(C)C(C(=O)NC2CC3CC2C(O)C3O)C1 CCC(C)C(CC(=O)NCC1(C)NC(=O)NC1=O)NC(=O)CC(F)(F)C(F)F C1(NC(Cc2c(C)nc(C)s2)=O)CC2CCC(C1F)N2C(=O)C1=NNC(=O)CC1 CCCC(C(=O)N(C)CCNC(c1c[nH]nc1C1(O)CCOCC1)=O)OCC c1(NC(CC(C)NC(C2(C)C=CCC2)=O)C)ncc([N+](=O)[O-])cc1C(F)(F)F C(c1ccco1)=CC(=O)NC1CCCC1NC(C1CCCO1)=O C1(C(N2CC(C)C2)=O)CCC12CCN(C(=O)CSC(=N)N)CC2 C=CCCCCCC(=O)NC(c1ccccc1)CNC(c1ccc(C)s1)=O CC(C)CC(CNC(C1CC12CCCC2)=O)C(=O)N1CCC(O)C(C)C1 c1(N2CCC(C=C)C2)cc(NCC(c2ncccn2)C)nc(C(F)(F)F)n1 c1(CC(N2CC(CC)C(NC(=O)COCCOC)C2)=O)cnc(Cl)cc1C CC(C)(C(=O)Nc1cccc2c1OCC2)C1=CCN(C(C2CCSC2)=O)C1 c1(C(N(C2CN(C(=O)Cn3cnnn3)CC23CC3)C)=O)cc2c(Cl)ccnc2s1 CCCC(C(=O)N1CCN(C(=O)CN2CC(C)(C)C2)CC1C(F)F)C(C)C C12(CNC(CC3(C)CC(F)(F)C3)=O)CCC1CN(C(c1cc(Cl)ncc1O)=O)C2 N1(C(=O)C(=O)NCc2nccc3ccccc23)CCC2(COCCO2)C1 CC(C)(CC(=O)NCCOCCNC(N)=O)n1cccc1 c1(CC)n[nH]c(=NC2CCCC3CN(C(c4ccn(C)c4)=O)CC23)s1 CN1CCN(C(=NCCCN(c2ccccc2)C)NCCOC(F)F)CC1=O C(=O)(C(Cc1ccco1)C(=O)O)OC.n1(CC)cc(-c2cn(CCO)nn2)cn1 C1(NC(c2cc(C)ncn2)=O)CCCN(C(c2cccc(CO)n2)=O)CC1F N#Cc1ccccc1C(=O)NC1(CCC(=O)N)CCCC1.CC(O)C(F)(F)F.CCO c1(C(N2C(C=CC(=O)N(C)CC3CCOC3)CCC2)=O)occ2c1CCC2 CCCC(C(=O)NCC1(C)COCCN(C(=O)CC2(N(C)C)COC2)C1)C(C)C C(N=c1[nH]c(Cl)ncc1C)C1(O)CCN(C(C(CCC)CC2CCCC2)=O)CC1 C(C(=O)N=c1ccn(CC(N2CCC(O)(CO)CC2)=O)c(O)n1)c1cnc(C)s1 C(=O)(C(CC)CCOC)NC(C1OCCN(C(c2cc(CCC)on2)=O)C1)C N1(C(COCC(C)C)=O)CCC(N(C)C(C2CC3C=CC2O3)=O)C2(CC2)C1 C1(O)(CC#C)CCN(C(=O)C(CCNC(c2nocc2C)=O)OC)CC1 CC1(C)CC(=O)NCC1C(N1CC2CC1CO2)=O.C(=O)C(=O)N=S(C)(C)=O.C C1(CNC(C(=C)CO)=O)(CO)CC2CCC1C2 C1(OC)CC(NC(C23CCC(C2)C3)=O)CN(C(=O)C(C2CCCCC2)O)C1 C(=O)(C1=CC(C)(CC)C1)NC1(C(N(CCC)CC)=O)CC1 C(c1ccc(O)cc1)=CC(N1CC(O)C1)=O.C(=O)(C(CCO)N(C)C)N(C)C C(=O)(C(C)C(O)CC(C)C)NC1(CNC(C(C(CC)CC)F)=O)CCCCCC1 C1(C2CCN(C(C3CC(C)C3)=O)C2)CCCCN1C(C1CC(C(F)(F)F)C1)=O C1(C(=O)NC23CC(C(N(C(CSC)C)C)=O)(C2)C3)CCCCN1C C(CN=c1ccnc[nH]1)C1CCN(C(C2CCCCCC2)=O)CC1 C(C1CCc2cccnc21)NC1CCC(C(=O)OCc2ccncc2)CC1 C1(C(=O)NCCN(C(=O)Cc2ccco2)C)CCC2CC1CO2 C1(NC(c2cncc(COC)c2)=O)CC2(C1)CN(C(=O)C(F)C(F)(F)F)C2 C1(c2n(C(CC)(C)C)nnn2)(NCC2(CO)COC2)CCC2CCCC2C1 C1(NC(CC2CC(C)C2)=O)CN(Cc2cn(C3CCCC=C3Br)nn2)CCO1 c1(CC(=O)NC2(c3c(Cl)cccc3Cl)CC2)ccc2c(c1)OCCCO2 C1(NC(C(CSC)O)=O)CN(C(c2cscc2C(F)(F)F)=O)C2(CCC2)C1 c1(C(N(C(CNC(c2ccc(C(C)=O)o2)=O)C)C)=O)cccc(-n2cccn2)n1 CC(C)(O)C(F)C(=O)N1CCOC(CNC(=O)CCn2cccnc2=O)C1 C12(NC(c3cccc4oc(O)nc34)=O)CCCC1N(c1ncns1)CCC2 C1(C)(CNC(c2ncn(C)n2)=O)CN(C(=O)C)C(C)(C)C1.C(C)C1CC1 N1(C(C(c2ccc(Cl)cc2)(C)O)=O)C2CCCC1CN(C(=O)CC=C(Cl)Cl)C2 CC1CN(Cc2[nH]ccc(=O)c2O)C(C)CN1CCO N1(C(CC=C)=O)CC(CC(=O)NCCC2CCCC2)C(C)C1 c1(SCCC(=O)NC(CNC(COCCOC)=O)C)ccc(OC)nc1Br C=CCC(CC=C)C(=O)N1CCC(C(N2CCC3(CCO3)C2)=O)C1(C)C c1(CO)n[nH]cc1C(N1CCCC1C(C)(C)CNC(=O)Cc1ccoc1)=O c1(C(=O)OC)cc(C(=O)NC2CC(C)(NC(c3ccccc3)=O)C2)nn1C C(C)(CC(C)N=c1[nH]c(Cl)nc2c1COCC2)NC(C(C(CC)C)O)=O CN=S(C)(=O)c1cccc(C(=O)NCCC(O)CNC(=O)Cc2ccccc2)c1 CC(C)C(CC(=O)NC(c1nncn1C)CO)NC(C1CC(CF)C1)=O C1(CS(=O)(=O)N(C2CN(C)C(=O)CC2)C)CCCCC(F)(F)C1 c1(NC(C2C(NC(c3c(C)nc[nH]3)=O)CCC2)=O)cnncc1Br N1(C(C)C)CCCCC1C(N1CCC1CNC(c1cc(-c2ccco2)[nH]n1)=O)=O c1(C(N(CCN(C(c2ccn(CCCC)n2)=O)C)C)=O)cccc(Cl)c1OC c1(C(=O)Nc2ccc3c(c2)CCC3)nc2ncc(CCO)cn2n1 C1(C(=O)NCCF)C=CCN1C(=O)COCCOCc1cccnc1 C(=O)(C1Cc2ccc(Cl)cc21)NCCN(CC(C)O)C(c1ncn(C)n1)=O Cc1ncn(C)c1C(=O)NC(C1CN(C(c2cnn(C(C)C)c2)=O)C1)C N1(C(C(CC)OCC)=O)CCC(C(=O)NCCCc2nncn2C)C12CC2 N1(C(CC)=O)CC(NC(c2cc(-c3ccc(Br)cc3)no2)=O)C2CC12 c1(OC)ccc(C(=O)NC2CCCN(C(C3CC(C(=O)OC)C3)=O)C2C)cc1C C(=O)(C#CC1CCC2(CC1)OCCO2)N1CCC(NC(C(CC=C)(F)F)=O)C1C C1(O)(CNC(C(CC#C)O)=O)CCCN(C(c2cn(C)nc2-c2ccco2)=O)C1 CCC(CN)C(=O)N1CC(CCO)(CO)C1 C1(C(=O)NCC(C)NC(=O)CSc2n[nH]c(=N)s2)C(F)(F)C12CCC2 Cc1ccc(CC(N2CCN(c3cc(C4CC4)ncn3)C(C)C2)=O)c(Cl)c1 CC(C)(O)C(F)C(=O)NC1CCCC1NC(=O)CNC(=O)CC(F)(F)F CCC(C#N)(CC)C(=O)NCCCC(C)(C)NC(c1cc(C)c(CO)cn1)=O C(=O)(CC(C)(C)O)N(C1CCCC1)CCCNC(CC1C(OC)CC1)=O C1(C(N2CCC(N(C(=O)C(C)C=C)CC#C)CC2)=O)CC2C=CCC(C1)C2 CC(C)C(C)C(=O)NC1CC(CNC(=O)C(c2ccccc2F)(F)F)C1 C1(NC(C2(NC(C(CC)CN(C)C)=O)CCCC2)=O)CC2CC(OC)C2C1 c1(CNC(C2C(C)CCS2)=O)cccnc1CNC(=O)C(C)(C)C#N C1(Nc2ccc(-c3ccc(C)s3)c(Cl)c2)CN2CC(C)C1C2 CC1CCCC(OCC(=O)NCC2C3CN(C(c4ccc(F)cc4)=O)CC23)C1 N1(Cc2nnc(C(C)C)o2)CC2CN(C(c3c(Cl)cnn3C)=O)CC2C1 Cc1ccc(C(=O)NCC(C2CC2)NC(=O)C(C)(C)c2ccccc2)o1 c1(CN(C2C(CO)C3CCCC23)C(NCCCC)=S)ccc2c(c1)CCO2 N1(C(c2c(C)cc[nH]2)=O)CC(C)(C)CC1C(=O)NCc1ncn(C(C)C)n1 C1CN(C(C2CC(O)CN2C(C)=O)=O)C(C)(C)C1.CC=O.C(=O)OCC C1(C(=O)NC2CCC2)CC(C2CC2)=NO1.c1(C2(C=O)CCC2)cccnc1.C c1(C(=O)NCCN(CCOC)C(C2CCCCO2)=O)cnc2[nH]nc(O)c2c1 C1(C(N2CC(C)C2)=O)CCC2(CC1)NC(=O)NC2=O.CC(C)(C)C(C#N)C(=O)N C1(C(=O)Nc2c(C)nc(Br)cc2)C2CCCC1CN(C(c1ccc(CO)s1)=O)C2 Cc1nc2cc(NC(=O)CC3CCC(NC(=O)CN(C)C)CC3)cnc2[nH]1 CCC(C)C(C(=O)N1CC(CO)(NC(=O)CCOc2cccnc2)C1)N(C)C Nc1c(-c2noc(C3(C(F)(F)F)N=N3)n2)nc(O)nc1O c1(C(N2CCCC(O)(CCNC(CCC#C)=O)C2)=O)[nH]c(C)c([N+](=O)[O-])c1C N1(CCNC(Cc2nc(C)sc2C)=O)CCCN(C(=O)CN2CC3CC3C2)CC1 c1(C(C2C(C)CN(C(=O)CC3CCCC(F)(F)C3)C2)=O)cc(S(N)(=O)=O)cn1C N1(C(c2c(OCC)cc(Cl)cc2)=O)CCC2CCCC12.c1(C(=O)N)nnc(C)s1 [N-]=[N+]=NC1COCC1NC(C1CC(O)(C)C1)=O.c1(C=O)cc(C(N)=O)co1 N1(C(c2nnc3ccccc3n2)=O)CCC2(CC1)CN(C(c1cc(F)c[nH]1)=O)C2 C1(CC)CN(C)CCCN1C(=O)CC1C(NC(=O)CC2(C)CCOCC2)CC1O N1(C(C(N)=O)=O)CCOCC(NC(=O)CCCNC(=O)CCc2ccccc2)C1 C(=O)(C(F)C(=O)NCC(C)CNC(c1coc(C(N)=O)c1)=O)OCC c1(CC)cn(C2CC3(C(=O)NC4(C)CCSC4)CC23)nn1 c1(CC)ncncc1C(N1CCCC(C(=O)N(C(C)C(F)F)C)C1)=O c1(CC)ccccc1CCNC(=O)CCN1CCCC1.C(=O)(C)N.C(C)=O c1(OCC(=O)NCCC(=C)C)cc(Cl)ccc1C.C(=O)CC.[SH](C)(=O)=O c1(C(=O)NC(C)CC(C)NC(c2ccc(C(N)=O)cn2)=O)cc(O)cc(N)c1Cl C1(N(C)C)CCN(C)C(NC(N2CCNCC2c2ccnn2C)=O)C1 N1(C(C23CC(C)C2C3)=O)CCC(F)(C)C1.c1(C(=O)N)cncc(-n2cccc2)c1 Cc1cncc(OCC(=O)N(C2CCN(c3ccncc3)CC2)C)n1 N1(C(C(n2ncc(C)c2)C)=O)CCC(C=CC(=O)NC2CCOCC2C)CC1 c1(C(=O)NCC2(NC(c3cncn3C)=O)C(C)CCCC2)cccc2occc12 c1(C(N2CCN(C(CCSCCC)=O)C(CCO)C2)=O)ccc(S(C)(=O)=O)o1 CC1CC(NC(C2CC3(CCC3)C2)=O)CN(C(=O)C(O)Cn2cncn2)C1 N(C(=NCCC(C)F)NCc1cnnn1C1CC1)C(C=C)C c1(C(=O)NCCC2CCN(C(C(CCSC)O)=O)C2)ccc(O)c(C)c1C CCCCC(CC)C(=O)NC(C)(CNC(=O)C=Cc1cscn1)CO c1(OC)cc(C(N2CCC2C)=O)ccc1[N+](=O)[O-].C(=O)(C(F)=C1CCCC1)N Cc1nsc(N)c1C(=O)NC(CC(=O)NC1COCC1O)C1CC1 C1(C(=O)Nc2cc(C)c(Br)c(C)c2)Cc2ccccc2CN1C(=O)CC(F)(F)F c1(NC(C(c2cnn(C)c2)N(C(C(CCC)C)=O)CC)=O)ccc(F)c(O)c1 C12(C(=O)NCCCC(=C)Cl)CC(C)(CN1C(c1cc(C)n(C)c1)=O)C2 CC(C)(CC1CCOC1)C(=O)N1CCCC(N(CCO)C(C2CCOC2)=O)C1 CC(CCN(C)C)C(=O)NC(CNC(C1CCC(F)C1)=O)C(C)(C)C C1(CNC(C2(C#N)C(C)(C)C2)=O)CN(C(c2cccs2)=O)CC12CC2 C(=O)(CC(C)CNC(C1CSCN1C(=O)C(C)=C1CCCC1)=O)OC C(=O)(C1CCc2ccccc21)NC1C(C)CN(C(c2ncc(Cl)cc2F)=O)CC1 N1(C(C2OCC(C)C2)=O)CCCC(F)(C(=O)N(C)CCc2ccccn2)C1 N1(C(c2cc(C)c(C)nc2C)=O)CCC2CCN(C(=O)C3=CCCCO3)CC12 N1(C(CC(=C)C)=O)CCC2(NC(=O)CCOC3COC3)CC2C1 CCCCCC(C)CC(=O)NCCC1CCCN1C(=O)C=Cc1ccccc1 CC(C)C(F)C(=O)NCC(C)(C)OCCNC(=O)C.c1cccc(F)c1.O C1(C(N2CC(C(C)NC(Cn3ncc(CC)c3)=O)OCC2)=O)CCCCC(=O)C1 CCCCCC(C)CC(=O)N1CC2CC2C1C(=O)N(C)CCOC c1(C(N2CC(O)(C(C)NC(=O)C)C2)=O)cccc2cc(O)ncc12.C1CC1.S N1(C(CC(C)C)=O)CC(C)OC2(CCN(C(C34CCC(F)(CC3)C4)=O)C2)C1 C(C)(C)(CCC(=O)N1CC(C(N2CC3(CCOC3)C2)=O)C(F)C1)OC Cc1ccc(C(N2CC3CC2CC3NC(C23CC(C)(CCO2)C3)=O)=O)nc1O c1(CN(C(=O)NCC(N2CCSCC2)C)C)ccc(S(N)(=O)=O)cc1 C1(C(=O)NC)CCCCC1N=c1[nH]c(=NCCN(C)C)[nH]c2c1COC2 Cc1ccc(C)c(C(=O)CCc2cn(C(C)C(=O)NCCCC(C)CO)nn2)c1 N1(C(C(C)OCCC(C)C)=O)CCCC2CN(C(C3CCSC(C)C3)=O)CC12 c1(C(CN2C3(C(=O)OC(C)(C)C)CC3CCC2)O)ccc(O)c(Br)c1 C(=O)CC(CN(C)C)C(F)(F)F.C(C(C)C)NCC.C1(C=O)CC1.CC C12(NC(=O)COc3ccccc3)CCCN(C(C3(F)CCCCC3)=O)C1C2 C(=O)(CC(F)(F)C(F)F)NC(C)C(C)(C)NC(=O)CO.c1cccc(F)c1F c1(C(=O)NC2(C)CCN(C(c3cc(F)cc(F)c3)=O)CC2)cnc2c(c1)COC2 C(=O)(CCCCc1csc(CCC)n1)N(C1CCN(CC(=O)NC)CC1)CC#C c1(C(=O)NC2C(CNC(=O)CC=C(Cl)Cl)CC2)nccc2ccccc12 C=CC(CC(=O)N1CC(OCCNC(=O)Cn2ccnc2C)C1)c1ccccc1 C1(F)CCCN(C(=O)CCc2nncs2)CC1.c1(C(=O)NC)ccc([N+](=O)[O-])[nH]1 CC1=NNC(=O)C1CC(=O)NC(C)C.c1(C2CC(C=O)C2)ccc(Cl)cc1.N N1(C(C(C)OCC)=O)CCc2nc[nH]c2C12CCN(C(c1n[nH]c(O)n1)=O)C2 C1CN(C(=O)C(C)(C)C)CCO1.c1(CCC(=O)N(C)C)nnc(C(F)(F)F)o1 C(C(CC(C)C)N(C)C)NC(C(C1CN(C(COCCC)=O)C1)OC)=O N1(C(c2nn(C)c(Cl)c2)=O)CC2CCCC(CNC(C3CCCOCC3)=O)(C2)C1 CCCC(CCC)=CC(=O)NCC(C)CN(C(=O)CC1CC1C1CC1)C N1(C(C(C)OCC=C)=O)CC(N(C(=O)Cn2cnnn2)CC)CC12CCOCC2 C(=O)(C(C)CC(C)(C)C)NC1CN(C(C=C(C)C(C)C)=O)CC1C C(C(=O)N(C)Cc1ncccn1)(C(C)OC)NC(C1CN(CC)C1)=O c1(C(N2C(CNC(C3=NOC(C)C3)=O)CC2)=O)cc2c(Br)cccc2o1 C1(OC(C)C)CC(CC(N2CC(N(C)C)C(C)C2)=O)C1(C)C CCC(C(=O)OC)C(=O)N1CCCC(N(C)C(C2CCCS2)=O)CC1 C1(NC(C=CC(C)C)=O)CN(C(=O)CCc2cnoc2)CC1C1CC1 C(CN=c1nc(N(C)CCc2ccccn2)cc(C)[nH]1)C1(OC)CCC1 C1CC2CCC(C1)N2C(C12CCN(CC1)C2)=O.C(CC1CCCC1)(C=O)OC.N C1(F)(C(=O)OC)CC1C(=O)NCCCNC(=O)CCC1CCC1 c1(C(C)(C)C)cccc(C(=O)NCC2CCN(C(C3CC(F)C3)=O)CC2)n1 c1(NC(CC)=O)cccc(NC(C2(Br)CC2(C)C)=O)c1 n1(CC(=O)NCC(CN(C(=O)CNS(=O)(=O)NC)C)O)cc(CO)nn1 Cc1cnc2c(C(=O)NCC(C)NC(c3c[nH]nc3C3CCC3)=O)cccn12 N1(C(=O)NCC2CCC(=O)NC2)CCCC(CC2(O)COC2)CC1 N1(C(C(C(C)CNC(=O)CCN(C)C)F)=O)CCc2c[nH]nc2C1 N1(C(COCCC)=O)CCCC2CN(C(C3(CO)CCCO3)=O)CC12 c1(C(=O)NCC(C2CCCN(C(C(C)(C)O)=O)C2)(C)O)ccc(C2CC2)nc1O N1(C(=O)C(F)Cl)CC2C(c3ccccc3)(C1)CS2(=O)=O.c12cc-1c1cn[nH]c1c2 C12(COC)CCC(C(=O)N)(CC1)CO2.C1(C=O)C2CCC(=O)C12.C1CC1 N1(C(C2(C)CC(=C)C2)=O)CC2CC2(C(=O)NC(c2nncs2)C)C1 c1(C(N2CCCN(C(CCC#C)=O)C(C(C)C)C2)=O)cnc2ccncc2c1 N1(C(C(CC)O)=O)CCN(C)C(C(N2CC(OC)CC2CF)=O)C1 C1(NC(C2CC(=C)C2)=O)C=CCC(C(=O)NCC2CCCCC2)C1.CCO.O CCCCC(C)(F)C(=O)NCc1nc(C(=O)N(C(C)CC)C)c(C)o1 N1(C(CC2N(C)CCC2)=O)CCC(CC(=O)NC2CC(CO)C23CCC3)C1(C)C C1(C(N(CCCO)CCC)=O)CC(C)CN1C(=O)C(C)SC(C)C C1(NC(C2CC23CC3)=O)CCN(C(c2ccccc2CO)=O)CC1 c1(C(N(CCNC(=O)CCn2cccc2)CC)=O)ccc2c(c1)ncn2C.C C(=O)(CC1=CCCCC1)N1C(C)C(NC(C2CC2[N+](=O)[O-])=O)CC1 c1(C(=O)NC)c(F)ccc(Cl)c1[N+](=O)[O-].C1(F)CCN(C(c2nn[nH]c2Cl)=O)C1 Cc1cncc2cc(C(=O)NC(C)CCCCNC(=O)C(CCO)N(C)C)sc12 N1(C(c2cn(CC)nc2C2CC2)=O)CCC2(CC1)CN(C(C1CCCSC1)=O)C2 N1(C(c2c(CC)nccc2)=O)CCC2CCCN(C(=O)CCC(F)F)C2C1 c1(C(N2CC(NC(=O)CCN3CCC(F)C3)C3C(C2)C3)=O)ccc2n[nH]cc2c1 C1(C2CN(C(c3ccccc3F)=O)C2)(NC(c2cc(CC)n(CCO)n2)=O)CC1 c1(C(C(=O)NCC=C)N(CCF)CC)ccccc1COC N1(C(c2n(CCC)ccc2)=O)CC2CC(C(=O)NCCC(C)O)(C2)C1 C#Cc1cc(C(N2CCC3(NC(=O)Cn4cnnc4O)CC3C2)=O)cc(F)c1 c1(N2CCC(NC(C(c3ccccc3)N(C)C)=O)C2)ncc(C#N)cc1F C(C(F)(F)F)(CC(C)=CC(=O)NC(=O)CC=C(C)C)C1CC1 c1(CC)nonc1CN1CCCC1CC(N1CCSCC1)=O C1(CC(=O)NCC(C)N(C(C2CC(C(C)C)C2)=O)C)CCC(=O)C1C c1(NC2CCCC(C(C)C)C2)ccc(S(=O)(=O)NC(C)(C)CC2CC2)cc1Br c1(N(C2CC3CNC2C3)C)cc(C(N2C3CCCC2C3)=O)ccc1F C(=O)(CC(C)CC(=O)N1CC2CC2(C)C1)OC.C1(C(=O)N)CN2CCC1(C)CC2 c1(C(C)NC(C2(F)CN(C(COC(C)C)=O)C2)=O)cccc(Cl)c1 c1(NC(C2CC(OC)CN2C(=O)CC(C)C(F)F)=O)cc(O)cc(F)c1 C1(C(N2CC(C)=C(C)C2)=O)CC2CC1CC2NC(=O)C(F)OC(F)(F)F C1(NC(COC(CC)(C)C)=O)CCC2CN(C(c3cnc4n3CCS4)=O)CC2C1 CCCCC(C(=O)N1CC(C(=O)NC(CC(C)C)C(N)=O)CC1(C)C)C(C)C C#CC1(C(N2CCC(CC(=O)OC)C2)=O)CCN(C(c2occc2CC)=O)C1 C(C=O)(C(C)C)NC(=O)OCC.C1CC1.C1(C=O)(CC)CC1.C=O C1(C)(CCC(=O)NCc2c(C)csc2)CCCN1C(c1cc(=N)[nH][nH]1)=O CC(C)(CC(F)(F)F)C=O.C1(S(C)(=O)=O)(C(N2CCC(CC)C2)=O)CCC1.N c1(OCC(=O)N(C)CCNC(=O)C(C)(C)OC(F)F)cccc(Br)c1F c1(C(N2CC(CN(C(CCC)=O)C)C2)=O)cnc2ccc(C)cc2c1 C1(C=O)CC2CC1C1CC21.C1(COC(C)C(=O)N2CC(CC)C2)CCCCO1.N N1(C(C2(SC)CC2)=O)C2CCCC1CN(C(c1c(S(N)(=O)=O)cnn1C)=O)C2 C#CCC(CC(F)F)C(=O)N(CCC(=O)NC(C)C(C)O)CCCO C=Cn1nncc1C(=O)NCC(CO)NC(C1CC(=O)C1C(C)(C)C)=O CC1(C)C2CC1CN(C(=O)C(CC(N)=O)NC(=O)CC1CC=CC1)C2 CC1CC(NC(=O)CC2(C(N)=O)CC2)CN(C(=O)C(F)(F)c2cncs2)C1 c1(C(=O)NCC(C)(C)CC2CN(C(=O)CCC(N)=O)C2)ccc(CF)cc1 Cc1ccc(C(N)=O)cc1C(=O)NC1C2CN(C(C3CSC3)=O)CC12 N1(C(C2(C)CCOCC2)=O)CCC2(C1)CN(C(C1CC3OC(=O)OC3C1)=O)C2 c1(C(N2C3C(NC(C(=O)NC(C)C)=O)CC(C3)C2)=O)nncc2c1CCCC2 Cc1ccccc1OCC(N1CC=CC(NC(C2CC2C(C)(F)F)=O)C1)=O c1(C(N2CC(O)(C(C(N3CCC(C(C)O)CC3)=O)F)C2)=O)occ2c1CCC2 C(=O)(C1CCc2ccc(Cl)nc21)N(CCNC(=O)C(C)(C)CSC)CC C1(OC)(C)CCN(C(c2cc(C)nc(N(C)C)n2)=O)CC1.C(=O)C(C)N(C)C Cc1ncc(C(=O)NC(C)(C)CC(=O)NC2(C(O)CO)CCC2)cn1 Cc1c(Br)noc1C(=O)NC(C)C(CO)NC(C1CCCN(C)C1)=O CCC1=C(C(=O)NCC2CN(C(C3CCCSC3)=O)CCC23CCC3)SCCO1 c1(C(=O)OC)ccccc1CC(=O)N(CCCCNC(c1cnc(NC)s1)=O)C CCCC(C(=O)N1CCC(N(C(=O)CN(C(=O)COCC)C)C)CC1)C(C)C Cc1cc(C)nc(SCC(=O)NC2CCCC2NC(c2ncn(C)n2)=O)n1 c1(C(=O)NCCC(=C)CNC(=O)CC(C)F)cc2c(F)c(F)ccc2[nH]1 c1(C(=O)NC2CC(CNC(C)=O)C2)ccc(Cl)c(C(F)F)c1 N(C1CCCc2nn(C)cc21)c1cc(C)c(F)c(C)c1 N(C1CCc2c(F)cccc21)C(c1c2ccccc2nn1C)C N1(C(=O)C=CC2CCCO2)CCC2(CC1)COC(CNC(C13CC1C3)=O)C2 C1(C(N2C(C(N3CCC(C=C)C3)=O)CC2)=O)CC(=O)CC12CCC2 N1(C(C)=O)CC(NC(c2cnc(Sc3ccccn3)cc2C)=O)C(C)(C)C1 c1(C(N(C2CCN(C(C3CC4CCC3O4)=O)C2)CC)=O)cn(C)c(O)n1 Cc1ccc(C(=O)NCCC2C(C)CCCN2C(=O)Cc2nonc2C)c(F)c1 c1(NCC(CC)C)ncc(C)cc1S(=O)(=O)NCC(C)CN1CCOC1=O c1ccc([N+](=O)[O-])cc1.N#Cc1cccnc1NC(N1CC(O)CCC1CO)=O Cc1ccnc(C(O)C(=O)NCC(c2ccccc2)CO)c1 N1(C(CNC(C)=O)=O)CC(NC(c2sc(-c3ccccn3)nc2C)=O)C2CC2C1 C1(C(=O)NC2CN(C(C(C)n3cccn3)=O)C2)CCCN1C1CCCCC1 C1(NC(C(C=CC)O)=O)CN(C(c2cc(C(N)=O)cs2)=O)C2(CCOC2)C1 C1CN(C(c2ccnc(O)c2)=O)CC12CCC2.c1(C(=O)NC)snnc1C(F)F c1(C(=O)NCC2CC(C)N(c3ncns3)C2)ccc(=O)n(C)c1 O=C(CC(C1CC1)C1CC1)NCC1CC1CNC(C1CC(O)C1)=O N1(C(CCSCC(C)C)=O)CC(C)CN(C(C2(c3nccs3)CC2)=O)C(C)C1 N1(C(c2c(C(C)(C)C)noc2)=O)CCCC(NC(c2c[nH]nn2)=O)C1.C1CC1.C CCC(C)(C)CC(c1nnnn1CCSCC)NCC1(CO)CCOC1 C1(CNC(c2scc(C)c2)=O)CN(C(=O)C(C)n2cccn2)CCC12CCC2 c1(C(N2CC3C(NC(c4cc(N)c(Br)cc4)=O)(C3)C2)=O)cn2c(n1)CCCC2 C1(CCC)CN(C(C2CCCOC2C)=O)CC1NC(C1OCCCO1)=O C1(C)(CNC(c2cc(CCC)n(C)n2)=O)CN(C(C2CCC2)=O)C(C)(C)C1 N1(C(C(=C(C)C2CC2)F)=O)CC(NC(c2n[nH]cc2C(C)C)=O)C(O)C1 N1(C(c2c(C)c(F)c(F)cc2)=O)CC2CC(C)N(C(C3CCCOC3)=O)C2C1 C#CC1CCC(NC(c2c[nH]nc2CNC(=O)C=Cc2cncn2C)=O)C1 CCC(C(=O)OC)C(=O)NC1(C(=O)NCC2CCC(F)(F)C2)CCN(C)C1 C1(NC(c2cc(OC)cnc2)=O)CC2CCC(C1)N2C(=O)C(CCS(C)=O)OC N1(C(C2CCCN(C(=O)COC3CCOC3)CC2)=O)CCCC2CCCCC12 c1(C(=O)NC2CC2NC(C2CC(F)C2)=O)ccc2c(c1[N+](=O)[O-])OCCCO2 N1(C(C(F)=CC)=O)CCn2c(CNC(C3CCCCC3C)=O)nnc2C1 c1(C(N2CC(CN(C(=O)C=C(Cl)Cl)C)OCC2)=O)c(O)cnc2ccccc12 C1(C(=O)NCCC(C(C)C)NC(c2ncc(C)nc2)=O)CC2CCC(C1)O2 C(=O)(CC(C)CC(=O)NC1CCN(C(=O)Cc2ccc(C)s2)CCC1CO)OC C1(NC(C(C(C)C)C)=O)CCCCCCC1NC(=O)CCN(CCC(C)(C)C)C CCCCCC(CC)C(=O)N1CCN(C)C(C(=O)NOCCF)C1 C(=O)(C1=CCCC(C)(C)C1)N1CCC(NC(C=Cc2c(C)ncs2)=O)C(O)C1 C1(N(C(CCNS(CC)(=O)=O)=O)CCO)CCN(C(c2cc(CO)no2)=O)C1 N1(C(CCCC#C)=O)CCC(C#C)(C(=O)NCC2CC2Cl)CC1 CC1CN(C(c2cc(C3CC3)no2)=O)CC(C)N(C(=O)COCCN(C)C)C1 CN1CCC(CO)(CNC(C2CC(F)CCN2C(c2nocc2Cl)=O)=O)C1 c1(OC)ccc(N(C(=O)C(C)(C)N)CC(C)C#N)cc1.c1(CC)ccc(C)cc1 C1(NC(=O)Cc2cc(C(F)(F)F)n[nH]2)CCCC2CN(C(C3CCCO3)=O)CC12 N1(CC(=O)NCc2cccc(NC(c3cccs3)=O)c2)CC2CC(O)C2C1 CCS(=O)(=O)CC(=O)NC1COCCC1NC(C1CCN(C(C)=O)C1)=O C1(NC(CCN(C(=O)C=Cc2nccs2)CC#C)=O)CC1C1CC1C C(=O)(CC(O)CC(C)C)NC1CCC(NC(CSCc2c(C)noc2C)=O)C1 c1(C(=O)NCC2(COCC)CCC2)cc(O)nc2c1c(C)nn2C c1(C(N2CCCC(NC(C(C)C(C)(C)C)=O)CC2)=O)nccc2ccncc12 N1(C(C(CCC)C#N)=O)CC2CCN(C(C3(CCS(N)(=O)=O)CCC3)=O)CC2C1 N1(C(C2CCN(CCC#C)CC2)=O)CC2CCC2(CNC(=O)CN(C)C)C1 c1(C(CC(=O)NCC(C)NC(=O)Cc2cnc(O)nc2O)C)ccc(F)cc1F CC1C(C(=O)NC2COCCC2NC(c2sc(Cl)cc2Cl)=O)CCN1C CC(c1cccc(Cl)c1)=CC(=O)NCC1COCCN1C(C1OCC1(C)C)=O C12(CNC(C(C)Cn3ccnc3)=O)CCC1CN(C(=O)CCCC(=O)C1CC1)C2 C1(CC=O)CC(C)(C)OC(C)(C)C1.C12CC(C1)C2.C(C)(C=O)SC(C)C C1(CC(=O)NCC(C)(CO)OC)(NC(C2CCCC2C)=O)CCCCC1 c1(CNC(CC2CC(C)N(C(=O)C(=O)N(C)C)C2)=O)cccc(F)c1F C(c1cnn(C)c1)=CC(=O)NCCN(C(=O)C(O)CC1CCOCC1)C C(=O)(CCCC1CCC1)NC(C)C.c1(C2(C(=O)NO)CC2)cccnc1 C(=O)(C1=C(C)OCCC1)N.c1(C(N(CCCC)CC)=O)cc(C2(C)CC2)on1 C(=O)(CS(C)(=O)=O)NCCC1CCN(C(CCNS(CC)(=O)=O)=O)C1 c1(CC(N2CC(O)(CN(C(C(CCC)O)=O)C)C2)=O)ccc(S(N)(=O)=O)s1 Cc1[nH]ccc(=NC(=O)C2CCCN(S(=O)(=O)CC3CCC3)C2)c1F C1(CNC(c2ccc(N)c(F)n2)=O)CC2CCC(C1)N2C(C1CCOC1)=O c1(C(C(=O)N(CCCCO)C)NC(=O)C=CCO)ccnn1C O=C1CC(C(=O)N2CCN(C(C3CCN(c4ncccn4)CC3)=O)C3CC23)=NN1 c1(C(=O)NCC(C)CNC(C2(Br)CC2(C)C)=O)cccnc1O C#CCC(CC#C)C(=O)N(C(C)CNC(c1sc(C)c(Br)c1C)=O)CC O=C(C1CCOc2c(F)cccc21)N1CCC(CN=c2ccnc(C3CC3)[nH]2)C1 C(C(C)C(F)(F)F)N(C(CN(CC(=O)NC(C)C)C)=O)C.C(=O)C(C)C c1(C(=O)Nc2c(OCC)cccn2)ccc2c(c1)S(=O)(=O)N=C1N=CNN21 C1(C(N(CCC(=O)OC)C)=O)C(O)CCN1C(=O)C(C)N=[N+]=[N-] CN1C(=O)c2ccc(NC(N3CCN(Cc4ccccc4F)CC3)=O)cc2C1=O N1(C(COCC=C)=O)CCOCC1CC(=O)N(C)CC1COC(=O)N1 c1(C(=O)OC)cc(C)cc(NC2(c3nnnn3CC(F)F)CC(C(C)C)C2)c1C c1(CCC)nnsc1C(=O)NC1COCC1CNC(c1coc(Cl)c1)=O c1(C(N2CCN(C(=O)C(F)=CC3CC3)CC2)=O)n[nH]c2c1CS(=O)(=O)CC2 Cc1ccncc1C(C)(C)C(=O)N(C)CC1CCN(C(=O)C(F)n2cccn2)C1 C(=O)(CCCc1ccccc1)NC(CNC(CSCC#C)=O)C1CCC1 N1(C(COC)=O)CC(C(N2CC3CC(OC)C3C2)=O)CC(C)(C)C1 c1(OC)cc(S(=O)(=O)N2CC(C)OC3(CCC3)C2)ccc1[N+](=O)[O-] N1(C(C2(C(C)C)CCCN2C(c2nc(Cl)cs2)=O)=O)CCS(=N)(=O)CC1 CC(C(=O)N(C)OCC(F)(F)F)NC(=O)CC(F)(F)F c1(CNc2ncc(COC)s2)ccc(C2CC2)cn1 C(=O)(C(CC)C=O)OCC.C1(C)(C(N(CC(C)(C)C)C)=O)CC2(CC2)C1 N1(CC=CC(=O)Oc2c(C#N)ccs2)CCC(c2ccccc2)C(O)C1 C1(n2cc(CC(C=C)O)nn2)CN(C(=O)C(CC)OCC)CC1C(=O)O N1(C(C(C)OCCCC)=O)CCC(C)(NC(c2ccc(Br)nc2N)=O)CC1 c1(C(=O)NCC(CC(C)C)NC(C(CC#C)O)=O)ccc2occ(C)c2c1 CCCCCCC(F)C(=O)N1CCCC(O)(CNC(C2CC(C)(C)C2)=O)CC1 N1(C(c2c(C)csc2)=O)CCC2CN(C(c3cnn(C4CC4)c3C)=O)CCC2C1 C(C(=O)NC1CN(C(=O)C2=COCC2)CCC1C)(C(C)(C)C)NC(C)=O C1(C(N2CCC(OC)CC2)=O)CN(C(c2ccc(Cn3ccnn3)o2)=O)C(=O)O1 N1(C(C)=O)CCCCC1C(N1CCCC1CNC(=O)C(C)CN(C)C)=O N1(C(c2ccc(-c3ccccn3)s2)C(=O)N)CCn2c(cnc2Br)C1.C(C)OCC C1(C)(C(N2CC3CCC2C3)=O)CCC(F)(F)CC1.CC(C)C=CC(=O)N.C CCCC(CCCC1CC1)N=c1[nH]c(=NC(C)CCO)[nH]c2c1CCCCC2 N1(C(C2CC2)=O)CCN(C(C2CCCNS2(=O)=O)=O)C(CCO)C1.CC(C)(C)O C1(CNC(COc2cccc(C)c2)=O)CCCCN(C2CCNC2=O)C1 Cc1nonc1CNC(=O)CCN(C(=O)CCc1nc(=N)[nH][nH]1)CCCO c1(CCC(=O)NCC(C)NC(CC(=O)NCC#C)=O)cccc(F)c1 CC1CN(C(=O)CC2CSC2)CC(C)N(C(=O)CC(C)(C)c2cccs2)C1 c1(N(C)CC2CCCCO2)nc2c(c(=NCc3cc(Cl)ccc3Cl)[nH]1)CCC2 C1(CNC(C(=Cc2ccco2)C)=O)CC12CCC2.C1(C=O)C2CC3C(C2)C13 C1(CNC(c2cn(CCC(C)C)nn2)=O)CC(NC(=O)CCC#N)C12CCC2 N1(C(C2CC(=C)C2)=O)CCC2(CC1)CC2C=O.c1sc2c(c1C(N)=O)CCC2 Cc1cc(C(=O)NCC2CN(C(C3CCC(=O)N3)=O)CCO2)ncn1 C1(C(N2CCCC(NC(c3cnc(N(C)C)s3)=O)C2)=O)CCOCC1(C)C N#Cc1ccccc1S(=O)(=O)NCC1(O)CN(C(=O)Cc2ccccc2O)C1 N1(C(C(CC(=C)C)C)=O)CC2(COC(C)C2)C1.C1(C(=O)N)CC2(C1)CC21CC1 N1(C(C2C(CC)OCC2)=O)CCCCC12CC(NC(C1CC1)=O)C2.C(C)C.C C12(C(=O)NCCCC=C)COCC1CN(C(=O)CC(N)CCSC)C2 CN1CCC(C)(C(=O)N(CCC(N2CCC(OCCF)C2)=O)CC2CC2)C1 N(C(=NCCCF)N1CCc2cccc(C)c2C1)CC1(CC)CCOCC1 C#Cc1ccc(C2CC2C(=O)NCCC2CC2)cc1.C1(C(=O)N)CC(O)C1 c1(C(=O)NC(C2CCCCC2)CNC(C(C)SC)=O)c[nH]cc1C(C)(C)C N(C1CCC(NC(C2CC3(CSC3)C2)=O)c2ccccc21)C(C1=NNC(=O)C1)=O c1(NC(C(COC)OC)=O)cccc(NC(c2sc(Cl)cc2Cl)=O)c1 CC1CCC(O)(C(=O)NC2CCC(CN=c3[nH]nc(CO)s3)C2)CC1 c1(C(=O)NC2(COC)CCN(C(c3cccc(F)c3)=O)C2)ncnc(O)c1Cl CC(C)CC(F)C(=O)NCc1cn(CC2CC2)nn1.C(=O)C(F)C1CCOC1 C1(C(=O)NCCN(CCC)C(c2ccccc2N)=O)CCC2C(C1)C2(F)F.C N1(C(c2c(CC)occ2)=O)CCCC(C)(C)C1C(=O)NCCC(Cl)Cl C(c1ccco1)=CC(=O)NCCN(C1CCCC1)C(=O)CCN.C1CCCO1 O=S(=O)(CCNC(CC(F)(F)F)c1ccc(Cl)cc1)C1CC1 C1(CNC(C2(C)CN(C(C3(C)CC(=C)C3)=O)C2)=O)CCCC(C)O1 C1(COC)(CNC(=O)CC2CCC2)CCCCO1.c1(C=O)cnnn1C.N N1(C(c2cn(CC(C)C)nc2)=O)CCN(C(C2CC(=O)N(C)C2)=O)CC1CC Cc1ccc2oc(C(=O)NC3CN(C(c4ccon4)=O)C4(CCOC4)C3)cc2n1 Cc1nc(CNC(=O)CSC(F)(F)F)oc1C(=O)N.C1CC1.C1CC1 N1(C(c2cnc(C)[nH]2)=O)CC2CC(NC(=O)CCSC(F)(F)F)C2C1 c1(C(N(CCNC(CCN(C)CCO)=O)C)=O)c2c(nn1C)CCCC2 Cc1ccc(C(=O)NCCC(=O)NOCCCC(F)(F)F)cc1C c1(C(C)C)n[nH]c(=NC2CC3CC(C2)N(C(c2ccccc2OC(F)F)=O)C3)o1 c1(C(N2CCCC(N(C(CC(C)C3CC3)=O)C)CC2)=O)cc(F)c2cn[nH]c2c1 C(=O)(C1=CC2CCCCCC12)N(C)CCNC(c1ccc([N+](=O)[O-])cn1)=O N1(C(c2cn(C)nc2)=O)CCC(NC(C2CC(C)(C(C)(C)C)C2)=O)CC(O)C1 c1(-c2cc(OCC)c(C)cc2)n[nH]c2cccc(C(=O)NC(c3ccno3)C)c12 C1(F)(CNC(CCOCC#C)=O)CCN(C(C2CCC(C)(O)CC2)=O)CC1 C(C(O)C(=O)NC1CC(CNC(c2ccc(-c3ccc(C)o3)s2)=O)C1)OC N1(C(CNC(=O)NC)=O)CCC2(C(N3CCC(C)(C4CC4)C3)=O)CCCC12 CCCCCC(O)CC(=O)NC1CCCCC1NC(=O)Cc1cnn(C2CC2)c1 N1(C(c2n(CC)c(O)nc2)=O)CCC2(CCCN2C(c2ccsc2C#N)=O)C1 CC(C)(C(=O)NCCC1(CNC(C2CC2(Cl)Cl)=O)CC1)C1CCCO1 c1(C(N2CCN(C(C3CCC(=C)CC3)=O)C3C2C3)=O)cc(F)c(F)cc1Br c1(CNC(C=CCN(C(C(C)OCC=C)=O)C)=O)ccc(C)c(C)c1 C1(CC=O)CCC(=O)NC1=O.N1(C(c2[nH]cc(C(C)=O)c2)=O)CCC(C)(C)C1 C(C)(C1CCCCC1)=CC=O.CCC(C)C(=O)NCC(=O)NC1CCCC1.C C1(C)CCCN1C(=O)C=CC1CC1.c1(C=O)cnn(CC(F)(F)F)c1C.CC C1(O)(CN(C)C(c2cc(C3CCC3)[nH]n2)=O)CCN(C(C2CCCOCC2)=O)C1 c1(C(N(C(C)C)CCN(C)C(c2cnc(C3CC3)s2)=O)=O)nccc(N)c1Cl c1(CCC=O)ccnn1C.C(C(=O)NCCC1CC1)OC.C(C)(C)C.C=O c12ccc(F)c(c1F)C(=O)O2.C1(NCC)CN(C(c2nccs2)=O)C1 Cc1cc(N(S(=O)(=O)c2cccnc2)CC2CCCO2)cc([N+](=O)[O-])c1 CC(CN(C(=O)C(n1cnc2ccccc12)C)C)N=c1ccnc(C2CCC2)[nH]1 c1(C(=O)NC(C(C)NC(C2(CC#C)CCOC2)=O)CO)cncc(OC)c1C C(CCCCCN=c1ccnc(CC2CC2)[nH]1)NC(CC(CCCCC)C)=O C1(Nc2ccc(C(C)=O)cn2)CCC2CN(C(c3csnc3C)=O)CC12 C(=O)(C(CCN(C)C)N(C)C)N(CCC(=O)NCCC=C=C)C CN1CC(Nc2ncnc(NCCc3c[nH]c4ccccc34)c2N)C2(CC2)C1=O C(C(C)CC(=O)NCC1CC1CNC(=O)C=C1CCC1)OC c1(C=O)cc2n(c1)CCCC2.N1(C(C2C(C(=O)OCC)C2)=O)CC(C)C1 C1(C)(C(=O)NC(C)C(=O)NCc2cc[nH]n2)CC=CC1 N1(C(C(n2c(C)cc(C)n2)C)=O)CC(F)(F)CC1(C)C.c1(C=O)cnc(Cl)[nH]1.N CC1OCCN(C(C2COC(=O)N2)=O)C1C(N1CC(F)(CO)C1)=O c1(C=O)nn2c(c1C)CCCC2.C(=O)(C(C)C(=O)NCC1COCC1)OC.C c1(C(=O)NCC2(NC(C3CCCOC3)=O)CC2)cccn2nccc12 C1(C(N2CCC=C(CNC(C3C(C)OCCC3)=O)C2)=O)CC2(C1)CC(C)(C)C2 CC1(C)CC(C)(C)CN1C(C1CCCN1c1nccs1)=O.C(=O)(C1=CCCC1)N N1(C(C2CCCN(C)C2)=O)CC(C(=O)NCc2cccc(F)n2)C2(CCC2)C1 c1(CC(=O)NCC2CN(C(CCC)=O)C3C2C3)csc2ccccc12 c1(OC)cc(S(=O)(=O)N2CCC(c3cccc(C(F)(F)F)c3)C2(C)C)cnc1Cl N1(C(CCC(C)OC)=O)Cc2n[nH]cc2C1C(=O)NC(C1CCOCC1)C c1(-c2cc(C(=O)OC(C)(C)C)ncc2)ccc2c(c1)S(=O)(=O)NC(=O)N2 N1(C(CNC(c2c(OC)nsc2)=O)C)CCN(C(C2SCC=C2C)=O)CC1 C1(CCC)CCCN(C(=O)CC)CC1.n1(CC(=O)N(CC(C)C)C)cc(Cl)cn1 CCC(C)CCC(=O)N1CC(NC(=O)CN2CCSCC2)C(c2ccccc2)C1 C(=O)(C(F)C=O)OCC.C(=O)(C(C)Cc1ccccc1)N(C(C)C1CC1)C Cc1nc(C)c(C(=O)N(C(=O)CCNC(C2CC3CCC2C3)C)C)s1 C1(C(=O)NC(C)CCNC(=O)Cc2cnc[nH]2)CCC2(CCOCC2)O1 C1(CNC(c2nc(C)sc2C)=O)CN(C(c2cnn(C)n2)=O)CC1(F)CO CCCCC(C)CCC(=O)N1CC(CNC(c2cc(C)nn2C)=O)CC12CCC2 c1(NC)nc(C)ccc1C(=O)NCC(CC(C)C)NC(=O)C(C)CCCOC N1(C(C(CC(C)C)C)=O)CCN(C(C2CC(=O)N2)=O)CCC1C C(=O)(CCCN=[N+]=[N-])NCC1C(CC)CCN1C(C1CCOCC1)=O O=C(C1=C2CCN=C2NC=C1)NCC1CCCC1NC(c1ccc(F)cc1Cl)=O c1(C(=O)NCC2(C)CCCN(C(C(C)SC)=O)C2)ccc2c(n1)CCC2 Cc1cc(C)n(CCCC(=O)NCC2CC(NC(=O)CC3(C)CCCO3)C2)n1 CC(C)CC(O)C(C)C(=O)N1CCC(C(=O)N(C(C)CO)C)O1 CC1C(C(=O)N2CC(CNC(C3(CCCF)CC3)=O)CC(C)(C)C2)=NOC1C CP(C)(=O)CC(=O)NCC1CC2CC2N1C(C1CC1Cc1ccccc1)=O Cc1cnc2c(C(N3CC4C(C)C4C3)=O)c(C)nn2c1.C1(CC(=O)N)C=CCC1 N1(C(C2(COC)CC2)=O)CC2CCCC(C)C2C1.c1(C(=O)N)oc(C)nc1C c1(OCN2CC(OC(C3C(C)(C)C3)=O)C2)cccc2c1OCC2 c1(OC)c[nH]c2nc[nH]c(=NCC3CC4(CCCCN4C(=O)C(C)C(C)C)C3)c12 C(CCCC(=O)N(C(C)CN(C)C(c1cnc(C(C)O)s1)=O)C)OC c12cnc(nc1)N1CC(C1)NC2=O.C(=O)(C(F)CC1CCCCC1)OCC Cc1ncnc(C)c1C(=O)NC(C)CC(C)NC(C1CCCC(=O)CC1)=O Cc1c(C(=O)NCC(C)(C)CN(C)C(C2CC2F)=O)ccc(C(F)(F)F)c1F c1(C(=O)NCC(C)CNC(=O)COc2cccc(F)n2)cnn2c1CCC2 Cn1ccc(C(=O)NC2CC2NC(=O)O)n1.C12(F)CC1C2.c1ccccc1 C1(C=O)CC(=O)C12CCC2.C(=O)(CCCOCCO)N1CC(N(C)CC)C1.N C1(CC#C)(C(=O)NC2(C(=O)O)CC2)CCN(C(=O)OC(C)(C)C)CC1 C(=O)(C(CC(F)F)NC(=O)C=CC)NCC.C1(CC)(CC)CCCC1.O N1(C(C=CCC)=O)CCC(NC(=O)COc2ccc(Cl)cc2C)C(F)C1 C(=O)(C(C)(C)C(C)NC(c1ccnn1COC)=O)NCCCOC=C N1(C(=O)CSC2CC2)CCCC(F)(C(N2CC3CCC=CC23)=O)C1 Cc1cc(C(=O)N(CCC)C)ccc1S(N)(=O)=O.c1(C(=O)N)csc(C(F)F)c1 N1(C(CS(CC)=O)=O)CC(C2CN(C(C3CS(=O)(=O)C3)=O)C2)C1 c1(OC)nn(C)c(Br)c1C(=O)NCC(C)N(C)C(C1CCC(C)(C)O1)=O C1(CNC(C(C)N(C)C)=O)CN(C(c2cccc(-n3ccnc3)c2)=O)CCCO1 C1(NC(c2cn(CCC)nc2C)=O)CC2CCC1CN2C(c1sccc1F)=O C=CCC(CC(F)F)C(=O)N(CC(C)O)CCNC(c1cc2nccnc2[nH]1)=O CCCCC(C(=O)NC1COC(=O)C1)NC(=O)C(C)N1CC(C)C1 N1(C(C(N2CCN(c3ccc(C)c(C)c3)CC2C)=O)=O)CC2CCC(C1)C2(F)F C1(NC(Cc2c(C)con2)=O)CCN(C(=O)C(C)Oc2cccc(F)c2)C1C c1(OC(C)C(N2CCC(NC(=O)CCC3CC3)CC2C)=O)ccc(Cl)cc1Cl Cc1cccc(C(CNC(=O)Cc2ccccc2Br)NC(C2CC(C)CO2)=O)c1 C1(C(=O)NCC(C)(C)NC(CC(C)(C)C)=O)CCc2[nH]nc(O)c2C1 CCCCCCC(F)C(=O)NC1CC(CNC(c2cc(C#N)oc2C)=O)C1 C(=O)(CC1=CCCC1)N1C(C(C)NC(C(CC)F)=O)CCC1 c1(C2C(C=O)C2)cccc(Cl)c1.C(CO)(C(=O)NC1CCCC1)NC(N)=O.C C1(NC(CCCCC)=O)CN(C(=O)CC(F)(F)Cl)C2(CCCOC2)C1 N1(C(C2N(C(C(C)NC(=O)NC)=O)CCC(F)C2)=O)CC2CCCC2(CO)C1 OC1(Cc2ccccc2)CC2(CCN(Cc3cn4cc(Cl)cc(Br)c4n3)CC2)C1 c1(CN2CCC(=CC(=O)NCC(N3CCCC3)=O)CC2)cc(Br)cc(F)c1F C1(c2ccc(C)cc2)CCN(C(=O)C(=O)Nc2cnn(CC=C(C)C)c2)CC1C C1(NC(C2CN(C(=O)C(F)(F)C3CC3)CC2F)=O)CC(O)CC1O C1(C(N2CCN(C)C(CNC(=O)CC(=O)N(C)C)C2)=O)Cc2ccccc2N1 C1(CNC(c2cnc(CC(C)(C)C)o2)=O)CCN(C2CCNC2=O)CC1 CC1CN(C(C2(F)CCCC2)=O)CCC1N(C)C(c1cccc[n+]1[O-])=O C1(C=O)CCN(C(N)=O)CC1.C(CCCC)N(C)C(c1ccc(C(N)=O)o1)=O.N C12(CNC(Cc3scc(C)c3)=O)CCCC1CCN2C(=O)C1CC1 c1(N(C(N2CCCC(=C(F)CO)C2)=O)CC)cc(C)cc(C)c1 c1(C(=O)NC2CC(C)(NC(c3ccccc3)=O)C2)c[nH]c2cccc(F)c12 C1(NC(C2(CCC)CCC2)=O)CC(C(=O)NCc2nc(C)cs2)CC1O CCCC(C)CC(=O)NCCC(O)CNC(=O)CCC1CCC1 C1(CNC=O)CCC1.[nH]1cncn1.C1(C2CCC2)CC1.CC=O.C1CC1.O C1(COC)CN(CC(=O)NCC2CCCC2O)CC2(CCC2)O1.c1ccccn1 N1(C(CC(C)NC(=O)C=Cc2ccncn2)=O)CCN(C2CC2)C(=O)C1 n1(CC(=O)N)cnnc1O.C(=O)(C(C1CC1)C1CC1)NC(C1CCC1)C C1(C(=O)NC2(CC=C)CCN(C(=O)C(C)C(C)(F)F)C2)CCc2c[nH]nc2C1 N1(C(c2ncc(OCC)nc2)=O)CCC2CC2C1.c1(C=O)cc(O)cc(=O)o1.N CC1(C2(C(N3CC(O)CC3C(=O)NOCc3nc[nH]n3)=O)CC2)CC1 C#CC(CO)(CO)NC(C1C=CCN(C(=O)C=CC2CCOC2)C1)=O c1(C(=O)N)cnn2ncccc12.c1(C(=O)OCC2COCCO2)ccc(C=O)s1 C1(C(=O)NC2CCC(NC(C3C(C)(C)COC3)=O)CC2)CC2(C1)CC2(F)F C(=O)(CC(O)CC(C)C)N1C(COC)CN(C(c2cn(C)[nH]c2=N)=O)CC1 C(C)(C(=O)N)(C(C)C)OC.C1CC(=O)N(C2CN(C(=O)C)C2)C1.CC(C)C C1(CCCC)CCC(NC(=O)C(=O)Nc2cccc(Cl)n2)CC1 C(=O)(C(C(C)C)n1cncn1)NC1C(CNC(C#CCOC)=O)CCC1 c1(C(N2CCC(c3nc(C4CCC4)no3)CC2)=O)nc2ncccc2[nH]1 C1(NC(C2CCOCCN2C(c2cccc(Cl)c2)=O)=O)CC2(CCCO2)C1 c1(CNc2c(OC)ccc(C)c2)cccc(C2=Cc3ccccc3C2)n1 C(CCCCCNC(=O)CC1CCC1)NC(C1CCCN1C1C(C(C)C)C1)=O CC(C)(C)CC(=O)NCC1CCCCN1C(=O)C(c1ccc(Cl)nc1)(C)C C1(C(=O)NCCOCCC)CCC(C)(C)C1.C1(C(=O)N)CCCCC(=O)C1 n1(CCC)nnnc1CC1CCC1C(F)(F)F.C1(C)(CC)OCCO1.CCS Nc1cc2c(cc1C(N1CCC(CO)C(NC(=O)CS(N)(=O)=O)C1)=O)CCCC2 C1(NC(c2c(C)n[nH]c2)=O)CCN(C(=O)Cc2ccc(F)cn2)C12CC2 c1(OCC(=O)NCC#CCNC(C2CCOC2)=O)ccc(Br)cn1 N1(C(C(N2CCCC(O)C2)C)=O)CC(CO)C(CC(C)(C)C)C1 c1(C(N(C(C)C)CCN(C)C(C2CC(=O)CO2)=O)=O)cnc2c(c1)nnn2C N1(C(C2=C(C)OCC2)=O)Cc2ccccc2C1C(=O)Nc1cc2cnccc2[nH]1 CC(C)CC(O)C(=O)NC1(CO)CCN(Cc2cccc(C#N)c2)CC1 n1(CC(=O)NC(COCC)C(N2CCC(C)(CCO)C2)=O)ccccc1=O O1NC(=O)CN(C2CC2)C(=O)C1.c1(CC)csc(CC)n1 c1(C(N2CC(Cn3cc(C(O)C4CC4)nn3)C2)=O)ccccc1C1CCC1 C1(CNC(CSCC#C)=O)CN(C(c2ccc(O)nc2Cl)=O)C2(CCOCC2)C1 N1(C(CC(C(C)C)C)=O)CCC2CN(C(C34CC(CO)(C3)C4)=O)CCC12 c1(C(N(C2CCN(C(CC=CC=C)=O)C2)C)=O)ccc2c(c1)CC2 c1(CC)n[nH]cc1CNC(=O)COCCNC(=O)CC.CC(C)C.O N1(C(CSCC#C)=O)CCC2CN(C(C3CCCCC3C(F)(F)F)=O)CC12 N1(C(Cc2c(OC)ccc(F)c2)=O)CC2(CCCN(C(=O)C(C)(F)F)C2)C1 C1(NC(CC(=C)C)=O)CCCC1(C)NC(C1CCC(CS)CC1)=O.c1cc[nH]c1 N1(C(c2cc(C)nc(C)n2)=O)CC2CCN(C(C3CCn4ccnc4C3)=O)C2C1 c1(OC)ccc(CC(=O)NCCC(C)C)c(Cl)c1.C1(O)(C=O)CC(C)(C)C1.N C1(CC)CCCCN1C(c1cnn(C2CC2)c1)=O.C1(C=O)CC(=O)N(OC)C1.N N1(C(c2c(C)cccc2)CO)CC(C)Sc2ccccc21 C1(CCNC(C2CCCCC2O)=O)CSCCN1C(=O)C=Cc1cnc[nH]1 O(C=CC(=O)N(CCCNC(C1CCC1C(C)(C)C)=O)C)CC c1(C(N2CCN(Cc3cc4ccc(Br)cc4[nH]3)CC2)=O)cc(F)cc([N+](=O)[O-])c1 C(=O)C(C)(C)CCCC(=O)N1CCC2(CCCN(C(=O)C)C2)C1.[SH](C)(=O)=O.CO C1(c2onc(C)n2)CC12CCN(C(=O)NCC1CC3CCC(C1)N3C)CC2 CCC(CN(C)C)C(=O)NC1CC(C)C1.C(=O)(C(C)Cn1ccc(C)n1)N c1(C(N2CC3C(C(=O)NCc4c(OC)nn(C)c4)C3C2)=O)ncnc(C)c1C N1(C(C2(NC(c3n(CC)ccn3)=O)CCC2)=O)CC(C#N)(CCF)C1 c1(OC)cc(F)ccc1C(=O)NC1CCCC(CNC(C2COCCN2C)=O)C1 CC(C)C(F)C(=O)N1CCC(C(C)(C)C(=O)N2CC(NC(=O)C3CC3)C2)C1 C=CCC(C(=O)N1CCC(C)(NC(C23CCC(C2)C3(C)C)=O)C1)C(C)C C1(CNC(C(CC)C(C)C)=O)CC2(CO1)CN(C(c1ccn(C)c1)=O)C2 CCC(CC(=O)N1CCC(C(=O)N(C)CC2(C)CCCO2)C1C(C)C)C(F)F c1(CN2C(CCNC(C3CCC(F)CC3)=O)CCC2)cc(Cl)ccc1Cl N1(C(CCc2n(C)ccc2)=O)CC2CC1CCC2NC(C1CS(=O)(=O)C1)=O CCC(C)(C)CC(=O)N1CC(NC(=O)CC23COC(CF)(C2)C3)CC1(C)CC c1(OCC)ccc(NC(=O)C=C(C)C)cc1O.C1(C(=O)N)CCC(F)C1 CCC(C)(CNC(C1CN(C(=O)CCOCC(F)F)CC1F)=O)CC Cc1nc(C)n(O)c1C(N1C2CCC1C(NC(=O)CSCC(F)(F)F)C2)=O N1(C(COC)=O)CC(NC(c2cc(OC)cc(F)c2)=O)C2(CCOCC2)C1 CC(C)S(=O)(=O)C(C)C(=O)N1CC(NC(=O)CCC(F)F)CC1(C)C c1(-c2cc(OC)c(F)cc2)c[nH]c2nc(C(=O)Nc3cncc(Br)c3)ccc12 C1(C(=O)NC(CNC(c2c(C(=O)OC)c(C)on2)=O)C)CCC(C)C(C)C1 c1(C(=O)NC(CC(C)NC(c2ccc(C(N)=O)cn2)=O)C)ccnc(S)c1 C(=O)(CC(C)(C)CNC(=O)Cn1cc(C2CC2)nn1)NC(C(=C)C)(C)C C1(CNC(C(C(C)C)CO)=O)CN(C(c2cc(O)cc(=O)o2)=O)CC(C)(C)O1 c1(OC)c[nH]c(C(=O)NC2CN(C(C3CC3C#N)=O)CC2C)cc1=O CC1CCC2(CO1)CN(C(=O)CC1C3CN(C(C45CC(C#N)(C4)C5)=O)CC13)C2 c1(-c2cncc(OC)n2)ccc2nc(C(=O)Nc3cc(Cl)cnc3O)oc2c1 CCCC(C)CC(=O)NC1(C)CCCN(C(=O)C(C)(C)c2cnc[nH]2)C1 N1(C(c2c(OC)nccc2C)=O)CCCN(C(c2cnc(C)[nH]c2=N)=O)CC1C C1(C)(C(=O)NC2CCCN(C(CSSC)=O)C2)CCC(C)=C(C)C1 CCCCC(O)C(C)C(=O)N(CC(C)NC(c1c[nH]c(=N)c(C)c1)=O)CC C1(C(=O)NC(CN(C(c2cnc(SC)nc2O)=O)CC)C)CCC(=O)N(C)C1 c1(OC)ccc(CNCC(CC)C(=O)OC)nc1OC(C)C CC1(NC(C23CCCC2(C(N)=O)C3)=O)CCN(C(c2ccc(Br)o2)=O)CC1 C(=O)(CC(C(F)F)N(C(=O)C(N1CCC(OCCO)C1)=O)C)OC CC1(C)CCCC(C(=O)NCC2CCC(O)C2)O1.N1(CCC(=O)N)CCCCC1 C(c1cccc([N+](=O)[O-])c1)=CC(=O)N.CC1(O)CCN(CC(=O)NCCCO)C1 c1(C(N(C(CNC(C(C)OCCOCC)=O)C)C)=O)csc(Cl)c1O C1(OC)CC(NC(c2cn3c(n2)SCC3)=O)CN(C(=O)C(C2CCOC2)O)C1 c1(C(N(C(c2cn(Cc3cnoc3)nn2)C)C)=O)cccc2c1ncn2C c1(C(N2CCC(NC(c3c(C)nn(CCO)c3)=O)C2)=O)ccc(C(N)=O)c(Cl)c1 C1(C(N2CC3(CN(C(C4CCCC4)=O)C3)C2)=O)CC2CCC1CC21OCCO1 c1(CCC(=O)NC(CCCCNC(c2cnc(C)s2)=O)C)c(C)nc(O)nc1C c1(NC(=O)CN2CCOC2=O)cccc(NC(C2(F)C3CCCC23)=O)c1 CC(CSc1ccccc1)C(=O)NCC(F)CNC(=O)Cc1cncn1C N1(CCn2c(C(=O)OC)cc(C(=O)OC)n2)CCCC2(CCCCC2O)C1 N1(C(C(CC)n2cncn2)=O)CCC2(CC1)CC2CNC(C1(Cl)CC1)=O C(CCOCCO)(C=O)NC(C1(CC#C)CCCO1)=O.C1C(=O)NN=C1C.N C(=O)(C(C)CC(F)(F)F)NC1(C(=O)NC(COC)CCO)CCCC1 CS(=O)C=CC(=O)N1CCCC1CCNC(c1[nH]ccc1-c1ccccc1)=O N1(C(c2cnc(OC)s2)=O)CC2C(CC(=O)N(C3CCC3)C3CCC3)C2C1 C1(C(C)(C)O)(C)CN(C(c2cc(C3CCC3)on2)=O)C1.C1(C=O)CSCCS1.N c1(C(=O)NC(C(N2CCOCC2)C)C)cc([N+](=O)[O-])ccc1O c1(CC)ccc(S(=O)(=O)N2CCN(C(=O)Cn3cc(Cl)cn3)CC2)s1.CC=O.N C(C(CNC(=O)CC1CN(C)C1)S(C)(=O)=O)NC(CSC(C)C)=O N1(C(CC2N(Cc3cc(C)cc(F)c3)CCOC2)=O)Cc2cccc(C)c2C1 N1(C(C2(C(F)F)CCN(C)CC2)=O)CC2CC(NC(=O)C3CC3)CC2C1 CCCC(C)C(C)N=c1[nH]c(=NCCF)[nH]c2ccc(OC)cc12 C(C(=O)NCCC1COCCN1C(=O)CC1CCCO1)(c1ccccc1)=C(C)C C(=O)(CCC(=O)NCC)N(CC)CC.C1(CCCNC(=O)CO)CC1 c1(N(C)C(C2CCCN(C(=O)Cn3cnc(=N)[nH]3)C2)=O)ccc(F)cc1 c1(C(=O)NCCCCCCNC(c2c(C)nc(C3CC3)s2)=O)c(C)cnnc1O C1(NC(c2c(C)nn(C)c2)=O)CN(C(c2ccccc2Cl)=O)CC12CC2.C(C)C.O CN1CCN(C)C2(CCCN(C(c3cc4cccc[n+]4cc3Cl)=O)C2)C1 C1(C(N(c2c(CC)cccc2)C)=O)CCN(C(=O)C(C)SC(C)C)C(C)(C)C1 N1(C(C2(C)C(CC)CCC2)=O)CCC=C(C(=O)NC2(C)CCCCC2C)C1 C(=O)(CCCCCC#N)NC1CC2(CC(C(N(C3CCOCC3)C)=O)C2)C1 N1(C(CC(CC)C)=O)CCCC(NC(c2cccc(CS(C)(=O)=O)c2)=O)CC1 C1(C(=O)NCC2(OC)CCN(C(=O)C(C)CCO)C2)CCCC2(CC2)C1 S(=O)(=O)(c1cccc(C(=O)NC2C3CCCC23)c1)N1CC(C)(C)S(=O)CC1 N1(C(c2c(CC)n[nH]c2)=O)CCC(C(C)NC(c2coc(C)c2)=O)CC1 CN1C(=O)OC2CN(C(=O)C(C)(CO)NC(=O)C(C3(O)CCCC3)F)CC12 CC(CNC(=O)CN(C)C(=O)OC)C(F)C(=O)NC1COCCC1(F)F CC1CC(C(=O)NC2CC(CC)C2)CC(=O)N1.C(=O)(CC=O)N.C(C)(C)C c1(C(N2C(C)CCC(CNC(CCSC)=O)C2)=O)nc2ccccc2[nH]1 C1(C)(C(N2CCC(C)(NC(C=CC(C)(C)SC)=O)C2)=O)CC=C(C)CC1 N1(C(CC2ON=C(C)C2)=O)CC2CCC(C(=O)NC3CCC(O)C(O)C3)(C2)C1 c1(C(C(=O)N)OC)cccc(C(F)(F)F)c1.C1CC1.C(=O)CC1CSC1.C c1(-c2cc(SCCOC(CCC3CCC(C(N)=O)O3)=O)on2)cccc(Cl)c1 c1(OCC)ccccc1C(=O)NCCCNC(Cn1cc(C=O)nn1)=O.N c1(C(c2n(CCC)nnn2)Nc2cnccc2CC)cc(C(F)F)cc(C)c1 C#CC1(C(N2CC(CC(N)=O)C2)=O)CCN(C(C2CC2CCC)=O)CC1 N1(C(c2ncn(C(C)C)c2)C(=O)NCCC#N)CCCCc2ccccc21 Cc1ncc(C(N2CCC3(CC3C(=O)NC34CC3COC4(C)C)C2)=O)c(C)n1 Nc1c(Cl)ccc(C(=O)N(CC)C2CC2)c1Cl.c1(C2(C=O)CC2)ccccc1.N C1(C)(CCNC(c2c(C)c[nH]n2)=O)CCN(C(c2snnc2C2CCC2)=O)C1 C(CCC(C)CC(=O)N1CC2CCC(C1)N2C(c1csc([N+](=O)[O-])c1)=O)=C(C)C N1(C(C(C)CC(N)=O)=O)CCCCC2(CCN(C(C3CC4(CCCO4)C3)=O)C2)C1 c1(C(=O)N(CO)Cc2cc[nH]n2)noc2cc(-c3cnc(C(F)F)nc3)ccc12 C(=O)(C1=CC(C)(C)C1)NC1(CNC(C2C(=C)CC2)=O)CCCCC1 N1(C(=O)C=CBr)CC2CCC(Nc3ncnc4c3COC4)C2C1 CC1CN(C(c2cnnn2C)=O)CC(C)N(C(c2ccn(CC(F)(F)F)n2)=O)C1 c1(C(=O)NC(C)CN(C(=O)C(F)(F)c2cscn2)C)ccc(Cl)c(C#N)c1 C1CCC12CN(C(C1CCC1)=O)C2.c1(C(=O)OC)ccc(OCCCC=O)cc1.N CCC(C)CCC(=O)NCc1ccc(CO)cc1F.C1(C=O)C2CCC(F)(F)C12.N C1(CCC)CCCN(C(=O)CC2CC2(Cl)Cl)C1.n1(CC(=O)N)ccc(=O)cc1C C1(NC(CC(CCC)O)=O)CC12CCN(C(=O)CCc1cnc(C)s1)CC2 N1(Cc2ccc(C)nc2C)CCc2c(C(=O)Nc3cc(Cl)ncc3Br)n[nH]c2C1 n1(CC)ccc2nc(N3CCNCC3C(=O)Nc3cc(F)ccc3C#N)ncc12 N1(C(c2ccc(N(C)C)cn2)=O)CC2(CCN(C(=O)CCCS(C)(=O)=O)CC2)C1 N1(CC(N2CCCC(O)(CNC(c3[nH]cc(C)c3)=O)C2)=O)CCCCC(O)C1=O c1(C(N2CC3CC(NC(C(CC=C)C)=O)CC3C2)=O)ccc2c(c1)nnn2CC Cc1cc(C(=O)NCCCCCN(C(=O)Cc2cnn(C)c2)C)c(C)o1 c1(C(C)C)cc(C(=O)NC2CC(N(C)C(C3CC(C)(F)C3)=O)C2)n(C)n1 CN1CCOC(C(=O)NC2CC(CNC(c3nccc(F)c3Cl)=O)C2)C1=O N1(C(C(C(C)C)C)=O)CC(F)(F)CC1(C)CNC(c1cccc(OC(F)F)c1)=O Cc1ccc2c(cnn2C)c1-c1cncnc1C(=O)NCC#N C1(C(=O)NC2(C)CCC(NC(CCC=CC)=O)CC2)CCc2nnn(C)c2C1 Cc1c(F)ccc(C(N2CCCC2CCNC(=O)C(=Cc2c[nH]cn2)F)=O)c1N CCC(C)(C)CCCC(=O)N1CCC(C)C1C(=O)NC1CC(CCC(N)=O)C1 C1(C)CCCN1C(=O)CC(C)C(C(=O)C(=O)Cc1ccc(N)cc1)OC.N.C Nc1cnc(C(F)(F)F)cc1C(=O)NCC1CC2C(C1)C2(F)F C1(NC(CC=C)=O)CCN(C(c2cc(C3CC3)nn2C)=O)CC1C c1(CC)nc(C(=O)NC2CCC(CNC(C3CSC3)=O)C2)n[nH]1 C1(CNC(c2cnc(O)s2)=O)CCCN(C(=O)C)CC1.C1CCS(=O)(=O)C1 C(=O)(N=c1[nH]nc2[nH]ccnc1-2)C1C=CC(NC(c2c(C)cc(C)c(Br)c2)=O)C1 N1(C(c2scc(C)c2C)=O)CCC(NC(=O)CN(C)CCO)C2(CCC2)C1 c1(C=O)cc(C(C)C)nn1C.C(=O)(C(C)(C)c1ccn(C)n1)N(CCC)CC C1(CNC(C2CN3CCCC3CO2)=O)CCN(C(C2CCCO2)=O)CCC1(F)F c1(C(N2CCC(CC(=O)NCC3CCC(=O)N3)C2)=O)cc2n(n1)CCCC2 CCC(C)CCC(=O)NC1(C(=O)N(C(C)CCSC)C)CC(F)(F)C1 CC(CCNC(c1cnsn1)=O)CCNC(C1(C)CCCCC1)=O c1(C(=O)NC(CCNC(C2C(C)CC(C)O2)=O)C)csc2nnsc12 N1(C(c2c(Cl)ccc(OC)n2)=O)CC2CCCC2(NC(=O)CN2CC=CC2)C1 CC1CCCN1C(=O)CC.n1(CC=O)ccccc1=O.C(=O)CCN(C)CCO c1(C(C(=O)NC2C(CNC(Cc3ccn(C)c3)=O)CC2)(C)C)ccc(F)cc1 C=C(C)CC(C)C(=O)NCC(c1ccccc1)NC(=O)C=Cc1ccco1 Cc1cc(C(N2CCC(NC(=O)CC3CCC(=O)N3C)C(O)C2)=O)cnc1O CCC(CC)(CCNC(=O)CC(O)c1ccccc1)NC(c1cscc1C#N)=O Cc1cccc(F)c1C(=O)NC1CCCCN(Cc2cc(Br)cs2)C1 c1(C(=O)NC2CC(C)(CNC(CCc3n(C)cnc3)=O)C2)c[nH]cc(Cl)c1=O C(CN=c1ccnc(C2CC2)[nH]1)OCCNC(C=CCOC)=O c1(C(N2CCCC(CCNC(=O)CC3CNC(=O)O3)C2)=O)cnc(O)c(F)c1 C1(NC(C(CCC)=CCC)=O)CCN(C(=O)CSCC(N)=O)C(C)C1 C(=O)(C(C(C)(C)C)n1cc(CS(C)(=O)=O)nn1)NCC1CN(C)C(=O)C1 Cc1cc(O)c(F)cc1NC(C1CCCC(NC(=O)CCO)CC1)=O.CC(F)F c1(N2CCC(CCC)C2)nc(=N)[nH]c(=NCc2ncc(C)s2)[nH]1 c1(C(=O)NCC2(Nc3cccc(C)c3)CCOCC2)cc(C)nc(C)n1 c1(C=O)ccnc2c(Cl)c(C)ccc12.C1(NC(C=CC=CC)=O)CCCC1.N C1(C(=O)NC(CNC(C(C(=C)Cl)(C)C)=O)C(C)(C)C)CCc2nc(C)nn2C1 N1(C(CN(C)C)=O)CCN(C(C23CCC2C3)=O)C(c2ccnn2C)C1 N1(C(c2nc(C)sc2C)=O)CCC(N(C(=O)C#CC2CC2)C)C(C)C1 c1(C(=O)NC(C)CC2CN(C(c3cnsc3)=O)C2)cccc(CCN(C)C)c1 CC1(C)CC(C(=O)NC2(c3nn[nH]n3)CC2)CCN1C(=O)C(F)(F)CO CC12CC(C(=O)N)(C1)C1(CCC1)O2.C1CN(C(=O)CCc2cnoc2)CC1O.C C12(C(N3CCCC3)=O)CCCC(CO1)C2.c1(CC)scnc1C(=O)NCCO c1ccc2ccccc2c1.C1(CC(=O)NCC(C2CC2)NC(=O)C)CC12CC2 C1(C)(C(N2CC(CC(=O)NC)(OCC)C2)=O)CCN(C)C1.C1CCCS1 C1(NC(CN(S(CC)(=O)=O)C)=O)CN(C(C2(C)CCCN2C)=O)CC1C Cc1nc2cccc(C(=O)NC(C)CCCNC(=O)C(C)OC(C)(C)C)n2n1 N1(C(C2(COC)C=CCC2)=O)CC(NC(=O)CCC(N)=O)C(O)C1 C(=O)(C1COc2ccccc21)NC(C)(C)CCNC(c1ccc(C(F)F)o1)=O c1(N(CCOC)CCNC(C2CCC(O)C2)=O)nc2cccc(C)c2o1 c1(C(N2CC(C(C)NC(C(CC)SC)=O)C2)=O)cc2n(n1)CCCC2O c1(OCC(=O)N(c2ccc(C)cc2Cl)c2nncn2C)ccc2c(c1)CCOC2 c1(CC)ncncc1C(=O)NCC1CCCN1C1CCN(c2cnn(C)c2)C1=O CC(C)CC(C)CC(=O)N1CC(C(C)NC(c2cc(C3CCC3)on2)=O)C1 CCCCC(C(=O)NC)NC(=O)CCC1CCN(C(=O)C(C)(C)F)CC1 CCC(CC)CCCC(=O)NC(CC(=O)NC(C)C(C)C)C(C)OC N1(C(CSCC#N)=O)CCC(C2CCN(C(=O)C3=NNC(C(F)(F)F)C3)CC2)C1 C1(NC(c2ccc(Cl)o2)=O)CCCCC1NC(C1CC(CC(F)(F)F)C1)=O N1(CCNC(C2CCOC2C2CC2)=O)CCCCC1.C(C1CCCC1)=CC=O c1(C(=O)NCC(C)(C)OC)ccc(O)c(C)c1.c1(C(=O)N)c(C)noc1C C#Cc1ccc(C(N2CCCC2C2(O)CN(C(c3cscn3)=O)C2)=O)cc1 c1(C(N)=O)cc(NC(C2CC=CC(NC(=O)CC3CCC(O)C3)C2)=O)ccn1 Cc1cccc(C(=O)N(C(CNC(=O)Cc2ccn(C)c2)C2CC2)C)c1C N1(C(CC(C)OC)=O)CCC(NC(=O)C=CCOc2ccccc2)C12CC2 C1(C(N2CCC(N(C)C(C3(C4CC4)CCCO3)=O)C2)=O)CCC(C)(C)C1 N1(C(C(C)C)C(=O)OCCC2CC2C(F)(F)F)CCS(=O)(=O)CC1 c1(C=O)cccn2cnnc12.c1(OC)cc(N)ccc1C(=O)NC1(CC)CC1.N c1(NC)c(C(=O)NC2CN(C(=O)C=Cc3nnn(C)n3)CC2C)cccc1F c1(NC(CC2CC(NC(c3cccc(C)c3N)=O)C2)=O)ccc2ccoc2c1 N1(C(C(C)(C2CC2)OC)=O)CCC2C(CCN2C(c2ccc(N)cc2F)=O)C1 N1(C(CC(C(C)C)OCC)=O)CCC2(CC1)CC(NC(c1nccn1C)=O)CO2 S(=O)(=O)(c1c(Cl)cccc1Cl)NC1CN(C(c2c(C)nc(C)s2)=O)CC(C)C1 N1(C(C(C)C(F)(F)F)=O)CCc2ccccc2C1CNC(=O)C=Cc1ccco1 C=CCCC(CC(C)C)C(=O)N1CC(SCCC(=O)O)C1 c1(C(C(=O)N(CCCN(C(=O)C(CO)N(C)C)C)C)(C)O)ccc(F)cc1 C(=O)C(C)(F)C(C)(C)F.N1(C(CC(=O)NCC)=O)CCCCC1C(C)(C)C CCCCCCC(C)(CC)C(=O)N(CC(O)CN(C(=O)CN(CC)CC)C)C c1(C(N2CCC3(CCCC3N)C2)=O)cc2ccc(O)cc2[nH]1 C1(CC)CCN(C(c2cccc(OC)n2)=O)C(C(=O)NOCC(C)O)C1 C1(C(N2CCC(OCCNC(CSCC=C)=O)C2)=O)CCC(C2CC2)CC1 c1(Cc2n(CC=C)nnn2)cc(Cl)cnc1NCC1(SC2CC2)CC1.O c1(C(=O)NCC2CCCN(C(CC(C)F)=O)CC2)cn2c(n1)C(C)CCC2 CCCCCCCCCCCCCC(=O)Nc1ncc(CCC2CCCOC2)s1 N1(C(C(CC)CO)=O)CCN(C(c2c(C)nn(C)c2C)=O)CC(C)(F)C1 CC1(C)CC2(CC2C(=O)N)C1.C1CC12CCC2.C(c1cccs1)=CC=O.C C1(O)(CC(=O)NCC2CN(C(C3CCOC(=O)N3)=O)CCO2)CCCCC1 c1(CC)cc(C(=O)NCC2C3CN(C(=O)Cn4ccnc4C)CC23)ccc1Cl c1(C(N(CC(O)CN(C)C(c2cn(C)nn2)=O)C)=O)ccc(-n2cccn2)cc1 C(C)(C)(C(C)NC(c1cc(C2(C)CC2)n[nH]1)=O)NC(CCOC)=O N1(CC(C2CCOC2)OCC)CC(=O)N(Cc2cc(C)c(Br)cn2)C1=O CCC(COC(c1cccn1Cc1ccccc1)=O)CC N1(C(C(N2CCNC2=O)C)=O)CC2(C=C(C(=O)N3CC(O)C(F)C3)CO2)C1 N1(C(Cc2cc(C)no2)=O)CCCC(N(CCO)Cc2sccc2C)C1 CC1CN(C(c2ccn(CC(F)F)n2)=O)C(C)CN1C(=O)CSc1ccncc1 c1(C(C#C)NC(C23CC(NC(C4CC4Cl)=O)(C2)C3)=O)ccc(F)cc1 CC(CC#N)C(=O)N(CCNC(=O)Cn1cccnc1=O)CCOCCO C(C)(C)(CC(=O)NCCS(N)(=O)=O)N(C(C(C)SCCCC)=O)C C1(NC(C(C2CCN(C(C(c3ccn(C)n3)C)=O)C2)(C)C)=O)C(O)C2CCOC12 CCC(CC)C(C)C(=O)NCCCN(C(C1CC(C(F)F)C1)=O)CC N1(C(c2cn(CC=C)nn2)=O)CC(NC(c2cnccc2OC)=O)CCC(O)C1 Cn1ncc2c1CC(C(=O)NCC1CCCC(C)C1)CC2.C1(F)(C=O)CCC1.N c1(C(N(C)CCO)=O)cccc2sncc12.C1(C(N(CC)C)=O)CC2C=CC1C2 [SH](=O)(=O)c1c[nH]c(C(=O)NC)c1.C1(O)CCN(C(c2cc(C)on2)=O)C1.CN N1(CCCCCOC)CCC(C)(NC(=O)CC(C)C2CCCO2)C1 C(c1ccc(Cl)cc1Cl)=CC(N1CC2N(C(c3ncc(CCC)cn3)=O)C2C1)=O C1(C(C)C)CCCCC1NC(C1(CCNC(=O)CCc2cnc[nH]2)CC1)=O CC(CCC(C)(C)C)C(=O)NCC(N1CCN(C(C2(C)CC=CC2)=O)CC1)=O C(C(C)(C)CC(C)C)N(c1nccc(N(C)Cc2cnc(C)s2)n1)C1CCCCC1 Cc1cc(CN2CCCC(O)(C(C)C)C2)c2nn(C)cc2c1 C1(CNC(C(CC)C#N)=O)CC(C)CN(C(=O)CC(C)(C)C#N)C1 C12(NC(C(C)SC)=O)CCCCC1CN(C(=O)Cn1nnnc1C)C2 C1(O)(CNC(C(CCSC)O)=O)CCN(C(=O)C(C(C)C)n2ncc(N)n2)CC1 N1(C(c2cc(=N)[nH]c(=N)[nH]2)=O)CC2=C(C1)CN(C(=O)C(CO)NC(N)=O)C2 N1(C(C2CCN(Cc3c(OC)cco3)CC2)=O)CCC(O)CC1C(=O)O C1(C=C)(CC(N2C(CCC#C)CCC2)=O)CN(C(C2(CC)CCOC2)=O)C1 c1(C(=O)NC(C)CNC(C2CC23CC3)=O)cnc(-c2cccnc2)s1 N1(C(C(CSC)O)=O)CCOC2(CCCN(C(=O)CN3CC=CC3)C2)C1 CN1C(=O)CC(NC(=O)C(c2ccoc2)NC(c2cncnc2)=O)C1=O C(=O)(C(C)CCN(C)C)NCCCNC(C)=O c1(CC(=O)NCC2C(NC(c3cc(C)ns3)=O)CCC2)cccc(C)c1F C1(COC)CN(C(=O)C(C)(C)c2ccn(C)n2)CCN1C(=O)C1=CCCCO1 c1(CC=O)cnc2cccnn12.N1(C(CNC(=O)OCC)=O)CC2CC2C1.C C1(NC(c2cc3nc(C)sc3[nH]2)=O)CCN(C(C2CCCN2C)=O)C12CCCC2 C1(c2cn(CC(=O)NCC(Br)=C(C)C)nn2)CCC(C)=CC1C C(CS(=O)(=O)CC(=O)NC1CCC(NC(=O)C(C)n2cccn2)CC1)OC c1(OCC(=O)NC2CC(NC(C3CCCC3C(F)F)=O)C2)ccc(Cl)cc1 c1(CC(N2CCCN(C(CC=C)=O)CC2CO)=O)coc2c(C)c(Cl)ccc12 C1(C(=O)NCC2N(C(c3c(Cl)ccc(C)c3)=O)CC2)CC2CCC(C1)C2(F)F c1(C(=O)NC(c2nc[nH]n2)CC)oc(CNC(c2c[nH]c(=O)cn2)=O)cc1C C1(OC)CCN(C(C2(F)CCN(C(c3ncccn3)=O)C2)=O)C12CCC2 CC1COCC(C(=O)NCCn2cnc(C(N3CCC3CC3CCCC3)=O)c2)O1 C1(CN(C(=O)CCn2ccnn2)C)CCCN1C(=O)CCOCC1CC1 C(=O)CCC(=O)NC1CCCN(C(=O)CC)C1.C(=O)C(C)(C)C.C1CC1.CO C1(O)(c2ccc(C)cc2)CCN(C(=O)CC2CNCCN2)CC1 c1(OC)cccc2c(CNc3cc(C)c(Br)c(C)c3)c(C)[nH]c12 C1(NC(C(C2CC2)OCC)=O)CCCC1CNC(c1sccc1)=O.C Cc1[nH]c(=N)nc(O)c1CCC(=O)NCCC(O)CNC(=O)C1CC1 C1(N(C(COC)=O)CC(C)C)CCN(C(c2cnn(C)c2C(F)(F)F)=O)CC1 CCCC(C(=O)NCC(C1CCCN1C(=O)CCC(=O)CC)(C)C)C(C)C c1(C(=O)NCC2OCCC2C(=O)NC(c2ncc[nH]2)CO)nccc2[nH]ccc12 c1(C(N2C(C(N3CCC(C)(O)C3)=O)CC(O)C2)=O)n[nH]c2ccccc12 c1(C(N2C(CNC(C(C(C)(C)O)F)=O)CC(C)(C)C2)=O)ccn2nccc2c1 C=C(C)CCC(C)(c1nnnn1C1CCOC1)NCc1ccc(C(F)(F)F)s1 c1(C(=O)NC(CN(C(CC=CC)=O)C)CC)c(N)sc(C)c1C C#CCCCC(C)C(=O)NC1CCCC(NC(c2nc(C)n(-c3nc[nH]n3)n2)=O)C1 C(=O)(CCCC(C)(C)C)N1C(CNC(C2CCC(O)CC2)=O)CC(OC)C1 C(=O)(CC(C(C)(C)C)NC(=O)C=Cc1ccsc1)NC(COC)CO C(C)(C(CC(=O)NCc1nccc(C)c1F)NC(=O)C(F)C(C)(F)F)OC C(=O)(C(C(C)C)SC)NCC(CNC(C1(CCOC)CCC1)=O)O C(=O)(CCCC1CCC1)NC1CCC(CCCC)C1.C1(C(=O)N)CCC(F)(F)C1 c1(NCC2C(C)CN(C(=O)C(C)(C)CO)CC2)ncc([N+](=O)[O-])cc1Br n1(CC)cnc2c(NC3CCCC3CO)nc(N(C)Cc3ccoc3)nc12 C#Cc1cc(C(=O)N(C)CCOCCN(C(=O)CCC(=O)NC)C)ccc1C C1(C2CC2)(C(N2C(CC)CC2)=O)CN(C(=O)CC2CCCC2)C1 C(=O)(C(C(C)C)n1cccc1)Nc1nc(C(C)(C)NCCOC(C)C)no1 N1(C(c2cnc(C(C)C)nc2)=O)CC2CCCC(C1)N2C(C1(F)CC1C)=O CC(C(C)(C)C(=O)NCC1CSCCO1)NC(=O)CCCCC1CC1 C1(O)(CC(=O)N)CCCN(C)C1.c1(C(C(=O)N(CCC)CC)C)ccncc1C C1(CC(N2CC(NC(C3(C)C=CCC3)=O)C2)=O)CCCS1(=O)=O CN1CCCC1C1COCCN1Cc1cn(C2CCSC(C)(C)C2)nn1 Cc1nc(C)c(CNCC2CN(C(=O)Nc3ccccn3)CCO2)[nH]1 c1(C(N2CCCC(O)(CNC(CCC(N)=O)=O)C2)=O)nnc(O)c2c1CCCC2 c1(NC(N2CCC(CC=C)C2)=O)cccc2c1OC(C)(C)C2 C1(C(N2C(C3(NC(CCC#C)=O)CC3)CCC2)=O)CC(=O)N(O)C1 N1(C(CC(C)C(F)(F)F)=O)CCCC12CCN(C(=O)Cc1cccn1C)CC2 Cc1nc2c(C(N3CCCC(NC(C4CCS(=O)(=O)N4)=O)C3C)=O)cccc2o1 N1(C(c2c(C)ncnc2)=O)C2CC1CN(C(C1CC1C1CC1)=O)C2 C=CCC(CC=C)C(=O)NCCCNC(=O)Cc1ccc(CO)cc1 C(CCSC)(C(=O)NC1CC(N(CC(C)C)C)C1)OC Cc1n[nH]c(=NCCCOC2CCN(C(C3CCCC(O)C3)=O)CC2)s1 N1(C(CC(CC#C)NC(c2ccccc2)=O)=O)CC(=O)N(C)CC1C C12(CC)CC1CN(C(C1(C3CCCN3C(C3CC(=O)CS3)=O)CC1)=O)C2 C1(CNC(=O)NC2(COC)CCOC2)CN(c2ccccc2)C(=O)O1 N1(C(CS(C)(=O)=O)=O)CCN(C(C2(O)CCSC2)=O)CC1CS(C)(=O)=O c12c(Br)ccnc1OC2.C1(CC(=O)N(C2CC(OC)C2)C)CCCC1O C1(C(=O)Nc2cccnc2)CC(F)CN1Cc1ccc(OCC2CCO2)cc1 Cc1ccccc1NC(=O)C(N1CCCC(CC(N)=O)C1)c1cnn(C2CC2)n1 C1(C=O)CCCCC1NC(=O)NC(c1ccc(OCF)cc1)C.C(C)(C)C.O C(CN=c1[nH]c(=NCc2cnc[nH]2)[nH]c2c1CCCC2)c1c(F)ccc(F)c1 CCC(CC(F)F)C(=O)NCCC(c1cccs1)NC(=O)C=CCO c1(C(N(C(CNC(c2c(CC)nn(C)c2)=O)C)C)=O)cnc2n(c1=O)CCS2 c1(C(=O)NCCC2CCN(C(COCC#C)=O)C2)coc2c(F)c(Cl)ccc12 Cc1ccc(OCC(=O)NCC2(O)CN(C(C3CCCCC3)=O)C2)c(Cl)c1.N CCC(C(C)(C)C(=O)O)NC(c1cnc2ncnn2c1)=O N1(Cc2c(C(=O)OCC)n[nH]c2)CCC(O)(C(=O)Nc2ccc(Br)cn2)C1 C1(C(=O)NCC(CC(=O)NCCF)O)CC2(C1)CC(O)C2 c1(OC(C2(Cc3cc(Cl)cc(Cl)c3)CC2)=O)cc(Cl)cc(Cl)c1Cl C(N=c1cc[nH]c(-c2nccs2)n1)C1C(C)CCN(C(C2(C)CC(C)C2)=O)C1 c1(C(C(=O)NCCCC)N(C)CC2CC2C)ccnc(Cl)c1F Cc1ccccc1-n1c(SCCCC(=O)O)nnc1C C1(C)CCCC1.C1(N(C(=O)CC2CCC2)C)(C(N)=O)CCC1.C(=O)(C)N c1(C(=O)N)ccn(CCF)c1.c1(C(N(CCC)CC)=O)ccc(-c2ccco2)[nH]1 c1(C(=O)NC2CCC(NC(C(C3CCOC3)OCC)=O)CC2)ccc(O)cc1C C12(CNC(CP(C)(C)=O)=O)CCC(CN(C(c3cc(CO)[nH]n3)=O)C1)C2 n1(CC)c(C)cc(C(=O)N(C2CCCN(C(C3CC(O)CN3C)=O)C2)C)c1C C(CN=C(NC(C1CC1)C1CC1)NCC(c1ccsc1)C)OC.C1CC1 c1(CCC)cc(C(=O)NCC(O)CNC(=O)Cc2cnn(C(F)F)c2)no1 C(=O)(C(S(N)(=O)=O)c1ccccc1)NC1C=CCN(C(C2OCCN(C)C2)=O)C1 C1(CC=C)(C(=O)NC(C(F)F)C(C)C)CCCN1C(=O)C(C)O.CCC(C)C C1(O)(C(N)=O)CCCN(C(C2CCC(O)CN2C(=O)CCc2ccoc2)=O)C1 c1(C(C)OCC)nc(C(C(=O)NCCSC)N(CC#N)CC)cs1 c1(C(N(CCOC)CCNC(c2cccs2)=O)=O)cc([N+](=O)[O-])c[nH]1.O C1(C2CCCN(C(=O)CC3CCOCC3)C2)(NC(C2N=C(C)SC2)=O)CC1 c1(CCC(=O)NCC2CCN(C(=O)Cn3cncn3)C2)nc(-c2cccs2)no1 c1(NC(CC2N(C(COC)=O)C3C2CCC3)=O)cc(C)c(F)c(C)c1 N1(c2n(Cc3cc(N)cc(F)n3)nnn2)CCC2(C1)CC(F)(F)C2(F)F C(CC(=O)NOCCC(F)F)=CCNC(C1CN(C)C1)=O C1(C(=O)NCCOc2cccc(C(=O)OC)c2)CCC(S(C)(=O)=O)CC1 Cc1ccc(CCC(=O)NCC2CN(C(C3CCCO3)=O)CCCO2)cc1Cl C1(CCNC(=O)CCc2nncs2)COCCN1C(C1CCS1(=O)=O)=O [N-]=[N+]=NC1CCCCC1N1CCN(C(C2CCNC(C(F)(F)F)C2)=O)CC1 C1(F)CCC1.c1(CC=O)csc(-c2ccc(C)o2)n1.C(C)(C(=O)NC)SC CCCC(CNC(=O)Cn1cncn1)C(=O)NCC1(O)CC(CO)C1 C1(CC)SC(C)CC(N2CCC(O)C(C(N3CC4CCCC3C4)=O)C2)C1C Cc1cc(C(=O)NCCCN(C)C(c2ccc(-c3cn[nH]c3)nc2)=O)ccn1 c1(-n2cc(CN(C(C3CC(C(C)C)OCC3)=O)O)nn2)ccccc1S(N)(=O)=O C(C1=CCCN(C)C1)NC(COC1(C)CN(C(C(CSC)C)=O)C1)=O C(=O)(C1CCCc2cc(O)ccc21)N(C)CC1N(C(CCC=C(C)C)=O)CCC1 C(=O)(C(C)N=c1[nH]c2ccccc2s1)NC1(CO)CCN(C(C(C)(C)OC)=O)C1 N(S(=O)(=O)Oc1ccccc1)C1(C(C)NC(=O)CN(C2CCCC2)C)CC1 N1(C(c2cc(N)c(N)nc2)=O)CCC2(CC1)CC2NC(C1CC12CCCCC2)=O c1(CNC(c2ccc(C(C)C)o2)=O)cccc(OC(F)F)n1 c1(C(N2C(CNC(C(C(C)(C)O)F)=O)CCCC2)=O)cccc2c1CC(C)(C)C2 N1(c2ccnc(N3CCCC3)n2)CC2CCN(Cc3cscn3)C2C1 C1(C(=O)NC(C)(C(=O)NCCC(F)(F)F)C2CCC2)(OC)CC(C)C1 c1(C(C(=O)NCCCCO)N(c2ccccc2)C)ccc(C(F)F)nc1 CCCCC(O)C(C)C(=O)NC1(C(N2CCC23CCSCC3)=O)CCN(C)C1 c1(C(=O)NC(C)CCNC(=O)C(CO)N(C)C)ccn2ncc(Br)c2n1 C=CC(C)(CC)C(=O)N(CCNC(c1ccc(Br)c(C(C)=O)c1)=O)CC C(=O)(C(C)(C=C)CC)NCc1ccc(CNC(C(CC#C)O)=O)cc1 C(=O)(C1=CN=C2N=CNN2C1)N1CCCC(CNC(CC(C)SC)=O)C1 n1(CCN2CCC(C(N3CC=CC(O)C3)=O)C2)cnc([N+](=O)[O-])c1 c1(N)cccc(OC(F)(F)F)c1.c1(C(CCO)NC(C2CC2)=O)cccc(F)c1 Cc1ncnc(C)c1C(=O)N(C)CCNC(c1c[nH]c(C(N)=O)c1)=O C(CCC(=O)N(C(CNC(c1csc(=N)[nH]1)=O)C1CC1)C)N(C(C)=O)C N1(C(C2N(C(C(CCCC)F)=O)CC(=O)C2)=O)CC(O)C(O)C12CCC2 c1(C(=O)NC2(C(=O)NC3CC(CCOC)C3)CC(O)C2)ccnc(C)c1 N1(C(c2c(C)ccc(C)c2N)=O)CC2(C)CN(C(=O)C3=CCSC3)CC2(C)C1 C12(C(=O)NCC(=O)OCC)CCCC1CCN2C(=O)C(C1CCCCC1)F c1(OCC(=O)NC(CC2CCN(C(CC=C)=O)CC2)C)ccc(C)cc1Cl C1(C)(C(N(C(C=C)C)C)=O)CC(O)CN1C(c1cc(O)ccc1F)=O c1(C(=O)NC2C3CN(C(C4C(C)C4)=O)CC32)c(F)ccc(Cl)c1F Cc1ccc(Br)c(CC(=O)NCCN2CCSC(c3ccccc3)C2)c1 c1(CNC(C(F)=C(C)C)=O)c(C)nn2c1CN(C(=O)CSC(F)F)CC2 C1(NC(c2c(C)noc2N)=O)CCN(C(C2CCCC2)=O)CC1c1ccccc1 C1(C(=O)OCCC#CC)CC2(C1)CC1(CCC1)C2 C1(C(=O)NCC(C(=O)NC(c2ncnn2C)CC)N(C)C)CCOCC1(C)C c1(CCC=O)ccc(F)c(F)c1.c1(OC)ccccc1C(=O)NCCC1CC1 C1(NC(CCN(C(=O)CC2CCSC2)C(C)C)=O)CCn2ccnc2C1 c1(OC(c2cc(CC)c(F)cc2)=O)cnc2onc(C)c2c1 c1(C(=O)NC2C3CN(C(c4n(C)nnc4)=O)CC32)ccc(I)c(F)c1F c1(C(N2CC(CN(C(c3c(C)cn(C)n3)=O)C)C2)=O)cnc2n[nH]c(C)c2c1 c1(NC)ccc(C)cc1C(N1CC2CCC2(CCNC(=O)CC(F)F)C1)=O N1(C(C=CCN(C)C(C2Cc3nccn3C2)=O)=O)CCC(C#N)CC12CC2 C1(S(N)(=O)=O)(C(=O)NCC(C(C)C)NC(=O)C(C)C#N)CCCC1 C1(C(C)C)CN(C(=O)CCc2ccc(O)nn2)CCN1C(=O)C(C)CC(N)=O c1(C(N(C)CCOCCN(C)C(C2CSC2)=O)=O)sccc1-n1cnnn1 C1(C(N(C2CCN(C(C(CCCC)O)=O)CC2)CCC)=O)CC=C(C(C)C)CC1 C12(NC(c3c(C)coc3)=O)CCC(C1)N(C(c1c(C(F)(F)F)noc1C)=O)C2 c1(CC(N2CC(CC(=O)NC3(C#N)CC3)C2)=O)c[nH]c2ccc(F)cc12 C(CCCCCNC(C1(COC(C)C)CC1)=O)NC(CCC=CC)=O N1(C(c2c(CC)ncnc2)=O)CCN(C(=O)C=Cc2ccoc2)C(C2CCC2)C1 O(NC(=O)C(C(C)NC(C1CC(CF)C1)=O)C(C)C)CCC(C)C C(=O)(C1CCCn2nccc21)N1CC2C(CNC(c3nc(Cl)ncc3Cl)=O)C2C1 CC1CN2CCN1CC2C(=O)NC1(C)CCN(C(c2cc(F)cc(F)c2N)=O)C1 CC1(CNC(=O)C(O)Cc2cnc[nH]2)CCCN(C(C2CSCC(=O)N2)=O)C1 Cc1cc(C(=O)NCCC2CCCC2)n(C)n1.c1(C(=O)N)ccc[nH]1.N(C)C O=S(=O)(c1ccncc1)N1CC2CC1CN2Cc1cnc(Cl)nc1Cl C1(NC(CC(=O)OCC)=O)CCN(C(c2cc(Br)cc(Br)c2)=O)C12CCC2 N1(C(CSCC)=O)CC=CC1(C)C(=O)NCC1(CO)CC1 C1(CNC(C(n2cc(C)nc2)(C)C)=O)CCCCC1.C(=O)C.C(=O)C1CC1 c1(OC)cc(CNC(C2CCCC2NC(c2cnn[nH]2)=O)=O)on1 C1(C(N(CCCNC(CSCC#C)=O)C)=O)CCOC(C)C1 C(=O)(CC(C)(C)C(=O)NCC1(C(=O)N)CC12CCC2)OC.C1CC1.C C1(N(C(C2C(C)=CCS2)=O)C)CN(C(c2ccc(C(N)=O)cc2)=O)CC1(C)C C1(NC(CCC=CC)=O)CCC(C)(C)C1.C1(CC=O)CN(C(C)=O)C1.N C1(C(N(CCCNC(=O)C(O)C(C)C)CC)=O)Cc2nncn2C1 c1(C(=O)NC(CNC(c2ccc(C)cc2C)=O)C2CC2)cc(O)cc(N)c1Cl c1(C(=O)NC(CCC=C)C(=O)N(CCCCCCC)C)cc2ccccc2o1 C(C(C(=O)NOCCC1CC1)NC(=O)C(C)C(F)F)OCC c1(CC(=O)NC2CN(C(c3ncnc(O)c3Cl)=O)CC23CC3)cccc(O)c1F CC1OC2CCC1(C(N1CCOC(C(N3CCN(C4CC4)CC3)=O)C1)=O)C2 C1(NC(c2n(C(C)C)ncc2)=O)CCN(C(=O)CC2(C)CC2)C(C)C1 C1(CNC(CCCC#C)=O)CCC2(CCC2)CN1C(c1cc(C(C)C)[nH]n1)=O c1(CC)nc(C)oc1C(=O)NCC1(C)CCCN1C(c1scnc1Cl)=O C1(C(=O)NCCC(=C)CNC(=O)CCNC(C)=O)CCCCC1OC Cc1nc(CCNC(C2CN(C(c3ccc(O)nc3)=O)CCO2)=O)c(C)[nH]1 C1(N(C(C(C)=CC2CC2)=O)C)CCCCC1NC(c1c[nH]ccc1=O)=O C1(C(N2CC3C(NC(c4cc5ccsc5s4)=O)C3C2)=O)CC2(CCCCC2)CO1 C1(C(N2CC(CC(=O)NC3CCc4nn[nH]c4C3)C2)=O)CCc2ccccc2N1 S(=O)(=O)(c1ccc(C(=O)NCCCO)cc1)NC(c1ccc(F)cc1)C(C)C C1(C(=O)NCCc2n(C)ccn2)C=CCCN1C(=O)CC1COC(=O)C1 C1(C(N2CC(CNC(CCCC)=O)CC2(C)C)=O)CC12CCC(=O)CC2 c1(CC(=O)N(C)CC2CCCCN2C(c2ccc(F)o2)=O)c[nH]c2ccccc12 Cc1nnc2c(C(=O)NCC(C)(C)CN(C(=O)Cc3c[nH]nc3O)C)cccn12 N1(C(Cn2c(C)ccn2)=O)CCOC(CNC(=O)CCCc2ccccc2Cl)C1 c1(CC(N2C(C(N3CCC(CCOC)CC3)=O)C(O)CC2)=O)cccc(C#N)c1 C(=O)(CCC(=O)NC1CC(C)C1)NCC=C.C1(C(=O)N)CCC1.C1CC1 N1(C(C(C)=C(C)C)=O)CCCC(CO)(NC(=O)CN2CCC(N(C)C)CC2)C1 C1(COC)CCCN(C(=O)CCC2CCC(=O)C2)C1.C(=O)CCC1CC1(F)F Cc1ccc(CN(CC(=O)O)C(C2CCC(F)C2)=O)cc1 C1(OC)CN(C(C2CCC(=O)O2)=O)CC1NC(=O)C=CC(C)C c1(C(=O)NCC2CCC(C)CN2C(C2C=CC=CC=C2)=O)cccc2cc[nH]c12 c1(C=O)cc(C(C)C)ccc1F.N1(C(c2n(CC)ncc2)=O)CC(F)CC1C.N c1(C(=O)NCCC(=C)CNC(C2CCC(C)C2)=O)ccc(C)c(Br)c1C CC(C)(CNC(=O)Cn1cnc(=N)[nH]1)C.c1(C=O)cscn1.CC(F)F.N c1(CN(C(C(C(=O)OCC)F)=O)CCCC(=O)OC)c(OC)ccc(Cl)c1F C(=O)(C#CC1CCCCO1)NC1CCCN(C(C(CC(C)C)(F)F)=O)CC1 S(=O)(=O)(c1cnccc1NC)N(C)CC1(C(F)(F)F)CC1.C1C=CCC1.C N12CC(C(O)C1)C2=O.N1(C(C=CC)=O)CC(N(C)CC)C1.C(CO)OC C#CCCCCCC(=O)NC(CC=C)CC(=O)N(C)CC1CCCS1 c1(C(C)C)nc(C(=O)NC(CC2CC2)C(=O)N(C)CC2CCOC2)co1 CCCCCCNC(c1cccc(NC(=O)C2CC2)c1)=O.C1(C=O)CCCO1.N c1(C(=O)OC)cc(CNC2CN(S(=O)(=O)CC)CC2C#N)c(Br)cn1 C(CC(C(=O)NCc1ccco1)N(C)CC1CCCN(C(C)C)C1)SC c1(C(=O)NC(C(=O)NC(CC(=O)NC)C)c2ccco2)cccc[n+]1[O-] C1(C(=O)NCC(C)N(C(c2ccc(NC)cc2)=O)C)CC12CC(C)(C)C2 C(=O)(CC(O)CCCC)NCc1c(C(=O)NC(CCCC=C)C)cccn1 c1(N2C(C)CC(NC(Cc3nc(C)c(C)s3)=O)C2)ncc2c(n1)CCCCC2 Cc1cc(C(=O)NC(C)C(C)C(=O)O)cc(O)c1 C(=O)(C(CCc1ccccn1)N1C(CC)CCC1C)NCC(=C)C N1(C(C=NOC)=O)C2CCC1CC(CNC(=O)C(C)Sc1nnnn1C1CC1)C2 C(CCCCC(=O)N1CCC(C(N2CCC(C(C)C)(CO)C2)=O)C(C)C1)OC C(CC(C(=O)N)NC(=O)OC(C)(C)C)=CC.c1ccnc(C(F)(F)F)c1 C(C1CCCO1)=CC(N1CCC(N(C(=O)CCc2ccncn2)CCO)C1)=O c1(CNC(C2C3CC2N(C(c2cnn[nH]2)=O)C3)=O)cnc(O)nc1O CC1(C(=O)NC2CCC(NC(=O)CSS(C)(=O)=O)CC2)CCCCNC1=O c1(C(N2C(CCCNC(CC3C(CC)C3)=O)CCC2)=O)ncc(C)cc1F c1(C(=O)NC2(C)CCN(C(C3CCS(=O)(=O)C3)=O)C2)ccc2c(c1)COCO2 c1(C(=O)NCCN(C(=O)C(=O)NC2CCCCC2)CCC)ncccc1O.O c1(C(N(CC(=O)NCCOC)C)=O)ccc2c(C(=O)N(C)C)n[nH]c2c1 N1(CC=O)CC(C)CC1C.c1(CNC(=O)NCCCC)cscc1OC.N C1(NC(CNC(C(C)(C)C)=O)=O)CCC(N=c2[nH]ccnc2F)CC1 CCC(C)CC(C(=O)N1CCC1CC(=O)NC)NC(c1ccc(SC)o1)=O CON(C)CCCN=c1nc2c(cnn2-c2ccccc2)c(N)[nH]1 c1(C(N2C3(CN(Cc4c(OC)cccn4)C3)CC2)=O)ccnc2c(Br)cccc12 N1(C(Cc2c(C)cnn2C)=O)CCC(C)C(F)(F)C1.C(=O)CCC1CC1(C)C.N Cn1cc(NC(=O)C(=O)NCc2sc(Cl)cc2Cl)c(-c2cccs2)n1 C(=O)(CCCN=C(NCC1CCCO1)NC1CCN(S(=O)(=O)C2CC2)CC1)OC c1(C(=O)NCCC(C)NC(C2CCC(C)(C)O2)=O)ccsc1S(N)(=O)=O C(=O)C1=C(C)NC2=NCCCC2=C1.C1(C(C(=O)N)OC)CCOCC1.CC=CC c1(C(=O)NCC(CC)NC(=O)C(c2nc(F)ccc2Cl)C)ccc(C)c2c1CCC2 CC1CCn2ncc(C(=O)NC(CCN(C(=O)C=C(Cl)Cl)C)C(C)(C)C)c2C1 O=C(C(O)CC(F)(F)F)NCCCC1CCN(C(C2SCCCS2)=O)CC1 C(=O)(CC(F)(F)C(F)F)NC(CCC(=O)NC(CCC)CCO)C C(=O)(CCC(=O)N1CC(OC)CC1CNC(c1coc(CO)c1)=O)NCC N1(C(C(c2ccc(Cl)nc2)C)=O)CC2(C1)CN(C(C1(c3cnccn3)CC1)=O)C2 O=C(C1CCc2nccn21)NC1CN(C(=O)Cc2cn[nH]c2)C2(CCCC2)C1 N1(C(COCCC#C)=O)CCCC(C(=O)NC(C)COCCOC)C1 c1(C(N2CC3C(CN(C(=O)C(C)(C)C(F)F)C)C3C2)=O)cc(F)c(F)cc1F Cc1ccc(C)c(N2CC(C(N3CCCC3C(=O)NC(C)(C)C)=O)CC2=O)c1 CC1C(C)N(C(c2cncc(F)c2)=O)CCN1C(=O)C=CCn1cncn1 c1(CC(N2CCN(C(CC(C=C)C)=O)CC2CC)=O)c[nH]c2ccc(F)cc12 Cc1cnc2n1CC(C(=O)NCCNC(c1ccc(Br)c(O)n1)=O)CC2 c1(C(N2CC(NC(COC)=O)CC(C)(C)C2)=O)c2c(c[nH]c1=N)CCC2 c1(C=O)ccc(C(C)=O)nn1.C1(C(C)C)CC1C(=O)N(CCC)CC C(=O)(CCCS(N)(=O)=O)NCCC(C)N(C(c1c(C)nc(Cl)cc1)=O)C c1(C(=O)NCCCOCCNC(Cn2c(C)nnn2)=O)cnn2c1C(C)CCC2 CCS(=O)(=O)C=CC(=O)N.C1CC(C)(C)CN1C(c1nc(C2CC2)cs1)=O.C CC1(C(=O)NCCC2CCN(C(c3n[nH]cc3Cl)=O)C2)CNC(=O)N1 N1(C2CCC(C(=O)OC)C2)CCN(C)C(CO)C1.C1(=O)C(C(C)C)N1 C12(C(N3CCCC3)=O)CC3CC(CC1C3)C2.C(C(=O)NC)(C(C)C)OCC.C C1(CNC(CN(CCC)C)=O)CN(C(=O)C#CC2CC(F)(F)C2)CCC12CCC2 CC(C)C(F)(CNC(c1ccn2cncc2c1)=O)C(=O)NC(CCO)C(F)(F)F c1(C(C)C(=O)NCC(F)CNC(=O)CC2CS(=O)(=O)C2)ccc(F)cc1 c1(SC)ccc(NC(C2CN(Cc3cc(F)ccc3F)CCC2O)=O)cc1F C1(CC(=O)NCCC2(O)CN(C(C3CCCC3)=O)C2)COc2ccccc2O1 c1(NC(C)=O)ccc(N2CCC(NC(=O)C(C)Cc3ccccc3C)C2)cc1 C(=O)(C1CCCc2ncnn21)N(C1CCN(C(c2csnn2)=O)C1)C CC1CC(NC(c2cc(-c3cnn(C)c3)on2)=O)CN(C(=O)C=O)C1.C1CC1.N C1(NC(C(C)OC2CCCCC2)=O)CN(C(=O)C(C)(O)C2CCC2)CC1(C)C C(CCCCC(=O)NCCn1cnc(C(=O)NC2CNC(=O)OC2)c1)N(C)C C(=O)(CCCCC(N)=O)NC1CN(C(C(C=C=C)C)=O)CC12CC2 c1(NC(C2CCCC(NC(=O)CCCCBr)C2)=O)c(C(F)(F)F)cccc1Br C1(C(=O)NC2CSC2)CCCCN1C(C1OC2CCC1C2)=O N1(C(Cc2ccc(C)cc2)=O)CC=C(C(=O)NCCC(C)C(C)(C)C)C1 Cc1ccc(C(=O)NC2CC3(C2)CN(C(C2C(C)CC2C)=O)C3)c2ncccc12 C1(C(N(CCC)CC)=O)CCC1(C)C.C(O)(C(F)(F)F)C1(C=O)CCC1.N C(=O)(CCC(C)(C)[N+](=O)[O-])N1C(CNC(CCC#CC)=O)C=CC1 C12(NC(c3cc(Cl)c[nH]3)=O)COCCC1CN(C(c1csc(Cl)c1)=O)C2 CP(C)(=O)CCC(=O)N1CCOC(CC(=O)NCCC2CCC(=O)N2)C1 c1(C(=O)NC2(CO)CN(C(C(CC)c3ccccc3)=O)C2)ccc(=O)n(C)c1 CC1=NOC(C(=O)NCC2CCN2C(c2cc(C)nn2C)=O)C1C C1(NC)CCN(CCCCCNC(C2(NC)CCCC2)=O)CC1 C1CC2CC1N(C(C1CC1)=O)C2.c1(CC)nc(C)c(C(=O)NC)s1.C=O C1(C(=O)Nc2cc(C)c(O)cc2)COC2(C1)CN(C(c1cnc(O)cc1O)=O)C2 C1(N(C(c2c(COC)noc2)=O)C)C2CN(C(C3(C)C=CCCC3)=O)CC12 C1(NC(C(C=C)O)=O)CCC(C)(NC(=O)CN2C(=O)CCC2=O)CC1 C1(NC(c2ccc(C(C)=O)[nH]2)=O)COC2(C)CC1C2.C(=O)C(C)(C)N(C)C C1(CC(=O)NCC2C=CCCC2)CCN(C(c2cnc(Cl)nc2)=O)CC1 c1(C(=O)NC(CCCC)CNC(=O)CC2CC2)cc(OC)nc(C)c1 c1(CC(=O)NC(c2ccc(F)c(F)c2)COC)cc(Cl)c(Br)cc1F CN1CCc2nc(C(=O)NC3CN(Cc4cc(F)cc(F)c4Br)CC3F)sc2C1 N1(C(C2CC(=C)C2)=O)CC2CN(C(c3cc(SC)ccc3O)=O)CCC12 C1(C(=O)NCC(C)C(C)(C)C)CNC(=O)CN1C(c1cnns1)=O CC(CC(F)F)C(=O)NCCC1CC(NC(=O)COCc2ccnn2C)C1 N1(C(C(=O)N(C)C)=O)CCN(C(=O)COCC(C)(C)CN)CC1 c1(C(=O)NCCC2CCN(C(C(CCC)CC)=O)C2)cccc([N+](=O)[O-])c1Cl CC1(NC(c2nccs2)=O)CC(NC(=O)C(O)c2cnc[nH]2)C1 c1(CC)ccc(C(N2CC3(CCN3C(=O)Cc3ncc(C)s3)C2)=O)c(F)c1 C1(C(N2C(C)CN(C(=O)C3=NNC(=O)C3)CC2)=O)CCc2nc[nH]c2C1 C1CCC=CCCC1.N1(C(C2C(OC(C)=O)C2)=O)CC(O)CC1CC(=O)NC c1(C(N(CCNC(C(CCCCC)CC)=O)C)=O)ccc2c(c1)CN(C)C(=O)N2 C(=O)(C1=C(C)CCOC1)N1CC=CC(C(=O)NCC(=O)NCCC)C1 C1(CNC(c2ccc(O)nc2)=O)CC(O)CN1C(=O)CC12CCC(CC1)C2 C(=O)(C1CCCc2nn(C)cc21)NCC(C)(C(C)C)NC(COC(C)=O)=O c1(C(=O)OC)c(C)oc2ncnc(N)c12.N1(C)CC2CC2C1.C1(Br)(C=O)CC1 n1(CC)nc(C(N2CC3CC3(NC(=O)Cc3ccc(O)cc3)C2)=O)c(C)n1 C(C)(CCC(=O)NCC1(SC)CC1)NC(c1cc(CC)no1)=O C1(C=O)CCc2cnnn2C1.S(=O)(=O)(CC(=O)NC1CCCC1)N(CC)CC CC1COCC(CNC(=O)C(C)N(C(c2cnncc2O)=O)C2CC2)O1 Cc1ccc(C(=O)NCC2CN(C(=O)CC3(O)CCCOC3)CC23CC3)nc1O C1(CC)C(CN(c2ccccc2Cl)C(=O)C=CBr)CCN1C(=O)Cn1cccn1 c1(CC)ccc(F)c(C(=O)NC2CC23CC(NC(C2CCCS2)=O)C3)c1 N1(C(C(=O)NC(=O)NCC)C)CC=C(CC)CC1.C1(C)(C=O)CCCO1.N C1(OCC)CCC(C(=O)Nc2ccc(NC(=O)OC(C)(C)C)cc2)CC1 c1(OC)ccc2[nH]c(CNC3CC3C=O)cc2c1.c1ccc(F)nc1C(N)=O C(=O)(C(C(=O)O)C(C)(C)C)NCc1ccc(-n2c(C)ncc2)c(F)c1 C(C)(C)(CCCCNC(=O)CC(C)C(F)F)NC(Cc1nc(C)sc1)=O CCCCCC(CC)C(=O)NC(C1CCCN1C(=O)C=C(C)C)(C)C C1(C)(C=O)CC(=O)N(C)C1.C1(CNC(CSC(C)C)=O)CC(F)C1.C C1(NC(c2cc(OC)ncn2)=O)CC2(CCC2C(=O)OC(C)=O)C1 Cc1cc(CNc2cnc(F)cc2C(=O)NCC2CCN(C)CC2)cnc1C N1(C(CC)=O)CC2(CC2)CC1.C1(F)(C=O)CCS(=O)(=O)C1.C(=O)NC.N C1(C)(C(N2CCC(C(C)(C)NC(C(C)CO)=O)CC2)=O)CCC(F)(F)C1 C1(C(=O)NCC2CCCN(C(C(=O)Nc3ncc[nH]3)=O)C2)Cc2cscc2C1 c1(C(=O)NCCC2CCN(C(=O)C3=CC(O)CCC3)C2)ccc2cc[nH]c2n1 c1(C(N2CC(N(C)C(C3CCCCC3O)=O)C2)=O)cnn2cccc(Cl)c12 N(C1CCc2cc(CNC(C3(C)CCCC3)=O)ccc21)C(C1C(OC)C1)=O N1(C(C2N(CC)CC2)=O)CC(C(=O)NCc2nc(C)ccc2C)CC1(C)C c1(C(N(C2CC(NC(C3(C)CCOC3)=O)C2)C)=O)cc2ccccc2c(O)n1 Cc1nc(CCCC(=O)N2CC(N(C(=O)C=Cc3cccs3)C)C2)cs1 c1ccc(N)c(C)c1F.CCC(C)(C(=O)N)NC(C1CC2(C1)CC2C=O)=O c1(C(=O)NC2CC3CC(NC(=O)CC4(CO)CC4)C3C2)c[nH]c2cnccc12 C(CN=C(NCC(F)F)N1CCC(C)(C(N)=O)C1)c1ccc(OCCC)cc1 C1(C(N2CCC(NC(C(CC)(F)F)=O)C2C)=O)C2CCC(C2)C1C(F)F C1(CC(C)NC(c2n[nH]c(C)c2F)=O)CC2CCC(C1)N2C(=O)CCCC(C)C Cc1cccc(CC(=O)NCC2CC2C)c1Cl.c1(C(=O)N)cc(N)cc(O)n1 C1(CNC(C=CC(CC)C)=O)CN(C(=O)CCOC)CCCO1.C1CCCO1 C1(C(=O)NC)CC(O)CN1C(c1cc(Cl)c(Br)s1)C(=O)Nc1ccccc1O C1(NC(c2c(C)cc(Cl)nc2N)=O)CN(C(=O)CC2CCOC2)CC2(CCC2)C1 N1(C(C(CC2CC2)OC)=O)CCC2C(C(=O)NCCc3nnc(C)s3)C2C1 C(=O)(C1=CC2(CCN(C(C3CC4CC(=O)C3C4)=O)C2)C1)N.CC(CC)N1CCC1 c1(CNC(c2ccc(C)cc2)=O)cccc2c1CN(C(=O)CCn1cccc1)C2 N1(C(CC2CCC(NC(C(CC)CC)=O)C2)=O)CC2CC1CS2=O c1(C(=O)OC)ncnc(N2CCOC(C(=O)NC3CCC(C)CC3)C2)c1F C1(C(=O)NC(C(=O)NCc2c(C)noc2)C2CCCO2)CCCSC1C Cn1cc(C(=O)NC2(CO)CCN(C(=O)C(C)(C)C3CCOC3)C2)ccc1=O Cc1cc([N+](=O)[O-])cnc1C(N1CC2CCN(C(=O)C(=O)NC3CC3)CC2C1)=O c1(CC)nc(C)c(CC(=O)NC2CCCC2NC(C2CCN2C)=O)c(C)n1 C=CC1OCCCC1C(N1CCC(CC)(NC(c2csc(C(F)F)n2)=O)CC1)=O c1(CC(=O)NC(CNC(C2(CC=C)CCOC2)=O)CC)cccc(C)c1 O=CCC(CCCC)Cc1ccccc1.C1(O)(C(N(CCC)C2CC2)=O)COC1 C(=O)(CC(C)(C)C(F)(F)F)NC1C(C)CN(C(c2cncn2C)=O)CC1 N1(C(Cc2nc(CC)sc2)=O)CCOC(CNC(c2ccc(C)s2)=O)C1 N1(Cc2cc(OC)cc(OC)c2)CCC2(CCCN(C(C3CC3(C)C)=O)C2)CC1 c1(C(N2CC(C(N(CC=C)CC=C)=O)(COC)C2)=O)n[nH]c(C)c1Cl c1(-c2n(CC(C)C)ncc2)cc(C(=O)NC2CN(C)CC2(C)C)ncc1F c1(C(N2CC(NC(c3n(CC)cnn3)=O)C2)=O)cn(C)c2c(cnn2C)c1=O C(=O)(C(C)(C)N=[N+]=[N-])NCC1C(C)CN(C(=O)Cc2ccon2)C1 c1(C(N2CCCC(C)C2CNC(=O)CS)=O)cccc2c1OCCC2.C(C)(C)C C1(C(N(CC(C)C#N)CC)=O)CCCN1Cc1nc(O)n[nH]1 Cc1ccc(C(C)C)c(NC(=O)NCC(C)CN(C)C)c1.N1CCOC1=O C(=O)(C1=C(Cl)CCCC1)NC(C(=O)NC(COC)C1(C)CC1)CCCOC C1(CC)CN(C(c2ccn(C(C)(C)C)c2)=O)C1.C(C)(C=O)OCCOC C1(C(=O)NC2CN(C(CCNC(=O)C=CCl)=O)CC2F)CCn2cnnc2C1 c1(C(=O)NC2CC(CCNC(c3n(C)c(S)nn3)=O)C2)cc2ncccc2[nH]1 C1(C(=O)NC(CCNC(CCc2onc(C(C)OC)n2)=O)C)CC2CCC(C1)O2 C1(C(=O)NCC(N2CCCCC2)=O)(NC(C2N(C)CCC2)=O)CCN(C)C1 c1(C(N(CCNC(C2C3COCC23)=O)C2CC2)=O)ccc(O)nc1Cl C(CC(C)(O)NC(=O)CCc1ncnn1C)N(C(CC)=O)C N1(C(c2c(CC)noc2C)=O)C2CCC(C2)C1C(=O)NC(C)C(C)(C)CO C(=O)(CCCCC(C)C)NCC(CNC(c1c(NC)nc(C)cc1)=O)(C)OC c1(CC)nn(C)cc1C(=O)NCC1CCC(N(C)C(c2sncc2C)=O)CC1 c1(C(N2CCC(N(C(c3cccnc3C)=O)CC)CC2)=O)cc(C)c(C)cn1 Cn1c(C(=O)NCC(C)(CO)NC(C2(c3ccno3)CCC2)=O)ccc1[N+](=O)[O-] C(=O)(C1=CCCN(C(C2CCC3(CC3)C2)=O)C1)NCc1cccc(OC)n1 CN1Cc2ccc(C(=O)NCC(CO)NC(C3CNC(=O)C3)=O)cc2C1 C=CCC(CC=C)C(=O)N1CC(OCCC(=O)NC2(CC(N)=O)CC2)C1 C1(N(C(C2CCCC2)=O)Cc2cccs2)CCC2(CC2)C1 c1(C(N2C(CNC(Cc3c(C)n[nH]c3)=O)CCCC2)=O)n[nH]c2c1CCCCC2 CCN=C(NC1CC1Oc1ccc(F)c(F)c1)N1CCCC(CC2CC2)C1 Cn1c(Cl)cnc1C(=O)NC1CN(C(=O)COC2CCCOC2)C1 c1(OC)ccc(C(N2CCC(C)C2)CNC(=O)C(=O)N)cc1.C1(N)CC1.C C1(O)(CC)CCCN(C(C2(C(C)C)COC2)=O)C1.c1(OC)sccc1C(=O)N CC(CCC(C)(C)C)NC(C1CC(C)CCN1C(C1CC1C(N)=O)=O)=O c1(C(N2C(C)(CCC)CC2)C(=O)NCc2ccco2)cc(Br)c(Cl)s1 C(c1cccnc1)=CC(=O)NCCC(C)OC.C(=O)C(C)CC1CCCC1.N Cc1c(Cl)ccc2[nH]c(C(=O)NC(C)CNC(=O)C(c3cncnc3)C)cc12 C1(NC(C2CCCOCC2)=O)C=CCN(C(=O)CC2OCCO2)C1 c1(C(=O)NC2CC(NC(c3cnn(CC)c3Cl)=O)C2)cc(C#N)n(C)n1 C1(C(=O)NCC=CCNC(CN2CCC(C)C2)=O)CC(C)(C)CN1C c1(CNC(c2cccc(OC)c2)c2nnnn2CCSC)ccc(N)c(Cl)n1 C1(CNC(CCC)=O)CN(C(=O)Cn2cc(C3CC3)cn2)C2(CCC2)C1 C(C(C)(C)C)NC(C(c1ccnn1C)C)=O.C1(CC(=O)N)CC(n2cnnc2)C1 C(=O)(C1CCc2ccccc21)N(CCC(N1C(C(N(C)C)=O)CC1)=O)C1CC1 c1(C(=O)NCC2CN(C(C(C3CCOCC3)OC)=O)CC2O)c(C)cnnc1O c1(C=O)ccc(C(C)(F)F)cc1.N1(C(C)=O)CCC(C(=O)NC(C)CC)C1.N C1(CCC=O)NC(=O)NC1=O.C1(CC)CCN(C(C2(N(C)C)CC2)=O)CC1.N N1(C(CCCC)=O)CCCC(C(C)(O)CNC(=O)C(F)(F)C2(O)CCC2)C1 C1(NC(=O)Cn2cnc([N+](=O)[O-])n2)CN(C(C2CC(F)(F)C2)=O)CC12CCCC2 O(NC(=O)CCN(C(c1c[nH]c(=NC)s1)=O)C1CC1)C(C(=O)OC)C C1(C(N2CCC(NC(c3occ(OC)c(=O)c3)=O)C2)=O)CCc2nnnn2CC1 C(=O)(C(O)CC(N)=O)NC(C1CN(C(c2cccnc2-c2ccncc2)=O)C1)C CC1COCCC1C(=O)N(CC(C)(C)NC(=O)CSc1nc[nH]n1)C c1(OC)nc(N2CCC(NCc3cccc(CO)n3)C2)ncc1C C1(C(=O)N)(COC)C=CCN1C(C1CC(=O)C1(C)C)=O.C1C=CCC1.C CC(C)CC(C(=O)NC(C)CCO)C(N)=O.C1(C=O)(C=O)CC1.C(C)(C)C N1(C(COC)=O)CCC(C2(O)CN(C(c3cc4cccc(C)c4nn3)=O)C2)CC1 N1(C(C2CCN(C(C)=O)C2)C(=O)NC)CCC(N(C)CCc2ccccn2)CC1 Cc1cc(Br)c2ncnc(NCC3CCCC(F)(F)C3)c2c1 N1(C(C2N(C)CC2)=O)CCC(C(O)CNC(=O)Cn2cc(C(F)F)cn2)CC1 C1(O)(C(CNC(c2c(OC)scc2)=O)C)CCN(C(c2cnc(OC)nc2)=O)C1 Cc1cnc2nc(C(N3CC4C(NC(c5cncnc5)=O)C4C3)=O)nn2c1 C1(C2CCCC2)(C(=O)NCC(CN(C)C(c2ccc(=O)oc2)=O)O)CCNC1=O CCC(CC(=O)N1CC2(CCCCN(C(c3cnc(O)s3)=O)C2)C1)CC(F)(F)F C1(C(N2C(C(=O)NCC(C3CCCC3)OC)CC2)=O)(C)CCCC1.C1CC1 c1(C(N2CC(NC(C3CCN(CCC)CC3)=O)(CO)C2)=O)cccc2nc[nH]c12 c1(C(N2C(CCCNC(=O)CC3CCCC3)CCC2)=O)nnn2c1CCC2 c1(OC)c(Cl)ccc2[nH]c(C(=O)NC(C)CS(=O)(=O)N3CCCC3)cc12 Cc1ccc(CCC(=O)N(C(CNC(=O)Cc2sc(C)nc2C)C2CC2)C)cc1 C1(NC(C2C(C(C)C)C2)=O)CC(O)C1CC(N1CCC(CCO)C1)=O c1(C(=O)NC(C(C)NC(=O)CCc2ccoc2)CO)cc(Cl)c(Cl)c(Cl)c1 O=C(CCC(F)F)NC1CCN(C(=O)COc2ccc(Cl)nc2)CC1 CCCC(CC)C(=O)NC1CC(C(=O)NCC2CCCC23CCC3)CC1O Cc1n[nH]c(C)c1C(C)CC(=O)NC1CC(CO)N(C(c2nncs2)=O)C1 CC1(C)OCCNC1C(=O)Nc1ncccc1N1CCOCC1 c1(C(=O)NCC2CCCN(C(C(C)O)=O)CC2)c(F)ccc2occc12 c1(C(=O)CNC2CCC23CCNCC3)ccc2c(c1)CCO2 N1(C(C2CCN(C(C)=O)C2)=O)CCC(CO)(NC(=O)C(N2CCOCC2)C)CC1 CCCC(C)(O)CC(=O)NCCC(CC)(CC)NC(=O)CC(C)(C)SC C1(NC(C(CCC)N(C)C)=O)CC(F)CN(C(c2cc(C)on2)=O)C1 C=CCCC(C(=O)N(C)CC1(C)CCCO1)NC(=O)CCC(C)(C)F N1(C(CCN(CCCCC)C)=O)CCC(F)C(NC(C2(CCOC)CCC2)=O)C1 C1(NC(c2cccc(C)c2C)=O)Cc2ccccc2C1NC(c1cnns1)=O CC(CS(C)(=O)=O)C(=O)NC1CCN(C(c2cnc(S(C)(=O)=O)s2)=O)C1C N#CC1CCCC(C(N2CCC(N(C(=O)CCc3ccncn3)C3CC3)C2)=O)C1 c1(C(=O)NC2(COC)CCN(C(=O)CCc3ccnn3C)C2)n[nH]c2c1CCC2 N1(C(C(C(C)C)C)=O)CC(CC(=O)NOC2CC2)C2(CC2)C1 CCC(C)(C)C(C)CC(=O)NCC1CN(C(c2csc([N+](=O)[O-])c2)=O)CCCO1 C(CCC(C)C(=O)N1CCC(C(C)NC(=O)CCC2CCCCN2C)CC1)OC CC(F)(F)C(C)(C)CNC(=O)CCC1(C)CCCN1C(=O)C1=CCOCC1 c1ccc(Cl)cc1.C(C)(C)(CCNC(=O)C)NC(C(C1CCCOC1)OC)=O c1(OCC)cc(Br)c(NC(=O)CSc2ccc(C)c(F)c2)cc1OC C1(C(=O)NC(C)CCN(C(=O)CC2CC(C(F)F)C2)C)CCN(C)CC1 N1(C(COCCCCCC)=O)CC2CC(C1)N(C(=O)CSSC)C2 N1(C(c2n[nH]c(C)c2Cl)=O)CCC2(CC(NC(C3Cc4cccnc4C3)=O)C2)C1 Cc1cc(N)ccc1C(=O)NC1(CO)CCCN(C(=O)CC2CCN(C)C2)C1 N1(C(CCCCC)=O)CCC(c2ccccc2)(NC(c2cc(CC)no2)=O)CC1 c1(CNC(c2n(CCCOC)nnn2)c2nccn2C)nccc2ccccc12 C1(C(=O)NCC(CC)OC)CCN(C(=O)c2[nH]nnc2C2CC2)O1 C1(C(=O)Nc2cncc(C(C)C)c2)C2CC1CN(CCOCc1ccccc1)C2 CCC(C)C(O)C(C)C(=O)NC(C)(C)CC(=O)NC.C1CC(=O)N1C CCC(C)C=CC(=O)N(CCC(=O)N(C(C)CC1CCCO1)CC)C(C)C N1(C(c2c(CNC(CN(C(C)=O)C)=O)ccs2)=O)CC(C)OC(C)(C)C1C CC1=C(C(=O)Nc2cccnc2C)C(c2cnn(C)c2)NC(=S)N1C C12(C(=O)NC3CCCN(C(CN(C(C)=O)C)=O)CC3)CCCN1S(=O)(=O)CC2 c1cccc(C#N)c1.n1(CC)cnnc1NC(c1nnnn1C1(C)CC1)(C)C.O C1(NC(C(COC)C)=O)CCC2(CC1)CC2.c1(C(=O)N)csc(-c2cn[nH]c2)n1 c1(C(=O)NC(c2nc[nH]n2)C)n[nH]cc1CNC(c1cncnc1)=O C(=O)(CCCC(=O)N1CCC(CO)(NC(=O)C(C)Cc2c(C)noc2C)C1)NC C1(NC(=O)COCCCF)CN(C(c2cnn3c2CCCC3)=O)CC12CCC2 C1(N(C)C)CCCCN(C(c2ccc(I)s2)C(=O)NCCC#N)C1 C1(C(=O)NC2CC(NC(C3(c4nc[nH]n4)CC3)=O)C2)(CO)CCCO1 C(=O)(CCCN(C)N=O)NCCC(C)N(C(c1c(C)nsc1)=O)C C1(NC(C2C(C)OCC2)=O)CCN(C(C2CCC(N=[N+]=[N-])C2)=O)CC1C c1(C(N(C)CCOCCN(C)C(C2(C)CCC2)=O)=O)cc(F)cc(F)c1O C1(SC)CN(C(=O)C=Cc2cc[nH]n2)CC1.C(c1ccccc1)=CC(C=O)C.N N1(C(CC2(OC)CCC2)=O)CCC(NC(c2ccncc2C)=O)C(F)C1 C12CCCC1CCN2C(c1ccc([N+](=O)[O-])o1)=O.C(c1cn[nH]c1)=CC(=O)NC c1(COC(c2c(N)c(Br)ccc2Cl)=O)cc(Cl)cc2cccnc12 C1CC(F)(F)CN1C(=O)C=CCn1cncn1.c1(C(=O)N)ccncn1.C c1(CCCC)ccc(CC(=O)NCC(C)CNC(=O)C(C)NC(C)=O)cc1 N1(C(COCC)=O)CCCC(NC(=O)C(O)C(F)F)C1C C(c1cccc(F)c1F)=CC(N1CCN(C(C2C(F)(F)C23CC3)=O)C2CCC12)=O C(=O)(CC1=CSC2=NCCN12)NC1C(C)(C)CN(C(c2ccc(Cl)cn2)=O)CC1 c1(C(CNC(CSSC)=O)NC(C2(OC(C)=O)CC2)=O)ccccc1 c1(N(CC(C)C#N)C)ccc(S(=O)(=O)NCC(c2ccc(Cl)cc2)(C)C)cc1F N1(CCCNC(C(=O)NCC(CC)(C)C)=O)C(=O)NC2(CCCC2)C1=O N1(C(CCOCCOC)=O)CCC2(CC1)OCCC2NC(C1CCS1(=O)=O)=O C1(CNC(c2c(C(C)C)cco2)=O)CCN(C(=O)CN2CCCC2C)CC1O C1(CCC)CC(C(=O)NCCN(C(=O)CO)CCC)CCO1.c1ccccc1C N1(C(CC(C=C)(C)O)=O)CCC2(C(=O)NCc3ccnc(OC)n3)CCCCC12 n1(CC)nc2c(c1C(N1CC(C)C1)=O)CCCC2.C1(C)(C=O)CC2C=CC1C2 c1(OC)ccc2c(c1)C(c1nc(C3CCCO3)nn1-c1ccncc1)CCC2 C1(N(C(=O)C(C)NC(=O)OC)CCC)CCN(C(=O)CCC2CCCN2C)C1 c1(OC)cccnc1CN=C(NCC(c1ccccc1)N(C)C)NC1CCCC1 C(C#CC(=O)N1CCCC1CN(C)C(c1cn(C)nc1OC)=O)(OCC)O N1(C(COCC)=O)CC2(C(=O)N(c3cccc(C)c3C)C)CC1CO2 c1(C(=O)OCC)cc(C)sc1NC(=O)C(N1CCC(c2cc(C)no2)C1)=O C1(Br)(C(=O)NCCC(C)NC(c2cnc(C(C)(C)C)[nH]2)=O)CC1(F)F c1(C(N(CCC(C)NC(=O)C=C2CCN(C)CC2)C)=O)cncc2c1CCC2 C#CCCCCC(=O)NN1CCCC1C(=O)NC(CC=C)C1CC1 Cc1nc(C)n(CCCNC(=O)CC(C)(C)NC(=O)CC2CC(=O)C2)n1 c1(C(=O)NCCN(C(c2nocc2C(C)(C)C)=O)CC)cc(C)ccc1F C=C(C)CC(C(=O)NC1CCC1NC)NC(C1(C)CN(C(=O)OC)C1)=O N1(C(c2c(N)non2)=O)CCC2CCCC12C(=O)NCCCOC(=N)O C1(C(N2CCCC(NC(C)=O)C2)=O)CC2(CCC2)C1.C(=O)(C(O)CC(N)=O)N n1(CC(C)NC(C2COC(=O)C2)=O)cc(-c2cccnc2)nn1 Cc1cccc(CNC(=O)C(C2CCN(C(=O)C(O)C(C)C)C2)F)n1 CC1CC(NC(C2(CNC(=O)Cn3cncn3)CCC2)=O)CCN1C C1(C(=O)NC(C(=O)NCC(F)F)c2ccoc2)(OC(C)C)CCC1 N1(C(c2cc(OC)ncc2)=O)CC2CC1CN2C(C1(CCF)CCOCC1)=O C(C)(CO)(CCF)NC(c1c(CNC(Cc2c(C)nsc2)=O)ccs1)=O N1(C(CC2C(NC(c3c(CC)cns3)=O)CCCC2)=O)CC(C)(C)OCC1C C#Cc1cccc(C(N2CCCC(F)(CNC(=O)CCCC(N)=O)C2)=O)c1Cl O=C1NC2(CCCC2)C(=O)N1CN1CCC(n2cc(Cl)cn2)C1 C(C(C(=O)NC1CN(C(=O)CC(C)n2ccnc2)CC1C)C(C)(C)C)OCC=C C1(CN(C)C(c2nonc2N)=O)CCCCN1C(=O)CNC=O C(=O)(CC(C)(C)CNC(c1n[nH]c(C)c1Cl)=O)NC(CN(CCC)C)(C)C c1(CC2(NCC(C(C)C)N)CCOC2)ccc(C(F)(F)F)cc1 Cn1cccc(C(N2CC(O)CCC2C(=O)NC2CC(CCF)C2)=O)c1=O Cc1nn(C)c(C)c1S(=O)(=O)NC(C1CC2CC2C1)C(=O)O c1(C(=O)NC(C)C(C)NC(C2CC(O)C2)=O)cccnc1N1CCCCC1 CCC(C)(O)CCNC(=O)CC1(N(C(=O)CCCC2CCC2)C)CC1 C(COC)(CC(=O)NCC1CSCCO1)NC(C1(COC)CC(=C)C1)=O Cc1[nH]nc2ccc(NC(=O)CC3CN(Cc4cnc5ccccc5c4)C3)cc12 N1(C(c2c(C)nc(Br)s2)=O)CCCC2CCN(C(=O)CCP(C)(C)=O)CC12 C1(NC(c2nccc(OC)c2)=O)CCN(CC23CC4CC2C3C4)CC1C S(=O)(=O)(CC(=O)NC1CCCCC1)NC.C1(=CC=O)CCC(C(C)C)CC1 C(C(CC(=O)NCCNC(c1cnn(C2CCOCC2)c1)=O)C(F)F)N(C)C N1(C(C(Cc2c(C)n[nH]c2C)C)=O)CC(NC(C2(CO)CC2)=O)CC12CCC2 N1(C(CC2CCC2)=O)CC2CC(C1)CN(C(C)=O)C2.N1(C=O)CC(O)CC1.CO N1(C(C)=O)C(C)CN(C(c2nc(C)c(C)cc2Br)C(=O)NC2COC2)CC1C c1(CC)onc(C2CCOCC2)c1C(N1CCCC(CN2CCOCC2)C1)=O C1(CNC(CCOCC)=O)CCN(C(=O)CC2(C(=O)OC)CC2)C1 O=C(CCCCO)NC1CCN(C(c2ncncc2F)=O)C1 c1(C(=O)NC2CCCN(C(c3c(CCC)n[nH]c3)=O)C2)cnc(S(C)(=O)=O)s1 c1(CCN(C)C)cnc2n1CCN(Cc1cc(Br)cc([N+](=O)[O-])c1)C2 c1(C(C(=O)NCC2CC2)N(C)Cc2sccc2Br)ccncc1F c1(CNc2cccc(CNC(=O)Cc3ccc(Cl)cc3)c2)cc(F)cc(F)c1Br Cn1ncc(C(N2CCC(NC(=O)C3=CCCCC3)C(F)C2)=O)c1S(C)(=O)=O c1(OC)ccc(I)cc1C(N1CCC(CN(C)Cc2ccn(C)n2)CC1)=O c1(CCC(=O)OF)ccc(C(=O)NCCC23CCCC2C3)cc1 C1(NC(C2(C)CCCN(C(C(CCC)OCC)=O)C2)=O)CC(C)CC(C)(C)C1 CC(C)(CCCOCC(=O)OCC)C(=O)C1CCOC1.C(C(F)F)N.CC c1(CC)c[nH]cc1C(=O)N(C)CC1(O)CN(C(=O)Cc2cccnc2)C1 c1(C(=O)NC2C(NC(c3c(C)noc3)=O)COC2)ccnc(C2CC2)c1 C(=O)(CCCS(C)(=O)=O)NC(C(C)C)CNC(=O)C=Cc1ccccc1F N1(C(C(CCC)C)=O)CC2CC(C1)N(C(c1ccc(N)c(Cl)c1O)=O)C2 C(=O)(C1c2ccccc2CN1Cc1cn[nH]c1)Nc1c(C(C)O)cccc1 C12(C(=O)NC(c3csc(C)c3)CC)COCC1CN(C(c1ccccc1)=O)C2 N1(C(C(CCO)NC)=O)CCC(CCNC(=O)CCc2ccsc2)CC1C c1(CC)ncnc(CC)c1C(=O)NC(C)CNC(=O)Cc1ccno1.C C(Cc1ccncc1)(C(=O)O)NC1CN(C(=O)OC(C)(C)C)C1 C1(Nc2ncc(C)c(C)n2)CCCC2CN(C(c3cccc(CO)c3)=O)CC12 CC(C)C(F)(F)CC(=O)NC1CC2CCC1C(NC(=O)C#CC(=O)N(C)C)C2 Cc1nc(NCCCOCCNC(=O)CC2CC3(CC3)CO2)cc2nncn12 N1(C(C2(C=C)CCC2)=O)CCC(NC(=O)Cn2ccnn2)C1C(C)(C)C CC1CCN(C(=O)COC2CC(F)(F)C2)CC1NC(c1nccnc1Cl)=O C1(C(=O)NCc2cc(F)cc(F)c2F)CCCC12CCN(C(c1ccoc1)=O)C2 c1(C(=O)NCC(CC(C)C)NC(=O)Cn2ccccc2=O)cc(C#N)n(C)n1 Cc1c(NC(=O)NCCCCCCCO)cccc1-c1ccccc1 c1(C(N(CC(C)C)C)=O)ccnc(N2CCN(C)CC2)c1.C(C=O)=CC=CC c1(C(=O)NCC(CC(C)C)NC(C2CCCC2C)=O)cnc2cc[nH]c2c1 C1(C(=O)NCCCC(C)NC(C2CC2C(C)(F)F)=O)OCCC1(C)C c1(C(N2CC(O)(C(C)NC(C(C)OC)=O)C2)=O)cc(Cl)ccc1C(F)F C1(CC)CN(C(c2cc(C3CC3)no2)=O)CCC1NC(c1nccc(Cl)c1C)=O Cc1cn2cc(NC(=O)C(=O)NCC3(CC4CC4)CC3)ccc2n1 C(CC(C)(C)C(=O)NC(C)C(OC)OC)Cc1cc(COC)ncc1 N1(CC(=O)N(CCOC)CCNC(=O)CC(C)(C)C)CCSC2CCCCC12 c1(C(N(CCCNC(=O)C(CO)c2ccccc2)CC)=O)cc(Cl)ncc1N N(S(=O)(=O)N1CCC(C)C1)c1c(C)n(C(N2CCOCC2)=O)cc1 C1(NC(CC=C(C)C)=O)CCCN(C(C2CC23CCC3)=O)CC1 C1(NC(C2CCC(OC)C2)=O)CCCCC1n1cc(-c2csc(C(=O)O)c2)nn1 c1(C(N2CCCC(CNC(CN(C(C(C)C)=O)C)=O)C2)=O)cccc2ccsc12 C(C(O)C(=O)NC(CNC(=O)C=C1CCCC1)C(C)C)=CCCC C1(CNC(CC=C)=O)CCN(c2nccc(Sc3ccccc3)n2)CCC1(F)F c1(C(=O)OC)ccc(C=CC(N2CCC(C)C2)=O)o1.c1(C(=O)N)cccnn1 CCC(C(=O)NC1CCC(CNC(=O)CCC2CC2(C)C)C1)C(C)C c1(C(=O)NCCN(C(=O)CC(C)(F)F)CCOC)cnc2c(c1)NCC2 C1(CCOC)CCCN(C(=O)C(CC2CCC2)NC(c2coc(C)c2)=O)C1 C1(C(=O)NCCOC(CC)CC)CN(C(C2CCN(C)C(=O)C2)=O)CC1(C)C C1(NC(CSCC(N)=O)=O)CCC2(CC1)CN(C(c1cc(Cl)c[nH]1)=O)C2 c1(C(=O)N)cccnc1.c1(C(N(C(C)C2CC2)C)=O)ccc(C(F)(F)F)o1 C(=O)(C1=COCCC1)NC1CC(C)(CNC(c2cccc(-c3nc[nH]n3)c2)=O)C1 C1(C(=O)NC2C(C(=O)NC(CCCCC)C3CC3)CCCC2)CC12CCCCC2 c1(C(=O)NCC(C)NC(C(CC)(C)C(N)=O)=O)c(C)cc(C)c(Br)c1C CCC(C)CC(=O)NC1CCC(CNC(=O)COCCOCCO)C1 C(=O)(C(C)CC(F)F)N(C1CCCN(C(CCCN(C(C)=O)C)=O)C1)C C(=O)(CN=c1[nH]c2ccccc2s1)NC1(C)CCN(C(CC2CC(CC)C2)=O)C1 C1(C(=O)NCC(CC)N(C(c2c(CC)nn[nH]2)=O)C)CC1C1(C)COC1 c1(CC(=O)NCC(CCOC)NC(CC(=O)NCC)=O)cn(C)nc1Cl Cc1csc(=NCC(=O)N2CCCCC(NC(=O)CCc3cncnc3O)C2)[nH]1 c1(C(=O)NC(CNC(c2c(C(C)C)ncnc2)=O)(C)CO)cnc2n1CCCC2 N(C1CCCc2ccc(F)cc21)C(=O)NC1CC1c1ccc2c(c1)OCO2 c1(C(N2CC3C(NC(CC(COC)C)=O)(C3)C2)=O)c(C)oc2ccccc12 Cc1cccc(C(N2CCCC2C(C)NC(=O)CN2CCCS2(=O)=O)=O)c1C C12(COC)CC(CN1C(c1c[nH]nc1)=O)C2.c1(C=O)ccc(F)c(N)c1.N c1(CC2(C(N(CC(C)CO)C)=O)CCC2)ccccc1 C=CCC(C)(C)CC(=O)NCC1(NC(=O)Cc2n[nH]c(=N)s2)CCCCC1 c1(C(=O)NCCC2(C)OCCO2)cncc(Sc2ccc(Br)cc2)c1 c1(CC)[nH]nc(C(=O)NC(C)CNC(c2ccoc2Br)=O)c1[N+](=O)[O-] N1(C(CC2CCC(NC(C(COC)C)=O)CC2)=O)CCN2CCOCC2C1 C(=O)(C(C)(C)CC(F)(F)F)N1CC(CNC(COCC)=O)C(C)CC1 c1(C(N2CC3N(C(C4CC(=O)NCC4)=O)C(CC3)C2)=O)cnc(O)c2cncn12 c1(C(N2CCC(O)(C(C)CNC(=O)Cc3ccccc3)C2)=O)cnccc1C#N N1(CC)CCC(C(C)C(=O)NC2(C(=O)OC)CC2)CC1 C1(CCC(=O)NCC=C=C)CCCCN(C(=O)C(C)(O)C(C)C)C1 C1(C(=O)N)CNC(=O)CC12CCC2.CCC(C)CNC(C1CC(F)(CO)C1)=O C1(C(N2C(CC)C(NC(=O)Cc3sc(O)nc3O)CC2)=O)CCCCC12CC2 CC1(C)CCC(F)(F)CC1C(N1CC=CC(NC(=O)COCCO)C1)=O C(=O)(CCCC(=O)NC)NC(C1CCCN(C(c2c(CC)nco2)=O)C1)C C1(NC(C=CCC)=O)C2COCC1CN(C(=O)COCc1nc[nH]n1)C2 N1(C(c2ncn(C)c2)=O)CC2CC(NC(c3cc(Br)n(C)n3)=O)C(C2)C1 N1(C(CC(C(F)F)NC(CCCN=[N+]=[N-])=O)=O)CC2(CCC2)CC1CO c1(C(=O)NCC2N(C(CC3N(C)CCOC3)=O)CC2)cccc2c1NC(=O)CC2 c1(OC)n[nH]cc1C(N1CC(O)(CCNC(=O)C(C)C2CCC2)C1)=O c1(N2C(CN(C(=O)CCC3CCCO3)C)CCC2)nccc(C#N)n1 N1(C(CN(C(c2n(CC#C)ccc2)=O)C(C)C)=O)CC(C(=O)O)C(CO)C1 N1(C(c2c(C)cnnc2)=O)CC(C)(C)CC1CNC(=O)CC1CCCOCC1 C1(C(N2CC(=CCC)C2)=O)CC(O)CCN1C(C1CCC(OC)C1)=O C(=O)(C1=CCC2CCC1N2C(=O)C(F)CCC(C)C)N1CCCCC(OC)C1 C(=O)(C(C)C(F)(F)C(F)F)NC1CCN(C(c2cc(CC)ncn2)=O)C1 C(=O)(CCCCCC#N)NC1(CO)CCN(C(C=CC(CC)=CC)=O)C1 CCCCCCCC(=O)NC(C)(C(=O)NC1COCC1N=[N+]=[N-])C1CCC1 N1(C(C2CC(C)C2)=O)CCN(C(c2[nH]nnc2C2CC2)=O)CC(C)C1 Cc1ccc(NC(C2(C)CCCN2C(=O)CC2CCC2)=O)c(S(=O)(=O)O)c1 C(C1CCN(C(C23CCC(O)C2C3)=O)CC1)=CC(=O)Nc1ccc(CC)cc1 C12(C(=O)NC(CC(=O)NC)C3CC3)CCN(C(C3CC=CC3)=O)CCC1C2 c1(OCC=C)ccccc1C(C)NC(c1cc(Br)co1)c1nnnn1CCCF C1(C(=O)NCCC(C)(C)O)CC2(CC2)CN1C(=O)CCCOC(F)F N1(C(CC(C)SC)=O)CCC(O)(CN(C)C(c2occc2C)=O)C1 Cc1[nH]c(C#N)cc1C(=O)N.C1(C(C)C)CCN(C(=O)C(C)(F)c2ccon2)C1 Cc1cnc2n1CCN(C(C1C(NC(c3cnn(C4CC4)c3)=O)C1(C)C)=O)C2 CC1(C)CC(C(N2CC(O)(C(F)(F)F)C2)=O)CCN1C(c1cnn2c1OCC2)=O C(C1c2ccccc2CCN1Cc1cnc(Cl)s1)NC(C1CCS(=O)(=O)C1)=O C1(CC)(NC(C(C(C)C)SC)=O)CCN(C(=O)COCC)CC1.CCO.O C(=O)(CCC(=O)N1CC(c2ocnc2CNC(c2nc(Br)c[nH]2)=O)C1)NC Cc1nsc(C)c1-c1cn(C2CC(NC(=O)C(F)C3CCC3)C2)nn1 Cc1ncc(F)c(NC2CC(CC(=O)Nc3cnncc3Br)C2)n1 c1(C(=O)OCC)c(NC(=O)C=O)sc2c1CCC2.C(Cn1cccn1)CC.N N1(C(c2nnc(CC)s2)=O)CCC(C)C(NC(=O)C(F)(F)C2CC2)C1 c1(C(N2CC3CC4CC3C2C4)=O)ccnc2ccnn12 c1(OC)ccc2sc(-c3nn[nH]n3)c(C)c2c1.n12ncc3ccc(cc13)C2=O N1(C(CNC(CCC)=O)=O)CC2CCCC1CN(C(c1ccnc(O)c1F)=O)C2 C1(NC(CC2CC(C)N(C(=O)CCc3cscn3)C2)=O)CCCCCCC1 c1(OC)ccccc1-c1oncc1C(N1CCCC1)=O.C1(=CC(=O)N)CCCC1 N(C(=NCCc1ccn(C(C)C)n1)N1CCC(C(F)F)CC1)CC(CC)C(C)C C(CCO)(C(=O)N1CCN(C2CCN(C(C3CCC(=O)N3)=O)C2)CC1)N(C)C C(C(=O)OCC1C2CCOCC12)(C(C)CC)C1CC(C(=O)OCC)C1 c1(C(N2CC(CC=C)C2)=O)ccccc1.C1(C)(C=O)CC1F.CCN(C)C.N c1(OC)ncnc(C(=O)N(CC(C)N(C)C(C2C3CCCCC23)=O)C)c1F N1(C(C2C(C)C2)=O)CC(C2CCN(C(C3CC(F)(CO)C3)=O)CC2)C1 C1(COC)CN(C(=O)C(C)(O)CC)CCN1C(=O)CCC(C)C c1(CCC)c(C(=O)NCC(C2CC2)NC(=O)Cc2ncoc2C)cnn1C C1(NC(C(CC#C)C2CC2)=O)COCCN(C(=O)COc2cc(C)on2)C1 c1(CC)cc(-c2ccc(C(C)CO)cc2F)c(C)cc1F C(=O)(C(C)(C)CC(=O)OC)NCC=C(C(=O)NCC(N(OC)C)=O)C CC(C)C(CC(=O)NCC1CC(C)(O)C1)NC(C1(O)CCOC1(C)C)=O C=CC(C)CC(=O)N(C(C)CNC(=O)C=Cc1csnc1C)CC C(=O)(C1=CC2C=CC(C1)C2)N1CC(OCCC(=O)N)C1.C1CC2(COCCO2)C1 N1CCC(C(=O)NCC2(N(C)C)CCOC2)CC1.N1(CC(=O)N)CCCOC1=O N1(C(C(CC)NC(N)=O)=O)CC2CC(C(=O)NCCC(F)(F)F)CC2C1 c1(CC(C(=O)OC(C)(C)C)NC(C)CC2CC2)ccc2ccccc2c1 N1(C(CN(C)CC)=O)CCCC(F)(CNC(=O)CC)C1.c1cc(F)ccc1F.S C1(CC=C)(N(C(C2CCCS2)=O)CC)CCN(C(=O)Cc2ccc(Cl)cc2)CC1 C(C(C)NC(=O)CCc1nc[nH]n1)(C(C)C)NC(CCCc1onc(C)n1)=O C12(CC(N3CCC3)=O)CNC(=O)C(C1)C2.Cn1nnnc1N1CC(C=O)C1.N C(C1CCN(C(c2ccc(O)cc2F)=O)CC1)=CC(=O)N(C1CCCCC1(C)O)C C1(C=O)CC(=O)CC(=O)C1.C(=O)(C(C)CC1CC1)N(C)Cc1nncn1C c1(C(N2C3CN(C(c4cncc(Cl)c4)=O)C(CC3)C2)=O)cn2cc[nH]c(=O)c2n1 C1(C(N(C(CNC(c2c(C)oc(CO)c2)=O)C)C)=O)CCC2CCCCC2C1 C(CC1=CCCCC1)NC(CC1OCCN(C(C(C)SCC)=O)C1)=O c1(C2C(C(N)C(N3CCC(CC(N)=O)C3)=O)C2)c(F)cccc1F N1(C(c2cn(Cc3cccc(OC)c3)nn2)=O)CCCCC1(CO)CO N1(C(C(n2ncc(C)c2)C)=O)CC(NC(=O)CN2CCC(=O)CC2)C(C)C1 N1(C(c2n[nH]c(C)c2Cl)=O)CCC(CCNC(C2(C(F)F)CC2)=O)C(F)(F)C1 CCCC(CC)CCC(=O)NCC(C)(CO)NC(c1cn(CCC)nn1)=O C(c1cccnc1)=CC(=O)N(C(C)C(=O)NOC(c1ccccn1)C)CC N1(C(C(C2CCCC2)OC)=O)CCN(C(c2cnc(Cl)[nH]2)=O)C2COCC12 N1(C(CC(CC)CC)=O)CC2C3CCC(C2C1)N(C(c1cc(O)nc(O)n1)=O)C3 N(S(=O)(=O)NCC1CC(F)(F)C1)(CCC)CC O=C(CCCCc1ccc(F)cc1)NCCc1nnc(-c2ccco2)o1 CC1C(=O)N(C)CCN1C(C1CCCN1c1cc(N(C)C)ncn1)=O N1(C(Cc2ccc(SC)cc2)=O)CC(C2CN(C(C3CC3C3CCC3)=O)C2)C1 CCC(CC(F)(F)F)C(=O)NC1CN(C(=O)Cc2cc(COC)on2)CC1(C)C CC1CC=C(C(=O)NC(C)CCNC(c2ccc(F)cc2F)=O)CC1 C1(CCC=C)(C(=O)NC(C)(C=C)CC)CN(C(C2CC2c2cncn2C)=O)C1 c1(C(=O)NC2CCCN(C(=O)COCCCF)C2)occ2c1CCOC2 CCC(CC)CCCC(=O)N1CC(C(=O)NCc2cccnc2O)C(C=CC)C1 CC1(C)CCCCC1(C)NC(C1CCC(NC(=O)CCCn2ccnn2)CC1)=O C(=O)(C(C)S(N)(=O)=O)NC1C2CN(C(COCC#C)=O)C1C2 c1(C(N2C(CNC(CN(C)C)=O)CC2)=O)ncccc1O n1(CCC)cc(C(=O)NC2CC(C(=O)NC(CN(C)C)C(C)C)C2)cn1 N1(C(CCC2CC(OC)C2)=O)CC(O)CC1CC(=O)NCCC1(C)CC1 N1(C(c2nn(C)c(Cl)c2)=O)CC(F)(F)CC1(C)C.C1(CC(=O)N)CC2(CC2)C1 N1(C(CC(C)OC)=O)CC(C)(C)CCC1CNC(=O)C(F)=C(C)C1CC1 CC1CN(C(=O)C(F)n2ccnc2)CCC1NC(=O)COc1ccc(F)cc1F C1(C(=O)NCC(CC)(O)CC)CCN(C(=O)C=Cc2ccc(C)o2)C12CCC2 C1CN(C(c2c(N)ccc(F)c2F)=O)CC(C)(C)O1.C1(COC)CC1C=O.N c1(NC(C2CCC(C)N(C(=O)OC(C)(C)C)C2)=O)ccc(Br)cc1C=O N1(C(C2C3CN(C)CC32)=O)CC(F)(F)CC1C(=O)NCCC1CCCC12CC2 N1(C(C2=CCC(C)CC2)=O)CCCCC2(CCN(C(c3ccncc3O)=O)C2)C1 C(=O)(C1Cc2c(Cl)cccc21)N1CC(O)C1.c1(CC(=O)NC)cc(F)cc(F)c1 CCC(F)(C(=O)OC)C(=O)NCC#CCNC(c1ccc(-c2ccccc2)[nH]1)=O c1(CC(=O)N)cc(O)nc(O)n1.C(C(O)CC)NC(C(C1CCOCC1)OC)=O CCC(C(=O)N(C)CC1CCCN1C(C1C2COCC12)=O)OC CC(C)CC(=O)C(=O)NCC12CC(CO1)N(C(C1CCS1(=O)=O)=O)C2 c1(C(=O)NC2CN(C(c3[nH]c(=NC)sc3)=O)C(C)CC2)ccc(F)c2[nH]ccc12 C1(CNC(C(C)OCCC=C)=O)CC(O)CN1C(c1cc(OC)n[nH]1)=O c1(N2CC(CC#N)N(C(c3cc(F)c(Cl)nc3Cl)=O)CC2)ncnc2cc[nH]c12 Cc1ncnc(NC2CCC(N(C(=O)C=Cc3cccc(CO)c3)C)CC2)c1F c1(C(c2n(CCCSC)nnn2)NC2CC2F)cccc(C)c1C Cc1ccc(C(=O)NCC2CN(C(=O)CN3C(C)CCC3C)CC2C)c(Cl)c1Cl c1(CNC(C(C)OC)=O)ccc(C)c(F)c1.C(c1cc[nH]n1)=CC(=O)N N1(C(C2(C#C)CCCC2)=O)CCC(C(=O)NCC2(F)CCC2)CC1(C)C N1(C(C(C)OCC=C)=O)CC=C(CNC(=O)CN2CCN(C)CC2)CC1 C1C2CC1N(C(=O)C(O)CCN(C)C)C2.n1(C(C)C=O)ccc(C(F)(F)F)n1.N C1(C(=O)NC2(CNC(CC=CC=C)=O)CC2)C2CCC1(c1cccs1)C2 N1(C(c2cc(CC(C)C)on2)=O)CC2CCOCC2(NC(=O)C=CCO)C1 N1(C(C(C(CC)C)N)=O)CCC2(CCC2NC(=O)CSc2ccncc2)CC1 c1(NC(c2cc(C)oc2)=O)cncc(C2CC2)c1 CCC(CCC(=O)N1CC2CCC2(CC(=O)NC(C)CCC(F)(F)F)C1)OC c1(C(=O)NC(C2(O)CN(C(C3(CC)CCOC3)=O)C2)C)cc(Cl)ccn1 Cc1cnc(NC2CC2C(=O)N(C)Cc2ccncn2)nc1-c1ccccc1F c1(C(=O)NCCNC(Cc2[nH]c(=N)sc2)=O)cccnc1Oc1cccnc1 N1(C(CCCN(C(=O)OC)C)=O)CCC(NC(c2cccc(Cl)c2)=O)C(O)C1 C1(C(=O)NCCCCNC(C2CCN(C(C)=O)C2)=O)CCS(=O)(=O)C1 C1(C2CCCN(C(=O)C(C)C3CC3)C2)(NC(c2ccc(OC)c(F)c2F)=O)CC1 c1(CNCC(CN(C)C)(C)C)cccc(Cl)c1N1CCOCC1 C(=O)(C(O)CC(F)(F)F)N.Cc1nn(C)c(C)c1CCC(=O)NC1CC(C)C1 C1(C(=O)NC(CC)CNC(=O)C(C)c2ccsc2)(NC(C)=O)CCOCC1 C1(NC(C(C)(C)OCC)=O)CN(C(c2cncc(C)c2)=O)CC1.C1CC1.C N1(C(CC(CC)C)=O)CCCC2(C1)CN(C(=O)Nc1ccc([N+](=O)[O-])c(C)c1)C2 Cc1cc(C(N2CCCCC2CNC(C2CCC2c2nc[nH]n2)=O)=O)cc(N)c1 C1(CC#C)(C(=O)NCCCc2cccnc2)CCN(C(=O)CCC(C)N(C)C)C1 C1(O)(C(N(CC(C)CNC(C2CCOCC2)=O)C)=O)CN2CCC1CC2 C(=O)(C1CCc2c[nH]nc21)Nc1cccc(CNC(CC(C)n2cccn2)=O)c1 CCC(CC)CCO.C1(C(=O)N)(C=O)CCN(C=O)C1.C(C)(C)C.C(C)(C)C c1(C(=O)NCC(C)NC(c2csc(C(F)F)c2)=O)ccccc1C(F)F c1(OCCCC)ccc(NC(=O)C(N2CCC(C)(CO)C2)=O)cn1 CCC(CCOC)C(=O)N1CC2CC1C2NC(C1CCCN1C=O)=O c1(CC)c(C(=O)NCc2ccoc2C(=O)NCCn2ncnn2)nnn1C N1(C(C2CC=C(C)CC2)=O)CCN2CCN(C(=O)CCc3csc(C)n3)CC2C1 C(CCCC(=O)NC1CC(NC(c2ccsc2Br)=O)C(O)C1)N(C)C c1(C(N2C(CCNC(C(C(CC)O)C)=O)CCC2)=O)cc(C#N)c2n1CCCC2 c1(C(=O)NCCC2(OC)CN(C(=O)C(C)C)C2)c[nH]c2cc(F)ccc12 CCC(COC)C(=O)NCCCC1CN(C(=O)C(C)(C)c2cncnc2)CCO1 c1(C2CN(C(C(C3CCC(OC)CC3)F)=O)C2)cc(O)cc(Br)c1 N1(C(C2(NC(C(C)NC(CC)=O)=O)CCCCC2)=O)CC2CC1CN2C N1(C(C(COC)(C)C)=O)CCC(C2CN(C(=O)C(C)Cc3cccc(F)c3)C2)C1 c1(C(=O)N)cc(F)c(F)c(N)c1Cl.Cn1cccc1C(=O)NC(C1CCCC1)C C(=O)(C(F)C(F)(F)F)NC(COCC)C.c12sccc1C(=O)N2 C1(CNc2cccc(OC(C(=O)NC)C)c2)(CO)CC2CCC1CC2 N1(C(C(C)OCCCC)=O)CC2CCCC(C1)N2C(c1ccc2[nH]ccc2c1)=O c1(CC)n[nH]cc1C(c1nnnn1Cc1nnn(C)n1)NCC(C)(C)F CC1(C)CC2(CCC2)C1.C1(CC=O)COCCN1C(=O)CC1CCCC(=O)C1.N Cc1[nH]nc(C(F)F)c1C(N1CC2CC1(C)C2)=O.C1(CC(=O)N)CCNC1=O C1(C(=O)NC(C(=O)N(C(CC)C2CC2)C)CN(C)C)CCOC(C)(C)C1 c1(Cn2ncc(NC(C(COC(C)C)N)=O)c2)ccc(Cl)cc1 c1(C(=O)NCC(CNC(=O)C(O)C(C)C)OC)cc(=O)c2ccccc2n1C n1(CC)cncc1CC1C=CC(C(=O)NCCN2CCOCC2)C1 N#CC1C2CC2CN1C(C1CCCC1NCc1cccc(-c2cncnc2)c1)=O C1(OC)OCCCC1NC(=O)C(N1CCC(O)(c2cc[nH]n2)C1)=O c1(OCC)cccc(-c2nc(CNC(c3nn(CCF)cc3I)=O)cs2)c1 C1(NC(C(=O)Nc2n(CC)ncc2)=O)CCN(c2cccc(Br)c2)C1=O N1(CCc2cn(CC(COC)O)nn2)CCN(C(=O)C(C)C(=O)O)CC1 C(=O)(C1=C(C)CC1)NCC1(CNC(C(C)SCC)=O)CC1(F)F C1(C(=O)OC)CC(O)CN1C(c1cncc(Br)c1)C(=O)NCc1ccccc1Br S(=O)(=O)(c1cccnc1)NCCC(N1CC2CCCC1C2)=O.C(=O)C.C1CC1.N c1(C(N2CC(NC(CN(C(C)C)C)=O)C(F)CC2)=O)ccc(S(C)(=O)=O)o1 N1(C(=O)CCn2c(=O)oc3ccccc23)CCCC2(CC1)CNC(=O)C2 c1(CC=O)ccc(C=O)o1.C(=O)(CC)N(CCC)CCO.C(C)(C)C.CO C=CCC(CC=C)NC(=O)C(C1(C)CC1)NC(c1ccc(O)cc1)=O N1(C(C2CC(OC)(O)C2)=O)CCC(C)(C)CC1.C1(CC=O)C(=O)ON=C1C c1(C(=O)NC2C(NC(c3cccc(CC)c3)=O)CC2)c(N)ccc(F)c1F c1(C(=O)NC2C(NC(c3cccc(OC)c3)=O)CCC2)cc(C)c(F)cn1 c1(-c2cnc(NC(C(CO)NC(=O)OC(C)(C)C)=O)s2)cccc(Br)c1 N1(C(C(n2cc(NC(CCC)=O)nn2)C)=O)CCCC(CCO)CC1 C(CC(=O)NNC(=O)C(=O)O)C(c1ncnn1-c1cnc(-c2ccccc2)nc1)=O CC(C)CC(C)C(=O)NCCCC(=O)NC1CCC1(C)C c1(C(=O)NCC2(C)CCCCC2)cc(S(C)(=O)=O)cs1.C1(C=O)CC(O)C1 C12(NC(C(C(C)C)O)=O)CCCC1N(C(=O)CC13CCC(CC1)OC3)CCC2 C(=O)(CC(Cc1ccccc1)C(F)F)NC(C)CNC(=O)C=C(Cl)Cl N1(C(c2c(C)n(C)nc2)=O)CCC2(CC1)COC(C)C2NC(=O)C1=COCC1 N1(C(C2C(CC(C)(C)C)C2)=O)CCC(C)CC1.c1(C=O)cccc(C2CC2)c1 CC(Cc1ccco1)C(=O)NCC(C)(C)CNC(=O)CSC(F)(F)F Cc1cc(F)sc1C(=O)NCC1CC1.c1(C=O)ccncc1.C(=O)(CC)N CS(C)(=O)=NC(=O)C(=O)NCCNC(=O)CCC1CCCC(O)C1 C1(C)(CNC(c2c(CCC)n(CC)nn2)=O)CCCN(C(=O)CC(C)F)C1 C1(CC=O)NC(=O)NC1=O.C(=O)(CCC1CC1)NCC(C)(O)C1CC1.N C(=O)(C(C)(C)CN(C)C)NC(c1cnn(C)c1)C(=O)N(CC#CC)C c1(C(=O)NCC2CCC(C(=O)NC(C)CCO)CC2)cc(O)c(O)c(Cl)c1 CCC(C)CC(C(=O)NCCC1CC1)NC(=O)CC=C(C)C CC1CCn2c(C(=O)NCCCN(CCCNC(C3CC34CC4)=O)C)cnc2C1 c1(C(=O)NC(CCNC(C(CC=C)C)=O)(CC)CC)ccc2nc[nH]c2c1F C1(NC(c2ccno2)=O)CCCN(Cc2ccc(-c3ccccc3)s2)C1 Cc1noc(Cl)c1CC(=O)NC(C1CCCN(C(=O)CCc2nccs2)C1)C C1(C(=O)NC(C(=O)Nc2c(C)nn(C)c2)C)CC2(CC2)CN1C C1(CNC(c2cccc(F)c2)=O)CCC2CN(C(c3cc(O)ncn3)=O)CC12 c1(C(N2CC3CN(Cc4c(C#C)cccc4)C3C2)=O)c(Cl)ccc2c1OCO2 c1(OC)ccnc(C(N2CCC(C)(NC(C3CC34CC4)=O)C2)=O)c1N c1(CN2C(C(=O)NC(C(C)(C)C)CO)CC3CC32)cc([N+](=O)[O-])ccc1O N1(C(c2c(CCC=C)cccc2)=O)CCC(c2ccccc2)OC(C)C1 c1(C(=O)NC2C3N(C(C(c4ccccc4)C)=O)C(CC3)C2)c(F)ccc(O)c1F C(C(C)(O)CC(=O)N1CCCC1)OC.C1(C2CC2)(C(N(C2CC2)C)=O)CC1 N1(C(C(OC)OC)=O)CC2(CCCC2)C1C(=O)NC(c1nncs1)C c1(N2CC(C(C)NC(c3n(C(CC)C)ncc3)=O)OCC2)ccccc1[N+](=O)[O-] C1(CC(=O)N(C(CNC(CC(CC)SC)=O)C)C)CCCC2(CCC2)O1 C1(CC(N2CCCC(CC=C(C)C)C2)C(=O)NC(C)C)COC(C)(C)O1 C12(C(=O)NCCOCCC=O)CCC(CC1=O)C2.C1CCC(C(N)=O)C1.N C1(c2n(-c3cccc(OC)c3C)nnn2)(NCC2CCC2)CC(C)N(C)C(C)C1 C1(C(N(C)CC2CCN(C(=O)CCCCCF)CC2)=O)CCC(=O)N2CCCC12 n1(CCCC(=O)NC)ccc(=NC(=O)C2CC2c2cc(C)[nH]n2)[nH]1 CCC(C)CC(C)C(=O)N1CC2(CNC(=O)CN3C(=O)CCC3=O)CCC1CC2 Cc1ccccc1C(=O)NCC(CC1CCCC1)C(=O)N1CC2C=CC2C1 N1(Cc2ccc(OC)cn2)CC2CC(C1)N2C(=O)CCc1ccc(C)cc1 C1(C(=O)NCC2(NC(c3n(CC=C)ccc3)=O)CC2)CCCC(C)O1 N1(C(COC(CC)CC)=O)CCC2(CCCN2C(=O)Cc2ccsc2Cl)CC1 C1(CC(=O)N(C)Cc2ccsc2)CCCN(C(=O)Cc2ccon2)CC1 CN1CC(C)(C(=O)NC2CCCC2NC(C2(O)CN3CCC2CC3)=O)CCC1=O Cc1csc(C(N2CCC(C(C)(C)NC(C3(C)CC(C)C3)=O)C2)=O)c1C C(=O)(C(C(C)C)c1cc(C)no1)NC(C(=O)NCC)CC Cc1ccc(C(N2CCC(C)(CNC(C3CCS(=O)(=O)C3)=O)C2)=O)cc1O c1(C(N2CC(NC(C=CC=CC)=O)C(SC)C2)=O)cc2c(s1)CCOC2 c1(C(N2C(CNC(C3CCC(C(N)=O)O3)=O)CC2)=O)cnc2ncccn12 C(=O)(C(CCN(C)C)NC(C1CC1C(F)F)=O)N(CCCC#C)C c1(C(c2cnco2)NCC2C(C)(C)C2)nnnn1CC(F)F N1(C(C2CC2F)=O)CC(CNC(C2(O)CCSCC2)=O)CC12CCC2 c1(C(C)NCC(=O)NC(c2c(C)cccc2)C(C)C)ccc(Cl)c([N+](=O)[O-])c1 c1(C(=O)NCc2c(C(=O)NC3CCC(C#C)C3)n(C)nn2)cnccc1C#N CCC(O)CC(=O)NC1C=CC(C(=O)NCCCn2cnnc2C)C1 CC(C)(CO)C(=O)NC1COCC1NC(=O)C(C)(C)c1cccs1 C(CN=c1[nH]c(=NCCC2CCSC2)[nH]c2c1CCCCC2)(C(C)(C)C)OC N1(C(C2C(C(C)C)N(C(=O)COC3CC=CC3)CC2)=O)CCC2C(=O)NCC2C1 CON(CCC(=O)NCCCCC1CCCC1)C(=O)C1CC=CC(O)C1 c1(CNC(=O)NC(C)CC(N)=O)ccnc(Oc2ccccc2)c1 c1(OC)ccncc1CC(N1CCC(OCCNC(c2cccnn2)=O)C1)=O N1(C(c2c(CC(C)C)nc(C)s2)=O)CC2CCN(C(=O)C(F)=CCCF)CC2C1 N1(C(C2N(C(C)=O)CCC2)=O)CC2CCCC(Nc3cc(=O)n(C)c(O)n3)C2C1 C(=O)(CCCC(C)(C)C#N)NC1(C)CN(C(CC2CCN(OOCC)CC2)=O)C1 c1(C(N2C(C(=O)O)CC(F)C2)=O)cccc2ncnn12 c1(CNC(Cc2c(CC)con2)=O)cncc(C(N2CCC2C2CCCC2)=O)c1 C1(C(=O)NCC(CN(C(CCSCC)=O)C)O)CN2CCN1CC2C N1(C(C2(C=C)CCC2)=O)CC2(CCN(C(C3CC4CCC3C4)=O)CC2)C1 c1(C(=O)NC2C(NC(=O)CC3CCCC3(F)F)C2)cc2ccccc2[nH]1 C1(CC(=O)NCC(C)(C2CC2)NC(C(C)CCO)=O)Cc2ccccc2N1 c1(COC)ccccc1CC(=O)NCC1CCN1C(c1oc(CO)cc1C)=O Cc1cc(CNC(=O)CC2(NC(=O)C(C3CCCCC3)O)CCC2)ccn1 Cn1nc(C(N2CCC(C3OCC3(F)F)CC2)=O)c2c1CCCC2 C1(C(=O)NCCC(Cn2cc(CC(C)(C)O)nn2)F)CCCCC1(F)F c1(CCC(=O)NCCCCC(C)NC(CC(C=C)C)=O)c[nH]c2cc(Cl)ccc12 C(=O)(CC(C(F)F)n1cccn1)NCc1c(C(C)C)ocn1 C1(C(N)=O)CCN(C(=O)Cc2cscn2)CC1F.C1(C=O)CCSCC1 c1(C(=O)NC2C3(CN(C(C(C)(O)C4CC4)=O)C3)CCC2)cnc2sccn2c1=O c1(CC)ncsc1C(=O)NCCN(C)C(C1CCC(C(N)=O)O1)=O C1(NC(C(C)(C)OCC)=O)CCN(c2cc(SC)nc(SC)n2)CC1C c1(CN2C(c3nc(C)on3)CCC2)cc2c(s1)CCCCC2 Cn1cc(Cl)cc1C(=O)NCC1CCN1C(=O)C=Cc1cncs1 c1(C(C)NS(=O)(=O)CCOCC2CCOC2)cccc(C(F)(F)F)c1O N1(C(CS(=O)(=O)NC)=O)CCCC(F)(F)CC1.C1(C=O)CCCN1C(C)=O.C C(=O)(C1=CCC(NC(c2cnn(C)n2)=O)C1)NCC(c1ccccn1)C c1(C(N2C(CCNC(C3ON=C(CC)C3)=O)CCCC2)=O)ccc(C)c(CO)c1 N1(C(C(C(=O)OCC)CC)=O)CCC=C(C(=O)N2CCC(C)(C)C2C)C1 C(CC(C)C)(C(=O)NC(CCF)C(=O)NCc1nc(C2CC2)n[nH]1)OC c1(CC)ncc2c(n1)CN(C(C1(C)CCN(C(=O)OC(C)(C)C)C1)=O)C2 N1(C(c2ccn3ccnc3n2)=O)CCC2(C=Cc3ccccc3O2)C1 CCC(CC(=O)NCC(CNC(c1cnc[nH]1)=O)OC)c1ccccc1 C1(CNC(c2ccccc2)CN2C(=O)NCC2)CCCOC1c1ccccc1 C1(O)(CNC(c2ccn(C3CCOCC3)n2)=O)CCCN(C(=O)CNC=O)CC1 C(=O)(CC=C(Cl)Cl)N1C(CCNC(=O)CC(F)F)CCC1 CC1(C)NC(=O)N(CC(=O)NC23CCN(C(C4SCCCS4)=O)CCC2C3)C1=O C(CC)(CCC(=O)N(C)CCc1ccccc1)NC(C(C)(C)OCC)=O N#Cc1cc2c(nc1N1CCN(CCNC(C3CCCS3)=O)CC1)CCC2 C(=O)(CS(=O)CCC(F)(F)F)OCc1c(C)cnn1CC1CC1 c1(C(=O)N)c[nH]nc1.C1(C(=O)OC)(C(=O)NCCCC)CC1C.C1CCCC1 C1(C2CC2)(NC(c2c(C)nc(-c3ncccn3)s2)=O)CCN(C(C2(F)CC2)=O)C1 c1(C(N2CC3(CC(CC(N4CC(O)C(F)C4)=O)C3)C2)=O)cc(Br)ccc1I C1CN(C(=O)C=CCN(C)C)CC(C)(C)O1.c1(OC)cccc(C=O)c1F.N c1(CC=O)cc2ccccc2o1.C(C)C(C)C.C(CC(=O)N)OCCOCC Cc1cc(C(=O)NCC2CCN(C(c3ccc(F)o3)=O)CC2)oc1Br C1(C(=O)NC2(CO)CC(F)(F)C2)COCCN1C(C12CSCC1C2)=O C(=O)(C(C(C)(C)C)c1cc[nH]n1)NCC(=C)CCNC(c1cnccn1)=O C1(NC(C2C(OCC)C2)=O)CCC2(CC1)CC2NC(=O)C(O)C(C)C c1(N(C2CCN(CCC)C2)C)cc(NC(C2CC2)C2CC2)ncn1 C1(CC)CN(C(c2cnn(CC)c2Cl)=O)CCN1Cc1ccc(C(C)C)c(Cl)c1 C(=O)(CCC(C)(C)O)N(CC(CN(C(c1c(C(=O)OC)cncc1)=O)C)O)C C1(C=O)CC12CCOCC2.C1(NC(Cn2cc(C(=O)NC)nn2)=O)COCCC1.N c1(C(=O)NC2CCC(NCc3ccc(Br)cc3CO)C2)cc(Br)cc2cc[nH]c12 c1(N(CCC)C)nc(=NCC2CCOCC23CCCC3)[nH]c2c1COC2 c1(C(N2CC(C(C(=O)NCC3(C#C)CCC3)O)C2)=O)ccnc(O)c1F C#Cc1cccc(C(=O)NCC2(CC)CC2)c1C.C(c1ccsc1)=CC=O.N C1(N(CCC)C=C(C)C2CC2)CCN(C(=O)CC2CCN(CC(C)C)C2)CC1 N1(C(C2(C#C)CCC2)=O)CCC(CO)(NC(=O)CCC=C)CC1 Cc1nn(C)c(Cl)c1-c1cn(CC2CN(C(CCC(O)CCO)=O)C2)nn1 CN=c1[nH]c(C(=O)NCC2(O)CCN(C(=O)Cc3ncc(C)s3)C2)cs1 CC(CO)(CO)C(=O)N1CC(F)CC1C(=O)Nc1nc(Cl)ccc1O c1(C=O)cc(O)ccc1C(F)(F)F.C(CCC(=O)NC1CCCC1)OCC.C N1(C(CC(=O)NC)=O)CCC(F)C(NC(=O)Cc2sc(S)nc2C)C1 c1(C(C)C)cccc(CNC(C2(n3ccnc3)COC2)=O)c1 c1(CC)cccc(C(=O)NCC2(C(N3CCC(C)(C=O)C3)=O)CC2)n1.N N1(C(C2C(CNC(c3ncc(C)cc3F)=O)CC2)=O)CC2COCC(C2)C1 C1(C(N(C(CC(=O)NC2C(C(C)C)CCCC2)C)C)=O)CCC(C)(C)CC1 Cc1noc(CN(C)C(C2CCC(CNC(C3CCCOC3)=O)C2)=O)n1 c1(C(C)OC)cn(C(C)CNC(C2CCS2(=O)=O)=O)nn1 C(c1cccc(F)c1F)=CC(=O)NC1CC(NC(c2c(C)cnnc2)=O)C1 C#CCC(O)C(=O)Nc1cccc(CNC(c2ccc(C(C)C)o2)=O)c1 C1(O)(CNC(c2csnn2)=O)CN(C(c2cn(CC3CCCO3)nn2)=O)C1 C(=O)(CS(=O)(=O)CCO)NC1CCN(C(C2CCN(S(C)(=O)=O)C2)=O)C1 c1(C=O)cc(C(F)(F)F)ccn1.C1(NC(CN(C)C2CC2)=O)CC(F)C1.C N1(S(CC)(=O)=O)CCCC1(C(N1CC2CC2(CO)C1)=O)C(=O)OC C(c1ccc(C)c(C)c1)=CC(N1CC(NC(C(CC)SC)=O)(CF)C1)=O N1(C(c2scc(C)c2)=O)CCCC(CN(C)C(C2CC2C(C)(F)F)=O)C1 N1(C(c2c(C#C)c[nH]n2)=O)CCCC(C)(C)C1CNC(c1[nH]cnc1CC)=O c1(C(COC)NC(C2CCCN2C(=O)Cc2ccccc2Cl)=O)ccc(C)cc1 C1(N(C(=O)CCC2CCC(=O)N2)CCCC)CCN(C(C2CCCCO2)=O)CC1 c1(C(C)=O)cnn(C)c1C(N1CC2C(C)C2C1)=O.C1(O)(C(=O)N)CCCCC1 c1(C(=O)NCC2CN(C(C(C=C)CC)=O)C(C)C2)cccc2c1CCC2=O CC(C(=O)NCC(C)CO)S(C)(=O)=O.c1(C(=O)N)cnc(C2(C)OCCO2)s1 C1(NC(C(c2ccccc2F)(C)C)=O)CC2CC1N(C(C1CCOCC1)=O)C2 CC1(CNC(c2cc(C(N)=O)no2)=O)CCN(Cc2ccc(Br)c(F)c2)CC1 c1(C(C(=O)NC(c2cn(CC)nn2)C)(C)O)ccc(F)cc1.C1(SC)CC1 C(=O)(C(CCCC=C)NC(=O)C(C)C(=O)OC)N1CCC(C#C)(O)C1 c1(C(N(C)Cc2cc(F)ccc2Cl)=O)ccc(S(C)(=O)=O)cc1Cl C(c1cccc(CO)c1)=CC(N1CC(C)C(NC(C2(C)CC2C)=O)C1)=O c1(C(=O)NC2C(NC(c3cc(Cl)c(Cl)s3)=O)C2)cc2ncccc2s1 C1(C=O)Cc2ccncc2C1.C1(CNC(C2(CN(C)C)CC2)=O)CCCC1.N N1(C(CC=O)=O)CCCC(N(C(=O)C(c2ccc(F)cc2)C2CC2)C)C1.CC.O c1(C(=O)NC(CCNC(c2c(SC)cccn2)=O)(C)C)nc(Cl)c(=O)[nH]c1N N1(C(c2c(C)nn[nH]2)=O)CCCC2C1CCCN2C(c1cc2occc2n1C)=O c1(C(=O)NCCC(C)NC(c2cc(Cl)c(Cl)c(Cl)c2)=O)cccc2cncn12 N1(C(c2cccnc2)=O)CCN(C(=O)C(O)CC2CCC2)C(c2cn[nH]c2)C1 O=C1CC(CC(=O)NC2(C)CCCN(C(C3(O)CN4CCC3CC4)=O)C2)=NN1 C1(NC(C(C2(C)CC2)NC(C(C)N2CCCC2)=O)=O)CCCCCC1(C)C Cc1ccc(F)cc1C(N1CCC(NC(C2C=CCS2)=O)C1C1CC1)=O c1(C(=O)NCC2CCN(C(C(CC=C)C)=O)C2)cc2n(n1)CCCO2 C(=O)(C(C)S(C)(=O)=O)NC1(CNC(C2(C#C)CCCC2)=O)CC12CCC2 c1(C(=O)NCCCN(C2CCCC(C(F)(F)F)C2)CC)ccc(Cl)c(Cl)c1 O=C(NNc1cccc(Cl)n1)c1cc2ncnc(C(F)(F)F)c2cc1Br C1(NC(c2ccc(=O)oc2)=O)CC2(C1)CCC2.C1(C=O)CCCS(=O)(=O)N1 C1(NC(CN2CCC(C)C2)=O)CCCCN(C(c2cc(N)cc(F)c2)=O)CC1 c1(SCC)ccc(C(N2CCCC2C(C)NC(=O)C#CC2CC2)=O)cn1 C=CCC(C)(CC)C(=O)NC1CCC(NC(=O)CCc2c(C)noc2Cl)CC1 c1(OC)cccn2ncc(C(=O)NCCc3ccc(Cl)cc3)c12 C1(CNC(C2(CCN(C)C)CC2)=O)CCCCC1.c1(C=O)c[nH]nc1OCF C(c1ccccc1)=CCCC(=O)NC1CC(CNC(=O)CCc2ccc[nH]2)C1 Cc1cccc(C2(C(=O)NC(C)CC3CCN(C(=O)C=C(Cl)Cl)CC3)CCC2)c1 C#CCCN=C(NCc1c(O)ncnc1O)N1CCC(NC(=O)OCC)CC1 CS(=O)(=O)C1CCCN(C(C2C3CCC(C3)C2NCc2cc(Cl)ncc2Br)=O)C1 C(=O)(C(CC)CC(C)C)NC(CNC(c1nc(CCC)sc1)=O)CC(F)(F)F c1(N2CCC(C(C)OC)CC2)ncc(C)cc1S(=O)(=O)N(C(CF)CF)C(C)C c1(C(N(C)CC2N(C(C(CC#C)O)=O)CCCC2)=O)c(Cl)cccc1Cl C(=O)(C1=CC(O)CC1)NC1(COC)CCCCC1.C(=O)C(F)CC(C)(C)C.N Cc1nc(NC(C2CCN2Cc2ccc(F)c(C(=O)O)c2)=O)cc(O)n1 CC(N=c1[nH]c(N2CCC(C3CCCC3)C2)nc2c1CCCC2)C1CCC1 Cc1cc(C(N2CCCC2CCCNC(c2nccnc2C(N)=O)=O)=O)n(C)n1 Cc1ncc(CC(=O)NC2CCCC2NC(c2csc(C)n2)=O)s1 c1(CNC(=O)CN2CCN(C(C3C4COCC34)=O)CC2)cc(Cl)c(Cl)cc1Cl C(=O)(CCC1=CCCCC1)NCC1N(C(c2c(N)c3c(s2)nccc3)=O)CC=C1 c1(OCC(=O)NC2CCN(c3n(C)ccn3)C2)ccc(-c2nn[nH]n2)cc1F Cc1cc(C(=O)NCCC2COCCN2C(C23COC(CF)(C2)C3)=O)n(C)n1 S(=O)(=O)(c1ccc(C(=O)NCCCC(C)CO)cc1)N1C(C=C)CCC1 CC(C(C)(C)C)=CC(=O)NCC(C(=O)NC(c1ccnn1C)C)N(C)C C1(CNC(c2ccnn2-c2ccccc2)=O)CCN(Cc2nc(CO)no2)CC1 c1(CC)nn(C)cc1C(=O)NCC1CC(NC2CC2C(C)(F)F)C1 C1(C(=O)NC(C2CCCC2)CN(C(=O)C2=CCOC2)C)CC2C=CC1CCC2 C=CC(C(=O)NC(C)C=CC(=O)NCC(C)(C)C=C)OC C1(N(C(C2C=CCC2)=O)C)CN(C(c2cn(C)ccc2=O)=O)CC12CC2.COC N1(C(c2nc(CC(C)C)sc2)=O)CCN(C(=O)CCCn2cccn2)C(C)C1C c1(C(=O)NC2CC(NC(CC(CC)(C)C)=O)CC2O)cccc(C#CC2CC2)c1 N1(C(CCOCCC)=O)CCC(N(C(=O)CCc2cnoc2)C)C1 CC1(CNC(=O)CC2CCC=CCC2)CCN(C(c2cc[nH]c(=N)c2)=O)CC1 Cc1[nH]cc(C(N2CC3CN(C(C4CC4C)=O)CC3C2)=O)c(=O)c1Br C1(OCCN2CCC(N(C(=O)C=C(C)C)CCC)C2)CCCCCC1 C1(C(=O)OC)C(C(N2CC(CCC)C2)=O)C2CCC12.c1(C(=O)N)ccccc1F C(=O)(C(C)(C)C(C)O)N(CCCNC(C(CC)NC(N)=O)=O)C1CC1 C1(CC=O)CC(C)N(C=O)C1.CCC(CC)=CC=O.C1CC1.C(C)(C)C.N C1(N(C(=O)C=CC(=O)N(C)C)CC)CCN(C(c2cccc[n+]2[O-])=O)CC1 c1(-n2ncc(C(N3CC(C4CC4)OC(C)C3)C(=O)N)c2)ccc(Cl)c(Cl)c1.CC N1(C(CC2(C#N)CC2)=O)CC(F)(CNC(c2c[nH]nc2C2CC2)=O)C1 c1(N(C2CCSC2)CCOC)ccc(S(=O)(=O)NCC2SCCS2)c(Br)c1 C1(C(N(CC#C)CCO)=O)CN1C(=O)CC CCC(C(=O)NC(CNC(=O)CCOC(C)C)CO)N1CCCC1=O CC1CCC(O)(C(N2CC3(C2)CN(C(c2cnc(Cl)[nH]2)=O)C3)=O)CC1 C1(CNC(c2ccc(O)c(Cl)c2)=O)CCCN(C(=O)CS)CC1.c1ccccn1 N1(C(c2c(OC)c(O)ccc2)C(=O)NCc2cccs2)CC2CCCCC2C1 C(C)(N=c1[nH]c(=N)[nH]c(=NC2CCC(CCC3CC3)CC2)[nH]1)c1c(C)n(C)nc1 N1(C(C(CC2CC2)NC(C(C(CC)C)N(C)C)=O)=O)Cc2ccc(C#N)cc2C1 c1(C(N2CCN(C(C)=O)CC2)=O)n[nH]c2c1CN(C(=O)Cc1cc(C)no1)C2 c1(C=O)cccc(CS(C)(=O)=O)c1.C1(C(=O)NCCC)(SC)CCC1.CC CCC(C)(C)CCCC(=O)NCCCCC(=O)NC(C)CCO CC1CN(C(c2ccn(C)n2)=O)CCCN1C(=O)CC(C(F)(F)F)c1ccon1 N1(C(c2c(C)scn2)=O)CCN(C(c2c[nH]nc2C(C)C)=O)CC1C CC1(CNC(=O)CCCCCNC(C2CCNC2=O)=O)NC(=O)NC1=O C(=O)(C#CC1CCCC1)N1CCCC(C(N2CCN(C(C#C)C)CC2)=O)C1C C(=O)(C(C(C)(C)C)C1CCC1)N1CC(OC)(CNC(=O)C(C)(C)CF)C1 C#CCCCCC(=O)NCC(C)(CO)NC(=O)C(C)Oc1cccnc1C(C)=O c1(C(=O)N)ccc2[nH]c(=N)sc2c1.C1(C(=O)NC(C)CC)CCN(C(N)=O)CC1 N(C(=NCCC1CCCCC12CC2)N1CCC2NC(=O)OCC2C1)CCOC N1(C(c2cccn(C)c2=O)=O)CCC2C(CCCN2C(c2ccsc2C#N)=O)C1 N1(C(C(CC)OC)=O)CCCCC1CCN(C(=O)Cc1ccc(C(C)=O)cc1)C C=CCCCCCCCC(=O)N(C(C)CN(C(=O)C(c1ccc(Cl)cc1)O)C)C N1(C(C(CNC(C2C(C=C)OCC2)=O)CCC)=O)CC2(CCC1CO)CC2 C(C(C)(C)C(=O)NCC1CCN1C(=O)CCc1cccc(OC)c1)OC C1(C)(C(=O)NCCN(C(CC2C(OC)CC2)=O)C)Cc2ccccc2N1 C1(CSC)(CNC(C2NCCCC2c2ccccc2)=O)CCOCC1 CC(C)CC(O)C(=O)NCC(CNC(=O)CCn1cnnn1)S(C)(=O)=O CON(CCO)C(=O)CN=c1nc(N2CCOC3(CC3)C2)c2c([nH]1)CCCCCC2 c1(C(=O)NC(CN(C(C(C)NC(c2ccccc2)=O)=O)C)(C)C)ncccc1O CC(C)C(O)CC(=O)NCCOC1CN(C(C2(C)C=CCC2)=O)C1 c1(CC)cnc(C)c(NC(=O)C(CNC(=O)CCC(C)(C)F)N(C)C)c1 C1(C)(CNC(CC(COC)C)=O)CN(CCc2scnc2C)CCO1 N1(C(C(CCC=C)(F)F)=O)CCC2(CC1)CCS2(=O)=O.C(=O)(C(F)=CC1CC1)N C(=O)(C(C(C)CC)OCC(F)F)Nc1c(OCC)nccc1 C1(NC(C=CCC)=O)CCN(C(=O)C(C)Oc2ccc(C)cc2)CC1O c1(C(N2CC(C)N(C(C3COCCO3)=O)CC2)=O)coc2c(Cl)cccc12 C1CC(C(F)(F)F)CN1C(=O)C(C(C)C)n1cnnc1.C(C(=O)N)SC(C)C C(=O)(C1CCc2ccccc21)NC1CC(C(=O)NCc2c[nH]c3ccncc23)C1 Cn1cc(OCOCCNC(=O)CN2CCC(CS(N)(=O)=O)C2)cn1 c1(C(N2C(CCCNC(C3CC4CCC4C3)=O)CCC2)=O)cc2ccsc2s1 c1(C(N2CC3(CCC(CNC(CS(CC)=O)=O)O3)C2)=O)cc2ccccc2cn1 N1(C(c2cc(OC)ncn2)=O)CCN(C(=O)CCC(C)SC)C(C(C)(C)C)C1 c1(C(=O)OCC(C2CCCCC2)OC)cnn(C(C)(C)C)c1 CC(C)C(C(=O)N1CCCC1CCCO)C(C)NC(=O)CC1CC2(CC2)C1 CCC(CN(C)C)CC(=O)NCCC(C)N(C)C(c1cc(CC(C)C)[nH]n1)=O N1(C(CC2CCCN(C(c3cc(CC)[nH]n3)=O)C2)=O)CCC(C)(CO)C(O)C1 C=C(C)CCCC(=O)NC1CCC(C)C1.c1(CC=O)c(C)nn(C(F)F)c1C.N C1(C(=O)NC2CCN(C(=O)C=C3CCOCC3)C2)CC12CCC(F)(F)CC2.C C=CC(C)(O)CC(=O)NC(C1CN(C(c2cc(-c3cnn(C)c3)on2)=O)C1)C C1(C(=O)NCC2CCCN2C(=O)C(O)C2CCC2)CCCS1(=O)=O c1(C(N2C(CNC(C(CC)n3ccnc3)=O)CCCC2)=O)n[nH]c2ccccc12 C=C(C)CC(C)C(=O)N(CCCN(C)C)CC.c1(C(=O)N)cc(N)cc(O)c1 c1(C(N2CCCC(C(C)NC(CC(CC)(F)F)=O)C2)=O)nccc2ccn(C)c12 c1(OC)ccccc1CC(=O)NC1(CNC(=O)CCC(C)OC)CC1 C(=O)(C#CC1CCOC1)N1CCN(C(c2sc(CC)c(C)c2)=O)CC1CC(F)F Cc1oc(S(C)(=O)=O)cc1C(N1CCC(NC(=O)C(C)C)C(F)C1)=O CCC(CC(=O)N(C)CC1CCCN1C(c1nc(OC)c(C)s1)=O)C1CC1 C1(C(=O)NCCCN(C(=O)C(c2ccccc2)O)CC)CCOCC12CCCC2 CCC(C)C(O)C(=O)N1CCOC(CCNC(c2cc(N)nc(Cl)c2)=O)C1 c1(C(=O)N)ccc(Cl)cc1C(F)F.C1(N(C(COCCC#C)=O)C)CCCCC1 Cc1ccc(OCC(N2CCC(C(C)NC(=O)CC(C)CF)CC2)=O)cc1C C1(C(N2CCOCC(C(=O)NC3CCN(C)C(=O)C3)C2)=O)Cc2ccccc2C1 c1(C(N2CC3C(NC(c4cc(O)ccc4F)=O)(C3)C2)=O)nccc2ccsc12 C1(C=O)CN(C(=O)CC2CC=CCC2)CC1(C)C.C(=O)(CC1CC1)O.CC Nc1nc2c(cc1C(=O)NC1CCCCCN(C(C3CCC(=O)N3)=O)C1)CCC2 N1(C(c2c(C)noc2)=O)CC2CCCC(C1)N(C(c1cc3ccccn3n1)=O)C2 c1(N2CC(CCO)OCCC2)nccc(=NCC2(CO)CCC2)[nH]1 N1(C(c2c(S(C)(=O)=O)cn(C)n2)=O)CC(C(=O)O)CC2COCCC12 C1(C(=O)OC)CCc2nc(NC(C3CCc4c(nnn4C)C3)=O)sc2C1 N1(C(c2ccccc2CO)=O)CCC2CC(CNC(C3(O)CC3)=O)CCC2C1 C1(NC(c2c(C)nn(CC(=O)Nc3ccccc3)c2Cl)=O)CCn2cnnc2C1 Cc1cnc(CCNC(=O)CCCCNC(C2CCC(N(C)C)C2)=O)cn1 Cc1cc(C(=O)NC2CCC(CNC(C3CC=CCO3)=O)C2)ccn1 N1(C(=O)CC2CCNC2=O)CCN(C(c2ncncc2Cl)=O)C(c2ncc[nH]2)C1 C1(NC(c2c(C)[nH]nc2C(F)F)=O)CC2(CCN(C(C3(F)CCCC3)=O)C2)C1 C1CN(C(c2ccccc2-c2ncnn2C)=O)C(C)(C)C1.C1(OC)CC1C(=O)N CCCC(O)C(CO)NC(C1CC(NC(c2cnc(C)nc2C)=O)C1(C)C)=O C1(OC)CC(CO)N(C(=O)CCC2CC2)C1.C1(CC(=O)N)CCC(C)(C)C1 Cc1ccc(C(N2CCCC2CCCNC(=O)COCc2ccnn2C)=O)cn1 C1(C(=O)Nc2ccccn2)CN(C(C2CCN(Cc3ccccc3)C2)=O)CCO1 Cc1ccc(C(=O)NCC(C2CCCCC2)NC(C2COCC2(C)C)=O)nc1 c1(CNCCCN(c2ccc(F)cc2F)C)ccc2nccnc2c1 N1(C(CCC(=C)Cl)=O)CCC(C)(C)C1CC(=O)N(C(C)CCC(C)C)C Cc1cc2cc(C(=O)N(c3ccc(C)nn3)C)ccc2[nH]1 C1(C#N)(CN(C)Cc2scnc2Cl)CCOCC1 N1(c2nc(CC)c(C)cc2C#N)CCC2(CC1)COC(C)O2 c1(C(C(N2CC(N(C(C(C)OC3CCCC3)=O)C)C2)=O)C)cc2ccccc2o1 N1(C(CCN2C(=O)CCC2)=O)CCC2CCC(C1)N2C(=O)CCCc1ccsc1 C(=O)(C1=CCN(C(=O)CC(C)(C)CC2CC2)CC1)NC1C(O)CCN(C)C1 CC1=C(C(=O)NC(C)CCNC(=O)C(C)CC2CCC2)COCC1 C=C1CCN(C(=O)CCCC(C)C)C(C(=O)NC(c2cn[nH]c2)C)C1 C1(C)(CNC(Cn2ccc(C)n2)=O)CN(C(=O)C)CCO1.C1(C=O)CCC1.N N1(C(C(C(C)C)NC(N)=O)=O)CC2CSCC2(C)C1.c12cn(nn1)C2 C(=O)(C(C#N)CCC)N1CCC(F)(C(=O)NCCCOCC#C)C1 c1(OC)ccc(CN(C)CCOc2ccc(F)cc2)nn1.c12ccccc1S2 c1(C(N2C(CN(C(c3n[nH]c(C)c3C)=O)C)CCC2)=O)[nH]nc2c1CCC2(C)C c1(C(N(C)CC2CCN(C(=O)C=Cc3cscn3)C2)=O)ccc(S(C)=O)cc1 c1(C(N2CC(C(NOC(CC)C)=O)OCC2)=O)noc(CC)c1C N1(C(CCC(C)OC)=O)CCCC(F)(CNC(=O)CN=[N+]=[N-])C1 c1(CC2CC2)cccnc1Cl.c1(C(=O)Nc2nc(C=O)cs2)ccc(Cl)nc1.N C1(N(C(C(COC)O)=O)CCNC(C2CC2)=O)CCCCCC1.N(C)(C)C N1(C(CNC(CC)=O)=O)CC(CCO)(NC(=O)C(C)CSc2ccccc2)C1 N1(C(C2(OC)CCC2)=O)CC(C(N2CCCC(C(C)C)CC2)=O)C(F)(F)C1 N1(C(C(CC)(CO)OC)=O)CCC2(CCN(C(=O)C(c3ccnn3C)C)C2)C1 CS(=O)C1(CNC(=O)C)CC1.C12CCCC1C2.C(=O)(CCC1CCCO1)N Cc1c(C(N2CCCC(C(C)(C)C(=O)NCC(C)(C)C3CC3)C2)=O)ccn1C N1(C(CC=CCC)=O)CCOC(C2CCC2)C1.N1(CCC)CCC(C=O)C1 C1(NC(c2ccc(C)cn2)=O)C2C3CCC(C3)C12.n1(CC(=O)N)nccn1 N1(C(CC(C)C)C)CCC2CC(C(=O)NCCC#N)C2C1 N1(C(c2n(CC=C)ccn2)=O)CC(NC(=O)COCCCOC)CCC1C CCC(CNC(C)=O)C=O.[SH](=O)(=O)C(F)(F)F.C1CCC1.C(=O)CC.N C(=O)(CCCCNC(c1ccc(=N)[nH]c1)=O)N(CCCC)C c1(CC)cc(C(=O)N)c(C)o1.C1(O)(C(C)C)CCN(C(=O)C=CC(C)C)C1 c1(C(=O)NC2(C)CN(C(C(C(C)OC)O)=O)C2)cccc2c1OCCC2 C(CN=c1ccn2ccnc2[nH]1)(N(C(=O)CCCc1ccc(Cl)cc1)C)C1CC1 N(C1CCCOc2ccccc21)C(=O)NCCF.C(C(C(F)(F)F)N1CCOCC1)N Cc1[nH]c(=NCC(C)(C2CC2)NC(C2C3C4CCC(C4)C23)=O)ccc1[N+](=O)[O-] CC1(C(=O)NCC2(F)CCC2)CC(C(F)(F)F)=NO1.C(=O)C.CCF.C Cc1ncccc1C=CC(N1CCC(CNC(=O)C(C)(C)CC#N)C(O)C1)=O N1(C(Cc2c(C)non2)=O)CCN(c2nnnn2C)CC1 c1(C(=O)NCC(C)NC(c2cccc(N3CCCC3)c2)=O)cnn2c1OCCC2 C#Cc1ccc(C(=O)NC(CC(=C)Cl)C(=O)NC(C)CCCC)cc1 C(=O)(C(C)(C)N1CCCC1)NCC(CO)NC(C(C1CC1)OCC)=O C(C)(C)(CN=c1nnn(C)[nH]1)NC(Cc1c(C)[nH]c2ccc(F)cc21)=O CCC1=C(C(=O)N2CCC(NC(c3ncnc(O)c3Cl)=O)C(F)C2)SCCO1 N1(C(C2N(C)CC(O)C2)=O)CCCC12CCN(C(=O)CC13COCC(C1)C3)CC2 N1(C(C(=O)NCc2cc(CC)n[nH]2)=O)CCC2(CC2)C1.N1CC2=CCC1CC2 C1(NC(COC2CCN(C(Cc3c(C)ccs3)=O)C2)=O)(CO)CCCCC1 N1(C(CCC=C)=O)CCN(C(c2ccc(-c3ocnc3C)cc2)=O)C2CC12 c12ccc(Cl)cc1O2.C=CCC(=O)NC1CCC1NC(=O)C(C)SC C1(C(N(CCC#C)C)=O)CC(NC(=O)C(C)C)CCO1 C(=O)(C(CC(F)F)N(C)C(c1ccnc(O)c1F)=O)NC(CC#C)CC#C N1(CC)CCN(c2cc(NCC3CC3C3CC3)nc(C(F)(F)F)n2)CC1=O C1(OCC)COCCC1CC(=O)NCCCCN(CCCS)C.C1CCC(=O)N1 C1(C(=O)NC(CNC(c2ccc(C)o2)=O)C2CC2)(OC)CCCSC1 n1(CC(=O)NC(C2CCCN(C(=O)CC3CCC3)C2)C)ncc(C#N)c1N C(=O)(C1=CCCCC1C)NC1CC(C(C)NC(c2c(C)oc(CO)n2)=O)C1 N1(C(c2cc(C)c(C)nc2)=O)CC2(CCN(C(=O)C(F)F)CC2)CC1C CC1(C)OCc2c1n[nH]c2C(=O)N.C1(C)CN(C(=O)C(O)C2CC2)C(C)(C)C1 C1(C)(C(N(C2CC(SC)C2)C)=O)CCCN(C(c2ccnc(CO)c2)=O)C1 C1(NC(C2C3(CC3)C23CC3)=O)C2CC3C(C2)C13C(C(CO)CCF)=O N1(C(CC(CNC(C(COC)C)=O)C)=O)CCC2(COC(C)C2)C1 c1(C(=O)NC2CC(O)(CNC(C(CCC)C)=O)C2)ccc2c(c1)C(=O)CCN2 C1(NC2CC(C#N)C2)CCN(C(=O)C(O)CN2CCCC2)CC1 Cc1cc(C(=O)NC2CCCC(NC(c3cnc(O)s3)=O)C2)c2ncccc2c1 C(=O)(CCC)N(CCOCCCC)CC.C1(C)(C=O)CC(F)(F)C1.O c1(C(=O)OCC)cncc([N+](=O)[O-])c1.N1(C=O)CCCC(n2cc(C)cn2)C1.N C(=O)(C(C)(O)c1cccs1)NCCCCN(C(=O)C(c1cscn1)N(C)C)C c1(OC)c(Br)cc(C(N2C(C(=O)NCCNC(C)=O)CCC2C)=O)cc1Br Cc1cc(=NCC2(F)CC(NC(=O)CC(C)CC(F)(F)F)C2)[nH]c(C)n1 c1(-c2cccc(OCC(=O)Nc3ccc(C(CC)=O)cc3)n2)cc(F)cc(Cl)c1 C(=O)(C#CC1(C)CCCO1)NCCC(=C)CNC(=O)C(CC)C(C)C C1(NC(=O)Cc2cnc[nH]2)CC(O)CN(C(c2ccc(F)c(C(F)F)n2)=O)C1 Cc1nc(C(=O)NC2CCC(NC(=O)CCC3CCCO3)CC2)c(C)s1 C(CC(C)CCNC(=O)CCCN(C)C)NC(C(C)CC1CC1)=O N1(CC(=O)N(C2CC(NC(=O)CC3(O)CCCCC3)C2)C)CCS(=O)CC1 c1(C(N2CCC(C(=O)Nc3c(OC)c(Cl)ccc3)CC2)=O)ccc(F)c(F)c1Br CCCCC(O)CC(=O)N1CCCCC1CN(C)C(c1c[nH]c(=N)o1)=O c1(OCC(=O)N(C2CCNC2=O)Cc2ccccc2)cnc(Cl)cn1 CCCCC(C)C(=O)N1CCC(C)C(NC(c2ccc(F)c(OC)c2)=O)C1 C1(C(=O)N)CCCN2CCCC12.CCC(COC)C(=O)NCC1(O)CC(C)C1 c1(-n2c(CN3C(=O)C(NCc4ccccn4)CC3)ncc2)c(F)ccc(Cl)c1F CC1CC2(CCC(CN(C=O)Cc3ccc(OCC4CCCO4)nc3)O2)CO1 C1(CC#C)(C(=O)N(CC(C)CNC(c2onc(C)c2C)=O)C)CC=CCC1 c1(C(N(C(C(=O)N(CC(C)C)CCO)C)C2CC2)=O)cc(F)cnc1O C(C)(c1ccco1)=CC=O.C(=O)(CCC1CCC1)NC(C#C)CC1CCCC1 c1(C(=O)NC(C)CCNC(=O)CC2CCC3CC3C2)cc2cnccc2o1 C(=O)(C1=CC(C)(C)C1)N1C(NCCn2cc(C3CCCN(C)C3)nn2)CCCC1 C1(NC(CC2(C=C)CC2)=O)CCN(C(=O)CN2CCCCC2)CC1 c1(C(=O)NCC2(C)CCN(C(C=CC)=O)C2)nn(C)cc1S(C)(=O)=O C1(NC(=O)COC2CC2)CC12CC(NC(c1cc[nH]c1C1CCC1)=O)C2 N1(C(c2cncc(C(C)C)c2)=O)CC2(C1)SCCC2NC(=O)C(C)c1ccsn1 C1(NC(C(CCC)NC(=O)CCN2CCCC2=O)=O)CN(C)C(C)(C)C1 C1(CCOC)CN(C(=O)CNC(C)=O)CCN1C(C1(C)CCCOC1)=O C(=O)C(C)(C)CC.CC1(c2ccccc2)CC(C=O)C1.C(=O)C=C1CCC1.N c1(C(=O)NC2C3CN(C(COC)=O)C2CC3)cc(C)c(F)c(C)c1 c1(-c2cc(CN(C(CC)C(=O)O)C)sc2)cc(S(=O)(=O)CC)ccc1OC C12(C(N3CCC(CC(=O)NC)C3)=O)CCCC1CCN2C(=O)C1=COCCC1 c1(CC(N2C(C)C(NC(=O)Cc3ncc(Cl)s3)CC2)=O)ccc(S(C)=O)cc1 c1(C(=O)NCC2C(NC(=O)CCCn3cncn3)CCC2)cc2ccccc2o1 CCC(CC(=O)N1CCC(C(C)(C)NC(=O)Cc2cc(C)[nH]n2)CC1)CC(C)C CCC(C(=O)OC)C(=O)N1CCOC(CNC(=O)CCC(C)(C)F)C1 c1(C(=O)NC2CCN(C(C=CCC)=O)CC2CC)ccc(C)c2[nH]c(C)cc12 c1(C2C(C(=O)N)C2)ccc(N(C)C)cc1.N1(C(CC=C(C)C)=O)CCC(C)C1 N1(Cc2n(CC)c(O)nn2)CC(=O)N(CC(c2ccc(F)cc2)(F)F)C1=O C1(NC(C=C(C)c2cccnc2)=O)CCN(C(=O)C(C)C2CCC2)CCC1(F)F C1(CC)CN(C(C2CCN(CC)C2)=O)CCC1C.C1(C(=O)N)CC(C2CC2)C1 c1(CC(=O)N)ccccc1[N+](=O)[O-].CC(C(=O)N1CCC(F)(C)C1)S(N)(=O)=O c1(CN=C(NCC2N(CC)CCC2)NC2CC2(F)F)cnc2c(Cl)cnn2c1 CCCC(O)C(=O)NCC(c1ccc(C)cc1)NC(c1ccnn1CCC)=O N1(CCCC)CCCCC1CNC(c1ccnc(CNC(C)=O)c1)=O Cc1nc(C)c(C(N2CCC(OC3CC(N(C)C)C3)CC2)=O)s1 C1(CONC(C(CC2CCC2)NC(CC2(C)CC2)=O)=O)Cc2ccccc2C1 C(C(C)(C)CC(=O)N1CC2CC(NC(C3(C)CCCS3(=O)=O)=O)C1C2)OC N1(CC(=O)OCC)CCCC1C.c1cc[nH]c1.C1(C=O)CCCC1C(C)C C1(C(=O)NCC=CCNC(=O)CCCc2ccncc2)CCC12CCCO2 CC(C)(C)C1=NOC(C)(C(=O)N)C1.C1CN(C(C2(n3cccn3)CC2)=O)CC1O N1(C(C2CN(Cc3ccc(CC)s3)C2)=O)CCCNC(=O)C1 CCCCCCCC(F)C(=O)N(CC(C)NC(=O)C(F)OC(F)(F)F)C N1(C(c2nc(C)[nH]n2)=O)CC2CC1CN(C(=O)CC1(C)CCCCC1)C2 C(=O)(C(F)(F)C(C)(C)O)NC(CC#C)CC(=O)NCC(C)CN1CCCC1 Cc1ccc(N)c(C(=O)NCc2ccnc(N3CCCCC3)c2)c1F C12(NC(c3n(C)c(S)nc3)=O)CCC1CN(C(=O)CCn1cnnn1)C2 CC#CCCCC(=O)NC1(CO)CCN(C(c2cnc(O)n2CC)=O)CC1 NS(=O)(=O)C1(C(N2CC(CCCCNC(c3csc(Cl)c3Cl)=O)C2)=O)CC1 N1(C(C(C)N2CCCC2)=O)CCCCC(C(=O)NC(c2ccccn2)C)C1 C1(C(C)C)CN(C(=O)COC2CCCC2)CCCN1C(C1CCN(C)C1=O)=O Cc1cccc2c(C(N3CCOC(CCNC(c4ccccn4)=O)C3)=O)n[nH]c12 C1(CNC(c2n[nH]c(C)c2Cl)=O)CC2CCC1N2C(=O)C(O)CC1CCCCC1 N1(C(c2cc(SC)oc2)=O)CCCC(C)(NC(c2cnn(CC(F)F)c2C)=O)C1 c1(NC(=O)CC2CCCN2C(c2cc(Br)c[nH]2)=O)cc2cccc(O)c2[nH]1 N1(C(CC(CC)C2CCC2)=O)CCN(C(C2(C(F)(F)F)CCCC2)=O)CC1CC C#CCC(CC(F)F)C(=O)N(CC(=O)NC1CCn2nccc2C1)C c1(C(CC)C)ccc(O)c(C(C(=O)NCCSCC)N(CC(F)(F)F)C)c1 C1(C(N(CCN(C(CCc2nnc(C)n2C)=O)C(C)C)C)=O)SC2C=CC1CC2 C(CCC(=O)NC(C1CCN(C(=O)C(C)(C)C)C1)C)N(C(C)=O)C N1(C(c2c(OCC)cccn2)=O)CCN(C(c2ccc(=O)n(C)c2)=O)C(CF)C1 c1(C(N2CCC(NC(COCCC)=O)C(CC)C2)=O)ccc2c(c1)CCN(C)C2 CC(C)C(C)C(C)CC(=O)NC1(C2CCCN2c2ncc(Cl)c(O)n2)CC1 c1(C(N2CC(C3OCCN(C(c4cc(CO)on4)=O)C3)C2)=O)cc2c(s1)CCC2 N1(C(C(C)CN)=O)CC2CN(C(=O)Cn3cncn3)CC12 C(=O)(C(CCC1CC1)NC(=O)C(O)CC1CCCC1)NCCCC N1(C(Cc2n(C)ccn2)=O)CC2CCC1CC2NC(c1n[nH]cc1Cl)=O Cc1ccc2[nH]cc(C(N3CC(O)CC3CNC(C3CSC3)=O)=O)c(=O)c2c1 c1(NC(c2ccc(C#N)cc2)CC(=O)Nc2nc(C)c(Cl)s2)[nH]cc2c1CCC2 C1(CNC(CC(C=C)(C)O)=O)CCC2(CO1)CCC2.C1(C=O)CC(F)(F)C1.N C1(CCC)CN(CC(=O)N(C)Cc2cscn2)CCN1Cc1ccccc1 C1(C(=O)NC(CC)C(=O)N(C2CCN(C)C2=O)C)CCN(OC)CC1 N1(C(c2oc(CC)c(C)c2)=O)CCOC2(C1)CN(C(C1CCC(C#N)C1)=O)C2 C(=O)(CC(C)(O)c1ccccc1)NC1(C)CN(C(CCSCCCC)=O)C1 C1(C(=O)NCc2nc(C)on2)CC12CCN(C(C1CCCC1)=O)CC2 C1(c2ccccc2)CCCN1.N1(C(C2(CCOC)CC2)=O)CCOCC1 c1(C(N2C(C)CC(C)CC2)=O)cccc2nn(C)cc12.C(=O)(C(F)OC(F)(F)F)N C1(C2CC2)(C(=O)Nc2ncc(Cc3cccc(C)c3)n2C)CC(=O)C1 n1(CCCOC)nc(C(C)C)nc1-c1cccc(OCC2CCCO2)c1 C1(O)(C(c2nnnn2C2CCCC2)N)CCC(C)(C)CC1.C1(OCC)CCCC1 CC1COCC1(c1nnnn1C)NCc1cccc(SC(F)(F)F)c1 C1(NC(c2c(C)c(=O)cc[nH]2)=O)CCC2CN(C(=O)CC3C(C)(C)C3(C)C)CC12 CC1CCC(F)(C(=O)NC2CC(NC(=O)C=CC3CCCC3)C(O)C2)CC1 c1(C(=O)NC2C=CCN(C(CCc3nnc(C)n3C)=O)C2)csc([N+](=O)[O-])c1 C1(C(N(CC(CNC(c2c(C)cco2)=O)O)C)=O)Cc2ccccc2CO1 N1(Cc2cn(C(CC(N3CCC(C)CC3)=O)(C)C)nn2)CCNC(=O)CC1C N1(C(CCC=CC(C)C)=O)CCCC2(NC(c3cc(O)n(C)n3)=O)CCCC12 N1(C(c2nc(C)sc2)=O)CC2CS(=O)(=O)CC2C1.c1(C(=O)N)cc(O)cc(F)c1 c1(C(=O)NCCC2CN(C(CSCC#C)=O)CC2C)ccc(C)nc1N N1(C(Cn2ncc(CC)c2)=O)CC2CCN(C(C3(C(F)F)CCC3)=O)CCC2C1 c1(OCC(C)C)nnccc1C(=O)N(c1cccnn1)CC1CNC1 CCCCC(O)CC(=O)N1CCCC1CNC(c1cccc(F)c1C)=O c1(C(N2CCN(C(N(C)C)=O)CC2)=O)ccc2ncc(Br)c(Cl)c2c1 N1(C(C2N(C(=O)CC(C3CC3)C3CC3)CCSC2)=O)CCCC2(CCCO2)C1 C#CCC(C)(C)C(=O)N1CC=C(C(=O)Nc2ccc(O)c(F)c2)C1 N1(C(C2C(CC(C)C)C2)=O)CCC1CC(=O)NCCOC(=N)O CC1=C(C)CC(C)(C(=O)NCC2CCCCN2C(c2ccccc2)C)CC1 C(N=c1cc(C(N)=O)nc[nH]1)C1N(C(C2C(C)(C)COCC2)=O)CCC1 CC(CC(=O)O)(C(F)(F)F)NC1CNCC2(CCC2)C1 N1(CC(N2CCOC(CNC(C3(CO)CCCO3)=O)C2)=O)CCC(O)CC1 c1(C(N2C(C)(CNC(=O)C3=CCSC3)CCC2)=O)cc(F)cc2cccnc12 C1(O)(CN(C(Cc2cc(C)ns2)=O)C)CCN(C(=O)C=CCn2cncn2)C1 c1(CC(=O)N(C2CN(C(=O)CCn3cc(Cl)cn3)C2)C)c(F)cc(F)cc1F N1(C(CSCCCC)=O)C2CCC1CN(C(C1CCn3nccc3C1)=O)C2 C1(C)(C(N(C2CC(NC(C3(c4ccsc4)CC3)=O)C2)C)=O)CC1(F)F Cc1cc(C(=O)N(C2CCN(C(=O)C(O)CC3CC3)C2)CCO)c(N)c(C)c1 CCCCC(O)C(=O)NCC1CCC1NC(=O)CC1CCCCC1 Cc1cncc(C=CC(=O)NC2CCC(C)CC2)c1.C1(CC(=O)N)C=CCCC1 C(N=c1nc2c(cnn2C)c(NCC2(Br)CC2)[nH]1)c1cc(C)cc(C)n1 C1(NC(N2CCC3(C(C(=O)OCC)C3)CC2)=O)COc2ncccc2C1 C(=O)(C(CCC)C(C)C)N.N1(C(C=CCN(CC#C)C)=O)CC(C)CC(C)C1 N1(C(c2ccc(C(=O)OC)n2C)=O)CCCC(NC(c2scc(C)c2C)=O)C1C C(=O)(CCCO)NCC1CCC1.C1(OC)CC(CCC(=O)NCC(C)C)C1 C(=O)(C1CCc2scnc21)N1CC2C(NC(C(C)CS(C)(=O)=O)=O)C(C2)C1 c1(C(c2n(C(CC)(C)C)nnn2)NCCC(O)CSC)nc(Br)ccc1OC c1(C(=O)NCCC2CCCN(C(C(CC)C)=O)C2)ccc(Cl)c(O)c1 C(=O)(C(F)C(F)(F)F)N.c1(N(CCC)C)ccc(C(N2CCOC(C)C2)=O)cn1 C1(C(=O)N)CCS(=O)CC1.n1(C(C)C)cc(C(=O)NCC2(C)CCC2)cn1 C1(NC(CC2(N(C(c3n(CCOC)ncc3)=O)C)CC2)=O)CCC(O)CC1 Cc1ccnc(C(=O)NC(C)(C)CCNC(=O)COc2ccc(Cl)cc2)c1 C1(CC#C)(C(=O)NCC2CC(SC)C2)CCN(C(=O)CCCC=C)C1 Cc1[nH]c(C(=O)NC2CCCC2CNC(c2nn(C)c(N)c2C)=O)c(C)c1C Cc1ccc2[nH]c(C(N3CC=CC(NC(C4CC(C)(C)CO4)=O)C3)=O)c(Cl)c2c1 N1(C(C(C(C)(C)C)OC)=O)CCC(NC(=O)C=C(C)I)C2(CCC2)C1 C1(C(N(CCCC)CC)=O)CCCNS1(=O)=O.c1(C(=O)N)ccsc1C(F)F N1(C(CC)=O)CC2CCOCC2(C(=O)O)C1.c1(CNC(COC)=O)ccc(O)o1 C1(C(=O)NC2(CCC)CC2)CC(NC(c2occc2CC)=O)CCO1 C1(CC)(CC)CC(NC(=O)C(C)CN(C)C)CN1C(C1CCCSC1C)=O c1(C(=O)N(C2CC3CNC2C3)Cc2cc3c(s2)CCC3)ccc2ccccc2n1 C1(COC)(C)CCCN1C(=O)Cc1cccc(C)c1.c1(C=O)cnn(C)c1N c1(C(N(CC(C)C(=O)NCCCc2cccnc2)C)=O)cccc[n+]1[O-] c1(NCCC2CCCN(C(C(C)CC3CCCC3)=O)C2)c[n+]([O-])ccc1[N+](=O)[O-] C(C(C)(C(=O)NCC1CC1CNC(c1cccc(Cl)c1)=O)OC)OC CC(C)CCC(O)C(=O)N1CCOCC(NC(c2cc(-c3ccco3)on2)=O)C1 n1(CC#C)c(C)cc(C(=O)NCCC2CC2)c1C.c1(C(=O)N)ccc(C)s1 C(=O)(CC(C)CC(C)(C)C)N.C(=O)(C1=CC(O)CC1)NCC(=O)NCC c1(C(=O)N)[nH]c2ccccc2c1C1CC1.C1(C(=O)NCCC)(CF)CC1(F)F c1(C(=O)NCc2ccc(-c3n(C)cnc3)nc2)cc(C(F)(F)F)cc(I)c1 C(=O)(C#CC(C)(C)CNC(=O)CC(C)(C)C)NC1(C)C(C)CCCC1 O=C(CC1=CCN(C(=O)C(O)c2ccsc2)CC1)NCC1(O)CC2CCC1O2 N1(C(C2C(C)(C)C2)=O)CCN(C(c2nocc2Cl)=O)CC1c1ccccc1Cl CCC(C)(C(=O)NCC(N1CC(C(N2CCCC2)=O)C1)=O)OC N1(C(c2ccc(F)c(C)c2Cl)=O)CC2(CCOCC2C(=O)NCCCN(C)C)C1 N1(C(CC2CC(N(C)C)C2)=O)Cc2n[nH]cc2C1C(=O)NCC1CCOC1(C)C C1(CC(=O)NCC(C)C#N)C2CCC(C2)N1C(=O)C=CC(C)(C)C.C c1(C(N(CCC)CCNC(c2cnc(C)cn2)=O)=O)ccc2nnnn2c1 N1(C(CN2CCCC(CC)C2)=O)CC=C(CCNC(=O)C(F)(F)C(C)(C)O)CC1 N1(C(C2(F)C(C)OCC2)=O)C2CCC1CC(CNC(C1CCC(=O)N1C)=O)C2 C1(NC(c2cc(CC)no2)=O)CCCCC1CNC(c1cnn(C)c1)=O.S C1(O)(CCNC(COCCSC)=O)CCCN(C(=O)C(C)CSC)C1 c1(CC(=O)N(Cc2ccco2)Cc2ncon2)ncc(-c2cccs2)o1 C(CC(C(C)(C)C)NC(C1CC(=O)NC(C)C1)=O)NC(C(N1CCOCC1)C)=O N1(C(C(CC)N(C)C)=O)CC(NC(c2cscn2)=O)Cc2ccccc21 N1(C(c2cccc(OCCOCC)c2)=O)CCC(Nc2ccncn2)C(F)C1 C1(NC(c2cc(C)[nH]n2)=O)CC2(C1)CC2C(N1CCN(c2cnccn2)CC1)=O N1(CC2(C)N=N2)CCN(c2cccc(CC#N)n2)CC1 C1(CNC(c2nn(C)c(O)c2)=O)(CO)CCN(C(C2CCC(=O)N2)=O)CC1 N1(C(C2(C#N)CCCC2)=O)CCN(C(=O)Cn2cc(Cl)cn2)C(CO)C1 c1(C(N(C(C)CCNC(=O)CC2CCC(=O)N2C)C)=O)cccc2nccnc12 C(N=c1ccc(C(F)(F)F)n[nH]1)C1CN(C(C=COCC)=O)C(C)C1 c1(NC2C(C)CCC2C)nc(N2CC3C4C=CC(C4)C3C2)c2ncsc2n1 c1(OC)ccccc1N1CC(C(=O)NCCOCC(N)=O)C1 C1(C)(OC)CCN(C(C2CC3CC2C2CC32)C(=O)Nc2ccc(F)cc2F)CC1 Cc1coc(C)c1C(=O)NCCN(C1CCCC1)C(c1cc(Cl)no1)=O Cc1c(C(=O)NC(C2CCCN2C(C2CCCCS2)=O)(C)C)cnn1CC(C)C C1(c2ccccc2)(CC(=O)N)CC1(C)C.C(=O)(CCc1cnoc1)N(CCC)C c1(C(N2CC(CC(C)NC(Cc3cnc(C)o3)=O)C2)=O)cccc(S(C)=O)c1 C1(C)(C(=O)NC(C(=O)NCCCCC(=O)OCC)C(C)C)CCCCCC1 c1(C(N2CCC(NC(C3=CC(C)(CC)C3)=O)CC2C)=O)occ2c1CCOC2 C(=O)(C(CCS(C)=O)N(C)C)NCC(CNC(c1c(OC)scc1)=O)CO C1(C(=O)NCC2CCCN(C(C(C)n3cncn3)=O)CC2)C2CCC3C(C2)CC13 CCCC(C(C)C)(c1nnnn1C1COC1)Nc1ccc(Cl)c(Br)c1 C(=O)(C(CNC(C1CC2(CCC2)CO1)=O)C(C)C)NC(C(=O)NC)C c1(NC(C2C(C=C)OCC2)=O)cc(Cl)cc(C#N)c1 N1(C(c2cccc(C)c2)C(=O)NCCCCCC)CCCCC1Cn1ccnn1 N1(C(=O)Nc2cc(CCC)nn2C)CC(CO)CC(F)C1 CC#CCCC(=O)NC1(CCCNC(=O)Cc2cccc(CC(F)(F)F)c2)CC1 C1CC2(CCC2)CN1C(c1ccccc1O)=O.c1(CC)onc(C)c1C(=O)NC CC1(C)OCc2cc(C#N)c(=NCC(C3CCCCC3)OCC(F)F)[nH]c21 C1CN(C(=O)CCc2cc(Cl)no2)C2(CCC2)C1.C(C)(C(=O)N)OCCC#C N1(C(CCCCC(=O)NC)=O)CCC2CCC(C1)N2C(c1ccnc(C)c1O)=O Cc1cccn2cc(C(=O)NC)cc12.C1CCCN1C(=O)C=CC=O.C1CC1 c1(CCNC(C2CCC(n3cc(COC)nn3)C2)=O)cccc(NC)c1 C1(NC(CC(CC)O)=O)(COC)CCN(C(C2CCCN2C(C)C)=O)CC1 c1(C(=O)NCC(CC)NC(=O)Cc2ccc(C)c(O)c2)ccc(N)c(N)n1 C1(CC)OCCC1C(=O)N.N1(CC=CC=O)CCCC1.C1(CC)CC1.C N1(C(C(C2CCCN(C(C(CC)C)=O)C2)(C)C)=O)CC2CCCC2C1 c1(C2CN(C(=O)NC(C(C)C)CN3CCOCC3)C2)ccc(I)nc1 Cc1cc(C)n(CCc2ccc(-c3ccc(C(=O)Nc4ccncn4)s3)cc2)n1 C(=O)(C1=NOC(C)(C)C1)N1CC(C)(NC(c2ccc(C)cc2F)=O)C1 c1(C(=O)NCC2N(C(Cc3cnc(C)[nH]3)=O)CC(C)CC2)nnn2c1COCC2 c1(SC)nc(Cl)cc(=NCC(C2CCCCC2)NC(c2ccnn2C)=O)[nH]1 C12(CC)CCC(C(=O)NCC3CC3(C)C)(CC1)CO2.C(=O)CC1CC1 c1(CCC(N2CCC(NC(C(C=C)(C)C)=O)(COC)C2)=O)c[nH]c2ccccc12 c1(C(=O)NC2CN(C(C34CC(CCC)(C3)C4)=O)CC2O)c(C)oc(C)c1C C(=O)(C(CNC(c1ncccc1N)=O)C(C)(C)C)N1CCC(COC)C1 N1(C(C2N(C)CCOC2)=O)CC2CCCC2(C(=O)NCCCS(N)(=O)=O)C1 C1(NC(C2N(C)CCOC2)=O)CN(C(C2CC(=O)C2(C)C)=O)CCC12CCC2 c1(C(=O)NC2CN(C(CNC(C)=O)=O)C2)cccc(N2CCOCC2=O)c1 C1(NC(C2CCC(OC(F)(F)F)C2)=O)CCc2nnc(C(F)(F)F)n2C1 N1(C(CNC(C(N2CCN(C)CC2)Cc2c(C)ncs2)=O)=O)CC2CCCC2C1 CC(C)C#CC(=O)N1CC(CC(F)C(=O)NCCCc2nnnn2C)C1 c1(C(=O)NC2CC(C)N(C(=O)C#CC3(C)COC3)C2)ccc2nc(CO)[nH]c2c1 N1(C(C(CC=C)NC(C)=O)=O)CC2CCN(C(=O)Cn3c(C)csc3=O)C2C1 C1(NC(c2cc(CC)c(Cl)cc2)=O)CCCC12CN(C(=O)C#CC1(C)COC1)C2 c1(C(=O)NCCC2(C(=O)NC(C(N)=O)C3CCCC3)CC2)ccco1.C N1(C(C2CC(=C)C2)=O)CCCC(C2CC2NC(C2CCc3ccccc3C2)=O)C1 Cc1ccc(NC(C2CC=CCN2C(=O)CC2CC3CC3C2)=O)cc1 C1(C2CCN(C(c3ccc(C#N)nc3O)=O)CC2)(NC(C(CCSC)O)=O)CC1 CC(C)CCC(F)C(=O)N1CCC(O)(CNC(=O)C(c2cccn2C)=O)C1 c1(CN(C(CC)C)C(=O)NCC2CCC(=O)N2)ccc(Cl)cc1 N1(C(C(CCC)N(C)C)=O)CCN(C(=O)C(C)Cc2cnn(C)c2)CC1C CN1CCC(C(=O)O)C1=O.c12ccccc1NC(=O)CCCc1cn-2nn1 C(=O)(CC(C)C(F)F)N1C(C(=O)NCCCOC(=O)NC)C(O)CC1 C(CO)(CC(C)CC)NC(CCC1CCN(C(c2c(C#C)c[nH]n2)=O)CC1)=O C1(CNC(=O)CCc2cnc(O)[nH]2)CC(F)CN1C(=O)COC1CCC1 C(=O)(C(CO)C(F)(F)F)NCC(=O)NC(CO)CC(F)(F)F c1(COC(C2CC3CC3C2)=O)ccc(C2(C(F)(F)F)CCO2)cc1 CCCCC(O)CC(=O)N(C(C(N1CCCC(CC)C1)=O)C1CC1)C N1(C(c2cc(CC)ncn2)=O)CC2CCC2(CCNC(c2nn(C)cc2N)=O)C1 Cc1ncncc1C(=O)NCC1OCCC1C(=O)N(c1ccc(Cl)cc1)C C(=O)(CC1=CCOCC1)N1CCCC(N(C(=O)C(C#N)C2CC2)CC)C1 C1(C(=O)NCCN(C(COCc2ncc(C)o2)=O)C)CC2(CC2)CO1 CC1C(C)N(C(c2cnc(S)n2C)=O)CCN1C(=O)Cn1cnc(Br)n1 c1(NC2(CNC(=O)CSc3ccccc3Cl)CCOC2)ncnc2ccsc12 CC(C)(C(=O)N1CCCC(C(F)F)C1)C1=CCN(C(=O)CNC=O)C1 C1(O)(CNC(Cc2ccc(OCC)cn2)=O)CCN(C(C2CC2F)=O)CC1 C1(NC(c2c(C)csn2)=O)CC2(C1)CC2C(=O)NCCC1CCCC2CC12 O=C1CC(C(=O)NC2COCCC2NC(=O)Cn2cnccc2=O)CCN1 C(C)(C)(CC(=O)NCCOc1ccccc1)NC(C(CSC)C)=O C(C(=O)NCC1CCOCC1)(C1=NOC2(CCC2)C1)NC1(C)NC(=O)NC1=O c1(CC)cc(C(=O)NCCC(O)CNC(=O)Cc2ccnn2C)oc1CC c1(C(=O)NC(C(C)OC)C(=O)N)ccc(C)c(O)c1.C1(CC)CC(F)(F)C1 C1(NC(C2(CC=C)CCC2)=O)CN(C(=O)C=CC2CCCN2C)CC1F C12(NC(c3cc(C)nn3C)=O)CCCC1N(CC(C)Cn1cccn1)CC2 C(=O)(CCCCCCC(=O)OC)NC1CCN(C(C(CC)NC(N)=O)=O)C1(C)C N1(C(C2CCC(=O)N2)=O)CCN(C(C23CCCN(CCC2)C3)=O)CC12CC2 c1(C(=O)N)cc(F)ccc1F.CC(C)(CO)C(C1CC1)NC(C1COCCC1)=O N1(C(C(C(C)C)C)=O)C2CCC1C(C)C(NC(=O)CCc1ccsc1)C2 C1(C=O)CCC(=O)N(c2ccccc2)C1.C(=O)(C(=O)NC1CC1)NCC.N c1(C(=O)NC(CNC(=O)C(c2ccc(Cl)cc2)CO)C2CC2)c(F)cncc1Cl CCCCC(C)C(=O)NCC1(COC)CN(C(c2cccnc2Cl)=O)C1 C1(C(=O)OC)CCC(n2nnnc2C(CC)(CC)NCC2CC(Cl)(Cl)C2)C1 C1(CC)CN(C(c2scnc2Br)=O)CCN1C(=O)Cc1nc[nH]n1 N1(C(=O)Cc2cc(C3CC3)no2)CCN(C(c2nc(CO)cs2)=O)C(CCO)C1 C1(NC(c2cc(C)c(Cl)s2)=O)CN(C(C2CC3C(C2)C3(F)F)=O)CCC1(C)C N1(C(c2cn(CC=C)nc2)=O)CC2CCN(C(c3ccccn3)=O)C2C1 C1(C(N2CCCC(C)(O)C2)=O)Cc2nccnc2CN1C(=O)C(F)(F)Cl C#Cc1ccnc(C(=O)NCC(O)CNC(C2CCC(O)CC2)=O)c1 c1(C(N2C(C)CC(CNC(c3ccc(CO)o3)=O)C2)=O)noc2c(F)cccc12 N1(C(C2CC(CC)N(C(C34CC(C#N)(C3)C4)=O)CC2)=O)CCC12CC(O)C2 c1(OCC)cc2c(s1)CCOC2CNC(C1CCC(NC(C)=O)CC1)=O CC(C)CC(CC(=O)N(C)Cc1ccon1)NC(=O)CC1CC(C)(C)CO1 c1(C(C(=O)NC(CC)C)N(C)Cc2ccon2)cc(F)cc(F)c1F C1(CCNC(CC2C(C)OCC2)=O)CCN(C)C(=O)O1 N1(C(C2(CC(C)=O)CCC2)=O)CC(C)OC(C)(C)C1.C(=O)C(C)(C)C(F)F n1(CC(=O)N(CC(CC)NC(=O)C(C)(C)C(=O)NC)C)ccc(C)cc1=O C1(C(N(C(C)C(=O)N(C(C)CSC)C)CC)=O)C=C(C)CS1 C(=O)(C(C(C)NC(=O)CCS(C)(=O)=O)C(C)C)NCC(C1CC1)SC c1(C(N2CC(C)(C)C(NC(c3ccns3)=O)C2)=O)cc2c(s1)CCC2=O c1(OC)nc(Cl)ccc1C(=O)NCCC(C)NC(C1(F)CCC(C)CC1)=O C=CCCCC(=O)NC1CC(CC(=O)NC2CCC3CCC23)C1(C)C C1(NC(c2c(C)nn(C)c2)c2nnnn2CCCF)CCC2CCCCC2C1 N1(C(c2ccn(CC(C)C)n2)=O)CCC(NC(C2CCCO2)=O)CC1 C1(NC(c2c(C)cccn2)=O)CC2CC(NC(=O)CC3CCCCC3(C)C)C1C2 n1(CC(N2CCC(C(C)NC(=O)CC3CC3C3CC3)C2)=O)cc(F)ccc1=O c1(N(C)CC2CCOC2)nnc(CS(C)(=O)=O)n1CCCN1CCOCC1 C(=O)(C1=C(C)OCCS1)NC1(C(=O)NC(CCOC)CO)CCC1 c1(OC)ccc(C)c(C(=O)NC2(CC)CC2)n1.O(C(F)(F)F)CC(=O)N CC(CCC(=O)NCC(O)CNC(c1ccc2c(c1)ncn2C)=O)S(C)(=O)=O c1(CC)cnc(Cl)nc1N(CCCNC(C1(F)CCCC1)=O)CC c1(C(N2CCC3(CN(C(CCC(CC)C)=O)C3)C2)=O)cnc(O)c([N+](=O)[O-])c1 C=C(CNC(c1cnn(CCNC(=O)CCCSC)c1)=O)C(F)(F)F C1(C(N2C3(C(=O)NCCCCC(C)C)CC3CC2)=O)CC2(C1)CC21CC1 N1(C(c2c(CNC(=O)C(O)Cn3cncn3)noc2)=O)CCC2(CCC2)C1 CC1(C)CC(CC(N2CCSCC2CCNC(=O)CC2(C)CCCO2)=O)CO1 CC1CN(C(=O)CN2CCCCC2)CC2(CCN(C(=O)CCCC(F)(F)F)C2)O1 C(=O)(CCN=c1ccc(C(F)(F)F)c[nH]1)NC1CCC(SC)CC1 C=CCCCCCCC(=O)N1CCC(CNC(=O)CC(C)CN(C)C)(OC)C1 c1(C(N2CCCCC2C)C(=O)NC(CC)C)ccc(-n2ccnc2)cc1 Cc1nc(N2CCOC(CN(C)C(C3CCN(C)C3=O)=O)C2)ccc1[N+](=O)[O-] CC(C)(CS(C)(=O)=O)C(=O)N1CCCC1CNC(C1CC2CC2C1)=O N1(C(=O)CC(c2ccccc2)C2CC2)CCC2(C1)CN(C(=O)C(Cl)(Cl)Cl)CCO2 N1(C(c2ccc(OC)c(Cl)c2)=O)CC(C)CN(C(=O)Cc2ncc(Cl)s2)CC1C C1(OC)C(NC(=O)NCC2CN(C(c3cc[nH]n3)=O)C2)CC12CCC2 c1(C(N2CC(CN(C(c3n[nH]c(C)c3C)=O)C)OCC2)=O)ccc(S(C)(=O)=O)s1 C(CC(C(=O)N1CCCC1CC(N1CC(C)(CF)C1)=O)OC)OC CCC(C)C(O)C(=O)NCC1(F)CCC(CNC(c2ccc(O)nn2)=O)C1 C(=O)(C(C)(C)C(N)=O)N1CCC(C2N(C(CC3CC3)=O)CCCC2)C1.CC=O.N N1(C(C2(c3cccc(N)c3)CCC2)=O)CCC2CNCC12 N1(C(c2ccc(=N)[nH]n2)=O)CC2CCN(C(=O)C(O)CCc3ccccc3)CC12 CC(C)CC(O)C(C)C(=O)N(CC(C)(C)NC(c1cc2cccnn2n1)=O)C c1(C(N(CCCNC(=O)CCc2cn(C)nn2)C)=O)cc(Cl)cc(Cl)c1 N1(C(CCCC)=O)CC2CCCCC2(CNC(c2cc(=N)[nH]c(Cl)n2)=O)C1 N1(C(c2c(C)cncc2)=O)CCCC2CCN(C(=O)CCc3ncc[nH]3)CC12 N1(C(CC2CCC(NC(C3CC=CCO3)=O)C2)=O)Cc2ccc(O)cc2C1 N1(C(C(CC)CC)=O)CC(NC(c2cnc(Cl)c(F)c2N)=O)CC12CCC2 c1(-c2cn(C)nc2)ccccc1CNCCCc1ncn(C)n1 c1(OC)c(C)cc(NS(=O)(=O)C(C)C(=O)N)cc1C.c1ccccc1CC(C)C CC(C)C(CO)C(=O)N1CC(C(C)NC(C2CCC(C(C)(C)C)CC2)=O)C1 N1(C(c2n(CC)nc(C(C)C)c2)=O)CCC(C#N)C1.c1(C(=O)N)nc(C)cs1 C1(NC(CS(CC)(=O)=O)=O)CC12CCN(C(=O)Nc1cccc([N+](=O)[O-])c1)CC2 C1(CN(C(C(CC)=CC)=O)C)COCCN1C(=O)CCc1cncc(OC)c1 c1(OC)cc(N)c(C(=O)NC23CC2CN(C(=O)CC2CSCCS2)C3)cc1O CC(C)(C)C(C(=O)NCCCc1cccnc1)n1cc(C2CCCO2)nn1 n1(CC)cnc2nc(N3CC4C(C3)C4(F)F)nc(NCCC34CC(CO3)C4)c12 c1(C(=O)NCC2CN(C(CNC(C)=O)=O)C(C)(C)C2)cc2nc[nH]c2cn1 C1(C)(CNC(C2(CCCC)CCC2)=O)CCC(NC(=O)C2=CCCC2)C1 c1(CC)noc(C)c1C(=O)NCC1CCCCC1.C(=O)(C)N.C(C)(C)C C1(C(N(CC(C)C)C(C)C)=O)CCCOC1c1ccccc1 C#CCC(CC(F)F)NC(=O)C(CC=CC)NC(c1ccoc1C)=O Cc1ccn(C(C)CC(=O)NCC2CCCN2c2nnc(CC(C)C)s2)n1 C1(NC(C2CC3(CCC3)CO2)=O)CCN(C(=O)Cn2cnnn2)C12CCC2 C1(CC)CCN(C(=O)CC2CCN(C(=O)CCc3cn[nH]c3)C2)C1C C1(C(N(CCOC)CC)=O)CCC2CC2CC1.c1(CC(=O)N)cc(C)sc1C c1(-c2n(-c3c(C)cc(Cl)cc3)nc(C3CC3)n2)nc(S(N)(=O)=O)c2ccccn12 N1(CCCCCNC(CN2C(C)CC2)=O)CCN(C(c2cocn2)=O)CC1 c1(C(N2C(C(=O)NC3CC3(F)F)CSCC2)=O)cn2cc(F)ccc2n1 C(=O)(C1=C(C)OCC1)NC(CNC(CCCCC)=O)CO N1(C(Cc2c(C)ccs2)=O)CCC(CC(N)=O)(NC(c2coc(CO)c2)=O)CC1 n1(CC(=O)NCC2CC(C)OCC2)ncc2ccccc12 CCC(C)C(=O)C(=O)N1CC(CC(F)C(=O)NCC2(C)CCCC2O)C1 c1(OC)cc2cc[nH]c2cc1-c1cnn(C)c1C(N1CCC2COCC2C1)=O S(=O)(=O)(c1cccc(=NC2CCc3c(F)cccc32)[nH]1)N1CCC(OC)(OC)C1 n1(C(CC)C)ncc(C(=O)NCCc2cnoc2)c1C=Cc1ccc(Br)s1 CCC(C)(O)C(=O)NCCn1cc(C(=O)NC2CC=CCC2)cn1 C(=O)(C1=NOC(c2ccccc2)C1)N1CC(NC(COCCN(C)C)=O)C(O)C1 C1(OCC)CN(C(c2cnc(S)n2C)=O)CC1C.C1(C2CC2)(C=O)CC1.N N1(C(CC)(CC)CC)C(=O)C(CC(=O)NC)SC1=Nc1cccc(CC2CC2)c1 C(C(N=c1ccnc(C2CC2)[nH]1)C1CC1)NC(c1cnc(C(F)(F)F)s1)=O c1(C(N2CC(F)(CNC(C(C)c3ccsc3)=O)C2)=O)cncc2nc[nH]c12 N1(C(COCC)=O)CC2CC(NC(c3c[nH]nc3-c3ccc(Cl)cc3)=O)C1C2 C1(NC(C2N(C(C)C)CCC2)=O)CCN(C(=O)Cc2cnoc2)CC1CO c1(CC)ccc(C(=O)N)cc1C(F)(F)F.C1CN(C(C2CC(O)C2)=O)CC1C C1(NC(C2(CCS(N)(=O)=O)CCC2)=O)COCCN(C(C2CC23CC3)=O)C1 c1(C=O)cc(=O)n(C)cn1.c1(OCC)ccccc1C=O.C12CC(C1)C2.N C1(C)(C(N(CCNC(C2COC(=O)N2C)=O)CC)=O)CC(OC)CN1C c1(CN2C(C(=O)NC(c3ccc(Br)cn3)C)CNCC2)cc(Br)c(F)cc1O c1(C(=O)NC(CNC(c2cn(CCC(C)(C)C)nn2)=O)CO)ccc(CO)cc1 N1(C(C(C)OCC#C)=O)CCOCC1CNC(c1cccc(F)c1)=O Cc1cc2ccc(C(N3CC(N(C(=O)CN4CCCCS4(=O)=O)C)C3)=O)cn2c1 N1(CC(=O)N(C)CC2N(C(COCC#C)=O)CCCC2)CCCCCC1=O c1(C(=O)NCC2(C)COCCN(C(C(C)N(C)C)=O)C2)cnc2c(c1)ncn2C C(=O)(C1CCCn2nccc21)NCC1N(C(c2cc(C#N)no2)=O)CCN(C)C1 c1(C(=O)NCCC(CNC(C(C2CC2)OC)=O)O)cc(F)ccc1C(F)F c1(N(C(=O)CN2CCCC2C2CCOCC2)CCCO)nccc(C(F)(F)F)n1 N1(C(c2nc(C)nc(O)c2)=O)CC(NC(=O)CCCC2CC2C)C2CCCC12 c1(N2C(C(C)C)CN(C(=O)C(C3CCC(=O)N3)C)CC2)ncc2ncn(C)c2n1 c1(C(N(CCN(C(C(CC)NC(C)=O)=O)C)C)=O)c(C)nc2cccnn12 c1(CCC=O)ccccc1C(N)=O.C(C)(C)(C=CC=O)SC.C1CCC1.N c1(CNC(C(=O)NCC(CC=C)c2ccccc2)=O)ccc(Cl)cc1C S(=O)(=O)(c1ccc(=NCc2cc3cc(Cl)ccc3o2)[nH]c1)N1CC(C)(C)SCC1 N1(C(c2ccc(C)nc2O)=O)CCN(C(=O)C(c2ccccc2F)C)C2CCC12 c1(CC(=O)NCC(C)N(C(=O)CC2CCC2)C)c(Br)ccc(F)c1F C1(CNC(C(C)OC)=O)CN(C(c2cccc(-n3ccnc3)c2)=O)CC1(C)C C(=O)(CCS(=O)(=O)c1ccc(F)cc1)N(C(C)CNC(=O)CC(C)C(C)(C)C)C c1(C(=O)NC2CC(C(CO)SC)C2)cc(C#N)ncn1 C1(NC(Cc2ccc(CCC)cc2)=O)CC(C)CN(C(C2C(OCC)C2C)=O)C1 c1(N2C3CN(C(c4ccc(C)o4)=O)C(C3)C2)nc(C(F)(F)F)nc2ccccc12 C1(C(CNC(CSC(C)C)=O)OC(F)F)CCCCC1.C(=O)CC.C(N)=O.N S(=O)(=O)(c1cc2oc(=O)[nH]c2cc1F)N1C(C(=O)Nc2ccccc2)CCC1 C(=O)(CC(F)(F)Cl)NCCNC(C1C(c2ccn(C)c2)C1)=O N1(C(C2(OC)CC2)=O)CC2C(C(=O)NCCCC3(O)CCCOC3)C2C1 c1(OC)ncc(Cl)cc1C(N1CCC(O)(CN(C)C(C2CCCC2)=O)C1)=O.C N1(C(c2c(CCC)nns2)=O)CCCC2CN(C(c3c[nH]c(=N)o3)=O)CCC12 CC1CCCN1CC(=O)N(C(CNC(c1sccc1-n1cnnn1)=O)C1CC1)C C1(NC(=O)Cc2ccc(Cl)s2)CCCCCN(C(C23CC=CC(C2)OC3)=O)C1 Cc1cc(C)n2ncc(C(N3CCC(C(C)Nc4ncccn4)C3)=O)c2n1 c1(C(=O)N)cnc2n1CC(C)CC2.c1(COC)nc(C(=O)NC(C)CO)co1 C1(NC(C(=Cc2cnc[nH]2)C)=O)CCN(C(c2ccc(Br)o2)=O)CC1F N1(C(CNS(N(C)C)(=O)=O)=O)CC2(CCCC2NC(=O)CCc2ccon2)C1 C(=O)CS(=O)(=O)CC(C)C.N1(C(C=C(C)C(F)F)=O)CC(C)OC(C)(C)C1.N C1(CNC(=O)NC2(COC)CC2)CCCN1C(=O)OC CCCCCC(C)CC(=O)NCCNC(=O)C(CS(C)(=O)=O)c1ccccc1 N1(C(c2ccc(C(N)=O)[nH]2)=O)CCOCC(CNC(C2C=CC=CC=C2)=O)C1 c1(CNC2CC(C(=O)Nc3n(C)ncc3Cl)C2)cc(Cl)ncc1Cl CC(CCCN=c1[nH]c(C2CC2)nc2c1CSC2)NC(C1CC2CCC1O2)=O C12(NC(CCCCC)=O)CCOC(CNC(=O)CC3CCCCC3O)(C1)C2 n1(CC)nc(C(=O)NC2(C)CCN(C(C3(C4CCCO4)CCC3)=O)C2)ccc1=O N1(Cc2n(C)ncc2Cl)CCOC(Cc2ccccc2)CC1 c1(C(=O)NC2CCN(CCC)C2)coc2c1CN(C(C1CC3CC1CC3=O)=O)C2 c1(C(N2CC(C)CC(NC(c3c(C(C)C)con3)=O)C2)=O)cnc2c(c1)COC2 C(N=c1[nH]c2ccc(F)cc2o1)c1ccc(CNC(c2ccc(O)nn2)=O)cc1 N1(C(c2c(C(C)C)cco2)=O)CC2(CC(NC(=O)C(C)CN(C)C)CO2)C1 C(CCN=c1[nH]c(=NCC2CS(=O)(=O)CCO2)c2ccc(C)cc2[nH]1)NCC C1(NC(C2CC3(CC3)C2)=O)CC2CN(C(c3ccc(O)cc3F)=O)CC12 C#Cc1cncc(C(N2C(C(N3CC(C)(C(=O)OC)C3)=O)CCC23CC3)=O)c1 C1(C(=O)NC2(CNC(Cc3ccn(CC)n3)=O)CC2)CCC(OC)CC1 CCC(CN(C(=O)COC1CCN(C(c2ccn(C)n2)=O)C1)C1CC1)CC c1(OC)ccc(Br)c(NC(C2CCC=CC2)=O)c1.c1(C=O)ccc2c(c1)CC2.N N1(C(CN(C)C2CC2)=O)CCCCC(NC(=O)CC2CCCC2(F)F)C1 c1(C(N2CCC(C(C)(C)NC(c3c(C)onc3)=O)C2)=O)ccc2c[nH]nc2n1 C1(F)CCN(C(c2csc(CC(C)C)n2)=O)C1.c1(OCC)cc(C(=O)N)on1 N1(C(C(C)CO)=O)CCCC(C2CN(C(C34C5CC(CC35)C4(F)F)=O)C2)C1 C(=O)(CC(C)(C)C)NCCC(C)C.C1(C=O)CC(=O)N(CCN2CCCC2)C1 C1(C(=O)NCC2CCCC2CF)(NC(CSCC)=O)CC(=O)C1 CCCC(C=O)NC(N)=O.C1C2CC1N(C(C1CN(S(C)(=O)=O)C1)=O)C2.N N1(C(c2c(C)onc2C2CC2)=O)CC(Nc2ncnc(Cl)c2F)C(C)(C)C1 CCC(C)(CC)C(=O)N1CCC(NC(C2(C)CCCC2C)=O)C(C)C1 C(CC(C(=O)NC1CCCC1)NCCN(C)C(C1CCCC1)=O)SC.N(C)C c1(C(=O)NCC(CCNC(C=C(C)C2CC2)=O)O)cnn2ccc(C)nc12 C#Cc1cc(C(=O)NCC(O)CCNC(=O)CN2CCC(OC)C2)ccc1C N1(C(c2ccc(C)s2)=O)CCN(C(c2ccnnc2O)=O)C(CC(F)(F)F)C1 C(CC(=O)N1CC(NC(=O)CN2CCS(=O)CC2)C(F)C1)(C(C)C)OCC c1(C(=O)NC2C(C)CN(C(c3cnsc3)=O)C2)ccc2c(c1)CN(C)C2 N1(C(c2ccn(CCC)n2)=O)CCC(O)(C(C)NC(=O)CN2CC(C)C2)C1 c1(C(=O)OC)nn2cccnc2c1NC(c1ccc(O)cc1)c1cnn(C)c1 Cc1cc2ccccc2nc1C(=O)NC1CC(C)CN(C(c2occc2Cl)=O)C1 N1(C(CN2CCN(C)CC2)=O)CCC(C2CCN(C(C3CC4(CCC4)C3)=O)C2)C1 c1(C(=O)NC2C(CNC(C=C3CCN(C)C3)=O)CC2)nnc(S)n1C C(CCC)(C(O)C(=O)N1CCC(N(C)CC)C1)NC(C(CC=C)CC)=O c1(C(=O)NCCN2CC(COC)C2)oc(SC)cc1C C(=O)(C(C)C(C)(C)C)N1CC(COC)(CNC(C2C3CCCOC23)=O)C1 N1(C(C(c2ccc(Cl)c(Cl)c2)C)=O)CC2CC1CC2.C1(C=O)CC(=C2CC2)C1.N c1(C(=O)NC2(C)CCN(C(CCSCCC)=O)C2)cc(C)cc(Br)c1O N(C(=NCCC(C)C)N1CCC(OCc2ccoc2)CC1)C(CC)C Cc1cccc(=O)n1CC(C)(O)C(=O)NCCCNC(=O)CC1CCOC1=O C(C(C)(C)C(C)(C)C)NC(CCC1N(C(Cc2c(C)con2)=O)CCC1)=O CCCCC(C)CCC(=O)NC1CCN(C(=O)C2=C(C)OCCC2)C1C(C)(C)C C1(OC)CN(C(c2cnc(C(C)C)n2C)=O)CC1.c1(CC(=O)N)cn(C)nc1C N1(C(c2c(C)n(C(C)C)nc2)=O)CC(C)CC1(C)C.C1(CC=O)CNC(=O)C1 C(C(C)(C)CC)NC(C=CC=CCC)=O.C(=O)(CCC(=O)N1CCOCC1)N Cc1ccnnc1C(=O)NCC1CCN1C(=O)CCCc1cccnc1 c1(SCC)ccc(C(=O)O)cn1.C1(=O)C(C(C)C)N1 n1(CC=O)cc(S(C)(=O)=O)cn1.C1(NC(CC(=O)N(C)C)=O)CCCCC1.C c1(OC)cc(Br)sc1NC(C1CCN(C(=O)COCC2CCOC2)C1)=O c1(C(N2CC(OC)(CNC(=O)CC(C)SC)C2)=O)nc(Cl)ccc1Cl CCC(CC(=O)NC(c1nocc1C(=O)NC1CCSCC1)C)OC C#CCCCOCC(=O)N(C(C)CNC(=O)CC1(C(=O)O)COC1)C Cc1ncc(C(=O)NC23CCN(C(C4(O)CC4)=O)CC2C3)c2c1OC(C)(C)OC2 Cc1ccc(NC(=O)C(=O)NC2CC2)cc1.c1(C=O)cnn(CCC#N)c1C.N C(CCC1CC1)(C(=O)N(C1CC2CC2C1)C)NC(C(CC)SC)=O c1(CC)c(C(N2CCCCC2)C(=O)NC(C)C)cn[nH]1.S(=O)(=O)(C1CC1)N c1(C(=O)NC(CNC(c2cc(OC)no2)=O)C)cccc(C(C)C)c1F N1(C(=O)CCC(F)F)CC23CCCC2(C1)CN(C(=O)COc1ccc(F)cc1)C3 CC(C)CC(C)(C)C(=O)N(CC(C)NC(C1CCCCC1)=O)C c1(C(N(CC(=O)NCc2cnc(CC)o2)C(C)C)=O)ncc(F)cc1N c1(C(N(C2CN(C(CC3(COC)CC3)=O)C2)C)=O)cc(O)cc(F)c1F c1(C(=O)NC(CC(C)C)CNC(=O)CC2=CCOCC2)ccc2c(c1)CCCC2 C1(NC(=O)Cc2ccc(F)cc2)CN(C(c2cc(Cl)ncc2F)=O)CC12CC2 C(=O)(C1CCCc2sc(NC(=O)Nc3ccc(Cl)c(C(=O)OC)c3)nc21)NC c1(C(N2CCCC(C(N)=O)C2)=O)cc2c([nH]1)CCCC2.C(C(=O)N)(C(C)C)SC c1(C(=O)NC(C2CCOC2)CNC(=O)COc2cccnc2)cnn2c1CCC2 C(=O)(C(CNC(=O)C(O)CC1CCCC1)CC(C)C)NC(CCCCC)C C1(OCC)CN(C(=O)C2=CCCC2)CC1CNC(c1cc(Cl)c[nH]1)=O c1(C(=O)OC)ccc(Br)nc1NC(C)C(C)n1cncn1 c1(C(N(C(CNC(C2CSCCS2)=O)Cc2ccccc2)C)=O)c[nH]c(Br)c1 c1(C(=O)NC(c2cnn(C3CCCC3)c2)CC)ccc(C(C)C(F)(F)F)cc1 c1(CN2CCC(C(=O)NC3CC(C)(C)C3)C2)ccc(N2CCCC2)nc1 c1ccccc1.C(C)(C(=O)N1CCC1CNC(=O)CCSCCCC)=C(C)C CC1CCC(CNC(=O)CCc2ccc(Cl)cc2)N(C(=O)COC2CC2)C1 C1(C(=O)NCC2(O)CCN(C(C(CCN(C)C)O)=O)CC2)CCc2nncn2C1 N1(C(c2nc(C(C)(C)C)[nH]n2)=O)CC2C(CNC(=O)C#CC3CC3)C2C1 N1(C(CC=CC=C)=O)CC2CC1(C(N1CCC(CC3CC3)CC1)=O)C2 C(C(CNC(=O)C=CCN(C(=O)CCC=CC(C)C)C)C(C)C)OC c1(C(=O)NC2CC(NC(=O)Cc3cc[nH]c3)C2)cnoc1C(F)(F)F c1(C(N2CC[Si](C)(C)CC2)C=O)cc(F)c(F)c(Cl)c1F.C(C)N(CC)CC c1(NC2CCN(C(c3cc(C)nc(Cl)c3)=O)CC2F)ncnc2cc[nH]c12 N1(C(c2scc(C)n2)=O)CCC2(CC(C(=O)Nc3ccnc(C(C)C)c3)=NO2)C1 c1(C(=O)NCC(CC(C)C)NC(CC(C)OC)=O)n[nH]c2ccc(C)cc12 CN1C(=O)CCCC1C(=O)N.C1(C)CCCN(C(=O)Cc2cc(C3CC3)no2)C1 C(C)(CSC)(C(=O)NCc1ccn(C)n1)NC(Cn1ncc(CC)c1)=O C1(NC(C(=O)OCC)=O)CC=CCC1C(=O)NCCc1cccnc1O C(=O)(CC(CC(=O)NCC)C(F)(F)F)OCC(=O)OCC.c1ccccc1 C1(CNC(c2cn(C)[nH]c2=N)=O)COCCN(C(C2(C)CCC(=O)N2)=O)C1 c1(C(F)(F)F)nc(-c2cc(CN3CCCC3Cn3cncn3)cs2)no1 CC(C(=O)N(C)CC1CCN(C(c2ccc(N)c(O)c2)=O)C1)S(C)(=O)=O CC1CCN(C(=O)C(CC(F)F)NC(c2ccc3cc[nH]c3n2)=O)CC1(C)C c1(CC)ccc(NC(C2CCN(C(=O)N)C2)=O)nc1.c1cscc1C(F)(F)F C1(CC)CN(C(c2sccc2OC)=O)CCC1NC(C1(C#N)CC1(C)C)=O C(c1nc2ccccc2s1)=CC(N1CC(CNC(C(CC)F)=O)C(C)(C)C1)=O C(CNC(c1cnc(C(C)C)nc1C)=O)(C(C)C(C)C)NC(CCCCSC)=O N1(C(C=CC(=O)NC2CCC(O)C2)=O)CC(C(=O)NC2CC2)CC(F)C1 C1(NC(c2c(C)nn(C(C)C)c2)=O)CN(C(C2CC3(CCC3)C2)=O)CCC1(C)C CN1CCN(CC(=O)NCCSCC(=O)NCC2CCCOC2)CC1 Cc1cc(OC(C)C(=O)NC2CC3CC2C2CC32)ccc1-n1cccc1 N1(C(C=CC)=O)CC2(CCN(C(c3cc(C=O)ccn3)=O)CC2)C1.C(C)(C)C c1(OC)ccc2c(c1)C(Nc1ccc3c(I)n[nH]c3c1)CC2 Cc1oc(S(N)(=O)=O)cc1C(N1CCCC1)=O.C1(C(N(C)C)=O)CC12CCC2 N1(C(c2c(CC)cco2)=O)CCN(C(=O)CCN2CCCC2=O)CC(CO)C1 N1(C(c2ccns2)=O)CCC2(CCN(C(C34CCC3CC4)=O)C2)C1 N1(C(C(CN(C)C)NC(=O)CCC2(C)N=N2)=O)CC([N+](=O)[O-])C1 c1(C(=O)N)cn2cnnc2cn1.C(CC(=O)N1CCCC1C)(C(N)=O)NC(C)=O N1(C(c2ccc(OCC)nc2)=O)CCC2C(NC(=O)CCSC)C2CC1 c1(CC)ccc(C(=O)NCCCCC(C)NC(c2c(C)nn(C)c2Cl)=O)c(C)n1 c1(N2CCCC(CNC(C(CC(C)(C)C)O)=O)C2)cc(S(C)(=O)=O)ncn1 C1(C(=O)NCCC(C)N(C(=O)CP(C)(C)=O)C)CCc2nn[nH]c2C1 c1(C(N(CCCN(C(C=CC)=O)C)C)=O)oc2c(c1C)C(=O)CC(C)(C)C2 C(=O)(C(CCC1CCC1)NC(=O)Cn1cnnc1)N(C)Cc1nc(=N)[nH][nH]1 CCCC(CC)C(=O)NC1(CCC)CCCN(C(c2nn(C)cc2N)=O)C1 c1(C(N2CC(CNC(C(CC)F)=O)C3(C2)CCC3)=O)c(C)cnc2ccccc12 CCCC(C(O)C(=O)NCCCC1CCOC1=O)NC(=O)CC1NC(=O)NC1=O c1(C(N2CC(C)(CNC(CCSCC)=O)OCC2)=O)cccc2ccnn12 C1(C(=O)OC)CC(N(C)C)CN(C(C2CCN(C(C)C)CC2)=O)C1 C(CC(C)(C)C)(C(=O)N(CC(N1CC(CC(F)(F)F)C1)=O)C(C)C)OC c1(NC(c2ncc(C(F)(F)F)[nH]2)=O)cccc2ncccc12.C12CCCC1NC2 N1(C(C2(NC(=O)C(O)C3CCCC3)CC2)=O)CC2CCC2C1 C(C(=O)N1CCCc2nncn21)N(C(=O)C(C)CCCC(C)C)CC N1(C(C2CCCC(C)C2)=O)CCN(Cc2ccc(F)cc2)C(C)C1 N1(C2CCCN(C(CC=CCC)=O)C2)CCN(C(C2CCCOCC2)=O)CC1=O c1(C(N(CCOC)C2CC2)=O)cn(CCNC(=O)CC(C)O)nn1 C1(NC(Cc2cn(CC)nn2)=O)CN(C(c2ccccc2F)=O)C2(CCOC2)C1 CCC(CO)C(=O)N1CC(NC(c2cccc(C(F)F)c2)=O)C(C)C1 c1(NCC2C(C(=O)OCC)C2(C)C)ccccc1-c1ccc(C)cc1 c1(C(=O)NC(C(C)NC(=O)C=CCO)C)cccc2cccc(Cl)c12 [SH](=O)(=O)CC=O.C1(CC(=O)N(CC)CC)CCCC1O.CC(=O)N.CCO CS(=O)(=O)C1CCN(C(C2CC(O)CN2Cc2ccc(C(N)=O)cc2)=O)CC1 C1(CC(=O)NCC2(CC)CCCC2)CCN(C(=O)C(=O)CC(C)C)C1(C)C c1(N2CCC(NC(C(c3ccccc3)NC(C)=O)=O)C2)ncnc2sc(Br)cc12 N1(C(CC(CC)C)=O)CCC2CN(C(=O)CCc3cn(C)nc3C)CCC12 C1(NC(=O)Cc2cnoc2)C2CC(NC(C3CC3C3CCC3)=O)CC12 C#CCC(C(=O)N1CC2C(CC(N3CC(c4nn[nH]n4)C3)=O)C2C1)C1CC1 Cc1cn2ccc(C(=O)NCC(C)(CO)NC(c3cc(Br)co3)=O)cc2n1 c1(C(=O)NC2CN(C(C3CCCC(=O)O3)=O)CC2O)ccc2c(n1)OCC(=O)N2 C1(CNC(COCC(=C)C)=O)CN(C(=O)Cc2ccc(F)nc2)CCCO1 N1(C(CCCC=CC)=O)CC2COCC2(C(N2CCC(c3ccon3)C2)=O)C1 c1(OC)ccc(C(=O)NCC(C)(CO)NC(=O)C)cc1[N+](=O)[O-].C(C)=O.O C(=O)(CC(F)(F)C(F)F)NC(C)CN(C)C(C1(C)CCC(=O)N1)=O C=C(C)C1CN(C(C2CC(CC)CCN2C(=O)CC2CC(OCC)C2)=O)CCO1 c1(C(=O)NC2C(CNC(C(C)SC)=O)CC2)ncnc2sccc12 N1(C(c2cnc(C(C)(C)C)o2)=O)CCN(C(c2ccncc2Cl)=O)C2CC12 c1(N(CC(CNC(c2c(CC)ncnc2)=O)C)C)ncnc2sc(C)nc12 c1(SCCOCC)ccc(C(=O)O)cc1C.C12CCN(CC1)CC(=O)NC2 N1(C(C=C(C)C(C)(C)C)=O)CCC(C2CCCN2C(C2CC(O)C2)=O)CC1 n1(CC)nncc1CN(C)C(=O)NCCN1CCCC1 c1cccc(S(C)(=O)=O)n1.C1(C(=O)N)CC12CCNC2.S(=O)(=O)(CC)N(C)C c1(NC(c2n(CC)nnn2)C2CN(C(C34CC(CO3)C4)=O)C2)ccccc1Cl CC1=CCC(C)(C(N2CCOC(CCNC(=O)Cc3ncccc3C)C2)=O)CC1 C=CC(C)(O)CC(=O)N(C(C)CNC(=O)C(CC)Oc1cc(Cl)cc(Cl)c1)C CC1CN(C(=O)CN(c2ccccc2)C)CCC1N(C)C(c1c[nH]nc1F)=O CC1(C)CC2(CCN(C(=O)CCc3ccc4c(c3)OCCO4)C2)CO1 c1(C(N2CC(F)CC(NC(c3cncc(Cl)c3Cl)=O)C2)=O)cn2c(n1)COCC2 C(=O)(C(C)CC(=O)N1CCOCC(C)C1)OC.c1(C=O)coc(C(C)(C)C)n1.N Cc1ccc(Cl)cc1C(N1CCC(CCNC(=O)C(C)C(C)(F)F)C1)=O Cc1nn[nH]c1C(=O)NC(c1ccccc1)C(=O)NCC1CCCO1 C(=O)(C(C)(C)CC(F)F)N1CCC(NC(CCc2nnc(C)n2C)=O)C(C(N)=O)C1 c1(CC(=O)NCc2nnn(C(C)(C)C)n2)ccccc1F CCC(CCC(=O)NCC1(COC)CCCCC1)NC(=O)CNC=O N1(C(C2C(NC(Cc3c(C)cnn3C)=O)CCO2)=O)CCC(C)C(O)C1 c1(OCC(N2CCCCC(NC(C(C)(C)CO)=O)C2)=O)ccc(C#N)cc1Cl c1(CC)ccc(CCN(CC(C)N2CCC2)C(=O)Cc2csc(C)c2)o1 N1(C(c2cccc(CCC#N)c2)=O)CCCCC(NC(=O)C(O)CC(N)=O)C1 CCCC(C(=O)NC1CN(C(=O)Cc2ccc(C)o2)CC12CCC2)S(N)(=O)=O C12(C(N3CCC4(CN(C(C5(C)CCCCC5)=O)C4)C3)=O)CCC(C1)S(=O)(=O)CC2 c1(CC)ccc([N+](=O)[O-])cn1.C1CC(C)(C)CN1 Cc1ccc(CCC(=O)N(C(CNC(=O)CC2(O)CCOC2)C2CC2)C)s1 C12(NC(c3c(OC)c[nH]n3)=O)CCC(C1)N(C(=O)Cc1cccc(C#N)c1)C2 c1(COC)ncc(C(=O)NCCCO)c(=N)[nH]1.c1(C=O)c(C)[nH]c(C)c1C.N CC(C)(C)CCC(=O)NCCC1(C)CCN(C(=O)CCCc2cnn[nH]2)C1 C1(C(=O)OC)CCCC(NC(c2sc(Br)nc2Br)=O)CC1 C12(CC(=O)NCCCCNC(c3cnc(C)o3)=O)CCCCC1C2(F)F c1(N2C(C(=O)Nc3ccc(C)cn3)CCC2C)ncnc(-c2ccccc2)c1C c1(C(=O)NCCN(C(C(COC)OC)=O)CC2CC2)cc(C#N)cs1 N1(C(COCCCCCCCC)=O)CCC2(CCCN2C(C2CC2(C)C)=O)C1 C1(NC(c2cn(CCCC)nn2)=O)CCCN(C(=O)Cn2cnc(=N)[nH]2)CC1F N#Cc1ccc(-c2cn(C3CN(C(C4CC(OC(F)F)C4)=O)CC3O)nn2)nc1 N1(C(c2c(C)nc(O)[nH]2)=O)CCC(C)N(C(=O)C2=CS(=O)CCC2)CC1 N1(C(C(CC(C)C)F)=O)CCOC2(CCCN(C(=O)CN3C(=O)CCC3=O)C2)C1 c1(C(=O)NCC2(F)CCN(C(C(C)O)=O)CC2)cc2cccnn2n1 N1(CC(C)CC2CCNCC2)CCC2(CC1)NC(=O)CO2 N1(C(C(N2CCSCC2)C)=O)CCCC2(C1)CN(C(C1(C#N)CCCCC1)=O)C2 N1(Cc2[nH]c(=N)sc2)CCCC(N(CC(c2ccccc2)O)C(C2CCC2)=O)C1 C(CCCC(C)NC(=O)C=CCOCC)NC(c1ccc(CC)s1)=O.O C1(CC)CN(C(=O)CCCC2CC2C)CC1C(=O)NCC(F)(F)CO C1(NC(CC(=C)Br)=O)CCCN(C(=O)CCC2CC2)C1C N1(C(c2cnc(C(C)C)s2)=O)CCCC(C)C1CNC(c1ccc(=N)[nH]n1)=O c1(CCC(=O)NCCCCCN(C)C(C2(C#N)CC2)=O)cccc2cnccc12 c1(CC)c(C(=O)N(CCCNC(=O)C(C2CC2)SC)CCO)nn[nH]1.C C(CC(C(=O)NCC1(F)CC1)NC(=O)COC(C)C)=CC C1(C(=O)NC(C(=O)OCC)CC)(CF)CCN(C(C2CC2Cl)=O)C1 N1(C(Cc2ncc(CC)[nH]2)=O)CC(NC(=O)Cc2cccc(O)c2)CC12CCC2 c1(C(=O)NCC(C)(C)CNC(=O)CC(=O)N2CCOCC2)occ2c1CCOC2 N1(C(C(CC)C)=O)CCN(C(=O)C2=NN(C)C(=O)CC2)CC12CCC2 c1(NC(C2(N)CCC(C)(C)C2)=O)ccc2ccccc2c1 S(=O)(=O)(c1ccc(F)cc1F)N1CCC(CC(=O)Nc2c(C)cc(F)c(F)c2)C1 C=CC(C)(CC)C(=O)NCCOCC.c1(C=O)cnc(CCC(F)(F)F)s1.N c1(C(N2CCC(CCNC(C(C3CCOC3)OC)=O)CC2)=O)cc(=O)cc(Cl)[nH]1 C1(NC(C(CCC)O)=O)CN(C(C2CC(OC)C2)=O)C2(CCCCC2)C1 C1(C(N2CC(NC(c3c(C)ncs3)=O)C2)=O)COc2c(OC(F)(F)F)cccc2C1 c1(C(=O)OC)cccc(NC23CC2CN(C(=O)C(N2CCC(OC)C2)=O)C3)c1 N1(C(C2C(C)C2)=O)CCCCCC(NC(c2cc(=N)[nH]c(Cl)n2)=O)C1 C(=O)(CC(O)CC(C)(C)C)NC(C(=O)NCC(C)N(C)C1CC1)CO C1(C(F)(F)F)(OC)CC2(COCCN2C(c2ccc(N(C)C)cn2)=O)C1 CC1OCCCC1C(=O)OC(c1cccc(C(F)(F)F)c1)C1CCOC1 c1(OC)cc(C(=O)NCC(C)(C2CC2)NC(=O)C(C)OC)c(F)cc1Br Cc1ccc2c(CC(=O)NCC3CCN(C(=O)CC4CCC(=O)N4)C3)c[nH]c2c1 CC(C)CC(C)OCCC(N1CC(C)(CNC(=O)CC2CC2(Cl)Cl)C1)=O C12(NC(CC=CC(C)(C)C)=O)CC(C)(C1)OC21CCC1.C(=O)CCCC#N.N c1(CC)ccc(O)c(C(=O)NC(C)CN(C)C(C2COCCC2(F)F)=O)c1 C1(C=O)CC2CCC(C1)C2.c1(C(=O)NCCCC)cc(CS(C)(=O)=O)on1.N C1(NC(c2c(CC)onc2)=O)CCCC12CN(C(C1(C#N)CCCOC1)=O)C2 C(CCC(O)C(=O)N(C1(CO)CC1)C)NC(c1c(C)nsc1C)=O N1(C(C(CCCNC(CS(CCOC)(=O)=O)=O)O)=O)CCOC2(CCCC2)C1 Cc1ccc(C(=O)C(=O)N2CCC2C2CCOCC2)cc1.n12cc(nn1)C2 C1(CN2C(O)CC2C(F)(F)COC2CCCCCCC2)CCOC2(CCCC2)C1 C(=O)(C1CCc2c[nH]nc21)NC(C(=O)N1C(CC)COCC1)CCC(C)C N1(c2nccc(OC)n2)CCCC2(NC(c3cscn3)=O)CCCC12 N1(C(C(CC=CCC)C)=O)CC(CNC(=O)C)C(C)(C)C1.c1cccnc1.N C(=O)(C#CC1(C)CCCO1)N(C1CCN(C(=O)C(C)C2CCC2)CC1)CCC CCC(CC)CC(F)C(=O)NC1(C)CCN(C(c2nc3cccnc3s2)=O)C1 c1(C(N2CCC(CCNC(C=CCCC)=O)CC2)=O)cc(N)c(Br)c(F)c1 C(CC1CCCC1)(C(=O)NCC1CC1CO)NC(=O)Cc1cncs1 Cc1cccc(C(=O)NC2CCC(NC(c3cc(Cl)ccc3F)=O)C2)c1[N+](=O)[O-] CCCS(=O)(=O)CC(=O)N1CCCC(NC(=O)Cn2ccc(C(F)(F)F)n2)C1C C1(NC(c2c(OCC=C)cccc2)=O)COC2(C1)CN(C)C2.C1CC2CCC1O2 c1(CCC)n[nH]c(=NC2C(C)CN(C(=O)CC3CCS(=O)(=O)C3)CC2C)s1 c1(C(N(CC(C)N(C(c2cc(OCC)no2)=O)C)C)=O)cnn(C)c1Cl CC1CC(NC(c2cc(Cl)c[nH]2)=O)CN(C(=O)C=CCN2CCC2)C1 CCC(c1ccccc1)=CC(=O)NCC(C)(C1CC1)NC(=O)CC(F)(F)F C(C(C)(C)CCS(C)(=O)=O)NC(Cc1c(C(c2nnnn2C)OC)con1)=O c1(Cn2c(-c3cc(C)sc3Br)nc(-c3cccc(Cl)n3)n2)ccc(C)c(C)c1 C1(CNC(C2(F)C(C)OCC2)=O)CC2(CC2)CN1C(=O)CC1CCC2CC12 c1(CN2CC3(C(C(N4C(C(=O)OC)CCC4C)=O)C3)C2)ccc(F)nc1F C1(NC(C(C)SC)=O)CCN(C(=O)CNc2ccc(C)cc2F)C12CCC2 N1(C(c2cc(C)sn2)=O)CCN(C(C2(C)CCC2)=O)CCC1C c1(CN2C(C(=O)NCCc3ccc(F)cc3)COCC2)cc(F)c(Cl)c(F)c1 C(=O)(CCCCCn1cc(-c2ccccn2)nn1)N(C)CC1CC1(C)C C(=O)(C(C)(F)C(C)(C)F)N(C)CC1(NC(C(C=C)C)=O)CC1 C1(=CC)CCN(C(=O)CC2CCCS2(=O)=O)CC1.c1(C=O)sccc1CCC C1(O)(Cn2cc(CCCSC)nn2)CCN(C(=O)CCc2nnc(S)n2C)CC1 CC1CN(C(=O)Cc2csc(S)n2)CCN1C(C1(C#N)CCCO1)=O C12(CN3CC(O)(CC)C3)CCCC(CO1)C2.c1(C2(CC=O)CC2)ccccc1 CC(C(C)C(=O)Nc1ccc(CCO)cc1)NC(=O)C=Cc1nccs1 CCC(CC)C(=O)NCC(=O)NCCC1CCC(NC(c2ccon2)=O)C1 C1(C(=O)NC2CCC(NC(CS(C(C)C)(=O)=O)=O)C2)CCc2nnc(O)cc2C1 C1(C(C)NC(=O)CN(S(C)(=O)=O)C)CCCCN1C(C1CCCCC1)=O C(N=c1[nH]c(N2CCC(CC(N)=O)C2)nc2c1COC2)C1(OCC)CCCSC1 C#CCC(CC(=O)Nc1cnc(CC)nc1)Nc1sccc1C C1(C(=O)NCC2N(C(CCCOC)=O)CC(OC)C2)CCC2(CCC2)CO1 N1(C(COC2CN(C(COCC(=O)NC)=O)C2)=O)CCC12CCC(O)CC2 C1(CNC(C2N(N=O)CCC2)=O)CC2(CCC2)C1.C1(C=O)CCC1.C1CC1 c1(C(N2C(Cc3cccc(N(C)C)c3)CCC2)=O)cc(Cl)c(Br)cc1Cl CC(CC(=O)N1CCC1C(N1CC(Cc2ccoc2)C1)=O)C(F)(F)F C1(NC(C(n2cc(Cl)cn2)C)=O)CN(C(=O)CC2CCC(F)(F)C2)CC2CC12 CCCC(C(=O)NCCC#CCO)NC(=O)CCC(N)=O CCCCC(O)CC(=O)N1CCOC(CCNC(=O)CN2CSCC2=O)C1 c1(OC)cc(C(N2CC(NC(=O)Cn3ccnn3)C(O)C2)=O)ccn1.N(C)C c1(OCCC(=O)N(C2(c3nccs3)CCCC2)CCCOC)ccccc1F c1(C(N2CCCCC(CNC(C3CSC3)=O)C2)=O)cccc2cnnc(O)c12 c1(CN2CCCC(C(C)NC(C3CCC(F)(F)C3)=O)C2)cc2cc(Br)ccc2s1 C(CN=c1[nH]c2c(c(=NC(C)CCN(C)C)[nH]1)COCC2)c1cc(C)cc(C)c1 CC1CN(C(c2cc(Cl)sc2Cl)=O)CCC1CNCC1CC(F)(F)C1 c1(C(=O)NC(CNC(C=NOC)=O)CC(C)C)cc2n(n1)CCCCO2 c1(C(N2C3(C(=O)NC4(CC#C)CCOCC4)CC3CC2)=O)cc(C)c(C)nn1 C1(CC=O)CCC(=O)NC1.CC(C)(CNC(C1CC1(Cl)Cl)=O)OCC.N c1(C(=O)NCCC2CCCN(C(C(C)OCC)=O)C2)cc2cccnc2s1 C1(C(=O)NC(CC)CCOC)CN(C(c2cc[nH]n2)=O)CC12CCC2 c1(C(N(C2CCN(C(c3ccc(OC)s3)=O)C2)C)=O)cc(C#N)ccc1C N1(C(CN2CCC(C)(CC)C2)=O)CCN(C(=O)CC23COC(CF)(C2)C3)CC1C C1(OCCCNC(CC=C=C)=O)COC2(C1)CN(C(C1CCC(NC)CC1)=O)C2 C(=O)(CC1OCc2ccccc21)NC(CC)(C)CNC(c1csc(C(C)C)n1)=O c1(C(=O)NC2C(C)(CNC(C(C(CC)O)C)=O)CCC2)cc2sccc2n1C N#CC1(C(N2CC3CC2C3C(=O)Nc2cccc(O)c2)=O)CCCC1 C1(CCC(c2nnnn2C2COC2)NCC(C)CCO)CCC(F)(F)CC1 C(CCCC(=O)NC(C)C(C)C)N(C(C(C)OCC)=O)C N1(C(C2CC(C)NC(=O)C2)=O)CC=C(C(C)(C)C(=O)NC2CCC2(C)C)C1 C1(CC)OCCC1C(=O)NC(c1cccnc1)C(=O)NC(COC)CCO c1(CNC(CSC)=O)cccc(SC)c1.C1(=O)C(C(C)C)N1C c1(-c2onc(C3(NC4CCC(OC)CC4)CCNCC3)n2)cc(Br)cc(Br)c1 Cc1nc2ncnn2cc1C(=O)N(CC(C)(C)CNC(=O)CCC(C)(F)F)C C1(OC)CCn2cc(C(N3CCC(NC(=O)CCSCC(N)=O)C3)=O)nc2C1 CC1CCN(C(c2cncnc2)=O)C(CNC(C2CC2c2ccsc2)=O)C1 c1(CCC)ccc(C(=O)NCCCO)cc1[N+](=O)[O-].C1(C=O)C(C)(C)C1(F)F.N C1(NC(c2c(CNC(c3ccc(OC)s3)=O)noc2)=O)CCCC(C)(C)C1 C(=O)C(C)CN1CCOCC1.N1(C(C2C(C=O)C2)=O)CC(CCC)C1.CC.O c1(NC2CC(NC(c3cc(C4CC4)on3)=O)C23CCC3)ncc([N+](=O)[O-])cc1F C(CCN(C)C(C1CCCCN1c1ncccn1)=O)(C(C)C)NC(CSSC)=O C1CCCC(C2CC2)C1.n1(CC#C)cnnc1C(=O)N(C(C)C(=O)N)C1CC1 C=C(C)C(CC(=O)N1CCC(C2OCCO2)C1)OCC C1(C(N2CCCCC(NC(c3ccn(C)c(=O)c3)=O)C2)=O)CC2C=CCC(C1)C2 C1(C(N(CCC)CC)=O)CCS(=O)(=O)C(C)C1.c1(C=O)cnc(C)nc1C.N c1(C(N2CC(O)(CN(C(c3snc(C)c3N)=O)C)C2)=O)ccc([N+](=O)[O-])cc1 C#Cc1ccc(CC(=O)NC2(C(=O)NCCCC(=O)OCC)CC2(C)C)cc1 C1(C(C)C)CN(C(=O)C(N2CCOC2=O)C)CC1C(=O)N.C1CC[Si](C)(C)C1.C O=C(CCCCCO)NNc1ccc(-c2ccccc2)cn1 C(CO)(C(C)(C)CO)NC(CC1C(C)CN(C(C2(C)COC(=O)N2)=O)C1)=O c1(C(CC)(C)C)ccc(OCc2cc(C(F)(F)F)on2)cc1 c1(C(=O)NC2C(NC(CCn3c(C)cc(C)n3)=O)CC2)noc2ccccc12 C1(C(N2CC(NC(C3(CC#C)CC3)=O)C2)=O)CC(C2CC2)C1 C(=O)(C(F)CCC(C)(C)C)N1CC(C(N2CCC(CN=[N+]=[N-])C2)=O)(CC)C1 C(=O)(C#CC1CCCC1)N1CCN(C(C2N(C)C(=O)OC2)=O)CC1CF C(C1=COCCC1)(c1nnnn1C1CCC1)NC(c1cccc(C)c1)C1CCCC1 N1(C(C2C(C)OCCC2)=O)CCCN(C(C2C3CCCCC23)=O)CCC1 CCCCC(CO)NC(C1CC(F)CN1C(C1CCC(F)(F)C1)=O)=O CCC(C)(CCNC(=O)CC1CCOC1=O)NC(=O)CCc1ccc(C)o1 n1(CCCC)nc(C(=O)NCC(O)CNC(=O)CC2(CO)CC2)ccc1=O CCN(OC)C(=O)C1C=CCN1C(C1CCC1(F)F)=O c1ccc(C(C)(C)C(=O)N(CC(O)CN(C)C(c2cn(C)nn2)=O)C)cc1.CC O=C(C1=CC2CCCC12)N1CCN(C(c2ccc3c(c2)OCO3)=O)CC1 CC(CC1CC1)N=c1[nH]c(=NCC2CC2(C)C)[nH]c2c1CSC2 C(CC(C(=O)N(CC=O)C)NC(C1CCN(C)C1CC)=O)=CC.C1CC1.N c1(C(N2CCC3(CC3)C2)=O)c[nH]c2cccc(F)c12.O=C1NC(C(=O)NC)CO1 CC(C)(C)C(O)C(=O)N1CC2CN(C(=O)Cc3ccccc3F)CC12 C1(C(=O)NCCOCCCC)(CNC(c2nc(Cl)cs2)=O)CCCO1 CCCCC(O)C(C)C(=O)NC1COCCC1C(=O)NCCOCCOCC C1(CC=O)CCCC2(CC2)C1.c1(C(N2CCC(C)(C)C2)=O)cc(O)nc(Cl)c1.N C1(NC(C(CSC)OC)=O)C2CN(C(=O)CCNC(C)=O)CC12 N1(CC(COCC)O)CCn2c(COC)nnc2C1 C1(C(=O)NCC(C)O)C2CN(c3cc(C(F)F)ncn3)CC12 c1(CNC(c2cccnc2O)=O)ccc2c(c1)CCC2NC(C1OCCCO1)=O c1(C=O)c(C)nn2c(C)cc(C)nc12.C(C)(C(=O)NCC(C)C)N(C(C)=O)C Cc1noc(C(=O)NC2CC(C)N(C(c3cc(C(F)(F)F)n(C)n3)=O)C2)c1C N1(C(C2C(C)(C)CO2)=O)CCN(C(c2cccc(C3CC3)c2)=O)CC1CO Cc1nn(C)c(NC(=O)CCC2CC(F)(F)C2)c1S(N)(=O)=O C1(CCNc2cc(NCCC3CC(OC)C3)ncn2)CCC2(CC1)CC2 c1(C(N(CC(C)NC(C2(C)CC3CCC2C3)=O)CC)=O)cc(C)c(C)cc1Cl C(=O)(C(C)CC(N)=O)NCC(CNC(COCc1nnc(C)s1)=O)(C)O C1(NC(c2ncccc2C2CC2)=O)CC2CCC1CN2C(=O)CCc1cccs1 c1(OC)noc(C)c1C(=O)NC1CCOCC1NC(=O)C(c1cnn(C)c1)C c1(C(=O)NC(C)C=CC(=O)NCC2(C)CC2(F)F)ccn2ccccc12 CN1C2CCCC1CN(C(C1CCC(NC(=O)C=CCO)C1)=O)C2 Cc1c(S(=O)(=O)NCc2ccc3[nH]ccc3c2)cnn1C(C)C N1(C(c2c(C)nc(CO)s2)=O)CCC(NC(=O)C=CCO)C12CCC2 C(CCCCCC(=O)NCC1CCCCC1NC(=O)CNC=O)SC CC(C)(O)CCC(=O)N1CC2(CO)CC1(CNC(=O)CSc1ccncc1)C2 C=CC(CC(=O)N1CC(CO)(NC(c2ccc(C(N)=O)s2)=O)C1)c1ccccc1 C1(NCC2N(C(c3cc(OCC)c(C)cc3)=O)CC2)CC(C2CCOCC2)=NO1 c1(COC)cccc(F)c1.c1(CC)nc(C(F)(F)F)c(C)s1.C(=O)(C=O)N N1(C(C(CC)O)=O)CCC(CNC(=O)C=CC(=O)N)C(F)(F)C1.C1CC1 C(=O)(C#CC1CCOCC1)NC1(CC=C)CCN(C(C2(C)COC(=O)OC2)=O)C1 C1(OC)CC(NC(C2CC3(CCC3O)C2)=O)CN(C(c2cc(C)oc2C)=O)C1 c1(C(N2CCC(C)C2CNC(C2(F)CC2)=O)=O)cc2c(s1)CCCCC2 c1(CC(=O)NCC2C(C(NOCC(=O)OC)=O)C2(C)C)cccnc1F c1(OC(C)C(N2CCC(N(CC(=O)NS(C)(=O)=O)C)CC2)=O)cccc(F)c1 C(=O)(NNc1cccc([N+](=O)[O-])c1C)c1c2cccc(OC)n2nc1 N1(C2CCC(NC(C3(C(N)=O)CCC3)=O)C2)CCN(C(C2(F)CC2)=O)CC1 O=C1CN(C(C2CCN(OC)CC2)=O)C2CCN(C(=O)Cn3cccn3)CC2N1 C(CC(C(=O)NC(C)CC1(O)CCC1)NC(=O)C(C)CSC)OC C(=O)(C(C)C(F)F)N(C1CC1c1ccc(Br)s1)CCNC(C)=O N1(C(C(CC)C(=O)OC)=O)CC2CC(C1)CN(C(c1cc(C)c(C)o1)=O)C2 CCCC(CC)C(C(=O)NCC(F)F)N1CCC(N2CCC(O)C2)CC1 N1(C(COCC(=O)NC)=O)CCC2C1CCCN2C(c1nc(OC)c(C)s1)=O C(=O)(CCCCn1cc(CC(C)(C)O)nn1)OCCNC(c1n(C)ncc1)CO c1(CS(=O)(=O)NC(C(C)OC2COC2)=O)ccc(Br)cc1 C(CC(C)(C)NC(=O)C=CC(C)C)=CC(=O)NCCC(=C)C CC1CC(CNC(C2CCCN2C=O)=O)CN1C(c1ncc(Cl)n1C)=O C(=O)(C(C)(C)C(C)O)NC(C)C=CC(=O)NC(C)CN1CCCC1 c1(C(N2CC=CC(NC(C3CCC(C)(F)CC3)=O)C2)=O)cc2cnccc2[nH]1 c1(CC)ccc(C(N2CC(C(=O)NCc3cc(OC)no3)C(C)C2)=O)cc1 C1(O)(C(N2C(CCCC)CCC2)=O)CCN(C2CCC(O)CC2)CC1 c1(C(=O)NCCCCCNC(c2c(C)cco2)=O)cccc2cc[nH]c12 C1(C(=O)NCC2C=CCCC2)CCN(C(c2cnnn2C2CC2)=O)CC1O c1(OC)ccc(CCN=C(NCc2ccnn2C)NC2(CF)CCC2)c(Cl)c1 C1(C(=O)OC)(COC)CCN(N2CCCC(OCC3CCC3)C2)CC1 CC1CCCC1(C(=O)NCCCc1cnn[nH]1)NC(=O)CN1CCCCC1=O c1(OC)ccc(C(N2CC(N(C(=O)C3=C(Cl)CCC3)C)C(F)C2)=O)c(F)c1N C1(NC(=O)C(F)C(F)(F)F)CCC2CN(C(c3cc(O)cc(Cl)c3)=O)CCC2C1 O=C1NCCC2CCCN(C(c3cn(CCN4CCCC4)nn3)=O)C12 c1(OC)cc[nH]c(=NCCCC(C)NC2CCN(C(=O)OC(C)(C)C)CC2)n1 C=C(C)C(O)CC(=O)N1CCC(NC(=O)C(C)Cn2cccn2)C(O)C1 C(C(COC)CC(=O)N1CC(NC(=O)C(C)(C)c2cnn(C)c2)CC(C)C1)OC C(CC(=O)NC(c1nc(C)no1)CO)(C(F)F)NC(c1n(CC)ccc1)=O N1(C2C3CN(C(Cc4cc(C)on4)=O)C(C3)C2)CCn2ncnc2C1 C12(CNC(c3c(CC)n[nH]c3)=O)CC1CN(C(c1cscc1OC)=O)C2 c1(N2CC(C)N(c3cc(C#N)ncn3)CC2)ncc2[nH]ncc2n1 c1(OC)ccc(C)c(C(N2CCOC(CN(C)C(c3ccccc3O)=O)C2)=O)c1 C(=O)(C1=CC2CCCCCCC12)N1CC(N(C(CCC(=O)N(CC)CC)=O)C)C1 Cc1ccc(C)c(CC(=O)N(C)CC2CCCN2c2cc(C)nc(C)n2)c1 N1(C(CC(C)c2ccco2)=O)CCN(C(=O)CCC(N)=O)CC(O)C1 c1(C(c2n(CCCSC)nnn2)NC(c2ccsc2)C2CC2)c(C)cncc1C C#Cc1ccccc1C(N1CCCC1CC(=O)NCC(C)C)=O CN1CCC(C)(C(=O)NCC2CCCCCN2C(c2coc(N(C)C)n2)=O)C1=O c1(-c2cncc(NCc3cc(C)sc3C)c2)c(F)cc(C(=O)O)cc1F C1(O)(C(N(CC(C)NC(c2n[nH]cc2-c2ccncc2)=O)C)=O)CCOC1 c1(C(N(CCN(C(c2cccnn2)=O)CC)CC)=O)n[nH]c2ccc(C)cc12 Cc1nc2cc(C(=O)NC3CC(CO)N(C(=O)Cc4ccn(C)n4)C3)cnc2s1 N#Cc1cccc([N+](=O)[O-])c1NC(CNC(=O)C=Cc1nccs1)C1CCC1 CC1CCN(C(=O)C(c2cncnc2)C)CCN1C(=O)CN1CCS(=O)(=O)CC1 c1(C(=O)O)cnc2c([N+](=O)[O-])cnn2c1 C(=O)CC(C)(C)C1CC1.c1(C(C)NC(=O)Cc2ccnn2C)cn(C)cn1.N C(=O)(C#CC1CCCO1)N1CCCC(CNC(c2ccsc2Cl)=O)CC1 c1(SC)cc(C(=O)NC(c2nc(C(=O)Nc3ccccc3)co2)C)co1 C1(NC(C2CC(=C)C2)=O)CCC12CCN(C(c1cn(C3CC3)nn1)=O)CC2 c1(C(N2C(C)CC(CNC(C3(C)CC(=C)C3)=O)C2)=O)cc(F)cc2nc[nH]c12 C1(NC(C(C2CC2)OC)=O)Cc2ccccc2N(C(=O)CC2CCN(C)CC2)C1 CC(C)CC(C)C(=O)NCC1C=CCN1C(=O)CCC(=O)N1CCOCC1 C1(OC)CN(C(C2CC(F)(CO)C2)=O)CC1NC(=O)Cn1cnnc1 N1(C(CN(CCOC)C)=O)CC23CCCCC2(C1)CN(C(c1ccon1)=O)C3 CC1CCCn2ncc(C(=O)NC3CCC3CNC(=O)C(C)(C)C)c21 c1(OC)cc(OC)c(C(=O)Nc2cccc(C(C)O)c2)c(F)c1 Cc1nc2[nH]ccc2c(=NCC2CN(C(=O)C(C)S(C)(=O)=O)CC3(CCC3)O2)[nH]1 C1(C(=O)NCC(C)N(C(c2c(C)cco2)=O)C)CCCC2(CCOCC2)O1 CC(C)(F)C(=O)NCC(c1ccccc1)NC(=O)CC12CCCC1C2 CN1N=C(C(=O)NCCCCn2cc(C3CC3CO)nn2)CCC1=O C=CC(C)(C)CCCNC(=O)CCCN(C(=O)CCCNC(C)=O)C C1(C(=O)NCCN(C)C(c2nccn2C)=O)Cc2ccccc2S1(=O)=O C1(CN=C(NC(C2CCCO2)C)NCc2ccco2)CC(C)(C)OC(C)(C)C1 N1(C(C2(CC)CCCO2)=O)CCC2CCN(C(=O)CNC(=O)C(C)(C)C)CC12 C1(C(N2CC(CCC)C2)=O)CCC(C)(C)OC1.c1(C(=O)N)cnc(C2CC2)nc1 CC1(C(=O)NC2CC2CNC(C2CCCS2)=O)CCC(F)(F)CC1 C1(C(=O)NCCc2cnc(C)[nH]2)C2CC1N(C(=O)C(F)CC1CCOC1)C2 c1(Oc2ccc(CN3CC(CC(CC)C)C3)o2)cncc(C(=O)O)c1 c1cccc(F)c1C.C(CC(C(=O)N1CC(CN2CCOCC2)C1)SC)OCC c1(C(N2CCC(C)(CCNC(C(C=CC)O)=O)C2)=O)cccc2c1C(=O)CC2 CCC(CNC(=O)CCCOC1CC1)(CC)NC(c1ccc(NC=O)cc1)=O C(=O)(C1OCCc2ccccc21)NCC1CCN(Cc2[nH]n(C)c(=O)n2)C1 N(C(=NCC(C)(C)C(C)(F)F)N1CCC2(C1)CC2(F)F)C(C=C)C N1(CC(=O)NC2CCC(NC(Cc3cnc(C)s3)=O)CC2)CCS(=O)(=O)CC1 N1(C(C=CSC)=O)CCC(C2CCCN(C(=O)COCC3CCOC3)C2)CC1 C(CCC(=O)NCC1(O)CC(NC(=O)C(O)c2cnc[nH]2)C1)=CC(C)C C(C(CC(C)(C)C)NCCCCC(=O)NC1CCNCC1)OC C1(C(N2CC(Cn3cc(CCN4CCCCC4)nn3)C2)=O)CC2COCC2C1 C(=O)(C1CC=Cc2ccccc21)N1CCCN(C(CCCCC#C)=O)CC1CO c1(C(=O)NC2(C)CCCN(C(COC)=O)C2)cc([N+](=O)[O-])cn1C C(=O)(C(CC=C(Cl)Cl)c1ccccc1)N1CC(C)C(CO)C1 C1(NC(CCCCCC)=O)CC2CC(C1)N(Cc1c(C)noc1C)C2 C(CCN=C(NCCSC)NC1CCC(=O)NC1)N(C(=O)OC)C C1(C(N(CCC(=O)NCc2cn(CC#C)nc2)C)=O)COCCC1C C(=O)(C(O)CC(C)C)NCC1CCCN(C(CCC(C)=O)=O)C1 C1(C(N2CCC(NC(c3cc(C)sc3)=O)C(O)C2)=O)Cc2c(C)cccc2N1 c1(C(N2C(CC(N3C(C#N)C4CC4C3)=O)CCC2)=O)cc2ccc(Cl)cc2s1 C1(NC(COC)=O)CC(O)CN(C(=O)C(O)CNS(C)(=O)=O)C1 C(=O)C(C)(C)CC(C)(C)C.C1(CC)CN(C(C2(C)CC(F)(F)C2)=O)CCO1.N CCCC(CC(C)C)C(=O)N1CCC(NC(c2ccc(CC)s2)=O)C(CO)CC1 c1(OC)c(C(C(=O)NC2CCOCC2)N(C2CCC2)CCN(C)C)ccnc1Cl Cc1nn(C)c(C)c1CCC(=O)NC.C1(C(N2CC=CC2)=O)COCC(C)(C)O1 C1(N(C(=O)CCC(=O)c2cccc(N)c2)CC)CCN(C(C2CC2CF)=O)CC1 N1(C(CC2C(CC)C2)=O)C2CC1CN(C(c1ncccn1)=O)C2 C1(C)(C(=O)NC(C)C(CO)NC(c2cnn(CCF)c2)=O)COCCO1 C1(O)(CN(C(c2cc(CC)sn2)=O)C)CCCN(C(C2CC3CC3C2)=O)C1 C1(C(=O)NC(CCC(=O)OC)C)CN(C(=O)C#CC(C)(C)O)CC1(F)F c1(C(N2CC(C)(CNC(CN3C(C)CC3)=O)OCC2)=O)ccc2cccnc2c1 N1(C(C(C(=C)Cl)(C)C)=O)CCCC(C2CC2NC(c2nc(C)ccc2OC)=O)C1 N1(Cc2cc(O)ncc2)CC2CCCCC2C1.C12(CCCCC1)CN2 C1(NC(CCOC(C)C)=O)CN(C(c2ccc(C(F)(F)F)o2)=O)CC1C N1(C(CCc2onc(CC)n2)=O)CCCC12CCCN(C(=O)C(C)N(C)C)C2 N1(C(c2n(CC)nc(C)c2)=O)CCn2c(CNC(=O)CC(C)CO)nnc2C1 C1(C(=O)NCC(C)(O)C2CC2)CC1C1CN(C(C2(C#N)CCCC2)=O)C1 N1(C(C=C=C(C)C)=O)CC2(CCCN(C(=O)CCC3CC3C)C2)C1 Cc1ccc(F)c(C(=O)NCC2C=CC(NC(=O)CCCCC3CCSS3)C2)n1 c1(NC(N2CCC(NC(c3occ(C(N)=O)c3)=O)C2)=O)cccc(O)c1F c1(C(N2CCOCC(NC(C=CC(C)C)=O)C2)=O)ccc2c(c1)C(=O)C(=O)N2 Cc1ccc(F)cc1CC=C.C1(=CC=O)CCN(CCc2ccnn2C)CC1 C1(C(=O)NC2(C3CC3)CCOC2)CCC2CCC1N2C(=O)CCC(CF)CF N1(c2nc(=N)nc(N3CCCC(OCC(C)C)C3)[nH]2)Cc2ccc(Cl)nc2C1 CC(C)(CC(=O)NCC12CCC(CC1)CN2C(c1cc[n+]([O-])cc1)=O)C(F)F c1(C(N(C2CCN(C(=O)CC(C)(F)F)CC2)CCCC)=O)cn(C(C)C)nc1C C1(n2cc(-c3c(C)cn(C)n3)nn2)CON(C(=O)C2(O)CC3CCC2C3)C1 c1(OC)ccncc1C(N1CCOCC1C(=O)NC1COCCOC1)=O C1(CC(=O)NC(CN(C(=O)COc2nc[nH]n2)CC)C)CC(CF)C1 N1(CCC(=O)NC(CC(C)NC(CCN(CCC)C)=O)C)CCC(C)CC1 C(c1cnn(C)c1C)=CC(N1CCC(CCOC)(NC(C2C=C2C)=O)C1)=O c1(C(=O)OCC2C(C)CC=CC2)cc(C(F)(F)F)cc(C(F)(F)F)c1 N1(C(C2CCCC(F)C2)=O)CCOCC2(COCCN2C(=O)Cc2nncs2)C1 c1(CC(=O)N(CCNC(C=CCCC)=O)C2CC2)sc(C)cc1C c1(C(=O)NCC2(F)CCC(NC(c3cscn3)=O)C2)c(F)ccc(Cl)c1F c1(C(N2CCC(C)(NC(=O)CCC3CCC3)C2)=O)cccc(Br)c1[N+](=O)[O-] C1(CN(C)C(c2csc(Cl)n2)=O)CCCCN1C(C1COC(=O)N1C)=O C1(Cl)(C(=O)NCCCN(C(=O)C(O)C2CC2)C)CCC1 C(C1CN(C(C2(O)CCOCC2)=O)CC1C(=O)NC(C)CCSC)=CC c1(CC)oc(C)cc1C(=O)NC1CCC(C(=O)N(C(C)CSC)C)CC1 CCCCC(O)C(=O)N1CC2(CC2)CC1C(=O)Nc1ccnc(F)c1C C(=O)(C(C)N(OC)C(=O)c1cnc(CNC(=O)C(C)COC)nc1)OC C1(CC)C(=O)NCCN1C(=O)Cn1cc(CNC(C2CC2CC)=O)nn1 C1(C)(C(=O)OC)CCN(C(=O)C(C2CCN(C(C3CCCN3C)=O)CC2)C)C1 c1(NC(CC2N(Cc3c(C)cccc3Br)CCOC2)=O)nc2ccc(Br)cc2s1 C(CN=[N+]=[N-])(C(=O)N1CCCc2ccnn21)NC(C(CCCC)O)=O C1(CCOC)CN(C(c2[nH]nnc2C)=O)CCN1C(c1cscc1C(C)C)=O C12(C(=O)NCC(C)(C)NC(c3cccc(Cl)n3)=O)CC=CCN1CCC2 c1(OC)cc(C)c(CNC2(CC(=O)Nc3cccnc3OC)CCC2)c(O)c1 C1(CC(=O)NCC(N(C)C(c2cnn(C)n2)=O)C2CC2)CCC(O)C1 N1(C(c2nc(CNC(CO)=O)oc2)=O)CCC(C)(C(N)=O)C1.CC=O.O c1(C(=O)NCCCN(C(CNC(CC)=O)=O)C2CC2)cnc2cc[nH]c2c1 N1(C(C(C)(F)F)=O)CCN(C(c2ccnc(C3CC3)n2)=O)CC1CC(F)(F)F Cc1cc(C)n(C(C)C(=O)NCC2(c3ccc(Br)cc3)CCOCC2)n1 CC1(C)COCC1C(N1CCC(C(C)(C)NC(=O)CCn2ccnn2)C1)=O C=CCC(CNC(C1CN(C)C1)=O)C(=O)N1CCC1 CC1CC2CN(C(=O)CN3CCCCC3)CC2N1C(C1CNC(=O)CC1(C)C)=O N1(C(C(C)C2CCC2)=O)CC2CC2(C(=O)NC2CCCC2CCO)C1 Cc1cccc2oc(C(N3CC(CO)(NC(=O)C4=COCCC4)C3)=O)cc12 N1(C(C(CO)NC(Cc2c(C)noc2C)=O)=O)CCC(O)C(O)C1 C1(NC(C2N(CC)CCC2)=O)(CO)CCN(C(c2cc(Br)c(C)o2)=O)CC1 N1(C(CCCNC(C(n2ccc(C)n2)C)=O)=O)CCC2OCCCC2C1 N1(C(CCCC=C)=O)CCC2(CCC(NC(=O)CNC(=O)NC)C2)C1 N1(C(c2csc(C)n2)C(=O)NCC)Cc2cnc(C3CC3)nc2C1 c1(C(N2CC3(CC(C(=O)NC(COC)COC)C3)C2)=O)cccc2ccccc12 CCCCC(O)CC(=O)N1CC(OCC)C(CNC(c2cccc(Cl)c2)=O)C1 C1(NC(C2N(C(c3cnn(C)c3Cl)=O)CCC2)=O)CCc2nncn2C1 c1(C(=O)NC2C3CN(C(C4CC(=C)C4)=O)C2C3)nc(Br)c2ccccn12 CC(CN=c1nn[nH]n1-c1ccc(F)cc1)NC(=O)C(C)CO N1(C(C(C2CN(C(c3csnn3)=O)C2)OC)=O)CCC(C)OC(C)C1 Cc1cc(C(=O)NC2(CNC(C3CCSC3)=O)CC2)c(Cl)cc1N N1(C(c2cnc(C)[nH]2)C(=O)NC2(C)CC2)CCc2ccc(C3CC3)cc2C1 c1(CC)[nH]c(=N)sc1C(N1CCOC(CCCNC(C2CCCNC2=O)=O)C1)=O C1(NC(CC)=O)COC2(C1)CN(C(c1cccc(C)c1)=O)C2.C(=O)C(F)(F)F c1(N(CC(C2CCC2)OCC)C)ncnc(N2CCC(CC(C)C)C2)c1C C(CCC(C)C)(C(=O)NC(C)C(=O)OC)N1C(CC)C(C)CC1 C(=O)(C(CCCC(C)OC)N1CCC(CCN(C)C)CC1)NCC=C C(=O)(CCC(C)(C)NC(=O)C=Cc1cccnc1)N(C)CC1(O)CCC1 c1(C(N2CC=CC(C(=O)NC3(CCCC)CC3)C2)=O)cc(C)ncc1C c1(C(N2C(CNC(C3CCC(F)CC3)=O)CC(C)(C)C2)=O)cnc2c(c1)CCC2 CCCC(CCCNC(=O)CN(C)CC)NC(=O)CCC(C)(C)N1CCOCC1 C1CCN(C(C23CC2CCC3(F)F)=O)CCC1(F)F.C(C(F)(F)F)=CC(=O)N.C C1(NCC(c2cc(F)cc(Br)c2)F)CC2(CCC(N)CC2)C1 c1(NC(C2N(C(c3c(C)cccc3Cl)=O)CCC2)=O)cnnc2ccccc12 c1(C(CC)N(C)C(=O)NCC(C)(CO)OC)ccncc1 N1(C(C(N2CC3CC3C2)C)=O)Cc2ccnn2CC1C(C)C.n12cc(nn1)C2 c1(C(N2CC3(CN(C(C4CCCC(N(C)C)C4)=O)C3)C2)=O)ccc2occc2n1 CC(CC(=O)NCC(O)CNC(c1cc(N)cc(F)c1)=O)CC(F)(F)F N1(C(=O)C=CI)CC2(C1)CN(C(C1C=CCCC1)=O)C2 c1(C(N(C)CCN(C)C(C2CCc3nncn3C2)=O)=O)cc(N)c(F)c(F)c1F CCC(CC(=O)NC1CC12CC(NC(=O)C#CC1(C(F)(F)F)CC1)C2)C(F)F c1(CC(=O)NCC23CC(CN2C(=O)CC2COCCO2)C3)c[nH]c2ccccc12 c1(C(=O)OC)cn(CC(N2CCC(c3cn(CCF)nn3)C2)=O)cn1 C1(C(=O)NC(C(CO)NC(c2c(C(C)C)ccs2)=O)C)CCC(F)CC1 N1(C(c2cc(SC)c(C)o2)=O)CC2(COC(C)C2)C1.CC(C)(C)C.C(=O)C.N C1(C(=O)NC(CC=C)C2CC2)CCCC(NC(=O)C(O)CCN(C)C)CC1 C1(NC(COC2CN(C(C=CC=CC)=O)C2)=O)CC(C)(CC)C1 N1(C(COc2cccc(COC)c2)=O)CCC(C2CC2)C1C.C(=O)C1CC1 C1(C)(CNC(c2scc(C)c2)=O)CCCN1C(c1csc(C(C)C)n1)=O c1(CC)ccc(C)cc1C(N1CCC(C)(NC(C2CC(C)OC2=O)=O)CC1)=O c1(C(=O)NC(C(C)NC(=O)Cc2ccc(Cl)s2)(C)C)cc(O)c2ccccc2c1 C12CN(C(C3CC4(C3)CC(F)C4)=O)CC(F)(C1)C2.C1(CC(=O)N)CCCCO1 Cc1nccc(C(=O)N)n1.c1(C(N2CC(O)(CC)C2)=O)cn(C(C)(C)C)nc1C C1(C=O)CC2(C1)CS(=O)(=O)C2.c1(C(N(CCC)CC)=O)cnc(O)cc1C C1CN(C(=O)Cn2cnc([N+](=O)[O-])n2)CC1(C)C.C(CC=O)NC(=O)OC.N Cn1ncc2cccc(CN3CCCCC3CCC(F)(F)F)c12.C(C)(C)C.C=O.N Cn1nncc1S(C)(=O)=NC(=O)C1(c2ccc(Cl)cc2)CCCCC1 CC(CNC(c1cn(CCO)nn1)=O)CN=c1nc2c(c[nH]1)ncn2C CCC(c1ccccc1)=CC(=O)N(C)CC1CCCN1C(c1cncn1C)=O c1(C(N2CC3CN(C(C(C)=O)=O)CC32)=O)cccc2ccnn12 C#CC1CN(C(C2Cc3cscc3C2)=O)CCN1C(C1COCCN1C)=O CC(C)(CNC(c1cc(C2CC2)no1)=O)CCNC(C1(C)CC=CCO1)=O N1(C(C(CCC)=CCC)=O)CC2CC(CNC(C3CC3[N+](=O)[O-])=O)C2C1 C1(CNC(Cc2nnc(C)o2)=O)CCC(C)(C)CN1C(=O)C1=CCCS1 CC(=O)CCCC(=O)NC1CCC(F)(CNC(c2ccnn2CC#N)=O)C1 c1(C(=O)NC2CN(C(c3cc(O)cc(O)c3)=O)CC2O)cnc(O)c(Cl)c1 N1(C(COC)=O)CCCC2(CNC(=O)CCCCC(N)=O)CCCC12 CCC(C(=O)N1CCC(C(C)CNC(=O)C=Cc2ccccc2)CC1)C(C)(F)F c1(CSc2n(CCOC)c(-c3cncc(Br)c3)nn2)nnc2n1CCN(C)C2=O c1(C(N2C(CNC(C3CC4C=CC3O4)=O)CCCC2)=O)ccc2c(c1)SCCN2 CCCCCC(F)C(=O)NC1(C(N2CCCC(C(N)=O)C2)=O)CC(F)C1 C1(CC(=O)NCC(CNC(C2CC(C#N)C2)=O)F)CCn2cncc2C1 Cc1ccc(C(N2CCC(O)(C(C)CNC(C3(Cl)CC3)=O)C2)=O)c(N)n1 CC(C)(CCCN)C(=O)N1CCN(CCc2cn(Cc3cccnc3)nn2)CC1 c1(C(=O)NCC(C)NC(C2CCn3c(O)nnc3C2)=O)cc(F)cc2nn[nH]c12 C(CCCc1ccccc1)(c1nnnn1C1CCOCC1)NCC=C1CCOCC1 C12(C(N(C)C)=O)CCC(NC(c3cc(F)ccc3Cl)=O)(CC1)CC2 CC(C)(O)C(C)(O)CNC(=O)CC1CCCN1C(=O)OC(C)(C)C CP(C)(=O)CC(=O)N1CC2CC2(NC(C2CCCCO2)=O)C1 c1(C(=O)NCCNC(C2(C)N(C)CC(OC)C2)=O)nc2cccnc2s1 c1(C=O)cccc2ccn(C)c12.c1(CNC(C)=O)ccc(C(=O)NCCC)s1 N1(C(CCC#CC)=O)CCC(c2ccccc2)(NC(C2CC3CCC3C2)=O)CC1 C1(CC(=O)N(CCC)CC)CCc2cnn(C)c2C1.C(=O)CC.[SH](C)(=O)=O C(CCCCCNC(=O)C(C1CCC(=O)N1C)C)N(C(C=C(C)C(C)(C)C)=O)C C1(C(=O)NC(CCC)c2nn[nH]n2)COCCC1NC(c1ccncc1CC)=O CCC(C)CCCCC(=O)NC1CC(N(C(=O)Cc2cncc(C)c2)C)C1 c1(OCCN(C)C)ccc(C(N2CC(C)CC(N)C2)=O)c(Cl)c1 Cc1cc(=NC(=O)C(=O)NC(C2CCCN2C(C2CC3CC3C2)=O)(C)C)[nH]o1 N1(C(C=C2CCC(C)CC2)=O)CCN(C(c2c[nH]ccc2=O)=O)C2CCCCC12 N1(C(Cc2nc(C)[nH]n2)=O)CCC(C)(C)C1C(=O)NCC1(CCO)CC1 C(=O)(C(C)(C)C(F)F)N.Cc1cn(CC(=O)NC2COCC2)nc1C(F)(F)F N1(C(Cc2cccc(OC)c2)=O)CCCN(C(C2CC2(Cl)Cl)=O)CCC1 C(=O)(N=c1cc(C(C)OC)[nH][nH]1)Nc1c(CC)cccc1 C1(CNC(c2cc(-c3cccs3)on2)=O)CCC12CCN(C(=O)CNC=O)CC2 c1(C=O)c(F)ccc(O)c1F.c1(NC(C2CCC2)=O)ccoc1C(F)(F)F.N N1(C(CCN(C)C(=O)N(C)C)=O)CCCC(CCCO)C1 c1(C(=O)NC(CNC(C(n2ccc(C)n2)(C)C)=O)C(C)C)cc(N)ccn1 C1(NC(CNC(CC)=O)=O)COCCN(C(c2sc(C3CCOC3)nc2C)=O)C1 C1(C(C)C)(C(=O)NC2COCC2NC(=O)COC2CCC2)CNC(=O)C1 c1(C(=O)NC(CC)CNC(c2ccsn2)=O)c(Br)noc1C1CC1 O=C1CCNC(=O)N1CCNC(C12CCCC1C2Br)=O C1(CC)(NC(c2cn(CCO)nn2)=O)CCCN(C(c2c(C)cccc2O)=O)C1 c1(C(N2CC3C(CNC(c4ccc(C=C)cc4)=O)C3C2)=O)cc(Cl)c(O)cc1C N1(C(c2oc(C)c(CO)c2)=O)CCC(NC(=O)CCS(C)(=O)=O)C(C(C)C)C1 C1(CC)CCN(C(c2coc(CO)c2)=O)C(C(=O)NCC(C)(C)CCO)C1 CC1CCN(CC(N2CCOC(CC(=O)NCC(C)(O)C3CCCC3)C2)=O)CC1 C(=O)(CC1=Cc2ccccc2C1)N1CC(C)CC(NC(C2(CC#C)CCC2)=O)C1 Cc1ccc(OCCC(N2CCOCC(CNC(=O)C(O)C(F)F)C2)=O)c(Cl)c1 c1(C(=O)NC2C(NC(C3(C)C=CCCC3)=O)COC2)cnc2c(N)cccc2c1 c1(C(=O)NCCC(C)N(C(=O)Cn2nccn2)C)cnn2cc(Br)cnc12 C1(C(N2CCC(OC)(CO)C2)=O)CCOCCN1C(=O)C(F)C(C)(F)F N1(C(COCCC(C)C)=O)CC2C(CO)C2C1.c1(C=O)cscn1.C(=O)(C)N c1(SCC)cc(C(=O)N)ccn1.C1CCCCC1.C1(C=O)(C(N)=O)CC1.C c1(C(N(C2CN(C(C3CC3(F)F)=O)CC2(C)C)C)=O)cnn2c1C(=O)NCC2 C1(NC(=O)CC2CCCN2C(=O)C=CC2CCCCC2)CC12CCCC2 Cc1cc(C#N)sc1C(N1CCCC1C1CC1)C(=O)NCCC#N C1(CC(=O)NCCCN(C(c2c(C)nco2)=O)C(C)C)CCCC2(CCC2)O1 CC(C)C(C)CC(=O)NCC1(C)CCCN1C(=O)CC1CC2CC2C1 Cn1nnc2c1CC(C(N1CC3CCC1CN3C(=O)CN1CCC1)=O)CC2 Cc1cc(C(N2CCC(n3cncn3)C2)C(=O)NCCC#N)on1 C1(C(C)C)CCC(C(=O)NCC#CC#CCO)N1C(c1ncc[nH]1)=O c1(CN2CCC(CC(=O)NC34CCC(C(F)F)(CC3)C4)C2)cnn2c1CCCC2 C(CC(O)CCC1(OC(C)C)CCC1)NC(=NC)NC(C)Cc1ccccc1 c1(C(=O)NCC#CCNC(CC2(OC)CCCCC2)=O)cc(C(N)=O)ccc1C CC1(C)OC(C(=O)NCCCCCCNC(=O)CO)C(C)(C)O1.C1CC=CC1 CCC(CCCC(=O)NCCC1CCCN1C)NC(C1C2CCCOC12)=O C1(CC)CN2CCN1C(=O)CC1(CCCCC1)C2=O.c1(COC)[nH]c(C)nc1C CC1CCN(C(=O)CN(C)C(=O)C2CC2)CC1NC(=O)C(F)C(F)(F)F C=C(C)C1OCCCC1C(=O)NC1CN(C(C2(C)CCCC2(F)F)=O)C1 C1(NC(c2cc(C)ncn2)=O)CC2CCCC(C1)N2C(=O)CC(C)C1CC1 c1(C(N2C(CC(=O)NCCCCCC=C)CC(F)C2)=O)cccc2ccnn12 c1(C(N2CCC(F)C2)=O)ccc([N+](=O)[O-])c(C)c1.n1(CC)ccnc1C(=O)N C(=O)(CC(C(F)(F)F)c1ccccc1)NCC1CCCC(C)(C)C1 C(=O)(N=c1cccn[nH]1)C1CCC(NC(C(C)Nc2ccc(CO)cc2)=O)C1 C1(CNC(C2CCN(CC)C2)=O)CN(C(c2cncc(C(C)C)c2)=O)CCO1 c1(NCCc2cncc(C)n2)[nH]c(=NC2CC3C(C2)C3(F)F)nc2sccc12 n1(C(C)C)cccc1C(=O)NCc1csc(C(=O)NC(C)C(=O)NO)c1 C1(C)(NC(CCN(C)C(c2ncc[nH]2)=O)=O)CCCCC1(C)C c1(C(N(C)CC2CCCN(C(C3COC(=O)N3)=O)C2)=O)cncc(F)c1Cl N1(C(C(=O)Nc2cnc(C)[nH]c2=N)=O)CCOC2(CCOCC2)C1 N1(C(c2scc(CNC(C3OCCN(CC)C3)=O)c2)=O)CCC12CCCC2 S(=O)(=O)(C1CCC(=O)CC1)NC1CN(C(c2cc(C)ncn2)=O)CC(C)C1 N1(CC2(COC)CCNCC2)CCC(O)C(CC(C)C)C1 Cc1ncc(CC(N2CC(CNC(c3[nH]cnc3C#N)=O)C(C)(C)C2)=O)c(O)n1 C=CCCCCCC(=O)N1CCC(NC(=O)C(C)(C)COC)CC1C c1(CNC(C(C(CC)C)C)=O)cnn2c1CN(C(c1[nH]cnc1C#N)=O)CC2 C1(C(N2CCC2)=O)CCCN(c2cnccn2)C1.C(C(=O)NC)=CC=CC CCC(O)C(C)C(=O)NCC1CC2(CC2)CN1C(=O)C(C)CCCOC c1(C=O)ccc(F)c(N)c1F.Cc1n[nH]c(C)c1C(C)C(=O)NCC(C)(O)C.N Cc1cn2c(=O)c(C=O)cnc2s1.C1(C)(OCC(=O)NCC)CCC1.CC C(=O)(CC(C)(C)CC(=O)NC12CCC(C(F)F)(CC1)CC2)OCC c1(NC(c2ccc(C(=O)O)[nH]2)=O)ncccc1C(=O)Nc1cn(CCCO)nn1 Cc1nc(C(C)(C)C)nc(O)c1C(=O)NCc1nc(-c2ccccc2)n[nH]1 C1(NC(C2C(C#C)C2)=O)CC(F)(C)C1.c1(C=O)c[nH]nc1-c1ccccc1.N CCCC(C)C(=O)NC1CCCCC1CNC(c1cc(N)c(C(=O)OC)s1)=O CCC(CC(=O)NCC#CC(=O)NC1CC1CCOC)C(F)F N1(C(C2CC(C#C)(O)C2)=O)CC2COCCC2(NC(=O)CCCC#C)C1 CC1CN(C(C2(NC(=O)CC3(C)CC3)CC2)=O)CCC1CO C(=O)(CC(=O)CN1CCCCC1c1ccc(Cl)cc1)OCC N1(C(C(CC)CO)=O)CC2CCCC(NC(=O)Cc3ccc(F)cc3Cl)C2C1 C(CC(C)C(=O)NCC(O)CCNC(=O)C(C)Cc1cnco1)OC c1(OC)ccc(F)cc1C(F)(F)C(=O)OCC1(c2ccc(F)cc2F)CC1 Cc1nc(NC(C2CC2C(C)(C)C)C)cc(N(CC(N)=O)C)n1 C1(NC(c2cnc(CC)s2)=O)CCCCCN(C(c2cc(C3CC3)no2)=O)C1 C1(CC(=O)OCC)COCCN1C(c1ccc(N(CC(C)C)C)nc1)=O N1(C(C(N2CC(C)C(CN)CC2)=O)=O)CCC(O)c2cc(Br)ccc2C1 c1(C(N2CCCC(NC(c3c(C)cc[nH]3)=O)CC2)=O)cnc2ncc(Cl)cn12 C=CCCCCCC(=O)NC1CC(C)(NC(c2cnc(Br)c(OC)c2)=O)C1 C1(OC)CN(C)CC1NC(c1[nH]ccc1C)=O.C(=O)CN(C)C1CC1.N C=CCC(CC(=O)NC(C)CCCCO)NC(=O)C(C=C)CC c1(N(CC(=O)OCC)C)ncc(S(C)(=O)=O)cc1Cl.c1ccc(F)c(Cl)c1 C1(C=O)CC(S(C)(=O)=O)C1.Cc1cc(C(=O)NCC2CCCCC2)sc1C.C c1(C(CCC(=O)NCC2C(N=[N+]=[N-])COC2)=O)c[nH]c2ccccc12 Cc1cnc(F)c(C(N2CC(NC(=O)C#CC(C)C)CC2C)=O)c1 O(N(C)C(=O)CNC(=O)CC1CC(C)N(C(=O)C)C1)CC.CC(N)=O.S N1(C(C(F)=CCC)=O)CC(C(N2CC(c3cc[nH]n3)C2)=O)C(C)C1 N1(C(C2(CC=C)CCCC2)=O)CCC(CO)C(NC(C2(C)CCN(C)CC2)=O)C1 c1(C(N2CCC(NC(C(C(C)C)(C)C)=O)C2C(C)(C)C)=O)coc2c1CCCC2 C1(CCNC(=O)CCOC2CCCOC2)CCN(C(c2cc[n+]([O-])cc2)=O)CC1 C1(N(C(C=CC(C)NC(C2CCS(=O)CC2)=O)=O)C)CCCC(C)(C)C1 C(C(CC(C)C)C(=O)NCc1c(C)coc1C)NC(CC(C(=O)OC)C)=O c1(C(N2CCC(CNC(CC(CC)CN(C)C)=O)C2)=O)ccnc2[nH]c(O)nc12 N1(C(CC2N(C(CC(C)C(F)F)=O)CCC2(C)C)=O)Cc2cc(O)nnc2C1 c1(C(N2C(CC)CSCC2)=O)ccc(C)c(C)c1.C(C=O)(C1CCC1)OCC.N CC1=C(C(=O)NCC2CC3CC3N2C(C2C3COCC23)=O)Cc2ccccc2O1 C(=O)(CC(=O)NC(C1(C(=O)NCc2cnc(C)s2)CC1)C)NCC c1(CCC(N2CCCC(CCNC(CC(C)C)=O)C2)=O)nc2cnccc2[nH]1 C(C(CCO)NC(C1CC(N(C(=O)CSC2CC2)C)C1)=O)OC C1(OC)CC2(C1)CC2C(=O)N(C)CC.C(=O)CN(C)C(C)=O.CC.O c1(OCCC)cc(F)ccc1NCc1c(C)noc1N C1(CN(C(=O)CC2COCCO2)C)CCCCN1C(=O)C(c1ccc(O)cc1)=O CCCCC=O.C12(CC1(F)F)c1nc(sc1)CNC2.CSC C#CC(CC(C)C)NC(=O)C(CC1CCCC1)NC(C1CCCN(C)C1)=O N1(C(C)=O)CCc2sc(CNC(C3CCCC(O)C3)=O)nc2C1 N1(C(C(NOCC)=O)Cc2ccccc2)C(=O)C2CCCCC2C1=O C(N=c1cc(C(C)(C)C)nc(Cl)[nH]1)C1CCN(C(c2c(S(C)=O)cccc2)=O)C1 Cn1cncc1C(N1CCC(N(CCO)C(C2CC2(C)C)=O)C1)=O Cc1cc(NC(=O)C(CN(C)C(c2ccncc2)C)N)cc(C)c1 C1(NC(c2cnc(CNC(C(C)SC(C)C)=O)nc2)=O)C(O)C2CCOC12 CCC(C)(CC)C(=O)NC1CC(NC(=O)C(C)=C2CCCC2)C1 c1(OC)ccc(NC(=O)NCCCNC(=O)N)cn1.c1ccc(Cl)cc1.C C1(C(=O)NC(C)C(=O)NCCc2cncn2C)CCC2(CCCC2)C1 CCC(C)C(C(=O)N1CCCCC1)N(C(=O)CCC(=O)C1CC1)C C(C)(CO)(C(F)(F)F)NC(COC1CCN(C(C2C(C)(C)COC2)=O)C1)=O C12(C(=O)NCCCNC(=O)CN3CCCS3(=O)=O)C3CCC(CC13)C2(F)F C(=O)(C1=CCCS1)NC1C(CNC(C2(CN(C)C)CC2)=O)CCC1 C1(CC)CCCCC1C(N1CC(C)(NC(=O)COc2ccc(O)nn2)C1)=O CC1CC(NC(c2cccc[n+]2[O-])=O)CN1C(c1ccc(C(F)(F)F)[nH]1)=O C1(NC(c2cc(CC)[nH]n2)=O)C2COCC1CN(C(C1CCN(C)C1=O)=O)C2 c1(OC)nsc(C(C(=O)NC2COC2)N(C2CC(O)C2)C)c1Cl N1(C(C2C(O)CCN(CC)C2)=O)CCC2(C1)OCCO2.c12cccc(c1)C1(CC1)N2 c1(C(=O)NCC(CC(C)C)NC(C(CCC(C)C)O)=O)cc2cc(Cl)ccc2[nH]1 N1(C(C2CC23CC(F)(F)C3)=O)CCC2(C1)CN(C(C1(O)CC1)=O)CCO2 CC(C)(C)CCCCC(=O)N1CCC(N2CCNC(=O)C2(C)C)CC1 C(=O)(CCCn1cccn1)N1CC(CCNC(=O)COCC2CCCO2)C1 C(=O)(C1=NOC2(CCC2)C1)N1CCC(NC(CCOC)=O)C1C C12(C(N(C)CC3COC(=O)N3)=O)CCCCC1OCC2 CCC(C)CC(=O)N1CCC1CNC(=O)CCCc1ccc(Br)cn1 Cc1ccc(N2CCOCC2)c(CNC(C2CCCC(C)(C)C2)=O)c1 C(=O)(C1=CCCOCC1)NCc1c(C(=O)Nc2c(CC)ccnc2)occ1 N1(C(c2c[nH]c3cnccc23)=O)CCC2CC(C1)CN(C(C1SCCCS1)=O)C2 c1(C2C(NC(c3c(CCOC)occ3)=O)C2)ccc(Br)c(Cl)c1 N1(CC)CCCCC1C(=O)NCCCC(C)(C)NC(=O)CCC1CC(C)C1 N1(C(CNS(CCCC)(=O)=O)=O)CCN(C(=O)C(CO)NC(N)=O)C2COCC12 C1CN(C(C2(C(F)F)CCC2)=O)CC12CCC2.c1(NCC)cccc(C=O)c1.N C(=O)(C(CC)(CC)CC)NCC(N1CCN(C(C(CC=C)C)=O)CC1)C c1(N(C)C)c(F)cc(C(N2CC(N3CCC(N)CC3)C2)=O)cc1[N+](=O)[O-] c1(N2CCC(CC=C)(NC(=O)COCCC)C2)ncnc2c1ncn2C CC(CS(C)=O)C(=O)N1CC(CNC(=O)CCCCCc2ccccc2)C1 Cc1cccc(CC(=O)NCC2CCN(C(c3ccccc3)=O)C2)c1.C(N)(=O)N N#Cc1ccc(OCC(=O)NC2CCCC2)cc1.C1(CC(=O)N)CCCC(=O)N1 c1(CCC)nccn1CCC(=O)NCC(C1CCOC1)NC(c1coc(C)n1)=O c1(C(N2CCOCC(CNC(C3CC=CCO3)=O)C2)=O)ccc(=O)n2c1CCC2 c1(CC(=O)NCC2OCCCN(c3ncc(C#C)cn3)C2)ccc2cnccc2c1 c1(C2C(CCCN(C(C)(C)C)CCCC3CCOC3)C2)cncc(Br)c1 C1(C(C)NC(C2(C)CC=CC2)=O)CCN(c2cc(C(C)(C)C)ncn2)CC1 c1(N2CCCC(CCNC(C(CC)C(C)O)=O)CC2)nc2cc(C)ccc2s1 c1(C(N2CCC3CN(C(CCOC)=O)C3C2)=O)ccc(F)c2c1OCC2 C1(C(N2CC(C)(NC(=O)CC3CCC(=O)C3)C2)=O)(CC)CCOC1 c1(C(=O)NCCC2(C(=O)NC3(C)CCSC3)CCCC2)cc2ncccc2[nH]1 Cc1cc(C(=O)NCC(C)(O)CNC(c2nn[nH]c2C(F)(F)F)=O)sn1 C1(C(=O)NC(CC)(C)CCNC(c2cc(C(C)C)on2)=O)CC2CCC(C1)O2 C1(Cn2cc(C(C)C3CC3)nn2)CCCN(C(C2CSC2)=O)C1 C(=O)(CC(C)C(F)(F)F)NC1CCN(C(c2c(NC)ccc(F)c2)=O)C1 C1(O)CN(C(c2cnn(C(C)C)n2)=O)C1.CCS(=O)(=O)NCC(=O)NC Cc1nc(C(N2CC(CO)(NC(c3cnn(CC(F)F)c3)=O)C2)=O)nn1C N1(C(C(CC)=CCCC)=O)CCC(C(=O)N(CC(C)(O)C2CC2)C)CC1 c1(C(C)(C(=O)O)NC(C(C2CCC2)OC)=O)ccc(Br)c(C)c1 CC(C)CCC(C)(c1nnnn1CC1CCCO1)NC1COC1 c1(C(=O)OC)cc(C(N2CC3(C)CC2CO3)=O)cc(C)c1.C1(C=O)CC1.N C1(CCNC(CCOC)=O)CC2CCC(C1)N2C(c1c(OC)ccnc1F)=O N1(C(C2CC2)=O)C2CCC1C1CC1C2.C1(CC=O)CCCS1(=O)=O.CCO C1(CNC(c2cc(CC)[nH]n2)=O)CC(C(=O)N(C2CCC(CC)CC2)C)=NO1 c1(OC)ccc2[nH]c(=NC3CCCCC3NC3CCCCC34CCC4)sc2n1 C1(COC)CC(C)N(C(=O)C(O)C2CCC2)C1.C1(C=O)C(C)(C)C1(F)F S(=O)(=O)(c1cccc(=NCC2(O)CCC2)[nH]1)NC(c1c(CCC)nns1)C.C N1(C(c2ccn(CC)n2)=O)CCOC(C)C1.C(=O)(C(F)(F)Cc1ccccc1)N Cc1cc(C(N2CCC(C)(CC(N3CCC(c4cc[nH]n4)C3)=O)C2)=O)ncc1F C1(C(=O)NCCC(C)N(C(CC=C=C)=O)C)CC12CC(O)C2 C1(CC(=O)NCC(=O)N(C)CC)CCN1C(=O)C(C)=CC1CC1 CC1CC(O)CN(C(=O)CCOCCNC(c2cc(O)n(C)n2)=O)C1 c1(C(N2CCN(C3CCCOC3)CC2)C(=O)NCCC2CC2)ccccc1CO c1(CNC(C2(CC)COC2)=O)csc(C(N2CCC(c3ccncc3)C2)=O)c1 CC1CCN(C(c2cccc3cnsc23)=O)CCN1C(=O)CCCCNC(N)=O CCC(CC)C(C)C(=O)N1CCCC1C.c1ccc(F)cc1.C(=O)(C=CC=O)N S(=O)(=O)(C1CC12CCC2)NC1CC(C(C)(C)C)SC1 C=CCC(C(=O)NCCSCC(=O)NC)N(C)C.N12CCC(C1)C2C c1(CNC(c2nnn(C)n2)c2nnnn2C2CC2)c(F)ccc(F)c1Br N1(Cc2c(C(=O)OC)n(C)nc2)CCc2cc(Br)sc2C1 n1(CC(N2CCC3(NC(C=C(C)C(C)C)=O)C(C2)C3)=O)nc2n(c1=O)CCCC2 N1(C(c2cnc(OC)nc2)=O)CCC(C(=O)NCC2CC23CCOC3)C12CCC2 C1(C=O)CCC2(CCCCC2)CC1.C(C(C)C(=O)NCC12CC(C1)C2)SC.N c1(OCC)cc(Cl)ccc1C(N1CCC1)=O.C1(S(N)(=O)=O)(C=O)CC1.C C1(C=O)CCC2(CCC2)O1.N=c1[nH]c(CCC(=O)NCC2(F)CCC2)cs1.C c1(C(N(C2CCCC2)CCCNC(C(C(C)C)C)=O)=O)cc(Cl)cc(Cl)c1N N1(C(C2(CC#C)CCOCC2)=O)CCC(NC(c2nccn2CC)=O)C(O)C1 C(=O)(C(C(=O)NC(C)CNC(c1cnoc1C)=O)C(C)C)OCC C(=O)(CCC(C)(C)C#N)NCC1CC(OC)CN1C(=O)C(C)=C1CCC1 CCCC(C(=O)OC)C(=O)N1CCC(NC(c2cc(C)n(C)c(=O)c2)=O)C1 CC(C)CCCC(=O)NCC1CC2CCC1N2C(C1CC1C)=O Cn1cc(-c2nc(C3CSc4ccccc4O3)no2)n2cncc2c1=O C(CC(C(=O)NCCCC1CCOCC1)NC(=O)CCc1nncs1)OC O(NC(=O)C(C(C)(C)C)NC(C1CC(N=[N+]=[N-])C1)=O)C(C(=O)OC)C c1(OCC)ccc2c(c1)CN(S(=O)(=O)c1ccc(OCC3CCCC3)cc1)CC2 c1(-c2nnc(C(C3CCN(C(C4(C)CC4(Cl)Cl)=O)CC3)=O)s2)cc(F)cc(F)c1 c1(CC(=O)OCC)sc(C(C)NCCN2CCCCC2)nc1C CC1CN(C(C2CCCCN(C(=O)CC(C)(C)C3CC3)C2)=O)CCS1=O C12(NC(=O)CN3CCC(O)CC3)CCCCC1CN(C(c1ccsn1)=O)C2 CC(C)(O)C(=O)N1CCC(C2CCCN2C(=O)CC2CC(=O)C2)C1 C=CC(C)(C)C(=O)N1CCCC(NC(=O)CSCc2csc(=N)[nH]2)C1 c1(OC)ccc(OC)c(C(=O)NC2CCC2NC(=O)CC)c1.C(=O)CO.N c1(C(N(CC)CC)=O)ccc(C)cc1.N1(C(c2ccc(F)o2)=O)CCCC1.S C1(N(C(CSC)=O)C)CCC(NC(=O)Cc2c[nH]nc2C)C1 C1(N(C(C2SCCCS2)=O)C(c2ccccc2)C)(CC)CCCC1 Cc1cc(C(=O)N(CC(C)C(=O)NCc2nc(C)c(C)s2)C)cc(C)n1 c1(C(=O)NC2(C(N3CCN(C)C(=O)C3)=O)CCN(C)C2)ccc(O)cc1F Cc1cc(C(N2CCC(O)CC2)C(=O)NCCCC2CC2)cc(Cl)n1.C(C)(C)C c1(CNC(C(CNC(C=C(C)C(C)(C)C)=O)O)=O)cc(C)ccc1O O=C1CCC(C(=O)NCCC2CN(C(=O)CCOc3ccccc3)C2)C1 N1(C(C2(C)CC(NC(CCC#CC)=O)C2)=O)CC2(C1)OC(=O)NC2C N1(C(C2(F)CCN(C(C3(OC(C)=O)CC3)=O)C2)=O)CC(S(C)(=N)=O)C1 C(CCC)(CCCNC(=O)CC1CCCN(CC(F)(F)F)C1)NC(C=CC)=O O(C=CC(=O)NC1CN(C(=O)CCO)C1)CC.n12cc(nn1)C2.C1CCOCC1 c1(C(N2CCC(NC(C(C)NC(C)=O)=O)CC2)=O)c(O)nnc(C)c1C C1C=CCN(C(=O)C(c2ccc(C(F)(F)F)cc2)F)C1.O=CCC1(CO)CC1.N c1(CNC2C(C(=O)NCCCCO)C2)cccc2c1oc1ccccc21 CC1CC(NC(=O)CSc2ccccn2)CC(C)O1.C(=O)CCN1CCC1C N1(C(c2coc(Br)n2)=O)CCCC(O)(CNC(C2CC(O)C2)=O)CC1 C(=O)(CCCC(C)(C)C)NCC(C1CCCCN1C(c1cc(C(F)F)[nH]n1)=O)C C=CC1(C(=O)NC2CC3(C2)CC3F)CN(C(=O)OC(C)(C)C)C1 C(CC(=O)NC1CC(C)(C)C12CC2)(C(F)F)NC(C1(OC)CC(C)C1)=O CC1CC(C(=O)NC(C2CN(C(=O)CSC(F)(F)F)C2)C)C(C)O1 N1(C(c2c(C(C)C)[nH]cc2)=O)CCN(C)CC1CNC(=O)CCCn1ccnc1 c1(C(N2C(C3CCN(C(C)=O)CC3)C(C)(C)C2)=O)ccc(Br)c(C)c1 C(=O)(CC(C)(C)CC(F)F)NC1C(C)CN(C(c2ccc(C3CC3)nc2)=O)CC1 C1(NC(C2C(C(C)C)(CC)C2)=O)CCOCC1NC(c1ccno1)=O.C c1(CC)ccc(F)c(C(=O)NC)c1.C1(C(N2CCCCC2)=O)CC(C)(C)CN1C CN1N=C(C(=O)N2CCC3(NC(c4ccnc5ccsc45)=O)CC3C2)CCC1=O C1(C(=O)NC2(COC)CN(C(C3CNC(=O)C3)=O)C2)CC12CCCC2 c1(CCC(N2C(CN(C)C(C3CCC3CF)=O)CCC2)=O)cccc(Cl)c1 c1(N2CCC(NC(C(c3cccc(Cl)c3)C)=O)C2(C)C)nc2cc(F)ccc2o1 CCCC(C(O)C(=O)NC(CC1CC1)C1CC1)NC(c1n[nH]c2c1COC2)=O N1(C(CC(CCC)NC(c2cc([N+](=O)[O-])c[nH]2)=O)=O)CCN2CCCC2C1 C1(NC(c2cnc(C)o2)=O)CS(=O)(=O)CC1NC(c1ccn(C)c1)=O C1(NC(c2ccc3c(c2)nnn3C)C)COc2ccccc2N(C)C1=O c1(C(=O)NC2C(NC(c3c(CC)n(C)cc3)=O)C2)ccc2nccnc2n1 Cc1cccc(C2CCN(Cc3cc(C)[nH]n3)C2C(=O)O)c1 c1(OC)ccc(C(=O)N(CC(O)CNC(c2nc(CN)sc2N)=O)C)nc1 c1(N2CCCC(=C)C2)nc(=NCc2cccc(Cl)c2)[nH]c2ncn(C)c12 CC1CC(NC(c2cccnc2N2CCOCC2)=O)CN1C(c1cc(F)n[nH]1)=O c1(SC)ccc2cc(C(N3CC=CC(NC(c4ccncc4Cl)=O)C3)=O)[nH]c2c1 c1(CCC(=O)NCC(CNC(C2(F)CCCC2)=O)CO)ccc2cccnc2c1 O=C(C1=NN(c2cccc(F)c2)C(=O)CC1)NC1CCN(Cc2cccnc2)C1 Cc1cc(F)c(Cl)cc1C(=O)N(C(C)C1CC1)C.C1(C=O)CCN(C)C(=O)C1 C(=O)(C1=CSCCO1)NCCOCCNC(c1cc(C)nn1C)=O N1(C(C(F)=CC)=O)CCCC(CNC(C2CCCCC(=O)N2)=O)CC1 c1(SCC(N2CCC(N(CCC)C(c3scc(C)c3C)=O)C2)=O)ccccc1O c1(C(=O)NC2C(NC(CC(C(C)C)O)=O)CCCC2)n[nH]c2nccc(Cl)c12 N1(C(COCC=C)=O)CC(NC(=O)Cc2ccccc2SC)C(C)C1 c1(CNC(CCC)C2CCCC2)cc(OC)cc(Br)c1 c1(NC(N(CCCC=C)C(C)(C)C)=O)ccc2c(c1)c(=O)c(Br)cn2C C1(CN(C(=O)OCC)CCO)CCCN(C(C)CSC(C)(C)C)C1 Cc1cnc(NCc2ccncc2F)c(S(=O)(=O)N2CCC(O)C(F)C2)c1 Cc1nn2ncccc2c1C(=O)NCCC(C)N(C(=O)CC1COC(=O)N1)C N1(C(CCC(CC)C)=O)CCC(NC(=O)C=CC2CCCCC2)C(C)(C)C1 C1(O)(C(=O)NC(CCCNC(C2(COC)CCC2)=O)CO)CCC(C)CC1 C(CCN=C(NCC1CCOC(C)(C)C1)NCC1(CO)CCC1)SC C1(C(=O)O)CC2(C1)CN(C(=O)Cc1cccc(Cl)c1)C2.CC(C)C.C(N)=O C1(C(=O)NCCC(=C)C)CCN(C(=O)C=Cc2ccncc2)CC1 C1(NC(c2[nH]cc(CN(C)C)c2)=O)CCC(O)C1.C(=O)CC(C)n1cccn1.N C(=O)(CCCCCN1CCOCC1)N.C1(CNC(COC(C)C)=O)COC(C)C1 Cc1nc(N)c(CC(=O)N(C(C)CCNC(C2(CO)CC2(F)F)=O)C)c(O)n1 N1(C(C=C(COC)C)=O)Cc2ccccc2CC1CNC(=O)C1=COCCO1 C1(NC(C(CC=C)C)=O)CC12CCN(C(=O)C(CC=C)C(C)C)CC2 C1(CC)(NC(C2CCC(O)CC2)=O)CCN(C(=O)C(CO)OC)CC1 Cc1ccc(NC2CC3(C2)CN(S(=O)(=O)C2CCCCC2)C3)c2cccnc12 N1(C(C(C)CN(C)C)=O)CC2COCCC2(NC(c2nc(C3CC3)cs2)=O)C1 C(=O)(C1=CC2(CN(C(=O)Cc3ccc(C#N)cc3)C2)OC1)NCC(C(C)O)C C1(CC)CN(C(=O)CCCC(C)C)CCN1C(c1ccc(O)cc1O)=O c1(OCC(N)=O)ccccc1C(=O)NC1CCCC(NC(c2csnn2)=O)C1 C1(C)(C(=O)Nc2c(C)cc(N)cn2)CC(C(F)(F)F)=NO1 c1(N2CCC(F)(C(=O)NC)C2)nc(=N)[nH]c(=NCCC(C(C)C)N(C)C)[nH]1 c1(N2CC3(OCC(NC(C4(CCO)CC4)=O)C3)C2)ncnc2cccnc12 N1(C(C(=O)NCC(C)(C(F)(F)F)OC)=O)Cc2c(F)cc(Br)c(Cl)c2CC1C c1(CNC(CC=C=C)=O)cnn2c1CN(C(c1cn(CCC(C)C)nn1)=O)CC2 c1(C(N)=O)ccnc(CNc2cn(C)nc2)c1.c1(C2(C=O)CC2)cccs1 C1(NC(C(C)C2CCC2)=O)CN(C(=O)COc2ccc(Cl)cc2)C2CCCCC12 c1(NCC(C(C)(C)C)NC(=O)CCCn2ccnc2)cccc(F)c1C#N C(C(CC(F)(F)F)NC(=O)Cc1cccc(Cl)c1F)NC(C(C(C)C)OC)=O c1(C(C)NC(=O)COC(c2nocc2C(C)(C)C)=O)ccc(Br)s1 Cc1ccc(NC(=O)CC2CCCC2)cc1C#N.C1(CC=O)CCC1.C(C)C.N C(CC(C(C)(C)C)NC(=O)CCn1cnc(=N)[nH]1)N(C(=O)C#CC1CC1)C C1(CC)CCCN(C(C2(NC(c3ncoc3C)=O)CC2(C)C)=O)C1 c1(CC(=O)N)ccc2sccc2c1.c1(OC)cc(C(=O)NC(C)CC)cc(F)n1 c1(OC)cccc(NC(=O)C(C(C)O)NC(C2CCNC2=O)=O)c1 c1(-c2nc(CC34CC(C(F)(F)F)(C3)C4)on2)cc(F)c(F)cc1Br C(=O)(C(C)(C)C(=O)N1CC2CCC2(CC(=O)NCCCC(C)C)C1)NC N1(C(C2CCC(C(C)C)CC2)=O)CCN(C(c2ccn(C(C)(C)C)n2)=O)C(C)C1 C1(CC(=O)NC(C2CCN(C(=O)CN(C)C3CC3)C2)C)(CC=C)CCCC1 N1(C(Cc2nc(C)sc2C)=O)CCC(NC(C2NC(=O)C3CC23)=O)C(O)C1 C1(NC(=O)NC(C(=O)OCC)C)CC2CC2N1.c1ccc(-c2nn[nH]n2)s1 c1(C(C)O)ccc(C(=O)N(C)CC2CCCN2C(=O)CCCC2CCCO2)cc1 N1(C(C2=CCC(NC(CCC=CC)=O)C2)=O)CC2CCCC(C1)N2C CCC(C)(C)CC(=O)NC1CC(C)(NC(c2ccc(-c3ccco3)nn2)=O)C1 C1(CC(=O)NCC2(CC)CCCO2)CC(C)(C)CN1C(c1cncs1)=O CCCC(C)(CC)C(=O)N(C)CC1CCN(C(c2cscc2OC)=O)CC1 CC1CS(=O)CCN1C(=O)CC(C)(C)NC(=O)COCC(F)F N1(C(c2c(C)cc(O)cc2C)=O)Cc2nccn2CC(NC(c2cnsn2)=O)C1 c1(C(=O)Nc2ccc(NC(C(C(C)C)O)=O)cn2)c(F)ccc(I)c1F C1(NC(Cc2ccc(C)s2)=O)CC2CC(C1)N(C(c1ccc(Br)o1)=O)C2 c1(C2(C(=O)NC(CCNC(C=NOC)=O)C)CC2)cc(C)cc(Br)c1 C1(c2noc(CCC=O)n2)CCCC1.C12(SCC)CC(CCC(F)(F)F)(C1)C2.N C1(NC(c2ccc(C)o2)=O)CCCC(NC(=O)C(C)NC=O)C1 c1(CNC(N2CCC(N(CC(C)C)C)C2)=O)cncc(S(C)(=O)=O)c1 c1(CC(C)C=O)cccc(Cl)c1.C1(CCC(=O)O)CC2(CCC2)C1.C1CCOCC1.N C1(C(N2CC(O)(CNC(c3cn(CCO)nn3)=O)C2)=O)CCc2nncn2C1 C(CC1=CCN(C(=O)CCCc2ccccn2)CC1)NC(c1ncccc1F)=O Cc1n[nH]c(C)c1CN1CCCC1CC(=O)NCC(c1ccco1)O C(=O)(C#CC1CCOCC1)NCC(CC)NC(c1cc[nH]c2nccc1-2)=O CC(C)C(F)(F)CC(=O)NC(CC(C)(F)F)C(=O)O c1(C(C(=O)NCC2CN(C(=O)CCC3CC3)C2)O)ccccn1 N1(C(C(C=C)OC)=O)CCCC(NC(C2CCOCC2(C)C)=O)C1CC N1(C(c2cncc(C)c2C)=O)CCC(C2CC2NC(=O)C(F)CC2CCC2)CC1 n1(CC(=O)NC2CC(C)(C)CN(C(=O)C3CC3)C2)c(S)nc2ccccc2c1=O C(C(C)(C)CC(=O)NCCC1CCN(C(=O)CCn2ncn(C)c2=O)C1)N(C)C C1(C)(C(=O)NC(CN(C(C(C)OCCOC)=O)C)C)COCCO1 CC1(C)CCC(C(=O)NCC2CC2C)CO1.c1(C=O)cc(C(F)F)ncn1 c1(N2CC3C(C(=O)Nc4cc(F)ccc4Cl)C3C2)cc(C2CC2)nc(Cl)n1 C(=O)C(C)CC(C)(C)C.C(=O)(C(F)C(=O)NC12CC(C1)C2)OCC.C Cc1cc(C2CC2)cnc1C(N1CCC(NC(=O)C(C)(C)C#N)C1C)=O C1CS(=O)(=O)CC1.c1ncccc1F.C(=O)C(C)(C)C.CP(C)(=O)COCC=O C1(C(=O)NC(CCC)(C)CC)C2CC(O)C(C2)N1C(=O)CSC1CC1 C12(CN(C(=O)NC(c3cccc(OC)c3)C)CC)CCCCC1C2 Cc1ccc(C=CC(=O)NC(C2CCCCC2)CNC(=O)C(C)O)o1 C(C(CC(C)C)NC(c1sccc1CC)=O)NC(CNC(=O)OCC)=O C1(NC(C2(C)CC=CCC2)=O)CC2CC(NC(c3ccc(CO)o3)=O)C1C2 C1(C(N2CCC3CN(C(c4ccc(Cl)cc4F)=O)C3C2)=O)CC12CCCCCC2 N1(c2cnc3nc(C)sc3n2)CCC(C2CCCN(Cc3ccccc3)C2)CC1 C12(CNC(N(CCC(F)(F)F)CC)=O)CC1CCN2C(=O)O.C(C)C N1(C(CSCC#C)=O)CCC(O)(C(C)CNC(=O)C(C)(C)N(C)C)C1 N1(C(c2n(C(C)C)ncn2)=O)CCN(C(c2ncoc2C2CC2)=O)CC1C1CC1 c1(NC(CCN(C(CCCCC)=O)CC)=O)ccc(F)cc1OC c1(CC)ccc(C(=O)NC2CCCCC2)cc1.C(=O)(C=CSC)N.C1(C)CCCC1 N1(C(=O)C2CC2)CC2(C(=O)N(c3ncnc4sccc34)CC)CC1CCO2 Cc1c(C(N2CC3CC2C3NC(=O)C(C)C(C)S(C)(=O)=O)=O)ccc2cncn12 N1(C(c2cc3sccc3[nH]2)=O)CC2CCN(C(c3cnccc3Br)=O)C2C1 C1(N(C(=O)C)CC)CCN(C(=O)CC)C1.c1ncc(C)[nH]1.C(C)CC(C)C.O N1(C(C)=O)CCC(F)C(NC(c2cc(Cc3cc(C)cc(C)c3)nn2C)=O)C1 N1(C(c2c(C(C)C)onc2)=O)CC2CCC1CN2C(C1CCOC1)=O N1(CC(N2CCCC2(C)C)=O)CCCCCCC1=O.CC(CC1CC1)C(=O)NC CC1CCCC(C(=O)NC2CCC(C(=O)NC(C)(C)C(=O)N(C)C)CC2)CC1 c1(C(N2C(CCC(C)(C)NC(C3C(C)C3)=O)CCCC2)=O)cc2sc(Cl)cc2[nH]1 CC(C)(Cc1ccc(Cl)cc1)CC(=O)NCC1CC1.C1(C)(C=O)CCOC1.N c1(CC)cc(C(=O)NC2CC(CC)C2)c2c(c1)CCO2.c1(C=O)nocc1C.N CC1(C)CCC(C(N2CC(C(N3CC4CC4C4CC34)=O)C(C)(C)C2)=O)CC1 c1(C(=O)NC(CNC(CCCCCN(C)C)=O)(C)C)cc2c(s1)CCCNC2=O N1(C(CC2N(C(CSCCCC)=O)CC3(CC3)C2)=O)CCn2nccc2C1 CCCCCC(O)C(=O)NCC1CCC(NC(c2nc[nH]c3nccc2-3)=O)CC1 C(CCCC(=O)N(C(C)CCNC(=O)CCc1ncccc1C)C)OC C(C(=O)N)(C(C)O)NC(C)=O.c1(C=O)cc(C(C)=O)c(C)o1.C1CCCC1 Cc1cc(=O)n(CCC(N2CC(NC(C3CC4(C)CC3CO4)=O)C(O)C2)=O)cn1 C=CCCCCCCC(=O)N1CCN(C(C2(C)CS(=O)(=O)C2)=O)CC12CCC2 N1(C(Cc2c(C)con2)=O)CCCC2C1CCN2C(=O)Cn1nc(C)cc1C(F)F c1(C(=O)O)cccc(CCN2CCOCC2c2ccc(Cl)cc2)n1 c1(NC(N2CC3CCN(C(c4c(C)ccs4)=O)C3C2)=O)cccc2nccnc12 C1(C(N2C(CN(C(=O)CCC3(O)CCC3)CO)CCC2)=O)CCc2ncncc2C1 C1(C)(CNC(C2N(CC)CCC2)=O)CCCN(C(C2SCC=C2C)=O)C1 N#Cc1ccc(NC(C2CC2NC(c2ccc(F)c(O)c2)=O)=O)c(F)c1 c1(C(=O)NCCC(C)NC(C(C(C)C)n2cncn2)=O)ccc2[nH]ccc2c1 c1(NC(C2CC23CN(Cc2cc(Cl)cnc2F)C3)=O)ccc2nc[nH]c2c1 C1(OC(C)C(=O)NC2(CF)CN(C(C3CC34CC4)=O)C2)CCCCC1 C1(NC(C(C)OCCC#C)=O)CC(C)(NC(=O)COC2CCCCC2)C1 Cc1cccc([N+](=O)[O-])c1C(N1CCC(CO)CC1)=O.C(=O)(C(F)=C1CCC1)N n1(CC(=O)NCC2CN(C(C3(CO)COC3)=O)C2)cc(Br)ccc1=O CC(C12CC3CC(CC(C3)C1)C2)=CC(=O)NC1Cc2cccnc2C1 C1(N(C(c2nccc(C)n2)=O)C)CCCN(C(C2CCCC(O)C2)=O)CC1 CC1CN(C(C2CN3CCN2CC3)=O)CCN(C(C2(C)CC2(Cl)Cl)=O)C1 c1(CC(=O)NCCC(=C)CNC(c2ncoc2C)=O)cccc(CC)c1 C#Cc1cc(F)c(C(=O)NC2CC(F)(F)CC2NC(=O)C(F)F)cc1F N1(C(=O)Cc2ccc(F)cn2)CCCN(Cc2cnc(Cl)c(Cl)c2)CC1 C1(NC(c2cc(CNC(C(C)OC(C)=O)=O)[nH]n2)=O)CCC(CCO)CC1 CC(CC(C)(C)O)NC(=O)C(C1(C)CC1)NC(c1cccnn1)=O C(=O)(C1SCc2cccnc21)N1CCN(C(CCCN(C)C)=O)C(CCO)C1 C1CC2CCC(C1)N2C(c1ccc(C(F)F)nc1)=O.Cn1nccc1C(=O)NC C1(OCCNC(CCN(C(CCC)C)C)=O)CCN(C(=O)C(C)(C)F)C1 C=CC(CC(=O)NC1CC1CNC(=O)Cc1cn[nH]c1)c1ccon1 c1(C(N(C(C)CN(C)C(C2(O)CCOC2)=O)C)=O)cccc(OC2CCC2)c1 CC(C(=O)Nc1cc(Br)ccc1N1CCCC1)C(C)S(C)(=O)=O c1(CC)cc(NC(=O)C(CCF)NC(c2c[nH]ccc2=O)=O)cnc1C C1(C(N2CC(C#C)C2)=O)CCN(C(=O)C=CC(C)CC)C(CC)C1 CN1CC(O)CC1C(=O)NCC(N1CC(O)C(O)C1)=O c1(OC)cc(C(N2CC(C(N3CCOCC3)=O)C2)=O)ccn1 C12(CC(=O)N(CCNC(c3c(CC)cccc3)=O)C)CCC(CC1)OC2 Cc1ccc2nonc2c1C(N1CCC(O)(CNC(C2(F)CCCOC2)=O)C1)=O n1(CC(=O)NC2(CNC(C3C(C)(C)CO3)=O)CCOC2)ncc2ncccc12 C(CC)(CC)(C(C)C)NC(CCN(C(C=CC)=O)CC)=O C12(C(N3C4CC(C4)C3)=O)CCCN(CCC1)C2.C1(C(=O)NC)CC12CC2(F)F C(=O)(C(C)(C)CCCO)NCC1CC(C)N(C(=O)CCc2ccc(Cl)nc2)C1 N1(C(c2ccc(F)c(C(F)F)c2)=O)CCC2CCN(C(C3CC=CC3)=O)C2C1 C1(CNC(C=CC(C)=O)=O)CN(C(=O)CCC2CC(C)(C)CO2)CCCO1 CC1CC=C(C(=O)NC(CN(C(=O)CO)C)(CO)CO)CC1.c1cccc(F)c1 CN1CC2CC1CN(C(C1(Cc3cccc(Cl)c3)CCOCC1)=O)C2 c1(OC)cc2c(cc1OC)N(C(=O)NCC1COC(C)(C)O1)CCC2 C1CC2(CCN(C(C34CC5CC(C(=O)N3)C4C5)=O)CC2)C1.C1(C=O)CCCO1.N C1(C)(CCNC(CN2CC(C)C2)=O)CCN(C(c2ccoc2C(C)C)=O)C1 C1(C)(CC)CC(NC(c2ccc(=O)oc2)=O)CN1C(c1cn(C)ccc1=O)=O c1(C(C(=O)Nc2ccccc2)N(C)Cc2cc(CO)on2)cccn2ccnc12 C1(CNC(C(C2CC2)OC)=O)CCCCC1.c1(C(=O)N)ccon1.C1CC1 c1(CC)ccc2c(CC(N3CC=CC3CNC(C3CC(F)C3)=O)=O)coc2c1 c1(C(=O)NCCCCN(C)C(C2(C3CC3)CCCO2)=O)ccc2ncncc2c1 N1(C(c2c(CC)ocn2)=O)CCCC(C(C)(O)CNC(c2cnns2)=O)C1 c1(C(N2CCC(NC(CCC(C)OC)=O)C2(C)C)=O)cnc2ccc(C)cc2c1 CN=c1cc(C(=O)NCCNC(C2CC(C)C2(C)C)=O)c(Br)c[nH]1 CCCS(=O)(=O)CC(=O)NC.c1(CC(N2CCC(F)C2)=O)cn2c(C)csc2n1 N1(C(C2C(C)(C)COCC2)=O)CCC(NC(c2csc(O)n2)=O)C2(CCC2)C1 Cc1nc(NCc2cc(C(C)(C)C)ccc2O)ccc1Br CC(C(C)(C)C(=O)NC1CCCCNC1=O)NC(C1CC(C)(C)C1)=O N1(C(c2cncc(-c3c(OCCCC)cccc3)n2)=O)CCC(O)C(F)(F)C1 C1(CNC(=NCCc2ccc(OCC)cc2)NCC)CCNCC1(F)F.C1CC1.O N1(C(Cc2c(C)ccnc2)=O)CC2(CCCC2NC(=O)CCCF)C1 c1(C(C(=O)OC)NCC(=O)N(CCOC)CC)ccccc1I C1(NC(C2(C)COC2)=O)CN(C(c2cc(Cl)ccc2F)=O)C2(CCOC2)C1 C(C(CC(=O)NC)NC(c1cn[nH]c1)C)NC(C(CC1CC1)OC)=O c1(C(=O)NCC2(C)CCN(C(=O)C(O)CC(F)(F)F)C2)c(F)ccc(Cl)c1N C1(NC(c2c(C(C)C)ocn2)=O)CCCCC1NC(=O)Cc1sc(O)nc1O C1(CNC(c2c(CC)cccc2)=O)CCC(C)N(C(c2cscn2)=O)C1 C(N=c1[nH]cnc(N)c1I)C1(c2cc(C)cc(C)c2)CCC1 c1(CCC(=O)NCC(CC)NC(c2c(CC)c[nH]n2)=O)cc(C)nc(C)c1 C12(C(=O)NCC=CCNC(CC3C(C)(C)C3(C)C)=O)CCC(CC1)CC2 C(=O)(C1Cc2ccc(F)cc21)NCC(CCNC(c1ccc(F)cc1)=O)OC C(=O)(C1CC(=O)Nc2cc(F)ccc21)OCc1onc(C)c1Br C(CCCCCC(C(=O)NCCC1(C)CC1)N1CCNC(=O)CC1C)OC(C)=O c1(C(N(C)CCO)=O)ccc2c(C(=O)Nc3nccc(F)c3F)n[nH]c2c1 c1(Sc2ccc(-c3n(C)nnc3)cc2)cc(N2CCSCC2)cc(Cl)c1 c1(CCC(=O)N(CCN(C(C(F)OC)=O)C)C(C)C)cc(C)ccc1Br CC(=O)CCC(=O)NC(c1ccnn1C)C(=O)NCCc1cnc(C)o1 c1(C(N2CC(CNC(c3ccc(O)cn3)=O)C2)=O)c[nH]c2ncc(Br)cc12 c1(CN2CCC(N(C(=O)CC)CCC)C2)ccc(O)nn1.C(=O)C.C(C)=O c1(OCC)ccc(CN2CCOC(CC(=O)NCc3cn[nH]c3)C2)cc1 Cc1ccc(CN2CCC(O)(CNC(C)C)C2)c(C)c1 C(=O)(C1=Cc2ccccc2C1)N1CC(CCCCNC(c2cncnc2)=O)C1 CCCC(C(=O)N(CCCCNC(=O)C(c1ccc(F)cc1)O)C)NC(C)=O N1(CC(C)C)CCN(C(C2(CCN(C)C)CC2)=O)CC1.C1(C=O)CCOC1.C CON(CC(=O)O)C(=O)N(CC(c1ccc(Br)cc1)O)C1CC1 C1(CNC(c2ccccn2)=O)CN(C(c2ccco2)=O)CC(C(F)(F)F)O1.C C1(OC)(CNC(c2cc(Cl)n[nH]c2=N)=O)CCN(C(C2CCOCC2)=O)CC1 C1(CN(C(=O)C2=COCC2)CC)CCN(C(c2cn(CCCF)nn2)=O)CC1 C12(CNC(Cc3onc(C)n3)=O)CC1CN(C(C1(c3ccccc3)CC1)=O)C2 c1(NC(CC(CC)C)=O)ccc2c(c1)CN(C(c1cnc(C)nc1)=O)C2 C(=O)(CC1=CCN(C)CC1)N1CCN(C(c2cn(CC)nn2)=O)CC(O)C1 C1(CN(C(=O)CC23CC(C2)C3)C)CCN(C(=O)C(C)(C)N(C)C)C1 c1(C(N2CCC(CCN(C(=O)CCSCC(N)=O)C)CC2)=O)ncncc1C#N N1(C(=O)NCC(C)CCCO)CCCC2(CCNC2=O)C1 c1(C(=O)NC2CCC(C)(CNC(=O)CCS(C)(=O)=O)C2)ccc2c[nH]nc2c1 C(C(CC(=O)NCCOCC(N)=O)NC(C1CCC(=O)N1)=O)OC c1(CN(C(=O)CCN2CCCCC2C(=O)O)C(N)=O)nc2ccc(F)cc2[nH]1 C#CC1(C(N2CCN(C)CC2CO)=O)CCN(C(=O)CC(C)(C)N(C)C)C1 c1(NC2C(C(F)(F)F)CCN(C(C(COC)C)=O)C2)c([N+](=O)[O-])c(C)n[nH]1.C c1(C(N(C2CCCN(C(CC=C)=O)C2)CCOC)=O)cc(O)cc(Cl)c1 CCC(CO)(C(=O)N(C1(C(=O)NCc2cc(C)cc(C)n2)CC1)C)OC c1(C(=O)OCC)sc2c(c1C(=O)Nc1nccnc1N(C)C)CCCC2 C12(NC(Cc3n(C)ncc3)=O)CCC1CN(C(=O)C(F)(F)c1cncs1)C2 c1(NCC2(CCNC(C3CCSC3)=O)CC2)c(F)cc([N+](=O)[O-])cc1F C(c1ccc([N+](=O)[O-])s1)=CC(N1C(C)CCC1)=O.Cc1nc(C)c(C(=O)N)o1 c1(C(=O)NCC(n2cc(CC(CC)(C)O)nn2)C)cnc(OCC(F)F)cn1 c1(CNCC(CC)Oc2ccccc2C#N)cc2ncccc2s1 N1(C(C(F)NC(c2nncs2)=O)=O)CCN(C(=O)CN2CCCC2)C(CCO)C1 C1(NC(Cn2c(C)ccn2)=O)CCCCN(C(=O)CCCC2CC2)C1 c1(OC(C)C)cccnc1C(=O)NC(C)CN(C(=O)CC(C)c1cccnc1)C N1(C(c2n[nH]c(C)c2O)=O)CCC2(CC1)CN(C(=O)CC1CC1)CC2CO C1(CCC)CN(C(C2CCC(C(C)(C)C)CC2)=O)CCN1C(=O)C=C(C)Cl C(=O)(C1=NN(C)C(=O)CC1)N(CC(C)CNC(c1nc[nH]c2ncnc1-2)=O)C CC1CN(C(=O)CCc2cc(Cl)cs2)CC1NC(=O)CC1(C)CCCC1 c1(CNCCS(N2CCCC(CSC)C2)(=O)=O)nc(O)c2ccccc2n1 c1(N2CCC(C)N(Cc3ccccc3)CC2)ccc(N=S(C)(C)=O)cn1 n1(CCC(=O)N(CC(C)NC(c2ccnc(O)c2)=O)C)cc[nH]c(=O)c1=O N1(C(CCC2CCN(C)C2)=O)CCC(NC(c2ccc(OC(F)F)nc2)=O)CC1 CCCCCC(F)C(=O)NCC1COC(C)(C)CN1C(C1CC=CCO1)=O CC1=C(C(=O)N2CC(NC(=O)C(O)C(F)F)CCC2C)CCC1 Cc1cc(CC(N2CCC(CO)(NC(C3CC3C)=O)C2)=O)ccc1CO N1(C(Cc2cc(COC)on2)=O)CCOC2(C1)CN(C(C1CCCC1O)=O)C2 N1(C(=O)CCOC2CCOC2)CCC2(CCCN(C(C3(CO)COC3)=O)C2)C1 CN1CC(F)CC1C(=O)Nc1cccc(NC(=O)CC2CC3(CC3)C2)c1 C(=O)(NNC(=O)COC)C1(OCC)CCOC1.c12ccccc1C(=O)N2 c1(C(=O)NCC2C(C)CN(C(C3CC4CCCC34)=O)CC2)ccc(F)c(C#N)c1 Cc1ccc(C(N2CCC3(NC(=O)CCCCC(C)C)CC3C2)=O)c(O)c1C C(CC(O)C(=O)N(CCF)CC)NC(C(CC)N(C)C)=O CCCCN=C(NCc1ccc(C)nn1)NCC1CCCC(=O)N1 n1(COC)ccc(C(=O)NCCC(C)NC(C2(CC3CC3)CC2)=O)n1 C(C=O)N(C)CCN(C(C1CC1C(C)(C)O)=O)C.C1CCC1.CC=C C1(C(=O)NCC(=C)CCNC(C2(CO)CCCC2)=O)CCC2(CCOC2)O1 C(CCN(C)C(C1CCC1(F)F)=O)(C(C)C)NC(C1(OC(C)=O)CC1)=O c1ccc(Cl)c(F)c1.Cc1c(C(=O)NCCN(C(=O)CF)C)cnn1CCO.O Cc1ccc2nsnc2c1C(=O)NC1COCC1NC(c1cc(F)ccc1O)=O CCCCCC(C)CC(=O)NCC(O)CC(=O)NC1CCC2(C(C)C)CC12 C1(C)(C)CC(=O)O1.n1(CC)ccc(CN2CCCC2Cc2cncn2C)n1 C(=O)(C(O)CC(F)(F)F)NCC(C(N1CCC(C2(C)CC2)C1)=O)(C)C C1(OCCNC(CNC(CC)C)=O)CN(C(C2CC(C)C2)=O)C1.C1CC1 N1(C(=O)OC(C)(C)C)CC=CCC1.c1(CCC=O)ccc(Cl)nc1.C1(N)CC1 Cc1cc(CN2CCC(C(=O)Nc3cnns3)C2)cc(C)c1Cl Cc1cc(N(C2CCCN(C(c3ccc(=O)n(C)c3)=O)C2)CCO)nc(C)n1 N1(C(c2c(C)snn2)=O)CC(NC(=O)CCc2ccc(CO)cc2)CC2(CC2)C1 C=C(C)C1OCCC1C(=O)N(C1CCCN(C(c2conc2C)=O)C1)CC Cn1cnc2cc(CC(N3CC4CC4(CNC(=O)CC4CCCC4)C3)=O)ccc12 C12(C(=O)NCCC3N(C(CCCC(C)O)=O)CCSC3)CCC(F)(CC1)CC2 Cc1cc(NC(=O)C(C2CCCC2)NC(C2CCN(C)CC2)=O)ccc1F C(CCCCCCCN)NC1(C(C)(C)C)CCC(F)(F)CC1 N1(C(c2ccc(CC)cc2)=O)CC2CCC(Nc3ccnc(CC4CC4)n3)CC2C1 C(=O)(CC(CN(C)C)C(F)F)N1CC(CCCC)N(C(=O)CCCC2CC2)CC1 C1(C(=O)NC2C(C(=O)NCCC3CCOCC3)OCC2)CCC(C2CC2)C1 C(=O)(C1=C(Cl)CCCC1)NC1(CN(C)C(C23CCN(CC2)C3)=O)CC1 C1(C(N(C)CC2CCN(C(c3nnc(C)s3)=O)C2)=O)CC(=O)NC1.C1CC1.C C=Cn1nncc1C(=O)NC1CC(NC(C2(C)CC2)=O)CC1O.c1ccccc1 CN1CCC(C#N)(C(=O)NC2CCCCC2N(C)C(C2CC(N(C)C)C2)=O)CC1 C1(C#CC(=O)NC2CCCCC2)(CC)COC1.c1(CC=O)cncn1C1CC1.N CC1CCCCCC1NC(=O)CC1CC(NC(c2ccccc2N(C)C)=O)C1 CC(C)C(C(=O)N(CCCO)C)NC(=O)CC1(C)CC1 c1(C(=O)NCC2N(C)CCN(C(CCCCSC)=O)C2)cc2cccnn2n1 C(=O)(C1=CC2(CCOC2)C1)NC(CCC)C(=O)Nc1cnc(C)c(Cl)c1 N1(C(C(CC=C)CC)=O)CCC(=O)NC2CN(C(c3ccoc3Cl)=O)CCC12 c1(SC)ncc(C(=O)NC(C)(C)C2CC2)n1C.N1(CC=O)CCNC(=O)C1 C12(NC(C(C)CNC(C3Cc4nccn4C3)=O)=O)CC3CC(CC1C3)C2 c1(C(=O)NCC(C)C)ccccc1NCCO.c1(C=O)cc(C(N)=O)ncn1 Cn1ccc(C(N2CCCC2CNC(C2CCCSC2)=O)=O)c1CC(=O)O C1(C(N)=O)CCN(C(C2CCN(C(c3ncsc3Br)=O)CC2)=O)CC1 CC1(C)C(C)CCN1C(=O)Cc1ccc(C(N)=O)cc1.C1(C=O)CCC1(C)C c1(C(=O)NCCCCC2CN(C(C(C(C)O)C)=O)C2)ccc2nccnc2c1 C(=O)(CCC(C)(C)N1CCOCC1)NCCNC(C1CC(C)SCC1)=O c1(C(=O)NCCCCCN(C(c2ccc(CCC)s2)=O)C)c(N)sc(C)c1C C1(CNC(c2cnc(C)[nH]2)=O)CC(C)N(C(=O)Cn2ncc(Cl)c2C)C1 c1(C(N2CC(O)(CNC(=O)C(F)(F)c3cncs3)C2)=O)cnc2nccn2c1 c1(C(C(=O)NCCCCCC)N(CC(=O)OC)C)ccc([N+](=O)[O-])cc1Cl N1(C(=O)CCc2cccc(Br)c2F)CC2CC(N3CCS(=O)(=O)CC3)C1C2 C#Cc1ccc(C(=O)NCC2CC2NC(=O)C(C)S(N)(=O)=O)cc1 C1(c2ccccc2)CCN(C(c2cc(C(F)F)[nH]n2)=O)C1.C1(OC)CC1C=O.N C(CCCCC(=O)NC1CC1NC(=O)CCn1ccc(O)nc1=O)NC(N)=O CCCCCC(=O)N1CCC(N(C(=O)C(COC)OC)CCC)C1 c1(C(=O)NCCC2N(C(C3OCCN(C)C3)=O)CCSC2)c[nH]cc(F)c1=O c1(Nc2ncc(C(=O)O)s2)cc(C)cc(C)c1.C1(C=O)CC(C)N(CC)C1 C(C(=O)N1CC=CC1C(=O)N(CC(C)(C)CN(C)C)C)(C(C)C)OCC N1(C(Cn2c(C)cc(C)n2)=O)CCOC2(CCCN(C(=O)Cc3cnns3)C2)C1 C1(C)(C(=O)NCCC(=O)N(C)C)CN(C(=O)C(CO)NC(N)=O)C1 C1(NC(CSCC)=O)C2CC3CC(C2)CC1(C)C3.c1(C=O)cc2scnc2[nH]1 C12(CNC(c3cc(OCC)n[nH]3)=O)CC1CN(C(c1ccc(O)cn1)=O)C2 C1(NC(c2cc(C)n(Cc3ccoc3)c2C)=O)CCCCN(C)C1=O CCC1=NOC(C(=O)N(CCC(=O)NC2CC23CC(O)C3)C)C1 c1(C(N(CC(C)C#N)CC)=O)cc(CNC(C2CC(C)C2)=O)nn1C C#CC1(C(=O)NC2CC2(C)C(F)F)CCN(C(c2cc(CCC)on2)=O)CC1 C12(C(N(CCNC(c3c(CC)csc3)=O)C)=O)CC(CO)(C1)OC2C c1(OC)ccc(OC)c2sc(Sc3cnc4c(c3)CCC(=O)N4)nc12 N1(C(c2cc3ccccc3c(O)n2)=O)CCC2(C1)CN(C(C1(Cl)CC1)=O)CCO2 C(C)(CO)(C(=O)NC1CC2(C1)CC2)OC.c1(C(=O)N)ccccc1.C1CC1 CCCCCCC(O)CCC(=O)NC(CNC(c1cc2n(n1)CCC2)=O)C(C)C CC(C)(C)C#CC(=O)N1CCCOC(CCNC(c2ccc(C(N)=O)[nH]2)=O)C1 C1(C(N(CCCNC(C2CC3(CC3)C2)=O)CC)=O)CCc2nsnc2C1 N1(C(C(CC)(C)CC)=O)CCC2(NC(C3CC4C(C3)C4(F)F)=O)CCCC12 c1(CCC(=O)NCC(CC)NC(c2ccc(F)s2)=O)ccc(N(C)C)nc1 Cc1cc(C)cc(C=CC(N2CCN(C(C3Cc4cccnc4C3)=O)CC2)=O)c1 CC#CCCCC(=O)NC(C1(O)CCN(C(c2onc(CC)c2C)=O)C1)C N(C1CCOc2ccccc21)C(=O)CSC(C)C(N1CCC2(CCCCCC2)C1)=O N1(C(C(c2ccc(F)cc2)C)=O)CC2CCC(NC(=O)C3=C(Cl)CC3)CC2C1 C(=O)(C1=NOC(C)C1C)N(CC)CC1CCCN1C(c1cc(C)n(C)n1)=O N1(C(c2cn(C)nc2)=O)CC2CC(NC(C3(Br)CC34CCC4)=O)CC(C2)C1 C1(C(N2CCC(N(C(=O)C#CC3CC3)CC#C)CC2)=O)CN2CCN1CC2 c1(CC)c(NC2CC(NC(=O)CC(O)CC)C2)ncnc1Cl C(=O)(CCCCCCNC(C1CC(n2cc(CC(O)COC)nn2)C1)=O)OC CC(C)CC(F)(F)C(=O)NCC1CC(NC(C2CC2(C)C(F)F)=O)C1 N1(C(C2CCN(C(CC)=O)C2)=O)CCN(C(c2ncncc2F)=O)C(C2CC2)C1 S(=O)(=O)(c1ccc(C)c(Cl)c1)N(C1(CC)COC1)C(C1(C)CCC1)=O C12CCCN(C1)C2.C1(CNC(c2cc(C3C(C)C3)on2)=O)CNC(=O)CO1 CCS(=O)CCNC(=O)CC1CCCN1C(c1ccnn1C)=O.CC(=O)OC C1(NC(Cc2ncc(C)s2)=O)CCOC2(CCN(C(C3(CO)CC3)=O)CC2)C1 N1(C(CC(CCCC)O)=O)CCC2CN(C(=O)CCc3ccnn3C)CCC12 C(=O)(CC1=C(C)NS(=O)(=O)N=C1C)NC1CCN(C(CCCCC#C)=O)CC1O N1(C(CCCCC#C)=O)CCC(C2CC2)C1CNC(=O)Cc1c(O)ncnc1O CC1COCC(C)N1CC(c1ccccc1Cl)C(=O)NC12CC(C(F)F)(CO1)C2 c1(C(N2CC(NC(C3C(C)(C)C3)=O)C2)=O)cccc(C(F)(F)C(F)F)c1 c1(CC)cc(C(=O)N(C(C)C(=O)NCCC(C)c2cn[nH]c2)CC)ncn1 C(C(C(C)C(C)C)NC(c1cccs1)=O)NC(c1c(C)nn(C(C)(C)C)c1)=O c1(C(N2CCC(N(C(c3cc(CC)on3)=O)C)C2)=O)ccc(-n2ccnc2)cn1 CC(N=c1cc(C(F)(F)F)c2ccccc2[nH]1)c1ccc(Br)cc1F c1(NCc2n(C)cnn2)ncc(S(=O)(=O)NCC(C)(CO)c2ccccc2)cc1Cl c1(C(C(F)F)NC(C2C(C)C2C)=O)cccc(C(F)(F)F)c1 c1(C(=O)NC(CC2CN(C(CC(CC)CN(C)C)=O)C2)C)cc(Cl)c(Cl)cc1C c1(CN2C(C(=O)Nc3ncc(C(=O)OC)s3)CN(C)CC2)c[nH]c2ccncc12 C1(C(=O)NC(c2ccc(Br)cc2)C(C)(C)C)CC12CCC(F)(F)CC2 C1CS(=O)(=O)C12CCN(C(C1(N(C)C)CCC1)=O)CC2.C(C)(CCC=O)OC.N C1(N(C(CCCCC)=O)C)CN(C(C2CCOC(CC)C2)=O)CCC1O N1(C(C(CC)Br)=O)CCCC(C(=O)NCc2ccnc(N3CCCC3)n2)CC1 Cc1cc(C(=O)NCC(C)CNC(=O)CSC(F)F)ncc1N Cc1ccc(NC(C2CC23CCN(C(=O)Nc2ccc(F)cc2C)C3)=O)c(Cl)c1 C1(Nc2c(-c3ccc(OC(C)C)cc3)n[nH]c2)CC2CC1CC2(F)F c1(C(=O)NC2CC(NC(C(C)CF)=O)C2)ccc(C(=O)C2CC2)cc1 c1(OC)ncc(NCC(C)CC(=O)N2CC(N3CCN(C)CC3)C2)c(C)n1 c1(C(=O)NCCNC(c2c(-c3ccc(C)cc3)noc2C)=O)cccc(O)c1C c1(C2(C(N3CC(C)C(NC(C4CCCO4)=O)C3)=O)CCCC2)cc(F)ccc1F C1(NC(C2(C(=O)NC)CC2)=O)CC(C(=O)NC2CCOCC2)CC1O C(=O)(C(C)N=[N+]=[N-])NCC1C(C(N(C(C(=O)OCC)C)C)=O)OCC1 c1(C(N2CC(C(C(=O)Nc3c(OC)cccc3)O)C2)=O)cc(O)cc(F)c1 C(=O)(C1=CCOCC1)NCC12C(CN(C(c3nc(C)sc3C)=O)C1)C2 Cc1c(CC(=O)NC(C(=O)NC2CC(F)C2)c2ccco2)cnn1C C(C(C)(C)OC(C)C)(c1nnnn1Cc1cccs1)NCC(C)(C)OC N1(C(c2n(C=C)ncc2)=O)CCN(C(c2ncccc2N)=O)CC1CC1CC1 Cc1ccc(CC(=O)N(C(C)C2CC2)C)c(F)c1F.C1(C(=O)N)CC2(CC2)CO1 O=C(C1CCCc2nn[nH]c21)NC1CC2CCCC(C1)N2C(=O)Cn1cnnc1 N1(C(C)C)CCCN(C(=O)C(CC2CCC2)NC(c2cnc(O)o2)=O)CC1 N1(C(C2(N3CCCC3)CC2)=O)CCCCC(C(=O)NCC2CCC2CO)C1 C1(CNC(CCN(C(C)=O)C)=O)CCN(C(c2oc(C(F)F)cc2C)=O)CC1 c1(OCC)ccc(CCC(=O)NC(C)CNC(=O)C(F)(F)CC)cc1 N1(C(CC(C)(C)C)=O)CC2(C1)CCCS2(=O)=O.C1(C=O)CCN1S(C)(=O)=O N1(C(C(COC)N(C)C)=O)CCC(CF)(NC(=O)CCc2ccc(SC)cc2)C1 S(=O)(=O)(c1[nH]c(=NCC23CCN(CC2)C3)ccc1Br)C1C(C)SCC1 c1(C(N2CCCC(CNC(CC(C)OC)=O)C2)=O)cc(=O)c2ccccc2[nH]1 N1(C(CC2(C)C(NC(CCC(C)OCC)=O)CCC2)=O)CC2CCC(CC2)C1 C1(CNC(=O)NC(CC)Cn2ccc(C)c2)CC2CCCC2C1 c1(CCC(N2C(C)(CNC(c3cc(C)ncc3)=O)CCC2)=O)ccccc1C#N CC1(C)C2CN(C(=O)CCC3(NC(C4CCC5(CC5)C4)=O)CCC3)CC12 c1(C(=O)OCC)cc(NCCCC2(C3OCCO3)CCOCC2)cc(Br)n1 c1(OC)ccccc1C(C)CC(=O)N1CC(C)(NC(=O)C2=CCCC2)C1 c1(C(N(CCCNC(C2(F)CC2C)=O)C(C)C)=O)cc(-c2ccco2)no1 C1(CNC(C(F)=CCC)=O)CN(C(=O)CC(=O)OC)CC12CC2 N1(C(CC(=O)NC2CC2)=O)CCC2CN(C(c3cnc(S)[nH]3)=O)CC2C1 CN1CCC(C(=O)NCC=C2CCSCC2)C1=O C(=O)(CC(CC(N)=O)CC(C)C)N1CCCN(C(CCC(CC)OC)=O)CC1 c1(NC(CN(CCC)C(C2CN(C)CC23CC3)=O)=O)cc(C#N)cn1C c1(C(N2CCCC2CCNC(C2CC(O)C2)=O)=O)cc(Br)n2ccccc12 c1(CC(N2CC3(C2)CN(C(c2ccc(C(F)F)s2)=O)C3)=O)ccn2cncc2c1 c1(OCC(=O)NCC(CCOC)NC(=O)COC)nn(C)cc1Br Cc1cc(C)cc(O)n1.C1(C)(C(N(CC=CC(=O)N)C)=O)CCC(C)CC1 CCC(CC(F)(F)F)C(=O)NCc1ccccc1.c1(C(=O)N)scnc1C1CC1 N1(C(c2c(CC)nccn2)=O)Cc2occ(C(=O)N(CCO)C3CC3)c2C1 c1(C(=O)NC2C(C)(C)CN(C(C3CC(F)C3)=O)C2)cn2cccnc2n1 c1(N2CCN(Cc3c(COCC(CC)C)cccc3)CC2)ccc(Cl)c(Cl)c1 c1(OC)ccc(C(=O)NC)cc1F.c1(C(N2CC(C)CC2)=O)cc(C)nc(Cl)c1 Cc1noc(CCC(=O)NCC2CCCC2NC(c2ccns2)=O)n1 Cc1nc2[nH][nH]cc-2c(=NCCC2CCCN(C(c3cc(O)ncn3)=O)C2)n1 C(=O)(C1CCCc2nn[nH]c21)NC1(CNC(C2(C#N)CCCC2)=O)CCOCC1 S(=O)(=O)(c1ccc(NCCC2CCSC2)cc1Cl)NCC(CCCCCCC)C CCCCCS(=O)(=O)CC(=O)NC1CN(C(=O)CC(C)COC)C2CCCCC12 c1(C(=O)OCC)ccc(Cl)cc1C(N1CC2CC1C2)=O.C(=O)C1=NOCC1.C CCC(C(=O)OC)C(=O)N1CCCC(C(C)NC(=O)COCC2CC2)C1 c1(C(N2CC(c3nccc(OCC)n3)C2)=O)cc2n(n1)C(C)CCC2 C(CCCCC(C(=O)NC(C)C)N1CCCCC1CC(c1ccccc1)O)OC N1(C(CN(c2cnccn2)C)=O)CCN(C(=O)C=CBr)C(CC(F)F)C1 C1(NC(CC2CC(NC(c3cnc(CC)nc3)=O)C2)=O)CCOCC1(C)C C(=O)(C(C)(C)CC#N)NCC(CC)(CC)NC(C12CCCC1C2(F)F)=O Cc1oc(C(=O)NC(Cc2ccco2)C(=O)NC2CC23CCCC3)cc1CO C(C(C)NC(c1ccc(C(=O)N(C)C)cc1)=O)(C(C)C)NC(CC)=O CC1(NC(=O)Cn2ncc(Br)n2)CCN(C(c2ccccc2C(F)F)=O)C1 CC1CC(C(=O)NCCCC2CCCN2Cc2nc(CS(C)(=O)=O)no2)CCO1 CCCCC(C)C(=O)NCCC1CCN(C(c2cccnc2OC)=O)C1 C=CC1CN(C(c2ccc[n+]([O-])c2)=O)CC1NC(=O)CCC1CCCN1C C(=O)(CCC1=NNC(=O)CC1)NCC1CCN(C(CC(=O)NCC)=O)CC1 CC(C)CC(C)(CNC(c1cccc(Cl)c1F)=O)NC(C1CCC(F)(F)CC1)=O C1(CNC(Cn2c(C(C)C)nnn2)=O)CN(C(C2CC2Br)=O)CCO1 N1(C(c2c(C)con2)=O)CCN(C(=O)C2=C(Cl)CCC2)C2CCCCC2C1 N1(C(CCCSC)=O)CCC(C)C(CC(=O)N(C2CC(F)(F)C2)C)C1 C1(NC(Cc2cn(C)nn2)=O)CN(C(=O)CCCNS(C)(=O)=O)CC12CC2 Cc1ccc(C2OCCCC2C(=O)NC2CC(NC(c3csc(C)c3)=O)C2)cc1 C1(CC(=O)NCCC2CCN(C(C34CC(C3)C4)=O)CC2)CC1C1CCCCC1 C1(C(N2CC(NC(c3c(OCCC)cccc3)=O)C(C)C2)=O)CCCC(C)(C)O1 C1(C(=O)N(CCO)CCO)CCC2(CC2)N1C(=O)CCC1CC1(F)F C=C=CCC(=O)NCC(C)(C)NC(=O)C(C)C1CCOC1 Cc1ncccc1C(N1CCOCC1CC(=O)NCC1(C)CC2(CC2)C1)=O CCC(C)(C(=O)NC1CCN(C(c2ccnn2CC(C)C)=O)CC1O)C(F)F c1(CNC(Cn2c(N(C)C)cc(C)n2)=O)cc(S(C)(=O)=O)co1 c1(NC(C2C(N(C(CCOCCOC(C)=O)=O)C)C2)=O)ccc(F)nc1 c1(C(=O)NCC2CC(NC(c3c(C)nc(CC)o3)=O)C2)cnc(C)nc1C C1(CC)C(C(=O)NCC=O)CCN1C(=O)C(C)C1(O)CCC1.C(N)(=O)N C(=O)(CCCCC(=O)N1CC(O)CC1CNC(=O)C(CCO)N(C)C)N(C)C c1(CC(N2C(CC)CCC2)=O)ccccc1F.CC(C(=O)N)NC(C1CCC1)=O O=C(CCCCCO)NC1CC1CNC(=O)CC(O)c1ccccc1 C1(NCC(=O)NC)CCN(Cc2ccc(Br)cn2)CC1 Cn1ncnc1CCC(=O)NCCOCC(=O)NCC1(C(N)=O)CCCC1 c1(C(=O)NCC2(O)CCN(C(CCc3cc(C)sc3C)=O)C2)c(C)cncc1C c1(OCCC(=O)NC(CCCNC(CCN(C)CC)=O)C)ccc(F)cc1Cl.O C1(CC(=O)N(C(C#C)Cc2ccc(Br)cc2)CCC)CCCC2(CC2)C1 c1(CNC(CCSC)=O)n[nH]c2c1CN(C(c1c(C)ccc3n[nH]cc13)=O)CC2 C1(CC)CCCCC1C(=O)NC1(CCC(=O)NCC2(F)CCOC2)CCC1 CC(C)S(=O)(=O)c1ccc(NC(=O)CN2CC(N)C2)cc1 CC1C(NC(c2ccnc(OC(C)(C)C)c2)=O)CCCN1C(c1cc[nH]n1)=O CC1CCc2sc(C(=O)NC3CN(C(=O)CCc4cc[nH]n4)CC3C)cc2C1 C(=O)(C(F)CC(C)(C)NC(C1CC(=O)NC(=O)C1)=O)Nc1cc(C)c(F)cc1 c1(C=O)ccc2c(c1)NC(=O)NC2.c1(CC)sc(=N)[nH]c1C(=O)N.CC(F)C N1(C(C(C(C)C)O)=O)CCCN(C(=O)CCC(F)(F)F)C(C(C)C)C1 CC1CN(C(C2CC2c2ccccc2)=O)CCN1C(c1nnc(S)n1C)=O C(=O)(CCCC(C)(C)NC(=O)C(C(CC)CC)OC)N(C)CC1CC(=C)C1 N1(C(=O)CC2(O)CCOC2)CCOC2(C1)CN(C(c1cnc3cccnn13)=O)C2 C1(C(N(CC(C)OC)C)=O)CC=CC(NC(=O)CC=Cc2ccccc2)C1 C1(C(=O)OCC)CN(C(c2ccc(Br)cc2O)=O)C2CCN1C2 C1(CC=C)(NC(c2cccc[n+]2[O-])=O)CCN(C(C2CSC(C)=N2)=O)C1 C1(C)(CC)CCCN(C(=O)CC2COCCN2C(=O)C(=O)NCC(F)F)C1 C1(C(=O)N)C2CC(O)C(C2)N1C(=O)C(F)C(F)(F)F.C12CC(F)(C1)C2 Cc1sc(Cl)nc1C(=O)NCCC1CCCCC1.C(=O)C(F)(F)CN1CCCC1 c1(NC(C(CN(CC(C)(C)OC)C)OCCO)=O)ccc(C)cc1 Cc1nc(C2CCC2)sc1C=O.C1(C=O)CCC(C(N)=O)C1.C(C)C1CC1.N c1(C(N2CCC(NC(C(CC)N(C)C)=O)(CF)C2)=O)cn2cc(C)sc2n1 C1(CNC(CCCC)=O)CCN(C(C2CCN(c3ccccc3)C2=O)=O)C12CC2 C(=O)(CC(C)CC(C)(C)C)N1CCCN(C(Cc2cn(CC)nc2)=O)C(COC)C1 N#Cc1ccc(C(N2CCC3(C2)CN(C(C2(O)CCSC2)=O)C3)=O)c(O)n1 N1(C(CCOCCOC)=O)CCN(C(C2CC2CC(C)C)=O)CC1C N1(C(CC(CC)C2CC2)=O)C(CC(=O)NCc2c(C)cccc2F)C2CCCC12 c1(C(=O)NC2(CO)CN(C(C(CC)N(C)C)=O)C2)ccc(Br)c(F)c1F C1(CC(c2cnc[nH]2)=O)CN(C(=O)Nc2sccc2-n2cnnn2)CCO1 C#CCC(C(=O)N1CCNC(=O)C1)NC(C1CC(OC)(OC)C1)=O N1(C(CC2CC(=C)C2)=O)CCSCC1C(=O)NC1CCOCC1F C12(NC(C(C3CCC3C(F)(F)F)N(C)CCF)=O)CCCC1C2 c1(CNC(=O)NCCC2(O)CCOC2)ccc(Cl)cn1 CC(C)(C)CC(O)C(=O)NC1CC2CCC1C(NC(=O)CC(F)F)C2 C(CC)(C(=O)NC(C1(O)CN(C(c2coc(O)n2)=O)C1)C)OCC C1(CC=C)(NC(=O)C(O)CSC)CCN(C(c2c[nH][nH]c2=N)=O)C1 c1(CC)c(C(N2CC3C(CN(C)C(c4ccc(Cl)s4)=O)C3C2)=O)cnn1C.O CN1C(=O)CCCC1C(=O)NC1CCN(C(=O)CC2CC3(CCO2)CC3)CC1 N1(C(c2cccc(NC(CC)=O)c2)=O)CC2(CCN(C(=O)CC(C)CF)CC2)C1 CC1CCN(N2CC(OC(=O)N(C)C)C2)C1N(C(c1ccccc1)=O)C c1nc(C(C)(C)C)nc(=N)[nH]1.C(c1ccsc1)=CC(=O)N(C(C)C)CCN N1(C(CC(C)c2cccnc2)=O)CC(F)(F)CC1(C)CNC(=O)Cc1cnco1 C1(C(=O)OC)CN(C(c2cc(NCc3cnco3)ccn2)=O)CC12COC2 N1(C(c2csc(C(=O)OC)c2)C(=O)NCCCC)CC2OCCN(C(C)=O)C2C1 N1(C(CCOC)=O)CC(NC(c2cc(-c3ccc(Cl)cc3)on2)=O)C2CC2C1 CCCC(C(=O)N(C(C)CC(N)=O)C)NC(c1ccnnc1C)=O N1(C(CN(C)C)=O)CCC2(CC1)CC2NC(=O)Cc1cc(Cl)cs1 c1(CC(=O)N(CC=O)C)ccn(CC(C)C)n1.CCC(C)N(C)C.C(=O)C N1(C(Cc2cc(C)sc2)=O)CC2(CC(C(=O)Nc3cnc(C)c(C#N)c3)CO2)C1 Cc1ccc(C(=O)NCC(C)(C)NC(=O)C(C)C2CCCC2)c(C(C)C)n1 c1(CC(C)C)ccc(C(=O)NCC2CCCCC2)cc1.C(=O)(C1=C(Cl)CC1)N C1(CC(=O)N(C2CN(C(CCOCC#C)=O)CC2(C)C)C)CCn2cncc2C1 N1(C(C2(NC(C3C(C)CCO3)=O)CSC2)=O)CC2(CC(N(C)C)C2)C1 C(c1ccc(F)c(C)c1)=CC=O.Cc1cc(C(=O)NCC2CC2)cc(Cl)c1 Cc1nc2c(s1)CC(C(N1CCC(C)C(O)C1)=O)CC2 C1(NC(c2n[nH]c(CC)c2Br)=O)CCCC(NC(=O)CC2(O)CCC2)CC1 Cc1ccc(N)cc1.c1ccncc1Br.c1(C2CCS2)nnnn1C1(C)CC1 N1(C(C(CSC)O)=O)CC2CCC(C(=O)NC(C)(C)CC(C)(C)C)(C2)C1 c1(C(N(CC(C)NC(C2CC(C)(C)C2)=O)C)=O)cccc([N+](=O)[O-])c1 CC1CC(C(=O)NCCCNC(=O)C(N2CCOCC2)C)CC(C)O1 C1(NC(C(C)(C)Oc2cccc(F)n2)=O)CCC(c2nn[nH]n2)CC1 c1(OC)ccc(C=CC(N2C3CN(C(c4ccc(Cl)cc4)=O)CC23)=O)c(F)c1 O=C1CSC(C(=O)NCc2n[nH]cc2C(=O)NCCC(O)C2CC2)C1 c1(C(N2CCCC(C(C)NC(Cc3cc(C)ncc3)=O)C2)=O)c[nH]c(=N)c(C)c1 c1(NC2C(C)SCC2)ncccc1S(=O)(=O)NCCCN(C)C1CC1 c1(C(=O)NCC2(COCC)CC2)ccc2cnnn2c1 C1(C)CCN(C(=O)N)C2(CC2)C1.c1(CCC)ccccc1CNC(C)(C)C C=C(C)CC(C(=O)NCC)NC(c1n[nH]cc1NC)=O.c1(C=O)ccco1.N C1(NC(C2NC(=O)OCC2)=O)CN(C(c2occ3c2CCC3)=O)CCC1CO c1(C(N2CCC(NC(c3c(C)ncn3O)=O)CC2C)=O)cc2c(Cl)nccc2s1 c1(-c2nc(C(Cc3ccc(C)cc3)C)on2)cccc(C)c1Cl C1(C=O)CCCC1(F)F.C1(F)(CNC(CN(S(CC)(=O)=O)C)=O)CCC1.C C(CCCCCNC(c1ccc(C2(O)COC2)cc1)=O)NC(=O)Cc1csnn1 O(NC(=O)CN(C1CC(C#N)C1)C(=O)Cc1ccns1)CC=C Cc1cc(C(=O)N(C(c2cn(-c3ccsc3C(=O)O)nn2)(C)C)C2CC2)on1 N1(C(C(C=CCCC)O)=O)CC2(CCCC2NC(C2(CC)CCC(O)CC2)=O)C1 c1(C(=O)NCC(CC)NC(=O)C(C)OC)cnc(C)c(N)c1.c1ccncc1 C1(O)(CC(=O)NC23CN(C(C(N4CCCCC4=O)C)=O)C(C2)C3)COC(C)(C)C1 n1(CC(=O)NC(C(C)SC)C)ccc(=NC(=O)c2cocc2C)[nH]1 n1(C(C(=O)NCC(C)NC(C2(C3CC3)CCCO2)=O)C)cnc(C#N)n1 c1(CC(=O)NCC(O)C)coc(-c2cccs2)n1.c1(C2C(C=O)C2)ccco1.N c1(C(=O)NCCC2N(C(c3nc(CC)oc3)=O)CCC2)cnn(C)c1CC C(=O)(CC(C)CC(=O)N1CCC(CNC(=O)C(C)CSC)CC1C)OC CCCCCCC(C)CC(=O)NCC(C1CC1)NC(C1(CCN(C)C)CC1)=O N1(C(c2nccc(C)c2)=O)CC2(CC(NC(C3CCCCN3N=O)=O)CO2)C1 Cc1cccc2cc(-c3ccc(C(C)O)cc3[N+](=O)[O-])cnc12 N1(C(c2cc(C#N)c(Br)cc2)=O)CCC2(CCC2NC(=O)C2CC2)CC1 c1(CC)cccc(CC)c1CSc1nc(C)nn1C(C1CC2CCC1C2)C CN1CCCC(F)(CC2NC(=O)N(Cc3cccc(-n4cncn4)c3)C2=O)CC1 c1(C(=O)NCC(CNC(CNC(C(CC)C)=O)=O)OC)cc([N+](=O)[O-])c[nH]1 CC1C(NC(c2ccc(N(C)C)cn2)=O)CCN1C(c1cc(F)n[nH]1)=O c1(NCc2c(C(C)(C)C)[nH]cn2)ccnc(-c2ccccn2)n1.C1(CCN)CCO1 c1(C(=O)NCC2CN(C(C3C(C=C)C3)=O)C2)ccc(C)cc1.C(C)=O.N C1CC2CCC(C1)N2C(=O)CC1CCCCC1(C)C.C1(CC(=O)NC)CCNC1=O C(=O)(CC(C(F)(F)F)c1ccccc1)NC1C(NC(C=CCC)=O)CC1 C1(C#N)(C=O)CC12CCOCC2.Cc1nc(C)c(C(=O)NCCC2CCC2)s1.N C(=O)(CC(C)(C)CN=c1[nH]c2c(c(=NCCS(=O)CC(F)(F)F)[nH]1)COCC2)NC N1(C(c2c(C)ccnc2Cl)=O)CC2(CCCC2NC(=O)C(C)CN(C)C)C1 C(=O)(C(O)CC(C)(C)C)NC1C=CC(C(=O)NCC(c2cnn(C)c2)C)C1 C1(C(F)(F)F)(OC)CCCN(C(C2CCCC3(CC3)C2)=O)C1 C1(NC(=O)COC(F)(F)F)CN(C(=O)CN2CCCS2(=O)=O)CC2(CC2)C1 N1(C(C(C)(C)F)=O)CC=C(C(=O)NCc2ncoc2C2CC2)C1 Cc1cc(O)ncc1C(=O)NC1CC(CCNC(=O)C(=Cc2c[nH]cn2)F)C1 c1(C(=O)NCC(CNC(=O)C=CC2CCOC2)CO)cc2ccccc2o1 CC(C)(O)C(C)(C)C(=O)N1CCCOC(CNC(=O)CC2CC(=O)C2)C1 c1(-c2n(C)ncn2)ccccc1C(=O)NC1COCC1NC(=O)Cn1cccn1 c1(CC(=O)NCC(COC)NC(c2nsnc2O)=O)nn(C)cc1Cl C1(NC(CNC(CC)=O)=O)C2CC3C(C2)C13C(=O)N(C1CCCCCCC1)C Cc1cc(F)ccc1C1CCN(CC2CSC2)CC1 C1CC2(CC2)CN1C(c1cc(Cl)c(Cl)n1C)=O.c1(SC)ccc(C(=O)N)o1.C N1(C(CN2CC(C)C2)=O)CC(NC(C2(O)CC2)=O)C(c2ccnn2C)C1 C1(C(=O)OCC)(NC(=O)CC2CCC3(CCC3)CC2)CC2(CC(F)C2)C1 C1(C)(CNC(c2ccc(CC)c(CC)c2)=O)COCCN(C(C2CCCC2)=O)C1 C(=O)(CCCCCCNC(C1C2CCC(=O)C12)=O)NCCC1CC(C)(C)OC1 C12(c3n(CC(=C)C)c(N4CCC(CCOC)C4)nn3)CC3CC(CC(C3)C1)C2 c1(-c2cn(CC3CCC(NC(C4(COC)CC4)=O)C3)nn2)ccc(C)nc1 N1(C(c2c(CNC(c3c(CCC)nco3)=O)occ2)=O)CC2CC1CS2 c1(N2CCN(CC(C)O)CC2)cnn(C(C)(C)C)c(=O)c1Cl c1(C(N2CC(NC(c3ncc(C)cc3C)=O)C(O)C2)=O)cc2cc[nH]c(=O)c2s1 C(=O)(C(C)(C)C1CCN(C(=O)CCC2CC2)C1)N(CCC)CC1CC1.O N1(C(C(=O)CN)=O)CCC2C(C(=O)O)C2C1.C1CCC1(C)C.CCO.C C1(C(N2CCN(C(CSC(C)C)=O)CC2CO)=O)CCOC2(CCCCC2)C1 N1(C(CC2CCCC(NC(C(CSC)C)=O)C2)=O)CCN(C)CC1CCO C1(C(N(CC(CC)O)CC)=O)(NC(c2cnsc2C)=O)CCCC1C N1(C(CC2(CC)CCOCC2)=O)CCCOC(CNC(c2csc(C)n2)=O)C1 CC1(C(=O)NCC2(O)CC(NC(C3CC(Cl)(Cl)C3)=O)C2)CCNC1=O C(=O)(C1=CS(=O)CCC1)Nc1ccc(-c2nnc(CCC(=O)O)o2)cc1 C1(C)CC(C(N2CCC(N(C(=O)C=CC(C)(C)C)CCO)C2)=O)CCO1.C C1(C(N2CCC(CC)CC2)=O)CCN(C)C(=O)C1.c1(CCC=O)c[nH]c(=N)[nH]1.N Cc1[nH]nc2ncc(C(=O)NC34CCC(C3)N(C(=O)CC3CCCCC3)C4)cc12 C1(C(N(CCC#C)CC)=O)CN(C(C2(F)CCOCC2)=O)CCN1C Cc1ccc(C(N2CC(CNC(=O)C(=O)Nc3ccc(N)cc3)C2)=O)cc1 C(=O)(C1=CC=NC(=O)C1)N1C(CNC(Cc2cnc(C)s2)=O)CCCC1 Cc1nc(C(C)C)oc1C(=O)NC1CN(C(=O)C(F)(F)c2cnn(C)c2)CC1C Cc1cc(C(N2CCN(C3CCCN(C(=O)C(C)(O)C(C)C)C3)CC2)=O)cc(C)n1 CC1(CC(=O)NCCC2CC(NC(c3csnc3Cl)=O)C2)CCOC1 c1(CC(N2CCN(C(CCC)=O)C3C2CC3)=O)c[nH]c2nccc(Cl)c12 CC(C(CO)NC(C1CN(C2CCCCC2)C1)=O)NC(c1nncs1)=O C12(CC=O)CCCCC1C2(F)F.C(CC(=O)NCCC1CC1)N(C)CCO.C c1(C(C)NC(=O)C(=O)N)ccc(Cl)c(C(F)(F)F)c1.C1(CC)CCC(C)C1 C1(C(N(CC(C(C)C)OC)C)=O)CN(C(C2CC(OC)C2)=O)CCO1 N1(C(C(=O)NCC)C(C)C2CCOC2)CCCN(C(c2ccc(F)cc2)=O)CC1 c1(OC)nc(C(=O)NC2CC2C)sc1C.C(c1csc(C)n1)=CC(=O)N C=C=CC(C)C(=O)N1CCOC(C(=O)NCc2cc(C3CC3)on2)C1 c1(CC)ccc(F)cc1.C1(CC(=O)N)COCCN1C(c1cncn1C(C)C)=O CC(N=c1nc[nH]s1)C1CCCCN1C(=O)Cn1cc([N+](=O)[O-])cn1 CP(C)(=O)CC(=O)N1CCC(CF)(NC(C2CCSCC2)=O)C1 C=CCC(C(=O)NC1CC(CNC(=O)C(C)=CC2CC2)C(O)C1)C(C)C C1(NC(C(N2CC3C(N(C)C)C3C2)=O)=O)CC2CCC1CC2=O c1(CC(=O)NC(C2CCCN2C(c2ns[nH]c2=O)=O)C)nn(C)cc1[N+](=O)[O-] c1(C(=O)NC(C)COCc2ccccc2)ccc(Cl)c(F)c1O c1(C(=O)NCC(C)NC(=O)CSc2ccc(F)cc2)cccc2nc(O)[nH]c12 CC1(C)CCCCC(C(=O)NC2CCCC2NC(c2c[nH]c(=O)cn2)=O)C1 N1(C(C(C)N(CC)CC)=O)Cc2occ(C(N3CCC3)=O)c2C1.[nH]1ccnn1.C N1(C(C2CC(SC)C2)=O)CCC2CN(C(=O)C(O)C(C)C)CC2C1 Cc1sc(C(=O)N(C)C(c2ccccc2F)C)cc1Br N1(C(CCC#CC)=O)CC2CN(C(c3cc(O)cs3)=O)CCC12 S(=O)(=O)(c1cc(F)c(F)cc1F)N1CCC(CNC(CCCCC(=O)OC)=O)C1 C=CC(C)(O)CC(=O)N1CCCCC(NC(c2c(OC(F)F)cccc2F)=O)C1 N1(C(C(=Cc2ccco2)C)=O)CC2CC(NC(c3nccc(Cl)c3F)=O)CC2C1 C1(C(=O)NCCCCCCF)CC12CCN(C(c1csnn1)=O)CC2 C1(C(N2C(C(=O)NC(C(=O)OC)C(C)OC)CC2)=O)CC2CCCC2C1 CCCC(CC)CCC(=O)N1CCN(C(=O)CC2=NN(C)C(=O)C2)C(CCO)C1 C1(C(N2CCC(F)(F)C2)=O)C2CCCCCCC12.C(C)(C(=O)N)OCCOC C1(C(C)C(=O)NC2CC(CO)C2)CCN(C(=O)CCCc2nncn2C)C1 c1(N2CCN(C3(C(=O)OC)CCOC3)CC2)c(C#N)c(C)nc2ncnn12 c1(OC)cc(Cl)ccc1C(N1CC(F)CC1C(=O)Nc1cncnc1C)=O c1(C(N2CCC=C(CNC(CC3N(C)CCCC3)=O)C2)=O)cc2cccnc2[nH]1 C1(C(C)NC(C2CCCC2)=O)CCCN(C(=O)C=CSCc2ccco2)C1 c1(C(C)NC(C(=O)NC2CC(C)OC2)=O)ccc(N2CCOC2=O)cc1 Cc1ccc(N)cc1C(=O)NC(C)CCCNC(c1nccc(F)c1Cl)=O c1(CC(N2CCC(C3N(C(C)=O)CC3(C)C)CC2)=O)csc2ccccc12 c1(C(=O)NC(CN(C(=O)CC(C)C(C)C)CC)C)ccc2c(O)ncnc2c1 C1(NC(c2c(CC)c[nH]n2)=O)CCN(C(=O)Cc2c(C)cnn2C)C1(C)C CC1(NC(C2CC(O)(c3ccccn3)C2)=O)CCCN(C(=O)Cc2cnsc2)C1 c1cc(Cl)ncc1.C1(C=O)CCN1C(=O)C.[SH](C)(=O)=O.CCC1CC1.N c1(C(=O)NCC2CN(C(c3snc(C)c3N)=O)C(C)C2)c(F)cccc1F c1(CNC(C2CCC(C)C2)=O)ccccc1.C1(C(N(C)C)=O)CC(C)(C)CO1 CN1CCCN(C(=O)Cn2cnc(Br)c2Br)c2ccccc21 C=CCC(C)C(=O)NC1COCC1C(=O)NCCCS(C)=O c1(NC(CCNc2c(C)cc(Br)c(N)c2)=O)sc2c(c1C#N)CCC(C)C2 N1(C(CC(CC)CC)=O)CCCN(C(=O)CCc2cccc3c2OCO3)C(C)C1 C1(C(=O)NCC2(O)CC(C(=O)NCCc3ncon3)C2)Cc2nccn2C1 C1(C(=O)NCC(O)CCNC(c2cc(C=O)co2)=O)(CC)CNC(=O)C1 c1(CNC(c2c(C)c[nH]n2)=O)cc2n(n1)CCN(C(c1scc(C)c1Cl)=O)C2 Cc1ccc2c(c1)CC(C(=O)NCC(C)Cc1ccccn1)N2 C1(C(N(CCNC(c2cc(C(N)=O)no2)=O)CC)=O)CCCC(C)C1 N1(C(CCC(CC)C)=O)CC2(CCCN(C(c3ccc(CC4CC4)cc3)=O)C2)C1 N1(C(CC(=O)OC)=O)C2CCC1CC(C(=O)Nc1cnc(C)[nH]1)C2 C(=O)(C1=CCCN(C(c2cccc(CC#N)c2)=O)C1)NC1CN(C)NC1=O C(C(COC)C(=O)NCCN1CCN(C(c2occ(C)c2C)=O)CC1)OC N1(C(C(C)CC(N)=O)=O)CCC(NC(=O)C(C)(C)c2cnn(C)c2)CC(C)(C)C1 N1(C(C(C)N(C)C)=O)CC2(C1)CN(C(c1ccc(Cl)c3c1OCC3)=O)CCO2 C=CCC(CC)C(=O)N1CCC(C(C)C(N2CCN3CCC2C3)=O)CC1 CCCC(CCCNC(=O)Cc1c(F)cncc1Cl)NC(=O)C(C)N(CC)CC C12(NC(=O)C=Cc3cocn3)CCCC1N(C(c1cscc1F)=O)CCC2 C12(NC(CCc3c(C)cccn3)=O)CCN(C(c3c(N)cccc3Cl)=O)CC1C2 C=CCC(CC)C(=O)N1CCCC(C)C1CNC(c1ccnn1CC1CCC1)=O c1(N(C)CC2CCN(C(C3(C)CCCOC3)=O)C2)cc(C(N)=O)nc(Cl)n1 c1(C(=O)NC2CCC(N(C(CCOC)=O)C)C2)c(OC)cncc1Br CCCC(C)CC(=O)NCCCC(C)(C)NC(c1ccc(Cl)c(OC)c1)=O C(CCCNC(=O)CCOC1CCCC1)OC.c1(C=O)ccco1.N(C)C.N N1(C(CCC=CC)=O)CC(CNC(=O)COc2cnn(C)c2)CC12CCC2 C12(N(C(CC)=O)C)COC(C=O)(C1)C2.c1nnc(C(C)(C)C)s1.CC.CO CCC(CC)CC(F)C(=O)N1CCC(O)C(NC(=O)C(c2c(C)noc2C)C)C1 CCCCCC(C)(C)C(=O)N(C(CNC(C1(C)CCN(C)C1=O)=O)CC)C c1(OC)ccc(CCC(=O)NC(C)CC(C)NC(=O)C=C2CCC(C)C2)cc1 N1(C(C2C(C=C)C2)=O)CC(OC)CC(NC(=O)CCc2c(F)cccc2Cl)C1 c1(C(N(C2CCN(C(C3CC4CC4C3)=O)CC2)CC)=O)ccc(OC)c(O)c1 c1(C(N2CCN(CCO)CC2)C(=O)NCC=C)ccc(F)c(Br)c1F CCC(C)(COC)C(=O)N.C1(CC)CCCN(C(C2(c3ccn(C)n3)CC2)=O)C1 Cc1cccnc1C(=O)NCCCCC1CCN(C(=O)CC(=O)NC2CC2)CC1 C1(C2CCC2)(NC(C2(CCNC(c3cc(C)sc3)=O)CCC2)=O)CC1 c1(NC(CC(CC)N(C)C(C2CCCC(F)C2)=O)=O)ccc2c(c1)CCO2 c1(C(C)C)nnc(N2CCCC2CNC(=O)CSc2ccccn2)o1 Cc1noc(C)c1C(C)C(=O)NCCC1CCCCN1C(=O)CCn1ccnn1 C1(C(N2CC(F)(CNC(c3c[nH]c4ccccc34)=O)C2)=O)CCc2nc[nH]c2C1 c1(C(N2CCN(C(C3(C)CSC3)=O)CC2C2CC2)=O)ccc2nn[nH]c2c1 c1(C(N(C(CNC(C2N(CC)CCCC2)=O)C)C)=O)ccccc1N=S(C)(C)=O C1(C(=O)NC(CCCCNC(c2c(CC)onc2)=O)C)CC(C2CCCC2)C1 C(=O)(C1=C(F)CN(C(=O)C2=C(C#N)CCC2)CC1)N(C)Cc1cccnc1 N1(C(C2C(C#N)C2)=O)CCC2(CCC(NC(c3ccc(CO)s3)=O)C2)CC1 C(CCCCC(=O)NC)NC(c1c(COC)ocn1)=O.c1cccc(N(C)C)c1 C(=O)(C(CC(C)CC)NC(c1cc(CC)nn1C)=O)NCCCC(=C)C N1(C(c2cnc(OCC)s2)=O)CCN(C(=O)CC2CC(OC)C2)CC1CCO Cc1cc(C(=O)NCCCCC2CCCN(C(=O)C#CC3CC3)C2)c(C)o1 C12(CC)CC(CSc3nc(-c4ccccc4C)nn3CC(C)CO)(CO1)C2 n1(CC(N2CC(CCCCNC(C(C)SCC)=O)C2)=O)cnc([N+](=O)[O-])n1 c1(C(N2CC(COC)C2)=O)cc(N)ccc1Cl.c1(C(=O)N)cccs1.C1CC1 N#Cc1cc(C(=O)NC2CC2NC(c2ccc(C(F)F)cc2)=O)c(N)nc1O [SH](=O)(=O)C1CC1.c1(N(C(=O)COC(=O)C)CCOC)ccncn1.N C1(NC(CCc2cc(OC)no2)=O)CN(C(=O)C=C(C)Cl)CC2CCCC12 Cn1cnc2c1CCC(NC(=O)C(=O)NCc1cc3c(s1)CCOC3)C2 c1(C(=O)NCC2(F)CN(C(C(OC)OC)=O)C2)cncc(S(N)(=O)=O)c1 c1(C(=O)NC23CC(C(=O)NCCCCCO)(C2)C3)ccc2cc[nH]c2c1Br C1(NC(=O)Nc2n(Cc3ccc(OC)cc3)ncc2)C2Cc3ccc(Br)cc3C12 CCC(C)(COC)C(=O)NCc1cocn1.c1ccccc1 C1(NC(c2cccc(C)c2)=O)CCCCCN(C(c2snnc2C)=O)C1 CC1CC(N(C)CCN2CCCCCC2)CN1Cc1ccccc1 c1(C(C)C)ccc(C(=O)NC(C)CCNC(C2COC(=O)N2C)=O)cc1F C1(NC(CCCOCC=C)=O)CN(C(=O)Cc2ccc(C)s2)C2(CCC2)C1.C N1(C(C=C(CC)CC)=O)CCn2c(CNC(C3(C)CCCCC3)=O)nnc2C1 C1(N(C(C2C(=C)C2)=O)C)CCC2CN(C(c3ccc(N)c(N)n3)=O)CC12 CC1CC(CNC(c2cnc(C(F)F)s2)=O)CN1C(=O)CCc1cc[nH]n1 Cc1ccc(Cc2ccc(C(=O)O)o2)c2nc(NCc3cccc(O)c3)cn12 N1(C(CC=CC)=O)CCC2CCN(C(=O)CCCC3CCCO3)CC12 CCCN=C(NCCC1CCCN1CCOc1cccc(C)c1)N1CCC(C)(F)C1 c1(C(=O)NC(C)C(C)(C)NC(c2ccc3occc3c2)=O)ccc2ncccn12 c1(CNC2CC(C(=O)Nc3nc(C)c(Cl)cc3)C2)cc(C)c(O)cc1C C1(CNC(CC2CC(=C)C2)=O)COC(C)(C)CN1C(c1cc(C)ccc1C)=O CCCC(C(=O)NC(CNC(c1cccc(-n2cc(C)cn2)c1)=O)C1CC1)OC Cc1cnc(COCC(=O)N(CC(O)CN(C(=O)Cn2nccn2)C)C)o1 c1(C(=O)NCC(CNC(C(CC)SC)=O)CO)cc2cc([N+](=O)[O-])ccc2[nH]1 C1(NC(C(CCC2CCC2)NC(C(N2CCNC2=O)C)=O)=O)COCCN(C)C1 N1(CC2CC(OC)C2)CCC(C(=O)N(C2CC2)Cc2ccc(Cl)s2)CC1 C(=O)(C(F)C(F)(F)F)NC(CNC(c1c(SC)cccc1)=O)(C)C1CC1 CC(C)C(F)C(=O)NC(CO)C(=O)NCC1CCOC1=O C1(C(=O)NCC2C(C(C)C)C2)CCCN1C(=O)COc1ccon1 N1(CC(C2CC2)OCC)CCN(C(c2cc(C(C)N)on2)=O)CC1 c1(C)c[nH]c2ccccc12.CCS(=O)(=O)CC(=O)NCC1CC1CNC CCCCCCCC(=O)N1CCOC(C(=O)NCCCC(C)C)CC1 C(=O)(CCCCCF)NC1(CNC(c2ccc(OC)cc2)=O)CCOC1 Cc1cc(N)c(C(=O)NCC23CCC(CC2)N(C(c2cnsc2)=O)C3)c(F)c1 N1(Cc2ccc(SC)s2)CCC2(CC1)CC(NC(C1CC(=O)N(C)C1)=O)CO2 Cc1ccc(C(=O)NCCCCC(=O)N(c2ccc(F)cc2)C)n1C CCCC(C)CC(=O)NC(CCN(C(=O)CNc1cccnc1)C)C(C)(C)C c1(CC)cc(CN2C(C(=O)Nc3[nH]cnc3C(N)=O)CC3CC23)ccc1O Cn1c(CC(=O)NC2(CF)CCN(C(C3CC3F)=O)C2)nnc1S N1(C(CC(C)O)=O)CC2CC1C2C(=O)NC(Cc1ccccc1)CO c1(C(C(=O)NCC)N(c2ccccc2)C)ccc2ncccc2c1.C1CCO1 C1(CN(C(C2ON=C(C)C2)=O)C)CN(C(=O)C(C(C)C)C2CCC2)CCO1 CC(C)CC(C)C(=O)NCC1(NC(c2ccoc2CC(N)=O)=O)CCCCC1C N1(C(C(=O)NCCOCCCC)=O)CCC(O)C1.C(=O)CCC1CC1(C)C N1(C(c2c(NCC)scn2)=O)CCOC(C(C)NC(c2cccc(C)c2)=O)C1 Cc1nccc(CCC(=O)NCC2(C)CCN(C(=O)CCc3ccco3)C2)n1 Cn1c(CC(=O)NCC2(O)CCN(C(C3CC4(CC4)CO3)=O)C2)nnc1S c1(C(N(CCC)CC)=O)nc(C(F)(F)F)cc(O)n1.c1(C(=O)N)conc1 N(C(=NCCOc1ccccn1)NC1CCOCC1)CC1C(C)CCC1 C1(NC(C(C(=O)NC)(C)C)=O)CCN(C(C2CCCC2C2CC2)=O)CC1(C)C c1(C(=O)NC)cc(CNC(C2CN(C(c3ccoc3)=O)C2)=O)ccn1 C(=O)(CCC(C)(C)C#N)N(CC(C)(C)C(=O)N1CCCC1)C CC(C)(C(=O)NCc1ccc(-c2ccsc2)cc1)C1=CC2CCC(C1)N2 C1(COC)(NC(=O)CCCc2ccc(C)s2)CCCN(C(=O)C(O)CC(C)C)C1 N1(C(C2CC(O)(CC#C)C2)=O)CC(NC(=O)C(Cl)Cl)CC(C)C1 N1(C(C(C(C)(C)C)NC(C(C)C2(O)CCC2)=O)=O)CCc2ccccc2C1 c1(C(N2CCC(NC(C(CC)=CC)=O)C(O)C2)=O)cc(Br)c(F)cc1C C=CCCCC(C(=O)NC(C)(CSC)CO)NC(=O)C(C)C=C c1(NCc2ccc(C(=O)OC)cc2)ccc(C)c(-n2nnnc2C)c1.C(C)(C)O c1(C(N2CCC(CCNC(c3c(C)c[nH]n3)=O)C2)=O)nc(Cl)c(Cl)s1 N1(C(C2C(C)=CCS2)=O)CCC(C(C)C(=O)NCCc2ccns2)CC1 C1(C(=O)NC2(C(N)=O)CCC2)COCCN(C(C2CC=CCO2)=O)C1 C1(CNC(C(F)OC)=O)CN(C(c2ccc(-c3ccccc3F)o2)=O)CC1(F)F C1(OCC)CCN(C(C2(NC(=O)C=CC3CCCCC3)CC=CC2)=O)CC1C n1(CC)ccc(C(N2CCCC2C(N2CCC(OC)C2C)=O)=O)c1C c1(C(=O)Nc2nnc(-c3ccc(C)c(Br)c3)s2)cc(Br)c(F)cc1F N1(CC(c2n(C)ncc2Br)=O)Cc2[nH][nH]c(=NC(=O)c3ccc(Cl)c(Cl)c3)c2C1 N1(C(C(=Cc2ccc(F)c(F)c2)C)=O)CCN(C(c2cnn[nH]2)=O)C(C)CC1C C1(C#N)(C(=O)NCC2CC(NC(C=Cc3ccc(C)s3)=O)C2)CCCOC1 C(=O)(C(O)CCC(C)C)N1CC(CNC(c2c(C)ccnc2O)=O)C1 CC(C)(O)CCCNC(=O)C(F)CC1CCOC1.C1(=O)C(=O)NC2CN1C2 c1(C(=O)NCC(C(C)(C)C)NC(C(CC)COC)=O)c[nH]c(=N)nc1C N1(C(CC2CCCC(C#N)C2)=O)CC2(CCC(NC(C3(F)CCOC3)=O)CC2)C1 C(C)(C(=O)N)(C1CCC1)NC(C1(NC(C)=O)CCC1)=O.C1CNC(=O)O1 c1(OC)cncc(C(N2CCC(CC(C)(C)C)C2(C)C)=O)c1C N1(C(C2CN(C(CCC)C)C(=O)C2)=O)CCC2(CC1)CC(CNC(=O)C1CC1)C2 CN1CCc2cc(C(=O)NCCCNC(C3CC34CCC(F)(F)CC4)=O)sc2C1 c1(C(N2CC(CC)C2)=O)cc(F)c(C(F)F)cc1F.CC(C=O)OC.C1CC1 c1(C(N(C2CCN(C(C3C(C)CCC3)=O)CC2)CCOC)=O)ccc(F)c(F)c1 C(=O)(C1COc2ccc(Br)cc21)NCCCCN(C)C(C1CC(F)(F)C1)=O CC(C)C(C(=O)NC)NC(=O)C(F)(F)F.C1CCC1.C1(O)(C=O)CCC1 c1(CC)ccc(Cl)c(C(N2CCC(C(C)NC(=O)Cc3ccccc3F)C2)=O)c1 N1(C(C(CCCNC(C2(C)CC(=C)C2)=O)O)=O)CCC2CCN(C)CC12 c1(CNC(c2n(C(CC)(C)C)nnn2)C2C3COCC23)c(F)cc(F)c(F)c1F CC(C)(CS(N)(=O)=O)C(=O)NC1CCCN(C(=O)CC2(O)CCC2)CC1 N1(C(C2(C#N)CC23CCC3)=O)CC2CC(C1)C(O)C2O c1(OC)ccc(C)c(C(N2CC(C)C2(C)C)C(=O)NC2(C)CC2)c1 CC(C)C(CC(=O)NC1(CNC(=O)C(O)C(F)F)CC1)C(C)C C1(N(C)C(c2ccsc2Cl)=O)CC2CCC(C1)N2C(=O)Cc1ccnn1C N1(C(C)=O)CC(C)OC2(CCN(C(c3ccccc3C(c3ccsc3)=O)=O)C2)C1 c1(OC)ccc(-c2cn(C(C)C(N3CCCCC3C(C)(C)OC)=O)nn2)nc1 C1(CC(=O)NC(COC)C(C)C)CCCN(C(C2(CCF)CCC2)=O)C1 C1(C(=O)NC2(C)CCCN(C(C(C(C)C)NS(N)(=O)=O)=O)C2)CCCCC1C1CC1 C(=O)(C1=CCCC1C)N1C2(C(N3CCC(C)(C(C)C)C3)=O)CC2CC1 C1(NC(CNC=O)=O)CC2CC1CN(C(C1CC(F)C(=O)N1)=O)C2 Cc1cc(Cl)cc(C)c1OCC(N1CCC(C)CC1)=O.n1(CC(=O)N)ccnn1 C(=O)(C1=CS(=O)(=O)CCC1)N1C2CC(CNC(C(C)n3cncn3)=O)C1CC2 N1(C(=O)NCc2ccncc2Cl)CCC(S(=O)(=O)N2CCOCC2)C1 N1(C(Cc2cc(C)no2)=O)CCCCC1CN(C(=O)C=CC1CCCCC1)C C1(CCNC(=O)Nc2cccc(C(=O)OCC)n2)CCC(F)(F)CC1 CCC(CC(=O)NC(C)C(C)(C)NC(c1nccc2ccncc12)=O)C(C)(C)C C(=O)C1=CCS(=O)(=O)C1.N1(C(C2CC(C#N)C2)=O)CC(C(F)(F)F)CC1.C c1(C(N2CCC(CO)(COC)CC2)C(=O)NCCCC)ccc(C)cc1Cl N1(C(C)CC(=O)O)CCN(C(=O)CSc2nc(-c3cccnc3)no2)CC1 N1(C(c2ncc(OCC)cc2Cl)=O)CCCC2(C1)CCCN2C.C(=O)(C1CC1)N c1(C(=O)NC2C(CC)CN(C(=O)C(CC)(CO)OC)CC2)cc(F)c(C)cc1O CCCC(CNC(C1(C2CC2)CC1)=O)C(=O)N1CC(CO)C(O)C1 c1(CC)nc(C)c(C(=O)NCCN(c2nc(C)nc(C)c2C)CC)c(C)n1 N1(C(C(C=C)(C)CC)=O)CCCCCC(NC(c2cnc(C(F)F)c(C)c2)=O)C1 C1(NC(CSCCC=C)=O)(CO)CCN(C(C23CCC(C2)C3)=O)C1 c1(C(N2C3C(NC(C(C)Cc4cnc[nH]4)=O)C(C3)C2)=O)cnc2c(c1)ncn2C Cc1ccc(C(=O)NC(C)(CO)C(=O)NCCS(C)(=N)=O)cc1C C1(CNC(CN(C(=O)C(N)=O)CC#C)=O)CCC=CO1 c1(N2CC(C(C)NC(Cc3c(C)nc[nH]3)=O)C2)ncnc2c(C)csc12 c1(C(=O)NC2(C)CN(C(c3c(C)sc(O)n3)=O)C2)ccc(S(C)(=O)=O)o1 C1(C(=O)NC(CCSC)C(=O)NCc2ccns2)CC(C)CC(=O)N1 N1(C(CCOC)=O)CCCN(C(C2CC2c2cn[nH]c2)=O)CC1C C1(C(C(=O)N(C)CC2(NC(=O)CNC(N)=O)CC2)O)CCCCCC1 C(C(CC(=O)N1CC2COCC2O1)C1CCC1)NC(CCCCCC)=O CCCCCC(=O)N1CCC(C)C1.Cc1cccc(NC(=O)C#CC(=O)N(C)C)c1 C(=O)(C(C)CC(C)(C)C)NC(CNC(c1scc(C)c1Cl)=O)C(C)C CC(C)C1CC(NCCC2(O)CCN(C(=O)OC(C)(C)C)C2)c2ccccc21 CC(CC(C)(C)O)NC(C1(C(=O)OC(C)(C)C)CC1)C C1(OC)CCC12CC(C=O)C2.C1(C(N2CC(O)(CC)C2)=O)CC2(C1)CC2F.N CN1CCC(N(C(=O)C(c2ccccc2)NC(C2CNC(=O)N2)=O)C)C1 Cc1ccc2cc(C(=O)NC(C)(C)CCCNC(C3CC4(CC4)C3)=O)[nH]c2c1 C(=O)(C(C)C(C)(F)F)N.C1(C(N(CC(C)O)CC)=O)CCN(C2CC2)CC1 N1(C(C(C)=C(C)C)=O)CC2(CCN(C(=O)CCC3COC(C)(C)O3)CC2)C1 C=CC(CC)CC(=O)N1CCCC1CN(C)C(c1cncc(CC)c1)=O C(CCCCNC(=O)Cc1nccs1)NC(CSCC=C)=O CCC(CC1CCCCC1)C(=O)N(C(C)CN(C(=O)C(C)(C)n1cccn1)C)C Cc1nn2c(c1C(=O)NC1CCN(C(=O)C=C(Cl)Cl)CC1C(C)C)CCCC2 C(C)(CCCC(=O)NC(C)(C)CSC)NC(c1c(OCC)nccc1)=O c1(C(=O)NCC2CC2)ccc2cnccc2c1.C(=O)C(F)(F)C(O)C1CC1.N c1(C(C)C(=O)NC2CN(C(=O)CC3CCOC3)C2)cnn(C)c1 C1(C(C(=O)N(CC(F)F)CC#C)O)CCC(F)(F)C1 C1(C)(CCC(=O)N(CCCNC(=O)C(Cl)=CCl)C(C)C)CCC(=O)N1 CCC(CC)CCCC(=O)N(C1CC(OC(C)C)C1)CC(N1CCCC1)C C=CC(C)(C)CCNC(C1(COC)CCCN1C(=O)CCC)=O.C(C)=O.N C1(CC(=O)NC2(C)CN(C(c3c(C)scn3)=O)C2)COCC(C)O1 CC1(C)CN(CCNC(=N)NCCOCC(F)(F)C(F)F)CCO1 CCC(CN(C)C)C(=O)NC(Cn1ccnn1)C(=O)NCc1cncn1C c1(C(C)C)ccc(N2CCCC2)c(-c2ccc(CNC(c3ccsn3)=O)nc2)c1 N1(c2ccnc(NCCCn3ncc(C)c3)n2)CCC2(CC1)CSC2 C1(C(=O)NC2CCN(C(CCCSC)=O)CC(O)C2)CCc2c(n[nH]c2C)C1 Cc1cc(C(=O)NCC(CC2CC2)C(=O)N2CCC23CCC3)[nH]c1C c1(NCC2S(=O)(=O)CCCC2)nccc(=NCC2CCCC23CC3)[nH]1 CC1(CNC(=O)C(c2ccc(F)cc2)F)CN(c2ncc(O)cn2)CCO1 C=C(Cl)CCC(=O)NOC(CC(C)C)C(=O)NC(C)C1CC1 N1(C(C(C)(O)CC(F)F)=O)CCCC2CN(C(C3(F)CCCCC3)=O)CC12 C1(NC(C(CC)CC)=O)CCC2CCN(C(c3cn4c(n3)CCCC4)=O)C12 c1(C(N(CC(CC)NC(=O)C(C)OC)CC)=O)nnn(C)c1C(F)(F)F c1(SCC(=O)NC(C)C(C)NC(c2cncnc2)=O)nccn1C(C)(C)C c1(C(N2C(C)(CNC(C(C)NC(CC)=O)=O)CCC2)=O)cc(C)c(C)cn1 c1(CN2CC3CC3C2)ccc(S(C)(=O)=O)o1.CC(C)C.C(=O)C=CC=O c1(C(N2CCC(NC(c3ccc(C)nc3)=O)C2C)=O)cnc(Cl)cc1N N1(C(CCn2ccc(C)n2)=O)CCCC12CCCN(C(c1nc(O)c(C)s1)=O)C2 C(=O)(C(=O)C(C)(C)CC)N1CCN(C(c2ccc(OC)cc2)=O)CC1C C(=O)(C1=Cc2ccccc2C1O)NCC(C(C)(C)C)NC(c1cnn[nH]1)=O c1(C(=O)NC(CN(C(c2c(CC)cno2)=O)CC)CC)cc(F)c(C)cc1Cl c1(C(=O)N)cccc(-n2ccc(C)n2)c1.C(CCC(=O)NCC(F)C)NC(C)=O CCCC(CC)CCC(=O)N1CCN(C(c2ns[nH]c2=O)=O)CC1CCO C(=O)(C1CCc2snnc21)NC(C1CCCNCC1)C C1(C(N(CC(C)NC(=O)Cn2cnnc2)C)=O)CC2CC1C1CC21 N1(C(CSC)=O)CCCC1C1CCCN1C(=O)COCc1ccccc1 CCC(CC(=O)N1CCN(C(c2ccc(Cl)cc2)=O)C(C)C1C)CC(C)C C(CCCC(C)NC(c1ccc(C(C)(C)C)nc1)=O)NC(CCCOC)=O C1(SCC(=O)N(CC(C)N(C(=O)CCc2ccon2)C)C)CCOC1=O N1(C(N2C(COC)CCOCC2)=O)CCc2nn(C)cc2C1.C1CC2CCC1CC2 C(=O)(C(C)C(C)(C)C)N(CCC(=O)NCCCNC(=O)OC)C c1(OCC(=O)NCC(C)CNC(c2ccc(Br)cn2)=O)ccc(F)cc1 c1(C(N(C2CCNCCC2C)c2cc(OC)ncn2)=O)ccc(F)cc1[N+](=O)[O-] CCC(O)CC(=O)N1CCCC1C(C)(C)NC(=O)CC(c1ccc(C)cc1)C N1(C(CCCC#C)=O)CCc2c(C(N3CCn4nc(C)cc4C3)=O)csc2C1 CCCCCC(O)CNC(=O)C(C)NC(C1CC(OC2CC2)C1)=O C1(C=O)CC(N(C)C)CCO1.c1(C(N(CC(C)(C)C)CC)=O)n[nH]c(C)c1C Cc1cc(=NC(=O)CN(C(=O)CCC(=O)N(C)C)C)[nH]c(Cl)n1 n1(CC)c(C(=O)N(CC(C)(C)CNC(c2ccccc2)=O)C)nc2ccccc12 C1(NC(C(C)SCC)=O)Cc2ccccc2C1NC(=O)C(c1ccncc1C)C N1(C(c2c(OC)cccn2)=O)CCN(C(=O)C(C)CC(F)F)C2CCCC12 N1(C(CSCCCC)=O)CC(C)CN(C(=O)CC2CCOC(CC)C2)C(C)C1 C1(C(=O)NC2(CCCC(=O)NC(C)CSC)CCC2)(OC)CCOC1 N1(CCNC(COC(CC)C)=O)CCN(C(=O)C=C2CCC(C)CC2)CC1 c1(C(N2CCC(C(C)(C)NC(C(CC)C)=O)C2)=O)c(Br)ccnc1OC c1(C(n2cc(CCNC(=O)C(C3CCS(=O)(=O)C3)C)nn2)C)ccc(F)cc1 C1CC(O)C1(C)C.C1(OCC(=O)N(C(C)C(=O)NC)CC)CCCCC1 N1(C(c2cc(C(=O)OC)c(C)n2C)C(=O)NC2CC2)CCN(C)C(=O)C1C C1(F)(C(=O)NCC(CC)C(C)C)CCN(C(C2(F)CCOC2)=O)CC1 c1(OC)cc(C(=O)NC2CC2)c(N)c(C)c1.C1(C(=O)N)COCC(C)(C)O1 C1(=O)C(C(C)C)N1.C(=O)(C(F)CC1CCC1)N1CC(CCC#C)C1 C1(N(C)C(C2CCCN2C(=O)CCC2CCC2)=O)CCCC1(C)O C1(NC(Cc2c(C)ncs2)=O)CN(C(c2cncc3c2CCC3)=O)CC1C1CC1 c1(OC)c(CC(=O)NC(C2CCN(C(=O)C(C)(C)SC)C2)(C)C)cccc1C#N C1(NC(CN(CCC)C(C2CC23CC3)=O)=O)CCCCC1NC(N)=O C(=O)(C(F)C(=O)N1CCCC(NC(C2CCCO2)=O)C1)OCC N1(C(C(C#C)(C)C)=O)CC2CCC1C(CNC(c1cnc(C)[nH]c1=N)=O)C2 C1CN(C(=O)CC)CC1C(F)(F)F.c1(C=O)cccs1.C(C(=O)N)SCC N1(C(CCN(C(C2C(C)CCC2)=O)C2CC2)=O)CC2(CCN2C)C1 C1(CNC(=O)CSCCC(F)(F)F)COCC1.c1(C=O)cn(CCO)nn1.C N1(C(CC2(C)CC2)=O)C2CC=C(C(=O)N(C3(O)CCC3)C3CC3)C1CC2 C1(NC(c2cc(C(C)C)n(C)n2)=O)CC2CN(C(=O)C(N3CCSCC3)C)CC12 N1(CCOc2cccc(OC)c2)C2CCC1CN(C(c1snnc1C1CC1)=O)C2 c1(-n2c(C3CCCOC3)nc(-c3ccn(C)n3)n2)ccc2ccsc2c1 C1(CNC(c2c(CC)n(C)nn2)=O)CC(C)CN(C(c2ccc(C#N)o2)=O)C1 CC1(C)OCCOC1CC(=O)NC1CCC(NC(=O)Cn2cnnn2)C1 C1(C(N(CCC(=O)NCC(C)CC2CCCC2)CCCO)=O)CC2CCCC2C1 c1(C(=O)OCC)ccc(C(=O)NC2CCCC2)cc1.C(=O)C=CCBr.C c1(NC(=O)C(CC2CC=CCC2)N2CCC2c2cccc(Br)c2)cccc(Cl)c1F N1(C(C2(C#C)CCN(C(c3oc(CC)nc3C)=O)C2)=O)CCC(C2(O)CC2)CC1 C(C(C)(O)CC(=O)N1CCC(OCC(=O)N(CCCF)CC(C)C)C1)OC c1(C(=O)NCC2C(NC(=O)C(c3ccc(Cl)s3)=O)COC2)cnc2n1CCOC2 C(CCC1CC1)(C(=O)NC(c1nncn1C)C)NC(c1c(C(C)C)cco1)=O N1(C(C(C)N(C(CC2(OCC)CCC2)=O)C)=O)CCC12CCSCC2 c1(NC2CC(NC(CCc3cc(C)no3)=O)C2)ccnc(CO)n1 Cc1nn(CCC(=O)N(C(C)CC)C)c(C)c1[N+](=O)[O-].C(C=C(Cl)Cl)=CC=O.N C(=O)(C1=COCCC1)N1CC(C)CC1.c1(OC)ccc(C2(C(=O)N)CC2)cc1.C C(C(F)C(=O)NCCC1CCC1)N(C(C1CCCN1C(C)C)=O)CC.N C1(NC(=O)CCC2CC2(Cl)Cl)CCN(C(C2CC2C2CCCCO2)=O)CC1.CC CC1CN(C(C23CC2CCN3C(=O)COC(C)(C)C)=O)CC(C(N)=O)O1 c1(C(N2CC(C(C)NC(C3CCC(CCCCC)O3)=O)C2)=O)ncc(N)nc1C CSC1=C(C(=O)NCC(=C2CN(C(c3cccc[n+]3[O-])=O)C2)F)CCCC1 N1(C(C(C)SCCCC)=O)CCOCCC1C(N1CC(C(=O)OC)(OC)C1)=O c1(C(=O)NCCCNC(C2CCC(OC)CC2)=O)cc2c(O)cccc2[nH]1 c1(CN(C)C)nc(C2CCCN2C(c2coc(NC(N)=O)n2)=O)no1 c1(C(N2CCCC(CNC(COC)=O)CC2)=O)cc(F)c(Br)cc1F C1(C(N2CCC(NC(Cc3cc(CC)no3)=O)C(F)C2)=O)CC2CSCC(C1)C2 c1(CC(=O)NCC2N(C(C(C)c3ccon3)=O)CC2)sccc1Br CC1=CCC(C(=O)NC(C2CCN(C(=O)CC3CC(C)(C)CO3)CC2)C)CC1 c1(CS(N2CCN(C3(C(=O)OC)CCCC3)CC2)(=O)=O)cccc(Cl)c1F c1(C(=O)NCCC(C)C)cc(O)cc(C#N)c1.c1(C(=O)N)ccc2c(c1)COC2 c1(C(=O)NCC2N(C(C(C)C)=O)CC(O)C2)cc2cc(Cl)ccc2s1 CCC(C)C(CC(=O)NC1CC2(C1)CC21CCC1)NC(c1ccc(Cl)cn1)=O Cc1sc(C(=O)NCC2C3CN(C(C4COC(=O)C4)=O)CC23)nc1O c1(C(N2CC3C(NC(c4cc(CC)[nH]n4)=O)(C3)C2)=O)cccc2c1NC(=O)C2=O CCCS(=O)(=O)CC(=O)N(CCCOCC)C.C1(C)(CC(=O)N)CC1(F)F c1(OC)cc(C(=O)NCC2(C)CCCN2C(=O)C(F)O)cc([N+](=O)[O-])c1Cl c1(C(=O)NCC(C)CNC(c2ncoc2C2CCC2)=O)nncn1C1CC1 C1(C)(C(=O)NCC2(F)CC(NC(C3C(C)CC3)=O)C2)CCC(F)(F)CC1 C1(OCC)CC(OC(=O)Cn2ccc(C)n2)C12CCCC2 C#CC(C)(C)C(=O)N1CC(OC)C(NC(c2cc(-c3cccs3)[nH]n2)=O)C1 C(=O)(CC(C)C(F)(F)F)NCC(CC(C)C)NC(=O)C(CO)NC(N)=O c1(NCCC2CCC(NC(CSc3n(C)cnn3)=O)C2)ncc2[nH]ncc2n1 O=C(C#CC1CCCO1)NCCN1CCN(C(c2cc3scc(Cl)c3[nH]2)=O)CC1 C1(C(N(CC(=O)NC)C)=O)CN(C(=O)C(C)OC)CC12CCC2 c1(C(=O)NC2C3CN(C(c4c(CC)nccn4)=O)CC32)ccc2cc[nH]c2c1 c1(C=O)cc(S(=O)(=O)N(C)C)c[nH]1.C(=O)(C(C)(C)C(=O)N)NC.CCCC N1(C(CNC(CCC)=O)=O)CC2CCC(C1)N2C(C)C(=O)Nc1ccc(O)cc1 Cc1ccc(S(=O)(=O)NC2CC(C)CC(C)C2)cc1OC(F)F N1(C(=O)NC(c2ccc(F)cc2)C)CCC(C(=O)N)C12CCCCC2.C(C)(C)C C1(NC(c2c(C)nc(CC)s2)=O)CCN(C(=O)CC2CC2(Cl)Cl)C12CCC2 C1(CC)CNC(=O)CN1C(C1CCC(CNC(c2nocc2C)=O)C1)=O C#CCC(O)C(=O)NCC1(F)CC(CNC(=O)CCO)C1.c1ccccc1 N1(C(CCCNC(N)=O)=O)CCC(CCC(=O)NCCc2cccs2)CC1 C(=O)(C(CCCC(C)C)N(C)Cc1nncn1C)NCCCCCC Cc1nn(CC(=O)NC2C3CCN(C(=O)CC(O)Cc4ccccc4)C23)cc1Cl N1(C(C2C(CC)CCC2)=O)CCC2CCN(C(c3cnc4ccccn34)=O)C2C1 c1(C(C(=O)NC2CC(C#N)C2)(F)F)ccc(-c2ccc(=N)[nH]c2)c(F)c1 N12C=CC(=NC(=O)C(OC(F)F)CNC(=O)C1)N=C2O.CC1CCCN1CCO c1(C(C(C)NC(c2ccc(C3(OC)CCC3)cc2)=O)O)c(Cl)cccc1Cl C1(N(CC)CC)CCN(C(=NCCc2ccccc2)NCCC(O)C(F)(F)F)C1 C12(NC(C3=C(C)CC3)=O)CCOC(C)(C1)C2.c1(C(=O)N)cc(N)cc(F)c1 CC#CCCCC(=O)N1CCC(C(N2CCC(C)=C(C)C2)=O)(CF)C1 N1(C(C2C=CC(NC(CCn3ccc(C)n3)=O)C2)=O)CC(C)(C)C1C1CC1 N1(C(CONC(CCC2C(C)C2)=O)=O)CC(S(C)(=O)=O)C1 c1(OCC)cccnc1C(N1CC(N(C(=O)C(O)CSC)CC)C1)=O N1(C(C2C(CC)C2)=O)CC(NC(c2cc(C)sc2C)=O)C2(CC2)C1 Cc1nnc2n1CCN(c1nnnn1CC1CCC3(CCC3)CO1)C2C CN1CC=C(CC(=O)N2CC3(CCCC(CNC(=O)CC4CC45CC5)O3)C2)CC1 C1(NC(CCC)=O)CCCN(C(=O)C=COCCC=Cc2cnc[nH]2)CC1 c1(CNCC2OCCN(C(=O)Nc3ccc(Cl)cc3)C2)cnc2cc[nH]c2c1 c1(C(=O)NCC2N(C(c3cncc(C)n3)=O)CC(O)C2)cnc2c[nH]nc2c1 c1(CNC(CCCCNC(C)=O)=O)ccc(CN(C)C)cc1Cl N1(C(CC(C)C)=O)CC2(CCCCN(C(C3CC3C3CCCC3)=O)C2)C1 N1(C(C2(SC)CCC2)=O)CCCC2(CCN(C(C3CCCNS3(=O)=O)=O)C2)C1 N(C(=NCC(C)(C)C1CCCC1)N1CCC2(CC1)CNC(=O)O2)C(CC)C CCC(CC(F)(F)F)C(=O)NCCC(C)N(C)C(c1ccc(F)c(OC)c1)=O c1(CCCC(=O)N(CCCNC(CSCC#C)=O)C)ccc2c(c1)OCO2 N1(C(c2ccc(CC)o2)=O)CCCCCC(NC(=O)C(C)(F)C(F)(F)F)C1 N1(C(C2(C)CC(F)C2)=O)CC2CCCC(C1)N2C(C1(Cl)CC12CCC2)=O C1CN(C)CCN1C(=O)C=Cc1ccnn1C.c1(OCC)nc(C(=O)N)co1 N1(C(c2cc(C)c(C)[nH]2)=O)CCCC(C)C1C.c1(CC(=O)N)cnn(C(F)F)c1 c1(C(=O)NCC2C3CN(C(C(C=CC)O)=O)C2C3)ccc2nn[nH]c2n1 C1(C(N2C3C(NC(c4c(C)cc(CO)o4)=O)CC(C3)C2)=O)CCc2nncn2C1 N1(CC(=O)NC(C)CNC(C2CCC(=O)O2)=O)C(=O)c2ccccc2CC1=O C(=O)(C(O)CC(C)(C)C)N(C)CC1CCN(C(C2CCCN2CC(F)Cl)=O)C1 C(=O)(C1=CCC2(COC2)OC1)NC.C(=O)(C(F)(F)CCC1CC1)N1CCCC1.C C1(C(=O)NC(C)(CNC(=O)Cn2cccc2)C2CCC2)CCCC(=O)N1 C12CC(C1)C2.C1(=CC=O)CCC(C)C1.CC(C(=O)N)N(CC(F)(F)F)C C1(C)(CCNC(COC)C(=O)OC(C)(C)C)CCOCC1 C12(CNC(Cc3nc(=N)[nH][nH]3)=O)CCCC1CCN2C(c1cn(C(F)F)cn1)=O C1(c2cn(C)nc2)CSCCCN1C(=O)CCC(=O)c1ccnc(C(=O)O)c1 c1(OC)c(C(=O)NC2CC(O)CN(C(c3cnc(Cl)s3)=O)C2)c(C)nn1C c1(C(N2CCC(NC(C3(C(N)=O)CC3)=O)CC2)=O)c(O)nc2ccccc2c1Cl O(NC(=O)CCC(N)=O)C(CC)CC.N(C)C c1(CC)ccc(NC(C23CC2CCN3C(c2coc(COC)n2)=O)=O)cc1O C1(C(=O)NC2C(C)CCN(C(=O)C(O)C(F)F)C2)CCc2nnc(O)n2C1 c1(OC)cc(CN2CC3CC(C2)N3C(c2nc(C)cnc2C#N)=O)cc(Cl)c1O CC1C(NC(c2ncnc3ccsc23)=O)CC2CCC1N2C(c1cc(Cl)c[nH]1)=O Cc1cc2ccccc2cc1C(=O)NCCC(C)(C)NC(C1CC=CCO1)=O C(=O)(CS(=O)(=O)NC)NC1CC(NC(C2(OCC)CCOC2)=O)C1 c1(C(N2CC3C(NC(Cc4c(C)nc(S)s4)=O)(C3)C2)=O)c(F)ccc(Cl)c1F C(C)(C(O)C(=O)NCC(C1CCN(C(=O)C=CC2CCCC2)CC1)(C)C)OC CC1(C)C(NC(=O)CC2CC=CC2)CC1C(=O)NOCC(O)C(C)(C)C O=S(=O)(c1ccc(Br)cc1NCC1CCC(C2CC2)O1)N1CC2OCCOC2C1 C1(NC(C2C(C(=O)OC)C2)=O)C2CC1CN(C(=O)Cc1cn(C)nc1C)C2 N1(S(c2c(NCC(COC)(C)C)ccnc2)(=O)=O)CCC2CCN(C)C(=O)C2C1 C1(NC(C(COCC)O)=O)CN(C(=O)C(c2ccn(C)n2)C)C2CCCC12 c1(NC(=O)NC(C)CN2CC(C)(C)C2)ccccc1OCc1ccccc1 c1(OC)c(C(N2C(C(N3CCC(O)C(F)C3)=O)CCC2C)=O)cc(Cl)cc1Cl C1(OC)CC(NC(C2CCC(C)(C)O2)=O)CN(C(=O)CCN(C)CCO)C1 C1(C(=O)NC2CCCC2NC(C2(n3cccc3)CC2)=O)Cc2ccccc2O1 CC1=NNC(=O)C1CC(=O)NCc1c[nH]nc1C(=O)NCCCCC1CC1 C1(C(=O)NCCN2CCN(c3nc(SC)nc(Cl)c3)CC2)CCCC(F)(F)CC1 CC1CC(C(=O)NC2C(C)CCN(C(c3c[nH]c(=N)o3)=O)C2C)CCS1(=O)=O C1(C(=O)NC2C(C(C)(F)F)C2)(OC)CCN(C(c2cnco2)=O)C1 C1(CC#C)CN(C(C2(C)C=CCN2C(c2c[nH]nc2OC)=O)=O)CCO1 N1(C(COCC#C)=O)CC2CCCC(C1)N2C(c1ncccc1N)=O C(=O)(CC1OCCc2ccsc21)N1CCN(C(CCC(C)(C)C)=O)CC(O)C1 N1(C(c2n[nH]c(CC)c2Cl)=O)CCCCCC(NC(=O)COCCCOC)C1 c1c(OC(F)F)ccnc1F.c1(CNC(=O)OC(C)C)ccc(C(=O)N)cc1 C(CC(C)(O)C(C)(C)CNC(C1(NC(C)C)CCOCC1)=O)OC N1(C(C(CC=C)C)=O)CC(F)(F)CC1(C)CNC(=O)C(O)CC(C)(C)C Cc1nn(C)cc1C(C)C(=O)N(CCCNC(=O)Cc1nc[nH]n1)C C1(CCC)CN(C(c2nnn(-c3cccc(C)c3)c2C)=O)CC1NC(=O)CCF N1(c2snc(CC)n2)CC2(CCC2)CC1CNC(C1(F)CC1)=O C1(=O)CCCCCCN1.Cc1cc(CC(C)NC(=O)COC2CCCOC2)n[nH]1 N1(CCc2ccc(OC)cc2OC)CCOC(C)(C#N)C1 CCCC(CCC)CC(=O)N1CCOC(CNC(=O)COC(C)(C)CC)C1 C1(CNC(C(C)Cc2cnco2)=O)CCCC(C)C1.c1(C=O)cc(N)ccn1.N C(=O)(CC(F)(F)CS(C)(=O)=O)N1CC2C(CNC(CSC)=O)(C2)C1 C=CC(CC)C(=O)NCC1(C(=O)NC(COC)C2CC2)CCCO1 C(=O)(C1=COc2ccccc2O1)NC1CCCC(NC(C(C)n2cncn2)=O)C1 c1(OCC)ccc(C(CN)Nc2nc(C3CCOC3)c(C)s2)cc1 C1CN(C(C2CCCN2C)=O)C2(CCC2)C1.c1(CSC)cccnc1C(=O)N.C C1(C(=O)OC)N(C(=O)C(=O)NCc2[nH]nc3ncccc23)CCCC1(C)C Cc1cccc(CCn2cc(CC(C)(C)C(F)F)nn2)c1 CC1CC(NC(c2csc(Cl)n2)=O)CN(C(=O)CCc2cc(F)ccn2)C1 c1(C(N(CCOCCN(C(CCCOCC)=O)C)C)=O)cc2n(c1)CCOC2 C(=O)(C(Cc1ccccc1)C(C)Nc1ccc(NC(N)=O)cc1)OC c1(CC)cc2c(c(=O)o1)C(c1cccnc1C(=O)O)NC(=O)N2C C1(NC(CC=CC=C)=O)CC2CC(C1)CN(C(=O)Cc1cnc3cccnn13)C2 CC(C)CC(CC(C)C)C(=O)NC(C1CCOC1)CNC(c1cnn(C)n1)=O c1(C(=O)NCC2(F)CC(CNC(C(CC)(C)C)=O)C2)ncccc1N=[N+]=[N-] c1(C(C)C)ccc(C(=O)NCC2(NC(c3cc(Cl)no3)=O)CC2)c(O)c1 N1(C(c2cc(C(C)C)on2)=O)CC(NC(C2CC(n3cnnc3)C2)=O)CC(F)C1 C1(C(C)(C)CNC(c2cc(C3CCC3)[nH]n2)=O)COCCN1C(c1cnsn1)=O c1(CC(=O)NCC(C)N(C(Cn2c(C(C)C)ncc2)=O)C)cccc2nonc12 N1(C(C(=O)NCc2cccc(O)c2)=O)CC2CC(C1)c1cccc(=O)n1C2 C1(NC(C=CCC)=O)(CF)CCN(C(=O)Cc2nc(-c3ccccc3)nn2C)C1 C1(NC(CCOCC#C)=O)CC2CC(C1)N(C(=O)CCC(=C)Br)C2 C#Cc1ccc(C(=O)NC2CCCC(CNC(=O)C(C)(C)C(=O)OC)C2)nc1 N1(C(C(CC)C(C)C)=O)CCN(C(=O)COC2CCCC2)C2CCCC12 C1(C(=O)NCC2CCN(C(C)C)C2)CN(C(c2cnsc2)=O)CC1(C)C C1(C)(CC)CC(NC(=O)C2CC2)CN1C(c1cnc(CC2CC2)s1)=O C(=O)(C1=C(Cl)CCOC1)NCC1(O)CN(C(c2onc(CC)n2)C)C1 C#CCC(CC(=O)N(C(C)CN(C(=O)CCNC(=O)OC)C)C)c1ccccc1 C1(CNC(CCc2nc(C)c(C)[nH]2)=O)CC2(CCC2)CN1C(C1OCCC1C)=O C(=O)(CCS(=O)(=O)C(F)(F)F)NCCN(C(c1ccnc(OC)c1F)=O)C C(CCC(=O)NC(C)(C)C(C)NC(=O)CCC=C(C)C)NC(=O)OC CN1CCN(C(c2ccnn2CC#N)=O)CC1CNC(C1CCC(N=[N+]=[N-])C1)=O Cc1c([N+](=O)[O-])cnc(N2CCN(C)CC2C2CCCCC2)c1Br c1(OC)cnc(C(=O)NC(C)CC(=O)NCC2CCN(C(C)C)C2)cn1 C(=O)(CCCC(=O)C1CC1)N1CC(CC(=O)NCC(=O)OC)OCC1 c1(NC)ccc(C(=O)NC2CCC2CNC(c2cnns2)=O)c(Cl)c1 C1(CC)CCC(C(N2CC(CNC(=O)C(C)(C)C#N)(OC)C2)=O)CC1 c1(NC(C)C(=O)Nc2ccc(Br)cc2Br)cnc(O)c2ccccc12 N1(C(CN(C)C(C2C=CCS2)=O)=O)Cc2ccccc2C1 N1(C(c2ccc(C(C)=O)[nH]2)=O)CCN(Cc2cn(Cc3ccccc3)nn2)CC1 N1(C(c2ccc(C)c(N)c2)=O)CCC2CN(C(c3cc(C4CCC4)on3)=O)CC12 C12(NC(C(CN(C)C)O)=O)CCOCC1CN(C(c1ccn3c1CCCC3)=O)C2 C(=O)(CCC(C)CC)NCC(CCCC)NC(=O)CCCn1cncn1 N1(C(CCN(C(C(CSC)O)=O)CC2CC2)=O)CC2CCC(C1)C(=O)O2 N(C1CCc2ccccc21)(C(=O)Nc1cccc(-c2csnn2)c1)CCO c1(OC)cc(CN(C)Cc2cn(Cc3cnc(C(F)(F)F)s3)nn2)on1 c1(C(N2CCC(CNC(C(CC)C(C)C)=O)CC2)=O)cnc2ccc(F)cn12 n1(CC(=O)NCC(CN(C(=O)C=Cc2cccs2)C)O)ncc(O)nc1=O c1(NC(C2C=CCN2C(C2CC(O)C2)=O)=O)cc(Cl)cc(Br)n1 c1(OC)nc(C(=O)NC(C)CCCCNC(=O)C(O)CSC)cc2ccccc12 c1(CCCNCc2n(C)nnc2Br)nnc2n1CCCC2 C(=O)(CN=c1[nH]c(N(C)Cc2sccc2Br)nc2ccsc12)N(C)CC C1CCN(C(=O)C=CC2CCC2)CC1C.N1(C(=O)OC)CSCC1C(=O)N.C C1(C(=O)N(C(CO)C(C)C)C)(CC)CCN(C(=O)COC2CCCOC2)CC1 N(C1CN(C(=O)CCC2CC2)CCc2ccccc21)C(C(COC)NC(C)=O)=O C1(OC)(OC)CC2(COC(CNC(=O)Cc3ccc4ccoc4c3)C2)C1 CC1(CNC(C2CCC(=O)C2)=O)CCN(C(=O)CC(C)(C)c2ccccc2)CC1 c1(C(c2n(CC=C)nnn2)NC(C2CC(F)(F)C2)C)ccc(F)cc1 C1(CC=C)(NC(c2cccc(Cl)c2Cl)=O)CCCN(C(C2CC3(CSC3)C2)=O)C1 c1(OC(C)(C)C)ccc(C(C(F)F)OC(C2OCCC2(C)C)=O)cc1 c1(C(=O)NCCCNC(=O)C(F)C(F)(F)F)cc(Cl)cc(Cl)c1F Cc1cc(C(=O)NCCC2CCCN(C(=O)Cc3c[nH]nc3O)C2)nn1CCO C=CCCC(C=O)NC(=O)C=Cc1ccco1.C1(C=O)(C(=O)C2CC2)CC1 C1(NC(CC(C=C)C)=O)CN(C(c2nc(C)nn2C)=O)CCC1F Cn1c(=O)c(SCC2CCCC(C(=O)O)O2)nc2ccccc12 N1(C(C2CCC(=O)NC2)=O)CCCC2C1CCN2c1ncc2c(n1)NC(=O)C2 C1(C(N2CCC(NC(c3ccn(CC)n3)=O)C(F)C2)=O)CC(C)(C)CC(C)(C)C1 c1(CN=C(NCC(=O)OCC#C)NC(C)CF)cccc(C#N)c1 C1(C=O)CCCC(F)C1.c1(C(C(N2CC(CO)C2)=O)OCC)ccc(F)cc1.N C1(C(=O)N)COCCN1.c1ccnn1C.C1(C(N(C(C)C)CC)=O)(C)CC1 CCCCN=c1[nH]c(CC(=O)NCC2CCC(S(C)(=O)=O)CC2)cs1 C1(CS(N2CCN(C=O)CC2)(=O)=O)CCOCC12CCCC2 C(=O)(C(F)(CNC(c1cccc(C)c1C)=O)C(C)C)NCP(OCC)(C)=O C1(NC(c2cccc(C)c2Cl)=O)CCN(C(c2cnn3cc[nH]c23)=O)CC1(C)C c1(C(=O)Nc2ccc(C)c(SS(C)(=O)=O)c2)cc2c(F)ccc(Cl)c2[nH]1 CC(Cc1ccccc1)C(=O)NCCCN(CCCNC(C1CCO1)=O)C N1(C(c2nc(C(C)C)oc2)=O)CC2(CCN(C(C3CNC(=O)N3C)=O)C2)C1 N1(C(C2N(C(C)(C)C)CC2)=O)CC2CC1CN2C(C1(O)CCSCC1)=O c1(OC)cc(C=O)ccc1C.C1(C(N(CC(C)C)C)=O)CCCS(=O)(=O)N1.N c1(COCC)nc(N2CCSCC2CCNC(C2CCCC2)=O)cc(Cl)n1.O N1(C(c2c(C)noc2C(F)F)=O)CCCC(F)(CNC(=O)CCCC(C)C)C1 n1(CCC(=O)NCCC2N(C(C#CC(C)C)=O)CCCC2)cc(S(N)(=O)=O)cn1 C1(CC(=O)NCCC2(C)CC2(F)F)CN(C(c2cc(C#N)cs2)=O)CC12CC2 c1(C(c2ncc(C)s2)C)nnc(N2CCCC2c2cc(C#N)cs2)n1CC1CC1 c1(C(=O)NCC2N(C(C3N(C)CCC3)=O)CCOC2)ccc(N2CCCC2)cc1 O=C(C1CSc2ccccc21)NC1CN(C(C2CC3(CC3)C2)=O)C2CCCCC12 N1(C(C2N(CCC)CCC2)=O)CC(C)(C)CCC1C.C1(C=O)CC(N(C)C)C1 CCC(C)CCC(=O)NCC1(C(=O)NCCC2CCCCO2)CC(C)(C)C1 N#Cc1ccc(CC(=O)NC2CCC2NC(C2(C(N)=O)CCC2)=O)c(F)c1 c1(C=O)cc(C)cn2ccnc12.C1CC(F)(F)C1.C(CC)N(C(=O)C)CC.N C=CCC(C)C(=O)N1CCCC(CCNC(C2CCCC(O)C2)=O)C1 N1(C(CCc2nc(C)sc2)=O)CCC(NC(C2CC2(Cl)Cl)=O)C(CO)C1 C1(C(N2C(C(C)NC(Cn3c(C)ncc3)=O)CCC2)=O)CC(C)CC(=O)N1 C(=O)(N=c1[nH]oc2ncccc12)C1N(Cc2c(C)cc(O)cc2C)CCC1O c1(C(=O)NC2C(NC(=O)CCC3CC3(Cl)Cl)COC2)ccc(C(F)(F)F)cn1 N1(C(C2(F)CCN(C(c3ccc(O)cc3F)=O)C2)=O)CCc2sccc2C1 N1(C(c2nc(CCCC)sc2)=O)CC2CN(C(c3csc(C)n3)=O)CC2C1 Cc1cc(C(=O)NC(CO)C(C)NC(=O)C=CC2CCCO2)c(C)cn1 N1(C(CCC2N(C)CCC2)=O)CC2CC1C2C(N1CC=CC1(C)C)=O c1(-c2c(C=O)con2)ccc(Cl)cc1.C1(NC(C=CCOC)=O)CCCCC1.N C12(CN(c3ccnc(NC(C4CCCCC4)=O)n3)C)CCCN1CCC2 N1(C(C(C(CC)C)O)=O)CC(NC(c2cnn3c2CCCC3)=O)C2(CCC2)C1 C12(NC(C(C)N(C)C)=O)CC3CCC(C1C2)N3C(=O)Cc1ccc(Br)nc1 C=C(CC(C)C)C(=O)OCC(=O)N(c1ccc(Br)cc1)C(C)(C)C C(=O)(CC(C(C)C)Nc1cccc(C(F)(F)F)c1)OCCCSC C12(C(=O)N)CCC(F)(CC1)CC2.n1(CC(N2CC(O)CC2C)=O)ncccc1=O C1(CC(=O)Nc2ccc(F)nc2)C2CCC(C2)N1C(C1CCC(=O)N1)=O C1(NC(C(C(C)C)=O)=O)CC2CC1CN(C(=O)CC(C)C(F)(F)F)C2 CC1CCN(C(=O)C2=CCC2)C(CNC(c2cccc(N3CCCC3=O)c2)=O)C1 c1(C(=O)NC2CCN(C(c3c(C)nc(N)cn3)=O)CC2F)c(C)ccc(Cl)c1F N1(C(C(C)C)=O)CCN(C(c2nc(C(F)(F)F)cn2C)=O)C(CCO)C1 c1(NC(C)=O)ccc(F)c(C(N2CC3CNC(C3)C2)=O)c1 c1(C(=O)O)cc(NCC2(CO)CC3CC3C2)ccc1Br CN1CCCC1C=CC(N1CCN(C(=O)CN2CC(C)(C)C2)CC1)=O C1(C(=O)NC(COCC)C(C)C)CCCCCCN1C(=O)C(O)C(F)(F)F C1(CC)(NC(c2csnc2Cl)=O)CCN(C(=O)C=Cc2ccsc2)CC1 c1(C(N2CCC3(CC(NC(C4CC4F)=O)C3)C2)=O)cc2c3c(cccc3c1)CC2 N1(C(CN(CC#C)C(c2cocc2C(N)=O)=O)=O)CCC(C)C1.C(C)=O C1(N(C(=O)CCC2CC(NC(C34CCC(CC3)C4)=O)C2)C)CC(O)C1(C)C C(CSC1CC1)(C(C)C)(C1C=CC(COC)C1)c1nnnn1C.C1COC1 c1(OC)cc(C(=O)NC2CC(NC(=O)CCc3cncnc3O)CC2O)ncn1 c1(OCC)ccc(S(C)(=O)=O)cc1CN.C1CCN(C(N2CCOCC2)=O)C1 C1(C(=O)NCC2(O)CN(C(C(C3CCOCC3)C)=O)C2)COCCN1CC(F)F CCCCCC(C(=O)NCC1(O)CCN(C(=O)COCC)C1)C(C)C.CCO.O CN(CC1CCCCCC1)N1CC2(CCCC2)C1c1ccccc1 C1(NC(C(C)=C2CCC2)=O)CC(F)C1.C1(c2ccccc2)(C=O)CC(C)C1.C N1(C(c2ncc(C)c(C)c2)=O)CCC2CCN(C(C3CCCCC3)=O)CC2C1 C1(C(=O)NCC(CC)NC(=O)CCOC2CCCC2)CC12CCOC2 CCC(CC(=O)NC1CN(C(=O)C2=CC(C)(C)C2)CC1n1ccnn1)C(F)F C(=O)(CCC(C)(C)C)N1CCC(O)(C(C)CNC(C2(F)CCOCC2)=O)C1 C(CCCCC(=O)N1C(C(=O)NCC(c2ccccc2)(C)C)CC1C)=CC C1(C(N2CCC(N(C)C(c3cccnc3N(C)C)=O)C2)=O)CC(=O)NC1(C)C Cc1cc(O)ncc1C(=O)NC(CO)CCCCNC(C1CCC(=O)O1)=O CC(C)CCCCCC(=O)N1CC(NC(c2cc(Cl)cs2)=O)CC(O)C1 CCC(CC(C)C)C(=O)N.c1(C(N(C(C)(C)C)CC)=O)cc(O)c(O)c(Cl)c1 C12(C(=O)OCC)CCCC1N(Cc1cc(I)cc(I)c1O)CC2 c1(CC(=O)NC2CCCCC2NC(C2CC3(CC3)C2)=O)cnc2ccccc2c1 c1(C(=O)NCc2cnc(NC(=O)C(c3cccc(Br)c3)O)s2)cccc(F)c1Br c1(OC)c(F)cc(CN=c2[nH]c(C)c(C(=O)Nc3cncc(Cl)n3)s2)cc1F c1(OCC)ccc(C(=O)NCCCO)cc1.c1(C(=O)N)cccc(CC(C)C)c1 N1(C(C(CCC)C)=O)CC(NC(c2cn3c(n2)COCC3)=O)CC(F)(F)C1 c1(OC)ccc(F)cc1CCNC(C1(Cl)CC1(F)F)=O n1(CCCNC(CCN(CC)CC)=O)cc(C2(O)CCCC2)nn1 C=CCCCCCC(=O)NC1CN(C(c2cnc3cccnn23)=O)CC1(C)C c1(C(=O)NC2CN(C(CC(=O)NCC)=O)C(C)(C)C2)c(N)cc(Cl)cc1Cl C(=O)(C(F)(F)C(F)(F)C(F)(F)F)N(CCC)C.c1(C(=O)N)ccn(CCF)n1 C1(C(N2CCC(=CCNC(CCN(C)CC)=O)CC2)=O)CC2(C1)CC(F)C2 C(=O)(CCCCC(C)(C)C)N1C2(CC)CC(C1)C2.C12C3CCCC3N1C(=O)C2 c1(OC)ccc2c(c1)CCC2C(=O)NC(C)CN(C(=O)CC1CCC(C)CC1)C C12(C(=O)NCC(N(OCC)C)=O)CCCC1CCN2C(=O)Cn1cnnc1 N1(c2n(CCC#C)c(-c3ccc(CC#N)o3)nn2)CCN(S(C)(=N)=O)CC1 C(=O)(C(O)CN1CCCC1)NC(C(N)=O)C1CC1.c12coc(n1)NC2=O N1(CC(=O)NCC(CN(C)C(C2CCCOC2)=O)(C)C)C(=O)CCC1=O CC1(C)CN(C(c2ccc(CO)o2)=O)CC(C)(C)C1NC(C1CCCN1N=O)=O C(CCN=C(NCC1CC1C=O)NC1CC1)OC(C)(C)C.c1ccc(Cl)cc1 c1(C(=O)OC(c2cccc(CC(C)C)c2)C(F)F)ccc2c(c1)CNC(=O)N2 C1(NC(CCN(C)CCO)=O)CN(C(C2(CO)CCCCC2)=O)CC(C)(C)C1 C(CCSC)(C(=O)NC(CC1CCC1)CO)NC(C(C)OC)=O N1(C(CS(=O)(=O)N(CC)CC)=O)CC2CCC1C2.C(=O)CCC(C)N(C)C.N N1(C(C(COC)(F)F)=O)CCC(C2(O)CN(C(=O)C(N3CCSCC3)C)C2)CC1 C(C(C)(C)C(C)O)NC(c1nc(C(C)NC(c2ccc[nH]2)=O)oc1)=O C(CC(=O)N)(C1=CCCC1)OCC.C1(CC)COCCN1C(=O)CN(C)CCO C12(NC(c3c(C)nn(CCO)c3)=O)CCN(C(c3cc(CO)[nH]n3)=O)CCC1C2 NS(=O)(=O)C1CCC(NC(=O)Nc2ccc(Cl)c(C(F)(F)F)c2)CC1 C1(C)(NC(c2c(CC)nn(C)c2)=O)CCCCC1C(=O)NOCC(O)C(C)C c1(C(N2CC3C(NC(C(C)(C)CF)=O)C(C3)C2)=O)cccc2ncnn12 CC1CCN(C(=O)Cc2cnsc2)CC1NC(=O)C=CI C1(C(=O)Nc2cccc(C(=O)OCC)n2)CCN(Cc2cccnc2F)CC1O c1(C(N2CC(C)CC(C)C2)=O)ccc(S(=O)(=O)C2CCOC2)cc1 c1(CCC)c(C(=O)NC(CNC(c2ccccc2)=O)CCOC)nnn1C c1(C(=O)NC2CC(C)(CC)N(C(C3CC(O)C3)=O)C2)cnc2[nH]c(O)nc2c1 c1(NC(c2cn(C(C)C)nn2)c2nnnn2C(C)C)cc(Cl)cc(Br)c1 CCC(CC(F)F)C(=O)NC(C)CNC(c1ccc(OC)cc1C(F)(F)F)=O C12(C(=O)OC)CCC(C(N3CCN(C(C4CCC(C)C4)=O)CC3)=O)(C1)C2 C=Cc1cncc(C(N2CCC(C)C(NC(=O)Cc3ccccc3F)C2)=O)c1 Cc1cc(=NC(C)c2ccnc(Cl)c2F)[nH]c(N2CC3CCOC3C2)n1 c1(Nc2c(C)nc(CCNC(C(CC)(C)OC)=O)s2)ccc(F)cc1C C1(CC#C)(C(=O)NCC2CCC2)CC=CCC1.C1(C=O)CCC(C)(C)O1.N N1(C(C(C(C)O)N(C)C)=O)CCC2CC2(C(N2CC(O)C2)=O)CC1 N1(C(CCOCCCOC)=O)CC2CCN(C(=O)CCn3cccnc3=O)CC12 N1(C(C(C2CC2)OC)=O)CCC2C(CCN2C(=O)CCc2nc(=N)[nH][nH]2)C1 c1(CN(CCCC(=O)O)C(=O)NC2CCCSC2)cccc(F)c1 c1(C(=O)NCC#CCNC(CCCCOC)=O)ncn2ccccc12 c1(C(=O)OC)cc2n(n1)CCCN(C(c1ccc(F)s1)C(=O)NC(C)C)C2 c1(CC(=O)NC2CC3N(C(COC)=O)C(CC3)C2)ccc(Br)c([N+](=O)[O-])c1 C(=O)(CCn1ccnc1)NCC=CC(=O)N(C1CC(CO)C1)C c1(C(N2CC(O)(CNC(=O)CC3CC4CC4C3)C2)=O)cc([N+](=O)[O-])cnc1O N1(CCNC(C(C)OCCOC)=O)CCCN(C(C2CC(C)C2)=O)CC1 N1(C(C2C(C)CCO2)=O)CCCC(C(C)(C)C(=O)NCc2ccncc2Cl)C1 c1(C(=O)NC2CCCC(NC(=O)COC3CCOCC3)C2)cc2cnccc2[nH]1 C1(NC(c2nc(C(C)OC)oc2)=O)CC2CCC1N(C(c1cscn1)=O)C2 CC(N=c1ccc2c([nH]1)CCC2=O)C1CCN(C(=O)C(C)OCCN(C)C)C1 C1(NC(c2c(CC)nns2)=O)CCCC12CN(C(c1ccc(OC)c(O)c1)=O)C2 N1(C(CC2COCC(C)O2)=O)CC2(C1)CN(C(c1csnn1)=O)C2 C(=O)(C(C)CC(C)(F)F)NCCN(C(c1cnc(C(C)C)s1)=O)CC C1(C(=O)NCC(O)CNC(=O)CC(C)n2cccn2)(CC)CCCC1 N1(C(c2c(CC)cno2)=O)CC2CC(NC(=O)CO)C(C2)C1.c1ccccc1 c1(C(C)(C)C)nnn(CC(=O)NCC2CN(C(=O)C=CCF)C2)n1 C1(CNC(CC(C)C)c2n(CC=C)nnn2)(OCC)CC(C)(C)CO1 c1(N2CC(C(C)N(C3CC3)Cc3cncc(Br)n3)C2)ccc(C(=O)O)cc1O C(=O)(C(CC=C)CC(C)C)NC1(CC=C)CCN(C(=O)COC2CCCCC2)C1 C=CC1CCCC(NC(=O)CCC2CC(NC(=O)C(C)O)C2)C1 CC1N(C(c2ccc(CNC(=O)OC(C)(C)C)cn2)=O)CCCC1(C)C C1(CC)CC1N=c1nc2ncn(CCN(C)C)c2c(NC)[nH]1 Cc1cc(NC(C2(C)C=CCN2C(C2CS(=O)C2)=O)=O)cc(F)c1 C1(O)CCN(C(C2CC(=C3CC3)C2)=O)CC1.c1(OC)cncc(C(=O)NC)c1 C(=O)(C1CSc2ccccc21)NC(CC)(CC)CCNC(=O)CSCCOC N1(C(C2(CC=C)CCCCC2)=O)CCCC(O)(CNC(C2CC2(F)F)=O)CC1 CCCC(CCC)CC(=O)N1CCCN(C(=O)C=CC2CCCN2C)C(C)C1 C(=O)(C(F)C(F)(F)F)NC(CC=C)CNC(=O)C(c1ccccc1F)(F)F N1(C(CC2C(C)(C)CCO2)=O)CC2CCN(C(c3cnccc3Cl)=O)C2C1 C1(C(N)=O)CCCN(CCC(=O)NCC23CC(CN2C(C2CCO2)=O)C3)C1 C1(CC(=O)NC)CN2CCC1CC2.C1CC(O)CN1C(C1CC1c1cc[nH]c1)=O c1(C(N)=O)c(C(=O)NC2CC3(C2)CN(C(C2CNC(=O)N2)=O)C3)cccc1F N1(CC=O)CC(=O)N(C)C1=O.C1(CC=C)CCN(C(=O)CC2CC=CCC2)C1 N1(C(C2C(C)C2)=O)CC2CCN(C(c3coc(S(N)(=O)=O)c3)=O)CC2C1 c1(OC)cn(C)c(C(=O)NCC(O)CN(C)C(C2Cc3nccn3C2)=O)cc1=O Cc1cncc(C(=O)Nc2cccc(NC(=O)Cc3ccc(C(C)=O)s3)c2)n1 Cc1nc(-c2cccc(Oc3ccccc3)c2)ccc1C(=O)N(CCCO)CCCO N1(C(CC)C)C(=O)NC(c2ccc(C#N)nc2)C2=C1COC2=O C1(C(=O)NCC2(O)CCOC2C)(CC)CCCN(C(c2cc(Cl)no2)=O)C1 c1(C(N(CC(CC)NC(=O)CC2CC(=O)C2)C)=O)nc(CC2CC2)no1 CCC(C(=O)NC(CC1CCC1)C(=O)NC(c1ncc[nH]1)CC)OC C12(C(=O)NCC)CCCC1N(C(C13CC1CNC3=O)=O)CC2.CCC1CC1.O c1(C(C(N2C(CNC(COC)=O)CC2)=O)C)ccc(S(N)(=O)=O)cc1 c1(C(=O)NC(CCCCNC(C(COC)OC)=O)C)c(F)cc(F)cc1F c1(C(=O)NCC2CCC(NC(C(CC#C)(C)C)=O)C2)ccc(C)c2c1NCCC2 C1(CCN(C(CC2CC2)=O)C)CCN(C(=O)C=Cc2cn(C)nn2)CC1.CC C1(NC(c2cncc(N3CCCC3)n2)=O)CCCN(C(=O)C2=COCCO2)CCC1 CN1CCC(N(C(=O)CCC2CCN(C(=O)CCOCC(F)F)C2)C)C1 C1(C(C)C)CCN(C(=O)CCC(N)=O)C(CNC(=O)C=CSc2nc[nH]n2)C1 N1(c2c(C)cnc(C)n2)CC2C3CCC(C2C1)N(C(C1CCC(=O)N1C)=O)C3 N1(C(c2c(F)ncc(C)c2)=O)CCCC2(NC(=O)CSC(C)(C)C)CCCC12 N1(C(C(C)CO)=O)C(CC(=O)NC2COC(C(F)F)C2)C2CCCC12 Cc1cc(C(=O)NC2CN(Cc3cc(C)cnc3Cl)CC2(F)F)cc(C)c1 c1(OC)cc(C(=O)NCC2CCN(C(c3ncccn3)=O)C2)n(C)n1 N1(C(CN(CCOC)C(C2CCC(C)(O)CC2)=O)=O)CC(C)C12CCOCC2 C=Cc1cncc(C(N2CCN(C(=O)C=Cc3cccc(Br)c3)C3CC23)=O)c1 c1(C(=O)NC2(C3N(C(C(c4cnccn4)C)=O)CCC3)CC2)cnc2[nH]nnc2c1 Cc1ccc(C=CC(N2CCOCC2CCNC(C2CSCCS2)=O)=O)s1 c1(C(=O)NCCOCCCNC(c2c(C)n[nH]c2)=O)ccc(CO)nc1 C1(CC(N2C(CNC(C(C)CN(C)C)=O)C=CC2)=O)CCCCCC1 N1(CC)CCCCC1C(=O)NC1CC(=O)CO1 N1(C(=O)NCC(=C)C)CCc2cccnc21 c1(C(N2CC(C(C)NC(C(CC=C)C)=O)C2)=O)cc2c(C)nn(C)c2nc1C C1(NC(c2nnn(CC)c2C)=O)CCN(C(=O)C(C)NC(=O)OC)CC1(C)C C1CCC(C)CN1C(=O)CC1(N(C)C)CCCC1.c1(SC)ncc(C(=O)N)s1 CC(C)CC(CNC(=O)C=Cc1nccs1)NC(C12CC(C1)C(C)O2)=O c1(C(N2CC(CNC(C3CN(CC)C(=O)C3)=O)C2)=O)cc(Br)ccc1O N#CC1CCCC(C(=O)NCC(O)CC(=O)NC2(CCF)CCC2)C1 N1(C(CC2C(=O)NC(=N)S2)=O)CCOCC(NC(=O)CCCC2CCCO2)C1 C1(CC(N2CCN(CC(c3ccccc3Cl)=O)CC2)=O)CSC2CCCC12 c1(CSC)ccc(NC(C2CCCN(C(=O)Cn3nnc(C)n3)C2)=O)cn1 CCC(C)CCC(=O)NCC(COC)NC(C1CCN(CC(F)F)CC1)=O c1(C(N2CCC(C)(NC(=O)CC3=CCCC3)C2)=O)cc2cncn2c(O)n1 c1(C=O)cnc2sc(C)cn12.Cc1cnn(C(C)C)c1C(=O)NCCO.CC CC1=NOC2(CCC2)C1.C(C(=O)N(CC(=O)N)CC)=CCN(CC)CC Cn1cc(C(=O)NC2CC(CNC(=O)Cc3nncs3)C2)c(=N)[nH]1 c1(C(N(CC(C)NC(c2c(OC)n(C)nc2C)=O)C)=O)ccnc2cc[nH]c12 c1(C(=O)NCC(CC)NC(=O)C(CN(C)C)N(C)C)nc(=O)n(C)[nH]1 C1(NC(=O)CN2CC3CC3C2)CCN(C(C2CC2(F)Cl)=O)CC1 C1(CNC(COCCC)=O)CCC12CCN(C(C1CC1C(=O)OC)=O)CC2 c1(NC(=O)CC2(NC(=O)CN3CCOC3=O)CCC2)ncc(Br)cc1F c1(C(=O)NC(c2ccc(C)cc2)CNC(C(CCC)C)=O)cc2ccsc2n1C c1(C(=O)NC2C(CNC(C(C(C)C)NC=O)=O)CCC2)cccc2c1COC2 C1(CN=C(NC(c2cccs2)C)NCc2cnco2)CCc2c(nnn2C)C1 C1(F)(CNC(C(C)SC(F)(F)F)=O)CN(C(C2CC2c2cncs2)=O)C1 c1(C(=O)NC(C2CCN(C(C3CC3C#N)=O)C2)(C)C)ncccc1S(C)(=O)=O CS(=O)(=O)c1ccc(C(=O)NCCC2CN(C(=O)CN3CCSCC3)CCO2)[nH]1 Cc1cc(CC(=O)NCCC2(C(=O)NC(C)CS(C)=O)CC2)n[nH]1 c1(C(N2CCN(C(C3(C)CCSCC3)=O)CC2C2CC2)=O)ncc2ccccn12 C1(NC(C(Cc2ccccc2)OC)=O)CCCCC1NC(=O)CCc1cnoc1 c1(C(=O)NCC2CN(C(COC(CC)C)=O)C2)ccc(S(N)(=O)=O)s1.O c1(OC)ccc([N+](=O)[O-])c(=NCC2(C)CC2(C)C)[nH]1 N1(C(c2c(OC)cncn2)=O)CCC(NC(=O)C2=CCCC2)C(F)C1 c1(C(=O)NC2CCN(C(C(c3ccc(C)cc3)C)=O)CC2)ccnc(C)c1Cl N1(C(C2CC(O)(CC#C)C2)=O)CCC(NC(C2CCCOC2)=O)C(O)C1 c1(C(=O)NC(C(C)(C)NC(c2nc(C)oc2C)=O)C)ccc(C2CC2)cc1F C(=O)(Nn1ccnn1)C1N(C(C(=O)OCC)=O)CCCC1 CCC(C)CC(=O)C(=O)NC(C(N1CC(CO)C2(CC2)C1)=O)C1(O)CCC1 c1(SCCC(=O)NCC2CCCN2C(=O)C(Cl)=CCl)ccc(F)cc1 C=CCCCCCCC(=O)N1CCN(C(c2cnc(C)cc2C)=O)C2CCCC12 CN1N=CC(CC(=O)NCC(O)CCNC(c2ccnc(S)c2)=O)C1=O c1(CC)nc(NCc2cc(Cl)cc3c2OCC3)c(C#N)cc1C C1(C(C)NC2(CS(C)(=O)=O)CC(F)(F)C2)COc2ccc(Br)cc2C1 c1(CC=O)ccc2c(c1)OCO2.C12(C(=O)NC(CCC)C)CC(C1)C(C)(C)O2 C(=O)(CC(C(F)F)N(C=O)C)N1CC=CC(NC(CC=C)=O)C1.C(C)(C)C N1(C(CC(CNC(Cc2c(C)ncs2)=O)C)=O)CCCC2(C1)N=N2 C1(CC#C)(C(=O)NCC2CCN2C(=O)C(C)n2cnnn2)CCCC1 C(CC(CC)C(=O)N1CCC(F)CC1C(N1CCC12CC(C(F)F)C2)=O)=CC N1(C(C(C=C)(F)F)=O)CCCN(C(=O)CN2CC3CC3C2)C(C)C1 N1(C(CC=CC)=O)CCCC(C(=O)N(CC(O)CO)CCO)CC1 C(=O)(CN=S(C)(C)=O)N1CCN(CCN(C(C(C)OC2CCCCC2)=O)C)CC1 CC(C)(CCN=c1[nH]nco1)c1ccc(NC(c2cnn3c2CCCC3)=O)cc1 N1(c2nc(C(C)C)cc(C)n2)CCC2CCC(C1)N2C(c1cnnc(O)c1)=O c1(C(C)C)ccc(F)c(C(=O)NC23CC(C2)N(C(c2cc(F)ccc2Cl)=O)C3)c1 N1(C(C2C(OCC)C2)=O)CCCC(C2(NC(=O)C(O)CC(C)(C)C)CC2)C1 C1(C=O)CCN(S(C)(=O)=O)CC1.CC(O)CC.C1(C=O)(OCC)CCC1.N C12(C(N3CCC(NC(=O)C=Cc4cocn4)C3)=O)CC(CO)(C1)OC21CCC1 c1(C(N2CCC(C(N)=O)C2)C(=O)NC(CC)C)ccc2cccc(Br)c2n1 N1(C(C2(C(C)C)CCN(C(C(COCC)C)=O)C2)=O)CC2OCCOC2C1 C1(OC)CN(C(=O)CCc2cn[nH]c2)CC1NC(=O)C(C)C1CCC1 CC1(C(N2CCC(NC(=O)CSCC(F)(F)F)CC2)=O)CNC(=O)C1 c1(OC)cc(C(N2CCC3CCC(C2)N3C(=O)CC(C)F)=O)c2cnccc2c1 c1(CC)cnc(Cl)nc1N1CC2CC(NC(=O)CC3(OC)CC3)C2C1 C1(CC(=O)NCC(C)N(C(=O)C)C)CCC(=O)NC1=O.c1(C=O)ccco1 N1(C2(CNC(C(CC)O)=O)CCCC2)CCN(C(=O)C=CBr)CC1 Cc1cc(CCCC(=O)N(C(C)CNC(=O)C(c2cccc(Cl)c2)C)C)c(C)s1 C(=O)(CCCCF)NCC1N(C(C(C)(C)c2cncnc2)=O)CC1 Cc1cc(CC(=O)NCC(F)CNC(=O)C2=CCCCC2)ccc1F c1(OC)cccc2c1CC(c1nc(CCC(F)(F)F)nn1-c1ccc(Cl)nc1)CO2 C1(NC(CC(C)N(C)C)=O)CC(CNC(C2CCC(CO)CC2)=O)C(O)C1 N1(C(c2c(C(C)(C)C)n[nH]c2)=O)CCCC(CO)(NC(c2cncc(Cl)c2)=O)C1 Cc1cc(S(=O)(=O)NC(C)(C)C2CC2)sc1Cl C(C)(O)(CCN=C(NC1CCCC1)N1CN(C)C(=O)C1C)c1ccc(C)cc1 c1(C(C)C)c[nH]nc1C(=O)NC(C)CC1CN(C(c2ccnn2CCF)=O)C1 C1(NC(c2ccc(C)o2)=O)C2CC3CN(C(C4CCCCC(=O)N4)=O)C1C3C2 C1(CCNC(CCOCCN(C)C)=O)CCN(C)CC1.C12(CCCC1)C(=O)N2 c1(OC)ccc(C)c(C(=O)NC(C)C(CO)NC(C2CCC(C)(C)C2)=O)n1 N1(C(c2ccc(OC)o2)=O)CC2CC1CN2C(C1(Br)CC12CCC2)=O C(C(CC(=O)N1CC(NC(C2CCC(N(C)C)CC2)=O)C1)CC(C)C)NC(C)=O N1(C(CCN(CC)CC)=O)CC(NC(=O)C(C(C)C)O)CC(F)C1.CC(C)C C(=O)(CCCN(C)N=O)NCC1(C)OCCN(C(C(C2CCC2)OCC)=O)C1 c1(C(=O)NCCC(CNC(C(C(C)(C)C)SC)=O)O)nnc2n1CCCCC2 C(CCCCCO)NC(c1n(CCCOC)nnn1)c1ccn(C2CCCC2)n1 N1(C(CCC)=O)CCC2CN(C(c3cc(OC)ccc3Br)=O)CCC2C1 CC1CCN(C(c2cnc(N)cn2)=O)CCN1C(c1cc(Cl)c([N+](=O)[O-])[nH]1)=O c1(C(=O)NC2C3CC(NC(C(C4CCOC4)OC)=O)CC32)ccc2ncnn2n1 c1(OC)ncc(F)cc1C(=O)NCC1CN(C(c2cccc(CF)c2)=O)CC1O c1(C2(NC(=O)NCC3C(CC(C)C)C3)CC2)ncccc1F C1(NC(c2scc(C(N)=O)c2)=O)CC2CN(C(C3(O)CC3)=O)CC2C1 c1(C(N2C(CNC(CCSCCC)=O)CCCC2)=O)cccn2nccc12 CC(C)CC(CNC(C1(P(C)(C)=O)CC1)=O)NC(C1(C)CC=CCC1)=O C1CC(O)CN1C(=O)Cn1cccn1.c1(C(=O)OC)ncc(C(=O)N)s1.C CC(CCC(C)(C)C)C(=O)N1CC2CC(C(=O)N(C)CC3CCSC3)(C2)C1 C(=O)(C1=NNC(=O)CC1)N1CCC(C)(n2cc(-c3ccc(CC)s3)nn2)C1 N1(C(C2CCC(CC)CC2)=O)CCC(N=c2[nH]nc(C(F)F)s2)C(F)(F)CC1 C(C)(C(CC(=O)N(C)CCNC(C)=O)NC(C1CC2CCCC2C1)=O)OC C(=O)(C(CCC)OC)N(CC=CC(=O)N(CC(CCC)C)C)C CC(=O)CCCCC(=O)N1CCCC(C)(C(=O)NC2CCSC2)C1 N1(C(c2c(C)con2)=O)CC2CCC(C1CO)N2C(c1cn2ccsc2n1)=O C1(O)(c2cn(C3CCN(C(C(N4CCC(C)(CC)C4)=O)=O)C3)nn2)CCOCC1 CN1CCCC(NC(C2CCC3(CC3)N2C(=O)C(C)(C)C(N)=O)=O)C1=O N1(C(CC2(C#N)CCCCC2)=O)CCC(NC(C2COCCO2)=O)C(CO)CC1 N1(C(C2N(C(C3C(C)=CCS3)=O)CSC2)=O)CCC(O)C(CO)C1 C12(NC(c3nccc(C)n3)=O)CCCC1N(C(=O)CC1CCC3(CCC3)O1)CC2 Cc1n[nH]c(C)c1SCC(=O)N.c1(CCC(N2CC(CC)C2)=O)ccc(F)nc1 CC1COc2ccc(C(=O)NCCC(C)N(C)C(C3CN4CCN3CC4)=O)cc21 C(=O)(CCC(=O)NC(C1CN(C(=O)Cc2cc(CC)no2)CCO1)C)OCC CC1CN(C(c2csc(-c3cccnc3)n2)=O)CCN1C(C1(CO)CCC1)=O Cc1ccc(C(=O)NC2CCCC2NC(=O)C(O)C(F)F)cc1-c1cnn(C)c1 c1(C(=O)NC2CCC(N(C)C(c3ccc4c(c3)CC4)=O)C2)cc2ccsc2n1C c1(C(=O)NC(CC2CN(C(CN(C(C)=O)C)=O)C2)C)cc(Br)nn1C CC1CCCN1C(=O)NCc1nc(C(=O)N(C)C)no1 c1(C=O)ncccc1Cl.C(C(C)C1CC1)NC(C1(C(=O)OCC)CC1)=O c1(OC)ncc(-c2cn(CCNC(=O)CC3CCN(C)C3)nn2)cc1C N1(C(COC)=O)CC(C)(C)C1Cn1cc(CN2CCC(N(C)C)C2)nn1 n1(C(C(=O)NCCN(C(C(CC)NC(C)=O)=O)C)C)cnc2c(N)ncnc12 CC(C)C(O)C(C)C(=O)NC1CCCC1NC(=O)CCc1c(F)cccc1Cl CCC(C)C(O)C(=O)NC1CC(C)(NC(=O)CN2CCCC(CC)C2)C1 C1(C(C)NC(c2ccc(CN=[N+]=[N-])o2)=O)CCCN(C(c2cncc(F)n2)=O)C1 C#Cc1cn(C)nc1C(=O)NCCN(C(=O)CC)C.c1(CC=O)ccccc1 N1(C(CCCN(C)N=O)=O)CCC2CN(C(c3cccc(N)n3)=O)CCC2C1 C(C(C)(C)C(=O)NC)NC(C)=O.C12CC1CN(C(=O)CN1CCCCCC1)C2 Cc1nc(O)[nH]c1C(=O)NC(C1CCOC1)CNC(=O)Cc1cn[nH]c1 c1(OCC)ccc(-n2nc(CCC(C)(C)C)nc2Cn2ncnn2)cc1 C1C2CN(C(=O)CC3CCC(C)(C)O3)CC12.c1(CCC(=O)NC)c[nH]c(=N)[nH]1 C#CC1(C(=O)N(C)Cc2ccsc2)CCN(C(=O)CC2CC(=O)NC2=O)C1 CC(CC(=O)NC1CC(CCNC(=O)C(C)(C)C2CC2)C1)C(F)(F)F CC(C)(C)CC(=O)NCC(=O)NC1CC1C.N1(CCC(=O)N)CCCCC1 C(=O)(C#CC1(C)CCCO1)NC1(C(=O)NCC(F)C2CCC2)C(C)CCC1 c1(C(=O)N)cc2cc[nH]c(=O)c2s1.C(=O)(C=CC(C)C)N(C(C)C)CC CCC(CCC(=O)NCC(C)S(C)(=O)=O)NC(c1ccc(C(F)F)o1)=O c1(C(N)=O)cc(=NCC2CC(NC(C34CCC(F)(CC3)CC4)=O)C2)[nH]c(Cl)n1 c1(CNC(C2CCN(CC(C)C)C2)=O)ccccc1.C(=O)C(F)=C(C)C.C c1(C(=O)NC2CN(C(CN(C(C)C)C)=O)CC2O)nccc2ccsc12 CC(c1cnn(C)c1)=CC(N1CCOCC1CN(C(=O)CC1CCN(C)C1)C)=O c1(C(=O)NC(C)CCCNC(C2CC(O)C2)=O)ncnc(O)c1Cl C1(C)(CNC(CC(CC)C2CC2)=O)CN(C(c2nnc(C)cc2O)=O)CCO1 C(CNC(C1(C)CCOCC1)=O)(CC(C)C)NC(C1CC(=C)C1)=O.C1CC1 c1(C(N2CC(CNC(c3scc(COC)c3)=O)C2)=O)cccc(F)c1.C C=CCCCCN=C(NCC1CCCCC1)N1CCCC(CSC)C1 c1(CN2C(C(N3CCc4ccsc4C3)=O)CC(O)C2)cccc(F)c1Br N1(C(CCOCC#C)=O)CC(CCNC(=O)C(=Cc2cn[nH]c2)C)OC(C)C1 c1(OCC)ccccc1CCC(N1CC(N(C(=O)CCCCOC)C)C(O)C1)=O C1(C(N2C(C)CN(C(=O)CC(C)(C)C#N)CC2)=O)CCc2cc(F)ccc2O1 C1(CC=C)(NC(=O)C(C)C)CCCN(C(=O)CCC)C1.C(C)=O.C(N)=O.O C1(O)CN(C(C=CC)=O)C1.C1(CC=O)C2CCC12.CC(C)(C)OC=O c1(C(N2C(CNC(c3cccc(=O)n3O)=O)CC2)=O)cc2ccccc2cn1 C(N=c1cc(C(F)F)nc[nH]1)C1CN(C(c2ccc(C)o2)=O)CC1(C)C N1(C(C(F)=CCC)=O)CCC(C)C(CNC(c2cc(SC)ccc2O)=O)C1 C1(O)(CCC)CCN(C(C2CSCN2C(C2CC2(F)Cl)=O)=O)CC1 Cc1cccc(-c2cn(C3CC(C(=O)N(C)Cc4cnc(OC)cn4)C3)nn2)c1 c1(C(=O)NCC(C=C)O)nc(CNC(c2cncn2C(C)C)=O)oc1C C1(NC(C#CC(C)(C)C)=O)CCC2(CCN(C(=O)Cn3nnc(=N)[nH]3)C2)C1 c1(N2Cc3c(C)csc3CC2)nc2cccnc2c(=NCC(C(F)(F)F)C2CC2)[nH]1 C1(OC)CCC(c2cn(CCN(C(=O)CCC(N)=O)C3CCCC3)nn2)CC1 N1(C(C(CC(C)C)OC)=O)CC2(CCC2)CC1CNC(C1CCC(=O)N1)=O C(C(C(=O)NC(C)C(C)F)C(C)C)NC(c1c(C)csn1)=O Nc1cc(C(=O)NCC2(C)CC2)nc(O)c1.c1(C=O)c[nH]nc1.CC(F)F C1CN(C(c2cc(C)c(C)[nH]2)=O)CC(C)(C)C1.N1(CC)CCC1C(=O)NC n1(C(C)C)cc(CNC(C2CCN2C(C2C3COCC23)=O)=O)nn1 N1(C(c2c(CC)c[nH]n2)=O)CCN(C(=O)CN2CC=CC2)CC1C1CCC1 Cc1nc(NCc2cccs2)cc(=NC(C)c2cc(Cl)ccc2Cl)[nH]1 N1(C(C(C2CC2)OCC)=O)CCN(C(c2occc2CC)=O)CC(C)(C)C1 CS(=O)c1ccc(C(N2CCOCC2CCNC(=O)Cn2cc[n+](C)c2)=O)cc1 N1(c2ccnc(C(C)(C)C)n2)CCCC2(CCCN(C(C3(O)CC3)=O)C2)C1 CC1(CNCC(O)CC2CCCCC2)CCCCCCC1 c1(C(=O)N)ccnc2ccccc12.CC(CCO)NC(=O)CC(=O)NCC1CC1 c1(C(C(=O)NCC(CN(C)C(c2ccc(=O)oc2)=O)O)(F)F)cccc(F)n1 C1(CNC(=O)Cc2ccon2)CC2CCC1N2C(c1nn[nH]c1Cl)=O N#Cc1ncccc1NC(=O)C(N1CCCC(OCC2CCOCC2)C1)=O CC1(CNC(C2(F)CC=CC2)=O)COCCN(C(C2(O)CCCCCC2)=O)C1 CCC(C(=O)NCC(C(C)(C)C)NC(c1cc(Cl)cc(C)c1C)=O)C(F)(F)F C1(NC(C(C)N2CCC2)=O)CCC(NC(c2cn(CC(N)=O)nn2)=O)C1 C1(C(CNC(c2cc(C)sc2)=O)(C)C)CCCCN1C(C1(n2cncn2)CC1)=O CCS(=O)(=O)CC(=O)NC1CC(C)CN(C(C2(COC)CCCCC2)=O)C1 C1(CNC(c2csc(-c3ccccn3)n2)=O)CCN(C(=O)CCCc2cccs2)C1 C(=O)(C#Cc1ccccc1)N1CC(CC#N)N(Cc2cncc(Br)c2)CC1 C1(NC(C2(CC#C)CC2)=O)CCCC12CCC2.C(=O)C(C)(C)C1CCCC1.C Cn1nc(O)cc1C(N1CCC1)=O.c1(C2(C(=O)N)CC2)ccccc1.C(N)=O C(=O)C1CCCc2ncnn21.C1(CSCC(=O)N(C(C)C2CC2)C)CCCO1 c12ccccc1C(=O)OC2.N1(CCNC(=O)OC(C)(C)C)CCNC1=O C1(CC(N2CC(CC=C)(NC(c3nc(=N)cc[nH]3)=O)C2)=O)Cc2ccccc2N1 Cc1ccc2occ(CC(=O)NCC(O)CN(C(=O)C(C)CS(C)(=O)=O)C)c2c1 C(=O)(CC(C)C(=O)N(C)CC1CCCC1)OC.c1(C=O)sccc1C(F)F.N c1(C(=O)NCC2CCN2C(c2cccc(O)n2)=O)cc(F)ccc1C1CC1 CC1CN(C(C2(CF)CC2)=O)CC1(C)CNC(=O)Cc1csnn1 CC1CCC(C(=O)Nc2n(CC3CC3)ncc2)N1C(c1ccc(Br)cn1)=O O=C1CCCC(C(=O)NCCC2CCCCN2C(=O)Cc2ccsc2)C1 c1(CC(N2C(CNc3nc(SC)c(Br)cn3)COCC2)=O)cc(Br)c(C)cc1C c1(C(N(CCC(C)NC(=O)C=CC2CC2)C)=O)ccc(OC(F)F)cc1 CC1CC=C(C(=O)NCC(O)CNC(c2cc(N)c(Cl)c(O)n2)=O)CC1 C(CC(C)(C)CC(=O)N1CCC2C(NC(=O)CS(N)(=O)=O)C12)OC C1(C=O)C2CCC(C2)C1(C)C.n1(CC(=O)N(CCC)CC)nnc(=N)[nH]1.N C1(CC)CCOCC1(c1nnnn1C1CC1)NCCOc1cc(F)cc(Br)c1 N1(c2c(Br)cnc(C(C)C)n2)CC2(C1)SCCC2NC(c1cnn(C)c1)=O CCCS(=O)(=O)CC(=O)N1CC(COC)CC1CNC(C1C=CCCC1)=O N1(C(COC(C)C)=O)CCC2(CCC2)C(C)C1.C(=O)(C(C(C)C)n1ccnc1)N c1(C(N2C(CNC(c3ccc(C(C)F)cc3)=O)COCC2)=O)ccc(C#N)n1C C1(NC(C2C(C)(C)C2)=O)CC2CN(c3nnc(C(F)(F)F)s3)CC2C1 c1(C(N2C3CCN(C(CNC(=O)OC)=O)C(C3)C2)=O)cnn2cc[nH]c(=O)c12 C1(NC(COCC(N2CCCC2)C)=O)COC2CN(C(C3(C#N)CC3)=O)CC12 C1CN(C(=O)C(C)CS(C)(=O)=O)CCC1(C)C.c1(CC)cc(C)c(C(=O)N)o1 C1(C(N(CC(C)C)CC(=O)NCCN2CCOCC2)=O)CCCCC(=O)C1 CCC(CCOC)C(=O)NCC1C=CCN1C(=O)CCCN=[N+]=[N-] c1(C(=O)NCCC(CNC(COC(CC)C)=O)O)cc(Cl)c(N)cc1F c1(OC)ccn2c(C(N3CC(NC(=O)C(C)(C)CC#N)CC(O)C3)=O)cnc2c1 c1(OC)cc(C(N2CCCCC2CN(C(=O)Cc2ncc(C)s2)C)=O)cnc1O Cc1ncc(C(N2CC(C(C)NC(=O)C(C)CC(N)=O)C2)=O)c(C)n1 c1(C(N2CCN(C(c3c(C)scc3)=O)CC2C(C)C)=O)ncccc1N=[N+]=[N-] CC1CN(C(=O)CN(C)CCO)CCN1C(=O)C(C1CCCCC1)F CC1CCN(c2ccnc(N(C)CC3CCCOC3)n2)CCS1 N1(C(C(C(=C)Cl)(C)C)=O)CCC2(CCCC2NC(=O)CC)C1.C1(C=O)CCC1 C(CNC(c1ccnn1C(C)C)=O)(CC(C)C)NC(C1(OC)CCCC1)=O Cc1[nH]nc(C(N2CC(C3CN(C(C4CC(N(C)C)C4)=O)CCO3)C2)=O)c1C N1(C(CC(CCC)OC)=O)CC2CCC(C1)N2C(=O)C(C1CC1)OC C1(O)(C(C)NC(C=CC(C)=O)=O)CN(C(C2CC(n3cnnc3)C2)=O)C1 c1(C(=O)NC2CN(C(C3CC(C(=O)OC)C3)=O)C(C)C2)nnn2c1COCC2 N1(C(C(=O)NC(C(C)C)c2ccco2)=O)CCn2c(C3CCNCC3)nnc2C1 CCCC(C)CC(=O)N1CCCC1(C)CNC(=O)CCCc1ccc(C#N)cc1 c1(C=O)c(C)nn(C)c1Cl.c1(CCCC)nc(C(=O)NCC2CCCC2)cs1.N C1(OC(C2C(c3c(C)c(Br)ccc3)C2)=O)C2CCOC2C12CCCC2 C1(C(N2CC(C#C)(F)C2)=O)CN(C(=O)C(C)(C)CCOC)CC1(F)F N1(CC=CC(C)(C)NC(=O)CSCCC#N)CCCC(N=[N+]=[N-])C1 N1(C(C2(CC)CCN(C(C(COC(C)=O)C)=O)CC2)=O)CCC(C)C(C)(C)C1 C1(CNC(CC(CC)C)=O)C(C2CC2)CCN1C(=O)Cc1ccc(F)c(OC)c1 C1CCC2(CN(C(C3CCC3(F)F)=O)C2)O1.Cc1ccc(=O)n(CC(=O)NC)n1 c1(C(=O)NCC2N(C(C3(NC(C)=O)CCC3)=O)CCC2)cc(Cl)ccc1N C(CCN=c1[nH]c(Cl)ncc1C(F)(F)F)OCCNC(Cn1nc(C)oc1=O)=O CCCC(CC(=O)NCCCc1ccncc1)NC(=O)C(C)CC#N CCC(CC)(CC)C(=O)NCC(O)CCNC(c1cc(C(C)C)sn1)=O N1(C(C(C)OCC)=O)CCN(C(C2CCC(CC)CC2)=O)C2CCC12 c1(C2N(CC3(C)ON=C(C)C3)CCOC2)cc(Cl)c(F)c(Cl)c1 Cc1ccc(CCC(=O)NC2CS(=O)(=O)CC2NC(c2cnsn2)=O)cc1Cl Cc1cc(=NCCC2CCCC2O)[nH]c(N2CCC(NC(=O)OC(C)(C)C)C2)n1 c1(C(=O)NC2CC(C)N(Cc3ccccc3)C2)cc(F)cnc1Cl c1(-c2c(CN(C3CCC(O)CC3)CCO)cccn2)ccc2ccoc2c1 Cc1c(C(=O)NCCN(CC(C)O)C(c2cscn2)=O)sc2cccc(F)c12 c1(C(=O)NC2CCCN(S(C)(=O)=O)C2)ccc2ncnc(O)c2c1 C(CC(C)(C)C)(C(=O)N1CCC(NC(c2c(Cl)ccc(F)c2F)=O)C1)OC c1(C(=O)NCC2(C)CCCN2C(=O)C#CC2CCCO2)cncc2cnccc12 Cc1cc(C(N2CCC2Cn2cc(-c3cscn3)nn2)=O)nn1-c1ccccc1 C1(NC(C=CCCC)=O)CC2CCC1N(C(c1cc(OC)c(OC)cc1F)=O)C2 Cc1ncnc(C(=O)NC2CS(=O)(=O)CC2NC(=O)C)c1C.c1cn[nH]c1.O Cc1cc(F)cc(Cl)c1CN1CCC(F)(Cc2ccccc2)CC1 Cc1[nH]c(-c2ccco2)nc(=S)c1NC(=O)CP(C)(C)=O Cc1onc(-c2cccc(Cl)c2)c1C(=O)NC1CC1NC(=O)C.C1CCOC1 O=C1NCC(C(=O)NCC=CC(N2CCC(N3CC=CC3)C2)=O)N1 c1(CNC(CC(c2ccc(F)cc2)N)=O)cc(-c2ccncc2)ccc1F N1(C(COC)=O)CC(NC(C2(C)CCCO2)=O)CC(F)C1 N1(C(CC(=C)C)=O)CCC2(CCCN(C(C3CC4(C3)CC(C#N)C4)=O)C2)C1 O=C(CCC[N+](=O)[O-])NCC1CCC(CNC(=O)C(c2ccc(Cl)cc2)O)CC1 CC12CC(C(N3CCCC3)=O)(C1)C(C)(C)O2.c1(CC(=O)N)ccc2nonc2c1 C1(C(=O)NCC2(C)CCN(C(C(C)OCC)=O)CC2)CCc2nn(C)cc2C1 C(=O)(C1=C(C)OCC1)N1C(C)(CNC(CC2CCCC(OC)C2)=O)CCC1 N1(C(c2c(C)cno2)=O)CC(NC(=O)Cn2cc[n+](C)c2)CC(C)(C)C1 Cc1c(F)cc(C(N2CC(NC(c3c(F)cncc3F)=O)C2)=O)cc1Br C=CC(C)(CCOC)C(=O)NC1CCC(NC(c2cscc2Cl)=O)CC1 C(C)(C)(C(=O)N(C1CC(C#N)C1)CC(=O)NCC(CC1CC1)CO)SC c1cccc(Br)c1.C(=O)(CC)N(C(C)C1CC1)C.C(C=O)=CC=CCC.N C(=O)(C1=CCCOCC1)N1CCC(NC(c2c(C)nc(C)s2)=O)C1C(C)C CC1(NC(C2(NC(=O)O)CCC(C)(C)C2)=O)COC(=O)OC1.C(C)(C)C C1(C(=O)NCC2(C(=O)NC3CCCC3O)CC(=C)C2)CC2COCC2C1 C(=O)(C(C)(C)CCOC)NCC(CC)(C)NC(=O)C(C)OC c1(C(=O)NC2C(NC(C=C3CCN(C)C3)=O)CC2)cc(N)ccc1Br c1(CCCC)nc(C)c(CC(N2CCC(O)C2)=O)s1.C1(CC(=O)N)CCC12CCC2 Cc1cccc(-c2nc(CC3CCC4(CCC4)O3)no2)c1F N1(C(Cc2c(CC)cccc2)=O)CC(OC)CC(NC(=O)C(F)(F)C(C)O)C1 N1(C(Cc2ccn(C)n2)=O)C2CCCC1CN(C(=O)C(C)(O)C(C)(C)C)C2 C1(N(C(c2cnc(OC)nc2)=O)C)CCN(C(=O)C(O)C(C)C)CC1C C(=O)(C1CCCc2nccn21)NCC1CCN(C(CC2CCC(C)(O)CC2)=O)C1 c1(C(N2CC3C(NC(c4c(Cl)cn(CC)n4)=O)(C3)C2)=O)c[nH]c(=N)nc1C N1(C(C2CCCN(C(C3CC(=C)C3)=O)C2C)=O)CCC2(CCCCC2)C1 N1(C(CC(CNC(=O)C(C)(C)C)OC)=O)CCC2(CC1)N=N2 N1(C(Cc2c(C)ncs2)=O)CCCC12CCN(C(C1CC1F)=O)C2 CCCCC(O)C(C)C(=O)NCC1(CC(=O)NCCCN(C)C(C)C)CC1 Cc1cc(C(c2nnnn2Cc2cccs2)NCC(C)Oc2ccccc2)sn1 C1(CNC(c2ccc(CC)s2)=O)CN(C(=O)C(CC)C2CCOCC2)CC1C Cc1cc(C(N)=O)cc(C(=O)NCC2CCN(C(=O)CCn3cccc3)CC2)c1 C1(C(=O)NC2CCN(C(CCCC(=C)C)=O)C23CC3)CCCC2(CCCCC2)C1 N1(c2ncc(C#N)nc2)CC(NC(=O)C2=CCS(=O)(=O)C2)C2CCCCC12 C(=O)(CCC(CF)CF)N1C(CCNC(c2c(C)c(N)ccc2)=O)C(C)CCC1 n1(CC(N2C(NC(C3C(CC(C)(C)C)C3)=O)CC2)=O)nnc(C2CC2)n1 N1(C(c2nn(C)c(CO)c2)=O)CCC2(CC1)CCN(Cc1ncccc1Cl)CC2 N1(C(CN(C)CC)=O)CCCC(NC(C2(Cc3cccc(F)c3)CCC2)=O)C1 N1(C(c2[nH]cc(C)c2)=O)CC2(CNC(=O)C(C)C(C)C)CCC1CC2 c1(C(N2CC(C)CC(NC(C(CC=C)C)=O)C2)=O)cc(Cl)c(F)c(Cl)c1 C1(C)(C(=O)NC(C2CCCN2C(=O)CCc2nccn2C)C)CCC(=O)NC1 C1(NC(c2cccc(CCC)c2)=O)CCCC12CN(C(C1(C(=O)N)CC1)=O)C2 Cc1nc(C(=O)NC2COCCC2)c(C)o1.c1(C(=O)N)ccnn1C1CC1(F)F C1(C(=O)NCc2snnc2C)(COC)CN(C(C2CCCCO2)=O)C1 Cc1nonc1CC(=O)NC1CCC1NC(c1conc1C1(C)COC1)=O N1(C(CCN(CCCO)C(c2c(CC)occ2)=O)=O)CC(O)CC12CCOC2 CCS(=O)CC(=O)N1CCCC1(C)CNC(C1CC(NS(C)(=O)=O)C1)=O N1(C(C2(CC=C)CCOCC2)=O)CCC(C2CCN(C(=O)C=CSC)CC2)C1 C1(C(N2CCC(O)(CCNC(C=COCC)=O)C2)=O)CC2(C)CC1CO2 S(=O)(=O)(c1cccc(=NC2CCS(=O)(=O)C2)[nH]1)NCCCCCCC=C C(=O)(C(=O)C(C)(C)C)N1C(CC(=O)Nc2cnn(CC)c2C)CCC1 C1(O)(CCNC(C2CCN(C)C2)=O)CCCN(C(=O)C(F)(F)c2nccn2C)C1 c1(CCC)ccc(C(=O)NCCC2CCC(NC(c3cc(CC)sn3)=O)C2)[nH]1 CN1C(=O)CCC1(C)CNC(=O)Cn1cc(-c2cccc(C#N)n2)nn1 C1(NC(c2cnn(C(C)(C)C)c2N)=O)CC2CCC1C(NC(=O)C)C2.CCF.O N1(C(c2cc(CC)no2)=O)CC(C(=O)NC)OC(C)C1.C1(N(C)C)CCCC1 c1(CC(=O)N(CC(C)NC(CCC(=C)C)=O)CC)cncc2ccccc12 c1(C(N2CCC(CCC(C)C)CC2)=O)c(Cl)sc(Cl)c1C.C(C=O)OC(C)=O.N Cc1csc(C(=O)NC2CC(CC(=O)N(CC(F)(F)CO)C)C2)c1 c1(CC)cc(C(N2CCOCC(NC(=O)CCn3ccnn3)C2)=O)cc(Cl)n1 C1(NC(C2C3COCC23)=O)CC2CN(C(c3cccc4occc34)=O)CC2C1 Cc1cc(C2=CCCCC2C)cnc1NC(=O)CC1CC1 CON1CC(C(=O)NC2(CCCNC(=O)COC3CCOCC3)CC2)CC1=O N(C1CCc2ccc(Cl)cc21)(c1ccc(Cl)nc1)CCC(C)C c1(OC)cc(Cl)c(C)cc1C(N1CCC(C)C1)=O.c1(C=O)ccc(F)c(C)c1.N Cc1cc(=NCC2(NC(C3CCCN(C(=O)C(C)C)C3)=O)CCOCC2)[nH]cn1 CCCC(CC)CCC(=O)NC1CN(C(=O)CCc2cnoc2)CC1OC N#Cc1cccc(F)c1-c1cc(C(=O)Nc2scnc2C(N)=O)cc2[nH]ncc12 CS(=O)c1ccccc1C(=O)NCC(CNC(=O)CNc1ccccn1)CO C1(NC(COCC(C)C)=O)CCCCN(C(=O)Cc2csc(C(C)C)n2)C1 c1(C(=O)NCC(C#C)OC)c[nH]nc1CNC(c1n[nH]c(O)n1)=O C12(C(N3CCCC(C)(C(N(CCC)CCO)=O)C3)=O)CCC(CC1)NC2=O c1(C(C)CC(=O)N2CC(C(C)NC(=O)CNc3ccccc3)C2)cccc(F)c1 N1(C(Cc2nc(C(C)(C)C)sc2)=O)CCC(C)C12CCC2.C(=O)C=O.C1CC1.N C#CCC(CC(F)F)C(=O)N(CC(C)NC(c1ccc(O)nc1C)=O)C C1CCCN(C(=O)Cc2ccc(F)cc2)C1.C1(CCNC=O)CC(F)(F)C1.N N1(C(C(C)N(C)C)=O)CC(F)(F)CC1(C)CNC(=O)CC1CC=CCN1C C1(C(N(C)CC)=O)CC2C=CC1CC2.C(=O)CCC.C(=O)C(C)(C)C.CC.O CC(C)(F)C(C)(F)C(=O)N1CC2CC1CN2C(C1CCC(n2cccc2)CC1)=O C(=O)(C(CNC(c1ccc(Cl)o1)=O)CC(C)C)N(C(C)C(=O)OC)CC c1(C(=O)OCC)cc(SCc2ccnc(NC)n2)nc(C)n1 C(c1cncc(C)c1)=CC(=O)NC12C(CN(C(C3N(C(C)=O)CCC3)=O)C1)C2 N1(C(CC(C)C)=O)CCC2(CCN(C(=O)C(C)CC(C)(C)C)C2)C1.[SH](C)(=O)=O.N C(=O)(CN=c1cc[nH]cc1)NCC1CCCN(C(C2(OC)CCC2)=O)C1 C1(C(=O)OCc2c(CC)nccc2)CCC2(CCCCC2)C1 c1(C(N(CCNC(c2cc(OC)ccc2F)=O)CC)=O)nn(C)cc1[N+](=O)[O-] C(=O)(C1=Cc2ccccc2C1O)N(CCOC)CCNC(c1ccoc1C)=O c1(CNC(=O)CC2CCCCN2C(=O)CC2CCCO2)c(F)cncc1Cl Cc1ccc(CC(CO)NC(=O)NC2CCC(C#N)C2)c(C)c1 Cc1nc2ccccn2c1C(N1CCCC(CNC(c2cnnn2C)=O)CC1)=O N1(C(Cn2nc(C)oc2=O)=O)CCC(CNC(=O)C)C(C)C1.C1(C)CCCC1 Cc1[nH]nc(C(N2CC3CC3(C(=O)N(CCC(O)CO)C)C2)=O)c1C O=S(=O)(c1[nH]c(=NC2CCCCC2CSC)ccc1Br)NCC(Cl)=CCl c1(CNc2c(OC)cc(Cl)cc2)cnc(O)c2ccccc12 c1(C(=O)NCC(CC)(C)NC(c2coc3c2CCCC3)=O)n[nH]c2ccccc12 C1(C(=O)NCC(C)SC)C(CNC(=O)C(n2ccnc2C)C)C1(C)C N#CC1CCCCC1CNC(=O)Nc1cc(C(F)(F)F)cc(Cl)c1 C1(N(C(=O)COC2CCOC2)C)CCN(C(C2(CO)CC2(F)F)=O)CC1 C(C(C)C(C)(C)C)(c1n(CCSC)nnn1)NCCc1ccc(Br)c(OC)c1 c1(OCC)ccc(CO)cc1F.c12ccc(cc1)CCN(C)CC2 N1(CC(N2CCC(OC(=O)NCC)C2)=O)CCN(C(c2ccsc2)=O)CC1 Nc1c(C(N2C3CCC2C(CNC(c2cccc(O)n2)=O)C3)=O)ccc(Cl)c1F c1(CC(=O)NCC2CC(CNC(c3cscc3F)=O)CO2)noc2ccccc12 C1(NC(CS(CC)(=O)=O)=O)CN(C(C2(n3ccnc3)CCCC2)=O)CC1C1CC1 C1(OC)CC(CF)N(C(=O)C(O)CNC(c2csnc2C)=O)C1 c1(C=O)cc(C(N)=O)ccc1C.C(C(C)CC(=O)NCC1CC1C)OC.N C1(OC)CN(C(c2cccc(N)n2)=O)CC1NC(C1CCC(C(N)=O)N1C)=O c1(C(N2C(CNC(C3C(CC)C3)=O)CCCC2)=O)ccc(C)c(Br)c1F c1(C(=O)NC2CC(C)N(C(c3cnc(N)c(Cl)c3)=O)C2)ncn2ccccc12 c1(SCC)ccc(NC(=O)Nc2cc(C)cnc2F)c(C)c1 Cc1cccc(OCC(=O)N(CC(C)CNC(c2ccc(C)nn2)=O)C)c1 c1(OC)ccc(CCC(=O)NC2CC(NC(c3cc(Cl)ncc3N)=O)C2)cc1O N1(C(C2CCC(CC)O2)=O)CCC(C(=O)NCC2CCC2C)CC1(C)C N1(C(C2(C#N)CCC2)=O)CCC2CCN(C(c3cn4cccc(F)c4n3)=O)C2C1 c1(C(N2CC(NC(COCC)=O)C3(C2)CC3)=O)cn(C)c(=O)c2cncn12 C(CCCC(C)NC(c1ccncn1)=O)NC(C=C(C)C(F)F)=O CCCC(C(=O)N1CCC(C)C1CNC(c1ccc(OC2CC2)cc1)=O)OC N1(C(=O)CC2CC3(CCCC3)CO2)CC2OCCN(C(=O)Cn3cnnn3)C2C1 N1(C(c2c(CC)ncs2)=O)CCC(CO)C(NC(=O)CC2CCN(C)C2=O)C1 C(C)(CO)(C(=O)NCC1CCC1)NC(CC1CC(OC)C1)=O.C1CC1.C C1(CCNC(CC2CC(C)C2)=O)COCCN1C(=O)CCCc1ccccc1 N1(C(CCC(C)OC)=O)C(C(=O)N(C)Cc2ccsc2)CCC12CC2 N1(C(CCC2C(C)=NOC2=O)=O)CCCCCC(NC(=O)C(C)(C)S(C)(=O)=O)C1 c1(C(N2CCCC(C)(NC(C3CC4CCC4C3)=O)C2)=O)cc2ccsc2c(O)n1 C1(CC=C)(NC(c2csc(Cl)c2)=O)CN(c2nnc(-c3ccccc3)o2)C1 O=C1CC(C(N2CCCCC2C(N2CC3(CSC3)C2)=O)=O)CCN1 C(c1cnn(C)c1C)=CC(N1CCC(N(CCC)C(c2ccsc2C)=O)C1)=O Cc1cc(CNc2cccnc2C(N2CC(C)C2)=O)ccc1Br c1(NC2(CCNC(C3N(C)C(=O)CC3)=O)CCC2)nc2ccc(F)cc2o1 N1(C(CCCCC)=O)CCN(C(=O)C(C)OCc2ccc(C)cc2)CC1CC C(=O)(C1=C(C)CCCC1)NC1(CC=C)CN(C(c2ccsn2)=O)C1 C1(CC=C)(NC(=O)Cc2ccc(OC(F)F)cc2)CCN(C(=O)CCF)CC1 N1(C(C2CN(C(COCCC=C)=O)CC2C)=O)CCN(C)CC1C1CC1 CCCCCCC(CC)CN(C)N(CCN1CCCCC1)C1CCN(C)C1 C=C(C)C(C)(C)C(=O)NCC1OCCC1C(=O)NCCNC(=O)CO c1(-c2ccc(C#N)cc2)c[nH]c2cc(C(=O)N(CCCO)CCCO)ccc12 c1(OCC)cc(C=O)ccn1.C1(C)CCN(C(=O)CC)C1.C1(C=O)CCC1.N c1(CC(N2CCC(N(C(c3ccnc(Br)c3)=O)CC)CC2)=O)ccc(C)cc1O N1(C(C2CC3CC2C3)C(=O)NCC(=C)C)Cc2ccccc2NC(=O)C1C O=C(C1=C2CCN=C2NC=C1)NC1CN(C(C2CN3CCCN2CC3)=O)C1 N1(C(c2cc(CSCC)on2)=O)CCC(F)CC1.C(=O)C1=CC(C)(C)C1.C C(C)(C)(C(=O)N(C)CCNC(c1cn(C(F)(F)CO)nn1)=O)SC C(CC(C)(C)C(=O)NC1CCOC(C2CCN(C(=O)C#CC(=O)NC)CC2)C1)OC C(CN=c1[nH]cnc(Cl)c1C)C1C(NC(Cn2nnc(C)n2)=O)CCC1 c1(CN2C(C)(C)CC(CO)C2)sc2ccccc2c1Cl C(=O)(C(COC)CC(C)C)N1CC(C(=O)NC(CCCC)CO)C(F)(F)C1 N1(C(C(N2CCOC2=O)C)=O)CC2(CCCC2)C1C(=O)N(C1CC2(CC2)C1)C N1(C(C(=O)NC2(C)CC2)CC2CC2(Cl)Cl)CCCC(c2nc[nH]n2)C1 C1(CC#C)(C(=O)NCC(Cl)C(C)(F)F)CCN(C(=O)Cc2csnn2)C1 N1(C(c2c(OCC)nccc2)=O)CCN(C(c2ccnn2C)=O)C2COCC12 C1(CNc2nnc(Cc3ccccc3)s2)CN2CCCCC2CO1 N1(C(C(C#N)CC2CC2)=O)Cc2[nH]nc(CNC(=O)Cc3cccs3)c2C1 c1(C(=O)NC2CC(n3cc(CC(CC)(C)O)nn3)C2)nc(Br)n(C)n1 C1(C(=O)NC2(COC)CCCC2)CC(C)CN(C(c2cnnn2C)=O)C1 C1(NC(c2c(C(C)C)nn(C)c2)=O)CC2CCC(C1C)N2c1ccnc(C#N)n1 C(=O)(CN=S(C)(C)=O)N(C(CC)CC(=O)Nc1cccc(NC2CC2)c1)C C1(C(N(C2CCC(NC(C3(C)CCCOC3)=O)CC2)C)=O)CCN(C)C(=O)C1 CC1CN(C(=O)Cc2ccc(C(c3ccco3)=O)nc2)C(C(F)(F)F)CO1 Cc1nn(C(C)(C)C)cc1C(=O)OCC(C1(S(N)(=O)=O)CC1)=O C(=O)(C(C#N)C(C)(C)C)NCC(CN(C(c1c(C)n(CCO)cc1)=O)C)O c1(CC)ccc(C=CC(=O)NCC=CC)cc1.C1(C=O)CCCC(F)C1.N c1(OCC(C)C)cccc(CN=C(NCC(C)(C)C)NC2CC2)c1 CC1(CNC(=O)CCCc2ccccc2)CCCN(C(=O)Cn2ncnn2)C1 Cc1oc(S(C)(=O)=O)cc1C(=O)NCCn1ccnn1.C(=O)C1=CCOC1.C N1(C(C2(S(C)(=O)=O)CC2)=O)CC2(CCC(NC(C3CCCSS3)=O)CC2)C1 C(=O)(CC1NC(=O)c2ccccc21)NCC1C(C)(C)N(C(C2CCCO2)=O)CC1 Cn1cc2c(n1)CCCC2C(=O)NC1CCN(C(=O)C(N)=O)CC1 C(=O)(CCC1=NNC(=O)CC1)N1C2CC(CC(NC(CCOC)=O)C2)C1 c1(OCC)cccc(NCC(C)(C)NC(C2CN(CC)CCO2)=O)c1[N+](=O)[O-] c1n[nH]c2c1CCC2.C(CC(=O)N)OCCCNC(CNC(=O)OCC)=O CC1CCN(C(=O)CC(C)C)C1C(=O)N(C)C.C1(C=O)CCCN1C(N)=O.N n1(CC)cnc(C(=O)NC(C)CNC(=O)C(C)CSC(F)(F)F)n1 CCCCCC(C)(C)C(=O)NC1CCCC1CC(=O)NCc1c[nH]nc1C1CC1 C(=O)(CC(O)CCCCC)NC(C(=O)NC(C#C)C1CCC1)CC1CCOCC1 CCC(C(=O)NCCSC)N(C(=O)C(N1CCC(C)C1)=O)C C(CCC)(C(O)C(=O)NCCCCCC1CC1)NC(C(CCC)NC(C)=O)=O c1(NC(C2CCCCC23CC3)=O)ccc(-n2cccn2)c(F)c1 C(C)(CNC(C1CC1(c1ccccc1)C)=O)(C(C)C)NC(c1c(C)cno1)=O c1(C(=O)NC2C(c3ccc(C)cc3)CCC2)ccn2nnnc2c1 c1(SC)nc(C)cc(=NCC(CC(C)C)NC(=O)C=Cc2ccc(C3CC3C)o2)[nH]1 N1(C(C23C(NC(C(C)=CC=C)=O)CC(CC2)C3)=O)CC2(CCC(=O)O2)C1 N1(C(Cc2c(C(C)C)con2)=O)CCC(O)C2(CCCNC2=O)C1 C(CN=c1ccc(Br)c(S(=O)(=O)NCCC(N2CCOCC2)C)[nH]1)SC(CC)C C1(C)(CNC(COCCC)=O)CCCC1.c1(CC=O)cccc(C2CC2)c1 c1(C(N(C(C(=O)NCc2scc(C)c2)C)C2CC2)=O)cncc(O)c1 c1(C(=O)NC2CC(C)CN(C(=O)CCP(C)(C)=O)C2)cc2cnccc2cc1F c1(C(=O)N)cc(C(F)F)cs1.C(O)(C(F)(F)F)C1(C=O)CCC1.C(C)CO c1(C(=O)NC2(CC)CCCN(C(C3OC(C)CC3C)=O)C2)ccc(F)c(F)c1F C(CNC(c1cc(F)cnc1O)=O)(CC(F)(F)F)NC(c1c(C)nn[nH]1)=O CC1(C(=O)NC(CNC(c2ccc(=N)[nH]c2Cl)=O)CO)CCc2ccccc21 N1(C(C2C(C(N)=O)C2)=O)CCC2(NC(c3cnsc3)=O)CCCCCC12 C(=O)(C(F)(F)C(C)O)N1CC(CCNC(C(C(C)C)OCC)=O)C1 C(N=c1cc(Cl)nc(C2CC2)[nH]1)C1CN(C(c2c(CC)scn2)=O)CC12COC2 c1(C(N2CC(CC)N(C(c3cn(C)[nH]c3=N)=O)CC2)=O)c2c(nn1C)CCCC2 C(CC(CC)C(=O)NCC1CCCN(C(C2CCCC(C#N)C2)=O)C1)=CC CNS(=O)(=O)NCC(=O)NCCCC1(NC(=O)CC(C)C2CCCO2)CC1 C1(CNC(C2CCC2C=O)=O)CC2(CCCCS2(=O)=O)C1.C(C=O)OC CC(CNC1CC(=Cc2ccccc2)C1)C(C)(C)C CC1=C(C)CC(C(=O)NC2C3CC(NC(=O)C(C)=C4CC4)CC23)CC1 c1(CNC(C2C(OC)(OC)CC2)=O)ccc(CCC)cc1.C(=O)C1=CCSC1 C1(CNC(C(=O)OCC)=O)CN(C(c2cc(COC)[nH]n2)=O)CCC1C C(=O)(C1c2c[nH]nc2CN1C(C12CC1CNC2=O)=O)NC(CC=C)CO Cc1ccncc1C(=O)NC(C1CCN(C(C2CC3CCC2C3)=O)CC1)(C)C N1(C(CC2C(C)CCN(C(C3CC(=C4CC4)C3)=O)C2)=O)CCC2(CCC(O)C2)C1 N1(C(Cc2ncc(C)o2)=O)CC(NC(c2ccncc2Cl)=O)CC2(CCC2)C1 CN=c1[nH]cc(C(=O)NCC2(F)CCCC2)s1.C(=O)CC(C)n1ccc(C)n1.N C1(NC(c2n(CC)ccc2)=O)CCN(C(c2cn(C)c(C)n2)=O)CC1CO C=C=CCC(=O)NC(Cc1cn[nH]c1)C(=O)NC(c1cnn(C)c1)CC CC(=O)CC(C)(C)C(=O)NCCn1cc(C(=O)NCC(C)(O)C(C)C)cn1 N1(C(CC2C(C)=NNC2=O)=O)CC2=C(C1)CN(C(=O)CCN1CCCC1=O)C2 Cc1[nH]c(Cl)nc(=NCCC2CCCN2C(=O)C2CSc3ccccc32)c1C#N C(=O)C1=CS(=O)CCC1.C(c1cccc(O)c1)=CC(N1CCC(CC=C)C1)=O.N c1(C(N2C(CCNC(C3CC(OC)C3)=O)CC(OC)C2)=O)cccn2cncc12 N1(C(C2(CC)CC2)=O)CCC2(CC1)CN(C(c1cccc(S(C)=O)c1)=O)CCO2 C=C=CC(C)C(=O)NCC1CCCN1C(=O)CCc1ccc(OC)nc1 CCC(CC(=O)NCCCCC1CN(C(c2cccc3oncc23)=O)C1)C(C)C c1(OC)nc(C(N2CC=CC2CNC(=O)C(C)SC)=O)cc(O)n1 C1(CC)CCC(C(=O)NCC(O)CNC(=O)CC2CNC(=O)C2)O1 CCC(C)(COC)C(=O)N1CCC1CNC(C1Cc2cscc2C1)=O C1(C(=O)NCCC(F)(F)F)C2CC3C(C2NC(C2CCCO2)=O)C13 C1(C(N2CCC(n3cc(C4(OC)COC4)nn3)C2)=O)(C=O)CCOC1.C1CC1.N N1(C(Cc2cc(OC)c(C)cc2)=O)Cc2nccn2CC(NC(C2(O)CC2)=O)C1 C=C(C)CCCC(=O)NC1CCCC(NC(C2(C)CCNC(=O)C2)=O)C1 c1(C(=O)NCC(C)N(C(C(CC)OCC)=O)CC)cc2c(C)cccc2[nH]1 CCC(CC)C(C(=O)N1CC(C)(C)CC1CC(=O)NC(c1nncs1)C)OC C1(C=O)CC2(CCCC2)CO1.CCC(C)CNC(=O)C=CCN1CCCC1.N C12(C(N3CCCCC3)=O)CC1COC21CCC1.C(C)(C)(C=CC(=O)N)SC.C C(CCC(=O)N)OC.c1(CC2CC2)ccc(C)cc1.C12(C=O)CC(C1)NC2=O N1(C(c2c(NC)snc2C)=O)CCOCC(C)C1.c1(C=O)cnc(C(C)C)s1.N c1(CN2C(C)C(N3CCOCC3)CC2)cc(Br)cc(Br)c1N C1(CNC(Cc2c(C)ncs2)=O)CN(C(=O)CC2CC2(C)C)CC1(C)C C(=O)(CCN=c1[nH]c(NCC2CC2C(C)C)nc2ccccc12)NC C1(C(N2CCCCC2)=O)CC(C)(C)SC(C)(C)C1.Cc1sc(O)nc1C(=O)N.C C1(CNC(c2c(OC)c(C)ncn2)=O)CCCCN(C(=O)Cc2cccs2)CC1 c1(-n2cc(CC(C)N(C(=O)CC3CSC3)C)nn2)ccc(C(=O)O)cc1 Cc1ccc(CCC(N2CCN(C(c3cc(Cl)c(Cl)cn3)=O)CC2)=O)c(C)n1 C(=O)(C1=CCCCO1)NCC(C(=O)NCC(C)C(F)F)(C)C CC1C(NC(c2cc3n(n2)CC(F)C3)=O)CC2CCC1N2C(C1CC1(C)Br)=O N1(C(C(=O)NCCCC)C(C)C2CCOCC2)CCS(=O)(=O)C2CCCC12 CN1CCN(C(=O)CC2(C#N)CC2)CC1CNC(=O)C(F)(F)c1nccs1 c1(CC)nc2c(C(N3CC4CC3C4NC(=O)C(C)(C)C(N)=O)=O)ccnc2[nH]1 Brc1ccnc(OC2CCN(CCn3cc(C4CCCNC4)nn3)C2)n1 C1(NC(C(C)OC)=O)CC2C1CCN2C(=O)CCCn1ccnc1C Cc1c(C(=O)NC(C)CN(C)C(c2c(N)cccc2Cl)=O)cccc1Cl N1(C(C)C)CC(C(N2CCC(C)CC2)=O)CC1=O.n1(CC(=O)N)cnc(C#N)n1 C1(C(=O)NCCSC(C(=O)N(C(CC)C)C)C)SCC=C1C C(=O)(C(F)CC(C)(C)NC(c1c[nH]nc1C)=O)NCC(=C)CC c1(CC(COC)SC)ccc(F)cc1.C12(CCCSC1)CNC(=O)O2 c1(C(=O)NCCn2cc(CNC(C3C(C)CC3)=O)nn2)cnn2c1CCCC2 c1cnc(Cl)c(C)c1.c1(C(CC(=O)N2CC(NC)C2)NC(C)=O)ccc(F)cc1 CC1=C(C(=O)N2CC(C)(C(=O)NCC3CCC(F)(F)C3)CC2(C)C)COCC1 CCC(CC(F)(F)F)C(=O)N1CC(COC)(NC(C2CCC(N=[N+]=[N-])C2)=O)C1 c1(-c2nnc(SC(C(=O)OC)C(C)CC)n2C)ccc2oc(CO)nc2c1 c1(C(C)=O)ccc(Cl)c(S(=O)(=O)N2CCSCC2C)c1.c12ccc(cc1)c(=O)[nH]2 c1(C(N2CCC3(NC(C)=O)C(CC2)C3)=O)cc(S(N)(=O)=O)oc1C C1(C(C)C)CCCN(C(C)C(=O)NOC(c2ccccc2)C2CC2)C1 N1(C(CC(C)SC)=O)CC2CCC(NC(c3cccn(CC(C)C)c3=O)=O)(C2)C1 C1(NC(CCN(CC=C)C(c2cc(C#N)ccc2N)=O)=O)CC2CC1CC21CC1 C(C(C(=O)N1CC(NC(N)=O)C1)C(C)(C)C)NC(c1nc(C)n(C)c1)=O C(CCC(C(=O)NCCC(F)(F)CO)NC(=O)C=CC1CC1)OC CCCCC(CC)C(=O)Nc1ccc(NC(=O)C(=O)N(C)C)cc1C c1(C(C(N2CC(O)(C(C)NC(CCC)=O)C2)=O)F)ccc(C(F)(F)F)cc1 c1(C(=O)N)n[nH]c(C)c1Br.C(C(C)(C)C)N(C(=O)C=C1CCOCC1)CC c1(CSC)csc(C(C(=O)NC(C)(C)C)N(CCCCCN(C)C)C)c1 c1(OC)cc(C)ccc1C(=O)NCCCCC(CO)NC(=O)C(C)(C)CF Nc1ncnc2c1ncn2CCC(=O)NCC1CCC(c2ccccc2)O1 c1(C(=O)NCC2(CC(=O)NC(CCC=C)C3CC3)CC2)ccc(O)nc1 CCC(CC)CC(F)C(=O)NC(C)C(=O)NC(C12CCC(CC1)C2)C C1(C(N(CC(=O)OC)C)=O)CCN(C(C2(C)CC3CCC2O3)=O)C(C)(C)C1 C(=O)C(F)(F)F.C1CC(C(F)C=O)C1.CC(C)C.CCC1CC1.C(=O)O CC1(C)COc2ccc(C(N3CCC3CNC(c3cc(=O)cc[nH]3)=O)=O)cc21 N1(C(C(CC)C)=O)CC(NC(=O)C(c2ccccc2C(F)(F)F)O)C(O)C1 C12(NC(c3ccc(C(C)C)cn3)=O)CCCC1CN(C(C1OCCO1)=O)C2 Cc1cc(CCC(N2CC=CC2C(=O)N(CCC(C)C)C)=O)n[nH]1 C1(NC(C2NC(=O)C(F)C2)=O)CN(C(=O)C(F)(F)C(F)(F)F)CC1C1CC1 c1(OC)cc(N)c(C(N2CCC3(C2)CN(C(=O)C2=NOC(C)C2)C3)=O)cc1OC c1(C(N2CCN(C(C(C)CC(N)=O)=O)CC(O)C2)=O)ccnc2c1ncn2C N1(C(CNC(CC)=O)=O)CCC(C2CN(C(=O)C=Cc3cnc[nH]3)C2)CC1 C(c1cccc(O)c1)=CC(N1CCC1)=O.CCC(C)(C)NC(C)C(=O)NC c1(CN2C(C(=O)NCc3cc(Br)ccc3Cl)CC(F)C2)cc(Cl)cc(Cl)c1O O=C1CC(C(=O)N2CCC(NC(=O)C(F)(F)c3cscn3)CC2)c2ccccc21 C1(NC(C(C)=C2CCC2)=O)CCCCC1CC(=O)N.C1(C(C)(C)O)CC1.C N1(C(CC(=O)OCC)=O)CCC2(CC1)CC(C)C2.C1(CC(=O)N)COCCO1 C(=O)(C(C(C)C)NC(c1ccc(-c2cnccc2C)cc1)=O)NCC c1(C(N2CCC(O)(CC)C2)=O)ccnc(Cl)c1Cl.c1(OCC)nc(C=O)co1.N CCCCC(F)(F)C(=O)NC(C)CCCNC(C1CC(C(C)C)C1)=O C1(CNC(c2ccc(C3(C)CC3)cc2)=O)CN(C(c2cnc(Cl)[nH]2)=O)CCCO1 Cc1cc(Cl)c2ncc(C#N)c(N3CCC(NC(C4CSCCS4)=O)C3)c2c1 CCC(C)(C)C(C)CC(=O)NC1CCN(C(c2cc[nH]c2)=O)CC12CCC2 N1(C(c2c(CC)oc(C)c2)=O)CCC(NC(c2cc(=O)cc(Cl)[nH]2)=O)CC1C CCC(CC)CCC(C(=O)NCCCF)N1CC2CN(C)CC(C1)O2 C1(=C(C(=O)NCC(CO)NC(C2C(OCC)CC2)=O)F)CCCCC1 C1(C(N2CCC2)=O)CCCC2C1C2(F)F.C1(C(=O)NCC)CC2(CCC2)C1.O O=C1CCC(C(=O)NCC2(O)CCN(C(c3cccs3)=O)C2)CN1.C1CC1.C C1(C(=O)OC)CN(c2nc3ccccc3n2C(F)F)CC1C1CCCC1 C1(NC(c2c(CC)occ2)=O)CC2CC(NC(C3CC3C)=O)C1C2 C1(NC(C2C(C)CC(C)O2)=O)CN(C(c2ccccc2OCC#N)=O)CC1(C)C C(=O)(CCP(C)(C)=O)Nc1ncc(C(Cn2cc(-c3n(C)cnc3)nn2)=O)s1 c1(C(N2C(C)CC(NC(c3c(C)cno3)=O)C2)=O)ccc(S(N)(=O)=O)cc1 Cc1cc(CC(=O)NCC(C2CCC2)NC(C2CCC(=O)N2)=O)ccc1CO CC(O)C(F)(F)C(=O)N1CC(N(C)C(C2CN3CCN2CC3)=O)C(O)C1 c1(CNC(=O)NC2CCN(c3c(C)ccc(Cl)c3)C2)nc(C)c(C)nc1C c1(C(N2CCCC(NC(c3cc(C(C)=O)sc3)=O)C2)=O)cc(C)c(C)c(C)c1 CCC(=O)CCC(=O)N(C1CC(NC(c2cc(F)n(C)n2)=O)C1)C C1(C(N(CC(C)NC(C23CCC(C2)C3)=O)CC)=O)CCc2cnn(C)c2C1 c1c(F)cc(Br)cc1Cl.c1(OC)cccc(O)c1CNc1cc(C=O)n(C)c1.N Cc1nc(NCC(C2CC2)N(C)C(c2cc3ccccn3n2)=O)c2ccsc2n1 C(=O)(C(C(C)O)N(C)C)NCC1C(C(N2C(C(=O)OC)CC2)=O)CC1 Cc1cc(C)c(CC(=O)NC2CCCN(C(=O)C(O)C(C)(C)C)C2C)c(C)c1 C(CCC(CO)NC(C1CC1CCOC)=O)NC(CCCOCCOC)=O C1(NC(CC(=C)C)=O)CN(C(C2CCCCC2C(N)=O)=O)CCC12CCC2 C(CCF)(C(=O)OC)NC(C1C(NC(COCCC)=O)CCO1)=O C(C1=CCCN(C(=O)C(C)CC(F)F)C1)NC(c1cc(COC)[nH]n1)=O Cc1ccccc1C(C)CC(=O)NCC1(O)CN(C(=O)CN2CSCC2=O)C1 c1(CN2C(C3CCN(C(CCNC(C)=O)=O)C3)CCCC2)c(F)ccc(C)c1O Cc1ncc(CCNC(c2cc(CNC(=O)Cc3ccsc3C)cs2)=O)s1 c1(C(N2CC(C3N(C(CC(C)(C)O)=O)CCC3)(O)C2)=O)cn2ncccc2n1 C1(C(N(CC(F)Cl)C)=O)COCCC1NC(=O)CCC1CCCC1 CC1CCC(CCC(F)(F)F)N(C(=O)COC(=O)COC(F)(F)F)C1 C1(CCNC(C)=O)CCN(C(=NCCF)NCCn2nccn2)C1 N1(C(C2CC2C(F)(F)F)=O)CCN(C(=O)C(F)(F)C(F)F)C(CO)C1 c1(C(=O)NC2CN(C(C(C)P(C)(C)=O)=O)C3(C2)CCC3)ccc2c(c1)COC2=O N1(C(Cn2cc[n+](C)c2)=O)CCC(C2CCN(C(=O)CNc3ncccn3)CC2)C1 C1(C(=O)N)CCCC2(CC2)C1.c1(C(=O)NC2CCC2)cnn(C2CCOCC2)c1 C1(C(C2CC2)NC(Cn2ncc(N)c2)=O)CCC(N2CCCC2=O)CC1 N1(C(CC2(COC)CC2)=O)CC2CC1C2CNC(=O)CCCc1cncs1 C1(C(N(C(CC)CNC(=O)C2=CCCOC2)C)=O)CCC(N=[N+]=[N-])CC1 c1(SC)ccc(C=CC(=O)NC2CCC2)cc1.C1(C(=O)N)OCCN(C)C1=O c1(N2CCN(CCCC)CC2)nc(C(F)(F)F)nc(=NC2CC3CCCC3C2)[nH]1 c1(C(N2CCCC2COC)C(=O)NCCOCC)ccccc1OCC CC1C(NC(C2CCS(=O)(=O)N2)=O)CCN1C(=O)CCCCc1ccc(F)cc1 C1(C)(NC(c2cc(Br)ccc2OC)c2n(CCC)nnn2)CC2(C1)CC2(F)F C1(NC(c2c(C)nc(C3CCCO3)s2)=O)CC2CC1N(C(=O)C(C)(C)C1CC1)C2 c1(CNC2(C(=O)OC)CC(O)C2)n[nH]c2c1CCC2 N1(C(C(C(C)O)N(C)C)=O)CC2CS(=O)(=O)CC2(NC(C2CSC2)=O)C1 N1(C(C(CNC(=O)Cc2csc(C)n2)OC)=O)CCCC2(CC(O)C2)C1 c1(NC(CCC2N(C)CCCC2)=O)cccc(F)c1C(=O)O N1(C(CC(C)OC)=O)CCC(N(C(=O)CCC(C)=O)CCO)CC1 C(=O)(CCC(=O)NCCC1CN(C(C2CCCC2)=O)CCO1)NCCC c1(C(=O)NC2CCCN(C(C(CSC)OC)=O)CC2)ccc2n[nH]cc2c1 CC(=NO)C1CC(C(N2CCN(C(c3cscc3F)=O)C3(CCC3)C2)=O)C1(C)C Cc1cccc(O)c1C(=O)NCC1CN(C(c2ccnn2C2CCC2)=O)CCO1 c1(OC)ccc(OCCC(N2CCOC(CNC(c3sncc3C)=O)C2)=O)cc1 C1(C(N(CC(C2CC2)OCC)C)=O)CCC(C(=O)OC)S1 C1(C(=O)N(C)CC2CCOCC2)(CC)CCCN(C(C2CC2C#N)=O)C1 Cc1csc(C(=O)N(CCC(=O)NCC2CCC2(F)F)C(C)C)c1C C1(N(C(=O)C(c2ccnn2C)O)C)CCCN(C(c2ncnc(O)c2F)=O)CC1 c1(CC)ccc(C(C)C(=O)N)cc1.C1(CC(N2CC(CC)C2)=O)CC2CCC1O2 C1(NC(C2C(C)OCCC2)=O)CCN(C(C2CCCN(C)C2)=O)C1(C)C C1(NC(C2CC(C)C2)=O)CS(=O)(=O)CC1N=c1[nH]nc(O)s1 C1(C)(CNC(c2n(CC)ccn2)=O)CCN(C(c2cnn(CCO)c2)=O)C1 Cc1ccc(Br)c(NC(C2CCC(NC(=O)Cc3ccccc3F)CC2)=O)n1 C(=O)(C(O)C(C)(C)C)NCCCCN(CCC)C.c1(C(=O)N)ccc(N)cc1Cl C1(C(=O)NCCCN(C(=O)C(F)CC2CCC2)C(C)C)C(C)(C)C1(C)C c1(C(=O)NC2CCCC(NC(c3cn(C)c(O)n3)=O)C2)cnn2c(N)ccnc12 N1(C(C2(C)N(C)CC(O)C2)=O)CC=C(CCNC(c2c[nH]cc(Cl)c2=O)=O)CC1 c1(NC(C2C(CNC(CC(C)=C(C)C)=O)CCCC2)=O)cc(C)cc(C)c1O c1(C(N(C2CCN(C(c3c(CC)occ3)=O)C2)CCO)=O)cc(Cl)c(Cl)s1 N1(C(c2cccc(C#C)c2)=O)CC2C=CC1C(C(=O)NCCCCSC)C2 N1(C(C2C(C)(C)CCCO2)=O)CCCCCCC1C(=O)NC1CCN(CCF)C1 c1(C(CC(N2CCCC(O)(C(=O)OC(C)(C)C)C2)=O)O)nc2ccccc2[nH]1 c1(N2CCC(C)(CC)C2)cc(S(=O)(=O)NCC(C)(C)SC)ccc1C#N N1(C(CS(CC)(=O)=O)=O)CCN(C(c2ccnc(F)c2Cl)=O)C(C#N)C1 c1(C(=O)NCC(CN(C(=O)C(=O)NC2CC2)C)O)cnccc1Cl c1(N2CC(C)C(NC(=O)Cn3ccc(C(F)F)n3)CC2)ncnc2cccnc12 C1(CC=O)CCCN1C(C)C.C(C(=O)N(CC)C(C)C)C1CC1.CC.O Cc1ccc(Cl)c(N)c1C(=O)NC(CNC(C1C2CCCCC12)=O)C(C)C N1CCCCC1C.c1nnn(C)n1.CC C1(C(=O)NCc2nnc(C)s2)CC2(CCN(C(=O)CC(C)C(F)(F)F)C2)C1 c1(NC(C2CC(=C)CN2C(=O)CCCCN(C)C)=O)ccc(C)cc1COC c1(OC)cc2ncn(CN3CCC(c4ccc(Br)cc4F)C3)c(=O)c2cc1Br Cc1cc[nH]c1C(=O)NCC1(C(N)=O)CN(C(=O)CC(C)n2cccn2)C1 c1(COC)ncc(C(=O)N(C2CC2)Cc2nnn(C)n2)c(O)n1 CC1(C)CCCCC1(C)NC(c1coc(CNC(C2COCOC2)=O)n1)=O c1(C(=O)N)ccccc1Cl.CC(C)CCCNC(=O)CSCCC#N.C(N)=O C1(NC(COCC(=C)C)=O)CCCN(C(=O)COC(C)CC)C1 c1(C(N2CCC(NC(CC(C)(C)C(F)F)=O)C2)=O)ccc2c(c1)C(=O)CCCC2 c1(C(=O)NC2CC(C)N(C(=O)CC3(C)CCC3)C2)cc(Cl)cc(Br)c1 C1(C(CNC(c2cc(C)no2)=O)O)CCN(C(c2ncc(C(F)F)s2)=O)CC1 C(=O)(C#Cc1ccc(Cl)cc1)NC1CN(Cc2cc(OCC)ncc2Br)CC1F C1CC2CCCC(C1)N2C(C1CCN(C)C1=O)=O.C(=O)(CC(=O)N)OCC.C n1(CC)ncc(C)c1C(N1CCC(C(=O)NC(c2ccnn2C)C)C1)=O C1(C(C)NC(CC=CC=C)=O)CN(C(=O)COCc2ccncc2)CCO1 Cc1n[nH]c(C)c1C(N1CCC1C(=O)NCc1ccncc1)=O.[nH]1cccn1.C N1(Cc2cc(C)on2)CC(NC(C23CC(N(C)C)(C2)C3)=O)C(F)C1 c1(SCC(=O)NCC(CNC(CN2CC(C)C2)=O)O)nnc2ccccn12 c1(N(C)C)ccc(-c2nc(C(F)(F)F)cn2C)c(F)c1F C1(C(=O)NC(CN(C(CCSc2ccc(C)cc2)=O)C)C)CC12CC(C)(C)C2 N1(CC)CCC(NC(c2coc(CNC(c3scnc3Cl)=O)c2)=O)C(C)C1 CCC(CC)CCNC(=O)C(Cn1cncn1)NC(=O)C(=O)NC1CC1.O C12(C(N(CCNC(c3cncc(C)c3)=O)C)=O)CCC(F)(CC1)CC2 N1(C(c2nc(C(C)(C)C)sc2)C(=O)NCC2CC2)CCCN(C2CC2)CC1 C(CCC(=O)NC1(C)CC(NC(c2c[nH]cc2Br)=O)C1)=CCC=C c1(CCC)ncoc1C(N1CC(C(C)NC(=O)C(C)CN(C)C)C1)=O C#Cc1ccc(C(=O)NC2CCCCCC2NC(=O)C(C)C(F)(F)F)cn1 C1(CC(N2C(CNC(C3(CCC)CC3)=O)COCC2)=O)CCC(C)(C)CC1 c1(C(N2CCC(C(=O)Nc3cc(OC)ncn3)C2)=O)cc(I)c(F)cc1F c1(OC)cc(=NC(=O)NC2(c3cc(F)c(F)c(F)c3)CC2)[nH]n1C C1(C)(C(N(CCCN(C(C2CC(OC)C2)=O)C)C)=O)COCC1n1cccn1 c1(C(=O)NCC2N(C(CC(C)SC)=O)CC(C)(C)C2)cc2nc(C)ccc2o1 C12(CNC(c3ccc(C(=O)OC)cn3)=O)CCC(C1)N(C(=O)C(C)O)C2 CCCC(C(O)C(=O)N(CCOC)CC)NC(C1OCCCC1(C)C)=O c1(-c2onc(C(N3CCCC3)=O)n2)cccc(F)c1.CC1CC2(C(=O)NC)CC12 C(=O)(C#CC1CCCO1)NCC1C(NC(CN(S(N(C)C)(=O)=O)C)=O)C1 C(=O)(C(C)CC(C)C)NC(C1(CNC(c2ncn(CC)n2)=O)CC1)C c1(C(=O)N)cccc2[nH]nc(O)c12.c1(CNC(CC(C)F)=O)cc(O)nc(C)n1 N1(C(CCSC(C)C)=O)CCC2CCN(C(=O)CSC)CC2C1 c1(C(N2CC(CNC(C(c3c(C)nn(C)c3)O)=O)C(C)C2)=O)ccc(=N)[nH]c1Cl c1(C(N2CC(NC(C3(F)CCOCC3)=O)C(O)C2)=O)ccc2snnc2c1 C12(CN)CCCCC1CN(C(c1ccc(=O)n3c1CCC3)=O)C2 N1(C(=O)CNc2ccccn2)CCN(C(=O)Cc2cscn2)C2CS(=O)(=O)CC12 C(c1ccccc1OC(F)F)=CC=O.C(CC)NC(C1(CCO)CC1)=O.CC Cc1cc(C(N2CCCC(CNC(C3(C)CCCOC3)=O)C2)=O)nn1CCO C1(NC(c2cnc(C(F)F)s2)=O)CC2CC1N(C(C1CCCC1(F)F)=O)C2 C1(C(C)C)CCOCCN1C(c1ccc(Cl)cc1O)=O.C12CCCN(C1)C(=O)N2 Cc1cc(O)n2ncc(C(=O)OCC3CCCC(=O)C3)c2n1 C1(CCCNC(c2cnn(C3CC3)c2)=O)CCN(C(C23CCC2C3)=O)CC1.C n1(CC)ncc(C(=O)NC(CO)CCCNC(=O)C(N2CCCCCC2)C)c1C c1(-c2cn(CC(=O)NCCC(c3ccc(CO)cc3)O)nn2)ccc(Cl)c(Cl)c1 N1(C(C2(CC#C)CCCCO2)=O)CCC12CN(C(=O)CCn1cnnn1)C2 N1(C(CCC(=O)OCC)=O)CCCC2(CNC(=O)C(C)(C)CO)CCCC12 C(CC(=O)NCC12CC1CN(C(=O)C#CC1CC1)C2)(C(F)(F)F)OC c1(C(=O)OC)cccc(C(=O)NCC(C)C(C)C)c1.C1(C=O)C(C)C1C.N N1(C(c2cc(C3(C)COC3)no2)=O)CC(C)(C)CC1(C)C.C(=O)C=CCO.N CCCCCN(C(=O)C=CCNC(=O)C(C)c1cccs1)C C1(O)(C(N2CCN(C(c3nc(C)oc3C)=O)C(C)C2)=O)CCCC(C)(C)C1 N1(C(C#C)=O)CCC(NC(=O)C(CC)NC(=O)OC)C1(C)C.c1ccccc1 N1(C(C=CCN(CC#C)C)=O)CC(C)(C)CC1.c1(C=O)coc(C(F)F)c1 C1(O)(CC(N2CCC(O)C2)=O)COC(C)(C)C1.n1(CC)cnnc1C(=O)N.C Cc1cc(C(=O)NCC2CN(C(c3cc(-c4cccs4)on3)=O)C2)nc(C)n1 N1(C(CNC(=O)OC)=O)CC2CN(C(c3ncccc3N)=O)C2C1 c1(C(=O)NC2(C)CC(NC(CC(CC=C)(C)C)=O)C2)ccn2c(C)ncc2c1 c1(C(N2CC(O)(CCNC(c3c(C#C)c[nH]n3)=O)C2)=O)cc2cncn2c(O)n1 C1(NC(C(CC)CC)=O)CN(C(=O)Cc2csc(Br)n2)CC2CC12 c1(OC)c(C(=O)NC2CC(O)CN(C(=O)C(F)CC3CCCC3)C2)cccc1Cl C(CCC(N)=O)(C(=O)NNC(=O)Cc1ccccc1F)n1cc(COC)nn1 N1(c2ccnc(SC)n2)CC2(CCCC2NC(c2coc(Cl)n2)=O)C1 C1(CNC(C(C#C)(C)C)=O)CC2CCC(C1)N2c1nc(Cl)ncc1CC c1(C(=O)NCC2CCN(C(c3c(C)nn[nH]3)=O)C23CC3)c(Cl)nc2ccccn12 c1(C(=O)NCc2cnsc2)cccn1C1CCCC1 C(CNCC1(Br)CC1C(=O)O)(CC(F)(F)F)OC C(c1ccc(Cl)cc1)=C(C=O)C.C1CCC1(C)C.C(C(=O)N)NC(=O)OC c1(C(=O)NCC(CN(C(C(C)c2cccs2)=O)C)C)cc2c([nH]1)CCC2 N1(C(C(C)C(F)(F)F)=O)CCCC(C2(NC(c3ccc4oncc4c3)=O)CC2)C1 c1(C(=O)NC(C)CCCNC(=O)Cc2nn(C)cc2Cl)cc(N)c(O)c(F)c1 C(C(C)NC(c1n[nH]cc1Cl)=O)(C(C)C)NC(c1cnc(C(=O)OC)s1)=O c1(C(N2CCC2)=O)cnc(Cl)cn1.C1(CC)(C(=O)N)CCC1.CCOCC c1(C(=O)NC(C(C)NC(=O)C=CC(F)(F)F)(C)C)ccc(N(C)C)nc1 C1(C)(CC(=O)NCC=C)CCN(C(=O)CCC2CCOCC2)C1 C1(C(=O)NCCc2cc(C)[nH]n2)(CC)CCN(C(=O)Cc2nncn2C)C1 C1(C(=O)NC(C(=O)OC)CCF)CCCCCCN1C(c1cocn1)=O C1(C)(C(=O)NCC2(O)CN(C)C2)CCN(C(C2CCN(C)CC2)=O)C1 CCCCCC(C)(CC)C(=O)NCC1(COC)CCCN1C(=O)C(C)C(F)(F)F Cc1ccc(C)n1CCC(N1CCC(CCNC(C23CCCCC2C3)=O)CC1)=O C1(NC(CCC)(c2nnnn2C2CCOCC2)C2CC2)CC2CCOC12 C1(NC(c2c(N)nccn2)=O)C2CCC1CN(C(c1cnc(OCF)cn1)=O)C2 c1(C(C)C)n[nH]cc1C(=O)NC1CC1NC(=O)C(C1CCCCC1)F CC(C)(C#N)CCC(=O)N1CCC(CNC(=O)C=Cc2cocn2)C1 C1(NC(c2c(C)cc(CO)o2)=O)CC2CCC(C1)N2C1CC1 CN=c1[nH]cc(C(=O)NC(C(=O)NC2CCCC(O)C2)C2CC2)o1 c1(CC(=O)NC(C2CCCN2C(=O)Cc2csc(Cl)n2)C)ncc(Cl)s1 C1(CC(=O)NC(CC=C)CC)CC2(C1)CN(C(c1cccc(F)c1OC)=O)C2 c1(C(=O)NCCN(C(=O)C(O)CF)C2CC2)ccccc1.c1ccccc1.O N1(C(C(CCCC)O)=O)CC(CNC(c2cc3cnccc3o2)=O)CC(C)(C)C1 Cc1cccc(C(C)C(=O)N)c1.C(F)(F)C(F)(F)F.C12CC(C1)C2.C(=O)C N1(c2nnc(COc3c(OC)cccc3)n2CC2CCOC2)CC2CC1CS2=O N1(C(C(C)=O)=O)CC(F)(F)CC1(C)CNC(C1CCCC12CC2)=O N1(c2cccc(C(C)C)n2)CCC2=C(COC2=O)C1 CCC(C(=O)NCC(C(=O)NCCC(C)N1CCC1)OC)NC(N)=O CC(O)(C(=O)N1CCCC(NC(C2(c3ccno3)CCOCC2)=O)C1)C(F)(F)F c1(C(N2CCC(O)C2)=O)cncc2[nH]ccc12.C1(C(=O)N)CC2(C1)CC2(F)F.C C1(C(N2CCC(CCOC)C2)=O)C2CCC(C2)N1C(C1CCOCC1)=O c1(OC)ccc(C(=O)C(N2CC(NC(c3ccc(Cl)s3)=O)CC2C)=O)cc1 C(=O)(C(CC(C)(C)C)NC(=O)CSCC(F)F)N1CC(C(C)C)C1 C1(NC(c2c(C)cccn2)=O)CCCCC12CCN(C(C1CCCS1)=O)CC2 C1(CNC(C2CCC(C)(C)C2)=O)CCCN(C(=O)Cc2cscn2)CC1 Cc1ccc(C(=O)N(C)CC2COCCN2C(C2CC2C(F)F)=O)c(Cl)c1 c1(OC)ccc(C(F)(F)F)c(F)c1NC(=O)N.C(C)C(C)(C)c1ccccc1 N1(CC(N2CCC(=CC)CC2)=O)CCCNS1(=O)=O.CC1(C)COCC1C=O.N N1(C(C=CC(C)NC(=O)Cc2ccc(O)cc2)=O)CC(=O)NC(=O)C1 c1(C(=O)NCCSCC2CC(O)C23CC(F)(F)C3)cnc2ncc(Br)cc2c1 C1(CC=C)(NC(C2CC(C)=NO2)=O)CCCN(C(c2cncn(C)c2=O)=O)C1 C(C(O)C(=O)NC1(C(=O)NC2CC2C)CCC1)SC C12(NC(c3n(CC)ccc3)=O)CCN(C(c3ccsc3OC)=O)CC1C2 C=CC1CN(C(=O)C(n2cc(C)cn2)C)CC1NC(=O)CC=CCC Cc1nn(C)cc1C(=O)N(CC(C)NC(CC(C)C(F)F)=O)C Cc1nc2c([nH]1)C(C(=O)NCC=CC)CCC2.c1(C(=O)N)cc(Cl)c(Cl)n1C C1(NC(C2(C)CCOC2)=O)CN(C(=O)CCN2CCCS2(=O)=O)CC2(CCC2)C1 CC(C)C(C)(C)C(=O)NC1CCN(C(=O)Cc2cccc(C(F)(F)F)n2)CC1F CCC(C)CCC(O)CC(=O)Nc1cccc(CN=c2[nH]c(OC)ncc2Br)c1 C1(C(=O)OCC)CCCN(C(=O)C=CC(=O)N)C1.c1cc(C2CC2)nn1C c1(C(=O)NCCC(C)NC(c2cc(SC)oc2)=O)cc(C)c2occc2c1 CCC(C)C(=O)NCC(=O)NC1(C)CC1.c1(C=O)cc(CC(C)C)[nH]n1.N N#Cc1nc(NC(C2(C)CC2)=O)cs1.n1(CC=O)cc(C2CCOC2)cn1.N C(C(C(=O)N(CCCC(C)O)C)n1cc(C2CC(=O)C2)nn1)OCC.C1CC1.C c1(C=O)cnn(CC(F)(F)F)c1C.C1(CCC)CC1C(=O)N.C(C)C1CCC1 N1(C(C2N(C(CC(=O)NCC#C)=O)CCC2)=O)C2COCC1C2 N1(C(C(C)C2CCOC2)=O)CCC2(CC1)CCN(C(=O)CCn1ccc(=N)[nH]1)C2 C1(C)(NC(C(C)(C)OCCC)=O)CCN(C(C2CC2c2cncn2C)=O)C1 c1(C(=O)NCC(C)N(C(C2CCCN(CC)C2)=O)C)cncc(N2CCCC2)n1 C1(N(C(=O)Cc2cnsc2)C)CN(C(c2c[nH]nc2Cl)=O)CC12CC2 C1(C(=O)NC(c2cn(C)nn2)C(=O)Nc2ccc(F)nc2)CCCOCC1 c1(C=O)cn2c(C)cccc2n1.C1(COC)CC1C(=O)N(CC(C)O)CC N1(C(CC=CC=C)=O)CCC(CCNC(=O)CCCC(=O)N(CC)CC)CC1C C1(N(C(=O)C(n2cc(-c3cc[nH]n3)nn2)C)CC)CNCCC1(C)C CC1=C(C(=O)N2CCC(C)(CC(=O)N(C)CC3(F)CCC3)C2)CCO1 CC(C)CC(O)C(=O)NC1(CCNC(=O)C(O)C(C)C)CCCC1 c1(C(N(C(C)CNC(C2CCCCO2)=O)C)=O)cc2n(n1)CCO2 c1(C(N2C(CCCC)CCC2)=O)ccc(Cl)nc1NC(c1cc(C)c(C)[nH]1)=O CC(C)C(C)CC(=O)N1C2CCC(C2)C1CC(=O)NCc1cncs1 C1(NC(=O)COCC2CCCOC2)CN(C(c2cc[nH]n2)=O)C2(CCC2)C1 C(=O)(C1CC(=O)Nc2ncccc21)N(C1CCN(C(c2cn[nH]c2)=O)CC1)CC c1(CC(N2CC(NC(C3CN(C)C(=O)C3)=O)CC2(C)C)=O)ccc(F)c(Cl)c1F N1(C(C)C)CC2CN(C(=O)C(C)n3cnnn3)CC2C1 CON=Cc1ccc(C(=O)NC2(CO)CCCN(C(C3C4CCCC34)=O)C2)cc1 CCC1=C(C(=O)N2CC(CO)(NC(=O)CC(C)CC(F)(F)F)C2)CCCO1 C1(NC(C(CC)OCC)=O)CN(C(=O)CCCCC2CCCCC2)CCC1(F)F C1(C(=O)NC(C(C(=O)OC)C)C)CC2(CCN1C(=O)C(OC)OC)CC2 C1(NC(C2(CC#C)CCCCC2)=O)CCCN(C(=O)C(c2cnn(C)c2)O)CC1 N1(C(C=CCC)=O)CCC2(CCC2CNC(c2cccn2CC)=O)CC1 C1(C2CCCCC2)(n2cc(-c3c(OC)ncc(Cl)c3)nn2)CCCCC1 Cc1nccc(C(=O)NC2CCC2)c1N.c1(C(=O)N)ccc(C=O)[nH]1.CC(C)C Cc1cccc(O)c1CNC1(C#N)CCN(Cc2cccc(C(F)(F)F)c2F)C1 n1(CC=O)nc(C)[nH]c1=O.C(C)(C(C)(C)C)NC(C(CSCC)F)=O.N C1(CC(=O)N(CC(CC)NC(c2sccc2NC)=O)C)CCS(=O)(=O)C1 C#CCC(O)C(=O)NCC(CC)NC(c1cc(-c2ccc(OC)cc2)[nH]n1)=O C1(CCNC(C2COCOC2)=O)CCCN(C(c2cccc[n+]2[O-])=O)C1 c1(NS(C)(=O)=O)cccc(C(=O)NC2CC(C)C2)c1.c1(C=O)cn[nH]c1.C N1(C(C2(SC)CC2)=O)CC2CC1(CNC(=O)C(C)(C)C1CCCO1)C2 C1(NC(CC(C)SC)=O)CCN(C(C2CCCC3(CC3)C2)=O)CC1F c1(C(C(=O)NC(CNC(CC(C)O)=O)C2CCC2)CO)ccc(F)cc1 c1(C(=O)OCCSCc2ccccc2)cnn2ccc(O)nc12 CC1C2C(CCN2C(C2CCC(C)(C)CC2)=O)CN1C(C1CCC(F)C1)=O c1(CC(=O)N(C2CCCC2)C(C)CO)nncn1C c1(C(=O)NC(CC2CN(C(CC(C(C)C)C)=O)C2)C)c(F)cc(F)cc1Cl C1(C(=O)NC2CCC(NC(CCCC3(C)N=N3)=O)C2)Cc2cc(Cl)ccc2O1 C(=O)(C(O)CC(C)(C)C)NC(CNC(c1c(C)nn(C2CCC2)c1)=O)C(C)C C1(NC(CC(=C=C)C)=O)CC(O)CN(C(c2csc(CCP(C)(C)=O)n2)=O)C1 CCC(CNC(C1CC1(C)Br)=O)(CC)NC(=O)COC1CCN(C)CC1 N1(C(c2c(CNC(Cc3c(C)ncs3)=O)noc2)=O)CC2(C)COCC2(C)C1 C(=O)(C1=CC2C=CC1C2)NCC(CC)(C)C(=O)NCCC(F)(F)C(C)C C12(C(=O)NCC(CC)(CC)CC)CCCC1CCN2C(=O)CCc1cncnc1 C1(NC(C(C)CN(C)C)=O)CC2CCC1CC2.c1(C=O)cc(SC(F)(F)F)c[nH]1 C1(CNC(c2c(C)coc2C)=O)CC2(CC2)CN1C(C1CCCCCCC1)=O c1(OC)cc(C(=O)NCC2(NC(C3CCCOC3)=O)CCOC2)ccc1Cl C1(F)(C(=O)OC(C)=O)CCCCC1.CCC1C(=O)N2CC(C)(C2)c2cn1nn2 C1(C(=O)NC(C2CCCCC2)CC)CC(NC(c2cccc(C)c2)=O)CCO1 C1(C)(NC(C(C)CO)=O)CCN(C(=O)C(F)(F)C(F)F)CC1 c1(CN2C(C(=O)Nc3ccc(CC)nc3)CC3(CC3)C2)ccc(Br)c(OC)c1F C#CCC(C(=O)NC(c1cnn(C)c1)C)NC(=O)C(C)NC(N)=O C1(C)(C=O)CCCS1(=O)=O.c1(SCC)ccccc1C(N1CCC(O)C1)=O.C n1(CCC(=O)N(CC)CC)nc(O)c2ccccc12.C(=O)C(O)CC(C)(C)C.N c1(Nc2ccc(C(=O)NCC3N(C(C(C)O)=O)CC3)cc2)cccc(C#N)c1 c1(C(N)=O)ccnc(N(C2CC3(CNC3)C2)C(c2ccccc2)=O)n1 c1(OC)nn(C)cc1NC(=O)C(n1cc(-c2ccc(C3CCOC3)cc2)nn1)C C1(C(=O)NC(CN(C(CCN(C(CC)CC)C)=O)C)CC)CC(=O)N(C2CC2)C1 c1(C(=O)NC(CC=C)CNC(C2(CCOC)CC2)=O)cnc2ccnn2c1.C N1(C(CCC(=O)NC)=O)CCN(C(c2nnsc2N)=O)C2CCCC2(C)C1 C=CCCCC(=O)NC1(C(N2CCC(CCOC)CC2)=O)CCOCC1 Cc1ccc(Cl)c(F)c1C(N1CCCC(NC(C23CC(C)C2C3)=O)C1)=O c1(C(C)=O)ccc(NC(=O)CC2CCC2)c(F)c1.C1(CC=O)COC(=O)C1 N1(C(C(C)Cc2ccncc2)=O)CC2CCC1C(C(=O)NC1CCN(C)CC1)C2 C(N=c1ccnc(Cl)[nH]1)C1(C(C)(C)C)CCN(C(c2cnn3c2CCCC3)=O)C1 C(=O)C1=CCCOCC1.C1(C(=O)NCCC)(CN(C)S(N)(=O)=O)CCCCC1 CCC(C)(O)C(=O)N1CSCC1C(=O)NCC1(CC)CCCO1 CC1=C(C(=O)N2CCC(CCN(C(=O)C=Cc3cccs3)C)CC2)CCCC1 CC1CCCN1CC(=O)NCCc1n[nH]cc1C(=O)NC(C(O)CO)C1CC1 c1(NC2CCCC(NC(=O)OC(C)(C)C)CC2)c(Cl)cc([N+](=O)[O-])cc1Cl c1(NC(=O)NC(c2nnc(O)n2C)C)cc(F)cc(Cl)c1F Cc1nnc2n1CC(C(=O)Nc1ccnn1C(C)C(F)(F)F)CC2 N1(C(c2c(N)nccc2)=O)CC2CC1CN2C(C12COC(CSC)(C1)C2)=O CCC(C)(C)C(C)CC(=O)N(CCNC(=O)C(F)OC)CCOC Cc1nc(CCC(=O)NC(C)(CNC(c2ccoc2)=O)CO)[nH]c1C C#Cc1cc(C(=O)Nc2cccc(CNC(=O)C(C)NCC)c2)ccc1Cl.C CCC(CC1CCCC1)C(=O)NC(C)C(C)(C)NC(c1cc(CO)oc1C)=O CCCCC(O)C(=O)N1CCCC1(C)CNC(C1(CCc2ccccc2)CC1)=O C1(NC(CSCCC#N)=O)CN(C(c2ncn3ccccc23)=O)C2(CCOC2)C1 Cc1cccc(CC(=O)Nc2cccc(C(O)C(F)(F)F)c2)c1Br Cc1cc(N2CC(C)CC2C(=O)Nc2ccsc2)nc(C)n1 C1(CC(=O)NCCCN(C(COCCC=C)=O)CC)CSCCO1 c1(C(C(N2CCC(n3cc(CCC(C)(C)O)nn3)C2)=O)O)ccc(F)c(Br)c1 CCC(C)C(O)C(=O)NCCN(C(c1ncc(Cl)nc1Cl)=O)CC N1(C(c2c(CC)ocn2)=O)CCC(CNC(c2cnc(C)nc2)=O)C(C)C1 Cc1cc([N+](=O)[O-])cnc1N1CC(O)(CCNC(=O)C(O)Cc2cnc[nH]2)C1 c1(C(N(C(C(C)C)C)CCO)=O)ccc(S(=O)(=O)N2CCNC(=O)C2)cc1 c1(C(=O)NCCN(C(=O)CC2CCCC(O)C2)CC)sc2ncccc2c1Cl c1(CC(=O)NCCC2CCC2)ccccc1[N+](=O)[O-].C12(C=O)CC3CC1C2C3.N C1(NC(CNC=O)=O)CN(C(=O)C(C)SC(F)(F)F)C2CCCC12 C(=O)(C(CC)N(C)C)NC1CC(O)(CNC(C=C(COC)C)=O)C1.O c1(CNC(C(=O)N(C2CCCCCCC2)CCCC)=O)cc2c(s1)CCCC2 N1(S(=O)(=O)C2CC3CCC2C2OC32)CC2CC(F)(F)CC(C1)C2(F)F c1(OCC)ccc(NC=O)cn1.C12CC(C1)C2.C(=O)CCC1CC1(F)F CC(C)CC(C)(CNC(=O)C(C)C(F)F)NC(=O)C=Cc1ccco1 c1(C(N2CCC(N(C(=O)CC3CCCCC3)CC#C)CC2)=O)cnc(N)c(O)c1 c1(C(C(=O)N(CC(C)NC(CCN(CCCCC)C)=O)C)(C)C)c(C)noc1C c1(C=O)c(C)cc[nH]c1=N.C1(C(N2CC(CC)(OC)C2)=O)CC2(C1)CC(F)C2 C(=O)(CC=C(Cl)Cl)N(C(CNC(CC)=O)Cc1ccccc1)C C1(NC(c2cc(C)c(C)o2)=O)CCCN(C(=O)C(C(C)C)NS(C)(=O)=O)CCC1 C(=O)(CCCCCN(C(=O)C(C#N)C(C)C)C)N1CCC(C=C)C1 C(=O)(C(O)C(C)(C)C)NC1CC(N(C(c2scc(C)c2Br)=O)C)C1 c1(C(=O)OC)cc(NC(=O)C(=O)NC2CC3(COC3)C2)c(C)cc1F N1(C(C2CCCCC2)=O)CC2CC2(C(N2CCCC2c2ccc(Br)cc2)=O)C1 CC1(C)CN(C(c2ccc(C(F)F)cc2)=O)CCN1Cc1ccc(C(F)F)cc1 Cc1ccc2c(c1)SC(C(=O)NCCNC(C1CCc3nc(=N)[nH]cc3C1)=O)C2 C1(C(=O)Nc2cc(C)ccc2)CNC(=O)C(C)(C)C1.c1(C=O)nc(=O)n(C)[nH]1 CCC(CC)(C(=O)NCC(F)CNC(c1cc(N)cc(O)c1)=O)c1ccccc1 c1(C(N(CC(C)NC(=O)C(C)(C)F)CC)=O)ccc(C(=O)C2CC2)cn1 C1(CNC(C(CNC(c2n(CC)ccc2)=O)C)=O)OCCCC1(C)C c1(OC)c(C(=O)OC(c2cc(C3CC3)ns2)c2nnnn2C)[nH]c2ccccc12 c1(CCC)nn(C)cc1NC(C1CCCN(C(c2ccc(F)c(C)n2)=O)C1)=O.N N1(C(C(CC)C(=O)OC)=O)CCOCC12COCCN(C(=O)C(C)(C)C1CC1)C2 N1(C(C(CC=C)N(C)C)=O)CCC2(CCCN2C(c2cnc(C3CC3)[nH]2)=O)C1 c1(CC)cccnc1C(=O)N(CCCNC(=O)COCC(F)F)C1CC1 c1(C(N2CC3C(NC(C(C)SCC)=O)(C3)C2)=O)cccc(C2CC2)c1C C(=O)(C1CCc2cccc(O)c21)N1C(CCNC(CCC(C)C)=O)COCC1 C(N=c1[nH]c(=N)[nH]c(=NC2CC(=O)N(C)C2)[nH]1)c1nccc(C)c1F c1(C(N2CCOC(C)(C)C2)=O)ccc2[nH]cc(C#N)c2c1.CC1CC1C(=O)NC Cn1[nH]c(=NC(=O)N2CCC3(CC2)OCCO3)c2cccnc12 N1(C(C2(C)CC2)=O)CCOC(C(c2ccccc2)(C)C)C1.c12cn(nn1)C2 c1(C(N2CC3N(C(C(C)OCC)=O)CC(C3)C2)=O)ccc2nnc(C(F)F)n2c1 C(=O)(CCCCC(N)=O)N1C(C(=O)Nc2cccc(C)c2C)CC(OC)C1 c1(CC)cc(C(=O)NC2CCC(C)N(C(=O)COc3ccsn3)C2)c(C)nn1 c1(OC)cccc2c1OC(C(=O)NCC(C(C)C)NC(c1cc(C)nn1C)=O)C2 c1(OC)ccc(C(C(=O)NCc2ccccc2Cl)N(C)CC2CC2)cc1Cl c1(CC)ccccc1NC(=O)C(C)=CCNC(=O)C(C)N(C)C(C)=O NC(=S)c1ccc(NCCC2CC23CCOCC3)cc1 C1(C(=O)NC2(C)CN(C(CC(=C=C)C)=O)C2)CC2CC(OC)C2C1 O=C(C1=COCCC1)NC1CCCN(C(C23CCCC(CO2)C3)=O)CC1 C(=O)(C1=C2CCN=C2NC=C1)N(CCCN(C(c1onc(C)c1C)=O)C)C c1(C(N(C)CC2(O)CCN(C(c3ccc(O)nc3)=O)C2)=O)ccc2ncnn2c1 c1(CN(C)C)ccc(C(N2CCC(CNC(c3c[nH]c(Br)c3)=O)C2)=O)cc1 C1(C(=O)NC2CCC(NC(c3cnc(CCC)s3)=O)CC2)CCn2nccc2C1 S(=O)(=O)(CCC(F)(F)F)NC(c1cccc(Cl)c1)C(=O)NCCOC.O c1(C(=O)OCC(=O)N(C2CC2)Cc2ccc(C)cc2)csc2cncn12 C(=O)(C(C)CC=O)N1C(CNC(C2(C(F)(F)F)CC(=C)C2)=O)CC(O)C1 C1(CNC(Cc2cccc(CC)c2)=O)CN(C(=O)CC(=O)OC)CC(C)(C)C1 N1(C(C2(COC)CC=CCC2)=O)CCC2(CC1)CN(C(c1cc(C#N)cs1)=O)C2 N1(C(C(COC)(C)O)=O)CC2(C=C(C(=O)N3CCCC(CCO)C3)CO2)C1 CCCCC(C(=O)N1CC(OCCNC(=O)C(C)(O)C2CC2)C1)ON=C(C)C C1(NC(=O)C2=CCCCO2)CCC2(CC1)CCN(C(c1ccc(O)cc1F)=O)C2 CC1C(C(=O)NCC(O)CC(=O)NCC2(F)CCCCC2)CCN1C CC(C)C(O)C(C)C(=O)N1CC2CC2(C(=O)NCC2=NOC3(CCC3)C2)C1 N1(C(C(Cc2cc[nH]n2)NC(C2C(C#N)C2)=O)=O)CCC(O)C(F)(F)C1 N1(C(COCCCCC)=O)CCC(C)(C)C(NC(c2nccc3ccsc23)=O)C1 N1(C(C(=O)NC2CC2)c2nc[nH]n2)CC2CCCCC2(C(N2CCOCC2)=O)C1 C(=O)(CCC1=CCCCC1)NCC1CC(C(=O)NC2(CO)CC(OC)C2)C1 CCC(C)(C)C(O)C(=O)N1CCCC1C(C)(C)C(N1CCCC(C#N)C1)=O C1(NC(=O)CC(O)Cc2ccccc2)CCCN(C(c2scnc2Cl)=O)CC1 C1(C(=O)NCc2c(C)n(C)nn2)CN(C(=O)CC2CCSC2)CC1(F)F c1(C(N2CCC(NC(c3ccc(SC)o3)=O)C2)=O)ccc(O)nc1C.C1CC1.C CC1(C)C2CCC1(C(N1CCC3C(C1)CN3C(=O)Cc1c[nH]nc1O)=O)CC2 C1(C(N2CC(N(C(c3c(COC)c[nH]n3)=O)C)C2)=O)C2CC3CC(C2)CC1C3 c1(CC(N2CCC(NC(CCC(C)OC)=O)C2C)=O)cc(S(N)(=O)=O)cn1C c1(C(N2CC3C(C)C3C2)=O)cc(Br)c2[nH]nnc2c1.C(=O)(C(F)(F)C1CC1)N CC(CC(=O)NCC1CCN1C(c1ccc(C2CC2)nc1O)=O)P(C)(C)=O C1(NC(C(CSC)O)=O)CCN(C(c2cccc(C)c2Cl)=O)CC1O CP(C)(=O)COCC(=O)NCCC1(NC(=O)CCCC2CCC2)CCCC1 C(=O)(C1CCCc2c1ncn2C)N(C(C)CC)C1CC1.C(=O)(C(F)=C1CCCC1)N C(=O)(C1CCc2nccn21)N(CCCOCCN(C)C(C1CC12CCCC2)=O)C C(CC(C(C)(C)C)NC(=O)Cc1cc(C)no1)N(C(C1C(CC)C1)=O)C C(=O)(C(O)CCC(C)C)N(CC(C)O)CCNC(c1cccc(C#C)c1)=O C1(C(=O)NC(c2ccccn2)CC)CCN(C(=O)C(C)OCCC(C)C)CCO1 c1(C(N(CCC)CCNC(C2CC3C=CC2C3)=O)=O)cc(C)cc(Br)c1O O=C(C1=NOCC1)NC1CC(C(=O)NCC2CN(C3CC3)C2)C1 C1(C#N)(C(N2CCCC(C)(NC(c3c(SC)n(C)nc3)=O)C2)=O)CC12CCCC2 C1(C(N2C(CC)CCC2)=O)CCC2(CC2)N1C(=O)CC1(OC)CCC1 N1(C(CC2CCCN(C(c3c[nH]c(=NC)o3)=O)C2)=O)CC(O)C(C)(C)C1 c1(CC(=O)N)cn2c(n1)CCCC2.C1(C(=O)NCCCC)CCC(N(C)C)CC1 Cc1cccc2c(C(=O)NCC3CCCN(C(=O)Cc4nc[nH]n4)CC3)c[nH]c12 CC(CC(F)(F)F)C(=O)NC(Cn1cccn1)C(=O)NC1CC(=O)NC(=O)C1 N(C(=NCCCCC(F)(F)F)NC1CC(c2ccc(F)cc2)C1)CC(C)C1CC1 C12(C(=O)NC3(CNC(C(C)C(F)F)=O)CCCC3)CCC(CC1)C(C)O2 N1(CC)CCOC(C(=O)NC2CN(C(c3ccc(C(C)(C)C)cn3)=O)CC2C)C1 Nc1ccc(F)c(C(N2CCC(CO)(CNC(=O)CCC3CC3)CC2)=O)c1F C1(CNC(Cc2c(C)n[nH]c2)=O)CN(C(c2ncccc2C(F)F)=O)CCC1C CC1CN(C)CC1NC(c1ccc(CNC(C2CC23CCOC3)=O)nc1)=O c1(SC)cccc(F)c1C(N1CCC(n2cc(CC3(O)CCC3)nn2)CC1)=O CC1CCN(C(c2c[nH]c(C(F)(F)F)c2)=O)CC1CNC(=O)CCCC(F)F C1(NC(C(CC)NC(N)=O)=O)CN(C(=O)CC(C)SC)CC2(CCC2)C1 c1(CC(N2CCCN(C(C3CCC(CC)CC3)=O)CC2)=O)c[nH]c2cccnc12 C(=O)(C#CC1CCOC1)NC(CNC(c1ccc(C)c(Cl)c1)=O)C1CC1 C1(C(C)C)CC(C)CCN1C(c1cc(CNC(C2CC2(F)Cl)=O)[nH]n1)=O CC(C)(C)CC=O.c1(CC=O)cn(C2CC2)nn1.C(=O)CC.CC(F)(F)F.N Cc1cc(C#N)ccc1C(=O)N.C1CCC(C)N(C(=O)C)C1.C(=O)CC(C)(C)C c1(N2CCCN(C(C)=O)CC2)nc(N2CCCC(C)(C)C2)c2ncn(C)c2n1 C1(COC)CCCN(C(C2C=CCCN2C(=O)CNc2ccccn2)=O)C1 c1(OC)cc(C(=O)NC2CC2)cc([N+](=O)[O-])c1O.C(=O)C1=CC2CCC1C2.C C(=O)(CC(C)CC(C)(C)C)NCCCCN(C(c1c(CC)oc(C)c1)=O)C N1(C(COCC)=O)CCC2CCCN(C(c3cnc(C(F)(F)F)c(F)c3)=O)C2C1 Cc1nn(CC(=O)N(CC(C)NC(=O)COc2cccc(C(C)C)c2)C)cc1Cl CCC(C(C)CN(C)C)NC(C1(NC(=O)CC(C)OC)CCSC1)=O c1(C(N2CC(C)N(C(=O)C(C)CC3CC3)CC2C)=O)ccc2ccn(C)c2c1 O=C(C1=CCCN(Cc2c(Cl)ccc(Cl)c2F)C1)NCC(O)C(F)(F)F c1(C(=O)NCC(C(C)C)NC(=O)C(c2ccccc2F)O)ccc2c[nH]nc2c1 C1(C(N2CC(O)(CN(C(CCc3c(C)cccn3)=O)C)C2)=O)CC2CC1CC2O c1(CCNC(C(c2ccn(CC)n2)N(CC)CC)=O)ccccc1.C(C)C c1(CNC(=O)CCc2ccc(C(N3CC(F)(F)C3)=O)[nH]2)cc2ccccc2s1 Cc1cc(C(=O)NCC2CCCC2)c(S(N)(=O)=O)s1.C(=O)(CNC=O)N C1(NC(=O)C(F)=C(C)C)CCCN(C(c2cc(C(C)C)ccc2F)=O)CC1.CC c1(C(=O)NC(CCCNC(C(C)O)=O)C)cn(C)nc1-c1cnccn1 c1(C(=O)NCC2C(NC(C(C(CC)(C)C)O)=O)CC2)cc([N+](=O)[O-])cnc1C C1(OC)CN(C(=O)COc2ccccc2)CCC1NC(C1CNC(=O)CC1C)=O C1(C)(C(=O)NC(C)CC2CC2)C=CCN1C(=O)C=Cc1ccsc1 Cc1cnncc1C(=O)NC.C1(C(F)F)CCN(C(=O)CC)C1.[SH](C)(=O)=O Cc1ncc(C(N2CCSCC2C(=O)NC2CCCC2CN(C)C)=O)n1C c1(C(=O)N)ncc2c(F)cccn12.N#CC1(C(=O)NC2CCC2)CC2(CCC2)C1 Cc1noc2cc(C(=O)N)ccc12.C1CC2CC(C1)N(C(C13CC(C)(C1)C3)=O)C2 c1(C(NCCN(C(=O)CCCC(N)=O)CC)=O)cc(F)cc2nn(C)cc12.C n1(C(C)(C)C)ccc(C(=O)NCCCC2CCCN2C(C2C=CCCC2)=O)n1 c1(OCC)cccc(C(=O)NC2CCC(C)CC2)c1.c1(C(=O)N)ccnnc1S Cc1cc(CN(C(c2cc(C3CC3)on2)C(=O)NCCCF)C)n(C)n1 c1(C(N2CCC(C(=O)N(C(C)(C)C)CCO)C2)=O)c(C#N)cccc1[N+](=O)[O-] Cn1nc(C(=O)NCC(C)(CO)NC(=O)CC2CC3CC3C2)c(Cl)c1Cl Cc1cccn2ncc(C(=O)NCC3C=CCC3)c12.C1(C(=O)N)CC(F)(F)C1 C1(CNC(Cc2c(C)non2)=O)CC2CCC(C1)N2C(c1nccc(Cl)c1C)=O CC1(C)CC(=O)NCC1C(=O)N.C1CCCCN1C(=O)C=CCn1cncn1 N1(c2ncc(C)cn2)CC=C(CCNC(=O)C(F)(F)C(C)O)CC1 C(=O)(CCCN=[N+]=[N-])NCC1C(NC(c2c(C)nn(C)c2)=O)CCCC1 N1(C(CC(CCC)NC(C2CCC(C)(C)OC2)=O)=O)CCCN(C)CC1C c1(N2C(CCNC(c3ccc(N(C)C)cn3)=O)CCC2)nccc(C#N)n1 N1(C(Cc2c(C)ncs2)=O)C2CCC1CN(C(C1CC1C=O)=O)C2.C(C)(C)C.O N1(C(CNC(=O)OC)=O)CC(C2CCCCN(C(=O)CC3CCCC(C)C3)C2)C1 N1(C(C2(CCC)CCC2)=O)CC2CC(NC(C34CCOC3CCOC4)=O)CC1C2 c1(CC(=O)NCC2(C(C)NC(c3cnnn3C)=O)CC2)c(Cl)cccc1Cl C(C(O)C(=O)N=S1(=O)CCC2(CC1)OCCO2)N1CCN(C=O)CC1 Cc1nc(F)ccc1CNC(=O)CC1CCN(C(=O)CC)C1(C)C.C1CC1.O n1(CCC(=O)N)c(C)csc1=O.C1(CC)CCC(C(N2CC(O)(CC)C2)=O)C1 c1(CC(=O)N(C2CC(NC(Cc3c(C)nn(C)c3)=O)C2)C)cccc2c1OCO2 c1(-c2nc(C)[nH]n2)cccc(C(=O)NCCCNC(C2CCOC2C)=O)c1 C(CCN=c1nc(N2CC=CC2)c2ccccc2[nH]1)C1CN(C)C1 c1(CN2CC3(CN(C(=O)C=Cc4cccs4)C3)C2)cccc([N+](=O)[O-])c1F C1(F)(C(=O)NCC=CCC(=O)NC2C(C)COC2)CC=CCC1 C1(CNC(CCc2cc(C)on2)=O)CN(C(=O)C(C)(C)C)CCO1 CC1(C)CN(C(=O)CCSc2ccccc2)CC1C.c1(C(=O)N)cccc(O)n1 N1(C(C=CC(C)C)=O)CCCC(C2CCN(C(=O)C#CC3CCCCC3)C2)C1 C=CCC(C)C(=O)NC1(CF)CCN(C(c2cccc(NC(=O)OC)c2)=O)C1 C(=O)(C(CCC1CCC1)NC(C1CC2CCC2C1)=O)NC(CCOCC)C C1(C(=O)N)C2CC2C2CC12.c1(C(N(CCC)CC)=O)oc(CC(C)C)nc1C C(CCC(C)(F)F)NC(C(C1CCCCC1)NC(C1(CC=C)CCOC1)=O)=O Cc1cc(I)c(C(=O)NCCN2CCN(C(=O)C(F)(F)Cl)CC2)cc1C CC(C)CC(C(=O)NCC1CC2(CC2)CO1)ONC(C1COCC1C(F)F)=O Cc1cc(F)cnc1C(=O)NCC(C)(C)CNC(=O)CCc1ccc(F)cc1F N1(C(CC(=O)OC)=O)CCN(CC(C)NC(=O)CCN(C2CCCCC2)C)CC1 CC1(C)C(C(=O)NCc2nc(C=O)co2)C1(C)C.n1(C2CC2)cccn1.N Cc1cc(C(N2CCC2CNC(C2CSC2)=O)=O)no1 N1(C(C(C)OCC#C)=O)CC2(C1)CN(C(C1CNC(=O)CC13CCC3)=O)CCO2 Nc1cccc(Cl)c1C(=O)NCC1CCCC1NC(C1C2COCC12)=O C1(NC(C(C)N2CCC2)=O)CC2CCC(C1F)N2C(c1ccc(O)nc1)=O CC1CN(C(=O)C=C2CCOCC2)CC1(C)CNC(C1CCC=CCCC1)=O c1(C(CC)OC)ccc(C(N2CC(O)C2)=O)c(O)n1.C(=O)C=C1CCC1 N1(C(c2ccccc2CO)=O)CCCC12CCN(Cc1c(Cl)cc(Br)cc1Cl)CC2 C1(CNC(CC(=C)Br)=O)(NC(c2cccc(C)c2)=O)CCCCC1C C1(CNC(c2nncc(OC)c2)=O)CCCCN(C(=O)CC(O)C(C)C)C1 N1(C(C2N(C(CC(CCOC)(C)C)=O)CC(=O)C2)=O)CCN2CCCCC1C2 C1(N(C(c2cncc(C)n2)=O)C)CN(C(c2ccc(F)c(CO)c2)=O)CCC1C c1(C(N2CCCC(Br)C2)=O)cc2n(n1)CCCN(Cc1cc[nH]n1)C2 C1(C(=O)NC2CC(CCNC(=O)Cc3cn[nH]c3)C2)CC12CCCC2 Cc1nc(Br)sc1C(N1CCCC1CCCO)C(=O)NC1CCOC1 CCC(Cc1ccccc1)C(=O)N1CC2C(C(=O)N(C)CCNC)C2C1 C(c1ccc(C)s1)=CC(=O)N(CCC)CCNC(=O)C(O)C1CCCC1 C(=O)(C(CC(C)C(C)(C)C)N(C)Cc1cccs1)NCCOC Cc1c(C(=O)NCC2CCCCC2)sc2cncn12.C1(C=O)CN(C)C(=O)N1.N c1(CN(C(C(=O)OCCCCCC)=O)C)cccc(OC2CC2(C)C)c1 C(=O)(C1=CC2(CCOC2)C1)N1C(C(C)(C)NC(c2cncc(C)c2)=O)CCC1 N1(C(CC)=O)CCC2CC(NC(=O)CCC[N+](=O)[O-])CCC2C1 C1(NC(c2c(C)ccc(OC)c2)=O)CN(C(=O)C(O)C(C)(C)C)CC2(CC2)C1 Cc1ccc2c(c1)CCC2C(=O)NC1CN(C(c2ccc(C)c3c2CCC3)=O)C1 C(C)(C(=O)NCC1CCC(C(=O)NC(c2ccco2)C)C1)(C1CC1)OC CC(C)CC(=O)N(C(C)CCNC(=O)C(c1ccc(Cl)s1)C)C Cc1ccc(NC(=O)NC2CC(=O)N(c3cn[nH]c3)C2)cc1C Cc1cnc(NCc2cccc3c2OCC3)c(S(=O)(=O)NC2(CCF)CCC2)c1 c1(C(N(C2CCN(c3ncnc4c3nnn4C)C2)CC)=O)cc(C)c2[nH]nnc2c1 N1(CCC(=O)NC2CC2NC(C2COC(=O)O2)=O)CCCS1(=O)=O C=CCC(CNC(c1cn(C)nc1CC)=O)C(=O)N(C1CC1C1CC1)C N1(C(CC=C)=O)CC(C)(C)CC1CNC(=O)CSc1ccncc1 C1(NC(COC)=O)C(C)(C)CN(C(c2nn(C)c3c(=O)[nH]cnc23)=O)CC1(C)C C(CC(C(=O)NCC1CCSC1)NC(c1ncc[nH]1)=O)OCC c1(C(=O)NCC2CC(OC)CN2C(=O)CC(C)(C)O)ccc(Cl)c(C)c1N N1(C(c2c(CC)cncc2)=O)CCC=C(CNC(=O)Cc2cncn2C)C1 c1(NC(CCc2ccc(C3(C(N)=O)CC3)cc2)=O)cnc2ccccc2n1 C1(C2CC2)(C(=O)NCC2N(C(c3onc(CC)c3C)=O)CCC2)CCOCC1 N1(C(C(=O)NC(CC)CC)C)CCC(C)(NC(=O)CCC2CCCCC2)CC1 N1(C(C(CCSC)O)=O)CC(C)(C)CC1CNC(C1(C)CCCC1(F)F)=O C1(C(C(=O)NCCCCN(C(C(C)OCCCC)=O)CC)O)CCCCC1 c1(C(=O)NCC(C)(C2CCC2)NC(=O)CCc2nncs2)c[nH]c2cnccc12 c1(N2CCC(N(C(c3cnoc3C3CCC3)=O)CC)C2)ncc(C#N)cc1F c1(C(N2C(C)CC(COC)C2)=O)cc(O)ccc1F.C(c1cn[nH]c1)=CC=O c1(C(=O)OC)cccc2c1CCOC2C(=O)NCC(F)CNC(c1cnsn1)=O C(=O)(C(C)S(N)(=O)=O)NCC1CC(NC(CCCC#C)=O)C1 c1(OC)ncc(CNC2CCC(C(=O)Nc3ccc(Br)cc3C)CC2)cc1Br C(=O)(CC(C)(C)C)N1C(C(N(CCCNC(C(CC)N(C)C)=O)C)=O)CCC1 C1CC(F)(F)CC1.C(CC=O)OCCOCC.C(=O)C(C)=CC(C)(C)C C1(CNC(C2(c3cc(C)no3)CC2)=O)CCCN(C(=O)C)C1.c1ccncc1.S C(=O)(CCS(=O)(=O)C1CCCC1)N1CCC(NC(c2ccc(=N)[nH]n2)=O)C1 N1(C(c2nccc(OC)c2O)=O)CC2(NC(=O)CS(N)(=O)=O)CCC1CC2 N1(C(C2CC(SC)C2)=O)CC2CCC1C(CNC(C1CSCCS1)=O)C2 N1(C(c2c(NC(C)=O)scn2)=O)C(C)C2CC1C2NC(c1ccccc1C)=O C(=O)(C(F)(F)C(C)(C)O)N.C1(OC)(C)CCN(C(=O)CC)C1.C1CCCOC1 CCC(C)(CNC(=O)C(O)C1CCCC1)C(=O)NCCN1CCCC(O)C1 c1(C(N2CCCC(NC(C(C)(C)OC)=O)C2)=O)c(N)c(C)cc2c[nH]nc12 CC1CCC(O)(C(=O)NCC2CCC(C)CC2)CC1.C1(CC=O)CCCOC1.N C1CN(C(=O)CC2(C)CC2(F)F)CCCO1.c1(OCC)cncc(C(=O)N)c1 N1(C(CC(CC)C)=O)CC2OCC(NC(=O)C(c3ccc(F)c(F)c3)(C)C)C2C1 N1(C(c2cccs2)=O)CCC2(CC1)CC2C(N1CCS(=O)(=O)CC1)=O CC(F)(F)C(F)C(=O)NC1CCCN(C(=O)CC2CCC(C3CC3)O2)C1 C1(C(=O)NCC(O)CC2CCC2)CCN(C(=O)C2CC3CCC2O3)O1 C1(OC)CC(CNC(=O)CCc2cnn(C)c2)N(C(c2nocc2C)=O)C1 Cc1c(C(=O)N(C(C)CCNC(=O)C(F)OC(F)(F)F)C)cncc1N C12(NC(c3cccn4cnnc34)=O)CCCC1CN(C(=O)COC(F)(F)F)C2 c1(OC)ccc(Cl)c(Cl)c1CNC1NCC12CC2(F)F.C(c1ccccc1)=CC C(CCC(C(=O)N1CCCC1CC1CC1)NC(=O)CCNC(=O)CO)OC Cc1ccc(Br)cc1C(=O)OCC(F)C1CCC1 C(CCC(O)C(=O)NCc1nscc1Br)NC(C1CC2CC1CC2O)=O N1(C(C(C#C)(C)C)=O)CC2(CCCC2NC(=O)C(c2cc(C)ccc2C)CCl)C1 N1(C=O)CCC2(C1)NC(=O)NC2=O.C1(NC(=O)OC(C)(C)C)CCC1(C)C N1(C(CCC(C)SC)=O)CCOCC(NC(=O)COc2cccc(Cl)c2C)C1 C=Cc1cc(C(N2CCC(NC(=O)COCC3CCCC3)CC2C)=O)cc(F)c1 N1(C(c2nc(C)oc2C)=O)CCN(C(=O)C=Cc2cscn2)CC2(C)CCCC12 C1(NC(c2c(C)snn2)=O)CC2CC(NC(C3(C)COC(=O)C3)=O)CC2C1 C1(C)(C(=O)NCC(C)NC(CC=C(C)C)=O)CC=C(C)CC1 CC1CN(C(=O)C=C2CCOCC2)CC(C)C1NC(c1cnn2c1CCCC2)=O n1(CC)cc(C(=O)NC2CC(CNC(=O)Cc3conc3C)C2)nn1 C1(F)(CNC(CSSC)=O)CCN(C(c2ccn(C)c2)=O)CC1 C1(NC(Cc2ncn(C)c2)=O)COC2(C1)CN(C(=O)CN1CCC(C)(C)C1)C2 N1(C(COCCOCC#C)=O)CCC1(C)CC(=O)NCCC(=O)NC N1(C(C(C)(O)C2CC2)=O)CC=C(C(=O)N2CCC(O)C(O)C2)C1 CC1c2ccccc2CCN1N(CC1CCN(C(c2ccccc2)=O)C1)C1CC1 c1(C(=O)NCC2C(NC(=O)C=Cc3cscn3)C2)cc2c(s1)CCOC2 c1(-n2c(C(Cn3ncnn3)NCCCNS(NC)(=O)=O)nnn2)cccc(OC)c1 N1(C(CCCC(C)=O)=O)CCC(C(=O)N(C2COCC2O)C)C12CCC2 C1(C(=O)NCCCOCCC(=O)N(CCOC)CCO)CCCCC1C Cc1ccc(Br)c(CNC(C2(C)CCCN(CC3(C(F)(F)F)CC3)C2)=O)c1 CCN=c1[nH]c(C)c(C(=O)NCCN(C(=O)Cn2nccn2)C(C)C)s1 CC(C)C(C(=O)N)NC(c1ccco1)=O.C1(C)CCN(C(=O)C(O)C(C)C)C1 CN1CCC(C(N2CCC(CF)(NC(=O)CCCc3nncn3C)C2)=O)C1=O c1(N(CC(N2CC(c3ccccc3)C2)=O)C)ccccc1Br c1(CC)noc(C(=O)NCC=CC)c1C.c1(C(=O)N)cnn(C(C)C)c1Br Cc1csc(C(=O)NC2CCC(N(C)C(C34CC(C)C3C4)=O)CC2)c1C C1(NC(C(C)SC)=O)CC(CC(=O)NCc2ccc[n+]([O-])c2)C1(C)C N1(C(C2C(C)CC=CC2)=O)CC(NC(=O)CC2CCCC2)C2(CCC2)C1 C1(CC(=O)NC(CCNC(CCC)=O)C)C=NN(C)C1=O C1(NC(CC=CC)=O)CCC2CC1CN2C(=O)Cc1ccc(C)c(Br)c1 c1(C(=O)NC2CCN(C(c3nnc(C)s3)C)CC2C)c(C)nc(C(C)C)nc1C c1(C(=O)Nc2cc(C(C)=O)[nH]n2)cc(C)nc(N2CCCC2)c1[N+](=O)[O-] C(=O)(C(C)(C)C#N)NCCCC(C)NC(C(n1ncc(C)c1)C)=O N1(C(c2occ(C(N)=O)c2)=O)CC(O)CC1C1CC1.C1=CCNC1=O C=C(C)c1cn(CC(C2CCN(C(=O)C(C3CCCN(C)C3)(C)C)CC2)F)nn1 C=CCC(C)(C)CC(=O)NC1CC(NC(C2(S(N)(=O)=O)CCCC2)=O)C1 C12(CCNC(CCc3scc(C)n3)=O)CCC1CN(C(c1coc(C)n1)=O)C2 c1(NC2C(C)(C)C(CSc3ccccc3)C2)nccc2nccnc12 CC1CC(NC(=O)CO)CN1C(C1CCN(C2CC2)CC1)=O.c1ccc(F)nc1 C(N=c1c(Cl)c[nH]c2ccc(Cl)cc12)c1c(OC)ccc(Br)c1 C(=O)(C(O)CC(N)=O)NC(CC)(C)CNC(=O)C(N)=O N1(C(C2C3CC(=O)CC32)=O)Cc2occ(C(N3CCc4nn[nH]c4C3)=O)c2C1 c1(C(=O)OC)cc(NC(c2cccc(NC(c3ccnn3C)=O)c2)=O)cnc1Cl C(=O)(CCCCNC(=O)CCN(C)Cc1ccc(SC)cc1)OCC c1(C(=O)NC(C2CCCN(C(c3c(C)nsc3C)=O)C2)C)ccc2[nH]ccc2c1 c1(C(N(C2CC(NC(C(C)NC(COC)=O)=O)C2)C)=O)nocc1Cl CCCC(C#N)C(=O)NCC(CC(=O)NCCC1CCC1)OC c1(OCC(=O)NC2C(CNC(COCC(=C)C)=O)C2)cccnc1 C12(C(=O)NC(CCC)CC)C(NC(=O)Cn3nnc(C)n3)C3CC1C2C3 N1(C(c2c(C)nn(C)n2)=O)CCC(CC(=O)O)c2ccccc21 c1(C(ONC(=O)NCc2nccc(CCO)n2)=O)ccc(F)cc1 N1(C(C(C)OCCC#C)=O)CCC2(CC1)CN(C(C1(C)CCC13CCC3)=O)C2 CCCCC(=O)N1CCC(n2cc(CNC(=O)C(CN(C)C)N(C)C)nn2)C1 c1(C(C)=O)c[nH]c(C(N2CC(C(C)NC(C3CC4(CCC4)C3)=O)C2)=O)c1C N1(C(C=C(C)C(F)F)=O)CC(CNC(C2(C)CCCOC2)=O)C2(CC2)C1 N1(C(C(n2ccc(C)n2)C)=O)CCC(NC(=O)Cc2nocc2C)C1C Cc1nc2cc(C(=O)N(C3CCC(CNC(C4CCOC4)=O)CC3)C)[nH]c2s1 c1(C(=O)NCCC(CNC(=O)C=CC2CC2)O)ccccc1.c1cnccn1.O N1(C(=O)Nc2ncnc(SCC)c2Br)CCc2cc(C(=O)OC)ccc21 CCC(CC(=O)N(C)CC1CN(C(=O)C(Cl)=CCl)CC12CC2)C(C)(C)C c1(C(C(=O)NCC2CCCO2)N(CCC)CCN(C)C)csc(Br)n1 c1(C(N2CC=CC2)=O)nc2ncccn2n1.Cc1ccccc1NC(=O)C(=O)N.C c1(C(=O)NC23CCN(C(Cc4ncc(C)o4)=O)CC2C3)cc([N+](=O)[O-])cnc1C C1(C(N2CCC(N(C(=O)C(F)=CCCF)CCO)CC2)=O)CCc2ncsc2C1 N1(CC(=O)NC2(C)CN(C(C(C(C)C)n3cncn3)=O)C2)C(=O)CCCC1=O C12(COC)CCC(C(=O)N)(CC1)CO2.C1(C(N2CCC2)=O)CCCC(=O)O1 CC(C)C(CNC(=O)N)C=O.C1(C(N2CC(C)C2)=O)(N(C)C)CCCSC1 N1(C(C(CC)(C)O)=O)Cc2c([nH][nH]c2=NC(=O)c2cccc(C)c2O)C1(C)C C1(CNC(c2ncc(C)nc2)=O)CC2CCC1N(C(=O)C=C1CCCCC1)C2 O=C(NNc1ccc(Br)cc1Cl)NC1(Cc2ccccc2)CC1 CCC(COC)(CC)C(=O)NCC(C)CNC(c1cc(N)cnc1C)=O c1(C(N2CC(CCNC(C(C)n3cncn3)=O)C2)=O)cnc(C2CCCO2)s1 C12CC(CO1)N(C(c1cc(C(C)C)[nH]n1)=O)C2.Cc1nsc(C)c1C(=O)N.C C1(C(=O)NCCCC2(NC(C3N(C)CCOC3)=O)CC2)CC2CCCC(C1)C2 Cc1cnc(C(=O)NC2CC(CNC(C3(C4CCCCO4)CCC3)=O)C2)cn1 N1(C(=O)CCCCCF)CCC2CCCC12CNC(C1(O)CCCCC1)=O c1(C(N(C2CCN(C(c3c(C)snc3)=O)C2)CCO)=O)cc(F)c(F)cc1Cl N1(C(C(Cn2ccc(C)n2)C)=O)CC2=C(C1)CN(C(=O)C(C)(C)c1cnsc1)C2 C1(NC(CCNC(C)=O)=O)CC2CC1N(C(c1cc(C(F)(F)F)cnc1O)=O)C2 c1(C(=O)OC)cn(CC(=O)NCC2CC(CNC(=O)CCCF)CO2)nn1 C12(C(=O)NCC(C3CCOC3)NC(COCCC)=O)CC(CC(C)O1)C2 C1(CCC)CN(C(=O)CN(C)C(C)C)CC1NC(c1ncn(C)n1)=O C(=O)(C1CCCc2cccnc21)N1CCN(C(c2ccc(Cl)o2)=O)CC1 C(N=c1ccn(CC(=O)NCc2ccccc2Cl)c(O)n1)c1ccc(C#N)cc1 c1(OCC)ccc(Br)c2cc(C(=O)NC3CC(N4CCSCC4)C3)[nH]c12 c1(C(=O)NC(CC)CNC(C2CCC(C)(C)CO2)=O)cnn2c(=N)[nH]cnc12 N1(C(C(c2ccc(C)o2)C)=O)CCN(C(=O)CCN2CCCC2)CC(C)(F)C1 CC1CCN(C(=O)C=C(Br)Br)CC1NC(c1cnc(C2CC2)o1)=O c1(C(=O)NCC2CN3CCC2C3)n[nH]c2c1CN(C(C1CCC=CCC1)=O)C2 C1(NC(C(CC)C)=O)C(C)(C)CN(C(c2cc(C)nc(O)c2)=O)CC1(C)C c1(CC)csc(CNC(=O)C(C)CN(C(=O)COC(C)C)C)n1 n1(CC)cc(S(=O)(=O)N(C2CCCC3CC23)C2CC2)cn1 C1(NC(C2(CCCC)CC2)=O)CC2(C1)CN(C(C1CC(C)(C)CO1)=O)C2 N(C1CC2(CN(C(=O)CC3CCOC3)C2)n2ccnc21)C(c1c(C)n(C)nc1)=O c1(CCC)ccc(C(=O)NC2CC2NC(=O)C(C2CC(F)(F)C2)O)s1 C(CCN=C(NCC(C)CN1CCCCC1)N1CCCC(C)C1)SC c1(CC)ccc(F)cc1C(=O)NCC(C1CCN(C(c2cc(F)c[nH]2)=O)CC1)F CCC(C)C(O)C(=O)NCC1CN(C(c2coc(C#N)c2)=O)C1 N1(C(C2(C)N(C)CCC2)=O)CC2CCC(C1)N2C(c1n[nH]c(C(C)(C)C)n1)=O C1(CNC(C2C(CC)CCC2)=O)CN(C(=O)CCc2ccccc2Cl)CCN1C CCCS(=O)(=O)C(C)C(=O)N1CCC(C)(CNC(c2cc[n+]([O-])cc2)=O)C1 N1(C(C(C)CO)=O)CCCC2C1CCCCN2C(c1ccnc(CO)c1)=O C(=O)(C1COc2ccc(F)cc21)N1CC2C(NC(C3(OC)CCCC3)=O)(C2)C1 c1(CC)cc(C(=O)NC2CCCN(C(=O)CCOC(C)C)C2C)cn(C)c1=O c1(NC(C2N(c3cc(OC)nc(C)n3)CC(F)C2)=O)oc2ccccc2c1C CC(CNC(=O)C(C)C(F)F)C(F)C(=O)NCC(C)(C)CN=[N+]=[N-] c1(C(N2CCC(NC(C(CCCC)O)=O)C2CC)=O)coc2cc(F)cc(F)c12 c1ccc2c(c1)OC(C)(C)CC2=O.c1(OCC)ccc(C(F)(F)F)cc1.C=O.N N1(C(CCOCC#C)=O)CCC(NC(=O)C(C)=CC)CC1c1ccccc1 C(C(C)(C(N)=O)NC(=O)CCc1cn(CC2CC3CC3C2)nn1)OC CCCC(C(=O)NCC1C=CC(NC(c2c[nH]ccc2=O)=O)C1)N(C)C C1(NC)CC(F)(F)C1.C1(C(C)F)CCCN1C(=O)C1CC1 N1(CC(=O)NCC(CNC(=O)C(CO)N(C)C)OC)CCCCC1=O c1(C(=O)NC2C(NC(C(C)(O)C3CC3)=O)COC2)ccc(N=[N+]=[N-])cc1 N1(C(c2c(OC)oc(C)n2)=O)CCN(C(=O)C(F)=C2CCC2)C(C2CC2)C1 Cc1cnc(C(=O)NC2(CNC(C3CCCCS3)=O)CCOCC2)cc1C Cc1ncn(O)c1C(=O)NCC(CNC(C1CC2CCC2C1)=O)CO c1(C=O)nc(Cl)oc1C.c1(OC)cc(CN(C(=O)CC2(C)CC2)C)on1.N C1(CN(CC(=O)NC2CC2)C)CCCN1C(C1(C(N)=O)CCC1)=O S(=O)(=O)(c1ccc(B(O)O)cc1)Nc1cc2c(cc1)N(C)CCC2 c1(CC)noc(CCNC(C2(NC(=O)CC3(O)CCCC3)CCC2)=O)n1 c1(C(=O)OC)ccc(-c2cc(CN3CCCC3CCN(C)C)nn2C)c(Cl)c1 c1(C(N2CCC(C)(NC(CCCC(C)O)=O)CC2)=O)cccn2c(O)nnc12 C(C1CCCc2ccccc21)NC(c1cc(N2CCCC2)ccn1)=O C1(NC(CC2C(C)CCO2)=O)CCSC12CN(c1nc(Cl)ncc1C(N)=O)C2 c1(CC(=O)NCCCN(C(=O)CCCCCF)CC)cc(C)cc(C)c1 Cc1cc(C(=O)NCc2cc(C=O)cs2)cc(O)c1.C(CC1CC1)C1CC1 CC1(C)CCC=C(C(=O)NC2CCN(C(C3CC34CCOCC4)=O)C2)C1 c1(C(N(CC(=O)N(C(C#C)C)C)C(C)C)=O)cccc(F)c1O c1(C(N2CC(O)CC(NC(CCCSC)=O)C2)=O)cccc2ncc(C)cc12 C1(NC(C(CCO)N(C)C)=O)(CO)CCN(C(c2ocnc2C(F)F)=O)CC1 C12(C(N3CCC(C(C)NC(c4ccon4)=O)CC3)=O)CC(C(F)F)(CO1)C2 c1(C(=O)NC2(CO)CN(C(C(C)CC(N)=O)=O)C2)nccc2cccnc12 Cc1cc(C(=O)NC2CN(C(c3ccoc3)=O)CC2(F)F)c(C)cc1F C1(C(=O)NCC2CN(C(CC(C)(C)C)=O)CC2(C)C)CCCN2CCCC12 Cc1cc(CC(=O)OCC2(C#N)CCCC2)cc(F)c1 C(CNC(=O)CC(C)n1cccn1)(CCNC(=O)CCF)OCC c1(-n2cc(C(=O)OC)nn2)cccc(C(F)(F)F)c1Cl.c1(C2CC2)ccccc1Cl c1cc(C(N)=O)nn1C.C1(CC)CC1CC(=O)N(C1(CC(=O)N)CC1)C.C c1(CN(CC(C)OCC)C)cc2cccc(OC)c2o1.C1(C)C(=O)N1 c1(C(N(CCOCCCN(C(=O)Cc2csnn2)C)C)=O)ccnc(CO)c1 c1(COC)[nH]c(C(=O)NC2(CO)CCCCC2)cc1Br C1(NC(CC(C)(C)C(F)F)=O)COC2(CCN(C(C3CCC(=O)C3)=O)CC2)C1 C1(C(=O)NCC2(CC=C)CCCC2)CN(C(C2CCC(=O)CC2)=O)CC(C)O1 C1(C(=O)NCC2CCCS2)CCCN(C(c2cc(C(F)F)[nH]n2)=O)CC1 c1(C(N2CC(C)(CNC(CCSCC)=O)OCC2)=O)oc2ccccc2c1CC C#Cc1cc(C(=O)NCC2CC(CNC(=O)CCCC=C)CO2)ccc1Cl C1(C(=O)NC2(CNC(CC3N(C)C(=O)CC3)=O)CCC2)COC2COCC2O1 C#CC(C)(C)C(=O)N1CC(CNC(c2cccnc2)=O)C(C)C1 CS(=O)(=O)c1cnc2c(C(N3CCCCC3c3nc(C(=O)O)cs3)=O)cnn2c1 c1(C(C(=O)NCCCN2CCCC2)NC(CN(C2CCC2)C)=O)cnn(C)c1 Cc1cn2nc(C(N3CCOCC3CNC(C3CCC(C)C3)=O)=O)cc(C)c2n1 c1(SCC)c(OC)cccc1NC(N1CCOCC1c1cccs1)=O CC(C)C(O)C(=O)NC1(C(=O)NOCC(C)(C)O)CC1C c1(C(N(C(CC(=O)Nc2ccc(C(C)C)nc2)(C)C)C)=O)ccc2n[nH]cc2c1 N1(C(C(C(C)(C)C)N(C)C)=O)CC(NC(=O)CCC#N)C2(CCOCC2)C1 C(=O)CCC(C)C.C(=O)(CC)N(C)CC1(SC)CC1.C1CCCC1.C(=O)CO CN1CCCCC(NC(C23CCC(CN(C(c4cncs4)=O)C2)C3)=O)C1=O C1(C(N2CCN(C(Cc3c(C)cnn3C)=O)CC2C)=O)CCc2nn(C)cc2C1 C(CCCC(CO)NC(C1CC1C(=O)OC)=O)NC(CN(CCOC)C)=O c1(C(=O)NC2C(C)CN(Cc3ccccc3)CC2)cnc2scnc2c1 CC(CC(=O)OCc1cc(C2(C)CC2)n[nH]1)NC(=O)OC(C)(C)C N1(C(C2C(C#N)C2)=O)CCOCC1CCNC(=O)CCC1CCC1 C1(O)(CC(=O)NC2CC(C(C)NC(c3nc(CC)sc3)=O)C2)CCCCC1 C(=O)(C#CC1CCOC1)N1CC(C(=O)NCc2cc(C3CC3)no2)(CC)C1 C(=O)(C1=CCC(C)(C)CC1)NC(C(=O)NC(C(C)(C)O)C1CC1)(C)CO C(=O)(C(C)C(CC)CC)NCC(CC=C)NC(c1cnc(N2CCOCC2)s1)=O c1(C(=O)Nc2ccccc2)ccc(F)c(CN2CCC(O)C(F)(F)C2)c1F N=c1ccc(C(=O)NC2CC(NC(c3coc(C(F)F)n3)=O)C2)c[nH]1 N1(CCOC(=O)CN(C(=O)C)C)CCC(CC)CC1.c1ccsn1.CCO C1(C(=O)NCCCNC(C=C(COC)C)=O)CCC(C)S1 C1(NC(=O)Cc2ccc(Cl)s2)CCN(C(C2CC(=C3CCC3)C2)=O)CC1CO C1(CN(C)C(=O)NC2CC2)CN(C(C2(C)CCCNC2=O)=O)CC12CC2 N1(C(C=CC(C)(C)SC)=O)CCC(C(=O)NC)C(C)C1.c1c(C)cnn1C.C C(=O)(CC(C)(C)C)NC(CC(=O)OCC)C.C1(CC=O)CC(C)(C)CO1 N1(C(CC(C(C)C)O)=O)CC(C2CCN(C(c3ccc4nnnn4c3)=O)CC2)C1 c1(C=O)ccc(CC(C)C)cc1.CC(C(C)(C)C)=CC(=O)NC1CC1C.N N1(C(C2(C)CCC3CC3C2)=O)CC2(C=C(C(=O)N3CC(N=[N+]=[N-])C3)CO2)C1 C#CC1(N(C)C)CN(C(C2CCOC2CNC(c2ns[nH]c2=O)=O)=O)C1 CCCCC(C)CCC(=O)N1CCC(C(C)(C)NC(=O)C(CC)N(C)C)CC1 C1(NC(CCCCC)=O)CC2CCC1N(C(=O)CCCOCCOCCOC)C2 n1(CCN(C)C)ccc(C(=O)NC)n1.C1CCN(C(=O)CC2(O)CCOC2)C1 c1(OC)cccc(C(CNC(=O)C(C)c2cc[nH]n2)NC(C)=O)c1 C(=O)(C1=NOC2COCC12)N1CCCC(CCC)(NC(c2[nH]ccc2C)=O)C1 CC1CN(C(c2ccnc(C3CC3)n2)=O)CCC1NC(=O)C=CC1CCCO1 C1(CCC)CN(C(C2CCN(C(=O)CC)C2)=O)CC1.C1(C=O)CN(C(C)=O)C1 C1(C(C)(C)C)CCCCC1C(N1CC2C(NC(C3CCC(O)CC3)=O)C2C1)=O CC(C)CCC(C(=O)NCCCC1CC1)N1CCCN(C)CCC1 C(CCCCNC(=O)CNC(=O)CC1CCCC1)NC(CC1CC(C)C1)=O c1(C(=O)NC(c2cccs2)C)conc1.C(=O)CCC1CCCC1.C(N)=O.C C#Cc1ccc(CCCC(=O)NCC=CCNC(C2(C(N)=O)CC2)=O)cc1 C1CC2(CO1)CN(C(c1cnc(Cl)cn1)=O)C2.CN1CC(C)(C)CC1C(=O)N.C CC1(C(=O)NCCCOCc2ccccc2)CCN(Cc2cc(Br)c[nH]2)C1 C1(NC(COC)=O)CCCCCC1NC(C12CCC(CC1)C2)=O C(=O)(CC1CN(C)c2ccccc21)NC(C)CCNC(C1(CF)CC1)=O C(=O)(C1CCCn2cnnc21)NCC1(C)CCN(C(C2CC(O)C2)=O)CC1 CN1CCN(C(c2cncnc2)=O)CC1C(=O)NCC1(C)CCCOC1 c1(C(=O)NCCCN(C(c2c(C)cc(C)cc2O)=O)C)ccc2c(c1)C(C)CO2 C1CC(C)(C)CN1C(=O)CCCc1ncc(C)o1.C(=O)(C=CC=O)O.CC C1(N(C(c2ocnc2C(F)F)=O)CC)CCCN(C(C2CC2CF)=O)CC1 C1(C(NOCC(C)O)=O)(NC(=O)Cc2csnn2)CCN(C)C1 CP(C)(=O)COCC(=O)N(C1CC1)CC1CCCN1C(=O)CC1CCCO1 c1(NC(N)=O)ccc(C(=O)NCCC2CN(C(=O)CC3CC3)CCO2)cc1 S(=O)(=O)(c1cccc(C(=O)N)c1)Nc1c(Cl)ccc(OC)n1.C1CCCN1C.C C1(CC(=O)OC)CN(C(C)C(=O)N)C(C)(C)CO1.c1(C(C)=O)cccc(C)c1C CCC(C)CC(=O)NCCC1CCCN(C(=O)CC2CCC(=O)C2C)C1 c1(C(=O)NC2C(OC)CN(C(c3ccc(C)cc3C)=O)C2)nn(C)c2c1CCC2 CCCC(CCC)C(=O)N1CC(NC(c2cc(C(F)F)n(C)n2)=O)C(C)C1 CC1CC(NC(=O)CNS(=O)(=O)C2CC2)CN1C(c1coc(O)n1)=O N1(CC(=O)Nc2cccc(C)c2)CCC(C)(N(C)C(c2ccncc2)=O)CC1 C(c1cccnc1)=CC(N1CC(COC)(NC(=O)CCCN(C)C)C1)=O C1(C(=O)NC(C)CC2CC2)CC(O)CN1C(C1(C)CC1(C)C)=O N=c1[nH]cncc1C(=O)NC1CCN(CCNC(C2CC=CCC2)=O)CC1 c1(CCNC(c2ccc(C)s2)c2nnnn2C2(C)CC2)ccc(Cl)c(C)c1 c1(C(=O)NCCN(CCOC)C(C2CC2(C)C(C)C)=O)snc(Cl)c1Cl c1(C(=O)N)ncn(C)n1.C(C)(CC=C)NC(CNC(=O)OCC=C)=O N1(C(c2cncc(OC)n2)=O)CCC(C)C(F)(F)C1.C(=O)(CCn1ccnn1)N Cc1cc(=NC2CC3C=CCC(C3)C2)[nH]c(=NCCCN2CCC(C)CC2)[nH]1 C(=O)(C(F)CC(CC)CC)NC(COCC)C(N1CCN(C)CC(O)C1)=O CC(C(CO)NC(C1(N(C)C)CC1)=O)NC(C1(C#N)CC1)=O C=CC(C)(O)C(=O)N1CC(O)(CCNC(C2CC(=O)N(CC(C)C)C2)=O)C1 c1(CCC(N2CCCC(OCC(=O)O)C2)=O)c(F)cccc1F C1(N(C(CCC(=O)NCC)=O)C)CC2CC1N(C(c1cn(C3COC3)nn1)=O)C2 N1(C(C2=CCC(C)CC2)=O)CCCC2(CCCN2C(c2cnc3n2CCC3)=O)C1 N1(C(C)=O)CC2(C1)CN(C(=O)CN1CCC(C)C1)C2.C(COCC)OC.O c1(C(N2CCC(N(C(c3cnc(C)nc3C)=O)C)CC2)=O)cc(Cl)c(F)cc1O CN(C)NC(=O)CCC(=O)OCCOC(=O)COc1ccc(C#N)cc1Cl CN1CCC(C(=O)NC23CC(C2)N(C(C2CC(O)C2)=O)C3)C(c2ccnn2C)C1 c1(NC(C2(CNC(=O)C(CC)n3cncn3)CC(=C)C2)=O)cc(C)ccc1C CCCC(C)(O)C(=O)NCC(C)(C)CNC(c1cnn(C2CCC2)n1)=O C1(N(C(=O)Cc2cscc2F)CC)CCCN(C(=O)C(C)OCC(C)C)C1 O=C1NC2(CCSCC2)C(=O)N1Cc1noc(C2CC3CCC2CC3)n1 c1(C(=O)NCC(CNC(C(CC=CC)CC)=O)OC)snc2ccccc12 CC1(C)COCC1C.c1(C(=O)N)cc(CC)on1.c1(C=O)coc(C2CC2)n1 C(C(C)(CC(C)C)NC(C1(F)CCCC1)=O)NC(C1(CC#C)CCCO1)=O CC1C(=O)NCCN1C(C1C2CC1N(C(=O)CC1CCCSC1)C2)=O c1(NC(=O)CC2CCCN2Cc2cc(F)cc(I)c2)ccc2nc(O)cnc2c1 N1(C(=O)CSc2ccccc2)CCN(C(c2cccc(O)c2F)=O)C2CCC12 c1(C(=O)NCC2C(NC(c3c(CC)c(C)sc3)=O)C2)ccc(Cl)cc1N CS(=O)(=O)c1cccc(NNC(=O)C2(C(=O)CN3CCNC3=O)CCOCC2)c1 N1(C(C2C(OC)CCC2)=O)CC2CC(C(=O)N)C(C2)C1.c1(CC)[nH]c(C)nc1C N1(C(C2(F)CCCNC2)=O)CCOCC1c1ccccc1Br Cc1cc(C(=O)N(C(C)CCNC(=O)CCCn2cccc2)C)nn1C1CC1 Cc1c(Br)c(C)n(NC(=O)Nc2cc(F)c(N)cc2F)c(=O)c1C#N C12(C(N(CC(C)C#N)C(c3cc(O)nc(O)n3)=O)=O)CCC(CC)(CC1)C2 C1(C(=O)NC(C(C)C)(C)CO)CC2CCN(c3ncccc3C(=O)O)CC12 c12cccc(c1[N+](=O)[O-])N2.C(=O)(C(F)(F)C(F)F)N1CCN(C(C)CCO)CC1 N(C1CCCc2c(F)cc(F)cc21)C(c1nn(C)c(Cl)c1)c1nnnn1CCCl CCCCC(C(=O)N1CCC(NC(=O)Cn2cccc2)C(CO)C1)N(C)C c1(C(=O)N)cc2n(n1)CCN(C(c1cc(C(C)=O)c[nH]1)=O)C2.C1(CC)COC1 N1(C(C=CCOC)=O)CC2CCOCC2(NC(C2CC=CC2)=O)C1 C12(CNC(CCC#C)=O)COC(C1)C2.c1(C=O)cn(C)nc1C(C)(F)F.C CCC(C)CC(C)C(=O)NCC1CCC2(CN(C(C3(C=O)CCC3)=O)C2)O1.N C(=O)(C(F)C(C)CNC(c1cc(COC)on1)=O)NC(CC)(C)CC CC(C)C1=NOC(C(=O)NC2CCC(C)C2)C1.C1(C)CCOCC1.C(=O)(C)N Cc1cn2c(C)c(C(=O)NCC=CCNC(c3ccc(O)cc3C)=O)nc2s1 c1(C(C(F)F)NC(=O)NC(C#C)CC2CC2)cccc(OC)c1 C(=O)(CS(=O)(=O)CCO)NC(C(C(C)C)NC(c1cnc(O)c(Cl)c1)=O)C CN1CCc2cc(C(=O)NC3(C)CCN(C(=O)C=CS(C)=O)C3)sc2C1 c1(C(=O)NC2CC23CC(NC(C2CCCC2)=O)C3)cccc(C2CCOC2)c1 c1(C(N2CC(CC(C)NC(=O)CN3CCC(O)CC3)C2)=O)cccc2occc12 CC1CC(C)(NC(c2ccccc2)CNC(=O)OC(C)(C)C)CC(C)(C)C1 C(=O)(C1=CCCCC1)N(CCCNC(CCC1CCCN(C)C1)=O)C C1(C(=O)NC2(C(=O)NC(C#C)C)CC(O)C2)CCCCN1CC C(c1cnc(O)nc1O)=CC(=O)NCC1CCN(C(=O)C2=CCCOCC2)C1 N1(C(c2ccc(CC#N)cc2)=O)CC(NC(=O)CCc2cscn2)CC(F)(F)C1 c1(CCC(=O)NCCCN(C)C(c2n[nH]cc2F)=O)cc(Cl)cc(Cl)c1 C(c1ccc(Br)c(Cl)c1)=CC(N1CC(C)C(NC(C2CN(C)C2)=O)C1)=O C12(C(=O)NCC(C#C)C(C)C)CCCC1CCN2C(=O)C(C)C(O)C(C)C C1(C(N2CCC(NC(CCOCC#C)=O)CC2)=O)CC(C)CC(=O)N1 C(=O)(C(O)CC(F)(F)F)N.N1(C(C)=O)CC2(C1)CN(C(=O)CC1CCCC1)C2 C1(NC(N(C(C)Cc2ccccn2)C)=O)CC(=O)N(CC2CC2)C1 N1(C(CCN(CCCCC)C)=O)CC2(CNC(=O)C(C)(C)C(N)=O)CCC1C2 c1(N(C2CNCC2F)C(c2ccc3c(c2)CCC3)=O)ncc2cc(Br)cnc2n1 C(=O)(C(O)C(CCC)NC(=O)COc1cnn(C)c1)NC1(C=C)CCCC1 C1(C(CC)C)CCCCN1C(=O)C(=O)Nc1cccc(C(=O)N(C)C)c1 C1(C(N2CC(NC(=O)CCC3CCCC3)C2)=O)CCCCO1 N1(C(C=C(C)C(C)C)=O)CCCC(C(C)(O)C)C1.C12(CC=O)COC(C1)C2 C(=O)(C1=CC2(CN(C(=O)CC(C)C3CCCO3)C2)OC1)NCC(COC)(F)F c1(CC(N2CCN(C(Cc3cc(C)on3)=O)C(CO)C2)=O)c[nH]c2cnccc12 C12(C(N3CC(COC)CC3)=O)CC(C)(CN1C(=O)C=Cc1cc[nH]n1)C2 c1(C(N2C(CC)C(NC(=O)CN3CC4CC4C3)CC2)=O)snc2ccccc12 C(=O)C(C)(C)C(F)c1ccccc1.C1(C(=O)N)(NC(C)=O)CCC1.CC(C)C C(CCCCC(=O)NC1COCCN(C)C1)NC(Cc1c(CC)con1)=O CC(C)C(CNC(C1CS(=O)(=O)C1)=O)C(=O)NCCS(C)(=N)=O N1(CCC(c2nscc2Br)C)CCCOC1=O.c1(CN)nnnn1C1CCCCC1 C1(C(=O)NC(c2ccccc2)C(=O)N(CCSC)C)CC2CCCC2C1 C1(C(=O)NC2CC(NC(c3c(N)c(Cl)ncc3)=O)C2)CCOC2(CCCCC2)C1 c1(CC(=O)NC(C2CCCCC2)CNC(C(C)SC)=O)c(C)n[nH]c1C C1(NC(c2c(CC)[nH]nc2Cl)=O)CCN(C(c2ccc(F)c(F)c2)C)CC1(C)C c1(SCc2nc(CNC(CC(=O)OCCC)=O)sc2)cc(C)ccc1N c1(COCC(=O)NCCCC2CCOC2)ccccc1.C(=O)(C=O)NCC c1(C(C)=O)ccc(C(N2CCCC(CC(=O)NCC3(C)CCN(C)C3)C2)=O)nc1 c1(C(=O)N)cc2c(cc1Cl)OCO2.CC(C)CCOC(C)C(=O)N(C(C)CC)C c1(C(=O)NCCC2CCN(C(c3cc(C#N)oc3)=O)C2)ccc2c(c1)OCCC2 C1(CNC(c2n(C)ccc2)=O)CCCCN(C(c2nnn(C(C)(C)C)n2)=O)C1 C(=O)(C(O)CC(F)(F)F)NCC(c1ccccc1)CNC(C1CC=CC1)=O S(=O)(=O)(c1cccnc1NC1CC12CCOC2)NCCCCCC=C c1(C(=O)NC2CN(C(C3N(CC)CC3)=O)CC2C)nc(C2CC2)ncc1Cl CC(C)C(C(=O)N(C)CCOCCCNC(=O)CCn1cccc1)n1ccnc1 C(=O)(C(Cc1cn(CCC2CC2)nn1)NC(=O)C(c1csc(C)n1)=O)OC C1(CNC(c2cnco2)=O)COCCN(C(c2cc(-c3ccco3)on2)=O)C1 C12(C=O)CC1COC21CCC1.c1(C(N(CCC)CC)=O)c(C)coc1C(C)C C1(CNC(=O)CC2CCSCC2)CN(C(c2ccsc2Cl)=O)C2(CCC2)C1 c1(C(=O)NC2CN(C(C=C(CC)C)=O)CC23CCC3)ccc2nc(C)sc2c1 C1(CC(=O)N(CCC)C)CCCC2(CCOC2)O1.C(=O)(CC=CC(C)(C)C)N C(c1cncnc1O)=CC(=O)N.c1(C(N(C2CCCCC2)C)=O)nc(=O)n(C)[nH]1 c1(CC(C)C)ccc2cc(C(N3CCN(C(=O)CC(C)(C)O)C4CC34)=O)[nH]c2c1 C1(C(=O)NCC(CNC(COCCC=C)=O)F)CC2CCCC(C1)C2 CC1c2ccccc2OC1C(=O)NC1(C)CCCC1.C(c1cnc[nH]1)=CC(=O)N C1(C(=O)O)CCC2(CCC2)CN1C=O.C1(CCC)(C)CC1(F)F.C(C)(C)C N1(CC(=O)NCC2CN(C(COCCC(C)C)=O)C2)CCCCCC1 CC1CN(C(=O)C=Cc2nnn(C)n2)CC1NC(C1C2COCC12)=O c1(CC)nc(C)c(C(=O)N(C2CCCC(NC(=O)C(=O)N(C)C)C2)C)s1 C12(CNC(C3C(C#C)C3)=O)CCCC1N(C(c1c[nH]c(C)c(Br)c1=O)=O)CC2 c1(C(=O)NC(CC)CN(C(=O)C(O)CN2CCOCC2)C)cnn(C(C)C)c1F Cn1nnc(C(=O)NC2CC(C(=O)NC(C(N)=O)C3CCCC3)C2(C)C)c1N c1(CC)[nH]c(=N)sc1C(=O)NC(C)(C)C1CC1.C1(C(=O)N)CC=CC1 N1(C(C(c2cccnc2)NC(c2cnnc(O)c2)=O)=O)C2CCC1CC(O)C2 N1(C(COC)=O)CC2(CC(NC(=O)CCc3cncn3C)C2)C1 CC(C)CCCCC(=O)N(C1CN(C(c2cn(CCO)nn2)=O)CC1F)C c1(C(N2CC(O)CC(NC(=O)C=C(Cl)Cl)C2)=O)ccc2nccnc2n1 C1(C(N(C(C)C(=O)NC2CCN(CCCO)C2)C)=O)CCCC12CCC2 C1(C(=O)NC(CS)C)CCN(C(=O)CSCCN(C)C)C1C.CCS C(=O)(CCC#N)NC1(CN(C)C(c2cc(-c3ccccc3)ns2)=O)CC1 C1(CC)CCC(C(=O)NCC2CCCCC2NC(=O)C(c2ccnn2C)O)CC1 c1(CNC(COCC=C)=O)nc(C(=O)N(CC(O)CCC)CC)co1 C=CC(CCC)CC(=O)NCC1C=CCN1C(c1coc(C(N)=O)c1)=O O=C(CC(C(F)F)Oc1ccccc1)NC1CN(C(c2cccc(Cl)c2)=O)C1 c1(CC(N2CCCC(CN(C)C(C3CC(C)(C)C3)=O)C2)=O)ccc2occc2c1 c1(C(=O)NC(C)CN(C)CCc2ccccn2)cc2c(s1)CCOC2 N1(C(CCCCCC#N)=O)CCCC(C2CC2NC(=O)C(F)(F)CC2CC2)C1 N1(C(CCNC(=O)OCC)=O)CCC(CC)C1.C1(C)(C=O)CC=CCO1.O C1(CC=C)(C(=O)NC2(CCNC(C3CCOC3C)=O)CC2)CCCO1 C1(N(C)C(C2CC3(CCC3)C2)=O)CCN(C(=O)C2=CCCC2)CC12CC2 c1(NCCn2ncc(C(=O)NCc3cn(C)nc3)c2)ccccc1N1CCCC1 CC1(C)CCC=C1C(=O)NC1CC2CN(C(=O)C(=O)Nc3ccc(Cl)cc3)CC12 N1(c2ccnc(NCC(c3ccncc3Br)C)n2)CCC(C)=C(C)C1 N1(C(c2c(C)nsc2)=O)CCOC(C)(CNC(=O)Cc2cccc(Cl)c2F)C1 C=C(C)CC(C(=O)NOCC=C)NC(=O)CC(CC)CC N1(C(C2C(C)OCC2)=O)CC2(CCC2)CC1CNC(=O)C(F)(F)CO CC(C)C(O)CC(=O)N1CCCC(C(N2CCC(O)(C(N)=O)CC2)=O)C1C c1(CN(CC(C)NC(c2ccn(C(CC)CC)n2)=O)C)c(Br)cnn1C N1(C(C2(C(=O)NC3CC3)CC2)=O)CCCC(NC(C2CC=CCC2)=O)C1 C(=O)(CC(C)COC)NCCC(C)NC(CCCc1onc(CC)n1)=O C1(C(=O)NC(CN(C(C#CC(=O)N(C)C)=O)C)(CO)CO)CCC12CCCO2 O=C(CS(=O)C(F)(F)F)NC1CC=C(C(=O)N2CCN(CCO)CC2)C1 c1(CCCNC(CCC2C(C)=NNC2=O)=O)nc2cc(C)cc(C)c2[nH]1 N1(C(COCCCC(C)C)=O)CCN(C(C2(CF)CC2(F)F)=O)CC(C)C1 N1(C(C2(C(N(C)C)=O)CC2)=O)CCCC(O)(CCNC(=O)CCCC(F)F)C1 c1(C(=O)NCC2(OC)CN(C(c3nocc3C)=O)C2)nccc2c(C)cccc12 c1(C(=O)NC(COCC)C(=O)N)cc(C)cc(C)n1.N1(CCC)CCOCC1 C(=O)(CCCC#N)N(C(C)C(N1CC(O)C(O)C1)=O)C(C)Cc1ccccc1F C#CCCCCCCC(=O)N1CC(NC(=O)Cc2cncn2C)CCC1C C1(CC(=O)NC2(CNC(C3CCCCC3(F)F)=O)CC2)Cn2ccnc2NC1=O CCC(C)C(C(=O)NC1CCC1NC(=O)CCc1nncs1)NC(=O)OC c1(OC)ccc(Br)c(CN2CCCC(CC(=O)NC3CC(S(C)(=O)=O)C3)C2)c1 Cc1cncc(C(=O)NC(C2CC(NC(=O)C(C)NC=O)C2)C)c1 n1(CC(=O)NC2C(NC(c3cnc(C)s3)=O)CC2)[nH]cc2c(=O)ncnc1-2 C=C1CCC(C(=O)NCC2(F)CCC(NC(=O)C(CCO)N(C)C)C2)CC1 C(=O)(C(O)CC(N)=O)NCc1ncc(C(=O)NCC2(C)CCOC2)cn1 N1(CCC)CCCC(C(=O)NCCC2CCCN2C(C2CS(=O)(=O)C2)=O)C1 c1(CCC(N2CC(CC(C)NC(=O)CCN3CCCC3)C2)=O)ccc(=N)[nH]c1 c1(C(=O)NC(C(C)(C)NC(C(CC(C)C)OC)=O)C)cc2c(ncn2C)s1 C1(C)(CNC(C2C(C)C(=O)C2)=O)CCCN1C(=O)CC1CCC(C)CO1 CC1(C(=O)NCC(O)CNC(=O)CN2CCCNC2=O)CCCCCCC1 CCC(O)C(C)C(=O)N(CCC(C(C)(C)C)NC(=O)Cn1nc(C)c(C)c1C)C C1(CNC(C(F)=CC)=O)CCCCCN1C(=O)CCCc1sccc1C CN(O)C(=O)CNC(c1nnnn1CC1CCOCC1)CCc1cccnc1 N1(C(C(=O)Nc2c(OC)cccc2)C)CCOC(C)(C(C)C)C1 N1(CC)CCN(CC(=O)NCC2CCCCN2C(=O)C(C)C=O)C(=O)C1=O.O C1(C(N(C2CCN(C(=O)CC3CCCOC3)C2)CC#C)=O)COCC(C)O1 C12(C(N3C(CC)CCC3)=O)CC(CO)(CN1C(=O)CC1CC(O)C1(C)C)C2 C(=O)(C(C)(C)C(=O)N)NC.C1(CC)CCCN(C(c2sccc2C2CC2)=O)C1 N1(CC(=O)NC(=O)CC(C)C2CC2)CCCCC1=O.C(CC)N(CC)CC c1(OCCN2C(C(CC)O)CCC2)ccnc(C(C)C)c1 C(=O)(C(C)(C)CCF)NC(C(=O)NCc1cnc(C)[nH]1)Cc1cn[nH]c1 c1(N2CCN(c3snc(C)n3)CC2)nc(NCCSC)nc2c1CCCCC2 c1(C=O)c[nH]c2c(Cl)cccc12.c1(C(=O)NCC2CCC2)sccc1C(F)F C1(C(=O)NCCC2OCCN(C(Cc3ccn(CC)n3)=O)C2)CC(C(C)C)=NO1 C12(C(=O)NCC3N(C(=O)CSc4ccccc4)CC3)CCC(CO1)C2 C(CN=c1[nH]cnc(CC)c1F)(C1CCCC1)NC(C1C(C)=C1)=O C=CCC(F)(F)C(=O)NC1CN(C(=O)C(O)CCSC)C(CC)(CC)C1 C1(NC(c2c(C)n(C)nc2)=O)CCC2(CCN(C(=O)C(C)(F)C(C)(C)F)CC2)C1 c1(NCC(CCCOC)C)cc(=NCC2CC2(F)F)[nH]cn1 CCC(C)C(O)C(C)C(=O)N1CCC(N=[N+]=[N-])(C(=O)N)C1.C(O)(C(C)C)C1CC1 c1(-c2nc(C)on2)ccc(C(=O)NC2(C)CN(C(=O)CC3CCC(C)O3)C2)cc1 c1(C(N2CC(C)C(NC(C3CCCCC3)=O)C2)=O)cc2ccc(F)cc2s1 Cc1cn2cc(C(=O)NC3CN(C(c4cccc(C(F)(F)F)c4F)=O)C3)sc2n1 CC1(C)CC(NC(=O)Cc2cnoc2)CN(C(=O)C(F)(F)CCn2cccn2)C1 Cc1ccc(C(N2CCC(C(=O)Nc3ccc(Br)cc3CO)C(O)C2)=O)c(O)c1 N1(C(C(C)(C)F)=O)CCC2(C1)CN(C(=O)CCOc1ccc(Cl)cc1)CCO2 C(=O)(C1=CCCCC1C)NCC(CCC)C(=O)N1CC(C)C(C)(CO)C1 C(C1NC(=O)c2ccccc21)OC(C1(CCC(C)(C)C)CCOCC1)=O Cc1nocc1C(=O)NCC(C)(O)CNC(=O)C(C1CCCCC1)C Cc1n[nH]c(C)c1C(=O)NCC1C(C)CCN1C(c1ncccn1)=O c1(C(N2CC(C(C)NC(=O)C(C)(O)c3ccccc3)C2)=O)ncncc1Br c1(OC)cncnc1C(N1CCCCC1Cn1cc(C(O)C(C)(C)C)nn1)=O C(=O)(C(F)(F)c1nccs1)NCC(C)N(C)C(c1ccc(CO)o1)=O Cc1cnc2c(C(=O)NCCCCNC(C3CC4C(C3)C4(C)C)=O)cccn12 N1(CC)CCN(N2CC(N3C(=O)NC(C)(c4ccccc4)C3=O)CC(F)(F)C2)CC1 C12(C(=O)NCC3CCN3C(=O)Cc3cccnc3F)CCCN(CC1)C2 S(=O)(=O)(c1ccc(NCC(O)C(C)c2cccs2)c(Cl)c1)N1CCN(CC)CC1 C(=O)C(C)(C)C(N)=O.Cc1nc(C)c(C(N2CC(C)C(C(F)(F)F)C2)=O)s1 C1(NC(c2cn(CC)nc2C)=O)CC12CCN(C(=O)CCC1CCCO1)CC2 CC1=NOC(C(=O)NC(C2CCCN2C(c2nocc2Cl)=O)C)C1 C=CCCC(=O)NCC1CC(NC(=O)CC(C)F)C1 c1(C(N2CCC(F)C2)=O)cc(F)c(Cl)cc1F.c1(OCC)nc(C(=O)N)co1 C(=O)(C=C1SCC(=O)N1C)N.CC(C)CCCNC(=O)C(=O)NCCC(N)=O n1(COCC)nc(C)c(CC=O)c1C.C1(C(N(CC(C)O)C)=O)C2COCC12.N C(=O)(C(C#N)C(C)(C)C)NC1C(C(=O)NC(CCSCC)C)CC1 c1(C(c2n(CCC)nnn2)NC(Cc2ncnn2C)C(N)=O)cnc(C)cn1 c1(C(=O)NCC(C)CNC(=O)C(C)S(C)(=O)=O)ccc2c(c1)CN(C)C2 c1(NC(C(C)NC(C)(C)C)=O)cc(Cl)ccc1C(F)(F)F Cc1ccc(S(=O)(=O)NCc2c[nH]c3cccc(C(C4CCOCC4)=O)c23)cc1Br N1(C(C2N(C(=O)NC(C)C)CCC2)=O)CC2CCC1CN2C(C1(C)CC1F)=O C(=O)(C(C)N=[N+]=[N-])N(C1CCN(C(c2cc(Cl)cn2CC)=O)CC1)CC c1(C(=O)OC)c(OC)cc(NCc2ccc(C(=O)OC)cc2)cc1Br N1(C(C2CCC(C)(C)C2)=O)CCN(C(c2cc(O)cs2)=O)CC2(CC2)C1 N1(C(c2cnc(-c3cccs3)o2)=O)CCCC12CCN(C(C13CC1C3)=O)C2 CN1CCN(CCNC(C2(C)CCN2C(=O)Cn2cc(Br)cn2)=O)CC1 C(c1c(Cl)cccc1Cl)=CC(N1CCC(NC(Cc2nc(CC)sc2)=O)C1)=O N1(C(CC(=O)NC)=O)C2CCC1C(C)C2.C(=O)(C(C)CCc1cccc(F)c1)N C1(C(=O)NC(c2cncc(OCC(F)F)c2)C)C=CS(=O)(=O)C1 CCC(C(=O)NCCN(CC(C)O)C(c1cccc(N(C)C)c1)=O)C(F)(F)F C1(CNC(C2(C=C)CC2)=O)CN(C(=O)CCc2nc(=N)[nH][nH]2)CC12CC2 c1(C(C)O)ccc(Br)cc1NC(C1CN(C(c2ccccc2)=O)CCO1)=O c1(C(C)=O)cc(Br)ccc1CSc1nc(CCC2CC2)cs1 CC1SCCCC1C(N1CC(C)(C(=O)NC2(CO)CCSC2)C1)=O N(C1CCc2cccnc21)C(CCN(C)C(C1CCNC(=O)C1)=O)=O N1(C(CC(=O)NCC#C)=O)CCCC(F)(F)CC1.C1(C=O)CCC2(CC1)CC2.N C1(CC(=O)NCC(C)CNC(=O)C(C2CC2)N(C)C)CN2CCN1CC2 CC1(F)CCN(C(=NCc2cc(F)ccc2F)NC2CCS(=O)(=O)C2)C1 N1(C(c2c(C)nc(CCC)s2)=O)CCC2(CCCN2C(c2cc(CC)no2)=O)C1 N1(CC)CCC(CNC(N2CCCCC2)=O)CC1.C(=O)(C(F)(F)CNC)N CC1CC2CN(C(C3C(O)CCN3C(=O)C=CCN3CCC3)=O)CC12 CCC(CN(C)C)C(=O)N(C(C)CNC(=O)CCN1CCCC1)C CCC(CC)CC(=O)NC1CCCC1NC(=O)CC1(c2ccccc2)CCCO1 c1(C(=O)NC(CCNC(C(c2c(OC)cccc2)O)=O)C)ncc(C)cc1F c1(C(=O)NCC(CC)NC(=O)Cc2sccc2C)cnn(C)c1C1CC1 c1(C(=O)NC2C3(CN(C(CNC=O)=O)C3)CCC2)cc2ccc(Br)cc2[nH]1 N1(c2c(C)cncn2)CCC=C(C(=O)NCc2ccc(F)c(O)c2F)C1 C1(CNC(c2cc(C)nc(C)c2)=O)CN(C(=O)Cc2cnc[nH]2)C2(CCC2)C1 C1(O)(CNC(C(C)S)=O)CCN(C(c2cc(C(F)(F)F)nc(Cl)c2)=O)CC1 C1(C(=O)NC(CC=C)(C)C)CN(C(=O)CC23CCCC2C3)CCN1C c1(C(N2CCCC(C)(NC(C(COC)OC)=O)C2)=O)ccc(C)c2cccnc12 c1(OC)cc(CCC(=O)NCC2(C)CCC2)ccc1O.n1(CC=O)ccnn1.N CC(C)C(C)(C)C(=O)N1CCC(CO)C1.C1(C=O)CSCN1C(C1CCC1)=O.N C1(C(=O)NCC2N(C(C3CC(C)OC(C)C3)=O)CCC2)Cc2cc(F)ccc2O1 c1(CC)cc(C(=O)NC2CC(C)(NC(=O)CSC(C)C)C2)ccc1Cl C1(CC=C)(C(=O)NCc2ccc[nH]2)CCN(C(=O)CC(O)CC)C1 c1(C(=O)NCc2c(C(N(CCCCC(C)C)C)=O)occ2)cccc(F)c1O CCC(C(=O)N1CCN(C2CCN(C(=O)C(C)=C3CCC3)C2)CC1)C(C)(F)F N1(C(Cc2ccn(CC)n2)=O)CCC(C)(C)C1CC(N1CCCC(C)(OC)C1)=O CCCCC(C(=O)N(C)CC1CCSC1)NC(=O)CCOCCC Cc1cc(C(N2CCC(N(C(=O)COCC3CCC3)C)C2)=O)c(C)s1 C1(C#N)(C(N2CC(C(C)NC(=O)Cc3cc(Br)cs3)C2)=O)CC2CC2C1 c1(NCCN(C2CCCCCC2)C(CC(=O)N(C)C)=O)cc(Cl)cc(Cl)n1 CC1(NC(c2cc(C3CCCCC3)[nH]n2)=O)CCN(C(=O)Cn2cccn2)C1 c1(C(N2CCC(c3cn(CC(CC)O)nn3)CC2)=O)cccc(OC2CC2)c1F CC1CCN(C(=O)C=CSCc2ccco2)C1C.C1(C)(CC=O)CCCCC1.N C1(C2(NC(=O)C(C)CNC(=O)CCCCN(C)C)CC2)(OC)CCC1 C#CC1CCCCCC1.C1(CC=O)CC(C)(C)CN1C(C1C(C)(C)C1(F)F)=O.N c1(CC)c(C)noc1C.C1(C)(CC)CC(C(=O)NCc2cc(C=O)on2)C1 C(c1ccc(Cl)s1)=CC(=O)NC1(CC=C)CN(C(c2cnc(C)o2)=O)C1 N1(C(Cc2cnc(C)o2)=O)CC2CC(C1)N(C(c1ccc(CCO)cc1)=O)C2 c1(CC(N2C(CC)CN(C(C3CCCOC3)=O)CC2)=O)ccc2ccoc2c1 CCC(O)C(C)(C)C(=O)N1CCCC1CN(C)C(c1cc(N)c(O)c(F)c1)=O C1(C)(CNC(NCc2n(CCC)nnn2)=NCCCSC)Cc2ccccc2C1 C1(C(N2C(CNC(C3C(C=C)C3)=O)CC2)=O)COc2ccc(O)cc2O1 N=c1ncc(C(N2CCN(C3CN(C(C4(Cl)CC4)=O)C3)CC2)=O)c[nH]1 N1(C(c2ccc(C)cc2Cl)=O)CC2(CCCN(C(C3(C)CS(=O)(=O)C3)=O)C2)C1 O=C(Cc1nc2ccccc2[nH]1)NNc1ccccc1-c1nccn1CCF c1(CCC)cc(C(=O)N(CC)CC2CCCN2C(C2CCC=CO2)=O)n[nH]1 c1(C(=O)NCCN(CCOC)C(C2CCCC2C)=O)cc(Cl)cc(C)c1.O C#CC(CNC(=O)C(C)(C1CCC1)NC(c1cc[nH]n1)=O)CC CC(N=c1ccc(Br)c(S(=O)(=O)N2CCCOCC2)[nH]1)c1ccns1 C1(CC)CCCCCC1(c1nnnn1C1COC1)NCCOc1ncccc1Br N1(C(c2c(C(F)(F)F)nc(C)o2)=O)CCC2(COC2)C1.c1(CC=O)cscn1.N Cc1ccsc1CCCC(=O)NCC(C)(C)CNC(=O)CN(C1CCSC1)C C(C(CC(=O)NCCN1CC(=O)NC1=O)C1CCC1)NC(C(C)NC=O)=O CCN=C(NCC1(C2CCC2)CC1)NC1CCC(NS(C)(=O)=O)CC1 n1(CC(=O)Nc2cc(CCC)[nH]n2)ncc2cc(Br)ccc2c1=O C(=O)(CC(CN(C)C)CC)NC(CC)CN(C)C(c1cn(C2CC2)cn1)=O n1(CC(=O)NCC2CC3CCC2N3C(C2CC(=O)C2)=O)cnc2ccccc12 N1(C(CCNC(=O)NC)=O)CC2CC(NC(=O)CC(F)(F)F)CC2C1 CN1N=CC(CC(N2CC3C(CNC(c4ccnc(S)c4)=O)C3C2)=O)C1=O C12(C(N3CCCC(N(C(c4cc(O)cs4)=O)CC)C3)=O)CC(C)(CCO1)C2 C1C=CCN1C(c1cnn(CCO)c1)=O.c1(C(=O)NC)cnn(-c2nccs2)c1 Cc1cc(O)ccc1CC(=O)NC1CCCC1C.c1(C(=O)N)c(Cl)nn(C)c1Cl C(CCC(N)=O)C=O.C1CCC(=O)N1.CC1CC(C(=O)NC2(CO)CCC2)C1.N C1(NC(CCN2C(C)CCCC2)=O)CCN(C(c2ncccn2)=O)CC1F C1(CNC(CCCC#CC)=O)C(C2CC2)CCN1C(=O)CCS(C)(=O)=O c1(C(N(C2CN(C(c3c(C)occ3)=O)CC2O)C)=O)ccc2c(c1)C(C)(C)CO2 c1(C(N2CCC(O)(CCNC(C(CC)NC(N)=O)=O)C2)=O)cc(O)cc[n+]1[O-] C(=O)(CCCC(=O)NCC1(F)CN(C(=O)CC2(N(C)C)CCC2)C1)N(C)C C(=O)(C(CC(N)=O)NC(=O)CCCN1CCCC1)N(C1CCN(CC)C1)C C1(C(=O)NC2(CCC(=O)NCC3(OC)CCC3)CCCC2)COCCN1C Cc1c(C(=O)NC2CCC23CN(C(c2ccn(C)n2)=O)C3)oc2ccc(Cl)cc12 N1(CC)CCN(C(=O)C(COC)NC(C2CCCCC2O)=O)C(C)C1 C(C(=O)NCC)(C(C)C)OCC.C1CCN(C(=O)C(F)(F)C2CC2)CC1.O CC(C)CCCNC(C1(O)CCC1)=O.c1(CCC(=O)N)nc(-c2cccs2)no1 C1(NC(C=C(CCC)C)=O)CC(O)CN(C(=O)C2=COCC2)C1 Cc1c(F)cc(CN(C(C)Cc2cc3ncccc3s2)C)cc1F CCC(C)(C#N)C(=O)NC1CC(CCNC(=O)C=Cc2cncc(F)c2)C1 C1(C=O)CCN(C(C2CCN2C2CCCC2)=O)C1.C1(CC=CC)CCCC1O.N c1(N2CCC(N(CC#C)C(C3CC4(C3)CC4F)=O)CC2)ncnc2c1cnn2CC C1(NC(CC2(C(=C)F)CCC2)=O)COC2(C1)CN(C(=O)CC1(C)CCCO1)C2 N1(C(C2=C(C)OCC2)=O)Cc2nnn(C3CC3)c2C(C(=O)N2CCCC2C#N)C1 c1(CCC(N2C(CCCNC(C(OC)OC)=O)CCC2)=O)cc(F)cc(F)c1 N1(C(c2ccc(CC)s2)=O)CCC(NC(C2CC3CCC2CC3)=O)C(F)(F)CC1 CON(CCC(=O)NC1(C(N)=O)CCCC1)C(=O)C(O)c1ccnn1C c1(C(N2CC(NC(C(CCC)C)=O)C(C)C2)=O)cc2c(OC(C)=O)cccc2s1 O=C1CN(NC(=O)c2ccc(-c3ccc(Cl)s3)cn2)C(=O)N1 c1(C(=O)NCC2N(C(CCC(CC)C)=O)CCC2)cc2c(ccn2C)s1 C1(C(=O)NC2CN(C(C(=O)OCC)=O)C2)CCCC1c1ccccc1 c1(C(=O)NC2C(NC(CC3CCC(=O)N3)=O)C2)ccc(-n2cncn2)cc1 C1(C(C)C)CN(C(=O)CCCC2CC2)CCN1C(=O)CC1(N(C)C)COC1 N1(C(C=C(COC)C)=O)CCC2C(C(=O)NCC3CCCC34CCC4)C2C1 c1(C(N(CCN(C(CC(CCC)CC)=O)C)C)=O)nc2nc(C)ccn2n1 N1(C(Cc2scc(C(=O)OCC)c2)=O)CCCCC1C1CC1.C(=O)(C=O)N Cc1nc(CN(C)CC2CCCN(C(=O)CCC3CC(C)(C)CO3)C2)sc1C N1(CCC(=O)Nc2cccc(CNC(=O)C)c2)CCCS1(=O)=O.c1cn[nH]c1 C1(O)(CNC(CC(CC)(C)C)=O)CCCN(C(=O)C(C2CC2)OC)CC1 N1(c2ccnc(COC)n2)CCC2CCC(C1)N2C(C1(C)CC1Br)=O CC(C)C(C(=O)NC1CCC(NC(=O)C)CC1)NC(N)=O.c1nnc(S)s1 c1(C(N2C3CC(NC(=O)C=CCF)CC2CC3)=O)cnn2cccc(F)c12 C1(C=O)CC2(C1)CC2(F)F.C(C(C)(C)C=O)N(C)C=O.CCC(C)(C)CO.C C=C=CCC(=O)NCc1cn(C2CCN(C(=O)C(=O)NC(C)C)C2)nn1 c1(CCNC(c2n(CCOCC)nnn2)(C2CCCCO2)CC)ccc(Cl)nc1 CC(C(C)(C)C)=CC(=O)NCCCC(=O)N(CC(C)C)C C(=O)(C(C)CC(C)(C)C)NCC(C(=O)NCCC(C)O)C C1(C(N(C2CCN(C(=O)C=C(C)C)C2)CC)=O)(COC)CCOCC1 N1(C(CC(=C=C)C)=O)CC(CNC(c2nc(C)ccc2Br)=O)CCC1C c1(C(=O)NC2(CNC(C(N3CCNC3=O)C)=O)CC2)ccc2c(n1)CCC2 C1CN(C(=O)Cn2ccnn2)CCC1(F)F.n1(CC)nccc1C=CC(=O)NC c1(C(N2CCC(O)(CNC(C(CC#C)C)=O)C2)=O)cc2ccccc2nc1O C=CC1CCN(C(=O)C=CCNC(=O)CC2CCC(O)C2)CC1 CC(CN(C)C(C1CCCN1c1cnccn1)=O)N=c1[nH]nc(C2CC2)o1 c1(OCCC(=O)NC2CCC(O)CC2)ccc(F)c(F)c1F c1(NC(c2c(F)cccc2Br)C)[nH]c(=NC2CCC(=O)N(C)C2)nc2c1ncn2C C1(CNC(C(CC=CC)C)=O)(NC(=O)C(=O)NCC)CCCCCC1.O Cc1ccc(C(N2CC(F)CC2CNC(C2(C#N)CC2(C)C)=O)=O)nc1O C1(C(=O)N)CCC(C2CC2)C1.C1(CCC(=O)NC(c2nc[nH]n2)CC)CCCC1 C1CC2CC(C1)N(C(=O)CCCc1ccccn1)C2.CC(C(=O)N)OCC1CC1 c1(CNC(C2N(C(C(c3ccccc3)C)=O)CC(O)C2)=O)cnn2c1CCCC2 c1(C(=O)NC(CNC(C=C(CC)CC)=O)C(C)C)ccc(-n2cnnc2C)cc1 c1(C(N2CCC(N(C(c3scc(OC)c3)=O)C)C2)=O)cc(C)c(C(=O)OC)o1 C=CC(CC)C(=O)NNC(=O)C(C)(C)CCCCNC(=O)C(CC1CCCC1)CC Cc1ccc2c(c1)CC(C(N1CC(N3CCOCC3)C(O)C1)=O)O2 N1(C(C2(CF)CC(=O)C2)=O)CC2CC2(CNC(=O)C(O)Cn2cncn2)C1 C1(C(=O)OC)C(CNC(=O)NC(C)CS(C)=O)C1(F)F CCC(CNC(=O)CC(CNC(C1CC1(C)C(F)F)=O)OC)C(C)(F)F CC1=C(C)CC(C(=O)NCC=CCNC(c2coc(C3CC3)n2)=O)CC1 CC1C(C)N(C(=O)COCCF)CCN1C(=O)CCNc1ncccn1 C1(CC(=O)NCC(C)NC(c2ccoc2C2CC2)=O)CN(C)CC1O Cc1cnc(C(N2CCCC2C(N2CC(F)C(F)C2)=O)=O)cc1Br c1(C(=O)NC2CCC(NC(=O)CN3C(=O)CSC3=S)C2)cc(Br)c(Cl)cc1F CC(CN=c1[nH]c(=NCCCOC(F)(F)F)c2cc(Cl)ccc2[nH]1)C1CC1 Cn1c(C(N2CC3OCC(NC(C4CC4CF)=O)C3C2)=O)cc2occc12 C1(CCNC(c2ccn(C3CCCC3)n2)=O)CCN(C(=O)C(F)(F)CF)CC1 CC#N.N#CCSC(=O)CC1CC1C(F)(F)F c1(C(N2CCC(N(C(=O)C=CI)CC)C2)=O)cccnc1CO n1(CC(N2CC(OC)(CNC(=O)CN3CCCC3C)C2)=O)cnccc1=O C(C(O)C(F)(F)F)N(C(c1ccccn1)C)C(C)=O.CC(O)CO C1(C#N)(C(N(CC(C)NC(c2sc3sccc3c2Cl)=O)C)=O)CC12CCCC2 CC(C)CC(C)CC(=O)NCC1(NC(=O)C=Cc2cnc[nH]2)CCCC1 N1(C(CCC#CC)=O)CCC=C(C(=O)N(CC(N)=O)CC(C)C)C1 C(N=c1[nH]cnc(Cl)c1Br)C1(F)CC(NC(c2c(OC)nc(C)cc2)=O)C1 c1(C(N2CCCC(NC(CC(CC)SC)=O)C2C)=O)cc2cccnn2n1 CC1(C)C2CCC1(C(=O)NCC(CC(=O)NC(C)(CO)C(F)F)C1CCC1)C2 C1(NC(C(C)O)=O)CCCCC12CCN(C(c1ccc(C(F)F)cc1F)=O)CC2 c1cn(CCNC(=O)COCC2CCC2)nn1.c1(C(=O)N)cnc(F)s1 c1(C=O)cccc2c1CCN2.Cc1cnn(C(C)C)c1C(=O)NCC1CCC1.N C(=O)(C1CCCc2nn(C)cc21)NC(C1(O)CCN(C(=O)C=CCO)C1)C N1(c2c(C(C)=O)c(Cl)ncn2)Cc2nccn2CC(NC(C2CC2(C)C)=O)C1 C1CN(C(=O)C=CC(=O)N)CCCO1.C1(C(=O)NC2CC2)(OC)CCSC1 Cc1ccn2nc(C(=O)NC(C)(C)C(C)NC(=O)CSc3nncs3)nc2n1 C1(CN(C)C(c2c[nH]nc2-c2ccn(C)n2)=O)CCCN1C(=O)C=CBr N1(C(c2cc(C)nn2CCO)=O)CC2CC(NC(=O)C=Cc3cnc[nH]3)C(C2)C1 N1(C(C(C)(C)OC)=O)CCC2C(NC(c3conc3-c3ccccc3)=O)C2CC1 Cc1cc(C(=O)NC(C2CCCN2C(c2ncn(C)c2C)=O)C)n(C2CCC2)n1 N1(C(C(F)=C(C)C)=O)CCN(C(c2cnc(-c3cnn(C)c3)s2)=O)C(C(F)F)C1 N1(C(C(CO)OC)=O)C2CCC(C2)C1CC(=O)NCCCSCCO CCC(CC)C(F)C(=O)NCCCCC(=O)NC(C(N)=O)C1CC1 C1(CCC(=O)NC(CCOC)CO)CCCN(C(c2ccccc2O)=O)C1 C(CCC(=O)NCC1CC1(F)F)N(C)C(C1(C)C=CCC1)=O CC(Cc1cnn(C)c1)C(=O)N.C(=O)(C(C)Cn1cccn1)N(CCC)CCO C1(CNC(c2ccccc2F)c2n(C)nnn2)CCC(Cn2ccnc2)CC1 c1(C(N(CC(C)(C)NC(COC)=O)C)=O)cc2c(=O)[nH]ccn2n1 CCC(C)(C)C(O)C(=O)NCC(C1CCCC1)NC(C1CCC(=O)N1C)=O N(C)(C1CCc2c(F)cccc21)C(c1ccc(OC)nc1C)C(=O)NC(CC)C C1(N(C(CCC=C(C)C)=O)C)CN(C(=O)CCN2CCCC2)CCC1O C1(CNC(Cc2nc(C)c(C)o2)=O)CC2CCCC2N1C(=O)C(C)SC(C)C c1(CC)cc(C(=O)NC(COC)C(=O)N)c(C)o1.C1(CC)CC(F)(F)C1 N(C1CN(C(c2ccns2)=O)CCc2ccccc21)C(c1c(C#C)cn(C)n1)=O C1(C(N(CCC)C)=O)CC(=O)N(C2CN(C)C2)C1.c1(C(=O)N)c[nH]c(=N)s1 Cc1cc(=NC(=O)C(=O)NC2CCC(CNC(c3ccoc3)=O)C2)[nH]o1 S(=O)(=O)(c1ccc(N2CC3CCCC(C2)N3C)c(Cl)c1)N(CC(CC)C)C CC(C)CCC(=O)NC(C)C1CC1.C(=O)CC1CC1.C(C)(C)C.C=O.N C1(C(=O)NCCc2c(C)nc[nH]2)C(O)CCN1C(=O)C(C)NC(N)=O C1(C(C)NC(c2cnc(C)s2)=O)CN(C(C2(Cl)CC2)=O)CCO1 CN=c1[nH]c(C(=O)NCC2CC(C)N(C(c3csc(-c4nc[nH]n4)n3)=O)C2)cs1 C(=O)(CC(C(C)C)C(C)C)N1C(CN(C(c2cncc(C)c2C)=O)C)COCC1 C(=O)(C1c2c[nH]nc2CN1C(c1nonc1C)=O)Nc1ccc(C)c(C)c1C c1(C(N2C(CNC(CSSC)=O)CC2)=O)cnn(CCC#N)c1C N1(C(C(C)O)=O)CCC(C)(CCNC(=O)CC2(C(F)(F)F)CC2)C1 C1(NC(CC)=O)C2CC1N(C(=O)CCc1nc[nH]n1)C2 N1(C(c2cnc(Cl)c(F)c2)=O)CCC2C(CCN2C(c2cnc(Cl)c(Br)c2)=O)C1 c1(C(=O)NC2CCN(C(C(CCC)O)=O)C2)cnc(C(F)(F)F)cc1C CCCC(C(=O)N1CC2CC(NC(c3ccc4ccnn4c3)=O)C2C1)C(C)C c1(CC=O)cccc(F)c1Cl.C1(O)(C(C)(C)C)CN(C(=O)C(C)(C)C2CC2)C1 CC1(C)CN(C(=O)CNC(C2CC2)=O)CC1C(=O)NC1C(O)CC1O C1(CCNC(CC2(C)CC2)=O)COCCO1.C12(CCC1)CC=CC(=O)N2 CCC(CCC(=O)N1CC(F)(F)CC1C(=O)NC(c1ccc(F)cc1)C)OC c1(C(C)C)cnn(C)c1C(=O)NC1CCCC1CNC(=O)C(C)O C(=O)(C1CC=Cc2ccccc21)N1C2CN(C(c3c(C(C)C)onc3)=O)C(C2)C1 C1(C(=O)NCCC[Si](C)(C)C)CC2CCCC2N1C(=O)C(F)OC(F)(F)F c1(C(N(C(CNC(C2(OC)CCSC2)=O)C2CC2)C)=O)cnn2cccnc12 CC1C(=O)N(C)CCN1C(=O)CCn1cc(C(c2ccc(F)cc2)O)nn1 c1(C(=O)NC2C(CNC(=O)Cn3cnnc3)CC2)ccc2nc[nH]c2n1 C1(NC(c2c(SC)cccn2)=O)COCCN(c2nnc(C3CCCC3)s2)C1 Cc1ncc(CC(=O)NC2CC(C)(C(=O)NCC(C)Cc3cn[nH]c3)C2)s1 C(C)(N=c1cnc(F)c[nH]1)C1OCCN(C(C(c2ccc(OC)cc2)(C)C)=O)C1 C=CC(C)(CCOC)C(=O)NCCNC(=O)CS(=O)(=O)CCOC C1(F)(C(=O)OC)CCN(C(C23CCC(OC)C2C3)=O)C1 C1(C(=O)NC2C(CNC(c3ccc(N)cc3Cl)=O)CCC2)CCn2nnnc2C1 Cc1oc(S(=O)(=O)N(C)C)cc1C(=O)NC1(C)CCCCCC1.C(=O)C.N CC1CCN(C(c2cccnc2O)=O)CCN1C(c1ccnc(C2CC2)n1)=O c1(C(N2C3(CNC(C(C(CC)C)OC)=O)CC(C2)C3)=O)ccc2ncsc2c1 CC(C)CC(C)(O)C(=O)NCC1(O)CCCN(C(=O)Cc2cnc[nH]2)C1 C(=O)(CC(C)C(=O)N1CC(C(N2CCC(c3ncc[nH]3)C2)=O)C(F)(F)C1)OC C1(CC(=O)OCC)CCCCN1C(=O)C(n1ccnn1)C.c1(C)sc(C)cc1C N1(C(CCCNC(=O)OCC)=O)CC2CC(NC(C3(O)CCSC3)=O)C1C2 C1(C#CC(=O)NCC2CCN(C(C3CCCN3C=O)=O)CC2C)(CC)COC1 C1(CC)CCCN(C(C2C3CCC(C3)N2C(=O)C(C)(C)SC)=O)CC1 c1(OC)cccc(C2CCCN2C(=O)C(N2CCC(CCCO)C2)=O)c1 C1(NC(c2ccnc(C(F)F)c2)=O)CCCCC12CCCN(C(=O)CO)C2 c1(C(=O)NC2CC(CNC(C(CSC)C)=O)OCC2)cc2ccncc2s1 C1(COC)(C)CCCN1C(c1cc(C(N)=O)ccn1)=O.C(=O)C(C)CCO.N C12(C(N(C3CC(F)(F)C3)C)=O)CC1CCN2C(C1COCC1(C)C)=O N1(C(C(CC#C)O)=O)CCC(C)N(C(=O)Cc2cc(OC)ccc2F)CC1 c1(COCCN(C)C(C2CCCC2)=O)nccc(-c2ccnn2C)n1 C#CC1(NC(C2CCC(C(=O)CC)CC2)=O)CCCC1 C1(CS(C)(=O)=O)CCCN(CC(=O)NCCC2CC(=O)N(C(F)F)C2)C1 c1(C(=O)NCC2N(C(C(C)O)=O)CCC2(C)C)cc(Cl)ccc1Br Cc1cc(CC(=O)NC2CCCC(NC(C3COC3)=O)CC2)ccc1Cl c1(C(N(CC(CC)NC(C2CNC(=O)N2C)=O)C)=O)sc(S(N)(=O)=O)cc1C CC(C)C(C)C(=O)NCC(C)(C)C(=O)NCCCC1CCC1 C1(NC(c2ccc(C(C)C)o2)=O)CCOC(C(=O)NCCc2cc(O)ncn2)C1 N1(C(C(C)C2=CCCC2)=O)CCC2CCN(C(=O)Cn3ccc(O)nc3=O)C2C1 c1(CC)ccccc1C(N1CCC(C(C)(C)C)CC1)=O.C(C=C(Cl)Cl)=CC=O C(C)(C(C)(C)C)NC(COCC(=O)OC)=O.N1(CC=O)CCCCC1.N c1(CCC)ccccc1C(=O)NC1CC1CNC(=O)CC1CCOC1 c1(C(N(CCNC(=O)COC2CCC2)CC)=O)c[nH]c(Br)c1 CN1CCOCC1C(=O)NC1CC(C)(NC(c2nn(C)cc2Br)=O)C1 C=CC(O)(C(=O)N1CCC(CC(=O)O)(C(F)(F)F)CC1)C(F)(F)F N1(C(C(CC=C)C)=O)C(CNC(=O)CCc2cn(C)nn2)CC2CCCC12 c1(C2(C(N3CCC(NC(C=C(CCC)C)=O)C3)=O)CC2)ccc(F)cc1Br C1(NC(C(N2CCC(O)CC2)C)=O)C2CCN(C(=O)C=Cc3ccncn3)C12 N1(c2cc(OCC)ncn2)CCC(C2(NC(C3CN(C4CCOC4)C3)=O)CC2)C1 Cc1nc2cc(C(=O)NC3C4C5CCC(C5)C34)cc(Br)c2[nH]1 c1(SC)ccc([N+](=O)[O-])c(C(N2CC(C)C2)=O)c1.c1(C=O)cnn(C(C)C)c1 c1(NCC2(C)ON=C(C)C2)[nH]c(=NCC(F)(F)Cl)nc2scnc12 N1(C(CSCC)=O)CCCC1(C)CCC(=O)NC.C12(CCC1)CN(C)C2 C1(C(N2CC(COC)N(C(c3nocc3C)=O)CC2)=O)CC2CCC(C1)C2(F)F Cc1c(C(N2CCC(CNC(=O)C(C)CC(C)C)CC2)=O)oc2ccc(Cl)cc12 CC1(O)CCCN(C(=O)C(Cc2cn[nH]c2)NC(c2ccnnc2O)=O)C1 N1(CCC(=O)NCC2N(C(c3scc(C(C)=O)c3)=O)CC=C2)CCCCC1C c1(CNCCN2CCN(C(c3ccc(Cl)cn3)=O)CC2)ccc(Br)nc1Br C1(C(N2CCC(CO)(CNC(C3CCC4CC34)=O)C2)=O)(CC)CCNC1=O C1(OC)(C)CCC(C(C)(C)C)CC1.c1(CCC(C)C)cccc(Cl)c1.C(=O)N C1(C(N2CCOCC(C(C)C)C2)=O)CCC(C)(C)N(C(=O)NCCCl)C1 C(CC(C)C)(C(=O)N(C1CC1)CC1CC1)NC(C)=O CC1Cn2nc(C(=O)NC3CCC(NC(c4coc(O)n4)=O)CC3)cc2C(=O)N1 C1(C(N2CC=CC(NC(C(N3CCNC(=O)C3)C)=O)C2)=O)CC(=O)CC12CCC2 Cc1cc(C(N2CC(NC(=O)CCN(CC(F)(F)F)C)C(C)C2)=O)c(C)o1 C1CN(C(=O)Cc2nnc(C)o2)C(C)(C)C1.C(C)(C(=O)N)N(C(C)=O)C.C CCC(C)C(C)CNC(=O)C(Cc1ccoc1)NC(=O)C=CC1(C)COC1 c1(C(=O)OC)ccc(N2CCOC(Cn3nc(C)nc3C)C2)nc1 C1(NCC)CCCC(N=c2[nH]c(=NCCN(CC)CC)[nH]c3ccsc23)CC1 C1(N(C(CCCOC(C)C)=O)C)CCC2CN(C(c3ccn(C)c(=O)c3)=O)CC12 c1(OC)ccc(C)cn1.C1(C(=O)N)CC2CC2N1C(=O)C(c1cccc(Br)c1)O C1(NC(c2n(CC)ccn2)=O)(C)CC2CCC1CC2.C(=O)CN(C)CCO.N CCC(O)C(C)C(=O)NCC1(C)CCCN1C(=O)Cn1ncnn1 c1(NC2CCC(NC(c3ccc(CCC)s3)=O)C2)nc(SC)cc(C)n1 N1(C(CCn2ccc(C)n2)=O)CC2CC1(C(=O)NC(C)Cn1cccn1)C2 Cc1nnc(CC(=O)NC2CC2CNC(c2conc2C(C)(C)C)=O)o1 Cc1c(Cl)ccnc1C(=O)NCC(C)(C1CCC1)NC(C1CCOC1)=O c1(C(C(=O)OC)N(CCNC(CCC)=O)C)cccc2ccccc12 c1(C=O)cccc(C2CC(F)(F)C2)c1.CC(C=O)=CC1CC1.CCC1CC1.N Cc1cc(F)c(C(N2CC(CNC(=O)CCc3ccsc3)CC2(C)C)=O)cc1F C1(CNC(c2cnc(CC)s2)=O)CC2(CCN(C(c3cnc[nH]3)=O)CC2)C1.C CCCC(C)CC(=O)NC1CCN(C(=O)C=Cc2ccncn2)CC1CO c1(NC(CC2N(C(Cc3c(C)nsc3)=O)CC2)=O)cn(C)nc1Cl C(C(CC1CC1)C(=O)NCCCP(C)(C)=O)NC(C1(C)CCCO1)=O C1(CNC(C(CC)(C)O)=O)CC12CCN(C(C1CC(C(C)C)=NO1)=O)CC2 C1(CC)CCCN(C(c2cccc(Br)c2F)C(=O)NCCC#N)CC1 C1COCCN(C(=O)CC2(O)CCC2)C1.c1(C=O)ccc(Br)cc1C(F)(F)F.N C1(C(N)=O)COC2(CCN(C(c3cc(F)cc(Br)c3)=O)CC2)C1 CC(C)C(O)C(C)C(=O)N1CCN(C(c2nc3ncccn3n2)=O)C(C(C)C)C1 c1(OC)cccc(C(=O)NCCC2CCN(C(=O)C(O)CF)C2)c1N C(CCOC)(C(=O)NCC(O)CN(C)C)NC(CCN(CC)CC)=O c1(CCC(N2CC(NC(c3ccc[nH]3)=O)C2)=O)csc2ccccc12 Cc1ccoc1C(c1nnnn1C)NC(c1snnc1COCCO)C c1(-c2onc(-c3c(NC)cccn3)n2)ccccc1S(C)=O C(CCS(=O)(=O)Cc1ccccc1)CN1C(c2c(C)nn(C)c2)CC1 n1(CCC)cccc1C(=O)NC(CNC(=O)C(C1CC1)SC)CO C1(CNC(C(CC)=CC)=O)(CF)CC12CCOCC2 Nc1ccc(C(N2CCCC(F)(CNC(C3CC3C3CCCC3)=O)C2)=O)cc1Cl N1(C(C(N)=O)=O)CCN(C(C2C3CCC2CC3)=O)C2CC12 C1(NC(C(C#C)(C)C)=O)CC(O)CN(C(c2c(OC(F)F)cccc2F)=O)C1 c1(C(N2CC=CC(NC(Cn3cc(C(=O)NC)nn3)=O)C2)=O)cncc(SC)c1 Cc1c(C(=O)OCC(C23CC(C#N)(C2)C3)=O)cccc1Cl N1(C(C(C=C)(C)CC)=O)CCC2CN(C(=O)C(=O)C(C)(C)C)CC2CC1 C1(C(N2CC3C(NC(c4cncs4)=O)C3C2)=O)C2CC3CC(C2)CC1C3 N1(C(c2c(C)nco2)=O)CC2CCN(Cc3ncccc3[N+](=O)[O-])C2C1 C(=O)(CCCN=[N+]=[N-])NC1C(CC)CN(C(=O)C(c2cccc(O)c2)(C)C)C1 c1(CN(C(=O)C(=O)NC(c2ccccc2F)C)CC)ccc(Br)c(Cl)c1 Cc1scc(C(N2CC3CC3C2C(=O)NC(C(=O)N(C)C)C2CC2)=O)c1C c1(OCC(C)C)ccc(C(=O)Nc2cccc(-c3nnn(C)n3)c2)cc1 N1(C(c2cnn(C)c2F)=O)CC2(CCCN(C(=O)CCc3cnc[nH]3)C2)C1 O=C1CCN(C(c2cnc(C3CCCN3C(=O)Cc3ccsc3Cl)s2)=O)CCN1 C12(C(N3C(CC)CC3)=O)CC(CN(C(=O)CCN3CCCCC3)C1)C2 c1(NC(CC(C)NC(Cn2c(C)cnc2)=O)C)c(C#N)cnc2c(Cl)cccc12 C1(C(C)NC(C(C2CCCCC2)NC(CN(C)CC)=O)=O)CCOCC1 CC(C)(O)C(F)C(=O)NC1CCOC1C(N1CCCC(O)CC1)=O C1(CNC(CN(C(=O)CCc2ccccn2)C(C)C)=O)CCCN1C c1(C(=O)NC2C(C)C2(C)C)ccc(-n2cc(C3CCN(C)C3)nn2)cc1 CC1CN(Cc2ccc(S(=O)(=O)N3CCCCC3)cc2)CC2(CCOC2)O1 C1(CNC(C2(CSC)CC2)=O)C2CN(C(=O)CCNC3CC3)CC12 C1(C)(C(C)C)CN(C(C2CCOCC2NC(c2ccc(O)cc2F)=O)=O)CCO1 c1(C(=O)NC2(CO)CN(C(C(C)OCC)=O)C2)[nH]c2c(c1C)CCCC2 Cc1cccc(Cn2cc(C3(O)CN(C(=O)C(C)CSC(F)(F)F)C3)nn2)n1 Cc1cccc(COCC(=O)NC2CCCC2)c1.C1(C=O)(N(C)C)CC1.C c1(CC)cc(C(=O)NC2(CO)CN(C(C3CCCN3C=O)=O)C2)cc(O)n1 Cc1c(C(N2CCCC(F)(C(=O)NCc3cn(C)cn3)C2)=O)cccc1Br N1(C(Cc2c(C)scc2)=O)CC2(C(=O)NC3CCCC(C(N)=O)C3)CCC1CC2 c1(CNC(c2c(CC)nnc(C)c2)=O)cnn2c1CN(C(=O)C=CS(C)=O)CC2 C1(C(CNC(c2cc(COC)on2)=O)(C)C)CCN(C(c2cncn2C)=O)CC1 C(C(=O)NOC1CCC1)(c1cccnc1)NC(CC=CC)=O C=CC(C)(CCNC(=O)CCC1CCCCC1)C(=O)NC1CC1CC(=O)OC CC1=C(C)CN(C(=O)CCC(C)NC(=O)Cc2cccc(F)c2)CC1 C1(CN(C)C(c2sccc2CO)=O)CCN(C(C23CSCC2C3)=O)C1 N1(C(C=CC)=O)CCCCC12CN(C(c1n[nH]c3ccc(Br)cc13)=O)C2 N1(C(C=CC)=O)CC=CC(NC(C2(OCC)CCOC2)=O)C1 Cc1nc2c([nH]1)CC(C(N1CCC(NC(=O)C(C)S(C)(=O)=O)C1C)=O)CC2 C1(NC(c2sc3sccc3c2Cl)=O)CCC(O)CN(C(=O)CCn2ccnn2)C1 C1(C(=O)NC(C)CCC(C)(C)C)(CC)CCN(C(C2CC2(F)Cl)=O)CC1 N1(C(c2c(C)nsc2)=O)CCC2(CCCC2NC(=O)C(C)C(O)C(C)C)CC1 S(=O)(=O)(c1ccc(C(=O)OCC)o1)NC1(C#C)CCOCC1 N1(C(=O)NCc2cc(Cl)ccc2I)CCCC(O)(C2CC2)C1 C1(C(C)C)CCC(C(=O)NC(C)(C)C(C)C)CC1.C(=O)(C(C)(C)N(C)C)N N1(C(C(C)(C)OC)=O)CC2(C1)CN(C(c1coc(C3CC3)n1)=O)CC2CO c1(C(=O)NCC(CNC(c2c(CC)occ2)=O)CO)ccncc1N C(C)(CCCCNC(=O)Cc1c[nH]ccc1=O)NC(Cc1ccc(C)s1)=O N1(C(C(CC)(C)C#N)=O)CCC2CCN(C(c3csc(Cl)c3Cl)=O)C2C1 C=CC(C)(C)CC(=O)NC1CC12CCN(C(C1CCN(C)C1=O)=O)C2 C1(NCc2c(C(=O)OC)nn(C3CCOCC3)c2)CCC2C3C=CC(C3)C12 N1(C(CCC(C)O)=O)CCC(C2(NC(c3cc4cnn(C)c4s3)=O)CC2)C1 C1(CN(c2ccccc2)C(Cc2c(Br)ccc(C)c2)=O)CCC2(CO1)CC(O)C2 C1(NC(c2cccc(C3CC3)n2)=O)CC2CCC1N2C(=O)CCc1ccoc1 C1(NC(=O)C=Cc2ccncc2)CC2(CCC(NC(C3CC3(Cl)Cl)=O)CC2)C1 C=C1CCN(C(=O)C(C2CC2)C2CC2)C(C(N2CC(F)(CF)C2)=O)C1 N1(C(c2cccc(CC)c2)=O)CC2CCC(CNC(=O)C)C2C1.C(C)(=O)N C(=O)(CC(C(C)(C)C)NC(c1sccc1C#N)=O)NC(CC(=O)NC)C C12CCC(F)(CC1)C2.N1(C(C(C)OCCC=C)=O)CCCCC1CCC(=O)N.C N1(C(c2n(C)nc(O)c2)=O)CCCC(C)(CNC(C2CCS2(=O)=O)=O)C1 Cc1cc(C(=O)NC(C)(C)CCCC(=O)NC2CCCN(O)C2=O)cc(C#N)c1 c1(C(N(C)CCN(c2cnn[nH]2)C)=O)ccc(NC(=O)Cc2ccco2)cc1 C1(C(=O)NCCOCC=C)COCC1NC(=O)C(n1ccnc1C)C c1(NC)ccc(C(=O)NC2CCN(C(=O)Cc3ccco3)CC2)cc1 C1(C(C)NC(Cc2ccc(C)o2)=O)CCN(C(=O)CCCCn2ccnn2)CC1 c1(-n2c(C3C(C)CC3)nc(C3CC34CC4)n2)cc(Cl)cc(Cl)c1 c1(N2CCC(C)C(NC(C3CC(F)(CO)C3)=O)C2)nc2cccc(Br)c2o1 c1(C(C)=O)ccc(C(N2CC(NC(C3(CO)COC3)=O)C(F)C2)=O)c(Br)c1 C1CC(=O)N1.CC(C(=O)NCCCOCCC(=O)N(C)C)N(C)C c1(C(=O)NCCNC(C2C(CC)C2)=O)cc2c([nH]1)CCCC2.C1CC1.C S(=O)(=O)(c1cnc(O)c(F)c1)NC(C(CCC(=O)O)C1CCCCC1)=O c1(C2C(C=O)C2)ccc(F)c(F)c1.C1COCC1.C1(CC#N)(C(=O)N)COC1 C1(C=O)CCC(=O)N(C)C1.CN=c1[nH]cc(C(=O)NC2CC(C(F)F)C2)o1.N C1CN(C(=O)Cc2cc(C)nn2C)C(C)(C)C1.C(C(C(=O)N)N(C)C)OC.C Cc1cc(N2CCCCC2CNC(=O)C(C)CN2CCOCC2)n2nc(C)nc2n1 c1(C=O)cccc(S(N)(=O)=O)c1.C12(C=O)CCCC1CCC2.CC(C)C1CC1.N c1(C(N(CCCNC(=O)C#CC2CCCO2)C)=O)cccc2nn(C)nc12 N1(C(CC2C(C(=O)OC)CC2)=O)CC2CCC(C1)N2C(=O)C(C)(COC)CC Cc1ccc(C(=O)C(C)N(C)Cc2ccccc2)nc1.C12CN(CCO1)CCC2 C(CC(C)C)(C(=O)NC1CC(N(C)C(c2cn3ccsc3n2)=O)C1)OC N1(C(C(C)(C)n2cncn2)=O)CCCC(NC(c2ccc(O)nc2)=O)C1 c1(C(=O)NCC(C)(C)CNC(c2cnc(C3CC3)o2)=O)ccc(O)cc1Cl N1(C(CCCCC)=O)CCC(C)(C)C1C(=O)NC1C=CCCC1 c1(CC(=O)NC(CCCNC(CC(=C=C)C)=O)CCC)coc2ccc(C)cc12 N1(C(CCc2cc(OC)no2)=O)CC(NC(c2c[nH]nc2C2CC2)=O)C(C)C1 c1(C(=O)OC)ccc2c(=NCCCNCCSCc3cscn3)[nH]cnc2c1 CON(CCC(=O)N(C1CCOC1=O)C)C(=O)CC(C)(C)SC c1(C(=O)NC2(CC(=O)NC(C(C)N(C)C)C)CCC2)cc(=N)[nH][nH]1 c1(C(=O)NC2C(NC(c3n(C)ncc3)=O)COC2)cc2ccccc2cc1N N1(C(C(C)NC(COC)=O)=O)CCOC2CCN(C(c3cc(C)ccn3)=O)CC12 C1(CNC(Cc2nc(SC)sc2)=O)CCCN(C(=O)C(CC)n2cncn2)C1 CCC(CC(F)(F)F)C(=O)NC1CN(C(C2(CC(C)=O)CCCC2)=O)CC1O c1(N2CC=CC(NC(CC(C)(C)C3CC3)=O)C2)ncnc2sc([N+](=O)[O-])cc12 c1(C(=O)OCC(c2cccc(OC)c2)(F)F)ccc2c(c1)OC(C)(C)C(=O)N2 C(=O)(C(CC)CC=CC)NC(CC#C)C(=O)NCC1CCCCC1 C1(NC(c2nc(C)n(C)n2)=O)CCOC12CCN(C(=O)C(C)n1cccc1)CC2 c1(-c2c(C(=O)NCC34CC(NC(CC)=O)(C3)C4)nco2)ccccc1F C1(CNC(COC(CC)C)=O)C(O)C(O)CN1C(C1CCC(O)CC1)=O N1(C(CCCC(=C)C)=O)CCC2C(CCCN2C(c2cnc(C)nc2CC)=O)C1 C12(NC(CCc3c(C)ncs3)=O)CN(C(c3cnc[nH]3)=O)CC1CS(=O)(=O)C2 N1(C(C2(C#N)CCC2)=O)C(C(N2CCC(O)(CC3CC3)C2)=O)CC2CCCC12 c1(C(=O)NC(C2(O)CCN(C(=O)C(O)C3CC3)CC2)C)ccc2cnccc2n1 C(c1cccc(C#N)c1)=CC=O.c1(CC)cc(C(=O)NC2CCC2)ncn1.C c1(NC(C=CC)=O)c(-c2cn(-c3cncc(-c4ccncc4)c3)nn2)cnn1C C1(C(N(C)CC2N(C(C3(CC#C)CCC3)=O)CCC2)=O)(C)CC(C)(C)C1 c1cc2cc(Cl)ccc2o1.c1(OC)ccc(OC)c(C(=O)C(C)NC(=O)N)c1.C C(C)(C(=O)N(CCCCNC(=O)C(C)n1ccnn1)C(C)C)OCC(C)C N1(C(CC(C(=C)C)O)=O)CC2(C1)CN(C(c1ccoc1C(F)(F)F)=O)CC2CO N1(C(c2ccc(SC)o2)=O)CCCCC(NC(C2CCNC2=O)=O)C1 N1(C(c2sc(Cl)c(OC)c2Cl)C(=O)NC)CCn2ncc(Br)c2C1 CC1CC(N=c2[nH]nc(O)s2)CN1C(=O)C(Cc1ccccc1)C(C)C C1CCN(C(=O)CN2CCS(=O)CC2)CC1.N1(C(C2CC2)=O)CCC1.CCN c1(C(N=c2ccn(CCC)[nH]2)=O)cc(=O)n(C)c2ccccc12 c1(OCC)ccc(NC2(c3nnnn3C(C)C)CCCOC2)c(C)c1 c1(CC(=O)N(CC(C)NC(=O)CC2CCCC(C#N)C2)C)nc2ncccn2n1 N1(C(C=CC(C)(C)SC)=O)CCN(C(c2nocc2Cl)=O)C(C)C1C N1(C(CC2(CCC#C)OCCO2)=O)CCC2(CC1)CN(C(=O)COC)CC(C)O2 C(N=c1[nH]c(=NC(CSC)C(C)C)[nH]c2c1COC2)c1c(OC)ccnc1 S(=O)(=O)(c1cccc(C(N2CCN(C(=O)CC(F)F)C(C)C2C)=O)c1)NC(C)C CC1C(NC(C2CC(n3cnnc3)C2)=O)CCCN1C(C1CCCCNC1=O)=O N1(C(CS(CC)(=O)=O)=O)CCCCC2(CCN(C(=O)C(C)(C)C3CCOC3)C2)C1 C1(NC2(c3n(C(C)C)nnn3)COCC2C)CCC(C)(C)CC1 Cn1ncc2cc(-c3cnc4cc(C(=O)NC5CCC(F)(F)C5)[nH]c4c3)ccc12 c1(C(=O)NC(C2N(C(CCc3cc(C)on3)=O)CCC2)(C)C)cnc(Cl)cc1Cl N1(C(C2(F)CN(C(C3CCC(=O)C3)=O)C2)=O)CCCC(C2CCC2)C1 N1(C(C2C(C(C)C)OCC2)=O)CCC(C)(CNC(C23CC4CC2C3C4)=O)C1 N1(C(c2cnc(C)[nH]2)=O)CC(C)N(C(c2cc(C(N)=O)n(C)n2)=O)CC1C.CC C12(C(N(C(C)CC(N)=O)C)=O)CC(CN(C(=O)C(c3cnn(C)c3)=O)C1)C2 N1(c2c(CC)cccn2)CCN(N2CC3(CCCC3)C2CC)CC1 N1(C(Cn2c(CCC)ncc2)=O)CCC(C)C1.c1(CC=O)sc(S)nc1C.C1CC1 N1(C(c2c(CC)n(C)nc2)=O)CC2CC(O)C1C2NC(c1sc(C)nc1C)=O CC(CN(C)C(c1ccnn1CCF)=O)C(=O)NCC1CC1c1ccco1 C1(CN(C)CC)CCN(C(c2sccc2C)C(=O)NC2CCOC2)CC1 C(=O)(CCN1CCC(O)C1)N1C(CC(=O)NCc2cccs2)COCC1 c1(C(=O)NCC2C(NC(C(C)N(C)C)=O)C2)c(N)cc(Cl)nc1Cl C(CC1CC1)(C(=O)N1CCCCCO1)NC(C1CCCCC(=O)N1)=O C1(C(=O)NCC2COCC(C)O2)COCCN(C(=O)Cc2cncnc2O)C1 c1(C(N2CCC(OC3CN(C(C4CC4)=O)C3)CC2)=O)cnccc1Cl.C(F)F.O N1(C(C2CCC(N=[N+]=[N-])CC2)=O)CC(CO)C2(C1)CN(C(=O)C(O)C(F)(F)F)C2 N1(C(C2(CCCC)CC2)=O)CCC(CN(C(=O)CC2CCCN2C)C)C1 N1(C(C2CC3CC3N2C(=O)CCc2cn[nH]c2)=O)CCc2nc[nH]c2C1 C1(CCNC(C(C2CCC2)OC)=O)CCCN1C(=O)CCc1cnn(C)n1 CC(C)CC(CC(=O)NCC12CCCC1C2)NC(C12C=CC(CC1)C2)=O c1(CCC(=O)OC)cccc(C(F)(F)F)c1.C(=O)C(c1nn[nH]n1)C1CC1.N N1(C(C(c2ccc(C)cc2)=O)=O)CC(CNC(C2C(C)C2C)=O)C(F)(F)C1 CCC(F)C(=O)NC(C1CCCN1C(=O)COCc1nccn1C)C N1(C(=O)NCC(C)CCCO)CCCn2cc(Br)cc2C1 Cc1ccc(S(=O)(=O)Nc2ccc3nc(-c4ccncc4)nn3c2)cc1C N1(S(C)(=O)=O)CC2CC1CN2CC(=O)NC1COC(=O)C1 c1(C(=O)NCC(C)CNC(C2CCC3CC3CC2)=O)c(F)ccc2c1OCO2 c1(CC)ccc(C=CC(=O)NC2CCN(C(C3CCNC(=O)C3)=O)C2)o1 N1(C(C2OCCN(CC)C2)=O)CCn2ncc(CNC(=O)CC(C)OC)c2C1 C1(NC(c2cncc(C)c2C)=O)CCN(C(=O)C(C)CC2CCC2)CC12CCC2 c1(-c2onc(C(=O)NC(C)CN(C(=O)C(C)(Cl)Cl)C)n2)cccc(F)c1 C#Cc1ccc(NC(=O)CCCn2nnc(-c3ccccc3)n2)nc1C CCC(C)CC(=O)NCCC1CCC1.c1(C=O)sc(C)cc1OC(F)F.C1CC1 N1(C(C(C)S(N)(=O)=O)=O)CCN(C(C2CC(C)OC2C)=O)CC12CCC2 N1(Cc2ccc(-c3c(NC)nccn3)cc2)CC2(CCC2)OCC1C(=O)O c1(C(N(c2nc3cccnc3s2)C2(CN)COC2)=O)c(Cl)ccc(Br)c1F n1(CC(=C)Br)c(N2CCC(CSC)CC2)nnc1COc1ccc(Br)cc1 c1(C(N(CCC)C)=O)coc(CS(C)(=O)=O)n1.C(=O)C(C)N.CC(F)(F)F c1(C(=O)NCC(C2CCCCC2)NC(CC(C)SC)=O)ccc([N+](=O)[O-])cc1 c1(C(=O)NC2CC(C(=O)Nc3ccnn3C3CC3)C2)ccc(CO)cc1 c1(CC(=O)N)cccc(C)c1F.Cc1nn(CC(N2CC3CC3(C)C2)=O)c(=O)o1 C1(CCNC(CCC(=O)NC)=O)CCN(C(=O)C(C)CC(C)(C)C)CCC1(F)F C1(C)(C(=O)NCc2nn(C)c(C(N3CCC(F)(C)C3)=O)c2)CCC(=O)NC1 N1(C(c2nnc(C)s2)C(=O)NC(C(=O)OC)C)CCC2(CCSC2)C1 Cc1nn(C)c(C)c1CNc1cc(N2CCOC(C)(C(C)C)C2)nc(C(C)C)n1 Cc1ccc(C)c(C(=O)NCC23CC(CO2)N(C(C2CCC(=O)O2)=O)C3)c1 N1(C(C2C(CC)C2)=O)CCC(C)(C)C1C(=O)NCC(C)CC1CCCC1 N1(CC(=O)NCC(CC)NC(=O)C(C)(C)F)Cc2ccccc2C1 N1(C(c2cccnc2)=O)CC2CCC1CN2C(=O)CF.C12C3C4C5C3C1C5C24.N c1(CS(=O)(=O)NCC2CN(Cc3cccc(O)c3)C2)ccc(C(F)F)cc1 C1(C(=O)NCC(CC)NC(=O)C=Cc2ncco2)CCC2(CCOCC2)O1 C(C(CC(=O)NC(C)C(=O)NCC(C)C)OC)NC(c1cc(CC)on1)=O C(=O)(CCCCN(C)C)N1C(CC(=O)NCC2(COC)CCC2)CCC1 C(C(C(=O)NCCCN(CC(C)C)C)C(C)(C)C)NC(C(CSC)(C)C)=O c1(C(N2CCCC(C(C)NC(CSCC)=O)C2)=O)cc2n(n1)CCO2 c1(CNC(C(CC)c2ccccc2)=O)cc(NC(CCSC)C(=O)NC)n(C)n1 Cc1cc(C)c(CNC(C2(NC(=O)CC3CCOCC3)CC(C)C2)=O)cn1 CCC(CC(=O)N(C1CC(NC(c2c(C(F)(F)F)coc2C)=O)C1)C)OC C(CCC(=O)NCC1CC(NC(c2cnn[nH]2)=O)C1)=CC.c1ccccc1.C C1(NC(C2CN(CC)C(=O)C2)=O)CC2CCC(C1C)N2C(c1cc(C)[nH]n1)=O Cc1ncsc1C=O.c1(CC)cc(C(=O)N(C2CCCC2C(C)(C)C)C)no1.N N1(C(c2ccc(N)cn2)=O)CC(NC(=O)CCOC2CCOCC2)CC(O)C1 C(=O)(C1(C)CCc2ccccc21)NCC(CN=c1[nH]nc(COC)s1)C(F)(F)F c1(C(=O)NC(C)CCCCNC(=O)C(C)(C)C#N)cnn2c1C(C)CCC2 N1(C(C=CC(=O)N(C)C)=O)CC(C)C(O)C1.C(=O)(CCCc1nncn1C)N c1(C(=O)Nc2cccc(NC(C=CSC)=O)c2)ccc2c(c1)CCOC2(C)C C(c1cnc(C)nc1O)=CC=O.N1(C(C(COC)(C)O)=O)CCC(C)C(C)C1.N Cc1cc(CNC(=O)NCC(C)CC(C)C)cc(C)c1F c1(C(=O)NC2(CO)CCN(C(C(CC=C)C(C)C)=O)C2)ccc([N+](=O)[O-])c(O)c1 Cc1cc(O)ncc1C(N1CCCC1CN(C)C(C1(n2cccn2)CCC1)=O)=O C1(COC(C2(NC(C)=O)CC2)=O)CC(C)(C)C1C(F)(F)F Cc1noc(CCC(=O)N(C(C)C2CC2)C)n1.c1(C=O)ccnn1C(C)(C)C.N Cc1cc(C(=O)NC(C2CCN(C(c3scc(Cl)c3Cl)=O)C2)C)cc(C)n1 CC(C)(C)C(=O)C(=O)N1CCC(CO)C(NC(=O)C(=O)NCC(F)F)C1 O(N=Cc1ccc(OC)cc1)CC(=O)NCc1cc(OC)nc(OC)c1 C1(SC)CN(C(=O)C(c2cccnc2)O)CC1NC(=O)C(O)Cc1cnc[nH]1 c1(NC(c2n(CCC)nnn2)CCCOC)ccc(-n2ccnn2)cc1.C1CC1 c1(C(C)C)ccsc1C(=O)NCC=CCNC(C1CCN1C)=O Cc1ccc(C(N2CCC(CNC(=O)C(C)CC3CCC3)C2(C)C)=O)c(Cl)c1Cl n1(CC)ncc(C(=O)NCC2C3CN(C(c4cc(C)n(C)c4)=O)CC23)c1Cl N1(C(=O)NCc2ccc(CO)o2)CCC2(CC2)C1 C#CCC(O)C(=O)N(CCCNC(C1CCN(C)CC1)=O)C C(=O)(CCCCOC(C)(C)C)NCC1C(NC(C(C)SC)=O)CCC1 N1(C(Cc2ccc(C)cc2Cl)=O)CCOC2CCN(C(C3CCC3C)=O)CC12 C(CN=c1[nH]c2cccc(Br)c2o1)C1C(C)CCCN1C(=O)CC1CC1(C)C FC1(c2ccccc2)CCN(c2nnc(CCCc3cccc(Br)n3)o2)CC1 C1(CNC(c2c(C)nn(C)c2C)=O)CC2CCC(C1)N2C(C)C(N)=O CCCC(CNC(=O)C(CC1CCCC1)NC(c1ccc(C)cc1F)=O)CCO c1(NC(C(N2CC3CC(OC)C3C2)=O)=O)ccc(S(=O)(=O)C(C)C)cc1 N1(CCCCN(CCC(C)(C)C)CCO)CCC(=O)N(CCC2CC2)C1=O.CO C1(N(C(=O)CO)C)CCC(C(N2CCN(c3ncco3)CC2)=O)CC1 C(=O)(C(O)(C(F)(F)F)c1cn[nH]c1)NC1CN(C(C(=O)OCC)C)C1 N1(C(c2cnn(C)c2Br)=O)CCCC2CN(C(c3cocn3)=O)CCC12 C1(F)(CNC(C2=C(C)OCC2)=O)COCCN(C(c2c(O)nnc(C)c2C)=O)C1 C1(C)(CNC(c2c(C)onc2)=O)CCC(NC(=O)C=CCO)C1 N1(C(CCCOC)=O)CCN(C(=O)CCCNC(N)=O)C(CC(F)(F)F)C1 c1(C(=O)NCCCCCNC(C23COCC2C3)=O)cc2cccc(Cl)c2s1 C1(NC(C2(CC(C)C)CCC2)=O)CC2CC1CN2C(c1ccc(Cl)cc1Cl)=O C1(Cl)(C(=O)NC(CCNC(C2CC(SC)C2)=O)C)CC12CCOCC2 CC1(NC(=O)CCNC(=O)CCC2CCOC2)CCCOC1 CN=c1nc(C(=O)NCC2COC(CNC(=O)C=CCO)C2)cc(C)[nH]1 c1(N2CC(CNC(C3N(C)CCCC3)=O)OCC2)cnc(C#N)c(C#N)n1 CCCCC(C)(F)C(=O)NCc1cccc(CN(C(=O)CC(C)OC)C)c1 c1(CC(N2CCC(C)C(N(C(=O)C(O)C(F)F)C)C2)=O)cc(F)c(N)cc1F c1cccc([N+](=O)[O-])c1Cl.c1(OC)cc(Cl)ccc1C(=O)NC1CCC(NC)C1 C(=O)(C(CC(C)CC)NC(=O)C#CC1(CC)COC1)NCCC=CC C1(Nc2c(Cl)cc(C(=O)OC)c(C)c2)COc2cccc(OC)c2C1 CP(C)(=O)CC(=O)N1CCCC(c2cn(CCCCCCF)nn2)C1 CN1CCN(C(C2CC2C2CCC2)=O)CC1C(=O)NCCOC1CCC1 N1(C(C(CC)NC(C)=O)=O)CCC(C2(O)CN(C(c3cnc(=N)[nH]c3)=O)C2)CC1 c1(C(=O)NCCCNC(c2cscn2)=O)ccncc1C(F)(F)F.C1CC1 C1(C)(CCN)CN(CCCC=O)CCO1.c1(CC)cc(C(N)=O)n(C)n1 c1(CCC(=O)NC23C(CCN(C(CCC#N)=O)CC2)C3)nc2cccc(Cl)c2[nH]1 c1(C=O)ccsc1S(C)(=O)=O.C(CCC(=O)NCCC)OCCOCC.C CC(O)C(C)(C)C(=O)NCCC1CN(C(=O)Cc2nc(=N)[nH][nH]2)CCO1 C1(CNC(C(C)(C)OC)=O)CC2CCC(C1)N2c1nc(C)cc(C)n1 c1(SC)ccc(C)c(C(=O)NC2CCN(C(=O)C(C)n3cncn3)C(C)C2)c1 C(=O)(C(C)CC(F)(F)F)NCC(CC)NC(=O)CSc1ccc(OC)cc1 CN1CC=C(C(=O)N(C2CC(NC(c3cccc(C#N)c3)=O)C2)C)C1 c1(CC(=O)NC2C(C)CN(C(=O)CN3CCCOC3=O)C2)cccc(F)c1F c1(OC(C)C)nn(C)cc1NC(=O)C(C1CCCC1)NC(C)=O c1(C(N2CCCCC2)=O)ccc(F)c(Cl)c1.c1(C(N(C)C)=O)coc(C(F)F)c1 N1(C(c2c[nH]c(Br)c2)=O)CC2CCN(C(c3ccccc3)=O)CCC2C1 c1(NC(C2CCCN(C)C2)=O)ccc(S(=O)(=O)NC(C)(CO)CO)cc1 c1(C(N2CC(NC(CCc3ccnc(C)n3)=O)C2)=O)ccc2nc(Br)nn2c1 CN=c1[nH]cnc2cc(C(N3CCN(C(c4c[nH]nc4C)=O)CC3C)=O)ccc12 C1(NC(C)=O)CCC(N(C)C(c2ccc(-c3ccccn3)o2)=O)C1.C1CC1 c1(C(=O)NC(CNC(c2c(C)cc[nH]2)=O)CO)sc(-c2ccc(Cl)s2)nc1C N1(C(C(=O)Nc2ccc(C)cc2)=O)CCOCC(C(=O)NCc2ncccn2)C1 N1(Cc2[nH]cc(OC)c(=O)c2)CCCC2(CCN(C(=O)Cn3ncnn3)C2)C1 N1(C(CCC2C(C)C2)=O)CCOC2(C1)CN(C(=O)Cc1cc(O)ccc1Br)C2 N1(C(Cn2ccc(C)n2)=O)CCCC2(CCCN(C(C3CCSCC3)=O)C2)C1 c1(C(=O)NCC(CO)NC(CC2CC(OC)C2)=O)onc2ccccc12 C(=O)(CCCC(=O)N1CCC(CCC(=O)NC)C1)Nc1c(CC)con1 C1(CNC(=O)C2=CCCC2)CC2(CO1)CN(C(c1cnnn1C1CC1)=O)C2 C(=O)(CCCCNC(C1CCCCCC1)=O)NC(C=C)COC Cn1cnc2c1CCN(C(=O)C(F)C(F)(F)F)C21CCN(C(=O)C(C)(C)O)C1 Cc1nn(CCO)cc1C(N1CC(CNC(=O)C(c2ccccc2Cl)(C)C)C1)=O C12(OC)CCCCC(C(=O)N)(C1)C2.C1CN(C=O)CC1C(F)F.C(C)(C)C C1(C(N2CCC(CNC(C(C(=O)OC)OC)=O)CC2)=O)CCCC(C)(C)CC1 C(C)(C(O)C(=O)N(C)CCN1CCN(C(c2cnc(C(C)C)nc2)=O)CC1)OC C1(C(=O)NC(C)(CNC(c2c[nH]nc2[N+](=O)[O-])=O)CO)CCn2ncnc2C1 C(C=O)(C(=O)N)OC.c1(C=O)c(Cl)cnn1C(C)C.C(C)(C)C.C(C)C CCC(CC(=O)NCC(C(C)C)NC(c1[nH]nnc1COC)=O)C(C)(C)C N1(C(c2c(C)ccc(Br)c2)=O)CC2(CCCC2NC(=O)Cn2ccnc2)C1 c1(CSCCCC)nc(-c2ccnn2C)nn1-c1ccc(Cl)cc1 CN1CCC(C)(C(N2CCC(CO)(NC(C3CCC(=O)C3)=O)C2)=O)C1 n1(CCC(=O)NC2CCC(NC(c3cc(CC)n(C)n3)=O)C2)ccc(O)nc1=O c1(CNC(c2c(C)ocn2)=O)cc(C(N2CC3C(C(N)=O)C3C2)=O)n(C)n1 C(CCN=C(NCCS(=O)(=O)C1CC1)NC1CCCCC1)OC C1(CC(=O)N(CC(C)NC(C(C)Oc2ccccn2)=O)C)CCCCC1(F)F N1(C(CC2(C)CCCO2)=O)C2CCC1CC(NC(c1cccc(C(F)F)n1)=O)C2 C(CCC(=O)NC(C(=O)N1CC(SC(F)F)C1)c1ccoc1)SC c1(C=O)cc(F)n(C)n1.Cn1cc(-c2c[nH]cc2C(=O)NCC2CCC2)cn1 c1(C(N2CC(NC(C(C#C)(C)C)=O)C2)=O)ccc2c(c1)C(C)(C)c1ccccc1-2 Cc1nn(C)cc1C(N1CC(CC(=O)NC23CC(C)(C2)C3)CC1C)=O Nc1c(C(N2CC(CCCCNC(C3CC34CCC4)=O)C2)=O)sc(Cl)c1Cl C1(C(N(CCN(C(=O)CNc2cncs2)C)C)=O)CCCC1 C(=O)(C(O)CCCNC(C1CC2C(C1)C2(F)F)=O)NCc1c(C)csc1 Cc1cc(NC(=O)CN(C(C)CC(C)(C)O)C)ccc1Cl C1CN(C(C2(F)C(C)(C)C2(C)C)=O)CCN1C(=O)C.[SH](=O)(=O)CC.CO N#Cc1ccc2c(c1)CCCC2C(=O)NC1CCCN(C(=O)CCCC(F)F)C1 CCCC(O)C(=O)NC1CC(NC(C2C3CCCOC23)=O)CC1O CC(C)(N=[N+]=[N-])C(=O)NCC1(O)CCN(C(=O)Cc2ccc(F)cc2)CC1 c1(OC)ccc(CC(C)C(=O)NCC(C)C)cc1F.C(=O)(C)N.CCN(C)C N1(C(c2ccn(CC)n2)=O)CCC2CC2(C(N2CCCC(C)C2CO)=O)CC1 c1(C(N2C(C(=O)NC3CC3)CC2)=O)ccc(F)cc1I c1(OC)[nH]c(=N)ccc1C(=O)NCCCCNC(c1cc(C2CC2)no1)=O C1(C(=O)N(C)Cc2c[nH]nc2C)(COC)CN(C(=O)CCC2CCCO2)C1 c1(NC(C(c2ccn(C)n2)C)=O)cccc(NC(C2(Cl)CC2(C)C)=O)c1 C1(C(=O)N)COc2cc(F)ccc2C1.C(c1cscn1)=CC(=O)NCC1CCC1 CC1CC(NC(=O)CCc2ccnn2C)CCN1C(=O)CSCc1ncc[nH]1 CCC(C(=O)N1CCCC1Cc1cn(CCC(C)C)nn1)n1ccnc1 C(=O)(C(C)(C)C(=O)N1CC2CC2(CNC(C2CC23CCCCC3)=O)C1)OC c1(C(=O)NC(COCC)(C)C)sccc1NC(C1CC(C)CO1)=O c1(-n2c(-c3cc4ccccc4[nH]3)nc(C(C)OCC)n2)cccc2ccccc12 C1(CNC(c2cn(-c3cccnc3)nn2)=O)CCCN(C(=O)Cc2nc[nH]n2)C1 Cc1cc(C)c(C(N2CCC(CCC(=O)NC(c3nncs3)C)C2)=O)cn1 C1(C#N)(C(=O)NC(C(=O)Nc2cccc(C)c2)C)CCC(F)(F)CC1 c1(CNC(CCSC)=O)nn(C)c2c1CN(C(C1CC3CSCC(C1)C3)=O)CC2 c1(C(N2CCC(CCC(=O)N(C3CC3)CC)C2)=O)cn(C)c(=O)n1C CC1=CC(NC(=O)COC2CN(C(c3cc(C)ns3)=O)C2)CCC1 Cc1c(C(=O)NCCC(C)NC(C2CC(C)(C)C2)=O)cnn1C(C)C(C)C Nc1ccc(F)c(C(N2CC(O)(CCNC(=O)C)C2)=O)c1.C1CC(F)(F)C1 c1(C(N2CCC(CNC(c3nc(C)sc3C)=O)C2)=O)cc(O)ccc1C c1(NCCCC2(O)CCNC2)cc(Cl)c(O)c2ccccc12 N1(C(CCc2c(C)n(C)nc2)=O)CCN(C(=O)CN(C2CCCC2)C)C2CC12 c1(C(=O)NCCN(CCC)C(C2(C)CC2(Cl)Cl)=O)snnc1C C1(CC)(NC(=O)CC2CCC(C)O2)CCN(C(c2[nH]ccc2C)=O)CC1 Cc1sc(O)nc1C(N1CC(O)(CNC(c2snnc2C2CC2)=O)C1)=O C1(CNC(c2cc(C)oc2)=O)CN(C(c2cccc(Cl)c2Cl)=O)C(C)(C)C1 c1(CC(N2CC3N(C(C(CC)SC)=O)C(CC3)C2)=O)cccc2c1OCCO2 C(=O)(CCCC(C)(F)F)N1C(Cc2cccc(CSC)c2)CCC1 CON(CCC(=O)NCCC(O)C1CCCC1)C(=O)c1ccc(C)o1 C1(NC(c2ccc(OC)s2)=O)CCCCCC1NC(c1nccnc1N)=O C1(NC(CCC#CC)=O)CN(C(=O)CCC(C)c2ccccc2)C2(CCCCC2)C1 C1(C)(NC(C(C2N(C(C=NOC)=O)CCC2)(C)C)=O)CCCC(C)(C)C1 O=S(=O)(c1c[nH]ccc1=NC1CC2CCCCN2C1)NCCCOC1CCCC1 c1(C(c2n(CCOCC)nnn2)N)nn(C)cc1[N+](=O)[O-].C1(C)CCOC1.C c1(C(N(CC(CC)NC(c2coc3c2COC3)=O)CC)=O)cnn2c1CCC2 c1(CC)cccc(CC)c1CC(N1CC(CNC(=O)C2=CCCS2)CC1C)=O c1(Cc2nnnn2C2CCC2)csc2ccc(F)cc12.C(C(C)(C)CO)NC(C)C.S N1(C(c2ccc3c(c2)CC3)=O)CCC2C(C1)CN2C(C1Cc2ccccc2O1)=O c1(C(C)=O)cc(C(=O)NC2CC2)ccc1C.c1(C=O)ccc(-c2cscn2)nc1.N CC1CCC(NC(C2CC3CC2C2CC32)=O)CN1C(C1CC2(C1)CC2(F)F)=O N1(C(C(CC)CCOC)=O)CCN(C(c2c[nH]ccc2=N)=O)CCC1C C1(N(C(c2cnsn2)=O)CC)CCCN(C(=O)CCc2ncccn2)CC1 N1(C(COC(CC)(C)C)=O)CCN(C(c2ccn(C)c2C2CCC2)=O)CC1CF CC(C)CCCNC(c1cncn1C(C)C)=O.c1(CCC(=O)N)ccc(Cl)nc1 N1(C(CC2(NC(COC(C)=O)=O)CCC2)=O)CCn2nncc2C1 O=C(C1=COCCC1)NC1CC2CC1N(C(c1cc(Cl)nnc1O)=O)C2 C1(C(=O)NCC2CCN(C(C(C)C)=O)CC2O)CC1C1CCCCC1 C1(C(N2CCOCC(COC)C2)=O)CCc2ccc(F)cc2C1 c1(C(C)C)nc(NC(C)CCOC(C)(C)C)cc(=NC2CCCC3(CC2)CC3)[nH]1 Cc1cc(CCC(=O)NCC)n[nH]1.n1(CC(=O)N)cc(C2CC2)nn1.C1CC1 c1(NC(CC(CC)N(C(C(C(=O)OCC)F)=O)CC)=O)ccc2ncccc2c1 Cc1ncnc(NC(N2CC(C(=O)NC3CC3C34CC(C3)C4)C2)=O)c1C C(=O)(C(C)Cc1cnn(C)c1)NC(C1(NC(c2c[nH]cc2Br)=O)CC1)C C=CC(CC)C(=O)NCCCN1CCC(NC(C2CCC(OC)C2)=O)C1 C=CC1(C(=O)NCC2COC(=O)N2)CCN(C(=O)CCCC#N)CC1 c1(OCC)ncc(C(=O)NCC2(C)CCN(C(=O)CC)C2)cc1Cl.C1CC1 N1(C(C(CC)OC)=O)CCC(C2CC2)(CNC(=O)CN(S(C)(=O)=O)C)C1 CCC(C)C(C(=O)NCCC(C)c1cn[nH]c1)NC(=O)C(N)=O c1(OC)c(C=O)cc(F)cc1F.C1(CC=O)NC(=O)NC1=O.C(C)C1CC1.N c1(CSc2nccc(C(=O)NCC(C)OC)c2)ccnc(C(=O)OC)n1 C1(CC(=O)N(C)CC2(C)CC2)CC(O)C12CCC2.c1(C=O)nccn1C.N c1(CNC(NC(C)CCC(C)(C)C)=NCC2CCCO2)cccc(Cl)c1[N+](=O)[O-] Cc1noc(CCC(=O)N)n1.C1CCN(C(C23CC(C(=O)O)(C2)C3)=O)C1.CC N1(C(c2coc(C(C)C)n2)C(=O)NCC)CCC(CC)CC1.CC(F)(F)F.O CC1(C)Cc2cccc(C(=O)NCC3CCN(C(c4ccc[nH]4)=O)C3)c2C1 C1(NC(C(CC)SC)=O)C2CCC1N(C(=O)C(c1ccc(F)cc1)(C)C)C2 c1(C(=O)NCC2(C)CC(NC(C3CC3(C)C)=O)C2)cc(Cl)cc(Cl)c1Cl c1(C(=O)NC2CN(C(CSCC(=O)OC)=O)C(C)C2)cc(=O)n(C)cn1 C1(C(=O)NCC(=O)N(C)C)CC12CCN(C(c1ccc(O)cc1Cl)=O)C2 CC1CCC(CNC(c2ccc(N)cn2)=O)CN1C(=O)CCc1cscn1 c1(CC(N2CC(NC(c3ccn(CC)n3)=O)C2)=O)c(C)[nH]c2ccccc12 N#CC1CCCN(C(c2cnc(-c3ccsc3)s2)C(=O)NC2CCCCC2)C1 C12(NC(c3c(C)cns3)=O)CCC(CC1)N(C(c1oc(C3CCC3)nc1C)=O)C2 C1(O)(CN(C(C=CCOC)=O)C)CCCN(C(c2cnn(C)c2Cl)=O)C1 C1(N(C(C(C)n2ccnc2)=O)C)CCN(C(=O)CCN2CCOCC2)CC1 C(=O)(C1=CC2CCCCCCC12)NCCN(C(c1coc(Cl)c1)=O)CC N1(c2nnc(-c3cnn(CC)c3Cl)n2C)CCN(C)C(c2ccccc2)C1 c1(NC(=O)COCc2ccc3c(c2)OCO3)cc(F)c(-n2ccnc2)c(F)c1 C(CC(C)C(=O)NCC1CCCC(NC(=O)CCC2CC(F)(F)C2)C1)OC c1(C(N2CCC(NC(=O)Cc3ccc(F)cc3F)CC2)=O)cncc2c[nH]nc12 N1(C(C(CCCNC(C(CC)C)=O)O)=O)CCOCC(C)(F)C1 CC1(C)CCCCC1.N1(CC=O)C(=O)NC(C)(C)C1=O.C1(C)(C(=O)N)CC1 Cc1ccc(CCC(=O)NC2CCN(Cc3c(C)noc3C)C2C2CC2)c(Br)n1 c1(C(=O)NC(C(C)(C)C)CNC(=O)C#CC2CCCO2)cn2cc(Cl)cnc2n1 C(CCC(C)(C)CO)NC(c1nccc(OC)c1)c1nnnn1CCSC c1(SC)ncc(=NC2CCN(C(c3cc(C4CC4)nc(Cl)c3)=O)CC2)[nH]c1C c1(C(=O)NC2CCN(C(CC(=O)OC)=O)CC2F)cc(C)c(C)c(Br)c1 C1CCCOC1.C(=O)(C(C)Cc1ccccc1)N(CCNC(=O)CO)CC O(C=C(C#N)C(=O)NCC1(C)CCCCC1)CC.C(C1CCCO1)=CC=O.N C12(CNC(CC(C)(F)F)=O)CCCC1N(C(c1cnc3c(c1)NCC3)=O)CCC2 Cc1[nH]nc(C(N2CC(CC)C2)=O)c1C(F)(F)F.c1(CC(=O)N)cncnc1O N1(C(CC(=O)N(C)C)=O)CC2C(NC(c3cc(-c4ccccc4)cs3)=O)C2C1 C1(NC(C)=O)CCN(C(=NCCC2(C)CC2)NC(C)C2CC2)C1 N1(C(=O)NC(C2(OC)CCC2)C(=O)OC)CCCCC1C.C(=O)C(C)C.C C(=O)(CN=c1ccc(C#N)c[nH]1)N1CCC(C)(NC(=O)CC2CC(=O)NC2=O)C1 C1(C(N2CCC(O)(C(C)NC(C(C)=C3CC3)=O)CC2)=O)C2CCCCCCC12 C(C(CC(C)C)C(=O)N1CCC(C(=O)N(C)C)C1)OC.C12(CCCCC1)C(=O)N2 N1(C(C2N(C(c3c(CC)c[nH]c3)=O)C3(CC2)CC3)=O)CC2(CNC(=O)N2)C1 N1(C(c2cnn(CC)c2N)=O)CC(NC(=O)CC=O)CC12CCC2.C(C)(C)C.O C(=O)(C#CC1CCCC1)NCC1CN(C(C(C)CC2CCC2)=O)CC1(F)F N1(C(CSC(C)C)=O)CC2C(C(=O)N(CC(O)C(C)(C)C)C)C2C1 N1(C(CS(=O)(=O)N(CC)CC)=O)CCC(C)CC1.C(=O)C(C)SC(F)(F)F CCC(C)CC(C)C(=O)N(CC(C)(C)NC(C1CCC(NC(C)=O)CC1)=O)C C12(CNC(C3(C(N)=O)CC3)=O)CCC(CC1)N2C(C1CCCC12CCC2)=O Cc1nnc(O)c(C(N2CCN(C(c3cc(CO)ccc3Cl)=O)C(C)C2)=O)c1C c1(C(N2CC(NC(CC(c3ccc(C)cc3)C)=O)C2)=O)ccnc(F)c1Cl c1(C(=O)NCC(C)N(C(C2C(C#C)C2)=O)C)cc([N+](=O)[O-])cn1C C1(CC)C(NC(=O)COCP(C)(C)=O)CCCN1C(=O)C(C)=C(C)C CC1CCC(C)(C(=O)N(C)CC2CCCN2C(=O)C(C)C2CCOC2)CC1 C1(CNC(CSCCOC)=O)CN(C(c2ccc(-c3cccs3)s2)=O)CC1C C1(NC(c2ccc(OC)c(C)c2)=O)CC2(CCCN(C(=O)C(C)C3CCC3)C2)C1 N1(C(CNS(NC)(=O)=O)=O)CCC(NC(=O)CO)C(F)C1.c1ccc(Cl)cc1 c1(N2CC(C(N3C4CN(C)CC3CC4)=O)OCC2)ncnc2c1ccn2C CC1(C)OC(=O)CC1C(=O)NC1CC1CNC(=O)Cc1nc[nH]n1 c1(C(=O)NCC2=CCN(C(=O)CC3CC(F)C3)CC2)cc(Br)cn2ccnc12 C12(CC)CN(C(=O)C(C)C3CCCC3)C(CNC(c3ccccc3)=O)(C1)C2 N1(C(c2cnc(CC)o2)=O)CC(C2CN(C(=O)C(C)C)C2)C1.[SH](C)(=O)=O.N N#CC1CCC(C(=O)NCCCCCNC(=O)COc2ccc(Cl)cc2)CC1 C1(C(N2CCN(C(c3ccc(SCCC)cc3)=O)CC2)=O)CCC12CCCO2 C1(NC(=O)CCN2CCC(O)CC2)C2CC(O)C1N(C(C1CC3C=CC1O3)=O)C2 CC(C(F)C(=O)NCCCC1(NC(C2CC(F)(F)C2)=O)CC1)C(F)(F)F N1(C(CCN(C(C)C)C(c2cccc3ccoc23)=O)=O)CC2(CNC(=O)N2C)C1 C1(NC(C2C(C)C2)=O)CCN(C(c2nn[nH]c2C(F)(F)F)=O)C12CCC2 C(=O)(C1=NN(C2CC2)C(=O)CC1)NCC1CC(NC(COC)=O)C1(C)C C1(NC(C=CC(C)(C)SC)=O)CC(C2CCN(C(=O)C3=CCCOC3)C2)C1 C1(NC(c2cnn(C)c2-n2cccc2)=O)CN(C(c2cnn[nH]2)=O)CC(C)(C)C1 c1(CNC(C(c2nccs2)N(CC(CC)(F)F)C)=O)cccc(OC)c1 c1(CN2C(C(N(CC=C)CC=C)=O)CSCC2)ccc([N+](=O)[O-])cn1 Cn1ncc(C(=O)NCC2(CNC(C3(C)CCCS3)=O)CC2(F)F)c1N c1(C(N(CCC(C)NC(C2(C)CCCO2)=O)C)=O)cn(C)nc1C(F)F C1(NC(C=CCC)=O)CCCN(C(=O)CCc2ccc(C(=O)OCC)cc2)C1 N1(C(C2C(C)CCO2)=O)CCCOC(CNC(c2cccc(Cl)n2)=O)C1 c1(C(=O)NC(CC(C)NC(C(CCC)C)=O)C)ccc(S(C)(=O)=O)o1 c1(CNC(=O)NC(c2ccccc2O)CC)cnc(OC2CC2)cn1 C(=O)(CCC(C)(C)NC(c1cn(C2CC2)nn1)=O)NC(CCOCC)C C(=O)(C1CCOc2ccccc21)N1CCC2(C(NC(C=C)=O)CCC2)CC1 c1(CC)c(OC)cccc1NC(C1CN(C(=O)CO)CCO1)=O.CC(F)(F)F N1(C(C(C2CCOC2)OC)=O)CC=C(CNC(c2cc(C(C)=O)c[nH]2)=O)CC1 N(C1CCc2ccc(O)cc21)N1CCC(C(C)NC(=O)OC(C)(C)C)C1.CC CCCCCC(=O)N1CC(C(C)NC(=O)Cc2cccnc2O)C1 CC1CCCN(CCNC(CO)C(C)NC(=O)Cc2cccc(C(N)=O)c2)C1 N#Cc1ccc(C(=O)NC2CC23CC(NC(C2CC4(CCC4)CO2)=O)C3)cc1 CCC(CNC1(c2nnnn2CC2CC2)CCC2(CC1C)CC2)(CC)CCO C1(NC(C(CCSC)(C)C)=O)CN(C(=O)CNc2ccc(Cl)cc2)CC1C1CC1 CC(CC(=O)NCCN(C1CCCC1)C(c1ncn2c1CCCC2)=O)C(F)(F)F C=CCCCCCC(=O)NCC(CO)NC(c1cccc(OC)c1CC)=O c1(OC)ccc(Br)cc1C(C(=O)NC(C)(C)C)N(C1CCC(C)C1)C C#Cc1cccc(NC(=O)C(CO)NC(=O)CCCn2ccnc2)c1 CC1(C(=O)N)CCNC1=O.S(=O)(=O)(C(F)F)N1CCC1.C1CCN1C=O.C N1(C(C(CC)=CC)=O)CCCC(C)(NC(=O)CC2CCCN(C(C)C)C2)C1 C1(C2CC2)(CNC(CC(CCC)O)=O)CCN(C(c2cnc([N+](=O)[O-])n2C)=O)C1 Cc1ccc(F)c(C(=O)NC23CCN(C(c4cnoc4CC(C)C)=O)CC2C3)c1 N1(C(=O)CCc2nnc(C3CC3)o2)CCCCC2(CCN(C(=O)CC3CC3)C2)C1 C12(NC(C(c3cccc(Br)c3)C)=O)CCC1CN(C(=O)C=CCF)C2 CCC(CC(=O)NC1CCC1NC(c1ccc2c(c1)CC2)=O)C(C)(C)C c1(CN2CCC(N(C(C(=O)OCC)=O)C)CC2)cc(Cl)c(O)c(Br)c1 c1(C(N2CC3(CNC(c4ccco4)=O)CC(F)(C2)C3)=O)cnc2n1CCCCC2 N1(C(C2CCN(C(CCC=C)=O)C2)=O)CC2CC2(OC)C1 c1(C(C)C)cccc(CNC(=O)NN2CCCC(N3CCC3)C2)n1 C1(NC(=O)Cc2ccon2)CC2CC1N(C(c1ccn3ccsc13)=O)C2 S(=O)(=O)(c1ccc(NCCn2cccnc2=O)c(Br)c1)N(C)Cc1csnn1 CCC(CC(=O)NC1COCC1NC(c1ccc(S(C)(=O)=O)o1)=O)C(C)(C)C c1(CNC(N2CCC(C)(CC(=O)OC)C2)=O)ccc(C2CC2)cc1F c1(C(NCC)=O)ccc(C)nc1C1CC1.CCCCCOCC=O.C1CC1.N C1(C(=O)C2CC2)CCCCN1C(c1cnc(C(F)F)o1)=O.c1ccccc1 N1(C(C2=CC(C)C2)=O)C(C)CC2CN(C(=O)CCN3CCCS3(=O)=O)CC12.CC C(CO)(CC(F)(F)F)NC(c1cc(CNC(COC(C)=O)=O)nn1C)=O c1(C(N2C(C)(CNC(c3cn(CCC)nc3)=O)CCC2)=O)nc(OC)ccc1C c1(CNC(C(CC)NC(=O)CNc2ncccn2)=O)cc(C)cc(O)c1 C1(NC(c2c(CC)nns2)=O)COC2(CCN(C(c3cnc[nH]3)=O)CC2)C1 c1(C(N2CCN(C(CC(C=C)C)=O)CC2)=O)nc2c(cc1Cl)OCCO2 C(=O)(CC(CC)OC)N(CC(C)(C)CNC(=O)CC1(O)CCC1)CCC N1(C(C(C)C)=O)CCC(OC)CC1.C12(C=O)CC(C1)C2.C(C)(C)C.C=O C12(CNC(CCC(=C)C)=O)CC(CO1)N(C(=O)CC1CCC(O)C1)C2 c1(OC)cc(Cl)ccc1CC(=O)NCCN1CCC(NC(=O)C(C)CF)CC1 C(C(=O)N1CCOCC(NC(=O)CCS(C)(=O)=O)C1)(C(F)(F)F)OC(C)=O N1(C(CC(=O)OC)=O)CC(CNC(C2(F)CCOC2)=O)C(F)(F)C1 CCCC(C)CN(C)C(c1cc[nH]c1-c1ccccc1)=O N1(C(c2c(OCC)n[nH]c2)=O)CCCC2CN(C(c3cc(C)cc(Cl)c3)=O)CC12 c1(OC)ccc(S(N)(=O)=O)cc1C(=O)NC1CCCOC1 CC1CN(C)CC(C(=O)NC(C)(C)CCNC(c2cc([N+](=O)[O-])c[nH]2)=O)O1 C(C1=NOC2CCCC12)NC(C(C)(C)NC(C12CCC(OC)C1C2)=O)=O C(C(CC)(CC)C(=O)N(C1CCOC1=O)C)NC(C1N(CC)CCC1)=O c1(NC(=O)C(C(C)O)N(C)C)c(Cl)ccc(C(=O)N(C)CC)c1N c1(C(=O)NC2CC3CC2N(C(C2SC4C=CC2CC4)=O)C3)noc2c(F)cccc12 C1(C(=O)OC)(CNCCc2ccccc2)C=CCC1.C(=O)C(C)c1ccsc1 N1(C(C2C(CC)C2)=O)CC2CC(C1)CN(C(=O)CCOC(C)CC(C)C)C2 C(=O)(CC(C)(C)C)OC.C1(C=O)CC2(C1)CN(C(=O)C=C1CCC1)C2.N N1(C(C2CC3(CC(=C)C3)C2)=O)CC(CNC(=O)CC=C(Cl)Cl)N2CCC1C2 Cc1[nH]c(C)c(C(=O)NCC2CCN(C(C3COC(=O)O3)=O)C2(C)C)c1C CC1(C)CC(CNC(C2C3CCN2CC3)=O)N(C(c2ncncc2Cl)=O)C1 CCC(C(=O)N(C(C)CCNC(=O)CCSc1nccn1C)C)C1CCC(=O)N1 c12cc(C#N)ccc1O2.C1(CC)CN(C(C)=O)CCN1S(=O)(=O)CCCl c1(C(=O)NC2CC3(C2)CN(C(=O)CCn2cnnn2)C3)cc(F)c(F)cc1F c1(CC(N2C3C(NC(CCSC)=O)C(C3)C2)=O)noc2ccc(Br)cc12 N1(C(c2c(CC)scn2)=O)CCC(C)C(C)C1.N1(C(C(=O)N)C)C(C)CCC1C C#Cc1ccc(F)cc1C(=O)NC.C1(F)CCC1.c1(C=O)conc1C(C)C C1(NC(CC(=O)OC)=O)(CO)CCCN(C(c2cc(N(C)C)ccn2)=O)C1 CC1(NC(c2cccn2C2CCCC2)=O)CCCN(C(c2cccnc2N)=O)C1 Cc1cc(C(=O)NCC2CN(C(=O)CCCOc3cccnc3)C2)cc(=O)n1C Cc1cc(C(=O)NC2CCOC(c3cccc(F)c3)C2)c2c(n1)CCCC2 CCCC(O)C(CO)NC(c1ccc(CNC(c2ccc(C)nc2)=O)nc1)=O Cc1cc(=NCCC(F)(F)F)[nH]c(N2CC3CC(C2)N(C)C3)n1 c1(C(N2CCC(O)(CNC(C3CCC4CC4C3)=O)CC2)=O)ccc(Cl)c(F)c1F C1(CCNC(=O)CCc2cncs2)CN(C(C2CC2(F)F)=O)CCO1 C(C(O)CNC(=O)CSC(F)F)N(C(=O)CC1CC1(C)C)C Cc1ccnc(C(N2CCC(C)C2C(=O)NCC(n2cccn2)C)=O)c1N C(CCC1CCC1)(C(=O)N1CCC(CSC)C1)OC(=O)C(F)(F)F C1(C)(CNC(C2C(C(C)C)C2)=O)CC(F)(F)CN1C(=O)C(N)=O CCCC(CC)CCC(=O)NC1(CNC(c2ccnc(F)c2O)=O)CCCC1 C1(CC(=O)NCC(F)CO)C2CCCC2N1C(=O)CN1CCCC1 C12(CNC(c3cc(N(C)C)n[nH]3)=O)CC(CN1C(=O)C(c1ccccc1)F)C2 S(=O)(=O)(c1ccc(Br)cc1NCC(CO)C1CCC1)NCC(CC)CO c1(N2C(CNC(=O)C=Cc3nccs3)CCC2)ncnc2ccc(F)cc12 C(C(C)(C(=O)NCC1CN(C(=O)CCCOC(F)(F)F)CC1O)OC)OC C12(C(C(=O)O)NCc3cnsc3Br)CC3CC(CC(C3)C1)C2 [SH](=O)(=O)c1ccc2c(c1)OCO2.C1(C(CN)=O)(C(=O)OC(C)(C)C)CCCC1 C1(CC(=O)NCC(C2CC2)NC(c2ncccc2Br)=O)CCCNC(=O)C1 c1(C(=O)NC2CCN(C(CN(C)CC)=O)C2C)ncccc1S(C)(=O)=O c1(C(=O)NC2(CNC(C(Br)=C(C)C)=O)CCCCC2C)cccc2c[nH]nc12 C(=O)(CCS(=O)(=O)CC(C)C)N(C1CCN(C(c2cnc(C)n2C)=O)CC1C)C C1(C(=O)N(C)Cc2cccnn2)(CC)CCN(CC2C=CCCC2)CC1 c1(C(N2CCCC(N(C)C(C3CCC(F)(F)CO3)=O)C2)=O)ccc([N+](=O)[O-])cc1 Cc1ccc2n[nH]cc2c1C(=O)NCCN(CC(C)O)C(c1ccnnc1O)=O c1(CC(C)OC)nc(CC2CC2(C)C)n(-c2ccc(Br)nc2)n1 N1(C(c2cc(CCC)ncc2)=O)CCN(C(=O)C(C)(C)F)C(COC)C1 C(=O)(CCCC(=O)NCC1CC1NC(C1(F)CC2(CCC2)C1)=O)N(C)C N1(C(CSCCS(N)(=O)=O)=O)CCC2C(C1)CN2C(=O)CC.C1CCCOC1.O C=CC1(C(=O)NCC2(O)CCCOC2)CCN(C(=O)Cc2cn(C)cn2)C1 N1(CC)CC2(CN(C(c3cc(=O)n(C)cn3)=O)CC(F)(F)C2)C1 c1(C(=O)N)cccnc1-n1nc(C)cc1C.C(C(=O)NC(C)C1CC1)=C(C)C c1(CCCC#N)cn(C2CCC(C(=O)NC(c3cccnc3)C3CC3)C2)nn1 c1(OC(=O)NC2CCN(C(C)C(=O)Nc3ccccc3)C2)cc2c(s1)CCC2 C1CCN(C(C2(C)CC2)=O)CC1.c1(C(=O)NC2CC2)cc[nH]n1.[nH]1cccn1 c1(-n2cc(CC3CN(C(C4(C)CC4(Cl)Cl)=O)C3)nn2)ccccc1[N+](=O)[O-] C#CC1(O)CC(C(=O)NC2CCCC2)C1.n1(CC=O)cc(C2CCC2)nn1.C N1(C(CC2C(C)OCC2)=O)CCN(C(=O)CS(=O)(=O)NC2CC2)CC12CC2 C1(NC(Cn2nc(C)c(C)c2C)=O)C(C)CCN(C(C2CCCCC2O)=O)C1C C1(NC(CNC(=O)C2CC2)=O)CCN(C(=O)Cn2cc(CO)nn2)C1 N1(C(CSC(C)(C)C)=O)CCC2(CC1)CC(NC(C1CCC3(CC1)CC3)=O)C2 c1(CNC(=O)CCOCCNC(c2cccnc2)=O)ccn2nccc2c1 C1(C(NC2CCN(C(=O)C)C2)=O)CC(=O)NC(=O)C1.c1cncc(Cl)n1.CC C1(C(=O)NCCN(C(C(CC)SC)=O)C)CCN(Cc2ccncc2)CC1 C(=O)(C1=NN(C)C(=O)CC1)N1CCCC1(C)C.CC(C)CC(C)(O)C(=O)NC N1(C(C(C(C)C)SC)=O)CCCC2CN(C(c3conc3C)=O)CCC12 CC(=O)CCC(=O)N(C1CN(C(c2cnn(C)c2)=O)C1)C C1(NC(CC(C)(C)n2cc(CCCSCC)nn2)=O)Cc2ccccc2C1O C(Cc1ccccc1)(CCC(=O)OC(C)(C)C)NCc1n(C(C)C)nnn1 c1(OC)ccc(CN2CCC2C(=O)NC(c2cccnc2)C(C)C)cc1 Cc1ccc(CNC2CC(CC(=O)Oc3cc(F)ccc3C(F)F)C2)cc1C#N C1(C(=O)NCCC(C=C)C)CC12CCN(C(=O)C(C)(O)C1CCC1)CC2 C(C(CC(F)(F)F)NC(=O)CC(C)(C)C#N)NC(Cc1nc(C)sc1C)=O C(=O)(C1CNC(=O)c2ccnn21)N1C(CNC(=O)CCC2=CCCCC2)C=CC1 c1(CC(=O)NCC2(COC)CN(C(=O)CCC)C2)coc2cc(C)ccc12 c1(COC)ccc(NC(c2cnn(CC(=O)N(C)C)c2)=O)c(N)c1 C1(OC)(CNS(=O)(=O)CC2NC(=O)NC2=O)CCC(C)(C)CC1 N1(C(c2n(CC)nc(C)c2)=O)CCN(C(=O)C(C)c2cc[nH]n2)CC1CCO c1(C(N(CCC(=O)NC(CCOCC)C)CCO)=O)cnn(C)c1Cl c1(CC)csc(C(F)(F)C(=O)N(CC(N2CCCCC2)=O)C(C)C)n1 Cc1c(C(C)C(=O)OCCOCCCN)cnn1C c1(CNC(C2N(C(c3cc(C)oc3C)=O)CCC2O)=O)cnnc(C)c1C N1(C(C2(C#C)CCN(C(=O)C(C)CCCCC)C2)=O)CCC(F)(C#C)CC1 CCCCS(=O)(=O)CC(=O)N1CC2CCCC2(NC(=O)C(O)C2CCC2)C1 c1(C(=O)NCC(c2ccc(F)cc2)O)ccc(Cl)nc1NC(c1ccccc1)=O Cc1ccc(I)c(C(N2CCC(C(=O)NC(C)C)CC2)=O)c1 N1(C(C)C(=O)NCC2C=CCC2)CCCS1(=O)=O.C1(C=O)CC(C)(O)C1.N CS(=O)(=O)CCCC(=O)NCC=CCNC(c1csc([N+](=O)[O-])c1)=O c1(C(N(CC(C)NC(C=CCC)=O)CC)=O)cc(C)nn1C CC(CN(C)C(c1csc(F)c1)=O)C(=O)N1CCCC1C(N)=O c1(C(N(C2CCCCC2NC(=O)C2=CCOCC2)C)=O)ccc(OC(F)F)nc1Cl C1(NC(CSCCC)=O)C2CN(C(C3(c4ccnc(Cl)c4)CC3)=O)CC12 n1(CC)ncc(NC(C2CC2NC(=O)C2CC2)=O)c1C.c1cc(C)nn1C c1(C(=O)NC(COC)(C)C)c2c(nn1C)CCN(C(C1CCC(=O)NC1)=O)C2 CC1(C)CCC(C(=O)NC2CCOC(CNC(=O)C(C)(C)C3CCC3)C2)CC1 C#Cc1ccc(C(=O)NCCC(O)C(=O)N2CC(C)(C)C2)cn1 C1(CC(=O)NC2C=CCN(C(c3nccc(C)c3)=O)C2)COC(C)(C)CO1 c1(C(=O)NCCC2N(C(c3nc(C)nn3C)=O)CCCC2)[nH]cc2c1CCC2 c1(C(N2CCCC(NC(=O)CC3CCOCC3)CC2)=O)cc2cn[nH]c2cn1 N1(C(C(CCC)F)=O)CCN(C(c2sccc2C#N)=O)CC1CCC c1(C(N2C(CN(C)C(C3(C)CNC(=O)C3)=O)CCC2)=O)ccc(=O)oc1 C1(C(C)NC(C(C=C)C)=O)CCCCN1C(=O)CN1CCCCCC1 C1(c2cncc(C(=O)OC)c2)CCN(N(C)C(C)c2cnn(C)c2)CC1 c1(CC)occc1C(N1CCC(C(N2CCC(C(N)=O)C2)=O)C1)=O c1(SC)cc(C(N2CCC(n3cc(COCC(N)=O)nn3)C2)=O)no1 C1(C(N(C)CC2N(C(c3nc(C(C)C)sc3)=O)CCOC2)=O)CCC2(CC1)N=N2 C(CN=c1[nH]c(Cl)nc2c1CC(C)CC2)(C1CCCCC1)NC(CCSC)=O c1(C(=O)NC2CC(NC(C(c3ccccc3)SC)=O)C2)coc2c1CSC2 Cn1nc(C(=O)NCCCCNC(=O)CC(C)(F)F)cc1-c1ccccc1 Cc1cc(C2(C(N3CCC(C)C3)=O)CC2)on1.C1(C(=O)N)(C(F)F)CCOC1 CC1(CN(C)S(=O)(=O)NCC2CCCN2CC(F)F)CCC(F)(F)CC1 N1(C(c2[nH]cc(C#N)c2)=O)CC2CCC(N=c3[nH]c4c(F)cc(Cl)cc4s3)C2C1 c1(N(CCCCCO)C)ccc(S(=O)(=O)N(CC(C)(C)CO)C)cc1C#N C1(NC(C2C(C)C2C)=O)CCCCN(C(=O)CC2CCCN2C(C)C)C1 N1(C(CCC(=C)Cl)=O)CCC(C2CC2)(NC(=O)C(C)C(=O)c2ccccc2)C1 c1(C(N2CCC(N(CCC)C(c3ccncc3O)=O)C2)=O)ccc(C)c(C)n1 C1(C(=O)NCCC2N(C(c3cc(C)c(F)cc3)=O)CCC2)CC12CCOC(C)C2 C1(C(=O)NCC(CCNC(C(C(C)(C)O)F)=O)O)CN2CCCN1CC2 C1(NC(c2c(CC)n[nH]c2)=O)C2CC(NC(=O)C(C)N3CC(C)C3)CC12 N1(c2c(OC)cncn2)CC(NC(c2ccc(C(F)F)o2)=O)CC2(CC2)C1 c1(NC(=O)C(=O)N(C2CC2c2ccsc2)CC2CCOCC2)cccc(Cl)n1 CC(O)CCC(=O)N1CCC(C(C)NC(c2cccc(SCC#N)c2)=O)C1 C=C(C)CC(C(=O)OC)NC(C1CC(O)CN1C(C1CC(=O)N(C)C1)=O)=O CC1C(NC(c2ccc(CO)c(F)c2)=O)CCCN1C(=O)C=C(Cl)Cl C=CC(C)(C)CC(=O)N1CCC(OCC(=O)NC(c2ccncc2)(C)C)C1 C1(C(N2CCC(=CC)CC2)=O)CC2(CCC(F)(F)CC2)CO1.C(C)(C=O)SC.N Cc1nncc(C(=O)NCC(=O)NCC(=O)N(CC(C)C)C2CC2)c1C c1(OC)c(F)cc(C(=O)NC2CCN(C(=O)C=Cc3cccnc3)C2C)cc1Cl Cc1cc(=NCC(C)N2CC(C)OC(C)C2)[nH]c(=NCC(C)n2ccnn2)[nH]1 c1(N2CCC(=C)CC2)nc(NCc2cncn2C)c2ccsc2n1 c1(OC)cc(NC(C2CC2C(=O)Nc2ccnc(Cl)c2Cl)=O)cc(C#N)c1 N1(C(C(=O)NCC2CCCO2)C2C(C)C2)CCC(n2cc(Cl)cn2)CC1 n1(CC)cc2ccc(C(N3CCC3CNC(=O)CCc3cnco3)=O)cc2n1 c1(OC)ccccc1C(O)C(=O)N1CCC1.c1cccc(Cl)c1.C(=O)C(O)C=C.C c1(CC)cnc(C(=O)NC(C)C(=O)NCCc2cocn2)nc1 c1(C2N(CC(=O)Nc3ccc(Br)cn3)CC2)ccc(Br)cc1Cl CCC(CCC(=O)NCc1nc(C)co1)NC(=O)CCCC(OC)OC C=CCCC(F)(F)C(=O)NC1CC(OC)CN(C(c2c(C)ccn2C)=O)C1 c1(C(N2CCC(C3CN(C(CCCC)=O)C3)C2)=O)c[nH]c2cc(C#N)ccc12 C1(NC(CSCCCC)=O)CC2CC1N(C(C1C3CCC1(c1cnco1)C3)=O)C2 c1(C(=O)NCCC2CCN(C(C(C)NC(C)=O)=O)C2)cccc(C#N)c1 CON(CCC(=O)N1CCC1C1CCC1)C(=O)C1(C)CCC(=O)NC1 c1(C(N2C(CCCNC(CCCCCC)=O)CCC2)=O)cnc2ccnn2c1O c1(C(N2CCC2)=O)ccc2c(c1)C(C)(C)C(=O)N2.CC(CC1CC1)C(=O)N c1(OC)ccccc1C(=O)NCCN(C)C(c1c(C)c[nH]c1CC(N)=O)=O C1(NC(C2CCC(C)O2)=O)COCCC1NC(C1(N2CCCC2)CC1)=O N1(C(c2cn(CC)nc2)=O)CC(NC(C2CCS(=O)(=O)C2)=O)CC2(CC2)C1 C1(CNC(CN(C)C)=O)CN(C(C2(C)CCC(=O)NC2)=O)CC2(CCC2)O1 C1(CNC(c2c(C)ccnc2)=O)CCCCN(C(c2ccn(C)c2)=O)CC1 c1(C(N(CC(C(=O)OCC)C)C)=O)ccc2c(c1)CCN(C1CCCSC1)C2 C(=O)(C(C)C(C)(C)C)NC1CCN(C(CCCn2c(C)ncc2)=O)C1C(C)(C)C c1(CC)ccc(C)cc1C(=O)NC1CS(=O)(=O)CC1.c1(C=O)cncs1.N c1(CCC(N2CCC2)=O)n[nH]c2c1CCCC2.C=C1CC(C(F)(F)F)(C(=O)N)C1 N1(C(C(C(CC)C)C)=O)CC(NC(C2CN(C)C2)=O)C2(CCCC2)C1 C(CC(=O)NOC1CCCCC1)N(C(=O)C(C)O)CC(=O)OC c1(C(N(CC(CC)NC(C2CCC23CCC3)=O)C)=O)cc(F)cc(F)c1 c1(C(N2CC(CCNC(C3CCN(CCC)CC3)=O)C2)=O)cnc(C)nc1OC N1(C(CC2CCN(C(C)=O)C2)=O)CCCC(NCCN2CCCC2)CC1 C(CCC(CO)NC(C1CC12CC2)=O)NC(c1c(C)cns1)=O c1(C(N2CCC(CCNC(C3CSC3)=O)C2)=O)cnc(C2CCCC2)nc1O C(=O)(CC(O)CC(C)(C)C)N1CCCC(N(C(=O)C=Cc2cc[nH]n2)C)C1 CCCC(CCC)CC(=O)NC(C)(C)C(C)NC(c1cc2[nH]nc(C)c2cn1)=O N1(C(C=CC(CC)C)=O)CC(C)(C(=O)N)CC1(C)C.C1(CCO)CN(C)C1.C c1(C(N2CC(C(C)NC(=O)CCCCF)OCC2)=O)cncn(C)c1=O CN1CCCC1CCC(=O)N(CC(=O)NCc1cnn[nH]1)C1CCC1 CC1CCC(NC(=O)CC2CCCC(=O)N2)CN1C(=O)C(=O)C(F)(F)F N1(C(c2n(CC)nc(C)c2)C(=O)NCc2ccco2)CCc2noc(N)c2C1 C(=O)CC(C)(C)n1ccnn1.C(C(O)CN(C)C)OCC(C)C.C(C)(C)C.C N1(C(C(COC)NC(=O)C(=O)Nc2ccc(F)cc2C)=O)CCC2OCCC2C1 CC1CCCC(C(=O)NCCNC(c2cc(C#N)cs2)=O)O1 C1(C)(C(=O)NC2CCN(CC)C2C(=O)NC)CCC(=O)NC1 CCCCCC(C(=O)NCC(C)(C)CN(C(=O)COc1cc(C)on1)C)C(C)C N1(C(C(CCCC)O)=O)CCC2CN(C(=O)C(C)(F)F)CC2C1 c1(NS(CC)(=O)=O)ccc(C(=O)NCCC2CCC(C(F)(F)F)O2)cc1 N1(CCNC(c2cc(C)[nH]n2)=O)CCN(C(=O)CC2CCCC2(F)F)CC1 C12(CNC(c3ccns3)=O)CCCC(CN1C(c1cncc(Cl)c1Cl)=O)C2 S(=O)(=O)(c1cccc2nccnc12)NC1C(C(=O)Nc2c(C#N)ncc(C)n2)C1 c1(C=O)ccc(S(C)(=O)=O)o1.CC1CCCN1C(=O)C.N1(C=O)CCCC1.N C1(NC(C(CC)C(C)C)=O)C2COCC1CN(C(=O)Cc1ccccc1)C2 C(=O)(CCC(C)(C)C)NC(CN(C(C1(COCC)CCOCC1)=O)C)C.O C1CC(=O)N(C)C1=O.c1(C(=O)NCC(CC)NC(=O)C)cnc(OC)s1.O CCC(C)C(C(=O)N1CC(O)CC1CC)N(C(=O)Cc1c(C)ncnc1C)C CCC(C(=O)NCCS(N)(=O)=O)n1ccnc1.C1CC(=O)N(C)CCCO1 N1(C(c2nc(C)oc2C)=O)CC(C2CCCN(C(C3OC(C)CC3C)=O)C2)C1 C12(C(N3CC(O)C3)=O)CCC(CC1)OC2.C(C(C)(C)C(=O)NC)OC(C)C.C CCC(C#N)C(=O)N(CC(O)CN(C(=O)C(N1CCSCC1)C)C)C O=C(CCCC(=O)N1CCCC(N2CCCC2)C1)Nc1ccccc1 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c1(C(N(C2CCCN(C(c3ccn(C(C)(C)C)n3)=O)C2)C)=O)cc(O)nn1C C1(C(N2C(CNC(Cn3ccc(=N)[nH]3)=O)CC2)=O)CCC(=O)NC1 N1(C(C2(C)CCC(=O)NC2)=O)CCC2(CCN(C(c3cccc4occc34)=O)C2)C1 C12(CNC(C(CC)OCC)=O)CCCC1N(C(c1cnc[nH]1)=O)CCC2 CC1C=C(C(=O)N2CCC(CNC(=O)CN3CCCC3=O)C23CC3)CC1 N1(C(C(CC)O)=O)CC(Oc2ccccc2)CC1C(=O)NC.c1nc(C)c(C)[nH]1 c1(C(=O)NCC(C)CNC(=O)OC(C)(C)C)ncn(-c2ccccc2)n1 C(CC(C(=O)N)NC(=O)C(C)CC1CCC1)SC.C(C(C)(C)O)c1ccccc1 N1(C(c2ccc(C(N)=O)[nH]2)=O)CCC(NC(=O)CN2CC3CC3C2)C(CO)C1 C1(C=O)CCN(C)C(=O)C1.N1(C(c2c(OCC)scc2)=O)CC2CC2(C)C1 Cc1ccc(CC(=O)NC(CNC(c2ccsc2)=O)CO)s1 Cc1cc(NC(C)(C)C)ccc1SCC(C)C(=O)NS(C)(=O)=O C#CC1CC2(CC(C(N3CC(NC(c4cc(C(C)=O)on4)=O)C3)=O)C2)C1 CC1CCC(C(=O)NCCC(O)CO)N1C(=O)Cc1cnnn1C c1(N(C2CN(C(C)=O)CC2O)C(=O)C(N2CCSCC2)C)ccc(F)nc1 c1(C(N(C2CCCC2)CCNC(c2occc2F)=O)=O)ccc(OC(F)F)cc1 C1(C(=O)OCC)CCN(C(=O)CCC2CCCN2C(=O)C(OC)O)C1.C Cc1cc(CN2CC3CCN(S(=O)(=O)CCCCl)C3C2)cc(F)c1F N1(C(C2C(C)(C)C3CCC2C3)=O)CCC2CCN(C(C34CC(C3)C4)=O)CC12 c1(C(=O)NCC(CNC(CC(C)N2CCCC2=O)=O)(C)O)cnn2cccnc12 c1(CCC(=O)NC2C(NC(C3C(OC)C3)=O)CCC2)nc2ccccc2o1 c1(-c2cn(CC)nc2)noc(C)c1CC(N1CCC(CN)CC1)=O C1(CNC(c2cccnc2C(F)(F)F)=O)COCCN1C(c1cscn1)=O N1(C(c2cncnc2)=O)CCCCC1C1CCCN1C(=O)CCc1cccs1 CCC(C)C(C(=O)NC(C)(C)C=CC(=O)NCCC(F)CN=[N+]=[N-])OC CCC(CO)C(=O)NCC(CC(C)C)NC(=O)C=CCOC.c1ccccc1 N1(C(C2C(C)C2C)=O)CCC2(CCCC2NC(c2cc(C3(C)CC3)on2)=O)CC1 c1(N2CC(C#N)C(NS(=O)(=O)c3ccccc3Br)C2)ncnc2c(F)cccc12 N1(C(c2cc(C#N)oc2)=O)CCC2(CNC(C3CC4(CCC4)C3)=O)CCCC12 c1(C(=O)NC(CCCNC(C(CC)N(C)C)=O)C)c(C)nn(C)c1C(F)F Cc1nc(Cl)nc(Cl)c1NC(C1CC1C(=O)Nc1ncc(Cl)cn1)=O c1(C(=O)Nc2ncn(C)c2)cc(-c2cccc(CN(C)C)c2)cc2c[nH]nc12 CC1CN(C(C2CCN(C)C2)=O)CC(C)CN1C(c1cnn2cccc(Cl)c12)=O CC(C)(C)CC(C)(C)C(=O)NCC1CN(C(=O)Cn2cc[n+](C)c2)C1 C(C)(C)(CC(=O)NC1CCN(C(=O)Cc2cccc(C(C)C)c2)C1C)OC N1(C(CN2CCN(C(COC)C)CC2)=O)CCC2(CC1)OCc1ccccc12 c1(C(=O)NC(CNC(c2nc(COC)nc(Cl)c2)=O)C)ccc2nnnn2c1 C1(N(C(Cc2c(C)ccnc2)=O)C)CCCCN(C(c2cc(Br)n[nH]2)=O)C1 C1(NC(C(c2cccc(C#N)c2)C)=O)CCN(C(=O)C=C2CCCC2)CC1F c1(C(=O)NC2CN(C(c3nc(C)oc3)=O)C(C)CC2)cccc2c1C(=O)CC2 CCC(CC(=O)N1CC(C(C(N2CCCC2CF)=O)OC)C1)C(C)(C)C CCCC(C(=O)N1CCC(C(F)F)C1)S(N)(=O)=O.c1(C(=O)N)ccc(N)c(Cl)n1 CC1CC(C(=O)NOCc2ccccc2)CCN1C(c1coc(CO)c1)=O c1(C(=O)NCC(C)NC(=O)C(O)C2CCCC2)cc2sccc2s1 C1(N(C(c2cc(C)ncn2)=O)C)CCCN(C(=O)CC2CSCCO2)CC1 c1(C(=O)NC23CC(NC(C4(C)C(C)OCC4)=O)(C2)C3)ccc2c(c1)ncn2C N1(C(CC2(C)CC2(Cl)Cl)=O)CCCCC2(CCN(C(c3cc(Cl)c[nH]3)=O)C2)C1 C1(NC(=O)C=CC2CCOC2)COC2CCOC12.c1(C(=O)N)ccc([N+](=O)[O-])s1 CC(C(C)NC(C1(C(F)(F)F)CC1)=O)NC(=O)CCC1CC1(Cl)Cl N1(C(C(C)C#N)=O)CCCC(C)(C(N2CCOC(C3(C)CC3)C2)=O)C1 c1(C(=O)NC2CCCC2O)cc2ccc(Cl)nc2s1 C1(OC)(CNC(c2cnsn2)=O)CN(C(c2cn(CC(F)(F)F)nn2)=O)C1 c1(C(N2CCC(NC(COCC)=O)CC2COC)=O)ccc2nc(O)[nH]c2c1F c1(CCC(N2CCN(C3CN(C(CCC(=C)Cl)=O)C3)CC2)=O)cc(C)ccc1C N1(CC(=O)NCCCC(C)NC(c2cncc(C)c2)=O)C(=O)CCCC1=O C(=O)(C1=C(C)CCC1)NC1CN(C(C(CC)NC(c2ccco2)=O)=O)C1 Cc1cc(Cl)ncc1C(=O)NC1CN(C(=O)CC2COCCO2)CCC1F C1(NC(C2CCC3CC3CC2)=O)CCN(C(C2CC3(CSC3)C2)=O)C12CCCC2 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CCC(C)C(C(=O)N(C1(CC)CC1)C)NC(c1nc(O)sc1C)=O CCCC(CC)CC(=O)NCC(C(C)(C)C)NC(=O)CSc1ccccc1 C1(C(C)C)CC(NC(=O)C(CC2CCCC2)NC(C2CCCN2C)=O)CO1 C12(NC(c3cocn3)=O)COCCC1CN(C(=O)CCn1cc[nH]c(=O)c1=O)C2 C1(CC(N2CC(C(=O)NC)C2)=O)CCC(NC(=O)CC2CCCN2C)C1 C12(C(N3CC(NC(C(CC=C)CC)=O)C(O)CC3)=O)CCCN(CCC1)C2 C(=O)(CS(=O)(=O)C(C)C)NCC(=C)CCNC(=O)CSCCOC CC(C)(C(=O)NCCCCCNC(=O)CCC1CCCC1)n1cc(Cl)cn1 c1(C(=O)NCC2(NC(COCCC)=O)CC2)n[nH]cc1OC O=C(C1OCCc2ccccc21)NC1CCN(C(=O)C(c2ccc(O)cc2)=O)C1 n1(C(C)C)nccc1C(=O)N.C1CCCN1C(C1CC1(C)C(F)(F)F)=O.C c1(C(N2C(C)C(NC(C3CC34CCSCC4)=O)CCC2)=O)nc(O)nc(O)c1N N1(C(c2cc(CC)[nH]n2)=O)CCC2(CCN(C(=O)C(C)(C#N)CC)CC2)C1 n1(CC(=O)NC2CN(C(C(C)(C)N(C)C)=O)CC2(C)C)ncc2cccnc12 C(CCC(C)C(=O)NCC1CN(C(c2ccc(Br)cc2)=O)CC12CC2)OC C1(NC(=O)OC(C)C)CCC(N(C)N2CCOc3ccc(F)cc3C2)CC1 N1(C(C2CC(N(C)C)C2)=O)CCCC(O)(CC(=O)Nc2ccccn2)C1 c1(C(N2C(CNC(CN(CCC)C)=O)C(C)CCC2)=O)ccc2cncn2c1C C(=O)(C(C)(C)CC(F)(F)F)NCC12C(CN(C(C3CCCN(C)C3)=O)C1)C2 C(=O)C1CCCc2ncnn21.c1(C(=O)OC)cc(C(=O)N(C(C)C)C)c(C)o1.N 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C1(C(N(CC(C)NC(C2CCC(=O)N(C)C2)=O)C)=O)CN(C)C(=O)CCO1 N1(C(c2cncc(CC)c2)=O)CCC(NC(=O)C(C)C2CCCC2)C(O)C1 c1(C(N2C3CN(Cc4cccc(C(=O)OC)c4)CC32)=O)nccc2[nH]ccc12 C(=O)(C(C(=O)OC)OC)N(CC(=O)NCCOCC(=C)C)CC Cc1nn(C)c(C(=O)NCC2C3CN(c4nnc(CO)s4)CC23)c1Cl C(=O)(C#CC1(C)CC1)NC1C(CNC(c2c(C)nc(CC)s2)=O)CC1 C(=O)(C1=CC2(CCN(C(=O)CCC3CC3C)C2)C1)N1CCCC(C)(CC)C1 C1(O)(C(CNC(CCOCCCOC)=O)C)CCN(C(=O)CCc2nncs2)C1 N1(C(C(N2CCSCC2)C)=O)CC2(C1)CN(C(=O)C=CBr)CC2CO c1(CCC(=O)N(CCC(C)NC(=O)C(C)Cn2cccn2)C)cnccn1 CC(C)CCCCC(=O)N1CCCC(C(=O)NCCCC(=O)N(C)C)C1 CCCC(C)C(CO)NC(=O)CCN(C(c1cc(C)c(C)cn1)=O)C(C)C c1(C(=O)NCCCCC(=O)NC(c2ccccc2)C(C)N(C)C)ncc(F)cc1F c1(C(N2CC(N(C(CC)=O)C)C(O)C2)=O)ccc2c(c1)CCCCN2 CP(C)(=O)c1cnn(CC(=O)NC2CN(C(c3ccn4cnnc4c3)=O)C2)c1 CC(c1cccs1)=CC(=O)NCC1CC1(F)F.C(=O)C(O)CN1CCCC1.C CC(C)C(C)CC(=O)NCCC1CCCN1C(=O)CCC1CCC(=O)N1 c1(CC(C)C)ccc(C(=O)N)cn1.C1(C(N(CCC)C)=O)CCCC1C(C)C C12(C(N3CC4N(C(c5cc(C)c(C)s5)=O)C(C4)C3)=O)CCCC1CC(=O)C2 CCS(=O)(=O)CC1CN(C(=O)CC2CC2)C1.C1(C(CC)C=O)CCC(C)CC1.N c1(C(=O)NC(c2ccccc2Cl)C(F)F)nnc(O)c2ccccc12 N1(C(C(C(C)(C)C)NC(C(CC=C)C)=O)=O)CCn2nncc2C1 N1(C(CC2(OC)CCCCC2)=O)CCCC(NC(=O)CCCC2(C)N=N2)C1C c1(NC2CCC(NC(c3nc(C)oc3)=O)C2)ncnc2onc(C)c12 N1(C(C(C)SCC)=O)CCC2CCC(NC(=O)C(=O)N)C12.CC.C(C)=O C1CCC(OC(C2(SC)CCC2)=O)C1.C1(C=O)CN(C=O)C1.C(C)(C)C Cc1cc(C)c(C(=O)N(C2CC(NC(=O)C(=O)N(C)C)C2)C)cc1C N1(S(c2ccc(OCC)cc2)(=O)=O)CC(C#N)C2(C1)C(=O)Nc1ccccc12 c1(C(=O)NC2COCC2NC(C2C=CCC2)=O)cncc2sccc12 CCCCS(=O)(=O)CC(=O)N(C1CN(C(=O)Cn2ccc(C(F)F)n2)CC1F)C C(=O)(C1=CCCCCC1)N1CC(NC(C2(C(C)(C)C)CCCC2)=O)C(C(F)F)C1 CC1OCCN(C(=O)CCC2(C)CN(C(=O)COc3ccsc3)C2)C1CO c1(CNC(C2CCN(C(CCOC)=O)C(CN)C2)=O)cccc([N+](=O)[O-])c1 c1(C(=O)NCCN(C(=O)C(C)CS(C)(=O)=O)CC)cn2cccnc2n1 CCCCCCC(F)C(=O)N(CCC(C)NC(c1cn(CCC2CC2)nn1)=O)C O=C(COc1ccccc1Cc1cccnc1)NNC(=O)C1(O)CCSC1 C(CN=c1[nH]c2cccc(F)c2s1)(C1CC1)NC(C1(C=C)CCC1)=O C12C(CNC1C(=O)N(C(C)C(C)S)CCO)O2.CC=CC CC(C)(CC1CCOC1)C(=O)NC1CCC1C.C(=O)(CCSC(F)(F)F)N c1(C(=O)NC(CNC(c2n(CC)ncc2)=O)C(C)C)cnc(C)cc1C c1(OCC)ccc(N)c(C(=O)NCC(C)(O)C)c1.c1(C=O)cccc(Cl)c1F n1(CC=O)nc(C)ccc1=O.c1(OCC)ccccc1CCNCC.CC.O C(C(=O)NC(C)C=CC(=O)N(C)Cc1cscn1)(C1CC1)OC Cn1nnc(CNC(C2CC(C3CC3)C2)=O)c1C(=O)NCc1cncs1 CC1CN(C(C2C(F)(F)C23CCC3)=O)CCCN1C(c1ccc2occc2c1)=O C1(NC(c2ncccn2)=O)CN(C(=O)CC23CC(C2)C3)CCC1C(F)(F)F C1(C)(CNC(c2cc(CC)ncn2)=O)CCN(C(C2(CCO)CC2)=O)CC1 C(=O)(CC(C)CC(=O)OC)NC(CN(C(c1c(C)cc(C)cc1C)=O)CC)C Cc1cc(S(=O)(=O)NC2(c3ccccc3)CCOCC2)sn1 C1(CNC(=O)CCCOC)CCN(C(=O)CC(F)F)CC1.C1(C=O)CCC1 Cc1cc(CNC(=O)OC(C)(C)C)n[nH]1.c12ccc(o1)C(=O)NC2 c1(C(N(C)CC2(O)CN(C(C(COC)(C)C)=O)C2)=O)nncc2c1CCCC2 CC(C)CC(O)C(=O)NC12CC(C)(C1)C2.c1(C(=O)N)ccccc1.N(C)C c1(OC)ccnc(NC2CCN(C(=O)C(C)CC3CCCC3)CC2)n1 N=c1ncn(CCC(=O)NCC2OCCC2C(=O)NC2CC(Cl)(Cl)C2)[nH]1 N1(C(c2c(CNC(CC3CCC(C)O3)=O)ccs2)=O)CC2CC3CC2C1C3 Cc1cc(CN2CCCC(c3cn(Cc4cccnc4)nn3)C2)ccn1 C1(NC(C(C=C)O)=O)CCN(C(c2ccn(CC(F)(F)F)n2)=O)C(C)C1 C(=O)(CN=c1[nH]c(C)cs1)N(C1CCN(C(c2cc(C)sc2C)=O)CC1)C N#CC1CC12CCN(C(=O)C(CC1CCC1)NC(=O)CCc1ncccn1)CC2 c1(CC)cc(C(F)(F)F)ccc1C(N1CC2CCC2C1)=O.c1(C(=O)N)ccns1 N1(C(c2c(C)ccnn2)=O)CC2CCC1C1CN(C(=O)CN3CC4CC4C3)CC21 N1(C(c2ccc(CC)nc2C)=O)C(CNC(C2(S)CC2)=O)CC2CCCC12 CC1CN(C(=O)CCc2ncc(C(C)(C)C)o2)CCC1N(C(=O)C=CCO)C c1(C(=O)NC2CCC(NC(c3cccc(C#C)c3)=O)C2)cnc2n1CC(C)CC2 C(=O)(C1CCOc2c(F)cccc21)NC1CN(C(C2(C)CC2)=O)C2(C1)CCCCC2 CC1OC2(CO)CC1(C(=O)NC(C)C(C)NC(=O)Cc1ccc(Cl)cc1)C2 C1(C2CCN(C(=O)C(C)(C)C3CCOC3)CC2)(C(=O)NCCSC)CCOCC1 c1ccccc1.CC1CCOC1C(N1CC(O)(CNC(=O)C)C1)=O.C(C)=O Cc1cc2nc(Cl)[nH]c(=NC(C)c3cn(C)c4ccc(C)cc34)c2s1 N1(C(c2c(C)cc[nH]2)=O)CCCC12CCN(C(c1csc(C(C)C)n1)=O)C2 c1(CSC)cnc(C(C(=O)NC2CCC2)N(C2CCC2)C)s1.C1CCOCC1 N1(C(COCC#C)=O)CCC(C2CC2)C1C(N1CCC1CF)=O C(=O)(CC(C)(C)CC(F)F)NCC1CC(OC)CN1C(=O)CCn1ccnn1 C1(CC(=O)N(CC(C)C(=O)N2CCC2C2CCCCC2)C)C(C)(C)C1(C)C c1(CC)cnc(O)c(C(=O)NCC(C)(CC)NC(=O)CCN(C)CCO)c1 N=C1NC(=O)C(CC(N2CC3CC2C3)=O)S1.c1(C(=O)N)cnn(C(F)(F)F)c1 c1(N(C)C)ccc([N+](=O)[O-])cc1C(=O)NC1CCC(C)(C)CC1.C(=O)C(F)F Cc1nccnc1NC(=O)NCCC1CCCN(C(=O)CC2(C)CC2(Cl)Cl)C1 N1(C(C(CCCC)O)=O)CCC2C(C1)CN2C(c1cnc(-c2ncccn2)s1)=O c1(C=O)ccc(N)c(O)c1.c1(CNC(C2(CCOC)CC2)=O)ccccc1 C1(NC(CSC)=O)CCC(C(=O)N(C(C)CC(C)C)C)C1 C(C(C)(C)C(=O)N1CC=CC(C(=O)NOCCCF)C1)OC c1(C(N2C(CC)C(C=O)CC2)=O)ccc([N+](=O)[O-])o1.C1(CCC)C=NNC1=O.N C1(CNC(=O)C=C(Cl)Cl)CCC2(CCN(C(c3nnn4ccccc34)=O)CC2)O1 C1(C(F)(F)F)(C(=O)NCCCNC(c2cnn(CCF)c2)=O)CCCC1 C1(C(N(C)CC2CCN(C(COC)=O)C2)=O)COc2cc(F)ccc2O1 C1(CC)C(C(=O)N(C)Cc2occc2C)CCN1C(c1csnn1)=O c1(CN(C(C)COC(C2CC2c2ccccc2)=O)C)nc2ccccc2s1 N1(C(CCC(C)OCC)=O)CCCC(O)(C)C1.n1(CC=O)cnc([N+](=O)[O-])n1 c1(C=O)ccc(F)c(F)c1F.CC1CC1C(=O)NCCCOCC.CCCO.N c1(OC)ccc(C(C(=O)NCCCCCO)N(C)C)cc1F c1(C(N(CCNC(=O)CCCC2CC2)CC2CC2)=O)cncc(F)c1 c1(C(=O)NC(C)C(CO)NC(=O)C(O)C(F)(F)F)cccn2cc(CO)nc12 N1(C(c2c(OC)nccc2)=O)CC(C)N(C(=O)CCCN=[N+]=[N-])CC1C c1(CC)noc(C(=O)N(C2CCCN(C(c3sncc3C)=O)C2)CCF)c1C c1(CC(=O)NC(C2CCCN2C(=O)C2=C(Cl)CCC2)C)ccccc1S(C)=O c1(C(=O)NCC(CC=C)NC(=O)CCc2ncccc2C)cc(C)c(O)nn1 c1(C(N(CC)Cc2ccccc2)=O)sc2[nH]cnc(=S)c2c1C C=CCC(C)C(=O)N1CCC(N(C(=O)CCCSc2ccc(Cl)cc2)C)C1 C=CC(CC)C(=O)NCC1(C(=O)NCC(C(O)CO)C2CC2)CC1 CCS(=O)(=O)CC(=O)NC(C)CC(C)NC(=O)C(c1cccc(F)c1)C c1(C(=O)NC2CCCN(C(c3cnns3)=O)CC2)ccccc1S(=O)C(F)(F)F c1(CC)ccc(C=CC(=O)NCC2CN(C(=O)C(C3CCCCC3)O)C2)o1 N1(C(C(CC=C)C)=O)CCC(O)(C2(NC(c3cc(CC)no3)=O)CC2)CC1 c1(OC)ccc(CCNC(C2CC23CN(Cc2ccnc(Br)c2)C3)=O)c(Cl)c1 C(=O)(C(F)(F)C(F)(F)F)NC1CCN(C(c2c(C)[nH][nH]c2=N)=O)C1 c1(CNC(C2(O)CN(C(c3cc(OCC)no3)=O)C2)=O)cccnc1S Cc1cc(CC(N2CC(C)C2C(=O)NC(c2nnc(C)s2)C)=O)n[nH]1 c1(CN(C=O)CC2COCC3(CCC3)O2)cccc2c1OCCCO2 C1(NC(CSC)=O)CC(CNC(c2cnc(O)n2C)=O)C12CCC2 N1(C(CCCC=C)=O)CC2CC(NC(c3cc(-c4cnn(C)c4)no3)=O)C(C2)C1 c1(NC(C(C)NC(C(COC)N(C)C)=O)=O)ccc(Cl)nc1 N1(C(CNC(=O)OC)=O)CC2(C1)CN(C(C1(CO)CC1)=O)CCO2 C(C)(C)(CCC(=O)NCC1CCC(C(N2CCCC2C(C)(C)O)=O)C1)N(C)C c1(C(=O)NC2C(NC(C(C)OC)=O)CCC2)nccc2cc(Br)ccc12 C=CC1OCCCC1C(=O)Nc1ccc(Oc2ccccc2)c(O)c1 Cc1ccc(SCC(=O)N(C(C)CNC(=O)CCc2ccnn2C)C)cc1N C1CCCCN1C(c1cccc(N)c1)=O.C1(CC(=O)NC)C=CS(=O)(=O)C1.C C1(C)(CNCC2(C)CC2(Cl)Cl)C=CCN1C(=O)OC(C)(C)C CC1(CO)CCCN1C(=O)C(=O)Nc1ccc(OCc2cocn2)cc1 CC1(C)CC=CCN(C(C23CCCC2CCN3C(=O)CCS(C)(=O)=O)=O)C1 CC1CN(C(=O)CC2CC(F)CN2C(c2cc(C#N)c[nH]2)=O)C(C)C1C CC1CN(C(c2c(Cl)ccc(O)c2Cl)=O)CC(C)N(C(c2csnn2)=O)C1 N1(C(CNC(C(CC)C)=O)=O)CC2(NC(=O)CSc3nnnn3C)CC1C2 C(CCCCNC(=O)C(O)C1CCCC1)N(C(=O)C(C1CC(F)(F)C1)O)C C1(NC(CCc2n(C)cnc2)=O)CCC(NC(=O)CC2(C(F)(F)F)CC2)CC1 c1(C(=O)NCCC2CN(C(c3cc(C)ns3)=O)CC2C)c[nH]c2cnccc12 N1(C(C2(CC)COC2)=O)CCCC(N(C(=O)CC2CCCO2)CC2CC2)C1 c1(C(=O)OC)nc(C(=O)N(C)CCN(C(=O)CCF)C(C)C)co1 N1(C(COC)=O)CC(C)CCC1CNC(=O)Cc1cnn(C(C)C)c1 Cc1ccc(SCC(=O)NC2CCCN(c3nnc(CC(F)(F)F)s3)C2)cc1C N1(C(c2c(C)nc(O)[nH]2)=O)CCC(CCNC(=O)Cc2cscn2)CC1C c1(C(N2CC(C)(NC(c3c(CC)c[nH]n3)=O)C2)=O)c(C)cccc1Cl C1(NC(c2c(C)cn(C)n2)=O)CN(C(C2(C)CC2Br)=O)CC(C)(C)C1 N1(CC)CC(CO)C2(C1)CN(c1nc(NCCCO)c3ccsc3n1)C2 C1(CCC)(NC(=O)CCN(C)CCO)CCN(C(C23CCCC2CCC3)=O)CC1 c1(C(=O)OC)ccc(C(N2CC(C)(NC(=O)CCCc3ccsc3)C2)=O)nc1C N1(c2nc(OCCOC)c(C)cn2)CCc2nc(Br)sc2C1 c1(C(CNC(C(CC)F)=O)NC(c2cc(Cl)c[nH]2)=O)cccc(Cl)c1 CCCC(C)(CO)NC(C1CCC(NC(=O)COC(C)=O)C1)=O Cc1ccncc1CCNC(=O)CC1CCN(C(=O)C(=O)NCC(F)F)C1 N1(C(C2(OC)CCCC2)=O)CCC(CN(C)C(c2cc(C3CC3C)on2)=O)CC1 C(N=c1cc(C)nc(COC)[nH]1)C1CCN(C(CCCC#CC)=O)C1 c1(C(=O)NC2CC(NC(C(c3ccnn3C)C)=O)C2)cccnn1 N1(C(C2N(C(CN(C(C)C)C)=O)CCC2)=O)CCN(C2CC2)C(C)C1 CS(=O)(=O)c1c(NC(N2CCCc3ccnc(O)c32)=O)cccc1F N1(C(C2(C#C)CC2)=O)CC(C)CC12CCC2.c1(CC(=O)N)cc(F)c(C)cc1F C1(NC(CC=CC)=O)CCN(C(=O)Cc2cnn(C3CC3)c2)CC12CCC2 C1(C(N(C2CCCC2(F)F)C)=O)CCN(C(c2nnc(O)nc2O)=O)C(C)(C)C1 N1(CC(=O)NC2CCCC2NC(=O)CC2COCCO2)CCN(C2CC2)C1=O c1(OCC)cc(C(N2CC3(C2)CN(C(c2cccc(O)c2Br)=O)C3)=O)ccc1F C1(CCN(C(C(COCC)C)=O)C)CCN(C(=O)C(C)Cc2ccccn2)CC1 N1(CC(=O)NCC(C)(CO)NC(=O)C(F)=CCF)CCN(C2CC2)C1=O CC(F)(F)CCCCNC(C1CC=CCC1NC(c1ccc(C#N)[nH]1)=O)=O C1(NC(CCN(C(CC2(NC(C)=O)CC2)=O)C2CC2)=O)CCOCC1C c1(CC)c(C)cccc1S(=O)(=O)NC1CCS(=O)(=O)CC1 C=CCCCCC(=O)N1CCC(F)C(NC(c2ccnc(C(C)(F)F)c2)=O)C1 c1(NCC(COC)(C)C)c(Cl)c(C)nn1CC(F)F C1(C(=O)NC2CC(NC(c3c(C)cno3)=O)C2)COc2cc(Cl)ccc2C1 c1(C(=O)N)cc2c(nn1)OCCS2.c1(C(=O)NC2CCC2)ccnc(C2CC2)c1 C(=O)(C(C#N)C(C)(C)C)NC(C(=O)NCCCCCC=C)CCC1CCC1 c1(CN2CCC(C)(C(=O)Nc3c(F)cccc3Cl)C2)c[nH]c2ccncc12 C(c1sc(Cl)nc1Cl)=CC(=O)NC(CNC(c1cccc(CCC)c1)=O)C N1(C(C2CC(OC)(OC)C2)=O)CC(C(=O)NCCN2CC=CC2)CC1(C)C c1(C(N(CC(CC)NC(=O)CNC=O)C)=O)cncc(Br)c1C c1(OC)cc(C(=O)NC2COCC2NC(=O)C(C)c2ccsn2)cc(Cl)c1 c1(C(=O)NC2(CC)CCCN(C(C3(C)CCC3)=O)C2)cccc2c1CCCC2 Cc1nc2cccc(C(=O)NC3CCCN(C(=O)CC(C)C)CC3)n2n1 c1(C(=O)OC)ccnc2c1CCC2NC(=O)Cc1ccccc1F.C1CO1 c1(C(N2C(C3(NC(CSCC#C)=O)CC3)CCCC2)=O)cccc2c1COCC2 c1(Oc2c(C(N(C(C)C)CC)=O)cco2)ccncc1.C(C)=O.C(C)=O C1(NC(c2scc(C(C)(F)F)n2)=O)CCC12CN(C(=O)CC1CCOCC1)C2 C1(N(C(c2ccc(OC)s2)=O)C)CCN(C(c2cncnc2C)=O)CC1C c1(C(=O)NC2CC(CNC(COC(CC)C)=O)C2)c(C)cc(OC)cc1C C=C(C)CC(C)C(=O)N1CCC(=CCO)CC1.CC=C N1(C(C2CCC(n3cc(-c4scc(C)n4)nn3)CC2)=O)CC2(CCOC(=O)N2)C1 c1(C(=O)NC(C(C)(C)NC(c2cc(C)c(O)nc2)=O)C)nc2c(s1)CN(C)CC2 O=S(=O)(c1ccc(C(F)F)cc1Cl)NC1CC2C(C1)C2(F)F Cc1ccc(-c2cn(C3CCN(C(=O)CCC4CCN(C)C4)C3)nn2)c(Cl)c1 C1(CNC(=O)C2=CCOCC2)CCC2CN(C(=O)Cn3cccn3)CC12 CC(CNC(=O)CCC1CC(NC(=O)CN2CCCC2C)C1)C(F)(F)F Cc1cccc(C(=O)N(CC(=O)N(C)C(C2CCCC2)C)C2CCC2)c1F C1(C)CCOC1C1CC1.C(C(=O)NCC(=O)NC(=O)OC)(OC)OC N1(C(c2cc(C(=O)OC)[nH]c2)=O)CCC(CC)CC1.C1(C)(C(=O)N)CCCOC1 c1(OC)ccc(CC(=O)NCC2CCN2C(C2(C#N)CCCC2)=O)cn1 c1(C(=O)NC2C=CCN(C(CC(=C)C)=O)C2)cc2ncccc2[nH]1 N1(C(C2CC(CC)(CC)C2)=O)CCN(C(=O)CC(C)SC)CC2(CC2)C1 c1(NC(C2CSCN2C(=O)CCc2nncs2)=O)cccnc1C1CC1 C1(C(C(=O)NC)O)CCS(=O)(=O)CC1.N1(C(C=CC(C)C)=O)CC(O)C1.C C1(C(=O)NC2CCCC(NC(=O)C3=CCOCC3)C2)COc2cc(F)ccc2C1 c1(NC(C2CCC(n3cc(C(C)(C)C)nn3)C2)=O)nccc(Cl)c1Cl C1(C(N(CC(O)C2CCC2)C)=O)CCN(C(C2CCCCC2(C)C)=O)C(C)(C)C1 C(c1cc(F)cc(F)c1)=CC=O.C12(NC(C3N(C)CCC3)=O)COC(C1)CC2 S(=O)(=O)(c1ccc(Br)cc1N1CCC2(CNC(=O)C2)C1)N1CCC(=C)C1 c1(C(=O)NCCC2CCN(C(C(C=C)(C)CC)=O)C2)ccc(S(C)(=O)=O)s1 c1(CC)cc(C(=O)NCC2CCCC2NC(c2ccccn2)=O)cc2c[nH]nc12 c1(OC)ccnc(C(=O)NCCOCC)c1.c1(CC(=O)N)sc(S)nc1C c1(CSCCCOc2cnccc2)n[nH]c2c1COC2 c1(OC)c[nH]nc1C(=O)N(C)CC1(O)CN(C(=O)CCc2cccs2)C1 C=C1CCC(C(N2CC(NC(=O)CCC(=O)c3ccc(Cl)cc3)C(C)C2)=O)CC1 c1(OC)ccc(F)c(C(=O)NCC2CCN2C(c2ccnc(S)c2)=O)c1O N1(CC)CC(NC(=O)CCc2ccccc2C(F)(F)F)C(N)C1 N#Cc1ccc(C=CC(=O)NC)cc1.C1CC2CCC1N2C(C1C2CCCC12)=O c1(NCC(CC(C)C)OCC)[nH]c(=NCC2CC2)nc2c1ncn2C CCCCC(O)CC(=O)N1CCOC(CC(=O)NC(Cc2ccco2)CO)C1 N1(C(CC=CC=C)=O)CCN(C2CCCN(C(=O)C(C)c3ccco3)C2)C(=O)C1 C1(C=O)CCCN1C(=O)C(C)(C)C1CCN(C(=O)CCc2cnn[nH]2)C1.CC.N C1(CNC(c2cc(CF)on2)=O)COCCN(C(C2(O)CCCCC2)=O)C1 N1(C(CC2(COC)CC2)=O)CCC(O)(C(C)CNC(c2ccc[nH]2)=O)C1 C(=O)(CCC(C)(C)C)NCCCCCNC(c1cc(C)nn1C(C)(C)C)=O c1(C(=O)NCC(CCNC(C2(CC#C)CC2)=O)O)cc(F)c(N)cc1O O=S(=O)(c1cccc(N2CC(F)C(F)C2)n1)NCC1CC2CCC1CC2 c1(CN2C(C(=O)Nc3c(OC)ncc(Br)n3)C=CC2)ccc(Cl)cc1[N+](=O)[O-] C1(C(N2CC(CC)C2)=O)(COC)CCCCO1.c1(C=O)ccc[nH]1.N(C)C.N CC(C)C(C(=O)NC(C)C(=O)N(C1(C)CC1)C)c1ccc(Cl)cc1 n1(CC)ccc(C(=O)NCC=CC)cc1=O.C1(C(=O)N)CC2(CCC2O)C1 CC1=C(C)CC(C)(C(=O)NC2CN(C(C3(C)CCC(C)(C)CC3)=O)CC2F)CC1 c1(-c2nc(C)c(O)cc2)ccc2nc(C(N3CC4CC3CN4C)=O)sc2c1 c1(C(=O)NCC2CCCN(C(C(CC)OC3CCCC3)=O)C2)cnc(C)cc1C N1(C(C=CC=CC)=O)CCCC2(NC(=O)C(CC)OCC)CCCC12 C1(C(=O)NC2CCN(C(C3OCCN(C)C3)=O)C2C2CC2)CC2(C1)CC2(F)F Cc1nn2c(C(N3CC=C(CNC(=O)C(C)C(C)C)CC3)=O)c(C)nc2s1 Cc1cc(C(=O)NC(C)CNC(c2ccon2)=O)c(C)n1NC(N)=O C(CC(C)C)(C(=O)NC1(C(=O)NCCN2CCCCCC2)CC(F)C1)OC c1(C(=O)NC(C2CCN(C(C3CC(=O)N(O)C3)=O)CC2)C)ccc(C#N)n1C N1(C(C2C(C)OC(=O)N2)=O)CCN(C)C(C(=O)NCCCn2cnnn2)C1 c1(C(N2CCC(C)(CNC(CCOC(C)=O)=O)C2)=O)cc2cccnc2s1 CC1(C(=O)Nc2cncc(CO)c2)C=CCN1C(C1CC2CC2C1)=O C(C)(N(C)N1CCOCC(C2CCC2)C1)c1ccc(OC)cc1 c1(CC)oc2ccccc2c1CC(=O)N(CC(C)N(C)C(C1CNC(=O)C1)=O)C c1(C(=O)NCC23N(C(CSC)=O)CCC2CCC3)cccc2c(C)c(C)[nH]c12 c1(C(=O)OCC)coc(C(=O)N)c1.CC(C)C.C(=O)C(C)C.C(C)=O C1(NC(c2cnc(SC)o2)=O)CCCC1(C)NC(=O)CC1COCCOC1 c1(CC(=O)N(CC(C)C)C)nccnc1C.C1(OCCOC)C(C=O)C1C.N C(=O)(C(C)C(O)CC(C)C)NCC1(OCC)CN(C(=O)CCCCSC)C1 c1(C(N2CC3C(NC(=O)CCF)(CCOC3)C2)=O)cc2c(Cl)cc(Cl)cc2[nH]1 C1(C)(NC(c2nc(C#N)cs2)c2n(C(C(=O)OC)C)nnn2)CCCCC1 C(=O)(CCCC(C)(C)C)N(CCC(=O)N(CC#C)CCO)CC#C C(=O)(C(C)(CC)CO)NCC1C(C(F)F)CN(C(c2c(CC)n[nH]c2)=O)C1 C1(C(=O)NCC(C(C)C)NC(=O)C(C)Sc2nncn2C)CCn2ncnc2C1 C1CCC2(CNC2)OC1.c1(C(C)NC(=O)N)ccccc1.C(C)(C)(C)NC.C C12(NC(CCC)=O)CCCC1N(C(=O)CCc1ccc(O)c(Cl)c1)CC2 N1(C(CC(CC)(C)C)=O)CCC(C2CCN(C(c3cnc(=N)[nH]c3)=O)C2)C1 c1(C(=O)NC(CC(C)NC(c2cnc(C)nc2C)=O)C)cc(=O)n2nccc2[nH]1 c1(C(N2CC(NC(C(CCC)S(N)(=O)=O)=O)C2)=O)oc2c(c1C)C(=O)CCC2 C12(OC)CCC(NC(=O)CC3(O)CN(C(c4ccc(C)[nH]4)=O)C3)(CC1)C2 N1(C(CC(CC2CC2)NC(C2(C(CC)=O)CC2)=O)=O)CC2CCCCC12C c1(-c2onc(CCc3ccc(C)cc3)n2)cc2c(Br)n[nH]c2cc1F c1(C=O)ccc(=O)n(C)n1.Cc1csc(C)c1C(N1CC(C(N)=O)(C)C1)=O c1(CNC(C(COCC)n2cc(C3CCC3CN)nn2)=O)ccc(F)cc1 N1(C(=O)C(N2CCC(OCc3ccccc3)C2)=O)CC2C3C=CC(C3)C2C1 C1(NC(C2CCCCC2c2cccnc2)=O)CCN(C(C2CC(O)C2)=O)CC1 c1(N2CCN(C(CN(C3CN(C(C)=O)C3)C3CC3)=O)CC2)cc(C)ccc1C C(=O)(CCCCC(C)(C)C)NC(C(=O)NC(CC(C)C)CO)(C)CO N1(C(CC2CC(N(C)C)C2)=O)CCCC1CNC(C1(c2ccccc2)CCC1)=O N1(C(C)=O)CCC2(CC(C(N3CC4(CC(N(C)C)C4)C3)=O)C2)C1.C(C)OC.O C1(C(N2CC(NC(C(CCC)NC(N)=O)=O)C(C)C2)=O)CC2(C1)CC2(F)F c1(C(N2CCC(C)(C)C2C)=O)cccc([N+](=O)[O-])c1N.c1(CC(=O)N)cnoc1 C(=O)(C1CCc2ccccc21)NC1(CNC(=O)Cc2ncc(Cl)s2)CCOC1 c1(COCCOC)ccc(CNC2CCN(Cc3ccc(Br)s3)CC2)cc1 N1(C(C2(C(C)C)CC2)=O)CC(NC(=O)C(O)C(C)C)C2(CC2)C1 C1(C(c2nnnn2C2CC2)N)CN(C)CC1c1cccs1.c1(OC)nscc1.C N1(C(c2ccc(C)cc2)C(=O)NC2CCCC2)CC(C)OC(C)(C(F)F)C1 c1(C(=O)NC2(C)CN(C(C3(C)CC3Br)=O)C2)cnc2n1CCOC2 Cc1ncc(N)cc1C(=O)NC1CCN(C(=O)C(C)Sc2ccccc2Cl)C1C CCC(CN(C)C)CC(=O)NCC(CNC(c1ccnc(C2CCC2)c1)=O)CO C#CC1(CNC(=O)CCOCCCNC(=O)CN2CCOC2=O)CCC1 O=CN1CCCC1C(=O)NC1CCOC(C(=O)NOCCCO)C1 N1(C(C(C2CCN(C(C3C(C)CCC3)=O)CC2)C)=O)CCN2CCCCC2C1 c1(C(N2CC(CNC(c3cc(OC)n(C)n3)=O)C3C2C3)=O)ccc(C)c(N)c1 CC1OC2(C)CC1(C(=O)NCC(CC(F)(F)F)NC(=O)C(c1ccccc1)O)C2 N1(C(c2cnc(OC)nc2C)=O)CCN(C(=O)CCn2ccnn2)C(C)C1C N1(C(CC(C)(C)C2CC2)=O)CCC2(CC1)CCN(C(C1(C)CC3CCC1O3)=O)C2 CC1CCN(C(=O)C=Cc2ccccc2)C(CNC(=O)C#CC(=O)N(C)C)C1 CCCCCC(CC)C(=O)NC1CC(C)(NC(c2cc3ccc(Cl)nc3s2)=O)C1 CN1CCCCC(NC(C2CC=CC(NC(C3(F)CCCCCC3)=O)C2)=O)C1=O N1(c2n(CC(=C)C)c(CC(C)(C)CC(C)O)nn2)CCOCC12CNC(=O)OC2 Cc1nc(CC(=O)NC2CCC2CNC(=O)C=C2CCOCC2)n[nH]1 C=C(C)CCCN=c1ccnc(N2CCC(Oc3ccncc3)C2)[nH]1 n1(CC)cc(CC(=O)NC2CCC2NC(c2cc(C(C)=O)[nH]n2)=O)cn1 C1(CCNC(COC)=O)CCCCN1C(=O)C(O)Cc1ccccn1 c1(C(N(CC(C)NC(=O)C(C)(O)COC)CC)=O)cnc(O)c2ccsc12 c1(NC(C2CN(C(=O)CC(C)NC(N)=O)CCO2)C)cc(O)nc(O)n1 C1(N(C(c2c(CC)noc2)=O)C)CS(=O)(=O)C1(C)C.c1(C=O)csc(Cl)n1 C1(CC)N(C(=O)C(Cc2cc[nH]n2)NC(=O)C(C)=C(C)C)CC1(C)C c1(C(N2CC(=C(CNC(=O)C=Cc3cccnc3)F)C2)=O)ccc2c(c1)CCN2 N1(C(CCC2CCC(=O)N2)=O)CCC(NC(c2csc(-c3cccs3)n2)=O)CC1 C(=O)(C(O)CC1CCCCC1)NC1CC(NC(=O)CSC2CCCC2)C1 c1(C=O)cccc(C)c1.C1(NC(COC)=O)CC(SCC)C1.C(=O)(C)N N1(C(c2ncn(CC)n2)=O)CCC(NC(=O)COc2ccc(CO)cc2)CC1C c1(NC(C2CC(OC)CN2Cc2cccc3c2OCO3)=O)nc2c(s1)CCCC2C CC1(C)CCC(CC(N2CCC(C)(CC(=O)NC3CC(F)(F)C3)C2)=O)O1 Cc1cccc2c(C(=O)NC3CC3NC(=O)C[SH](=O)=O)n[nH]c12.C(C)(C)C C1(CNC(CCC#C)=O)(OCCNC(=O)CC(C)C)CCOCC1 CN1CCC(C)(CNC(C2CCC(C)CC2)=O)CC1.c1(C=O)cc(O)nn1C.N c1(OCCOC)cccc(CC(N2CC(C(=O)NC3(CO)CCC3)C2)=O)c1 N1(C(c2c(C)nc(O)cc2)=O)CC2(CCCC2)C1C(=O)N1OC2CCC1C2 C1CC2COCC(C1)C2.C1(C=O)CC2C=CC1C2.CC(C=O)NS(C)(=O)=O.N c1(C(N(C2CCCN(C(=O)C3CC3)C2)CC)=O)cc(S(C)(=O)=O)ccc1C c1(C(=O)NC)cccc(C(=O)N(C)CC2CCCN2C(c2cccc[n+]2[O-])=O)c1 C1(C(=O)NCC2CC3(CN(C(CCC#C)=O)C3)C2)CCCCN1S(N)(=O)=O C1(OCC)CCC(CNC(C2CCN(c3cc(C(C)=O)ncn3)CC2)=O)CC1 c1(C(=O)NCC2CN(Cc3ccc(C(=O)OC)[nH]3)C2)cc(C)ccc1I N1(C(c2c(SC)ccs2)=O)CCCC12CCN(C(=O)CC(C)C(C)C(C)C)C2 C=CCC(C)(C)CC(=O)NCC.C(=O)CC(F)(F)F.C1CCN(C(=O)CC)C1.O C(CC(C)C(=O)NC1CCCC1C(=O)N(CC(C)OC)C(C)C)=CCC C1(C(=O)OC)N(C(c2ccc(C#N)o2)C(=O)NC2(C)CC2)CCCC1(C)C c1(N(C)C)cccc2c1CN(N1CCC(C)(C)C1c1ccnn1C)C2 c1(C(=O)NC(CCNC(c2nn(CC)nc2C)=O)C)c(Cl)ccc(F)c1F c1(C(N2C(N(C(=O)CC)C)CC(F)C2)=O)ccnc2cc[nH]c12.C(=O)C1CC1.N N1(C(C(C)C2CCC2)=O)CC2CCC(C1)N2C(c1cn(C2CCCCC2)nn1)=O c1(COCC(=O)NC2CN(C(=O)Cn3cnc(Br)n3)C2)ccccn1 C(CC(C)(C)NC(=O)Cc1c[nH]nc1O)N(C(=O)C(N1CCCC1)C1CC1)C c1(C(=O)NCC2C(NC(c3ccc([N+](=O)[O-])s3)=O)C2)ncc2n1CCCC2 c1(OC)cc(C(C)OC(=O)CC2CC3(CCNCC3)CO2)ccc1S(C)(=O)=O C1(NC(CCCCC(=O)NC)=O)CCS(=O)(=O)C12CN(C(c1ccc(F)s1)=O)C2 c1(C(C=O)(C)C)cccc(N)c1.N1(CCC)CCCC1.C1(C(=O)N)(CC)COC1 N1(C(c2occ(C)c2)=O)CCN(CCN2CCCC2=O)CC1C C1(CC)CCC(C)CN1C(=O)C(C)(C)CNC(c1cc(OC)cnn1)=O C(=O)(CC(O)CNC(c1ccc(Cl)o1)=O)NCC1CC(CN=[N+]=[N-])C1 N1(C(C(C)N(C(CCSC)=O)CC2CCCOC2)=O)CCC(OCC(N)=O)C1 C(C1=CCN(C(c2ccnc(CO)c2)=O)CC1)NC(CC(=O)N(C)C)=O CC(CC(C)NC(C1CN(C)C1)=O)NC(C1CCCN1S(C)(=O)=O)=O c1(C=O)c(C2CC2)cccc1F.C1(C(=O)NC2CC(C)C2)CC2(CCCO2)C1 CC(C(=O)N1CC2CC2(NC(=O)CCc2ccccc2)C1)P(C)(C)=O Cc1n[nH]cc1CN(C(=O)CC1CCC(NC(C2CC2(C)C(F)F)=O)C1)C c1(C(N(C(c2ccccc2)CNC(C(C)O)=O)C)=O)cc(Cl)ccn1 C1(CNC(=O)CCn2ccnc2)CN(C(=O)COC(F)F)CC1O c1(C(N2CC(CNC(C3CC(O)(CC#C)C3)=O)C2)=O)cc(C)cnc1C c1(NC(c2cnc(CNC(c3cc(C)sc3)=O)nc2)=O)ccc(F)c(O)c1 C1(NC(c2cnc(OC)s2)=O)CC2(C1)CC(NC(=O)CCC1CCOCC1)C2 N1(C(C(F)OC)=O)CCC(C2CC2)(CNC(c2cc3n(n2)CCC3)=O)C1 C1CCCN(C(c2scnc2C(C)(C)C)=O)C1.c1(CC(=O)N(C)C)nonc1C CC(C)C(O)C(C)C(=O)NCC1CN(C(=O)C(C)(C)N2CCOCC2)CCN1C c1(CN(CCCCC)C2CC2)noc2c1CCCC2 C1(OC)CC(O)CN(C(=O)C#CCNC(=O)C(C2CC2)C2CC2)C1 N1(CCSc2ncccn2)CCC(C2(c3c(CC(=O)O)cnc(O)c3)CC2)CC1 Cc1ccc(C(=O)N(CCNC(=O)CS)C(C)C)c(C)c1.C1CCOC1=O c1(OC)cc(O)c(CN2CCC(C#N)(NC(C3C4COCC34)=O)C2)cc1OC c1(C(=O)NCCCCOC)cn(C)c(=O)n(C)c1=O.c1(C=O)ccc(=O)oc1 Cc1ccc(Cl)c(Br)c1CC(=O)NC1(CO)CC(C)CC(C)(C)C1 S(=O)(=O)(c1ccc(Cl)cc1)N1CCC2CN(C(c3c(F)ccc(F)c3Cl)=O)CC21 C#CC1(O)CCN(C(c2cn(CCNC(c3cc(C)nnc3C)=O)cn2)=O)CC1 Cc1cc(CO)oc1C(=O)NCCC(C)NC(C1CCCC1(F)F)=O C1(CCC)(CO)CCCN(C(C2CCN(C(C)=O)CC2OC(C)(C)C)=O)C1 O(N(C)C(=O)CNC(=O)CCNC(c1cccnc1CC)=O)CC CCCC(C)C(=O)N1CCOCC1CNC(=O)CCN1CCCC1=O C1(C(N2CCC(NC(=O)CC3(C(F)(F)F)CC3)C2)=O)CCc2ncccc2C1 N1(C(c2c(C)nco2)=O)CCCC(NC(=O)CS(=O)(=O)N(C)C)C(F)C1 C1(C)(CNC(CC2CCC(C)(C)O2)=O)CCCN(C(C2CC(=O)CCO2)=O)C1 c1(CC(C)N(C(=O)CCC2CC2(F)F)CC)cc(Cl)ccc1Cl N1(C(CC(=C=C)C)=O)CC(NC(=O)C(O)CSc2ccccc2)C2(CCC2)C1 Cc1ccc(OCCC(=O)N(C)CC2CCCN(C(=O)CCC#N)C2)c(C)c1 c1(C(=O)NCC(CC)NC(=O)Cc2cc(-c3ccccc3)on2)c(C)coc1C N1(C(C(C)Cc2ccc(F)c(F)c2)=O)CCN(C(c2nncs2)=O)C(C)CC1C c1(N2CCN(Cc3c(C(=O)OC)snn3)CC2)nccc2c(N)cccc12 C(=O)C(F)n1cccn1.C1(CC)(CNC(C2(CC(F)F)CC2)=O)CC1.N C1(N(C)C(C2CC2C(F)F)=O)CN(C(=O)CCc2ccc(Cl)cc2)CC1(C)C CC(C)CC(CC(=O)N(C1CN(C)C1)C)NC(=O)CCC1CCC(=O)C1 Cc1cccc(-c2cn(C3CC(NC(=O)CC4CCCN(C)C4)C3)nn2)c1 C1(C(NOCCCOC)=O)CC2CC1CN(C(c1cc(Cl)no1)=O)C2 C1(C(=O)NC(CN(C(=O)CC(F)F)CC)C)CCc2cn(C)nc2C1 c1(CC(=O)N(C(C)CN(C(=O)CC2CCCCC2O)C)C)cccc([N+](=O)[O-])c1 C1(NC(CC2CC(CC)C2)=O)CCCC(C(=O)NCC(CO)C(N)=O)CC1 n1(CCC)cc(C(=O)NCCC2CCC2)c(C)n1.C(C)(C1CC1)=CC=O C1(CCC=C)(C(=O)NCCC(C)OCC)CN(C(c2cc(C)on2)=O)C1 C1(COC)(C)CCN(C(=O)Cc2ncc(Cl)s2)C1.C1(CC=O)OCCO1.N C#CCCCC(C)C(=O)NCc1ccc(C(=O)NCCCOCCOC)nc1 c1(NC(=O)CC2COCC2O)cccc(NC(C2(O)CC(CF)C2)=O)c1 C(C(C)CC(F)(F)F)NC(C)C(c1ccccc1)N N1(C(=O)Cc2cccc(F)c2)CCc2sc(C(N3CC4CCC3CC4)=O)cc2C1 Cn1nc(CNC(C2CC2[N+](=O)[O-])=O)cc1C(=O)NCCC1CC1 Cc1cc(=NCc2cccc(N(C)C)n2)[nH]c(=NCCn2ccnn2)[nH]1 c1(C(N2CCCC(OC)C2C)C(=O)NC(CC)C)ccc(C(=O)OC)c(C)n1 CCC(C)(C(=O)N(C)CC1CCN(C(=O)COc2ccc(Cl)cc2)C1)C(N)=O C(=O)(CCC(=O)C(C)(C)C)NCC(CNC(C(c1cccc(Cl)c1)OC)=O)C c1(OC)cc(F)ccc1CN(C)C(c1cc(SCc2ccccc2)on1)=O C=CCCCCCCNC(=O)C(C)CN(C)C(c1ncsc1C)=O N1(C(C=CCOC)=O)CCC2C(C(=O)NCc3nonc3C)C2C1 C1CCN(C(C2CC2)=O)C1C(F)(F)F.C1(C(=O)N)(NC(C)=O)CCCC1 CCCCC(C)CCC(=O)NC(C)CCNC(c1cccc(OC(F)(F)F)n1)=O C(=O)(C(C1=Cc2cc(Br)ccc2OC1)N1CCC(C)(O)CC1)NC(C)C C=CCC(CC=C)C(=O)N1CCC(C(C)C(=O)N(CCC(F)(F)F)CC)C1 c1(OC)cc(C(N2CC(C)(NC(c3ccc[n+]([O-])c3)=O)C2)=O)sc1Cl C1(NC(=O)CCC2CCC2)CN(C(C2(C3CCCCO3)CC2)=O)C2CCCC12 C(=O)(C(C(C)(C)C)NC(=O)C=Cc1ccccc1)NC(C)C(=O)NO N1(c2c(C(=O)OC)c(C)cc(C)n2)CCC(C2CCN(C(=O)C(C)O)CC2)C1 C(=O)(C#CC1CCCOC1)N1CCN(C(c2cc(C)nc(C)n2)=O)C(CCO)C1 c1(CN2CC3C(C(=O)NC(c4ccccc4)CCO)(C3)C2)ccc(Cl)cc1Cl C1(C(=O)OC(C)(C)C)COC2(COC2)C1.C(CC1C(=O)N1)NCC N1(C(c2c(C)noc2)=O)CCC=C(CNC(=O)C(N2CCOCC2)C)C1 C(=O)(CC(O)CNC(=O)C(C)(CO)NC(c1cn[nH]c1)=O)OC c1(N2CCN(CC)CC2)nc(N2CCCC(C(=O)N(C)C)C2)nc2sccc12 N1(C(=O)CCC2CCOC2)CCOC2CCN(C(=O)C(F)(F)CC3CC3)CC12 Cc1sc(Br)nc1CC(=O)NC(C1CCCN1C(=O)CC(C)(C)C)C Cc1cc(C(=O)N(C)CC2CCCCC2)nc(C)c1.C1(C(=O)N)CC12CC(O)C2 N1(C(C(CC)OC2CCCC2)=O)CC2(CCC1C)CC2.C(=O)C.C(C)(C)C.N N1(C(C(CN(C(C2CC(C)=C(C)CC2)=O)C)C)=O)CCCC2C(O)CC12 C1(CNC(C(N2CCCCC2)C)=O)CC(C)N(C(=O)CCc2nccs2)C1 C1(CNC(C(C=C)C)=O)CCCN(C(c2cc(C(C)=O)c[nH]2)=O)C1 c1(C(N2CC3(CC(NC(CC(C=C)(C)C)=O)C3)C2)=O)[nH]c2c(c1C)CCCC2 CC(C(=O)N(CC(=O)NCC(Cl)=CCl)C)C1C(NC)C1 c1(C(=O)Nc2cccc3c[nH]nc23)cc2n[nH]cc2cc1-c1c(O)cccc1O c1(C(N2CC(NC(=O)C(F)=C(C)C)CC(OC)C2)=O)cnc2[nH]cncc1-2 N1(C(COCCC#C)=O)CC(C(=O)NCCc2nc(C)oc2C)CCO1 CC1OC2(C(=O)NCCC3CC(NC(c4cc(Cl)ccc4N)=O)C3)CCC1C2 C12(CNC(C3CC(=O)C3)=O)CC1CN(C(=O)CCCO)C2.c1ccc(Br)cc1 CCS(=O)CCNC(=O)CC1(N(C(=O)CCC=C(C)C)C)CC1 c1(NC(C)=O)ccccc1CN=C(NC)NCc1cc[nH]n1.C1CCCO1 N#CC1CCCC(C(=O)NCC2CC2C)C1.N1(CC=O)CCC(=O)NC1=O C(=O)(C1=NN(C)C(=O)CC1)NC1CN(C(c2c(C)onc2)=O)CC1C.C1CC1 c1(C(N2CCCC(N(C(=O)C(O)C3CCC3)CC)C2)=O)cc(Cl)c(Cl)cc1N c1(C(N(C2CCCN(C(=O)C(F)C3CCC3)C2)CC)=O)cnc(C#N)s1 C1(CNC(C2(C)CCCN2C(=O)CCc2cncnc2)=O)CC(O)C12CCC2 C1(C(N(CCCCCC)C)=O)CCCCC1(C)NC(=O)CC C=CCC(C)C(=O)N1CCCCC1CNC(=O)CC1CCC(C)(C)O1 S(=O)(=O)(c1cccc(C(C)(C)C)c1)NC(CC(CC)(C)C)C(=O)OC C(CCCC(=O)NC1CCC(NC(c2cc(C)sn2)=O)C1)SC C1(CNC(C2C(OCC)C2C)=O)CC(N=c2nc(C(C)C)[nH]s2)C1 C1(NC(c2cc(C)n(C)c2)=O)CC2(C1)CC(NC(C1Cn3ccnc3N1)=O)C2 CC(C)(CNc1cc(NC2CC=CC2)ncn1)C(F)F C(=O)(C1=CCCC1(C)C)N1C(CNC(C(C(C)O)C)=O)CCC1 C=CC(C)(CCOC)C(=O)NCc1ncccc1C(N1CC(C2CCCO2)C1)=O N1(C(C2N(CC)C(=O)CC2)=O)CC(NC(=O)C(F)(F)COC)CC(F)C1 N1(C(C2(COC)CC2)=O)CCCC2(CCC2)C1.C(=O)C(C)(C)N1CCCC1.N CCC(c1ccc(C)cc1)=CC(=O)NCC12CC(C1)C2.C1(C=O)CC=CCC1 C1(C(=O)NCC2OCCN(CC)C2)CCc2nnnn2CC1 CCCC(C)(O)CC(=O)NCC=CCC(=O)NC1(C)CC(F)C1 Cc1n[nH]c(C)c1C(C)C(=O)NCC1(O)CN(C(c2ccno2)=O)C1 N#Cc1cccc(CC(=O)NC(c2ccccc2F)CNC(C2COCO2)=O)c1 c1(CC(=O)N(CC(C)O)CC)ccccc1CN.C(C1CCC1)=CC=O C1(CN(C)C)CCCC1(C)NC(C1N(C(C(C)(C)OC(C)=O)=O)CC1)=O c1(CC(N2CCC(C)(NC(CCC(C)C)=O)C2)=O)cccc([N+](=O)[O-])c1 C1CCOC2(CCS(=O)(=O)C2)C1.c1(C(=O)OCCC)ccc(NC=O)cc1.N C#Cc1c(F)ccc(NCC2OCCC2(C)C)c1F C=CC(CCC)CC(=O)NCC1(F)CCCN(C(=O)C(O)(C2CC2)C2CC2)C1 n1(CC)c(SCCO)nc2ccc(F)cc2c1=O CC1(C(N2CCC(O)(C(C)(C)CNC(c3ccc(C)o3)=O)C2)=O)COCCO1 C1(NC(c2c(C)nc(CCC)o2)=O)CN(C(C2CCC3(CCC3)O2)=O)CC12CC2 C=CC1(CC(=O)NCCC2CC2C)CN(C(C2CCCN2C=O)=O)C1 CC(C)C(O)C(C)C(=O)NCCC(=O)NCc1ccccc1C(F)F c1(C(=O)NCC(CCCC)NC(=O)C(O)COC)cnc(C)c(N)c1 N1(C(c2c(C(C)C)ncs2)=O)CCC2(CCCC2NC(=O)C2=NNC(=O)C2)C1 C(=O)(C(C(F)(F)F)C(F)(F)F)OCC(=O)NC1Cn2c(C)nnc2CC1 N1(C(CC(C)OC)=O)CC2(CCN2C(c2ccc(=N)[nH]c2Cl)=O)C1 C1(NC(CC(COC)(C)O)=O)CN(C(C2CCCC(C)(C)C2)=O)CC2(CC2)C1 C1(NC(CSC)=O)CCN(C(c2cccc(-c3cnn(C)c3)c2)=O)CC1CO N1(C(CC2(C=C)CCC2)=O)CC(NC(=O)CCC(=O)NC2CCCC2)C(C)(C)C1 C1(C(=O)NC(CNC(C2N(CC)CCOC2)=O)C(C)C)(C)CC2(CCC2)C1 CC1CN(C(C2CC(Cl)(Cl)C2)=O)CC1NC(c1cc[nH]c1)=O C(CC(C)(C)C(=O)NC(C)CCCCNC(=O)C1=CSCS1)OC N1(C(C(CC)(C)C)=O)CC=C(CNC(=O)CC(C)SC)CC1 C1(N(C(C(CC)NC(N)=O)=O)CC)CCN(C(=O)CCS)CC1.c1ccccc1 c1(CC)ccc(C(C)C(N2CCCCC2CNC(c2ccoc2C)=O)=O)cc1 N1(C(CSCC(C)C)=O)CC(C)C2(CC2)C1.c1(CC=O)cccc(Cl)c1Cl.N C(C(O)C(=O)N)SC.c1(CCC(=O)N(CC)C2CC2)nnc(C2CCCC2)o1 c1(NC(C(C)N(C(=O)CN2CCSCC2)CCC)=O)ccc(O)c(Cl)c1 C1(N(C(c2c(C)ccn2C)=O)C)CCCN(C(c2cnc(NC3CC3)s2)=O)CC1 C1(NC(C2CC(OC)(OC)C2)=O)COCCC1C(N1CC(N(C)C)C1)=O c1(C(N2CCC(C)(NC(c3cc[nH]c(=N)c3N)=O)C2)=O)cc2cc(Cl)ccn2n1 C1(C(=O)NCCCCCCN(C(CCSCC)=O)C)Cc2ccc(F)cc2C1 c1(C(N2CC3CCC(C2)N3C(=O)C=Cc2cnc[nH]2)=O)ccc2c(=O)[nH]ccc2c1 C(CNC(c1ccc(O)nc1Cl)=O)(CC(F)(F)F)NC(=O)CCC1CCOC1 CC(C)CC(O)CC(=O)NCC1CCCCCN1C(=O)CC1CC=CC1 C(=O)(CCC(F)(F)C(F)F)N1C(C)CCC(CNC(c2c(C(C)C)nco2)=O)C1 c1(C(=O)NCC(C)(CO)NC(CCCCC=C)=O)cc(Br)c(C)nc1O C1(C(=O)OCCS(=O)(=O)NC2C(C)C2)CC(F)(C)C1.c1ccccc1.O Cc1nnc(O)c(C(=O)NC2CCC3CN(C(=O)CCn4cccn4)CC23)c1C c1(CC(=O)NC2(C3N(C(c4c(C)nco4)=O)CCCC3)CC2)ccc(Cl)c(Cl)c1 C1(NC(c2cc(COC)[nH]n2)=O)C2CCCC12.C(=O)C(CC)N(C)CCC.N N1(C(C(CC)CC)=O)CCOCC(C)(CNC(C2(F)CCS(=O)(=O)C2)=O)C1 C1(NC(CC2C(OCC)COCC2)=O)CC(F)(F)C12CCC2 N1(C(CCCCOCC)=O)CC(C(=O)Nn2cccn2)CCC1(C)C N1(C(C(C)(C)C2CCC2)=O)CC2(CCC2NC(=O)CCc2ccon2)C1 N1(C(C(C)NC(CC)=O)=O)CCC(NC(C2CN(CC(F)(F)F)C2)=O)C1.C C(=O)(C1CCc2cc(Br)ccc21)N1C2CC(CNC(CN(C)CC)=O)C1CC2 C(CCCCN=[N+]=[N-])NC(C(C)(CO)NC(=O)CC1CCOC1)=O c1(C(N(C2CCN(C(=O)CC3CCCCO3)C2)C)=O)cccc2ncnn12 C(N=c1[nH]c(=N)[nH]c(=NCCN2CCC3(CC2)CC3)[nH]1)c1c(C)cncc1 CS(C)(=O)=Nc1cccc(C(=O)NC2CCCC2NC(=O)Cc2ccsc2)c1 c1(CC)cc[nH]c1C(=O)NC(C1(C)CC1)C.C1(C)CCC1.C(=O)(C)N C(=O)(C(F)C1CC1)NCC1(N(C(=O)C=C2CCC2)C)CC1 C1(C(=O)NCc2cc(C(=O)NCCc3n(C)ccn3)on2)CCCC(=O)N1 N1(CCOCCNC(CN2CC(=O)NC2=O)=O)CCC(C2CCC2)C1 C12(C(N(CC(C)NC(Cn3c(C(F)F)cc(C)n3)=O)C)=O)CCCC(CO1)C2 Cc1conc1CC(=O)N(CC(C)CNC(C1CCCC1C)=O)C C12(C(N3CC(C)(OC)C3)=O)CC(CO)(CN1C(=O)CCOCCS)C2 C1(NC(CSCC)=O)CS(=O)(=O)CC1.c1ccc(C)cc1C.C(=O)(CC)N Cc1cc(C(=O)NCC(C)(C2CC2)NC(=O)CO)c(C)n1C.C1CC=CC1 N1(C(c2c(C)nccn2)=O)CCC2(CCCC2NC(=O)CCc2ccsc2)C1 C1(C(=O)NCCN(C(C)C)CC)CC2CC2N1C(C1(C#N)CCC1)=O N1(C(C=C(C)C(C)C)=O)CCN(C(=O)CCc2ccoc2)C(C2CC2)C1 c1(C(N(CC(C)NC(c2nc(CCC)oc2)=O)C)=O)snc(Cl)c1Cl C1(C(=O)NCC2(c3cc[nH]n3)CC2)COCCN(C(C2CCCSC2)=O)C1 C(CC(CC)C(=O)N(C1CCCN(C(=O)C2=COCCO2)C1)CC1CC1)=CC Cc1nn(CC(=O)NC2CC(C)(NC(C3CC=CC3)=O)C2)c(C)c1C=NO c1(N2CCN(C(C(=O)NC(CC)(C)C)c3nccs3)CC2)cc(F)ccc1F N1(C(c2cc(CC)ncn2)=O)CC(CNC(C2(C)CCCS2)=O)CC(CC)C1 c1(C(=O)NC2C3(C)CN(C(c4cc(C)n(C)n4)=O)C2C3)cccn2ccnc12 c1(CC)nc2ccccn2c1C(N1CCC(NC(=O)C(C)=C(C)C)C1)=O C1(C(N(C)Cc2cn(C(C(=O)OC)C)nn2)=O)CCN(C2CCCCC2)CC1 c1(CC)cccc(C(=O)NC2C3CC2N(C(=O)C(F)C2CCC2)C3)c1O c1(C=O)cncs1.CCCCNC(=O)C=CCOC(C)C.C(C)(C)C C1(NC(CCCCC#C)=O)CC2CC1CN(C(c1c(OC)cccc1OC)=O)C2 Cc1cccc(O)c1C(N1CC2CCC2(C(=O)Nc2ccc(Br)cc2CO)C1)=O N1(C(CSCCC(C)C)=O)C2CCC1CN(C(=O)C(C)(C)C1CCC1)C2 C1(NC(CCOC)=O)CCCCC1NC(=O)CC1CCCN(C(C)C)C1 CN1CCC(C(=O)NC(CCF)C(=O)NCC2(F)CC(O)C2)CC1=O Cc1cc(C(=O)NC(Cc2ccco2)C(=O)NC)cc(O)n1.c1nnc(O)n1C C1(Nc2cc(C(N)=O)ncn2)CC(NC(c2ccc(Cl)o2)=O)C12CCC2 N1(CC2CCN(C3CCCC3)CC2)CCN(CC2CC2)C(C#N)C1 CC(C)C(C(=O)NC(C)CC1CN(C(=O)C(C#N)=CC2CC2)C1)n1cnnc1 C1(NC(c2ncn(C(C)C)c2)=O)CCCN(c2ncc(O)cn2)CC1 Cc1cc(CNC(N2CCOC(C(C)O)C2)=O)ccc1-n1cccn1 c1(C(=O)NC2CN(C(COc3ccc(C)nc3)=O)C2)cc(N)c(F)c(F)c1Cl c1(C(=O)Nc2cccc(NC(c3c(C)oc(Cl)n3)=O)c2)ccn2cnnc2c1 C1(OC)CC(NC(c2cc(Br)co2)=O)CN(C(=O)COC2CCOC2)C1 C1(NC(C2C(C)CC=CC2)=O)CN(C(=O)C(F)(F)C2CC2)C(C)(C)C1 N1(C(C=CC(C)(C)SC)=O)CCCC2CN(C(=O)CN3CCN(C)CC3)CCC12 N1(CC)CCCC1CC(=O)NC(CNC(C1(CC)CC1)=O)C1CCC1 C(COC(C)=O)(C(=O)NOC1CCC1)NC(COCCCC)=O Cc1cc(C(=O)NC2CC3CN(c4nccc(C)n4)CC23)nc(C)c1 N1(C(c2ccc(C)s2)=O)CC(NC(=O)CC2CC3CCC2O3)C2CCCC12 C1(NC(=O)CCn2cc(Cl)cn2)CCN(C(c2coc(Br)c2)=O)CCC1CO Cc1cc(Cl)cc(N)c1C(=O)NC(C)CNC(c1c(C)ncn(C)c1=O)=O c1(C(=O)N)ccc(S(N)(=O)=O)c(N)c1.CC(C)(C)C(O)C(=O)N1CCC(C)C1 c1(C(=O)NCCC(C)NC(C2(C#N)CC23CCCC3)=O)cccc2nncn12 C1(NC(C2CCC(C(C)(C)C)CC2)=O)CC12CCN(C(C1(O)CC1(C)C)=O)CC2 C(CCOCCO)(C(=O)NC(c1ccccc1C)C)NC(C=NOC)=O c1(SC)ncc(C(N2CCC(O)C2C(=O)NC(C2CCNCC2)C)=O)c(Cl)n1 C1(C(=O)NCC(C)F)(NC(c2cn(C3CC3)cn2)=O)CCOCC1 N1(C(C(C)(C)C)=O)CC2(CCN(C(=O)CCc3cn[nH]c3)C2)C1 CS(=O)(=O)c1ccc(NC(c2ccc(C3CNCCO3)cc2)=O)cc1 c1(C(N2CCCC(NC(C3(C)CC(C#N)C3)=O)C2)=O)csc2c1CCCC2 n1(CCCn2c(C)ncc2)c(N2CCC(CC(C)C)C2)nnc1CC1CC1 c1(C(=O)NC(C(C)NC(C2CCC(CCC)CC2)=O)CO)cc(F)cc(F)c1O c1(C(=O)NCC2(C)CCCC2)ccc([N+](=O)[O-])cc1Cl.C1(C(=O)N)CC(F)C1 N1(C(C2CC3CN(C(C4CC(SC)C4)=O)CC3C2)=O)CCCC12CCOCC2 C1(NC(CSCC#C)=O)CN(C(c2cc(C3CCCCC3)[nH]n2)=O)CC1(C)C CC1CN(C(c2cncc(C(C)(C)C)c2)=O)CC1(C)C.C(=O)(CS(N)(=O)=O)N c1(C(=O)NC(CCC=C)(C)C)coc2c1CN(C(=O)C(C(C)O)N(C)C)C2 C1(NC(c2c(C)ccc(Br)c2)=O)CCCC12CCN(C(c1ccc(Cl)cc1)=O)C2 c1(NC(C2CCCN(Cc3ccc(I)cc3O)CC2)=O)ncc(Br)cc1O c1(CC(N2CCN(C(c3c(C)coc3)=O)CC2CO)=O)cccc2c(C)csc12 C(=O)(CCC(F)F)NC1(C)CN(C(=O)CCc2cccc(C(F)(F)F)c2)C1 N1(C(CN(C(C)=O)CCO)=O)CCC(N(C(=O)Cc2cscn2)C)C1 C#Cc1ccc(C(=O)N(C2CCN(C(=O)Cc3ccns3)CC2)CCOC)o1 C(=O)(C(CC)C(=O)N1CCC(O)C(NC(=O)C(=O)NCC(F)(F)F)C1)OC Cc1sc(C(N2CCCC2C2CCN(C(C3CC3C(N)=O)=O)CC2)=O)c(C)c1C c1(C(=O)N)ccc(-c2cccs2)nc1O.C1(CC(=O)N(C)CC)CC2(CC2)CO1 c1(C(N(C(C)CNC(C2CC(N(C)C)C2)=O)CC)=O)cnn2ccsc12 c1(C(=O)C(F)F)cccc(OC(C2(Cl)CC23CCC3)=O)c1 Cc1cc(O)ccc1CC(N1CC(NC(c2cc(Br)ccc2Br)=O)CC(F)C1)=O C1(NC(Cc2cnc(C(C)(C)C)o2)=O)CCN(Cc2cnccn2)CC1O Cc1ccc(CCC(=O)NC2CCCN(C(C3CC(F)(CO)C3)=O)C2C)cc1Cl N1(C(C(CCF)NC(C2C(C)(C)NC(=O)C2)=O)=O)CC2(C1)CC1(CCC1)C2 N1(C(CCCCOCC)=O)CC(NC(=O)COc2ccc(CC)cc2)CC(O)C1 N1(C(C(CCC)CC(C)C)=O)CCC2CN(Cc3ncc(Cl)n3C)CC2CC1 N1(C(C2C(CCC)C2)=O)CC(C(=O)N)C2(CCC2)C1.C1(C)CCC(O)CC1.C c1(NC2(C3CN(C(C(C)OCC)=O)C3)CC2)nc(C)cc(C)c1C#N CCC(C)C(CC(=O)N(C1CCN(C)CC1)C)NC(=O)C(F)n1ccnc1 C(CCNC(c1cc(C)ccn1)=O)(C(C)C)NC(C(=Cc1cnc[nH]1)C)=O c1(C(=O)N)ccncc1Cl.CC1(C)CC(C(O)CNC(=O)CCc2cnc[nH]2)C1 N1(C(c2ncc(C)nc2)=O)CC(NC(c2ncnc(O)c2Br)=O)CCC1C C(=O)(CS(F)(F)(F)(F)F)NCC(C)CNC(C1CCC(=O)N1)=O CC1(C)CN(C(c2c(F)cc(F)cc2F)=O)Cc2ccc(Br)cc21 N1(C(CC(C)C)=O)CCN(C(=O)CCn2c(C)csc2=O)CC1C1CC1.CCS CC(CCNC(C1CC1(Cl)Cl)=O)CCNC(C1(C)CC=CCO1)=O c1(CC(N2C(C)CC(NC(C3(CCF)CCC3)=O)CC2)=O)ccc2c(c1)OCO2 C1(CCNC(c2c(F)cccc2Cl)=O)CCCN(C(c2cnc(S)nc2)=O)CC1 N1(C(c2cccc(C)c2O)=O)CC2CC(NC(C3CCCCC3O)=O)C(C2)C1 c1(NC(C23N(C(c4c(CC)nn[nH]4)=O)CC(C2)C3)=O)cc(COC)ccc1C N1(C(c2[nH]cc(C)c2C)=O)CCCC12CCN(C(=O)C(C)Oc1ccccc1)C2 Cc1nc2ccccn2c1C(=O)NCC(C)(C)C.C1(C#N)(C(=O)N)CC12CCC2 C1(C(N2CCC(c3nc(C4CC4)no3)CC2)=O)CC12CCOC2 c1(OCC)cccc(CN2CCC(=O)CC2)c1 c1(SCCC(=O)N(C2CCN(C(C(CC)SC)=O)C2)C)ccccc1Cl c1(OC)ccc(Cl)c(C)c1C(N1CCC(NC(c2nnn(C)n2)=O)C(O)C1)=O N1(C(Cc2c(C)cccn2)=O)CCC(N(C)C(c2csc(O)n2)=O)C(C)C1 Cc1sc(S(=O)(=O)N2CCCC(C)C2)cc1[N+](=O)[O-].N(C)(C)CCO Nc1c(O)ccc(Cl)c1C(N1CCC(NC(c2ccncn2)=O)C(F)C1)=O C1(C(=O)NC(c2ncnn2C)C)CSCCN1C(C1C2(CC2)C12CC2)=O Cc1ccc(F)c(N)c1C(N1CCC2CCCC12)=O.C1(C(=O)N)CCS(=O)(=O)C1 C1(CNC(c2cnc(C)[nH]2)=O)N(C(=O)C2=CCS(=O)(=O)C2)CCCC1(C)C Cc1nc(C=CC(N2CCCC(N(C)C(c3cccc[n+]3[O-])=O)C2)=O)[nH]c1C C1(C2(O)CCN(N3CCOC3c3cccc(O)c3)C2)(C(N)=O)CCC1 CN1CCC(N(C(=O)C(O)C(F)(F)F)CCC(C(F)F)N2CCOCC2)CC1=O C(CCC(CO)NC(=O)Cc1ccccc1Cl)NC(C(C)n1cncn1)=O n1(CC(=O)NC)nnc2ccccc12.N1(C(C2(CN(C)C)CC2)=O)CCCC1.C N1(C(c2c(C)cc(C)nc2)=O)CCn2c(CNC(c3ncoc3C)=O)nnc2C1 Cc1cn(C)c(C(N2CCCC2C=Cc2cccs2)C(=O)NC2CC2)n1 c1(C(N(CCCNC(c2ccncc2F)=O)CC)=O)c(C)ccnc1C C1(O)(CNC(C(COC)OC)=O)CCCN(C(c2ccn3c2CCCC3)=O)CC1 N1(C(CCOCCOC)=O)CC(CC(=O)NC(C)CC(C)C(F)F)C2(CC2)C1 c1(C(N2CC(CC(=O)Nc3cccc(C(F)(F)F)c3)C2)=O)cc(Br)ncc1F N1(C(c2c(OC)ccc(Cl)c2C)=O)CCOC2CN(C(C3CC3C#N)=O)CC12 c1(CC(N2C(CNC(C(C=C)O)=O)CCCC2)=O)cn2c(C)csc2n1 c1(N2CCC(CSC)C2)cc(C)c(S(=O)(=O)NCC(c2ccccc2)C)cn1 C(=O)(CCC(C)(C)N(C)C)N1CCC(C)(CNC(C(CC)CC2CCCC2)=O)C1 Cc1nc2[nH]c(C(=O)NC3CC(NC(=O)C(C#N)C(C)C)CC3O)cc2s1 C1(CC(=O)NC2CC(CO)N(C(c3cnn[nH]3)=O)C2)CCC(O)CC1 C1(CC)CCC(C(=O)NCC(C(=O)N)N(C)C)O1.c1(CC2CC2)nn[nH]n1 c1(C(=O)NC(C)CCNC(=O)C(F)CC2CCC2)c[nH]c2cc(Cl)ccc12 C1(C(=O)NCCCCC#C)COCCN1C(=O)C(C)n1cncn1 S(=O)(=O)(c1csc2ccccc12)N1C(C(N2CC(CC)OCC2)=O)CC(F)C1 C1(CC(=O)NC2C=CCN(C(C(=CC3CCCC3)C)=O)C2)CCC(C)(C)CO1 c1(C(=O)NC2CC(O)(CNC(CCC#C)=O)C2)cn(C(C)C)nc1C C12(CCC(=O)NCC(CNC(c3ccoc3C)=O)OC)CCC(CC1)C2 C1(C(N2C(CNC(CCSCCCC)=O)CCC2)=O)CCCc2ccccc2C1 C1(C(N2C(CC(C)C)CC2)=O)CCN(C(=O)CCn2ccnn2)CCO1 Cc1cn(CC(N2CC(O)(C)C2)=O)c(=O)nc1O.c1(C(=O)N)ccc(C)c(N)c1 c1(COC)cc(C(=O)NC2CC2CNC(C2CC(OC)C2)=O)ccn1 C(=O)(C(C)(O)C(C)c1ccccc1)NCCCC.n1(C(C(=O)N)C)nc(C)cc1C C1(C)(C(=O)NC(CC)CNC(=O)CCc2cc(C)[nH]n2)CC2CCC1C2 S(=O)(=O)(c1cccc(Cl)n1)NC1CN(C(c2ccc(O)c(O)c2)=O)CC1O c1(CC)nncn1NC(=O)C1N(C(=O)CC2CCCC2O)CC12CCCC2 N1(C(C2(C)CC(C)OC(C)C2)=O)CCN(C(C2CCS(=O)(=O)N2)=O)C2(CCC2)C1 C(=O)(C(C)(C)C(C)(C)C)NC1(C2N(C(CC3CCN(C)CC3)=O)CCC2)CC1 c1(CC(N2CCC(NC(=O)C(c3ccccc3)O)C2)=O)ccc(Cl)c(Cl)c1 S(=O)(=O)(c1cc(F)ccc1F)N1CCC2(N(C(CC3C(=O)NC(=O)N3)=O)CC2)CC1 C1(NC(c2cnc(OC)o2)=O)CN(C(C2CC2c2ccc(C)o2)=O)CC1C c1(N(C(C(=O)NC)C)C)cnc(OC(F)F)c(C)c1 Cc1[nH]nc(CO)c1C(N1CCOC(C(=O)NCc2cnco2)C1)=O N(C(=NCCNCc1ccccc1)N)C(c1ncn(C)n1)C.[SH](=O)(=O)C(F)F C(=O)(C(=O)C(C)(C)CC)N(C(C(=O)NC(CC=C)CC(F)F)C1CC1)C C1(CNC(C(C)NC(C2CCC2)=O)=O)CCN(C(C2CC(F)(F)C2)=O)C1 CC(=O)C(C)CC(C)C(=O)N1CCC(F)CC1C(=O)N(CC(O)CF)C N1(C(CC(C=C)CCC)=O)CCCC12CCCN(C(=O)Cn1nnc(=O)[nH]1)C2 C1(NC(C2(COC)CCCCO2)=O)COC2(C1)CN(C(c1csc(O)n1)=O)C2 C1(CC)CCC(C(=O)NC2CCCC2NC(=O)C(C)CCOC)CC1 c1(NC(c2nnc(S)n2C2CC2)=O)nc2c(F)ccc(Br)c2s1 c1(C(=O)NCCCCN(C)C)nc(C2CC2)n(-c2ccccc2Cl)n1 c1(C(N2CCCC(CC=C)C2)=O)ccnc2[nH]c(O)nc12.C(=O)(C=C1CCC1)N C1(NC(c2nn(C)c(OC(F)F)c2)=O)CS(=O)(=O)CC1NC(=O)CCCC#N c1(C(N2CCN(C(C3C(CC)CCCC3)=O)C(C)C2)=O)ccc2c(n1)CCCC2 Cc1nc(O)c2ccc(C(N3CCC(NC(=O)C(F)F)C3C)=O)cc2n1 C(=O)(C1=CCC(C)CC1)NC1(CC)CCCN(C(=O)CCCN2CCCCC2)C1 N1(C(C2=NNC(=O)C2)=O)CCCCC(NC(C2C3(CCC3)C23CCC3)=O)CC1 Cc1c(C(N2CC3CC2CN3C(=O)NC2CCC(C)CC2)=O)cncc1Br CC(C)C(CNC(C12CCN(CC1)CC2)=O)C(=O)NCCC1C=CCC1 c1(C(=O)NCCC2=CCN(C(=O)CO)CC2)nccc2c(Cl)cccc12 C(C)(C(=O)NC1CCC1NC(c1cnc(N(C)C)s1)=O)(C1CC1)OC c1(C(=O)NCC(N(C(=O)C(C)(F)F)C)C2CC2)ccccc1-c1ncnn1C Cc1cn2c(n1)CC(C(N1CCN(C(c3ccc(C)[nH]3)=O)C(CCO)C1)=O)CC2 n1(CC(N2CC(C(C(=O)NCc3nncn3C)OC)C2)=O)cnccc1=O CS(=O)(=O)c1ccc(O)c(NC(c2ccc(C(F)(F)C(=O)O)cc2)=O)c1 CCCCCC(O)CC(=O)N1CCC(n2cc(C(C)(C)OC(C)=O)nn2)C1 N1(C(CCCCOC)=O)CCCC(O)(CNC(=O)C(C)(C)c2cnco2)C1 N1(C(C2CCC(C)(C)CC2)=O)CCCN(C(=O)CCC2CCC2)C(CO)C1 c1(C(=O)NCCCOCCNC(C2CCN(C)C2=O)=O)cc2cn[nH]c2cn1 C1(C(NOCCCOC)=O)CC2(CCC2)CN1C(c1csc(CO)n1)=O c1(CCC)nc(C)c(C(=O)NCC(C)C(C)C)o1.C1(N(CC=O)C)CCSC1 c1(C(=O)NCCN(C(=O)C=Cc2cncc(O)c2)C)c(Cl)cccc1[N+](=O)[O-] C1(C(N(CC)C)=O)CC(=O)CC12CCC2.C(=O)(CC)N(CC=O)C.CC.O c1(CC)n[nH]cc1C(=O)NC1(C)CC(C(=O)N(C(C)C(C)C)C)C1 c1(-c2nnc(CO)o2)ccc2nncn2n1 C(=O)(C(C)S(N)(=O)=O)NCC1(NC(c2c(NC)cnnc2)=O)CC1 C1(NC(Cc2ncc(C)s2)=O)CCCN(C(=O)CCCc2nccs2)C1C C1(C(=O)NC(C)Cn2cc(C3CCOC3)nn2)CCCN(c2ccn(C)n2)C1=O N1(CCNC(=O)CC2CCNC2)CCCCCC1 c1(OC)ccc(OC)c(CC(C)NC(=O)N(C2CCCC2C)C)c1 C(=O)(C(C)C(C)(C)C)N1CC(C(N(CC#C)CC)=O)C(CC)C1 c1(CC)ccc(C(N2CCCC(CC(=O)NC3CC34CC(OC)C4)C2)=O)cn1 CC1CCCC(C)N1C(=O)C(=O)NCCN(C)C(c1cc(C2CC2)ccc1F)=O N1(C(C(C2CCCCC2)C)=O)CCC(NC(=O)C2=CCOCC2)C(F)C1 c1(NC(C2CCN(C(=O)CC3(O)CCCCC3)C2)=O)nc(O)nc(O)n1 c1(C(C)C(=O)NCCN(C(=O)CC2CCCN2C)C2CC2)cccc(Cl)c1 c1(C(=O)NC(CNC(C(CC)(C)C(N)=O)=O)CO)ccc2nc(C)oc2c1 C(=O)(CCC(=O)N1CCCC1)N(C)CC1N(C(C(c2ccn(C)n2)C)=O)CCC1 C=CCC(C)(C)CC(=O)N(CC(=O)NC1Cc2cscc2C1)CC C(=O)(C1=CCC(F)(F)CC1)N1CCCC(NC(C2(c3cccs3)C(C)C2)=O)C1 Cc1c(C(=O)NCC(CO)NC(=O)CCOC)ccn1C1CC1.C1CCC1 c1(N2CCC(CC(=O)OCC)C2)ccncc1C(F)(F)F C1(C(=O)NC2(c3ccccc3)CC2)CCCC12CN(C(=O)NC1CCCCO1)C2 C1(CC(=O)NCC(CC)NC(=O)C(=Cc2ccccc2)OC)CCC=CCC1 c1(C(N(CCN(C(C)C)C(C2CC3C=CC2C3)=O)C)=O)ccc([N+](=O)[O-])n1C N1(C(CC2N(CC)CCOC2)=O)CC2CCC(C1)C(NC(=O)C(F)C(F)(F)F)C2 C1(C(=O)NCC(CC)NC(C=CC)=O)CCCCCNC1=O C=C=CC(C)C(=O)N1CCSCC1C(=O)N(CCOC)CCOC C1(NC(=O)NC2(CO)CCSCC2)CC2CC1CC2O CCC(C)CC(C(=O)N(CCCC(C)O)C)NC(=O)C(C)C(O)C(C)C C1(N(C(=O)Cc2cccc(O)c2)C)CN(C(C2CCCCN2N=O)=O)CC1(C)C CN1C(=O)CCC1C(N1CCCC(CCNC(=O)C(c2ccccc2Cl)O)C1)=O C(=O)(C(C)(C)CCF)N(CC(=O)NCC1CCC(C)C1)C1CC1 CC1C(C)N(C(c2ccc(Br)s2)=O)CCN1C(c1ccc(N)cc1O)=O N1(C(C(C=C)c2ccccc2)=O)CCCC(N(CCO)C(C2CC=CCC2)=O)C1 C(CCCCCNC(=O)CCCN1C(=O)CNC1=O)NC(C(C)C1CCOC1)=O C1(NC(CN(C(C)C)C)=O)CCCC1C(=O)NCCCOCC.C(N)=O c1(OC)cc(Cl)c(C)cc1C(N1CCC(CC)C1)=O.c1(C=O)cc(C#N)cs1.N N1(C(c2c(C)cc(N)cc2)=O)CC2CCC(C1)N2C(C1CCC2(CCOC2)O1)=O c1(-n2ncc(C(=O)NC(C3(O)CN(C(C(F)OC)=O)C3)C)c2)cccc(Cl)c1 c1(CC)cnccc1C(N1CCC(OC2CN(C(=O)CC3CSC3)C2)CC1)=O c1(C(c2nnnn2CC2CC2)NCC=C(C)C)cc(CO)ccn1 C1(C(N(C)CC2(NC(Cc3c(C)nc[nH]3)=O)CC2)=O)CC2CCC(C1)C2 C1(C)(C(=O)NC(CC)CNC(c2cn(CC3CCOC3)nn2)=O)CCNC1=O c1(OC)cccc(F)c1CC(=O)NC(C1CCCCC1)CNC(c1cnn[nH]1)=O C12(CN(C)CC)COCC1CN(C(=O)Cn1cccc1)C2 Cc1ccncc1CC(=O)NC(C)(C)C(=O)Nc1cnn(C2CCC2)c1 C1(C(=O)NCC(C)(C)C)COC2(CCN(Cc3ncc(Br)cc3Br)CC2)C1 C(=O)(C#CC1CC1)N.C(C(C(=O)NC1CC1)N(C)C)OC(C)C.C1CCC1 c1(C(=O)NCC2C(NC(CCC(=C)Br)=O)CCC2)ccc(C)cc1OC Cc1ncc(N)cc1C(=O)NCCN(C1CCCCC1)C(=O)C(C)C1CCC1 c1(OC(C)C)ccc(OC)c(CN2CC3(CC3)CC2Cc2ccccc2)c1 c1(CN(CC(CC)C)Cc2ccc(Cl)cc2)c(F)cnc(Br)c1C c1(C=O)cccc(Cl)c1C.C(C(=O)NC(C)C1CCC1)(C1CCC1)OCC.N c1(C(=O)NCC2(F)CC(CNC(C3(C)C=CCC3)=O)C2)ccccc1F C12(NC(C(CC)n3nccc3C)=O)CC1CN(C(c1cnc(O)o1)=O)C2 C(COC)(CC(=O)NC1CCC(F)(F)C1)NC(C1(CCCC)CCC1)=O c1(CC(N2C(C(=O)NCC3OCC(=O)NC3)COCC2)=O)ccn2nccc2c1 Cc1nc(-n2nc(CCOC(C)C)nc2C2CC2c2ccsc2)n(C)n1 c1(C(N(C)CC2CCCN2C(=O)C=CCO)=O)ccc(F)cc1[N+](=O)[O-] c1(C(N(CC(C)C)C)=O)cn(C)nc1-c1ccccc1.C1CC1C=O.COC c1(C2C(NC(c3c(Cl)csc3Cl)=O)C2)ccncc1Cl C1(NC(c2cnn(C3CC3)c2)=O)COC2(CCN(C(=O)CSC(F)F)C2)C1 C=CCC(CC)C(=O)NCc1nc(CNC(=O)CCN2CCCC2=O)cs1 c1(CNC2(CC(=O)Nc3ccc(F)cc3F)CCC2)c[nH]c2nccc(Br)c12 N1(C(C(C)C2CC2)=O)CC(CNC(=O)CCNc2ncc(F)cn2)C(C)C1 c1(C(=O)NCCC(CNC(C2ON=C(CC)C2)=O)O)cnc2ncnn2c1C CC(C)(C)C(C(=O)NCC#CCNC(C1CCCCC12CC2)=O)NC(N)=O C(=O)(C1=Cc2ccccc2OC1)N1CCCC(CCN=c2[nH]cnc(C)c2Br)C1 C(CN=c1[nH]c2c(c(=NCC(CSC)OC)[nH]1)COCC2)N(CCC)C1CC1 Cc1nc(NCC(c2ccc(F)c(F)c2)C)cc(N2CC3C(C2)C3(F)F)n1 c1(C2C(C(N(CCCCNC(=O)CCC3CCCO3)C)=O)C2)cccnc1 c1(C(=O)NC(C)(C)C)ncc(Cl)s1.n12cc(nn1)C(C)(C)NC(=O)C2C C(=O)(CCC1=CCCCC1)NC(CC(=C)Cl)C(=O)NCC(O)CC(F)(F)F CN1CCC(C)(C(N2CC(NC(=O)COc3ccc(Cl)cc3)C(F)C2)=O)C1=O CN=c1cc(C(=O)NCC(CNC(=O)C(F)CC(C)C)OC)cc[nH]1 C1(CNC(C=NOC)=O)CC(F)(F)CN1C(=O)CC1COCCO1 C(C)(C)(C(=O)N1CC(CCNC(C2CCN2S(C)(=O)=O)=O)C1)SC c1(OCC)cncc(C=O)c1.c1(C(NCC)=O)cnn(C2CC2(F)F)c1.N C1(NC(CC(C=C)C)=O)CCCN(C(c2cncc(C)c2C)=O)C1C c1(C(=O)OCC)cc2cc(NC3COc4cccnc43)ccc2o1 C#CCCCCC(=O)NCCC(C)NC(C1(C)COC(=O)OC1)=O c1(C(N2CC(NC(C(C)SCC)=O)C(n3cccn3)C2)=O)cc2occc2n1C N1(C(c2c(OC)ccc(F)c2)=O)C2CCC1CN(C(C1C=CCC1)=O)C2 c1(CC)ccc(OCC(=O)N)cc1.C(C)(C)CCN(C(=O)CC)C.C(C)=O C(C(O)CC(C)C)NC(C1(NC(c2ccc(CC)o2)=O)CCSC1)=O Cc1nc2ccc(C(N3CCN(C(=O)CC4CN(C)C4)CCC3C)=O)cn2n1 C1(C(C)=O)C(CC(=O)NC(C2CCOC2)CNC(C2CC2)=O)C1(C)C.C CC(C)CC(C)(CN=c1nn[nH]n1C)NC(C1CC(C)(C)C1)=O C1(C(N2CCC(NC(=O)CC=C(Cl)Cl)C23CC3)=O)OCC2COCCC12 C1(O)(C2(C)CC2)CN(C(=O)C(c2ccco2)NC(=O)CC2CCC2)C1 c1(CNC(C(C)N(C(=O)C(C(C)C)C2CCC2)CC)=O)ccc(C)cc1O c1(C(N2CCC(OC)C2)C(=O)NCCC#N)ccc2cc(Br)ccc2n1 N1(C(C2OCCC(C)C2)=O)CC(C)(C)CC(C)(C)C1.C(=O)CN(C)C(N)=O.N c1(NC(=O)NC(C)(CCF)C(=O)O)cnc2[nH]nnc2c1 C1(C(=O)NC(C2CCCN2C(=O)CO)C)Cc2c(F)cccc2O1.c1ccsn1 N1(CC)CCOC(c2nc(-c3cncs3)nn2-c2cnn(CC)c2)C1 C1(NC(C(CC)(C)C)=O)CCCCN(C(=O)CC(C)n2ccc(C)n2)CC1 CCCC(C(=O)NCC1CC1[N+](=O)[O-])NC(C1CC1(F)F)=O c1(C(=O)NC2(COC)CCCN(C(C(CC=C)(C)C)=O)C2)ccc2ncnn2n1 C1(C(=O)OCC)(NC(=O)CCCOC)CCCCC1.C(=O)(C(C)OCOC)N Nc1c(F)ccc(F)c1C(=O)NC1CCN(Cc2ccccc2)C1(C)C O=C1CN(C(C2CCCCC(F)(F)C2)=O)C2CCN(C(=O)CSC(F)F)CC2N1 C1(CC(=O)N(CC(COCC)(C)C)C)CN(C(=O)C(O)CC)CCO1 Cc1cn2cc(-c3ccc(C(=O)NCCCN4CCC(C)CC4)cc3)nc2s1 c1(C(=O)NCC(O)(C2CC2)C2CC2)cc2c(s1)CCC(c1ccccc1)C2 C(=O)CS(=O)(=O)N1CCCC1.C(C(O)CC)N(C(=O)C(C)(C)N1CCCC1)C.N N1(C(c2cnc(CC)s2)=O)CC2CC(NC(=O)C(F)(F)c3ccccc3)C2C1 CN=c1[nH]c(=NCC2CN3CCN2CC3)[nH]c(=NCC2CCCC3(CCC3)C2)[nH]1 C1(C2CC2)(C(=O)NCC(N(OC)C)=O)CN(C(C23CCC(CC2)C3)=O)C1 N1(C(CSCCOC)=O)CCCC1C(=O)NCc1[nH]nnc1C O=C(C1=CCN(C(C2CCN(C3CC3)C2)=O)C1)N1CC2CCC1C2 c1(C(N(C2CCN(C(=O)C(C)C(C)O)C2)CC)=O)cnc(OC)c(Cl)c1 N1(C(CC)=O)CCC(CNC(=O)Cn2nc(C)c([N+](=O)[O-])c2C)C(F)(F)CC1 c1(C(=O)NCCCC(C)NC(CC(CC)(C)C)=O)cc2ccc(F)cc2s1 N1(C(CCN(C(C)=O)C)=O)CC=CC(NC(=O)C(F)(F)C2CC2)C1 c1(C(C(=O)N(C)Cc2cn(CCOCC)nn2)CC)cccc(Cl)c1 C(=O)(C(C)(C)C(C)(F)F)NC1CCC(NC(CSCCC(C)C)=O)CC1 Cc1ccc(C(N2CCC(C(O)CNC(C3CCCOC3)=O)CC2)=O)cn1 c1(C(C(=O)NC(C)CCNC(c2ncccc2F)=O)O)ccc2ccccc2c1 C(=O)(C1=CC2(CCN(C(C3CCC(C)(C)C3)=O)C2)C1)N1CC(C)(C)SCC1 CCCCCC(F)C(=O)NC1(CC)CN(C(c2cc(C)c(O)nn2)=O)C1 CCCC(C(=O)NC1CCC(CCNC(=O)CSC(C)(C)C)C1)OC c1(C(N(CC(C)N(C(=O)CN2CCC(C)C2)C)C)=O)ccc(O)c(Br)c1 Cc1ccn(CCNC(C2(O)CCN(C(=O)CN3CCCCC3)CC2)=O)c(=O)c1 N1(C(C(CC=C)OC)=O)CCC(CNC(C2CCOC2C2CC2)=O)CC1C C1(C(=O)NCC(C(C)C)NC(C(Br)=C(C)C)=O)OC2CCCCC2C1C Cc1cc(CC(=O)N(C2C3CN(C(C4CCCN4C)=O)CC23)C)cc(O)n1 c1(C(=O)Nc2ccc(OC)cc2OC)csc2c1CCN(S(=O)(=O)CC#N)C2 N1(C(c2cccc(Cl)n2)C(=O)NC(C)(C)C)CCCCC1CC1CCCCC1 CC1CC(N(C(=O)C(C(C)(C)C)NC(c2csc(=N)[nH]2)=O)C)CC(C)C1 c1(C(N2CC(NC(C3(S(N)(=O)=O)CC3)=O)CC(C)C2)=O)ccc(C#N)cc1F N1(C(c2c(C)noc2)=O)CC2CN(C(=O)CC(C)P(C)(C)=O)CC(C1)O2 Cc1[nH][nH]c(=N)c1C(N1CCN(C(c2ccc(CC3CCC3)cc2)=O)CC1)=O N1(C(c2nc(Br)n[nH]2)=O)CCC(C2CNC2)CC1 c1(OC)cc(Br)ccc1CNC(C1CC1C(=O)Nc1cncc(Cl)c1C)=O c1(CNc2ccc(OC)c(OC)c2)c(Br)ccc2c1OCO2 N1(C(CC=CC)=O)CCCCC1C(C)NC(c1sccc1C(=O)OCC)=O C1(CC)CCC(C)N(C(=O)CSCCNC(=O)CCN2CCOC2=O)C1 N1(C(C(C)OC)=O)CC(NC(c2ccc(Cl)o2)=O)CCC1C C1(C2CCCN(C(C3(CO)COC3)=O)C2)(NC(C2CCN3CCOCC23)=O)CC1 c1(OC)ccc2cnc(C(=O)NCCCC)cc2c1.C1(C)(C(=O)N)CC2(CC2)C1 N1(C(C(C)C2CC2)C(=O)OC(C)(C)C)C(=O)C2CCC(O)CN2C1=O O=C(C1CCCc2cncn21)NCC1(O)CCN(C(C2CSC2)=O)C1 C1(O)(CNC(c2ccc(CC)s2)c2nnnn2CC2CCOC2)CCOCC1 C1(N(C(C(C2CCOC2)OC)=O)C)CCC(NC(c2ncsc2C(C)C)=O)CC1 O([Si](C)(C)C(C)(C)C)CC(C)C1CCC1.C1(C(C)=O)CCc2cscc2C1 c1(C(=O)NC2CCC(CC(=O)NCC(CCC)O)C2)cccc(C)c1 C1(CNC(c2nc(Cl)cs2)=O)CCN(C(c2csnc2C2CC2)=O)CC1 c1(OC)ccccc1OCCN(C)C(C1(C)CCCN1C(=O)C(C)C)=O CC(CCCNC(=O)CCc1ccsc1)NC(c1ccnn1C1CC1)=O c1(OCC)cc(C(N2CC(CNC(=O)C3CC3)CC(C)O2)=O)ccc1O Cc1cc(C(=O)NC(C(=O)NCC(CC2CC2)CO)c2ccoc2)oc1C c1(CNC(c2cc3cnccc3[nH]2)=O)cccn2nnnc12 C1(C(NOCC)=O)(CC)CCCN(C(c2cnc(=N)[nH]c2)=O)C1 [N-]=[N+]=NC1(C(=O)NCCCF)CCN(C(=O)CC2CC3(CC3)CO2)C1 c1(C(N2CCC(C(C)NC(C=CS(CC)(=O)=O)=O)C2)=O)nccc2ccccc12 CCC(CC(=O)N(CCCC(=O)NC(C)C(C)(C)O)C)C(C)C c1(OC)ccc(C(C)CC(=O)NC(C)(C)CO)cc1.c1(CC(=O)N)sccc1C c1(CC)cccc(C(N2CC(C(C)NC(=O)C(CC3CCC3)SC)C2)=O)c1F N1(C(C(C)OC2COC2)=O)CC2CCN(C(C3(C)CCC(=O)NC3)=O)CCC2C1 Cc1ccc(C(N2CCN(C(c3csc4nccn34)=O)C(C)C2)=O)nc1C c1(NC(C2OCC(C)C2)=O)cccc(NC(c2cnc[nH]2)=O)c1 CC(C)(C)C(F)(F)CNC(=O)NCC(c1ccccc1Br)(F)F N1(C(CC(C)(C)N(C)C)=O)CC(NC(c2c[nH]cc2C(F)(F)F)=O)CC(O)C1 N1(CC=C)C(=S)NC(c2cscc2F)C2=C1CN(c1ccc(F)cc1)C2=O N1(C(C2N(C(c3cc(OCC)n[nH]3)=O)CC=C2)=O)CCOCC(C)(F)C1.[S+]C CN1CCC(F)(CNC(=O)C(CCC2CC2)NC(=O)CS)C1.CC(F)F c1(C(N2CCCC2)=O)ccc(S(N)(=O)=O)c(F)c1.CC1=NOC(C)(C(=O)N)C1 C1(C)(C(N2CCC(C)(CO)C2)=O)CCC(F)(F)CC1 C12(NC(c3n[nH]cc3F)=O)CC1CN(C(c1ccc(Nc3nccs3)cc1)=O)C2 CS(=O)CCC(=O)N1CCC(N(C(=O)CC2CC(CC3CC3)C2)CCO)CC1 N1(C(c2nc(CCCC)sc2)=O)CCN(C(=O)C(O)c2ccco2)CC1C(F)F C#Cc1ccnc(C(=O)N(C)CC2CCN(C(c3ccc(OC)nc3)=O)C2)c1 C1(F)(CNC(C2CCC(O)CC2)=O)CCN(C(C2CCC3(CCC3)O2)=O)CC1 C(CCS(C)(=O)=NC(=O)C1CCC12CCOCC2)(C(C)(C)C)OC(C)(C)C c1(CN(CCN(C(c2cc(C(C)=O)[nH]n2)=O)C)C(C)C)cccc(C#N)c1 C(N=c1[nH]c(=NCC(C)(C)CCCO)c2[nH]ccc2[nH]1)C1(CCOCC)CC1 C1(C(=O)NC(C(N2C(C)(C(C)C)CC2)=O)C2(O)CCC2)CCCN1C=O CN=c1[nH]nc(CC(=O)NC2(CNC(=O)CCC3CCC(=O)N3)CCOC2)s1 Cc1cccc2sc(C(=O)N(CCCN(C(=O)CC(C)(C)N(C)C)C)C)c(Cl)c12 C1(C(=O)NC(C(=O)NCCCc2nc(C)[nH]n2)CCF)C2CCC(F)(F)C12 N1(CC)C(=O)CCC1C(N1CC(C)CC1C)=O.c1(CC(=O)N)cccc(N)c1 C(=O)(C(C)C(O)C(C)C)NC1(C)CC(NC(c2ccc(OC)c(C)c2)=O)C1 c1(C(N2CCCC2(C)C)=O)ccc(Cl)c(Cl)c1O.c1(OC)cc(C=O)n(C)n1.N N1(C(C(N2CCC(C)C2)=O)=O)CC2(CCC(NC(C3(C#N)CC3)=O)C2)C1 CC(C)C(C(=O)N1CCCC1C)N1CCCS1(=O)=O.C(c1nccs1)=CC=O.N N1(C(C(NOC)=O)=O)CCC(n2cccn2)(NC(C23CCC(C)(C2)OC3)=O)CC1 C1COC2(CCN(C(C3CN(C(=O)CO)C3)=O)C2)C1.O=CC.C=O.C1CC1.N N1(C(CC2CCC2)C(=O)NC2CC(CO)C2)CCOC(C2CCOC2)C1.CS CCCCC(C)(F)C(=O)NC(CCOCC)C(C)C C=CCCCC(=O)N(CCNC(=O)CC(CC)OC)Cc1ccccc1 CC(C)(C(=O)N=c1ccn(-c2ccc(F)cn2)[nH]1)C1(O)CCOC1 NS(=O)(=O)c1cc(C(N2CCC(NC(C3C=CCC3)=O)C23CC3)=O)co1 c1(OCC)ccc2c(c1)C(NC(=O)NCc1ccc(OC)nc1)CCO2 c1(NC(C2C(NC(=O)CN3CC=CC3)CCOC2)=O)ccc(O)c(=O)cc1 O=C(O)C(CNC(=O)CC(Cl)Cl)C1CCCCC1 C(=O)C1CC(=O)Nc2ncccc21.c1cc(C)cc(C)c1.CCCCNC(=O)C(C)C CC1(C)CC(NC(c2occc2Cl)=O)CN1C(c1cc2c(s1)CCC2)=O CCC(C(O)C(C)C)NC(C1CC2(CC2)CN1C(c1ccc(C#N)s1)=O)=O c1(C(N2CC(Cc3ccc(Cl)cc3)C2)=O)ccc2ccccc2c1F n1(CC(=O)NCC2CCC2)cc([N+](=O)[O-])cn1.c1ccsc1.C1(C=O)CC1 C(=O)(C(=O)C(C)(C)C)N1CCC(O)(C(C)NC(C2CC(C)(C)C2)=O)C1 c1(C(N(C)CC2(F)CCC2)=O)ncc2cnccn12 c1(C(N2CC(C)CC2)=O)ccn(C)c(=O)c1.c1(CC)ccc(C(=O)NC)nc1 N1(C(c2ncc(C)nc2)=O)CCCOC(CNC(=O)CCCN=[N+]=[N-])C1 c1(COC)ccc(C(=O)N(CCCC)C)[nH]1.C1(n2cccc2)(C(=O)N)CCCC1 C12(NC(c3n[nH]c(C)c3C)=O)CCCCC1N(C(c1c[nH]c(C(N)=O)c1)=O)CC2 c1(C(N2CC3CCCC3(C=O)C2)=O)ccc(S(=O)(=O)CC2CC2)cc1.C1CC1 C=CC(C)(C)C(=O)NC1CCC(C)(CNC(c2oc(C)nc2C)=O)C1 C(=O)(C1(C)OCCc2ccccc21)NCC(CN(C(=O)CCCS(C)(=O)=O)C)O c1(OC)ncccc1CNC(=O)NC1C(Oc2nc(C)cs2)CC1O C1(C(C)NC(C=C(C)C2CC2)=O)CN(C(=O)C(C2CC2)C2CC2)CCO1 c1(C(N2C(CNC(C(C=CC)O)=O)COCC2)=O)cccc(F)c1Br N1(C(C(C(C)C)NC(N)=O)=O)CCC2(CCCN(C(=O)C(F)F)C2)C1 N1(C(c2n(CC=C)ccn2)C(=O)NCCOCC)CCCCC1CCC c1(C(=O)NCC(CNC(CCCc2onc(C)n2)=O)O)c(N)sc(C)c1C C#CC1CN(C(=O)CC2CC(CC)C2)CCN1C(=O)CCCC(=O)N(C)C c1(NC2C(C)c3c[nH]nc3CC2)c(F)cc([N+](=O)[O-])cc1F c1(C(N2C(C)CN(C(CCC#C)=O)C(C)C2)=O)ccc(S(=O)(=O)C(F)F)cc1 N1(C(Cc2c(C)ccs2)=O)CCCCC12CC(NC(=O)CC1CC13CC3)C2 Cc1cc(C(N2CC(NC(=O)COC)C(O)C2)=O)cc(C)c1Cl.c1ccncc1 C(=O)(C(C)N(OC)C(=O)CC(C)(C)C1CCN(C(c2csnc2C)=O)C1)OC c1(OC)ccncc1NC(=O)C(C1CCOC1)NC(c1ccc(C)nn1)=O CC1CN(C(c2ccc(Cl)s2)=O)CCCN1S(=O)(=O)CCCl N1(C(C2C(C)(C)OCC2)=O)CCC(C(N2CC(C(=O)N(C)C)C2)=O)C1(C)C C12(CNC(C3(C)C(C)OCC3)=O)CN(C(=O)C(C)n3cncn3)CC(F)(C1)C2 Cc1nn(C)c(C)c1NCC(=O)NCC1CCCCN(C(=O)CC(C)F)C1 c1(-c2c(C(=O)NCCCN(C(C(C#C)(C)C)=O)C)cn(C)n2)ccc(C#N)cc1 N1(C(CCNC(=O)OCC)=O)CC(C)(C)CC1C(=O)NC.C1(O)CCC1 O=C(CC=C(Cl)Cl)NCC1(F)CCC(NC(=O)C(O)C2CCC2)C1 C12(C(=O)NC(COC)C(C)C)CC1CCN2C(C1CCC1(OC)OC)=O c1(C(=O)Nc2ncccc2C2CC2)cccc(-n2cc(-c3cn[nH]c3)nn2)c1 c1(C(N2CCN(C(C3(CC)CC3)=O)CC2CCO)=O)cc2c(cn1)COCC2 N1(C(c2ncc(F)cc2F)=O)CCC2(CC1)CC2C(N1CC2CCC(O)C2C1)=O C1(C)CCN(C(=O)CC)C1.C(CCC(=O)N)N(C(=O)OCC)C.C(C)C.C S(=O)(=O)(c1cc(Br)c(F)cc1F)N(C)CC1CCCN(C(C2(C)COC2)=O)C1 c1(OC)cc(C)cnc1C(=O)NC12CCC1CN(C(=O)CCCc1nccs1)C2 C12(NC(c3cc(C)c(C)[nH]3)=O)CCCC1N(C(c1nc(O)sc1C)=O)CC2 N1(C(CN(C)CCO)=O)CC2(CCCCN2C(=O)CCc2nnc(S)nc2O)C1 Nc1cc(F)c(O)cc1C(N1CC(F)(CNC(=O)C(F)n2ccnc2)C1)=O c1(C(N2CC(C)CC(CC)C2)C(=O)NCCCSC)ccc(S(N)(=O)=O)cc1F C(=O)(C(O)C1=CCCCC1)N1CC(COC)C1.C1(CC=O)CC(C)(C)CO1.C c1(C(CCC=C)C)nc(-c2cccc(Br)n2)nn1CC1CCCCC1 N1(C(c2cccc(CC)c2)=O)CCC2(CCN(C(=O)CSC(C)C)CC2)C(C)C1 c1(C(=O)NC2C(OC)CN(C(C(CC)O)=O)C2)ccc(OC(F)(F)F)c(C)c1 Cc1ccc(Cl)c(OCC=O)c1.C(=O)C(C)CSC(F)(F)F.C1(CC)CC1.N N1(CC(C)NC(c2nnc(S)n2C)=O)CCN(C(c2ccn(C)n2)=O)CC1 c1(C(=O)OC)cc2c(=NC(CCOC)c3ccc(N(C)C)cc3)nc[nH]c2n1C c1(C(=O)NCCC(C)S)ccnc2c1ccn2C C(c1ccc(C)cn1)=CC(=O)NCC1OCCN(C(CC(=O)OCC)=O)C1 C=CCCCCC(=O)N1CC(OC)CC1CNC(=O)CCc1ccccc1Br CC1CN(C(=O)Cn2ccnn2)CC1NC(c1ccccc1C(C)(C)C)=O c1ccn(C)c(=O)c1.CC(CC1CC1)C(=O)NCC1(C(=O)NC)CC1 C1(C(N(C(C)C)CC)=O)COC(C)(C)CO1.c1(C=O)ccccc1.C(C)=O C1(CC)C(C(=O)NC(CC2CC2)C(=O)N)CCCN1C(=O)CC(C)C(F)F C#CCC(C(=O)NC(c1n[nH]c(CC)n1)C)NC(C1CCC2CC12)=O N1(C(C(C)(C)F)=O)CC(NC(=O)C=Cc2cn[nH]c2)C(N=[N+]=[N-])C1 N1(CC2CCC(CCC)CC2)CC2(C1)CN(c1nc(OC)cc(OC)n1)C2 N1(C(CC2CC(CC)OCC2)=O)CCC2(CC1)CCN(C(=O)CSCC(N)=O)C2 c1(C(N(C2CC(C)(C)C2)C)=O)coc2c1CN(C(C1CC1(F)Cl)=O)C2 c1(N2CCC(N(OC)C)CC2)nc2ccccc2c(=NCCC2CCCO2)[nH]1 c1(C(N2CCC(NC(C3CCCC(C)C3C)=O)C2)C)ccc2ccccc2n1 CCCC(C)NC(=O)C(C)(C)NS(C)(=O)=O.C1(CC(=O)N)CC1(Cl)Cl Cc1nc(C2CC2)cc(=NCCSC(F)(F)F)[nH]1 C(CS(=O)(=O)CC(=O)N1CCC(NC(=O)Cc2ccc(C)c(F)c2)CC1C)OC c1(CN(C2CC(O)CN2C)C)cc(Br)ccc1[N+](=O)[O-] N1(C(CC2C(C)CCCC2)=O)CCCC(C)(CNC(C2(O)CC(C)(C)C2)=O)C1 C1(C)(C(=O)NC(C)CC2CN(C(C3(CCO)CC3)=O)C2)CC=CCO1 C(=O)(C1COc2ccc(Cl)cc21)NC1CCCN(CC(COC)O)C1 C1(NC(C2CCCC2)=O)CN(C(=O)C(O)Cc2ccccn2)CC12CCC2 C1(NC(=O)COCCCF)CN(C(c2c[nH]nc2-c2cccs2)=O)CC1O c1(C(CC)=O)ccc(Cl)c(NC(=O)CN2C(C)CCC2C)c1 c1(C(N)=O)cc(C(=O)NC2CCCC(NC(=O)Cc3cn[nH]c3)C2)ccc1O C(=O)(C(F)(CC)C(=O)OC)N1CC(NC(C2C(CC)CCCC2)=O)C1 c1(OC)ccc(Cl)cc1C(=O)NCC(C)NC(c1ccc(-c2csnn2)cc1)=O C1(C(N2CCC2)=O)C2CCC(O2)C1C(F)(F)F.n1(CCCOC)cc(C)nn1 N1(S(C2(CC)CC2)(=O)=O)CCOC2(CC1)CCS(=O)(=O)C2 C12(C(=O)NC3C=CCN(C(Cn4cnc(C(N)=O)n4)=O)C3)CCC(C)(CC1)C2 c1(C(=O)N)ccc2[nH]ccc2n1.c1(CNC(Cc2cnc(C)s2)=O)ccccc1C C12(CNC(=O)CCNC(=O)CC3CC34CCCC4)CCC(CC1)OC2 C1(NC(CS(CC)=O)=O)CC(F)CN(C(=O)CCc2ccc(Cl)c(Cl)c2)C1 C1(C(N(C2CCN(C(C3CC(F)(F)C3)=O)C2)CC)=O)CCN(C2COC2)C1 c1(CN(C(=O)C(C)=CCNC(c2ccccn2)=O)CC)occc1C c1(C(=O)NC2CN(C(c3ccc(CSC)cc3)=O)C3C2C3)cc(C)cc(O)n1 N1(C(C(C)SC)=O)CCCC2(C1)CN(C(c1cccc3c1CCC3)=O)CCO2 c1(C(=O)NC2CN(C(c3cccc(OC)n3)=O)CC2O)ccc(C)c(F)c1 c1(NC(c2cc(OC)nn2C)=O)ccc(OC)c(F)c1.N1(C)CCOCC1 C(=O)(C(C)C(C)(F)F)NCC(CC)(C)NC(=O)C(=O)N(C)OC N1(C(CNS(NC)(=O)=O)=O)CCCOC(CNC(c2csc3nccn23)=O)C1 CCCCCCCC(=O)NC(CN(C)C)C(N1CCOCC1CC1CC1)=O N1(C(c2c(CC)[nH]c(=N)s2)=O)CCN(C(c2sccc2CO)=O)CC2(CC2)C1 Fc1ccc(Br)cc1NCCCOCCCC1CNC1 Cc1ccc2sc(NC3CCC4CN(C(=O)C=Cc5cccnc5)CC34)nc2c1 N1(C(c2ccc(CC)[nH]2)=O)CCC(C)C1C(=O)Nc1cccc(O)c1 c1(NC(C2N(C(C=C(COC)C)=O)C(C)C2)=O)ccc(C)cc1CO C1(CCCC)CN(C(=O)COCC2CC2)CCN1C(=O)CN(C)C C1(CC(=O)NCC(CC)(C)O)CCN(C(C2CCCN2C)=O)C1(C)C CC1(C)CC(C)N(C(c2cc3n(n2)CCC3)=O)C1.C(c1ccc[nH]1)=CC(=O)N N1(C(C(CC=C)(C)C)=O)CC2CCCC(NC(c3cc(CO)c(C)o3)=O)C2C1 C(=O)(C1CCCc2ncc(C)n21)N1C2C(NC(c3cc(C)nnc3)=O)CC(C2)C1 C(=O)(C1COc2ccccc21)NCCN(CCC)C(c1ccnc2ccsc12)=O N1(C(c2cc(C)no2)=O)CC(F)(F)CC1C(=O)NC(c1ccc(Br)cc1)C C1(N(C(=O)CC2CC2C)C)CCC(NC(=O)Cn2cc(C(C)O)nn2)CC1 c1(CNC(=NCC2CCC2)NCC2CCC(C)O2)ncccc1C(C)OC c1(C(C)NC(N(CC#C)CC2CC2)=O)ccc(C(F)(F)F)nc1C c1(C(N2C3CN(C(c4ccc(C)o4)=O)CC32)=O)ccc2cc[nH]c2c1 N1(C(c2ccc(=N)[nH]n2)=O)CCCC(CO)C1.C1(C(=O)N)CC(=O)N(C2CC2)C1 C1(NC(CCC#C)=O)(CF)CCN(C(c2cnn(C)c2CC)=O)C1 c1(-n2cc(COC(C)=O)nn2)ccc(F)c(NC(=O)CC(=O)N2CCCC2)c1 N1(C(C2COCC(C)O2)=O)CC23CCCC2(C1)CN(C(C1CC2CC2C1)=O)C3 C(CCOCCO)(C(=O)N1CCC(F)(CF)C1)NC(C1CCSCC1)=O n1(CC(N2CCN(C(c3cc(O)cs3)=O)C3CCC23)=O)ncn2cccc2c1=O C=C(C)CCCC(=O)N1CCOCC(CNC(c2ccc(OC(F)F)cc2)=O)C1 c1(SC)cccc(C(N2CC(NC(=O)C=CC(F)(F)F)CC(O)C2)=O)c1Cl c1ccc(O)c(C(C)(C)C)c1.CCC(C)(C)C.CC(=O)NC.CN(C)CC.O c1(C(=O)OC)c(NCC2CN(C(=O)CC3CC4C=CC3C4)CCO2)ncnc1Cl Cn1cnc(Br)c1C(N1CCNCC1)C(=O)N(C1CC1)C1CC1.C(C)(C)C.C N1(Cc2c(Br)cc(C)c(C)n2)CCCCC1C1(C)CCCO1 Cc1c(C(=O)NC(CO)C(C)NC(=O)C(C)CC(C)(C)C)sc2cc(F)ccc12 N1(C(c2c(SC)cccc2)=O)CCC(=O)C2(CCC2)C1.N12CC(C1)C2 C1(NC(CCN(C)CCO)=O)CN(C(C2(C)CC2(F)F)=O)CCC1(C)C CC(C)CC(C(=O)NC1CC1(C)C)ONC(C1CCCCCN1C)=O C1(C(=O)NCC#CCNC(=O)CSc2ccccc2O)CC12CC(O)C2 N1(C(c2c(COC)cco2)=O)CCN(C(c2cnc(OC)s2)=O)CC2(CC2)C1 c1(NC(C(C)(CO)NC(C2C(C)(C)C2)=O)=O)ccc(F)c(O)c1 C12(C(N3CCC(C(C)C(=O)NCCC4(O)CCCC4)CC3)=O)CCC(C1)C2(C)C C=C=CCCC(=O)NC1C2CN(C(c3ccc(CN(C)CC=C)o3)=O)CC12 c1(C(C)NC(N(CC(CC)C)Cc2ccccc2)=O)cc(F)ccc1F CC1(C)CCC(C(N2CCC(C)(NC(c3cc(C4CC4)ncn3)=O)C2)=O)OC1 c1(OC)ccc(C(C)C(=O)NCCNC(=O)C(F)=CCCF)c(OC)c1 C1(C)(NC(C(C)N2CCCC2)=O)CCCCC1C(=O)NOCCC1CC1 C1(OC)CC(CNC(=O)CCC)N(C(=O)C(=C2CCCCC2)F)C1.C(N)=O c1(C(=O)N)c2c(nn1C)CCCC2.c1(C(N(C(C)C)CC)=O)cc(O)nc(O)n1 C1(CC)CN(C(=O)CC2CCC(=O)N2)CCC1.C(=O)(C(C)(C)CC1CC1)N c1(OC)ccc(CC(=O)NCC2CC(OC)CN2C(C2CC(C)C2)=O)cc1Cl C1(NC(CSC)=O)CCN(C(=O)COC2CCCOC2)C1(C)C C1(OC)CN(C(=O)CONC(C2CCC(C)CC2)=O)CC1F c1(C(N2CCCC(F)(CNC(c3cc(CO)on3)=O)C2)=O)cccn2nnnc12 C12(CC3(CS(=O)Cc4ccccc4)CCCC3)CCC(CC1)CO2 N1(CCC#C)CCN(C(c2cc(C(=O)OC)cc(F)c2)=O)C(C)C1 N1(C(=O)CCC2COCCN2)CCN(c2ccncn2)CC1 Cc1[nH][nH]c(=NC(=O)c2nccc(F)c2Cl)c1C(=O)OC(C)(C)C N1(CC(N2CCCCC2)=O)C(=O)CC(C)(C)C1=O.C(CC(=O)NC)SCC c1(SC)ccc(CCC(=O)NCC23CC2CN(C(c2csc(CO)n2)=O)C3)cc1 Cc1cc(C(=O)NCC(CNC(c2coc(O)n2)=O)CO)ccc1C#N N1(C(N(CCOC)CC)=O)CCC1(C)C1CCCCC1 c1(N2CCC(C(N3CCC(C#C)CC3)=O)(C(C)C)C2)ncnc2scc(C)c12 c1(C(=O)NCCCNC(c2c(CC)nns2)=O)ccc2c(c1)C(C)(C)CO2 C1(C=O)C2(CC2)C12CC2.C(c1cccs1)=C(C)C(=O)NCCCOCC.N c1(CC(=O)NCCOCCCNC(C2CCSC2)=O)ccnc2ccccc12 N1(C(c2ccc(OCCC(=O)OC)cc2)=O)CC2CC2(C)C1.C(=O)C=O.N c1(C(=O)NCC(C)NC(=O)Cc2nnc(O)s2)cnn2c1CCCC2 C1(CC(=O)NC2CC(CNC(c3cnnc(Cl)c3)=O)C2)CC2CCC1C2 C(=O)(CC(C)(C)C)NC(C)C(CO)NC(C1CC1(C)C(F)(F)F)=O C1(C(N2C(CCNC(CN(C)C3CC3)=O)COCC2)=O)CCCCC12OCCO2 C(C(=O)NCc1cc(C=O)co1)(C(C)C)OCC.c1(C(C)C)ncccn1 C(=O)(C(CCc1cccc(F)c1)N(C)CC1(F)CCC1)NC(C(=O)OC)C C1(C(=O)NC(c2ccc(C(C)(C)C)cc2)CCC)CN(C)C(=O)N1 N1(c2c(C(C)=O)cnc(C)n2)CCC2(CCN(C(C3CCCO3)=O)CC2)C1 c1(OC)ccc(C(=O)NC(C2CCCN(C(=O)Cc3cnsc3)C2)C)nn1 N1(C(C(CN(C)C(C2CCCCCCC2)=O)(C)C)=O)CC2C=CC1CC2 c1(C(N2C(CCNC(=O)CC3CC=CC3)COCC2)=O)ncc(C2CC2)cc1F C1(C(=O)Nc2c(C(=O)OC)scn2)CC12CCN(C(c1ccc(C)nc1)=O)C2 CC(C)C(C)C(=O)NC(C)CN1CCN(C(C2(CC(F)F)CC2)=O)CC1 CN1CCN(C(C2CCCCN2C(=O)CCc2ccccn2)=O)C2(CCC2)C1 c1(C(=O)NC(C)(CNC(=O)C2=CCCC2)C2CC2)ccc(N)cc1Br O=C(C1=CS(=O)CCC1)NCCN1CCC(NC(C2CC3(CCCO3)C2)=O)CC1 N1(C(C2N(C(C)=O)CCC2)=O)CC(C)CCC1CNC(=O)CC1OCCCO1 Cc1cc(CCC(=O)N2CC(CNC(c3cc(CO)on3)=O)C2)cc(C)c1 C1(C(N(C)Cc2cn(C)nn2)=O)CC(NC(=O)CCCC2CCC2)C1(C)C C1(CN(Cc2nc(C)sc2)Cc2ccccc2)CCCS(=O)(=O)C1 CC1(C)CN(C(=O)COC2CCCC2)CC(CNC(=O)C2=CCCOCC2)O1 Cc1cc(N)n(-c2ccc(NCc3nccn3C(C)C)cc2)n1 C1(C(N(CCOC)CCNC(=O)C(=Cc2c[nH]cn2)F)=O)CC12CCCC2 C(=O)(C(C)CC(C)(F)F)N1CC(C)(NC(c2c(C)nc(-c3nc[nH]n3)s2)=O)C1 Cc1cc(C(=O)NC(C2CC(NC(C3CCC3C(N)=O)=O)C2)C)cnc1C Cn1nnc2cncc(C(N3CC(NC(C4(C)CCOC4)=O)C3)=O)c12 N1(C(c2cc(C(=O)OCC)sn2)=O)CCN(C(=O)CCS(C)=O)CC1 N1(C2CN(C(=O)Cc3cn[nH]c3)C2)CC(NC(=O)CCN2CCOCC2)CC1=O C(=O)(C(C)(C)CN(C)C(C1CC(F)(F)C1)=O)NCCc1cnc(C)o1 C1(C=O)CCn2cc(C)nc2C1.C1(NC(C2(CC#C)CCC2)=O)CC(F)C1.C N1(c2cc(NCCCN3C(=O)COCC3)ncn2)CCc2n[nH]cc2C1 c1(CN(C(C2(N3CCCC3)CC2)=O)C2CC2)ccc(OC(F)F)cn1 c1ccc([N+](=O)[O-])c(C)c1.C(CCCC(=O)NCC1COC(CO)C1)OCC c1(C(=O)NCC(C(C)C)NC(c2occ3c2CCCC3)=O)ccn2nccc2n1 Cc1cc(C(N2CC(NC(=O)COC3CCC3)CC2)=O)ccc1C(F)(F)F Cc1cc(C(=O)NC(CNC(=O)CCOC(C)C)CO)nc(C)n1 C(=O)(C1=CCOCC1)N1C(C(N(C2C(C)C2)C)=O)C=CC1 Cc1ccncc1CC(N1CCCC(C(C)NC(C2CC(=O)CO2)=O)C1)=O c1(-n2c(C(C)Nc3c(C)noc3C)nnn2)ccc(C(F)(F)F)cc1Cl N1(C(Cc2c(C)noc2C)=O)CCC(O)(C(N2CCCC(CCO)C2)=O)CC1 C(C1=CCCN(C)C1)NC(C(c1ccnn1C)NC(C(CC)C)=O)=O c1(N2CC(CC(C)NC(c3cccn4nnnc34)=O)C2)ncc2ncnc-2[nH]1 C=CCC(C)(CC=C)NC(C1CCCC1NC(C1CC(F)(CF)C1)=O)=O C12(C=O)CCCN(CC1)C2.N1(N(C2CC(C=O)C2)C)CCC(O)CC1 CCCC(C)(O)CNC(C1CCCC1CNC(=O)CN(C)C(=O)O)=O C1(NC(C(CCC)O)=O)C(C)(C)C(NC(=O)CC2COCCO2)C1(C)C C1(C(=O)NCC(C)(C(C)C)NC(c2c(C)nc(O)s2)=O)COCC(C)(C)O1 C1(C(=O)NCCCN(C(c2cncc(CO)c2)=O)CC)CCN2CCCC2C1 CC1CN(C(=O)C(CN)CCOCCO)CC(C)O1 C1(C(=O)NCC2(C)CCCN(Cc3nc(C(F)F)no3)C2)CCc2c[nH]nc2C1 C1(CC)(CC)CCN(c2cnccc2Oc2ccccc2)CC1 c1(OC)ccc(F)cc1CCC(=O)Nc1c(Br)cncc1Br C1(C(=O)NC2CCC(C)(NC(=O)CCCCC#N)CC2)CC2CCCN2C(=O)N1 c1(C(=O)NC23CCC(N)(CC2)C3)ccc([N+](=O)[O-])cc1I.c1cc(Br)ccn1.C C1(C(=O)N(C)CCn2cncn2)(NC(C2CC(C)C2)=O)CCN(C)C1 c1(C(=O)NCC2CN(C(c3cc(OC)nn3C)=O)C(C)C2)ccc(O)c(O)c1 N1(C(CCc2cc(C)on2)=O)CC2COCCC2(NC(C2CC2C)=O)C1 C12(NC(c3c(C)nc(C)o3)=O)CCCC1N(C(=O)CCc1cccc(F)c1)CC2 CC1(C)CCN(C(c2ncncc2Cl)=O)C1C(N1CC(C2CCCO2)C1)=O CC(CC(=O)NCC(F)C)P(C)(C)=O.n1(CC=O)cccc(C(F)(F)F)c1=O N1(C(c2c(C(C)C)ccs2)=O)CC(NC(=O)C(O)Cc2cnc[nH]2)CC(C)C1 c1(C(N2C(C)CN(C(=O)CC3COC(=O)C3)CC2)=O)cc2cc(F)ccc2o1 CC(C)CC(O)CC(=O)N1CC(O)(C2(CNC(=O)C=CC=C(Cl)Cl)CC2)C1 N1(C(C=CC)=O)CCC(C2CC2)(C)C1.c1(C=O)cccc(Br)c1C(N)=O.N c1(OC)cc(C(=O)N(CCCCNC(=O)C=C2CCOCC2)C)cc(F)c1 C1(C(=O)NC2(C)CN(C(=O)C=CC3CCOC3)C2)CC2(C)CC1CO2 c1(C(N2CCN(C(C)(C)C)CC2)=O)c(OC(F)F)cccc1Cl Cc1ccc(C(N2CCOCC2CNC(=O)CCC(F)(F)F)=O)cc1I C1(CNC(CC2CC(CC)OCC2)=O)CC(C)(C)CN1C(c1nc(Cl)cs1)=O N1(C(c2cc(C)c(C)[nH]2)=O)C2CCC1(CNC(=O)C=CC1CCCO1)CC2 C1(C(=O)NC(CC)CNC(=O)C=C2CCC2)CCC2(C1)CC2(F)F C1(C(=O)NCc2cc(C)sc2)(NC(C2CCC(F)CC2)=O)CC(F)(F)C1 C1(C)(C(N(C)CC2CCCS2)=O)CN(C(C2CC3(CC3)CO2)=O)C(C)(C)C1 Cc1coc(C)c1C(=O)NC1C=CCN(C(=O)CCCOC(C)C)C1 Cc1c(C(=O)NC2CN(C(=O)COCc3ccccc3)CC2O)ccc(F)c1F C1(NC(C(C(C)C)C)=O)CCC2(CC1)CCN(C(=O)CC(=O)NC1CC1)C2 N1(C(CN(CC(C)C)C(C2CCC(C)(C)CC2)=O)=O)CCC2(CC1)CC(O)C2 CC1CC(NC(=O)CP(C)(C)=O)CN(C(=O)COC2CCC2)C1 c1cc(CN(C2CC2)CC)c[nH]1.C1(C=O)CCCN1C=O.C(C)(C)C.N N1(C(Cc2cn(C)nc2)=O)CCC(O)CC1C(N1CCC(C(N)=O)C1)=O C12(C=O)CCN(C1)S(=O)(=O)C2.Cc1cc(CCC(=O)N)no1.C(C)C1CCC1 C(c1cccc(O)c1)=CC(=O)NC(CC)(CNC(c1cnc(O)o1)=O)CC C(=O)(CC(C)CC(C)(C)C)NC1CCCCN(CCC(C)F)C1 C1(NC(c2ncc(NC)nc2)=O)CN(C(=O)C=C(C)C(F)F)C(C)(C)C1 C1(NC(c2cnc(CC)[nH]2)=O)CC2CC(NC(=O)Cc3cnc(C)s3)C2C1 C1(C2CCCCC2)(C(N2CCC(C)C(NC(=O)CCSC3CCCC3)C2)=O)CC1 CC1CC(C(=O)N(C)Cc2ccoc2)N1C(=O)C=Cc1cscn1 CN1CC(N(C(=O)C(=O)NC2COCC2N(C)C)C)C(O)C1 c1(CC(=O)NC2C(CC)N(C(=O)C3=CCCC3C)CC2)ccc(C)c(C)c1 C1(CC(=O)NC2(C)CC(NC(C3CC(SC)C3)=O)C2)CCCC(=O)N1 S(=O)(=O)(c1ccccc1)NC(C)C(=O)N.C1(F)(C(NC)=O)CCC1.C1CC1 C=CCCCCCCCC(=O)NCC1CC(NC(C2CC3(C2)CC(C)(C)C3)=O)C1 C12(C(=O)NCC#CCNC(CCSC)=O)CC(C(F)F)(C1)C2 O=C(CCCCCNC(C1CC1C1CCCC1)=O)NCc1ncc[nH]c1=O c1(C=O)c(C)nn(C)c1Cl.Cc1cscc1C(=O)NCC1(F)CC(C)C1.N C(=O)(CC(C(F)(F)F)NC(=O)CCc1nccs1)NCC(COC)(C)C C1(NC(c2c(C(C)C)cco2)=O)CCC2CN(C(C3CCN(C)CC3)=O)CC2C1 c1(CC(=O)NC2C(NC(C(CCCOC)C)=O)CC2)ccc(F)c(Cl)c1F N1(C(c2csc(C3CC3)n2)=O)CCN(C(=O)CC2(O)CCC2)C2CC12 CN1C(=O)CCCC1C(N1CC(O)(C)C1)=O.c1(C(=O)N)coc(C(N)=O)c1 c1(CCC)c(C(=O)NC(C2CN(C(C3C=C(C)CS3)=O)CCO2)C)cnn1C C1(O)(CNC(C2C=CCCC2)=O)CCN(C(c2cc(Cl)cs2)=O)CC1 N1(C(c2ccco2)=O)CC2CCC(C1)N(C(=O)COCc1cccc(Cl)c1)C2 N1(C(c2ccc(CC)o2)=O)CCCC(C(=O)Nc2cc(O)cc(F)c2)CC1 c1(C2(C)C(C(=O)NC(C)Cn3cc(-c4cncnc4)nn3)C2)ccccc1F C1(CNC(c2occ(C)c2C)=O)CC12CCN(C(=O)CN(C1CCCC1)C)CC2 CC1CC(C(N2CCC(NC(C3(CN(C)C)CCCC3)=O)CC2)=O)CCS1 N1(C(c2c(CC)scc2)=O)CC2CCC2(NC(=O)CC2CC(C)=NO2)C1 C1(NC(CC(COC)(C)O)=O)CN(Cc2ccccc2)C2(CCC2)C1 C#Cc1ccc(F)c(C(=O)N(C)C)c1.C1(C(N2CCCC2)=O)CC2(C1)CC(F)C2 N1(C(c2ccc(CC3CC3)s2)C(=O)NCCC#N)CCc2c(Br)cccc21 C1(C(=O)NC(CNC(C2CN(OC)C(=O)C2)=O)(C)C)Cc2ccncc2N1 c1(OC)cc(O)ccc1NC(=O)CN1CCN(C(=O)CCC)CC1.C(C)(=O)O CCCCC(CC)CC(=O)N1CCC(C(N2CC(c3nncn3C)C2)=O)C(O)C1 C1(O)(CC)CCN(C(c2cnc(C(N)=O)s2)=O)C1.N(S(N)(=O)=O)CC=O C12(CC)CCC(C1)N(C(c1cncc(O)c1Cl)=O)C2.C1(C=O)CC1C=O.CO C1(C(N(CC)C(C)C)=O)CCCC1C1CC1.n1(CC(C)C)ccc(C(=O)N)n1 N1(C(C(CC)c2ccccc2)=O)CCN(c2cnccc2C)CC1 N1(C(C(CNC(C)=O)(C)C)=O)CC(NC(c2cnn(C)c2Cl)=O)CCC(O)C1 Cc1cccn2nc(C(=O)NC3CN(C(=O)C=CC(C)(C)C)CC3C3CC3)cc12 C1(C)(C(N(CC)C)=O)CC=CCC1.c1cc(C(=O)N(CCC)C)on1.COC c1(CCC)ncc(NC(=O)CCC(C)NC(=O)C(C)c2cc[nH]n2)cn1 N1(C(C2CC(O)CCN2C(c2cccs2)=O)=O)CCC2(CC1)CC(F)(F)C2 CC1(C)CC(O)CN1C(C1CC=CCC1)=O.c12ncccc1NC2=O C(=O)(C(C)(C)C(C)O)NCC(CNC(Cc1c(OC)cccc1)=O)CO C(=O)(C(C(C)(C)C)NC(=O)Cc1ccnc(O)c1)NCCCCCCC C1(COC)CCCN1C(=O)C.C(=O)(C=COCC)NCCC.C1CCOC1.O N1(C(C2C3(CCN(Cc4ccc(C)cc4Cl)CC3)C2)=O)CCC2(CC1)CC2(F)F C(=O)(C1=CC2(CCOC2)C1)N1C(C)CN(C(=O)C(C)OCCN(C)C)CC1 C1(C(=O)NCCC2(C)CC2(F)F)CCC12CCC2.n1(CC(=O)N)[nH]cnc1=N C(=O)(C(O)C(C)c1ccccc1)N1C(CNC(C(n2cc(C)nc2)(C)C)=O)CC1 c1(C(=O)NCC2(O)CC(CNC(C(C)CF)=O)C2)ccc(C(F)F)nc1 c1(C(=O)NC(CC)CN(C(=O)C(C)(O)CC)CC)nnn2c1COCC2 C1(CC)CC(CC(=O)NCCC2CC2)CCO1.C(=O)C(F)CC1CCCCC1.N CN1CC2(CC2)CC1C(=O)NCC1(O)CCCN(C(=O)CCCCCN(C)C)C1 N1(C(c2c(C)nn(C)c2)=O)CCC(NC(=O)C=Cc2cccnc2)C(O)C1 C1(C(=O)NCC(COC)(C)C)CCC(C)(C)N(C(c2cscc2C)=O)C1 c1(C(=O)NC(CC(CC)C)C)ccc(Cl)c(F)c1 c1c(N)cccc1[N+](=O)[O-].C1(C(=O)NCC(N2CCC2C(=O)N)=O)CCCCC1 Cn1cnc(C(=O)NCC2C3CCC(C3)N2C(=O)CCN2CCCCC2)cc1=O C=CCC(C(=C)C)C(=O)N1CC2(CCC(NC(c3ccc(Br)c(C)c3F)=O)C2)C1 C1(NC(C(C2CCCCC2)OCC)=O)CCCC1NC(=O)C(O)CSC CCC(C(=O)NCC(C1CC1)N(C(=O)CCc1scnc1C)C)C1CCOCC1 C12(CNC(=O)C=CC(F)(F)F)CCCC1CCN2C(c1cn2ccnc2cn1)=O N1(C(C2(NC(C)=O)CCC2)=O)CC2CCN(C(=O)CCc3cccs3)CC2C1 Cc1nc(Cl)c(C)c(=NCC2CC(F)(F)C2(C)C)[nH]1 c1(C(N2CC=C(C(=O)NCCN(C(CC)C)C)C2)=O)cccc2cncn12 N(C)(S(=O)(=O)N(C)C)CC(=O)N(C1CCCN(C(=O)CC(C)CF)C1)CC C1(C(N2CCC(O)(CNC(C(C=C)CC)=O)CC2)=O)CN2CCCC2CO1 C(C(C)(O)C(=O)NC1CCCC(CC(=O)NCc2ncccc2C)C1)OC C1(CC)CCCC1C(=O)N(CCNC(c1c[nH]nc1CO)=O)C.C1CC1 C=CC1(C(=O)NCC(F)(F)C(C)C)CCN(C(C2CCCCC(=O)C2)=O)C1 c1(C(N2C(CCC)CN(C(=O)C(C)CCOC)CC2)=O)cc(C)c(C)cc1Cl N1(C(CCC=C)=O)CCCC(CCNC(C2(CCC)CCNC2=O)=O)CC1 N1(C(C=C(CC)C)=O)CCCC1C(C)(C)CNC(=O)CCC1CCCN1C N1(C(C2C(C(C)(C)C)C2)=O)CCCCC1CC(=O)C=CCN1CC=CC1 c1(CNC(C2(n3cc(C(CC)(O)CC)nn3)CC2)=O)cccc(N(C)C)c1 C1(NC(C(C)(C)OC)=O)CCCN(CC(=O)NCC(c2ccccc2)C)CC1 c1ccccc1[N+](=O)[O-].n1(C(C)C)cnc(C(N2CC(C)(NC(=O)C)C2)=O)c1.O c1(CCC)cc(C(N2CCCC(NC(C3(C#N)CC34CCC4)=O)C2)=O)cc(O)n1 CN1N=C(C(=O)NC2CC(C(F)F)C2)CCC1=O.C1(O)(C(C=O)F)CCCC1.N C1(O)(CNC(CCc2n(CC)ccn2)=O)CCN(C(=O)CS(=O)(=O)CC)CC1 N1(C(COC2CCN(C(C3(C)CC4C=CC3C4)=O)C2)=O)C2CCC1CC1(C2)N=N1 N1(C(CC(CCC)C)=O)CCC2(CC1)CC2NC(c1sc(Br)nc1C)=O N1(C(c2ccc(CC(=O)Nc3n(CCC)ccc3)nc2)=O)CC(C)CC(C)C1 N1(C(C(C(C)C)C)=O)CCCOC(CNC(c2cnc(Cl)n2C)=O)C1 c1(C(=O)N)cnc2c(c1)c(C)nn2C.C(C)(CCC)NC(C(C)NC(C)=O)=O c1(C(C2CC(F)(F)C2)C)nnnn1CCC1(C)CC1.C1(CSC)CC1.C C(N=c1cc(C(C)(C)C)nc(Cl)[nH]1)C1C(C)CN(C(=O)CCCCCN(C)C)CC1 c1(C(=O)NCc2ccccc2O)nc2ccc(-c3ccn4ccnc4c3)cc2o1 C1(C)(CNC(c2ccc(CC)[nH]2)=O)CCN(C(C2CC2C)=O)C1 c1(NC(C)CNC(=O)CC2CC(C)CC(C)(C)C2)ncnc2[nH]cnc12 N1(C(C(CC)(C)NC(=O)OC(C)(C)C)=O)CCC2(CC(O)C(O)CO2)C1 C1(C(=O)NC23CC(C2)C3)CC1C1CCCC1.C1(C=O)CC(n2cnnc2)C1.N C(C(C)CN=c1nc(N(C)Cc2cnccn2)c2[nH]ccc2[nH]1)OCC C(CCCCC(=O)NCC1NC(=O)NC1=O)NC(c1c(C#N)ccs1)=O C(=O)(CCC(C)NC(=O)CCOC(C)C)NC(C#C)(C)C1CC1 C12CCCC(CC1)NC2=O.C1(CC)(CO)CN(C(=O)CC2OCCO2)C1 N1(C(c2cc(C3CCC3)on2)=O)CCC(NC(C2CC(F)C2)=O)C(O)C1 c1(OC)cccc(C=CC(=O)NC2CC2)c1.C(C1CCCN1C)=CC=O.C C(=O)(CC(CC)C(C)C)NCC(CC)NC(c1c(-c2ccncc2)noc1C)=O N1(C(Cc2c(C)occ2)=O)CCC(C(=O)NCC2(C)CCCO2)=C(F)C1 Cc1nc2c(s1)CCCC2CNC1(c2nnnn2C2CC2)COC2(CCCC2)C1 N1(C(CCC(=O)NCCC)=O)CC2CCC(C2)C1.c1(C(=O)N)cc(C)cc(O)c1 N1(C(c2ccc(C)c(Cl)c2)=O)CCC(NC(c2cnoc2)=O)C(C)(C)C1 c1(C(=O)NCC2N(C(c3cc(C)ns3)=O)CCCC2)cc(Cl)ccc1OC(F)F Cc1nc2ccnn2cc1C(=O)NC(C)(CNc1ncc(Br)c(O)n1)C1CC1 C1(CCc2cn(C(C)C(=O)N3CCC3)nn2)CCCN1C(=O)CN1CCOCC1 C(=O)(CS(=O)CCC(F)(F)F)NCC(CC=C)NC(c1cccc2occc12)=O C12(C(=O)NCCCCCN(C(C(CSC)OC)=O)C)CC(C)(CCO1)C2 C1(C(=O)NCC2CCN(CCC)C2)OC(=O)C2(CCC2)C12CCC2 c1(C(C(=O)NCC2CC2)N(C)CCOCCO)cc(Cl)cc(Cl)c1Br N1(C(c2n(CC)c(O)nc2)=O)CCC2(COC(C)C2)C1.C1(C(=O)N)CCC(C)O1 C1(NC(c2cc(C)c(C)[nH]2)=O)CN(C(=O)CNC(=O)C2CC2)CC2(CC2)C1 CCC(C)(C(=O)NC(C)CC)NC(=O)OC(C)(C)C.c1(C=O)ccsn1 C1(C(=O)NC2(CNC(c3cscc3Cl)=O)CCOCC2)CC2(CCCO2)C1 C1(C(=O)NCC2CC(F)(F)CN2C(C2COCCO2)=O)CCCCC12CCC2 C(C(COC)C(=O)N1CCCC(C)C1)OC.n1(CC=O)cncn1.C(=O)C.N c1(OC)ccc(F)c2[nH]c(C(N3CC(NC(c4c(N)cccc4F)=O)C3)=O)cc12 C(=O)(C1=C(Cl)CCCC1)N1CC(C(=O)NCC(C2CCC2)OC)N(C)CC1 C1(C)(CC(=O)N(CC(CNC(CC=C)=O)O)C)CCCC1 c1(C(N2CC(C(=O)Nc3cc(C)nn3C)C(O)CC2)=O)c(O)ccc(Br)c1O C1(C2CCN(C(c3cnc4[nH]cnc4c3)=O)C2)(NC(C(C(C)C)SC)=O)CC1 C1(NC(=O)Cc2cn[nH]c2)CCCC(C(N2CC(O)(c3cnn[nH]3)C2)=O)CC1 C1(CNC(C(C)CCO)=O)Cc2ccccc2CN1C(=O)CN(S(C)(=O)=O)C C(=O)(CCC(C)(C)C)N1CC2C(CC(=O)NCC(CCC)OC)C2C1 C12CC(C1)C(C)O2.n1(CC)cc(C(=O)NC)nn1.C(=O)CCO.C(N)=O C1CCC2(CN(C(C3(F)CC4(CCC4)C3)=O)C2)O1.Cn1c(Cl)cnc1C(=O)N c1(C(N(CCCNC(Cc2cc(C)nn2C)=O)C2CC2)=O)ccc2c[nH]nc2n1 CC(C)CCCC(=O)NCCN(C)C(C1(CC(F)(F)F)CC1)=O Cc1c(C(=O)NCC(C)NC(=O)C)sc2ncnc(N)c12.c1(CC)cccs1.O C1(CCC)CN(C(c2cc(COC)[nH]n2)=O)CCN1C(=O)CC1CC(F)C1 C1(CC(N2CCCC(NC(C3(N(C)C)CCC3)=O)C2)=O)OCCCC1(C)C C1(S(C)(=O)=O)(C(N2CCCC2)=O)CCC1.C1(CC(=O)NC)(CC)CCC1 c1(C(=O)NC2C(NC(C(COC)C)=O)CCCC2)c(C)n(C)c2ccccc12.O C12(C(=O)NC(C(=O)NC)CC3CC3)CC3CC1C2C3.C1(C=O)CCNC1 c1(CNC(C=CCN(C)C)=O)nc(C)cs1.C1(C)(C(=O)N)CC1(C)C C1(C(N2C(C(=O)NCCSC(C)(C)C)CC(O)C2)=O)OCCCC1(C)C Cc1ccc2cc(C(N3CCC(CC(N4CC5C(C(N)=O)C5C4)=O)CC3)=O)sc2c1 c1(C(C)=O)ncc(C(=O)NCCCCCc2cn(CC3CCC(=O)O3)nn2)s1 c1(NC(CC2(NC(C(CC)CC)=O)CCC2)=O)ccc(C#N)c(F)c1 C1(N(C)CC)CCN(C(C2C=CC(NC(C3(C)CCCC3)=O)C2)=O)C1 CS(=O)(=NC(=O)C(O)c1ccncc1Br)c1ccccc1Br Cc1ncc(S(=O)(=O)NCC(N2CCN(C3CC3)C(C)C2)=O)s1 c1(C(=O)NCC=CCC(=O)NC(c2ncc[nH]2)CC)ccc2occc2c1 Cc1[nH]c(=NCc2ncc(Br)cn2)sc1Cl C1(NC(=NCC=C)NCCOCCSC)CCc2nc(CC)nn2C1 N1(C(c2ccn(CC)n2)=O)CCN2C(=O)C(NC(C3C4CCC3CC4)=O)CC2C1 C(=O)(C1COc2ccc(Cl)cc21)N1CC(NC(c2cc(SC)oc2)=O)CC1(C)C S(=O)(=O)(c1ccc(=NCC2CC3CCC3C2)[nH]c1)N(CCCCC=C)C Cc1cccc(NC(C2C3CC2N(C(=O)Cc2c(C)n[nH]c2C)C3)=O)c1[N+](=O)[O-] c1(C(=O)Nc2ccc(OC(F)(F)F)nc2)n[nH]cc1C1=CCCCC1 N1(C(C(CC(C)(C)C)O)=O)CCC2(CC1)OCCC2NC(c1coc(Br)n1)=O C(=O)(C(C)(C)C(C)(C)C)NC(CNC(c1ccnc(C)c1C)=O)C(C)C(C)C C1(CS(=O)(=O)NCc2nc(C(C)(C)C)on2)CCC(F)(F)CC1 C(C(C)(C)CC(=O)NOCC(C)O)NC(c1n[nH]c(C)c1C)=O C(=O)(C(C)C(O)CC(C)C)NC1C(C(=O)Nc2ccc(OC)nc2)COCC1 Cn1cc(C(=O)NCCC2(CNC(c3ncccn3)=O)CC2)n(C)c1=O CC(C)CC(CNC(=O)CCC(CF)CF)C(=O)N1CCCC1C(C)O C1(NC(c2c(C)nc(CC)s2)=O)CN(C(C2CC2(F)F)=O)CCC12CCC2 c1(OC)ccnc(C(=O)NCC(CO)NC(=O)Cc2c(C)nn(C)c2C)c1.O N1(C(c2c(-c3cn(C)nc3)ocn2)=O)Cc2c(F)ccc(F)c2C1 c1(C(N(CCCNC(Cn2nc(C)oc2=O)=O)C)=O)cc2cc(C)c(Cl)cc2[nH]1 c1(CN2CC3(CCC(C(=O)NCCCCN(C)C)O3)C2)ccc2ccccc2c1Br c1(C(C(=O)NC2CCCC2)N(C2CCS(=O)(=O)C2)CC=C)cc(Cl)ncc1Br Cc1cnc2n1CC(C(=O)NC1CCC1NC(=O)CCc1ccccc1Cl)CC2 c1(C(=O)NC(C2CCN(C(CSCC)=O)CC2)C)c(OC)cccc1Cl c1(C=O)cnn(C2CCC2)c1.O=C(CCOC1CC1)NCCOCCC.N C1(NC(CCC=CC)=O)CC2CCC(C1F)N2C(=O)CCN1CCCC1 c1(C(C(=O)OC)NCC2(OCC)CCCCC2)ccc(C#N)cc1Cl c1(OC)ccc(C(=O)Nc2[nH]nc(OC)c2C#N)cc1F.C12CN(CCS1)C2=O S(=O)(=O)(c1ccc(C#N)c(NCC(C2CCCCC2)F)c1)N(C1CC(=C)C1)C CC1CCC(C)(C(=O)NC2CCCC2)C1(C)C.c1(C(=O)N)cnc(C2CCC2)o1 CC(C)CC(C)C(=O)NC(C1CN(C(=O)C=Cc2cc[nH]c2)C1)C c1(OC)cccc2cc(C(N3CCC3CNC(C3CCCC(=O)O3)=O)=O)[nH]c12 Cc1cc(C(N2CCC(CO)(CNC(=O)CC34CCCC3C4)C2)=O)ccc1F c1(C(=O)NC2CCCCN(C(C3C(C)CCO3)=O)C2)c(N)cc(Cl)nc1Cl C1([Si](C)(C)C)(CNC(CC(C)NC(C2CCCOC2)=O)=O)CC1 C1(NC(C2(C)CC(C)OC(C)C2)=O)CC2CCC(C1C)N2C(c1ccncc1)=O c1(CCC(=O)N(C2CCN(C(C(C)NC(CC)(C)C)=O)C2)C)ccc(O)nc1 c1(-c2c(C(=O)NC(C)C(N)=O)cc(OCC)nc2)cc2ccc(OC)cc2[nH]1 C(=O)(C(C)CC(=O)OC)N1C(CN(C(C(CC)F)=O)C2CC2)CCC1 c1(CCC(=O)NC(C)CCNC(=O)CCC(C)O)cccc([N+](=O)[O-])c1 c1(C(N2CCN(C(=O)CC3CCCCC3)CC2C(F)F)=O)cncc([N+](=O)[O-])c1 C1(C(=O)NC2C(CNC(c3scnc3Cl)=O)CCCC2)CC2(C1)CC(O)C2 C(=O)(CCCCCF)N1C(CNC(=O)Cc2ccc(Cl)cc2)CCCC1 c1(C(=O)NC(CC)CNC(=O)C(F)CC)c(OC)cccc1F C(=O)(C(CNC(c1nonc1CC)=O)CC=C)NC(C#C)C1CC1 c1(CC)cc(CC(N2CC(C)C2C(=O)NC(CO)CCOC)=O)on1 N1(C(c2c(C)ccc(C)c2)=O)CC(C)CN(C(c2cnc(C)cn2)=O)C(C)C1 c1(C(C)OCC)ncc(C(=O)NCCC)s1.C(=O)(C(C)(C)C1CCCO1)N c1(N2CCC(C)(C(=O)Nc3ncc(C)c(F)c3)C2)ncnc2ccc(I)cc12 CC1CCN(CCC(N2CC=CC(NC(c3ccns3)=O)C2)=O)CC1 O=C1Cc2cc(C(N3CC(C(=O)Nc4cccc(Cl)c4Br)C3)=O)c(Cl)cc2N1 c1(C(N2CCC(N(C(C3CC(OCC)C3)=O)C)C2)=O)ccc(CC)cc1C C1(C)(CCC)CCC(N(C(=O)CC(F)(F)F)CC(C)C)C1.CCC=O.CC=O.N C1(CCC)CN(C(=O)CN2CCN(CC)CC2)CCN1C(c1cc(C)n(C)c1)=O N1(C(=O)C=CC2CCCC2)CCCC12CCN(C(C1(C3CC3)CCCO1)=O)CC2 c1(CN(CC(O)CO)C)c(NC(c2ccc(C)cc2)=O)cccc1F c1(CCC(=O)NC2CC(NC(C(CCC)OC)=O)C2)cccc(S(N)(=O)=O)c1 Cc1cc(C(=O)NC(CNC(C2CCC(C(N)=O)N2C)=O)CC(C)C)ncc1F CC1COCC(CC(=O)NCC2(NC(c3ccc(C(F)F)o3)=O)CCCC2)O1 C(c1ccc2c(c1)CCO2)=CC=O.n1(CC)nncc1C(=O)N.C(C)(C)CO C1(C(=O)NCC2CCN(C(=O)C)C2)(OC)CCCC(C)(C)CC1.CC(N)=O CCC(CC)(CO)C(=O)NC1CC1C.c1(C(=O)N)nccc(-n2ccc(C)n2)n1 CC1N(C(C2CC(NC(=O)C(O)CN(C)C)CCO2)=O)CCCC1(C)C c1(N2CC(C(=C)C)OCC2)nc(=N)[nH]c(=NC(CC2CCC2)c2ccccc2)[nH]1 N1(CC2N(Cc3c(C)nns3)CCC2)CCc2sccc2C1 c1(CN=c2[nH]c(COC)c(C)s2)sc2ccccc2c1Br.S1(=O)(=O)CCN1 C(CCC)N(C(C=CC=CCC)=O)CC.CCC(C)C.C(=O)C.C=O.N C1(C(N(C(C)C)C)=O)CC12CCC(C)(C)CC2.c1(C=O)cc(N)c(Cl)c(O)c1.N N1(C(c2c(C(C)C)noc2)=O)CC=CC(C(=O)NC2CCCC2O)C1 C12(C(=O)NCC(C(C)C)NC(=O)CC(C)C(C)C)CC(C)(C1)OC2(C)C CC1CN(C(C2CCC(=O)C2)=O)CC(C)N(C(c2nn[nH]c2C(F)(F)F)=O)C1 Cc1cc(C(=O)NC2CN(C(c3cnoc3C3CC3)=O)CC2C)c(C)n1C c1(N(C)C)cccc(C(N2CCCC2C2(O)CN(C(C3CCOC3)=O)C2)=O)n1 c1(C(N2C(C(C)NC(=O)CN3CCCCC3)CCC2)=O)cc2cccc(F)c2s1 C1(CC(N2CCC(NC(C34OC(C)C(C3)C4)=O)CC2)=O)CCC(C)(C)CC1 c1(Oc2ccc(NC(=O)NCc3ccnc(Cl)c3)cc2)ccc(F)cc1Br CC(CCN=c1[nH]c(N(CC2=CCCOC2)C)nc2ccccc12)S(C)=O Cc1nsc(N)c1C(=O)NC(C1CN(C(c2scnc2Cl)=O)CCO1)C Cc1cc(-n2c(SCCN3CCCC(C)C3)nnc2-c2cnn(C)c2)ccc1Cl C1(NC(C2(CC(C)C)CCC2)=O)CCCC1CNC(c1ccco1)=O c1(C(=O)NCCCCCCN(C(C(C(C)SC)O)=O)C)ccc(C2CC2)c(F)c1 N1(C(Cn2c(C)ncc2)=O)CC2CC(NC(C3CCS3(=O)=O)=O)C1C2 c1(CC(=O)NCCNC(C(C)SC(C)C)=O)c[nH]c2c(Br)cccc12 CC(O)C(C)C(=O)NC12CC(NC(=O)CC3CCC(=O)N3)(C1)C2 Cc1cnn2cc(C(N3CCC(CO)(NC(=O)CO)CC3)=O)cnc12.C1CC1.C C(=O)(C(CNC(C1CCSCC1)=O)C(C)(C)C)N1CC(C)C(C)(CO)C1 C(=O)(C#CC(C)(C)CNC(C1CN2CCC1C2)=O)NC(C)C(O)C(F)F c1(C(=O)OC)cc(C)[nH]c(=NCC2C(C)CCCN2C(c2sc(F)cc2C)=O)n1 CC(C)C(O)CC(=O)NCC1(O)CC(C(N2CCC3CCCC23)=O)C1 Cc1nc2sccn2c1C(=O)NCC(C)(C)CNC(=O)CCC1CC1(F)F C=CCC(C)(O)C(=O)N1CCCC(C(C)NC(=O)Cc2ccc(O)cn2)C1 c1(C(=O)NCC(C)OC)cc2n(n1)CCC2.C1(C=O)CC(C2CC2)=NO1.N C1(O)CCN(C(C23COC(CS(C)(=O)=O)(C2)C3)=O)CC1.CC(C)(O)CC=O.N c1(NC(CCC)(CC)c2nnnn2CC2CCCO2)ccc2nn(C)cc2c1 C1(CCNC(c2cc(O)nc3c2CCC3)=O)CSc2ccccc2O1 C1COCC(C)O1.c1(CNC(C2CC(OCC)C2)=O)ccoc1C(=O)N C=CCC(F)(F)C(=O)NCC1CCN(C(=O)CC2CC(C)=NO2)CC1 CC(C)C(C(=O)N1CCCC(CCCO)C1)NC(c1ncccc1Br)=O N1(C(C2(C(=O)NC)CC2)=O)CCCCC(C(=O)N(C2CCSC2)C)C1 C1(C#N)(C(=O)NCc2ccc(C(=O)NCCNC(C)=O)o2)CCCOC1 N1(C(c2cccc(SC)c2)=O)CCN(C(=O)Cn2ccc(C(F)F)n2)CCC1C C#CC1(N2CCN(C(c3noc(-c4ccccc4)n3)C)CC2)CCOCC1 N1(C(COC2CC(NC(C(CC)C#N)=O)C2)=O)CCNC(=O)CC1 C1(C(=O)O)CN(C(C2CCC(C3CC3)CC2)=O)CC12CS(=O)(=O)C2 c1(C=O)cccc(S(C)(=O)=O)c1.N1(C(C(C)NC(CC)=O)=O)CCOCC1C CC(CNC(C1CC(C)(F)C1)=O)CC(=O)N1CC(O)C(O)C1 C1(NC(C2CC=CC2)=O)CCN(C(=O)C=CC=C(Cl)Cl)C12CCC2 c1(CC)c(N(C2CCN(C(c3cc(C4CC4)on3)=O)C2)C)ncnc1Cl c1(C(N2C(C3(O)CN(C(c4nc(C)sc4)=O)C3)CCC2)=O)ccc(C)c(C)c1Cl CC1SCCCC1C(=O)NC(Cc1ccoc1)C(=O)NCC(c1nccs1)C C1(OC)CCC(C)N(C(C2CCC3(CC3)N2C(C2CCCN2C(C)C)=O)=O)C1 N1(C2(C=O)CC2)CCOCC1.C1(C=O)(CNC(C2CC2(Cl)Cl)=O)CCC1 Cc1cn(C)cc1C(=O)NC(C)C1CC1.c1(C=O)cc(-c2cccn2C)[nH]n1.N N1(C(CCC(CC)OC)=O)CCC2(CC1)CN(C(C1(C3CC3)CC1)=O)CCO2 C#CCC(O)C(=O)NC1(CCC(=O)NC23CC(C2)C3)CCC1 C1(N(C(CNC(=O)OCC)=O)C)CCN(C(C2CC3(CC3)CO2)=O)CC1 CS(=O)(=O)c1cncc(C(N2CCCC2CC)=O)c1.C1(C2CC2)(C(=O)N)CC1 c1(CC)c(C(=O)N(CCC(=O)NCCCN2CCOCC2)C(C)C)cnn1C N1(C(CCC2N(C)CCC2)=O)CCC(C2CC2)C1CNC(=O)Cc1cscn1 c1(-c2ccc(C#N)s2)cnc2ccc(C(N3CC4CC4C3C#N)=O)cn12 N1(C(CC2CC(C)C2)=O)C2CCC(C2)C1CNC(c1ccc[nH]1)=O C#CCC(O)C(=O)N1CCC(O)C1C(=O)NC1CCCNC1=O n1(CCCC)nccc1C(=O)NC1(CO)CN(C(=O)CC23CCCC2C3)C1 c1(CCC(=O)NC(CN(C(C(C=CC)O)=O)CC)C)cccc(F)c1Cl N1(CCCCCNC(C=C(CC)C)=O)CCN(C(c2cocc2C(N)=O)=O)CC1 C1(C(N2C(C(=O)NCc3c(CC)n[nH]c3)CCC2)=O)CC(=O)CCO1 C=CC1(CNC(=O)Nc2ccncn2)CCC1 C1(C)(C=O)CCC(F)(F)CC1.N1(C(C(COC(C)C)(C)C)=O)CC2CC1CC2.N C1(NC(=O)C(c2ccccc2)O)CCCCC1C(=O)Nc1cncc(F)c1 C(=O)(C(O)CCC(F)(F)F)N(CC(O)CNC(C1CCCC(=O)N1C)=O)C Cc1cc(S(N)(=O)=O)c(-c2ccc(O)c(C#N)c2)c([N+](=O)[O-])c1C CCCC(C(=O)N(C)C)NC(C1(CC)CCCN1C(=O)C(C(C)C)C1CCC1)=O CC1C2CC(C2)N1C(c1cc(Cl)n(C)n1)=O.c1(C=O)conc1C1CCCO1.N C=CCC(C(=O)NC12CC1CN(C(c1cnn(CCF)c1)=O)C2)NC(C)=O c1(C(=O)NC2CC(O)(CNC(CC(CC)OC)=O)C2)nn(C)c(C)c1Cl C1(OC(C)=O)CCN(CC(=O)NC(C2CC2)C2CC2)C(CO)C1 c1(CCN(CCC(=O)O)C(c2ncc[nH]2)CC)cccc(Cl)c1 C(CCCCCCCOC(c1sccc1S(=O)(=O)NC(C)(C)C)=O)OC CN1CCOC(C(=O)NCCC2CCN(C(=O)CCC3CCCCO3)CC2)C1=O N1(C(c2cc(C)cc(O)c2)=O)CC2CC(C)CC1C2.C12(C(=O)N)CC(F)(C1)C2 C(=O)(C(C)(C)CN(C(=O)CC1(C)CC1)C)NC1CC(=C)C1 C12(NC(c3n(CC)ncc3)=O)CC1CN(C(=O)CCc1cncc(C)c1)C2 C1CC2CC1CN(C(c1ccnn1CCF)=O)C2.C1(C(=O)N)(CC)CC(C)(C)C1 N1(C(CCC=CC)=O)CC2(CCOCC2)CC1CNC(=O)C=CC(C)C c1(NC(C2(C)CCN2Cc2ccc3occc3c2)=O)cccc2ccccc12 C1(NC(CC=CC=C)=O)CC2CN(C(c3cnc(NC(C)=O)o3)=O)CC2C1 C(=O)(C(CC)C(=O)NC(C)C1CC1)OCC.c1(C=O)cc(C(F)F)cs1 c1(C(N(C2CN(C(c3ccc(Br)c(F)c3F)=O)C2)C)=O)ccc(N)c([N+](=O)[O-])c1 N1(C(CC=C(C)C)=O)CC2(C1)SCCC2NC(c1nsc2ccccc12)=O C1C2CCC(C2)C1C(=O)NC.c1cc(C)on1.C(C=O)NC(=O)OCC CC(C)CCC(CO)NC(C1(F)CN(C(=O)CCC2CC2(F)F)C1)=O N1(C(CC2C3CN(C(C(C=C)(C)O)=O)CC32)=O)CCS(=O)C(C)C1 C1(C2CCC2)(CC)CCN(C(C2CC(Cc3ccsc3)C2)=O)C(=O)O1 Cc1cccc2oc(C(=O)NC3(CF)CCN(C(C4CCCC4(F)F)=O)C3)cc12 C12(NC(c3c(CC)con3)=O)CCC(CC1)N(C(C1CC=C(C)CC1)=O)C2 C1(CNC(N(C)Cc2c(OC)ccc(OC)c2)=O)CCC2(CCOC2)O1 C1(NC(C(C2(C)CC2)NC(CC2CC(OC)C2)=O)=O)CC=CCC1 c1(N2CC=CC(NC(C3C(OC)CCC3)=O)C2)ncc2cccnc2n1 CCCCCC(O)C(=O)N1CC2CC(N(C(=O)C(CC(C)C)NC(C)=O)C)C1C2 c1(C(=O)NC(CNC(c2cccc(CC)c2)=O)C2CC2)cnn2ncccc12 N1(C(C(C)NC(N)=O)=O)C2CCC(C2)C1C(=O)Nc1cncc(CO)c1 c1(NC(C(CCCOC)NC(CC2CC(=C)C2)=O)=O)cnc2cc[nH]c2c1 c1(C(=O)N)ccc(S(=O)(=O)CF)nc1.C1(CNC(CC)=O)(C)CC12CCC2 Cn1cc(S(=O)(=O)NCC(O)COc2ccccc2)cn1 N1(C(c2cnc3c(c2)COC3)=O)C2CCC1CN(C(C1(n3nccn3)CC1)=O)C2 c1(C(=O)NCC(CNC(C2(O)CCOC2)=O)OC)cnc(O)cc1O C1(CN(C(C2(CN(C)C)CC2)=O)C)CCCN1C(C1CCC1CF)=O c1(CC(N2CC(NC(c3ccnnc3)=O)C2)=O)cnn(-c2ccccc2)n1 c1(C(N(CCNC(C2CS(=O)(=O)C2)=O)CC)=O)nnn2c1CSCC2 c1(C(=O)NCC2CCN(C(C3OCCN(C)C3=O)=O)C2)ccnn1C1CCCC1 N1(C(CC(COC)NC(=O)CNC(C)=O)=O)Cc2cccc(F)c2C1 N1(C(C=Cc2ncc(C)[nH]2)=O)CCCN(C(C2CCn3cnnc3C2)=O)C(C)C1 C1(CCNC)CCN(C(=O)CC2(C(=O)OC)CC2)C1C N1(C(CC2N(CC)CCC2)=O)CCC(NC(c2nc(=O)n(C)[nH]2)=O)C12CC2 C1(c2nnnn2CC2CC2)(NC2C(Cn3cncn3)C2)CCC2CCCC2C1 C(C)(CC(F)(F)F)NC(C(=O)NC(C)CCc1ccc(I)cc1)=O N#Cc1cc(S(N)(=O)=O)ccc1NC(=O)NCC1CC1.c1cccc(Br)c1 N1(C(C(CNC(Cc2c(C)occ2)=O)CC2CC2)=O)CC2(COC(C)(C)C2)C1 c1(OC)cccc(O)c1C(N1CCOC(C(C)NC(c2n[nH]c(O)n2)=O)C1)=O c1(CNC2CCN(C(CC(C)OC)=O)C2)ccc(Nc2ccccc2)cc1 Cn1nc(CC(=O)NCC2(CNC(=O)CCCc3ccccn3)CCC2)cc1Cl C1(C(=O)N)CC2(CCC2)C1.C(C(=O)N(CC)C1CC1)(C(C)C)OCC [SH](=O)(=O)c1c(C)noc1C.N1(C(CC(=C)C)=O)CCC(NC(=O)CN)C(C)C1 CC1CN(C(c2c(Cl)csc2Cl)=O)CCC1NC(=O)CNC(=O)C(C)(C)C c1(NC(C2C(C(=O)Nc3nc(C)c(O)cc3)C2)=O)cnnc2ccccc12 C=CCC(C)(C)CC(=O)N1CCC(CCNC(=O)Cc2ccn(CC)n2)C1 N1(C(C(=O)OC)C2CC2Cl)CCN(C(c2ccncc2Cl)C(=O)NC(C)C)CC1 C1(NC(=O)C(C2CCOCC2)F)CN(C(C2CC=CCC2)=O)CC1O Cc1ccc(C(O)CCNCC2CC2C(=O)O)s1 C1(CNC(CCC#C)=O)CC2(CC2)CN1C(=O)C=Cc1ncc[nH]1 Cc1nc2ccc(C(N3CC4C(CNC(C5(C)CC5(F)F)=O)C4C3)=O)cc2[nH]1 C(=O)(C1=NOC2(CCOC2)C1)N1CC2C(NC(C(NOC)=O)=O)(C2)C1 N1(C(C2C(=O)OCC2)=O)CCCC(O)(c2cn(CCO)nn2)CC1.N12CC(C1)C2 C(=O)(C(=O)NCC(C)(C)NC(=O)C(O)C1CCCC1)N(C)C C(=O)(CCCCC(C)(C)C)NCC(CO)NC(C(C)(CO)OC)=O N1(C(CSCC(=O)OC)=O)CCC2CCC12.C1(C)(C=O)CCC(C)(C)C1.N CCC(C)CN=C(NCC1(c2ccc(OC)cc2)CC1)NC1CCS(=O)(=O)C1 c1(C(N2CC=CC(NC(C3(CO)CCC3)=O)C2)=O)cc2ccc(O)nc2s1 CCC(C)CC(C(=O)NCc1ccncc1OC)NC(C1CS(=O)C1)=O c1(N2CCC(C)(SC)C2)nc(=NCC2CSCCO2)[nH]c2ccsc12 c1(C(=O)NC2CCN(C(CSC(C)C)=O)C2C)noc2c(F)cccc12 c1(NC(C2C(C(=O)Nc3ccc(C)nc3C)C2)=O)c(F)cccc1C#N C1(C(=O)N)CC12CC2(F)F.n1(CC(=O)NCCC)cc(CN2CCCC2)nn1 C1(S(C)(=O)=O)(C=O)COC(=O)C1.C1CCC(F)C1.C(C(=O)NC)=CC c1(CC=O)cnc2ccccc2c1.C#CC1(C(=O)NCCC2(C)CC2)CC1.N c1(C(N2CCC(NC(C3(n4ccnn4)CC3)=O)C2)=O)cc2n(n1)CCCC2 C1(C(N2CCC(N(C(=O)C3=CCCS3)CC)C2)=O)CCC2C(C1)C2(F)F Cc1cn(C2CCCCC2)[nH]c1=NC(=O)C(=O)Nc1cnn(CC(F)F)c1 Cc1c(-c2noc(CCc3cccc(F)c3Cl)n2)cccc1[N+](=O)[O-] C(=O)(C(CC1CCCC1)N(C1CC=CCC1)CCO)NC(c1ccsc1)C C#CCCCC(C)C(=O)NCC1=CCCN(C(c2cc(C#N)cn2C)=O)C1 N(C(=NCCCc1ccsc1)NCCN1CC(C)OCC1C)CCSC CS(=O)(=O)c1sccc1C(=O)NC1CC1NC(c1ccc2nc[nH]c2c1)=O CCC(C(=O)NCC(O)CCNC(c1cc(C(C)C)no1)=O)C(C)C Cc1cnc(C)c(C(N2CC(NC(c3nc(C)n(C)n3)=O)C(O)C2)=O)c1 n1(CC)cc(CNC(=O)CN(C(=O)C(C)n2cccc2)CC(C)C)nn1 C(C)(C(C)(C)C(=O)NC12CC(C)(C1)C2)NC(C(C=C)CC)=O N1(C(=O)CCc2nc(C(F)(F)F)no2)CCC(S(=O)(=O)c2cccc(F)c2)CC1 C1(NC(C(N(C(C2N(CCC)CCC2)=O)C)C2CC2)=O)CCCCCCC1 N1(C(c2n(CC)nnc2)=O)CCC(NC(c2ccc(Cl)o2)=O)C1C C1(C(=O)NCC(CNC(C(C)OC2CCCCCC2)=O)(C)C)CCCCC12CC2 C1(C(C)NC(c2ccn(CCC)n2)=O)CCCN(C(c2ccoc2C(C)C)=O)C1 n1(CC(=O)NC2C(NC(C(CC(C)C)O)=O)CCC2)ncc2ccccc2c1=O CCC(C(=O)NC1COCC1NC(C1CC=CCC1)=O)n1nccc1C C12(C(N(CCN(CC=C)C)CC)=O)COCC1CN(C(=O)CC(O)(CC)CC)C2 c1(N(C)C)ccc(S(=O)(=O)NCCSCC(=O)Nc2nccs2)cc1[N+](=O)[O-] C1(C=O)CC2(CCCCC2)C1.c1(COC)ccc(C(=O)N)[nH]1.C1CC(CC)C1 Cc1cncc(C(N2CC(NC(c3cc(C4CCCC4)nn3C)=O)C(O)C2)=O)n1 Cc1ccnc(C)c1C(N1CC(NC(C2(O)CC2)=O)CC(C)C1)=O CC1CC(NC(=O)NCCCP(C)(C)=O)c2cc(C(F)(F)F)ccc21 C#CC1(O)CCCC(NC(C2CCC(C(=O)N(C)C)CC2)=O)C1 C12(NC(c3ccc(C)cc3C)=O)CCCC1N(C(c1oc(C)nc1C)=O)CC2 CC(C)C(C)C(C)CC(=O)N.C12CC(CN1C(=O)CC1CCS(=O)(=O)C1)C2 N12CCCCC(C1)NC(=O)C1(CC1)C2=O.c1(C(=O)NC)ccc(Br)cc1.CO C1(C(N2CC=C(CNC(C3C(C)CC3)=O)CC2)=O)CCc2cnnn2C1 C1CCN(C=O)CC1(C)C.c1(CC)cnc(-c2ccoc2)s1.C(C)(C)C.C(=O)N CC(C)CC(C)C(=O)NCC(C)(C)CC1CN(C(C2CC(C)N(C)C2)=O)C1 CCCC(C)CCCC(=O)NCC1CCN(C(c2cc3sc(Cl)cc3s2)=O)C1 C(=O)(CCc1cnc[nH]1)OCC=C(C)C.C(=O)CCO.C(=O)C(F)(F)F.N CC1COCCN(C(=O)CC2CCCCN(C(=O)C(c3cncnc3)C)C2)C1 c1(C(N(CC)C)=O)ccc([N+](=O)[O-])cc1.CCC(COC)C(=O)N.C(C)(C)C C(=O)(C(O)C(F)(F)F)N1CCC(CC(C)NC(CCc2nnc(C)n2C)=O)CC1 C(N=c1cc[nH]cc1S(=O)(=O)NCC(C)Cc1cccs1)c1ccnc(C)n1 CC(CCCC(F)(F)F)N=c1[nH]c(=NCCCCC2CC2)c2c(F)cccc2[nH]1 CN1CC(=O)N(CC(N2CC(F)(c3cn(CC(C)(C)C)nn3)C2)=O)C1=O C1(C(=O)NCC(CC)(CC)NC(CC=CCC)=O)CCCC12NC(=O)NC2=O C(=O)(C1=CCCN(C(=O)C2=CCCSC2)C1)NCCc1c(C)noc1C c1(C(=O)NC(=O)CCSc2ccccn2)ccc(Br)cc1 n1(C(C)C)cnc(C(=O)N)n1.c1nc(C(=O)NC(C)C)co1.C1CCCO1.C N1(C(Cn2cc(CNC(C=CCOC)=O)nn2)=O)CCOC2(CC2)C1 C1(NC(=O)Cn2cccn2)CCCCN(C(=O)Cc2cncc(Br)c2)C1 Cc1cccc(C(N2CC(NC(=O)CS(=O)(=O)N(C)C)CC(C)C2)=O)c1N c1(C(=O)NC2(C)CN(C(Cc3cc(C)nn3C)=O)C2)ccc2c(c1)COC2 c1(C(N2C(C)(CNC(CN(CC)CC)=O)CCC2)=O)oc2ccccc2c1Br Cc1cc(C(=O)NC2CC(F)(CNC(C3CCC(F)C3)=O)C2)oc1Br N1(C(c2ccc(COC)o2)=O)CCC2C(NC(C3CN(C(C)C)C3)=O)C2C1 C(CCCCC(=O)NC1CN(C(c2cc(C)sc2C)=O)CC1OC)OCC C1(C(N2CC(O)(CNC(CCC=C)=O)C2)=O)CCC12CCCO2 N1(C(C=CCOC)=O)CC(NC(=O)CC(O)c2ccccc2)C2(CC2)C1 C1(C)(C(N2CC(C)(CNC(C=CC)=O)C(C)C2)=O)CCCCCCC1 c1(OC)ccc(F)c(C(=O)NC2CN(C(=O)CC3CC(=O)NC3=O)CCC2O)c1 Cc1nn(C)cc1CC(=O)N(C)CC1CN(C(=O)Cc2csnc2C)CCO1 C(CC(C)(C)C(=O)NCC1(C)CCOCC1)OC.C(=O)C(C)(C)n1cnnn1 C(CC(C(C)(C)C)NC(=O)C(C)C)N(C(c1c(C)nc(O)s1)=O)C Cc1cncc(-c2cn(CCNC(=O)COC(F)(F)F)nn2)n1 C1(C(=O)N(c2ncccn2)CC2CC2)CC2C=CC1N(C(C1CCC1)=O)C2 C(CC(CC)C(=O)NCC=CC(=O)NCc1cn(C)nn1)=CC N1(C(CC=CCC)=O)CC2(C1)CN(C(c1ccccc1CC(=O)OCC)=O)C2 n1(CC)ccc(C(=O)NCC(CCOC)NC(=O)CCCC2CC2)c1C c1(CCC(=O)NCC(CC=C)NC(C2CCOC2(C)C)=O)ccc2c(c1)OCO2 CC(C)CCCCCC(=O)NC1COC2(C1)CN(C(C1(C#N)CCCOC1)=O)C2 S(=O)(=O)(c1cc(C(=O)O)n[nH]1)NC(c1ccncc1Br)C C1(C(N(C2CN(C(Cc3c(C)nc[nH]3)=O)C2)C)=O)Cc2cc(F)cc(F)c2O1 c1(NC(CC2N(c3nc(SC)c(F)cn3)CCOC2)=O)ccc2oncc2c1 c1(CC)n[nH]c(=NC2(CNC(c3cncn3C)=O)CCOCC2)s1 C1(C(=O)NCC(C)F)CC2(CC2)CN1C(=O)C=Cc1cc[nH]c1 N1(C(CCCOC)=O)CC(C)(C)CC1C(N1CCC(C)(O)C1)=O c1(CC(=O)N(CC)CC2CCCN2C(=O)CCC2CC2)nc(Br)sc1C C1(C(C)C)CN(C(c2csc(-c3cnn(CC4CC4)c3)n2)=O)CCS1 C1(C(=O)NCCNC(C2CC(N(C)C)C2)=O)CC=CCC1 N1(C(c2ccc(CC)cn2)=O)CCCC(NC(=O)CCc2cncc(F)c2)C1C C=CC(C)(O)CC(=O)NC(CC1CC1)C(=O)NCc1ccc(CO)o1 N1(C(C2CCN(C(c3nc(C)oc3)=O)CC2(C)C)=O)CCC2(CCOC2)CC1 c1(NC(C(=O)NCC(C(C)(C)C)(C)O)=O)ccc(F)c2ncccc12 Cn1nc(C(=O)NCC(C)(C)NC(c2coc3ccccc23)=O)c2c1CCCC2 N1(C(C2NC(=O)OCC2)=O)CCN(C(c2ccncn2)=O)CC1CF c1(OC)ccccc1C(CNC(c1cc(F)n[nH]1)=O)NC(=O)C(C)O C1(NC(=O)CC2CCCCC2)CC2CC1CN(C(c1ncc(Br)cn1)=O)C2 C12(C(=O)NC3CCCN(CC)C3)CC3CC(C)(C1)CC(F)(C3)C2 C1(C(NOCCCC)=O)CC2CN(C(c3ncncc3C)=O)CC2C1 c1cccc(F)c1Cl.N1(Cc2ccn(CC)n2)CCOC(CNC(=O)C=O)C1.N n1(CC)nc(C2CC2)cc1C(=O)N(C)CCOCCNC(=O)C(N)=O Cc1[nH]c2c(C(=O)NCC(c3cccc(F)c3)O)cccc2c1C c1(C(=O)NC2CC(C)N(C(c3cnc(C(F)(F)F)s3)=O)C2)nccc2occc12 C1(C(=O)NCC2CC2Cl)(CC)CCN(C(C2CCC(=O)NC2)=O)CC1 CC(C)CS(=O)(=O)CCC(=O)NC(C1CN(C(=O)CN2CCCC2=O)CCO1)C c1(CC=O)ccc(O)nc1.C1(CNC(CN(c2cnccn2)C)=O)CCCC1.N C(CN=c1nc(N2CC3CC3(c3ccccc3)C2)cc[nH]1)C1CCC(C)(C)O1 N(C1CN(C(c2cnn(C)c2CCC)=O)CCc2ccccc21)C(CC=C)=O C1(CNC2C(c3c(C)n(C)nc3)N(C)C(=O)C2)CCC2(CC1)NC(=O)N(C)C2=O N1(C(c2c(C)cc(OC)nc2)=O)CC(C)CN(C(=O)CCS(N)(=O)=O)C(C)C1 N1(C(c2c(CC)ccs2)=O)CCCCC(C(=O)NCC(C)(O)C2CC2)C1 c1(CCC(=O)NC(CC)CNC(=O)C(N2CCCCC2=O)C)cc(F)cc(Cl)c1 N1(C(COC2(C)CCCC2)=O)CCOCC1CCNC(c1ncc(Cl)s1)=O C1(CCC(=O)N(CC)C)CCN(C)CC1.CC1CCC(=CC(=O)NCCO)C1 CC(C)C(CCC(=O)N(C)C(c1nccs1)C)NC(=O)C(C)C c1(C(N2CCCC(CN(C)Cc3ccns3)C2)=O)cc2sccc2s1 O=S(=O)(c1cccc(N2CC3C(C2)C3(F)F)n1)NC1CN2CCC1C2 c1(C(C)=O)ccc(C(=O)NCCC2CCC2)cc1Cl.C1(C)(CC=O)CC1F.N Cn1ncc(Cl)c1C(=O)NC1CN(C(c2ccn(C(C)(C)C)n2)=O)CC1O C(=O)(C1=NOC(C)(C)C1)N(CC(=O)N(CC(C)C#N)C1CC1)C.CC.O C1(NC(c2c(CC)ocn2)=O)CC2CC1CN(C(C13CCCC(CO1)C3)=O)C2 c1(C(=O)NCC2C(NC(C(CC#C)C)=O)C2)cc(Br)c(F)cc1OC C(=O)(CC(C)CC(=O)OC)NC1CC2(CC(NC(CCC(CC)C)=O)C2)C1 Cc1cc(Cl)c(C(=O)NCCC2CCC(NC(=O)Cc3nnc(O)s3)C2)s1 c1(OC)cc(O)ccc1NC(=O)C(=O)N(C1CCN(S(C)(=O)=O)C1)C C1(NCCOCCOC)CC2C(NC(=O)C=CC(=O)OC)C2C1 C(CCCCC(=O)N1CCC12CN(C(C1CCCCC1(F)F)=O)C2)OC N1(C(c2c(C)n[nH]c2)=O)CCC(C)C1CNC(=O)Cc1ccc(Br)cc1 Cn1nc(C(N2CCC(C)(CCNC(C3(CF)CC3)=O)C2)=O)ccc1=O C1(NC(=O)CCC2CCC(=O)N2)CCN(C(=O)C2=CCCS2)CC1F c1(NC(C(CC(C)C)NC(C(C(C)C)OC)=O)=O)cc(C#N)cnc1C N1(C(C(C=C)CC)=O)CCC(N=[N+]=[N-])(C(=O)NCC2CCN2CC)C1 Cc1cc(C(=O)NC2CN(C(=O)C(C)OC(C)(C)C)CCC2F)cc(C)c1C c1(C(=O)N)cc([N+](=O)[O-])c2nsnc2c1.CC1CC(C(=O)NC2(C)CCC2)C1 c1(C(N2C(C=O)CC3CC32)=O)ccc(Br)cc1S(C)(=O)=O.c1(CC)nccs1.N c1(C(=O)NC(CC)CNC(c2cnn[nH]2)=O)cn(CC(=O)NC)nn1 c1(C(NOCC(=O)N(C2CCC3(CC3)C2)C2CC2)=O)cn2c(n1)CCC2 C(C)(C)(C(=O)NOCC1CC1)C1CCCN(C(Cc2scc(C)c2)=O)C1 c1(CC(N2CC=CC2C(N2CC3COCC3C2)=O)=O)ccc([N+](=O)[O-])cc1F c1(CS(Cc2ccc(C)o2)=O)nc(C2CCCO2)nn1-c1ccc(Cl)cn1 N1(CCC(=O)NCCCN(C(c2occc2Br)=O)C2CC2)CCC(F)C1 N1(C(C2N(C)C(=O)OC2)=O)CC(F)(F)CC1(C)C.C(=O)(C=CC(N)=O)N CC(C)C(C(=O)N)NC(=O)C(F)(F)F.C1CCCN1C(=O)CN1CCCC1=O c1(C(=O)NC2CCN(C(c3cc(C)nn3C)=O)CC2F)cc(F)cc2c1CCC2 Cc1cccc(C)c1NC(=O)C=O.C1(O)(CC)CN(C(c2[nH]nnc2C)=O)C1.N Cc1c(C(N2CCC3CN(C(C4CC(=O)N(C)C4)=O)CC23)=O)ccc(F)c1F N1(C(c2[nH]cc(C(C)=O)c2)=O)CCCC12CCN(C(=O)C1=C(Cl)CCC(C)C1)C2 N1(C(c2c(C)cn(C)n2)=O)CCCC1(C)C.c1(C=O)coc(CS(C)(=O)=O)n1.N C1(OC)CCC(CC(=O)NC(CNC(C2(CO)CCCCO2)=O)C2CC2)CC1 C1(CNC(C2(OCC)CCC2)=O)CN(C(c2cnc(C)o2)=O)CC1(C)C c1(CC)ccccc1C(F)(F)C(=O)NCC(C)CN(C)C(c1n[nH]cc1F)=O c1(C(=O)NC(CNC(C(CC)(C)OC)=O)C)cc(C(C)(C)C)n(C)c1C Cc1cc(C(=O)NCCc2ccc(C)cc2)ccc1Cl.C1(C)(CC=O)CC1F.N C1(C)(C(=O)NC)CCN(C(C2CC2(C)C(F)(F)F)=O)CC1 c1(CC)ccc(C(=O)NCCC(C)NC(C2(COC)CCCO2)=O)cn1 c1(C=O)cc(Cl)cc(Cl)c1[N+](=O)[O-].c1(C(N2CC(C)(C)C2)=O)cc(Cl)ncc1Br.N O=C(C1=NOC(CNC(c2ccc(Cl)s2)=O)C1)NCCc1nncs1 C1(C)(C(N2CCC(CSC)C2)=O)CC12CCN(C1C3CNCC1C3)CC2 c1(CC)nc(C(=O)NCC2(O)CN(C(C3CC3)=O)C2)cs1.C(C)C.C c1(C=O)cc(C(C)(C)C)ccc1O.C(C)C(=O)N(C(C)CC)C.C(=O)NC.N Cc1cc(CNC2CCOCC2C(=O)NC(P(C)(C)=O)c2ccccc2)ccn1 c1(C(N2CCN(c3cc(C4CC4)[nH]n3)CC2)=O)ccc2c(c1Br)OC(F)(F)O2 N1(c2cc(CC)nc(C)n2)CCC2(CC1)CC(O)C2 CCN=c1[nH]c(C(N2CCCC(CNC(=O)CC(CC)C3CC3)C2)=O)cs1 CC1CC(NC(C2COCCO2)=O)CN1C(=O)CCNC(N)=O C(=O)(C1=Cc2ccccc2OC1)NC12CCC(CN(C(CSCC=C)=O)C1)C2 N1(C(c2scc(C(C)=O)c2)=O)CC=C(C)CC1.c1(C(=O)N)csc(C(N)=O)n1 c1(CC(=O)NCC2(Cc3ccc(Br)cc3)CC2)ccc(OC(F)(F)F)cc1 n1(CC(=O)NCC(C)(CO)CO)cc(C(=O)ON)cc(Br)c1=O N(C(=NCCCC1CC1)N1CCC(Oc2ncc(C)s2)CC1)CC1(SC)CC1 C1(CNC(Cc2c(C)n[nH]c2)=O)CCCCN(C(c2cn(C(C)(C)C)cn2)=O)C1 c1(C(NC)=O)nn(C)c2ncc(S(C)(=O)=O)cc12.C1(OC)CCC(C)(C)CC1.C CC(C)C(C)(CNC(=O)CC1CCC(=O)N1)NC(C1CCC(=O)O1)=O C(=O)CC(C)CC.N1(CC(N2CC(OC)C2)=O)C(=O)CCC1=O.C(C)=O.C C1(C(N2CC(O)(CCNC(=O)CC3CCCO3)C2)=O)OCC2COCCC12 c1(OC)cc(F)c(C(=O)N(C)CC2CCN(C(=O)CSC)CC2)c(F)c1F C1(NC(C(=O)NCC)=O)CCN(CC2(c3ccccc3)CCN(C)CC2)CC1F C1(CC(N2CC(O)(C(C)NC(=O)CNC(N)=O)C2)=O)CCCCCC1 CCCCCC(C)CC(=O)NCCNC(=O)C(C)(C1CC1)OC c1(C(C)NC2COC3(CCOC3)C2)[nH]nc2c1CCC2(C)C CC(C(=O)N1CCOC(CNC(=O)C=Cc2cccc(C)c2)C1)S(C)(=O)=O Cc1ncnc(O)c1C(=O)NC1CC(Cn2ccnc2)C1 Cc1cc([N+](=O)[O-])ncc1C(N1CCC(NC(c2cnn(C)c2)=O)C12CCC2)=O Cc1ccc(CCC(=O)NCCC2CC(NC(c3cc(CC(C)C)c[nH]3)=O)C2)s1 c1(-n2c(C(=O)NC(C(=O)OCC=C)C(C)C)ccn2)c(Cl)cccc1Cl C(C(C)(CC)C(=O)N(C)CC1CCCC1(C)C)NC(CCCSC)=O C(=O)(CCCC(=O)NC1CC(C)CN(C(c2sccc2SC(F)F)=O)C1)NCC c1(C(N2CCCC(N(C(CC)=O)CCF)C2)=O)ccc(Cl)c(S(C)(=O)=O)c1 N1(C(c2c(C)onc2)=O)CCC2CN(C(C3CC3CF)=O)CC12 C1(N(C)C)CCCC(c2nnnn2C(C)(C)CC)(NCCCCCCF)C1 C1(NC(=O)CCC(N)=O)CN(c2n(C)nc(C3CC3)c2)CC12CCC2 CC(C)CC(C)C(=O)NCCC(C)(C)CNC(=O)C(O)CCc1ccccc1 C(=O)(C(C)(C)CCNC(=O)C#CC(C)(C)C)NCC(CC)N(C)C N1(C(C=COCC)=O)CCN(C(=O)CC2OCCCC2(C)C)CC1CF C(=O)(C1CSc2ccccc21)NC1CC(NC(Cc2cn(CC)nn2)=O)CC1O Cn1cc(-c2cn(-c3ccc(C4CC4)cc3)nn2)c(C#N)n1 CC1CCC(O)CN1C(C1CCC(NC(c2ccc[n+]([O-])c2)=O)CC1)=O CCC(C)(CNC(=O)COCC1CCCO1)C(=O)N1CCC(C=O)CC1.O CC(C)C(O)C(C)C(=O)NCCCCC1CCCN(C(C2(C(N)=O)CC2)=O)C1 Cc1cc(F)cc(C(=O)NC2CCC(NC(c3ccc(Cl)cn3)=O)CC2)c1O N1(CC)CCCC(C(=O)NC2(CNC(C3CC(C)C3)=O)CCOC2)C1.O N1(C(N)=O)CCCC(C(=O)N(CC)C)C1.C1CCCCN1C(=O)Cn1cnnc1 c1(C(=O)NC2CC(C(=O)Nc3c(C#N)ccc(O)c3)C2)cccc2c1CC(=O)N2 C(=O)(C(C)C(CC)CC)NCC(C(=O)NCc1n(CCC)cnc1)O C(=O)(C#CC1CCC1)N(CC(O)CN(C(=O)Cc1ccc(O)nc1)C)C S(=O)(=O)(c1ccc(Br)c(O)c1)NCC(c1cnc(C)nc1)=O c1(OC)ccc2[nH]cc(C(=O)NCCN(C(=O)C=CCF)C(C)C)c2c1 Cc1c(C(=O)NCCC2(O)CN(C(C3CC(F)(F)C3)=O)C2)cnn1C C1(NC(C2(C)C(C)(C)C2)=O)CC(C(=O)NC(CO)CCC2CC2)C12CCC2 c1(C(N2CCC(COCCO)CC2)C(=O)NCC=C)cn2ccc(Br)cc2n1 N1(C(=O)OC(C)(C)C)CC(C(=O)NCCC(N2CCCC2)=O)CCC12CCC2 N1(C(C(C)=CC)=O)CCC(CCCCNC(C2CCCN2C(C)=O)=O)CC1 S(=O)(=O)(c1cscc1C(F)(F)F)NCC(C)(C)C1CC1 c1(C(C(=O)NCCCF)N(CC(F)Cl)C)cnc(C(C)(C)C)s1 C1(CC(CO)NC(=O)NCC(=O)N(C)C)CC(F)(F)C1 Cc1nc(O)nc(C)c1CCC(=O)NCCC(C)N(C)C(C1C2CCCOC12)=O c1(OC)ccccc1C=CC(N1CC(CNC(c2cc(C)ccn2)=O)CC1C)=O CCC(CCCC(=O)N1CC(O)(C)C(O)C1)NC(=O)C(C)(C)F C1(C2CCCN(C(=O)CCc3ccc(O)cc3)C2)(NC(C(C)SC)=O)CC1 Cc1sc(C)c(C(=O)N(CCC(C)NC(=O)C(C)(C)C(C)O)C)c1Br c1(C(N2C(C(C)NC(CC(CC(C)C)C)=O)CCC2)=O)ccc2ncncc2c1 n1(CC(=O)OC(c2nnc(-c3ccc(F)cc3)s2)C)ncc2ncccc12 c1(C(=O)NCc2c(C(=O)NCC(CC)CO)con2)cn(C)cc1C N#CC1CC2(CC(C(N3CCN(C(C4CCC(=O)N4)=O)CC3CO)=O)C2)C1 CS(=O)(=O)C1CCC(C(=O)NCCCC)CC1.C1(CC(=O)N)CC(=O)NC1=O C(=O)(C1COc2ccc(F)cc21)NC1CN(C(c2cccc(C)n2)=O)C(C)CC1 c1(CCC(=O)N(CC(C)NC(C23CCCC2C3)=O)C)cnn(C)c1 N1(C(=O)C(O)C2CCC2)CCCC(C(N2CCCC(CC3CC3)C2)=O)C1 N1(C(CC)=O)CC(CCNC(c2ccnc(C)c2C)=O)OC(C)C1 c1(C=O)cc(C(N)=O)ccn1.c1(C(C)NC(C(C2CC2)SC)=O)ccccc1 N1(C(CCC#CC)=O)CC(N(C)C(c2cc(=O)cc[nH]2)=O)C2(CC2)C1 C(C#Cc1cn(CC2(C(F)(F)F)CC2)nn1)NC(c1ncccc1Cl)=O N1(C(C2(C#C)CC2)=O)CCC2(C=C(C(=O)NC(C)(CC=C)CC=C)C2)C1 C1(CNC(c2cc(Br)ccn2)=O)CCCCN(C(=O)Cc2cscn2)C1 C1(NC(c2cc(C(=O)OC)sc2)=O)CC(C)N(C(C2CNC(=O)N2)=O)C1 N1(C(CCC)=O)CCCCC1C(N1CCCC(NC(C23CC(C2)C(C)O3)=O)C1)=O c1(N2CCC(OCCNC(C3CC(CC)OCC3)=O)C2)nnc(C)c(C)n1 C1(NC(c2ccc[nH]2)=O)CCN(C(C2CCCS2)=O)CC1CO C(N=c1[nH]cnc2cccc(F)c12)C1(NC(c2c(C)nn[nH]2)=O)CCCCC1C C(=O)(C1=CCC(NC(C2(F)CCCCCC2)=O)C1)N(CCC)CCC N1(C(CCC)=O)CCC(C(=O)N(C)CCN(C)C(C2CN(C)CC2C)=O)CC1 c1(NCCCOC(C)=O)c2c(nn1-c1cccc(Cl)c1)CSC2 CCC(O)C(C)(C)C(=O)N1CCC(CCC(N2CC3C(C2)C3(C)C)=O)C1 C(=O)(CCCC(C)CC)N1C2(CNC(C(CCC)OC)=O)CCC1CC2 O(NC(=O)C(C(C)CC)N(C)C(C1CCCC(=O)C1)=O)CCOCC#C C12CN(CCC1F)C2=O.c1(NC(C=CCOC)=O)cncc(-c2ccoc2)c1 C1(NC(c2cnc(CC)[nH]2)=O)CCCCN(C(c2c(N)cnn2C)=O)C1 c1(C(=O)NC(CNC(c2cncc(C(C)=O)c2)=O)C)cnc2ccncc2c1 Cc1cncc(CC(=O)NC(C)(CO)C(=O)N(CCC(O)CO)C)c1 c1(OC)cccc(CN2CC3(CCN3C(=O)CCc3ccc(C)cn3)C2)c1OC C#CC1(C)CCCN(C(=O)NCC2CC3(CCCCC3)C2)C1 N1(C(C=C2CCN(C(c3nccc(C)c3)=O)CC2)=O)CCCC(F)CC1 Cc1cc2oc(=O)cc(CNc3ncc([N+](=O)[O-])cn3)c2cc1Cl C1(NC(c2c(CC)nns2)=O)(CO)CCCN(C(=O)C(C)(COC)CC)C1 c1(C(N2CC(N(C(C(CC=CC)CC)=O)C)C(O)CC2)=O)ccc2nc[nH]c2c1 c1(C(=O)NCC2(NC(C(CC)C(C)O)=O)CC2)ccc(S(C)=O)cc1 C1(NC(CSCCN(CC)CC)=O)CCCCC1.c1(C=O)coc(Cl)c1.C C(=O)(CC1=CCCC1)N1C(CC(=O)NCC2C(C)(C)CCO2)CCCC1 N1(C(c2c(-c3c(C(=O)OC(C)C)nccc3)ncs2)=O)CCCC(C)(CO)C1 c1(C(N(C(C)C2CC2)C)=O)snnc1C1CC1.C1(O)(CC=O)CCCC1.N C1(CN(C(C2(OCC)CCC2)=O)C)CCCCN1C(=O)C(C(C)C)OC c1(N(C)C)ccc(C(=O)NC2CCCN(S(C)(=O)=O)C2)c(Cl)c1 c1(C(=O)NCC(CC)NC(=O)C(C)CNc2ccccc2)cc(C)cc(Br)c1 N1(C(CCNC(COC)=O)=O)CCC(CCCCNC(=O)CN2CCC2C)CC1 C(=O)(CC(C)C(C)(C)C)NC1(CC)CCN(C(c2cccc[n+]2[O-])=O)CC1 C(=O)(C(C(C)(C)C)NC(c1c[nH]nc1CC)=O)NC.C(=O)CC.C(N)=O c1(OC)ccc2c(C(=O)NC)c[nH]c2c1.C12CC1CN(C(c1coc(C)c1)=O)C2 c1(C(N2CCC(CNC(Cn3nnc(C)n3)=O)CC2C)=O)cnc2ncccn12 C1(C(=O)NCCC(C)SC)CN(C(=O)C(=O)CC(C)C)CC1C1CC1 c1(C(=O)NC(c2scc(C)n2)C)ccc(-c2ccsc2)cc1 c1(C(=O)NCc2c(OCCCOC)cccc2)cc(C=O)n(C)c1 CN1CC(OC)CCC1=O.C(=O)C(C)(C)CC#N C1(C)(NC(c2c(CC)cn(C)n2)=O)CCCN(C(=O)Cc2conc2C)C1 c1(C(=O)NC2(CC=C)CCCN(C(=O)CCOCC)C2)cnc2cccnn12 C1(NC(=O)Cc2ccns2)CCC(CNC(C2CCCCC2O)=O)CC1 c1(C(=O)NCC=CC(=O)NCC(C(C)C)OC)nc(C)oc1C C1(C=O)CCS(=O)(=O)C(C)C1.C1(CN(CC)CC)CC2(C1)CC(O)C2 C1(CC(=O)N(CC(=O)N(CCC)C)C(C)C)CC(NC2CC2)C1(C)C CCC(C(=O)NC1CC(CNC(c2cnccc2C(F)(F)F)=O)C1)C(C)O N1(C(CC(CC)C)=O)CC2CCC(NC(c3c4c(nn3C)CCOC4)=O)CC2C1 c1(C(=O)NC(CC)C)nc(CNC(=O)CN2CCNC2=O)oc1C C1(CNC(C(CC)NC(N)=O)=O)C2CN(C(=O)C(O)Cc3cnc[nH]3)CC12 N1(C(c2nc(CC(C)C)sc2)=O)CCC(NC(C2CCCNS2(=O)=O)=O)CC1C c1(C(=O)NC2CC3(CN(C(C(CC=C)C)=O)C3)C2)cc(OC)c(OC)c(Cl)c1 CC(CC(C)(F)F)C(=O)N1CCN(C(c2ccc(C)cc2)=O)C(C)C1.C(N)(=O)N c1(CNC(C(CC#C)O)=O)nnc2n1CCN(C(c1cnn(C3CCC3)c1)=O)C2 c1(CNC(=O)NCCOc2c(C)cccc2C)cnc2ccc(C(F)F)cn12 N1(C(C(c2ccc(O)cc2)C)=O)CCOC(C(=O)Nc2ccc(Cl)nc2)C1 C(=O)(C(O)CNC(=O)C(C)CN(C)C)N(C(COC)C)C Cc1cc(C=O)cnc1OC(F)F.C1CC2(C1)CN(C(=O)C(O)CN(C)C)C2.N N1(C(c2cccnc2O)=O)CCC2CCCN(C(=O)CN3C(=O)CCC3=O)C2C1 N1(C(C(C)OC)=O)CCc2cc(CNC(C3(F)CCCC3)=O)ccc2C1 C1(C(N2CC(N(C(=O)CC3CC=CC3)C)C(O)CC2)=O)CCC2CC1C2(C)C C1(C(N2CCC(C(C)(C)NC(CCC(=O)NC)=O)CC2)=O)CC2CC(=O)C1C2 C1(NC(=O)NC(C(=O)OC)(C)C2CC2)CCOC(C)C1 N#Cc1ccc(C(N2CC3(CC(C(=O)Nc4cccc(F)c4I)C3)C2)=O)c(Br)c1 c1(OC)ccccc1C(=O)NCCCNC(=O)CC1CCCOCC1 C(C(=O)N=S(=O)(CCO)c1cccc(Br)c1)Oc1cccc(OC)c1 C1(NC(COCC=C)=O)CCCCC12CCCN(C(C1CSCN1C(C)=O)=O)C2 C(C)(C)(C(C)CC(=O)N1CCC(C(C)C)(C)C1)NC(c1c(CCC)n[nH]c1)=O Cc1c(N(CC(C)C(C)C)C)ncnc1N1CC(N(C)C)C2(CC2)C1 C1(OCC(=O)OC(C)(C)C)CN(N2CCCC(O[Si](C)(C)C(C)(C)C)C2)C1 N1(C(C)C)CC(CN(C)CC2CCCN2C(C2CCC(C)CC2)=O)CC1=O c1(OC)cc(C(=O)NCCOC2CN(C(C3CC3(Cl)Cl)=O)C2)sn1 CCC(C)(CNC(c1cc(Br)cs1)=O)NC(=O)CC1CCCOC1 CCC(CC)C(=O)N1CCN(C2CCN(C(=O)Cc3cc[nH]n3)C2)CC1 CC(C)CC(O)CC(=O)N1CCCC(CC(N2CC(CO)(CF)C2)=O)C1 CC(C)(C(F)(F)F)OC1CCC1C(N1CCCCC1C)=O.C(=O)CCCC#N.N c1(C(=O)NCC(=O)NC2CC2)coc(CNC(=O)CCCF)n1 N1(C(c2cc(C)[nH]n2)=O)CC2CCC(C2)C1.c1(C=O)cc(C)n(C(C)(C)C)n1.N CC1(CCC(N2CCCC(n3cc(-c4cccnc4F)nn3)C2)=O)NC(=O)NC1=O C1(NC(C(CCC)(C)CC)=O)CCC2CN(C(=O)CNC3CCSC3)CCC2C1 N1(C(C(C)C)=O)CCC2(CC1)CC(C(=O)N1CCc3n[nH]cc3C1)=NO2 C1(C(C=O)N(CC(C)OCc2ccccc2)CC)CCCC1(C)C.CC(C)C.N CCC(F)(F)C(C)(C)C(=O)NC1CCC(CCNc2ncn(C)c(=O)c2Br)C1 CC(C)C(C(=O)N(CC(C)(C)NC(c1cnc(Cl)[nH]1)=O)C)n1ccnc1 Cc1cc2occ(CC(=O)NCC3CCCCN(C(=O)C=CCO)C3)c2cc1C N1(C(C(CC(=O)OC)C)=O)CC2CCCC(N(C)C(c3cc(C)n(C)n3)=O)C2C1 CC1=CC(C(N2CC=CC2CNC(C2(C(N)=O)CC2)=O)=O)SC1 CCCC(CCNC(c1ccc(-n2cc(C3(C4CC4)CC3)nn2)cc1)=O)CCC N1(c2nccc(C)n2)CCc2sc(C(=O)Nc3cn(C)cn3)cc2C1 N1(C(c2nn(CC)c(C)c2)=O)CCC2(NC(=O)CC3CC(F)(F)C3)CCCC12 C1(NC(CC2N(C(c3c(C)nccc3)=O)CC3(CC3)C2)=O)CC2CC1C(O)C2O Cc1cccc(C(=O)NCC(C)(C)NC(=O)CC2CCC(C3CC3)O2)c1 Cn1ccc2cccc(C(=O)NOCCCCCc3cn(CC(=O)O)nn3)c12 N1(C(=O)C(O)Cc2cccc(Cl)c2)CCN(C(=O)CC2CC2)C(C2CC2)C1 N1(C(=O)NC2CN(C)C(=O)C2)CC2(C1)CN(Cc1ccc(C(F)(F)F)cc1)C2 c1(C(N(CC(=O)NCC)CC#C)=O)cc[nH]c1NCCCc1ccccc1 CCCC(C(O)C(=O)NC(c1ccccn1)CC)NC(c1ncn(C)c1C)=O CC(CN(C)C)CCC(=O)N1CC(C(=O)NCC2C=CCC2)C(C)(C)C1 CN1CCC(C(N2CCC(CF)CC2)=O)(NC(c2cc(O)cs2)=O)C1 CCCC(C(=O)NCC1CC1CNC(=O)CN(CC)CC)OC N1(C(CC(CC)(C)C)=O)CCCC1C1CCCN1C(c1conc1C)=O Cc1ncccc1C(N1CCC(OCC(=O)N(C2CCC2)C(C)C)C1)=O c1(C(N2CC(C(C)C)C2)=O)cc(CNC(=O)C)on1.C1(C(=O)N)CC1C C1(NC(C(C)OCCC(=O)Nc2ccccc2)=O)CCCC1CF.C(N)=O O=C1Nc2ccc(C(N3C4CCC3CN(C(C3COCCO3)=O)C4)=O)cc2C1=O CC1=C(C(=O)N2CCC(NC(c3cc(C(C)(C)C)[nH]c3C)=O)CC2C)CCO1 C1(C=O)CCCC(C(N)=O)C1.c1(C(=O)OC)c[nH]nc1C(=O)NC1CCC1 C(C(C)(C)CC(=O)O)NCC(c1c(OC)cccc1)C C1(CNC(=O)C(=O)Nc2ccccc2)CCCCC1Nc1nc(Br)cs1 c1(C(N2C(C)CN(C(C3(CF)CC3(F)F)=O)CCC2)=O)cc2c(s1)CC(C)(C)C2 C1(CC)CC(C)(C)CN1C(=O)CCn1cc(CN2CCC(F)CC2)nn1 c1(C(N2C3CN(C(C(C)(C4CC4)OC)=O)CC2CC3)=O)cc(F)cc2ccoc12 C1(CC(=O)NCCCN(C(c2c(OC)cccc2)=O)C)CCC2(CCC2)CO1 CC1(C(N2CCCC(CCNC(=O)Cc3cncs3)CC2)=O)CCC(F)(F)C1 CCCCC(C(=O)N1CC(N(C)C)C(C)(C)C1)NC(C1C=CCS1)=O c1(C(N(CC(C(=O)NC(CSC)C)C)C)=O)nn(C)cc1Cl C(CC(C(=O)NOCC(=O)N(C)C)NC(C1CCC1C)=O)OCC Cc1sc2ncc(C(N3CC(OCCNC(C4CCCC4)=O)C3)=O)c(=O)n2c1C c1(C(=O)NCC(CC)NC(=O)CCCC(=O)N(C)C)sc(C)c(Br)c1C C(=O)(C(CNC(C1CCCCO1)=O)CC(C)C)N1C2(CC(COC)C2)CC1 c1(C(COCCOC)NC(=O)C(C)c2ccsc2)cccc(Cl)c1.CC=O.N N1(C2C3(CC(S(=O)(=O)NC)C3)C2)CCc2c(Cl)ccc(OC)c2C1 c1(CC(N2C3C(C(=O)O)C(C3)C2)=O)ccccc1F.CC1(C(F)F)CC1C=O c1(CCC)ccccc1C(=O)NCCCC1CCCCN1C(=O)C(CSC)OC C1(C(C(=O)NCC(C(=O)NC)C)C)CCN(C(=O)Cn2ccnc2)CC1 C1(CC(=O)NC(CNC(COCCCOC)=O)(C)CC)CCOCC1(C)C CCC(C)C(O)C(=O)NC(C)CC1CCN(C(=O)COc2ccc(Cl)nc2)CC1 c1(C(=O)NCC2CN(C(C(CC(CC)C)C)=O)CC2C)cc2c(cn1)OCCC2 C1(NC(COCCN(C)C)=O)COCCN(C(=O)CCCc2ccccc2)C1 c1(OC)cccc(F)c1-c1cccc(NCc2sc(Br)nc2Br)n1 C1(C(N(CC(CN(C(c2ccc(OC)cc2)=O)C)O)C)=O)COC2COCC12 Cc1cn(C)nc1C(=O)NC1CCOCC1C(=O)NC1(CCO)CCCC1 c1(OC)ccc(CC(=O)N(C(C)CNC(C2(C(C)=O)CC2C)=O)C)cn1 C(=O)(C1Cc2ccc(Cl)cc21)NCCc1c(OCC)c(Cl)ccc1 c1(C(=O)NC(C(=O)OC)C(O)C(C)C)cc(C)nc(O)c1[N+](=O)[O-] C(=O)(C1=C(C)NC2=NCCCC2=C1)N1CCC(CCOC)(NC(=O)CO)CC1 C(=O)(CCCCC(F)(F)F)NCC1(C)CCCN1C(c1ccc(N)c(O)c1)=O N1(C(C(C2CCOCC2)C)=O)CCC2CN(C(=O)C(C)(C)C3CCCC3)CCC12 c1(C(=O)NC(CC)CNC(=O)COC(C)(C)C)cccc(Br)c1N N#Cc1cncnc1C(=O)Nc1cccc(NC(=O)CNC(N)=O)c1 C1(C(c2ccc3cc[nH]c3c2)=O)CCc2nnn(C3CCC3)c2C1 CC(C)CCC(=O)N1CC=CC1CNC(=O)C(F)(F)C.C(=O)(CC(C)C)N CCCS(=O)(=O)C(C)C(=O)NC1COCC1NC(C1(CF)CCOCC1)=O c1(NC(C(CC)c2ccccc2)=O)ccc(F)c([N+](=O)[O-])c1 c1(OC(C)C)ccc(N)c(C(=O)NC2CC2)c1.N1(CC=O)CCC(C)C1.N N1(C(c2c(C)cc(CC)o2)=O)CC(C)N(CC)C(C)C1 c1(C(C=O)N(C)C)ccc(Cl)cc1.C=C1CC(C(=O)N)(CF)C1.C1COCC1 C1CC2CCC(C1)N2C.C(=O)(C(C(=O)NCc1c[nH]nc1C=O)OC)OC.N c1(C(=O)NC2C(C)N(C(c3ncc(Cl)cc3O)=O)CCC2)coc2ccccc12 CCC(C)C(O)C(C)C(=O)NC(C)(CNC(=O)CCC)C(C)C.C(C)(=O)O C(CC(C)CCO)NC(C1CCN(C(C(n2ccc(C)n2)C)=O)C1)=O Cc1cc(O)ccc1C(=O)N.C1CC(C)(C)CN1C(C1CCC(N=[N+]=[N-])C1)=O.C c1(CC)nnc2n1CCCC2CC(N1CC2CC2(NC(=O)C=O)C1)=O.C1CC1.N C12(NC(c3scc(C)c3)=O)CCCC1N(C(c1ccc(C#N)cc1)=O)CC2 N1(C(C(CC)F)=O)CCC2(CC1)CN(C(c1ccc(CC3CC3)s1)=O)CC(C)O2 Cc1ccc(C)c(OCCC(=O)NC)c1.C1(C=O)CC(=O)NC(C)C1.C1CC1 c1(OCC(=O)NCCN(C)CCO)ccc(F)cn1.c1ccc(C=O)cc1.N C(CCCCCCC)N.C(C)(C(C)CO)N(C(C=CC=CC)=O)CC c1(CSC(C)C(N2CCC(NC(=O)CCN3CCCC3)C2)=O)ccccc1 C(=O)(C(C(C)(C)C)N(C)C)N1CC(NC(COC(CC)C)=O)C(CO)C1 C1(F)CCN(C(c2c(C)noc2C(C)C)=O)C1.CCC(C)C(=O)NCC(=O)N c1(C(=O)NC(C2CCN(C(C(c3ccccc3Cl)C)=O)C2)(C)C)ccccc1O C#CC(C(C)O)NC(=O)CN(C1CC(C#N)C1)C(=O)CC12CCCC1C2 C(=O)(C1c2c[nH]nc2CN1C(=O)CN(C)C(C)C)N(CCCCC(C)C)C N1(C(C2CCC(C(=O)OC)C2)=O)CCOCC(CNC(=O)CCC(C)SC)C1 Cc1ccc(C(=O)NC(C)(C)CCNC(c2ccc(C3CC3)cc2F)=O)nc1C N1(C(c2ccc(CCCC)cc2)=O)CC2OCC(NC(=O)C(C)SC)C2C1 C1(NC(C)=O)C2CC1(C)CN2C(=O)Cc1ccc(C)c(C)c1 C1(C=O)(C(=O)NC)CC12CC2.C1CCCN1C(=O)C.C(C)(C)C.CC.O c1(C(C(=O)NC2(C)CC(NC(CC(C=C)C)=O)C2)C)cn(C)c2ccccc12 C1(CC(=O)N(C(CC)C(=O)NCC(C)(CC)CC)C2CC2)CCCC12CC2 Cn1nncc1CCNC(=O)C(CO)NC(=O)CSc1cn[nH]c1 c1(C(CNC(=O)Cc2cccc(Cl)c2)NC(C(CC)C)=O)cc2ccccc2o1 c1(C(=O)NC(C2(O)CCN(C(C3(C)CCSCC3)=O)C2)C)cccc2nc[nH]c12 C1(CC(=O)NC(c2nc(CC)[nH]n2)C)CCCCN1C(=O)Cc1ccc(C)s1 C1(SC)CC(C(=O)NCCN(C2CCCC2)C(COCCOC)=O)C1 C1(NC(CCC2(C)CCC(=O)N2)=O)CC2CC1CN2C(c1cccc(N)n1)=O C1(NC(=O)NCC(N2CCN(C)CC2)C)CCn2nnnc2C1 C#CC1(OCC(=O)NC2CCCC2NC(C2(CC)CCOC2)=O)COC1 CC(c1ccc(F)cc1)=CC(=O)NC(C)CCCNC(c1ccccc1O)=O c1(C(=O)N)ccnc(Cl)c1F.C1(O)(CC)CN(C(C2CCC2c2nc[nH]n2)=O)C1 C1(NC(C(C(C)C)O)=O)C2CCN(C(c3ccc([N+](=O)[O-])s3)=O)CC12 N1(C(CCN(C)CC)=O)CCC(F)(C(=O)N(CC(O)(CC)CC)C)C1 N1(C(COCCCC(C)C)=O)CC2(CC(NC(=O)C(O)C(F)(F)F)CO2)C1 C(CCS(=O)(=O)Cc1cn(CC(=O)O)nn1)NCc1n(C(C)C)ncn1 C(=O)(CC(C)(C)C(F)F)NCCCN(C(CC1C(C)=NNC1=O)=O)CCO Cc1cc(Cl)c(Cl)cc1C(N1CCC(C(C)NC(=O)Cc2cscn2)C1)=O Cc1cccc(C(N2CCN(C(=O)C=CC3CCC3)CC2)CN2CCCC2)c1F c1cc(=O)n2oc(C)cc2n1.C1(C(C(=O)NC(C)C)OC)CCC(F)(F)CC1.N C1(CC)CN(C(c2cc(Br)c(C)o2)=O)CCN1C(=O)CC1CC=CCC1 C(C)(CO)(C(=O)NCCCCNC(=O)CC1CCC=CCC1)NC(C)=O C1(CC)CN(C(c2nnc(C)cc2O)=O)CCC1NC(c1[nH]ccc1C1CC1)=O c1(CC)c(C(=O)NC(C)C(C)C(=O)NCC2(CCOC)CC2)nnn1C N1(C(C2CN(C(c3c(N)cncn3)=O)CC2(F)F)=O)CCc2cc(F)ccc21 C#Cc1ccccc1CNC(=O)C(CC(=C)Cl)NC(c1cncc(C=C)c1)=O C1(C(=O)NC2CCC(CC(=O)NC3CCC4CC3CO4)CC2)CCCCC1(F)F C(=O)(CCC(=O)NCCC)N(C1CCN(C(c2cnn(C)c2N)=O)CC1)CCC c1(CNCc2c(C)nn(C3CCC3)c2)c[nH]c2cnc(Cl)cc12 N1(C(C2C(C)(CC)C2)=O)CCn2c(C)nnc2C1.C(=O)C(C)(C)CC(C)(C)C c1(CNC(=O)CC2CCC(=O)N2)cccc(C(=O)NC)n1.C1C2CCCC12 C1(N(C(C=CC(C)NC(C(C2CCC2)OCC)=O)=O)C)CCN(C)C1 C1(NC(=O)COCC(F)F)C2CN(C(C34CCC(C3)C4)=O)CC12 C(C(C)(C)CNC(=O)C(C)N(C(c1ccc(CO)o1)=O)C1CC1)OC C1(CCC#C)CCCN1C(=O)CN(CCC)C(c1coc(C2CC2)c1)=O c1(SC)c(C(=O)N(CC(O)CN(C(=O)CC(C)(C)O)C)C)cnn1C N1(C(c2cn(C3(C(=O)N(C)C)CC3)nn2)C)CCC(CN=[N+]=[N-])C1 CC1(C)NC(=O)CCC1NC(=O)CC1CCN1C(=O)C1=CCCCCC1 Cc1cnc(C)c(C(=O)NC(C2CCCCN2C(=O)CC2CSC2)C)c1 c1(N(C(C2(C)CC2)=O)CC)ccc(O)c(C)c1.C1(CC=O)CCCSC1.N N1(C(CCc2c(C)csc2)=O)CC2(CCC(CNC(=O)C(C)C3CCOC3)O2)C1 N1(C(CCCCSC)=O)CCC(NC(C23CCCC(CO2)C3)=O)CC(O)C1 c1(CCC(=O)NC(CNC(CSCCCC)=O)C)ccc(OC)cc1Cl C1(CNC(CCCC)=O)CCC2(CCC2)C1NC(=O)Cc1ccc(C)cc1Cl N1(C(CCCCOC)=O)CC(C(=O)NCCOC2CCCC2)CC12CCC2 c1(C(N2C(C(C)NC(c3ccoc3Br)=O)CCC2)=O)cc2cnccc2o1 CN1C(=O)CCC(NC(=O)C(C2(O)CCC2)NC(c2ccncc2N)=O)C1=O C(=O)(CC(O)CC(C)C)N(C1CCN(C(=O)C(C)C2CCC2)CC1)CCC C(C)(CCC(=O)N1CCC(CCC(=O)Nc2nc(C3CC3)n[nH]2)C1)SC C12(NC(C3C(C)CCS3)=O)CCC(CC1)N(C(=O)COCc1nc[nH]n1)C2 N#Cc1c(NC2(CCNC(C3(O)CCC3)=O)CCC2)cccc1F N1(C(C(C)(C)F)=O)CCC(F)C(NC(c2nc[nH]c2C(F)(F)F)=O)C1 N1(C(c2cc(C(C)C)[nH]n2)=O)CC2CCC1C(C(N1CCC(O)(CO)CC1)=O)C2 c1(C(N2CC3N(C(C(C(COC)C)C)=O)C(CC3)C2)=O)ccc2ncccc2n1 N1(C(CCOCCN(C)C)=O)CCCC1(C=O)OC.C1CCC1.CC.C(N)=O CC(C)C(C)CCNC(c1ccn(C(F)F)n1)=O.N1(CC(=O)N)CCCCCC1 CCC(C(=O)NC(C1CCN(C(c2cc(F)cnc2O)=O)CC1)(C)C)C(C)(F)F C(=O)(C(F)C(F)(F)F)NC1CC(c2n(C)nnn2)C1 c1(NC(CCNC(=O)Cn2ccnc2)Cc2ccccc2)cc(C(F)F)ncn1 CCCC(C(O)C(=O)NC(COC)CCCC)NC(=O)C(C)(C)C1CCCO1 CC1CC(C(=O)NCCCCCNC(=O)CC2CCCOC2)CC(C)C1 N1(C(C2CC(C)OC2)=O)CC2CN(C(=O)CCCCC3CCCCC3)CC2C1 c1(C(N2CC(SC)C(NC(C3CCC3)=O)C2)=O)cc(C)n(C2CCOCC2)c1C N1(C(C(F)=C(C)C)=O)CCC(C)C(CNC(c2nccc(Cl)c2F)=O)C1 c1(C(N2CCC2)=O)cc(C(=O)C(F)(F)F)ccn1.CC1CC(C(=O)NC)CO1 CC1C(C(N2CC(F)(C)C2)=O)C(O)C(=O)N1C.c1(C=O)ccc(S(C)=O)cc1 c1(C(N2CCC3CCN(C(CC(C)CF)=O)C3C2)=O)cc2c(nc1O)CCSC2 C1(OC)(C)CCN(C(C2CC(CCO)C2)=O)C1.c1(C=O)cc(C(C)C)[nH]n1.N Cc1cccc(C(F)(F)C(=O)NC2C=CCN(C(c3cc[nH]c(=N)c3)=O)C2)n1 C1(C)(NC(c2cnn(C(C)C)n2)=O)CCN(C(c2cscc2C2CC2)=O)C1 CC1CC(CCNC(C2CC(=O)NC(=O)C2)=O)CCN1C(c1cnn[nH]1)=O CCC(C)(C)CC(=O)NCc1ocnc1C(=O)NC(C)(C)CCN(C)C N1(C(CC2CC(=C)C2)=O)CCCC1C(=O)N(C)CC1CCCOC1 C12(NC(c3c(C)nc(C)s3)=O)CCCC1N(C(=O)Cc1cccnc1)CC2 C(=O)(CC(C)C(=O)O)N(CCC)C(C1CC1Cc1ccccc1Cl)=O c1(C(=O)OC)csc(C)c1NC(C1CC(F)CN1C(=O)C(C)(C)C)=O Cc1ccc2c(c1)N(C(=O)CCN(CCO)C(C1CCC(N=[N+]=[N-])C1)=O)CC2 N1(C(CC2CCCN(C(CC3(OCC)CC3)=O)C2)=O)CCN(C)CC(C)C1 C(=O)(C(O)C(C)c1ccccc1)N(CCCNC(c1cn(C)nn1)=O)C(C)C N1(C(c2nc(C)[nH]n2)=O)CCN(CCNC(=O)CS)C2(CCC2)C1.c1cnsc1 C(=O)(C1CC(C)(C)Oc2ccccc21)NC1CN(C(C2CC3(CC(C#C)C3)C2)=O)C1 c1(C(N2CCC(NC(C3C(C)CCC3)=O)(CF)C2)=O)ccc(O)cc1F Cc1cc(Cl)nc(Cl)c1CN1CCC(NC(c2ccccc2C#N)=O)C1 C(CC(CC)C(=O)N(CCCCCCNC(=O)Cn1cc(F)ccc1=O)C)=CC C1(C)(C(=O)NCC2(C)CCN(C(CCCCCC)=O)CC2)CC2CCC(C1)S2 c1(C(=O)NC(C2CCOC2)CNC(Cc2cnc(C)[nH]2)=O)cc(=N)[nH]c(Cl)n1 C1(CNC(c2c(C)nccc2)=O)CCN(C(C2CCCN2C)=O)CC1O C1(N(C(CC=CC)=O)C)CN(C(=O)C(N2CCNC2=O)C)CC1(C)C c1(C(N2CCOCC2C(=O)OC)C(=O)NC(C(=O)OC)C)cccc(F)c1C C1(C(N2C(CC)CN(C(=O)CC3(C)CC3)CC2)=O)CN=C2N=CNN2C1 C(=O)(CC(F)(F)F)N.Cc1cnc(CC(=O)NCCC(O)CNC(=O)CC)o1 c1(C(N2CC(F)(CNC(C=C(C)C(C)(C)C)=O)C2)=O)cc(Cl)c(N)cc1F C12COCCN1C2=O.C(C(=O)NCCNC(C1CC1OC)=O)=CC C(c1cccc(Cl)c1)=CC(=O)NC(C(C)C)CNC(=O)C(C)N1CCC1 c1(OC)ncccc1CC(=O)NC(CN(C)C(C1CCCS1)=O)(CO)CO c1(N(C)C)c(F)cc(-c2noc(-c3c(F)cc(-n4cncn4)cc3F)n2)cc1F C1(C(N2CCC(O)C2)=O)OCC2COCCC12.C1(C(=O)N)CC2(C1)CS(=O)(=O)C2 CC#CCC(C(=O)NCCOC(C)=O)NC(=O)CC1CC=CCC1 c1(OCCC)ccc(CSCC)cc1.C1(C)C(CC(=O)OC)N2CCC(C2)O1 N1(C(C)=O)CCC2(C=C(C=O)C2)C1.C(CC1CC1)CO.C#CCOCCO N1(CCC)CCCC(C(=O)NC(C2CCN(C(C3(C)CC(=O)C3)=O)C2)C)C1 Cc1[nH]c(C#N)cc1C(=O)NC1CCCC1NC(C1CC12CCOCC2)=O C(C1CCc2ccc(OC)cc21)NC1C(=O)NC(C(=O)C2CC2)C1 c1(C(=O)NCCNC(C2=C(C)CCC2)=O)ccc2nc(Br)nn2c1 C(=O)(C1=CCN(C)C1)NC1CC(C(C)NC(=O)CC2CCCCO2)C1 n1(CC=C)cc(C(=O)N)nn1.C(=O)(C(C)(C)c1csc(C)c1)N(CC(C)O)C CN1CCCCC1CCC(=O)N(C1CCN(C(c2cc[n+]([O-])cc2)=O)C1)CCO C(=O)(CCC(=O)N(CCNC(=O)C1CC1)C)NC.c1cn(C(C)C)nn1 c1(C(N2CCC2C)=O)c(F)ccc2nc[nH]c12.C1(C(=O)O)(OC(C)=O)CC1 CCC(C)C(O)C(=O)NCCOCCOC1CC1 c1(NCCC=C=CC)ccc(S(=O)(=O)NCC2OCCO2)cc1F C1(CNC(c2c(CC)cco2)=O)CN(C)CCN1C(c1cc(C)n(C)c1C)=O C(=O)(C(C)(C)CCF)NC(C1CCCN(C(c2n(CC#C)ccc2)=O)C1)C C(CC(C(C)(C)C)NC(C1CNC(=O)N1)=O)N(C(=O)CCc1cnn(C)c1)C C(=O)(C1CCCc2ccnn21)NCC(CC)NC(=O)C(N)=O C1(NC(C(C)N(CCC)C(c2c[nH]c(C(=O)OC)c2)=O)=O)CC(C)OC1=O C#CC(CNC(C12CCC(CC1NC(=O)CCN=[N+]=[N-])C2)=O)CC(C)(C)C c1(N(C)C)cc(CNC(=O)CCOc2cccc(Cl)c2)ccn1 C1(NC(C(C)N(C)C(=O)OC(C)(C)C)=O)CN(C(=O)CCCCCF)CC1(C)C c1(C(=O)NC(CC=C)CNC(C2(O)CCSC2)=O)cn(C)c(=O)n1C N1(C(CCCN(C(c2c(C)ccs2)=O)C)=O)CC(O)C(N=[N+]=[N-])C1 C1(NC(c2scc(C(C)=O)c2)=O)CC2(CCC(NC(c3ccnnc3)=O)CC2)C1 C1(CC)CCC(C)CN1C(=O)C(CCC1CC1)NC(=O)CC(C)COC O=C(C1CCCc2nncn21)N1CC(N2CCN(C(C3C4CCC34)=O)CC2)C1 c1(NC(C(C2CCN(C(C3CN(C)C3)=O)C2)F)=O)cc(Cl)cnc1O n1(CC(=O)NCC(CNC(C(C)SCC)=O)CO)sc(=O)c2ccccc12 c1(C(N2CC3C(NC(CCC#CC)=O)C3C2)=O)cccc(S(N)(=O)=O)c1 C1(O)(C(C)NC(COCCCC)=O)CCN(C(=O)C(O)C(C)CC)CC1 C1CN(C(c2cncc(O)c2Cl)=O)C(C)(C)C1.C(CC(=O)N)NS(C)(=O)=O.C c1(CNC(=O)CCOCCCNC(C2CCC2C(=O)O)=O)cccnn1 C1(C(N2CCC(O)C(NC(=O)C(=Cc3ccco3)C)C2)=O)(OC)CC2CCC1C2 N1(C(C(CNC(c2cc(C(=O)OC)[nH]c2)=O)(C)C)=O)CCNC(=O)CC1 C1(C(N2CCC(CCCNC(c3scc(C)c3)=O)CC2)=O)CCN(C)C(=O)C1 C(=O)(CCCN=[N+]=[N-])NC(CC1CN(C(c2c(C)nn(C(C)C)c2)=O)C1)C c12ccc(cc1)S(=O)(=O)N1CCCC21.c1(C(C)(C)C)[nH]c(=N)ccc1Cl c1(C(=O)NC2(C)CCN(C(C3(O)CC4CCC3C4)=O)CC2)cnn2ccncc12 C1(NC(C(CC=CC)C)=O)CCC12CCCN(C(=O)C(C)=C1CCCC1)C2 N1(C(=O)CC2CC(C(F)F)C2)CC2(CCN2C(=O)C(O)C2CC2)C1 c1(C(=O)NC(CNC2(CCF)CC2)CO)ncnc2sccc12 C1(NC(c2ccncc2F)=O)(CO)CCN(C(c2cnn3ccsc23)=O)CC1 c1(C(=O)NCC(C)N(C(c2cc(C(C)C)c(F)cc2)=O)C)c(F)cc(Cl)cc1F c1(CC)ccc(C(N2CC3C(NCc4cn(C)nc4C)C3C2)=O)cc1 CC1(C)CC(NC(c2ccc(-c3ccccc3F)[nH]2)=O)C(C)(C)O1.C(C)(C)(C)O C1(N(C)C(c2ccc(Cl)o2)=O)CCCN(CC(=O)NCCC#N)C1 CC1CC=C(C(=O)N2CCCCCC(NC(C3CC(C#N)C3)=O)C2)CC1 c1(C(=O)NC2C(NC(c3cc(C)nnc3)=O)C2)[nH]c2cc(Cl)ccc2c1C Cc1ccc(O)c(C(=O)N(C(C)CCNC(C2CC2[N+](=O)[O-])=O)C)c1 N1(C(C2(C)CCN(C(C(COCC)C)=O)CC2)=O)CCC(C2CCOC2)C1 Cc1ccc(C)cc1.c1(CC=O)ccccc1CS(N)(=O)=O.C1CC1C=O.N C(=O)(CC(C)CC(F)(F)F)N1C2C(CNC(C3C(CC)CCC3)=O)C(C2)C1 c1(NCC(=O)OC)cn(CC(=O)NC(C2(C)CC2(Cl)Cl)C2CC2)nn1 N1(C(c2occ(C)c2)=O)CCC(C2CC2)C1C(N1CCC1C(C)O)=O C#Cc1cncc(C(=O)NC2CCCCC2)c1.C1(CC(=O)N)CC(=O)NC(=O)C1 N1(C(C(C2CC2)SC)=O)CC2CC2(CNC(=O)CN(C)C(C)C)C1 Cc1ccsc1C(=O)NC1(C)CN(C(c2scnc2Br)=O)C1 c1(OC)cc(I)ccc1C(=O)NC1CCN(C(c2ccc(Br)cc2)C)CC1 Cn1c(CC=Cc2[nH]nc(N3CCN(C=O)CC3)n2)cnc1Cl.c1ccccc1 N#Cc1cccc(N2CCCC2C(=O)NC2COCCC2NC(C2(O)CC2)=O)c1 c1(C(N2C3CN(Cc4ccc(OC(C)=O)cc4)CC32)=O)cccc2cnccc12 C1(C=O)CC(=O)NC1(C)C.N1(C(C)C(=O)NCC2(F)CCC2)CCC(O)CC1 C1(NC(COCC#C)=O)CC2CCC1N(C(C1(C)CCN(C)C1=O)=O)C2 c1(N2CCCN(c3ncccn3)CC2)ncnc2n[nH]cc12.Brc1cscn1 Cc1c(NCCC2CCC2)ncnc1NCC(C1CCN(C)C1)N1CCCC1 N1(C(c2cc(C)nn2C)=O)CCC2(CCCCC2NC(C2CCCCC2)=O)CC1 N1(C(c2cnn(CC)c2C)=O)CCN(C(c2sc(CO)nc2C)=O)C(C)C1 N1(C(Cn2ccc(C(=O)OC)n2)=O)CCOC(C)C1.C(=O)(CCC)N.C(N)=O N1(C(C2(C)N(C(c3n(C)ncc3)=O)CC2)=O)CC2CC(C1)O2 C1(NC(C(CO)NC(N)=O)=O)CC1C1CCCN(c2ccc3c(n2)CCC3=O)C1 Cc1cc(C)c(C(N2CCC(NC(=O)Cc3ccc(S(C)=O)cc3)C2)=O)c(O)n1 C1(CCC)(NC(C2CC2F)=O)CCN(C(=O)C(C2CCC(F)(F)CC2)O)CC1 C(=O)(CCCC(C)NC(c1cocn1)=O)N(CCCCC)CCOC N1(C(CC=CC=C)=O)CC2CC(NC(c3cnn(-c4ccccc4)c3C)=O)C1C2 C1(NC(C(C)OCCN(C)C)=O)CN(C(C2CC2(F)F)=O)CCC12CCC2.C CC(C)CC(C)CC(=O)NC12CCC(C(N3CCOC(C(C)(C)C)C3)=O)(CC1)C2 CC1CCN(C(c2ccc(=O)oc2)=O)CC1CNC(c1cc(Cl)ncc1F)=O C(=O)(CCC(=O)NC1CCN(C(c2cc(C3CC3)ncn2)=O)CC1)N(C)C c1(C(=O)NC(CC)CN(C(=O)C=NOC)C)cncc2sccc12 C(=O)(CC(F)(F)F)N(C1CCN(CCCNC(=O)C(O)Cc2cnc[nH]2)C1)C CC1(C)C(c2cccc(Cl)c2)CCN1CC(c1ccccc1)N1CCCCC1 C1(NC(CSCCCC)=O)(CO)CCCN(C(c2ccc(C3(C)CC3)cc2)=O)C1 C(=O)(C#CC1CCC2(CC1)OCCO2)NCC1N(C(CCC(=O)NC)=O)CCC1 O=C(N1CC2COCC2O1)C1CCN(C(=O)C23CCCC2CCC3)O1 C1(N=[N+]=[N-])(C(=O)NC(C(C)(C)OC)C)CCN(C(C2CCC3(CC3)C2)=O)C1 N1(C(c2cnn(C)n2)=O)C2CCC1CC(CNC(c1ccc(N)c(Cl)c1O)=O)C2 CCC(O)(CC(=O)N(C(C)COc1ccc(Cl)cc1)C)c1ccccc1 C1(C(=O)NC(C)CN(C)C(c2ccc3[nH]ccc3n2)=O)CC(F)(F)CCC1(C)C c1(CC)cc(C(=O)NCCC2CCN(C(c3cnco3)=O)C2)c(C)o1 c1(C(=O)NC(CCOC)C(C)C)ccc([N+](=O)[O-])cc1OC N1(C(C2=NOC(C)C2)=O)CCN2CCN(C(c3ccnc(F)c3O)=O)CC2C1 c1(C)ccccc1.C1(N(CC(=O)OC)C(=O)NCCCO)CCC(C)(C)C1 c1(NC(C2CCCN(C(=O)CC3CC=CCN3C)C2)C)cc(O)nc(=O)n1C C1(OCC#C)CCN(C(c2conc2C)C(=O)NCC2CCOCC2)CC1 Cc1ccc(C(=O)NC)n1C.C12CC(CN1C(=O)CCCC1CCCC(=O)N1)C2 Cc1ccc(CNC(C2(C#N)CC(C)C2)=O)cc1 C1(N(C(C(=O)N(C)C)=O)CCF)CCCN(C(=O)COCc2ccncc2)C1 CC12CC(CC(=O)NCCCCCCNC(=O)C(C)(C)N(C)C)(CO1)C2 CC(O)(C(=O)NCc1nc(CNC(C2CC(F)C2)=O)cs1)C1CCC1 c1(C(N(C)CC2(NC(C3C=CCCC3)=O)CC2)=O)cc2c(Cl)cccc2s1 c1(C(CC2CC2)N(CC(CC)OCC)C)cc(C)cc(C)c1 N1(C(CC2CCN(C)C2)=O)CCN(C(c2cc(C3(O)COC3)on2)=O)CC1 c1(C(N2CCCN(C(=O)CSC(F)F)C(CO)C2)=O)cnc2c(c1)CCCC2 C12=CC(=NCCC(C(F)(F)F)N1)NC=N2.CCCS(=O)(=O)NC(C)COC N1(C(CNC(C)=O)=O)CC(NC(=O)CSC(C)(C)C)CC(F)(F)C1 N1(C(c2cc(C)n(CCO)n2)=O)CCC(C)(C)CC1.C(=O)CN(C1CCC1)C.N N1(C(C)=O)CCCC2C1CCN2C(=O)CCNC(C1CCC(=O)N1)=O C1(C(N(C(C)C)CCNC(=O)C2CC2)=O)CCCCC1.C(=O)C(Cl)(Cl)Cl c1(CNC(C2CC3CC3N2C)=O)ccccc1-c1ccncc1.c1ccc(Cl)cn1 C1(NC(c2cc(CC)on2)=O)CC2CCC1N2C(=O)CCO.C(=O)C(F)(F)F CC(C)CCC(C(=O)N(C)Cc1cnn(C)c1)NC(C1OC2CCC1C2)=O C(C(=O)N1CCCO1)N(C(C)C)CC1(CS(C)(=O)=O)CCOCC1 C1(C(=O)NC2(C)CCN(C(C3CC4C(C3)C4(F)F)=O)C2)CCc2nnnn2CC1 c1(OCC(=O)NCC(CC)NC(C2CCCS2)=O)cc(C)ccc1Cl C(C(=O)NCCC1(NC(=O)C)CC1)(C(C)C)n1ncc(C)c1.C1CCCOC1 c1(NCC2CC(NC(c3cc(C)nnc3O)=O)C2)nnc2c(c1C#N)CCCC2 Cc1cc(CC(N2CCCC2C2CCN(C(C3(C)CC3)=O)C2)=O)ccc1[N+](=O)[O-] C1(NC(C2C(C)(C)CN(C(c3cc(O)cc(=O)o3)=O)C2)=O)CC2CCC(C1)C2O c1(C(N2C(CCCC)CN(C(=O)C=C(C)CCC)CC2)=O)cccn2cnnc12 C1(O)(C(C)NC(c2ccc(CO)cc2)=O)CCN(C(c2ccoc2Br)=O)CC1 C(C1=CCN(C(c2cnc(C)c(N)c2)=O)CC1)NC(C(C)OCCCCCC)=O c1(CCOC)nsc(N2CCCC2CN(C(=O)CC2CCCC2C)C)n1 C1(n2cc(CSCCNC(c3c(OC)cncn3)=O)nn2)CCCCC1(F)F c1(CC)ccc(F)c(C(N2CC(CC)C(C)C2)=O)c1.C(=O)(C(C)(C)N=[N+]=[N-])N C=C(C)CCC(C(=O)NCC(=O)NC)N(CC(F)F)C(C)C C(=O)(CC1OCCc2ccccc21)NCC1C=CC(NC(C(C)(C)C(F)F)=O)C1 C1(NC(C23OCC(CC)(C2)C3)=O)CC2CC1N(C(c1cc(Cl)ccc1C)=O)C2 c1(C(=O)NCc2c(C(=O)NCC(CC)C#N)con2)ccc(COC)cc1 c1(CC)ccc(N)c(C(=O)NC2CC(NC(=O)C(O)CC)C2)c1 c1(OC)cc(C(N2CCC(C)(C)C2)=O)cnc1O.n1(C(C(=O)N)C)cc(Cl)cn1 C1(NC(=O)CC2CCCC2)CC2CC(C1)CN(C(C1C=CCC1)=O)C2 C1(CC=O)CCC=CCC1.C1(CN(C)C)CCC(C(=O)NCC(C)C2CC2)O1 C(c1cccc(F)c1Cl)=CC(=O)NCc1ccc(CC=C)cc1 c1(C(N2CC(C(C)NC(=O)C(C)(C)C#N)C2)=O)cnn2ccn(C)c12 Cc1cccc2c(C(N3CCC(O)(CN(C)C(c4ccsc4Cl)=O)C3)=O)cnn12 C(CCCCC(=O)NCC(CC(N1CCCC(O)CC1)=O)C1CCC1)OCC C1(CNC(=O)COCCF)CCCC(NC(C23CCC(CC2)C3)=O)C1 n1(CC)nnc(C(N2CCC3CC23C(=O)NCC(F)(F)CC2CC2)=O)c1C C(=O)(N=c1[nH][nH]cc1-c1ccc(F)cc1)c1ccc(OC)cc1OC.C1(=O)CN1 N1(C(c2ccc(C)c(Br)c2)=O)CC2CC(C)N(C(c3cc(C)c(C)o3)=O)C2C1 CC(C)C(C)C(=O)NC(C)CN(C(=O)C=Cc1ccc(I)o1)C c1(OCC)cccc(CNC(C2CN(C(C3CCCCS3)=O)CCO2)=O)c1 N1(C(COCCC)=O)CCN(C(c2cc(C)no2)=O)C(c2cnn(C)c2)C1 n1(CC=O)c(C)cc(O)cc1=O.C(C(F)C(=O)N)N(CC)CC.CC(C)CO c1(CCN(C(c2nncn2C)C(=O)NCc2ccc(F)s2)C)cccnc1 c1(NCc2n(CCC)ccn2)[nH]c(=NC2CC=CC2)nc2scnc12 C1(OC)CC2CC1CN(C(C1CCCN1C(c1[nH]ccc1C1CC1)=O)=O)C2 c1(C=O)ccc2ncn(C)c2n1.N1(C(C=CCOCCOC)=O)CCCC1C.N C1(CNC(C2(CC)COC2)=O)CN(C(=O)C(C)(C)n2ccc(C)n2)CCCO1 Nc1sc2c(c1C(=O)NCC1CC1)CCC2.C(=O)(C(F)(F)c1cscn1)N C12(NC(C(C)n3cccn3)=O)CC3CCC(C1C2)N3C(=O)C(C)(C)C C1(F)(CNC(C(CCSC)NC=O)=O)CCN(C(=O)C(C)CO)CC1 c1(C(N2C3(C(=O)NCCc4cc(C)no4)CC3CC2)=O)ccc(C)c(C#N)c1 C1(CNC(CCc2c(C)ncs2)=O)CCN(C(C23CCCC2C3(F)F)=O)C(C)C1 C1(C=O)CC2C=CC1C21CC1.C1(CC(=O)N(CCC)CC)CN2CCN1CC2.N CCCS(=O)(=O)C(C)C(=O)NCC1CC2CCC1N2C(=O)CCC(F)(F)F N1(C(C(CCOC)(C)C)=O)CC2CCC1C(CNC(=O)CC1(O)CCOC1)C2 CC1CN(C(=O)CC2CSCCS2)CCN1C(c1cc[nH]n1)=O CC1CN(C(=O)C(N)=O)CCC1C(=O)NC(C)C(C)O CC(CC(C)(C)C)C(=O)NC1CCC1NC(c1ccc([N+](=O)[O-])s1)=O C(=O)C(C)=Cn1ccnn1.C(c1ccccc1)=C(CC)C(=O)NCC1CC1C.N CC1(C)OCCOC1CC(N1CC(NC(=O)CC(C(F)F)N2CCOCC2)C1)=O N1(C(C2C(C(C)C)CCC2)=O)CCCN(C(c2cccc3c[nH]nc23)=O)CC1C c1(C(=O)NCC2CC(NC(COCC)=O)C2)ccccc1C1CCCC1 N1(C(c2c(NCC)scn2)=O)CC2CC(C1)C2NC(C1CCCCC1C)=O c1(CC(N2CCN(C(COC)=O)C(CS(C)(=O)=O)C2)=O)c[nH]c2cccc(C)c12 c1(OC)cc(CCNC(=O)CCC2(OC)CCCCC2)ccc1[N+](=O)[O-] c1(C(N(CC(C)NC(C=C(C)C(F)F)=O)C)=O)c[nH]ccc1=O C(=O)(CC(C)C(C)(C)C)N1C(C)C(NC(c2ccc(CO)s2)=O)CCC1 C(=O)(C(CC)CC(C)C)NC(CN(C(C1(CCCC)CCC1)=O)CC)C(C)C C(N=C(NC1CCOCC1)N1CCc2nnc(O)cc2C1)c1c(C)nn(C)c1C N1(C(c2c(C)cns2)=O)CCCN(C(C2(C)COC(=O)C2)=O)CC1C CC(O)(CNC(=O)CC1CC(NC(c2ccn(C(F)F)n2)=O)C1)CCO C1(C(N(C2CCCOC2)CC)=O)CSCCN1c1nnc(C(C)(C)C)o1 N1(C(CC=CCC)=O)CC(O)CC1CNC(c1cn(C2CCOC2)cn1)=O C(CCC(C)C(=O)NCC(CNC(=O)Cc1ccc(Br)nc1)OC)OC N1(C(c2nn(CCCC)c(=O)cc2)=O)CCN(C(=O)C(C)OCC)C2CCCC12 c1(NCC(C2CC2)OC)cc(C#N)ccc1F.c12nc(cn1C)N(C)C2 CC1(C(=O)NCCCC(=O)NCCCCO)CC1(F)F C1(C(=O)NCC(CO)NC(c2cc(Br)co2)=O)CC2(CCCC2)CO1 N1(C(C2CNC(=O)N2)=O)CCC(NC(c2ccc(O)nc2Cl)=O)C(F)C1 C1(CCNC(c2c(CC)ncs2)=O)C(C)CCCN1C(c1ccc(O)nc1Cl)=O N1(C(C2CN(CC)C2)=O)CC2CC2(C(=O)N(CCC(Cl)Cl)CC)C1 N1(C(c2n(CCC)ncc2)=O)CCCC(C)(C)C1C(=O)N(C)CCC1CCCO1 C1(O)(C(C)NC(=O)CC2(C)CCCCC2)CCN(C(=O)C(O)c2ccsc2)CC1 C1CN(C(c2cnco2)=O)CC2(CCC2)C1.c1(CC(=O)N)ccc(C(F)(F)F)nc1 N1(C(=O)Nc2cccc(C)c2)CC2(CCC(NC(c3cnc(O)c(Cl)c3)=O)C2)C1 S(=O)(=O)(CCC(=O)N1CCC(CN(C)C(C2CCCS(=O)(=O)C2)=O)C1)NC C(c1ccc(F)c(C)c1)=CC(=O)NCc1c(OC)cccc1.c1ccccc1.C CC(C)(C)C(C#N)C(=O)N1CCC2(CC1)CC2NC(=O)CC.[SH](C)(=O)=O.N CN1CCC(C2CCCN(CC3CC4(CCCO4)C3)C2)CC1 C1(C(NON2CCC(C)C2)=O)CCN(C(=O)C(C)Cc2cnc[nH]2)C1(C)C C=CCC(C(=O)N1CC(C(=O)N(C2(C(=O)OC)CC2)C)C(C)C1)OC Cc1cc(N2CC(NC(C3CCCN(C)C3)=O)CC3(CC3)C2)n2ncnc2n1 C1(C2CCN(C(c3cc(Cl)cnn3)=O)CC2)(NC(c2ccc(C)c(O)c2)=O)CC1 C(C)(CCC(F)(F)F)NC(CCC1CCC(NC(C(CSC)OC)=O)C1)=O N1(C(C(CCC)NC(=O)CCc2cnoc2)=O)CCCCC(COC)C1 C1(NC(c2scc(OC)c2)=O)CCCCN(C(c2[nH]nnc2C(F)F)=O)C1 c1(C(=O)NCc2c(C(=O)NC3CC(CCC)C3)scc2)cc(C)on1.O c1(NC)nc(C(=O)NCC2CCCCC2)ccc1[N+](=O)[O-].C(=O)C(C)(F)F.C N1(C(C(=O)N)(C)C)CCN(C)CC1.C1(CNC(C2C(CC)C2)=O)CCC1 CCCCC(C)CCC(=O)N1CCC(NC(=O)C(C(C)C)NC(=O)OC)CC1 C1(NC(c2c(C)noc2C(F)(F)F)=O)CCC2CN(c3ncns3)CC2C1 C1(NC(C2CCC(CC)O2)=O)CCN(C(=O)C=C=C(C)C)CC1C C12(NC(c3cccc(C)c3C)=O)COCCC1CN(C(=O)CC(=O)N(C)C)C2 N1(C(C(C)SC)=O)CCC2(CCC(CNC(=O)CC3CCOCC3)O2)CC1 N1(C(c2c(C#C)c[nH]n2)=O)CC(C(=O)NCCNC2CC2)C2(CCC2)C1.C C(=O)C(F)(F)F.C1(C=O)(C(=O)NCC)CC1.C(=O)C.C(C)C.C CC(CC(=O)NC1CCCN(C(c2ccc(N)cc2C(F)(F)F)=O)C1)C(F)(F)F c1(C(=O)NCCC(C(C)C)NC(C2CCCSS2)=O)ccc(C2CC2)c(Cl)c1 c1(CC(N2CC3C(C(N4C(CCOC)CCCC4)=O)C3C2)=O)cc(Br)ccc1Br CC1(F)CCC(C(=O)OCc2nc(-c3cccc(C(F)F)c3)no2)CC1 C1(CN(C)C(c2cscc2F)=O)CN(C(c2cscc2C(N)=O)=O)CCO1 O(NC(=O)CC1CCCN1C(c1sccc1COC(C)=O)=O)CCCC#C N1(C(C2CCC(=O)O2)=O)CC(NC(C2CC2F)=O)C2(CC2)C1 c1(C(=O)NC(C(CO)NC(c2cnc(C)o2)=O)C)ccccc1S(=O)C(F)(F)F N1(C(c2c(C#N)scc2)=O)CCCN(CCNC(C2CC(C3CC3)C2)=O)CC1 C1(F)(CNC(=O)C(C2CCC2)C2CCC2)CCN(C(C23COCC2C3)=O)C1 c1(CC(C)C)nc2cccc(C(=O)N(CC(O)CO)CC(C)(C)C)c2[nH]1 N1(C(Cc2c(C)cc(Br)cc2)=O)CCC2C(CCN2C(c2cnco2)=O)C1 CCCCCCCCCCCCN(C)CCSc1cn(C(C)CC)nn1 C1(C(N(C2CCCC2O)C)=O)CC1C1CN(C(=O)CC2(C)CCCCC2)C1 c1(N(C2CNCC2F)C2(c3ncc(C)c(Br)c3)CC2)ncnc2ncc(Br)cc12 c1(C(=O)NC(C2CCCN(C(c3ccccn3)=O)C2)C)cnc2ccccc2c1 c1(NC(=O)CC2CCN(Cc3ccc(Br)[nH]3)C2)nccc(Br)c1O C1(CCNC(C2NC(=O)OC2)=O)CCCN(C(C23CCC(C2)C3)=O)C1 c1(C(N(C2CN(C(=O)C(O)C3CC3)C2)C)=O)csc2nccn12 C(=O)(C(C)CC(C)C(C)=O)OC.C12(CO)CCN(C1)C2.c1ccccc1 N1(C(CC(C)SC)=O)CCc2[nH]nc(CNC(=O)C(c3ccc(C)cc3)C)c2C1 CC(C)CC(C)C(=O)N1CC2CC2(CNC(c2cc(F)cnc2O)=O)C1 C1(NC(C=C2CCC(C)C2)=O)CCCN(C(c2csc(Cl)c2)=O)CC1 C1(NC(C(C)C2CC2)=O)CCN(C(=O)Cn2cc(S(N)(=O)=O)cn2)CC1(C)C Cc1c(CC(=O)N(CC(C)(C)NC(=O)Cn2ccnc2C)C)cnn1C c1(CC)n[nH]c(CC)c1CC(=O)NCC1CC(NC(c2ccccn2)=O)C1 C1(NC(CNC(C)=O)=O)CC(=O)N(CN)C1.C1CC2CC2C1.c1ccco1 c1(N(C2CC3CNC2C3)C(c2scc(C)c2C)=O)ccc(F)c(C(F)F)c1 c1(C(=O)NCCN(C(CCCC(C)=O)=O)CC(C)O)cc2cc(Cl)ccn2n1 c1(C(=O)NCCC2OCCN(C(C(CC=C)CC)=O)C2)cc(Cl)cc2c1CCC2 O=C(CCC(=O)N(C1CCc2nc(Br)sc2C1)C1CC1)CCC(=O)c1cccs1 C1(C)(CC)CCCN(C(=O)CCCC(C)NC(=O)C2=C(Cl)CCC2)CC1 CC(CC(=O)N1CCC(c2cc[nH]n2)C1)C(C)(C)NC(C1CC(F)(F)C1)=O C(=O)(C(F)CCC(C)(C)C)N1C(CCC)CN(C(=O)CCc2cnoc2)CC1 C123CN(CC1CCO2)C3=O.c1(CNC(COC)=O)nn(C)c(Cl)c1Cl C1(NC(=O)C(c2ccc(Br)cc2)O)COCCN(C(C2CC(O)C2)=O)C1 C(CCC1CC1)(C(=O)NC1(C(=O)NC)CC1)NC(C(C=C)O)=O N1(C(c2cn(CC)nn2)=O)CC2(C1)CN(C)C2.CC(C)CC1(C(=O)N)CC1 c1(C(=O)NCc2csc(C)n2)ccc([N+](=O)[O-])o1.C1(C=O)CC1(Cl)Cl.N c1(C(C)C)cncc(C(=O)NCC(O)CCNC(=O)C(C)CC2CC2)c1 c1(NC2C3CCC(F)(F)C2C3)nc2cc[nH]c2c(=NC2CC3CCCCN3C2)[nH]1 Cc1csc(C(=O)NC2CCOCC2NC(=O)C)c1Cl.c1(C(=O)N)ccccn1 N1(C(c2c(SC(C)C)cccc2)=O)CCC2(CCC2CNC(=O)CCF)CC1 C1(CC(=O)NC(C2(C=O)CC2)C)CCCN(C)C1.C1(C)(CC)CC1(F)F S(=O)(=O)(c1cc2c(cc1)CCC2)N(CC(=O)OCc1ccccc1)CCC.O N1(C(c2c(C)nc(O)s2)=O)CCC(C)N(C(c2cocn2)=O)CC1 C(=O)(C(O)CC(C)(C)C)NC1C(O)CCN(C(c2ncc(C)cn2)=O)C1 C(=O)(CCCCC(C)CC)NCC(C)N(C(CC(CCC)(C)O)=O)C C12(NC(c3c(C)nc(O)s3)=O)CCCC1CN(C(C1CC1c1ccccc1)=O)C2 N1(C(COCCC)=O)CCC(CC(=O)N(CC(n2ccnc2)C)C)CC1 CC1C(C)N(C(c2nscc2Br)C(=O)NCC(F)F)CCS1=O c1(CC(=O)N(C(C2(F)CN(C)C2)=O)C)ccc(-c2cn(C3CCC3)nn2)cc1 N1(C(C2N(C)CCOC2)=O)CC=C(CC(=O)NC(C(N)=O)C(C)(C)C)CC1 CCCC(C)(O)CC(=O)N(C1CC(C#N)C1)CC(=O)N(CCC(F)(F)F)C CC#CCC(C(=O)NC(=O)CN1CCCC1=O)NC(=O)C(CCCC)N1CCCC1 N1(C(c2c(CC)noc2)=O)CC2CCN(C(C3CC(O)(C(F)F)C3)=O)CC12 c1(C(N2CCCC(CN(C)Cc3c(C)n[nH]c3C)C2)=O)c(Cl)cccc1I c1(C(=O)NC(CC(C)NC(C2(C)CC2(F)F)=O)C)ccc(C#N)cc1 c1(C(=O)NC2C(CNC(C(C)NC(N)=O)=O)C2)cc2n(n1)CCCN2 C1(CNC(c2cccnc2S)=O)CC(C(=O)NCC2CCCSC2)=NO1 CC(C)CCCC(=O)N1CCN(C(=O)CNC(C2CNc3ncnn3C2)=O)CC1 c1(C(=O)NC(CC=C)CNC(=O)C=CCCC)ccc2ncccc2c1Br CC1(C(=O)Nc2nccs2)CCCN1C(C1CCC(C(F)(F)F)CC1)=O C1(NC(C2C(CCOC)C2)=O)CC2CCC1CN(C(=O)CCCN=[N+]=[N-])C2 c1(C(C)=O)cc(C(=O)NCC2(NC(=O)C(F)C3CCOC3)CC2)no1 C12(NC(C(c3ccc(C)cn3)(F)F)=O)CCCC1CN(C(=O)Cn1ccnn1)C2 c1(CC)cc(=NCC2(F)CC(NC(=O)C(C)CSC(F)(F)F)C2)[nH]c(C)n1 CCCCCC(C(=O)N1CCN(C(=O)CCc2cccs2)CC2(CC2)C1)C(C)C N1(CC)C(C)CN(C(=O)CC2CC3(C2)CN(C(=O)C(C)CC(F)F)C3)CC1C CCC(C)CCCCC(=O)NC1(C(N2CCCC(C#N)C2)=O)CC1C C(C)(CCC(C)C)NC(N(c1ccccc1)CCCC)=O CC(C)C(O)CC(=O)N1CCC(C(F)F)(CNC(c2cn(C)nn2)=O)C1 C1(CCC(=O)NC2(CNC(CCc3n(C)ncn3)=O)CCOC2)CCCCCC1 c1(C(=O)NCC(C)(C)OCCNC(c2cnco2)=O)[nH]cc2c1CCC2 c1(OC)ccc(C(CO)NC(C2CCN(C(c3nc(C)sc3C)=O)CC2)=O)cc1 C1(CN(C(C(C2CCCCC2)C)=O)C)CCCCN1C(=O)CCC1(C)CC1(F)F N1(C(C2CC(C(C)=O)C2(C)C)=O)CCC(C)CC1C.c1(CC(=O)N)cn(C)nn1 C12(C(N3CC(NC(c4cc(OC)ns4)=O)C(C)C3)=O)CCC(C)(CO1)C2 c1(NC(=O)NC)ccc(-c2noc(C3CCN(C(=O)CC(=O)O)CC3)n2)cc1 c1(CCC(=O)N(C(C)CNC(=O)C(C)C)CC)nc(C2CC2)no1 C1CC2CCCC2C1.C1(CC(=O)N(C)CCOCCC(=O)N)CCC(=O)N1.C C1(C(=O)NC(C=CC(=O)NC2CC(OCC)C2)C)CN(C)C(=O)N1 C1(C(C)C)N(C(C2CC(C)(F)C2)=O)CC12CCN(C(=O)C(C)C1CCOC1)CC2 c1(OC)ccc(F)c(C(N2CCC(CC)C2)=O)c1Cl.N1(CC(=O)N)CCC(C)C1 C1(CNC(c2cccc(CC)c2)=O)CCN(C(C2(C)CCCCC2)=O)CC1C C1(C(=O)NC2(C)CCC(C)C2)CN(C(=O)CC2CCC(C)(C)O2)CCC1(C)C C1(C(N2C(C3CCN(C(C(C)SC(C)C)=O)C3)CCC2)=O)CC2CCCC(C1)C2 c1(CN2CC(CC(=O)OC)(OC)C2)cc(Br)c(O)c(Br)c1 N1(C(=O)CN(C(C2CCC3CC23)=O)CC2CC2)CC2(CC(O)C2)C1 CC1(C)CCCN1C(=O)Cn1cc(C2CC2)nn1.C1(CC(F)F)(C=O)CCC1 c1(C(C)NC(C2(F)CCN(C(=O)CC3(C=O)CCCO3)C2)=O)ncccc1F c1(C(N2CC3CC3C2)=O)sc(C)c(C)c1C.C(=O)(CCC=O)NCCCOC.N c1(C(=O)NC(CCCNC(C2(CC#C)CC2)=O)C)cncc(Cl)c1Cl c1(C(N2C3CC(C2)C3)=O)c[nH]nc1[N+](=O)[O-].c1(C(=O)N)ncc(C(F)F)cn1 CC1CN(C)C(=O)CN1C(=O)CC1CC1CNC(c1cccc(O)c1F)=O C=CCCCC(=O)NCC1CCCC(CNC(=O)CCc2cc(Cl)no2)C1 C1(N(C(c2ccc(C)o2)=O)CCF)CCCN(C(C2(C)CC2(C)C)=O)C1 N#Cc1cccc(NCC(=O)N)c1.C1C2CN(C(=O)CN3CCC(F)C3)CC12.C C=CCCCCCC(=O)NCC1CCCN(C(=O)C(C(C)C)SC)C1 C1(C(N2C(CNC(C(CC)CC)=O)CCCC2)=O)CCC(C)(C)CO1 N1(C(C(C)OCCOCC)=O)CCCCC1C1CC1.c1(C=O)ccn[nH]1.N N(C)(C1CCc2ccc(Cl)cc21)CC1OCCN(C(C2CN(C)C(=O)C2)=O)C1 C1(CC)CN(C(c2cc(C)cc(C)c2)C(=O)NC2(C)CC2)CC(C)S1=O c1(OC)ccc(CN2CC3CN(C(c4cnc(Br)s4)=O)CC23)nc1Br N1(C(c2onc(CC)c2C)=O)CC(NC(c2ccc(Cl)o2)=O)CC12CCOC2 c1(C(N2CCC(OCCNC(=O)CO)C2)=O)cc(-c2ccccc2)cc(Cl)c1O N1(C(c2c(C)ncs2)=O)CC2CCC1CN2C(c1ccc(COC(C)C)cc1)=O N1(C(C(C)=C2CC2)=O)CCCC2CN(C(=O)Cn3nnnc3C(C)C)CC12 c1(OC)ccc(Cl)c2c1CCCC2N(C)C(N1CC2OCCOC2C1)=O c1(C(N(CC(N2C(C(N(C)C)=O)C3CC3C2)=O)C)=O)cnc2ccccn12 C1(C=O)CCc2nc[nH]c2C1.N1(CC)C(=O)CCC1CC(=O)NC(C)(C)CC.N C1(NC(CCc2ncc(C)[nH]2)=O)CN(C(C2CCNC2=O)=O)C2(CCCCC2)C1 CN=C(NCC1(F)CCC(c2ccccc2)CC1)N1CCC(O)C(C)(C)C1 N1(C(c2ccc(NCCOC)cc2)=O)CC2CCN(C(=O)C=CBr)CC2C1 C1(C)(CNC(CC2CN(C)C2)=O)CCCN(C(c2ccc(N)c(Br)n2)=O)C1 C1(C)(CNC(C(CC)(C)CC)=O)COCCN(C(=O)C(c2ccccc2F)C)C1 CC(C(=O)N1CCCC(CCNC(C2CN3CCN2CC3)=O)C1)C1=CCCC1 CN1CCC(C#N)(C(=O)NCC(C)(C2CC2)NC(=O)CCS(C)=O)CC1 Cn1nc(C(=O)NCC2CCCC2NC(=O)C(F)F)cc1C1CC1 CC1C(C(=O)NCc2nocc2C(=O)NCCC2C=CCC2)CCN1C CCC(CC(=O)N1CCC(CO)(CNC(=O)CO)C1)C(C)C.CCCN(C)C N1(c2c(C#N)cccn2)CC2CC(NC(c3cccnn3)=O)CC2C1 C(=O)(CC(C)CC(C)C)NCC1C(NC(c2c(CC)n(C)cc2)=O)CCC1 C(CN=c1cc[nH]cc1S(=O)(=O)N1CCN(C)CC1)(C(C)C)NCC(C)C C(CC1=CCN(C(c2ccnnc2)=O)CC1)NC(c1cc(CC)cc(Cl)c1)=O C1(CN=[N+]=[N-])CN(C(C2CCCCN2C(=O)C#CC2CC2)=O)CCO1 O=C(NOCC=CCl)C1=CC2(CCN(C(=O)C3=NOCC3)C2)C1 c1(C(N2CCC(C(C)(C)NC(=O)CC)C2)=O)ccc2c(n1)CCCC2.C(N)=O.N CC(C)(C)C(O)CC(=O)NC1(C)CC(NC(=O)CCCN2CCCCC2)C1 N1(C(CC2CCCN(C(CSCC(=O)OC)=O)CC2)=O)CCC2(CC1)CN(C)C2 CC1(C)CCOC(CC(=O)NCC2C=CCN2C(=O)C2=NOCC2)C1 C1(O)(CNC(C(C)OC)=O)CCN(C(c2cccc(-c3cnn(C)c3)n2)=O)C1 N1(C(CCn2c(C)cc(C)n2)=O)CC(NC(C2CC3(CCC3O)C2)=O)C(C)(C)C1 Cc1ccc(C(=O)NC(CC(C)C)C(=O)NCCN2CCCCC2)c(C)c1 C(=O)(C1OCCc2ccccc21)NC(CCNC(Cn1c(C)cc(=O)cc1)=O)C c1(COC(c2cc(C)nc(C)c2)=O)ccc(N)cc1[N+](=O)[O-] N1(C(c2ccc3ocnc3n2)=O)CC2C3COCC3C2C1 C1(NC(C(C2CN(C(=O)CCC3CC3)C2)OC)=O)CCN(C(C)C)CC1 Cc1nc(C2(NC(=O)CC=CCNC(=O)C(C)C#N)CC2)n[nH]1 c1(CNC(CC2(NC(c3cncc(OC)c3)=O)CC2)=O)ccc(C)cc1C C=C(C)CC(C)C(=O)N1CC2C(CNC(=O)CCc3cnc(C4CC4)o3)C2C1 N1(C(CSCCCC)=O)CCC(CCCNC(C2CCCN2C(=O)NC)=O)CC1 N1(C)CCc2nc(Cl)[nH]c2C1.c1(COCC)nc(OCC)cc(N2CCCC2)n1 c1(C(=O)NCCC2(C)CCCO2)cc(CNC(c2ccc(O)nn2)=O)ccn1 c1(CNC(Cc2nc(SC)sc2)=O)cc2ccccc2nc1N1CCC1 N1(C(c2ccc(OC)o2)=O)CCC2(CC1)CN(C(=O)CC1(OC)CC1)CC2C n1(CCN(C(=O)Nc2ccc(OCC)c(O)c2)CC)cnc2[nH]ccc2c1=O C1(C(CNC(C(CC)C)=O)(C)C)CCCCN1C(=O)Cc1ccc(C(C)C)cc1 n1(CC(C)(C)CO)nc(-c2cncnc2)nc1-c1cccc(C2(C)CC2)c1 c1(C(N2CCC(C(F)(F)F)C2)=O)cccc(C)c1C.c1(CC)cc(C(=O)N)n[nH]1 Cc1ccccc1CC(C)C(=O)N1CC(NC(=O)C(O)CN(C)C)C1 C(=O)(C(O)CC(F)(F)F)N1CCCC(NC(c2cc(SC)c(F)cc2)=O)CC1 C(=O)(C(C)C(C)(C)C)NCCC1CC(NC(C(C#C)(C)C)=O)C1 S(=O)(=O)(c1ccccc1)N(CCCCNC(C(C)C)=O)C.C(C)(C)C.C=O.N N1(C(CCCCSC)=O)CCC2CCN(C(C3COC4CCCCC34)=O)C2C1 c1(Cn2c(-c3c(Cl)cnc(Cl)c3)nc(CCCO)n2)cccc2c1CCCC2 C1(NC(C2CC(C)(F)C2)=O)CC2CCC1CC2NC(c1cnc(O)s1)=O N1(C(c2cn(CCC)nc2C)=O)CC2(CCC(CNC(=O)CC(C)CCC)O2)C1 N1(C(C=CC(=O)NCCCCCC)=O)CCN(C(C2CC2[N+](=O)[O-])=O)CC1 C1(c2ccccc2)CCCN(N2CCOC(c3ncno3)C2)C1 c1(C(N2CCOCC2)=O)c(C)cc(Cl)cc1C.C1(C(=O)OC)CC1C(=O)N.C C1(NC(C23CC(CN(C(C(CC=C)C)=O)C2)C3)=O)CC1C1CCCCC1 c1(C(=O)NC2CN(C(CC3CC(=C)C3)=O)CC2O)cc(Br)ccc1C Cc1cn2cc(C(=O)NNC(N)=O)ccc2n1.C1CC(C(C)C)CCCn2cc(nn2)C1 c1(CN(C)C(c2ccc(C)cn2)=O)ccc(Br)cc1.c1(C(=O)N)cc(O)no1 c1(CN2CCC(N(C(c3sncc3C)=O)CC)C2)ccc(N2CCC(O)C2)cc1 CC1CC(C(=O)NC(C2(O)CCCCC2)C(N2CCC(C)(C)C2)=O)CCO1 N1(C(c2ncc(Cl)cc2F)C)CC2=C(C1)CN(CCC1CCOC(C)(C)C1)C2 C(=O)(CC(C)C(C)C(C)C)NC1CN(c2ncc(C(=O)OCC)c(C)n2)C(C)C1 c1(C(=O)NC2CN(C(C3C(F)(C(=O)OC)C3)=O)CC2F)ccc(Cl)cc1F c1(CNC(C#CCNC(C(C=C)O)=O)=O)cncc(OC)n1 c1(OCC(C)C)ccccc1C(=O)NCC1(O)CC(NC(=O)C=CBr)C1 c1(CN2CCCC(NC(Cc3ncc(C)s3)=O)C2)c(F)cc(C(F)(F)F)cc1F C1(C(=O)NC2CCN(C(c3[nH]cc(C#N)c3)=O)C2)CC2(CCOC2)C1 C1(C)(C(=O)NC(C(C)C)CNC(c2cnc(Cl)s2)=O)CCC(=O)CC1 C1(CNC(C(CC)n2ccnc2)=O)CN(C(=O)C(C2CC2)SC)CC(C)(C)C1 n1(CC)cc(NC(C2CC(CCNC(c3ccccn3)=O)C2)=O)ccc1=O.O N1(C(C2N(C(C(CC)C(F)(F)F)=O)CC3CC32)=O)CCCC2(CCOC2)C1 C1(C(F)(F)F)(C=O)CCOCC1.C(=O)(C(F)(F)c1nccn1C)N(CC)CC N1(C(c2c(C)nc(C)[nH]2)=O)CCCC2CN(C(C3CCCN3C=O)=O)CC12 c1(C(N(CC(CNC(C(COC)O)=O)C)C)=O)cccc2c1ncn2C c1(C(=O)NCC2N(C(C3(CC=C)CCOC3)=O)CCC2)sccc1C#N C1(OC)CN(C(=O)CC2CCC2(C)C)CC1NC(c1cn[nH]c1)=O N=c1ccc(C(=O)NCCC2CC(C(N3CC(O)CC3C(F)F)=O)C2)n[nH]1 c1(NCc2ccc(OC)c(Br)c2)ncccc1[SH](=O)=O.C1(C(C)N)CC(F)(F)C1 c1(C(N(C)CC2(NC(=O)CCS)CC2)=O)cccc2sccc12.C1CCCC1 C1(CNC(c2n[nH]c(C)c2O)=O)CC(C)(C)CCC1NC(c1cc(F)c[nH]1)=O CC(CNC(=O)CC(C)O)C(=O)NC1CCN(CCF)C1 c1(C(N2C3C(CNC(C4CCC4)=O)C(C3)C2)=O)noc2c1CCCC2 N1(C(CS(CC)=O)=O)CCOCC(C(=O)Nc2cccc(OCF)c2)C1 c1(CC(=O)NC2CCN(C(C3CSCN3C(C)=O)=O)CC2)ncn(C)c1C.C c1(C(=O)N)cncs1.C1(NC(=O)C=CC(F)(F)F)COCC1C.C1CC1 C(C(=O)N1CCSCC(C)C1)(C(C)(C)O)NC(Cn1c(C)ccn1)=O c1(OCC=C)ccc(C(=O)NC2COCCC2NC(C2CC2C)=O)cc1O c1(C(=O)NC2(CNC(C3C(C)OC(=O)N3)=O)CCOC2)cccc(F)c1Cl C1(CCNC(C2(CC)CCC(=O)N2)=O)CCCN(C(=O)O)CC1.C(C)(C)C N1(C(CSc2nc(C)[nH]n2)=O)CCC(C)(C)C(NC(=O)Cc2cnccn2)C1 c1(OC)cc(C(F)CNC2CC(c3nc(C(C)C)no3)C23CCC3)ccc1Cl c1(C(C)C)cnc(C(C)(C)C)s1.C12CCCC1CNC2=O N1(C(C2CCN(C(CC(CC)OC)=O)C2(C)C)=O)CC(C)CCCC1C C1C(C)(C)C1(F)F.C(C)(C=O)(N(C(CN(C(C(C)C)=O)C)=O)C)C1CC1.N c1(C(=O)NC(C2CCCN(CC(=O)N3CCC3)C2)C)cnc2c(c1)nnn2C c1(N(C(=O)C(C)Cc2cnn(C)c2)CC(=O)NC)c(C)cccc1Cl c1(C(=O)NC2C(OC)CN(C(=O)CCC=CC(C)C)C2)cn(C)c(=O)n1C O=NN1CCCC1C(=O)NC(CNC(=O)C)CO.c1(CC)cccc(F)c1.O c1(C(N2C(CN(C(C=CC)=O)C)CCCC2)=O)c(Cl)cccc1[N+](=O)[O-] N1(C(C2CCC2)=O)CCN(C2CCCN(C(C34CCCC(CO3)C4)=O)C2)C(=O)C1 n1(CCCC)ccc(C(=O)NCC(C)C2CC2)n1.C1(CC(=O)N)CCC(C)C1 C1(C2(O)CCOCC2)(CNCC2(C#N)CCC2)CCC1 c1(NC(CN(C)C(c2ccc(C#N)o2)=O)=O)cnc2ccnn2c1 c1(OC)cc(C(N2CCCC(N(C)C(C3CC3C)=O)C2)=O)c2c(c1)OCC(=O)N2 C1(C(N2CCN(C)C(CNC(=O)CC3CCCC3O)C2)=O)CC2(CCOCC2)C1 c1(NC(=O)OC(COC)C)cnc2onc(C3CCCC3)c2c1 c1(C(N(C)CC2CCN(C(C(CC)(C)COC)=O)C2)=O)cc(Cl)c2n[nH]cc2c1 N1(C(c2n(C)ccc2)=O)CCCC(C(=O)NC2C=CC(O)C2O)CC1 c1(C(=O)NC2CCC(NC(C(C(C)C)OC)=O)C2)c(C)cccc1Cl c1(C(=O)NCC2N(C(C3(C#N)CCCO3)=O)CC2)ccc2c(Br)cncc2c1 CCC(CC)C(C(=O)NC(C)(C)C)N(C(c1cc(C)co1)Cc1ccccc1)C C(=O)(C(C)(C)CCn1cc(CC(C)(C)C(=O)O)nn1)NC(C)CC1CC1 C1(CO)CCC(C(N2CCOC(CO)C2)=O)CC1.C12CC1C(=O)NC2C.CC N1(C(C(C2CC2)SC)=O)CC2CC1CN(C(c1ccn(C)c(=O)c1)=O)C2 CCCC(C)(O)CNC(=O)CC(C)CNC(=O)CCc1ccccc1 C(C(C)(C)C(=O)NCc1ccccn1)NC(c1c(C)cns1)=O c1(C(N2CCCC(C(C(=O)N(CCC)C)C)C2)=O)ccc(C#N)cc1C c1(CC)cc(F)c(NC(c2ccnc(C)c2)=O)c(F)c1.c1(C=O)ccsc1Cl.N c1(SC)nc(O)nc(C)c1C(=O)NCC1(F)CCN(C(=O)C)C1.C1CC1 CC1CC(NCC2CCC2(F)F)CC(C(F)(F)F)C1 C(C)(CCC(=O)NC1COCC1NC(=O)CSc1cn[nH]c1)OCC N=c1nc2cc(C(=O)NC3CC3NC(=O)C3=CCCSC3)ccn2[nH]1 c1(C(C(=O)NCCC(C)(C)NC(c2ccc(=N)[nH]n2)=O)O)ccccc1Br C(C(C)(CC)C(=O)NC(CC1CC1)C1CC1)NC(C=C(C)C(C)C)=O CC(C)CC(C)(O)C(=O)N(C)CC1CCC(CNC(c2nccnc2N)=O)CC1 c1(C(N2C(CN(C(=O)CCO)C)COCC2)=O)cc(N)cc(F)c1.C1CCC1 CN1CC(CC(=O)NCC(c2ccccc2)NC(c2ccncc2N)=O)C(O)C1 CC#CCCCC(=O)NCC1(F)CCN(C(=O)C(n2ccc(C3CC3)n2)C)C1 C1(CNC(C2(C)CCCN(C(C(C)SC)=O)C2)=O)CCc2ccccc2O1 Cc1ccc(C(=O)N(CC(C)(C)NC(c2cnc(-c3cccnc3)s2)=O)C)nc1 C12(CC=O)CNC(=O)C(C1)C2.CC1CN(C(c2cn(C)nc2CCC)=O)CC1 Cc1cccc2c(CCNC(C3CCC(N4CCN(C)CC4)CC3)=O)cccc12 C1(C(=O)NC(C(=O)N(C2(C#C)CC2)C)CC2CCC2)CCCC(C)(C)C1 CCCC(C(=O)NCCC1(O)CCCC1)NC(=O)C(C)(C)n1cncn1 N1(C(C(OC)OC)=O)CC2(CC2)CC1C(=O)NC1COCC1CO C(=O)(C1c2c[nH]nc2CN1C(c1cn(C)nn1)=O)N(CC)Cc1ccon1 C1(N(C(C(C)OCCCC)=O)C)CN(C(c2cc(O)nc(O)n2)=O)CC1(C)C C#CC1(NC(C2C(C)CCN2C(=O)Cc2ccc(F)cc2)=O)CCC(C)CC1 c1(OCC)ccc(CNC(=O)NCc2[nH]nc3c2COC3)cc1Cl c1(OCCNCCC)ccc(F)cc1[N+](=O)[O-].CCCNC=O.C(C)(C)C Cc1c(Cl)cnn1CC(=O)N(CCC)C(C)C.C(=O)(C(C)(C)C1CCCCO1)N C(CC(C)(C)NC(c1csc(=N)[nH]1)=O)=CC(=O)NC(C)CN1CCCC1 N1(C(C#CC(=O)N(C)C)=O)CCC(NC(=O)CC2CC=CC2)C(O)C1 N1(C(c2snnc2C2CC2)=O)CC2C(C1)N2C(=O)C=Cc1ccsc1 C1(C(=O)NCCCCC)CC2CC1CN(C(c1ccnc(C)n1)=O)C2 N1(C(C2(CC)CCCO2)=O)CC(NC(c2cnc3n2CCOC3)=O)C(C2CC2)C1 C1(C2N(C(CC)=O)CCC2)CCN(c2nccc(OC)n2)CC1 C12(CCC1)C(=O)N2.C(=O)(CCNC=O)N(CC(=O)N(C)C)CC#C C1(C(N(CC(C)(C)NC(c2c(CC)[nH]nn2)=O)C)=O)CN2CCCC2CO1.C c1(C(N2CC(NC(c3cc(C)n(C)c3)=O)CC(OC)C2)=O)ccc2ccoc2c1 C(=O)(C(C)CC(C)CC(C)C)N1CC(O)(C(C)NC(c2ccc(OC)cn2)=O)C1 c1(OC(C)C)ccc(CC(N2CCCC2CNC(=O)CCCC#N)=O)cc1 Cn1cc(Br)c(-c2cn(C3COCC3NC(=O)Cc3csc(C4CC4)n3)nn2)n1 c1(C(=O)NCC(C)CN(C)C(C2(C)CCC(=O)N2)=O)cc2sc(Cl)cc2s1 n1(CC)cc(Cl)cc1C(=O)NCC(C)N(C(=O)Cc1cncc(O)c1)C N1(CC)CC2CCCCC2(C(=O)OC(CCCCN)C(=O)NC)C1 c1(C(N2CC(OC)CC2)=O)ccc2nc(Cl)nn2c1.C1(C=O)CN(C(N)=O)C1.N C(N=c1[nH]cnc(Cl)c1CC)c1ccc(CNC(C(C)OCC)=O)c(F)c1 C1(C(C)NC(=O)C(C)(C)C2CCCC2)CCN(C(=O)CC2CC3CC3C2)C1 N1(c2nc(C(C)=O)c(C)s2)CCC(CNC(=O)CC2CC3CCC2C3)C(C)C1 c1(CN2C(C)(C(N(CC)CC3CCC3)=O)CC2)ccc(F)c(Br)c1 c1(OC)cccc(C(=O)NC2CC2C(=O)Nc2cc[nH]c2)c1 CCC(C)C(O)C(=O)N1CC(C)(NC(c2c[nH]c(=N)c(C)c2)=O)C1 c1(C(N2CC3CCN(C(CC(C=C)(C)C)=O)C3C2)=O)ccc2c(c1)NC(=O)CS2 c1(CC(=O)NC(CN(C(c2cncc(C(C)C)c2)=O)C)C)cc(Cl)cc(Cl)c1 C1(NC(CC2C(C)CCO2)=O)CCS(=O)(=O)C12CN(C(c1cnn(C)c1Cl)=O)C2 Cc1nc(C(=O)NCC2(F)CCC2)c(C)o1.c1(C=O)c[nH]nc1C1CCCO1 N(C(=NC)N1CCC(NC(N)=O)C1)CC(c1c(OC)cccc1)(C)C CC1CCC(C(=O)NCC2(CNC(=O)C(C)(C)n3cncn3)CCCC2)O1 CC1(CC(=O)NC2(CCC(=O)NC3CC(=O)NC3=O)CCC2)CCCCC1 Cn1ccc(C(N2CCN(C(c3ccc(=O)n(C)n3)=O)CC2C(F)F)=O)cc1=O CCCN=C(NCC(CC(C)C)OC(F)F)N1CCCC(C(=O)OC(C)(C)C)C1 c1(C(N2CCC(NC(Cc3cc(CC)no3)=O)C(C)C2)=O)ccnc2ncnn12 N1(C(CN(C(C)=O)C)=O)CCN(C(=O)C)CC1.n1(C2(C(=O)N)CC2)cccc1 CC1(C)CCC(C(=O)NC2CC(NC(=O)Cc3cc(Cl)ccc3Cl)C2)CO1 N1(N(CCCN(C(=O)CCc2ccccc2)C)C)CCN(c2nnc(O)s2)CC1 CC1(C(=O)N2CC(F)(CNC(C3CCCCO3)=O)C2)COc2ccccc21 Cc1ccc(CC(N2CC(NC(=O)CSc3nnc(S)s3)CC2C)=O)cc1C C(c1ccc(O)c(C(F)(F)F)c1)=CC(=O)N.C(C)(CC)N(CCC=C)CC c1(CNC2C(C(=O)Nc3n(CC)ncc3)C2)ccc(OC)nc1Br c1(C(=O)NC(C)CN(C)C(C2CC2Br)=O)cnn(CCF)c1 C(=O)(C1=CCCCC1C)N1CC(C(C)NC(c2ccc(CCC=C)cc2)=O)C1 Cc1cc2[nH]c(C(N3CC4CC4(CNC(C4(C)CCC4)=O)C3)=O)cc2o1 C1(C(F)F)(OC)CCN(C(c2ccnc(C)c2)C(=O)NC2CC2)C1 C1(C(=O)OC(C)C(N2CCSC2C(F)(F)F)=O)CCC(C)C1 C=C=CC(C)C(=O)NCC1C=CC(NC(=O)C=C2CCCC2)C1 C1(C(=O)NC2CN(C)C(=O)C2)C2CC3C(C2NC(C2CCOC2)=O)C13 C(=O)(C1=CC2CCC1C2)NCC1(NC(C2C(C)=CCS2)=O)CCCCC1 Cc1csc(C(N2CCC(OCCNC(=O)Cn3cnccc3=O)C2)=O)c1Cl c1(C(=O)NCCC(=C)CNC(c2ccc(CC)cc2)=O)cc(C(C)C)oc1C Cc1cncnc1N(C)CCN(C(=O)CCc1nc(O)n[nH]1)C(C)C N1(CCOC)CC(C(=O)NCCC(C)NC(=O)CCc2ncc(C)[nH]2)CC1=O C(=O)(CCC(=O)Nc1ccccc1)NC1C(CNC(CC=C)=O)C1 C=CCCCCCCNC(C1CCCN(C(C2(C(C)(C)O)CCC2)=O)CC1)=O C(=O)C(C)(C)CC(F)(F)F.CC(O)C(C=O)N.CC(F)C.C(N)(=O)C=O.N N1(C(C(C)(O)Cn2ccccc2=O)=O)CCCC12C1CCC2C1 Cc1[nH]nc(C(F)F)c1C(=O)NCC(=O)NC1CC1F C12(NC(CSCC)=O)CC1CN(C(c1cnc(-c3ccccc3)cn1)=O)C2 C1(CNC(CC(C)(C)O)=O)(C)CC12CCN(C(C1(O)CC(F)(F)C1)=O)CC2 C1(C(CNC(=O)Cc2ccco2)O)CCCN1C(=O)CC1(C(F)(F)F)CC1 N1(C(C(C)C#N)=O)CCN(C(c2c(C(F)(F)F)nn(C)c2Cl)=O)CC(CO)C1 CC(C(=O)NCCOC(C)(C)CNC(C1CNC(=O)C1)=O)C(F)F c1(CNC(C(c2ccccc2)NC(C=C(C)C)=O)=O)csc(CC)n1 c1(C(=O)NC2COC3CN(C(CCSC)=O)CC32)ccc2c(c1)NCCC(=O)N2 N1(C(CC2CC(=C)C2)=O)CC(C)(C)OCC1C.c1(C(=O)N)cc2n(c1)CCSC2 N(C1CCCc2nc(-c3ccc(F)cc3)sc21)Cc1c(C)nn(C)c1N1CCC1 C(=O)(CC(C)C(=O)NCC1(NC(=O)C#CC2(C)CC2)CCOC1)OCC c1(C(C=O)N(CC(=O)OCC)C(C)C)cn(-c2ccccc2)cn1.CC.N c1(C(C)=O)ccc(NC(C2CCCN2C(c2csc(C#N)c2)=O)=O)cc1Cl C12(CNC(=O)CC3CC4(CCC4)C3)CCCC1CN(C(C1CNC(=O)N1)=O)C2 C(CN=c1[nH]c2ccc(Br)cc2o1)C1CCC(NC(c2c(C)sc(O)n2)=O)C1 N1(C(c2c(C)nc(O)[nH]2)=O)CCC2(CNC(c3cccs3)=O)CCCC12 CN1CCC2C1CCCN2Cc1cccc(C(=O)N(c2ccccc2C#N)C)c1 Cc1ccc(CC(N2CC(NC(=O)CC3CC3)CCC2C)=O)cc1Br C1(NC(C23CC(CNC(=O)C=Cc4cc[nH]n4)(C2)C3)=O)CCCC1(F)F C1(NC(c2c(C)nc(C(C)C)s2)=O)CN(C(c2ccns2)=O)CC12CCOCC2 c1(C(N(C2(C(=O)NCC(CC=C)OC)CC2)C)=O)cc(F)ccc1C(C)C C=C=CC(C)C(=O)N1CCC(C(=O)NOC(C)C=C)C1C(C)C C1(C(=O)NCCCN(C)C(C2(O)CCC2)=O)CCC1(C)C O=C1C(N2CC(F)(c3cccnc3)C2)CCCN1c1ccc(Br)cc1 N1(C(c2c(C)sc(Cl)n2)=O)CCC2(CCC(CNC(=O)CC3=CCCC3)O2)CC1 Cc1nc2cc(C(=O)N(C)CCNC(=O)CC3(CO)CC3)cc(Br)c2[nH]1 Cc1csc(=O)n1CCC(N1CC2CC2(NC(=O)CO)C1)=O.C1CCCOC1.C C1(CNC(C(COCC)(C)C)=O)CC(C(=O)N2CCOC3CC23)=NO1 CC1OC2CCC1(C(=O)N(C1(C(N3CCCC(C)C3CO)=O)CC1)C)C2 c1(NC(C2C(C(=O)OC)C=C2)=O)cccnc1.C1(=O)C(c2ccoc2)N1 C1(C)(NC(COCCCC)=O)CCCN(C(C2CC(F)(F)C2(C)C)=O)C1 c1(C(N2C(CN(C(=O)Cc3cn[nH]c3)C)COCC2)=O)cc2ccnn2cn1 C(CCN=c1nn[nH]n1C)N(Cc1cc(C)on1)Cc1ccc(C(C)(C)C)s1 c1(OC)ccc(C(=O)NC2CC(O)(CNC(c3c(Br)cnn3C)=O)C2)cc1 N1(C(C(C)N(C(C(C(C)C)NC(C)=O)=O)C)=O)CCC(=O)N(C)CC1 CC(C)(C)C#CC(=O)N1CC2(C1)CN(C(c1coc(C3CCCCC3)n1)=O)C2 C1(C(N(C(COC)C)C)=O)C(C)CCN1C(=O)CC1CC2CCC1C2 C1(n2cc(C(C)NC(=O)CC(c3ccccc3CO)C)nn2)CCC2(C1)CC2(F)F N1(CC)N=C(C(=O)N(CCCNC(C2CCN3CCCC3C2)=O)C)CCC1=O N1(C(COCC)=O)C2CCC1CN(C(=O)C(C1CCOCC1)OCC)C2 C(CC(C)C)(C(=O)NCC1CCOC1=O)N(C(C(COC)N(C)C)=O)C c1(CC(=O)NCC2(C(=O)NCC3CSC3)CC=CC2)cnccn1 c1(NC(C(c2ccco2)NC(=O)CC2CCOCC2)=O)cncc(CO)c1 C12(CNC(CNC(CC)=O)=O)CCC(CC1)N(C(c1ccc(Cl)[nH]1)=O)C2 N1(C(CC(CC)C)=O)CCCC(O)(CNC(=O)C2=CCC(C)CC2)CC1 CC1CC2CN(c3nccc(N(C)CC4CCC5(COC5)O4)n3)CCN2C1=O C1(NC(CNC(Cc2scc(C)c2)=O)=O)CN(C)C2(CCC2)C1 C(=O)(CC(C)O)N(CC(C)NC(c1cnc(C(F)F)s1)=O)CC.C(C)=O N1(C(C(CSC)C)=O)CCC(C2(NC(c3nc(Br)c[nH]3)=O)CC2)CC1 C(=O)(CN1C(=O)Cc2ccccc21)NCc1cccc(CN(C)C)c1 C=C(C)CCCC(=O)NC(C1CCN(C(c2cscc2SC)=O)CC1)C C(=O)(C(CC1CCOCC1)NC(C1CC2CC2C1)=O)NCCOC N1(CC)CCN(C(C2CCC=CC2NC(=O)CC(C)(C)O)=O)CC1C N1(C(=O)CC2CN(C(c3ccc(Br)s3)=O)C2)CCc2c(Cl)cc(Cl)cc2C1 c1(C(=O)NC2CC(C(N3CC4CCCC4C3)=O)C2)ccc2c(c1)CCN2 C1(C(=O)NCC2CCC(C(N(C(C)CO)C)=O)C2)CCCN(C)C1 c1(CC)nnc(C)cc1C(=O)NC1CC2CC1N(C(C1CCN(C)C1C)=O)C2 c1(OC)cc(C(=O)NCC2CC2NC(=O)CC(O)CC2CC2)ncc1Br C(=O)(C(C)(C)C(F)F)NCC1C(NC(c2cn(C)nc2C2CC2)=O)C1 C1(C(=O)NCCCC(C)NC(C=Cc2ccc(C)o2)=O)CCC2(CCOCC2)O1 C=CCC(C(=O)NCC(CNC(=O)CCC(C)(F)F)S(C)(=O)=O)C(C)C C1(C(F)(F)F)(C(N2CC(n3cnc(=N)[nH]3)C2)=O)CS(=O)(=O)C1 C1(C(=O)NC(c2cccc(NC3CCN(CC)CC3)c2)=O)COc2cscc2O1 C1(CC=C)(NC(=O)CCOc2ccccc2Cl)CCN(C(C2(F)CCOC2)=O)C1 c1(C(=O)NC2CCCN(C(C3(O)COC3)=O)C2)noc2ccc(Cl)cc12 C1(C(C)(C)C)CN(C(=O)C#CC2CC2)CC1C(=O)NOCCC1CC1 N1(C(C(CCOC)OC)=O)CC(NC(=O)COc2cc(Cl)ccc2Cl)CC1(C)C C1COC2(CCN(C(=O)C(CO)N(C)C)CC2)C1.C(C(=O)N)(C(C)O)NC(C)=O N1(C(c2c(C)snc2)=O)CCC(O)(C)C1.C1(c2ccccc2)(C(=O)N)CC1(F)F CC(C)CC(CNC(=O)CC12COCC(C1)C2)NC(=O)CS.C1CCCO1 N1(C(c2cscc2-c2ccccc2)=O)CC2(CCN(C(C3CC(O)C3)=O)CC2)C1 c1(C(=O)NCC2C(Nc3ccc(C#N)nc3)CCCC2)cccc2c1C(=O)NC2 C#Cc1ccc(F)c(C(=O)N(CC(CC)NC(c2ccncn2)=O)CC)c1 C1(CO)CCC(F)(F)CC1.C1CCCCC(=O)NCCN1CCC.C1CC1.C N1(C(C(C)S(N)(=O)=O)=O)CCNC(=O)CC1C(N)=O c1(NC(CCN(CC#C)C(c2cccc(CO)n2)=O)=O)cccc2c[nH]nc12 c1(-c2ccc(C)cc2C#N)n[nH]c2ccc(C(N3CCC(O)C(F)C3)=O)cc12 Cc1cccc2c1N(C(=O)C(C1CCCCC1)NC(C1COCCC1C)=O)CC2 C1(NC(c2ncc(CC)s2)=O)CC2(CCCCN2C(C2(C)CC2Br)=O)C1 Cc1cc(Br)sc1C(=O)NC(C)C(CO)NC(c1c(C)cnn1C)=O C(=O)(CCC(C)(C)N(C)C)NCC1(C)CC(NC(C2=C(C)CC2)=O)C1 C1(CC)COCCN(C(C2(C)CCN(C(c3sccc3OC)=O)C2)=O)C1 N1(C(CC(C)F)=O)Cc2nccn2CC(NC(=O)C(C)(C)N(S(C)(=O)=O)C)C1 C1(NC(CCC2(C)CCC(=O)N2)=O)CC2(C1)CN(C(c1cccc(C#N)c1)=O)C2 c1(C(=O)NCC(C(C)C(C)C)NC(c2nnc(C)s2)=O)cccc2c1CCOC2 c1(NC(C)=O)cccc(C(=O)NC2CC2CNC(c2ccnnc2)=O)n1 CCS(=O)(=O)CC(=O)NCCC(O)CNC(=O)C(c1ccc(F)c(F)c1)C c1(C(=O)NCC(CNC(c2ccoc2C)=O)OC)c(C)[nH]c2ccc(Cl)cc12 C1(C(=O)Nc2cn(CC)nc2C)CN(C(=O)C(C)(C)C)CCC1(F)F c1(OC)nccc(C(C)(C)NC(N2CC(CC(O)C(=O)O)C2)=O)n1 N1(c2cc(NC3CCC4CN(C)CC4C3)ncn2)CCC(C2CCOCC2)C1 N1(C(Cc2c(OC)ccnc2)=O)CC2(CCN(C(=O)C(C)C3CCCO3)CC2)C1 C1(NC(Cc2c(CC)con2)=O)CN(C(=O)Cc2ccoc2C)CC1OC CC1CCN(C(c2cnn(C)c2N)=O)C(C)C1NC(=O)CC(C)(O)C1CC1 C=CCC(C)C(=O)NCCOC1CCN(C(=O)CC2CCN(CC(F)F)CC2)C1 Cc1cc(CC(N2CCCC2C(=O)O)=O)c(C)n1-c1ccc(OC(C)(C)C)cn1 S(=O)(=O)(c1ccc(NCc2ccsc2Cl)c(Br)c1)N1CCS(=O)(=O)CC1CCO N1(C(C2(OCC)CCOC2)=O)CC2CCCN(C(c3cc(Cl)cnc3C)=O)C2C1 C1(C(=O)NC2(C=C)CCCC2)CCN(C(C2CC3(CCC3)C2)=O)CCO1 c1(C(=O)NC(C(C)C)CCN(C)C(C2CCCC(C)C2)=O)cnc(Cl)c(Cl)c1 C12(NC(C3CC4CCC4C3)=O)CCC(CC1NC(C1CN3CCC1CC3)=O)C2 N1(C(c2occ(C)c2)=O)CC(NC(=O)Cc2ccc(Cl)cn2)CC12CCC2 Cc1nsc(C)c1C(=O)NC1CCCC(NC(c2csnc2C2CC2)=O)C1 C1(NC(CCCC)=O)CC2(CCC(NC(=O)CC3CCC(F)(F)C3)CC2)C1 c1(C(N2CCN(C(C(CCOC)C)=O)CC2CF)=O)cnc2c(ccn2C)c1 c1(CCC(=O)NC(C(C)NC(C2CCCC(O)C2)=O)C)cc(F)cc(F)c1 C1(CC(=O)NC(C2CCCCC2)CNC(c2ccno2)=O)C=CCCC1 c1(C(=O)Nc2cccnc2CO)nsc2cc(-c3cn[nH]c3)ccc12 c1(N2CCC(C)(C(=O)O)CC2)nnc2n(c1=O)CCC2 C1(C(N2CCCC2)=O)CC2CCC(C1)S2(=O)=O.c1(C=O)ccnc(C2CC2)c1.N C(CN=c1[nH]n2cc(C)nc2s1)N(C(=O)C(C)CC(C)C)CC c1(C(=O)NCC2C(CNC(C#CC(C)(C)C)=O)C2)coc2c(F)cccc12 N1(C2C(NC(=O)CCc3cn[nH]c3)COC2)CCN(C(C23CCC2C3)=O)CC1 c1(C(=O)NCC(C)N(C(C2C(=C)C2)=O)CC)csc(CCCC)n1 C1(C(=O)NCCN(C(C(c2cccc(C)c2)F)=O)C2CC2)CCCCCC1(F)F N1(C(c2c(C(C)C)ccs2)=O)CCC(CNC(C2CCCOC2)=O)C(O)C1 C1(CCC(=O)Nc2ccc(N(C)C)nc2)CCCCN(C(=O)Cc2ccns2)C1 C1(C(=O)NC(C)CCNC(=O)CC2(CO)CCC2)CC(O)(C#N)C1 C1(C(=O)NC(c2ccccc2)(C)C)CC2(CC2)CN1c1nccc(C(F)F)n1 N1(C(c2csc(Cl)c2)=O)CC2C3CCC(C2C1)N(C(c1cc(O)ccc1O)=O)C3 C1CCC(C)N(C(C2CC(S(C)(=O)=O)C2)=O)C1.Cc1onc(C2CC2)c1C=O c1(C(C(N2CCC(CNC(CC3(OC)CC3)=O)C2)=O)(F)F)cccc(F)c1Cl N1(C(Cc2ncn(C)c2)=O)CCC2(C1)CN(C(c1cc(Cl)cc(Cl)c1)=O)C2 CCCC(F)C(=O)NCCC1(C)CCN(C(c2csc(C)c2N)=O)C1 c1(C(=O)NC(C)CCCNC(=O)Cc2cc[nH]n2)cncc2cccnc12 C1(C(=O)NC2CC(C3CCC3)C2)CN(C(c2ccnnc2O)=O)CC1(F)F C12(C(=O)NC3C(C=C)COC3)CCN(C(=O)CCC(C)(C)OC)CCC1C2 C1(CCOC)(NC(=O)CCc2nccs2)CCN(C(=O)CCn2cccn2)C1 CC(C)CC(CNC(=O)C(C)C1CCC1)NC(=O)CCC12CCC(CC1)C2 CC1CC=C(C(=O)N2CC(NC(c3cc4ccccc4s3)=O)C3(CCC3)C2)CC1 c1(CC(C(=O)NCC2CN(C(CN3C(C)CCCC3)=O)C2)O)c(F)cccc1Cl CCCCC(CC)CC(=O)NC1CCCCN(C(C2(C3CCCO3)CC2)=O)C1 Cc1ccc(SCC=O)cc1.C1(C(N(CC)C)=O)(C(=O)N(C)C(C)C)CC1 N1(CCN(C)C(c2cnn(C)c2CO)=O)CCN(C(C2(CF)CC2)=O)CC1 c1(CNC(N2Cc3ccc(Cl)cc3C2)=O)ccc([N+](=O)[O-])c(F)c1 N1(C(C(C2CC2)OC)=O)CCC2CCC(NC(C3CCN(C(N)=O)CC3)=O)C1C2 c1(CNC(C(C)(C)N(C)C(=O)OC(C)(C)C)=O)ccccc1I C1(CC)CC(F)(F)CN1C(C1CCC(F)(F)CO1)=O.c1(C=O)cccc(Cl)c1.N c1(NC(c2ccc(NCc3cccc(OC)c3O)cn2)=O)cc(C)c(O)c(C)c1 C(CC(C)(C)C(=O)NCC1CCN1C(=O)C(n1ccnc1C)C)SC c1(C(C)(C)C)cc(C(=O)NCC(CO)Nc2cc(C3CC3)ncn2)ccn1 C1(C(C(=O)N(CCSC)CC)C)CCN(C(=O)CCc2cn[nH]c2)C1 CC(O)CCCCCC(=O)N(C)CCN(C(=O)C=CC1(C)CCOCC1)C c1(C(=O)NC2CN(C3CN(C(C(C=C)O)=O)C3)C(=O)C2)nn(CC)c2c1COCC2 CC1(CNC(C2CC(N)(CO)C2)=O)COCCO1 NS(=O)(=O)C1(C=O)CC1.C1CC2(C1)CC2.C(=O)CN(CCO)CCO.N Cc1nc2ccc(C(=O)NC(c3cccc(Cl)c3)C(=O)O)cc2n1C N1(C(CC(C)F)=O)CC=CC(NC(=O)Cc2csc(C3CCCC3)n2)C1 C1(F)(c2cn(C(C)C)nn2)CCN(C(=O)CCOC2COC2)C1 C1(F)(C(=O)NCC(CC)(CC)NC(c2cnc3c(c2)CC3)=O)CCC(C)CC1 C12(CNC(C(F)=CC)=O)CCC(C1)N(C(=O)CNS(N)(=O)=O)C2 c1(C(N2CCCC(NC(C(C)(C)N(C)C)=O)C(F)C2)=O)ccn2[nH]c(=N)nc2c1 c1(OCC)ccc(C(=O)NCC(CC)NC(=O)CC2CCCCO2)cc1C C1(C#N)(C=O)CC2(CC2)C1.n1(C(C)C)nccc1C(=O)N.C1(O)CCC1.C c1(C(N(C(CNC(C(C)O)=O)C)C)=O)ccc(Br)cc1OC(F)F c1(C(=O)NCCC2CC(NC(c3ccc(C(C)=O)s3)=O)C2)cccc(F)c1 c1(C(=O)NCC=CC)ncnc2c1CCC2.c1(C(=O)N)n[nH]cc1C1CCC1 N1(C(CNC(=O)NC2CC2)=O)CC2CC1CN2C(C1(O)CCCCCC1)=O CC(C)P1(=O)CCN(C(=O)C(N)CCN2CCOCC2)CC1 CCC(C)CC(C)C(=O)N1CCCC1C=CC(=O)NCC1(CC2CC2)CCC1 C(C(Cc1ccncc1)C(=O)O)NCCCC(=O)NCc1ccccc1 N1(C(=O)CSc2ccsc2[N+](=O)[O-])CCCC2C1CCN2C(C1CCCO1)=O C(=O)(CCCCCF)N1CC(O)(C(C)NC(C(C)SCC)=O)C1 Cc1ccc(C(C)C)cc1C(=O)NC1CC(C)N(C(c2cc(CO)on2)=O)C1 CCCC(C(=O)NC(C)CNC(=O)CCNC(N)=O)c1cccc(Cl)c1 C1(CC)CCCCC1C(=O)NC(C(=O)NC1CCC(N(C)C)C1)C(C)O Cc1cnccc1C=CC(=O)NC1CC1C.c1(C(=O)N)csc(CC(C)C)n1 C(=O)(C1=CCCC1C)N1C(CNC(c2c(C)coc2C(C)C)=O)CCCC1 c1(CN(C(c2ccsc2C2CC2)C(=O)NCC2CCOC2)C)ccc(F)cc1 Cc1c(N)ccc(C(N2CC(CNC(=O)CCC3CC3(F)F)C(O)C2)=O)c1C C1(C=O)CCCOCC1.C(=O)(CCn1cncn1)N(CC(=O)N(CC)CC)C Cc1nc(C)c(C(N2CCCC2(C)CCC(=O)NCCOC2CCCCC2)=O)o1 O=C1CCC(NC(=O)CNC(C2C3CCC2(c2ccco2)C3)=O)CN1 C12(NC(C3C(C)N(C)CC3)=O)CN(C(=O)CN3CCCCC3)CC1CS(=O)(=O)C2 N1(C(C=CC)=O)C2CCC1C(CO)N(C(c1cc3cccc(C)c3s1)=O)C2 n1(CC#C)cccc1C(N1CC(C(O)C(=O)NCC(c2ccnn2C)O)C1)=O C(=O)(C1=C(C#N)CCC1)N(C)CC.C1(CC=O)CCCCC1(C)C.C1CCCC1.N C1(CC(=O)NCCCN(C(C(N)=O)=O)C2CC2)CCC2(CCC2)O1 CC1CCN(C(=O)CC2CCN(C(c3cncn3C)=O)CC2)C1CO C(C(=O)OC)(C(C)C)NC1(CSC)CCC1.C1=CCNC1=O N1(C(c2c(C)n(-c3ccccc3)nn2)=O)CC(C)(C)c2cccc(Br)c21 c1(CCNC(C(C)=C2CCC2)=O)cccc(Cl)c1.C(=O)(C(C)CN(C)C)N N1(C(C)=O)CCCC(C(N2CC=CC2CNC(C2(CF)CC2(F)F)=O)=O)C1 c1(C(=O)NCC2(O)CN(c3ncnc(C)c3Br)C2)nc2ncccn2n1 C12(C(N(C(CC)C3CC3)C)=O)CCC(CN(C(=O)CC(C)(F)F)C1)C2 c1(C(N(CC)CC2CCCN2C(=O)CNC(=O)NC)=O)cnccc1Br C1(CNC(=O)CCC2CCCC(=O)N2)CN(C(C2CC=CC2)=O)CCCO1 C#Cc1ccccc1C(N1CCC(OC(C2CC(=O)N(C(C)C)C2)=O)C(O)C1)=O N1(C(c2ccn(CCC)n2)=O)CCC(C2CC2)C1C(N1CCOC(C#N)C1)=O C1(NC(C2(CC)CCCC2)=O)CCN(Cc2nnnn2-c2ccccc2)CC1C C(N=c1[nH]c2c(c(=NCC3(C)CC(F)(F)C3)[nH]1)CCC2)c1nccc(N(C)C)c1 CC(C)=C=CC(=O)NCC1(NC(c2ccc(CN=[N+]=[N-])o2)=O)CCCC1 N1(C(=O)NC(C)Cc2ccc(Br)cc2)CCOCC1(C)Cc1ccccc1 C1(C(=O)NC2CCN(C(c3c(C)ccc(C)n3)=O)C(C)C2)CCc2c[nH]nc2C1 C1(NC(COc2cn(C)nc2)=O)CC2CCCCCCC12 CN(C(c1ccc(F)cc1)c1ccco1)N1CCN(CC(C)(C)C(F)(F)F)CC1 CCCCC(C(=O)NC1CC1(C)C(F)F)NC(c1ccccc1O)=O N1(C(C(C)=C(C)C)=O)C2COCC1CC(NC(C1CCCN(C(N)=O)C1)=O)C2 c1(C2(C(=O)NC(CC)CNC(=O)CC(C)F)CC2)cc(OC)ccc1C CC1CCCN(C(c2csc(CNC(=O)C(C)(C)CO)c2)=O)C1CCO CCCCCC(C)CC(=O)NC1(C(=O)NC2CC(=O)N(C)C2=O)CCCCC1C C1(NC(C(CC)C(C)C)=O)CC12CCC(NC(c1cc(C)sc1C)=O)CC2 CC1(C(=O)NC2CN(C(C34CCC(C3)C4)=O)CC2n2ccnn2)CCC(O)CC1 CCC(C)C(CNc1cccc(C(=O)N(CCC(N)=O)C)c1)OC C1(NC(C2CCN3CCCC3C2)=O)CC2CCC1CN2C(c1cnsc1)=O c1(C(=O)NCC2N(C(COC(CC)(C)C)=O)CCOC2)sc2ccccc2c1C N1(C(c2c(N)snn2)=O)CC(C(=O)NCCCN2CCC2)CC12CCC2 c1(C(N2CCC(CCOC)(NC(c3ccc(C)[nH]3)=O)C2)=O)cnccc1C#N Cc1ccn2ncc(C(=O)NCC3CCN(C(=O)CCC4CC4C)C3(C)C)c2n1 C(=O)(C1c2c[nH]nc2CN1C(=O)CCC(C)(C)C)NC(C)CS(N)(=O)=O c1(N(C)CCC2CC2)nc2c(c(=NCC3(c4ccccc4)CCCC3)[nH]1)CSC2 N1(C(c2cc(CNC(CC3C=NN(C)C3=O)=O)ncc2)=O)CCCC(C)(O)C1 C1(C(=O)NCC(C)CN(C)C(c2cc(CCO)on2)=O)Cc2ccccc2CO1 C(CCCC(c1nnnn1CCCSC)NCCOCc1ccc(Br)cc1)SC C1(NC(Cc2c(C(C)C)con2)=O)CCOCC1C(=O)NCC=CC1CC1 Cc1cc(=NCC2(C(F)F)CC3(CCC3)C2)[nH]c(=NCC2CC(F)(F)CO2)[nH]1 n1(CC)c(C(N2CCC3CCCC23CNC(C2CCC2)=O)=O)nc2ccccc12 c1(NCCCNC(C2(CC#C)CC2)=O)ncccc1C(=O)OC CCCCCCCCC(=O)NCCCN(C(=O)C(O)CC(N)=O)CC1CCCC1 Cn1ccnc1CCNC(=O)CC1CCN(C(=O)CCn2cnnn2)C1 N1(C(c2ccc(CO)o2)C(=O)NC2CCCCC2)CCc2cc(Cl)ccc2C1 C(=O)(NNc1ccc(O)cc1)C1NCC1.N1(C(=O)OC(C)(C)C)CCCC1CN N1(C(c2nc(C)sc2C)=O)CCC(C)C(CNC(c2cc(C#N)c[nH]2)=O)C1 C1(N2CCC(CC(=O)N(C)C)C2)CC(C(=O)NC2CCCC2)C1(C)C C1(CC(=O)NCC(CC)(C)NC(C2C=CC=CC=C2)=O)CCOC(C)(C)C1 C1(NC(CCCN(C)C(c2cc(C3CC3)on2)=O)=O)CCN2CCC1C2.ClCC N1(C(CC(C=C)C)=O)CC2(C)CC1(C(=O)NC(Cn1cncn1)CC)C2 CC(CC(N)=O)C(=O)N(C)CC1(O)CN(C(C2(CF)CC2)=O)C1 CC(C)CC(C)CC(=O)NC1CN(C(=O)CCOCCN(C)C)CC1F N#Cc1cc(C(=O)NCC=CCNC(=O)C(C2CCC2)C2CCC2)on1 N1(C(C(CC)OCC)=O)CC2(CC2)CC1CNC(c1cc(CF)on1)=O Cc1cc(C(N2CCN(CC(=O)N(C)C)CC2)C(=O)NCC2CC2)ccc1CO C1(O)(CC(N2CC(O)(CC)C2)=O)COC(C)(C)C1.C(=O)C#CC(=O)NC CCCC(CC)CCC(=O)N1CCCCC(CC(=O)NCc2cccc(C)n2)C1 N1(C(C2CC(NC(c3n(CC#C)cnn3)=O)C(O)C2)=O)CC(C)CC(C)(C)C1 C(=O)(CCC(C)NC(c1cnc(Cl)n1C)=O)N1CCC(COC(C)=O)C1 C(CS(=O)(=O)CC(C)C)NCc1nnn[nH]1.C1(C2CCCO2)(CC)CCC1 c1(OC)ncccc1C(=O)NCC(C(=O)NCCN1CCOCC1)N(C)C C1(CC)(CNC(N2CCC(Nc3cc(OC)ccn3)C2)=O)CCCOC1 C1(CNC(c2ccc(C)o2)=O)CCC2CN(C(=O)C(C)Sc3ccccc3)CC12 S(=O)(=O)(c1ccc(Cl)c2nonc12)N1CC(N(S(CC)(=O)=O)C)C1 Cc1nc(=N)[nH]c(C)c1C(=O)N(C)CC1CN(C(c2cc(Cl)cc(Cl)n2)=O)C1 c1(N(C(=O)C(F)CCC2CN(C=O)C2)C)ccc2scc(Br)c2c1.C(C)(C)C.O C1(NC(c2c(C)cco2)=O)C2CCCN(CC(O)COC(C)C)C2C1(C)C c1(C(=O)NC2(c3ccc4ccccc4c3)CC2)ccc2ccc(O)nc2n1 Cc1noc(C)c1C=CC(N1CC(N(C)C(c2csc(C)c2N)=O)C2(CC2)C1)=O N1(C(C(COC)OC)=O)CCC2(CC1)CN(C(=O)C=Cc1ccccc1Cl)C2 c1(CNC(C(C)=CC)=O)cn(CC(=O)NCC2(N(C)C)CC2)nn1 c1(CC)ccc(OC)c(NC(=O)Nc2cc(N3CCCCC3C)ccc2O)c1 Cc1cc(Br)oc1C(=O)NC1CC(C)(NC(=O)C(C)n2cccc2)C1 CCC(C)(C)C(O)C(=O)N(CCC(=O)NC1CN(C)CC1C)CCO C1(C(N(CC(CCC)C)C)=O)CCN(C(=O)CC(C)(C)CCC)C(C)(C)C1 c1(CN2CCC(CC(=O)N(C)Cc3cccc(N(C)C)c3)C2)ccc(Br)cc1 N1(C(C2N(CC)CCOC2)=O)CCC(C)(CNC(=O)Cn2[nH]cnc2=N)CC1 C1CC2(COC(C)(C)C2)C1.C1(C(N2CC2=O)=O)CCS(=O)(=O)C1.CCC.O C(=O)(CC(C)C1CCCCC1)NC(C1CCCC1)CNC(COCCCC)=O c1(CC(=O)NC2(CNC(=O)CCCC3CCCC3)CCC2)ccc(Cl)cc1F O=C(C1=Cc2ccccc2C1O)NC1CC1NC(c1cc[nH]c1)=O C(c1cc2ccccc2o1)=CC(N1CCC(C(C)NC(COCCCC)=O)C1)=O O(NC(=O)C(CC1CCC1)NC(c1ccc(C)cc1)=O)CC(=O)OC CC1CCCN(C(c2ccon2)=O)C1CNC(=O)CCC1(O)CCC1 C=CCC(C(=O)OC)N(C)C(c1ccc(OC)cc1)C C1(CC)CN(C)CC1NC(=O)NCc1cnn(CC2CC2)c1 c1(C(=O)NCCC(=O)NC(CCC)C(=O)NC)c(F)ccc(Br)c1C Cn1ccc(C(=O)NC(CNC(C2(c3ccccc3)CC2)=O)CO)c1 C1(CC)CCC(C(N2CCC(COC)(NC(=O)CC3CCCOCC3)C2)=O)CC1 CC1(C)CCC(C(=O)NCC2(C(=O)NC3(C)CC4(CC4)C3)CC2)O1 C1(CNC(c2noc3ncccc23)=O)CC2CCCC2N1C(c1ccccc1)=O C1(NC(Cc2nc(C)[nH]n2)=O)C=CCN(C(C2CCCN2c2ccccc2)=O)C1 C1(C(=O)OCC)CCCC1NC(=O)C(O)C1CN(C(c2c[nH]nc2C)=O)C1 C1(C=O)CCN(S(=O)(=O)N(C)C)CC1.C(CSC)(C(=O)NC(C)CC)OC CN1CC(O)CCC1C(=O)NC1(CCNC(C2CCCCCCC2)=O)CC1 N1(C(c2c(C)ccnc2)=O)CC2CC1CCC2NC(=O)CC1CC=CCC1 C=CCC(C(=O)NCc1nc(CNC(c2ccc(Cl)cn2)=O)cs1)OC CC1C(NC(c2cnc(C3CC3)nc2)=O)CCCN1C(c1ccsc1C#N)=O C1(NC(CNC(C)=O)=O)CCN(C(=O)Cc2cccc(C)c2Cl)C(C2CC2)C1 C(O)(CCC(c1csc2c1CCCO2)C)(C(F)(F)F)c1ccc(C)o1 Cc1[nH]nc2ncc(CNc3cc(C(F)F)cc(C(F)F)c3)cc12 N1(C(c2cnn(CC)n2)=O)CC2(CC(NC(=O)Cn3cnnc3)C2)C1 C1(C(=O)NCc2c(C)nns2)C2CC2CN1C(C1C=CCCC1)=O C(=O)(CCC(=O)N1CCC(CCC(=O)N(C)Cc2cc(C3CC3)no2)C1)NC N1(C(c2c(C)onc2)=O)CCN(C(c2ccc(C(=O)N(C)C)cc2)=O)CC1 c1(Cc2ncc(C)s2)nc(CN2CCC(CN(C)C)C2)[nH]c1-c1ccccc1 CC1OC2CCC1(NC(c1nc(C(C)C)no1)C)C2 C(N=c1cc(-c2ccc(Br)cc2)nc[nH]1)n1nnn(-c2cnn(CC)c2C)c1=O c1(OCCC(=O)N(c2ccc(I)cc2)C)ccc(Cl)c2c1C(=O)NC2 C1CCCN(C(c2cnc(C(C)C)nc2)=O)C1.C(=O)(C(C)(O)C1CC1)NCC c1(C(=O)NCC2CCC(NC(CCC#CC)=O)CC2)ccc(O)c2ncccc12 C(C)(C)(CC(=O)NCC1COC(C)(C)C1)N(C(CCN(C)C)=O)C c1(C(N2CCC(n3ccnc3)C2)=O)ccncc1-c1ccc(F)cc1 CC(CO)C(C)N=c1[nH]c(=NCC2C3CC2NCCNCC3)c2[nH]ccc2[nH]1 N1(C(C2=C(C)CCC2)=O)CC(O)(C2(CNC(c3cc(F)cnc3O)=O)CC2)C1 C(=O)(C(C)C(F)(F)C(F)F)N1CCC(NC(c2nccc(C)n2)=O)CC1C CCC(CC)(CC)C(=O)N1CCN(C(c2n[nH]c3c2CCCC3)=O)C(C(F)F)C1 C1(C(=O)NCC2CC(NC(C(C)c3ccco3)=O)C2)CCCC12OCCO2 C1(C(C)C(=O)Nc2cccc(C(=O)Nc3ccccc3F)c2)CCN(CC)CC1 c1(C(=O)N)nsc2c(Cl)cccc12.c1(CC)cc(CC(=O)NCC2CC2)on1 c1(NCCC2CCC(NC(C3N(N=O)CCC3)=O)C2)nc(Cl)nc2sccc12 C(=O)(C(C)(F)C(C)(C)F)NCCC1CCC(NC(CC(C)O)=O)C1 Cc1ncn(C)c1C(N1CC2C(NC(c3ccc(C4CCOC4)s3)=O)C2C1)=O N1(C(C(C(C)C)=O)=O)CCC2(CC2NC(c2ccc(SC(F)(F)F)cc2)=O)C1 c1(C(=O)NC2CCN(C(CCC)=O)C2)sc(C)nc1OC C12CCC(C(N3CC4(C3)CN(C(=O)CC3CCC(C)C3)C4)=O)(CC1)CO2.CO Cc1nc(Br)oc1C(N1CCC(NC(C2COC(=O)N2C)=O)C1)=O Cc1cc(C(=O)NCCC2CN(C(c3cc(C(C)(C)C)n[nH]3)=O)C2)cn1C c1(CC(=O)NCC(COCC)CO)ccc(F)cc1C.C1(OC)C(=O)N1 C1(NC(C(c2n(C)ncc2)O)=O)COCCC1NC(=O)C.C1CC(F)(F)C1.O N1(C(C2(OC)CCCCC2)=O)CC(C(=O)NCC(C)C(C)(F)F)CCC1(C)C N1(C(CCC(=O)N2CCCC2)=O)CCC2(C1)CN(C(=O)C1CC1)C2 c1(OC)ccc(Cc2nnc(NC(=O)COCc3ccccc3)s2)c(C)c1 C1(C(=O)NCC(C)N(C(=O)Cc2ccno2)C)CCN(C2CCCCC2)CC1 C1(C(=O)NC2CCCC(CNC(C3CC4C=CC3C4)=O)C2)CN2CCC1CC2 C1(NC(c2cn(C)nc2)=O)CCN(CCNC(C2(O)CCCCC2)=O)CC1 C(=O)(C1CCCc2c[nH]nc21)NC(CCCC)CNC(=O)CCc1cnc(C)o1 c1(C(=O)NC2C3CN(C(C(CSC)O)=O)CC2C3)c(O)cc(F)cc1F O=S(=O)(c1ccc(NC2CCSC2)nc1)NC1(c2ccc(F)cc2)CCOC1 Cc1cc(C(=O)NCC2(O)CCN(C(C3(C)CC3)=O)CC2)c2cccnc2c1C C#Cc1ccc(C(=O)N(C(CNC(=O)CC(C)OC)CC)C)nc1 c1(C2C(C(N3CC(N(C(c4c(C)occ4)=O)CCO)C3)=O)C2)c(F)cccc1Cl c1(-c2cn(CC3(CC4(CC)CC4)CC3)nn2)ccc2c(ccn2CCO)c1 Cc1cc(=NCCS(=O)C(C)(C)C)[nH]c(N2CCC(OCC(C)C)CC2)n1 c1(CNC(CC2(C)N(C(CS(CC)=O)=O)CC2)=O)cc(=O)cc(C)[nH]1 Cn1c(NC(=O)CC2(c3nc4ccccc4s3)COC2)nc2cc(Br)c(Cl)cc12 C1(CC(=O)NCCC2(NC(C(CCO)N(C)C)=O)CCCC2)CCCCC(=O)N1 CCC(C)C(=O)C(=O)N1CCC(CC(=O)NCC2(COC)CC2)CC1 C1(NC(c2ncn(C)c2)=O)CC(NC(c2cc(N)ccc2O)=O)C12CCOCC2 c1(C(=O)NCC(CC)NC(c2csc(COC)c2)=O)ccoc1Br C=CC1(CC(=O)NC2CCN(CC)C2=O)CN(C(C2CC(C)(O)C2)=O)C1 c1(C(F)(F)F)ccc2nc(CCc3noc(C4CCC5(CCOCC5)O4)n3)[nH]c2n1 C1(C(N2CC(C(N3CC(CC)C3)=O)(SC)C2)=O)CCCC2(CC2)C1 c1(OC)ccc(OC(F)(F)F)cc1NC(=O)NC1CCC1(C)c1ccccc1 c1(-c2cn(CCCNC(c3n(CCCC)ncc3)=O)nn2)c(Br)cnn1C N1(C(c2c(C)con2)C(=O)Nc2ccc(F)cc2)CCn2cnnc2C1C c1(N(C(=O)CCSC2CC2)CC)ncc(CO)cc1Cl C(CC(=O)N1CC(C)CC1(C)C)(C(F)(F)F)c1c(C)nn(C)c1C.C(=O)(CO)N c1(OC)c(C=O)c(C)nn1C.C1C2CN(C(C3CCN(C(N)=O)CC3)=O)CC12.N S(=O)(=O)(c1cccc(Cl)c1C)Nc1c(Cl)ccc(OC)n1 N1(C(c2ccc(C)cc2N)=O)CCC(CNC(c2cccnc2C)=O)C(F)(F)C1 c1(CC(=O)NCCC(C)N(C(C(C)SC(C)C)=O)C)ccc([N+](=O)[O-])cc1 CN1CC=C(C(=O)N2CCC(O)(CN(C)C(C3CC3(F)F)=O)C2)C1 CC(C(=O)NC12CCCC(NC(C3CCN(C)C3=O)=O)(C1)C2)C(C)(F)F N1(C(C2OCC(C)C2)=O)CCC2(CCCN2C(c2cnc(C#N)s2)=O)CC1 CC1CC(NC(=O)C=Cc2nc[nH]n2)CCN1C(=O)C(N)=O C1(C(CNC(c2nnc(C)s2)=O)O)CCN(C(c2[nH]nnc2C(F)F)=O)CC1 N1(C(C2C(C)(C(C)C)C2)=O)CCCCC(NC(C2CCCC(O)C2)=O)C1 C(=O)(C1CCCc2nc[nH]c21)N1C2(CNC(=O)CCc3cnn[nH]3)CCC1CC2 N1(CC(CN)Cc2cccnc2)CC(CO)C2CCCC12 Cc1noc(C)c1C(c1nc(-c2cccc(Cl)n2)nn1C1CCOC1(C)C)C c1(C(N2CC(NC(c3cc(C)sc3)=O)C(C3CC3)C2)=O)cc2cccc(F)c2o1 C(C1c2ccccc2CCN1c1ncnc(Cl)c1Br)NC(CCCS(C)(=O)=O)=O c1(NC(CC)CNC(=O)Cc2cnccc2Cl)ccnc2nc(C)nn12 c1(C(=O)NCC(O)Cc2ccccc2)ccc(Cl)cc1-n1cccc1 CC(C)(CNC(=O)CCSC(F)(F)F)NC(C1CCC1c1nc[nH]n1)=O C=CC1CCCC(NC(=O)CCC(CC)NC(=O)CC=CCC)C1 C1(C(=O)N)CC(=O)N(C2CC2)C1.C1CC2CC2N1C(=O)C(C1CCCCC1)F C1(CNC(C(CCOC)C)=O)CN(C(c2nccn2C(C)C)=O)CC(C)(C)C1 c1c(N)cccc1Cl.C1(NC(CC)=O)CCCC(NC(=O)CC2CC(CC)=NO2)C1 Cc1cc(C#N)cc(C(N2CCN(C(=O)CC(C)P(C)(C)=O)CC2C)=O)n1 CC(C)C(C)C(=O)NCCOCC.c1ccccc1.c1(CCC=O)cncnc1.N c1(C=O)cnc(N)c([N+](=O)[O-])c1.C(C(F)C(=O)N)N(CC)CC.C(C)CCO CCC(N=c1[nH]c(=NCc2cc(Br)cn2C)[nH]c2cc[nH]c12)c1ccccc1F c1(C(=O)NC2(CO)CCN(C(c3ccnc(OC)n3)=O)C2)cccc([N+](=O)[O-])c1 C1(CCC)(NC(C2CCCNS2(=O)=O)=O)CCCN(C(=O)Cc2cccnc2)C1 c1(-c2c(NCc3cc(OC)nc(OC)n3)ccnc2)c(C)ccc2ccccc12 N1(C(c2nccc(N(C)C)c2)=O)CC(NC(C2CCCCS2)=O)CC(F)C1 C1(c2c(C(N(CCn3ncc(C)c3)C)=O)c[nH]n2)CCN(C(C2CCC2)=O)CC1 S(=O)(=O)(c1ccccc1-c1ccccc1)NCC(=O)Nc1ccc([N+](=O)[O-])cc1O Cc1nc(C(=O)N)c(C)n1C1CC1.C1(C=O)CCOC(C)(C)C1.C(C)(C)CO c1(CNC(c2c(CC)cc[nH]2)=O)ncccc1C(=O)NC1CCC1O c1(C(=O)NC2CCN(C(C3(C)CC4(CC4)C3)=O)CC2CO)cc2cnccc2o1 C1(N(C)C(C2CCC2(F)F)=O)CN(C(c2nccc(Cl)c2F)=O)CCC1O c1(C(=O)NC2C(NC(C(CC)OCC)=O)CCC2)cccnc1CC CN=c1[nH]c(C(=O)NCC2CCN(C(=O)C(c3cncn3C)O)C2)cs1 CC(C)C(C#N)C(=O)N1CC(C)C(C)(C)C1.c1(C=O)c[nH]cc1C(C)(C)C.N c1(CNC2C=CC(C(=O)Nc3c(OC)cc(Br)cc3)C2)cccc2c1OCCO2 C(Cc1ccccc1)(C(=O)N(c1csc(C(F)(F)F)n1)Cc1ccccc1)OC c1(-c2c(C)cc(Cl)cc2)cnc2n[nH]c(Br)c2c1 n1(CCOC)ncc2ccc(NC(=O)CC3(N)CCC3)cc12 C1(CNC(C(c2ccc(F)cc2)C)=O)CN(C(C2CC2F)=O)CCC12CCC2 N1(C(c2cc(Br)cc(C)c2C)=O)CCCC2(C1)CN(C(=O)C=Cc1cccs1)C2 N#Cc1ccc(CN2CCC(CC(=O)NCCc3ccncc3)C2)cc1Br N1(C(CCCC(C)=O)=O)CCC2CCC(NC(=O)CCC(C)C)C1C2 c1(C(=O)N)cc2ncccc2[nH]1.C1(NC(C(C)OCCC=C)=O)CCC(C)CC1 CCC(C)(C)CC(=O)N1CC2CC(CNC(c3cc(OC)ccc3N)=O)C2C1 Cc1nc(CC(=O)N(C2CC(NC(C3CCOC3)=O)C2)C)cs1 CCC(CC)(C(=O)NC1CC2CN(Cc3c(OC)ncnc3C)CC2C1)C(=O)O C(C(Cl)C(C)(F)F)NC(C1(CC)CN(C(=O)CC2OCCC2C)C1)=O c1(CCC(N2C(CNC(C3CCO3)=O)CCC2)=O)cc(F)c(F)c(F)c1 Cc1cc(Br)cc2cc(C(=O)NCC(C)CNC(c3ccsc3)=O)oc12 CC(CS(C)(=O)=O)C(=O)NCCC(C)(C)C.C1(C=O)CCCN1c1nccs1.N c1(C(N2CCOC(C)(C)C2)=O)ccc2c(c1)NC(=O)CN2.C(C(=O)N)OCC N1(C(Cc2n(C)ncc2)=O)CCN(C2CCN(C(C3(C)CCC(=O)N3)=O)C2)CC1 c1(C(=O)NC(C(=O)Nc2c(C)scc2)CN=[N+]=[N-])cc2ccncc2[nH]1 c1(OC)ccc2c(c1)CCN(C(c1cnc(Br)s1)C(=O)Nc1ccccc1OC)C2 CCCC(C(=O)NC(CC1CCOCC1)C(=O)NC1CCCC(C)(C)C1)C(C)C N1(CC)N=C(C(=O)NCC(COC)NC(=O)CCCCOC)CCC1=O c1(C=O)ccc(N)c(Cl)c1.C1(NC(CCN(CC)CC)=O)CC(C)C1(C)C c1cc2nn[nH]c2cc1[N+](=O)[O-].c1(C(=O)OCC)ccc(CNC2COC2)[nH]1.C C(=O)(C(O)(C(C)C)C(F)(F)F)NC1CCC(NC(c2cc(C)n(C)c2)=O)CC1 c1(-c2ccc(C(N3CCC3(C)C)C(=O)NCC=C)o2)ccccc1F C1(C(N2CCC(C(C)NC(c3cnn(C(C)C)n3)=O)C2)=O)Cc2cscc2C1 N1(C(CN(C(CC)C)CC(C)C)=O)Cc2occ(C(N3CCC3)=O)c2C1.N C(=O)(C1=CC2(CCOC2)C1)NCCC(C)NC(c1nnc2ccccn12)=O c1(NC(C2CCN(C(CCC=C)=O)C2)=O)cnc(OC)c(O)c1 c1(C(=O)OC)cnc2c(c1)N(C(N1CC(C)CC1c1ccccc1)=O)CCO2 CCCCCC(C1CC1)NC(=O)Nc1nccnc1CC1CCCN(CC)C1 C1(CNC(C2CC3CCC(C2)S3)=O)CN(C(=O)CSC(F)F)C2COCC2O1 c1(C(=O)NC2C(C)CCN(C(=O)C(N)=O)C2)csc2c1CCCC2 C1(O)(C(C)CNC(=O)C(C)(C)c2cscc2Cl)CCN(C(C2CCCCC2)=O)C1 N1(C(c2c(SC)cccc2F)=O)CCN(C(=O)CSC2CCCCO2)CCC1C C#CC(CC(C)(C)C)NC(C1COCCC1NC(c1nonc1N)=O)=O N1(C(CCC)=O)CC(CNC(=O)C(C)(C)n2ccnn2)CC1(C)C c1(C(C)=O)cc(C(N2CCC(CCNC(C3CCCCCC3)=O)CC2)=O)c(C)o1 C(=O)(CC(CC)C(F)F)N1C(CC=C)(C(=O)NC2CCCC2C#N)CCC1 C(=O)(CCCCC(C)(C)C)NC1CCC(C(=O)NC(C#CCCC)(C)C)CC1 C1(N(C(C=COCC)=O)C)CN(C(=O)Cc2nc(C)cs2)CC1(C)C CCCCCCCCCC(=O)N1CCC(NC(=O)CN(C)CCO)C(CO)C1 C1(C(=O)NCCC2CN(C(C(C)C3CCCC3)=O)C2)CCOC1C(F)(F)F Cc1ccc2sc(=NCC3CN(C(=O)CCNC(=O)CO)CC3(C)C)[nH]c2c1C C1(CC=C)(NC(=O)CC(F)F)CN(C(=O)Cc2nnc(C)o2)C1 c1(C(=O)NC(C(C)NC(C2COC(=O)C2)=O)(C)C)nccc(C(F)(F)F)n1 CC(C)CC(F)(F)F.c1(C(=O)N)c[nH]nc1CC.C1(C(C)(F)F)(C=O)CC1 N1(C(Cc2c(C)cccc2Cl)=O)CCC2(C1)CN(C(=O)C)C2.C1(C(=O)N)CC1C C1(CC(=O)NC2(C3N(C(c4ccc(C)s4)=O)CCC3)CC2)COCCOC1 N(C(=NCCCOC)NCC1CCCN(C)C1c1ccnn1C)C(C#C)C C1(NC(C(c2ccccc2)C)=O)CN(C(C2(C)CCCS2)=O)CC1(C)C C(CN=C(NCCOC1CCSCC1)NC1C(C)C1(F)F)SC N1(C(C2CN(C(C)=O)C2)=O)CC2(C)CN(C(c3csc(C)c3C)=O)CC2(C)C1 n1(CC(C)C)nccc1NC(=O)C(C1CC(F)(F)C1)N N1(C(c2cnn(C)c2C(F)F)=O)CCCC2(C1)C(O)CC2O C1(c2n(CC=C)nnn2)(Nc2ccc(C3CC3)nc2)CCC2(CC1)CNC(=O)C2 n1(CC)nc(C(=O)NCC2CC(C)N(C(=O)CC3(CO)CC3)C2)cc1O C#CCC(CC(F)F)C(=O)N1CCOC(CC(=O)NC2(C)CCCC2(C)C)C1 c1(NC(=O)NC(c2nc(C(=O)OCC)[nH]n2)C)ccc(N(C)C)c(Cl)c1 c1(C(=O)NC(CC=CC)C(=O)NCC2CCC(CC)O2)cc(O)ccc1C C1(NC(=O)Cc2cccnc2Cl)COCCN(C(=O)CC2CCCCO2)C1 N(C1CCC(NC(C2(CF)CCC2)=O)c2ccccc21)C(C(CC)(C)C(F)F)=O c1(C(N)=O)ccc(C(N2CCOCC2C(=O)O)=O)cc1.C1CCCCC1 CC(CC(C)(C)C)C(=O)NC1CCC(C(=O)NCCOC(=N)O)CC1 CCCCC(O)CC(=O)N(CC(C)C(=O)N(C)CC1(OC)CCC1)C c1(CC=C)ccccc1C(=O)NCCc1ccccc1OC(F)(F)F CC(C(C)C(=O)NCc1nc[nH]n1)NC(=O)CCCC1CC1C c12nccnc1C(=O)N1CCC(CC1)C2.C1(C(N(C(C)C)C)=O)SCCCS1 CC1(C)Cn2[nH]c(=NC(=O)N(C3CC3)Cc3cncs3)cc2CO1 C=Cc1cnn(C)c1C(=O)NCCC1CCN(C(c2nocc2C2CC2)=O)CC1 Cn1cc(S(N)(=O)=O)cc1C(=O)NC.C1CCOC1.C(=O)CCC1CCOC1 C=CC1(C(=O)NCc2nc(C)no2)CCN(C(=O)CN2CCNC2=O)CC1 C1(CC)CN(C(=O)COc2cccnc2)CCN1C(C12CC(C1)C2)=O c1(C(=O)NC2C(C)CN(C(=O)CN3C(=O)CCC3=O)CC2)c([N+](=O)[O-])cnn1C CCCCC(O)CC(=O)NC1CC2C(NC(=O)CCc3ccc(N)cn3)C2C1 CCC(CNC(=O)CCC(=O)N1CCCCC1)N=c1ncnc2[nH][nH]c(C)c1-2 N1(c2cc(NC3CCOC(C)C3)nc(C)n2)CCC2(CC1)CN(C)C(=O)CO2 CN1CC(=O)N(CC(N2CC3C(CNC(=O)CCCC#N)C3C2)=O)C1=O C1(C(=O)NCC2N(C(Cc3n[nH]c(=N)s3)=O)CCC2)CCC2(CCOC2)O1 N1(C(c2c(C)cno2)=O)CCN(C2CN(C(=O)C(N3CCNC3=O)C)C2)CC1 Cc1nc(CNC(=O)C(C2CC=CCC2)NC(=O)C=CC2CCC2)co1 n1(CC(=O)NC2CCCC(CNC(c3nccc(C)c3)=O)C2)ncc(O)nc1=O N1(C(CC=CCCCCC)=O)CC(NC(=O)CCCCN2CCCC2)CC(F)(F)C1 c1(OC)cc(CNC(C2CC3CC3N2C(c2ncc(Br)cc2Cl)=O)=O)ccc1F c1(C(N(C)C)=O)cc(S(=O)(=O)N(C)Cc2ccccc2)c[nH]1.c12ccccc1N2 C(=O)(C(C)C(C)(C)C)N1CCC(N(C)C)C1.C1(C)(C=O)C(C)(C)C1(C)C C1(NC(=O)CC2CC2C(F)(F)F)COCC1Nc1ncccn1 c1(C(N2C3(CNc4nccc(SC)n4)CCC3CC2)=O)ccc2c(n1)CCC2 c1(CC)ccc(C(=O)NC2CCOCC2NC(=O)CCP(C)(C)=O)cc1F C1(S(N)(=O)=O)(C(=O)NCC2N(C(CCc3nc(C)c(C)o3)=O)CC=C2)CCC1 N1(C(c2c(C)cccn2)=O)CC=C(CNC(C2CC3CC2C2CC32)=O)CC1 C1(C(N2C(CCN(C(=O)C3=CCC3)C)CCCC2)=O)CCn2nncc2C1 C(=O)(C(C)(C)C(=O)N1CCSCC1C(=O)N(C(C)CC)C)OCC CC(C(C)(C)C(=O)Nn1cncn1)NC(=O)CCCCN(C)C c1(C(=O)NC2CC(C)N(C(c3nc4ccccn4n3)=O)C2)cccc2nn[nH]c12 c1(NCCC2CCC(NC(C3CC(C)=C(C)CC3)=O)C2)nc(C)nc(O)c1C c1(NC(C2(CNC(=O)C(C)=CCC)CC(=C)C2)=O)ccc(O)c(Cl)c1 C(=O)(C#CC1(C)CCCO1)N(C(CNC(Cc1c(C)cc(Br)cc1)=O)C)C C#Cc1nc(C(N2CCC(O)(CNC(c3ccco3)=O)C2)=O)cs1 C1(CNC(=O)C(c2ccc(Cl)cc2)=O)CC2CCC1N2C(c1ncc(F)cn1)=O CCCC(O)C(=O)N1CCC(C(C)CNC(=O)COCCOCC)CC1 C(=O)(C1CCCn2ccnc21)NCCOC1CCN(C(C(CC(C)(C)C)O)=O)C1 N1(C(C2CC(CC)(CC)C2)=O)CCC(CC(C)NC(C2(F)CCCOC2)=O)CC1 n1(CCOCC)nnnc1C(c1nc(C)cs1)NCC=C.c1(N)ccccc1 C(C(C)CC(=O)NC(C)(C)CCN(C)C)NC(c1c(NC)cncc1)=O c1(OC)cccc(-n2nc(C(C)C)nc2C2CCCN2C)c1 C#CCC(C)(C(=O)N(C)CC=C)NC(c1ccn(C)c1)=O c1(CC)conc1CC(=O)NCCN(C1CCCCC1)C(=O)C(F)C1CC1 C1(NC(C(CC=C)CC)=O)CN(C(=O)Cc2cn[nH]c2)CC12CCC2 C1(CNC(C(c2ccc(F)cc2)(C)F)=O)COCCN1C(C1CC2CCC1O2)=O c1(C(N2CCC2(C)C2CC2)C(=O)NCCCC)cc(Cl)cc(Cl)n1 c1(C(=O)NC2C(C)CN(C(=O)CCc3cncs3)C2)c[nH]c2c(C#N)cccc12 c1(C(N(CCC)CC2CCN(C3(C)CCOC(C)C3)C2)=O)ncc2[nH]ncc2n1 c1(C(=O)N)cc(O)cc(=O)o1.C1(NC(c2cn(CCC=C)nn2)=O)CCCCC1 C12(C(=O)NCC3CN(C(C45CC(F)(C4)C5)=O)C3)CCCC(=O)N1CCC2 C=CCC(CC=C)C(=O)N1CCCCC1CC(=O)NC1CCC2(CC1)N=N2 CC1CN(C(C2CC2(C)C(F)F)=O)CCCN1C(=O)COCC(F)F Cn1cnc(C(=O)NCC(=C2CN(C(c3c[nH][nH]c3=N)=O)C2)F)c1 CCC(C)(C)CCCC(=O)NCCC1CCCN1Cc1cccc(C)c1 CC(C)CC(C(=O)NC1(CCF)CC1)ONC(C1CCCCCC1)=O C1(C(=O)NC2CCN(C(CNC(=O)OCC)=O)C2)CCc2nnn(C)c2C1 N1(C(=O)OC(C)(C)C)CC2(CCCC2)CC1CNC(C1(C)CCOCC1)=O c1(C(=O)NC2(C)CCN(C(c3cnc(C(C)C)s3)=O)C2)cnc(O)c(F)c1 C1(N(C(C=NOC)=O)CC(C)C)CCN(CC(=O)N(C2CCC(=O)N2C)C)CC1 N1(C(Cn2c(CCC)ncc2)=O)CCC(NC(c2ccc(C)nn2)=O)C(F)C1 c1(C(=O)OC)cnc(NC(C2CC3CC(=O)C2O3)=O)c(Br)c1 N1(C(C2CC(O)(CNC(C(CCC)(C)C)=O)C2)=O)Cc2cccc(C)c2C1 c1(C(=O)N)ccc(S(F)(F)(F)(F)F)cc1.C1(CNC(C=NOC)=O)CCCCC1 c1(C(=O)NC2CCN(C(CNS(NC)(=O)=O)=O)CC2C)nn2c(c1C)CCCC2 C(C1=CCN(C(C2CCCCO2)=O)CC1)NC(c1n(C)nnc1Br)=O c1(C(C)NC(CN(C(C(C)C)=O)C)=O)ccc(C)cc1.C(=O)(C1=CCOC1)N c1(CCC(=O)NCC(CNC(C2CCOC2C2CC2)=O)OC)ccccn1 C1(C(N2CC(CNC(C3CCOC3)=O)C3(C2)CC3)=O)CN2CCCN1CC2 c1(CC)ccc(C(N2CCC(NC(C3SCCS3)=O)CC2C)=O)cc1C#N C1(CC)CN(C(C2CC3CCC2O3)=O)CCC1NC(=O)CNC(=O)NC c1(C(N(C2CCN(C(=O)C(C)(O)CC(C)C)CC2)CC)=O)cnc2ccccn12 N1(C(c2ccc(CC)cc2)=O)CC(OC)CC(NC(C2(C)CCN(C)CC2)=O)C1 c1(C(N2CCC3(C(C(N4C(C)(C)CC(O)C4)=O)C3)C2)=O)c(O)cc(O)cc1O CCC(CCCC(=O)Nc1cccc2c1CCO2)NC(=O)CC(C)(O)CCC N1(C(CC(C)CNC(c2cc(CO)ccn2)=O)=O)CC2CCCC(C2)C1 CC1CC=C(C(=O)NCC(CC2CCCC2)C(=O)Nc2cnsc2)CC1 N1(C(C2CN(C)C(=O)N2)=O)CCCC(C(=O)NC2CCCNC2=O)CC1 C(c1cccc(F)c1Cl)=CC(=O)NCC(C)NC(C1(C)CCCOC1)=O N1(C(C(C(C)O)C)=O)CC2CCC(CNC(C3CC=CCC3C)=O)C2C1 c1(C(C(=O)NCC(F)F)N(C)Cc2cc(CC)no2)ccccc1Br C#CC1CN(C(c2ccc(C3CC3)s2)=O)CCN1C(=O)C(COC)CC Cc1cc(=O)n(C)nc1C(=O)NCC.C1(CC(=O)N)CCCCCO1.C1CC1 CN1CCCC2CN(C(C3(C4=CCN(C(=O)OC(C)(C)C)CC4)CC3)=O)CCC12 C(c1cccc(F)c1)=CCC=O.CCCC(C)C.C(C)(C)(C=CC(=O)N)SC Cc1c(NCc2cccc(O)n2)nc[nH]c1=NCc1nc(-c2cccnc2)cs1 C1(CC(=O)NC(C)CN(C)C(c2ccc(C(=O)N(C)C)s2)=O)CCOCC1 CC1(C(=O)NC2CC(CC(=O)N(C3CCCC3)CCO)C2)CC2C=CC1C2 c1(C(=O)NC(C(c2ccc(Cl)cc2)OC)C)ccc(S(C)(=O)=O)c(F)c1O CCC(COC)C(=O)N1CCC(CCNC(c2cc(CCO)on2)=O)CC1 C=CCC(CNC(c1c[nH]nc1C(F)(F)F)=O)NC(=O)C(F)C.C=O.N c1(OCC)cccc(OCC(=O)NCC(O)C)c1.C1(CC=O)CCC=CCC1 c1(N2C(CN(C)C(c3cc(CF)on3)=O)COCC2)nc(Cl)ncc1[N+](=O)[O-] c1(N2CCC(C)(NC(C3=C(C)CCC3)=O)C2)nc(C(F)(F)F)nc2[nH]cnc12 O=C(CCC(CF)CF)NC(C(=O)NCc1ccnc(O)c1)c1ccco1 C1(NC(Cc2nc(C)sc2)=O)CCCCN(C(c2ccc(O)c(Br)c2)=O)C1 c1cccc(Cl)c1O.C1(CNC(c2cccn2C2CC2)=O)CCC(C(=O)N)O1 CC1CCC(NC(=O)CCC2CCCC(O)C2)CN1C(C1CCCN(C)C1)=O c1(C(C(=O)NCC(CNC(c2c(Cl)ncc(C)c2)=O)C)C)cc2ccccc2s1 c1(NC(C)CCNC(c2ncc(F)cc2F)=O)ncc(Cl)cc1[N+](=O)[O-] C(=O)(CC(C)C(F)(F)F)NC(C1CCCC1)CNC(c1c(C)[nH]c(C#N)c1)=O N1(C(CC2C(C)OCC2)=O)CCC(C)(C)C1C(=O)N(C(C(N)=O)C1CC1)C c1(OC)cnc(F)c(C(=O)NCC2CCCC2)c1.C1(C=O)CCC(C)(C)CC1 CCC(O)(CC(=O)NC(C1CN(C(=O)C(C)(C)COC)C1)C)c1ccccc1 C1(C(=O)NCC(C(CC)N(C)C)=O)CNC(=O)CC12CCOC2 C1(C(N2CC(O)C2)=O)CCC(C)NC1=O.N1(C(C)=O)CC(OCC(=O)NC)C1 N1(C(C2N(CC)CC2)=O)CCC(NC(=O)C(n2ccc(C3CC3)n2)C)C1(C)C C(=O)(C(C)(F)C(F)(F)F)NCC1(C)CCCN(C(c2c(C)nc[nH]2)=O)C1 C1(CC=O)CCN(C)C1=O.C(CCCc1ccccc1)NC(C(=O)NCC)=O N1(C(CC2(COC)CC2)=O)CCCCC(N(C(=O)CC2C(=O)NN=C2C)C)C1 C1(NC(=O)NC2CC3(CC3)C2)CC2(CCC2)C1 N1(C(c2c(=O)ccn(C)c2)=O)CCCC2(CCN(C(=O)COC(F)F)C2)C1 CN1CCC(N2CC(NCC3CC4CCCC34)CC2=O)CC1 c1(CC)cc(NCC2CCCN(CCC3CCOC3)C2)n2ncnc2n1 C(=O)CC(C)(O)C(F)(F)F.C(C(=O)N(C)CCOCCC)N(CCOC)C C(=O)(C(C)CC(C)C)NC1CC2(CC(OC)C2)C1.C(=O)C(C)(O)C(F)(F)F C1(CC)CCN(C(=O)CCOC(C)=O)C(C(N2CC(C#N)(CCF)C2)=O)C1 C1(O)(CN(C(C(CSC)C)=O)C)CCCN(C(=O)C=Cc2c(C)coc2C)C1 N1(C(c2cnoc2C)=O)CC(C)CN(C(=O)CN(C)S(N)(=O)=O)C(C)C1.C C=CCC(C)(C)CNC(=O)C(F)C1CC(NC(=O)CC2(C)CCCCC2)C1 c1(C(=O)N)cc([N+](=O)[O-])n[nH]1.C1(CC(N2CCC(F)C2)=O)CC(O)C12CCC2 N1(C(C(C)SC(CC)(C)C)=O)CC2C3CCC(C(NC(=O)CCSC)C3)C2C1 C(=O)(CCCC(=O)N1CCC(C2CCCCN2C(c2ccc(O)nn2)=O)C1)OC C1(NCC(COCC)O)CCOC1N(C)CC CC1C(C(=O)Nc2cccc(CCO)c2)CCN1C(c1cnn(C)n1)=O CC1CC(NC(=O)CCC=Cc2ccccc2)CCN1C(=O)CSC(F)F CCC(O)C(C)C(=O)N(C1CCN(C(=O)C=C(C)c2cnn(C)c2)CC1)C C1(F)(C(N(C2(C=O)CC2)C)=O)CCCCC1.C1(C(=O)OCC)CCCC1.C CC(C)(C#N)CCC(=O)N1CC(NC(=O)C=Cc2ccsc2)C2CCCC12 C1(NC(CC2C=NN(C)C2=O)=O)CCN(C(c2ccc([N+](=O)[O-])o2)=O)C1(C)C C(=O)(C(CCSC)NC(N)=O)NC(C1N(C(COC)=O)CCC1)(C)C CN1CCCC1C(=O)NCC1CCC1.C1(CC=O)CCC(C(F)(F)F)O1.N N1(C(c2ncc(C)nc2)=O)CCC2(CCCN(C(C34CSCC3C4)=O)C2)C1 N1(C(=O)Nc2c(C(=O)OC)nc(Br)cc2)CCN2C(=O)OCC2(C)C1 CN1CC(=O)N(CC(=O)NC2(C3CN(C(c4cccc(F)c4Cl)=O)C3)CC2)C1=O N1(C(C(CC2CC2)OC)=O)CCC2CCCC12C(=O)NCC1CCN(C)C1 CC1(C)CC(NC(C2CCCC2)=O)CN(C(c2ccc(-n3ccnc3)nc2)=O)C1 c1(NC(CNC(=O)CS(=O)(=O)C2CC2)C2CC2)ccc(Cl)cc1[N+](=O)[O-] Cc1nocc1C(=O)NCC1CCC1NC(=O)CSCCN(C)C C(C1=NOC2CCCC12)NC(CC(CNC(c1[nH]cc(C)c1C)=O)C)=O c1(NC(C(C=C)O)=O)ccc(C(C)NC(c2cccc(C)c2)=O)cc1 C(c1ccccc1C#N)=CC(=O)NCC(CNC(C(C(C)O)(C)C)=O)O c1(N(CC(Cl)Cl)C)ncccc1S(=O)(=O)NC(Cc1nccs1)CO C12(C(=O)NCC(C(=O)NCc3cnn(CC)c3C)C)CCCN(CC1)C2 CC1CN(C(C2CC2NC(c2ccc(O)c(O)c2)=O)=O)CCC1O CC(CNC(=O)Cc1ccoc1)C(=O)NC1C(O)CC1O C1(CCNC(=O)OC(C)(C)C)CCCCC1C=O.c1ccc(C(F)F)nc1.N C1(C(N(CCC=O)CCCO)=O)CCC(=O)CC1C.C1(C(=O)N)CC1.CCC c1(C(=O)NC2CCN(C(c3n(C)nc(O)c3)=O)CC2F)cc2n(n1)CCCC2O C(C=O)(C(C)(C)C)OC.Cc1ccn(CC(=O)NCC2CN(C(=O)O)C2)n1 C1(C(NOCC=C)=O)C(CC)CCN1C(=O)COC(C)=O c1(C(N2CCN(C(C(C)n3cccc3)=O)C3(C2)CC3)=O)ccc2c(c1)CCOC2 N1(C(C2(C=C)CCCC2)=O)CCOCC(C(=O)NCCOC2CC=CC2)C1 c1(OC)c(Cl)cc(C(=O)NC2CC2NC(C2CCCC2(C)C)=O)cc1Cl C1(C(=O)NCc2c[nH]nc2C(N2CC(CCO)C2)=O)CC2C=CC1C2 C1(C(=O)NC2CCC(NC(c3c(C#N)ccs3)=O)CC2)CCCCC1(F)F N1(C(CC=CC=C)=O)CCC(CO)(NC(=O)C(C)Cc2ccc(OC)cc2)C1 C(=O)(C(F)C(C)(C)O)NCC1(C(N2C(CC(C)C)COCC2)=O)CC=CC1 c1(C(N2CC(N(C(CCNC(=O)NC)=O)C)C2)=O)ccn2ccnc2n1 CCC(C)C(C(=O)N1CC(OCCO)C1)NC(C1C(C)OC(C)C1C)=O c1(C(N2CCC(CC=C)(NC(c3ncoc3CC)=O)C2)=O)cc(F)cc(N)c1N Cc1cc(C(=O)NC)n(C2CCOCC2)n1.c1(CC(N2CCC2)=O)cnn(C)c1 C1(CCC)CN(C(C2(C)CCCS2)=O)CC1NC(=O)CC1(CO)CC1 C1(NC(C2COCCO2)=O)CCC12CCN(C(c1ccoc1Cl)=O)CC2 C1(NC(c2c(C)cccn2)=O)CCSC12CN(C(=O)CC1CCCC(=O)N1)C2 c1(C(=O)OC)cc(C(=O)NC(C)(C)CCC)ccc1F.C(=O)(C(C)C(C)C)N c1(CNc2ccc(CCCCC)cc2)ccc2ncccc2n1 c1(OC)cccc(C(N2CCC2C(=O)NC(c2nccs2)C)=O)n1 C1CN(C(=O)C(O)P(C)(C)=O)CC2(CCC2)O1.c1(CC)noc(C)c1C(=O)N N1(C(CC(C)OC)=O)CCN(c2nc(Cl)ncc2Br)CC(O)C1 C1(C(=O)NC2C(OC)CCOC2)CN(C(=O)C(=O)CC(C)C)CC(C)(C)C1 CC1(C)CN(C(=O)CCc2ccc(Br)cc2Cl)CC(C)(C(F)(F)F)O1 c1(CC(=O)N(C2CCN(CCn3ncc(C)c3)C2)C(C)C)ccccc1I c1(C(CNC(C(=O)NCCCN(CCOC)CC)=O)O)cc(O)ccc1F Nc1ccc(-c2cn(Cc3noc(C4CCN(C5CC5)CC4)n3)nn2)nc1 S(=O)(=O)(C1CCCNC1)NC(c1ccc(CC)cc1)CC(C)C c1(-c2cn(C3CCN(C(=O)Cc4ccsc4)C3)nn2)ccc(OC(F)(F)F)cc1 c1(C(C)C)ccccc1-n1nc(C(O)CC)nc1C1CC1Cl C1(C)(C(N2CC(C)C2)=O)CCN(C(=O)CC2CCSC2)CC1 C1(CNC(Cn2c(C)nnn2)=O)CN(C(c2ccnn2C2CCC2)=O)CCC1C c1(CNC(=O)CC2CCSCC2)ccc(C(=O)NCC2CC2(Cl)Cl)cn1 c1(C(=O)NC(C(C)NC(c2ccnc(OC)c2F)=O)C)ccc(C=NOC)cc1 C1(CC)C(=O)N(C)CCN1C(C1CN(C(=O)CCc2ccc[nH]2)CC1(C)C)=O CC1CC(CNC(=O)C(C)c2cccs2)CN1C(c1conc1C1CCC1)=O C1(NC(CCC(=O)NC)=O)C2CC3CN(C(C4CC(n5cccn5)C4)=O)C1C3C2 c1(NC(CC2(C)CN(C(C(C)(C)C)=O)C2)=O)c([N+](=O)[O-])ccc(F)c1F O=C(CCC=CBr)NCCCCCNC(c1conc1C1CCCO1)=O N1(C(C(C)CN(C)C)=O)CC(C2CCCN(C(C34CC(CN3CCC)C4)=O)C2)C1 C1CCN(C(=O)C=C2CCOCC2)C1.C1(Cl)(C(=O)OCC)CC1C=O.N CC(=O)n1ncc2c(NC(c3coc(CC4CC4)n3)=O)cccc12 c1(CC=O)ccc([N+](=O)[O-])cc1Cl.CC1COC(C(=O)N)C1.C12CC(C1)C2.C C1(C)(C=O)CN(C(=O)CCN2CCOC2=O)C(C)(C)C1.CCCC(=O)N(C)C.N C(=O)(C1=C(Cl)CCCC1)NC1CCC(CCC(=O)NCC(C)SC)C1 C(CCCCC(=O)NCC(O)CCNC(=O)C(C)CN1CCOCC1)NC(C)=O CCCC(CCC)NC(=O)C(C1CC=CCC1)NC(=O)Cn1nc(C)cc1C C1(F)(CNC(C=C(CC)CC)=O)CCCN(C(C2(CF)COC2)=O)C1 CCC1=C(C(=O)NCC(F)CNC(c2nc(O)c(C)s2)=O)SCCO1 C(CS(=O)(=O)c1ccc(F)cc1)C(=O)NCc1c(C(=O)O)nc(C(=O)O)cc1 C(=O)(C(C)(C)C(C)(C)O)N1CC(C(=O)NCC2(CCC=C)CC2)C(C=C)C1 Cn1cncc1NC1(C(=O)NC2CCC(NC=O)C2)CC1.C(C)(C)C.O c1(CNC(Cc2c(CC)con2)=O)ccc(NC(C23CCCC2C3)=O)cc1 C1(C(=O)NCC(C)NC(=O)Cc2c[nH]c(=N)nc2O)CC2(CCOC2)C1 C(C(COC)C(=O)NC1(C(N2CCN(CCO)CC2)=O)CC(F)C1)OCC N1(C(C(=O)NCCCC)CC2CCCC(C)(C)C2)CCS(=O)(=O)C(C)C1 C(=O)C(C)S(=O)(=O)C(C)C.c1(CCC)ccc(N)c(C(=O)N)c1.C1CC1.C c1(CNC(C2CC2(C)C)CC)nc2ccc(F)c(F)c2[nH]1 c1(C(C(=O)NCC(=O)NC2(C(=O)OC)CC2)F)ccccc1 CC(C)CCC(O)C(=O)NC(CCN(C)C)C(=O)N(C1CCCC(C)C1C)C c1(OCC)cc(C(N2CCCC2CCC(=O)N2CCC2CC(=O)OC)=O)on1 Cc1ncc2c(n1)CCC(NC(N1CC(O)C(O)C1(C)C)=O)C2 Cc1ccc(C(C)C(=O)NC2CC2CNC(c2cncs2)=O)cc1.C1CC1 Cc1cc(CC(N2CCC3C(NC(=O)C(F)=CCCF)C23)=O)c(C)s1 N1(C(=O)CCC2CCCOC2)CCCN(C(c2cnc(C(F)(F)F)nc2)=O)CC1 C1(NC(C(CCC)N(C)C)=O)CN(C(=O)CSCc2nccs2)CC12CCC2 c1(OC)c(CN2CC3CC2CS3=O)cc(Cl)cc1Cl N1(C(Cc2c(C)n[nH]c2)=O)CC2(CNC(c3cnc(C4CC4)s3)=O)CC1CO2 c1(C(C(=O)NCC2(CNC(CC)=O)CCCC2)C)c(Cl)cccc1Cl C(=O)(C1CCCc2cccnc21)N(CC(C)(C)Nc1ncnc2[nH]cnc12)C c1(C(=O)NCC2CCN(C(COC(C)=O)=O)C2)cn2ccc(F)c(C)c2n1 C1(NC(C2(C(C)C)CC2)=O)CCC(O)CN(C(c2nn[nH]c2C(F)(F)F)=O)C1 c1(OCCC(CC=C)(C)C)ccc([N+](=O)[O-])nc1 Cn1cc(C(=O)NC2CCC2NC(c2ccsn2)=O)nc1O C12(C(N3CC(O)CCCC3)=O)CC3CC(C(=O)N1)C2C3.C1(C(=O)N)CC(O)C1 CCCC(C(=O)OC)C(=O)N1CCCCC1CNC(=O)C(C)(O)C1CCC1 Cc1ccc(Cl)c(C(=O)NCCC2CC2)c1O.c1(CCC(=O)N)ccc(Cl)cc1 C1(CC)CN(C(=O)CCc2nc(C)no2)CC1C(=O)NCC1CCCC(C)O1 C#CCN(OC)C(=O)C(Cc1cn[nH]c1)NC(c1ccc(C#N)n1C)=O c1(C(N2CC(NC(C3(C)CC(F)(F)C3)=O)C(CO)C2)=O)n[nH]c2c1CCOC2 c1(C(=O)N)ccc(C)nc1O.C(=O)(CC(C)(O)Cc1ccccc1)N(CC)CC C1(CNC(c2ccc(CCF)cc2)=O)CCCC(NC(c2cccnc2S)=O)C1 c1(CNC(N2CCC3(CCC3)C2)=O)ccc2cccnc2n1 C1(NC(c2cc(OCC)ncc2)=O)CCC(C)CC1.C1(CC=O)CCSCC1.N C1(C(=O)NCC(C2CCCC2)NC(C(N)=O)=O)CC(Cl)(Cl)C1 CC(CNC(c1ccccc1)=O)S(C)(=O)=O.c1(C=O)ccc(C2CC2)cc1.C N1(C(C=CCC)=O)CCCC2CN(C(c3nn(CC)cc3[N+](=O)[O-])=O)CC12 Cc1occ(C(F)(F)F)c1CC(=O)NC1(C)CCCC1.C1(C=O)CCC(F)C1 N1(C(C(CC(=C)Cl)NC(c2cc(CC)no2)=O)=O)CC2(CCC2(C)C)C1 CC1(C)CN(C(=O)Cc2c[nH]ccc2=O)CCC1NC(c1ccno1)=O c1(C(N2C(C(=O)NC(COC)C)CC(F)C2)=O)cccc([N+](=O)[O-])c1O C1(C)(CC)COCCC1NC(C1(NC(c2cc([N+](=O)[O-])n[nH]2)=O)CCC1)=O N1(C(C(c2cn(CC)nc2)=O)=O)CCCC2(CC2)C1.C1(C(=O)N)CCCC(O)C1 c1(NC(c2c(CC)[nH]nc2)=O)ccc(NC(=O)C(C)(C2CC2)O)c(C)c1 c1(CC)ccc(C(N2CCCC(CCO)C2)=O)cc1 c1(C(N(C)C)=O)ccc(OCC(C)(C)COC2CCOCC2)cc1 c1(CC)c(C(=O)NCCNC(c2cc(C3CCOCC3)nn2C)=O)cccc1F Cc1c(C(=O)NCC(O)CC(=O)NCc2ccc(CO)o2)cccc1O n1(CC(=O)N)nnc(=O)[nH]1.C(C(=O)N1CC(CC)C1)(C1CCOC1)OCC C1(NC(CCc2cnc(C)s2)=O)CCN(C(c2cnc(C)[nH]2)=O)CCC1CO C(CCCC(=O)N1CC=CC1CF)N(C(c1c(C)scn1)=O)C N1(C(CC2(C)CCCC2)=O)CC2(CCCCN2C(c2ccnc(Br)c2F)=O)C1 N1(C(=O)OC(C)(C)C)CC(C2(OC(C3CCN(c4ncccn4)C3)=O)CC2)C1 CCCCC(CNC(=O)COc1ccc(Cl)cc1)NC(C1(C)CCCOC1)=O c1(OC)ccc(OC(C)C(=O)N2CCC2C(=O)Nc2ccc(O)cc2)cc1 C1(C(N(CC)Cc2csc(-c3ccccc3)n2)=O)CCCOC1CC(=O)O C1(NC(C(C2CCN(C(=O)C(c3ccnn3C)C)CC2)C)=O)C(C)(C)C1(C)C c1(C(=O)NCC2CCN(C(=O)CN3CCCCC3=O)C2)n[nH]c2ccc(Cl)cc12 CCC(C)(CNC(c1coc(C)c1)=O)C(C)O.C1(O)(CC(=O)N)CCCC1 N1(C(=O)C=Cc2ccc(C(F)F)o2)CCC2CN(C(C3CCOC3)=O)CC2C1 CC1CCN(C(=O)CSCc2ncc[nH]2)CC1CNC(C1OCCCO1)=O c1(OC)cnc(Cl)cc1C(=O)NC1CC(NC(C2CCC(=O)C2)=O)CC1O O=C(C1=CS(=O)(=O)CCC1)NCC1CCC(NC(c2nncs2)=O)C1 N1(C(CC2CCN(C)CC2)=O)C2CCC1CC(NC(C1(F)CCOC1)=O)C2 c1(OCC)cc(NC2CCCC(NC(=O)CCC(C)C)C2)ncn1 Cc1cc(C)c(C(=O)NC2CCC(O)C2)c(C)c1.c1(C=O)nn(C)c(C)c1Cl.N C1(CCC)(NC(c2ncc(OC)cn2)=O)CCCN(C(=O)C(C)(C)c2ccsc2)C1 CCC(CC(=O)N(C1CCCC1)CCNC(=O)C(N1CCCCCC1)C)C1CC1 c1(C(C(=O)NCC(n2ccnn2)C)(F)F)c(F)cccc1F.N(CCO)CCO.C CC(CC(N)=O)C(=O)NCCC1(O)CCN(C(=O)C=C2CCCCC2)C1 C(=O)(C(F)(F)C(F)(F)C(F)F)N(CC(=O)Nc1cn2cc(C)nc2cc1)C C1(C(=O)NCCOC)CC2CCC1N2C(=O)CCc1ccc(C2CC2C)o1 C1(NC(C2CCCN(C(N)=O)C2)=O)CN(C(C2CNC(=O)O2)=O)CC2(CCC2)C1 C(C1CN(C(=O)C(C)(C)N(C)C)CC1C(N1CCC(c2cc[nH]n2)C1)=O)=CC c1(SC)ccc([N+](=O)[O-])cc1C(N1CCC(N(CCC(F)(F)F)C)C1)=O C1(C(=O)NCCC#C)CCN(C(=O)C=NOC)C12CCC2 C(=O)(CCC(C#N)NS(=O)(=O)C1(CC2CC2)CC1)OC(C)(C)C Cc1cc(OC(C)C)c(-c2cc(C(=O)Nc3ccc(Cl)c(Br)c3)n[nH]2)cc1C c1(NC(CC(CC)O)=O)nc(Cl)ccc1C(=O)Nc1cnc(OC)nc1 C(=O)(C(C)(C)CN(C)C(C12CCC(C1)C2)=O)N(CCC=C)CC CC1CC(NC(c2cccc(C3CC3)c2Cl)=O)CCN1C(=O)Cc1cc[nH]c1 C1(CCC)(NC(=O)C(c2cccc(OC)c2)C)CCCN(C(=O)CCCOC)C1 C1(CC(N2CC(C)SCC2)=O)CC(C)(C)CN1C(=O)C#CC(C)(C)O C1(O)(CNC(C2(CO)CC(C)(C)C2)=O)CCCN(C(c2ncncc2Cl)=O)CC1 c1(C(=O)N)nn(CC(F)F)cc1[N+](=O)[O-].C1(NC(CCSCC)=O)CCCCC1 c1(C(N2CCN(c3cncs3)CC2)C(=O)N(C)C2CC2)ccc(Cl)c(Cl)c1 C1(c2nnnn2C2CCCC2)(Nc2c(C)n[nH]c2C)CC(O)C1(C)C CCCCC(C(=O)NC(C)C(C)n1cccn1)NC(=O)C(C)CSC C(N=c1nc(N2CCC(C3CC3)CC2)c2c([nH]1)CCC(C)C2)c1c(OC)ccs1 N1(C(C(C(CC)C)O)=O)C2CCCC1CN(C(c1ccc(C)c(C#N)c1)=O)C2 C1(NC(C(COC(C)C)(C)C)=O)COC2CCOC12.C(=O)(C)N.C(C)(C)C Cc1ccc(N(C)C(C2CCOCC2NC(c2cnn[nH]2)=O)=O)c(C)c1 CC1C2CC(C2NC(=O)CCCSc2ccccc2Cl)N1C(=O)C#CC(C)(C)O C(=O)(C(C)C(C)(F)F)N1CC(CN(C(C2(CCOC)CCCC2)=O)C)C1 c1(CC(=O)NC2(CNC(=O)CC3CC3)CC2)cc(C2CC2)no1 N1(C(CCCC=C)=O)CC2CC(NC(c3ccc(S(C)=O)cc3)=O)CC1C2 C1(NC(C(=O)N(CC(c2cc(C)c(O)cc2)O)C)=O)C2Cc3c(Br)cccc3C12 C1(NC(c2cc(C)sc2)=O)CCC12CCN(C(=O)C(C)c1ncco1)CC2 Cc1c(C(F)(F)F)n[nH]c1C=O.C1C(Cl)(Cl)C12CC2.C1(O)(CC)CN(C)C1 N1(C(C(C(C)C)F)=O)CCC(O)(CN(C(=O)CCC2CCCN2C)C)CC1 CC(C)CC(C)CC(=O)NCC1(C(=O)NC2CC(F)C2)CC=CC1 c1(C(=O)OC)c[nH]c(C)cc1=NC(C)CN(C)C(c1cccn2nncc12)=O c1(C(=O)OC)cc(Br)ccc1NC(C1CC1NCc1c(F)cccc1I)=O N1(C(=O)Cc2ccc(F)c(Cl)c2)CC(C2CCCN(C(=O)C(Cl)(Cl)Cl)C2)C1 C(CO)(CCCCNC(C1(C)SCCCS1)=O)NC(COC(CC)(C)C)=O c1(C=O)cccc(S(=O)(=O)N2CCC(O)(C=O)CC2)c1.C1CCS(=O)(=O)C1 CC(C)C(C(=O)N1CC(F)(CNC(C23CSCC2C3)=O)C1)NC=O CC1CN(C)CC1N=c1[nH]c(=NCc2cc(Br)ccn2)[nH]c2c1SCC2 N1(C(C=CSC)=O)CC(CNC(=O)C(C=O)C(C)C)C2(CCC2)C1.C(C)(C)C N1(C(C(C)OC)=O)CCN(C(c2cc(C3CC3)ns2)=O)C2COCC12 C1(NC(COCCC(C)C)=O)CCCC(C)C1.c1(CCC=O)cncc(O)c1.N C(=O)(C(C)CC(=O)OC)NCC1(C(=O)NCCCC#C)CCOCC1 C12(NC(=O)Cc3ccccn3)CCOCC1CN(C(=O)C#CC1CCCOC1)C2 C1(C)(CNC(C2(CC)CC2)=O)CCCN1C(=O)C=C1CCN(C)CC1 Cc1cc(N2CCCC(C(c3ccc(Br)cn3)O)C2)nc(-c2ccncc2)n1 CN=c1nc(N2CCC(C)(C(N)=O)C2)[nH]c(N2CC(CO)C3(CC3)C2)n1 Cc1cc(C(=O)NC2CCN(C(=O)C(C)(C)O)CC2)cc(O)c1 C1(C(=O)NC(C)CCNC(=O)C(F)=CC2CC2)CCC2CC1C2(C)C CC1(C)CC(N(c2cc(Cl)nn2-c2ncccc2Cl)CC)CN(C=O)C1.C(C)(C)C C1(CC)(CNC(C2CC2C)=O)CCN(C(=O)CCC=O)CC1.C(C)(C)C.C C1(NC(c2ccnc(C)c2C)=O)COC2CN(C(=O)CC3CCOCC3)CC12 N1(C(C=CCN(CC)CC)=O)CCCC2(CC2)C1.C(=O)C(C)CC(C)(C)C N1(C(c2c(OC)n[nH]c2)=O)CC(CNC(C2(C)CCOC2)=O)C2(CCC2)C1 CC(C)C(C(=O)NC1(C)CN(c2ncnc(=N)[nH]2)C1)NS(C)(=O)=O N1(C(c2n[nH]c3c2COC3)=O)CCC2CCCC12C(=O)NCc1ccc(Cl)o1 c1(C(=O)NCCC2CC(C)N(C(=O)CS(C)(=O)=O)CC2)cc2c(cc1N)CCC2 C=CCCC(C)(C)CC(C=CC(N1C(C(=O)NCC)CC(F)CC1)=O)=O c1(CC)ccc(NC(C2CN(C(=O)Cc3cscn3)C2)=O)cc1I c1(C(N(C2CC(NC(=O)CCc3nccn3C)C2)C)=O)cnnc(C2CC2)c1 C(=O)(CC(C)(C)C)N.CCCCNC(C1CC(O)C1)=O.C(C)(C)C.C=O CC1=CCCN(C(=O)C(CO)NC(=O)CC(O)C2CCCC2)C1 C(=O)(CC1=NNC(=O)C1)NC1(CC=C)CCN(C(=O)CCCCN2CCOCC2)C1 c1(C(=O)NCC2N(C(CCCOC(C)C)=O)CC3(CC3)C2)cccc2c1OCC2 C1(C=O)CC(C(C)(C)C)=NO1.C1(CCNC(C2(CC)CC2)=O)CCC1.N N1(CC(=O)NC(C)CCCc2cccnc2)CCS(=O)CC1 C1(NC(C(C)OCCOCC)=O)CCC2(CC1)CC2.c1cccc(F)c1C#N c1(CN2CCOCC(C(=O)NC(CC(=O)OC)C)C2)ccc(F)c(O)c1F N1(C(C2CC(CC)OCC2)=O)CC2CN(C(=O)C(C)CCCOC)CC2C1 N(C(=NCCF)N(C)Cc1nnnn1C)Cc1c(C)cc(Br)cc1 N1(C(CC=CC)=O)CC(C)N(C(=O)Cc2cc(C)on2)C(C)C1 CC(C)CC(CNC(=O)CSCCOCCF)C(=O)Nc1cscn1 CCCCCC(F)C(=O)NC12CC(CNC(=O)C(O)Cc3ccccc3)(C1)C2 C=CC1(CC(N2CC(O)(CNC(c3n[nH]cc3-c3ccncc3)=O)C2)=O)CCC1 CC1CN(C(c2cccc(SCC#N)c2)=O)CCN1C(C1(CO)CCCO1)=O C(C(CC1CCCC1)C(=O)NCc1cnc[nH]1)NC(=O)C=C1CCC1 c1(C2OCCN(Cc3ccc(=O)n(C4CCNC4)n3)C2)cc(F)c(Cl)cc1Cl c1(C(C)C)ccc(Br)c(CNC2CCCC(O)C2)c1 c1(C(=O)NCC(C)N(C(C(CC)C(F)(F)F)=O)C)n[nH]c2c1CS(=O)(=O)CC2 C1(NC(CCCCC(N)=O)=O)Cc2ccccc2C1NC(=O)CC1C=CCC1 C#Cc1ccc(CN(C(C)CO)C)c(F)c1F.c12ccc(c(OC)c1)OC2 Cc1cccc2ncc(C(=O)NC3CCC(CNC(=O)CCc4cncs4)C3)n12 c1(NC(CC)C2CC2)nccc(N2CCC(CSC)CC2)n1 C1(C(=O)O)(NC(=O)NCCc2sccc2Cl)CC2CCC1C2 CCC(CCCC(=O)OC)NC(c1cc(Br)c(NC(=O)OC(C)(C)C)s1)=O c1(N(C)C)ccc(C(=O)NCC2CCCN2C(c2cnccc2Br)=O)nn1 C(C(=O)NCCC1(C)CC1)(C(C)(C)O)NC(CC(CC)OC)=O N1(C(c2ncc3[nH]ncc3n2)=O)CCC2(CNC(C3(O)CC3)=O)CCCCC12 Cc1nc(C2CC2)ncc1C(=O)NCC(O)C.c1(C=O)ccn(CC(C)C)n1.N CC1CCN(C(c2ccn(C3CC3)n2)=O)CC1C(=O)NCCCNC(N)=O CC(=O)n1ncc2nc(NC3(c4ccccc4[N+](=O)[O-])CCC3)ncc12 CCCCC(CC)C(=O)NC1CC2(C1)CN(C(=O)CC1Cc3ccccc3O1)C2 CN(O)C(=O)CNC(=O)C(C1CC1)N(C)C(C1CCNC1=O)=O c1(C(=O)NC(C)C(C)NC(c2cnc3[nH]ncc3c2)=O)n[nH]c2c1C(=O)CCC2 N1(C(CC(C)SC)C(=O)NCC2CC2)CC2CCCC1C2 c1(C(N2CCCCC2CC(C)O)C(=O)NC)cc(OC)c(OC)c(OC)c1 c1(C(CNC(c2nc(Cl)cs2)=O)NC(Cc2c(C)ccs2)=O)ccccc1F CC1CN(C(C(=O)NCC(F)F)c2cnn[nH]2)c2cccc(Cl)c2O1 C1(CNC(C2CCN(c3ccccc3)C2)=O)CCOCC1.C1(O)(C=O)CCC1.N C(=O)(N(CCCO)OC)C1(CF)CCN(C(C=CC(CC)C)=O)C1 C(=O)(C(CC(C)C)C1CC1)N1C(CC2N(C(CCCC)=O)CCC2)CCCC1 CC(F)(C(=O)N1CC(NC(c2cc3cccnc3o2)=O)C(O)C1)C(F)(F)F C1(C)(CC=O)CCN(C(C2CC3C=CC2O3)=O)C1.n1(CC=C)cc(C)nn1.N N1(C(CCCOCC)=O)CC2CC(NC(c3c(OC(F)F)cccc3F)=O)C2C1 N1(C(C(=O)N(C)C)=O)CCC(C(N2CC(CC3CC3)C(N)C2)=O)CC1 N12CC3COCC3(C1)C2=O.n1(CC)cc(CC(=O)NC(C)CC(=O)OC)nn1 c1(C(=O)NC(C)C(C)(C)NC(=O)CCC2CC2)scc2c1CCCC2.C1CC1 C1(C(N2CCC(N(C(=O)Cc3cnoc3)CCC)C2)=O)CC(=O)N(O)C1 C12(C(=O)NC3(CNC(C4(CC#C)CC4)=O)CCC3)CCCCN1CCC2 C(C(C)(C)CC(=O)N(C)Cc1noc(C)n1)NC(c1nc(OCC)oc1)=O N1(C(C2OCCN(CC)C2)=O)CC2(CCN2C(c2ccccc2C(C)(F)F)=O)C1 N1(C(CC(CNC(=O)COC2CCOC2)O)=O)CCCN(CCO)CC1 C(=O)(CCS(=O)(=O)NC1CC1)N(C(C)CN(C(=O)CCCC1CC1)C)C C1(CC)C(NC(c2ccc(C3CC3)cc2)=O)CCCN1C(c1csc(O)n1)=O n1(CC=C)cc(C(=O)NCC(C2CCCC2)NC(C2(O)CCSC2)=O)nn1 C(N=c1[nH]cnc2[nH]ccc12)C1C(NC(=O)CCn2cncn2)CCC1 C1(CC=C)(NC(c2cnnc(O)c2)=O)CCN(C(C23CCC(CC2)CO3)=O)CC1 Cc1ccc(OCC(=O)NC2CCN(C(=O)CC3COCCO3)C2C2CC2)nc1 CP(C)(=O)c1cncc(C(=O)NCC2(O)CCCN(C(c3ccoc3)=O)CC2)c1 CSC=CC(=O)N1CCCC1C(C)(C)NC(=O)CCN(CCC(C)(C)C)C C1(C(=O)Nc2ccnc(-n3ccc([N+](=O)[O-])n3)c2)CCC2CNCCC2C1 C12(CNC(C(c3cccc(C)c3)O)=O)CCCCC1N(C(=O)O)CC2.C(C)(C)C C1(CSC)CCC(NN2CCC(CC#N)CC2)CC1 C1(CN(C)C(c2csc(CC(F)(F)F)n2)=O)CCCN1C(=O)CCCF c1(NC(c2c(C)nns2)C)[nH]c(=NCc2ccc(Br)c(C)c2)nc2c1cnn2C Cc1ccc(C(=O)NC2CC(C)CN(C(C3CCC=CCC3)=O)C2)c(Cl)c1C C1(NC(c2ncc(C)nc2)=O)CCCC2CN(C(C3(O)CCSCC3)=O)CC12 CCCCC(=O)NC1CC1CNC(=O)CN(C)Cc1ccccc1 C(C)(C)(CC(=O)NC(CCF)C(=O)NCc1ncc(C)o1)OC CC(C)C(O)C(=O)N1CCC(CCCNC(c2cnn(C(C)C)c2N)=O)CC1 c1(OC)ccccc1-c1ccc(C(=O)N(CCCO)CC2CC2)s1 CC(O)C(F)(F)C(=O)N1CC=C(C(=O)N2CCC2C2CCC2)C1 C1(C)(C(N2CCC(OCCN(C)C)CC2)=O)CCCC1(F)F C12(C(=O)OC)COCC1CN(CC1CCCN(C(C)C)C1)C2 C12(C(N3CC(NC(c4ccc5c(c4)CC5)=O)C(O)C3)=O)CCC(CC1O)C2 C1(CNC(CC=C(C)C)=O)C(C2CC2)CCN1C(c1cccnc1)=O.C1CC1 c1(CC(N2C(CNC(C(C3CCC3)OC)=O)CC2)=O)cn2cccc(C)c2n1 C(CN(C)C)(C(=O)N1CC(C)(C(=O)OC)C1)NC(C1CC(=C)C1)=O C1(C#N)(C(=O)NC(c2ccccc2)C(=O)NCC(C)CN(C)C)CCCC1 N1(C(c2cc(C)c(C)nn2)=O)CCCC1C1CCCN1C(c1cc(C)n(C)n1)=O C1(OC)CCC12CC(C(N1CC=C(CNC(C3CC3C(F)F)=O)CC1)=O)C2 C1(CC)CCOCCN1C(c1oc(CNC(C2CC2)=O)cc1C)=O.C1CC1.C C(=O)(C1Cc2ccc(F)cc21)NC1C(NC(c2ccc(OC)nc2)=O)CCCC1 c1(OCC(=O)NCC(C(C)(C)C)NC(=O)C(F)F)cccc2ccccc12 Cc1coc(C2CC2)c1C(=O)N(C)CC1CN(C(=O)Cc2csc(Cl)c2)C1 C1(N(C)C(C2CSC2)=O)CCCCN(C(C2(C)CC(C)(C)C2)=O)C1 C1(C(=O)NCCSc2nc(C)[nH]n2)C(C)CCN1C(=O)CN1CCOCC1 c1(C(C(=O)NCCCF)N(C(c2nncn2C)C)C)cccc2c1COCC2 c1(C(=O)NC(CN(C(C(CCCC)O)=O)C)C)ncn2c1COc1ccccc1-2 CC1C(NC(=O)C=Cc2cncs2)C(C)CCN1C(=O)Cn1ncc2ncccc12 CC(C)C(CN(C)C)C(=O)N1CCN(C(c2cccc(CCO)c2)=O)CC1C c1(C(=O)OC)cc([N+](=O)[O-])c(NC(=O)CC2CNCCO2)s1.c1ccnnc1.C CC1(C)CN(C(c2n[nH]cc2[N+](=O)[O-])=O)CCC1NC(c1scnc1C1CC1)=O CC1COC(C(=O)NCC2(F)CC(NC(c3cn(CCCC#N)nn3)=O)C2)C1 Cn1c(O)nc(NC2(CNC(=O)CCc3ccccc3)CC2)cc1=O c1ccc(C=O)cn1.C(=O)(CCC(C)OC(C)(C)C)NCC1CN(CC)C1 O=C(C1CCc2c(Br)cccc21)N1CCCC1c1ccc(F)cc1F C1(NC(=O)CCn2ccnc2)CCN(C(=O)Cc2c[nH]ccc2=O)CC1F C1(NC(CC(C)SC)=O)CCCC1(C)CNC(c1ccc(C2CC2)nc1)=O c1(OCc2cc(C)on2)ncccc1S(=O)(=O)N1CCCC(CN2CCCC2)C1 CCC(C)(C)CC(=O)OC.C1CNC1CC.C(C)C CC(C)(C)CC(O)CC(=O)NC(C1CC(F)(F)C1)C#N c1(C(N(C2CCN(C(c3coc(CO)c3)=O)CC2)CC#C)=O)ccc(Cl)c(F)c1 C1(NC(c2nc(C)oc2)=O)(C)CCC(C)(C)CC1.n1(C2(C=O)CC2)cncn1 C(c1ccc(C)cc1)=C(C=O)C.c1(C(N(CC)CC)=O)ccc(C#N)o1.CO N1(C(c2nccc(C)n2)=O)CCCC(CNC(=O)C(C)OCCC(C)C)CC1 C12CCCC1CN(C(=O)C(C)S(C)(=O)=O)C2.C1(C(=O)N)(OC)CC(C)(C)C1 c1(OC)c[nH]nc1C(=O)NCCC1CCC1.c1(C2C(C=O)C2)ccccc1.N N#Cc1cc([N+](=O)[O-])ccc1N1CCCC1CCNC(c1ccoc1)=O O(NC(=O)C(=O)N=c1cc(C)o[nH]1)N(C(CCC(N(OC)C)=O)=O)C1CCCC1 C(C(=O)NCCCCCC)(C(C)C)NC(=O)OC.c1(C=O)cnn(C2CC2)c1 c1(CCC)ccc(N)c(C(=O)NCC23CC2CN(C(C2CC(O)C2)=O)C3)c1 C=CC(F)(F)C(=O)NCC1CCCCN1C(=O)CC1(c2ccccc2)CCCO1 N1(C(=O)NS(CC=C)(=O)=O)CCC(CC2CC2)CC1 Cc1ncc(C(=O)NCCc2cc(C(=O)NC3(C4CC4)CC3)no2)n1C C1(O)(CC(=O)NC2CC(C(F)F)(NC(=O)C(F)n3ccnc3)C2)CCCCC1 N1(C(C(CCC)NC(C)=O)=O)CCc2sccc2C1CNC(=O)CC(=O)N(C)C c1(C(=O)NC(C(C(C)C)NC(c2c(Cl)cc(C)s2)=O)C)cc2cccnc2[nH]1 N1(C(C(C2CN(C(COCCC=C)=O)C2)O)=O)CCC(CC(C)O)CC1 N1(C(c2c(C)nn(CC(F)F)c2)=O)CCC(N(C)C(c2cnn[nH]2)=O)C(C)C1 c1(OC)cc(C)cnc1C(N1CCC(NC(=O)CCOCC(F)F)C1(C)C)=O CC1CN(C(c2ccc(Cl)s2)=O)CCN1C(C1CC(C(F)F)C1)=O Cc1cc(C(=O)NC2CCCC2C2CC2)c2c(c1)CCO2 c1(C(C(=O)NC(C(C)(C)C(=O)O)c2ccccc2)S)nc2ccc(Cl)nc2[nH]1 c1(C(N(CC(CC)NC(=O)C(C(C)O)N(C)C)C)=O)ccc(N(C)CC)nc1 C1(C(N(CC(CC)NC(=O)CNC(C)=O)CC)=O)CCCC1C(C)C c1(C(N2CC(NC(C=C(C)Cl)=O)CC23CCC3)=O)ccc(S(N)(=O)=O)cn1 CCC(CCCC(=O)NCCC1CN(C)C1)NC(=O)C(C)C CCC(COC)C(=O)NC(C)CC(=O)NC(CCO)C1CC1 Cc1nccc(N2CC3C(C2)N3C(c2cnon2)=O)n1 N1(C(C)=O)CC(O)CC1C(=O)N.C1CCN(C(=O)C(C)(C)n2cnc(C)c2)C1 CC1(C)C(C)(C(N2CCC(C)(C(N3CCC=C(Cl)C3)=O)CC2)=O)C1(C)C CCCC(CC)CCC(=O)N1CC(CC(=O)NCC(C)C#N)CC1(C)C C1(CNC(CNC(CC)=O)=O)C(C)CCN1C(c1cn(C)nc1OC)=O Cc1cc2n(n1)CCN(C(C1CCC(NC(=O)C(C)CO)C1)=O)C2 C1(OCC(N2CC(NC(C(c3ccccc3C)OC)=O)C2)=O)CCCC(C)C1 C(=O)(CCCn1ccnn1)NC(C1CN(C(c2csc(Br)n2)=O)C1)C c1(C(=O)NC(CNC(=O)C=CC2CCCCC2)CO)cc(F)cc2ccoc12 C1(C(=O)NCC(n2cc(-c3ccn(C)n3)nn2)C)CCCC2C1C2(F)F c1(C(N2CCC(CNC(C=CCCC)=O)C(C)C2)=O)cccc2c1NC(=O)CO2 c1(C(=O)NC2C(NC(C(CSC)c3ccccc3)=O)CC2)cc(F)cnc1O CN(C)NC(=O)CCC(=O)NC1(C2CCCCN2C(c2cnc(S)nc2)=O)CC1 N1(C(=O)CC2(O)CCCCCC2)CCC2(C1)CN(C(C1(C(F)(F)F)CC1)=O)C2 C1(C(N2CC(OCCCCC)C2)=O)C(C)CCN1C(c1nc(C)sc1C)=O N#Cc1ccccc1F.N1(CCNC(=O)COc2ccccc2)CCC(CCO)C1 Cc1nc(-c2ccc(Cl)cc2)sc1C(=O)NC.C1CCCCN1C(=O)CC1CC1 c1(C(=O)NC(CCNC(c2c(F)cc(C)cc2F)=O)C)ccnc2c1ncn2C N1(C(C(C(C)C)SCC)=O)CCN(C(=O)CCN(S(C)(=O)=O)C)CC(O)C1 C12(NC(c3ccc(-c4ccccc4F)o3)=O)CCCN(C(=O)C=CCF)CC1C2 C1(C)(C(=O)N)CC(O)CN1C(=O)CCC1CC1.C(COCC)OCC N1(C(c2c(CC)nn(C)c2)=O)CC(NC(c2ccccc2C)=O)C2CC2C1 c1(C(N2CC(NC(=O)C=Cc3cccs3)C3C2C3)=O)cc2ccccc2[nH]1 c1(-c2nc(-c3c(C)cccc3)sc2)cc(Cl)nc(C)n1 N1(C(CN(C)CCO)=O)CC(NC(c2cccc3sccc23)=O)C2CCCCC12 C(C(COC)CC(=O)NCc1cscn1)OC.C(C(F)(F)F)=CC=O.C N1(C(CCC=CC)=O)CCC2(CC1)CC2CNC(=O)C(CCC)OC c1(NCC(CC)C)ncc(S(=O)(=O)NC(c2ccc(C(F)(F)F)nc2)C)cc1Cl c1(OCC)ccc(N)c(C(=O)N(CCCC)C)c1.C(=O)C(C)Cn1ccnc1.N c1(C(=O)NC2C(NC(c3ccc(C(N)=O)cc3)=O)C2)cc(Cl)ccc1[N+](=O)[O-] c1(CC(=O)N(CCOC)CCNC(=O)CC)cc(F)ncc1Br.C(N)=O c1(C(N2C(CC)CN(C(=O)Cc3nc(=N)[nH][nH]3)CC2)=O)cc2nccn2c(O)n1 CC1(NC(C2CC2CNC(C2SCCS2)=O)=O)CC2(CCC2)C1 C1(CC(N2CC=CC(NC(CCC(N)=O)=O)C2)=O)CCCCC12CC2 c1(C(C(N2CC(C(CC)C)OCC2)C)=O)ccc(OC)c(C)c1 C=C(C)CC(C)C(=O)NCC(C)NC(=O)C(c1cccc(Br)c1)(F)F c1(C=O)cn2c(n1)CCC2.C1(CN(C)C(c2cccs2)=O)CC(F)(F)C1.C c1(C(C(=O)NCCC)N(CC=O)CC)cnc(N(C)C)o1.c1csc(C)c1 Cc1nc(-c2cccs2)sc1C(=O)NCC(CNC(=O)Cc1nc[nH]n1)CO C1(C(=O)NCC2CCC3(CC3)C2)CC2(CCN1C(=O)CC1=CCOCC1)CC2 C=CC1(O)CCN(C(c2nccc(OC)c2C)C(=O)NC)C1 C12(C(N3CC(C(=O)NCCOCC#C)(CC=C)C3)=O)CCCC(CO1)C2 N1(C(c2c(C)sc(O)n2)=O)C(C(=O)NOC(C)(C)C)CCC12CC2 c1(OC)ccc2[nH]cc(C(=O)NCC(C)CNC(c3cnc(Br)s3)=O)c2c1 C(=O)(CCC(CC)SC)NCCN1CCN(C(c2cc(CCC)[nH]n2)=O)CC1 C1(NC(C2(N(C)C)CCC2)=O)CC2CC1N(C(=O)CCc1ccccc1Br)C2 c1(CC)[nH]c(C(=O)NC2CCCC2CNC(c2c(C)nsc2N)=O)nc1Cl Cn1cc2c(C(=O)NCC3CCCCNC3)cc(F)cc2n1 C(=O)(CCC(C)(C)C#N)N1CCCC(N(C(=O)CS)CC)CC1.c1nnc(S)s1 CC1CCC(=CC(=O)NC2C=CCCC2C(=O)NCc2ccnc(Cl)c2)CC1 N1(C(C(CC)CN(C)C)=O)CCN(C(C2CNC(=O)O2)=O)CC1CCO C=C(C)c1cnccc1NC(=O)N(CCC(=O)OC(C)(C)C)CC(C)C Cc1ncc(N)cc1C(=O)NCC1CCC(NC(=O)Cn2nccn2)C1 N1(C(c2cnc(F)c(Cl)c2)=O)CC2CC(C1)N(C(=O)Cn1cc(CO)nn1)C2 CC1CCCCC1(CNC(C1CC2(C1)CC21CC1)=O)NC(c1cc[nH]n1)=O N1(C(C(CC)c2ccccc2)=O)CC=C(CCNC(c2cc[nH]c(=N)c2)=O)CC1 CN1CCCCC(C(=O)NC(C)(C)C2CC2)C1=O.c1(C(=O)N)cc[nH]c(=N)c1N C(=O)(CS(=O)(=O)C(C)C)N1CCC(CCC2N(C(COCC)=O)CCC2)CC1 C1(CC(=O)NC(c2ncc(C)s2)(CC)C)CCC(C2CCNCC2)O1.C(=O)N.C S(=O)(=O)(c1c(Cl)nc2cc(Cl)ccn12)N1CCCC(Cc2n(C)ncc2)C1 N12CCCC1(Cc1ccccc1)C2=O.CC(N)CCC.C(=O)O N1(C(c2c(COC)ncs2)=O)CCC2CCC12C.c1(C=O)cc(C)cc(C)c1 C1(NC(c2ccn(CC)n2)=O)CC(NC(=O)Cc2cc(C)on2)C(O)C1 CN1CCN(C(=O)CC2CC2C(F)(F)F)CC1c1cc(F)cc(F)c1 c1(C(N2CC(O)(C(C)NC(CC(C)F)=O)C2)=O)csc(=NC2CC2)[nH]1 C(=O)(CCCC1CCC1)NCCCC(C)C1CC1.C1(C(=O)N)CC1C(N)=O Cc1ncc(CC(N2CCCC2C(C)NC(c2ccns2)=O)=O)o1 c1(C(N(C2CCCCN(C(=O)CC3COC(=O)C3)C2)C)=O)cccc2nc[nH]c12 Cc1cnc(C(=O)Nc2ccc(F)c(F)c2Cl)cc1C#N C(CC(=O)N1CCOC(C#N)C1)(C(F)(F)F)NC(C(C(C)C)SCC)=O c1(CCC(N2C(CCNC(CSC)=O)CCC2)=O)c(C)nc2ncnn2c1C c1(C(CN2C(c3onc(C)n3)CCCC2)=O)c[nH]c2cccc(C)c12 c1(C(=O)NCCCCN(C)C(c2ccnnc2)=O)ccnn1CC1CCC1 c1(C(=O)NC2CN(C(C(COC)O)=O)CC(C)(C)C2)c(Cl)ccc2c1OCO2 c1(C(N(C)CCNC(c2cnc(Cl)c(N)c2)=O)=O)cccc2c1CNC2=O C1(CNC(CC(C)(C)O)=O)CC2(CO1)CN(C(=O)Cc1cccnc1)C2 C(=O)(C(C)(C)C(N)=O)N(C1CCN(Cc2ccc(CF)cc2)C1)C CC(C)C(C)CC(=O)NCC(C)(C)OCC(=O)NCC1CC(O)C(F)C1 C1(CNC(C2CCCN(C)C2)=O)CN(C(C2CC(F)(F)C2)=O)CCC12CCOC2 C(=O)(C(F)(F)C1=CCOCC1)NC(CC=C)CNC(C1CN(C)C(=O)N1)=O N1(C(C2CN(C)C(=O)N2)=O)CCCC(N(c2cncc(Cl)n2)C)CC1 C1CC2CCC(C1)N2C(=O)Cc1ccc(Cl)nc1.C1(C(C(=O)N)O)CC(F)(F)C1 C(=O)(C(CC)C(C)(C)CC)NCC(C(=O)NC(C#C)C1CC1)(CC)CC c1(C(C(=O)NC2CCC(CNC(C3CCCCO3)=O)CC2)=O)cc(Cl)cc(Cl)c1 c1(-c2n(C(C)C(F)(F)F)nc(Cn3cncn3)n2)cncc2sccc12 N1(CC2(C)CCC(=O)N2)CCC(=O)N(CCc2noc(C3CC3)n2)C1=O C1(NC(C2(CC)CCCCC2)=O)CCN(c2nc(C(F)F)nc(=N)[nH]2)CC1F c1(CC)cc(N2CCCC(C(C)NC(C3(C)CC3)=O)C2)nc(C)n1 c1(OC)ncc(C(=O)N(c2cc(NC(C)=O)ncn2)C2CCNC2)cc1C c1(CC)cccc2[nH]c(C(=O)N(C)CCNC(C3C4CCCOC34)=O)cc12 C(C(COC)CC(=O)NCCC1CSCCN1C(=O)CC1CCC1)OC C(=O)(CC(C(F)(F)F)C1CC1)N(CCC(C(C)C)NC(c1c(C)n(C)cc1)=O)C C1(C(N(CCCCCNC(C2(CC3CCC3)CC2)=O)C)=O)Cc2ccccc2S1 CCC(C)(C)CC(=O)N1CCCC(C(C)C(=O)NCCn2ccnn2)C1 C1(C(NOC(C=C)C)=O)N(C(=O)C(C)Cn2cccn2)CCCC1(C)C c1(N2CC(C)(NC(C(C)C3CCOC3)=O)C2)ccc2nnc(C3CC3)n2n1 N1(C(Cc2c(C)non2)=O)CCN(C(=O)CCN2CCCC2=O)C2(CCC2)C1 C1(C(=O)NCC23C(CN(C(C=CCCC(C)C)=O)C2)C3)C(C2CC2)C1(F)F c1(C(N(CCC)CCNC(=O)CC23CCCC2C3)=O)ccc2ncc(C)n2c1 c1(C(=O)NC(C)(C)C)ccc(NC(c2ccc(-c3nccs3)cc2)=O)cc1 c1(C(N2CCC(C(=O)NCC(CC)(C)CC)C2C(C)C)=O)cccc(C)c1N c1(CNC(c2c(C)nc(-c3ccc(C)nc3O)s2)=O)cc(C)c(C)cc1C c1(N2CCC(NCC3CCC(=O)C3)C2)ccccc1Br c1(NC(C(C)CC2CCCCC2)=O)cccc(CNC(=O)C(C)c2ccsc2)c1 C1(NC(c2cnns2)=O)CCOCC1C(=O)NC(CO)CCCO N1(C(C(C)(C)OC)=O)CC2ON=C(C)C2C1.c1(CC(=O)N)ccc(C)c(C)c1 c1(OC)cc(C2CC2)ccc1C(=O)NC1(C)CCCN(C(C2OCCC2C)=O)C1 C1(OC)CCN(C(CC2CCCCC2)C(=O)NCC2CCCO2)CC1 c1(OC)c(C(=O)Nc2cncc(C(C)(C)F)c2)cc(Cl)cc1C C(C(=O)NCCCN=[N+]=[N-])(C(C)O)NC(c1c(CC)non1)=O c1(C(C)(C)C)ccc(NC(C2CCCN2Cc2cc(Br)co2)=O)cc1 CC1(C)CC(CNC(C23CCC(C)(C2)OC3)=O)N(C(C2C=CCS2)=O)C1 Cc1ccc(CC(=O)NCCC(C(C)C)NC(c2c(Br)noc2C)=O)cc1 C=CC1CCCN(C2CN(C(=O)CC(C3CCCN(C(=O)NC4CC4)C3)C)C2)C1 C(N=c1nc(N2CCC(n3cncn3)C2)c2ncn(CC(F)(F)F)c2[nH]1)C1(OC)CC1 N1(C(C2(CC)CC2)=O)CCCC2(C1)CN(C(=O)C1=CCC(F)(F)CC1)C2 N1(C(CCCCCC(C)O)=O)Cc2[nH]c3ccccc3c2CC1c1ccccc1 C(=O)(CCC(F)(F)F)N.C1(C(=O)NC2C(C)C2)CCCC1.C(=O)C(C)(C)C N1(C(CCC(C)O)=O)CCC2CC(CNC(=O)C(C)CN(C)C)CCC2C1 Cc1cc(CC(=O)NCC(C2CCC2)NC(=O)CC(F)(F)F)cc(C)c1 c1(C(=O)NCC(CCNC(c2cnccc2OC)=O)OC)cc(C#N)oc1C C(=O)(C(C)(C)C(F)(F)F)NC1C(CO)CCN(C(C=Cc2c(C)nccc2)=O)C1 CC(O)CC(C)(C)CNCc1ncccc1CN CCC(CC(F)(F)F)C(=O)NC(C)(CNC(=O)CCCCC(C)C)C1CCC1 C(=O)(C(C)(F)C(C)(C)F)NCC(CCCC)NC(c1cnc(C2CC2)[nH]1)=O c1(NCC2(NC(C3CC4(C3)CC(F)C4)=O)CCCC2)nc2cccc(F)c2s1 CC1C(NC(=O)CCCc2ccncc2)CCN1C(=O)CC1CCCN1C(C)C N1(C(c2cccc(C(=O)OC)c2)=O)CCCCC(SC)C1 c1(C(=O)NCCC2CCN(C(COC)=O)C2)cnc(OC)c(OC(C)=O)c1 C1(C(N(C(C(=O)OCC)C)C)=O)C(C)CCN1C(=O)CC1(CC)CCC1 c1(NC(=O)CCC2CCCN2C(c2cc(F)ccc2Cl)=O)ccc(Br)cc1Cl N1(C(CC2CC(=C)C2)=O)CCC(C2CCCN(C(c3c[nH]c(C)cc3=O)=O)C2)C1 C12(C(N(CC(CC)NC(c3cscn3)=O)C)=O)CCC(OC)C1CC2 Cc1cc(=NC2CC(NC(c3c[nH]nc3[N+](=O)[O-])=O)C2(C)C)[nH]c(C2CCC2)n1 C#CC1CCCCN1C(=O)CC1CN(C(C2(CC=C)CCOC2)=O)CC12CC2 c1(C(=O)NC(CN(C(C(=Cc2cnc[nH]2)C)=O)C)(C)C)ccc(C)c(CO)c1 C1(C(=O)NCC2CC(NC(c3cocn3)=O)CC2O)CCOC2(CCC2)C1 O=C(C(F)(F)Cc1ccccc1Br)Nc1ccc(-c2ccccc2)cc1 N1(c2nnc(C(C)(C)C)o2)CCCC2(NC(=O)C(C)(C)c3ccccc3)CC2C1 c1(C(N2CCC(NC(C=C(C)c3ccsc3)=O)C2)=O)cccc2c1OCC2C N1(C(CC(=O)NCC)=O)CC(F)CC1CC(=O)NCCN1CC2CCC1C2 N1(C(c2ccc(CC)o2)=O)CC2CC(NC(=O)CC(C)C)C(C2)C1.C(=O)N CCC(C(C)CN(C)C)NC(C1CC2(C1)CC2F)=O C1CC2(CO1)CN(C(=O)C)C2.C(=O)CC(C)C.C(CC(=O)NC)SCCCC C(=O)(CC(C)(C)C)N1CCC(N(C(C(C)Cc2cnco2)=O)CC2CC2)C1 Cc1cc(C(=O)NCC2(n3cccn3)CCOCC2)[nH]c1C N1(C(c2c(C)ccs2)=O)CC(CC(=O)NCCc2ccncn2)C(C)C1 C=CCC(CC(C)C)C(=O)NC1CC2(NC(c3cnccc3C)=O)COC1C2 c1(C(=O)NC2CC(C)N(C(c3cnc(NC4CC4)s3)=O)C2)ccn2nccc2c1 C(c1cn(C)cn1)=C(C(=O)N(CC(C)C)Cc1ccc(Br)cn1)F c12nc(cc(C)n1)ON1CCN21.c1(OC)ccccc1CCNC(C)=O N1(C(CCOC)=O)CCN(C(=O)CN2CCC(N(C)C)CC2)C2(CCC2)C1 C12(OC)CCC(C(=O)N(CC(C)CNC(=O)C(C)C(C)O)C)(CC1)C2 C=C=CC(C)C(=O)NC1CCC(C(=O)NCC(C)(C)C2(O)CCC2)CC1 C(=O)(CCCC(F)(F)Br)NCC(C)NC(c1cc(C)c(Cl)cc1)=O CN1N=C(CC(=O)NC2(C)CCN(C(=O)Cc3cccc(Cl)c3F)C2)CC1=O c1(N2CC(OC)(CNC(=O)CCc3ccc(O)nc3)C2)nc(Cl)ncc1Br CN1CCC(c2ccc(Br)cc2)(CNCc2cccc(Br)c2O)CC1 C1CN(C(=O)C=Cc2cnn(C)c2)CC1.c1(C=O)nc[nH]c1C(C)(C)C.CC N1(C(CCCC(=C)C)=O)Cc2ccc(C(C)NC(C3CCCC3CC)=O)cc2C1 CCCC(CC)CC(=O)N1CCN(C(=O)CC(C)C(C)C)CC1c1ccccn1 C1(NC(c2c(C(C)C)n[nH]c2)=O)CCCC2CN(C(=O)C(C)CBr)CC12 C1(NC(c2cc(CO)on2)=O)(CO)CCN(C(c2scnc2C2CC2)=O)C1 N1(C(CC(CNCc2ccc(SC)o2)O)=O)CCCC(O)(c2cnn[nH]2)CC1 Cc1nc2c([nH]1)C(C(=O)NCC1CCC(O)C1)CCC2.C(=O)C(C)(C)C1CC1 c1(NC(C(c2cn(C(C)(C)C)c(C)n2)OC)=O)cccc(N2CCCC2=O)c1 C1(CCC)(NC(=O)Cc2cn[nH]c2)CCCN(C(C2CC2CC(C)(C)C)=O)C1 C=CC(C)(O)C(=O)NCC1CCC(NC(c2coc(OCC)n2)=O)CC1 c1(CNC(c2cccc(COC3CC3)c2)=O)ccnc(OC(F)(F)F)c1 N1(Cc2cc(C)c(C(F)(F)F)cc2)CC2CN(C(C3CN(C)CCO3)=O)CC2C1 C1(CC)CCN(C(=O)COCCCF)C(C(N2CC(OCCOC)C2)=O)C1 N1(C(C(C)O)=O)CCC(C)(NC(=O)CCc2cccs2)C1 C(=O)(CCC(C)(C)C)NC(C(=O)OCC)C1CC1.C(=O)CCC(C)=O.N CC1=C(C(=O)NCC2CCN(C(C3CC34CC4(F)F)=O)C2)CCCO1 C1(C2CCCN(C(=O)CCc3cnoc3)C2)(NC(C2CSCCS2)=O)CC1 N1(C(C2(c3ccccc3Cl)CC2)=O)CCOC(CCNC(C2CCOC2)=O)C1 C1(C(=O)NCCC2CNC23CCC3)CC(C2CCNC2)C1 C1(C(=O)NCc2cc(C(C)C)no2)CCC(NC(=O)CC2COCCO2)CC1 N1(CC(=O)NC)C(=O)CCC1=O.C1CC(F)C1.c1(C=O)n[nH]cc1C1CC1 C1(C(=O)Nc2c(C)noc2)CNC(=O)CN1C(C1CC2COCC2C1)=O c1(-c2ccc(C(N3CCC4C(NC(c5csc(Cl)n5)=O)C43)=O)o2)ccc(F)cc1 N1(C(c2cc(C)oc2)=O)CCC2(C1)CN(C(=O)CC1(C)CC1(F)F)CCO2 C12CN(C(C3(O)CC3)=O)CC1CS(=O)(=O)C2.c1(C(=O)N)ccc2nccn2c1 CC1(C)CC(=O)NCC1C(=O)NC1CN(C(=O)C)CCC1F.C(=O)C(F)(F)F c1(OC)cc(F)c(F)cc1S(=O)(=O)NOCCN.C(CCC)NC(=O)C1CC1 c1(C(=O)NC(C2CN(C(=O)CCNC(=O)CO)CCO2)C)cccc(F)c1 CN1CC=C(CC(=O)NCC2CN(C(=O)CCc3cnco3)CC2(F)CO)CC1 C1(C=O)CC2(CC2)C12CC2.n1(CC(NS(N)(=O)=O)C)cc(CCCCC)nn1 c1(C(N2CCC(CC(C)NC(C3(C)CCOC3C)=O)CC2)=O)cnc(Cl)cc1N C1(Br)(C(=O)NCCCN(C(c2cc(C)co2)=O)CC)C(C)C1C c1(CC)nc(C(=O)N)c(C)o1.CCC(C)(C)C.C(=O)C.C(=O)CN(C)C c1(CC=O)cccc(Cl)c1F.N1(C(C2CC(CC(=O)OC)C2)=O)CCCC1.C n1(CCC)ccc(C(=O)N(C)CCn2cc(C)nn2)n1.C1(C(=O)N)CCOCC1 C(=O)(CN=c1[nH]c(C)cs1)N1CC(NC(c2c[nH]nc2C2CC2)=O)CC(OC)C1 CC(C)CC(CNC(=O)CCN1CCCCC1C)NC(c1nc(C2CC2)cs1)=O N#Cc1ccccc1OC1CN(C(=O)C(=O)NCC(=O)NC2C3CCCC23)C1 c1(C(N2CC(O)(CN(C(C=CCC)=O)C)C2)=O)ccn2cncc2c1 c1(C(CO)NC(C2CC3CC3N2C(=O)CCc2ccccc2)=O)ccc(F)cc1 c1(C(=O)NCC23OCCCC2C3(F)F)cccc(S(=O)(=O)CC(F)(F)F)c1 C1(C(=O)NC(C(=O)NC2COCC2F)C2CCCC2)OC2CCC1C2 c1(C(N(C2CCN(C(=O)CC3CCC3)C2)CCC)=O)cc(C2CC2)on1.C Nc1cc(Cl)ccc1C(=O)NCC1(O)CN(C(c2cc(C(F)F)on2)=O)C1 N1(C(C2ON=C(C)C2)=O)CCC2CC1CN(C(=O)CCCC(C)(C)C)C2 CC(C)CC(C)(CNC(=O)CC1CCC(F)(F)C1)NC(c1ccsc1)=O C1(C(=O)NCC=C)CC(C)CN1C(=O)CC1CCC1 CCC(C(=O)NC(C1CCN(C(C2CCC(O)CC2)=O)CC1)C)C(C)C CN1CCC2(CC1)CN(C(C1C3CCC1(c1cncs1)C3)=O)c1ccccc12 C1(NC(C2CC(CC)C2)=O)CCC(F)(F)CC1.C12(C(=O)N)CCN(CC1)C2 C1(C)(C(=O)OCC)CC12CCN(C(=O)C(=O)Nc1cc3[nH]cnc3cc1F)CC2 c1(C(=O)NCC(CC)NC(c2ccc(C)c(O)n2)=O)cc2ccc(Cl)nc2s1 Cc1ccc(C(=O)N(CCC(C)NC(=O)CC2CNC(=O)C2)C)nn1 C(=O)(C(C)(C)C(=O)NC)OCC.C1CN(C(=O)CC)CCO1.c1cccnc1 CN1C(=S)NC(c2cccc3cccc(Br)c23)C2=C1C(C)(C[Si](C)(C)C)NC2=O C1(NC(=O)C=Cc2ccco2)CN(c2ncc(I)cn2)Cc2nccn2C1 c1(CCC)n[nH]cc1C(=O)NCCCOCCC(N1CCC(C(N)=O)C1)=O O=C1CCC(CCC(=O)NC2(CNC(c3ccc(Br)s3)=O)CCC2)N1 N1(C(C2C(CCOC)C2)=O)CC2CC1(C(=O)N)C2.c1ccccn1.C(C)=O CCC(CC)CC(F)C(=O)N1CC2C(CN(C(=O)CN3CCNC(=O)C3)C)C2C1 c1(NCC(NNC(=O)c2ccc(C)cc2)=O)cc(NC(N)=O)c(F)cc1C c1(CN(CCCc2cn(CC)nc2)C=O)ccc(Cl)n1CC Cc1ccc(C(=O)NC2C3CC2N(C(=O)C(C)c2cncs2)C3)nc1O N1(C(CCS(C)=O)=O)CCCC(C2CN(C(c3cnn4ccccc34)=O)C2)C1 c1(C(N(C)CC2CCCCN2C(=O)CSc2cn[nH]c2)=O)ccc2cccnn12 CCC(CNC(c1ccnn1C1CCC1)=O)CC.c1(C=O)cn(C(C)C)cn1.N N1(C(c2ccc(C(C)=O)[nH]2)=O)CC2CC(NC(c3c(C)ncn3O)=O)CC(C2)C1 C1(CC=O)COC2(CCC2)CO1.Cc1ccc(C(=O)NC(C)(C)C2CC2)[nH]1.N N1(C(C(C)NS(CC)(=O)=O)=O)CCCN(C(=O)Cc2cc(F)ccc2Cl)C(C)C1 C(CC1=CCN(C)CC1)NC(C1CN(C(c2c(C)nns2)=O)CC(C)O1)=O Cc1ccc(C(=O)NC(C)(C)CN(C)C(C2SCCC2C)=O)o1 N1(C(=O)COCC2CC2)CCCCC1C1CCCN1C(=O)COCC(F)(F)F c1(C(C2CC2)NC2CC3CC3C2)ccc(C2CC2)nc1O c1(C(=O)NCC2CC(C)N(C(c3cscc3C#N)=O)C2)ccc(=O)n2c1CCC2 c1(CNC(C=C(C)C)=O)ccc(N2CCCCC2)cc1.C1(C=O)CC(C)(C)O1 c1(CCC(=O)NC2CC3CC2N(C(C2(F)CC=CCC2)=O)C3)ccc(F)cc1F c1(C(C)NC(C2CCCC2)=O)ccnc(F)c1.c1(C(=O)N)ccc(C2CC2)o1 c1(-c2nc(C=Cc3ncc(C(=O)Oc4ccccc4)[nH]3)on2)c(F)cccc1F C#CC(C(C)OC)NC(=O)C(C)N(C(=O)CC1CC(=C)C1)CC c1(C(C(=O)NC2(C(=O)NC(C#C)(C)C3CCC3)CC2)C)cnn(C)c1 CCC(CC(C)C)C(=O)NCC(C)(C)OCC(N1CCN(C)CC1CC)=O N1(C(C(CC)NC(N)=O)=O)CC(C)C(C)(C(N2CC(C)(CCO)C2)=O)C1 C1CCN(C(=O)C)CC1C.c1(C[SH](=O)=O)ccccc1.C(C=O)=CCOC.N N1(C(C2C(C=O)C2(F)F)=O)CCC(C2CC2)C1.c1(CC=O)n[nH]c(C)n1.C C1(CC)(NC(c2cccc(C(N)=O)c2C)=O)CCN(C(=O)C=C(C)Cl)CC1 c1(CCC)c(C(N2CCOC(CNC(c3ccoc3Cl)=O)C2)=O)nnn1C c1(C(=O)NCC2CCCN2C(=O)C2=C(Cl)CC2)cc(Cl)cc(Cl)c1Cl c1(C(N2CCC(NC(C(C)OCCOCC)=O)C2C)=O)cccc(O)c1Cl c1(CC)[nH]nc2ccc(C(=O)NCC(=O)CC(C)C)cc12 C(=O)(C1=CCN(C)C1)N1CC(CNC(C(CO)N(C)C)=O)C(CO)C1 C1(C2(NC(c3cc(SC)no3)=O)CC2)CCCCN1C(=O)Cc1c[nH]ccc1=O c1(NC(=O)CC(O)c2ccccc2)cccc(NC(=O)C(F)(F)CC2CC2)c1 C#CCCCCC(=O)NCC(CC(=O)NCc1cc(C(C)C)on1)C1CCC1 c1(NC(C2(F)CCN(C(c3c(C)oc(C)c3C)=O)C2)=O)cnc2ccccc2c1 C(=O)(C1=CC(O)CCC1)N1CC(O)(CC)C1.c1(C=O)ccc(F)c(C(N)=O)c1 c1(NC(CC2CCCC(NC(C(CC)O)=O)C2)=O)cccc(F)c1C c1(C(=O)NC(CC=CC)C(=O)NCC2(O)CCOC2)ccc(C)c(C)n1 Cc1ccc(CCNC(=O)C(CNC(=O)C(C)OC2CCCC2)N(C)C)s1 CCC(C)C(C(C(=O)NC1(C)CC1)N1CCC1(C)CCN(C)C)OC.C1CC1 N1(C(CN(C2CC2)CC)=O)CCC2CCC(C1)N2C(=O)C(O)Cn1cncn1 c1(N2CC(C)(C3CC3)OCC2)ccc(S(=O)(=O)NCc2ccncc2)cn1 C(=O)(CCC(F)F)NCC1(COC)CN(C(c2ccncc2Cl)=O)C1 c1(C(=O)OCC)cccc(NNC(=O)NC2CN(c3ncccn3)CCO2)c1F n1(CC)nnnc1C(c1nc(COC)cs1)NCCSCC(F)(F)F CCCCC(CC(=O)N1CCOC(C2CCC2)C1)NC(C1CCC(=O)O1)=O c1(CC(=O)N(C)CC=CC(=O)NC2C[Si](C)(C)C2)cncnc1 C1(CNC(C2(C=C)CC2)=O)(NC(=O)Cc2c(CC)noc2)CCCCC1C CCCN=C(NCC12CC(C)(CO1)C2)NC(C)C c1(OC)ncc(C)cc1CNC(=O)NCc1cnc(N2CCOCC2)nc1 CCC(COC)(CC)C(=O)NC(C)CCN(C)C(c1ncoc1C)=O N1(C(=O)OC(C)(C)C)CC(C=O)C(F)(F)C1.c1nn(CC(F)(F)F)cc1Cl.N C1(C(=O)NCCCOC(=O)NC)CCN(C(=O)CC2CCOC2(C)C)O1 CC1(C)CC(C(N2CCCC3(CO)CCCC23)C(=O)NC2(C)CC2)CC(C)(C)O1 c1(NC(=O)OC)ccc(CN2CCCC(C(C)C(=O)NC(CO)CO)C2)cc1Cl C=CC1(C(=O)NC(C)C(O)C(F)F)CCN(C(c2cc(C)cc(C)n2)=O)CC1 CC1CN(C)C(C)CC1NC(=O)C(C1CC1)N(C)C(c1cc(O)ccc1F)=O Cc1cc(=NCC2CN(C(C3CCCCO3)=O)CC23COC3)[nH]c(C)c1C#N C1(CCC)CN(C(=O)C(C)(C)F)CCN1C(=O)COc1cc(F)ccc1OC Cc1c(C(=O)NCC(C)(O)CNC(=O)C(C)Cc2ccccc2)[nH]ccc1=O n1(CC=O)ccc(=O)c([N+](=O)[O-])c1.CC(C(=O)N(CCC)C)C1CC1.CC.O S(=O)(=O)(c1ccc(Cl)c(Cl)c1)N1CC2N(C(C3CC4CCC3O4)=O)C2C1 c1(C(N2CCCC(CN(C(CCOC)=O)C)C2)=O)ccc(OC)c(C(F)F)c1 C1(C2CCCN(C(C3CC(F)C3)=O)C2)(NC(=O)CS(=O)(=O)C2CC2)CC1 Cc1cc(C(=O)NC2(CNC(c3ccccc3)=O)CCOC2)c(N)c(F)c1 n1(CCc2ncn(C)c2)cc(C(=O)NCc2nnnn2C2CC2)c(O)nc1=O Cc1cc[nH]c(=N)c1C(=O)NCC(C)NC(C1(C)CCN(C)C1)=O N1(CC)N=C(C(=O)NC2CC(O)C2)CCC1=O c1(C(N2CCN(C(C3N(CC)CCCC3)=O)CC2CO)=O)ncc([N+](=O)[O-])n1C C1(C(N2CC(C)(C)CC2)=O)CN(CP(C)(C)=O)C1.CCCC(C(=O)N)OCC.C C(CCS(N)(=O)=O)c1cn(CCNC(CCCN(C(C)C)C)=O)nn1 CCCC(CCC)CC(=O)NC(C)(C)CN(C(=O)C1=C(Cl)CC1)C c1(CNC(CN(C(=O)CC2CCCNC2=O)CC#C)=O)cnc(OC)cc1C Cc1cc(C(N2CCOCC2C(=O)NCCC2(O)CCC2)=O)ncc1N c1(C(=O)NCC(C)N(C)C(c2cc[nH]n2)=O)cnccc1C1OCCO1 Cc1nc([N+](=O)[O-])cn1CC(=O)Nc1cc(N2CCCC(C(N)=O)C2)ncn1 c1(C(N2CC(CN=c3[nH]cnc(C)c3F)OCCC2)=O)ccc2c(cnn2C)c1 CON1CC(C(=O)N(C)CC2CN(C(c3ccncc3Cl)=O)CCO2)CC1=O c1(C(=O)N)c(F)cc(Cl)cc1Br.c1(C(N2CC(O)C2)=O)ccc(Br)c(Cl)c1Cl.C C1(NC(C(n2cc(Cl)cn2)C)=O)CCCC(NC(C2CCCOC2C)=O)C1 C1(C)(C(=O)NC(c2ncccc2F)C)C=CCN1C(=O)CCCF C1(C(=O)NCCCC(C)NC(=O)CCC2OCCO2)CCC(F)(F)CC1 c1(C(=O)NCCCNC(C2(O)CCCC2)=O)cnc2ccccn2c1=O C1(NC(=O)Cc2ccc[nH]2)CCC2CN(C(=O)CC34COCC(C3)C4)CC2C1 C1(C(=O)NCC2(NC(C(C3CCOCC3)C)=O)CC2)C(C#N)C1(C)C CCCC(CC)CC(=O)N1CC2CCN(C(=O)CCc3ccccc3Cl)C2C1 CCC(C)(CC)C(=O)N(CC(C)C(=O)NCC(C)C(C)(F)F)C C(=O)(C1=NOC2COCC12)N1CCC(C(N(CCC(O)CO)C)=O)C12CC2 C(=O)(CCCC(C)=O)N(C(CNC(c1c(N(CCCC)C)cccc1)=O)C)C c1(CCC(=O)N)cccc(F)c1F.Cc1oc(CO)cc1C(=O)NCC=CC N1(C(C2(NC(C)=O)CC2)=O)CC2CCCC2C1.n1(C(C=O)C)cc(Cl)cn1.C CCC(CN(C)C)CC(=O)N1CCN(C(=O)C2=CCCC2)C(CC(=O)NC)C1 C1(C(N2CCC3(C(NC(c4nnc(C)o4)=O)C3)CC2)=O)Cc2ccccc2CN1 C1(C(N(CC(=C)C)Cc2ccc(CC)cc2)=O)CCc2cnn(C)c2C1 N1(C(C2CCC(NC(CCCC#N)=O)C2)=O)CCC2(CSC2)C1 C(C(CO)C(F)(F)F)NC(C1(CC#C)CCN(C(c2cc(F)ccc2F)=O)C1)=O c1(C(c2nnnn2C2CCCC2)NC2CC(CCOC)C2)cc(Cl)cs1 C(=O)(C1CCCc2n[nH]cc21)NC(C)(C)CNC(C12CCCC(C)(C1)OC2)=O N1(C(C2CN(C(C(COC)COC)=O)CC2C)=O)CCCC(O)CC1 C1(NC(CCSC)=O)C2CCC(C2)C1C(=O)NCc1cn(C)nn1 N1(CC)CC(C(N2CCC(C)(C)C2)=O)CCC1=O.c1(C=O)ccc(O)c(Cl)n1.N CN1CCC(C)(C(=O)NCCCN(CCCCNC(=O)Cc2ccsc2)C)C1 Cc1cccc(C(F)(F)C(=O)NCC(C)C2CC2)c1.c1(CC(=O)N)nocc1C c1(C(=O)NC(C)CCNC(C2CCC(F)(F)C2)=O)nc[nH]c2ncc(Br)c1-2 C1(C(N2CCC(C(C)NC(c3cc(O)n(C)n3)=O)C2)=O)CC2(C1)CC(F)C2 c1(C(N2C3C(CNC(C4(C)CCCC4)=O)C(C3)C2)=O)cnc2c(F)cccc2c1 CN1CCC(C)(CNC(=O)CC2C3CN(C(C4(Cl)CC4)=O)CC23)C1 C1(CC(N2C(C)(CC(=O)NCCN3CCOC3=O)CC2)=O)CCOC1(C)C c1(C(=O)NC2C=CCN(C(c3c(C)noc3)=O)C2)cn(C)ccc1=O CCC(CC(=O)N1CCC1C(=O)NCc1ccc(C)o1)C(F)F Cc1ncc([N+](=O)[O-])n1CC(=O)NC1CCN(C(=O)CC2CCCC2(F)F)C1 Cc1cc(NC(=O)CCC2CCN(C(C3CC(F)(CF)C3)=O)C2)c(C)c(C)c1 N1(C(C(CN(C(C(CC=CC)C)=O)C)C)=O)CCC2CCN(C)CC12 C(C)(CC(F)(F)F)NC(C(C)C)=O.C1(C(=O)N)CCN(c2cccc(F)c2)C1=O c1(CC(=O)NC2CCC(Nc3nc(C)cc(C)n3)CC2)ccc2c(c1)NC(=O)C2 CCC(CN(C)C)CC(=O)NCc1cc(C(=O)NCCC(O)C(=O)OC)co1 CC(C)(C(F)(F)F)OCC(=O)N.C(=O)CC(F)(F)F.CC(C)CO.C(=O)C C(=O)(CCCCc1ccccc1O)N(CCNC(CCSCC)=O)CC C1(C(=O)NCC2CC23CCOC3)CNc2ccnn2C1 CCCC(C)(O)C(=O)NCC(C)(C)OCCNC(=O)CCCC=O.C(C)C.N c1(C(N2C3(CN(C(CN(C)C)=O)C3)CCCC2)=O)cnc(O)c2c1NCCC2 C(=O)(CC(CC)C(F)F)N1CC=C(C(=O)NC2(C#C)CCOC2)C1 CCCC(C)CC(=O)N1CCCCC1CCN(C)C(c1cc(CCCO)on1)=O n1(CC=O)ncn2cccc2c1=O.C1(C=O)CS(=O)(=O)C1.CC(C)C1CC1.N C(=O)(C1CCC(=O)c2cccn21)N1CC(CC(C)NC(c2c(C)cc(C)o2)=O)C1 c1(C(N2CCC(=CC(=O)NC3CCNC3=O)CC2)=O)cnc2cccc(Cl)c2c1 CC1(C(=O)NCCSCCO)CCCN(C(C2CC(=O)NC(=O)C2)=O)C1 C12(C(N(CC(C)CNC(=O)C(C)(C)CN(C)C)C)=O)CCCC(C1)OC2 C=CC(CCC)CC(=O)NCC1CCCN1C(C1(c2ccc(Cl)nc2)CC1)=O C(=O)(CC(C)C(C)C(C)C)NCC#CCNC(Cn1nc(C)c(Cl)c1)=O C1(CNC(c2ccc(CNC(CC(C=C)C)=O)s2)=O)CCCC2(CC2)C1 C1(C(N2CCC(CNC(CCC#CC)=O)C2)=O)CCCCC1(C)C N1(C(C(c2ccncc2)C)=O)CCC(O)(C(C)NC(=O)C(=O)NC2CC2)C1 C1(NC(c2c(COC)ncs2)=O)CN(C(=O)C(Cc2ccccc2)OC)CC1C N1(C(CC(COC)(C)C)=O)CC2(CCN(Cc3nc(C)cs3)CC2)C1 C(=O)(C(C)(C)CC(F)F)NC1C(C)(C)CN(C(c2cnncc2O)=O)C1 c1(NC)c(C(N2CCC(C)(C)C2)=O)cccc1F.c1(C(=O)N)cc([N+](=O)[O-])n[nH]1 C1(C(N2CCC(CNC(C3(C)CCC(=O)N3)=O)C2)=O)CC2CCCCN2C1 C(=O)(C(F)CCC(C)C)N1CCC(CC=C)(C(N2CCC(F)(CO)C2)=O)C1 C1(C(=O)NCc2cc(C)[nH]n2)CCCN1NC(=O)c1ccc(O)cc1F C(=O)CC(C(F)(F)F)P(C)(C)=O.CN1CCOCC1C(=O)NC1CC(F)C1.C C(CCC(C(=O)N(C)Cc1cccnn1)NC(=O)CC1CC2(CC2)C1)OC CC1(CCNC(C23CC(NC(=O)CC4CCSCC4)(C2)C3)=O)CC1(F)F c1(-n2c(C=O)ccn2)ccc(C)cc1.C1(C(=O)NC2CC2)(OCC)CCC1 C(=O)(CCCCC(F)(F)F)NCC1CC(NC(C(CC)(C)C#N)=O)C1 c1(C(=O)Nc2c(NCC)ccc(Cl)c2)cc([N+](=O)[O-])c(C)cc1Cl C(=O)(CC(C)C)N(CCNC(=O)C(C)SC1CCCC1)CC.C(=O)N c1(C(N2CCN(C(C(C)NC(=O)OC)=O)CC2C)=O)cc2cc(C)ccc2o1 N1(C(c2cc(C)sc2C(F)(F)F)=O)CCCC(C)(NC(C2CCCN(C)C2)=O)C1 Cc1cc(C(=O)NC(C)(C)CCCNC(c2ccc(F)cc2N)=O)nc(O)n1 C(=O)(CS(=O)(=O)CCC)N1CC(C=C)C(NC(C2CSCCS2)=O)C1 C1(CC)(NC(=O)CN2CCCS2(=O)=O)CCN(C(=O)CC2CSCCO2)CC1 C1(NC(c2ccc(SC)cc2)=O)CCC2CN(C(=O)C3=COCCO3)CCC2C1 c1(NC(=O)NCCCCSC(C)=O)cc(O)nc(C2CCOCC2)n1 C1(C(N(CC(C)NC(=O)COC(C)(C)C)C)=O)CCC2(CCC2)O1 C1(CC)CN(C(c2ccc(C(F)(F)F)o2)=O)CCN1C(C1CCCC(C)(C)C1)=O C(CC(CC)C(=O)N1CCN(CC(N2CCC(C)(NC(C)=O)C2)=O)CC1)=CC CCCCC(CC(=O)NCC1CCC2(CC2)CO1)NC(c1cnc(OC)cn1)=O c1(COC)ccccc1.C1(C=O)CC(O)CN1C(c1cc(C(F)(F)F)cs1)=O C=CCC(CC=C)C(=O)NCC(C)(C)C#CC(=O)NC(CCCCC)C1CC1 c1(C(N2CCC(OC)C2)C(=O)NC2CC2)n[nH]c(C)c1Br C1(CNC(C(CSC)C)=O)CC(C)CCN1C(=O)CN(C)S(N)(=O)=O CC1CN(C(c2ccc(O)nc2Cl)=O)CC(C)N(C(=O)C(C)CCN(C)C)C1 c1(OCC)cc(C(=O)Nc2oncc2C#N)c(-c2cncc(C(=O)NC)c2)cn1 CC(C(C)(O)C(=O)N1CC(CO)(NC(=O)CCCN(C)C)C1)c1ccccc1 Cc1cc(C(=O)NC2(CCC)CC2)c(N)cc1F.C1(C)(CC=O)CC1(F)F.N C1(NC(c2cc(C)sn2)=O)CC2CC1N(C(=O)CN(C)S(=O)(=O)N(C)C)C2 N1(C(c2cccc(NC)n2)=O)CCC(CNC(=O)C(=O)N(C)C)CC1C C12(NC(c3[nH]cc(CC)c3)=O)CCCCCC1N(C(c1c(Cl)n[nH]c1C)=O)CC2 c1(OCC)ccnc(Sc2cnn(CC(O)CN3CCOCC3)c2)n1 N1(C(c2nc(C(C)=O)sc2)=O)CCOCC1CN(C(=O)CN1CCC(C)C1)C C1(=CC(=O)NCCCN2CCOCC2)CCN(CC2CC3(CCC3)C2)CC1 C1(C(C)NC(=O)C=Cc2cnc[nH]2)CCCCN1C(C1C=CCC1)=O Cc1nn(C)c(-n2cncn2)c1C(=O)NCCNC(c1ccccc1Cl)=O c1(C(=O)NCC2N(C(Cc3cc(C)cc(C)c3)=O)CC=C2)c[nH]c2cccnc12 Cc1cnncc1C(=O)NC1CCC1NC(C1(C)C=CCC1)=O C1(CN(C)C)CCN1C(=O)CCC1CC(NC(=O)CCC2(C)CC2)C1 Cc1cc(C(=O)NC2(CNC(C3CC(O)CN3C)=O)CCOC2)c(O)nn1 N1(C(c2ccc(COC)s2)C(=O)NCCSC)CCC(C)(F)C1 C(=O)(CCCCNC(=O)CN1CCC(OC)CC1)OCC C1(CC(=O)NC2(C(=O)NCCC3CCOCC3)CCSC2)CCCC1O CC1OC2(CNC(c3cocn3)=O)CC1(NC(C13CC(F)(C1)C3)=O)C2 Cc1c(C(=O)NC2CN(C(=O)CC3CCCCC34CC4)C2)ccc(Br)c1F C1(CC(=O)NC2C(NC(C3(CC=C)COC3)=O)CCCC2)Cc2ccccc2O1 c1(C=O)cccc(Cl)c1.c1(C(N2CC(CC=O)C2)=O)nc(C)ncc1Br.CC.O CS(=O)(=O)c1nccc(N2CC(O)(CCNC(=O)C(C3CCOCC3)O)C2)n1 C1CCCCCCC1.C1(C(=O)NC)CCN(C(=O)C(CC#N)c2ccccc2)CC1 N1(C(CCC(=O)NC)=O)CC2(CCC(C)O2)C1.c1(C(=O)N)cc2cc(Cl)sc2[nH]1 C1(NC(C(C)NC(C(CC)OC)=O)=O)CC(=O)N(C2CN(CC)C2)C1 Cc1[nH]nc(C(=O)NCC2CN(C(c3c(Br)cnn3C)=O)CC2C)c1Cl CC1CN(C(c2ccc(C(N)=O)cc2)=O)CCC1.C1(C(=O)N)CC2C(C1)C2(C)C C1CCC2CN(C(C3(F)CCC3)=O)CCC2C1.c1(C(=O)NC)cc(C2CC2)no1 N1(C(Cn2cc(C(C)O)nn2)=O)CCN(C(c2ccc(Br)o2)=O)C(CCO)C1 C1(C)(C(=O)NCCCN2CCN(C(CC(C)OC)=O)CC2)CCC12CCC2 C1(C(=O)NCC(=O)NC(C)CN(C)C(C)C)(OC)CCC(C)C1 Cc1c(C(=O)NC2CSC2)[nH]c2ccc(C3=CCCC3)cc12 c1(C(=O)NC(C)Cn2cc(C3CC3)nn2)nc(-c2ccccc2)cn1C c1(C(=O)NCC(C)CN(C(=O)C#CC2(C)CC2)C)cc2ccc(Br)cc2[nH]1 Cc1nc2cc(C(N3CC4C(NC(C5(C(C)(C)O)CCC5)=O)C4C3)=O)[nH]c2s1 N1(C(c2cc(C(N3CCN(C(C)=O)CC3)=O)n[nH]2)=O)CC(CO)C(C)(C)C1 N1(C(CC(CC)C(C)C)=O)CC2CCN(C(=O)CCC3CCOCC3)C2C1C C1(NC(COCCC)=O)CCC2(CC1)CCN(C(=O)C(C)(C)c1ccc(Cl)s1)C2 C1(C(N2CCCC(CC)C2)=O)CN(C(=O)CCc2nncn2C)C(C)(C)C1 C1(CNC(CC)=O)CCC2CN(C(c3coc4c3CSC4)=O)CCC2C1 N#Cc1ccc(C(N2CCN(C(=O)CCC3CCOC3)CC2CCO)=O)nc1 N1(C(C=C(C)C)=O)CC2(C)CC1(C(=O)NCC(C)(C)n1ccnc1)C2 Cc1cc(CC(N2CCC(n3cc(C4CC(F)(F)C4)nn3)CC2)=O)cc(Br)c1 CCC(CCC(=O)N1CCC(CO)(NC(c2ncc[nH]c2=O)=O)C1)OC C1(NC(C(=O)NCC2N(CC)CCC2)=O)CCC2(CC1)N=N2 CCCCCCCC(=O)NC(C1(CNC(=O)CCCCC(N)=O)CC1)C Cc1cn2c(n1)C(C(=O)N1CCC(F)C(NC(c3cnn[nH]3)=O)C1)CCC2 CCC(F)(F)CN(C(=O)C(Cc1cc[nH]n1)NC(=O)CCNC(N)=O)C c1(CC(=O)NC2CN(C(C(CC=CC)C)=O)CC2O)cc(C)cc(F)c1 c1(C=O)ccccc1.C(C)(C(=O)N(C)CC1(C)CC1)SCCCC.C(C)C C(N=c1[nH]c(=NCCCN2CCCC2)[nH]c2cccnc12)C1(OC)CCC(C)C1 c1(CN(C)C(c2coc3c2CSC3)=O)c(F)cccc1F C(CN=c1[nH]c(Cl)ncc1C)C1CCN(C(C=CC(CC)=CC)=O)C1 C12(CNC(c3cccc(C)n3)=O)CCC(CNC(=O)CCCF)(CC1)OC2 c1(CNC(CC(C)c2ccco2)=O)cnn(C)c1C=O.CCC(C)(O)C1CC1.N c1(C(N2CC(CNC(c3cc(C)c(C)o3)=O)C(C)C2)=O)ncnc2c1cnn2C C(=O)(CCCC(=O)NC(C)C(C)NC(=O)CC(C)CC1CC1)NCCC CC1(C(=O)NCCC2CCN(C(=O)CCc3ccncc3)CC2)CC2CC2C1 n1(CC=C)cc(C(=O)NCc2nc(C)cs2)nn1.c1(C(C=O)O)ccccc1 C(=O)(CCN=c1[nH]ccs1)N1C2CC(NC(=O)Cc3cc(F)ccc3F)(C2)C1 C1(C)(NC(C(c2ccccc2)C)=O)CCCN(C(C2CCN2C2CCCC2)=O)C1 C(=O)(CCCCC(=O)NCC(C)=CC(=O)NC1(CO)CCOCC1)OC c1(-c2nnc(N3CCC(CC)C3C)n2CCC2CC2)c[nH]c2ccccc12 N1(C(c2cnc(C)[nH]2)=O)CCC(NC(C2CN(S(N)(=O)=O)C2)=O)C2(CCC2)C1 c1(CC(=O)NC2C(CNC(C(Cc3c(C)nc[nH]3)O)=O)CC2)ccccc1Cl C=Cc1cnc(NC(=O)Nc2cccc(N3CCOCC3=O)c2)nc1 C(C)(CS(C)(=O)=O)N(C(c1c(C)cco1)C(=O)NCC1CCOC1)C c1(CC)cccc(C(N2CCC(O)(CNC(c3cnns3)=O)C2)=O)c1C c1(C(N(CCCN(C(C2C(C)C2C)=O)C)C)=O)cccc([N+](=O)[O-])c1 CC(C)CCC(=O)C(=O)N1CC2CCC(CNC(=O)CC3(O)CCOCC3)(C2)C1 N1(C(c2c(C)cc(F)s2)=O)CCN(C(=O)CC2CCC(=O)NC2)CC(C)C1 C(=O)(C(C)CC(C)C)NC1C2CCN(C(CCCOC)=O)C21 Cc1nn(CCS(=O)(=O)Nc2ncncc2OC(C)C)c(=O)o1 c1(OC)cnc(Br)cc1C(=O)NCC(C1CC1)NC(=O)Cc1c[nH]nc1C CC1CC(C(=O)NCC(CO)NC(=O)CSC(F)(F)F)C1 C1(C(=O)NCC2CCC(NC(=O)C=CC(F)F)C2)CC2CCC(C1)S2 CC(O)CCN=c1[nH]c(N2CCN3CCOCC3C2)nc2c1CCCCC2 N1(C(C=CC(C)(C)SC)=O)CCCC2C1CCN2C(c1c(C)cc(Cl)cc1N)=O C1(S(C)(=O)=O)(CNCC2OCCN(S(C)(=O)=O)C2)CC1C(F)(F)F N1(C(C2C(C)C2)=O)CC(C)CN(C(C2CC(=O)N2)=O)CC1C C1(C(=O)NC(CCOC)CO)CCN(C(=O)COC)CCO1.C1(O)CC1 N1(C(Cn2nnc(C)n2)=O)C(C)CC2CC12.C12(C(=O)N)CCCC1(C(N)=O)C2 C12(C(=O)NC3C(NC(Cc4cccc(C)c4C)=O)COC3)CCC(=O)N1CCS2 Cc1cc2c(C(=O)NC(C)C(CO)NC(c3cnc(C)c(N)c3)=O)cccc2[nH]1 c1(C(N2CCC(CNC(c3cc(C)sc3)=O)C23CC3)=O)cnn2c1NCC(C)C2 Cc1cccc(-c2nc(C(N3CC(CC(N)=O)C3)=O)cs2)c1 c1(-c2c(OC)ccc(C)c2)nccc2c(Br)cccc12 c1(OC)ccccc1CCNC(c1ccsc1C(F)F)=O.C1(C=O)CC1.N N1(C(CC2CCN(C(C3(NC(C)=O)CC3)=O)C2)=O)CCCC(O)CC1 CS(=O)(=O)c1coc(C(N2CC(C3CN(C(=O)CC4=CCCC4)C3)C2)=O)c1 c1(C(C)O)cc(-c2cc(NC(C3CCC3)=O)ccn2)ccc1F N1(C(C=COCC)=O)CCN(C(=O)C(n2ccc(Br)n2)C)CC1CF C(=O)(C(C)(CO)CO)OCC(C(=O)N1CC(OC(=O)NCC)C1)C c1(C(=O)NC2C(C)CCN(C(c3n[nH]cc3Cl)=O)C2)ccn2ncnc2c1 N#Cc1c(OC2CCN(C3CCOCC3)CC2)cccc1Br c1(CSC)ccc(CNC(=O)NCC(C)NC=O)cc1F.C(C)(C)C c1(OC)ccc(Cl)cc1N(CCC(F)(F)F)CC(=O)NC(C)(C)C C=C(C)c1cncc(C(C(=O)NC)N(C(C)COCC)C)c1.c1ccccc1 C1(C(=O)NCCCOCCCNC(=O)C=C(Cl)Cl)CC2CCC1O2 CC1CC(=O)NCC1C(=O)NCC1(O)CCN(C(=O)CCc2cncnc2)CC1 C1(NC(CC(CC)CC)=O)CCCCN(C(c2c(C)noc2C2CC2)=O)CC1 c1(C(=O)NCC(C(=O)NCc2scc(C)c2)C)ccc(=O)n(C)n1 S(=O)(=O)(c1ccnn1C1CCCC1)NC(c1ccc(OC)c(-c2ccncc2)c1)C CC(C)CS(=O)(=O)CC(=O)N1CCC(C)C1CNC(c1c[nH]cc1Br)=O C#Cc1cc(C(=O)N(C(C)CNC(=O)C(C)CC=CC)C)cc(Br)c1 c1(C(N2CCC(N(C(=O)C=C3CC3)CC)C2)=O)cc2ccccc2cc1O CC1CCN(C(c2sccc2Cl)=O)CC1CNC(CCC(=O)N1CC(CO)C1)=O c1(C(N2CCCC(C)(NC(c3cc(Cl)no3)=O)C2)=O)nnn2c1CCCC2 C1(C)(C(=O)N)CCCNS1(=O)=O.N1(C(c2scc(OC)c2)=O)CCCCC1CC N1(C(=O)NCc2c(C)nn(C3CC3)c2)CCOCC(C)(O)C1 CON1CCC(CC(=O)NC2CC2NC(=O)C=C(C)Cl)CC1 Cc1cnc(C(N2CC3CC2C3NC(=O)CS(=O)(=O)C(C)C)=O)cc1C#N N1(C(c2n(CCC)ccc2)=O)CCC(NC(=O)C=C2CCC(C)CC2)C1CC N1(C(C=C2CCC(C)CC2)=O)CCC2(CC2)CC1C(N1CC2CC1CS2=O)=O N1(C(=O)CCC)CC(=O)NC(C)C1.c1(C(C)C)ccc(-n2cc(O)c(C=O)n2)cc1 C(=O)(C(CN(C)C)NC(c1ccc(C2CC2)s1)=O)NC(C)C(N)=O c1(C(C=O)C)cc(F)cc(F)c1.N1(CC(=O)NCC)C(=O)CCCC1=O.CC C12(C(=O)NCC3C(C(=O)NC(CC)(C)CC)CCC3)C=CC(CC1)C2 c1(SC)cc(C(=O)NC2CC(F)C2)nn1C.N1(C(C=O)=O)CCC(C)CC1.C C(=O)(C1CCCc2nc[nH]c21)NCC(CCCC)NC(C1(C)CC(F)(F)C1)=O Cc1c(F)ccc(C(=O)N(C)CC2CCCN2C(=O)C(C)C(C)C)c1N CC1(C)CCCC1(C)NC(=O)C(C1CCC1)NC(=O)Cc1cncnc1O C=C(C)CN=C(NCC1CCC(C)(CC)O1)N1CCc2nnc(O)cc2C1 N1(C(c2n(C(C)C)nnc2)=O)CC2CCN(C(=O)CC(C)n3ccnc3)CC2C1 n1(CC=O)ccccc1=O.c1(CNC(CSC(C)(C)C)=O)csc(C)n1.N C1(NC(C(C)OC)=O)C2CC(NC(=O)C(C(C)C)NC(C)=O)CC12 c12ccc(cc1)CNC(=O)NC2.C1(C(=O)OC)CCCO1.C(C)=O.C C1(C(=O)NCCCCNC(c2c(C)cc(=O)oc2C)=O)Cc2c(C)cccc2O1 C12(NC(c3nc(Br)c[nH]3)=O)CC1CN(C(=O)CC13CCCC1C3)C2 N1(CC(=O)NC2(C(N(CC(CCC)O)C)=O)CCC2)CCNC(=O)C1 N1(C(C(C(CC)C)N)=O)CCC2(CC1)CC(NC(=O)Cc1nc(C(C)C)no1)C2 c1(C(=O)NC2(CCCNC(=O)Cc3cscn3)CC2)ncc(C2CC2)cc1F c1(CN2CCC(NC(C(C)CS(C)=O)=O)CC2)ccc2c(c1)CCCC2 C1(C=O)CC(C)(C)CC(C)(C)C1.C(=O)(C(C)CC(=O)NC1CC(O)C1)OC C1(CNC(c2csc(Cn3ccnc3)n2)=O)CN(C(=O)C#CC2CC2)CCCO1 S(=O)(=O)(c1cccc(NC(c2nocc2Cl)=O)c1)N1CC(N)C1 CC1(C)OC(C)(C)C1C(N1CC2CCC2C1)=O.c1(C=O)ccc(C(F)F)s1.C C1(CC)OCCC1C(=O)NC(C)CC(C)NC(=O)C(C)(C)c1ccccn1 C1(NC(C2C(CC(C)C)C2)=O)C2CN(C(C3CC(O)C3)=O)CC12 C1(CCNC(COC)=O)C(C)CCCN1C(C1CCN(C(=O)C2CC2)CC1)=O c1(C(=O)NCC2C(NC(=O)CC3(CO)CC3)CCCC2)nccc(F)c1Cl C1(CNc2cccc(NC(=O)NC(CC)(CO)CO)c2)CC2C(C1)C2(F)F C1(C(=O)NCC(COC)C)C=CC(NC(=O)OC(C)(C)C)C1 c1(C(N(C2CCN(C(=O)Cc3cnns3)C2)C)=O)cc(Br)cc2c1OCC2 N1(C(C2C(C=C)C2)=O)CCC2(CCCCC2NC(c2ccc(C)c(Cl)c2)=O)CC1 N1(CC(=O)OC)CCCc2cc(OC)ccc21.C1(=O)C(COC2CCOCC2)N1 N1(C(C(=O)NC2(CCO)CC2)=O)CC2(CC2C(F)F)C1 N1(C(C(C)(C)OCC)=O)CC2CCN(C(C3CC(=O)N(C)C3)=O)C(C2)C1 C#CCC(CC#C)C(=O)NC1(CC=C)CCN(C(=O)CN(CC)CC)C1 c1(C(C)=O)ccc(S(=O)(=O)N2CCCCC2C(=O)NCCC2CCOC2)cc1 N1(C(c2cc(CC)n(C)n2)=O)CCC2(CC2)C1.n1(CC(=O)N(C)C)nnnc1C c1(C(=O)NC(C(=O)NCc2nnn(CC)n2)C)cc(C#N)cn1C c1(C=O)coc2c1C(=O)NCC2.CC1CCCN(C(=O)COC2CC2)C1CC.N c1(OC)ccc(Cl)c(C)c1C(=O)NC1CCN(C(c2nc(O)sc2C)=O)C(C)C1 C1(CNC(COCCC)=O)CC2(CC(NC(=O)CO)C2)C1.C1CCC1 CCC(CC)=CC(=O)N(CC(C)NC(=O)COCC1CCCO1)CC c1(CC)cnn(CC(=O)NCC2CCCN2C(=O)C(=Cc2cccs2)C)c1 C1(CNC(c2on(C)c(=O)c2)=O)CCC12CCN(C(=O)CCn1ccnn1)CC2 N1(C(C2Cn3c(C)nnc3C2)=O)CCCC12CCN(C(C1(C)COC(=O)C1)=O)C2 Cc1cc(O)nc(C)c1C(=O)NCCCC(C)NC(c1cccc(C2CC2)n1)=O C(=O)(C(S(C)(=O)=O)C1CC1)NC(CCCNC(c1ccc(OC)nc1)=O)C c1(NC2CC(C)Oc3c2cccc3)cc(=O)c2ccccc2n1C c1(C(=O)NCC2=CCN(C(C(C)CC(F)F)=O)CC2)cc(Cl)c2c(c1)OCCO2 c1(C=O)c(F)ccc2nc[nH]c12.Cc1cc(C(=O)NC2(C)CC2)nn1CCO.N N1(C(C(COC)(F)F)=O)CC2CC(NC(=O)C=C(C)c3ccco3)C1C2 Cc1nc(C(N2CC(CNC(c3nc(C4CC4)cs3)=O)C(C)C2)=O)[nH]c1C N1(C(c2c(C)nc[nH]2)=O)CCC2CCC(NC(c3ccsc3S(N)(=O)=O)=O)C1C2 c1(C(=O)N)cnc(C2CC2)nc1O.n1(CC(=O)N(CC)CC)cnc(=N)[nH]1 [SH](=O)(=O)c1ccccc1.C1(NC(CNC(=O)OC)=O)CCC1.N(C)(C)C C1(NC(C=C(CCC)CCC)=O)CCCCCN(C(=O)COC2CCCCC2)C1 N1(C(c2cccc(OC)c2)=O)CCN(C(C23CC=CC(C2)OC3)=O)C(C2CC2)C1 C(=O)(C(C)(F)C(C)(C)F)NCCCCNC(C(c1c(C)n[nH]c1C)C)=O c1(NC(CN(CCOC)C(c2n[nH]c(C)c2O)=O)=O)ccc(C)nc1 Cc1nn(CC(=O)N(CCC)CC)c(C)c1[N+](=O)[O-].C(=O)C(C)CC1CCC1 CCCC(C(=O)N1CCCC(CNC(C23CCC(C2)C3)=O)C1)C(C)C c1(C(=O)NCC2CCN(C(COC)=O)C(C)C2)cc2cccnc2nc1C C1(NC(C(=O)NCC)=O)CC2(CCCN(C(=O)C(O)Cc3cnc[nH]3)C2)C1 c1(C(=O)NCC(C2CCC2)NC(C(C)=CC)=O)ccc2nnc(C)n2c1 c1(C(N(CC(C)CNC(=O)COC(C)(C)C)C)=O)cnc2n1CCOC2 Cc1ccc(O)c(CNC(=O)CC2CN(C(=O)CO)CCC2C)c1.CCC(C)C Cc1n[nH]c(C)c1SCC(=O)N(CC(O)CN(C(=O)CCc1ccncn1)C)C C1(N(C)C)CN(C(=O)CC2(C)CCCO2)CC1C.C1(C=O)CCC(C)(C)O1.N N1(C(C(CCC)C#N)=O)CC2(CCC2)CC1CNC(=O)CCc1cscn1 c1(C(CC(C)NC(CC)CC)O)ccccc1 C1(C(=O)NC2CCN(C(c3c(C)nn[nH]3)=O)C2)Cc2nncn2C1 c1(C(C)O)ncc(C(=O)NCCO)s1.C(C1CCOC1)=CC(=O)N(CC)C CS(=O)c1ccccc1C(=O)NC1CC(CCNC(=O)C=O)C1.C1CC1.N C1(C)(CC)CCCN(C(=O)CC2(C)CC2)CC1.c1(C=O)cncn1C(C)C.N CCCCC(CCCC)C(=O)N(CC(C)O)CCNC(c1cc(C)cc(F)c1)=O c1(SC)c(C(=O)NC2CCC(C)(C)C2)cccc1F.c1(C=O)nc(O)c(C)s1 c1(C(=O)NCC(CC)NC(=O)C(c2ccc(F)cc2)(C)F)ncnc(C)c1Br C(=O)(CC(C(C)(C)C)NC=O)N1CCC(C)C1.C1CC(=O)N(C)C1.C(C)(C)C C1(NC(C(CN(C)CC)C)=O)CN(C(c2ncsc2C(C)C)=O)CC1OC c1(C(=O)NCC2C(NC(CC(C)CN(C)C)=O)COC2)ccc2cnsc2c1 c1(C(=O)NCC2N(C(CCCCCSC)=O)CC=C2)cc2nccnc2cc1C N1(C(C(=O)NCCOC)=O)CCCCC(NC(=O)CC2CCSC2)CC1 N1(C(c2ccc(CC)s2)=O)CCC2(CC(C(=O)N(C3CC(O)C3)C)C2)C1 N1(C(C=CC)=O)CCC(C)N(C(C2CCCN2Cc2ccsc2)=O)CC1 C(CCCC(=O)NCCC1COCCN1C(C1OCCOC1C)=O)OCC c1(C(N2CCCC(C)(NC(C3CNC(=O)N3)=O)C2)=O)cc2cc(O)ccc2[nH]1 N1(C(C2=C(C)CC2)=O)CCN(C2CCCN(C(=O)CC3CCOCC3)C2)C(=O)C1 N1(C(=O)NC(C(C)C)C(=O)N2CCCCC2)CC2CC(=O)CC(C2)C1 c1(N(C(NOC)=O)C2CC2)ccc(C(F)(F)F)c(F)c1Br N1(CC)CCCC(C(N2CC(NC(=O)CCC3(C)CC3(F)F)C(C)C2)=O)C1 C1(CNC(CCc2[nH]c(=N)sc2)=O)CCCN(C(=O)Cc2ccccc2O)C1 Cn1cc(C2CCN2C(c2ccc(C(C)(C)C)s2)=O)cn1.n12cc(nn1)C2 c1(N2CCCC(c3c(C)cccc3)C2)nc(C2CC2)nc2ccsc12 CN=c1cc(C(=O)NC2CCN(C(=O)CCSc3ccccc3)C2C)cc[nH]1 c1(OCC)ccc(C(N2CCN(C(=O)CS(N)(=O)=O)C(CF)C2)=O)c(F)c1 C1(NC(c2cc(C(C)C)nn2C)=O)CC2CN(C(c3ccc(F)nc3F)=O)CC12 N1(C(CN(C)C2CC2)=O)CCC2(CCOCC2)C1.C(=O)C1=CCS(=O)(=O)C1.C N1(C(c2cnc(SC)s2)=O)C2CCC1CN(C(=O)Cc1cnnn1C)C2 N1(C(c2cc(OC)cc(C3CC3)c2)=O)CC2CC(C(=O)O)C(C2)C1 Cc1cc(=O)ccn1CC(=O)NCC1CC(NC(C2(C)CCCC2)=O)C1 N1(C(C2CCCOC2)=O)CCC2(CC1)CCN(C(=O)C(c1ccc(Cl)cc1)O)CC2 c1(C(=O)NCCN(C(=O)CCc2cc(C)no2)CC)ccc(C)n1C C(=O)(C(F)CCC(C)C)NC1CC(C(N(C(C#C)C)CCCC)=O)C1 C(=O)(C1CCc2c(Cl)cccc21)N1C(C#C)CN(C(c2ccsc2)=O)CC1 c1(OCCCC(=O)NCC(CO)NC(C(CC)NC(N)=O)=O)ccccc1C N1(C(C2OCCN(C)C2)=O)CCC2CC1CN(C(c1cnc3n1CCC3)=O)C2 c1(C(N2CCN(C3CNC3)CC2)=O)cc2ncccc2[nH]1 C1(C(=O)NCC2(C)CC(C)C2)(CC)CCCN(C(=O)CCC(=O)NC)C1 c1(C(=O)NCC(N2CC(C)OC(C)C2)=O)ccc(N=NC(N)=O)cc1 c1(C(=O)NC(CN(C(CCC(=C)Cl)=O)C)C)ccc(F)c(C(F)(F)F)c1Cl C1(CCNC(=O)C=CC)(NC(C2(COC)CCCC2)=O)CCOCC1 N1(C(C2C(C)C2)=O)CC(NC(c2cc(CN(C)C)c[nH]2)=O)CC1(C)C C(=O)(C1=CC2CC(C1)CC2O)N(C1CCN(C(C2(CCF)CC2)=O)C1)C c1(C(=O)NCCC(C(C)C)OCC)ccc2c(c1)nc(C)n2CCO c1(OC)cc(C)c(CCNC(N2CCC3(C2)CC3(F)F)=O)cc1OC c1(C(N2CC3CC(NC(c4cc(C5CC5)on4)=O)C3C2)=O)cc2ccccn2n1 Cc1oc(S(N)(=O)=O)cc1C(=O)NC1CC2(C1)CCC2.C(=O)CC(F)(F)F CC(CC1CCCO1)N=c1ccc2cc([N+](=O)[O-])ccc2[nH]1 C(=O)(C1=CC(O)CCC1)NCC1(C(C)C)CCN(C(CCn2c(C)ncc2)=O)C1 C(CN=C(NCC1CCCO1)NCC1CCCC1(F)F)C1C(F)(F)C1 c1(C(N(CCNC(C(c2ccccc2)SC)=O)C(C)C)=O)cncc2nc[nH]c12 N1(C(COC(C)=O)=O)CCC2(CCN(C(c3cc4ccc(Br)cc4[nH]3)=O)CC2)C1 N1(C(Cc2c(C)cccc2)=O)CCCC2(CCN(C(=O)CC(C)C(C)(C)C)C2)C1 O=CN1CCOCC1C(=O)NC1CC12CCN(C(=O)C(F)C(F)(F)F)C2 C1(CNC(C2CCOC2)=O)CCCCN(C(=O)C(O)C2CCC2)C1 CCC(C)C(=O)N(CCC(=O)N1CC(CC)(CO)C1)OC C1(CNC(c2ccn(Cc3ccncc3)n2)=O)CCC2(CCOCC2)O1 c1(OC(C)C)cccnc1C=O.C1(CC)CCN(C(=O)C(C)CC2CC2)CC1.N CCCCC(CC)C(=O)NCCC(C(C)C)NC(=O)C(=O)NC(C)C O(NC(=O)C(CC1CCOCC1)NC(C1CCCC(=O)CC1)=O)C(C)(C)CO N1(C(C(CCC)C#N)=O)CCC2(CC1)CC2NC(c1c(Cl)cc(Cl)cc1Cl)=O C(=O)(CCC(=O)N1CCCC(CCCO)C1)NC(CC)(C)CNC(=O)C(C)(C)C N1(C(C(CCCC)O)=O)CCC2CN(C(=O)Cn3ncc(Cl)c3C)CCC12 c1(CNC(C(c2ccccc2Cl)N)=O)cnc(Br)c(F)c1 N1(C(C2N(C(C(C)C(F)F)=O)CC(F)C2)=O)CCCOCC1C Cc1cnc(C=CC(=O)NCC2CC(F)CN2C(C2CC(C)(O)C2)=O)[nH]1 C1(NC(C(F)=CC)=O)C2CC3CN(C(=O)CC(CC)C4CCC4)C1C3C2 N1(c2snc(C(C)C)n2)CC2C(CNC(C3(c4cccc(Cl)c4)CCC3)=O)C2C1 c1(CC)cccc2nc(C(N3CCC4CCCC4CC3)=O)sc12 C1(CNC(C(CC(=C)C)OC)=O)CCC2(CN(C(c3ccnc(C)c3N)=O)C2)O1 N1(C(C(C)OCCN(C)C)=O)CCC(C)(C)C(NC(c2cncc(N)c2)=O)C1 Cc1ccc(Cl)c(C(N2CCC(CCN(C)C(C3CC(Cl)(Cl)C3)=O)CC2)=O)c1 c1(C(=O)NCC(CC)NC(C2CC2F)=O)cc2c(Br)cccc2c(=O)o1 C1(NC(c2c(CC)n[nH]c2)=O)COC2(CCN(C(c3cnn(C)n3)=O)C2)C1 C1(C(N2CC(CNC(c3cc(C)oc3)=O)C(C)CC2)=O)CCCC2CCCCC12 C1(C(=O)NC(COCC)C)CCOC1CNC(C1(CC)CC1)=O C1(C)(COC)CCN(C(=O)C(CC2CCOCC2)NC(=O)Cn2cccn2)C1 Cc1nc(C(C)C)ncc1C(=O)NCC1C2CN(C(C3CC3C#N)=O)CC12 c1(C(=O)NC(CNC(C(C=CC)O)=O)CCOC)cc(Br)cnc1C1CC1 CC1CN(C(c2cc(Cl)c(Br)[nH]2)=O)CCC1NC(=O)CCn1ccnn1 c1(C(C=CC=O)=O)ncccc1O.CC(C)CO.C(C(F)(F)F)C1(C=O)CC1 N1(CC)CCOCC1C(N1CCC(O)(C(C)NC(=O)CC2(C)CC2)C1)=O N1(C(CN(C)C)=O)CC(F)(F)CC1Cn1cc(CCO)nn1 N1(C(c2cc(C)[nH]c2)=O)CCC(C)C(NC(=O)C(c2ccccc2Cl)C)C1C Cc1cc([N+](=O)[O-])cc(C(=O)NC2CC(C)N(C(=O)CCCF)C2)c1Cl c1(C(N2CCCC(C(N3CCC(C)(OC)C3)=O)C2)=O)ccc(F)c(C)c1F C=C(Br)CC(=O)NC1(CCO)CN(C(=O)C(C)NC(C2CCCCC2)=O)C1 c1(C(N2CCC3CN(C(c4cscc4Br)=O)CC32)=O)ccc2c(c1)OCCO2 c1(OCC)cc(-c2ccc(=NCc3cccc(CN(C)C)c3)[nH]c2)c(F)c(F)c1 C1(NC(C(N2CCC(O)CC2)C)=O)(CF)CCN(C(=O)CC2COC(=O)N2)C1 C(=O)(C(F)C(F)(F)F)N1CCC(n2cc(CNC(C(C)C3CCC3)=O)nn2)CC1 CCCC(C)(CCC)C(=O)NCC12CC(NC(c3cnc(C)cn3)=O)(C1)C2 N1(C(C(CC)NC(C)=O)=O)CC2C(CC(=O)NC(c3ccc(C)nc3)C)C2C1 C(=O)(C(C)(C)CS(C)(=O)=O)N1CCC(NC(c2n(C)nc(O)c2)=O)CC1 c1(-c2c(C(=O)NCC(c3ccc(F)cc3)OC)n[nH]c2)ccc(F)c(C#N)c1 C(C)(C(=O)N1CCC(N(CCCn2nc(C)nc2C)C)CC1)(C(C)C)NC(C)=O c1(C(=O)NCC2N(C(C=CSC)=O)CCCC2)ccc2n[nH]c(C)c2c1 C(Cc1ccc(C(F)(F)F)cc1)(C(F)(F)F)N(CCCOCC)C c1(C(N2C(C)(C)C(C)CC2)=O)cc2ccccc2o1.C1(C)(CC=O)CC1(Cl)Cl.N N1(C(CCn2ccc(C)n2)=O)CCCCC(NC(C2CCCO2)=O)CC1 C1(CNC(c2ccc(C(F)(F)F)[nH]2)=O)C2CCCC1N(C(=O)CCC(F)F)C2 n1(CC(=O)NCC23CC(NC(=O)Cc4ccoc4)(C2)C3)cc(Cl)cn1 C(=O)(C1=C(CC)OCCS1)N1C(C)CC(OC)C1.c1(CC(=O)N)ccc(Cl)cc1 Cc1ccc2[nH]c(C(=O)N(C)CC3CCCN(C(=O)C=C4CC4)C3)cc2c1F c1(C(N2CCC(O)C2)=O)c(C)oc(C)c1S(N)(=O)=O.C(CC(=O)N)=CC=C.C C1(CC(=O)NCC(COC)C)CCN(C(=O)C(=O)N(C)C2CC2)C1 C=CCC(C(=O)Nc1cccc(C(N)=O)c1)NC(c1cncc(C)c1)=O C(C)(C)(C(=O)NCC1(NC(c2csnn2)=O)CCC1)SC C1CC(F)CN(C(=O)C)C1.C(=O)C(C)(C)C.C(C)(C=O)N(CCOC)C.N Cc1nc2cc(C(=O)NC3CN(C(C4CC4F)=O)CC3C3CC3)cnc2s1 Cc1sc(C(=O)NC23CC(C2)C3)cc1S(N)(=O)=O.C1(C=O)CC12CCC2.N C(=O)(CCCCC(C)(C)C)NC(CNC(c1n(C)nc(Br)c1)=O)C1CCC1 CC1(C)CCCC(CC(=O)NCC(C)(C2CC2)NC(=O)C=CC=C(Cl)Cl)C1 c1(CNC(=O)NC(c2ncccc2Cl)C)ccc2nsnc2c1 c1(C(N(CCC#C)Cc2ccc(C3CCCNC3)cc2)=O)ccc(Br)cc1 C(C1Cc2ccccc21)NC(C1(C)CCCN(C(CCSC)=O)C1)=O c1(NCC(CC)(C)NC(c2ccnc3[nH]ncc23)=O)c([N+](=O)[O-])cnn1C C1(CC)CCCCC1C(=O)NCC(N1CCN(C(=O)C(O)C2CCC2)CC1)C c1(OCC(N2C(C)(C)C(CNC(=O)CC(F)F)CC2)=O)ccccc1[N+](=O)[O-] c1(OC)ccc(C(=O)NC2CCCN(Cc3cc([N+](=O)[O-])c[nH]3)C2C)cc1C C(=O)(C1=CCCN(C(=O)CC2CCC(C)O2)C1)N1C(CSC)CCC1 c1(OC)ccc(C(N2CCC(N(C(=O)C(C)C(F)F)C)C2)=O)c(Cl)c1OC N1(C(c2ccc(C(F)F)cn2)C(=O)NCCOC)CCc2c(F)ccc(O)c2C1 c1(C(N2CCCCC2C2CC2)=O)cc(C(N2CCCC(N3CCC3)C2)=O)ccn1 C1(C(=O)NCCO)N(C(c2cccc(O)n2)=O)CC12CCCC2.C1CCCC1.C Cc1[nH]nc(C(=O)N)c1C.c1(C(C2C(C(N(CC(C)C)C)=O)C2)=O)ccccc1 CC(C)CC(CC(=O)NC1(c2cccs2)CC1)NC(c1ncccc1N)=O CC1(C)CC(C(=O)NC)=NO1.C1(O)CN(C(C2(c3ccccc3)CCOC2)=O)C1 C1(C(C)NC(=O)C=C2CCC2)CCCN1C(=O)Cc1csnn1 Cc1sc(C(=O)NCCOCCOCC)cc1.C1CCCO1.C(=O)C.N N1(C(CC(C)O)=O)C2CCC1CN(C(c1cc3c(s1)CCC3)=O)C2 c1(C(=O)NC23CCN(C(c4cccc(Cl)c4)=O)CC2C3)occ2c1CCOC2 C(=O)(C1CCCc2sccc21)N1C2(Cn3cc(CC(=O)O)nn3)CC(C1)C2.C.O N1(C(c2cnccn2)=O)CCC2CC(NC(c3csc(Cl)c3)=O)CCC2C1 Cc1ccc(C(=O)NC23CC(CNC(c4cccc(Cl)c4F)=O)(C2)C3)cc1Cl c1(CN2CCC(NC(c3c(C)nc4sccn43)=O)CC2)ccc2ncccc2c1 c1(C(=O)NC(CCC(=O)NCc2cn(CC)nn2)C)cccc2ccoc12 C(=O)(C(C)(C)C(C)NC(=O)CCCNC(C)=O)N(C(C)C(C)C)CC C(=O)(C(C(C)NC(c1oc(C)nc1C)=O)C(C)C)NC(c1ncccn1)CC CCCC(CC)CCC(=O)N1C2CCC(C2)C1C(N1CCC(CC)C1)=O C1(CC)(NC(c2cccc(CNC(c3conc3C)=O)c2)=O)CC(F)(F)C1 Cn1nc2c(c1C(N1CCN(C(c3cc(C(=O)NS)ccn3)=O)CC1)=O)CCC2 c1(C(=O)NCC2C3CN(C(C=CC=CCC)=O)CC32)cn2ccnc2s1 N1(C(c2c(CCC)nns2)=O)CC(CNC(c2csc(C#N)c2)=O)CC1C c1(C(=O)NCCNC(C(C)C2CCC2)=O)cncc(-c2ccccc2F)c1 C(=O)(N1CC(O)CCO1)C12CC(NC(c3ccncc3Cl)=O)(C1)C2 c1(NCCSCCC#C)ccn2nccc2n1 c1(C(=O)NCC(C)NC(=O)CC2CCC(C)(C)CC2)cccc2c1CCC2 C1(NC(c2n(C)nc(O)c2)=O)CC(NC(c2ccc(F)o2)=O)C12CCOCC2 C1(CCNC(CC=CC(C)(C)C)=O)CCN(C(=O)CC2(O)CC2)C1 C1(CNC(=O)CC2(CNC(c3ccc(CO)[nH]3)=O)CC2)CCCC12CC2 C1(C(=O)NCC(CCNC(C(C)O)=O)O)(C(F)F)CCN(C)CC1 C1(CNC(=O)NCC(C(C)C)O)CCCC1(F)F C1(C)(NC(C2(CNC(c3cc(CC)[nH]n3)=O)CCCC2)=O)CCC(C)C1 N1(CC(=O)N(C)CC)CC2C3CCC(C2C1)N(C(C1CC1C1CC1C)=O)C3 CONC(=O)C(C)(C)C1=CCN(C(c2[nH]ccc2CC2CC2)=O)C1 CCC(C)C(O)CC(=O)NCCC(C)(C)CNC(=O)Cc1cccc(O)c1 C(CC(C(C)C)NC(c1ccc(C2CCCC2)cc1)=O)NC(C1CN(CC)C1)=O N1(CC(c2cccc(C(F)(F)F)c2)F)CCC2COCCC12 N1(C(C(C)(C)c2sccc2Cl)=O)CC2CC2(NC(c2cccc(O)c2)=O)C1 N1(C(c2c(Cl)ccc(C)c2)=O)CC(CO)C2(C1)CN(C(=O)CCC1CC1)C2 c1(C(N(C)CC2CN(C(c3ccoc3)=O)CCO2)=O)ccc2c(c1)nnn2C Cc1ccc(C(CNC(c2cc(C)c(C)s2)=O)NC(c2cc(F)c[nH]2)=O)cc1 C1CC2CN(C(=O)C(C)(C)C(N)=O)CC12.C(C)(C=O)(C1CC1)NC(C)=O.N c1coc(C(=O)N(C)CCN(C(=O)C(c2cccnc2)C)C(C)C)cc1=O.CO N1(C(C2N(C(c3ccc(C#C)o3)=O)CCC2)=O)CC2CC(CO)C(C2)C1 CCC(C)(COC)C(=O)N(CC(=O)NC1CC2(CCC2)C1)C1CCC1 C(=O)(C1=Cc2ccccc2C1)N1CC(C(N2CCC(NC(=O)O)C2)=O)(CC)C1 Cn1nnc2c1CC(C(=O)NC1CC(CNC(=O)Cn3cnccc3=O)C1)CC2 N1(C(C(c2ccco2)NC(CCc2n(C)ncn2)=O)=O)CCOC(C2(C)N=N2)C1 Cc1cc(F)sc1C(=O)N(CCNC(c1ccc(F)o1)=O)C1CC1 Cc1cc(Cl)ncc1CC(N1CCC(C(C)(C)NC(c2scnc2Cl)=O)CC1)=O c1(C(=O)NC2C(C)CN(C(=O)Cn3cc(Cl)cn3)C2)ccnn2ccnc12 C1(C(N(CCCCCNC(C2COC2)=O)C)=O)CCCC(c2ccccc2)O1 CCS(=O)(=O)c1ccccc1CC(=O)NC1CCN(C(=O)CC(C)(C)C#N)C1C c1(C(N(CCC)CCNC(=O)CCCC2CC2)=O)cnc(N(C)C)c(Cl)c1 N1(C(C(C)CC2CCCCC2)=O)CCN(CCOCCO)CC1 N1(C(c2cnc(CC)nc2)=O)CC(N(C(=O)CCCF)C)C(C)(C)C1 c1(C(=O)NCC2CCCN2C(c2cccc(I)c2F)=O)c(F)cc(Cl)cc1F C1(C(N2CC(C)=C(C)CC2)=O)CN(C(C2CC2C2(C)COC2)=O)C2(CCC2)C1 c1cnc(NC(c2nnnn2CCS)C2CCCC2)c(C2CC2)c1.c1ccccc1 c1(SC)ccc(C(=O)N(CC(C)(C)NC(=O)CC(O)C2CCCC2)C)s1 C1(C(N(C(C)CCNC(C2CCCCCC2)=O)C)=O)CC2CCC(C1)O2 N1(C(C(CSC)C)=O)Cc2occ(C(N3CCC4(CCO4)C3)=O)c2C1 Cc1sc(O)nc1C(=O)NC1(C(=O)NOCCC(F)F)CCN(C)C1 c1(C2C(C=O)C2)cccc(Cl)c1.c1(COC)nc(C(=O)N)co1.CC(C)CO C1(NC(C(C2CN(C(C)=O)C2)OC)=O)CCCC12CN(C=O)C2.C(C)(C)C c1(C(=O)NCC(C)NC(COCCCOC)=O)cccc2c1OCC(=O)N2 c1(CC)cccc(C(=O)NCCN2CCN(C(=O)CCc3ccnn3C)CC2)n1 C1(CNC(CC(C)C)=O)=CC(=O)C(N=c2[nH]c3ccc(F)cc3o2)=C1 Cc1[nH]c2ccccc2c1CCC(=O)NCC(C)CNC(c1ccc(Cl)cn1)=O C1(NCCCn2cnc(C)c2C)CCC(=O)N(C)C1 c1(C(N2CC(Cc3ccc(F)cc3)C(C)C2)C(=O)NC(CC)C)c(Br)cnn1C Cn1nc(C(F)(F)F)cc1C1CCCC1.N1(C)CCC1C(F)(F)F N1(C(C(=Cc2ccccn2)C)=O)CC2CCC1CN2C(=O)C(C)(C)CC#N C1(NC(C2(CC)CCN(C(=O)CCC(C)C)C2)=O)CCN(C)CC1(C)C CCCCC(O)CC(=O)N1CCN(C(c2nnccc2C)=O)CC(C)C1 c1(C(=O)NCC(CC)NC(CNC(CC)=O)=O)oc(-c2cnn(C)c2)nc1C C1(NC(c2scc(OC)c2)=O)CC2CCC1CC2NC(C1(CO)CCCO1)=O N1(C(Cn2nnc(C)n2)=O)CC(C)N(C(c2conc2C)=O)CC1C N1(C(C2CCC(C)(C)O2)=O)CCC2C(C1)NC(=O)CCN2C(c1cnns1)=O C1(C(N2CCCCCC2)=O)CCCN(c2nnnn2Cc2cccc(Br)c2)C1 C(CCC(C)CCOC(=O)C(F)(Cl)Cl)=C(C)C C(=O)(CC(O)CCCC)N(C1C2CN(C(COCC=C)=O)CC21)C C1(NC(c2c(CC)oc(C)c2)=O)CC(C(=O)N(CC(O)CO)C)C12CCC2 O=C1CC(C(=O)NC2CCN(C(=O)Cc3c[nH]ccc3=O)CC2CO)CC(=O)N1 CC1CSCC1NC(=O)C(c1cccnc1)NC(=O)CCCc1cnn[nH]1 c1(C(=O)NC2CCCCN(C(C(C(C)C)(C)C)=O)C2)cc(O)ccc1[N+](=O)[O-] N12CCCC(F)(C1)C2=O.c1(NC(c2c(OCC)n[nH]c2)=O)ccc(OC)cn1 C1(NC(C2CC(N(C)C)C2)=O)CCCN(C(C2CN3CCC2CC3)=O)CC1 C1(CC(=O)NCC(C)NC(c2ccnc(S)c2)=O)CCn2cncc2C1 CC(CC1CC1)CC(=O)NC(CC1CC1)CC(=O)Nc1cccnc1 c1(C(=O)NCC(C)(C)CNC(=O)Cc2cnns2)cnc2c(c1)CCOC2 c1(C(N2C3CC(CN(C(CCC(C)SC)=O)C3)C2)=O)ccc2nc(C)cn2c1 c1(C(N(C(CCNC(c2cc(OCC)ncc2)=O)C)C)=O)ccc(O)c(O)c1 N1(C(=O)NC2CCC=CCCC2)Cc2nc(C3CC3)nc(O)c2C1 c1(C(N2CCC(c3cn(C(C)C)nc3)C2(C)C)=O)ccc2c(c1)ncn2C c1(C(N2C(CNC(CC3(C=C)CCC3)=O)CC2)=O)ccc(C(F)F)cc1 C=CCCCCCC(=O)NC1CC(F)CN(C(c2cnc(OC(C)C)cn2)=O)C1 C(=O)(CS(=O)CC)NCC(CNC(C=CC=CC)=O)OC N1(CC(=O)NCCCN(C(=O)CC2COCCO2)C(C)C)CC(C)(C)C1 N1(C(c2cc3cn[nH]c3cn2)=O)CC(C2CCCN(C(C3CCC4CC34)=O)C2)C1 N1(C(c2nc(CC)oc2)=O)CCCC2CN(C(c3nn(C)cc3Cl)=O)CCC12 C1(CNC(Cc2cc(OC)no2)=O)CCCCN(C(C2(C)C=CCC2)=O)C1 C12CCC(CC1)OC2.CC(CN(C)C)CC(=O)NCC1CC1CC(=O)N.C c1(OCC)ccc(COC(c2cncc(OC)c2C)=O)cc1Br CCC(C)(COC)C(=O)N1CCC(O)(CN(C(=O)CCCc2ccc(C)s2)C)C1 N1(C)CCC2(CC1)CS(=O)(=NC(=O)C1(S(C)(=O)=O)CC(O)C1)C2.CC(C)C c1(NCCCC)ccccc1C(=O)NCC(C)CNC(c1cnc(O)s1)=O C(CCN=c1cc(C)[nH]cc1C(=O)OC)N(c1cccc([N+](=O)[O-])c1)CCC c1(C=O)cn[nH]c1.C(C)CCNC(=O)C.N1(CCC)CCCC1.C(=O)N.N n1(CC=C)cc(C(=O)NC2CCC(CNC(=O)CC3CCCC3O)C2)cn1 CN1CC(CCO)(CNC(=O)CCC2CC2)C1.C(C1CCC1)=CC(=O)N N1(C(COC2CN(C(C3C(C)(C)C3)=O)C2)=O)C2CCCC1COC2 N1(C(CNC(CC)=O)=O)CC2(CCCC2NC(c2ncc(F)cn2)=O)C1 n1(CC(C)NC(c2c[nH]c(C(c3ccccc3)=O)c2)=O)cc(C2(O)CSC2)nn1 C1(C(N2CCC(NC(Cn3nnc(C)n3)=O)CC2)=O)COC2(CO)CC1C2 CC1CN(C(c2cc(C3CCCN3C)[nH]n2)=O)CCN1C(=O)C(F)=CC1CC1 C(=O)(C(F)C(=O)NCC#CC(=O)NCCC(C)OC)OCC c1(CC)nnc(S(C)(=O)=O)s1.c1ccccc1.C(CCN(C(=O)CO)C)NC C1(OCC)CCC(C(=O)N(CC(C)NC(=O)Cc2cccc(Cl)n2)C)CC1 N1(C(c2ccc(OC)nn2)C(=O)NC(C)C)CC(CO)OC(C)C1 C1(NC(C(C(C)C)OCC)=O)CCN(C(=O)C(F)F)CCC1CO N1(C(C2C(C)C2C)=O)CCC(OC2CN(C(=O)CC3CC4(CC4)C3)C2)CC1 C1(NC(Cc2c(C)con2)=O)CCCCCC1NC(=O)CCc1cccc(O)n1 c1(-c2cn(C(CC)C(N3CCC(C#N)C3)=O)nn2)cc(Cl)cc(Cl)c1Cl N1(C(C(CCOC)NC(c2ccc(C)[nH]2)=O)=O)CC(F)CC(F)C1 C1(C(=O)OC)CCC(C(N2CCC(C(C)NC(c3cc(Cl)ns3)=O)C2)=O)CC1 Cc1nc(C(N2CC(C)(CCC(=O)NC(c3ccccn3)CO)C2)=O)co1 c1(C(=O)NC2CN(C(=O)CC3(CC(=O)O)CCCC3)CC2F)c(F)cccc1Cl Cc1cc(C(=O)C(=O)NC(C)CCCNC(=O)C(F)=C2CCC2)ccc1F Nc1cccn(CC(=O)NC2CC(NC(C3CCC4(CC4)C3)=O)C2)c1=O C#Cc1cc(C(N2CC(CNC(=O)CN(C)C(C)C)CCC2C)=O)cc(N)c1 CC(c1ccccc1C)=CC(=O)NCCOCCCNC(c1ncc(Cl)s1)=O CC1(C)CN(C(=O)CN2C(=O)CNC2=O)CCC1NC(c1c[nH]nc1[N+](=O)[O-])=O N1(C(CC2(C=C)CC2)=O)CCC(NC(c2nccc(CC(=O)OC)n2)=O)CC1C c1(CC)cnoc1C(=O)N(C(C)CNC(=O)C(C)(C)n1cnnn1)C c1(C(N(C2CCCCN(C(C(C(C)C)OCC)=O)C2)C)=O)[nH]nc2ncccc12 Cc1nn(CC(=O)NC2CC3CC2N(C(=O)C(C)C2CCC2)C3)c(C)c1[N+](=O)[O-] c1(C(N)=O)csc(C(=O)OCCC2CCC(=O)N2)c1 c1(C(N2CC(F)CC(NC(=O)C=Cc3cc[nH]c3)C2)=O)ccc2c(c1)OCCC2 c1(C(=O)NC2(c3ccc(C(C)(C)C)cc3)CCCCC2)ccc2c(c1)NCC2 C1(CC(N2CCC(OCC)C2)=O)CN(C(c2ccn(C3CC3)c2C)=O)CCC1C C1(NC(c2c(NC)cccc2)=O)CCN(C(=O)COC(F)F)CCC1(F)F C(CC(C)(O)CNC(=O)C(CCN(C)C)NC(=O)C(C)C(C)C)OC c1(C(=O)NCC2CCCC(CNC(C(CCC#C)O)=O)C2)ccn2cccc2c1 Cc1cc(O)c(Cl)cc1C(=O)NC(C)C(C)NC(=O)C.c1cccc(Cl)c1.O c1(C(=O)NCC(CN(C)C(C2CCc3nn[nH]c3C2)=O)O)nn(C)c2c1CCC2 C1(C)(C(N2CC(C)(C)C(NC(C3(C#N)CCC3)=O)C2)=O)CCCCC1(F)F C(=O)C(F)(F)C(O)C(C)C.C1(CSC)CCN(C(=O)CC2CCCCC2)CC1.N CCCCC(O)CC(=O)N(C)C(c1cn(C(C)CO)nn1)C c1(C(=O)N)cc(N)cc(F)c1.CC(C)(C(F)(F)F)NC(=O)CC1(C)CC1 C1(C(N2CC(N(C)C)C2)=O)CCC(C2CC2)N1C(=O)Cc1cncs1 N1(C(c2c(C)cco2)=O)CC2C(NC(C3CCN(S(C)(=O)=O)CC3)=O)C2C1 c1(OCC)cncc(NC(C2CCN2C(c2cccnc2OC)=O)=O)c1 C12(C(=O)NCC(C(=O)NC(CN(CC)CC)C)C)CC(C)(CCO1)C2 N1(C(C(C(C)C)NC(=O)OCC)=O)CC2CCC1C2.c1(C=O)cnn(C)c1 N12C3CCC(C1CC3)C2=O.Cc1cc(C(=O)NC2CCN(C(C)C)C2)[nH]c1C N1(C(c2c(CNC(c3c(CC)nco3)=O)ccs2)=O)CC2CC1CO2 N1(C(C(C=C=C)C)=O)CCCC(O)(CCNC(c2cccc(F)c2)=O)C1 C(C)(C)(CC(=O)N1CCC(CCCCCNC(C2COC(C)(C)C2)=O)CC1)SC O=C(C#Cc1ccccc1Cl)N1CCn2c(CO)nnc2C1 C(=O)(C(CCC(N)=O)N=[N+]=[N-])N1CCCC(CN(C)C(c2ncccc2F)=O)C1 CCC(C)C(=O)C(=O)NC1CC2CCC1(C(=O)NC1(CC)CCCCC1)C2 c1(OC)ccc(C#N)cc1CN1CCSCC1C(=O)Nc1cc(Br)cnc1F N1(C(c2cnn(C)c2Br)=O)CC2CC1CC2NC(=O)CN1CCCC1 C1(NC(CSCCOC)=O)CCC(F)(CNC(=O)Cn2cccc2)C1 Cc1cc(C)n(CC(N2CC(N(C(=O)Cc3cnsc3)C)C(C)(C)C2)=O)c(=O)n1 C1(N(C)C)(CC)CCN(C(=O)CC(C)CNC(C2SCC=C2C)=O)C1 N1(C(c2c(C)snn2)=O)CCC2(CCCCC2NC(=O)CN(C)C2CC2)C1 N#Cc1nc(=NC2CC(NC(=O)CCc3cc(F)ccc3F)C23CCC3)cc[nH]1 Oc1ncnc2ccc(NCCNCc3ccc(O)cc3Cl)cc12 c1(C(N2CCCC(CCOC)C2)=O)ccc(C)c(C)c1F C(CNC=O)(C(C)(C)C)NC(C1(C)CC1)C.S(C(F)F)N c1(C(C(=O)NCCC(C)NC(C2CCCC(CF)C2)=O)O)ccc(F)c(F)c1 C1(CC(=O)NCCCC)CCCC1NC(=O)C.C1(C)(OC(C)C)CCCC1 c1(OCC)cc(C(=O)NCc2c[nH]nc2C(=O)NCCN=[N+]=[N-])on1 Cc1ccc(F)c(CNC(=O)NCC2(N3CCOCC3)CCCOC2)c1 c1(CNC(C2CCC(NC(c3[nH]cc4c3CCC4)=O)C2)=O)cc(F)cc(F)c1 CC1CN(C(=O)Cc2ccc(F)nc2)CC1(C)C(N1CCCC1CCCO)=O CCCC(C(=O)NC1(CC(=O)NC(C)(C)CCF)CC1)OCC C1(Cl)(C(=O)OC)CC12CCN(C(c1scnc1Cl)C(=O)NC1CCC1)CC2 Cc1ncoc1C(N1CC(C(N)=O)(CNC(c2cc(Cl)cs2)=O)C1)=O c1(C(N2C(C(C)NC(c3n[nH]c(C)c3O)=O)CCC2)=O)snc2ccccc12 CCC(C)C(C(=O)N1CCCC(NC(c2cc(-c3ccco3)c[nH]2)=O)C1)N(C)C C1(C(=O)NCC(CCCC)NC(c2cc(C)sc2C)=O)C2CCC1(C)C2(C)C c1(C(=O)NC2CCC(CCNC(C34COCC3C4)=O)C2)cnn2c1CCCC2 c1(CNC(C2(C)CC2F)=O)ccc2c(c1)CCN(C(c1ccc(N)cc1O)=O)C2 C1(OC)CCC2CCN(C(C34CC(c5ccccc5)(C3)C4)=O)C1C2 C1(C(=O)OC(C)C(=O)NC(=O)Nc2ccccc2)CCCC2(CCOCC2)O1 CC1CN(CCNC2CN(C(N)=O)C2)CCC1NC(=O)Cc1ccsc1 c1(C(=O)NCC2CCN(C(C3OCC(=O)C3)=O)C2)noc2c(F)cccc12 Cc1cc(=NC(C)C2CCCCC2)[nH]c(=NCc2cn(-c3ccccc3)nn2)[nH]1 C12(NC(=O)CN3C(=O)CCCC3=O)COCCC1CN(C(=O)C1=CCC1)C2 C(CC[Si](C)(C)C)NC(c1nn(CC)cc1Br)c1n(C(CC)(C)C)nnn1 C(=O)C1=CC2CCCC12.c1(OC)ccc(C(=O)C(=O)NCC=CC)cc1.N C1CCS(=O)(=O)C1(C)C.c1(-n2cc(CN(C)C(=O)NC)nn2)ccccc1Br C1(NC(c2c(C)cno2)=O)CCCN(C(=O)Cc2ccc(C(N)=O)nc2)CC1F CCC(CC)(CCNC(=O)CCC(C)OC)NC(C1COCCC1(F)F)=O c1(CC(N2CC=CC(NC(C(N3CCOCC3)C)=O)C2)=O)cccc2cn[nH]c12 c1(CN2C(C(=O)NCC3CNCCO3)C=CC2)cc(F)c(Cl)c(F)c1 c1(CC=O)ccc2sccc2c1.N1(C(C(COC)NC(C)=O)=O)CCC(C)C1.N c1(CC(N2CC3C(C(=O)NCc4c(C)n(C)nc4)(C3)C2)=O)ccc(Cl)c(Cl)c1 c1(C(=O)NC2CN(C(CC(=O)OCC)=O)C3C2C3)cnc2c(C)cccc2c1O CC1CN(C(=O)CC2CC=CCN2C)CCCN1C(=O)CC1=CCCCC1 c1(C(N2CC(CCCNC(C(C)OC)=O)OCC2)=O)oc2ccccc2c1Cl Cc1ncnc(N(C(C)CNC(=O)CCCc2ccc(Cl)cc2)C)c1F C1(NC(C)=O)CCC(C(=O)NC2C3CC2N(C(=O)C(C)(F)F)C3)CC1 c1(-c2ccc(C(=O)NCC3CN(C(C4CC4(F)Cl)=O)C3)s2)ccccc1F N1(C(CCNC(=O)NC)=O)CCC(C2CC2)C1.C1(O)(C2C(=O)N2)CCCCC1 c1(C(=O)NCCCN(C(C=C(CC)CC)=O)CCO)ccc(C)c2c1CCCN2 CCCC(CC)C(=O)NCC(C1CCN(C(=O)CCOCCCOC)CC1)C c1(C(=O)NCCC(C)(C)NC(C#CC(C)C)=O)cc(Cl)cc(Cl)c1O c1(C(=O)NC2C(CNC(CC3N(C)CCCC3)=O)CCC2)cc(O)nc(O)c1 N1(C(C(C=C)OC)=O)CCC(O)(C(C)NC(=O)CNC(=O)C2CC2)C1 c1(C(c2n(CCOC)nnn2)NC2(CC3CONC3=O)CC2)ccc(F)cc1 N1(C(C=CC)=O)CC=C(C(=O)NCC2(OC)CCSC2)CC1 c1(C(N2CC(C)C(NC(=O)CO)C2)=O)coc(S(N)(=O)=O)c1.C1CCCC1 C1(CC(N2CC(C(C(=O)N(C3CC(C)C3)C)O)C2)=O)(CO)CCCC1 S(=O)(=O)(CC(=O)N1CCC(O)(CC)C1)NCC.C1(C(=O)N)CC1C1CC1C C1(CCC(=O)N(C2C(CCC)C2)C2CCC2)CCN(C(=O)Cc2cn[nH]c2)C1 c1(OC)cc(N)ccc1C(=O)NC.c1(C=O)c[nH]nc1C1CCOC1.C1CC1 C1(CC#C)(C(=O)NCCn2cccn2)CCN(C(=O)CCc2ncccc2C)C1 O=C1CCC(NC(C23CC2CCN3C(c2ccnn2CCF)=O)=O)CN1 C1(NC(C2C(=C)C2)=O)CC2CCC1N2C(=O)C=Cc1ccccc1C CCC(COC)C(=O)NCCn1cc(CNC(=O)C(c2ccccc2)F)nn1 CC(C)CC(CC(=O)NC(C)(C)CC(C)(C)C)NC(C1CCOCC1(C)C)=O CC1(C)CN(C(c2ccns2)=O)C(CNC(=O)C=Cc2ccccc2C#N)CO1 C1(NC(C(c2ccc(C)cc2)C)=O)CC2CCC1C(NC(c1cn(C)nn1)=O)C2 C1(CCOC)CN(C(=O)Cc2ncc(C)o2)CCN1C(=O)CCC(C)(F)F c1(C(N2CCC2)=O)ccc2c[nH]nc2c1.Cn1nc(C(C)(C)C)cc1C(=O)NC N1(C(c2cc(Cl)cc(Br)c2)=O)CCCC2C1CCN2C(c1ccc(F)nc1F)=O c1(C(=O)NCC2CC2(F)F)cccc(-c2cn(-c3ccc(CO)nc3)nn2)c1 C(=O)(C(C(=O)NCC(=O)NCC=O)OC)OC.C1(C=O)COCC(C)O1.N C(=O)(C(C)(O)CCN(C)C)NCC1CN(c2ccc(OC)cc2)C(=O)C1 N1(C(c2ncoc2C(F)(F)F)=O)CCN(C(C2CC2(Cl)Cl)=O)C(C2CC2)C1 N1(C(c2ccc(C(C)=O)c(Br)c2)=O)CC2CC(NC(=O)C#CC3CC3)CC1C2 CCCC(C(O)C(=O)N1CCC(CC(C)C)C1)NC(c1ccsc1Cl)=O N1(C(C(C(C)O)NC(COCC(C)C)=O)=O)CCCC(C)(C)CC1 C1(CC(N2CCC2)=O)CCC(=O)NC1.C(C=O)(C1CCCC1)OCC.CC.N C(CNC(=O)Cc1cnns1)(C(C)C(C)C)NC(c1c(C)noc1N)=O CC(F)(F)CC(=O)NCC1(F)CCN(C(=O)CC2CC2(Cl)Cl)C1 N1(C(CCN(C(=O)C=CC2CCOC2)C)=O)CC(C)(C)C1C1CC1 c1(CCC(=O)NC2C(NC(c3c(COC)cc[nH]3)=O)CCC2)ncccc1C N1(C(c2n(C)c(O)nc2)=O)CC(C2CCN(C(=O)CN3CC=CC3)CC2)C1 C(CCCCCN=c1[nH]c(Cl)ncc1[N+](=O)[O-])NC(CC1CC(C)(C)OC1)=O CC1CN(Cc2ccc(-c3ccc(F)cc3)cc2)CC2(CCOC2)O1 C1(NC(C(CCC)OCC)=O)CC2CC1N(C(c1ccc(C)c(N)c1)=O)C2 C(CCN(C)CCNC(C1(C(=O)N(C)OC)CC1)=O)(C(=O)NC)OC C1(NC(C=CC)=O)COC2(C)CC1C2.C(=O)C(O)(CC)c1cccc(Cl)c1.N c1(COC(c2n(CC)ccn2)=O)cc(-n2cccn2)ccc1C C1(C(N(C2CC(CSC)C2)C)=O)CC(NC(C2CCOC2)=O)C1(C)C c1(C(=O)NCCN(C(c2cc(OC(C)C)no2)=O)CC)cc(Cl)c[nH]1 C(=O)(C#CC1(C)COC1)NC(COC)C(=O)NC(CCO)C1CCCC1 c1(C(C)OC(c2ccc(CC)nc2)=O)ccc(OC)c(Br)c1 Cn1nc(CC2CCN(C(C3(CC(N)=O)CCNCC3)=O)CC2)c2c1CCC2 C(C(CC(=O)NC1CC(CC)C1)C(F)(F)F)N(C)C.C(=O)(CCc1csnn1)N c1(CC)nocc1C(=O)NCC1CCCC1.C1(C=O)CCOC1C1CC1.C c1(C(N2CCCC(O)(C(F)F)C2)C(=O)NCCC2CC2)cc(F)nc(F)c1F C1CN(C(c2cc(Cl)ncc2O)=O)CC(C)(C)O1.C1(C(=O)NC)(OC)CCCC1 c1(NC(=O)C2CC2)ccc(C(N2CCC2CNC(=O)CCCCF)=O)cc1 c1(C=O)cc(C)n(C)c1.n1(CC(=O)N(CC(=O)OCC)C)ccnn1.C c1(C(NC)=O)cc(C(N)=O)[nH]n1.c1(C(N2CCC2)=O)ncn(C(C)(C)C)n1 N1(C(CNC(Cc2nc(=N)[nH][nH]2)=O)C(F)F)CCN(C(=O)Cc2cccs2)CC1 CC1CCCCC1N(C)C(c1ccc(CNC(C2OC3CCC2C3)=O)s1)=O N1(C(c2ccc(CC)cn2)=O)CCCC(CC)C1C(N1CCC(OC)C(C)C1)=O C1CCN(C(c2cc(C3CC3)oc2C2CC2)=O)CC1(C)C.C=C1CC1C(=O)N N1(C(CN(C2CC2)CC)=O)CCC2(C1)CN(C(=O)Cc1nc(=N)[nH][nH]1)CCO2 N1(C(c2cc(C)cc(O)c2)=O)CCCN(C(C2CCCC2P(C)(C)=O)=O)C(C)C1 c12cccc(c1F)C(=O)NC1CC(C1)CC(=O)N2.c1(C(=O)OC)sccc1Br N1(C(c2c(C)n(C)cn2)=O)CC2CC1CN2C(c1snnc1C(C)C)=O c1(C(C)NC(CCC2(NC(COC)=O)CCCC2)=O)[nH]c(C)nc1C N1(C(C(CC)COC)=O)C2CCC(C2)C1C(=O)NC(C)(CO)CC(C)C c1(CNC(C2(C(C)NC(c3c(C)nn[nH]3)=O)CC2)=O)cccnc1Cl c1(C(N2C3CC(CNC(C4C(C)(C)CCC4)=O)(OC3)C2)=O)cnn2cnnc2c1 c1(C(N2CCC(O)(CCNC(C(CC)F)=O)C2)=O)cc2cc(Cl)ccc2n1C CC(C)(CCCNCC=CCOC1CCOCC1)C(=O)N1CC2CC2C1 c1(C(N2C3CC(NC(=O)CC4CCC4)CC2CC3)=O)cc2ccnc(Cl)c2[nH]1 C1(C(=O)NCC2(CCC)CCC2)CC2CC1CN(C(c1cncc(CC)c1)=O)C2 c1(C(=O)NC(CNC(Cc2c(OC)ccc(Cl)c2)=O)C)cc2c[nH]cnc-2n1 c1ncccc1C=O.C1(C(N(C(C)C2CC2)C)=O)CC1[N+](=O)[O-].CC(C)C.O C1(NC(CN(CCC)C)=O)CC2CCC(C1)N2C(=O)CC(c1cccc(F)c1)C C(CCP(=O)(c1ccccc1)c1ccccc1)NC(C(=C)C)=O C1(C(=O)NC(c2ccc(C)nc2)CC)Cc2ccc(C)cc2S1 c1(NCC)ccc(Cl)cc1C(=O)NCC1CN(C(C2CN(C)C2)=O)CCO1 n1(CC(N2CC3C(NC(C=C(COC)C)=O)(C3)C2)=O)cccc(C=O)c1=O c1(NC(C(C)C)CCNC(C2CCC2(C)C)=O)ncnc2[nH]c3ccccc3c12 Cc1nn(C)c(C)c1C(=O)NC1CCN(Cc2cc(OC(F)(F)F)ccc2Br)C1 N1(C(C)=O)CCOC2(CCN(C(=O)CC3CC3(C)C)C2)C1.C#CCOCCO c1(OCC)cc(C(=O)NC2(C)CN(C(C3CNC(=O)N3)=O)C2)ccn1 c1(OC)ccc(C)nc1C(=O)NCC(O)CN(C)C(c1cccc(F)c1)=O.O N1(C(c2cc(Br)n[nH]2)=O)CC2CC1CN2C(C1CCC=CCCC1)=O c1(C=O)cc(C(F)F)ccc1F.C(c1cn[nH]c1)=CC(=O)NC1CC(O)(C)C1 c1(OC)ccc(C(=O)NC2CN(C(c3ccc(Br)cc3N)=O)C2)c(C)n1 c1(CCNC2(c3n(CCCF)nnn3)CCC=CCC2)cc(Cl)ccc1Cl C1(C(N2CCC(NC(C3N(CC)C(=O)CC3)=O)C2C)=O)CCC(C)(C)CC1 c1(CC)[nH]nc(C(=O)NC(C)C(C)C(=O)NC(C)CCn2cncn2)c1C C1(C(=O)OC)CCC(C(=O)N)C1.n12cc(nn1)C(C)N1CC(C1)C2 C1(CC)CC(C)CN1C(=O)CN(C(c1sccc1F)=O)CC CC(C)C(C(=O)NCCNC(c1ccccc1)=O)NC(N)=O.c1ncccn1 C1(NC(=O)COCCc2ccccc2)CCCN(C(=O)CNc2nccs2)CC1 c1(CNCC23C(CN(C(c4c(CC)nccn4)=O)C2)C3)ccc(O)c(F)c1 CC(N=c1cc(C#N)nc(C2CCOCC2)[nH]1)c1csc(-c2cnn(C)c2)n1 N1(C(C(CC(C)C)O)=O)CCOC2CN(C(=O)C(C)(C)c3ccccn3)CC12 N(C(=NCCOC(C)(C)C)N1CCC(CC(=O)NC2(C)CCC2)C1)C(C)C Cn1ccnc1SCCC(=O)NCC1CCCN1C(C1(O)CCSC1)=O N1(C(CN(C)CC)=O)C(C)CC2CN(C(C34CC(F)(C3)C4)=O)CC12 N1(C(=O)Cc2cc(OC)cc(F)c2)CCC2CN(C(=O)Cc3c[nH]nc3O)C2C1 c1(OCC)oc(C)nc1C(N1CCC(CC)C1)=O.C(=O)(CCC1CCC1)N C1(CNC(C(C(C)C2CC2)O)=O)CCCN(C(c2cc(F)ccc2F)=O)CC1 C1(CNC(C2CCN(C(=O)C3(C#N)C(C)(C)C3)O2)=O)CC2CCCC(C1)C2 Cc1cc(C)c(C=O)c(S)n1.C1(C)(CC=O)CCS(=O)(=O)N1.C1CCCC1.N c1(C(=O)NCC23C(CN(C(CP(C)(C)=O)=O)C2)C3)cc(C(F)(F)F)ccc1N CCC(C(=O)N1CCCC1CC(N1CCC1(C)C(=O)OC)=O)NC(C)=O CCC(C)(CO)C(=O)N1CC(N(C)C(c2nn(C(F)F)cc2Cl)=O)C(C)(C)C1 C(C(CN=c1[nH]c(C(F)(F)F)nc(=NCC(C)(C)OC(F)F)[nH]1)C(C)C)OC c1(Cn2cc(C(C)NC)nn2)ccc(C(=O)NC(C)(COC)C2CC2)cc1 CC(C(=O)N(CCCNC(C1CCCC1O)=O)C1CC1)S(C)(=O)=O C1(C(N2CCCC(CNC(=O)CCCC3CCC3)CC2)=O)CCc2nnnn2C1 C1(C(=O)OCC)C=CCN1C(=O)C(CO)NC(N)=O N1(C(CC(=O)N(C)C)=O)CC2CC(NC(c3coc(C4CCCCC4)n3)=O)C1C2 N1(C(C(C)OCCCC)=O)CCN(C(=O)CC23CCCN2CCC3)CC2(CC2)C1 C1(CNC(c2cc(C#N)oc2)=O)CN(C(c2ccc(CCF)cc2)=O)CCCO1 C12(NC(Cc3ccc(C(=O)OC)cc3C)=O)CCCC1CN(C(=O)C(N)=O)C2 CP(C)(=O)CCC(=O)N1CCOCC(NC(c2nccc(Cl)c2O)=O)C1 N1(C(C2(COC)CC(=C)C2)=O)CC2CCC2(C)C1.C(=O)CCCCC1CC1.N N1(C(C(C(C)O)(F)F)=O)CC2CCOC2(CNC(=O)CC)C1.[SH](C)(=O)=O.N C(CN=C(NC1CC1)N1CCC(N(C)CCO)C1)c1nc2cccc(C)n2c1 N(C(=NCCCNC(=O)OC)N1CC(C(F)F)C2(CCC2)C1)C(C=C)C C1(NC(c2ncc(Cl)cc2Cl)=O)CN(C(C2CC3CCC2O3)=O)C2(CCC2)C1 Cc1cc(C)n(CC(C)NCC2NCCCS2)n1 C1CN(C(c2ccc(C)s2)=O)C2CC12.c1(C(=O)OCC)ncc(C(=O)N)s1 N1(C(C(Cc2cnn(C)c2O)C2CC2)=O)CCC2(CCOC2)CC1.c1(=O)c(=O)[nH]1 C=CCC(C)(O)C(=O)NCC(C)(C)OCC.N12CCCC1NC(=O)C2 C(CSC(F)F)(C(=O)NCC1CC(C)C1)NC(CC1CC(CC)C1)=O c1(C(N2CC(NC(C3(OC(C)C)CCOC3)=O)C(C)C2)=O)cc([N+](=O)[O-])cn1C C(CNC(=O)CC(C)C1CC1)(CC(F)(F)F)NC(c1cc(C)sn1)=O C(CN=c1[nH]ccc(=NC2CC3(C2)C(F)(F)C32CCC2)[nH]1)SC(C)C C1(NC(C2CC(OC)C2)=O)CCC(N(C)C(C2CCC(C)(C)O2)=O)CC1 c1(C(=O)NCC(N(C(C(CC)C(C)O)=O)C)C2CC2)cnn2c1NCC(C)C2 c1(NC(CC2(C)CCN(C(C3CN(C(C)=O)C3)=O)C2)=O)c(O)cccc1F N1(C(c2cc(C)c(F)nc2)=O)CCC2(CCCN2C(c2ccc(N)c(F)c2)=O)C1 c1(C(=O)NC2C(NC(c3ccoc3)=O)C2)c(Br)n[nH]c1Br C(c1c(F)cccc1F)=CC(=O)NC1C2CN(C(c3ccc(C)c(O)n3)=O)C1C2 N1(C(c2n(C)ncc2)=O)CC(CNC(=O)COC)CC1(C)C.C1CCCOC1 CCCC(CC(C)C)C(=O)NC1CCCC(CC(=O)NC2CC3CC3C2)C1 N1(C(c2[nH]cc(C)c(=O)c2)=O)CC(C)N(C(c2ccc(C#N)cn2)=O)CC1C C(=O)(C(C)(C)C(C)(C)O)N1CCC(NC(c2cc(C(C)(C)O)on2)=O)C1 Cc1coc(C)c1C(=O)NCC1CCN(C(c2nc(Cl)sc2Cl)=O)C1 c1(OC)cc(CN)ccc1NC(=O)C(N)CC1CCCO1 N1(C(C2C(C(C)C)CCO2)=O)CCN(C(C23CC(CO)(C2)C3)=O)C2(CCC2)C1 c1(OC)ccnc(Cl)c1CN1CC(C)(C(=O)NCCOC)C1 N1(C(c2n(C=C)ncc2)=O)CCCC(NC(=O)C(C)CC(=O)OCC)CC1 c1(OC(=O)C(F)(F)F)ccc2nc(NCc3c(OC)cccn3)sc2n1 C1(C(=O)NCc2cc(C)c(C)nc2)N(C(c2cnnc(C)c2)=O)CC12CCCC2 N1(C(C(C2CCN(C(C3(O)CCOC3)=O)CC2)C)=O)CCOC(C)CC1 CC1C(NC(=O)C(=O)NC2CC2)CCN1C(=O)CCCc1ccsc1 C(=O)(CCCCN(C)C(c1ccccc1F)=O)N1CC(CCOC)C1 N1(C(=O)CCC(F)(F)F)CCCC2(CCN(C(c3ccc(C4CCCO4)[nH]3)=O)C2)C1 c1(C(=O)NC2CCCN(C(C3CC4(CC4)C3)=O)C2)cc(O)ccc1Br C1(O)CCOC1.c1(C(C(=O)NC(C2(C(=O)NC)CC2)C)C)cnn(C)c1 Cc1nc(=N)[nH]cc1C(N1CCCC(NC(=O)C(C)(C)C2CCCCC2)C1C)=O N1(C2CCC(C)C2)CCN(C(C(=O)NCCC2(C)CC2)c2cncs2)CC1 C(C(C(=O)N(CCCCNC(=O)CCCN(C)C)C)NC(C)=O)OC O=C(O)CC1OCCc2sc(C(N3CCC4CC3C(=O)O4)=O)cc21 C1(NC(CC(CC)OC)=O)CN(C(c2c(F)cccc2Cl)=O)CCC1F c1(CCC(=O)N(CC(C)O)CC)ccc(O)nc1.C1(C(=O)N)CC2(CC2)C1 C#CC1(O)CCCN(C(c2ccc(-c3cn(-c4ccc(Br)cc4)nn3)cc2)=O)C1 C1(NC(c2ccon2)=O)CC(C2CCN(C(c3ccc(F)o3)=O)C2)C1 N1(CC(CC)C)CC=C(CNC(=O)CCN=[N+]=[N-])CC1 CC1(C#CC(=O)N2CCCCC2CCNC(=O)COC2CCOC2)CCCO1 c1(OC)cc(C(=O)N(C)CCN(C(=O)CC(C)O)C)c2ncccc2c1 N1(C(=O)CC2CCCO2)CCC(C(=O)N(C2CCCC2)CC2CC2)C1 CN1CC(CC(=O)NCCCOCCN(C)C(c2cc(Cl)c[nH]2)=O)C(O)C1 C1(C(=O)OC)CC2(CC(OC(c3cc(C(C)C)ccc3C)=O)C2)C1 CC(C)CCCNC(c1cccc(OC(F)F)c1)=O.C1(C)(CC(=O)N)CCCO1 CC(C)CCC(C)N=c1nc2sccc2c(NCC(Cl)(Cl)Cl)[nH]1 c1(CNC(C2CCCC(F)(F)C2O)=O)ccc2cccc(Cl)c2n1 c1(C(C)(C)C(=O)NCC(O)CNC(=O)Cc2cnco2)ccc2c(c1)OCCO2 C1(C)(C(=O)NC2CCC(=C)CC2)COCCN1C(c1ccccc1)=O.C(C)(=O)N C1(CCC(=O)NCC2(C(=O)NCC3CCC(C)O3)CC2)CCC(=O)N1 C(c1cc(C)c(C)cc1C)=CC(=O)N(CC)CC.c1(C=O)ccnn(C)c1=O C1(N(C(C(C(C)C)OCC(C)C)=O)C)CC2CCC(C1)N2C(=O)CN(C)C c1(-c2cn(CCC(=O)NCCC3CNCCO3)nn2)cccc([N+](=O)[O-])c1 CC(C)(C(=O)N1CCC(NC(C2CC(C)(O)C2)=O)C(CO)C1)C(F)(F)F CC1CCN(CC(=O)NC(c2ccccc2)C)CC1NC(C1CCC2(CCC2)O1)=O CC(C)CCC(C(=O)NCC1CC2(CCO1)CC2)NC(C12COCC1C2)=O CC1(NC(C2(c3cccnc3)CC2)=O)CC(NC(C2CCC(=O)C2)=O)C1 C1(N(S(CCOC)(=O)=O)C2(CO)CC2)CCC2(CCNC2)CC1 c1(CC)ccccc1-n1cc(CC2CCCN2C(c2cc(C)oc2C)=O)nn1 N1(C(CCOCC)=O)CC(NC(c2ccc(C(F)F)nc2O)=O)CCC1C C1(C(=O)NCc2c(C)cnn2C)CN(C(=O)C(C)c2cccs2)CC1(F)F CC1CCCCC1CNC(c1ccc(C(N)=O)cn1)=O.C(=O)CCC(C)(C)F.N N1(C(C2(CC#C)CCN(C(=O)CCOC)C2)=O)CCCCC(C(=O)OC)C1 C1(C(N(CCCNC(C2(SCC)CC2)=O)C)=O)CC2CCC(C1)C2O N1(c2nc(C)nc3c2c(C)cs3)CCc2cc(O)ccc2C1C C(CC1CCC1)(C(=O)N(c1cnn(C)c1)C)NC(C(C)NC(C)=O)=O C1(C=C)(C(=O)NC(C#C)C)CCN(C(c2cc(OC)ccn2)=O)C1 CCC(C)(O)C(=O)NC1CCCC1C(=O)NC1CCN(C)C1=O C=Cn1ncc(C(N2CC(O)CC2C(=O)NC2(C(N)=O)CCCC2)=O)c1N C1(CC(=O)NC2CCN(C(CCOC(C)=O)=O)C(C)C2)CSc2ccccc2O1 C12(CC=O)CNC(=O)C(C1)C2.c1(CC(=O)N)ccc(O)cc1.C1CCCC1.C c1(C(N2CCOCC(NC(CC3C(C)C3)=O)C2)=O)cccc2ncnc(O)c12 C1(CC(N2CCC(C(N(C)C)=O)C2)=O)CCN(C(c2n[nH]c(=N)[nH]2)=O)C1(C)C c1(CNC(=O)NC2CCCc3c(C(=O)O)n[nH]c3C2)c[nH]c2cc(Cl)c(Br)cc12 Cc1cc(C(=O)NC(C2CCCN2C(=O)CCc2ncc[nH]2)(C)C)ncc1CO C1(c2n(CCCC)nnn2)(NC2CC3CC3C2)CC2CCCC(C2)C1 C12(CNC(c3c(CC)occ3C)=O)CC(C1)C(C)O2.C(=O)C(C)CCC C(=O)(C(C)(C)CCCF)NCC1CC2CN(C(c3c(CCC)nco3)=O)CC21 C(N=C(NC1CC1)NC1CCN(c2ccn(C)n2)C1)C1CC(=C)C1 Cc1cc(NC(C2CC2NC(c2cccc3nccnc23)=O)=O)cc([N+](=O)[O-])c1 N1(C(c2cc(C)oc2)=O)CCC(C2CCCN2C(=O)C(C(C)C)OC(C)C)CC1 C1(C(=O)NC2CCC(N(C(CC(C)NC(N)=O)=O)C)CC2)CCn2nncc2C1 C1(N(C)C(C2CC(CF)C2)=O)CCCCC1NC(=O)C(C1CCCCCC1)O c1(C(=O)NCC(CNC(C(CCOC)C)=O)(C)O)cccc2oc(C)nc12 C1(C(=O)OC)(C(N2CC(n3cc(C4COCC4O)nn3)C2)=O)CCOC1 N1(C(CC2C(C)CCC2)=O)CC(C)CN(C(=O)COc2cccc(Cl)c2)CC1C C1C(O)C(O)CN1C(=O)CCn1cncn1.c1(C(=O)N)ccn(C(F)F)n1.C CC#CCC(C(=O)N1CCC(F)(F)C1)NC(c1cc(C)nc(O)n1)=O c1(NC(C2CCC(NCc3cscn3)C2)=O)ccc(-c2cn[nH]c2)cc1 C(=O)(CCCC(C)C)NCC1CN(C(C(COC)OC)=O)C(C)C1 C1(C(=O)NCC(O)CN(C)C(C2(O)CCCCC2)=O)(OC)CCCCCC1 Cc1cc(C)c(CCNC2(C(=O)NC3CCCCC3C3CC3)CC2)cc1C c1(NC(CN2CC(CC)C(c3ccc(C)cc3)C2)=O)ccc(Cl)c(Br)c1 C1(C(=O)NCCNC(C2=CC(C)C2)=O)Cc2nccn2C1 C1(CNC(CCc2cc(C)n(C)n2)=O)C(C2CC2)CCN1C(=O)CCC1CC1 C(=O)(C1=CC2(CCN(C(=O)Cc3cnns3)C2)C1)NC(C#CC(C)C)(C)C CCC(CC(=O)NCC(O)CO)NC(C1C2CCC(=O)C12)=O C1CCC2(CN(C(=O)C=Cc3nnn(C)n3)C2)O1.Cc1ccn(CC(=O)N)n1.C Clc1cc(OCc2cnc(-c3ccccc3)s2)cc2c1OCCO2 N1(C(c2n[nH]c(C)c2Cl)=O)CCC2CC1CN(C(C1CC1CC(C)(C)C)=O)C2 c1(C(N2CC3CC(NC(=O)COc4cccnc4)C3C2)=O)cnn2c1CCCN2 CCCCC(C)C(=O)NC1CCCC1CC(=O)NCC(C)CC1CCC1 Cc1ccc(C(=O)NCCCC(C)(C)NC(=O)CCCCC#N)c(=O)n1C CCCCCCCCCC(=O)NC1CCCCN(C(=O)CC2COC(=O)C2)C1 C1(C=O)CC2CCC(C1)S2(=O)=O.C(=O)(C(O)C(C)(C)C)N(C)CC.CC.O C=C(C)C1OCCC1C(=O)NCCC(C)(C)NC(=O)CC(c1c(C)noc1C)C C1(NC(C(CSCC)NC(=O)CC(Cl)Cl)=O)COC2(CCCC2)C1 C1(NC(c2cc(C)n(C)c2)=O)CC(O)C(C)(C)C1 c1(C(N2CCCC(CN(C(CSCC#C)=O)C)C2)=O)ccc(Cl)cc1OC C1(N(C(C(CC)OC2CCCC2)=O)C)CC2CCC(C1)N2C(C1CC(C)(F)C1)=O Cc1[nH]nc2c1CN(C(=O)NCc1nc(Br)sc1C)CC2 S(=O)(=O)(C(C)CNC(C1CN(c2ccccc2)C1)=O)NC.c1ccccc1.O N1(C(C(CC)COC)=O)CCCN(C(c2cc(C)n(C)c2)=O)C(CO)C1 C1(F)(C(=O)NCc2ccc(C)s2)CCCN(C(=O)C(C)NC=O)C1 Cc1nc2c(N3CCCC(C(C)NC(=O)CN4CCCC4)C3)ncnc2[nH]1 c1(C(N2CCSC(C)C2C)C(=O)NCCOC)cc(F)c(Cl)cc1Cl C1(C2CC2)CCSCC1.C(C(=O)NCCC1(C=O)CC1)OCCN(C)C.N c1(C(N(CC(=C)C)C)=O)ccc2c(n1)CN(C(C1CC(C)(C)CCO1)=O)CC2 c1(OCOC)cccc(C(N2CCC(C(C)C(N3CC(O)C(F)C3)=O)CC2)=O)c1 Cc1ccc(C(=O)NCC=CCNC(=O)C(C)(C)C2CCCCO2)c(C)n1 CC(C)CC(CN=c1[nH]c(N2CCCS(=O)(=O)CC2)nc2ccsc12)N1CCCC1 c1(C(=O)NCCN(C(c2cccc3c2CCO3)=O)CC)cc2cc(Cl)sc2[nH]1 Cc1cccc(Cl)c1C(=O)NC1CC(C(=O)Nc2ncc(Br)cn2)C1 N1(C(C(=O)N(C)C)=O)CCOC(CC2CC2)C1.N12CCCC(C1)C(C)(C)C2=O c1(C(=O)NCCC2CCC(NC(c3n[nH]cc3Cl)=O)C2)ccc2c[nH]nc2n1 c1(-c2onc(-c3ccc(C(C)C)nc3O)n2)ncnc2sccc12 CC1CN(C(=O)Cn2ncnn2)CCN(C(C2CC3CCCC(C2)C3)=O)C1 C(CC(F)CN=[N+]=[N-])NC(C1CC(O)(CNC(C(C)CN(C)C)=O)C1)=O c1(C(=O)NC(CNC(C2(C)CC(C#N)C2)=O)C2CC2)cc(Cl)cc(Cl)c1O Cc1nc(C(F)(F)F)ccc1-c1ccncc1.C1(C(C#N)N(C)CC)CCCOC1 c1(C(N2CCCC(OC(C)=O)C2)C(=O)NC)cnc(C2CCOCC2)nc1 C=C(C)CN=C(NCCc1c(C)cccc1Cl)NC(c1cccc(Cl)c1)C C=C(C)CN=C(NC1CCC1)N1CCC(C(F)(F)F)(CC(=O)NC)C1 CCCCS(=O)(=O)CC(=O)NC1CC2(C1)CC2NC(=O)Cc1cc(C)cs1 C1(C)(C(=O)NCC(C)NC(c2cc(C3CCCC3)no2)=O)CCC(=O)NC1 CC1(C)CN(C(c2cn(CCNC(=O)COc3cccnc3)cn2)=O)C1 c1(C(=O)NCC(CC=C)NC(C2(CC#C)CCCOC2)=O)ccc2ncnn2c1 Cc1ccc(C(=O)NCC(N2CCN(C(c3cnsn3)=O)CC2)C(F)F)nn1 c1(NC2(CO)CCN(Cc3ccc(F)c(F)c3)CC2)ncc2ccc(Br)cc2n1 C1(N(C(C#CCNC(C2CN(C)C(=O)C2)=O)=O)C2CC2)CC2CCC(C1)O2 c1(CC(=O)NC2(CC=C)CN(C(=O)CCc3ccncn3)C2)c(Cl)cnn1C C(C)(C)(CN=c1cc(Cl)nc(C(C)C)[nH]1)N1CCN(C(C(C=C)(C)CC)=O)CC1 CC(CCC(F)(F)F)(c1ccccc1)NCCCP(C)(C)=O Cc1nc2ccc(C(N3CC(NC(=O)Cc4ccc(O)nc4)C(O)C3)=O)cn2n1 c1(C(N(CC(C)C)C)=O)ccc2c(n1)CCOC2.c1(C(=O)N)nncn1C1CC1 C(C(=O)NC1(C)CCCC1)(C(C)C)OCC.C1(CC=O)CCCC(=O)C1.N N1(C(c2cn(CCNC(c3csc(O)n3)=O)nc2)=O)CC2CCCC1C2 c1(OC)cc(CNC2CCN(C(c3[nH]c(C)nc3C)=O)C2)c(F)c(F)c1F N1(C(CC2CCN(C(=O)CC3CCCO3)CC2)=O)CC2C(C1)C2(F)F C(C(=O)NCC(C)C1CC1)(C1CCCC1)NC(C)=O.C(=O)CCc1nccs1 c1(N2CC(C)(C)OCC2)ccc(S(=O)(=O)N2CCS(=O)C(C)(C)CC2)cc1F C(CC(C)C)(C(=O)NC)NC(c1c(CC)onc1C)=O.C1(O)CCC(C)C1 C1(OCC)CCCCN(C(=O)C(COC)OC)C1.c12sccc1C(=O)NC2 c1(C(=O)NC(C2CN(C(C3CC(C#N)C3)=O)CCO2)C)cccc(Cl)c1F c1(C(=O)NC2C3CN(C(C4(CC5CC5)CC4)=O)CC23)cc(O)ncc1Br C1(O)(CNC(C2(C)C=CCCC2)=O)CCCN(C(c2ccc(C#N)[nH]2)=O)C1 C1(CNC(c2ccn(CC)n2)=O)CCC(F)(F)CC1.c1(C(=O)N)ccon1 N1(C(c2n(CC)cnc2Cl)C)C(COC)CC2CCCCC12 c1(CC(N2CC(C=O)C(F)C2)=O)c[nH]c2cnccc12.Cc1cnncc1CC(=O)N C(C(COC)CC(=O)NCC12CC(CO1)C2)OC.c1(CC=O)cc[nH]c1.C C1CC2(C1)CN(C(=O)CC13CC(C1)C3)C2.O=C(C=O)NCC(F)(F)F.N C(=O)(C(F)(C)C(C)C)N1C(COC)C=CC1.C1(C=O)CC(=C2CCC2)C1 N1(C(C2(NC(=O)O)CCCC2)=O)CCC2(CCOC2)C(CO)C1.c1ccco1.C C(=O)(C1CCCc2nn(C)cc21)NCC(C)NC(=O)C1CCCc2cccnc21 c1(C(C(=O)NCC=C)N(C(C)CC)C)ccc(OCCC2CC2)cc1C.S N1(C(C2(C)C(C)C2)=O)CC2CC2(Cn2cc(-c3cccc(Cl)c3)nn2)C1 c1(C(=O)NC2CC(NC(C=C(C)c3cccs3)=O)C2)cc(F)cc2ccoc12 C(C(C)(C)C(=O)NC1CC1)OC.N12CCN(CC1)CC1CCC(C1)C2=O CC(CO)C(=O)NC(C)(C)CC=CC(N1CCC(C(N)=O)C1)=O C(=O)(CCCCC(N)=O)N1CCC(NC(C(C)N(C(=O)OC)CC)=O)CC1 C12(C(N3CCC(CCNC(C(C)(C)c4sccc4Cl)=O)C3)=O)CCCC(CO1)C2 C(=O)(C(C)(C)C(C)C)NC1C(NC(C(c2cccc(OC)c2)C)=O)COC1 C(=O)(C1=CCCC1(C)C)NCCN(C(c1c(C)cnn1C)=O)CC.CCO.O c1(C(N2CCC(NC(c3c(C)n(C)nn3)=O)C(C)C2)=O)cc(Cl)cc(Cl)c1N N1(CC)CC2CCCC(Nc3cc(C(C)C)ncn3)C2C1.C1(C2CCC2)C(=O)N1 c1(OC)cc(C(N2CCN(C(=O)C=CBr)C(C(C)C)C2)=O)cc(C#N)c1 N1(C(CC(OCC)OCC)=O)CCOCC(NC(=O)CC(C)COCC)C1 C1(N(C(Cc2cc(C)nn2C)=O)C)CC2CCC(C1)N2C(C1CC(N(C)C)C1)=O c1(C(C)C)ccc(O)c(C(=O)NC23CC(C2)C3)c1.C1(C=O)CCOC(C)C1.N C1(NC(C2(CC=C)CCC2)=O)CC2CC2C1.N1(CC=O)CC(=O)NC1=O.N C(=O)(CCCF)NCC(C(=O)N(C1CC(CO)(CO)C1)C)C1CCCO1 c1(C(N2C(C)(CC(=O)NC3(C)CC(=C)C3)CC2)=O)cnc2cc[nH]c2c1 c1(CNC(C(CC=C)NC(COC2(C#C)COC2)=O)=O)cnc2n1CCC2 Cc1cnn(C)c1CNC(C1CCCCC1)=O.C(=O)(C(O)CN1CCOCC1)N CCCC(C)(O)C(=O)N(CCNC(c1cc(N2CCOCC2)nc(Cl)c1)=O)CC C1(C(N2CCCC(CNC(C(C(C)C)F)=O)C2)=O)CCCCC12OCCO2 N1(C(=O)CSc2cccc(Cl)c2)CC2OCCN(C(=O)CCCC(F)F)C2C1 C1(O)(C(N(C(CNC(c2c(C)ccc(C)c2)=O)C)C)=O)CCCC(C)(C)C1 C1(CC=O)CCC(C)(O)CC1.C12CC1CN(C(=O)C(F)C1CCC1)C2.CCO Cc1ccc2nc(C(N3CCN(C(=O)C(O)C(C)C)CC(O)C3)=O)cn2c1 N1(C(C(C(C)O)(F)F)=O)CCC(C2CN(C(=O)CCC3CC3)C2)CC1 N1(C(c2c(C)nn(C)c2)=O)CC(C(N2CC(N(C)C)CC2(C)C)=O)C2(CC2)C1 C(C(CC(C)C)C(=O)N(C1CCC(=O)N(C)C1)C)NC(C(OC)OC)=O c1(C2CCN(C(C(=O)NC34CC(COC)(OC3)C4)=O)C2)c(F)cccc1F N1(C(CC(=O)OC)=O)CC(NC(c2cnc(CC(C)C)s2)=O)CC12CCC2 C1(C(=O)NCC2ON=C(CC)C2)CCN(C(=O)C2CN(C(=O)OC)C2)O1 c1(C(=O)NC(CN(C(c2cncc(C)c2)=O)CC)C)cc(O)c(F)cc1N Cc1nc(CNC(=O)C(C2CCCN(C(=O)Cc3ccco3)C2)C)c(C)s1 CC1CCCN(CC(C)NC(c2cc(C3CC3)nn2C)=O)C1 c1(C(c2c(OC)cccc2)OC(=O)NC2CCCCC2C)ccc(F)c(Cl)c1.O CCCC(CCC)C(=O)NC(C1CN(C(C2CCOC(C)(C)C2)=O)CCO1)C C1(C)(CNC(c2c(C)cco2)=O)CN(C(=O)C(F)CC(C)C)C(C)(C)C1 C(=O)(CC(CC)OCC)N(CC(=O)NC1CC(C=C)C1)C(C)C c1(C(N2C(CC(C)O)CCC2)C)ccc(Br)cc1 c1(OCCOCC)cc2c(cc1CN1CCCC(N(C)C)C1)OCO2 C1(NC(C(CC(=C)C)NC(=O)CCCCOC)=O)CC2CC1OC(=O)N2 O=C1CC(C2CCN(c3nccc(N4CCC(CN5CCCC5)CC4)n3)C2)CN1 c1(CC)ccc(Cl)cc1C(=O)N(CC(C)(C)CNC(c1ccncc1C)=O)C N1(C(C2CC(C)(NC(c3ccoc3Cl)=O)C2)=O)CC2CC(O)CC2C1 c1(C(=O)O)cc2cc[nH]c2cc1C(=O)Nc1ccsc1C(N1CCC(O)C1)=O c1(CC=O)c(C)cccc1C.C(C(C)(C)C(=O)N(CCCO)C)OCC.CC N1(C(CCN(CC)CC)=O)CCC(F)(C(=O)NC(CO)CCCO)CC1 C1(CC(=O)NC2(CCC(=O)NC3CC34CCC4)CCCC2)NC(=O)NC1=O CCC(CC(=O)N1CCC(N(C(=O)CCCOC(C)(C)C)CC)C1)C(F)F C1(C(=O)NC(CNC(c2cc(C)ns2)=O)(C)C2CCC2)CCc2nnn(C)c2C1 Cc1ccn(C)n1.N1(C(C)=O)CC2C(N(C(=O)CC34CCC(CC3)C4)C)C2C1.N c1(C(=O)NC2COC3(CNC(C4CSCCS4)=O)CC2C3)cccc2cncn12 C(=O)(C1=C(C)N(C)c2nnnn2C1)NCC(CC)NC(c1cccc(F)c1Cl)=O C(CC(C)(C)C)(C(=O)NC(CCSC)C(=O)NC(C)CCC(C)(C)C)OC CC1=CCC(C(=O)NCC2CCN2C(c2ccc(C(=O)OC)s2)=O)CC1 CC1CCc2sc(C(=O)NC3CC3C)cc2C1.c1(C(=O)N)occc1C1CC1 Cn1cnc(C(=O)NCCC2(NC(c3cc(C(N)=O)[nH]n3)=O)CC2)c1 c1(C(=O)NC2C(CNC(COCCCCCC)=O)C2)cc(Br)cn2ncnc12 C(CCC(C(=O)N1CCC(CC(F)F)C1)NC(=O)C=Cc1cc[nH]n1)OC C1CCC(C)N(C(=O)C)C1.c1cc(C#N)oc1C.C(C(=O)N)=CCN(C)CC CC1(C)C(O)CCN1C(=O)CN(C1CCC1)C(c1ccccc1)=O c1(C(=O)NCCC2OCCN(C(c3cnc(OC)s3)=O)C2)cn2ccsc2n1 C(=O)C(C)(C)C(C)(F)F.Cc1ncc(C=CC(N2CCC(O)(C(C)C)C2)=O)s1 c1(CN(C(c2cc(CC)[nH]n2)=O)C)ccc(Br)c(F)c1 CN=C(NCCCCc1cccc(F)c1)NC1Cc2ccccc21 N1(C(CC2C(C)(C)C2)=O)CCC(C)(CC(=O)NCCc2ccns2)C1 c1(CCC)nc(C)c(C(NC(=S)Nc2ccccc2F)=O)o1 N1(C(c2ccc(CCC)cc2)=O)CCC2(COCCN2C(=O)C(S)C(C)C)C1 c1(CC)cc(C)cc(O)c1.C1(C(=O)N)CC1(C)C.N1(CCC=O)CCOC1=O C(=O)(CCCCCCCCC1CC1)NCC(C)CNC(=O)CC1CSC1 Cc1[nH]nc(Cl)c1NC(C1CN(Cc2ccccc2C(=O)O)CCO1)=O c1(OC)ccc(CC(=O)NC(C)CCNC(=O)C(C)(C)c2nncn2C)cc1F CCCC(C)(C)C(=O)NCCN(C(c1cnoc1CC)=O)C1CC1 N1(C(c2nnc(C)s2)=O)CCC(CF)(NC(=O)CCC(C)N(C)C)C1 Cn1nc(C(=O)NC2CCC(CNC(=O)CCP(C)(C)=O)CC2)c(Cl)c1Cl C1(OC)CC(NC(c2ccc(C)nc2C)=O)CN(C(=O)C(C)c2cc[nH]n2)C1 C1(NC(c2n(C)ncc2Cl)=O)C2CC3CN(C(c4ccc(Cl)c(O)c4)=O)C1C3C2 c1(C=O)nn(C(C)(C)C)cc1Cl.c1(C(C)=O)cc(C(=O)N)co1.CC(C)(O)C C1(C(=O)N)C2CCC3(COC(=O)C13)O2.CC(C)CCCN(C(=O)C1=CCSC1)C N1(C(c2n(CC)ccc2)=O)CCN(C(=O)Cc2cc(C)sc2C)C2CCCCC12 CC(C)C(C)CCNC(=O)CN(C)C(C)C.c1(CCC=O)ccc(F)cc1.N C(CC(C)C)(C(=O)NCCCCC(C)NC(=O)C(C)C)OC.c1(C=O)ccco1 C1(N(C(c2c(OC)cccc2)=O)C)CCCN(C(C2(C(N)=O)CC2)=O)CC1 C1(C(=O)NCC(CN(C(c2c(CC)nccn2)=O)CC)O)CCCC12OCCO2 C1(NC(C2CC(C)C2)=O)CC2CN(C(=O)C(C)(C)c3cnsc3)CC2C1 CC(C)C(C)C(=O)N1C(C(=O)N(C)CCN2CCCC2)CC2CC12 N1(C(C(=O)Nc2ccc(F)c(Br)c2)=O)CC2CC(C1)CS(=O)(=O)C2 N1(C(C(C)OC(C)(C)C)=O)CCCC(F)(C(N2CCCCC2C)=O)C1 c1(N2CCC(CC(=O)NCC(C)(O)CCCO)C2=O)cccc([N+](=O)[O-])c1 N1(C(c2cccc(OC)c2)=O)CC2CN(Cc3c(Br)cnn3C)C2C1 C=CCC(C)(C)C(=O)NCC1CCCCC1.c1(C(=O)N)ccc(CC(N)=O)cc1 N1(C(CCC)C)CC(C(=O)NCC2(F)CCC2)CC1=O.C(=O)C=C1CCC1 c1(C(=O)NCCNC(c2cc(C)c(O)nn2)=O)c[nH]c2cc(F)ccc12 Cn1nc2c(c1C(=O)NC1CC3CN(C(=O)C4=NOC(C)(C)C4)CC3C1)CCCC2 c1(C(=O)NCCC2CCC(NC(CC(=C=C)C)=O)C2)cc2ccncc2c(O)n1 N#Cc1c(Cl)nsc1NCCC1CC(NC(=O)CC2CCC(=O)NC2=O)C1 Cc1c(Cl)ccc(C(N2CCC(O)C(NC(=O)C(C)C(C)(F)F)C2)=O)c1Cl Cc1cc(C(N2CC3(CCC3CNC(C3CC3F)=O)C2)=O)c(N)c(Cl)n1 CC(C)(CO)C(c1ccccc1)NC(=O)CS(N)(=O)=O Cn1c(Cl)cnc1C(F)(F)C(=O)NCCC1(O)CN(C(c2ccccc2)=O)C1 C=CCCCC(=O)NC1(C)CC(C(=O)NC(CO)CCC)C1 N1(C(c2ccn(CC)c(=O)c2)=O)CC(C)CN(C(c2c(C)cnn2C)=O)C(C)C1 N1(C(C2OC(C(=O)OC)C(C)C2)=O)CCCC(CNC(c2ccccn2)=O)CC1 C(CC1=CCN(C(c2ccc(Cl)cc2O)=O)CC1)NC(C(C)C(F)F)=O C(=O)(C(C)(C(C)C)NCc1cn(CC(CC)O)nn1)NCCSC Cc1ccc(Cl)cc1.c1(CC(=O)N(C(CN(C(C(C)O)=O)C)C)C)cc(C)no1 C1(NC(C(C)CN(C)C)=O)CC1C1CCCN(C(c2ccc(C#N)s2)=O)C1 C1(CC)CCN(C(=O)CC=CC(C)(C)C)C1C(=O)NCc1cnccc1C CC(CO)(C(=O)NCCC1CC(F)(F)C1)NC(c1c[nH]ccc1=O)=O C1COC2(C1)CN(C(=O)Cn1cnc([N+](=O)[O-])c1)C2.C1(C=O)(CC)CCC1.N C1(C#N)(C(N2CCC(NC(CC=C=C)=O)(CC)CC2)=O)CC12CCOCC2 C12(C(=O)NC(C3(C)CC3(F)F)C)CCC(CC1)CO2.C1CCCCC1C=O.N C=C(C)CC(C)C(=O)N1CCSCC1CCNC(=O)CN(C)C1CC1 C(=O)(C(C)(C)C(O)CC)NC(CC=C)CNC(=O)Cc1cnc(O)nc1O c1(C(=O)NC(CCCC)CNC(=O)CSCC(C)C)coc2ccccc12 C12(NC(=O)C(O)Cc3ccccc3)CCCC1N(c1nc(Cl)ncc1CO)CC2 n1(CC(=O)NCC(C)NC(=O)CC2CC3CCC(C2)N3C)cc2ncccc2n1 c1(NC(C2N(C)CCCC2)=O)nc2c(s1)CC(NC(=O)C#CC(=O)O)CC2 N1(CC(C)C)CC(C(=O)N(C2CN(C(=O)CC3CC3)CC2O)C)CC1=O C1(CCCC)CCCN1C(=O)C(Cc1ccoc1)NC(=O)CN1CCCC1=O c1(CC(=O)NCCN2CCN(C(C(CC)(C)F)=O)CC2)ccc(C)c(C)c1 c1(C(N2CCC(NC(c3csc(Cl)n3)=O)C2)=O)cc(F)c(Br)cc1F c1(CCC(N2CCC(n3cc(CC(CC)(C)O)nn3)C2)=O)cccnc1Cl CCC(C(=O)OC)C(=O)N1CCC(NC(=O)C(=Cc2ccncc2)C)C(F)C1 C(CCC(F)(F)F)N(C)C.C1(C(=O)NC(C)C(=O)N)CS(=O)(=O)C1.C=O C1(C(=O)NCC(CC)NC(c2ccc(SC)cc2)=O)CCc2n[nH]cc2C1 c1(C=O)cnn2c(=O)cc[nH]c12.Cc1ccnc(C(=O)NC2CC(C)(C)C2)n1.N c1(OCC)ccc(CCNC(=O)NOc2ccc(Cl)cc2)cc1 C(=O)(C(CO)C(F)(F)F)N1CC(C)CC1.c1(CC(=O)N)cccc(C(F)(F)F)c1 C12(CNC(C(CSC)OC)=O)CCCC(CN1C(=O)C)C2.c1ccccc1Cl Cc1cc(C(N2CCOC(C)C2)=O)c(C)n1-c1cnn(C)c1.C1(C(=O)N)CC1C C1CC2CC1CC21CC1.Cc1oc(CNC(C2(C#N)CCOC2)=O)nc1C=O.N C1(NC(COC(CC)(C)C)=O)CCCC1.C(=O)CCC=CCc1ccccc1.N C(=O)(C(O)CC(F)(F)F)NCC=C1CCN(C(C2CC(C)OC2=O)=O)CC1 c1(SCCC)ccc(C(=O)NCC(C)N(C)C(C2(O)CCOCC2)=O)cc1 C1(CCOC)CN(C(=O)Cc2cc(OC)no2)CCN1C(=O)C(C)C1CCCC1 c1(C(C)C)ncsc1C(=O)NCCOC1CCN(C(c2cc(F)cs2)=O)C1 N1(C(c2cc(C(C)(F)F)n[nH]2)=O)CCC2CN(C(C3CC3F)=O)C2C1 C(CC(C(=O)NC(C1CCCN1C(=O)C=C(C)c1ccsc1)C)OC)OC c1(CC)c(NC(c2cnc(C(C)(C)C)o2)=O)cccc1C c1(C(=O)NC2(CC=C)CCN(C(c3cccc(Cl)c3)=O)C2)ccc2c(n1)CCC2 c1(C(=O)N(c2ccncn2)CC2CNC2)cn(C2CCC2)nn1 C(=O)(C1CCCn2ncnc21)N1CCC(C)(CNC(=O)Cc2nccs2)C1 Cc1c(C(F)(F)F)n[nH]c1C(=O)NC.C1CCCC1.C(=O)C(F)(F)C1CC1 c1(C(=O)NCC(C)N(C(=O)CCC2CC(C)(C)CO2)C)ccccc1N(C)C C(CCCC(c1nnnn1CCCC1CC1)NCC(C)(C)CC(F)F)(OC)OC C1(n2c(=O)cc(C)nc2C)CCN(N2CCCC2CC(C)(C)C)CC1 c1(CC(C(=O)N)NC(c2cc(SC)no2)=O)ccc(Cl)cc1Cl.C1CSC(C)C1 C1(C=O)CCN(C(=O)CC2CCN(C)CC2)C12CCC2.CC(C)C(O)C1(C)CC1 Cc1cc(C(=O)NC(CNC(C2CCC(F)(F)CC2)=O)CO)cn(C)c1=O N1(CC)CC(C(=O)N(C)CCNC(=O)CC2CCCC(OC)C2)c2ccccc21 C1(O)(CN)CCCS(=O)(=O)C1.CN(C)CCOCCO CCCCCC(=O)NCC(=O)NC(C)C(C)NC(c1cc(C(C)=O)c[nH]1)=O C1(CCNC(c2csc(C(F)F)c2)=O)CCN(C(C2C=CCCC2)=O)C1 c1(C(C)(C)C)nc(=NC2CN(C(=O)CCC3CC3(F)F)CCC2(F)F)s[nH]1 c1(C(N2CCC(CNC3CC(CO)C3)C2)=O)ccc(-c2csnn2)cc1 CC(C)(CCC(=O)NCCN1C(=O)CNC1=O)NC(=O)CC#N C1(C(=O)NCCc2c(C)nn(C)c2)CCCCC1C.C1(C=O)CC(N(C)C)C1.N c1(C(N(C(CNC(C(c2ccc(N)cn2)C)=O)C)C)=O)ncn2cccnc12 Cc1ccc(=N)[nH]c1C(=O)NCCN(C(=O)C=CC(C)(C)C)C C(=O)(C(C)(C)CN(C(=O)COC)C)N1C(CCC)CCC1 Cc1nc2ccc(C(=O)NCCNC(=O)CNC(=O)C3CC3)cc2[nH]1 c1(SC)nc(Cl)cc(=NCC(C)NC(C2Cc3nnc(C)n3C2)=O)[nH]1 C1(CCN(C)C(C2CC3CCC3C2)=O)CCN(C(=O)CC2CCC23CCC3)CC1 C1(C(=O)NC2CN(C(c3snc(C)c3N)=O)C2)CCC(=O)N2CCCC12 c1(C(N2C(C)(CCC=O)CCC2)=O)ccc(C)cc1C.C1(C(=O)OC)CCC1.N N1(CC(c2cn(C)nc2)=O)CCCC(NC(=O)CC2(C)CCOC2)C1 C(C)(CN=c1[nH]c(=N)[nH]c(=NCCCN2CCCCCC2)[nH]1)(C1CC1)OC N1(C(C(C(C)C)O)=O)C2CCCC1CC(NC(C1CCCCCN1C)=O)C2 N1(C(C2CCN(C)CC2)=O)CC2CC(NC(c3ccc(Cl)c(F)c3)=O)C2C1 C(=O)(C1=NOC(C)(C)C1)NCC(C(C)C)(C)NC(=O)C(O)CC1CCCC1 C1(C#N)(COC)CN(C(C2(NC(c3ccc(Cl)o3)=O)CC(F)C2)=O)C1 c1(CC(=O)NC2C(CNC(c3c(C)cnn3C)=O)C2)cc(O)ccc1Br c1(-n2cc(CCCC(=O)O)nn2)ccc(C(F)(F)F)cc1.C=C1CC(C(=O)N)C1 c1(OC)cc(CNCC2CCCN2C(=O)CCc2cccc(Br)c2)cc(F)c1 CC(CC(N)=O)C(=O)NCC1(NC(c2cc(C(F)(F)F)n[nH]2)=O)CCCC1 c1(CC(C(=O)N)O)ccc2ccccc2c1.C1(CNC(CC2C(C)C2)=O)CCC1 S(=O)(=O)(c1ccc(N2CCSC3(CCC3)CC2)c(F)c1)NCCNC(C)=O CN1CC(O)CCC1C(=O)NOCC(=O)NCC12CCCC1OCC2 C1(NC(C(C)O)=O)CCN(C(N)=O)CC1.N1(CCn2ccnn2)CCN(C)CC1.C S(=O)(=O)(c1ccc(C#N)cc1)NCCCOc1c(C)cccc1C.C(C(C)F)N N1(C(C(=O)NCCCSC)c2cnn[nH]2)CCSC2CCCC12 C(C)(C)(CC(F)(F)F)NC(C(C1CCN(C(c2cc(CC)[nH]n2)=O)CC1)C)=O C1(NC(C2CC=CC2)=O)CCCCC12CCN(C(=O)C=Cc1cncc(F)c1)C2 CC1c2c[nH]nc2CCC1C(=O)NCCC(C)(C)NC(=O)CCn1cnnn1 C1(CC(=O)NCCCCCN(C)C)CCCN(C(c2ccc(O)nn2)=O)CC1 N1(C(=O)C=CCNC(C2(O)CCCCC2)=O)CCC(=C(F)F)CC1 CN1CCC(NC(=O)NCC2CCN(CC(F)F)C2)C1=O Cc1ccn2ncc(C(=O)NCCOCCN(C)C(C3CCC(C)O3)=O)c2c1 c1(OC)ccc(C(=O)NC)cc1C.c1(C=O)cn(C(C)(C)C)cn1.C1CCC1 S(=O)(=O)(CC(=O)NCC1CC(C)N(C(c2cccnc2S)=O)C1)NCC CC1CC2(CCN(C(=O)Cn3cnc(=N)[nH]3)CC2)CN1C(=O)CCc1ncc[nH]1 C12(CNC(C(OC)OC)=O)CCCC1CCN2C(=O)CN1C(=O)CCCC1=O CCCC(C(=O)NC1CN(C(=O)CN2CCCOC2=O)CC1OC)C(C)C C1(C(=O)Nc2cc(C)c(F)cc2)CC12CCN(C(C1CCCOC1)=O)CC2 C1(C(=O)NC)CCN(C(=O)C(C2(O)CN(C(c3nonc3N)=O)C2)F)C1 c1(C(=O)OC)cccc2oc(=NCC(C3CC3)NC(c3ccc(F)cn3)=O)[nH]c12 C(=O)(C1=NOC2(CCC2)C1)NC(C)C=CC(N1CC2C(C1)C2(F)F)=O C1(C(=O)NCCC(C(=O)N)OC)CCCCC(=O)C1.C1(N(CCC)C)CCCC1 CC(C)(CC(=O)NCCC1CC(C(=O)NC2CC(=O)N(O)C2)C1)C1CC1 C12(C(N3C(C=C)CC3)=O)CCC(NC(=O)CC(C)(C)CC)(CC1)C2 CC1=CCC(C)(C(=O)NC)CC1.C1CCCC1.c1(C=O)c[nH]c(C(F)(F)F)c1 Cc1ccc(C)c(C(=O)NC2C=CC(C(=O)NC34CC(C3)C4)C2)n1 N1(CC)C2CCC1CN(C(=O)C(CCOC)NC(=O)CC(C)SC)C2 C12(CNC(c3cc(C)on3)=O)CC1CN(C(=O)Cc1csc(C3CC3)n1)C2 N1(C(c2c(C)n(C)cc2)=O)CC(NC(=O)C(F)C2CCCC2)C2CCCC12 C#CC1CC2(CC2)CN1C(=O)C(C1CCCC1)NC(c1c[nH]c(=S)cn1)=O C1(CC)C(NC(=O)Cn2cccnc2=O)CCCN1C(c1cccc[n+]1[O-])=O N1(C(C(C(CC)C)C)=O)CCN(C(c2ncnc3ccsc23)=O)CCC1C C1(CCNC(C=C(C)C2CC2)=O)CCCN(C(=O)C(C)C2CCCO2)C1 c1(C(N2CCC(NC(C=CC=CC)=O)C(C)C2)=O)ccc2c(c1)C(=O)CCS2 N1(C(C2(F)CCC(C)CC2)=O)CC2CC(C1)CN(C(C1CCC(F)(F)CO1)=O)C2 N1(C(C2=C(C)OCC2)=O)CC2CN(C(C3(C)CCCC3)=O)CCC12 C(=O)(CC(C(C)C)NC(=O)COCCC(C)C)NCC(CC)OC c1(CC(C)C)cc(C(N2CCCC(NC(=O)CC3(C)CCCO3)C2)=O)n(C)n1 C1(NC(c2ccn(CCC)n2)=O)CN(C(=O)C=CCF)CCC1C c1(C(=O)NCC(C)NC(c2ccc(CC)cn2)=O)sc2nnc(S)n2c1C c1(C(=O)NC(C)CCNC(=O)C#CC2CCC2)cn2c(Br)cccc2n1 c1(NC(=O)CC2CN(C(c3ccno3)=O)CCO2)ncnc2c1ncn2CCO C(C)(C)(CCCC(=O)NC1(C)CC1)NC(CN1CCC(CC)C1)=O.C1CCC1 n1(CC(=O)NCC2(F)CC(NC(c3scc(C)c3)=O)C2)ccccc1=O Cc1cccn2c(C(N3CCC(C)C3CNC(c3ccnc(F)c3)=O)=O)cnc12 CC1CC(CNC(=O)NCCOC(=N)O)CC(C)(C)C1 C(=O)(CC(C)C)NC.C=C1CC(C(=O)NOCC2CC2)(C(=O)NC)C1 c1(C(C)=O)cc(C(=O)N)ccc1C.C1CC(C)N(C(=O)Cc2nnc(O)s2)C1.C N1(C(CNS(CC)(=O)=O)=O)CC(NC(=O)C(CO)N(C)C)CC12CCCCC2 c1(C(=O)N)sccc1Cl.C1(C)(C(N(C(C)C2CC2)C)=O)CC1C(F)(F)F c1(C(N2CC(O)(CNC(CSCCOC)=O)C2)=O)ccc2cn(C)nc2c1 c1(OC)ccc2c(c1)CCCC2NC(C1CC(F)(F)CO1)C C1(C(=O)NC(COCC)C(=O)NC2(CCO)CCC2)CCC(C)(C)OC1 N1(C(c2cscc2Cl)=O)CCC2C(C1)CN2C(C1(c2cc[nH]n2)CC1)=O C(CCc1cccs1)NC(COCCC=C)=O.C1(C(=O)N)CN(C(C)=O)C1 C1(NC(c2c(NC(CC)=O)cccc2)=O)CC(F)(F)CC1.C(=O)(C1CC1)N C1(C(=O)NC(CC)CNC(c2coc(O)n2)=O)CCCCC1(C)C N1(C(C(COCC)C)=O)CCC(N(C(=O)CC=C(Cl)Cl)C)CC1 C1(NC(Cn2nnc(C)n2)=O)CN(C(C2CC(=O)C2(C)C)=O)CC2(CCC2)C1 c1(C(=O)NCCCC2N(C(C=C3CCN(C)C3)=O)CCC2)nccc2[nH]ccc12 N1(C(C(=O)NCC)=O)CC(CNC(=O)Cc2ncoc2C)OC2COCC12 N1(C(C=Cc2cnc(C)s2)=O)CCC2CCCN(C(c3cc(F)cs3)=O)C2C1 c1(C(N(CC(CC)NC(C2CCN(C)C2)=O)C)=O)cscc1C C1(C(=O)OCC)CN(C(=O)NCC2CC(F)CN2C)c2ncnn2C1 S(=O)(=O)(c1ccc(CC(=O)N(CC(O)C)C)cc1)NC.C(=O)(CCCC(C)=O)N CC(CC(=O)Nc1cn(CCC2CC2)nn1)S(=O)(=O)c1ccc(F)cc1 CC1(C(=O)Nc2ncc(Cl)nc2Br)CCCN(C(C23CC(C2)C3)=O)C1 C(=O)(C1COCc2ccccc21)N(C1CCCN(C(c2cnc(C)[nH]2)=O)C1)CC c1(NC(CNC(c2nc[nH]c2)=O)C)ccccc1.c1(COC)ccc(Cl)cc1.C C(=O)(CC(C)CC(=O)N)OC.C1CN(C(=O)C=C(C)c2cccs2)C(C)(C)C1 C(=O)(CC1C(=O)Nc2ccc(Cl)cc21)NCCC(C)NC(C12CC3CC1C2C3)=O c1(NC(c2n(C)nnn2)(C)Cc2ocnc2C(F)F)ccc2c(O)nc(O)nc2c1 c1(NCC(C2CC2)NC(C2(C)CC2(F)F)=O)ncc2c(n1)CCOC2 C1(C(=O)NC(C(C)NC(c2c(C)snn2)=O)C)CC(=O)N(c2ccccc2)C1 C1(CCC)(NC(c2cnc(O)c(C)c2)=O)CCCN(C(=O)C(F)C(C)(F)F)C1 C1(NC(COCc2onc(C)n2)=O)CCCC12CN(C(c1ncccc1O)=O)C2 C12(C(N3CCC(C(CC)C)CC3)=O)COC(C1)C(NC(C1CC(C)(C)C1)=O)C2 C(=O)(C1=C2CCCN=C2NN1)NC1C(N(C(C(CC=CC)CC)=O)C)CCCC1 Cc1cc(C)nc(Cc2cccc(NC(=O)NC3CN(C4CC4)C3)c2)n1 C1(CNC(C(C)OC)=O)CC12CCN(C(=O)CNS(=O)(=O)N(C)C)CC2 C(=O)C(C)(C)CC(C)(C)C.C(=O)(C(C)C(C)(C)C)N(C)Cc1ccccn1.N N1(C(CC2C(C)OCC2)=O)CCC2(C(=O)NC3(C)CC=CC3)CCCC12 CCC(O)C(C)(C)C(=O)NCC12CC(NC(C3CCCOCC3)=O)(C1)C2 c1(C(=O)NCC(CNC(CC2N(C)C(=O)CC2)=O)(C)O)cc2c([nH]1)CCOC2 c1(C(=O)NCC2C(NC(CN(C(C)=O)C)=O)C2)sc(C)cc1.C1CC1 C1(NC(CC)=O)COC2(C1)CN(C(c1ncc(C)cc1OC)=O)C2 C(=O)(C#CC1CCCO1)NCC(C)(C1CCC1)NC(c1cc(Cl)c(F)cc1O)=O CCCC(O)C(=O)NCCOCCNC(=O)CSC(F)F c1(SCC)ccc(C(=O)NC23CC(CNC(=O)C(C)O)(C2)C3)cn1 C1(NC(COC2CCN(C(CC(C=C)CC)=O)C2)=O)CC(C)(C)C12CCC2 c1(OC)ncc(C(N2CCC(C)C2C)=O)cc1C.n1(CCC(=O)N)cc(Cl)cn1 C1(CNC(c2n(CC)cc(Cl)c2)=O)C(O)C(O)CN1C(c1ccnnc1C)=O Cc1ncc(C(N2CCN(C(=O)C(O)CC(C)C)C(CO)C2)=O)c(=N)[nH]1 CC(C)C(CNC(c1ccc(NC(N)=O)s1)=O)NC(C1CC2CC1C2)=O N1(CC)CC(C(=O)NC2(CO)CCCN(C(C3(O)CCCCC3)=O)C2)CCC1=O C1(C(=O)Nc2cncc(C)c2)CCN(C(C2CC(=O)NC2(C)C)=O)C12CCC2 c1(CC(=O)NCC2C=CCCN2C(c2cn[nH]c2)=O)ccc(Cl)cc1Cl CCC(CCOC)C(=O)NCC1CC(NC(C2CC3C=CC2CC3)=O)C(O)C1 c1(C(C(=O)N(CCCCCNC(COC)=O)C)(C)F)ccc(F)cc1 c1(C(N2CCC(C)C(CNC(=O)C(C)(C)CO)C2)=O)cc2nc(O)[nH]c2cc1N c1(NC(c2ccsc2)C)ncnc2c1ncn2C1CC1CCCCC(=O)O Cc1cccc(C(=O)NC2CN(C(C3CN(C)C3)=O)CC2C#N)c1Br c1ccc(N(C)C)c([N+](=O)[O-])c1.C=C1CC1C=O.C(=O)C.CC=CC.N N1(C(c2ccc(=N)[nH]n2)=O)CC(CNC(C2CCC3(CCC3)O2)=O)C2(CC2)C1 O=[N+]([O-])c1cccc(Oc2cc(Cl)ccc2CNCC2C3(CC3)C23CC3)c1 CC(CCc1ccc(F)cc1)C(=O)N1CCC(NC(=O)C=Cc2cc[nH]c2)C1C C1(NC(=O)C2CC2)CC2CC1N(C(=O)CCc1nc(-c3ccncc3)no1)C2 CC(C)C(O)C(C)C(=O)NCCOCCCN(C)C(N)=O.C(=O)(CCC)N c1(C(=O)NCC2C(CNC(CC3(C)CCC3)=O)C2)sc(Br)cc1F CC1Cn2nccc2CN1C(C12CC1CCCCC2)=O c1(OC(C2CCCC(C)(C)C2)=O)c(Cl)cc(Cl)cc1Br N1(C(C(CC)(C)OC)=O)CCC(O)(CCNC(=O)C(O)C2CCCC2)CC1 C1(O)(CNC(CSCCC)=O)CCCN(C(=O)CCOC2CCOC2)C1 C12CCN(C(c3cc(C)ccn3)=O)CC1C2.c1(COCC)nc(C)c(C=O)s1 C1(C(=O)NC(C(=O)NCc2cccnc2Cl)c2ccco2)C2CCC(F)C12 CC1(C)CN(C(=O)Cc2nc(C3CC3)cs2)CCO1.CC(F)(F)F.C(=O)C.N C1(CN(C(C(CSC)O)=O)C)CCCCN1C(c1ccnc(N2CCCC2)c1)=O N1(C(C(CSCC)NC(=O)CCc2ccccc2)=O)CCC(C)(NC)C1.C=O Cc1nc(C(C(=O)NCCCC2CC2)N2CCC2c2cccc(Cl)c2)oc1C c1(COC(=O)COCCC2CCN2Cc2cscc2Br)ccc(F)cc1 c1(C(C)C)ncoc1C(=O)NC1CCCC1C.C(=O)(C(C)Cn1ccnc1)N C(=O)(CCC=C(C)C)NC1CCN(C(c2ccc(C3CCCCC3)o2)=O)C1.CC c1(C(N(C2CCC2)C)=O)cc(CNC(=O)COCC2CCOC2)[nH]n1 c1(C(N(C)CCNC(C2CCCCNC2=O)=O)=O)cc2cc(Cl)ccc2o1 CN1CC(C(=O)NCC2COCCN2C(=O)CC2(O)CC2)c2ccccc2C1=O N1(C(C=CC(CC)C)=O)CCN(C)C(C(=O)NCCCOC)C1 N1(C(c2c(C)cco2)=O)CCCC2(C1)CN(C(c1cc(F)cc(F)c1N)=O)C2 Cc1cccnc1CNC(=O)CNC(c1c[nH]cc1C1CC1)=O Cc1[nH]c(=N)nc(O)c1CCC(=O)NC1CC(C)N(C(=O)Cc2cccs2)C1 C1(CNC(C(C)NC(CC)=O)=O)CN(C(C2(CCOC)CC2)=O)CCO1 N1(C(C(C)SC)=O)CCCC2(C1)C(NC(=O)Cc1csc(C)n1)CCN2C N1(C(C2C(c3ccccc3)(C)C2)=O)CC2(C1)CN(C(C1CCC3(C1)N=N3)=O)C2 CC(C)CC(C(=O)N1CC(OCC(=O)N(CC(O)C(C)(C)C)C)C1)N(C)C C(=O)(C(C)CC1CC1)N(CCCC)C(C)CC.C12(C(=O)N)CCN(CC1)C2 c1(C(=O)NCC(CNC(c2c(C)cc(C)o2)=O)CO)ccc(F)c(CO)c1 c1(C(N2CCC(CC(=O)NCc3cnc(C(C)C)s3)C2)=O)c[nH]c2cnccc12 c1(C=O)ccc(-c2nc(=O)o[nH]2)cc1.C(C)(C)(CC)NC(C1C(C=C)C1)=O.N C1(NC(C(C)(C)OC(C)C)=O)CN(C(=O)CC2CC3(CC3)CO2)CC1O c1(OC)cccc(F)c1CN1CCN(CC(=O)Nc2ccnc(Br)c2F)C(=O)C1 C1(C)(Cc2cn(Cc3cc(C)nn3C)nn2)CCN(C(=O)C=CS(C)=O)CC1 c1(OCC)ccc(Cl)c(NC(=O)CSc2ccccc2N)c1 c1(C(=O)OC)cnc(C(=O)NC(C)C2CC2)cn1.c1(C(=O)N)cnccn1 c1(C(C(=O)NCC(C)CNC(C2CCCN2N=O)=O)C)ccc2c(c1)OCCO2 C(=O)(C(C)(C)CCC#N)NCc1cc(C(N2CC(C(=O)NC)OCC2)=O)n[nH]1 N1(C(Cn2cc(C3CC(N(C)C)C3)nn2)=O)CCC(C)(C#N)C1 C1(C(NNC(=O)NCCCNS(=O)(=O)C2CC2)=O)C(F)(F)C12CCOCC2 C1(NC(=O)CC(c2ccccc2)C2CC2)(CNCc2ccccc2)CCCCC1 C(=O)C(F)(F)C(C)O.CC(C)C.C1(CC=O)CCC1.C(C)(C)C.C=O.N N1(C(CCSC)=O)CCC(NC(=O)CC2(C#N)CCOCC2)C(C(C)C)C1 CC1CN(C(C2(C)CC(C#N)C2)=O)CCCN1C(C1CC2(CC2)CO1)=O N1(C(c2n(CC)cnn2)=O)CCCCC1CCNC(=O)C(N1CCCCCC1)C Cc1ncc2c(n1)CCN(Cc1cccc(OCC(F)F)n1)C2 Cc1nc(N2CCN(C(c3c[nH]nc3C3CCCO3)=O)CCC2C)c(C)c(O)n1 c1(N2CCC(O)(C(C)NC(=O)Cc3ccc(Cl)nc3)CC2)cccc(F)c1C#N N1(C(c2n(C(C)C)ccc2)=O)CCCC2(C1)CN(C(=O)COCC(F)F)CCO2 N1(C(C(C)n2cncn2)=O)CC(CNC(c2ccoc2)=O)C(C)(C)C1 N1(C(c2c(C)nc[nH]2)=O)CC2CCC1C(NC(c1cc(Cl)cc(Cl)c1)=O)C2 c1(C=O)cc(C)c2[nH]nnc2c1.C1(C)(CC)CC(C(=O)NCC2CC2)C1.C C=CCC(C(=O)NCc1ccoc1C(N1CC(O)CC(O)C1)=O)C(C)C c1(C(=O)NC2C(C)CN(C(C3CCOC3)=O)C2)cc2n(n1)CC(C)(C)CO2 C(=O)(C(CC(C)C)C(C)C)N1CC(CC)C(NC(=O)C(O)Cc2ccccn2)C1 c1(CC(CO)CCC=O)cccc([N+](=O)[O-])c1.CC1(C)CC1S CCC(CC)C(F)C(=O)N1CCC2(CC1)CC2CNC(c1ccc(OC)o1)=O CN1CCN(C(C2(CNC(C3CC4(CSC4)C3)=O)CC=CC2)=O)C2CC12 C1(CC(=O)N(CC(F)F)CC)CCN(C(c2[nH]ccc2C)=O)C1 N1(C(C2C(CC)C2)=O)CC2CC1C2NC(=O)C(c1cccc(F)c1)C CC1CN(C(C(=O)NCC2CCC2)C2CCOC2)CC1Cc1ccc(F)cc1 C1(CC)C(C(=O)NC(c2ccc(F)cn2)C)CCCN1C(=O)C(C)n1cccc1 C1(NC(C2(F)CCN(C(Cc3nc(C)sc3)=O)C2)=O)COC2(CCCC2)C1 C1(C)(C(=O)N)CCC(=O)NC1.Cc1cccc(CCNC(C2CC2(C)C)=O)c1 c1(C(N2CC3(C(NC(C=C(C)C)=O)CC3)C2)=O)cnc2[nH]cnc2c1 Cc1ccc(C(=O)NCC2CC2NC(=O)CS(N)(=O)=O)c(F)c1C C1(C(=O)NCC2N(C(CCn3ncc(C)c3)=O)CCCC2)CCc2nncn2C1 Cc1ccc(O)cc1C(N1CC(O)CC1C(=O)NCCc1cccnc1F)=O C1(C(N2CCCC2C2(O)CN(C(C)=O)C2)=O)(CC)CCCN1C(=O)CO CC1(C)Cc2cc(C(N3CC(CCNC(C4CC5CCC4C5)=O)C3)=O)ccc2O1 C12(C(N(CCN(C(=O)CN(c3cnccn3)C)C)C)=O)CCOC(C)(C1)C2 C(=O)(C(C)C(O)CC(C)C)N(C(CC)C(=O)NC1CCC2(CC1)CC2)C c1(C(N2CCC(OCC(N3CC(=C)C3)=O)C2)=O)cc(C#N)ccc1C C(Cn1cccn1)(C(=O)NCCc1nncn1C)NC(C(C)OCC#C)=O n1(CC)ccc(C(=O)NCC2CC(NC(C3CCOC3C)=O)C2)cc1=O C(=O)(CCC(C(C)C)NC(=O)CC)NCc1cn(CC)nn1.C(C)(C)C.O Cc1ccnn1CC(=O)NCC1CCC1NC(=O)CCc1nc(=N)[nH][nH]1 C1(CN(C(Cc2nnc(C)o2)=O)C)CCCCN1C(c1ccnnc1O)=O Cc1nnc2n1CC(C(=O)NCC=CC)CC2.c1(C=O)cnn(C2CC2)c1Cl.N C=C(C)CCCC(=O)N1CCC(N(CCOC)C(C2CC(C)OC2C)=O)CC1 C1(C=O)CCn2c(C)cnc2C1.C1CC(O)C1.C1(C(=O)N)(COC)CC1.C C1(C)(CC)CCCN(C(=O)C(CC(C)C)N(C)C(C2CCC(CC)O2)=O)C1 N1(C(C2CC(OC)C2)=O)CCC(C)(C)C1C.C1(CC=O)COC(C)(C)CO1 C(C(=O)N1CC(O)CC1C)(C(C)C)NC(c1c(C(C)C)cc[nH]1)=O.C(N)=O c1(C=O)ccc(NS(N)(=O)=O)nn1.C1(CC)CCN(C(=O)CC2C=CCC2)C1 CC1C(NC(C2CC2(F)F)=O)CCCN1C(=O)C(c1nc(F)ccc1Cl)C c1(CC)c[nH]nc1C(=O)NCCC=CCCCC1CN(C(=O)C)C1.C(C)CC CCCCCCC(CC)NC(C1CC2CCC(C1)N2C(C1(F)CCC1)=O)=O N1(C(CCC2C(C)(C)C2)=O)CCCC(NC(=O)CCCc2nccs2)C1 Cc1nc2ccc(C(=O)N(C3CCN(C(c4cccnc4O)=O)CC3)C)cc2[nH]1 Cc1cc(=NCc2ncc(Cl)n2C)[nH]c(=NCC2CCC(C3CC3)C2)[nH]1 N1(C(C(C)OCC=C)=O)CCN(C(c2c(O)noc2C)=O)CC1CC1CC1 c1(OC)nc(Cl)cc(=NC(=O)CCc2ncc(-c3ccc(CSC)cc3)cn2)[nH]1 C#Cc1ccc(C(=O)NCC(CC=C)NC(=O)C(C)(CC)OC)c(F)c1 C(=O)(C(C)(C)CF)NCC1(C)CC(NC(Cc2cc(C)sc2)=O)C1 c1(C(N(CC(C)O)CCNC(CCC(=C)Cl)=O)=O)ccc(F)c2ncccc12 C1(COCC)CCN(C(c2sccc2C)C(=O)NCCC#N)CC1 c1(OC)ccc2c(N3CCN(C)C(CO)C3)nc(=NCc3csc(C)n3)[nH]c2c1 c1(C(CC)(C)O)cn(C(C)CNC(c2ccc(-c3ccco3)s2)=O)nn1 CCCCCC(=O)NCC1(F)CN(C(C2CCCN(C(=O)C3CC3)C2)=O)C1 C(=O)(C1CCCn2ccnc21)NCCN(C(c1n(C=C)nnc1)=O)CC c1(OC)c(C(=O)N(CCCCNC(=O)CC(C)(C)C)C)cccc1Br Cc1cc2ncc(C(=O)NCC3CC3NC(c3ncccc3Cl)=O)cc2[nH]1 c1(NC(c2n(CC=C)nnn2)CCCSC)ccc(F)cc1CO Cc1ccc(C)n1-c1c(C(=O)NC2CCC(c3ccccc3)O2)cnn1C CCC(C)(C#N)C(=O)N(CCCNC(c1cnc(C(F)(F)F)cn1)=O)C CC(CNC(=O)C=Cc1ccco1)C(F)C(=O)N1CC(CO)C(C)(C)C1 N1(C(C2CCN(CC)CC2)=O)CC2OCCN(C(=O)C=C(C)C(C)(C)C)C2C1 c1(CC)ccc(C)cc1NC(c1nc(C)oc1C)=O.C1(C=O)CC(=O)CS1.N C1(NC(c2cc(C)[nH]c2)=O)CCCC2CN(C(c3nnn(C)n3)=O)CC12 C12CCCN1C(=O)CC1C=CC(C1)NC2=O.c1(CN(C)C)ncsc1C C1(NC(c2c(OCC)n[nH]c2)=O)CN(C(=O)CC2CCCCCC2)CC1C1CC1 C1(NC(CC23CC(C)(OC2)C3)=O)CC1C1CCCN(C(c2nccs2)=O)C1 c1(CN(CCCNC(C2(C)CC2F)=O)C)ccc(OC2CC2)cc1 C1(CN(C(=O)CSCc2cccs2)C)COCCN1C(=O)CS(N)(=O)=O Cc1ccc(C=CC(=O)NC(CCOCCO)C(N2CCC3(CC2)CC3)=O)cc1 C1(C2(O)CCN(C(C3C=CCC3)=O)CC2)(NC(C(CC)CC(C)C)=O)CC1 C1(NC(C(CCC)NC(N)=O)=O)CC2CCC1N2C(c1cccn1CC)=O Cc1ccc(OCC(=O)NCCNC(c2nn(C(C)(C)C)cc2Cl)=O)cc1C c1(OC)ccc(C)c(C(=O)NCC(C)CNC(c2cc[nH]c(=N)c2)=O)n1 Cc1nc(C2CCC2)oc1C(=O)NC1(C)CN(C(=O)C)C1.CCN(C)C.S N1(C(C2(C=C)CC2)=O)CCC(C(C)(C)C)(CNC(=O)Cc2cn[nH]c2)C1 S(=O)(=O)(CCCC(=O)OC)NCC(=O)N(C(C)C(c1ccccc1)O)CC c1(C=O)cc2ccccc2o1.C1CC2(C1)CC2.C(=O)(C(F)(F)F)NCC=O.N C=CC(C)(O)C(=O)N1CCOC(CCCNC(=O)C=CS(C)=O)C1 CN1CCC2CN(C(N3CCCC(Cc4ccccn4)C3)=O)CC12 N1(C(C(CC(=C)C)OC)=O)CCCC12CCN(C(=O)C(C)CCCC)C2 Cc1noc(C)c1CCC(N1CCCC1CCC(=O)NCCC(C)C)=O CC1CCCC(C)N(C(C2CCN(C(c3coc(N(C)C)n3)=O)CCO2)=O)C1 C1(NC(C2C=CC(NC(C3COCOC3)=O)C2)=O)CCC2(CCC2)C1 Cc1csc(C(=O)NCC(C)(C)NC(=O)CN(C2CCSC2)C)c1C N1(C(CCCSC)C(=O)NCCC2(C)CC2)CCc2nnnn2CC1 N1(C(c2ccc(C(C)C)o2)=O)CCCC(CCNC(C2CCCN2C(C)C)=O)C1 CCC(C)C(O)C(C)C(=O)NCC(C1CCOC1)NC(c1cnc(Cl)cc1N)=O C1(C(N2CC(N3CCN(C(CC)=O)CC3)C2)=O)CC2(C1)CC21CC1.CC(C)C.O CCC(CCCC(=O)N(C1CCOC1=O)C)NC(=O)CCCC(=O)N(C)C C1(C(N2CCCC(NC(c3cc(N)cc(O)n3)=O)C2)=O)CCC2C(C1)C2(F)F C1(O)(C=O)CCN(C(=O)Cc2cccc(C#N)c2)CC1.c1(C(=O)OC)cccs1 C(=O)(C1CCCc2c1ncn2C)N1CCC(NC(C2CCN(CC)C2)=O)CC1C N1(C(C2=CCC(C)(C)CC2)=O)CCN(C(c2ccc(Cl)c(N)c2)=O)CC2(CC2)C1 CN1N=C(C(=O)N2CCC(C(N3CCC4(CC(CO)C4)C3)=O)C23CCC3)CCC1=O Cc1ccc(C(=O)NCC(C2CCC2)NC(C2CCCC(=O)O2)=O)cc1Cl c1(CCC(=O)N(CCCNC(CC=C(C)C)=O)C(C)C)cccnc1Br C1(c2ccccc2Cl)(C(=O)NC(C(C)C)CNC(=O)C(C)C#N)CCOCC1 c1(C(C)=O)ccc(N2CCC(CC(C)NC(=O)CCC3CCCCO3)CC2)nc1 c1(OC)ccc2cc(CNC(c3nnnn3CC3CC3)CC3CC3)ccc2c1 c1(OCC)ccc(OC2CCCC2)cc1NC(c1cc(OC)c(Cl)cn1)=O C#CCC(CC(=O)NCC(C)C(=O)OCC)NC(=O)C(C1CCOCC1)=O CC(C)(CNC(C1CCC1)=O)CCNC(C1COCCO1)=O.C(C)(C)C.O C1(CC)CN(C)CCN1C(=O)CC1C=CC(NC(C2C3CC(=O)CC23)=O)C1 C(CCCC(=O)N(CC(C)N(C)C(c1cccc(-c2nccs2)c1)=O)C)SC c1(CC=C)cccc(C(=O)NC2CCOCC2C(=O)N)c1.C1(C(O)CO)CC1 Cc1nn(C)c2ncc(C=CCCCN=C(NCCF)NC3CCC3)cc12 c1(C=O)ccnc2ccc(F)cc12.CC(F)C.CCCCOC(=O)C=CC=O.N N1(C(=O)CSc2cccc(Cl)c2)CCC2(CC1)CN(C(c1cscn1)=O)CCO2 c1(OC)ccc(S(=O)(=O)NCCN2CCO2)cc1 c1(C(=O)NCC(CC)NC(=O)CC2CCC(=O)C2)ccc(C(=O)OC)cc1 c1(OC)ncc(C)cc1C(N1CCCCC1C(=O)NC)=O.c1ccc(O)c(O)c1 n1(CC(=O)NCCC(=C)CNC(=O)Cc2ccccc2)cccc(O)c1=O C1(CNC(C=Cc2n(C)cnc2)=O)CC2CN(C(=O)CC(O)C3CCCC3)CC12 c1(C(NOCC(CC)C)=O)cccc(CNC(C2CC2F)=O)n1 CC(C(=O)NCC1CCN1C(=O)Cc1cnns1)C1CCCC1 c1(OC)cccc2c1CCC(NC(=O)NC(c1ccc(OC(F)F)cc1)C)C2.OC c1(C(C(=O)NCC)N(C2CCN(CC(C)O)CC2)C)ccc(Br)c(OC)c1 C1(CNC(CSCC=C)=O)CCCC12CCN(C(=O)CC1CCCN1C)CC2 c1(C(N2C(CNC(c3cc(Cl)ncc3Cl)=O)COCC2)=O)ccc2c[nH]nc2c1 C1(CNC(C2CCN(CC#C)CC2)=O)COCCN(C(c2ncccc2Cl)=O)C1 C1(NC(CC(C=C)C)=O)CCC2(CC1)CN(C(C1CCOCC13CCCC3)=O)C2 CC1CCC(NC(c2ccc(CCF)cc2)=O)CN1C(=O)CCCn1ccnc1 N1(C(CC2(C=C)CCC2)=O)CC(CNC(=O)Cc2cccnc2)CC(C)C1 C1(C=O)CCC(C)(F)CC1.C(=O)(C1=CC(C)(C)C1)N1CC(COC)(C)C1 c1(C(=O)NC2C(NC(C3=C(C)OCC3)=O)CCC2)cc(=O)n2nccc2[nH]1 c1(C(=O)NC(CC=C)CNC(c2cc(C)sc2C)=O)c(C)oc2ncnc(O)c12 N1(C(c2cccc(N)c2F)=O)CCC2(CCN(C(C34CCC(CO3)C4)=O)C2)C1 c1(C(=O)NCC(F)CNC(=O)C(O)CC2CC2)ccc(N2CCOCC2)cc1 c1(C(=O)NCC(C)N(C(c2nc(CC)sc2)=O)C)ccc(Cl)c(F)c1F c1(CC(c2ccn(C)c2)NC(=O)CCOCC2CC2)ccccc1F c1(C(N2CC3C(CN4C5CCCC4CNC5)C3C2)=O)cc2ccncc2cc1F n1(CC)nccc1C1CC1C(=O)NCCN1CCC(C(F)(F)F)C1 CCCS(=O)(=O)CC(=O)N1CC(CNC(=O)C(CC)CC(C)C)C(C)(C)C1 C(=O)(C1=CS(=O)CCC1)NC1C(C)N(C(=O)CC23COC(C)(C2)C3)CCC1 c1(OC)cc(OC)cc(CC(=O)NC2CCCC2NC(C2(C)C=CCC2)=O)c1 C1(NC(C2CC(SC)C2)=O)CN(C(c2cnc(CC(C)(C)C)s2)=O)CC1C Cc1cc(C(N2CC(N3CCN(C(=O)C(C)S(C)(=O)=O)CC3)C2)=O)c(C)cc1Cl N1(C(c2c(C#C)cnn2C)=O)CCC2(CC1)CC(NC(=O)C(C)N1CC(C)C1)C2 C(=O)(C(CC1CCCC1)NC(=O)CC1CCSCC1)NC(C(C)O)C c1(C(=O)NC2C(OC)CN(C(C3CCCO3)=O)C2)cc2cc(Cl)ccc2o1 c1(OCCCC)ccc(C(N2CCN(C(C)(C)C)CC2)C(=O)NCC)cc1 C12CCCN(C1)C(=O)c1ccn2n1.C(=O)(CCCn1cncn1)OCC CC1(C)CCN(C(=O)Cn2cnnc2O)C1CC(=O)NCc1nc(=O)o[nH]1 C(CCC(C(=O)NC1CCOCC1)N(C(C)C(C)(C)CO)C)SC.C1C(=O)N1 c1(C(=O)NCC2CC(NC(C3CCC(C)S3)=O)C2)cc2oc(Br)cc2[nH]1 N1(C(c2c(C)nns2)=O)CC2CC1CCC2NC(c1nn(C)c2c1CCC2)=O C1(N(C(C(CC2CC2)OC)=O)CC2CC2)CCCN(C(=O)C(F)F)CC1 c1(NC(C(=O)N(C2CCN(C(CC(CC)C)=O)CC2)C)=O)ccc(Cl)c(F)c1 c1(C(N2CCCC(C(C)NC(Cc3ccn(CC)n3)=O)C2)=O)cc2n(n1)CCC2 c1(OC)cc(C(=O)NCC(CO)NC(c2cnnn2C2CC2)=O)ccc1Br c1(C(=O)NCC2C(NC(=O)CCCF)C2)cccc(Cl)c1Br N1(C(CC(CC)OC)=O)CCc2ccc(C(=O)NCCC3(O)CCOC3)nc2C1 N1(C(C(C)OCC)=O)CC2CCC1CN2CCN(C1CC1)CC c1(CC=C)cccc(OC(c2nc(C3CC3)cs2)(C)C)c1 N1(C(C(C)=CC)=O)CC2CCCC2(NC(c2csc(C3CCCO3)n2)=O)C1 c1(C(=O)NC(C)CCNC(=O)C=Cc2ncco2)cc(O)ccc1Cl C1(CC(=O)N(C(C(=O)N(CC)Cc2cccnc2)C)C)CC(O)C1(C)C N1(C(C2C(CCOC)C2)=O)CC(O)(CN(C)C(C2CC23CCC3)=O)C1 CC(C)(C)CN(C(=O)Cn1cnc(C(F)(F)F)n1)C.C(C=O)C1CC1.CC CCCCCC(CC)C(=O)NC(CNC(=O)COC(F)F)CC(C)C N1(C(C2CC(C#N)(O)C2)=O)CC2CCC(NC(=O)C=Cc3cnccn3)CC2C1 C1(NC(c2ocnc2C(F)F)=O)CCC(CNC(C2(F)CC2)=O)C1 c1(C(N(CC(C(N2C(C(=O)OC)C(C)CC2)=O)C)C)=O)cccc(F)c1N C1(NC(C2CCCC2)=O)CCCCC1NC(C1(C2CC2)CCCO1)=O CCCC(C(=O)N(C)CC=CC(=O)N(C(C)C(C)C)C)OCC CCCC(C#N)C(=O)NC(C)CC(=O)N1CC(C)(C)C1 N1(CC(N2CCC(CCNC(=O)CCN3CCC(F)C3)C2)=O)C(=O)CNC1=O Cc1cc(NC(C2(C)CC=CCC2)=O)cc(Cl)c1 c1(CC)ccc(C(=O)N(C2CN(C(C3CCCN3C)=O)CC2(C)C)C)c(F)c1 c1(OC)cc(CC(=O)NC2CCN(C(C3(C)COC3)=O)CC2F)ccc1C N1(C(C(C)=CC2CC2)=O)CC(CNC(=O)CCCCN(C)C)OC2COCC12 C(CCCCCCCO)n1cc(C2C(C(=O)NCCOc3cn(C)nc3)C2)nn1 c1(NC(c2n(C)ncc2)=O)ccc(=NCc2cc3ccccc3s2)[nH]c1 C1(NC(C(CCOC)(C)C)=O)C2CCN(C(c3cc[n+]([O-])cc3)=O)CCC12 C(C(C)(C)C(=O)N1CCOCC1)OC(C1(Cl)C(C(C)=O)C1)=O C1(CNC(C(C)CF)=O)(NC(c2ccn(CC#N)n2)=O)CCC(F)(F)CC1 c1(SC2(C)CCN2C)nc(Cl)ccc1Cl.C1(c2cn(CC)nn2)CNC(=O)CO1 CN1C(=O)CCC1C(=O)NCC1(CNC(=O)CCC(N)=O)CC12CCC2 C1(C(=O)OC)SC(C)CC(N2CCCC(C)(C(=O)N(C)C)C2)C1C c1(C(N2CCC(F)C2)=O)coc2c1C(=O)NCCC2.C(C(=O)NC)(C(C)C)SC c1(C(=O)NCCC2(O)CCCN(C(CCC(N)=O)=O)C2)c(N)cccc1[N+](=O)[O-] CC1(C)CCC(C(=O)NCCOCCCNC(=O)Cc2cccnc2F)OC1 Cc1oc2ccccc2c1C(=O)NCCC1(NC(C2CC3CC3C2)=O)CCC1 C1(NC(C(COC)OC)=O)COC2(C1)CN(C(C1CCC1)=O)C2.c1cnn[nH]1.C c1(CC(=O)NCC2C(NC(c3cncc(C)n3)=O)CCC2)cccc(F)c1Cl C(=O)(CC1=CCN(C)CC1)NCC1N(C(C(CC2CC2)OC)=O)CC(O)C1 c1(CNC(CC)CCOC)cc(Cl)ccc1Br CC1(C(N2CCC3(C2)CN(C(C2(C#N)CCCO2)=O)C3)=O)CCCCNC1=O C1(NC2(c3n(CC(F)F)nnn3)CCCSCC2)CCC(C2CCC2)CC1 Cc1cccc(OCC(=O)NC2(CNC(C3CC3(Cl)Cl)=O)CCC2)c1C C(C(C)CN(C(=O)CC1CC(CNC(=O)CC2CCCO2)C1)C)OC C1(CCC(=O)NC2CC3CC3C2)CCN(C(=O)C=Cc2cccnc2)CC1 c1(C(=O)NC23C(CN(C(COCC=C)=O)C2)C3)ccc2cccnc2c1 C1(C(=O)NCCNC(CCOCCOCCOC)=O)(CF)CCCOC1 C1(NC(C2N(C(c3ccc(NC)cc3)=O)CCSC2)=O)C2CCN(CC2)C1C C(C(C)(C)C(=O)NCC1OCCC1C(=O)N(CCCC(=O)OC)C)OC C1(c2ccccc2)(C=O)CC2(CC2)C1.C(C)C=O.C1CCC1.C(=O)OCC C=CCC(CNC(c1ccoc1Cl)=O)NC(c1ccnn1C1CCOCC1)=O N1(C(C(COC)(C)O)=O)CC2CC(CNC(=O)Cc3cccc(F)c3)C2C1 C1(NC(C(C)N2CCCC2)=O)CCCCCN(C(c2cncc3nc[nH]c23)=O)C1 CCC(CNC(c1n[nH]cc1[N+](=O)[O-])=O)N=c1[nH]nc(C)o1 C1(C(=O)NC(C2(O)CN(C(C3(Cl)CC3)=O)C2)C)COC(=O)N1C N1(C(CCSCCC)=O)CCC2CCN(C(=O)CC(C)(C)CCOC)CC12 C1(C(=O)N)CN(C(c2ccc(Br)cc2)=O)CC1(F)F.N(C)(C(=S)NCC)CC N1(C(CSCCOC)=O)CC2(CCC2)CCC1.C1(C=O)CCN(C(C)C)C1.C C1(C2NC(=O)N(C(C3CCCCO3)C#C)C2=O)CC2(CCOCC2)CO1 C1(C(=O)NC(CCCC)CC)C(CC)CCCN1C(=O)COC1CC=CC1 c1(CC)cc(F)ccc1C(=O)NCC(O)CCNC(=O)C=CS(C)=O N1(C(C(C2CC2)OCC)=O)CC(C)OC2(CCN(C(=O)CCCF)CC2)C1 C1(O)(CN(C(=O)C(F)CC2CCC2)C)CN(C(c2cccs2)=O)C1 N1(C(C(CC)C#N)=O)CCCCCC1CNC(=O)Cn1cncc1C C(=O)(CCCCC(=O)NC(C)C=CC(=O)NC1C2CCCOC12)OC S(=O)(=O)(c1ccc(Cl)c(F)c1)N(CC(CCC)C)C.C(C)(C)C.C(=O)C1CC1 c1(SC)cc(C)ccc1C(=O)N.C1(C(N(C2CCCC2)CC)=O)CC1C1CC1 Cc1nccn1CCC(=O)N(CC(C)CNC(C1CCCC1F)=O)C C1(NC(c2c(C)ccs2)=O)CCN(C(=O)Cc2ccccc2)CC1C(C)C CC1CCN(CC(=O)NC2COCC2NC(c2cc(=O)cc[nH]2)=O)CC1 c1(SC)ccc(N)cc1C(=O)N.C1CC(C)N(C(c2ocnc2C(F)F)=O)C1 c1(CC)cnc(C(N2CC3C(C)C3C2)=O)cn1.C1(CC(=O)N)CCC(=O)N1C c1(C(C(=O)NCCOC)OC)ccccc1NC(c1nncs1)=O C1(C(=O)NC2C(C)COCC2)C2CCCC2CN1C(=O)CC1CCCC(=O)C1 Cc1ccc(C)c(SCC(=O)NC(C)(C)CO)c1.C1(C=O)CC(OC(F)F)C1 C1(NC(CC(C)(C)CC(F)F)=O)Cc2ccccc2N(C(C2CC3CC3C2)=O)C1 C(F)(F)(C(F)(F)F)CC.C1(CC(=O)NCC)COC(C)(C)C1 Cc1nc([N+](=O)[O-])cn1CC(=O)NCCCO.c1(C=O)cscc1C(F)(F)F.N c1(CC(N2CCC(NC(CCNC(C)=O)=O)C2(C)C)=O)cccc2ccncc12 c1(C(N(CCCN(C)C(C2(c3cccnc3)CCC2)=O)C)=O)ccc(Cl)o1 C1(CC=C)(NC(=O)CC2C=CCC2)CCN(C(c2snc(Cl)c2Cl)=O)C1 N1(C(C=C(C)Cl)=O)CC(NC(=O)C(C)(C)c2ccnn2C)CC2(CC2)C1 CN1CC2CCN(C(C3(CNC(C4CC5(CCO4)CC5)=O)CCC3)=O)CC2C1 C1(C(=O)NC2(CNC(=O)CC3CSCCO3)CCCC2)CC2(CCC2O)C1 CC(C)(O)C(C)(C)C(=O)N1CCC(OC2CCCC2)C1 c1(C(C(=O)N(C)CC2CCN(C(C(CC)F)=O)C2)(C)C)ccc(Cl)nc1 Cc1nc(C(=O)NCC2CC2NC(=O)CC(C)N(C)C)ccc1[N+](=O)[O-] N1(C(CC(COC)C)=O)CCC2C(C1)NC(=O)CN2C(=O)CN(C)C(C)=O CC(C)CC(O)CC(=O)N1CCN(C(=O)CCOc2ccc(F)cc2)C2CC12 CCCCCC(CCCCC)C(=O)N1CCCCC1C(=O)NCc1nn[nH]n1 c1(NC(=O)NCC2(C)CCCN2c2ccc(C#N)nc2)ccc2ncnn2c1 O=C(C#CC1CCCCC1)NC1CC(O)C1CC(=O)N(C1CCCC1)C1CC1 N1(C(c2n(CC)ccn2)=O)CCC(C(N2CCC(N=[N+]=[N-])C2)=O)C(C)C1 c1(NC(c2ccc(NCc3cc(C)n(C)n3)cn2)=O)ccc2nc(O)[nH]c2c1 N1(C(C(C)N(C)C)=O)CC(CNC(C2(Cl)CC2(C)C)=O)OC(C)(C)C1 CC(C)C(C(=O)NCCN1C(=O)CCC1=O)C(C)NC(C12CC1CNC2=O)=O c1(OC)c(C(C)=O)cc(Cl)cc1-c1ccc(-c2nccn2CCC(C)OC)cc1 c1(OC)ccc(-c2cncc(C(=O)NC3CC(F)C3)c2)c(OC)n1 C(=O)(CC(C)C(F)(F)F)N1C(CNC(C(CC)(C)F)=O)CN(C)CC1 c1(C(N2CCC(OC)(C)C2)=O)coc2ccc(F)cc12.C(=O)C(C)C(F)(F)F.N C12(CNC(Cc3c(C)cccc3C)=O)CCCC1CCN2C(=O)C1CC1 N1(C(C(C)(C)c2cnco2)=O)CCC(C2CC2NC(C2CCCCO2)=O)CC1 Cc1cc(C)c(C(N2CCN(C(c3cc(C)sc3C)=O)C3CC23)=O)c([N+](=O)[O-])c1 C1(C(NOC(C=O)C)=O)CC(O)(C(=O)N(c2ccncc2)C(C)(C)C)C1.CC c1(C(=O)NC2C(NC(=O)CCc3c(Cl)cncc3Cl)C2)n[nH]c2ccccc12 N1(C(C(C2CCC2)OCC)=O)CCC(N(C)C(c2cncnc2)=O)C1 O=C(NOCC1CCCC1)C(CC1CCC1)NC(C1CC12CCC2)=O CC1=C(C(=O)N(C)CC2CCCN2C(=O)Cc2coc(C)n2)SCCO1 C1(OC)CCN(C(C2(NC(=O)C=CC(C)(C)C)CC2(C)C)=O)CC1(C)C c1(CCNC(C2CC2NCc2ccccc2O)=O)ccc(Cl)cc1F CCC(F)(F)C(C)(C)C(=O)NC1CCC1NC(=O)CCc1ncccc1C CC1CCCCN1CC(=O)NCCN1CCC(NC(=O)CCc2cnn(C)c2)C1 c1(C(=O)NCC(COC)NC(=O)C(c2ccccc2)(F)F)ccnc(S)c1.O N1(CC(n2cccn2)C)CCC(CC(=O)NCCSC(C)(C)C)C1 c1(OC)cccc(Cn2nnnc2C(c2ccc(C)s2)NC(C2CCCC2)C)c1 c1(C(C2CCCO2)N(c2c(OC)ccc(C#N)c2)C)nc(O)c2ccccc2n1 C#CC(CNC(=O)C(CC1CCC1)NC(=O)CC1OCCO1)CC CCC(C)C(O)C(C)C(=O)NCc1c[nH]nc1C(=O)NCC(C)CN(C)C CC(C)C(CO)C(=O)N1CC(NC(=O)Cn2cnnn2)C(C)(C)C1 C1(C(C)C)CCCCC1N=c1cc(NCCC#N)nc(COC)[nH]1 c1(CCCNC(C(CCN)OC(C)C)=O)[nH][nH]c(=N)c1C#N c1(N2C(CNC(C(C(CC)C)NC(C)=O)=O)CC3(CC3)C2)ncnc2cc[nH]c12 C(CC(C)(C)C(=O)NCC1CC(F)C1)OC.C(C1CCCC1)=C(C=O)C.C C1(NC(C(C)OCC(F)(F)F)=O)CCN(C(c2occc2F)=O)C1C C1(C(N(CCCC)C)=O)CC2CCC(C1)S2(=O)=O.C1(C)CCCC1.C(=O)(C)N c1(C(N(CCCCNC(c2nc(OCC)oc2)=O)C)=O)cccc(F)c1N S(=O)(=O)(c1nc2ccccc2s1)NCC(C1CC=CCC1)=O C1(C(=O)NCC(C2CCN(C(Cc3c(C)nc[nH]3)=O)CC2)C)CC2C=CC1CC2 C1(NC(CC(C=C)c2ccccc2)=O)CCN(C(=O)Cc2cnc(C)[nH]2)C(C)C1 c1(C=O)ccc(F)c(C)c1.c1(NC)nccnc1NC(c1ccn(CC)n1)=O.N c1(CC)[nH]nc(Cl)c1C(=O)N(C(CNC(C1CC=CCC1)=O)CC)C C1(NC(CNC(=O)OCC)=O)CC12CCCCC2.C1(C(=O)N)CCCCO1 c1(C(N2CCC(CN3CCCCC3)CC2)=O)cccc(Cl)c1C(F)F C1(C(=O)NC2CC(NC(CCNC(COC)=O)=O)C2)CN(C)CC(C)O1 C(=O)(CC(C)(C)C(F)F)NCc1cccc(NC(Cc2ccc(C)c(F)c2)=O)c1 N1(C(CC2OCCN(C(C3CC(C)N(C)C3)=O)C2)=O)CCC(C)(C#N)C1 N1(C(=O)NC(c2nc3c(s2)CC(C)CC3)C)CCCc2cccc(C(N)=O)c21 C12(NC(Cn3ncn(C)c3=O)=O)CCN(C(=O)CC(C)(C)C3CC3)CC1C2 c1(C(N2CC(NC(=O)CSCC(F)F)C(CO)CC2)=O)occ2c1CCCC2 c1(C2N3CC(C(O)C3)NC2=O)cc(F)ccc1C.C1(NC(C)=O)CCOC1 C1(NC(CCCSC)=O)CCCOC12CCN(C(=O)C(c1cnn(C)c1)O)CC2 CC1=C(C(=O)N2CCN(C(c3c[nH]nc3C)=O)C(CC(C)(C)C)C2)CCO1 c1(C=O)ccc(F)c(C#N)c1.C1(CNC(C2(CCCC)CC2)=O)CCCC1.N N1(C(c2c(C)nccn2)=O)CC(C(=O)Nc2conc2C)CC1(C)C C(=O)C(C)S(=O)(=O)C(C)C.c1(CC)cnc(O)c(C(=O)NC2CCOCC2)c1 C1(C(C)NC(c2cnn(-c3ccccc3)n2)=O)CCCN(CC2CCC(=O)N2)C1 C1(C(=O)NCC(C2CCCC2)NC(=O)C=CCO)CC2(CCC2)CO1 C(CO)(CCCNC(=O)Cc1ccccc1SC)NC(C1(CC)CCCO1)=O CC1COCC(CC(N2CC(CNC(=O)COCP(C)(C)=O)C2)=O)O1 O=C(CS(=O)(=O)CCO)NCC12CC(CO1)N(C(c1ccc(O)cn1)=O)C2 CCC(C)C(C(=O)Nc1cc(C)ns1)N(CC(=O)OC)C(c1ccccc1)C N1(C(C=CC)=O)CCOC(C(N2CCC2COC)=O)CC1 Cc1cc(C)c(CNC2CC(C(=O)Nc3cccc(CO)n3)C2)c(C)c1 c1(N2CCC(c3c(C(=O)OC)cccc3)C2)cc(C)nc2c(C(=O)OC)cnn12 CCCC(C(O)C(=O)NCC(O)CC(C)C)NC(c1c[nH]c2ccccc12)=O c1(C(=O)NC2CCC(C(=O)NCCOCCO)C2)c(Cl)cc(Cl)cc1Cl O=C(NN=c1ccc2nccn2[nH]1)c1n[nH]c2c(I)cccc12 Cc1nc(C)c(CC(N2CCN(CCS(C)(=O)=O)CC2)=O)s1 C1(NC(CCn2c(C(C)C)ncc2)=O)CCCN(C(C2CCC(C)O2)=O)CC1 N1(C(c2c(C)snn2)=O)CC(CC(=O)NC2CN3CCC2CC3)CC1(C)C C1(F)(C(=O)NC2C(SC)CN(C(c3cnn(C)c3)=O)C2)CCN(C)CC1 N1(C(c2cc(CCC)ncc2)=O)CC(NC(c2cccc(=O)n2C)=O)C(C)(C)C1 CC1(C)CCN(C(C2CCCCC23CCC3)=O)CC1C.C12(C=O)CC(F)(C1)C2.N CC1CC(C(N2CCN(c3ccccn3)CC2)=O)N(CC2(c3cccs3)CC2)C1 C1(C)(C(=O)NCC(=CC(=O)NOCC(O)C(C)C)C)CCCC1O N1(C(C2CCN(C)C(=O)C2)=O)CCC(C2CC2)(CNC(=O)C=O)C1.C1CC1.N c1(C(N2CCC(NC(C(C)NC(C)=O)=O)C2)=O)n[nH]c2ccc(Br)cc12 C1(CC(=O)NC(CCC)CNC(=O)COCCOC)CCCN(C)C1 C(=O)(C1CCCn2nccc21)NC1(CC=C)CCN(C(=O)Cn2cc(Cl)cn2)C1 C(=O)(CS(=O)(=O)C(C)(C)C)NC(CNC(COC)=O)C1CC1 Cc1cc([N+](=O)[O-])ccc1CNc1c[nH]nc1C(=O)NC(c1cnccn1)C CCC(CC)C(=O)NCCC1COCCN1C(c1ccn(CCC(F)(F)F)n1)=O C#CCC(C)(CC)C(=O)NCC1CCN1C(=O)CC1CCN(CC(C)C)C1 Cc1scnc1C(=O)NCC1CCCC1NC(=O)CC(C)N1CCCC1=O Cc1nc2ccc(C(=O)NCC3CCN(c4ccc(C(=O)O)cn4)CC3)cc2[nH]1 C1(C)(CNC(C(CSC)C)=O)CCCN(C(c2cc(C(F)F)cs2)=O)C1 CC(C)C(C(=O)NCCC(C)NC(=O)CCc1sccc1Br)C1CCC1 Cc1cc(C(N2CC(CNCc3c(Cl)ccnc3C)C(C)C2)=O)cc(Cl)c1 C(C)(CCCN=c1[nH]cnc(Cl)c1F)NC(CC(CC)CC(F)(F)F)=O C12CCCN(C1)C2=O.C(C(CC)NC=O)NC(COCCOCC#C)=O N1(C(C2N(CC)CCC2)=O)CCN(C(=O)CC2(C)CCCCC2)CC1C1CCC1 C(=O)(C(F)CC1CCCCC1)NC(CN(C(=O)CCC=CC(C)C)CC)C C1(NC(C2C3(CCC3)C23CCC3)=O)COC2(CCN(C(=O)CCC3CC3)C2)C1 Cc1cc(C(F)(F)F)nc(N2CCC(C)(C)C2)n1.C1(CC(C)C)(C(=O)N)COC1 Cc1cnc(NCC2CCCCN2C(c2ccc(C3CC3)cc2)=O)nc1 Cc1cc(S(N)(=O)=O)oc1C(=O)NCCNC(C1(C)CC=CCC1)=O c1(OC)cc(C(=O)NCC2(F)CCCN(C(=O)CCCCCBr)C2)cnc1Br N1(C(C(CCC)N(C)C)=O)CCC2(CCC(NC(=O)C3=NOC4COCC34)C2)C1 CC1CN(C(c2sccc2Br)=O)CC(C)C1NC(=O)CN(C)C C1(CC(=O)NC(CCC)CNC(=O)COC)CCN(C)CC1 C1(NC(C(C)(C)c2ccno2)=O)CCCC(NC(=O)CN2CCOCC2)C1 c1(C(=O)NC(C)CNC(=O)C(F)(F)c2ccccn2)ccc2ccnc(Cl)c2n1 CCC(C)(CNC(C1CCC1C(=O)OC)=O)C(=O)NC(CO)C1(O)CC1 N1(C(CCCN(C(C)C)C)=O)CCN(C(=O)C=Cc2ncco2)C2COCC12 C1(NC(C(c2ccc(F)cc2)(C)N(C)C)=O)CN(C(C2CC(O)C2)=O)CC1(C)C CCC(CC(F)F)C(=O)NC(C)(C)CN1CCN(C(C23CC2C3)=O)CC1 C12(NC(C=CC)=O)CCOCC1CN(C(=O)CC(c1ccc(OC)cc1)C)C2 C1(C(N2CCCC(N(C(c3ocnc3CC)=O)CC)C2)=O)CCn2cncc2C1 C1(CC=O)OCCCC1(C)C.c1(CCC)ncc(C(=O)NCC2COCC2)s1.N C(CC(=O)N(C1CCC1C)C)(C(F)(F)F)NC(Cc1cccc(C)c1)=O CC1(C)CN(C(c2cccnc2N)=O)CC1NC(c1ccoc1)=O N1(C(C2CC(C)OC2)=O)CC2CCC1CN2C(=O)Cc1ccon1 C1CCCN(C(=O)Cn2nnc(C3CC3)n2)CC1.Cc1nn(C)cc1C(=O)NC C1(C(=O)NCC2CC2(F)F)CCC2CCC1N2C(=O)C=CC1CC1 Cc1ncc(N)cc1C(=O)NC1CCCCC1NC(C1OC2CCC1C2)=O C1(C(=O)NC(CNC(=O)OC)C)CC(N=[N+]=[N-])CN1C(=O)CC(C)(C)O Cc1cccnc1CCC(=O)NC1CC(NC(=O)Cc2ccco2)C1 c1(CC(N2CC(C(N(CCC)CCC)=O)C(C)CC2)=O)c[nH]c2nccc(Cl)c12 C1(CC(N2C(CN(C)C)CCC2)=O)C2CCC(C2)N1C(C1CCC(=O)O1)=O C(=O)(C1=NOC(CNC(C23CSCC2C3)=O)C1)N1CCC(C#C)C1 c1(OC)ccc(CCNCCC(CNC(N2CCCC2)=O)OC)cc1O c1(C(C)C(=O)NC2CCC(NC(c3ccc[nH]3)=O)C2)ccc2ccccc2c1 C1(C(N2CCCC(C(C(=O)NC3(CC=C)CCOC3)C)C2)=O)CC(C)CC(=O)N1 Cc1cc2c[nH]nc2cc1C(=O)NC1CCN(C(C2(C)CC(C(C)C)=NO2)=O)C1 CCC(N=c1[nH]c(=NC(C)c2ccc(Br)s2)[nH]c2ccsc12)c1nncn1C CC1CN(C(c2ccc(F)o2)=O)CCC1CNC(c1cnn[nH]1)=O Cn1cnnc1.C(CC(=O)N)SCC1CCN1C(=O)CSC1CC1 N1(C(=O)CCF)CCN(C(c2ccc(C3CC3)nn2)=O)C(c2ccncc2)C1 Cn1nc(C2CCC2)cc1CNC(c1ccccc1)CC1OC2CCC1C2 Cc1nc(C)c(C(=O)NCC(C)C(C)C)[nH]1.c1(C=O)cc(C)c(C(C)C)s1.N Cc1ncc(C=CCNC(N2CC(c3noc(C)c3C)(O)C2)=O)s1 CC(=O)CCCC(=O)N1CCCC(CCNC(C23CC(CN2C2CC2)C3)=O)C1 CC1(C#CC(=O)N2CCCC2CCNC(c2ccc(C(F)(F)F)[nH]2)=O)CCCO1 C1(NC(CC(C)(C)C#N)c2nnnn2C2(C)CC2)COC2(C1)CC1(CNC1)C2 N1(C(c2c(C)nn[nH]2)=O)CCC2(NC(=O)COC3CCC(F)(F)CC3)CC2C1 n1(C2CCC2)cc(CCCC)nn1.CC(C=O)OCCOCCOCCO.N C1(C(=O)NCC=CC)CCN1C(=O)C(C)OCCOC c1(C(=O)NCCCN(C(CCOc2ccc(C)cc2)=O)C)cccc(S(C)=O)c1 c1(C(N2CCC3(C(NC(C4CCC(C)O4)=O)C3)CC2)=O)ccc2c(c1)nnn2C C12(CNC(C3CC3(C)C)CC)C3CCC(CC13)C2(F)F c1(OC2CCN(C(=O)NC3CCN(CC#C)CC3)CC2)cccc([N+](=O)[O-])c1 N1(C(C(C)(C)NC(=O)Cc2ccc[nH]2)=O)CCN(CC(=O)N(C)C)CC1 C12(CNC(CSCC)=O)CC(CNC(=O)CCS(C)=O)(CO1)C2 CCC(C(=O)NCC1CCCN(C(c2cn(C)nc2C2CCC2)=O)CC1)C(C)C CN=c1nc(N(C)CC2CCN(C)CC2)[nH]c(=NCC2(C)CC2Br)[nH]1 C1(CNC(CN(C(C)=O)C)=O)CC12CCN(C(C1CN3CCCC3CO1)=O)CC2 c1(OC)c(C(=O)NCC(C)NC(=O)CCCCCN(C)C)occc1=O Cc1nn(C)cc1C(C)C(=O)NC1CCN(C(c2cc[nH]c(=N)c2)=O)C1 C1(C(=O)NC(CNC(C2(CCCC)CC2)=O)(C)CC)CCCC(F)(F)C1 C1(CC)CN(C(c2cnc(O)c(F)c2)=O)CCC1C.C1(C=O)NC(=O)OC1C.N O=C(C=NN1CCCCC1)N(C1C2CCC(C2)C1C(=O)N=c1cco[nH]1)CCO C(C(C)CC(=O)NC(C)(C(=O)NCC1CC1)C1CCC1)OC c1(SC)nc(N2CC(C)(C)CC2C)ncc1C.c1(C=O)cnn(C(C)(C)C)c1.N CC1CC(C(N)=O)c2ccccc2N1C(=O)C1=NOC(C)C1 C1(O)(CNC(CN(C)CC)=O)CC(C(=O)NC(C2CCCC2O)C)C1 C(=O)(C(=O)C(C)(C)C)N(C(C)CCNC(=O)C=Cc1ccc(Cl)s1)C Cc1cccc(C(CNC(C2C3CC4C(C3)C24)=O)NC(=O)C2=CCSC2)c1 C1(C(N2CCC(C(C(N3C(C=C)CCC3)=O)C)CC2)=O)Cc2nccn2C1 c1(C(N2CC3C(CNC(CCC(=C)Cl)=O)(CCC3)C2)=O)[nH]c2ccccc2c1Cl Cc1nc2ncnn2c(C)c1C(=O)NC(C)CCNC(c1ccc(F)cc1N)=O C1(O)(C(C)CNC(C2(CF)CC2)=O)CCN(C(c2ncncc2Cl)=O)C1 CCCC(CNC(=O)Cc1csc(C)n1)C(=O)NCC(C)Cc1cn[nH]c1 C(CN=c1[nH]c(=NCc2ncco2)[nH]c2c1CSC2)(C1CCOC1)OC c1(C(=O)NCCN(C(=O)CC2CCOC2)C)cc2c(Cl)ccnc2s1 C(=O)(CC(C)(C)O)NC1CC(F)(CNC(c2nc(CCCCC)sc2)=O)C1 N1(C(C2C(C)C2)=O)CCC(C(F)F)CC1C.C(=O)CC(C)(C)C.C(=O)C.N Cc1[nH]nc(Cl)c1C(=O)NC.C1(CCC=O)CCC(=O)NC1.C12CC(C1)C2 c1(C=O)ccc2c(n1)NC(=O)CO2.N1(CC(=O)N(C)C)CCCC1=O.C1CC1 C(=O)(C1=C(Cl)CCOC1)NCCC(C(C)C)NC(=O)C(F)(F)c1nccs1 C1(CC=C)(C=O)CCCN1C(=O)C(N1CCOC1=O)C.C1CC1C(C)(C)C.N CON1CCC(C(=O)NC(C(=O)NOC(C)(C)CO)c2cnn(C)c2)C1 Cc1cn2cc(CNC(N3CCC(CC(=O)O)CC3)=O)nc2s1 C12(C(=O)NCC3C(C)CN(C(c4cccc(=O)o4)=O)C3)CCCC1CCC2 N1(C(C=C(CCC)C)=O)CCOCC1CN(C(=O)C(CC)NC(N)=O)C c1(C(C(=O)NCCCCCN(C(=O)CCC2(C)CC2)C)(C)C)c(F)cccc1F c1(CC)[nH]nc(Cl)c1C(=O)NCC(CC(C)C)NC(C1(OC)CCCSC1)=O Cc1cc(N2CCC(CC(C)NC(C3CCC3)=O)CC2)nc(C(C)(C)C)n1 C=C(C)C(CC(=O)NCC(C)NC(c1ccc(C(F)F)o1)=O)OCC c1(-c2cc(C)cc(F)c2)ncn2c1CN(Cc1ccc(Cl)cn1)CC2 C(CN=[N+]=[N-])(C(=O)N1CCC(O)C1C)NC(C1CC(C)N(C)C1)=O Cc1cc(C(=O)O)cc(=NCC23CCC(CC2)OC3)[nH]1 c1(C(=O)NCC(CC=C)NC(=O)CCOCC)ccc(OC)c(Cl)c1F CC1CCC(CN(C)C(=O)NCCC2CCC2(F)F)CC1 CC1(C)CCN(C(=O)C2=CCN(C(c3ccc(C(F)F)o3)=O)C2)CC1CO C(=O)(C1=NOC2COCC12)N(C(C)C)CCN(C)C(c1ccc(F)cc1F)=O C12(NC(C(CCC)N(C)C)=O)CCCCC1CN(C(c1cc(C)ncn1)=O)C2 N1(C(c2cc(C)[nH]c2C)=O)CC(CNC(c2ccccc2Cl)=O)N2CCC1C2 N1(C(CC2(NC(C)=O)CC2)=O)CCCC1C(C)(C)NC(C1CCOC1C)=O C1(NC(CC)=O)C2CC1N(C(C1CSCN1C(c1nncn1C)=O)=O)C2 C1(CN=C(NC(C)C)NCC2CCN(c3ccc(Cl)cc3)C2)CCCC(F)(F)C1 C1(OCCNC(=O)CCc2cnoc2)CCN(C(c2cc(CO)on2)=O)C1 C1(=CC(=O)NC23CCN(C(CC4CN(C)C4)=O)CC2C3)CCCCC1(C)C c1(C(=O)NCC(C#C)(C)C)oc(CNC(c2cc(OC)ncn2)=O)nc1C Cn1nc(C(N2CCOC(CC(=O)NC(c3cccc(Cl)c3)CO)C2)=O)cc1O c1(C(=O)NCc2c(C(N(CC(C)O)CC)=O)[nH]cc2)c[nH]c2cccnc12 N1(C(CSCCOC)=O)CC(NC(c2cc(C=O)nn2C)=O)CC2(CC2)C1 CC1(C(=O)NC(C)C2CCC2)OC(=O)c2ccccc21.C(=O)(C1=C(Cl)CCC1)N C(N=c1nc2sccc2c(NCCN(C)C2CC2)[nH]1)C1CC2N(C)C(CC2)C1 c1(C(=O)NC(CCNC(C(C)Oc2ccccc2Cl)=O)(C)C)n[nH]c2c1COC2 c1(OC(C2N(C(c3ccn(CCOC)n3)=O)CCC2)=O)cccc2c1CCOC2 c1(NC(C(CC=C)CNC(=O)CCNC(=O)COC)=O)cnn2ncccc12 N1(c2cc(NC3CC(OC(C)(C)C)C3)nc(C)n2)CCC(C2CNC(=O)C2)C1 c1(OC)cc(CC(=O)N)c(F)cc1O.C(C)C1CC1.C(=O)CN(CC(C)C)C N1(C(C2CC3(CCC3)CO2)=O)CCCC(C2CC2NC(C2(F)CCOC2)=O)C1 N1(C(c2cc(Cl)cnc2C)C(=O)NC(CC)(C)C)CCc2ccsc2C1C C12(CC)CCC(CC1)N2c1nnc(C)n1Cc1ccc(C)cc1C N1(C(c2c(Cl)cc(C)s2)=O)CC(NC(=O)CCCCC)CC(C)(C)C1.C(N)(=O)N Cc1ocnc1CC(=O)NCCCCNC(c1cnoc1C1CCC1)=O C1(C)(CNC(C2C(CNC(C(C)=C(C)C)=O)OCC2)=O)CCCCCC1 CC(CCC(C)(C)C)C(=O)N1CC2CC1C2NC(=O)CCCCCc1cccs1 CCCCCCCCCCC(=O)N1CCCSc2ccc(F)cc21.C(C)(C)C C(C(CC)(CC)NC(c1csc(C2CCCCC2)c1)=O)NC(CCC=C)=O C(O)(CN=c1ccc(Br)c(S(=O)(=O)N2CC(C)C(F)C2)[nH]1)c1ccc(C)c(F)c1 CCC(C)(CC)CN=c1[nH]c(=NCC2CSCCO2)[nH]c2c1CCCCCC2 N1(C(CNC(CC=C=C)=O)=O)CCN(C(C2CC2c2ccccc2Br)=O)CC1 C1(NC(CCC)=O)C(C)CN(C(C2(c3cccc(F)c3)CCC2)=O)CC1C CCCC(O)C(=O)NC(C)CC1CN(C(=O)CC2CCC2(C)C)C1 C1(CC)CCNC1C(=O)NC(C)CCCN C=CC(C)(C)CC(=O)N(C)CC1COCCN1C(=O)CC1COC(C)(C)C1 N1(CCCC(=O)N(CCNC(C2CCNC2=O)=O)CC)C(=O)CN(C)C1=O Cc1nc(NCC(C)(C2CC2)NC(c2csnn2)=O)ncc1Br N1(C(C2N(C)CCCC2)=O)CC2(CCN2C(c2ccccc2F)=O)C1 C1(CNC(c2ccncn2)=O)CC2CCC1N2C(=O)C=CCN1CCCCC1 c1(CC(=O)N(C)CCOC2CCCCO2)cccnc1C(F)(F)F N1(C(Cc2nc(C)sc2)=O)CC(NC(C2CCC3(CCCC3)C2)=O)C(C2CC2)C1 c1(C=O)cc2ccc(Cl)cc2o1.CC(C(=O)NCC)NC(=O)CC1C=CCC1 C1(C(=O)NC(CC(C)NC(C=NOC)=O)C)CCN(CC(C)C)CC1 C1(CC(N2CCC(C(CNC(C=NOC)=O)F)CC2)=O)CCc2ccccc2C1 C1(O)(C(C)C)CCCN(C(=O)N(C(C)(C)C)CCNC2CCCSC2)C1 Cc1cc(C(=O)NCC2(NC(c3ccc(N)cn3)=O)CCC2)cc2ccoc12 C1CCN(C(c2cc(C)n(C)c2C)=O)C1(C)C.C1(CCCC)(C(=O)NC)CCC1 C(C(C)(O)CC(=O)NCCC1(NC(=O)C(CO)N(C)C)CCC1)OC c1(C(N2CC3(C(NC(=O)COC4CCOC4)CC3)C2)=O)cnc2ccccc2n1 C1(NC(c2cnc(CC3CC3)s2)=O)CCC12CN(C(C1CC13CC3)=O)C2 N1(C(C(CO)NC=O)=O)CCC(C2CC2)(C)C1.c1(C=O)cccs1.C1CC1 C#CCC(CC(F)F)C(=O)N1CC(C)(C=O)C(C)(CO)C1.C(=O)(O)NC C(=O)(C(F)(F)C(F)(F)Cl)N1C2CC(NC(C)=O)(C2)C1 c1(C(=O)NCCC(C)NC(C=CC=CC)=O)cc(F)c(C=O)cc1F CC1(C)CC(NC(=O)C(=O)N)CCS1.C1CC(=O)N(C2CC2)C1c1ccccc1 C#Cc1ccc(Br)c(C(=O)NC2(C)CC2)c1.C(c1ccncc1C)=CC(=O)N C1(NC(c2ccc(C(C)=O)o2)=O)C2COCC1CN(C(=O)Cc1nocc1C)C2 c1(C(=O)NCCC(=O)NCC(CC)NC(=O)CC(C)C)ccccc1OC c1(C(=O)NC(C)(C)CNC(c2ccncc2)=O)cnc2cc[nH]c2c1 C(=O)(C1=CCOCC1)NCC1C(C)CN(C(c2c[nH]ccc2=N)=O)C1 CCCC(C)(C)C(=O)N(CCCNC(=O)CCc1cc(O)cc(C)c1)C1CC1 c1(C(=O)Nc2cc(Cl)ccn2)csc2c1CCN(Cc1ccc(O)cc1F)C2 C1(NC(CC(CC)SC)=O)CCCCCC1NC(c1cc(CCO)on1)=O CC1(NC(C2CCCC(F)(F)C2)=O)CCN(C(c2cc(C(F)(F)F)ns2)=O)CC1 c1(OC)ccc2c(c1)OCC(C(=O)NC1CCC1NC(C1COC1)=O)C2 C(CC(C)(C)NC(C1CCOC1C1CC1)=O)NC(CCN(C)CCO)=O c1(C(N2C(CC(N3CC(S(C)=O)C3)=O)CC(F)C2)=O)cn2ccccc2n1 CC(N=c1[nH]c(=NCc2ccco2)[nH]c2c1CSC2)C1CN(C)CCN1C C1(CC(N2CCCCC2)=O)CCCC(C)(C)O1.C1(C(=O)N)(SCC)CC1.C CC(CCCCN=c1[nH]cncc1Br)NC(=O)C#CC(C)(C)C N1(c2nnc(CCC)s2)CCC2CCC(C1)N2C(c1ccn2nncc2c1)=O CC1CN(C(=O)COc2ccccc2Cl)Cc2ccccc21 Cc1cn2[nH]c(=NCC(C(C)(C)C)NC(c3cnn4cc[nH]c34)=O)sc2n1 CCCCC(O)CCC(=O)N1CCC(C(C)(C)CNC(=O)CC2CC2(C)C)CC1 C(=O)(CCCC1CCC1)N(CC(=O)NCCNc1ccccn1)CCOC c1(C(=O)NC2CCC(C(=O)NCC(O)Cc3ccccc3)C2)cc[n+]([O-])cc1 N(C(=NCCS(=O)(=O)c1ccccc1)N1CCC(C)C1)CCN(C(C)C)C(C)C c1(C(=O)NCCCN(C(c2n[nH]cc2C2CCC2)=O)CC)scnc1C N1(C(=O)Cc2cnc(C(F)(F)F)s2)CC2CCN(C(c3ncccn3)=O)C2C1 c1(C(N(C2CCCN(Cc3ccc(C)c(C)c3)CC2)C)=O)cn2cccnc2n1 C1(NC(=O)C=Cc2nccs2)CCN(C(c2cn(CCCF)nn2)=O)C12CC2 C1(C(N2C3CN(C(C#CC(C)C)=O)C(C3)C2)=O)CCC2CCCCC2C1 C(C(=O)N(CCC(=O)N(C)C1CC1)CC)(C(C)C)OCC c1(OC)cnc(Cl)cc1C(=O)NC1CCN(C(c2ccc(C)cc2O)=O)C1 N1(C(CC(C(=O)OC)C)=O)CC(NC(c2cccc[n+]2[O-])=O)C(N=[N+]=[N-])C1 C(C(=O)NCCC)(C(C)C)N(CC)CC.c1(CCC(=O)N)ccc(=N)[nH]c1 CCC(CO)C(=O)N1CC(CO)(NC(=O)Cc2sc(SCC(C)C)nc2C)C1 C12(C(=O)NC3(CC)CCC3)CC(CN(C(c3ncnc(O)c3F)=O)C1)C2 C1(C(CNC(C2C(C)C2)=O)NC(=O)C(C)N(C)C)CCCCC1 C1(C(=O)NC2(CNC(c3cnoc3)=O)C(C)CCCC2)C2CCCCCCC12 c1(CN2CCC(F)(C(=O)NC(C)C#N)CC2)c[nH]c2nccc(Br)c12 C12(NC(c3ccc([N+](=O)[O-])o3)=O)CCC(CC1)N(C(C1CCCC(O)C1)=O)C2 CC1C(NC(=O)CC(O)CN(C)C)CCCN1C(=O)COC1CCOCC1 c1(CC=O)ccc2oc(C)nc2c1.S(=O)(=O)(CC(=O)N(C1CCCC1)C)NC.N c1(-c2cn(CC(=O)OCC)nn2)cccc2ccccc12.n12nc(C)nc1C2 N1(C(c2c(C)cco2)=O)CCN(C(C2C(F)(F)C23CCC3)=O)CC1CC1CC1 CCC(CC(=O)NC1CC(C)N(C(=O)C=CCOC2CCOCC2)C1)SC c1(C=O)nc[nH]c2nccc1-2.CC(C(=O)NCCCOCCO)NC.C1CC1 N1(C(C2CCN(C)C2)C(=O)NCC)CCN(C(C2CCCCC2)=O)CC1 c1(COC)ccc(NC(=O)NCC2(O)CCN(C)C2)cc1F Cc1ccc(F)cc1-n1nc(-c2nccs2)nc1C1CC1C c1(C(=O)NCCCN(C)C(c2cc3cnccc3[nH]2)=O)cc2c(Cl)cncc2o1 c1(C2CCN(c3n(CC)c(CC4CCS(=O)(=O)C4)nn3)CC2)ccccc1C#N CCCCC(O)CC(=O)NC(C1CC(NC(=O)CCCCOC)C1)C CC(C)CC(C(=O)Nc1cc(N2CCNC2=O)ccc1F)C(C)C C1(OC)CNCCC1(CO)OCc1cc(-c2ccccn2)nn1C N1(CC2N(C(Cn3cc(C=CC)nn3)=O)CCC2)CCn2nc(C#N)cc2C1 C1(C(N2CCC(N(C(C34CCC3CC4)=O)CC)C2)=O)CC(=O)N(C2CC2)C1 c1(OC)ccc2[nH]cc(CNCc3cccc(C(F)(F)F)c3C)c2c1 Cc1cc(C(=O)NCC(C)(C)C(N2CCCOCC2C)=O)nc(O)n1 C1(NC(CSCC(N)=O)=O)CN(C(c2cc(F)c(F)cc2N)=O)C2(CCC2)C1 C1(CC(C)C)(C(=O)NCC(C(F)F)c2ccccc2)CCNCC1 C1(NC(c2c(CC)nc[nH]2)=O)CCCCN(C(c2coc3ccccc23)=O)CC1 c1(NC(CCC#C)(C)c2nnnn2CCOC)c(C)cccc1C Cc1ncc(C(N2CCCN(C(=O)C=CC(C)C)CC2)=O)c(C)n1 c1(C(N2CC3C(NC(C4(C)CC5CC5C4)=O)C3C2)=O)c(F)cccc1Cl c1(CNc2nc(C)nc(N3CCC(N4CCCC4)C3)c2)cnc2ccsc2c1 Cc1cc(NCC(c2ccc(F)cc2)C)n2ncc(C)c2n1 C1(CNC(C2(CC=C)CC=CC2)=O)CCC(C)CN1C(c1ccnnc1S)=O CN1C(C)(C)C(C(=O)NCC23COC(C(F)(F)F)(C2)C3)CS1(=O)=O C#Cc1cccc(CC(=O)N(C(CC)CC(N2CCSCC(C)C2)=O)C)c1 C1(NC(C=C(CCC)C)=O)C(C)CCN(C(=O)C(C)CC(N)=O)C1C CC1CCN(C(c2cc(C(N)=O)cn2C)=O)CC1NC(C1CC(C(F)F)C1)=O N1(C(CC2C(C)C2)=O)CCCC(CNC(=O)CCc2cnc[nH]2)C1 N1(C(=O)CSc2cn[nH]c2)CCN(C(=O)CC2CCS(=O)(=O)C2)C(CCO)C1 C1CN(C(=O)CC2(C#N)CCC2)CC1(C)C.c1(OC)cc(CC(=O)N)ccn1.C CCC(C)CCCC(=O)NCC(CC(F)(F)F)NC(c1cc(SC)ccc1C)=O c1(C(=O)NCC(CC=C)NC(=O)C(C)CC(N)=O)ccc2cccc(F)c2n1 c1(C(N(CCNC(=O)CCCC2CC2)CC)=O)ccc(OC)c2cnccc12 C1(CNC(COCCCC)=O)CN(C(C2CN(C)C2)=O)C2(CCC2)C1 c1(C(=O)NCC2(F)CCCN(C(CCC(CC)C)=O)C2)c(C)nn2cccnc12 C(=O)(CC(C=C)CC)NC1CC(F)(CNC(CN2CCCC(CC)C2)=O)C1 C(C(C)C(C)C)NC(C1(C(C)(C)OC)CC1)=O.n1(CC=O)cnnc1O.N C1(C(N(CC(CN(C(C(c2ccncc2)C)=O)C)O)C)=O)COC(=O)C1 c1(C(N2CC3CC3C2)=O)cc2c(C)cc(C)cc2[nH]1.C(C)(C(O)C(=O)N)SC.C C(C)(CCC(=O)N(C1CCC1)CCOC)NC(C(C)OCCOC)=O C(CC)(CC)(CCO)NC(C1OCCN(C(Cn2ncc(CC)c2)=O)C1)=O Fc1ccc(C2CC2N(c2nnc(C(F)(F)C(F)F)s2)C2CCCC2)cc1 c1(COC)nc2n(n1)CCCC2NC(=O)NC1(C)C2CCCCC12 C=Cn1nccc1C(=O)NC1CCOC(C(=O)N(CC(CC)CC)CCC)C1 N1(C(c2c(OCCC)cccn2)=O)CCC2CN(C(=O)CC(F)(F)C(C)C)CC12 CC(=O)CC(C)(C)C(=O)NC1CCOC(C(N2CCC=C(Cl)C2)=O)C1 c1(C(N2C(CNC(Cc3c(C)cnn3C)=O)CCCC2)=O)nn(C)cc1[N+](=O)[O-] CC1CC(NC(=O)CN=S(C)(C)=O)CN(C(C2COCC2(C)C)=O)C1 C1(C(=O)NC(C2CCCCC2)CNC(C2(C#N)CC2)=O)CCCN1CC(F)F c1ccc(F)c(F)c1.C1(C(c2n(C(CC)C)nnn2)NC)CC(S(C)(=O)=O)C1 n1(CC(N2CC(O)(CNC(C(C)C(F)F)=O)C2)=O)ccc(=O)n(C)c1=O CC1(C)OOc2cc(-c3ccc(NS(=O)(=O)c4ccccc4F)nc3)ccc21 C1(C(N2CC(F)C2)=O)CCN(C2CCSC2)CC1.c1(CC)nnsc1C(=O)N.C n1(CC=C)ncc2c(O)nc(=NCCNC(=O)Cc3ccccc3CC)[nH]c12 C1(C(N2C(C=C)CC2)=O)CCC(C)N1C(=O)CCCN(C)C c1(N2C3CN(C(c4cc(OC)cc(Cl)n4)=O)C(C3)C2)ncnc2c1CCCC2 c1(CC=O)ccc2nn(C)cc2c1.C(C)(C)(C)NC(C=CC=CC)=O.N c1(C(=O)OCC)ccccc1.c1(C(=O)NCCCOCCN)ccco1 C1(NC(C2=C(C)CCC2)=O)CC1C1CCCN(C(c2cc(CC(C)C)[nH]n2)=O)C1 C1(NC(CCCSC)=O)CC2CCCC(C1)N2C(c1ccn2[nH]c(=N)nc2c1)=O C1(CNC(C2CC(SC)C2)=O)COCCN1C(c1cnoc1C)=O C1(NC(C2CCOC2)=O)(CO)CCCN(C(c2ccnc(OCCO)c2)=O)C1 N1(C(C(C)C)=O)CCC(CO)C(NC(c2ncccc2OCC(F)(F)F)=O)C1 CCCCCCCCC(=O)N1CCCC(CNC(=O)CCCN2CCOC2=O)C1 c1(C(=O)NC2CCCN(C(C=C(CCC)C)=O)CC2F)ccc2c(c1C)CCC2 N1(C(C2(OC)CC2)=O)CC(C)C(NC(c2ccc3ncsc3c2)=O)C(C)C1 N1(C(C2(C)CN(C(=O)Cc3ccc(F)c(Cl)c3)C2)=O)C2CCCC1COC2 CC(C)CCC.C(C(F)(F)F)C1(C=O)CC1.C(=O)CN(CCN(C)C)C.N C1(C(N(C)CCOC2CC2)=O)CCCN(C(C2CC(O)C2)=O)CC1 c1(C(=O)NCC(CNC(C2CCCN(C)C2)=O)OC)ccc(Br)c(O)n1 N1(C(C2OCCN(C)C2)=O)CC(N)CC12CCCCCC2 n1(CCC)nc(C)c(C(=O)NC2COCC2)c1C.C1(CC(=O)N)CCOC1(C)C N1(C(=O)NC(CC)C(C)(C)O)C2CCCC1CC1(CC1)C2 N1(C(C2(C)ON=C(C)C2)=O)CCC(C)C(O)C1.C(=O)(C(C)(C)N1CCCCC1)N N1(C(N(C2CCOC2)C)=O)CC=C(c2c[nH]c3cnccc23)CC1 N#Cc1cnc(C(N2CCC(NC(=O)CC3CCC3(F)F)C(F)C2)=O)c(Cl)c1 c1(OC)ccc(C(=O)NC2CN(C(=O)CC3CC(C(F)F)C3)C2)cn1 c1(C(=O)NCC2N(C(C3NC(=O)OCC3)=O)CC2)cc2cc([N+](=O)[O-])ccc2[nH]1 N1(C(c2cc(CCNC(=O)CC(Cl)Cl)on2)=O)CC2C=CC1CC2 c1(C2CCN(C(C3(C)SCCCS3)=O)CC2)nc2ccccc2o1 CC1(C(=O)N(C)C)CCCN(C(=O)CCn2cc(-c3cncc(N)c3)nn2)C1 N1(C(C2CCC(C)N2C(=O)CCc2ccccc2)=O)CCCC(C)(CN(C)C)C1 C(=O)(C(CCC(C)C)NC(=O)C(C)OC(C)=O)NC(C=C)C1CCC1 C1(C(=O)NCC(C)N(C)C(c2ccc(-n3ccnc3S)cc2)=O)CCOC1(C)C CCCC(C(C)CC)N1c2nnnn21.CCCS(C)(=O)=O.C1(C)CC1 C(CN=c1[nH]c2c(c(=NC3CCN(C4CCCC4)C3)[nH]1)CCC2)=CC C1(C(=O)NCCCCCN(C)C(c2c(Cl)cnn2C)=O)CC12CCCCC2 c1(NC(CC2CCN(Cc3ccc(C)[nH]3)C2)=O)cccc(C2(C)CC2)c1 c1(C(=O)NC(C(C)NC(c2cc(Cl)c(Cl)n2C)=O)C)[nH]nc2ncccc12 O=CN1CCN(C(C2CC2NC(=O)Cc2ccc(Cl)cc2)=O)CC1 C1(CC)CCCN(CC(=O)N)C1.C12CC(C1)N(C(C1CCN(C(C)C)CC1)=O)C2 CCCCC(CCC)NC(C1C=CCN(C(=O)CCc2nccs2)C1)=O n1(CCNC(=O)NC(C2CSC2)C)cncn1 N1(C(C(CC)NC(C)=O)=O)CCNC(C(N2CCN(CC)CC2)=O)C1.C(C)=O c1(CC(=O)NC2CCCC(NC(C3(CC)CCC3)=O)C2)nccc2ccccc12 c1(CC(=O)NC2C(NC(CSC)=O)COC2)c[nH]c2cccnc12 n1(CC)cc2ccc(C(=O)OCC(N3CC(=O)N(C)CC3C)=O)cc2n1 C(N=c1cccc(S(=O)(=O)N(C)CCC(CCO)C(C)C)[nH]1)c1n(CC)ccn1 CS(=O)CCC(=O)NCC1CC(NC(c2nccnc2N)=O)C1 c1(OC)cc(C(=O)NC(C2CCN(C(c3ocnc3C(C)C)=O)C2)C)sc1Cl c1(CC(=O)NCC2CCN(C(c3cnn[nH]3)=O)CC2O)cc(Cl)cc(Cl)c1 N1(C(c2c(C(C)C)c[nH]n2)=O)CCC2OCCN(C(=O)C(C)CS(C)(=O)=O)C2C1 C(CC(C)C)(C(=O)N1CCCC1C(C)NC(c1c[nH]nc1C(F)F)=O)OC c1(N2CC(CCCCCNC(=O)CCN3CCOCC3)C2)ncc2c(n1)COC2 N1(C(c2c(C)n(C)nc2)=O)CC2OCCN(C(C3CC4CCC3CC4)=O)C2C1 c1(C(N2CCC(CCNC(C3(C)CC3)=O)C2)=O)nc(Cl)c(Cl)c(N)c1Cl C12(C(N3CCC(OC)(C)C3)=O)CCN(CC1)CC2.c1(C=O)occc1C(C)C c1(C(=O)NCC2CN(C(C=C(CC)CC)=O)C2)oc2ccccc2c1OC C(C(C(=O)NCC1CCCO1)N1CCC=C(Br)C1)(C1CCC1)OC C1(C(=O)NCC(C(C)C)NC(C(COCC)C)=O)CCc2c[nH]nc2C1C C1CC2OC1C1CC21.CC(C)CC(=O)N(CC(=O)NCC1(C=O)CCC1)C.N C1(CNC(C(CC=C)(C)C)=O)CC2(CCC2)CN1C(=O)CC1CC(F)(F)C1 C(=O)(C(C)CC(F)F)N1CC(C)C(CNC(c2ccn(C3CCCC3)n2)=O)C1 C12(CCNC(c3ccc(OC)cn3)=O)CCC1CN(C(c1cc[nH]c1)=O)C2 C1(=CCNC(c2cc(=O)cc[nH]2)=O)CCN(C(c2ccc(CO)nc2)=O)CC1 N1(C(CNC(CCN(C(C(C)C2CCC2)=O)C)=O)=O)CCN(C)CC1 c1(C(N(C)CC2(O)CN(C(C3CC4(CCOC4)C3)=O)C2)=O)cccc2ccsc12 C1(NC(C(CC)OCC)=O)C2CC(O)C1N(C(c1cccc(C)c1Cl)=O)C2 Cc1ccc(NC(C2CCC(C)CN2C(C2CCSCC2)=O)=O)c(C)c1O C1(NC(Cn2cc(C(C)O)nn2)=O)CCCC12CCN(C(=O)CCC(C)O)CC2 C1(F)CCN(C(C23CCC(CO2)C3)=O)CC1.C1(C(=O)N)CC(=O)C12CCC2.C N1(CCNC(C)=O)CC(C)OCC1C.N12CCC(CC1)c1nncn1SCC2=O c1(CCC(=O)N)ccccc1F.CC(CNC(C1CC(OC2CC2)C1)=O)CO N1(C(C(C2CC2)OCC)=O)CCC(C(=O)NC(CO)CCO)CC1 CC1CCc2ncc(C(=O)NCCc3nc4cc(C(F)(F)F)ccc4s3)n2C1 C12(CC(=O)NC3CCN(C(c4nc(CC)oc4)=O)C3)COC(C)(C1)C2 Cc1cc(C(=O)NCC)c(C)cn1.c1(CC(=O)N(CC)C)cc(F)ccc1C.O C1(CC(=O)NC2CCC(NC(CC(C)=C(C)C)=O)CC2)CN2CCN1CC2 CC1C(NC(=O)C(C)c2cccs2)CCCN1C(=O)CC(F)F n1(CC)c(C(N2CCCC2C(=O)NCCC(C)CO)=O)cnc1O c1(C=O)ccc(C2CC2)cc1F.CC(C)C(C(=O)N1CCC1)NS(C)(=O)=O.N C1(C2(O)CCOCC2)(CN2CCCC(Cn3c(C)nc(C)n3)C2)CCC1 CC(=O)CCC(=O)NC(Cc1cn[nH]c1)C(=O)NC(C)C(C)(C)CN(C)C N1(C(c2c(C)nn[nH]2)C(=O)NCC2CCCO2)CC2CCCCCCC12 Cc1ccc(NCC2=CC(=O)OC2)c(Br)c1 c1(C(N2CCCC(CC=C)C2)=O)c[nH]nc1S(N)(=O)=O.C(=O)(CC(C)C1CC1)N c1(CSC)cc(C(N2CCC(C)(CNC(=O)CC(C)C(C)C)C2)=O)ccc1F c1(CNC(C=C(C)c2ccco2)=O)cc2n(n1)CCN(C(=O)C=CS(C)=O)C2 c1(OC)cc(CC(N2CCCC(NC(c3ccncc3I)=O)C2)=O)ccc1O C1(O)(CN(C(c2c(C)cno2)=O)C)CCCN(C(=O)C=Cc2cnc[nH]2)C1 c1(CN2C(C)(C(=O)Nc3ccc(Cl)nc3)CCC2)cc(F)c(Cl)cc1O C1(CC=C)(NC(C2CC2c2ccccc2C)=O)CCN(C(C2(F)CCC2)=O)CC1 C1(CCn2cc(CCCOC)nn2)CCCN(C(C2CCC2C(F)F)=O)CC1 c1(C(N2CCC(C(F)(F)F)C2)C(=O)NC(CC)C)cc(F)c(F)c(OC)c1F CC(C)CC(CNC(=O)NC1CC(CS)C1)N1CCOCC1 Cc1cccn2nc(C(=O)NCC3CN(C(=O)CCC4CCOC4)CCO3)cc12 C1(N(C(c2cc(C)c[nH]2)=O)CC)CCCN(C(C2CCCN2C)=O)C1 C1(NC(CCc2nc(=N)[nH][nH]2)=O)CN(CC(N2CCOCC2)=O)CC12CC2 C1(CC)CCCN(CC(=O)N(C)CC2(NC(=O)C(C(C)C)SC)CC2)C1 N1(CCCCOc2ccc(C)cc2)CC(C(=O)OC(C)(C)C)CC(C)C1 c1(C(=O)NC2C(NC(Cc3cccc(C)c3)=O)CCOC2)cscc1S(C)(=O)=O c1(C(N2C(C)CC(CNC(C=CCCC)=O)C2)=O)cccc(OC)c1N C(=O)(C(C)(C)CCC#N)N1C2CC(CNC(C3(C#C)CCCC3)=O)C1CC2 c1(CC(=O)NCC2C(NC(c3cnn(C)c3Cl)=O)CCC2)cccc2cn[nH]c12 C1(c2cn(CC3CC(CC(=O)OCC)C3)nn2)CCC(=O)CC1 N1(C(c2sc(Br)cc2Cl)C(=O)NCCC)CC(C)(C)CC1CC(=O)OC C1(C(=O)OC)CN(S(=O)(=O)Cc2c(C(=O)O)cnn2C)CC12CC2 C(c1ccccn1)=C(C)C(=O)NC(CNC(=O)Cn1ccnc1C)CO N1(C(C(CO)NC(=O)COCC(F)F)=O)CCC(C2(O)CC2)CC1 C(C(CC(C)C)NC(C1(CO)CCC1)=O)NC(C1(C=O)C(=C)CC1)=O.C CN=C(NCCC(=O)OC(C)(C)C)NC1CCCCC1 S(=O)(=O)(c1cnc(Cl)nc1)N1CC(NC(C2CC(=O)NC2)=O)C(O)C1 C1(NC(C(C)N(CC(F)(F)F)C)=O)CC2(C1)CC2.c1(CC(=O)N)cnoc1 N1(CCN(C2CC2)CC)C2CCC1CC(C1CCO1)C2 C12(CNC(CCC(C)OC)=O)CCC(CC1)C(C)(C)O2 CC(C)CCCC(C)C(=O)N1CCC(F)(C(N2CCC3(CNC(=O)N3)C2)=O)C1 c1(C(N2C3(CN(C(c4cnco4)=O)C3)CCCC2)=O)cc(F)cc2cnccc12 C1(CNC(C(C2CC2)SC)=O)CC2COCC2N1C(=O)Cc1cnn(C)c1 C(=O)(C(=O)C(C)(C)CC)NCC(=O)NCC(=O)NCC(CC)CC CCCC(O)CC(=O)NC1CN(C(c2cnc(O)n2C)=O)CC1C(F)F CCC(CNC(C1(NC(C2CC2C(N)=O)=O)CCN(C)C1)=O)C(C)C CCC(CC)CC(F)C(=O)NCC1CCCN1C(c1coc(SC)c1)=O C(=O)(CCCCCn1cnnn1)NC1CN(C(COc2cn(C)nc2)=O)C2C1C2 C1(CNC(CC=CC=C)=O)CCN(C(c2cnc(Cl)c(Cl)c2)=O)C1(C)C CCCCCC(O)C(=O)NC1CC2CCC1(NC(=O)CN1OC(C)(C)CC1=O)C2 C(C(C)(C)CNC(C1CCC2CC12)=O)C1CN(C(CC=C)=O)C1 C1(CCCN(CC(CC)OC(F)F)C(=O)OC(C)(C)C)CCCC1(C)C c1(Cc2c(CNC(N(C(C)S(C)(=O)=O)C)=O)cccc2)cccc2cc[nH]c12 C1(c2cn(CC3CCOCC3)nn2)(NC(C2CCCN2C2CC2)=O)CCCOC1 CCCCCC(O)C(=O)N1CCCC(C(=O)NCC(Cl)C(C)(F)F)C1 N1(C(c2cn(C)nc2O)=O)CCCC2(C1)CN(C(=O)C(C)(C)F)CCO2 CC1CC(C(=O)Nc2cccc(C3CN(CC(=O)NC(N)=O)C3)c2)CCS1 C(c1ccc(F)c(Cl)c1)=CC(N1CC(CCNC(C2(CC)CC2)=O)C1)=O N1(C(C2CCN(C(CC)=O)C2)=O)CCOC2(C1)CN(C(C1(O)CC(C)(C)C1)=O)C2 c1(C(C)=O)ncc(-c2cn(CC3C=CCN3C(=O)CC3CC(C)=NO3)nn2)o1 c1(CCC(=O)NC2CCC(NC(c3n(CC)c(O)nc3)=O)C2)ccc(F)cc1F C(CC(=O)NC(C)(C)CNC(=O)CC(C)(C)C)(C1=CCCC1)OCC.S CN1CCCC(F)(C(=O)NC2CC(CC)C2)C1.C(=O)(CCC)N.[SH](C)(=O)=O C1(C(N(CCCCN(C(C(C)c2ccsc2)=O)C)C)=O)CC(F)C(=O)N1 CC1CCCCN1C(=O)CCNC1CCN(CC(=O)Nc2cccc(F)c2)CC1 C#CC(C(=O)Nc1ccccc1Cc1nn[nH]n1)C(C)C N1(C(C)=O)CS(=O)(=O)CC1C(=O)NC(C1CN(C(c2sccc2C)=O)C1)C N1(C(CCOCC)=O)CCN2C(=O)C(NC(=O)CCN3CCN(C)CC3)CC2C1 C(=O)(C1=NNC(=O)C1)NCCOCC(=O)NC(Cc1ccco1)CO C1(OC(=O)C(c2ccccc2Cl)F)CCC2CC1OC2=O c1(C(=O)N)ccn2nccc2c1.C1(CC=C)CCN(C(C2C3(CC3)C23CC3)=O)C1 O=C(C1=CCSC1)NCC(C1CCN(C(=O)CCOCc2ccccc2)CC1)F C(=O)(CC(C)C(=O)OC)NCC(C(=O)NC(C#C)(C)C)O C1(NC(c2nc(C(C)C)sc2)=O)CCCCC12CCN(C(=O)C(F)(F)C(F)F)C2 Cc1cn2c(CC(=O)NCCCCCNC(=O)CC(=O)NC3CC3)csc2n1 N1(C(CC(C)CN(C)C)=O)CC2(CCCCN2C(C2CC=CCC2)=O)C1 C1(O)(C(=O)NCC(CNC(CC(C)c2ccco2)=O)F)CCCCCC1 C1(NC(COCC)=O)CN(C(c2ccc(N3CCCCC3)cc2)=O)C2CC12 c1(C(=O)NC2CC3(CN(c4ncnc(C)c4Br)C3)C2)cccc2c1OC(F)(F)O2 C12(C(N(C3CCN(C(=O)C=CSC)C3)CC)=O)CCCCC(F)(C1)C2 n1(CC)nc(C)c(C(=O)NCC(C)C(C)C)c1Cl.C(=O)(CC(C)n1ccnc1)N CC1(C)CCN(C(C2(C)CC=CCC2)=O)CC1CNC(C1(C)C=CCCC1)=O Cc1sc(=O)n(CC(=O)NCC2CC3CCC2N3C(c2c(Cl)cnn2C)=O)c1C C1(C(=O)NCC)CCNCCC1Nc1nc(C)c(CCF)s1 C1(CNC(c2cc(C)ncc2)=O)CC2(CC2)CN1C(c1ncccc1N)=O Cc1ccn(C(C)C(=O)N(C)CC2CCCN2C(=O)Cc2csnn2)n1 c1(C(=O)OCc2ccc(F)c(F)c2F)cccc2c(Br)cccc12 c1(C(=O)NC2C(C)(C)C(CNC(c3csc(Cl)c3)=O)C2)ccn2ccnc2c1 C(C)(C)(C(C)C)NC(C(CNC(C1(COCC)CC1)=O)OC)=O.S C=CC(C)(O)C(=O)N(C)CCOCCN(C(=O)C(O)C1CCC1)C c1(CC)cnc(C(=O)NC(C2CCCN(C(=O)C(F)(F)CC3CC3)C2)C)nc1 C(C(C(=O)NCC(C1CCCCC1)NC(=O)CC1CCCC1OC)OC)OC c1(C(N2CC(NC(C(CSC)OC)=O)C(C)CC2)=O)cc2ccncc2c(O)n1 n1(CC=O)nc(C)cc1C(F)F.c1(CC)sccc1C(=O)NC.C1CC1 C1(C)(NC(c2sccc2Br)C)CCCCC1C(=O)O CCC(CC)C(C(=O)N(C(C)C(=O)N(C)C(c1ccncc1)C)C1CC1)OC Cc1c(C(=O)NC(C)(CNC(c2ccc(N(C)C)cc2)=O)CO)cccc1Cl NS(=O)(=O)CCCCCCN=c1cccc(S(=O)(=O)N2CC3CC2CS3)[nH]1 c1(Cc2nnnn2C2CC(F)(F)C2)csc(C2CC2)c1.C(C)(C)C1CC1.C Cc1noc2nc(C(=O)NCC3CN(C(=O)C=Cc4cocn4)CC3C)ccc12 c1(C(=O)NCCCN(C(=O)C(F)OC(F)(F)F)C)ccc(C2CCCOC2)cc1 S(=O)(=O)(c1cccc2scnc12)N1CC2(CC(C(N3CC4CCC(C3)O4)=O)C2)C1 c1(C=O)cccc(-c2ccccc2)n1.C1(NC(C=CC=CC)=O)CCCC1.C C1(CC)CC(O)CCN1C(=O)CC1CC(NC(=O)C=C(C)COC)C1 CCC(CC)CC(F)C(=O)NC12CCC(C(=O)NC3C4CCCC34)(CC1)C2 N1(C(C(=O)N(C(CNC(C=C(C)C)=O)C)C)C)CCP(C)(=O)CC1 c1(C(=O)NCC2(C)CCCN2C(C2CCCCC(=O)N2)=O)c(O)cccc1Cl CCCC(CC)CCC(=O)N1CCOCCC1C(=O)NC1CC1C(F)(F)F CC1C(NC(=O)C(=O)N)CC2CCC1N2C(c1ccn(CC#N)n1)=O.CC(F)F N1(C(c2cnc(C(C)C)s2)=O)CC(O)CC1CNC(C1CCCC1(C)C)=O n1(CCNC(CSCC#C)=O)ccc(C(=O)NC(COC)CCO)c1 C1(NC(C(CCOC)C)=O)CN(C(=O)C2=CCS(=O)(=O)C2)C2(CCCCCC2)C1 C(CCF)(C(=O)NCC1NC(=O)NC1=O)NC(c1c(CC)con1)=O c1(C(=O)NC(C)CNC(C2CCC2(F)F)=O)ccnc2c(C(N)=O)cnn12 N1(C(c2nn(C)c(Cl)c2)=O)CC(C)(C)OCC1CNC(c1csnc1Cl)=O Cc1ncc(CCC(=O)N(C(C)CCNC(C2(C#N)CCOC2)=O)C)c(O)n1 c12ccc(Cl)cc1[nH]c(=O)[nH]2.c1(C(COC)CCO)ccc(C(C)(C)C)cc1 C(=O)(N1CCC(C(=O)NCc2ccc(C)nc2)O1)c1c(SC)csc1 C12(NC(COC)=O)CCCCC1N(C(=O)C(C)SC)CC2.Cc1cc(C)cc(C)c1 CC1CC(N=c2ccnc(C(C)(C)C)[nH]2)CN1C(c1ccnc2ccccc12)=O N1(C(CCCCCOCC)=O)CCC(C2CCN(C(=O)C(C)(C#N)CC)CC2)C1 N1(C(Cn2nc(C)oc2=O)=O)CCCOC(CNC(C23CC=CC(C2)OC3)=O)C1 C1(C=O)CCC(=O)N(C)C1.C(=O)(CCCN(C)C)N.C1(C(C)OC)CCCC1 CC1(N(CCCO)C(c2cc(C(F)(F)F)ncc2F)=O)CC2(CCC2)C1 C(CCNC(C1(C)CSC1)=O)(C(=O)NC1CCC=CCC1)OC N1(C(Cc2c(C)cco2)=O)CCN(CCNC(=O)N(C)C)C(c2nn[nH]n2)C1 C(N=c1nc2c(cnn2C(C)C)c(N2CCC(C3CC3)CC2)[nH]1)c1cncc(C)c1 C1(O)(CN(C(C(c2ccco2)NC(c2nc(CC)sc2)=O)=O)C)CCCCC1 CCCC(C)(C)CC(=O)NCCCCC(C)NC(=O)C=CCN1CCOCC1 Cc1c(C(=O)N)cc(C2CC2)n1C.C1(C=O)C(C)(C)C1(F)F.C1(CC)CC1 c1(CC)cccc(CC)c1CNc1cc(NC2CCOC(C)(C)C2)ncn1 C1(C(=O)N)C(C2CC2)CCN1C(=O)Cc1ccsc1.c1scnc1C1CC1.C C1(C(N2C(CN(C(C(CSC)(C)C)=O)C)COCC2)=O)CCCC(C)(C)O1 C12(NC(c3cccs3)=O)CC1CN(C(c1ccc(CO)o1)=O)C2.CC(F)(F)F C12(C(N3CC(CC(C)NC(CC(C)OC)=O)C3)=O)CC(C)(C1)OC2(C)C C1(NC(COC2CN(C(C(CSC)C3CCC3)=O)C2)=O)CCC2(CCC2)O1 C1(C(N2CCC(N(C(=O)C=CS(C)=O)CCO)C2)=O)(OC)CCSCC1 c1(C(=O)NC2CCC(CC(=O)NCC(CC)(C)CO)CC2)nccc(C)c1F C1(C)(CNC(c2cnn(C)n2)=O)CN(C(C2CC2C2CC2)=O)C(C)(C)C1 CN1CCC(C)(C(=O)NCCCCN2CCCN(C(c3cnsc3)=O)CC2)C1=O c1(C(N(C2(c3ccccc3)CNC2)Cc2ccn(C)n2)=O)ccn2ncnc2c1 C(N=c1ncc(C(=O)C(F)F)c[nH]1)C12OCC(NC(=O)CSC(F)(F)F)(C1)C2 C1(C(C)C)C(C(C)C)CN1C(c1ccc(C)o1)=O.c1(CCC=O)ccnn1C.N C1(CCC)CCCN(C(=O)CC(C(F)F)NC(=O)C(CC)N(C)C)CC1 N1(C(CCCOC)=O)CCC(C)(C)C1CC(=O)NC1(CCO)CCOC1 N1(C(c2snc(C)c2N)=O)CC2(CCC(NC(C3CC(O)C(F)C3)=O)CC2)C1 C(=O)(CC(C)(C)CNC)N(c1ccc(CNC(c2cccnn2)=O)cc1)C CC1CN(C(=O)CCC2CCCN(C(=O)C(=O)C3CCCC3)C2)C(C)(C)C1 c1(C(=O)N)c(C)n[nH]c1C.Cc1ccn(C(C)C(N2CC(C(N)=O)(C)C2)=O)n1 CC(C)C(C#N)C(=O)N1CC2(CCN2C(c2cc(-c3cccs3)[nH]n2)=O)C1 Cc1cc(Br)ccc1CN1CC(C)(CC(=O)NCc2occc2Br)C1 N1(C(c2c(C)cn(C)c2)=O)CC2(CCCC2)C1C(=O)NC1CCCC1(F)F C1(NC(Cc2c(C)con2)=O)CCN(c2nnc(C3CC3)o2)CC12CCC2 Cc1ccc2oc(-c3cnc(CC(=O)Nc4c(C)nc(Cl)nc4Cl)nc3)cc2c1 C1(C(=O)NC(CCN(C(c2c(C)ccn2C)=O)C)C(C)C)CCCN2CCCC12 C=CC(C)(O)C(=O)N1CCC(c2cn(Cc3cc(C)cnn3)nn2)C1 C(CCCCNC(=O)Cc1ccon1)NC(C1C(C(C)C)C1)=O C1(NC(COC(C)=O)=O)CN(C(=O)CCc2ncc(F)cn2)CC1C1CC1 CC(C)CCCN=c1[nH]c(N(C)CCN2CCN(C)CC2)nc2c(F)cccc12 Cc1nn(C)cc1CC(=O)NCC1(NC(=O)CCN2CCCCCC2)CC1 CC1CC(NC(=O)COCCF)CN1C(c1cncc(-n2ccnn2)c1)=O c1(CCC=O)ccc(F)cc1F.S(=O)(=O)(CC=O)NCC.C1(CC)CCC1.N N1(C(C(CC2CC2)OC)=O)CCC(C)(C)C1C(=O)N.C1CC2(CCC2O)C1 N1(C(CC2ON=C(CC)C2)=O)CC2(CCCC2NC(c2cnc(SC)s2)=O)C1 c1(C(=O)NCC(CCCC)NC(c2c(C#C)c[nH]n2)=O)ccc([N+](=O)[O-])s1 CC1CCSCCN1C(=O)CC(C1CCCC1)NC(=O)C#CC1CC1 Cc1ccc2c(c1)CC(C(N1CCC(CNC(c3snnc3C)=O)C1)=O)S2 N1(C(C2(C#C)CC2)=O)CC2(CC(CC(=O)NC(CO)CCC=C)C2)C1 N1(C(C2(C(=O)NC)CC2)=O)CC(C)C(C)C1.C1(C=O)CCC(F)(F)CC1.C C=CCC(C)(C)C(=O)NCC1(F)CCN(C(c2cc(O)cc(F)c2)=O)C1 c1(OC)cc(C(N2CC(CNC(=O)C(C)(C3(C)CC3)OC)C2)=O)ccn1 c1(C(=O)NC2C(C)CN(C(c3ccc(C(F)F)o3)=O)C2)nccn2nccc12 C1(CNC(CC2(C)CC2)=O)CN(C(=O)C=Cc2ncc[nH]2)CCC12CCC2 C1(NC(=O)CC2CCCN(C(C3(C(F)(F)F)CC3)=O)C2)C2CCCC1CC2 c1(CC(N2C(CNC(c3scc(C)c3Cl)=O)CC2)=O)c[nH]c2ncccc12 N1(C(C(C)S(N)(=O)=O)=O)CC2CCC(N(C(=O)CC3(N(C)C)CCC3)C)C2C1 S(=O)(=O)(c1nc(N2CCCC(CCN(C)C)C2)ccc1Br)NCCC(=O)N(C)C CC(C)(C(=O)NC1CC(C)C1)OCc1ccccc1.C1(O)(C=O)CCOC1 C1(CNC(C(C(C)O)C)=O)CCC2CN(C(c3ccn4c3CCCC4)=O)CC12 CN1CCC(C(N2CCC(C)(NC(C34COCC3C4)=O)C2)=O)(C(F)F)CC1 CCCC(CC(C)C)C(=O)NCC1(C(=O)NCC)CCCCC1.C1CC1(F)F.O c1(C(=O)Nc2ccc3sccc3c2)cccc(O)c1[N+](=O)[O-] C1(F)(C(=O)NCCc2cc(F)ccc2Br)CS(=O)(=O)CC12CCC2 C(=O)(CC(C)CC(=O)N1CCC(C)C1C(N1CC(O)(C2CC2)C1)=O)OC Cc1[nH]c2ccc(C(=O)N(C)CCNC(c3c(Cl)ccc(F)c3N)=O)cc2c1C c1(C(=O)Nc2n(C)nnc2)n[nH]c2c1CCN(C(c1cnc(Cl)s1)=O)C2 Cc1cc(C#N)ccc1C(=O)NCCNC(c1c(C)cc(C)oc1=O)=O CCCCCC(CC)C(=O)NC1(C)CC(NC(c2noc3c2COCC3)=O)C1 c1(-n2c(C)c(C(=O)NC3(c4cccc(Br)c4)CCC3)cn2)ccc(F)c(F)c1 CCC(CCCC(=O)N(C1(C(=O)OC)CC1)C)NC(=O)Cc1ccsn1 CC(CNC(c1ccoc1)=O)CNC(=O)C(C)C1CC1 C1(NC(C2(C)CC(F)C2)=O)CC2CC1N(C(C13CC(C)(CCO1)C3)=O)C2 c1(C(=O)NCC2CC(F)(CNC(CCCC=C)=O)C2)cc2c(C)n[nH]c2cn1 Cc1cc(-c2cn(C3(C(=O)NCCc4cc(Br)cs4)CC3)nn2)ccc1Cl c1(OCC(=O)NC(C(C)NC(=O)C=Cc2cccs2)C)cccc(Br)c1F c1(CC)nnc2c(C(=O)NC(C)C(C)C)cccn12.C1(Cl)(C=O)CC1(F)F.N c1(CC(N2CCC(OC)(CNC(=O)CC(O)CS)C2)=O)ccc2c[nH]nc2c1 Cc1c(C(=O)NC2CC3(C2)CC(NCc2cc(F)ccc2Br)C3)cccc1Cl c1(NC(CC2CCC(C#N)C2)=O)ccc2c(c1)CCCN2 C(N=c1[nH]c2c(c(=NC(C)C(C)N3CCCC3)[nH]1)CCC2)NC(C(C)C)=O C1(C(=O)NC(C(C)(C)NC(Cn2ncc(C)c2)=O)C)CCC2CC2CC1 C(=O)(C(CNC(=O)C=C1CCCCC1)N(C)C)NCC(n1cccn1)C CCCC(C)(CC)C(=O)NC1CN(C(c2ccc(C(N)=O)c(Cl)c2)=O)CC1(C)C c1(C(=O)NC2CC(CNC(C(CCSC)O)=O)C(O)C2)ccnc(Cl)c1OC C#Cc1ccc(Cl)c(C(N2CCC(C(C)NC(=O)C(C)(C)C#C)C2)=O)c1 Cc1cccc(NC(=O)C=O)c1.C1(C(N(CCC)C2CC2)=O)CCCN1C=O.N c1(C(N2CC3C(NC(=O)COCC4CCOC4)C3C2)=O)ccc2nsnc2c1 N1(C(C2N(C(C(C(C)C)OC)=O)CCC(C)(C)C2)=O)CCCCCCCCC1 C(=O)(CCC(F)(F)CN=[N+]=[N-])NC(C(=O)OC)Cc1cc(F)cc(F)c1 C(=O)(CCCC(F)(F)CO)NC1C(CNC(c2cnc(OC)nc2C)=O)C1 CS(C)(=O)=Nc1nc(C(=O)NC)cs1.C1CCCN(C(C2CC(F)(F)C2)=O)C1 CC1OCCN(C(c2cncn(C)c2=O)=O)C1C(=O)NCC(F)F N1(C(C2CCN(CC)CC2)=O)CCC2CC2(C(N2CC(O)C(O)C2CO)=O)CC1 C1(C(N(C)Cc2cccc(C)n2)=O)CC2CN(C(=O)Cn3nnnc3C)CC2C1 C1(CNC(Cc2c(C)nsc2)=O)(Cn2cc(C3CCCCO3)nn2)CC12CCC2 Cc1nc(C2CCOCC2)ncc1C(=O)NCC1CCCN1C(=O)C=CCO C1(C(=O)NC2C(C(N3CCN(CCO)CC3)=O)OCC2)CC2COCC2C1 c1(C(=O)NC(C(=O)NCc2c(OC)nsc2)Cn2cccn2)ncncc1N N1(C(CCC(C)(F)F)=O)CCC2(C1)CN(C(c1ccnn1C(F)F)=O)CCO2 C1(SCCN(C2CCC(C)CC2)CC)CC2(CCOC2)CO1 C(=O)(C(C(=O)OC(C)(C)C)C(C)(C)C)N1C(C)CCN(C(=O)C=CBr)CC1 N1(C(CN2C(C)CCC2)=O)CCC(CNC(c2cc([N+](=O)[O-])n[nH]2)=O)C1(C)C C1(O)(NC(C2C=CCN(C(=O)CCN3CCCC3)C2)=O)CCCCCC1 N1(C(c2[nH]c(=N)sc2)=O)CCCC(F)(C(=O)NCC2(O)CC(O)C2)C1 N1(c2cc(CC)nc(C)n2)CC(NC(C2CC(=O)NC(=O)N2)=O)CC2(CC2)C1 c1(C(N2C(C)CCC(NC(c3ccc(C4CC4)s3)=O)C2)=O)cc(F)c(O)c(Cl)c1 C1(C=O)CN(C(c2cc(C(C)=O)c[nH]2)=O)C2(CCC2)C1.C(=O)(CC)O.CC c1(COc2cc(C(C(=O)NC)N(C3CCOC3)CC)sn2)cccc(F)c1 Cc1c(C(=O)NCC(C2CCCC2)NC(=O)C(C)(C)F)oc2c1C(=O)CCC2 c1(C(=O)NC2C(NC(CN(C)CC)=O)C2)cn2c(n1)CCCC2C N1(C(c2c(CC)nco2)=O)CCCC2(CCN(C(C3(OC)CCC3)=O)C2)C1 C1(C)(C(=O)NCC(CC(C)C)NC(c2cn(C)cn2)=O)Cc2ccccc2N1 C(=O)(C(F)(F)C(F)(F)F)N1CCC(NC(c2cc(C(F)(F)F)n[nH]2)=O)C1 N1(c2nc(C)nc(O)c2C)CC2(C)CN(C(=O)C=Cc3cccnc3)CC2(C)C1 C1(CNC(c2c(C)nc(C)[nH]2)=O)CCN(C(=O)CN2CC=CC2)C12CCC2 N1(C(C(COC)(C)O)=O)C2CCC1CC(C)C2.n1(CC=O)nc(C)c(C)c1C.N c1(C(=O)N)cc(Br)c(F)cc1O.C1(NC(C2(CC)CC2)=O)CC(F)(C)C1 C(=O)(C1=NOC2COCC12)NC1C2CN(C(C(C(C)C)OCC)=O)C1C2 N1(C(C(C2CCCC2)OC)=O)CC(CNC(=O)CC#N)C2(CCC2)C1 c1(C(N(C2CC2)Cc2c(Cl)ccc(OC)c2)=O)cc2ncccc2o1 c1(NC(CC2(N(C(COCCOC)=O)C)CC2)=O)cscc1C C12(CNC(C)=O)CCCCC1N(C(C1C3CNC(=O)C13)=O)CCC2 C1(CNC(c2c(C)[nH]cc2)=O)C(C)CCCN1C(=O)CCCN1C(=O)CNC1=O Cc1ccccc1S(=O)(=O)CC(=O)N=S(C)(=O)c1ncc(Br)s1.C1(=O)CO1 C1(C)(NC(COCC(C)C)=O)CCN(C(=O)CCc2ccccc2C#N)CC1 C(=O)(C(O)CC[S+](C)C)NCCOCCN(C(=O)CCc1ccc(Cl)cc1)C C1(C)(NC(c2cc(C(C)C)no2)=O)CCCN(C(=O)Cc2cncn2C)C1 c1(C(=O)NCC2N(C(CC(C)OC)=O)CCC(C)C2)ccc(N=[N+]=[N-])cn1 N1(C(C(C=C)(C)CC)=O)CCC2(COC(C)C2)C1.c1(C(=O)N)sccc1C(F)F N1(C(CCOC(C)=O)=O)CC2(CCN(C(C3CC3(Cl)Cl)=O)CC2)C1C(C)C c1(C(=O)NCCOC2CN(C(C(n3c(C)ccn3)C)=O)C2)ccc(O)cc1 C(=O)(CCCC(C)(F)F)N1CCC(N(C(C2CC2(Cl)Cl)=O)CC)C1 c1(C(=O)NC2COCCN(C(c3nc(CCC)oc3)=O)C2)ccc2nccn2c1 N1(c2nc(CC)nc(C)c2)CCCC1C1CCCCN1C(=O)C(C)(C)C1CC1 C(CC(=O)N(C(C)CC(=O)OC)C)(C(F)F)NC(CC=C)=O c1(NC(CN)=O)cccc(C(=O)OCC(C(CCCC)=O)=O)n1 Cc1ccc(CC(N2CCC(CNC(C34CCC(C3)OC4)=O)C(C)C2)=O)cc1C c1(C(N(C)CC2(O)CCN(C(C(CC)CC)=O)C2)=O)ccc2nnc(O)n2c1 O=C(C1=CCCCC1)N1CC2CC2(CNC(C2(c3cc[nH]n3)CCOCC2)=O)C1 CC(C)(C)C(O)C(=O)N1CCCC1CN(CC(=O)NC1CCOC1)C1CC1 c1(NCC(C)CNC(c2n[nH]c(O)n2)=O)cc(S(C)(=O)=O)ncn1 CN1CC2CC1CN2C(C1C(O)CCN1C(C1CC(CF)C1)=O)=O CCC(CCCC(=O)NCc1nc(C)cc(C)n1)NC(c1cc(COC)[nH]n1)=O c1(C(=O)NCCN(C)C(C2COC3(CCC3)C2)=O)ccn2ccnc2n1 c1(C(N2CC3(OCC(NC(C(C)C4CCC4)=O)C3)C2)=O)cc2nc[nH]c2cc1F c1(CC=O)c(C)cccc1Cl.C(C)(CO)(C(=O)N)NC(C)=O.CCCC1CC1 C1(NC(N2CCC(C)(C(=O)OCC)C2)=O)Cc2ccccc2C1 c1(C(N2CC(CC(=O)N(C3C=CCC3)CC)OCC2)=O)cc(C)ccc1OC S(=O)(=O)(CC(=O)N1CCC(c2cn(C(C)CO)nn2)C1)NCC c1(OC)cc(C(=O)NC2CCCC2C)c2c(c1)CCO2.C(=O)C.CC(N)=O c1(N(CCN(C)C(C2(c3ccc(Br)cc3)CC2)=O)C)ncccc1C#N C(=O)(C1=NOC2COCC12)NC(c1cn(C)nn1)C(=O)NC(c1cnc[nH]1)C Nc1ccc(C(=O)NCC2CN(C(=O)C=Cc3cscn3)CCCO2)c(O)c1Cl C12(NC(CCC#C)=O)CCC(CNC(c3c[nH]cc3C(C)=O)=O)(C1)OC2 c1(C(N2CCN(C(C3ON=C(CC)C3)=O)CC2CO)=O)cc2ccc(F)cc2[nH]1 Cc1cc(C(=O)NC(CO)CCCNC(=O)C(C)S(N)(=O)=O)nc(O)n1 C(=O)(CC(C(=O)NC1CN(C(=O)C#CC(=O)NC)CC1C)N1CCCCC1)OC c1(C(=O)NC(CNC(C(COC)OC)=O)(C)C)c(C)nc2ncnn2c1C C1(NC(CCOC(C)C)=O)CCCC12CN(C(=O)C(c1ccc(F)c(F)c1)O)C2 c1(C(N2C(C)(CNC(=O)CSc3n[nH]c(O)n3)CCC2)=O)csc2cncn12 CCC(CCOC)C(=O)NC(C)(C)CNC(c1ccc(-c2ccccc2)cc1)=O c1(C(=O)NC2(CF)CCN(C(C3(C)ON=C(C)C3)=O)C2)cnn2ccncc12 N1(C(CCCN(C)C)=O)CC(NC(C2(C3CCC3)CC2)=O)CC(O)C1 c1(CC)cnccc1C(N1CCCC1CCNC(=O)C(C)CN1CCCCC1)=O C=CCC(C)C(=O)N1CCC(C)C1CNC(=O)CC1(C(F)(F)F)CC1 c1ccccc1C.C12(CCC)CC(C(=O)N)(C1)C2.C(C)(C)C1CC1.C(=O)C CCC(C)(O)C(=O)NCC1(O)CCN(C(c2ccc(OC)nn2)=O)C1 C1CCN(C(=O)CC2C=CS(=O)(=O)C2)C1.C(=O)CCCN1CCCC1.CO.C N1(C(C(C=C)CC)=O)CCCC(C(N2CCN3CCC2C3)=O)(CC)C1 c1(C(=O)NC2CN(C(C3(C#C)CC3)=O)CC(O)C2)cc(Cl)c(C)cc1[N+](=O)[O-] CC(CNC(C1(C)C=CCC1)=O)C(F)C(=O)NCCOCC1CCC1 c1(CC(=O)NCCCN(C(c2n[nH]c3c2CCC3)=O)C2CC2)cncnc1O Cc1csc(C(=O)NCCCCCn2cc(C(C)(O)CCO)nn2)c1 c1(N2CCN(CC3CC3)CC(C)C2)cccc2c1CCN2C(=O)OC(C)(C)C CC1(C)CC(NC(=O)CSS(C)(=O)=O)CN(C(C2CCCCO2)=O)C1 O=S(=O)(c1cccc(N2CCOCC(O)C2)n1)NCCCOCCCO c1cc(C)ccc1[N+](=O)[O-].C=Cn1nccc1C(=O)NCCCCNC(=O)CC.O N1(C(C(C)OCCC#C)=O)CCC2(CCC2)CC1.c1(C(=O)N)cn2c(n1)CCC2 CC1=NN(CC(=O)N2CCS(=O)(=O)C(CC)C2)CC1.C(=O)CC(O)CN(C)C.N CCC(CC(=O)NC(CCSC)C(N1CC(=O)NCC1C)=O)C(C)(C)C c1(C(N(C2CN(C(C=C(C)C3CC3)=O)CC2(C)C)C)=O)csc2c1CCC(C)C2 N1(C(C)=O)CC2CCCC1C2.C(=O)CC.[SH](C)(=O)=O.C(C)N.C(=O)C1CC1 CCC(CNC(=O)CC1(C)CCN1C(=O)C(CC)SC)CC(C)C N1(C(c2c(SC)ccs2)=O)CCC2(CC1)CC2NC(=O)CCC1CCCOC1 c1(C(N(C)CC2CCCN2C(c2ccnc(S)c2)=O)=O)ncc(Cl)cc1F c1(CC)ccc(F)c(C(N2CC(NC(=O)C(CC)NC(C)=O)C(F)C2)=O)c1 N1(C(c2ccnc(C)n2)=O)CC(C)CN(C(c2cc(Cl)ccc2F)=O)CC1C Cc1nc2cccc(C(=O)NCC3C(C)CCCN3C(=O)Cn3ccnn3)c2s1 C(CCC(O)C(=O)NCC1(C)CCCC(=O)N1)NC(C1ON=C(CC)C1)=O N1(C(c2n(CC)ccn2)=O)CCOC2CCN(C(c3cc(OC)ccn3)=O)CC12 c1(CCCC(=O)N(CCNC(C2CCCCO2)=O)C2CC2)ccc(Br)cc1 C1(NC(c2c(CC)nc[nH]2)=O)CC2CC1CN2C(=O)CCn1nc(C)cc1C Cc1cc(Br)c(Cl)cc1NC(=O)Cc1sc(N2CCOCC2)nc1-c1cccs1 CC(C)CC(C)(C)C(=O)NC1CC2CCC1N(C(C1(C)CCCC1)=O)C2 N1(C(c2ccncc2)=O)CC2(C)CC1(C(N1CCC3C(C(N)=O)C3C1)=O)C2.CO C(=O)C(CC)=Cc1cn[nH]c1.C(C(=O)NCC)(C1CCCC1)OCC.CC.O CC1CC(C(=O)NCC(F)(F)F)N(C(=O)CC(=O)Nc2ccn(C)n2)C1 C1(C(C)O)COCCN1C(C1CCOC1CNC(C1CCC(=O)O1)=O)=O N1(C(C(C)OCCOC)=O)CC(C)C2(C1)CN(C(=O)CCCC)C2.C(N)=O C1(N(C(CNS(NC)(=O)=O)=O)C)CN(C(C2CCCN2C=O)=O)CC1(C)C Cc1ccn2cnc(C(=O)NC3CCN(C(c4ncccc4O)=O)C3C)c2c1 CC1CC(O)CCN1C(=O)C(F)CC1CN(C(c2cnc(N)cn2)=O)C1 C1(CCC)CN(C(c2csnc2Cl)=O)CCN1C(=O)CCn1nc(C)nc1C N1(C(C2(C)CCCN(C(c3ccc(Cl)cn3)=O)C2)=O)CCn2ccnc2C1 C1(NC(C(N2CCSCC2)C)=O)(CF)CCN(C(c2cccc(N(C)C)c2)=O)C1 CCCCC(O)CCC(=O)NCCN(C(=O)CCCN1C(=O)CN(C)C1=O)CC O=C1NCCCc2occ(C(N3CCC(C4CCCO4)CC3)=O)c21 C1(C)(CNC(C(c2c(C)noc2C)C)=O)CCN(C(=O)C#CC2CCC2)CC1 c1(C2CCC2)ccccc1.C1CC(F)C1.O=CCSC.C(=O)CC1CC1.N N1(C(C=Cc2c(C)cccc2F)=O)CCC(C2(C)CC2)CC1.c1(CNC)ccco1 N1(C(CCC(C)C)=O)CC2CS(=O)(=O)CC2(NC(=O)C=C2CCOCC2)C1 C1(C(N(CCN(C(C)C)C(c2cccnc2)=O)C)=O)Nc2ccccc2C1(C)C CC(C)C(CNC(C1CCCCS1)=O)C(=O)NCC1CCOC1=O Cc1sc2nc(SCCOC(=O)CC3CCCC(=O)N3)nc(O)c2c1C c1(CN2CCCC(C(=O)NC(c3cc(F)cc(Cl)c3)C)C2)cnc2cc[nH]c2c1 N1(C(C(n2ncc(C)c2)C)=O)CC2CC1CN2C(=O)COC(=O)C(=O)O N1(c2c(C)c(NCc3nccs3)ncn2)CCC2(CNC(=O)C2)C1 c1(C(=O)NC2C=CC(CNC(Cc3n(C)nnc3)=O)C2)cnn2cccnc12 C12(NC(CN(C)CCO)=O)CCCC(CN(C(=O)CCn3ccnc3)C1)C2 CC1CCC(NC(=O)CC(F)(F)F)CN1C(=O)C=CCOC1CCOCC1 C(=O)(C(CO)C(C)(C)C)NC(C1OCCN(C(C(C)Sc2nncn2C)=O)C1)C C1(C(=O)NCCC(C(=O)OC)C)CCC2(CC2)N1C(c1cncc(C)c1)=O c1(NCC2CCC(O)C2)nccc(=NC2CC(F)(F)C2)[nH]1 c1(-n2cc(CC3N(C(c4csc(Cl)c4)=O)CCC3)nn2)cccc(F)n1 c1(C(=O)NC(c2cn(CC(C)(C)O)nn2)C)ccc2c(c1)NC(=O)CC2 c1(C(CC(C)(C)C)NCc2ccc(C)o2)nc2ccccc2s1 c1(NC(C2CC3CC3N2C(c2ccc(O)c(I)c2)=O)=O)cc(Cl)c(O)c(Cl)c1 C[Si]1(C)CCC(CNC(C2C=CCN2C(C2CC3CC3C2)=O)=O)C1 c1(C(N2CCC(O)(CCNC(=O)CC3CSCCS3)C2)=O)n[nH]c2ccccc12 O=C(CCCCC(F)(F)F)NCC(C1CC1)NC(C12CCC(F)(CC1)C2)=O C12(NC(c3nn(C)c(OC(F)F)c3)=O)CCN(C(C3(F)CCCCC3)=O)CC1C2 N1(C(c2n(C)ncc2)=O)CCCC12CCN(C(C1(O)CCCC(C)(C)C1)=O)CC2 N1(CC(N2C(CC(=O)NCC(COC)C)CC2)=O)CCCCC1C c1(CCC(N2CCC(O)C2)=O)csc2nc(C)cn12.C=CC1(C(=O)NC)CCC1 C1(C(=O)NC(c2cnnn2C)C)CC(F)(F)CN1C(=O)Cn1ccnc1 C1(NC(COCC=C)=O)CC2CC(NC(c3cc4c(s3)CCOC4)=O)CC2C1 C1(CC(=O)NCCN(CCC)C(C2(CC)CCCCCC2)=O)CCOCC1(C)C n1(CC)nc(C(=O)NCC(C)C(=O)NCC2(C)C=CCCC2)cc1C Cc1oc(C(C)C)cc1C(=O)NOC(c1nn[nH]n1)C c1(CN2C(C(=O)Nc3c(C(=O)OC)n[nH]c3)C(O)CC2)c(Cl)cc(O)cc1Cl C1(OC)CCOCC1OC(c1cc(C(N2CCN(C)CC2)=O)nn1C)=O c1(C(N2C(CNC(C3CC4CCC3CC4)=O)CC2)=O)ccc2cnccc2c1 N1(C(C(CNC(=O)C(O)Cc2ccccc2)CC2CC2)=O)CC2(CCC2O)C1 c1(C(N2CC(N(C)C(C3CC3(F)F)=O)C2)=O)c(Cl)cnn1C1CC1 c1(C(=O)NCCCNC(=O)CCn2cnc3ccccc23)ccn2cncc2c1 CC(C)CCC(=O)NC1CCCC(NC(c2cc(C3CCOC3)[nH]n2)=O)C1 N1(C(C(F)=CCC)=O)CCCCC(CNC(c2ccc(CC)cc2)=O)C1 c1(C(=O)N)ccc2nn[nH]c2c1.CC1(C)CN(C(C23C=CC(CC2)C3)=O)CC1C c1(C2(OC(=O)CNC(C(=O)C(CO)c3ccccc3)=O)CC2)ccccc1 CCC(C)CCCCC(=O)NCc1ccnc(C(=O)NC2COC(C)(C)C2)c1 c1(C(=O)NCCCCC2CCCN(C(C(CC)O)=O)C2)c(C)nn(C)c1Cl C1(=CC=O)CCC(C)(C)CC1.C1CCCC1.C(=O)(C=CC)N(C)CC.N C12(CNC(c3c(C)cns3)=O)CCCC1N(C(c1ccccc1)=O)CCC2 C(CC(C(=O)NCCC(F)(F)F)NC(=O)C(C)C(F)F)OC C(=O)(CC(c1ccccc1)C1CC1)NC(C1CCCN1C(C1CC=CC1)=O)C N1(C(C2(COC)C=CCN2C(c2cocc2C)=O)=O)CC(C#N)C2(CCC2)C1 N1(C(CCC=C)=O)CCC2(C)CN(C(=O)C(O)CCCCC)CC12 C1(C(=O)NC(CC)C)CC(F)CN1C(c1cnc(C(C)C)o1)=O N1(C(CCn2ncn(C)c2=O)=O)CC(C)(C)CC1(C)C.C12(C(=O)N)CCC(C1)C2 C1(CNC(CNC(CCC)=O)=O)CCCN(C(c2ccnn2C(C)C)=O)CC1 c1(NC(C2C(C)N(C(=O)C=C3CCC3)CC2)=O)cc(Cl)ccc1O S(=O)(=O)(c1ccc(F)c(F)c1F)N(c1ncc(OC)cn1)C1CNCC1(F)F c1(CCOC)n[nH]c(=NCCCC2CC(NC(=O)CO)C2)s1.c1ccc(C)cc1 C1(NC(c2cccc(CC)c2)=O)CCN(C(=O)CCN(C)CC)CC1(C)C N1(C(C)=O)CCC(C)(CC(=O)N(C(C)CN(C)C)C)C1.Cc1ncsc1CO CCCCC(C)C(=O)NCC(C1CCCN1C(=O)CCC(C)=O)(C)C Cc1nn(C)c2sc(C(=O)NC3CCN(C(C4(C)C=CCC4)=O)CC3)cc12 CCCCC(CC)(c1nnnn1CC1CC1)NC1CCCC1CCO c1ccc(N(C)C)cc1.c1(N(c2ncc(C(C(=O)NCC)N)s2)C)ccccc1 CC1(C)CCCC(C(=O)NCCC2CN(C(c3cc(N)c(Cl)cn3)=O)CCO2)O1 c1(C(=O)N)ccn2ccnc2n1.c1(C(N(C(C)C)CC)=O)cnn(C(C)C)n1 Cc1ccc(F)cc1S(=O)(=O)N1CCOCC1CNCc1ccnc(Cl)c1Cl C=C(C)C1CN(C(=O)C(C2CC=CCC2)NC(=O)CP(C)(C)=O)CCO1 C1(C2CCN(C(=O)Cc3cn(C)nn3)C2)CC1.C(CC=O)N(CC(F)(F)F)C.N C(C(CC(C)C)C(=O)NC1CCC2(CC2)C1)NC(C(CCO)OC)=O N1(C(c2cn(CC=C)nn2)=O)CC(CC(=O)N(CC(C)OC(C)=O)C)CC1C C(=O)(CCS(=O)(=O)Cc1ccccn1)N.CC1CC1C(=O)N(CC)C1CC1 Cc1cc(C(=O)NCC2CCCCN(C(=O)CCN3CCC(F)C3)C2)nc(O)n1 N1(C(c2c(C)cnnc2)=O)CC2(CC2)CC1C(N1CCCC(C)(N(C)C)C1)=O N1(C(c2cc(C)ncn2)=O)CCCC(C2CC2NC(C2CCC(F)(F)CC2)=O)C1 c1(SC)ncc(C(N2CC(NC(=O)CCC3CCC(=O)N3)C(F)C2)=O)n1C c1(OC)c[nH]nc1C(=O)N(C1CC(NC(=O)CCCSC)C1)C Cc1ccc(CC(=O)N(C)CCOCCN(C)Cc2cncc(Cl)n2)c(Cl)n1 c1(C(=O)NC2CCN(C(c3ccc(Br)cn3)=O)CC2)cnc2ccccc2n1 c1(C(N2C(C(C)(C)NC(c3cccc(CO)c3)=O)CCC2)=O)cc2cscc2s1 C(c1ccccc1F)=CC=O.N1(C(C(C)OCCN(C)C)=O)CC(C)C(C)C1 C1(NC(C2CC(C#C)(O)C2)=O)CCN(C(=O)C(c2cscn2)N(C)C)CC1C N1(CC)CCc2c(F)ccc(F)c2C1.c1(OC)cc2c(cn1)-c1csc(c1)CS2 N1(C(C2(CNC(C(C)c3ccsc3)=O)CCCO2)=O)CC2CCC(C1)C(=O)N2 C(C(CC(=O)N1CCC1c1cccc(F)c1)NC(=O)C(C1CCOCC1)=O)OC CC1(C)CC(NC(=O)C=CS(C)(=O)=O)CN(C(=O)Cc2ccc(O)cc2)C1 C1C2CCCC1N(C(c1snnc1C1CC1)=O)C2.N1(CC(=O)NC)CC2CC2C1 C1(C(=O)N)CC2CCC1CC2.c1(C(=O)NCC(C)C)cn(C)nc1-c1nccs1 C1(NC(=O)C)CCCC12CCN(C(=O)C1CC1)CC2 C1(C(C)NC(c2c(C)ocn2)=O)CN(C(C2CNC(=O)N2C)=O)CCO1 C1(NC(c2cc(C)sc2C)=O)CC2(CCC(C)OC2)C1.C(=O)(C1=COCCC1)N c1(C(=O)NC2C(NC(CCSC)=O)CCOC2)cc2c(=O)[nH]c(C)cn2n1 CC(Cn1cncn1)N=c1cc(NCCC2CSCCS2)nc(C(F)(F)F)[nH]1 C1(C(N2CC(c3ccccc3)(NC(CS(=O)(=O)NC)=O)C2)=O)CCOCC1(C)C C1(CNC(C(CC)(C)O)=O)CC2CCC1N2C(c1oc(CO)cc1C)=O C(=O)(C(C)(F)C(C)(C)F)N1C(C(=O)N)CCC12CC2.C(C(C)C)OCC C1(C(N2CC(C)(C)C2C2CC2)=O)CCCN1NC(=O)c1nccnc1N.C1CC1 c1(OC)ccc(C(=O)N(C)CCNC(C2CCN(C)C(=O)C2)=O)cc1Cl c1(C(N2CCC(CNC(C(C)=C3CC3)=O)CC2C)=O)ccnc2ccsc12 C12(C(N(C3CCOCC3)C)=O)CC1CCN2C(c1ccsn1)=O c1(C(N2CCC(CN(C(=O)C(F)(F)CO)C)CC2)=O)cccc2oncc12 CC1CN(C(c2ccc(C3CCC3)nc2)=O)CCC1NC(=O)CC(C)(C)C C1(CNC(CCN(C)CCO)=O)C(C2CC2)CCN1C(C1CCCC1)=O CN1CCCC(NC(=O)C(C)CC2CC2)C1=O.c1(C(=O)N)cc(O)cc(=O)o1 C1(c2cn(C(C)C)nn2)CC2CCC(C1)N2C(=O)CCCc1nc(C2CC2)no1 C1(NC(C)=O)CCCN(C(=O)C(C)(C)CNC(=O)C(C)=C(C)C)C1 N1(C(Cc2cnc(C)[nH]2)=O)CCC(C)C(N(C)C(c2ncc(Cl)cc2O)=O)C1 C1(C(=O)OCC)C2CCN(C(=O)NCCCn3cccn3)CC12 C(=O)(C(CC(C)SC)N(C(C)C(=O)OC)C1CC1)NCCCC Cc1nc(CNC(=O)C(C2(C)CC2)NC(c2cnn(CCF)c2)=O)no1 C1(NC(C=CCCC)=O)CCCC(c2nccn2C)C1 CCCC(CCC)C(=O)N1CCC(c2cn(Cc3cnns3)nn2)C(O)C1 C(=O)(CC(C)(C)C(F)(F)F)NC(C1OCCN(C(c2cnc(C)n2C)=O)C1)C C1(C(=O)NCC(C)CNC(=O)Cc2nnc(C)o2)(CSC)CCOCC1 c1(CNC(Cc2c(C)ccc(I)c2)=O)ccc2c(c1)OC(C)(C)O2 Cc1nn(C(C)(C)C)cc1C(N1CCCCC1CC)=O.C1(CC(=O)N)OCCO1 N1(C(C2C(CC)OCC2)=O)CCN(C(c2cc(OC)ncc2Cl)=O)CC1C c1(CN2C3C(C(=O)Nc4ncc(C#N)nc4)C(C3)C2)cnc2ccc(F)cn12 C(C)(C(C(=O)N1C(C(=O)N(CCO)CCn2ccnn2)CC1C)N(C)C)OC N1(C(C2(C)CCCCC2)=O)CCCN(CCNC(C2CCC2(C)C)=O)CC1 c1(CC(=O)N(CC(C)C)C)cnc(C)nc1O.c1(CC)nc(C)c(C=O)o1.N CC(C)C(CC(=O)OC(C)(C)C)NC(=O)CCc1ccccc1Cl c1(C(=O)OCC2N(C(=O)OC(C)(C)C)CC(O)C2)cccc(C#N)c1Br C(C#Cc1ccccc1)N(C(CC)C)CC(=O)O C(=O)(C(C)CC(F)(F)F)NC1C(NC(Cc2nc(C)sc2)=O)CCOC1 c1(C(=O)Nc2c(C(=O)OC)cc(C#N)cc2)ccc2sc(C)nc2c1 C(CCCCCCCO)=CC(=O)N(CCC(C)NC(=O)C(C)C1CCC1)C C(=O)(C(O)CC(F)(F)F)NC1C(NC(CC(C)(C)O)=O)CCC1 c1(CC)nc(C)c(C(N2CCCC(N(C(=O)C(F)=C(C)C)C)C2)=O)c(C)n1 C1(C(=O)Nc2c(OCC)cccn2)CCC2(CN(Cc3ncn(C)n3)C2)O1 c1(C(C)C)ccc(C(N2CCCC2CCNC(C2CC23CC3)=O)=O)c(O)n1 C#CC1(C(=O)N(C(CCO)C(F)F)C)CN(C(=O)C(c2cnn(C)c2)=O)C1 C1(N(C)C(c2cnccn2)=O)CN(C(c2c[nH]nc2Br)=O)CC1F C(=O)CS(=O)CCC(F)(F)F.c1(SCC)cnc(C(=O)O)cn1.[nH]1ccnn1.C N1(C(c2sc(Cl)cc2Br)C(=O)NC(c2ccccc2)C)CCC2(CNC(=O)N2)C1 N1(C(CCNC(COC)=O)=O)CC(NC(=O)CC(F)F)CC(C)(C)C1 Cc1cc(CNC(=O)C(CO)N(C)C)oc1C(=O)N.c1(CC)cncc(F)c1 C(=O)(C(C)(C)C(F)F)NCCc1cccc(OC)c1.C(=O)(CC1CSC1)N Cc1cc(Cl)cc(C(=O)NC2COCC2NC(C2CCc3ncnn3C2)=O)c1C C(c1ccccc1Cl)=C(C(=O)N)C.C(CC(C)C)NC(C1(OCC)CCC1)=O Cn1cc(C(N2CCNCC23CCC3)=O)c2cc(Br)ccc12.N1CC2CC1CN2C Cc1cccc(Cl)c1CN1C2CCC(C2)C1C(=O)NC1CONC1=O Cc1ccc([N+](=O)[O-])c(N2CC3CCC2CN3C(c2cccc(O)n2)=O)c1 c1(OC)cccc(CCCn2nnnc2NC(c2cncc(F)c2)C)c1 C(=O)(CC(C)N1CCCC1=O)NCCN(C(C(C)SC)=O)CCCN(C)C C12(NC(C3CCCOC3)=O)CCCCCC1N(C(=O)C=CC1CCC1)CC2 C1(C(=O)NC(COC)C(N2CC(F)CC(F)C2)=O)CCCC(=O)N1C CC1(C)OC(=O)CC1C(=O)NCC1CCCN1C(c1coc(O)n1)=O c1(N2C(C)CC2C(=O)Nc2cc(O)nn2C)ncc(C(C)(C)O)cn1 CCC(CCC(=O)N1CCC(C)(CNC(c2cc(C(C)C)n(C)n2)=O)CC1)OC c1(C(=O)NCC2(O)CN(C(C3(CCCC)CCC3)=O)C2)cc(O)ncc1Br C1(C(N2CCC(C=O)C2)=O)CCC2CCC(=O)N2C1.c1(C(=O)OC)cc(Cl)sc1 CC#CCCCC(=O)N(CCCOCCNC(=O)CC1(C(F)(F)F)CCC1)C C1(C(=O)NCC(CN(C(C=CCO)=O)CC)(C)C)CCOCC1.CC=C c1(OC)c(C(N2CCCC2CNC(C2C3CCCC23)=O)=O)c(C)nn1C C1(C)(C(=O)NCCCCN(C(=O)C(F)C2CCC2)C)CCC(=O)NC1 c1(C(=O)NCC(C)(C2CCC2)NC(C2OCCO2)=O)nc(C2CC2)ncc1Br c1(NC(CC2CCCN(C(C3(C)CCCN3)=O)C2)=O)ccc(C#N)c(Cl)c1Cl c1(C(=O)NCCN(C(=O)CC)C)ccc2c(c1)NS(=O)(=O)C2.C1CCCC1 N1(C(C2CCCN(C(=O)Cn3cnnc3O)C2)=O)CCC2(CCCCO2)C1 CC(C)CC(F)C(=O)N(CC)C1CC1.C(=O)CC(C)N(C)C=O.C(C)(C)C C(=O)(C1COc2cc(C)c(C)cc21)NCC(=C)CCNC(=O)CC(F)(F)F C(=O)C(F)CC(C)C.C1(C2CC2)(OC)CCC1.c1(C=O)ccc(C(C)=O)o1.N N1(C(c2cc(CC(C)C)on2)=O)CCCN(C(=O)CC2CCC(F)(F)CC2)CC1 C(CCCCNC(=O)CCc1ccncc1)NC(CC1(C)CC1F)=O c1(CC(N2CC(C)N(C(=O)C)CC2C)=O)cc(Cl)c2c(c1)OCCO2.C(N)=O.N c1(NC(=O)NC2CCC(OC(C)C3CC3)CC2)cccc2c(Cl)ccnc12 C(=O)(C(C)(C)CN(C)C(c1cnn(C)c1Cl)=O)NCC1(CO)CC(C)C1 c1(CC)c(C(=O)NC2(CO)CCN(C(=O)C(C)N)C2)nnn1C.C(C)(C)CC c1(C(N2CC(N(C)C)C(CO)C2)=O)ccc(N=[N+]=[N-])cn1.C1(=O)CN1 C1(N(S(CC)(=O)=O)Cc2ncccc2Br)C(C)OCC12CCNCC2 c1(C(N(C2CCCN(C(COCC=C)=O)CC2)C)=O)cc(Cl)c2[nH]c(O)nc2c1 CCCC(C(=O)NC(c1cccnc1)C(=O)NC1CC(=O)N(C)C1)N(C)C CCCC(O)C(=O)NC12CC(C1)N(C(=O)C(C)n1cnnn1)C2 C1(CC(=O)NCC=CC(=O)NCc2cscn2)CC2CCC1C2 N1(C(CCCCCCC)=O)CC(C)CN(C(c2ncc(F)cc2C)=O)CC1C Cc1nn(C(C)C)c(C)c1C(=O)NC1(CO)CN(C(=O)COC(F)F)C1 O=C(CCc1cscn1)NCCCN(C(=O)CCC1CC1(F)F)CCO C(CN=c1[nH]nc(O)s1)C1CCCN(C(C(C(C)(C)C)NC(N)=O)=O)C1 O=C(N=c1[nH]nc(-c2cccc(F)c2)s1)c1cn(C2CCOC2)nn1 c1(C2CC2)ccc(C)cc1.C1(CC(=O)NC(C=O)C2CC2)CC2CC2C1.C c1(-c2cn(CC(CC(C)C)NC(CNC(CC)=O)=O)nn2)cc(Br)cc(C)c1Cl Cc1nc(C(C)NC(=O)CC2CCN(C(=O)CN3CC=CC3)C2)cs1 C1(C)(C(N(CC(CC)NC(=O)CCCn2cncn2)CC)=O)CCOC1C c1(CC(=O)OC)ccc(Cl)c(NC(C2CCN2c2ncc(SC)cn2)=O)c1 C1(N)(CC)CCCN(C(c2cnc(O)cc2)=O)C1.C(=O)(CCC(C)SC)NCC Cc1nc(C(C)(C)C)[nH]c(=NCC(C2CC2)NC(c2nccn2C(C)C)=O)c1C C1(CC)C(C(=O)NCCC2CC(=O)N(C)C2)CCN1C(c1cccnc1O)=O C1(F)(C(N2CC3C(CNC(C(C)c4cccs4)=O)(C3)C2)=O)CCCC=C1F c1(C(=O)NC(C)CCNC(=O)C(C)Cn2ccnc2)ccccc1C#CC1CC1 C1(NC(c2ccc(C)n2C)=O)CCCCN(C(c2ccnn2C(C)C)=O)C1 C1(NC(CCN(C(C=Cc2ccc(C)o2)=O)C(C)C)=O)CCN(C)C1(C)C C(C=O)(C1CC1)OC.C1(CC)CC(C=O)C1.C(C)CC1CCC1.C1CC1.N C(=O)(C(F)(CNC(C1COCCN1C1CC1)=O)C(C)C)NC1(C)C(C)CCC1 C(CC(=O)N1CCCC1)(C(C)(C)C)NC(CC1C(C)=NNC1=O)=O.C1CCC1.C C1(C(=O)NC2CCN(C(C3C(C(C)(C)C)C3)=O)CC2F)CCC(N=[N+]=[N-])CC1 N(C(=NCCCc1ccc(Cl)cc1Cl)NCc1nnc(CO)s1)C(C1CCOC1)C CC#CCCC(=O)N1CCC(n2cc(-c3cncs3)nn2)CC1 c1(SCC(=O)NCC2CC(NC(C3(CC)CCC3)=O)C2)ccccc1Cl Cc1ncccc1C(=O)NCC1(NC(=O)CN2CC3C=CC2C3)CC1 C1(NC(C(CN(CC)CC)F)=O)CCC(CN(C(=O)C(C)O)C)CC1 C=CC(C)(O)CC(=O)N(CCCN(C(=O)CC1(c2ccccc2)CCC1)C)C c1(C(C)OC(=O)CCc2ccc(Br)c(Cl)c2Cl)nc2ccccc2n1C c1(N2CCCC(CC=C)(NC(=O)CCC(C)C)C2)ccc([N+](=O)[O-])c2nonc12 N1(C(c2ccc(SC)s2)=O)CCN(C(=O)CC2(O)CCN(C)CC2)CC(C)(F)C1 Cc1ccc(C(C)NC(C2CCCN(C(C3CCC(C)(C)C3)=O)C2)=O)nc1 C1(NC(COC)=O)C2CC1N(C(C1CC=CCC1C(=O)OC)=O)C2C C1(C(=O)NC2CN(C(c3cn(CCCF)nn3)=O)CC2O)CCC2(CCC2)CO1 N1(C(C(C)Oc2cccc(F)c2)=O)CCC2(CC1)CC2NC(C1(C)CCC1)=O C(c1cccc(Br)c1)=CC(N1CC(CC(C)NC(C(C)(CO)OC)=O)C1)=O C1(C(N2C(C3(O)CN(C(CCc4n(C)cnc4)=O)C3)CCC2)=O)C(C)(C)C1(F)F N1(C(CSC(C)C)=O)CCCC2(CNC(=O)CN3CCOCC3)CCCC12 C=C=CC(C)C(=O)NCC1(OC)CCN(C(C2(CC(F)(F)F)CC2)=O)C1 c1(OC)ccc2c(c1)CCC2C(=O)NC1CC1NC(c1ccc(=O)n(C)c1)=O C(CC(=O)NCc1ncoc1C)(C(C)CC)NC(c1cnc(CC)nc1)=O C(C(C(=O)NC(CN1CCCC1)CC)NC(C1CCS1(=O)=O)=O)OCC CCCC(C(=O)NCC1CCC1NC(c1scnc1C)=O)C(C)C c1(C(N(CC(CN(C(C2CC2)=O)C)O)C)=O)ccc([N+](=O)[O-])c(N)n1.CC c1(OC)ccc(C2(NCC3CCCN3c3ccncn3)CC2)c(Cl)n1 C(=O)(C1=C(CC)OCCC1)N(C)CC1N(C(c2cncc(OCC)c2)=O)CCC1 C(CCN=c1nc(N2CCCC(CSC)C2)cc(C)[nH]1)OC c1(NC(C(C)(N(C(C=CC=CC)=O)C)C2CC2)=O)cc(C)ccc1O CC1=C(C(=O)NCC(C)CNC(=O)CC(C)(O)C(F)(F)F)Cn2nnnc2N1C c1(CC(=O)N(C)CC2N(C(C(C)c3ccon3)=O)CCC2)cccnc1Br C(=O)(C1=CC2(CCN(C(=O)CC3=CCCCC3)C2)C1)NC1CC(C)(C)C12CC2 c1(C(N(C2CCN(C(CC(C=C)C)=O)C2)CC)=O)nc2nccc(C)n2n1 N1(C(c2[nH]ccc(=N)n2)=O)CCN(C(=O)Cn2nc(Cl)ccc2=O)CC1CCO C1(NC(C=C(C)C(C)C)=O)CCCC(CNC(c2ccn(CC#N)n2)=O)C1 c1(C(=O)NC2(CN(C)C(C3CCCCC3)=O)CC2)ccc2nc(O)[nH]c2n1.C N#CCCCCC(=O)N(CCNC(c1cc(Cl)no1)=O)Cc1ccccc1 N1(CC=O)CCc2sccc2C1.c1(C(N(C)CCOCC)=O)cnn(C)c1Cl.N c1(C(=O)NC(C2CN(C(=O)C(F)(F)C3CC3)C2)C)cc(O)c2ccsc2c1 C(=O)(C(CO)C(C)(C)C)N1C(C(C)NC(c2ccc(O)cc2F)=O)CCC1 c1(C(N2C(CN(C(C(C=C)O)=O)C)COCC2)=O)cccc2ncnc(O)c12 c1(C(=O)NCC2OCC(CNC(c3cnsn3)=O)C2)c(F)cccc1Br N1(C(c2c(C)ncs2)=O)CCOC2(C1)CN(C(C13CCC(C1)OC3)=O)C2.CO.C c1(CC(=O)NCC2CCC2)ccc(O)c(Cl)c1.C12(CC=O)CCC(CC1)C2 c1(CNCC2CCC(C(NOC)=O)C2)csc2c1CCCC2 c1(CC(=O)NCC(C)CN(C(=O)Cc2ccc(F)cc2)C)ccc(Br)cn1 C(=O)C(C)C(C)S(C)(=O)=O.C1(NC(C(C)OCC(C)C)=O)CCCCC1.N c1(-c2ccc(CN(C3CCS(=O)(=O)C3)C(C)(C)CO)cn2)ccc(Cl)cc1Cl Cc1ccc(C(N2CC(O)CC2CNC(c2ccnc(CO)c2)=O)=O)nn1 N1(C(=O)NCc2ccc(OC(F)(F)F)cc2)CCC(=O)N2CCCCC12 C(N=c1[nH]cnc(Cl)c1F)C1CCCCN(C(=O)CCc2c(F)cccc2Cl)C1 C12(CNC(c3c[nH]c(=S)cn3)=O)CCC1CN(C(C1CC13CCC3)=O)C2 C(=O)(C(C(C)NC(=O)Cn1ncccc1=O)C(C)C)Nc1cccc(CC)c1F N1(C(CC2(OC)CN(C(=O)C(c3cnn(C)c3)C)C2)=O)CC2CC2(COC)C1 CCC(CC)(CO)C(=O)N1CC(C(=O)NOCCCCF)C(F)C1 N1(C(c2n(CCC)ncc2)=O)CC(NC(=O)CC2CCCOCC2)CC(O)C1 N1(C(C=CCCC(C)C)=O)CC2(CCCN(C(c3nccnc3N)=O)C2)C1 C1(NC(CCN(C(c2cc(OC)ns2)=O)CC)=O)CCN(C(C)C)CC1 CC(C(=O)NC1CCN(C(c2cnn(-c3ccccn3)c2)=O)C(C)C1)S(C)(=O)=O C(=O)(C1OCCn2ccnc21)NCC(N(C(=O)Cn1cnnc1O)C)C1CC1 N1(CC)CCCC1C(=O)NC1(CCC(=O)NC2CCNC2=O)CCC1 C(C(C)C(=O)NOC(c1ccccc1)C)N(C(c1c(CC)ncnc1)=O)C CN1CCN(C(=O)CC2CCOC2)CC1CNC(C1(F)CCOCC1)=O N1(C(C2CC(OC)C2)=O)CCC(C(F)(F)F)C(NC(c2cnn(C)c2)=O)C1 C#Cc1cc(C(=O)NC2CCN(C(=O)C(c3cc(C)ccn3)(C)C)C2)ccc1C C(=O)(C1=CCCSC1)NC(CNC(C(COC)NC(C)=O)=O)C1CC1 NC(CO)CC(=O)Nc1ccc(CN2CCCC2=O)cc1 C1(C(=O)NCC(c2ccccc2F)NC(CC(C)F)=O)CCC2(CC1)CC2(F)F c1(OCC(=O)NCC2C(C)CN(C(=O)CO)C2)ccc(S(C)(=O)=O)cc1 c1(CNC(=NCC)NCC(c2ccc(Cl)cc2)n2cccn2)ncc(C)cc1C C1(COC)(NC(=O)Cn2cccn2)CN(C(=O)CCC2CC2C)C1 N1(C(C23CCC(NC(CN(C4CCCC4)C)=O)(CC2)C3)=O)CC(O)CC12CCC2 c1(NC(C2CC2C(=O)Nc2cc(F)c(Cl)cn2)=O)cccc(F)c1[N+](=O)[O-] C1(NC(c2c(N(C)C)cncc2)=O)COCCN(C(C2CNC(=O)O2)=O)C1 c1(OC)cc(C)ccc1NC(=O)C(N1CCC(N2CCNCC2=O)CC1)=O c1(CCC(N2CC(C(C(=O)NC(CCC)C3CC3)O)C2)=O)ccncn1.C1CC1 CCCCC(O)C(=O)NCC(CC(F)(F)F)NC(c1cncnc1C1CC1)=O c1(N(CC)Cc2ccccc2)ccc(C(=O)NCC2CC2)cc1 CC1(C(N2CCN(CCO)CC2)=O)CCCN(C(c2cc(C3CCC3)on2)=O)C1 CCC(C)C(O)C(=O)NCCCCC(C)NC(c1ccc(C(F)(F)F)[nH]1)=O C#CCC(C)(CC)C(=O)NCCCC1CN(C(c2ccc(=NC)[nH]c2)=O)CCO1 c1(NC(C#CC)=O)cnc(Cl)cc1C(=O)Nc1nc(C(=O)OC)cs1 N1(C(C)C)CCCC(N(C(=O)CCCc2nccs2)C2CC2)C1.C1CO1 c1(OCCCC)ccc(CN2CCCC2(C)c2ccccc2)cc1OC Cc1cccc(CCS(=O)(=O)NC(C)C(=O)OC(C)C)c1 CC1CCCN(C)N1C(=O)N=c1ccn(CCC#N)[nH]1.C1CCCC1 Cc1ccc2c(c1)C=C(C(=O)NC(C)CNC(=O)Cc1cc(F)ccc1C)CO2 c1(C(=O)NC(CC(C)Nc2ncccn2)C)cccc2c1NC(=O)CO2 N#Cc1cc[nH]c(=NCCC2CCC(NC(c3cnn4c3CCC4)=O)C2)n1 c1(C(=O)NC2N(C)CC2)ccccc1-c1cccc(C(N2CCCCC2)=O)c1 C1(C(=O)NCCCCC#C)CC2(CCC2)CN1C(c1cc(C)cs1)=O C1(C2(NC(c3c(C)ccs3)=O)CC2)CCCCN1C(=O)CCCC1CCCO1 c1(CC)cc(C)c(C(=O)NC(C(N2CC3C(CO)C3C2)=O)c2ccco2)o1 N1(C(C2CN(C(CCN(CC)CC)=O)C(C)(C)C2)=O)CC(C)C12CCOCC2 C#CCCCCCC(=O)NC(C)CN(C)C(c1conc1C1CCCO1)=O C1(=C(C)C)CN(C(=O)C(C)=CC(C)(C)C)CC12CC2.C1CN(C)CCO1.C=O.O N1(C(c2c(C)c[nH]n2)=O)CCC(C2CC2)C1C(N1CC(Cc2ccoc2)C1)=O c1(C(=O)NC2C(NC(C(C(C)O)(C)C)=O)CCC2)ccc2nnn(C)c2c1 C1(OCC)(CC)CCN(c2nnnn2Cc2ccccc2OC)CC1 CC1(NC(=O)CCOCC(F)F)CCN(C(C2C(C)(C)C2(C)C)=O)C1 N1(C(c2ncnc(C)c2C)=O)CCC2CN(C(=O)C=CCCC(C)C)CC12 c1(OC)ccc(CC)cc1.C1(C)(C=O)CCC(C)C1.C1(=CC=O)CCCC1.N CCN=C(NCCC1COC(C)(C)C1)NCC1(CC)CCCC1 Cc1ncc(CC(=O)N(C2CCN(C(C3CC(F)(CF)C3)=O)C2)CCO)s1 N1(C(CC2C(C)(C)C2)=O)CC2(CCN(C(C3CC(=O)C3)=O)C2)C1 c1(C(=O)NC(CC)CNC(=O)CCC2CCCN(C)C2)c(Cl)sc(C)c1C N1(C(c2c(C)n(C)cc2)=O)CC(O)CCC1C(N1CCS(=O)CC1C)=O CC(CC1CC(F)(F)C1)C(=O)N(C(C1CCCN1CC)C)CC.c1ccccc1 c1(C(N2CCC(NC(C(=C(C)C3CC3)F)=O)C2)=O)coc2c1N(C)C(=O)CCC2 C#CC1CN(C(=O)C(C)(C2CC2)N(C)C(C2CCC(C)O2)=O)C1 Cc1ccc2c(c1)C=C(C(=O)N1CC3(NC(c4cccs4)=O)CCC1CC3)CO2 c1(C=O)ccc2c(c1)OC(C)(C)C(=O)N2.CCS(=O)(=O)NC(C)C=O.CC C1(CC(=O)NC(c2cnn(C3CC3)c2)C)CN(C(c2ccncc2)=O)CCO1 C(=O)(C(C)(C=C)CCO)C(CC#C)=O.OCOCC c1(NC(C)=O)ccc(NC(C2CCCN(C(C3(C)COC3)=O)CC2)=O)cc1C c1(C(=O)NCC(C)C)ccc(C#N)cc1O.C1(C=O)CCCC(C(C)(C)C)C1.N C1(NC(Cc2c(C)con2)=O)C=CCN(C(C2(N3CCOCC3)CCCC2)=O)C1 CCCC(C#N)C(=O)N1CC(C2CN(C(=O)CCOC3CC3)CCO2)C1 CS(=O)(=O)c1cc(C#N)ccc1CN1CCCC1C(N1CCC(O)CC1)=O CCCCC(CC)C(=O)NCC1CN(C(=O)CSCc2nc3ccccc3[nH]2)C1 N1(C(COCCC#C)=O)CC(O)(C2(CNC(C3(C)CCCN3C)=O)CC2)C1 C1(N=c2ccn(CCC3CC3)[nH]2)(c2n(C(C)C)nnn2)CCC(C2CC2)C1 C1(C)(C(N(C)Cc2ccco2)=O)CN(C(C2CCC=CCC2)=O)C(C)(C)C1 CS(=O)CCN=c1[nH]c(=NCc2nn[nH]c2)[nH]c2c1CCC2.c1(S)ccccc1 CC1Cc2c(F)cccc2CN1C(c1cc([N+](=O)[O-])ccc1I)=O c1(C(=O)NC(CNC(CC(OCC)O)=O)CO)coc2ccc(CC)cc12.C C#Cc1cc(NC(c2occc2COC)c2nnnn2CC2CCCO2)ccc1C N1(C(CC(CCCCCC)C)=O)CCc2ccccc2C1CCNC(=O)CCF C1(NC(=O)CC2CC2)COCCN(C(C2CC=CCO2)=O)C1 CCCC(C)CCCC(=O)N1CCN(C(c2cc(CC)n(C)n2)=O)CC1C C1(CC(C)(C)C)C(=O)N1.CC(CC(=O)NCCCC1CCC1)n1ccnc1 c1(C(=O)NCCCNC(c2c(C)ccnc2)=O)cc(F)c(Br)c(Cl)c1 c1(C(=O)NCC(CNC(c2nc(OC)oc2)=O)O)cnc(N)c(O)c1 c1(CN(C)C)cccc2c1N(CC(c1cccc(I)c1)C)C(C)(C)C(=O)N2C C(=O)(CC(C)P(C)(C)=O)N(CCNC(=O)CCCCc1ccccc1)CC.C CCCC(CCCO)C(=O)N(CC(C)NC(=O)C1=CCCO1)C C1(CNC(C(COC)NC(c2ccncc2)=O)=O)COCC(C)O1 Cc1ccc(N)c(C(=O)NCCC2(NC(C34CCCCC3C4)=O)CCCC2)c1 Cc1cc(F)cc(C(N2CC3CC(NC(=O)CN4C(=O)CNC4=O)C3C2)=O)c1N C(CC1=CCN(C(c2nccc3n[nH]cc23)=O)CC1)NC(c1ccc[nH]1)=O Nc1cncc(C(=O)N(C2CC2)CC2CCCN(C(c3ccnnc3S)=O)C2)n1 CC1CC2(CCN(C(=O)C(CSC(C)(C)C)NC(=O)C)C2)CO1.CC(F)F C(C(=O)N(C1CCN(C(C2(C(F)(F)F)CC=CC2)=O)CC1)C)(C(C)C)SC CC1(C)CCC(=CC(=O)NCC2(NC(=O)CCC[N+](=O)[O-])CC2)CC1 C(=O)(C(C(C)(C)C)OC)N1CCC(N(C(CS(=O)(=O)NC)=O)C)CC1 N1(C(C(CCC)c2ccccc2)=O)CC2CC(C1)C2NC(=O)COC.C1CCC1 Cc1cc(NC(=O)C(O)CCNC(=O)CC2CCN(C)C2=O)cnc1F Cn1c(=NC(C)(CCC(=O)O)c2ccc(Cl)cc2)n(CCO)c2ccccc12 C1(CC=O)SC(=N)NC1=O.Cc1cc(OCC(=O)NCC2CC2)no1.C c1(C(N2CC(NC(CCSCC)=O)(CO)C2)=O)csc2c(OC)cccc12 N1(C(C2CC(=O)C2)=O)C(C(N2CC(O)(c3nn[nH]n3)C2)=O)CC2CC12 C=C1CCC(C(=O)NCC2CCCCN2C(=O)CNC=O)CC1 N1(C(CSCCCC)=O)CC2CCC(NC(C3CCCCC(=O)N3)=O)(C2)C1 C(C)(C(=O)NOC(CO)CO)N(C(CC=C)=O)C O=C(NNc1ccc(F)c(F)c1)NC1CC(C(O)C(F)(F)F)C1 N1(C(Cc2n[nH]c(=N)s2)=O)CCCC(CCCCNC(=O)CC2CCOC2)C1 C1(NC(Cc2c(CC)con2)=O)CCC2CC1CN2C(c1ccc(F)cc1O)=O N1(C(C=CC(N)=O)=O)CCCCC(NC(c2cc(C3CC3)nnc2O)=O)C1 N1(C(CCCc2onc(CC)n2)=O)CCN(C)CC1CNC(=O)C(C)CC(C)C C1(CC(=O)NC(C2CC(NC(C(C)=C(C)C)=O)C2)C)CSCCO1 N1(C(c2n(C)cc(Cl)c2)=O)CC(C)CC12CCC2.c1(C(=O)N)cnc(C2CC2)o1 N1(C(CCC)=O)CCCC(O)(CCNC(c2cnoc2C2CCC2)=O)C1 C(=O)(C(C)C(=O)OC)NCC(C(=O)N(CCCC)CC1CCC1)C c1(NCC2C(C)CCN(C(=O)CC3CCC(C)CC3)C2)ccc([N+](=O)[O-])cc1Cl c1ccc2c(n1)CCC2=O.C1(C(=O)NCCOCCC)C(F)(F)C12CCC2.N N1(C(C(c2cn(C)nc2)NC(=O)CCc2nc[nH]n2)=O)CC(C)(C)C1C1CC1 C(CNC(c1cn[nH]c1)C1CCC1)(CO)OC CC(C)CC(CNC(=O)CC1CCCN(C)C1)C(=O)NC1(CO)CC=CC1 C12(CNC(c3c(C)ocn3)=O)CCC(CC1)N2C(C1(C)CC1F)=O C(CNC(=O)C(C)SC)(CCNC(=O)COc1ccsc1)OC c1(C(=O)NC2(C)CC2)ccc2c(c1)OCCO2.c1(C(=O)N)cccc2nncn12 C(CC(=O)N1CCC(C(=O)NC2CC(C)(O)C2)O1)c1ccc(C)o1 C(CC(C)C)(C(=O)NC(C)C=CC(=O)NCCC(C)C(F)(F)F)OC CN=c1[nH]c(=NCC2CCC(O)C2)[nH]c(=NCCC(F)(F)Cl)[nH]1 C(=O)(CC(C)CC(C)C)N1CCN(C(CCCc2onc(C)n2)=O)CC1C(F)F C(c1ccccc1[N+](=O)[O-])=CC=O.c1(SC)ccccc1C(=O)NC.C1CC1 Cc1cc(Cl)c(C(N2CC(CCNC(=O)C(F)CC3CCC3)C2)=O)cn1 N1(C(CC(C=C)C)=O)CCN(C(=O)CCCC#N)C(c2cccc(F)c2)C1 N1(C(c2c(C)n(C)nn2)=O)CCC2(CC1)CC2CNC(=O)CC1=NNC(=O)CN1 C12(Nc3nc(C)c(C)s3)CCCC1CN(C(c1cc3c[nH]nc3s1)=O)C2 C(=O)(C(O)CCCNC(=O)C(F)C(C)C)NCC(CO)OC C1(NC(c2ccc(C(C)(F)F)cn2)=O)CN(C(=O)CC2(C)CCCO2)CC12CC2 N1(C(C(=O)N(C2CC2)Cc2n(C(C)C)ccn2)=O)CC(CO)C2CC12 C1(NC(CC(CC)SC)=O)CC2CC(C1)CN(C(C13C4C5C1C1C3C4C51C)=O)C2 N1(C(CC(CC)SC)=O)CC2(CO)CC1(C(N1CCC(COC)C1)=O)C2 c1(C(=O)NC2C(C)CN(C(c3ccoc3)=O)C2)cnc2n1CCOC2 C1(C(c2n(C(C)(C)C)nnn2)NCC=C2CCSCC2)C2CC3CC(C2)CC1C3 CC1CCC(NC(=O)C=CC=O)CN1C=O.c1nnc(O)s1.C(C)(C)C.N O(NC(=O)C(O)C1=CCCCC1)CCNC(=O)C=CC1CCOC1 Cc1ccc(S(=O)(=O)NCCc2cncnc2)cn1 C1(C(=O)NC(C(=O)NC2CC(CC)C2)Cn2ccnn2)CC2(CSC2)C1 c1(NC(CC)=O)cccc(C(N2CC(C)(NC(C3C4COCC34)=O)C2)=O)c1 Cc1cc(C(=O)NCC(C)N(C(=O)CCOC2CCOCC2)C)cnc1C(F)F C(CC(=C)C)(C(=O)N1CCC2CC12)NC(c1n(C=C)ncc1)=O c1(C=O)ccc(S(N)(=O)=O)o1.N1(C(C(C)CO)=O)CCCC(F)C1.CC(=O)N N1(C(C(C(C(C)C)O)(F)F)=O)CCC(C2CN(C(=O)C3CC3)C2)CC1 c1(OCC)cccc2[nH]c(CNC(=O)C(C)SC3(c4ccccn4)CC3)cc12 N1(C(CCC2N(C(C3CC(C)(CC)C3)=O)CCCC2)=O)CC(F)CC(F)C1 c1(NC(CCC2N(C(c3c(C)sc(O)n3)=O)CCC2)=O)ccc2c(c1)CCC2 C1(C(=O)NC2C3(CC(NC(=O)CCC(F)F)C3)C2)CCn2ccnc2C1 N1(C(c2nc(CC)oc2)=O)CC(NC(c2sc(F)cc2Cl)=O)CC2(CCC2)C1 c1(C(N2CC(C)(c3cn(-c4cnn5ccsc45)nn3)C2)=O)nc[nH]c2ncnc1-2 CC1CN(C(=O)COC2CCN(C)CC2)CCN1C(c1csc(C2CC2)n1)=O CN1CCC(C)(C(=O)N(CCCCCNC(=O)CCCc2ccsc2)C)C1 c1(C(=O)NC2(CO)CCCN(C(c3c(CC)ccs3)=O)C2)cn2c(n1)COCC2 C(=O)(CCCn1cc(C(O)C(C)(C)C)nn1)NCC(C)(C)C1CC1 CC(C(CCc1ccccc1)NC(c1cnc(O)o1)=O)NC(=O)Cc1csnn1 c1(C=O)ccnc(Cl)c1O.Cc1c[nH]cc1C(=O)N.C1(CC=CC=O)CCC1 c1(CC)cc(OCc2ccccc2SC(c2ccc(Br)cc2)C(=O)O)ccc1O c1(C(=O)OC)cnc(C(=O)NCCCCC(C)NC(=O)CCC2CC2)c(N)c1 c1(C(=O)NCCCN(C)C(C2CCC3C2C3(F)F)=O)cc([N+](=O)[O-])n[nH]1 c1(CCN=C(NC(C#C)COC)NCC(C)C)c(C)[nH]c2c(C)cccc12 Cc1cn2c(n1)CCC(C(=O)NC1CC(O)CN(C(c3sc(F)cc3C)=O)C1)C2 C(=O)(C1=CS(=O)CCC1)N.C1(NC(c2c[nH]nc2C(F)(F)F)=O)CCCCC1 c1(NC(C(n2c(-c3c(OC)nccc3C)ncc2)C)=O)ccc2occc(=O)c2c1 C1CCCN(C(C)=O)C1.c1ccn[nH]1.C1(OCC)CC(CC(=O)N)C1.CC=O C1(O)(C(=O)NCC2CCC(F)CC2)CCc2ccccc2C1 N1(C(c2coc(CC3CC3)n2)=O)CCC(F)C1.C12(C(=O)N)CCC(CC1)C2 CC1(C)C(NC(C2CCCCC2(C)NC(=O)Cc2cnoc2)=O)CC1(F)F N1(C(C2C(C)CC2)=O)CCC(C(C)(C)NC(c2ccccc2)=O)CC1.C1CC1.O c1(C(=O)NCC23C(CN(C(c4ccnc(C)c4C)=O)C2)C3)ccc(C)c(F)c1F C1(CC(N2CCC(SC)CC2)=O)CCCC12CN(C(c1ncc(F)cc1F)=O)C2 CC1CCCN(C(c2c(Cl)nsc2Cl)=O)C1C.C1(C=O)(C=O)CC1.C1CC1.N N1(C(C2CC(SC)C2)=O)CCC(O)(CC)CC1.c1(CC(=O)N)ncc(Cl)cc1F C1(C(=O)NC(C(=O)NCCc2n(C)nnc2)CC2CCC2)CCC2(CC2)C1 c1(CC(=O)NCCNC(C2C(COC)C2)=O)cccn1C.C1CC1.C c1(NC2CCCN(C(c3c(C)c(Cl)cnc3)=O)CC2)ncc([N+](=O)[O-])cc1Cl n1(CC)nc(C(=O)NC2(C)CN(C(=O)C=CC(=O)N(C)C)C2)c(Br)n1 C1(OC)(CNC(c2csnn2)=O)CCN(C(C2CC2C2CC2C)=O)C1 CC(C(=O)OCC1CC1)OC1CN(C(=O)C(=O)N(C)C)C1 c1(C2C(NC3CCN(C(c4cn(C)nc4)=O)C3)C2)cc(F)cc(F)c1 CCC1=C(C(=O)NC2CC(OC)CN(C(=O)CC(C)CN(C)C)C2)SCCO1 C(CC(C(=O)NCCC1CC(C)(C)C1)NC(=O)CC1CCCO1)OCC c1(COCC(=O)NCC2(O)CN(C(=O)COC(F)F)C2)ccncc1 C1(NC(C(CCN(C)C)NC(CC2(OC)CCC2)=O)=O)CN2CCC1CC2 Cc1ccc(C(N2CCC(CCN(C)C(c3ccc(C)s3)=O)CC2)=O)c(O)n1 Cc1nc(C(F)(F)F)ccc1C(=O)NC.C1COCCN1C(=O)Cc1cccs1 C1(NC(CC2(C=C)CC2)=O)CN(C(=O)CCc2cc(C)nc(C)c2)CC2(CC2)C1 N1(C(C(CC)(C)O)=O)CCc2ccc(-c3cc(C(F)(F)F)ccc3F)cc2C1 C1(NC(C(C(C)C)c2cnn(C)c2)=O)CCN(C(c2ccc(Cl)cc2)=O)CC1F N1(C(CCC=CCC=C)=O)CCCN(C(=O)C(COC)OC)CC1 c1(CC)nccc(C=O)n1.C1(C(N2CC(C(N)=O)C2)=O)CCC(N(C)C)O1.N C1(C(C)NC(=O)Cc2ccsc2)CCN(C(=O)Cc2ccnnc2O)CC1 c1(C(=O)NCC2(CNC(CC(COC)O)=O)CC2(F)F)c(C)ncn1OC C#CCCN=C(NCC(c1ccc(C(F)(F)F)cc1)O)NCC(C)CC(C)C N1(C(C2(C)CCC(=O)C2)=O)CC(CNC(c2scnc2Cl)=O)C(F)(F)C1 C12(NC(c3cn(CC)nc3)=O)CCOCC1CN(C(c1nc(Cl)cs1)=O)C2 N1(C(c2[nH]cc(C)c2)=O)C2CCC1CC(C(=O)NCC1(C)CCCC1O)C2 N1(C(C(CSC)O)=O)CCC(CNC(C2CCCN2CC(F)(F)F)=O)CC1 c1(C(N2CC3(CCN(C(=O)CC4CCC(O)C4)C3)C2)=O)cc([N+](=O)[O-])cnc1O c1(C(=O)N)cc(S(N)(=O)=O)co1.c1(CC)cc(C(=O)NC(C)CC)nn1C N1(C(C2CCC(C)(C)C2)=O)CCCN(C(c2ccc(F)c(O)c2F)=O)CC1CO c1(CCC=O)ccc(Cl)cc1Cl.C(C=O)OC.C1CC1.C(=O)(C1CC1)NC N1(C(C(C)(C)SC)=O)CCN(C(C2CCCC(O)C2)=O)CC(C)(F)C1 C=C(C)CC(C)C(=O)NC1CN(C(=O)CCCSC)CC1c1ccccc1F C1(C(c2ccon2)=O)OCCC1CNC(C1CN(C2CCC2)C1)=O.C1CC1 C1(NC(CN(C2CCC2)C)=O)CC2(C1)CC2NC(=O)CC1C=CCC1 N1(C(CNC(C)=O)=O)CC(NC(c2csnc2Cl)=O)CC(O)C1 CN1CCN(C(=O)CCOCC(F)F)CC1C(=O)NCC(C)(CO)CO CC(CC1CC1)C(=O)NCCCCNC(=O)COC1CCCOC1 C(=O)(C1=CCCCCC1)NCCC(CNC(c1cc(O)nc(O)n1)=O)OC N1(C(C(CC)(C)F)=O)CCC2(CCOCC2)C(CNC(=O)Cn2cnnn2)C1 CC1(C=CC(N2CCN(CC(N3CCC(NC(N)=O)C3)=O)CC2)=O)CCOCC1 C(=O)(C(C)(C)S(C)(=O)=O)NC1CCN(C(CC(=O)NCC)=O)CC1CC CC(C(=O)NCC1CN(C(C2(N3CCCC3)CCC2)=O)C1)n1cccn1 C1(C(=O)NCC2CN(C(=O)CCCc3ncco3)CC2O)COC2(CCC2)C1 C1(NC(c2c(C)nns2)=O)CCC(F)(CNC(=O)C(C)(C)n2cnnn2)C1 Cc1nc2ccc(NC(=O)C(N3CCC(O)C(c4ccccc4)C3)=O)cc2s1 c1(C(=O)Nc2cccc(-c3cnn[nH]3)c2)cnc2ccc(Br)cc2c1 C(=O)(C(CC)CC(C)C)NCC(C(=O)NC(CCC)C(C)(C)C)N(C)C C(CN=c1[nH]c2ccccc2o1)(C1CC1)NC(CCCCOCCC=C)=O CN1CCC(C(=O)NC2CC3CC(NC(=O)CC4(C)CCCCC4)C2C3)CC1=O c1(-c2n(C)ncc2)cnc2cc(C(N3CCNC(CO)C3)=O)ccn12 c1(C(=O)NC2C=CCN(C(CCC(=C)Cl)=O)C2)cnc(CO)nc1C Cc1ccnc(C(=O)NCC(CC2CC2)C(=O)N2CC(O)(C(F)(F)F)C2)c1F CC1CN(C(c2nc(C(C)(C)C)n(C)n2)C(=O)NCc2ccco2)CCO1 Cc1ccnc(C(N2CCOCC2CC(N2CCC(CC3CC3)CC2)=O)=O)c1F C1(C)(C(=O)NC(COC)C2CC2)CCCN(C(C2(C(C)=O)CC2)=O)C1 c1(C(=O)NCCN(C(C)C)C(C2(CF)CCC2)=O)c(F)ccc(O)c1F n1(CC(N2CCS(=O)(=O)CC2)=O)ccc2cc(C3=CCNCC3)ccc12 CC(C)(C)CC(CO)NC(C1CC(F)CCN1C(c1ccc(CO)nc1)=O)=O N1(CC)CCN(C(C2CCCCC2CNC(C2(C)CC2C)=O)=O)CC1=O CC(CN=c1cc[nH]cc1S(=O)(=O)N1CCSC1(C)C)c1ccsc1 C(c1ccc(C)cn1)=CC(=O)N(C(CNC(Cc1cccc(CC)c1)=O)C)C N1(C(CCC(=O)NCCC)=O)CCCC(O)(CNC(C2CC2C)=O)C1.S c1(CC(=O)N(CC(O)CN(C)C(C2CCS2(=O)=O)=O)C)ccccc1Cl c1(C(=O)NC2C(C)CCN(C(C(CC)CC)=O)C2)ccc2c(c1)COC2 n1(CC(=O)NC)[nH]c(=NC(=O)Cc2cn(C)nc2C)cc1C C(=O)(C(C(C)O)N1CCCCC1)N(C1CCN(C(Cc2c(C)non2)=O)C1)C c1(NC(C(=O)NCCCN2CCCNC2=O)=O)ccnc(Cl)c1I C1(C(N(C)CCNC(C2CC2c2cnc[nH]2)=O)=O)CCC1(F)F N1(C(CC(C=C)C)=O)CCCCC(CNC(c2snnc2CC)=O)C1 C(c1ccccc1C#N)=CC(=O)NCCC1N(C(C(C)CF)=O)CCCC1 C12(C(=O)NCC#CC(=O)NCCCC(=O)NC3CC3)CCCC(CO1)C2 C1(NC(C(c2cccc(C)c2)C)=O)CC2(CCN(C(C3CC34CC4)=O)C2)C1 Cn1nnc2c1CCC(C(N1CCC3CCC(C1)N3C(=O)Cc1ccns1)=O)C2 C(=O)(C1=NNC(=O)CC1)N1CCN(C(CSC2N(C(C)(C)C)CC2)=O)CC1 Cc1cc(C(=O)NC2(CNC(C3CCCCCCC3)=O)CCOCC2)ncc1F Cc1nn(CC(=O)NC2COCC2NC(=O)C2=CCCCO2)c(C)c1Br C1(C2(NC(c3cc(Br)c(C(F)(F)F)[nH]3)=O)CC2)CCCCN1C1CCCC1 C(=O)(C(=O)CC(C)CC)NC(CC(=O)NCC(C=C)O)C(C)C c1(C(N(CCNC(=O)CC(C)=C(C)C)CC)=O)cccc(C(N)=O)c1F CC(C)CC(CNC(=O)C=Cc1ccccc1)C(=O)N1CCC(OC2CCC2)C1 C(=O)(NNc1ccncn1)Nc1c(C)c(Cl)c(Br)cc1 C1(CNC(c2ccc(F)s2)=O)CC(NC(C2COCCO2)=O)C12CCC2 C(=O)(C1=CCOCC1)N(C1CCCCN(C(c2cccc(C3CC3)c2)=O)C1)C Cc1ncc(C(=O)NC2(CCC(N3CCC4(CCO4)C3)=O)CCCC2)c(=N)[nH]1 C1(CC#N)CCCN(N2CC3(CC(O)C(O)CO3)C2)C1 c1(NC(CNC(CC2C(C)(C)CC2)=O)=O)ccccc1.C1(C(=O)N)COCCO1 CN1CCCC2(CCN(C(=O)C=Cc3cc(Br)c4c(c3)OCO4)C2)C1 c1(C(N2CCN(C(c3cnc4ccccn34)=O)C3CC23)=O)cc2cnccc2o1 C=CCCC(=O)N(CC(=O)N(CC(O)CC)C)CC1CC1 c1(C(N(CC(CNC(C2CC(CC)(CC)C2)=O)C)C)=O)cccc2c1NCCC2 C1(C2N(C(C(C)NC(c3ccco3)=O)=O)CCC2)CCN(C(=O)C2=CCC2)CC1 CCC(CCCC(=O)N1CCCC2(CC1)N=N2)NC(C1CN2CCN1CC2)=O C1(CC(=O)N)COC(C)(C)CO1.CCCC(C(=O)NC(C1CCCC1)C)N(C)C c1(CC)cc(C(N2CCC(O)C(NC(c3csc(Cl)n3)=O)C2)=O)cc(F)c1 Cc1ccc(-n2nnnc2CNc2cccc(C(F)C(F)(F)F)n2)cc1 N1(C(CC2C(C)CCN(C(=O)CCCCC3CC3)C2)=O)CC(=O)NC(C)(C)C1 c1(OCC)ccc([N+](=O)[O-])c(C(=O)NC2CC(C)N(c3cncc(Cl)n3)C2)c1 C1(CCC(=O)N(C(C)C(=O)NCC2CCCCS2)CCC)CCOCC1 c1(C(N(CCCC)CC)=O)cnc2c(F)cccn12.C1(O)(CC(=O)N)CCCC1 C#Cc1ccc(C2(NC(=O)C(C)CN(C)C)CC2)cc1Cl Cc1nc2cc(C(N3CCCC(NC(=O)Cc4cc[nH]n4)CC3)=O)ccc2n1C C1(CC)(CC)CCN(C(=O)C(CCNC(C2CCSC2)=O)OC)C1 N1(C(C(CC)C(C)(F)F)=O)CC(C)(C)C(NC(=O)C(O)c2ccsc2)C(C)(C)C1 CON(CCC(=O)NC1CC2(CCO1)CC2)C(=O)C(C1CCCC1)N(C)C c1(CC(N2CCC(C(=O)NC3CCC(=O)NC3=O)C2)=O)ccc2ncccc2c1 C1(NC(Cc2c(C)ccs2)=O)COCCN(C(=O)CC(C2CC2)C2CC2)C1 N1(C(c2oc(C(=O)OC)c(C)c2)=O)CCC(NC(=O)CC(C)(C)C)C(O)C1.S Nc1c(I)cc(F)c(NCC2CCCNC2=O)c1F C=CCCCN=[N+]=[N-].C(C(=O)N1CCCC1C(=O)O)C(C)C.n12cc(nn1)CCC2 S(=O)(=O)(c1ccc(Cl)c(Cl)c1)Nc1sc2ccc(C(=O)OC)cc2n1 N1(C(Cc2n(C)ncc2)=O)CCN(C(=O)CC2(CO)CC2)CC1c1ccncc1 Cc1ccc(C)c(CC(=O)NCC2CCN2C(=O)CN2CSCCSC2)c1 N1(C(C(C)(C)C)=O)CCCC(C(=O)NC2CCCCC2NC(=O)CNC=O)C1 c1(OC)cc(C(=O)NC)nn1C.C(=O)CC(C)C1CCC1.C1CC1.C(C)=O N1(C(C(=O)NCC2(OC)CCCCC2)=O)CC(O)(C#CBr)C1 Cc1ccc(C(C)C(=O)NC2(CNC(=O)Cc3ncccc3C)CCCC2)cc1 c1(CC(=O)NCC2CNC3CCCCC23)n[nH]c2c(Br)cccc12 C1(C(N(C2CCN(C(c3cc(C4CC4)on3)=O)C2)CCO)=O)CCOC(=O)CC1 c1(OCC(=O)NCC)cc(F)ccc1F.C1(C=O)CCCC1c1nc(S)n[nH]1.N N1(C(C(c2ccccc2Cl)OC)=O)CC2CC(C1)CN(C(=O)Cc1ccoc1)C2 c1(CN(C)CC2CCCN(C(c3ccc(Cl)c(I)c3)=O)C2)c(F)cc(Br)cc1Br CC(C)CCCCNC(N1CCC1CS(C)(=O)=O)=O N=C1NC(=O)C(CC(N2CCCC(C)C2)=O)S1.c1(C=O)cncnc1C(=O)O.N c1(C(=O)NCCCCNC(C2COCC(C)O2)=O)cccc2c1OCCC2 CN1CC(N=c2c(C#N)c[nH]c3c(F)cccc23)C1C(F)(F)F n1(CC(=C)C)nnnc1C(c1ccc(-c2cccs2)s1)NCc1cc(C)no1 CCCCCC(O)C(=O)N(CCN(C(=O)C(CC)C(C)O)C)C(C)C c1(N2CCC(CNC(COc3c(C)cccc3)=O)C2(C)C)ncc2ccnc-2[nH]1 CCCC(C(=O)OC)C(=O)N1CCCC(CC(=O)N(CC(F)Cl)C)CC1 c1(C(N2C(CNC(C(CCC)C)=O)(COC)CCC2)=O)cc2cccnc2s1 C(=O)(CCCCC(F)(F)F)N(C1CCN(C(c2n[nH]c(C)c2[N+](=O)[O-])=O)C1)C C(CCCCCNC(c1ccco1)=O)NC(=O)CCc1nnc(C(F)F)o1 C(=O)(C1OC(=O)c2ccccc21)NC1CN(C(CCC(=C)Cl)=O)C(C)(C)C1 n1(CC(=O)N(CCCC)CC)nc(C)ccc1=O.c1(C=O)cccs1.C(=O)C c1cnc(C)c(C#N)c1.c1(C(C#C)NC(=O)COCC=O)cccc(C)c1.O C12(NC(C(SC)SC)=O)CCCC1N(C(=O)CC(C)C(F)(F)F)CC2 Cc1ccc(C(=O)NC23CC(C)(C2)C3)nc1.c1(C(C(=O)N)O)cnn(C)c1 C1(C(=O)OC(CC)C(N)=O)CC2CCCCC2N1C(=O)OCC(C)(C)C Cc1cc(C(=O)OCc2nc(O)c3sccc3n2)cc([N+](=O)[O-])c1O C12(C(=O)NCC(CCCC)O)CC(CO)(CN1C(=O)CC1CCC=CCC1)C2 C(CCCCCCC(=O)N1CCCC(N(C)C(C)=O)C1)SC c1(C(N(CCCC(C)(C)C)C)=O)cn(C)c(=O)c(C)n1.C(CC=O)=CCC.N N1(C(CC(C)O)=O)CCC(C)N(C(=O)CC(C)C2CC2)CC1 N1(C(CC2(OC)CCOCC2)=O)CCCC12CCN(C(c1occc1C)=O)CC2 C1(C(N(C)CC=CC(=O)N(C(CF)CF)C)=O)C(C)(C)C1(F)F N1(C(Cn2ccc(C=O)n2)=O)CC2(C1)CN(C(=O)Cc1ncn3c1CCC3)C2.C c1(NC(c2cc(OC)ncc2F)=O)nccc2[nH]ccc12 C(=O)(CC(C)(C)SC)N(CC(CN(C(C(COC)N(C)C)=O)C)O)C Cc1cc(-c2nc(C(=O)NCC3COC3)c(C)s2)cc(F)c1 c1(NC(CC2(NC(C(C)SCC)=O)CCCC2)=O)cnc2ccccc2n1 C1(C=O)CCC(C)(C(=O)O)C1.Cc1nc(CC(=O)N(CCC)C(C)C)cs1.N c1(Cn2cc(CCS(N)(=O)=O)nn2)ccccc1S(N)(=O)=O C1(NC(C(C)CS(C)(=O)=O)=O)CC2CCC1CN(C(=O)CCN1CCOCC1)C2 C(c1ccncc1)=CC(=O)NC1CCOCC1NC(C1(CO)CCCCC1)=O C1(CC=O)CCS(=O)(=O)C1.C1C2CC1N(C(=O)Cc1ccc(OCF)cc1)C2.N C1(c2nnc(C)o2)COCCN1C(=O)CSc1ncc(-c2ccc(F)cc2)o1 N1(C(c2[nH]cc(C#N)c2)=O)CCC2CN(C(C3CC4(C3)CS(=O)(=O)C4)=O)C2C1 c1(C(=O)NC2C(NC(C(CC)O)=O)CC2)ccc(S(=O)(=O)CC)c(C)c1 N1(C(C(COC)NC(C)C(=O)OC)=O)CCc2sccc2C1 N1(CC2(OC(C)C)CCOC2)CCC(=O)N(CC(C)CC(F)F)C1=O c1(N(C)Cc2ccc(OC)cn2)ncccc1S(=O)(=O)N1CC(O)CCC1C N12CCC(C)(C)CC1C(=O)NCCCSCC2=O.N1(CC)CCCC1CF C1(C(N2C(CC(N3CCC(CC4CCC4)C3)=O)CC2)=O)CC2C=CC1O2 C12(NC(C(COC)N(C)C)=O)CC(C)(C1)OC21CN(C(=O)C(C)(CO)O)C1 C1(C(=O)NCC=CC(=O)N(CCCC)CCCC)CCCC1C(C)=O C1(C2(O)CCCOC2)(CNC(=O)C(F)(F)Oc2ccc(Cl)cc2)CC1 N1(C(C(C)=NOCC#N)=O)C2CC1CN(C(c1ccc(N)c(F)c1)=O)C2 C1(NC(=O)CNC(=O)C(O)Cc2ccccc2Cl)CCCCC1c1nc[nH]n1 c1(CC(=O)NCCC2N(C(C(CC)OC)=O)CCCC2)ccc2nc(O)[nH]c2c1 CC(CN(C(=O)CCCC1CCCO1)C)C(=O)N(C)CCOC(F)F C1(N(C(C(C)C)=O)C)CCC(NC(C23CCC(CC2)C3)=O)CC1 Cn1nc2c(c1C(N1C3CCCC1CN(C(C1CC4CC4C1)=O)C3)=O)COCC2 C1(CN(C(CC)=O)C)CN(C(C2(CCN(C)CC)CC2)=O)CCO1 C(=O)(CCC(CF)CF)N1CCC(CNC(C=Cc2n(C)ncc2)=O)C1 c1(CNC(C(=C)CN(C)C)=O)cc(-n2cc(C)cn2)ccn1 N1(C(C2C3CN(C(C4=C(C)CCC4)=O)CC32)=O)CCC(C2CC2)C1CO N1(C(c2cc(OCC)n[nH]2)=O)CC(CCNC(c2ccsc2)=O)C(C)C1 C#CCC(C)(C(=O)N1CCC1)NC(=O)C=C(C1CC1)C1CC1.C(C)=O.C CCCCC(O)C(=O)NC1CCN(C(=O)Cc2cc(F)ccc2O)C12CC2 C1(C(N(CCC#C)CCO)=O)CC(O)CN1C(=O)C(O)CC1CC1 C(=O)(CCCCCCN=[N+]=[N-])NCC(CC)Nc1ncnc2c1nnn2C CCCCN=c1nc(N2CCC(CCC(=O)NC)CC2)c2ncccc2[nH]1 Cc1nc2ncnn2c(C)c1CC(N1CCCOC(CNC(=O)C(C)CF)C1)=O N1(C(c2cnc(CC)nc2O)=O)CCC2CCC(C1)N2C(c1ccc(C)nc1)=O C1(CN(C(c2cnc(C)o2)=O)C)C2CN(C(=O)C(C)Cc3ccc(O)cc3)CC12 c1(C(=O)Nc2nc(-c3ccc(C)cc3CO)sc2C)c(C)cc(C#N)cc1Cl O=C(C1Cc2ccccc21)NCCC1(O)CCN(C(C2CCC2)=O)CC1 C(=O)(CCC[N+](=O)[O-])N.c1(CSCC)ccc(C(N2CCCCC2CC)=O)cc1 CC1CC(NC(=O)C(C)(c2ccccc2)N(C)C)CCN1C(C1CSCCS1)=O O=C(C1CCCc2sccc21)NC1CCN(c2cc(-c3ccccc3)ncn2)C1 N1(C(CC2(NC(c3c(CC)con3)=O)CCCCC2)=O)CCC(O)C(F)C1 c1cccc(C(N)=O)c1.CC(CCCO)NC(C1(n2cc(CN)nn2)CC1)=O.C C(CN=C(NCC(C)(C)C(F)F)NC(c1cccc(C)c1C)C)C1(SC)CC1 c1(C(=O)NCC(CNC(C2C(C)(C)C2)=O)F)cocc1C(N)=O C(=O)(C1=CN(C=O)CC1)N1CC(C)C1.C(=O)C=CC1CC1.C(C)(C)C.C N1(C(C=C(C)c2cccs2)=O)C2CCC1C(NC(=O)CCn1cccnc1=O)C2 C(=O)(NN1CCOCC1)c1cc(C#N)ncc1 C1(C(=O)NC2C=CCN(C(C3CCCC(=O)O3)=O)C2)CC12CC(F)(F)C2 N1(CCCNC(CN2CCC(C)C2)=O)CCN(C(C2CCC2(F)F)=O)CC1 CCCCC(O)C(=O)NC1CCCN(C(C2(COC)CCCC2)=O)CC1 c1(C(=O)NC(CNC(c2cnc(C(C)OC)s2)=O)CO)ccc(C)nc1N CC1C(C)N(C(=O)C=C2CCCCC2)CCN1C(=O)CCCn1cncn1 C1(NC(C2CCC(=C)CC2)=O)CCC(C)N(C(=O)Cc2c(Cl)cnn2C)C1 CC#CCCCC(=O)NCC1COC(CNC(=O)CCCCCn2cnnn2)C1 C1(CC#N)CCCN(C(c2ccnc(F)c2)C(=O)NCC2CC2)C1 N1(C(C2C(C)(C)CCC2)=O)CC2(CCCN(C(=O)C=Cc3ccc[nH]3)C2)C1 C(=O)(CCCC(F)(F)F)NCC1OCCN(C(c2n(C)ncc2C(F)F)=O)C1 c1(N2CCC(NC(c3c(C)cccc3O)=O)C(C)(C)C2)ncnc2n[nH]c(Br)c12 c1(C(N)=O)cccc(C(=O)NCC2(NC(C3CCNC3=O)=O)CCOC2)c1F N1(C(C(CNC2CC(C(=O)OC)C2)CC2CCCC2)=O)CCOC(C(F)F)CC1 Cc1cn2c(C(N3CC(NC(=O)Cn4cnccc4=O)C(O)C3)=O)c(C)nc2s1 c1(CNC(C2CC(F)(F)CN2C(c2ccnnc2)=O)=O)ccc2c(c1)CCC2 c1(C(=O)NCC(CC)NC(c2cnc(C)[nH]2)=O)n[nH]c2ccc(Cl)cc12 C1(CNC(C(CCC)C)=O)CN(C(=O)COc2nn(C)cc2Br)CC12CC2 C1(C(=O)NC2(CO)CCN(C(c3c(SC)cccc3)=O)C2)CC(=O)NC(C)C1 c1(C(C(=O)NC2COC2)N(CCCSCC)C)ccc(-c2cn[nH]c2)cc1 C(CCC(=O)NCC1CC1C(F)(F)F)OC.C1(C)(CC=O)CCCCC1.N c1(C(c2nnnn2CCC2(C)CC2)NC(CC)COC)cnc(OC)cc1C C1(C(=O)NCCC2CC(NC(C(=C(C)C3CC3)F)=O)C2)CNC(=O)C1 c1(CC)nn(C)c(C(=O)NCC2CN(C(=O)Cn3cncc3C)CCO2)c1Cl C(=O)(C#CC1(C)CC1)NC1C(C(C)C)N(C(C2CC(C(C)C)C2)=O)CC1 NS(=O)(=O)c1coc(C(=O)NCCCCNC(C2CC3(COCCO3)C2)=O)c1 N1(C(C2CCCN(CC)C2)=O)CCOCC(C(=O)NCCCn2cnnn2)C1 C1(CC(N2CCC(OC)CC2)=O)C2CCC(C2)N1C(c1csc(=N)[nH]1)=O C#CCCCCCC(=O)NCC1CN(C(c2cc(F)ccc2O)=O)CCC1C C(=O)(CC1CCc2ccccc21)NCCN(C)C(C12CCC1CC2)=O c1(C(=O)OC)cc2cc(NC(=O)NCC(C)(C)CN(C)C)ccc2s1 N(C(=NCCCCl)NCc1nc(C2CCCCC2)no1)C1CC(C)(F)C1 CCC1=NOC(C(=O)NC2(CO)CCN(C(c3cc(C)no3)=O)C2)C1 C(C(CC(C)C)C(=O)N=c1cc2ccccn2[nH]1)NC(C(C(C)C)OCC)=O c1(C(N2CCC(O)(CC)C2)=O)ccc([N+](=O)[O-])cc1.C12CC(C=O)(C1)C2.C Cc1cc(C(N)=O)cc(C(=O)NCC(C)CO)c1.C1(CC=O)CCC(C)(C)O1 CC(C)CCCC(C)C(=O)N(CCC(C)(C)NC(=O)C(C1CCOCC1)F)C Cc1cccc(F)c1C(=O)NC(C1CCN(Cc2ncsc2Br)C1)C Cc1cc(C)c(CNC(=O)CC(C)NC(=O)C(C)NC(=O)C2CC2)s1 c1(COC)ccccc1CC=O.C12CC1CN(C(C1(C(F)F)CCCC1)=O)C2.N N1(C(COCc2nnc(C)s2)=O)CC(CNC(=O)CCO)CC1C.C1CC1 Cc1cccc(C=CC(N2CC(NC(c3ccnnc3S)=O)C3(CC3)C2)=O)c1 CC1(C)C(CC2CC2)CCN1C(c1cc(Br)no1)=O.c1cn[nH]c1.C(=O)(C)N c1(C(N2C(C)CN(C(CCC(=C)Cl)=O)C(C)C2)=O)cc2cc(F)cc(F)c2[nH]1 Cc1cnc(C(=O)NC(C)C(C)C(=O)N2CC(O)CC2CO)c(F)c1 C1(CNC(Cc2cc(C)ns2)=O)C2CN(C(c3cc(C(N)=O)cn3C)=O)CC12 N1(C(CC2(OCC)CCC2)=O)CC(CNC(C2CC2C)=O)(COC)C1 CC(C)CC(C(=O)NC1CC(CNC(=O)C(C)(C)C(C)O)C1)C(C)C C(=O)(C1CCc2ccccc21)N(C(=O)CN1CC2CC2C1)Cc1cc(C)ncc1 C1(C(=O)NC2(COC)CCCC2)N(C(c2[nH]ccc2C)=O)CCC1(C)C CC(CC(F)(F)F)C(=O)NCC1CCC(NC(C23CCN(CC2)CC3)=O)CC1 C1(CNC(CNS(C)(=O)=O)=O)CC12CCN(C(=O)CCCS(N)(=O)=O)CC2 C(CCC(C)(C)NC(=O)CCC)NC(C(C1CC1)SC)=O.C1CCC(C)CC1.O C1(C(=O)NCCCCNC(c2ccc([N+](=O)[O-])o2)=O)CCCCC1(F)F C1(CC(=O)NC(C(=O)NC2C(OC)CCC2)C2CC2)CC2(CC2)CO1 Cc1ccc(C(=O)NCC2CCCN(Cc3cncc(Cl)c3)C2)c2ncccc12 c1(OC)cc(C(N2CC(NC(=O)C(C)(C)CF)C(C)C2)=O)c(Cl)cn1 N1(C(c2c(C)ccnc2)=O)CC(O)CC1(C)C(=O)NCCc1ccc(F)nc1 Nc1ccc2nccc(C(N3CCC(O)(c4nc(C5CC5)no4)C3)=O)c2c1 N1(C(Cc2cc(C)sc2)=O)CC(CNC(=O)C(C)C(F)F)OC2COCC12 N1(C(CC2CCC(C)C2)=O)CC2(CCCCN2C(c2cnn[nH]2)=O)C1 c1(N2CCC(CC=C)(NC(c3ccc(C4CC4)s3)=O)C2)nc2ccc(Br)cc2o1 Cc1cc2cc(C(=O)N(CCNC(C3(CCF)CC3)=O)C3CC3)oc2cc1C CC(C)C(F)C(=O)NCCN(C(=O)C(O)Cc1ccccc1)CCO.CCO c1(OC)ccc(C(=O)NCC2(C)CN(C(c3c(Cl)ccnc3Cl)=O)C2)c(I)c1 c1(C(=O)NC2CC(C)(CC)N(C(c3c[nH]nc3C)=O)C2)cncc2[nH]ccc12 C(CNC(=O)CNC(=O)C(F)n1ccnc1)(CO)N(C)C c1(CC(=O)NC(C(C)NC(C(CSC)OC)=O)C)ccc2c(c1)CCCO2 C(C)(C=O)(C(C)C)NC(C)=O.C1CCN(C(C2CCC(=O)CC2C)=O)C(C)C1.N CC1CCC(C(=O)NCC(C)CNC(=O)C(O)c2ccsc2)CC1 c1(C(N(CCCCCNC(C(CC(C)C)OC)=O)C)=O)ccc([N+](=O)[O-])n1C N1(C(c2n(CC#C)ccc2)=O)CCC(O)(CC)C1.C(=O)(C=O)N.CCC(N)=O c1(NC(CC2(C)CCN(C(CCC3(C)CC3)=O)C2)=O)ccc2c(c1)OCC2 CC(O)CCCCCC(=O)NC1(CF)CCN(C(c2cc(C#N)ccc2N)=O)C1 Cc1cc(C#N)ccc1CNC(CC(C)C)C(N)=O CC1(CNC(C2(CNC(C3CCCS3)=O)CCCC2)=O)CCCCC1 C1(CCC)CN(C(=O)Cc2ccon2)CCN1C(C1CC(CC)=NO1)=O c1(C(c2nnnn2C2CC(F)(F)C2)NC2(CC)CCOC2)ncccc1F CCC(C)(C)CC(=O)N(C1CCN(C(c2scnc2COC)=O)CC1C)C N1(C(C(C2CCN(C(c3c(CC)noc3)=O)CC2)C)=O)CC(C)(C)C2CCCC12 C1(N(C(CN(C(C)(C)C)CC#C)=O)C)CC(=C)C1.C1CO1 N1(c2ccc(Cl)cc2)CC(N=c2[nH]c(=NCc3cc(Br)cs3)c3sccc3[nH]2)C1 c1(CC)noc(C(=O)NC2(CN(C(=O)CC3CCCC3C)C)CC2)c1C Cc1nncn1NC(=O)c1ncoc1CNC(=O)C(C)C1CC1 Cc1ncn(C)c1NC(c1ccccc1)=O.C1(C=O)CCN(S(C)(=O)=O)C1.N c1(C=O)cc(Cl)c(N)c(Cl)c1.C(=O)CC(F)(F)F.CCCC(C)NC(=O)C.N N1(C(Cc2ccc(C)cc2)=O)CCCC2(CCCN2C(C2CCC=CO2)=O)C1 N1(CCCC(=O)OC(C)C)CCC2(CC1)CC2C(=O)NCc1nn[nH]n1 N1(C(=O)COCC(F)F)CCC2CN(C(c3c(F)cc(Cl)cc3F)=O)CCC2C1 Cc1cn2cc(C(=O)N(CCC(C(C)(C)C)NC(=O)CCF)C)cc(F)c2n1 CCC(CC)C(C(=O)N1CC(=O)NCC1C(=O)NCCSCCO)OC N1(C(c2c(CC)cccc2)=O)CCC(NC(c2cnc(C)o2)=O)C(CO)C1 CC(CC(=O)NC1CN(C(c2scnc2C(C)(C)C)=O)C1)CC(C)(C)C c1(-c2cnc(COC)[nH]2)ccc(F)c(F)c1C c1(C(=O)NC(CNC(C2CCN(c3n(C)ccn3)C2)=O)(C)C)cc(Cl)sc1Cl N1(C(C2(COC)CCCO2)=O)CCN(C(c2ccc(=N)[nH]c2)=O)C(CCO)C1 C1(CN(C(=O)CSc2nccn2C)C)CCCN1C(C1CC2CC2C1)=O C(C(C)(C)C#CC(=O)N1CC(=O)NC2(CC2)C1)NC(c1c(C)noc1N)=O Cc1cc(Br)ccc1CC(N1CCC(O)(C(C)NC(c2ncn(C)n2)=O)C1)=O C1(COC)CCN(C(=O)C=CC(F)(F)F)C1.C1(C=O)(C2CC2)CCCO1 c1(CCC)n[nH]cc1C(=O)NC(C(=O)N(C)CCOC(F)F)C1(C)CC1 C1(CNC(C(C)=C2CCCC2)=O)CN(C(=O)C(O)C(C)(C)C)CC(C)(C)O1 c1(C(=O)NCC(C)(C)NC(C2CCN(C)C2)=O)cc([N+](=O)[O-])ccc1O c1(C(=O)NC2CCN(C(c3scc(C)n3)=O)CC2F)cc2ccncc2[nH]1 N1(C(C(c2ccccc2)C)=O)CCN(CCNC(=O)C=CBr)CC1CCO Cc1cc(NNC(=O)c2cccc3[nH]nc(O)c23)ncn1 C(=O)(C1CCCc2sccc21)N1CC(O)CCC(NC(c2n(C)c(S)nc2)=O)C1 C1(NC(C2C(C(C)=O)C2(C)C)=O)CCC(C(N2C3CSCC2C3)=O)CC1 Cc1c(C(N2CCC(O)(C(=O)Nc3cc(Cl)ncc3F)C2)=O)cccc1Cl CN1CC(O)CCC1C(N1CCC(CC(=O)NCC2(O)CCSC2)C1(C)C)=O N1(C(COCCOCCOC)=O)CCC2(CC2)C1.C1(C(=O)N)CC=CC1 C(C)(C)(CCCNC(=O)CN1CCOC1=O)NC(Cc1ccc(C)s1)=O N1(C(CCS(N)(=O)=O)=O)CC2CCCC2C1C(=O)NC1CC2CC2C1 C1(CC)CC(N=c2[nH]c3ccc(S(=O)(=O)NC(c4csc(C)n4)C)cc3s2)C1 C1(C(N2CC(NC(C(C(C)C)NC(C)=O)=O)C(C)C2)=O)CCC(N=[N+]=[N-])CC1 CC1C(NC(c2coc(Cl)n2)=O)CCCN1C(C1OCCN(C)C1=O)=O Cc1ccncc1C=CC(=O)NCC(O)CNC(C1CC(O)CN1C)=O N(C1CCCc2n[nH]cc21)C(C=C(CNC(C1N(CC)CC1)=O)C)=O C1(CN(CCNS(NC)(=O)=O)CCN)CCCC(P(C)(C)=O)C1 C1(CC)CN(C(C2CC(N3CCCC3)C2)=O)CCN1C(C1CCN1CC)=O c1(C(=O)NCC(CN(C)C(C2CC3(CSC3)C2)=O)O)ccc(F)cc1O C#CC1CCCN(C(C)C(=O)NC(C)C(=O)OC(C)=O)CC1 c1(C(=O)NCC2N(C(c3c(C)cco3)=O)CCN(C)C2)cnc2[nH]nnc2c1 C(=O)(C1Cc2ccccc21)N(CCC(O)C(C)(C)C)C(CN1CCN(C)CC1)=O c1nnc(C(C)(C)C)n1C(C)(C)C.C(=O)CC(C)O.CCCCNC(=O)C c1(OCC)ncc(C(N2CCC(CC(=O)NC(C)(C)C(N)=O)C2)=O)cn1 Cc1ccc(-c2nnc(CCC(=O)OCCOCCOCC(C)C)o2)cc1 N1(C(c2nsc3c(Cl)cccc23)=O)CC2CCCC1CN(C(C1CC(O)C1)=O)C2 Cn1cc(C(N2CCN(C3CN(C(=O)CC4CCC(O)C4)C3)CC2)=O)c(O)n1 c1(-n2ccc(C)n2)ccccc1C(N1CCC(NC(C2(Cl)CC23CCC3)=O)C1)=O c1(OC)cccc(C=CC(=O)NC2CC(C)C2)c1.c1(C=O)ccc(C)nc1O c1(C2C(N(CC(C)C)C(=O)NC3COCCO3)C2)cccc(C(F)(F)F)c1 C1(C(N2C(C)CC(NC(=O)CCc3cn[nH]c3)C2)=O)CCCCS1(=O)=O C1(CC=O)CCCS1(=O)=O.n1(CC(=O)NCC)cnc(C(F)(F)F)c1.C N1(C(CCc2ccc(C)s2)=O)CCC2CCN(C(=O)CC3=CCCCC3)CC12 C1(C(C)C)CN(C(C2(N(C)C)CCCSC2)=O)CCN1C(=O)CCC#N CC1CN(C(=O)C2=CCOC2)CCC1CNC(=O)CCCc1cccs1 C1(C(=O)NC2CC2CC(C)(C)C)(NC(c2c(C)c[nH]n2)=O)CC(F)(F)C1 c1(C(N(C)CCNC(=O)CCC2CCC(=O)N2)=O)ccc2c(c1)CCCC2 C(C)(CCC(=O)N(CC(C)(C)CO)C1CC1)NC(c1c(C)n[nH]c1)=O C1(NC(C2C(C(C)=O)C2(C)C)=O)CCOC(C(=O)NCc2snnc2C)C1 c1(C=O)conc1C(F)(F)F.c1(C(N(CCC)CC)=O)cc(N(C)C)c[nH]1 C1(O)(CNC(CC2N(C(C)C)CCC2)=O)CCN(C(C2(C)CCOC2)=O)CC1 C(=O)(C1CCc2ccccc21)N1CCC(NC(C2CC=CCO2)=O)C(F)C1 Cc1ccc2cc(C(=O)NC(C)CCNC(c3cc(Cl)c(Cl)n3C)=O)cn2c1 N1(C(c2cnc(CC)nc2)=O)CCC2CN(C(=O)C3=CCCSC3)CCC2C1 C12(CNC(C(C)OCCCCCC)=O)CC1CN(C(C1(CC)CC1)=O)C2.O C1(C(=O)NCCCN(C)Cc2cncc(OC)c2)CCc2nncn2C1 C(CCCC(=O)N(CCNC(C1CCCN1C=O)=O)C1CC1)OC C1(C(=O)NC(C(=O)OCC)C2CC2)CCCCC1.c1(C=O)cnc(O)o1 C(=O)(C(C(CC)CC)OC)N(CCNC(CC=CC)=O)C(C)C c1(OC)cccc(C(O)C(=O)NCC2CC2NC(c2ccc(C)o2)=O)c1 N1(C(C(c2ccc(Br)cc2)C)=O)CC(NC(=O)CN2CCOCC2)CCC1C c1(OC(C)C)cncc(C(=O)N(C)CC2CC2)c1.C(=O)C(F)=C(C)C.C N1(C(C(C)N(C(=O)C=C2CCSCC2)CC2CC2)=O)CCN(C2CC2)CC1 C1(C(C)C)CN(C(=O)Nc2ccc(C3(O)COC3)cc2)CCS1 CC(C)C(C(=O)NC(C)(C)CCNC(C1SCCS1)=O)c1ccc(F)cc1 C(CN=c1[nH]ccc(C#N)c1[N+](=O)[O-])(N(C(C(C(C)C)OC)=O)C)C1CC1 N1(C(c2sc(Br)c(C)c2C)=O)CC(NC(C2CCCO2)=O)CCC(O)C1 c1(OCC(=O)NC2C(NC(C(C=CCCC)O)=O)CCCC2)ccccc1C#N C1(NC(C(CC)COC)=O)CCC2(CCN(C(C3(O)CCCCC3)=O)C2)C1 C1(CCNC(CC(C)N2CCCC2=O)=O)CCCN(C(=O)COC2CCOC2)C1 CCC(CC(C)C)C(=O)N1CCCN(C(c2cnn(C(C)C)c2F)=O)CC1C Cc1cnn(C)c1C(=O)NCC1(C)CCN(C(=O)C=C2CCC(C)C2)C1 C1(NC(CC(C=C)(C)C)=O)CCCC12CCN(C(=O)C(F)CN(CC)CC)CC2 C1(F)(C(N2CC(O)(C(C)NC(CN3C(C)CC3)=O)C2)=O)CCCCC1 N1(C(C(C(C)OC)NC(=O)C=Cc2cccnc2)=O)CCn2nccc2C1 C(C)(C(=O)NNC(=O)CC(C)C)n1cc(-c2c(OCCOC)cccc2)nn1 C1(CC(=O)NC2(C(C)C)CCC2)CN(C(c2cnnc(O)c2)=O)CCC1C C1CCS(=O)(=O)C12CN(C(c1c(Cl)csc1Cl)=O)C2.C1(CC=O)COC(=O)N1.N c1(C(N2CCC(N(CCC)C(c3cc(Cl)n(C)n3)=O)C2)=O)ccc2nc[nH]c2c1 C=CCC(C(=O)N1C(C(=O)N(C2COCC2O)C)CCC1C(C)C)C(C)C CC(CS(C)(=O)=O)C(=O)N1CC2CCC(C1)C2NC(c1ncncc1Cl)=O c1(C(=O)NC2CN(Cc3c(C)cc(C#N)cc3)CC2F)cc2cc(Cl)ccc2[nH]1 C(=O)(C(CCC(N)=O)n1cc(C(O)CC(C)C)nn1)NCCCC(=O)OC C1(CCC)CN(C(C2(n3cc(C)cn3)CC2)=O)CC1C=O.C1CC(O)(CO)C1 c1(CC)cc(F)c(C(=O)NC)c(F)c1.C1CN(C(=O)CCn2ccnc2)CCO1 c1(C(=O)NC2CCC(NC(C=Cc3cncc(C)c3)=O)C2)c[nH]c2nccc-2c1 N1(C(c2ccc(Cl)c(C)c2N)=O)CC2CCCC(C1)N2C(C1C=CCCC1)=O N1(C(C2(Br)CC2)=O)CCC(C(O)CNC(C2CCC(O)C2)=O)CC1 C(=O)(CC(CC(C)C)NC(=O)CN1CCCCC1)N(CC(=O)NCC)C C=Cn1ncc(C(N2CCC(C)C(CC(=O)NOCc3nc[nH]n3)C2)=O)c1N.OC N1(CCNC(CN2C(C)CCC2)=O)CCCN(C(=O)Cc2ccn(C(F)F)n2)CC1 Cc1noc(C)c1C(C)CC(=O)NC1(C)CCC1.C1(C=O)CCC(F)(F)C1.N C1(Cl)(C(=O)NC2(CN(C)Cc3ccccc3)CC2)CC12CCC2 C1(NC(C=NOC)=O)CC2CC(C1)N(C(=O)CCC1(C(F)(F)F)CCCCC1)C2 c1(OCC(CCC)NC(=O)NCC=C)ccccc1OCC N1(Cc2ccc(-c3c(C)ccnc3)cc2)CCCC(O)(C(N2CCCC2C)=O)C1 Cc1cc(CCC(=O)N(C)CC2CCC(NC(C3CCCC3)=O)CC2)ccn1 Cc1cc(C(N2CC(C)(NC(C3CCCC4CCCN34)=O)C2)=O)c(O)c(C)c1 c1(CC)ccc(C(N2CCC(CN(C(C3SCCC3C)=O)CC)CC2)=O)cc1 N1(C(c2c(OC)nn(C)c2)=O)CCC(Nc2cc3nncn3cn2)C(C)(C)C1 CN=c1nc(N(C)CCc2ccccc2)[nH]c(=NCCCC2CC2(Cl)Cl)[nH]1 C1(C(CC)NC2(CO)CC2)CCC(C)CC1.C(=O)C(C)(C)C1CC1 c1(C(=O)NC(CC)(CC)CCNC(=O)C(C)C2CC2)cc(Cl)cc(Cl)c1N c1(NC(C)=O)ccc(C)c(CN2CCCCC2C(c2ccccc2)C2CCC2)c1 C1(CC(=O)NCCCn2c(C)nnc2)CN(C(C2C=CCCC2)=O)CC12CCC2 CC1CCc2[nH]nc(C(N3CC4CN(C(=O)C5=COCCC5)CC4(C)C3)=O)c2C1 CN1CCCC(CC(N2CCCC(C(=O)NCCc3cn[nH]c3)C2)=O)C1 c1(C(C(=O)N(CC)CC2CCN(C(C)C)C2)F)ccc(Br)cc1Cl CCC(C(=O)N1CCC(C(C)CNC(c2ccc(C(C)=O)cn2)=O)CC1)C(C)C c1(N2CC(CC(C)OC(CC3OCCN(C(C)C)C3)=O)C2)nc[nH]c2ncnc1-2 C(F)(F)(C(=O)NN1CCCCCC1)c1c(C)cc(C)cc1C C(=O)(C1=C(C)OCCC1)N1C2(C(N3C(CCCC)CCC3)=O)CC2CC1 C(CCC(C)C(=O)N1CCC(NC(=O)CCCn2cccn2)C(O)C1)OC C=Cn1nncc1C(=O)NC1CCN(CCNC(C2CC3CCC2C3)=O)CC1 C1(OC)(CNS(=O)(=O)C2CCCC2)CCS(=O)(=O)C1 N1(C(CC(=O)NCC)=O)C(C(=O)NC(C)C(F)F)CCC12CC2 CCCC(C(=O)NCC1(NC(=O)CC2CCCC(C)C2)CCC1)OC c1(-c2c(C)cnc(F)c2)cc(C(=O)Nc2ccc3c(c2)COC3)c2n[nH]cc2c1 CC(C(C)(C)NC(=O)CCc1ccsc1)NC(=O)C.C1(C(=O)N)CCCC1 C1(CC)C(NC(=O)C)CCCN1C(c1nonc1N)=O.C(=O)(CC(C)(C)C)N N1(C(COCCSC)=O)CCC(CCCCNC(=O)Cc2cnsc2)CC1 n1(C(CC)C)cc(C(c2nnnn2C(C)C)NCC(c2ncc(C)s2)C)cn1 c1cc(C)c(C)nn1.C1(NC(C=CC(CC)C)=O)CC(O)C1CC(=O)NC c1(C(=O)NCC=CCNC(CC(C)n2ccnc2)=O)ccc(C2CC2)nc1 CC1(C)CN(C(c2csc(CO)n2)=O)CC(C)O1.C1(C)(C=O)CCNC(=O)C1.N c1(-c2n(-c3cccc(SC)c3)nc(CC(C)(C)CO)n2)c2ccccc2nn1C N1(C(C2C3(CC(NC(CCN(C)C)=O)C3)C2)=O)CC2CC(F)CC2C1 c1(NC2(CN(C)C(C3(C)CC=CCC3)=O)CC2)cc(C#N)ccc1[N+](=O)[O-] C1(NC(Cc2cc(=N)[nH]cc2)=O)COCCN(C(=O)C2=CCC2)C1 N1(C(C(CCC)(C)C)=O)CC2(CCC(NC(=O)CCCCCCSC)O2)C1 Cc1ccc(C(=O)NC)c(C)n1.C1C2CN(C(c3cc(C(C)C)nn3C)=O)CC12 c1(C(=O)NC(C)C(C2CCCCC2)NC(=O)CCF)conc1C1CCC1 C1(C(N(CCN(C(C(C=C)c2ccccc2)=O)C)C(C)C)=O)CN(C)CC(C)O1 C#Cc1ccc(CNC(=O)C(=O)Nc2cccc3cc[nH]c23)c(F)c1 c1(C(N2CC(OC)C(NC(C3COCC3(C)C)=O)C2)=O)cnc(O)c(F)c1 C(=O)(CCCCCF)NC1CCC(NC(c2n(C)nc(O)c2)=O)C1 C(=O)(C(C)C1=CCCC1)N1CCCC(O)(CNC(Cc2nc(C(C)C)sc2)=O)C1 c1(CC)c(C(=O)N)[nH]c2ccccc12.C1(C(N(CC(C)C)C)=O)CC2(CCC2)C1 c1(C=O)occ2c1CCC2.C(C)(C)C=O.C1CCC1.CCCNC(=O)NC CC1CCC(N(C2CCC2)CCN(C)C)CC1 N1(C(=O)NC(C(=O)OC)C)CCCn2nc(C(N3CCC(F)(F)C3)=O)cc2C1 C(CS(=O)(=O)c1ccc(F)cc1)NC(=NCCCC)NC1CCC(SC)C1 C1(C(C)C)CN(C(C2(C)CCCN2)=O)CCN1C(=O)CCc1cncnc1 C(=O)(C(F)(F)C(O)c1ccccc1)N1CCC(C(c2ccccn2)=O)C1 C#CC1CCCCN1C(=O)C(CNC(C1(CC)CCCO1)=O)C(C)C Cc1ccc2sc(C(=O)NCC3CCN(C(=O)Cc4nccs4)CC3C)cc2c1 CC1CCCC=C1C(=O)NC1CC(CC(=O)N(C)CCc2ncccn2)C1(C)C CC(C)CCC(C(=O)NC1CCC12CCC2)NC(C1CC(CC2CC2)C1)=O.C C1(C(=O)NCC(C)(C2CCC2)NC(C(C(C)(F)F)F)=O)CCOCC12CCC2 Cc1nc(C2CC2)ccc1C(=O)NC1CCCC1.C1(CC=O)COC(=O)C1.C N1(C(c2c(CC)csc2)=O)CCN(C(=O)COCc2ccccc2C)C(C)C1C N1(C(c2ccc(C#C)o2)=O)C2CCC(C2)C1CC(=O)NC1CSC1 C12(C=O)CCC(CC1(F)F)C2.c1(CNC(C2COC2)=O)cccc(C)c1.N C1(C(=O)NCC2(O)CCN(C(C(C)SC(C)C)=O)CC2)CCn2ncnc2C1 Cc1nc2cc(F)cc(C(=O)N(CC(C)N(C)C(=O)C3CC3)C)c2nc1C C1(NC(c2cnn(CCO)c2)=O)CCCN(C(=O)Cc2n[nH]cc2Br)CC1 N1(C(c2scc(C)c2)=O)C2CCC1CN(C(c1c[nH]c(=N)c(C)c1)=O)C2 c1(CCCC(=O)NCC2C(NC(COCCCCC)=O)C2)ccc(F)cc1F N1(Cc2nc(NC(c3cc(OC)c(CO)cc3)=O)sc2)CCn2ncnc2C1 C1(C(N2CCCC(NC(C(CC=C)C)=O)CC2)=O)CC(C)(C)CC(C)(C)C1 N1(C(CCC(=C)Cl)=O)CCC2(CC1)OCCCC2NC(C1C2COCC12)=O c1(CN2CCCC(C)(C(=O)NC(CC)CO)C2)ccc(C)c2ccccc12 C1(C(=O)NC(C#C)C2CCC2)CCOCCN1C(C1CCC(C2CC2)C1)=O C(N=c1[nH]c2c(c(=NCCCCS(N)(=O)=O)[nH]1)CSC2)c1cnnc(C)c1C N1(C(c2cc(CC)on2)=O)CCCC2C1CCCN2C(=O)CCCC(C)(C)CC c1(C(C)C)cc(C(=O)NCC2CC(C)N(C(=O)C3=NOCC3)C2)ccc1F N1(C(c2nc(C(C)C)oc2)=O)CC2C(C1)N2C(=O)C(c1ccccc1)O c1(CC)cccc(N2CCCC(NC(c3cc(C)oc3CC)=O)CC2)c1[N+](=O)[O-] c1(C(=O)NC(C)CNC(=O)CC2CCCO2)cccc(SC(F)(F)F)c1 C(=O)(C1CCCc2nnn(C)c21)NC(C)CNC(=O)C1CCCn2cncc21 CC(C)CN=C(NCC1(O)CCC(C)(C)CC1)NC1CCCC1c1ccccc1 Cc1nc(C(N2CC(C3CN(C(=O)C=CCF)CCO3)C2)=O)oc1C C1(C(=O)NCC2CCCN(C)C2=O)CC12CCN(C(c1nc(Cl)cs1)=O)CC2 c1(C(=O)OC)cccnc1N(C1CCN(C(c2oc(C(C)C)nc2C)=O)CC1)C Cc1c(C(=O)N(CC(O)C)C)ccn1C(C)C.C(=O)(C=CCN(C)C)N C1(NC(c2cccnc2)=O)CC2CCC1N2C(c1ccc(C(F)(F)F)cn1)=O CCCC(C(C(=O)NCCOCC)N(C)Cc1cc(C)no1)OC N1(CC(=O)N(C2CCCN(C(c3c(Cl)nsc3Cl)=O)C2)C)CCCNS1(=O)=O c1(C(C)(C)C)ncc(NC(C23CC2CN(C(c2ccncc2O)=O)C3)=O)cn1 C1(C(=O)Nc2nc(C(C)=O)c(Br)s2)CN(C(=O)OC(C)(C)C)CC(C)(C)C1 CC1(C(=O)NC(C(=O)NCC2SCCS2)C2(O)CCC2)CCOC1 N1(C(CC(=O)NCC)=O)CCCC12CCN(C(c1c(OC)noc1C)=O)C2 C1(C)(NC(Cn2c(C)ccn2)=O)CCCN(C(=O)Cn2cnc(Br)c2)C1 CCC(C)(CC)NC(=O)C(Cc1cn[nH]c1)NC(c1cnn(C2CC2)c1)=O C1(OC)CN(C(=O)CCC(C)SC)CC1NC(=O)C(C1CCCC1)C1CCCC1 CC(CCNC(=O)C(C)Cc1cccc(Cl)c1)CCc1ccccc1 C1(NC(CCn2c(C)ncc2)=O)CCC(C)N(C(c2cc(N)nc(Cl)c2)=O)C1 CN1CCc2cc(C(N3CCN(S(=O)(=O)C(F)(F)F)C4CC34)=O)ccc21 CON1CC(C(N2CCCC2(C)C(=O)NCC2(C)CNC(=O)O2)=O)CC1=O c1(C(=O)NC(c2c(C)ccc(OC(F)F)c2)C)ccc(S(C)(=O)=O)c(F)c1O O=[N+]([O-])c1cccc(CS(=O)(=O)NCCn2ncc3ccccc23)c1 c1(C(=O)NCCC(C)N(C(C(C)Cn2ccnc2)=O)C)cc2c(o1)CCCC2 C1(C(N2CC(F)(CNC(=O)Cc3nnc(O)s3)C2)=O)CCOCC12CCC2 C(=O)(CC(C)(O)C(F)(F)F)NCC(CC(C)C)NC(=O)CNC(N)=O N1(C(CC(C)c2ccco2)=O)CC(=O)NCC1C(=O)NCc1ccc(Cl)cc1 Cc1c[nH]c2ncc(C(=O)NC3CC(C)CN(C(c4cncc(N)n4)=O)C3)cc12 C1(C(=O)NC(CNC(c2c(SC)cccc2)=O)C(C)C)CCOC(=O)CC1 C12(NC(c3n(CCCC)ncc3)=O)CCCC1CN(C(c1c(C)csc1Cl)=O)C2 Cc1c(Cl)ccc(-c2nc(-c3ccc(F)cc3)nn2-c2ccc(Cl)nc2)c1Cl c1(OC)ncncc1NC(C1CC(N(C(=O)CCC2CCCO2)C)C1)=O c1(C(N2CCC(O)(CNC(CCC=CC)=O)C2)=O)ccc(C(F)F)cc1F c1(-c2cc(NC(C3OCCN(c4cn(C)nc4)C3)=O)n[nH]2)ccc(F)cc1F C1(CCOC)CN(C(=O)COC(C)C)CCN1C(c1cc(O)cc(Cl)c1)=O c1(OCCCC)ccc(-c2noc(C(C3CCS(=O)(=O)C3)C)n2)cn1 c1(C(N(c2nccc(OC)n2)CC2CCNCC2)=O)cn2cccnc2n1 CC(C)(F)CCC(=O)N1CCC(OCCNC(C2COC(=O)C2)=O)CC1 S(=O)(=O)(c1cccc(=NCc2ccc(F)c(F)c2)[nH]1)N1CCC(CN(C)C)C1 c1(C2N(CC(C3(O)CCOCC3)(C)C)CCC2)cc(OC#N)cc(OC(C)(C)C)c1 Cc1ccc(=O)n(CC(=O)Nc2ccccc2SCC(F)F)c1 N1(C(C2C(CCC)C2)=O)CCC(NC(=O)C)C12CC2.c1cc(C)cc(C)c1.N C1(NC(C(C(C)C)c2ccccc2)=O)CC(O)CN(C(=O)C(F)=CC2CC2)C1 c1(C(=O)NC2CC(C)N(C(c3coc(N(C)C)n3)=O)C2)snc2ccccc12 Cc1ncc(Br)cc1C(N1CC(NC(c2ccc(=O)n(C)c2)=O)CC(O)C1)=O CC(C)C(CCN(C)C(C12CCCCC1C2)=O)NC(=O)C(F)=C1CCCC1 CC1CN(c2nnc(C(F)F)o2)CC1C(=O)NCC1CCC(N(C)C)CC1 c1(OC)cc(C(=O)NC2CC2NC(=O)CC2CCC(=O)N2C)cc(Cl)c1O c1(C(N2CCCC(C)(C)C2)C(=O)NCCSC)cnc(N(C)C)c(F)c1Cl.C c1(NC(C2C(NC(C3C(C)CCCC3)=O)CC2)=O)ccc(F)cc1O Cc1c[nH]cc(C(=O)NC23CCN(C(C4(C)CC(F)(F)C4)=O)CC2C3)c1=O CS(=O)(=O)C1(C(=O)NCC2CCN(C(c3cccnc3)=O)C2)CCCC1 Cc1nn2cc(C(=O)NC3CC4CC3CN4C(c3cc(Cl)cc(Cl)c3)=O)nc2s1 N1(C(C(C)(C)Cc2ccccc2)=O)CCC2(CCN(C(=O)C#CC3(C)CC3)C2)C1 C#CCCC(C(=O)Nc1ccccc1O)NC(=O)CCC(=O)NC C(=O)CC1CC1.C1(C=O)CCC1.C(COCC)OCC.C(C)=O.N C1(C(C)NC(C(c2ccccc2)OC)=O)CCCN1C(c1cc[nH]n1)=O C1(OC)CN(C(C2CCC2)=O)CC1.c1(C(=O)N)ccc[nH]1.C(=O)CC1CC1 C=C1CCN(C(=O)C=CCCC(C)C)C(C(=O)NC2(CCCCO)CC2)C1 N1(C(=O)Nc2n(C(C)C)ncc2)CCc2sccc2C1c1ccccc1 C1(CCC)CN(C(=O)CCC2CCCCO2)CCN1C(c1cc(C)on1)=O c1(C(N2CC3CN(C(CC(CC)C)=O)CC3C2)=O)cc(=O)n(C)c2ccccc12 C(C(=O)N(CCC(C(C)C)NC(c1cc(C)on1)=O)C)(C(C)C)SC Cc1nn(C)c(C(F)(F)F)c1C(=O)NCC(CO)NC(C1CCCCO1)=O c1(CN(C)C(c2ccc[nH]2)=O)cnn2c1CN(c1nc3cccc(Br)c3o1)CC2 C1(NC(C2C(OC)CC2)=O)CCN(C(c2ccc(OC)cc2OC)=O)CC1F C(=O)(CC(C)C)NCC(C)N(CC(C)SCC=C)C.C(=O)CC(C)C.N c1(OC)cc(F)ccc1C(=O)N.C1CC12CCN(C(c1ccc(C(C)C)o1)=O)C2 C1(C)(C(=O)NCCCCC(C)NC(C2C(=C)C2)=O)CCN(C)C1=O N1(C(C(CCN(C)C)NC(c2ccc(C)c(O)c2)=O)=O)CCC2(CCCO2)C1 N1(C(C(CCCC)N(C)C)=O)CC2=C(C1)CN(C(C1CC3(C1)CC3(F)F)=O)C2 N1(C(c2ccc(C=O)s2)=O)CC2CC2C1.C(=O)(CN(C)C(N)=O)NC.C N(C(=NCc1ccc(N(C)CCS(C)(=O)=O)nc1)N1CCC(C)CC1)C(C)C C1(C(N(C2CN(C(c3cccn3C)=O)CC2F)C)=O)CCCN(CP(C)(C)=O)C1 Cc1nc(Cl)ccc1NC(C12CC(C)(CN1C(C1(C)CNC(=O)C1)=O)C2)=O Cc1nc2c(s1)C(NC(=O)NCc1ncccc1O)CCC2 c1(C(=O)NC2(CCNC(COCC)=O)CC2)nccn2nc(C)cc12 CCC(C)(CO)C(=O)N1CCC(C)(NC(=O)CCc2cccc(C(F)(F)F)c2)C1 C1(CC(=O)N(CC(F)F)CC)CCN(Cc2ccc(-n3cccn3)cc2)CC1 C1(NC(C2CC(C#N)(OC)C2)=O)CC2(C1)CC(C(N1CCC3CC13)=O)C2 C1CC2(CCC2)CN1C(=O)C1=NNC(=O)CC1.Cc1ncsc1C=CC(=O)NC N1(C(CCCn2cc(C3(OCC)CCCC3)nn2)=O)CCCCC1CF c1(C(=O)NCC2CCN2C(=O)C=CCO)cc2c(ccc3ccccc23)[nH]1 C(=O)(C1=CCCOC1)N1CCN(CCN(C(c2cnc(C(=O)OC)s2)=O)C)CC1 CON(CC1CCCc2ccccc21)C(=O)CCN1CCC(OC(F)F)CC1 C1(CC(=O)NCCNC(C2CCC3CC23)=O)C(=O)Nc2ccccc2S1(=O)=O CC(C)(CCCNC(=O)CCC1CCCO1)C(=O)Nc1ccc(C2CC2)cc1 c1(C(N2CCC(Oc3ccncc3)C2)C(=O)NC2CCOC2)sccc1I c1(CC)c(C(=O)NC(c2cn(C)nn2)C=O)nnn1C.CC(C)CC1CCC1.N C1(C)(NC(c2nccc(CNC(CC(C=C)CC)=O)c2)=O)CCC(C)(C)CC1 c1(NCc2n(Cc3sccc3)nnn2)cncc(-c2cc[nH]n2)c1 C(=O)C(CO)C(C)(C)C.CC(C)(CC(F)C(=O)O)NC(c1cccc(C#N)c1)=O c1(CC(C)NC(c2ccoc2)=O)ccc(CNC(c2coc(O)n2)=O)cc1 C(CCC(O)C(=O)Nc1cccnc1)NC(C1CNC(=O)O1)=O C(=O)(C1=CCCCO1)N(C(C)CNC(c1csnc1C1CC1)=O)C c1(C(N2CCC(CNC(c3c(C)nc[nH]3)=O)C2)C)cc(Cl)sc1Cl N1(C(C(C=C)O)=O)CC(C)(C)OC2(C1)CN(C(C1CS(=O)(=O)CC(=O)N1)=O)C2 C(C)(C(C(=O)N(CC(C)C)C)N(C)C)OC.c1(C=O)oc(C(F)(F)F)nc1C c1(C(=O)NCCCN(C(C(CC=CC)C)=O)CC)cc(C)c2nc(C)nn2c1 CC1(C(=O)NC2CC2NC(=O)C2=C(Cl)CCCC2)COc2ccccc2O1 Cc1ccc(=O)n(CC(=O)NCC23CC(CO2)N(C(=O)CCC(N)=O)C3)c1 C1(C#N)(CC)CCN(C(=O)NCc2nc(C)co2)CC1 C1(CNC(CCC(=O)NC)=O)CCCCCN1C(c1cc(F)ccc1O)=O O=C(CCC(=O)N1CCOC(c2cnn[nH]2)C1)N1CCCC1.c12cn(nn1)CC2 C(=O)(CCC(C(C)C)NC(C1CC1C1CC1)=O)NC1(COC)CCC1 C1(C(N2CC(C)OC(C)C2)=O)CC2CCN(CC=C(Cl)Cl)CC12 Nc1cc(C(=O)NC2CCN(C(=O)C(c3ccccc3)O)C2)nc(O)c1 C(C(CC(C)C)C(=O)N1CC2(CCCC2)C1C(C)C)NC(C(COC)C)=O N1(C(C(=O)OCC)=O)CCS(=O)(=O)C(C(=O)Nc2cccnc2)C1 c1(CN2CCCC(NC(C(c3n(C)ccc3)=O)=O)CC2)ccc2cccnc2c1 Cc1ccc(-c2ccsc2)c2nc(C(=O)Nc3cccnc3CO)cn12 CC1(C)CC(NC(C2CC=CCO2)=O)CN1C(=O)CCCOc1cccc(F)c1 N1(C(C2CCCC(C)C2)=O)CC2(C1)CN(C(=O)CC1CC3(CC3)CO1)C2 C(CCC(F)(F)F)(c1ccccc1)NC(C12CCC1CNC2)=O Cc1ncc(C(N2CC=CC2(C)C(=O)N(C2CCC2C)C)=O)n1C C1(CC(c2ccccc2)NC(C(=O)NCC(CC)OC)=O)CCC(F)(F)CC1 C(CC(F)F)(C(=O)NC1(C)CC(C)(C)C1)N(C(CNC(C(CC)C)=O)=O)C CC(C)(C(F)(F)F)NC(=O)CCC1(C)CN(C(c2ccc(C(F)F)o2)=O)C1 C1(NC(=O)CC(F)(F)C(F)F)CCCCC12CCN(C(=O)CCCCCO)CC2 c1(C=O)ccc2c(c1)C(=O)C(=O)N2.CC(C)(C)CC.C1(Cl)(C=O)CC1(C)C C(C(C)(C)CC(=O)NC(C1(C(=O)NC2CCCN(C)C2)CC1)C)OC CCC(CNC(=O)C=Cc1cccs1)CC.c1(C=O)cc(C2(C)CC2)on1.N N1(C(c2c(OC)ccnc2F)=O)CCCC2(CCCN2C(C2(F)CCCC2)=O)C1 N1(C(CC(C)C2CC2)=O)CCN(c2ncc(O)cn2)CC(C)(F)C1 C1(C(N2CC(c3nc(C)on3)C2)=O)CC(C)CN(C(C2CC(O)CN2C)=O)C1 C1(C(=O)NC(CC(C)NC(C23CC(F)(C2)C3)=O)C)CCOCC12CCCCC2 Cc1ccc(C)c(C(=O)NCc2nc(C)c(C(N3C(CO)CC3C)=O)o2)c1 CCCC(O)CC(=O)NC1CC12CC(NC(c1ccc(Cl)cc1CC)=O)C2 CCCC(CC(C)C)C(=O)NCC1(O)CCCN(C(C2(C(N)=O)CCC2)=O)CC1 N1(C(Cc2c(C)con2)=O)CC(C2CCCN(C(=O)C3=COCCO3)C2)C1 C(=O)(C(CCC1CCC1)NC(c1nc(Cl)oc1C)=O)NC1CN(CC)C1 N1(C(C2(C(C)C)CCC2)=O)CCC(CO)(NC(=O)CC2COCCN2C)CC1 CC(CC(=O)N(C)CCC1CCCCN1C(=O)CC(C)(C)CN(C)C)C(F)F c1(CCC)c(C(=O)NC2CCCC(CN(C(=O)C(=O)N(C)C)C)C2)nnn1C Cc1cccc(CNC(C2(NC(C3(C)CC=CCC3)=O)CC2C)=O)c1 C#CCCCCCC(=O)NC1CCN(C(C2(CO)CCCO2)=O)CC1(C)C c1(C(N(C2CCN(C(C3C(C)C3)=O)C2)C)=O)nccc2ncccc12 c1(-n2cc(C3N(C(c4cc[nH]n4)=O)CCOC3)nn2)ncnc2ccccc12 C(C)(C)(CCCCNC(=O)CN(C)C1CC1)NC(CCc1ccc(C)nc1)=O C=C(CNC(=O)C(O)C1CN(C(=O)CCCC(C)CC)C1)c1ccccc1 C1(CC(=O)NC2C3(CC(NC(C=C(CC)C)=O)C3)C2)CCCCC1(F)F C1(NC(C(C)=C2CCC2)=O)CCC(CCNC(=O)CCS)C1.c1nnnn1C N1(C(CC2C(C)C2)=O)CCN(C2CCCN(C(=O)CCC(=O)N(C)C(C)C)C2)CC1 Cc1c(C(=O)NC2CC3CC(NC(=O)C(C)C(F)(F)F)CC23)nn2c1OCCC2 C1(CCNC(C2N(C(C=CCC)=O)CCC2)=O)CCCC1(C)C N1(C(C(=O)OC)C)CCOC(CN(C(=O)CC(C)S)C2CC2)C1.c1cccs1 Cc1cc(C(=O)NCC(CO)NC(=O)C2=CS(=O)CCC2)ccc1[N+](=O)[O-] CC(C(=O)N1CCCC1CNC(=O)C1=NN(C)C(=O)CC1)C(C)S(C)(=O)=O N12CCOC(C1)Cc1ccc(s1)CC2=O.c1(C(=O)N)ccc(O)cn1.COC c1(C(N2CC(C(C)NC(CCc3cc(C)sc3C)=O)C2)=O)ccc(O)c(C)c1C C12(C=O)C3CC(CC13)C2(F)F.N1(CC(C)C)CC(C(=O)NCCCC)CC1=O S(=O)(=O)(c1ccc(N2CC3CC2CC3O)c(F)c1)NC1CNC(=O)C1(F)F C1(NC(c2c(OC)c(C)sc2)=O)C2CCC1CN(C(=O)C(C)SC(F)(F)F)C2 c1(C(N2CCCC(CNC(C(CC=C)C)=O)C2)=O)nnc(O)cc1O N1(C(COCCCC#C)=O)CC(=O)NC2CN(C(=O)C(C)(C)C)CCC12 c1(C(N2CCOCC2c2cccs2)C(=O)NC)cccc2nonc12 C1(CC(=O)NCC(CNC(Cc2c(C)non2)=O)O)CC(C)OC1C c1(NC)cncc(C(N2CCC(N(C)C(C3(Cl)CC3(C)C)=O)CC2)=O)c1 c1(N2CC(C)OC(C)C2)nc(=NCC2CCCCCC2)[nH]c2cc[nH]c12 N1(C(Cc2c(C)nccc2)=O)CC2CC(CNC(c3nc(C)c(C)s3)=O)CC1C2 C12N(CC13CCCCCC3)C2=O.c12cccc(n1)NC2C(=O)O.C(C(F)F)OC C(CCCCC(=O)OCCOC)(c1nnnn1C)N(CCCNC(C(C)C)=O)C N1(C(C)=O)CC2CCC1C2.C(=O)C(F)(F)c1cnn(C)c1.C=CCOC=O.N N1(C(C)C)CCCC1C(=O)NC1CC(C)(CNC(=O)Cc2cncn2C)C1 N1(C(C=C(C)Cl)=O)CCC(CNC(=O)CCNC(=O)CO)C12CCC2 C1(C(=O)NCCCC(N2CCCC(CC)C2)=O)CC2(CCC2O)C1 CC(C)(C)C#CC(=O)NC1CCCC1(C)CNC(C1(N2CCOCC2)CC1)=O C(=O)(CCCC(F)(F)F)N1CCCC(CC)C1.C1(CS(C)(=O)=O)(C=O)CCC1.N C(=O)(C1=CCCC1)NC(c1ccccc1)C(=O)N(C)Cc1cncn1C CC1(C)CC(C(=O)NC2(CO)CCCN(C(=O)COC)C2)=NO1.C1CCOC1 C1(C(=O)NC(C=CC(=O)NCCN2C(C)CCCC2)(C)C)CC2CC1CC2O N1(C(c2c(C)sc(C)c2Br)=O)CCC2(CC1)CC(NC(=O)C(N)=O)CO2 c1(C(=O)NC(CN(C(CC2C(C)CCCC2)=O)C)(C)C)cc2c(s1)CCC2 C(=O)(C1CCc2nccn21)N1CCC(CN(C)C(c2occ3c2CCCC3)=O)C1 C(C)(C)CC.C(=O)C(F)(F)c1ccncc1.C1(C(=O)N)CC1C=O.C#CC C1(C(N(CCN(C(=O)C=CSC)CC)CC)=O)OCCOC1c1ccccc1 N1(CC2(CCNC(c3cc(CC)no3)=O)CC2)CCC2(C=C(C=O)C2)C1 Cc1nc2cc(C(=O)OCC3NCCC3C)ccc2n1C1CC1 C(=O)(CC(c1ccncc1)N(C)C)NC(C1CC1(C)C)C C(CCC(C)C)(C=O)NC(C)=O.C(C)(C(F)F)=CC(N1CC(CC)C1)=O.N c1(N2CCC(COC(CC3C(OCC)C3)=O)C2)cccc(C#N)c1 c1(C2C(=O)NCCCN2C)ccc(SC)o1.N1(CC)CCSCC1 c1(-c2ncn(C)c2C2OCCC2c2ccccc2)ccc(F)c(Cl)c1 N1(C(N(CCCNc2c(C)cc(F)cc2)C)=O)CC(C2CCCC2)C1 N1(Cc2cc(C(=O)OCC)n3c2cccc3)Cc2ccccc2C2(CC2)C1 CCCN=C(NCC(O)C1(C)CC1)NCC(F)(F)C1CCC1 C(=O)(N=c1[nH]nc(Cl)cc1C)C1N(C(=O)Nc2c(C)cc(C)cc2C)CCC1O N1(Cc2cn(CC=C)nn2)CCC(CNC(=O)C(F)(F)F)CC1.OC c1(COCCCN(C(=O)CC2CC2)CC)cn[nH]c1.CCC.C(=O)C Cc1sc(CNC2CC(N)C2)c(Cl)c1C(=O)O 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c1(C(=O)NC(C(C)NC(=O)CO)CCc2ccccc2)ccc(Cl)c2c1OCCO2 c1(C=O)c2c(nn1C)CCCC2.n1(CC)ncc(Cl)c1C(=O)NCC1CCC1 N1(C(Cc2c(CC)cccc2)=O)CCC2(CC1)CC2NC(c1cc(CO)on1)=O C1(C)(CNC(c2cnc(CC)s2)=O)CCCN1C(=O)Cn1cc(CO)nn1 c1(C=O)cnc(O)c2cncn12.C12(CNC(C(C)=CC)=O)CC(CCO1)C2 C1(N(C(CC2CCC(C)O2)=O)C)CCN(C(c2ccc(Br)o2)=O)CC1 N#Cc1cc(C(=O)NCCC(=O)NCc2ccccc2)ccc1[N+](=O)[O-] C1CN(C(C2CC3(C2)CC(F)C3)=O)CC2CC12.c1(C2C(C=O)C2)ccccc1.N C1(CNC(COC(CC)C)=O)CN(C(=O)CCCC2CCC2)CC(C)(C)O1 C1(C(=O)NCC2ON=C(CC)C2)C2CCCC2CN1C(C1CCCCC1)=O N1(C(CC=C(C)C)=O)CCCC(CCNC(=O)C(C(C)C)c2ccn(C)n2)CC1 N1(C(C2(C#C)CC(F)(F)C2)=O)CC2CCCC2(C(=O)NOCCCF)C1 CN1CCC(C(=O)NCC2CCCCC2C(N2CCC2CC2CCCC2)=O)CC1 C12(NC(=O)CN3CCSCC3)CCCC1CN(C(=O)CSC(F)F)C2 c1(CCCOC)cn(C2CCN(C(=O)C(F)CC3CCCCC3)C2)nn1 C1(NC(Cc2c(C)nc[nH]2)=O)CC2CCC(C1)N2C(C1(F)CCCOC1)=O N1(C(c2cc(C)c(O)nc2)=O)CC2(C=C(C(=O)NC3(C(F)(F)F)CC3)CO2)C1 c1(-c2cncc(SC)c2)cccc2[nH]nc(C(N3CCOC4CC34)=O)c12 N1(C(=O)OC(C)(C)C)CCC(C)(C(=O)NCC)CC1.C1(C#N)CCCOC1.N C1(C(=O)NCc2ccc(C(N3CC(CC)C3)=O)nc2)CCC(=O)N(C)C1 C(=O)(CCCNC(=O)C(C1CCCO1)NC(C1(C)CCCO1)=O)OC C1(NC(Cn2c(C)nc(C)n2)=O)CCCCN(C(=O)C(c2ccccc2)O)CC1 Cc1ncc(C(=O)NC2CCOCC2)c(C2CC2)n1.C12(C(=O)N)CCC(CC1)O2 C1(C(N2CCC(C3CCCN3c3ncncc3Br)C2)=O)CCCCC1C1CC1 N1(C(C(C)(C)C)=O)CCC(C(N2CCOC(C#N)C2)=O)C(O)C1 c1(CC(=O)NCCC2(OC)CN(C(c3nocc3C)=O)C2)c(C)nn(C)c1C c1(C=O)cnc(S)n1C1CC1.C12CN(C1)C2=O.O=C(CSC(F)F)N.CC CC(C)CC(C)(O)C(=O)NC.C1CN(C(C2(C(=O)N(C)C)CC2)=O)CCCO1 C(=O)(C1COc2ccccc21)N1CCC(CNC(C(C)OC)=O)C1(C)C C12(NC(C(C=C)CC)=O)C(C(=O)N(C(C)C(=O)OC)C)C3CC1C2C3 CCC(CNC(=O)C(F)(Cl)c1ccccc1)(CC)NC(C1CCCS1(=O)=O)=O N1(C(c2ccc(OC(C)C)cc2)CC)CCN(C2=NCCCS2)CC1 C1(COC)CN(C(=O)C(O)C2CCC2)C1.c1(C=O)ccccc1.C(=O)(C)N c1(C(N)=O)cc(=NC2CC(F)(CNC(c3ccnc4ccnn34)=O)C2)[nH]c(Cl)n1 C(C(C)(C)CC(=O)N1CCC(C(F)C(=O)NCC(Cl)C(C)(F)F)C1)N(C)C c1(C(N(CCCC)CCN(CC(=O)NCCCC)C)=O)ccc(C)o1 N1(CCC(N2CCCC(CCC=C)C2)=O)c2ccccc2Sc2ccccc21 N1(C(C2(CNC(c3c(C)n(C)nc3)=O)CCCO2)=O)CCCC(C2CC2)CC1 c1(C(N2CC(=C(C)F)C2)=O)cccc(=O)o1.CC1CC1C(=O)NCC=O.N Cc1cc(CNC(C2(NC(C3CCNC3=O)=O)CCC2)=O)nn1C C1(C(=O)N)CC(O)CN1C.C1(CCC(=O)N(CC(=O)OCC)C)CCCC1 Cc1nc(N2CCCCC(CNC(c3ocnc3C)=O)C2)c(C)c(O)n1 c1(OC)ccc(C(=O)NCCC2(O)CN(C(c3sncc3C)=O)C2)c(N)c1 C(=O)(CC(CCCC)NC(=O)CC1CC(C)=NO1)N(CC=C)CC1CC1 N1(C(CNC2CCCC2O)=O)CCCC(C)C1.c1(CC=O)cc(C)[nH]n1.CCS c1(OC)cc(C)c(C(=O)NC2(C)CCN(C(=O)CC(C)(C)C#N)CC2)cn1 c1(C(=O)NCC2(C)CCC(NC(c3cccnc3O)=O)C2)ncc(Cl)cc1F c1(OCC(C)C)ncccc1C(N1CCC=C(F)C1)=O S(=O)(=O)(c1ccncc1)N1CC(C)CC(NCc2c(OC)nccc2I)C1 C1(C(=O)OC)(C(c2nnnn2C2CCC2)NCCc2cnoc2C)CC=CCC1 C=CCCC(C(=O)N1CCC(O)C(O)C1)NC(=O)CC1C=CCC1 [SH](=O)(=O)c1ccc2oc(O)nc2c1.N#Cc1cccnc1C=Cc1ccccc1 c1(C(=O)Nc2c3ncc(C)nc3ccc2)cc2n(n1)CCN(C)C2=O N1(C(=O)Cc2ccc(C(F)(F)F)cc2)CC2CCC(C1)N2C(=O)C(O)O CC1(C)CCCC(C(N2CC(NC(C3CC=CC3)=O)C(C(F)(F)F)C2)=O)O1 CCCC(C(O)C(=O)N1CCCC1C(N)=O)NC(c1n[nH]cc1C)=O N1(C(C2CC(=O)NC2)=O)CCC(CF)(NC(c2cnc(C(F)(F)F)s2)=O)C1 N1(C(=O)OC)CCN(c2ccnc(N3CCC(OC)CC3)n2)CC(C)C1 CN1CC(C(=O)NC23CC(NC(=O)COC4CCCOC4)(C2)C3)NC1=O C(C(C)(C)C(=O)N1CCC2CCC12)NC(c1ccn(COC)n1)=O C1(C(=O)NCCC(CNC(Cn2c(C)ccn2)=O)O)CCN(C2CCSC2)CC1 C(=O)(CC(C)CCC=C(C)C)N.CCCC(C)CC(=O)NCC1(C)CCCCC1 C1(C(N2CC(CNC(=O)CCCc3ccccn3)C(O)C2)=O)CCCS(=O)(=O)C1 C(=O)(C(C(=O)N(CC(C)NC(c1c[nH]cc1-c1ccc(Cl)s1)=O)C)OC)OC c1(C(N(C2CN(C(=O)CC3CC(C)(C)C3)CC2O)C)=O)cnn2c1OCC(O)C2 C(CC1=CCN(C(c2sccc2Cl)=O)CC1)NC(C1(C)CCCCO1)=O Cc1nc2cc(C(=O)NC3CCCC(NC(=O)C(O)C4CC4)C3)[nH]c2s1 C1(CNC(C=COCC)=O)CN(C(=O)C2=C(Cl)CC2)CCC1C C(=O)(C(F)(F)CCn1cccn1)N1CC(NC(C(n2c(C)ncc2)C)=O)C(C)C1 O=C(CC(F)(F)C(F)F)N1CC(C2CN(C(C3COC(=O)N3)=O)CCO2)C1 c1(C(=O)NC2CCN(C(C(CC3CC3)OC)=O)C2)nnccc1C C1(NC(c2nc(CCC)sc2)=O)CC2CCC1N2C(=O)CC(C)(C)C.C(C)=O C1(C(=O)NCCCCC(=O)NC)CCCN1NC(=O)C1CNC(=O)O1 CC(C)CCC(=O)N1CC(O)CC1CNC(c1cccnn1)=O.C(C(F)(F)F)O C1(NC(C(CCC)OC)=O)CN(C(=O)CCCC(F)(F)F)CC2(CC2)C1 N1(C(=O)NC2C(CN(CCC)CC)C2)CCCC(C(=O)OC)C1 c1(CN(C(=O)CC2CCN(C(=O)C(C3CCOCC3)=O)C2)CC)cccnc1 C1CCCN(C(C2(F)CCS(=O)(=O)C2)=O)C1.C(C(=O)N)N(C1CC1)CC c1(C(N2CCN(C(C(C)CF)=O)C(c3ccncc3)C2)=O)cc[nH]c2nccc1-2 C1(NC(N(C(C)CCCO)C)=O)CNCCC1(C)C C(CCC(C)C(=O)N1CCN(C(=O)C2=CCCCO2)CC1C(C)(C)C)OC Cc1cncc(CNC2CCCC2C(=O)Nc2cccc(F)c2)c1 C1(N(C(=O)NCC(c2cnn(C)c2)C)C)CCN(c2ccncc2)C1 N(C(=NCC1CCC(C)O1)N(C)Cc1ncc(Cl)n1C)Cc1cc(C)on1 C1(NC(c2c(C)onc2)=O)CCCC(CNC(c2ccc(Cl)o2)=O)C1 Cc1cc(C(N2CC(C)(C(=O)Nc3cncnc3C)C2)=O)cc(Cl)c1 N1(C(C=CSC)=O)CCC(C2CC2NC(=O)C(C)Cc2ccccc2Cl)CC1 c1(CNC2CC(C(=O)N=c3cccn[nH]3)C2)ccc([N+](=O)[O-])c(O)c1 c1ccc(F)c(Cl)c1.CCC1=NOC(C(=O)NCC(C)(CO)NC(=O)CO)C1 C1(C(N(C(C)CN(C)C)C)=O)CC(C)CN(C(C2CSC2)=O)C1 N1(C(C(CCC)F)=O)CC2=C(C1)CN(C(=O)C=Cc1ncc[nH]1)C2 C1(F)(C(=O)NCC=CCOC)CCN(C(=O)Cc2cn[nH]c2)CC1 c1(C(N2CC(F)C2)=O)cc(C(F)(F)F)ccn1.CC(CN(C)C)C(=O)NC C1(NC(C(COC)C)=O)CS(=O)(=O)CC1Nc1nccnc1C#N C1(F)(c2cn(C3CCC(CC)C3)nn2)CCN(C(c2cc(F)ccc2O)=O)CC1 c1(C(=O)NCC(CC)(C)NC(c2cc[nH]c2C)=O)nnc(O)cc1O.C1CC1.C CS(=O)(=O)c1cccc(CN2CC(F)(F)CC2C(=O)NCCc2cnc[nH]2)c1 C(=O)(C(O)CC(F)(F)F)N1CC(C(=O)NCC(C(CC)C)CO)(CC)C1 C(=O)(C1=CCC(C)CC1)NCC1C2CN(C(c3nc(CCC)oc3)=O)CC21 C1(NC(CC2C(C)(C)COCC2)=O)CN(C(=O)CSCC(N)=O)CCC12CCC2 C1(C(=O)NCCC)CN(C(=O)OC(C)(C)C)CC1C1CC1 c1(C(=O)NC(CC#C)CCOC)[nH]c(C)c(C(C)=O)c1C(C)C CC1(C)CCC(C(=O)NC)CO1.C1(C)CCCN1C(=O)CC1CCCS1(=O)=O c1ccc(NC(=O)C(N)=O)c(Br)c1.N1(C(c2n(C)ccc2)=O)CCSCC1C=O CC(C)C(O)CC(=O)N(C)CC1(O)CCN(C(=O)CC2CCOCC2)CC1 N1(C(CCC(=O)NC)=O)CCN(C(C2CC3C=CC2CC3)=O)C(C(C)C)C1 c1(C(=O)NC(C2CN(C(=O)CCS(C)=O)CCO2)C)ccc2c(c1)CCO2 C1(C(=O)NCC2CCCN(C(C(C)NC=O)=O)CC2)CC2(C1)CC(C)(C)C2 c1(C(N2CCCC(N(C(C(C)(C)n3cccn3)=O)CCO)C2)=O)cncc(F)c1Cl c1(C=O)ccnc2[nH]c(C)nc12.C(C(=O)N(C(C)C)C)(C(C)(C)C)NC(C)=O c1(C(=O)NC2CC(CNC(C=COCC)=O)C2)cc2c(N(C)C)cccc2s1 c1(CC)c[nH]cc1C(=O)NC(C)C(C)NC(=O)C(C)(C)N1CCCC1 C1(C(=O)NCC(C)(C)C#N)CCCCN1C(C1(F)CC=CC1)=O CC(N=[N+]=[N-])C(=O)NCCC1CN(C(C2CCCOC2)=O)C1 N1(C(c2n[nH]c(=N)s2)=O)CCCOC(CNC(=O)C(C2CC2)C2CC2)C1 CC(C)CC(O)CC(=O)NC1CCC(CNC(=O)C(=O)NCCC(N)=O)CC1 C1(NC(C=NOC)=O)CCC12CCN(C(=O)Cc1sccc1Cl)CC2 C(=O)(CCS(C)=O)NC1(CCOC)CN(C(=O)Cc2ccccc2F)C1 N1(C(COCCCOC)=O)CCC2CCC(NC(=O)COC3CCCC3)C12 c1(C(N2CCC(C(C)NC(C3CCC3)=O)C2)=O)csc2c(O)ccnc12 C(C)(C(CC(=O)N1CC(c2ccccn2)C1)NC(C1CC(C)(C)CN1C)=O)OC Cc1ccccc1OCCN1CCC1CNC(=O)Cn1cccn1 Cn1nc(C(=O)NCC2CC2NC(=O)CSc2nncs2)c2c1CCSC2 C1(CNC(C(CC#C)CC#C)=O)Cc2ccccc2CN1C(=O)C(CC)SC C1(CC)CCCN1C(CNC(=O)NC)=O.C1CC(=C2CCC2)C1.CC=C.N C(CC)(CN=c1[nH]cnc(Cl)c1CO)(C1CC1)NC(C=C(C)c1ccco1)=O c1(CC(C(=O)N(CC(C)NC(=O)CCC2(C)CC2)C)C)ccc(F)cc1 CS(=O)(=O)CCCC(=O)NC1CCN(C(=O)CC2OCCCO2)C(C2CC2)C1 C1(CNC(C=CC(C)=O)=O)CCCN(C(=O)CCC(C)N2CCCC2)CC1 N1(c2ncc(C)s2)CC(C(=O)Nc2ccc(-n3cccn3)nc2)CC(F)C1 c1(OC(C(=O)NC(C)C(C)C)C)cccc(Cl)c1.c1(C=O)cnc(C2CC2)o1 C1(F)(C(=O)OC)CN(C(c2cc(F)ccn2)=O)CC1C1CC1 N1(C(COCC=C)=O)CC=C(CC(=O)N2CCC2CC2CC2)CC1 C(CCCC)(CC(=O)NC(c1ccon1)(C)C)NC(c1ncn(CC#C)n1)=O C1(CNC(C=C(C)C(C)C)=O)CCC(C)CN1C(c1ncc(C(F)F)s1)=O C=Cn1nccc1C(N1CCOCC1CN(C)C(c1occc1CC)=O)=O N1(C(c2nc(CC)oc2)=O)CCOCCC1C(N1CCOC(CC2CC2)C1)=O O=C(C1=COCCC1)NC1CC(CCNC(=O)C(F)(F)CCc2ccccc2)C1 C1(CNC(C2(F)CN(C(C(CC)O)=O)C2)=O)CC(O)C(O)C1 C1(CNC(C2(CC=C)CC2)=O)CN(C(c2cnc(N)cn2)=O)CCC1C Cc1c(F)ccc(C(=O)N(C2CN(C(C3CC34CC4)=O)CC23CC3)C)c1Cl C(=O)(CCC(=O)NCCC1CN(C(C2(n3cccn3)CC2)=O)C1)N(C)C c1cccc(Cl)c1.c12ccc(o1)C(=O)NC2.C(C(O)C)N(C)C.C(=O)(CC)N N1(C(CC2CC(=O)OC2)=O)CC2CCN(C(C3CCS(=O)CC3)=O)C2C1 Cc1cc(N(C)CC2CCCN2C(C2CCc3cncn3C2)=O)c(C#N)cn1 C1(CC)CCN(C(C2CN(C(N)=O)C2)=O)C1.c1(CCC=O)ccc(C)s1.CO C(=O)(CCN=c1[nH]ccs1)NCC1N(C(c2cnc(OC)nc2C(F)F)=O)CC1 Cc1cccc(C(=O)NC2CCC(c3ccc(F)c(F)c3)C2)c1Br N(C1CCc2cc(CNC(C34CC(F)(C3)C4)=O)ccc21)C(c1cnn(C)c1Cl)=O C(CC(C(=O)NC1CC2(CC2)C1)NC(=O)CC(C)N(C)C)OC CC12CCOC(CNC(=O)C(O)CCNC(c3sccc3Cl)=O)(C1)C2 C1(CNC(c2onc(CC)n2)=O)CC2(CCC2)CN1C(c1cncc(Cl)n1)=O C#CCC(C)(CC)C(=O)NCC(O)CCNC(c1cccc(COC)c1)=O c1(CCC=C)ccc(C(=O)NCC(C)CN(C)C(c2cc(SC)on2)=O)cc1 CCC(O)C(F)(F)C(=O)NC1CC(O)(CNC(C2(C)CCCC2)=O)C1.O c1(C(=O)NC(C2CCCN2C(C2CC3CCC2O3)=O)(C)C)n[nH]c2c1COCC2 C=CCC(C)(CC)C(=O)NC(C)CN(C(=O)Cc1ccc(F)c(Br)c1)CC N1(C(CC(C=C)(C)C)=O)CCCC2(CC(NC(c3cc(Cl)cnc3O)=O)CO2)C1 N1(S(=O)(=O)CCC(F)(F)F)CCc2cccc(-c3ccc4nc[nH]c4c3)c2C1 c1(CNC)n[nH]c2c1CN(C(=O)NCCOCCC1CCCC1)CC2 N1(C(CCC(C)O)=O)CCc2ccccc2C1CCNC(=O)CN1CC2CC2C1 c1(OC)cccc2c(CC(=O)NC3CN(C(=O)C(C)(C)SC)CC3O)coc12 CCCCCCNC(=O)C(=O)CCc1ccccc1.C1(C)(CC(=O)N)CC1(F)Cl c1(COC(C2C(N(C)C)COC2)=O)nc(-c2ccccc2)[nH]c1Cl C(=O)(CCCCCCCC1CC1)N1CCC(NC(CC(CC)SC)=O)CC(O)C1 c1(C=O)cnc(O)n(C2CC2)c1=O.CC(O)(C(=O)NC)C1CCC1.C1CCC1 c1(C(N2CCC(C)(NC(COC3CN(C(C)=O)C3)=O)C2)=O)cnn(C)c1C#N C1(NC(CC2(C)CCCC2)=O)CCCC(NC(=O)C(=O)NC2CC2)C1 N1(C(=O)NC(C)Cc2cccnc2)CCN(CCC(N)=O)CC1 CC1CCC(C)(NC(c2cc(CNC(=O)COC(=O)CO)ccn2)=O)C1 O=NN1CCCC1C(=O)NCC1(O)CCN(C(=O)Cc2ccccc2O)C1 CC1=CCC(C)(C(=O)NCC2CCN2C(=O)CO)CC1.c1c(Cl)cccc1Cl C(CCSC)(CN=c1[nH]c(=NC(C)CC(C)C)c2c(ncn2C)[nH]1)OC c1(C(=O)NC(c2cn(CCCSC)nn2)CCC)cccc(C(C)=O)c1 c1(CNC(=O)NC(CC)C(C)(C)O)c(F)cccc1F Cc1cc(=O)n2nc(CN3CC(O)CC3c3cccc(F)c3)sc2n1 c1(C(N(C2CCN(C(c3c(F)cncc3Cl)=O)C2)CC)=O)ccc2c(n1)NCC2 C(=O)(CS(=O)CC(F)(F)F)N1CC(N(c2ccccc2)CC(=C)C)C(C#N)C1 c1(N2C(C(=O)Nc3cccc(F)c3Br)CC(O)CC2)ncc2cccc(O)c2n1 C1(CC)CN(C(=O)C2=CCOCC2)CCN1C(=O)CCc1cc(C)no1 c1(C(N(CC(C(=O)NCCC(CC)(C)O)(C)C)C)=O)ccc(N)c(F)n1 Cc1cc(C(N2CC(NC(C3(c4cccc(Cl)c4)CC3)=O)C(C)C2)=O)nn1C Cc1cc2ncc(C(=O)NC3CCN(C(c4ncccc4O)=O)C3C)cn2n1 N1(C(C=CCCC(C)C)=O)CCC(C2CC2)C1CNC(=O)CCN1CCC1 CCC(CN(C)C)C(=O)NC1CCCCC1NC(=O)CC(=O)OC(C)(C)C N1(c2nnc(Cc3c(OC)cccc3)n2CCCN(C)C)CC(O)CCC1C C(=O)(C1=CC2CCCC12)N1CC(CC(C)NC(C(CCCC)O)=O)C1 c1(C(C(=O)NCC(C)O)N(C(C)=O)Cc2cscn2)ccc(F)cc1 N1(C(c2ccc(-c3c(F)ccc(OC)c3OC)s2)=O)CC2OCCCC2(CO)C1 C#CCC(C)C(=O)NCC1CCN(C(=O)C(C)C)CC1.c1(C(=O)N)ccccc1 c1(C(N2C(CNC(CCc3c(C)n[nH]c3C)=O)C(C)CC2)=O)cnn2ccsc12 c1(CCC(=O)NCC2CC2)cccc(F)c1F.c1(C=O)c(Cl)n[nH]c1C1CC1 Cc1nsc(C(N2CCC(C(=O)N(C)Cc3ncccn3)(CO)C2)=O)c1N c1(OC)ncccn1.C1(O)(C=O)CCN(C(C2CC(=O)N(C3CC3)C2)=O)C1.C C#CC1CN(C(C2(NC(=O)CC(C=C)CC)CC2)=O)CCO1 N1(C(C(CC=C)(C)C)=O)CC(C2CCCN(C(c3nn(C)cc3Cl)=O)C2)C1 c1(C2N(c3n(CCOCC=C)c(C(C)F)nn3)CCC2)cc2ccccc2o1 CCC(CC)(CC)C(=O)NCCC1(C(=O)NCC2(C)CCCCC2O)CC1 C12(CNC(C=C(C)C(C)C)=O)CCC(CC1)N2C(=O)C(O)Cn1cncn1 C1(C(=O)NCC2(SC)CC2)CN(C(c2cc(Cl)n(C)n2)=O)CCN1C Cn1c(C(=O)NC2(CCNC(=O)C=Cc3cnc[nH]3)CCOCC2)nnc1S C1(NC(c2nc(COC)sc2)=O)C=CCN(C(C2(C#N)CCCC2)=O)C1 c1(C(N2C(C(=O)NCc3ccccc3Cl)CC(F)C2)=O)c(Cl)ccc2c1OCO2 C(=O)(CCCCCC(C)(C)C)N1C2CCC(NC(CCC(C)OC)=O)(CC2)C1 C12(C(N3CCC(NC(C(C)OCC)=O)C(O)C3)=O)CCN(CC1)S(=O)(=O)C2 C1(C(NCCn2ccnc2O)=O)CN(S(=O)(=O)CC2CC(N)C2)CCC1O.C C1(C2CC2)(C(=O)NC2CCN(C(=O)CCCC3CC3)CC2C(=O)O)CCOCC1 N1(C(C(CC(C)C)(C)C)=O)CCOC2(C1)CN(CC1CCC1)C2 CC1COCC(CC(=O)N(C(C)(C(=O)NCC2CC3(CCC3)C2)C2CC2)C)O1 CC(O)C(F)(F)C(=O)N1CC(C(N2CC(N(C)CCO)C2)=O)OC(C)C1 C1(OC)CN(C(=O)CCC(C)SC)CC1NC(=O)CCCSC C1(NC(c2cn3cccnc3n2)=O)CN(C(=O)CC2C=CCC2)C2(CCCC2)C1 C1(CC)CN(C(C2(C)CCCCO2)=O)CCC1NC(c1ccnc(Cl)c1O)=O C12(NC(c3n(C=C)nnc3)=O)CCCC1N(C(c1cnc3ncccn13)=O)CC2 CCC(C)(C(=O)NC1CC2CCC(C1)N2C(c1cnc(=N)[nH]c1)=O)C(N)=O CC(C)(C)CC(F)C(=O)N1CCC1CNC(c1cc(O)ncc1F)=O CC1(C(N2CCC(C3CCCN3C(=O)Cc3cncc(O)c3)C2)=O)CCC(=O)N1 C#Cc1cnn(C)c1C(=O)NCC1=CCCN(C(=O)C(C(C)C)OC)C1 C1(NC(C(C(C)C)OCC)=O)CCCC12CN(C(C1(C)CCCCC1)=O)C2.O N1(C(=O)Nc2c(C)ccnc2Cl)CC2CCC(C1)N2C(c1ccc(OC)cc1)=O C1(C(N(CC(C)O)CCNC(Cc2cc(C)nn2C)=O)=O)CCC12CCOCC2 C1(NC(CNC(=O)OC)=O)CCCC1.n1(CC=O)nnc(-c2ccccc2)n1 c1(SCC#C)cccc(C(=O)NC(C)CCCNC(=O)CC(C)CC)c1 N1(C(COCCN(C)C)=O)CC23CCCC2(C1)CN(C(=O)CC1CCC1)C3 C(=O)(C(C)(C)S(=O)(=O)C1CC1)NC(C)CCNC(c1nccn2nccc12)=O O=C1CC(CC(N2CC(NC(=O)CNC=O)C(c3ccccc3)C2)=O)CC(=O)N1 CCC(C(=O)N1CCCC1C1(NC(=O)CCCc2ccccc2)CC1)n1ccnc1 C1(NC(COCC#C)=O)CC(O)CN(C(=O)CCc2c(C)ncnc2O)C1 Cc1cnncc1C(=O)NC(C1CCOC1)CNC(=O)COC1CCC1 N1(C(C2C(c3n(C)cnn3)CC2)=O)CCC(CNC(=O)CC(F)F)C12CCC2 N1(C(COCC(C)(C)C)=O)CCC2(CC1)CCN(C(c1ccc(Cl)nc1N)=O)C2 c1(C(=O)NC2CC(C)N(C(=O)CCc3cnc[nH]3)C2)cc(=O)c(O)c[nH]1 N(C1COc2ccc(Cl)cc21)C(C1C(C(=O)Nc2nc(C)c(C)s2)C1)=O N1(C(C(F)OC)=O)CCC2(CCCN(C(c3cccc4c(C)[nH]nc34)=O)C2)C1 C(=O)(C(F)(F)C(C)(C)O)NC(C)CNC(C1(C)CC1Br)=O c1(CC)cncc(C(=O)N(CC)C(C)C)n1.c1(C(=O)N)cnn(C2CC2)c1 c1(C(=O)NC(CCC(=O)NCCCC)C)cnc(O)cc1C Cc1nn(C)cc1CC(=O)NCC1CC(C)N(C(c2cc(C(C)C)no2)=O)C1 c1(OCC)cccc(-c2cn(C3CC(C(=O)N)C3)nn2)c1.CC(C)C.C(C)=O O=S(=O)(c1ccccc1Br)N(C1CCOCC1)C1CC1 N1(C(c2ccc(OC)cn2)=O)CCC(NC(=O)Cc2conc2C)C1(C)C N1(C(C(CCO)N(C)C)=O)CC2CC1CN(C(c1ccc(F)c(Cl)n1)=O)C2 c1(CC2NC(=O)N(CCc3nc(N(C)C)sc3)C2=O)ccnc2ccccc12 N1(C(CNC(CCCCC)=O)=O)CC(NC(=O)Cc2coc(CC)n2)CCC1C CC1(CNC(C2CCC(C(N)=O)C2)=O)CN(C(=O)COC2CC2)CCO1 c1(C(=O)NC2CCN(C(=O)CSC3CC3)C23CCC3)cccc2c1CCOC2 N1(C(CCCC#C)=O)CCC(CCNC(c2c(C)oc(Br)c2C)=O)CC1C CC(CN(C)C)C(=O)NCC(C)(C)CC1CN(C(=O)CO)C1.C1CCCO1 c1(C(=O)NC(CC=C)CNC(=O)C=CC2CC2)cccc(CCCCO)c1 N1(C(CC(C)SC)=O)CC2CCCC2(NC(=O)CN(C)C)C1.c1cccc(Cl)c1 CCCCC(C)(F)C(=O)NCC(CC(C)C)NC(C1(CCOC)CCC1)=O CN1CCC(CO)C12CCCN(CC(=O)N(c1ccc(Cl)cc1[N+](=O)[O-])C)C2 c1(N2C(C)CCN(C(=O)CCN3CCC(O)CC3)CC2)ncnc2scc(Br)c12 C1(NC(c2c(C)nco2)=O)CCCCN(C(C2CCC2c2ccc(F)cc2)=O)C1 C(CN=c1[nH]c(=NCC2(C)CC2Br)c2[nH]ccc2[nH]1)C1CN(C)C1 c1(NC(C2CC23CCN(Cc2cc(O)ccc2Br)C3)=O)ccc(O)c(F)c1F CC(F)(F)C(F)(F)CCOC(C1CCC(=C2CCC2)CC1)=O C(C)(C)(CC(=O)NC1(CS(C)(=O)=O)CCOCC1)n1cc(-c2nc(C)sc2)nn1 Cn1cnc2ncnc(NC(C3(c4cccc(-c5ccc(O)cc5)c4)CC3)=O)c12 C1(NC(c2n(CC)ccc2)=O)CCN(C(=O)Cc2cnc(C)o2)CC1CO Cc1nc(C(N2CC(F)(CNC(=O)Cc3cccc(F)c3)C2)=O)c(C)n1C c1(C(N2CC(O)CC(NC(C(C(C)(C)C)=O)=O)C2)=O)ccnc2[nH]cnc12 c1(C(=O)NCCN(CCC#C)C)[nH]c(C)c(C=O)c1C.C(=O)C(C)C.CCC CCCCC(O)CC(=O)NCC1CCN(C(c2[nH]c(O)nc2C)=O)CC1(F)F C1(N(c2c(OC)ccc(OC)c2)C(=O)C#CC(=O)O)COC2(CCNCC2)C1 N1(C(CSC)=O)CCN(C(=O)C=Cc2ccccc2F)C(C(F)F)C1 CCCC(C(=O)N1CCOC(CO)C1)NC(C1CC(CC2CC2)C1)=O N1(C(C(CC)CC)=O)CCCC(O)(CNC(=O)C(C)OCCOCC)CC1 N1(C(CCN(C)CC)=O)CCCN(C(c2cc(O)ccc2Br)=O)C(C)C1 CN1CCCC(O)(CC(=O)NCC2CC(O)CN2C(C2CCC(O)CC2)=O)C1 N1(C(CCCSC(C)C)=O)CCC(CO)(CNC(=O)CC2CCCN2C)C1 C1(NC(c2scc(CNC(C(CC)OC)=O)c2)=O)CC(C)CC(C)(C)C1 C#Cc1cc(C(N2CC(CNC(c3ccc(C)cc3)=O)C2)=O)cc(Br)c1 c1(CC)ccc(CCCC(=O)NCC2C=CCN2C(=O)Cc2cn(C)nn2)cc1 N1(C(c2cncc(SCC)n2)=O)CCN(C(c2nc(C)n(C)c2C)=O)C(CO)C1 C#Cc1cncc(C(=O)N(C2CCCN(C(=O)CCOCC)C2)C)c1.C(C)=O.N N1(C(C(C(C)C)(C)C)=O)C2CCC1CN(C(=O)Cn1cnccc1=O)CC2 C(=O)(CCCCCC)N1CC2(C(C(=O)NCCC#C)C2)C1 C1(C(=O)NCCCC(c2ccccc2)NC(CC(C)C)=O)CCCCCS1(=O)=O c1(-n2c(-c3ncoc3C)nc(CCCCOC)n2)ccc(F)c(Cl)c1 Cn1cc(C(=O)N)c2c(c1=O)CCCC2.C1(C)COCCN(C(=O)CC2CC2)C1.C O=C(CCCc1ccccc1)NC1CCN(C(C2CCCN2CC(F)(F)F)=O)C1 N1(Cc2onc(C(C)OC)n2)C2CCC1CN(C(=O)C(=O)NCCO)CC2 N1(C(CC2CCN(C(C(CCSC)O)=O)C2(C)C)=O)CCn2c(C)cnc2C1 c1(C(=O)NCCC2(C(=O)NCC3(CCCO)CC3)CCC2)sccc1F N1(C(CCCOCC)=O)CCN(C(=O)COCC2CC2)CC1C1CCC1 c1(CNC(CC2ON=C(C)C2)=O)ncc(C(=O)NCC(C)(CO)CO)cn1 c1(C(N(C2CN(C(c3nn(C)cc3Cl)=O)C2)C)=O)ccc(C(F)(F)F)cc1N N1(C(C(CCC)N(C)C)=O)CCC(C(N2CCC2CC2CC2)=O)(CC)CC1 c1(CC(=O)N(CCC)CCNC(c2snnc2C2CC2)=O)ccccc1.C c1(C(=O)NCCN(C(C(C)c2ccsc2)=O)C)cn(C)nc1C(C)(F)F C(C(CC(C)(C)C(=O)O)NC(c1ccc2c(c1)CCCC2)=O)OC.C(C)C(=O)N CS(=O)(=O)c1ccc(C(=O)NC2CCC23CCC3)s1.C(=O)CCC1OCCO1.N C1(NC(C(Cc2ccccc2)N(C)C)=O)CCCCN(C(=O)C(C)(F)F)C1 C(CNC(c1nnn(C)c1N)=O)(CC(=O)NCC1CCCSC1)OC C(=O)(N=S1(=O)CCN(C(=O)C(CCSC)O)CC1)OC.c1(CS)ccccc1 CN1CC(N=c2ccc(Br)c(S(=O)(=O)NC3CCCN(C)C3)[nH]2)CCC1=O c1(C=O)cnc(C2CC2)s1.C(=O)(C=CC(=O)N(C(C)C1CC1)C)N(C)C N1(C(CCCOc2ccc(C)cc2)=O)CCC(NC(=O)C(F)(F)C(C)O)C(F)C1 N1(C(=O)Nc2c(C)non2)CCCC(C(=O)NC2C3CC4C(C3)C24)C1 C12(NC(=O)CC3(O)CCC3)CCCCC1N(C(c1nsc3ccccc13)=O)CC2 C1(C(=O)NCC2(OC)CCN(C(C(=O)NCC)=O)C2)CCc2ccccc2C1 N1(C(C(CC)N(CC)CC)=O)CCC(C(C)CNC(c2ccnnc2S)=O)CC1 C(C)(CNC(C1(NC(=O)C(C2CCCCC2)F)CC(O)C1)=O)(CO)OC c1(OCC)ccc(Br)c(C(N2CCCC2CN2CC(C)CC(C)C2)=O)c1 N1(C(C(CC)CC)=O)CCCCC12CN(C(C1CCC1C(C)(C)C)=O)C2 N1(C(C2CCCS2)=O)CC2CC(C1)N2C(c1ccc(Cl)c(F)c1)=O C1(CNC(C(CCC)F)=O)CN(C(c2c[nH]nc2Cl)=O)CCC12CCC2 N1(C(C2(C)CC2(Br)Br)=O)CC(F)CC1c1nc(-c2ccnc(SC)c2)no1 CC1(C)CN(C(=O)C(Cl)Cl)CCC1C(=O)NC1CC2(C1)CC(O)C2 C1(NC(c2cn(CC(F)F)cn2)=O)CCN(C(c2cnccc2Cl)=O)C12CCC2 C=Cc1cc(C(=O)N(CCC(C(C)(C)C)NC(=O)CCC2CC2)C)cc(F)c1 C1(CNC(C(C)O)=O)CN(C(c2n[nH]c(-c3c(F)cccc3F)n2)=O)CCCO1 N1(c2nccc(C)n2)CC2CCC1C1CN(C(C3Cc4ccccc4O3)=O)CC21 C=C(Cl)CC(C(=O)NC(C)C(CC)CC)NC(=O)C(C(C)C)N(C)C Cn1cnc2c(C(N3CCC(C(F)CNC(=O)CO)CC3)=O)cccc12 C(CCCCC(=O)NC1CC2C=CC1C2)N(C(=O)CC1CCOC1(C)C)C C1(NC(CC(=C)C)=O)CC2CC(NC(=O)CCc3ccc(C(=O)OC)[nH]3)C2C1 CC1(C(=O)NCC(c2ccccc2)CO)CCN(C(c2c[nH]c(C#N)c2)=O)C1 N1(C(C2(C#C)CC2)=O)CCN(C(=O)CN2CCS(=O)CC2)C(C)C1 Cc1cnc(C(=O)N(C)CC2CCCCC2)nc1.c1(C(=O)N)coc(C(N)=O)c1 C(CSC)(C(=O)N1CCCC1CNC(=O)C(N1CCSCC1)C)OC N1(C(c2nn(CC)c(=O)cc2)=O)CC(C)(C)CC1(C)C.c1(C=O)cnc(S)[nH]1.N Cc1cc(C(=O)NC(C)C(CO)NC(c2n[nH]c(C)c2Cl)=O)sc1Br n1(CC)nc(C(=O)N(CCCNC(=O)C(C)CCOC)C(C)C)cc1C C(=O)(CC(C)F)N(CCCC=C)C Cn1nnnc1COC1CCN(C(=O)NC2(CCc3ccccc3)CCCC2)C1 N1(C(C(C2CN(C(C3CCC3)=O)C2)OC)=O)CC(C)(CCOC)C1.C1CC1 C(=O)(C(O)P(C)(C)=O)NC(C)CN(C)C(c1ccncc1Cl)=O Cc1cnc(C(N2CCC(O)C(O)C2)C(=O)NC2CCCC2)c(C)c1 N1(C(c2c(CC)ocn2)=O)CC2(CCC2)CC1C.C1(C(=O)N)CCN(C)C1=O C#CCC(C)(CC)C(=O)N1CCC(=CCNC(C2CCC=CCCC2)=O)CC1 C=CC(CCC)CC(=O)NCC(CNC(=O)CCc1cccc2c1OCO2)OC C(CCC(C)C(=O)NCC1(C)CCCN(C(c2ccc(CF)cc2)=O)C1)OC c1(C(N2CC(OCC(=O)NCC(CC)(C)Cl)C2)=O)ccc(O)c(C)c1 CCC#CCCN=c1[nH]c(=NCC(=C)C)[nH]c2ccc(OC)cc12 C=CCC(CC=C)C(=O)NCCC1=CCN(C(=O)CSCC(F)(F)F)CC1 Cc1ncc(C(=O)NC(C)(C)CNC(=O)C(C)Cc2ccnn2C)o1 c1(C(N(CCCNC(c2ccc(OC)s2)=O)CC)=O)coc2c1C(O)CCC2 C1(C(=O)N)CCCC(C#N)C1.C(C(C)(C)C)N(C)C(C1(c2ccsc2)CC1)=O Cc1nc(C(=O)N(C(C)CCNC(C2(c3ccccc3Br)CC2)=O)C)c(C)s1 Cc1ccc2c(O)c(C(N3CC4(CCC(C(=O)O)OC4)C3)=O)cnc2n1 N1(C(C(CCC)CC2CCCCC2)=O)CCCN(C(C2CC(OC)C2)=O)CCC1 N1(Cc2cnc(C(C)(C)C#N)s2)CCN(CC(=O)Nc2ccccc2)CC1 N1(Cc2c(C)c(F)ccc2)CCNc2ccc(O)cc2C1 c1(C(N(CCCCN(C(C(C(C)C)O)=O)C)C)=O)cc(N)cc(F)c1 N1(C(C=CC=CC)=O)CC2CCN(C(=O)COc3cccc(OC)c3)C2C1 CC1(NC(=O)CSCC2CCCO2)CCN(C(=O)Cc2ccc(F)cc2)C1 C1(C)(NC(C(C)Cc2ccccc2)=O)CCN(C(c2ccc(Br)nc2)=O)CC1 c1(C(=O)NCCCC(C)C)cnc(O)c(F)c1.C1(C(=O)N)CCCN1CC(C)C Cc1cccc(F)c1CN1CC(c2nc(C)c(C(=O)O)o2)C1 CN(C)S(=O)(=O)N1CCOC(C(N2CCCC2C)=O)C1.C(=O)C(F)(F)C1CC1 C(C)C(C)(C)CO.C(CC1CCC1)(C(=O)N)NC(C1C(CCOC)C1)=O Cc1ccc(-c2ocnc2C(=O)NC2CCCC2NC(=O)C(C)CC2CC2)s1 C1(C(CNC(c2cccs2)C)ON)CCCC1 c1(CN(CC(c2noc(C3CC3)n2)O)C)ccc(F)cc1F CN=c1[nH]c(=NCc2ccnc(C)n2)[nH]c(=NCCc2cccc(C)c2)[nH]1 C(=O)(C1=NNC(=O)CC1)N(CCC)CCOC.C(=O)(CC=O)N1CC(O)C1 Cn1cc(C#CCNC(=O)COCCNC(=O)C(O)CC2CCCC2)cn1 c1(C2(C)CCN(Cc3nc4ncccn4n3)CC2)nnc2n1CCCC2 Cc1cc(C)c(C)c(CN2CC(N3CCOCC3)C2)c1C N1(C(C(CCSC)O)=O)C2CCC1CC(CNC(C1CCn3ccnc3C1)=O)C2 c1(C(=O)NCCC2N(C(C=C(CCC)C)=O)CCCC2)ccc2c(c1)CCCC2 N1(C(C2(C)CC2(F)Cl)=O)CC2(CCN(C(C3CCCN3N=O)=O)CC2)C1 C(=O)(C(CC(C)C)NC(=O)CCC(C)(C)c1cccc(Br)c1)NC c1(C=O)cccc(S(C)(=O)=O)c1.N1(C(CC)=O)CC2(C1)SCCC2.C=CCO c1(SCCNC(C2N(C(=O)OC(C)(C)C)CC2)=O)c(O)cccc1O c1(CC)nc(Cl)c(C)c(=NC(C)C2CN(C(=O)CC3CC(=O)NC3=O)CCO2)[nH]1 N1(C(Cc2cc(C)no2)=O)CCCC2(CCN(C(c3c(C)cccc3Cl)=O)C2)C1 N1(C(CCn2c(C(C)C)ncc2)=O)CC=CC(NC(C2(CF)CCC2)=O)C1 CC1CN(C(=O)CC2CC2)CCC1.C(=O)(C1=CCOCC1)N.C(C)(C)C.C=O C12(OC)CCC(C(N3CCCC(N(C(=O)CCCF)CCO)C3)=O)(CC1)C2 C(=O)(C1=C(Cl)CCOC1)NC1CCC(CC(=O)NC(c2ncc[nH]2)CC)C1 C(=O)(C#CC1CCCC1)N1C(C(=O)NC(C2(C(N)=O)CC2)=O)CC2CC21 C1(F)(CNC(C(CC)O)=O)CCCN(C(C2CCN(CCF)CC2)=O)C1 c1(NC(C2CCCN(C(CCC(=O)O)=O)C2)=O)ccc2c(c1)COC2 N1(C(C=CC(=O)OCCCC)=O)CC2=C(C1)CN(C(=O)C(O)C(C)SC)C2 CC(C)CC(C)(C)CN.c1(Cc2nnnn2CCCC2CC2)cc(C(F)F)no1 N1(C(C(c2cnn(C)c2)C)=O)CC(NC(c2cc(C(N)=O)cs2)=O)C2(CC2)C1 N1(C(C2(N(C)C)CC2)=O)CCOC2(CCN(C(=O)C(O)Cc3cn(C)cn3)C2)C1 c1(C(=O)NCCC2CCN(C(C(C)(C)O)=O)C2)ccc2c(c1)NCCC(=O)N2 c1(C(=O)NC(C2CCN(C(C3CN(C)C3)=O)C2)C)c(O)cccc1F CCCC(C)(O)CC(=O)NCC1CC2CCC(C1)N2C(c1cc(N)ccc1Cl)=O N1(C(C(CC)C)=O)CCC(C)(C)C(C(=O)NC2(c3nc[nH]n3)CC2)C1 c1(NC(C2CC2c2ccc(Br)cc2)=O)cccc(C2CC2)n1 CC(C(=O)N1CC2CCC2(CNC(c2cncc(Cl)c2Cl)=O)C1)C(F)(F)F c1(C(=O)NCCCNC(=O)Cc2nnc(O)s2)cc2cccc(Cl)c2o1 CCCC(C)CC(=O)NCC1(CCNC(=O)C(F)(F)c2nccs2)CC1 N1(C(C2CC(=C)C2)=O)CC2CCCC2C1.C(c1ccc(C(N)=O)o1)=CC(=O)N C1(NC(c2cncc(SCC)n2)=O)CCCN(C(=O)C2CC2)C1C C1(NC(c2cnc3n2CCC3)=O)CN(C(=O)C2=C(Cl)CCC2)CC1C1CC1 c1(C(C(=O)NC2CCCC2)=O)ccc2c(c1)CCCC2.C1(C=O)(SC)CC1.C Cc1c([N+](=O)[O-])ccc(F)c1C(N1CCN(C(C2(C)CC2)=O)CC1C1CC1)=O N1(C(CN(C(=O)C=C(C)C(C)C)CCC)=O)C(C)CC2CCCC12 Cc1ccc(C(=O)NC2(C#N)CCN(C(C3(C)COC3)=O)C2)c(C)n1 N1(C(C(C)NS(CC)(=O)=O)=O)CC2CCC1C2NC(C1CC(F)(F)C1)=O c1(C(=O)NC2C(NC(C(=O)NCC)=O)CCCC2)ccc2[nH]cc(C#N)c2c1 C(N=C(NCc1noc(CC2CC2)n1)N1CCC(C)C1)C1C(C)C1 c1(CC)nc(C(N2CC(c3ccccc3)C2)=O)c(C)o1.c1(C(=O)N)coc(C)n1 n1(CC)nc(C(N2CCC(C)C2CNC(c2ncccc2F)=O)=O)ccc1=O N1(C(CCC)=O)CCC(CCNC(c2cnn(CC(F)(F)F)n2)=O)CC1C C(=O)(C(C)CC(C)(C)C)N1CCCC(CN(c2c(C)c(Cl)ncn2)C)C1 CC1(C(=O)NC2CCN(CCCNC(=O)CN3CC(C)(C)C3)C2)CCCC1O C1(C(=O)N)CCn2c(cnc2C(F)(F)F)C1.C(C)(C(=O)NC1CCC1)OC N1(C(C(COC)(C)C)=O)CCC(CCNC(=O)CCc2cnc(C)o2)CC1C c1(C(C(=O)NCC(C)C(C)C)N(C(C)C(=O)N)CC)ccc(O)cc1OC C1(NC(c2nnn(C)n2)=O)CCCC(NC(=O)CCCN2CCCC2)C1 c1(NC(=O)NC2CCCC(C(F)F)C2)ccccc1I C=CC(C)(O)C(=O)NCC1CCN(C(c2ccncc2SCC)=O)C1 CS(=O)(=O)CCCC(=O)NCC1CC1.c1(C2(C(=O)N)CC2)ccc(Cl)nc1 Cn1cc(C(=O)NCCN2CCN(C(C3CCCC3(F)F)=O)CC2)c(O)n1 c1(C(=O)NCC2CN(C(C(C)(C)C)=O)CC2C(F)(F)F)ccnc2[nH]cnc12 c1(-c2cc3ccc(Cl)c(F)c3o2)nc(C2CC2)nn1C1CCc2c(F)cccc21 c1(C(=O)NC(C(C)NC(c2cncc(CC)c2)=O)(C)C)ccc2nncn2c1 C1(N(C)C(c2cc(F)cc(Br)c2)=O)CCCN(c2ncccn2)CC1 C1(C(N2CCC(N(C(=O)C(C)n3ccnn3)CC)C2)=O)C2(CC2)C12CC2 Cc1ccc2cc(C(=O)NC3CC3NC(=O)CCOC3CCC3)nn2c1 Cc1ccc(C(C)(C)CC(C)C(C(C)C)CNC(=O)OC(C)(C)C)nn1 N1(C(COCCCCOCC#C)=O)CCN(C(=O)C(O)P(C)(C)=O)C(CC)C1 N1(C(C(C=C)(C)O)=O)CCN(C(=O)CC2CC(F)(F)C2)CC(O)C1 C(=O)(C(CCCC)CCCC)NC1CC(O)(CNC(C(C)OCC=C)=O)C1 C(CC(C)(C)C)(C(=O)NCCNC(c1ccoc1Cl)=O)OC N1(C(COCCCOC)=O)CC(C(=O)NCc2ncoc2C)C(C)(C)C1 C1CC(=O)N(C2CC2)C1.N1(CCN(C(=O)NC)C2CC2)CC2CCC1C2 c1(CC)ccc(C(=O)NC2CCCC2C)c(C)n1.c1(C(=O)N)cc(C)nn1C c1(CNC(C(CCCCC)C(C)C)=O)ccc2c(c1)CCN(C(=O)C=C(C)Cl)C2 c1(C=O)cnc(O)c2cncn12.c1(CNC(C2C(C)CC2)=O)ncccc1C.N C(=O)(C(CCC1CC1)NC(=O)CC1CCCCO1)NCC#CC C1(NC(C2CC(CC)C2)=O)CN(C(c2cnn(C)c2)=O)CC1C1CC1.C1CC1 S(=O)(=O)(c1csc2ccccc12)N1C(CC)CN(Cc2cnc(Cl)cc2Cl)CC1 c1(NC(CCOCCOCCOC)=O)cccc(OC)c1.c1ccc(C)o1 C12(C(=O)NC(C(C)NC(=O)COC(F)(F)F)(C)C)CCC(C)(C1)OC2 c1(C(N2CCC(NC(C3(OC)CC3)=O)CC2C)=O)ccc(N)c(F)c1F C1(CNC(c2ocnc2C(F)F)=O)CN(C(c2ccc(O)nn2)=O)CC12CC2 c1(CNc2cc(OC(C)(C)C)cc(Br)c2)cccc2ccsc12 C#CCCCC(C)C(=O)N1CC(NC(c2c(CC)nc(C)n2C)=O)CC(O)C1 Cc1c(C(=O)NCC(C2CCCC2)NC(C2C=CCC2)=O)cnn1C(C)C C1(C2CN(C(c3cn(C)c(=O)cn3)=O)C2)(NC(c2c(CCC)[nH]cc2)=O)CC1 N1(C(C2=C(C)CCC2)=O)CCC(C(=O)NCC(CO)N(C)C)CC1(C)C c1(C(N(C2CCCN(C(C)=O)CC2)C)=O)cnc2nc(Cl)ccc2c1 c1(C(=O)NC2C(C)N(C(=O)CCc3ccnn3C)CC2)ccc(P(C)(C)=O)cn1 N1(C(c2c(CC)nccc2)=O)CC2(CCC(Sc3cccc(C#N)n3)CC2)C1 C12(NC(CCC(=O)NCCC)=O)CCOCC1CN(C(C1CCCCC1O)=O)C2 c1(NCC)cccc(C(=O)NCCC(C)NC(=O)Cn2cncn2)c1 c1(CC)nc(C(=O)NC2(CCCNC(=O)C(C)(C)NCC)CC2)cs1 Cc1cccc(C(N2CCCC(CNC(=O)C(c3ncc(Cl)n3C)(F)F)C2)=O)c1O c1(C(=O)NCCCN(C(C2CC(CF)C2)=O)CC)c(C)noc1C(F)F c1(C(=O)NCc2cn(C3CN(C(C=NOC)=O)C3)nn2)sc(C)c(C)c1C c1(C(C(=O)NCC(F)F)N(C2CCN(C)C2=O)C)cccc2[nH]ncc12 Cc1cc(C(N2CCCCC2CN(C)C(c2cc(CO)on2)=O)=O)cc(N)c1O Cc1ccc(C)c(C(=O)NC2CCC(C(=O)NC3CN(C(N)=O)C3)C2)n1 N1(C(C(COC)O)=O)CC2CCCC(C1)N2C(c1cccc(C(C)(F)F)c1)=O N1(C(C2CC(C)OC2)=O)CCCN(CCCCNC(=O)C(F)=C2CCC2)CC1 C=CC1(C(=O)NC2CN(C(c3cc(SC)c(C)o3)=O)CC2C)CCOCC1 C(=O)(C(F)(F)C1=CCOCC1)NCC1C2N(C(=O)C=Cc3ncc[nH]3)C(CC2)C1 C(=O)(CC(C)(C)N(C)C)NC(C(=O)NC(c1nccs1)C)C1CCCC1 N1(CC(N2CCC(NC(CCCCSC)=O)C2)=O)CCn2nccc21 N1(C(c2cc(C)nn2CCO)=O)CC2CCC(N(C)C(c3ccns3)=O)C2C1 N1(C(CCC)=O)CC2C(CNC(c3cncn3-c3ccncc3)=O)C2C1 C1(CCOC)(NC(c2ccc(CC)[nH]2)=O)CCN(C(C2CC2C)=O)CC1 C1(NC(=O)CCC2(NC(c3cc(C(N)=O)c[nH]3)=O)CCC2)C2CCCCC12 N1(C(C2C(COC)C2)=O)CCCN(C(C2CC(=O)N(C3CCCC3)C2)=O)CC1 N(C(=NCCCF)NCC1(C)CCCOC1)Cc1cc(C)c(O)cc1 C1(CNC(c2n(C)ncc2Cl)=O)CCN(C(c2cccc(Cl)c2N)=O)CC1(F)F C1(NC(c2cncc(CO)c2)=O)CCN(C(=O)CC2CCOC2=O)CCC1(F)F N1(C(c2ccccc2)C)CCC(N(C)N2CCOC3CCCCC23)CC1 C(=O)C(=O)C(C)(C)C.N1(C(CC2CN(C(=O)O)C2)=O)CCCCC1.CC(C)C c1(C(=O)NC2(CNC(c3c(C)scc3)=O)CCOC2)cnnc(O)c1 N1(C(CN(C(COC)=O)C)=O)CCC(C(F)F)(CNC(C2CCCC2)=O)C1 C1(C(N(C(CC)CNC(=O)CCC2CCOCC2)C)=O)CN(CC)CCO1 C1(C(C)C)CN(C(C2CC(=O)N2)=O)CCN1C(C1CN2CCN1CC2)=O CCC(CNC(=O)C(C)(CO)NC(C1COC(=O)N1C)=O)(CC)CC C1(O)(CCNC(=O)CCc2cnn[nH]2)CCN(C(c2ccccc2F)=O)C1 c1(C(=O)OC)cccc2c1N(C(c1c[nH]nc1-c1cccc(Cl)c1)=O)CC2 C(CCC(C)C(=O)NCc1ccc(C(=O)Nc2cc(C)cc(F)c2)cc1)OC c1(CC(N)C(=O)N2CC(O)(c3cnn[nH]3)C2)ccc(O)cc1 C12(CCNC(C3CC(O)CN3C(=O)CCCn3cccc3)=O)CC(CCO1)C2 N1(C(CCCOC)=O)CCCN(C)CC1.C12(C=O)CC(c3ccccc3)C1C2 CCCCCCCC(=O)NC1CN(C(C2(OCC)CCOC2)=O)CC1CC CCC(C)C(O)C(C)C(=O)NC1(CN(C(=O)CC(C)(O)COC)C)CC1 c1(C(=O)NC2(C3N(C(C4CCC(=O)N4)=O)CCC3)CC2)ccc2cnoc2c1 c1(N2CC(O)(CNC(c3cc(CSC)c(F)cc3)=O)C2)nc(Cl)nc2sccc12 C1(CC(=O)NCCC(=O)NCC(C)C)CCCCN1C(C1COCCN1C)=O C(=O)(CC(O)CNC(=O)CN1CCCC1=O)N1CCC(C(N)=O)C1 c1(OCCO)ccc(OC)cc1.c1(C2(CN(C)C)COC2)ccccc1Br c1(C(C(=O)N(CCN(C(=O)CNC=O)C)C)O)cccc(F)c1.C1CC1 C(=O)(CC(CC)OC)NCCN(C(C1(CCC)CC1)=O)CCOCC c1(C(=O)NC2CN(C(=O)CC3CC3)CC3(CCC3)C2)nc2ccccc2cc1Cl c1(C(=O)NC2CN(C(C3(CCOCC)CCC3)=O)C2)cnc(C(C)C)o1 CCCCC(C(=O)OC(C)(C)C)NC(=O)NC1CCCC(O)C1 C1(N(CC(c2ccccc2)N(C)C)C)CCN(C(c2cscn2)=O)C1 CC1CC(NC(C2SC3C=CC2CC3)=O)CCN1C(c1cnn(C(C)(C)C)c1)=O c1(C(C)NC(C2CCC[Si](C)(C)C2)=O)cc2ccc(C#N)cc2[nH]1 N1(C(CC2CC(OC)C2)=O)CC2CCN(C(C3CCCN3C)=O)CC(C2)C1 CC(C)CC=O.CC(C)(C)C.C1(C=O)CCCC1C(F)(F)F.[SH](C)(=O)=O.N Cn1ccc2c(C(=O)NC3CCCC3NC(C3CC=CCO3)=O)ncnc12 N1(C(C#CC(C)(C)C)=O)CCC2(CC1)CC2CNC(=O)CCN1CCC1 C1(C(N2CCC(CCC)C2)=O)CCCN(C(c2c[nH]nc2Cl)=O)CC1 C(=O)(CCCC(=O)NC1C2CC3C1C3C2C(=O)N)OC.CCN(C)C(C)C c1(CC(=O)NC2(CO)CN(C(CC(CC)SC)=O)C2)nnc2n1CCOC2 N1(C(C2(C#C)CCCC2)=O)CC(C)N(C(c2ccc(OC)c(C)c2)=O)C(C)C1 C#Cc1c(NCc2c(C)nn(CC(=O)OC(C)C)c2C)cc(Br)cc1F C1(CNC(c2c(CC)ccs2)=O)CCCC2CN(C(=O)C(C)(C)CSC)CC12 c1ccc2c(c1)CCN(C(c1nc(Cl)cs1)=O)CC2.CC(C(=O)N)NC(N)=O.C C1(C(N2CC(CNC(CC3C(C)C3)=O)OCCC2)=O)CCc2nc(O)[nH]c2C1 c1(C(=O)NC2C(CC)CN(C(=O)C(N)=O)CC2)cccc2cnnn12 N1(C(c2c(CCNC(c3[nH]cc(C)c3)=O)n[nH]c2)=O)CC2(CCC2O)C1 c1(C(=O)NCC2CC3CC3N2C(c2cc(F)c[nH]2)=O)cnc2n1CCCCC2 CCC(C)(C#N)C(=O)N(CCCNC(c1coc(-c2cccnc2)n1)=O)C1CC1 C1(C)(C(=O)NCC(CNC(C(c2ccc(F)cc2)CC)=O)C)CC(F)(F)C1 CC(C)CC(C)CC(=O)NC1CC2(C1)CC(NC(c1cnn3cccc3c1)=O)C2 N1(C(C2N(C)CCC2)=O)CCC(N(C(=O)CSC(F)(F)F)CC2CCC2)CC1 C1(NC(c2cc(C(N)=O)[nH]c2)=O)(CNC(c2snc(O)c2Cl)=O)CCOCC1 N1(C(C(CC)CC)=O)CCC2(CC1)CC2NC(=O)Cc1cnc(C)[nH]1 Cc1nc(NCCc2ccc(F)cc2Cl)cc(N2CCCC(CS(C)(=O)=O)C2)n1 Cc1ccc(-c2cn(CC3CCN3C(c3cnnn3C)=O)nn2)c(F)c1 C1(NC(COCC=C)=O)(CNC(C2CC(CF)C2)=O)CC(F)C1 CC1(C)CCCCC1C(N1CC(NC(c2nnn(C(C)(C)C)n2)=O)C1)=O N1(C(Cc2c(C)n[nH]c2C)=O)C(C)CN(C(c2cnn(C)c2C#N)=O)CC1C C(C1Cc2ccccc21)NC(C1C(CNC(CCCN(C)C)=O)C1)=O c1(C(=O)NCC2(F)CN(C(Cc3c(C)scc3)=O)C2)cc2c(C)sc(C)c2s1 c1(C(N(C2CC(NC(C3CCC([N+](=O)[O-])CC3)=O)C2)C)=O)cc2ncccc2o1 CC(C)CC(C)(CNC(N1CCCN(c2ncccn2)CC1)=O)CO N1(C(CNC(c2c(C)occ2)=O)=O)CCN(C(=O)Cc2cscn2)C(C2CC2)C1 c1(C(=O)Nc2cncs2)cc2ncc(-c3ccnc(OC(F)F)c3)cc2[nH]1 Cc1cc(C(=O)NCC2C(C)CCN2C(=O)C=Cc2scnc2C)cc(Cl)c1 C#CCC(C)N(C)N1CCOC(c2ccccc2OCC)C1 Cc1cc(N)c(C(N2CC3CC2CCN3C(c2ccn(C)n2)=O)=O)cc1F N1(C(=O)C2=COCCO2)CCCC12CCN(C(C13COCC(C1)C3)=O)CC2 c1(C(=O)NC2CC(NC(C=C(C)c3cccs3)=O)C2)ccc(F)c(N)c1F Cc1cc(N2CCC3(CC2)CC3C#N)ncc1S(=O)(=O)NC1C2COCC12 C1(C(=O)N)CCC2(CCC2)O1.C1(NC(c2csc(C)c2)=O)CCC(F)(F)C1 N1(C(c2n(C)ccn2)=O)CCC(C2CN(C(=O)C(F)(F)c3ccccn3)C2)CC1 Cc1cccc2c(CC(N3CC(C)(C)CC3CNC(=O)C(N)=O)=O)c[nH]c12 C(C)(C(=O)NCc1ccc(C(=O)N)o1)(C1CC1)OC.c1(C(C)C)ncc[nH]1 C1(NC(c2ccc(COC)cc2)=O)CN(Cc2cccnc2C)CC1(C)C C1(NC(CC)=O)CN(C(=O)C(F)(F)CN(C)C)CC2CC12 N1(C(CSCCOC)=O)CCC2(CC2)CC1C(=O)NCC.c1ccccc1.O N1(C(C(C(C)SC)O)=O)CC2CCN(C(=O)CCNc3nnnn3C)CCC2C1 C(N=C(NC(C)C)N1CCC2C(C1)C2(F)F)c1cnc(COC)s1 N1(C(C2C(CC)C2)=O)CCN(C(c2cc(C3CC3)ncn2)=O)CC1C(C)C C12CC(CO1)N(C(c1ccc(CC(N)=O)cc1)=O)C2.C(C=O)SCCOC.N c1(C(N(CCNC(CCc2cc(C)on2)=O)C2CC2)=O)c(C)nc(CO)nc1C C1(C(=O)NC(C)C(N2C(CO)CC2CC2CC2)=O)CC(CO)C12CCC2 c1(C(N2CCC(O)C2)=O)cccc2c1OCC2C.C(C(=O)NC)N(C(=O)OC)C Cc1sc2ncc(C(=O)NC3CCC3NC(=O)C(C)(C)F)c(=O)n2c1C c1(OC)cc(C)c(C(=O)NC(C)C2CC2)c(F)c1.C1(C#N)(C=O)CC1.N Cc1cc(C(=O)N(C)CC2CN(C(=O)C=CS(C)=O)CCO2)n(C(F)F)n1 N1(C(c2ccc(OC)cn2)=O)CCCN(C(c2cc(Br)c[nH]2)=O)C(CO)C1 N1(C(C2C(C)C2)=O)C2CCC1CC(NC(=O)C=CC1CCOCC1)C2 C(=O)(CCCC(=O)NC1CC2C1CCN2C(c1ccnc(O)c1)=O)N(CC)CC CCC(CN(C(C1CCC1)=O)C1CC1)CC(C)C.c1(CCC(=O)N)cccn1C c1(NC(C)C)ccc(C(N2CCCC2)=O)cc1F.C(=O)(C(C)(C)C1CC1)NC.C C(=O)(C(C)(C)CCC#N)NCCCC(C(=O)NCc1nc(C)sc1)O c1(N2CC(NC(c3c(C)cco3)=O)C2)ncnc2c1cnn2-c1cccc(Br)c1 C(CO)(CCCNC(c1cc(Cl)n[nH]1)=O)NC(c1cn(C(F)F)cn1)=O CC#CCC(C)NC(=O)C(O)C1CN(C(=O)Cn2nccc2C)C1 N1(C(c2cc(C)c(Br)s2)=O)CCN(C(=O)COC2CCCCCC2)C2CC12 C1(C(=O)NCC2CN(C(C(C(C=C)C)C)=O)C2)CCC2(CC1)OCCO2 c1(C(CNC(=O)NC2CC2F)O)ccc(Br)cc1 C(=O)(C(C)(CSC)OC)NC1(CC)CN(C(C2CCS2(=O)=O)=O)C1 N1(C(C(CCC)=CCC)=O)CC(NC(=O)CC2CC(O)C2)CC2(CC2)C1.C C1(CNC(C2=CC(C)C2)=O)CC(C)CCN1C(=O)CCCCCN(C)C N1(C(C(C)(C)NC(=O)CC2CCC(=O)N2)=O)CCC(O)(C(F)F)C1 CC(C)(C)C(O)C(=O)NCC1(O)CN(C(c2ccc(Br)c(Br)c2)=O)C1 C(N=c1ccnc(NCc2ccc(F)cc2F)[nH]1)C1(OC(C)C)CCOC1 C1(COC)CN(C(c2cnn(C3CCC3)c2)=O)CCC1N=c1cc[nH]c(C#N)n1 N1(C(COC2(C#C)COC2)=O)C2CCC1C(F)CC2.N1(CC(=O)N)CC2CC2C1 C(=O)(C1CCCc2nccn21)N1CC(NC(c2sccc2Cl)=O)CC(C)C1 Nc1ccc(C(=O)NC2CCCN(C(c3ccc[nH]3)=O)CC2)nc1N CS(=O)(=O)c1cccc(NC(=S)NNC(c2ccc(F)c(S(N)(=O)=O)c2)=O)c1 c1(C(=O)NC(C(C)NC(CCn2ccc(C)n2)=O)CO)cncc2c1CCCC2 N1(CC)CCOCC1CC(=O)NCCCN(C)C(C1CCC(C)(C)C1)=O N1(C(C(CC(C)C)NC(=O)C=Cc2cn(C)cn2)=O)CC2(CCC(=O)NC2)C1 C=CCC(C)C(=O)NC1(CNC(c2oc(C3CCC3)nc2C)=O)CCCC1 C1(C(=O)NC2CCCC2CNC(=O)CS)(CC)CCCO1.c1ccncc1 c1(CCCC)ccc(CC2(OC)CN(C(=O)N)C2)cc1.C1(C(=O)CC)CC1.C c1(C(=O)NC2(C)CN(C(=O)C(F)C3CCC3)C2)ccc(N2CCCCC2=O)cc1 CC(C)(Cc1ccccc1)CC(=O)NC1CC2CC1N(C(C1(CCF)CC1)=O)C2 c1(C(N2C(C(=O)NCc3ccsc3)C=CC2)=O)cc(O)cc(O)c1 C1(C(=O)Nc2ccc(COC)cc2)CCN(C(=O)C2CC2)CCO1 c1(C(C)NCc2cnc(N(C)C)n2C)cccc(Cl)c1Cl C(=O)(N=c1ccn(-c2ccccc2C#N)[nH]1)c1ccc(CN2CC(C)OCC2)o1 C(=O)(C(C)(O)CC(C)C)NC1CC(NC(Cc2c(C)nc(S)s2)=O)C1 N1(C(C2CC3CSCC(C2)C3)=O)CCC2CC2(CNC(=O)C(F)(F)CO)CC1 c1(Cn2cc(C(Cc3ccccc3F)NC)nn2)ccnc(F)c1F C12(CNC(c3c(C)nccc3Cl)=O)CCCC1N(C(=O)C=C(Cl)Cl)CCC2 C12(C(=O)N)CCCC1CCN2C(C1CC(C2CC2)=NO1)=O.Cc1n[nH]c(C)c1C CC1(NC(C2CCCNC2=O)=O)CCN(C(=O)CCC(=O)c2cccc(Cl)c2)C1 N1(C(C(CC)C)=O)CCN(C(=O)CN(C)C(=O)OC)C2CCCC2(C)C1 Cc1ccc(C(N2CCC(C(=O)N(CC(C)C)C(C)(C)C)C(O)C2)=O)cc1C C(=O)(C(CNC(=O)CSCCOC)CC=C)N1CCC(CC#C)CC1 CC1=C(C(=O)NCC2CC2NC(c2cn(C)c(=O)cn2)=O)CCCO1 C1(C(N2C(CCCNC(CCCC(C)O)=O)CCC2)=O)Cc2ccc(F)cc2C1 CP(C)(=O)C(O)C(=O)NC1CCC(CNC(c2ccccc2O)=O)CC1 c1(C(=O)N)cc2cc([N+](=O)[O-])ccc2s1.C1CCN(C(C2(C(N)=O)CC2)=O)C1 N1(C(c2ccn(CC)n2)=O)Cc2ccc(C(C)NC(=O)CC(C)(C)F)cc2C1 C1(COC)CN(C(C2CCC(C(F)(F)F)CC2)=O)CCN1C(=O)CC(C)O C12(C(=O)NCCN(C(=O)C(O)C3CCCC3)CCC)CC1COC21CCC1 C(=O)CCCC=O.c1(C(N(CC)CC)=O)cn(C)nc1C(F)(F)F.CCC C1(C=O)CCCCC1C1CC1.C1(CNC(C2(NC(C)=O)CCC2)=O)CCCC1 CCCCCCCC(=O)N(C)CC1(CNC(=O)C)CC1.c1ccc(F)c(Cl)c1.O c1(C(=O)NC(CC(=O)OC)c2cncs2)cc(I)cc(I)c1I c1(-c2c(SCC3(CC)CC3)cco2)nc(-c2ccccc2Cl)nn1C(C)CC c1(-n2c(COC3CCOC3)nc(C3C(C)C3)n2)ccc(Cl)c(Cl)c1.c1nccn1C C1(C(C)C(=O)NCCCC2CCC2)CCCN(C(c2cnsc2)=O)C1 CC(C)C(C(C)NC(=O)CCCc1cnn[nH]1)NC(=O)CCOC1CC1 Cc1ccc(S(=O)(=O)CCC(=O)N2CCN(C(=O)Cc3csnc3C)CC2)cc1 C1(C(=O)NC(C#C)(C)C)CCC(C)(C)C1.C(=O)(C(C)C)N(CC=O)C.N c1(C(N2CC(C(N)=O)(CNC(C3CC3F)=O)C2)=O)cccc2c1CC(=O)N2 N1(CC(=O)N(C)C(c2ccc(Br)cc2)=O)CC2(CCC23CCC3)C1 N1(C(CC(=O)OC)=O)CCCCC1CN(C(=O)C(C)(C)n1cnnn1)C N1(C(CN(CC)CC)=O)Cc2occ(C(=O)NC34CCC(C3)OC4C)c2C1 C(=O)(CC(C(F)(F)F)NC(c1nnccc1C)=O)NC1(c2ncc(C)o2)CC1 c1(OC)ccc2c(c1)C(C(=O)NC1CC(=O)N(Cc3ccccn3)C1)CC2 c1(C(=O)NC(C(C)F)C)cccnc1CNC(=O)CCCOC1CCOCC1 C1(CCC)(N(C(C2CCN(C)C2=O)=O)CC)CCN(C(=O)C(O)C(C)CC)CC1 C(=O)(C#CC1CCOCC1)NC1CCC(CNC(Cc2cccc(OC)c2)=O)C1 N1(c2cc(NCCC3CCCO3)nc(C)n2)CCc2cccc(F)c2C1C c1(C(=O)NCCC(C)N(C)C(c2cncn2C)=O)cnc(O)c(Cl)c1 c1(CC)ccc(F)c(C(=O)NCC(CO)NC(c2cnc(OC)cn2)=O)c1 N1(C(CCCc2onc(C)n2)=O)CC2(CC(NC(c3ccc(O)cc3F)=O)C2)C1 C(c1cccc(Br)c1)=CC(N1CC(C(C)NC(CCOC)=O)C1)=O C1(C(=O)NCC(N(C)C(C2(C#N)CCCOC2)=O)C2CC2)CCc2n[nH]cc2C1 C(=O)(CC1COc2ccccc21)NC(C)(C)CCNC(=O)C1=C(Cl)CC1 N#Cc1ccc(C(N2CCC(NC(=O)C(Cl)(Cl)Cl)C(F)C2)=O)cc1 c1(C(N)=O)ccc(C(N2CC(NC(=O)Cc3ccoc3)C3CC3C2)=O)c(Cl)c1 CN1CC=C(CCNC(c2cccc(CS(=O)(=O)NC(C)(C)C)c2)=O)CC1 C12(NC(C3OCC(C)(C)C3)=O)CCC(C1)N(C(c1cc(N)c(F)cn1)=O)C2 c1(C(=O)NC2CCN(C(c3n[nH]c(C)c3C)=O)C2)cc(O)nc2ccc(F)cc12 c1(OC)cc(F)cc(C(N2CCC3(NC(=O)C4=CCOCC4)CCCC23)=O)c1N n1(CCC)nccc1C(COC(C)(C)C)NCc1nnnn1CC C=CCCC(C(=O)NC(C)C(=O)NC1CC1)NC(c1n[nH]cc1C#C)=O c1(N2CCC(NC(N)=O)CC2)ncnc2c1ncn2C1CC(CO)C(O)C1O C(=O)(C#CC1CCCCC1)N1C(CCN(C)C(C2OCCO2)=O)CCCC1 c1(C(=O)NC(C(C)NC(C2N(CC)CC2)=O)(C)C)cc([N+](=O)[O-])ccc1 c1(C(N(C)CC2CCCN(C(C3CC(CCO)C3)=O)C2)=O)c(F)ccc(F)c1F Cc1ccc(C(=O)NC(C)CCNC(=O)CO)nc1O.c1ccc(CC#N)cc1 C1(CNC(C2C(C)CC2)=O)CCN(C(=O)Cn2ccnn2)CC1O C1(OC(N(C)C)=O)CN(N2CCC(Cc3sc(O)nc3O)C2)CCO1 CCCC(C(=O)N(C1CCCN(C(C2CC3CCCC23)=O)C1)C)OC N1(C(CCCC)=O)CCN(C(C2CC(O)C2)=O)CC(CO)C1 N1(C(C(CC)N2CCCC2=O)=O)CCN(C(C2(C(C)C)CC2)=O)CC1 c1(C(N(CCCNC(C(C(CC)CC)C)=O)CC)=O)cc2cc(F)ccc2[nH]1 n1(CC(=O)NC2CCN(Cc3ccc(F)cc3Cl)CC2O)cc([N+](=O)[O-])cn1 C1(C(N2CC(OCCNC(CCC(CC)C)=O)C2)=O)CCc2n[nH]cc2C1C c1(C(=O)NCCCN(C(C(C)CC(F)F)=O)CCO)c(N)ccc2nccnc12 N1(C(c2ccc(OCC(=O)OCC3CCCO3)nc2)=O)CCC(O)C12CCC2 c1(CC(=O)N(C2CCN(C(c3c(CC)ncs3)=O)C2)CC)cnccc1C C1(C(N2CC(C(C)NC(=O)C(C)SCC(F)(F)F)C2)=O)CCCC12OCCO2 C1(CC(N2C(C)(CNC(C3(CCCF)CC3)=O)CC2)=O)CCCC12CC2 N1(C(CC(C)CNC(c2cc[nH]n2)=O)=O)CCC2CC1C(=O)O2 Cc1ccnc(C(=O)NC(C2CC=CCC2)C(=O)N)c1N.C1(C(N)=O)CCC1.C c1(CC)cc(C(=O)N(CCC(C)NC(C2(C3CCCO3)CCC2)=O)C)on1 Cc1ccc(C(=O)NC2CC(NC(c3cc4n(n3)CCC4)=O)C2)c(F)n1 CC1=C(C(=O)NCCC2CCC(NC(C3CC4(CCCCC4)C3)=O)C2)SCCO1 c1(C(=O)NCC(CNC(C2C(=C)C2)=O)F)cc(S(N)(=O)=O)sc1C C(=O)(CCN(OC)C(=O)CN(C)C(C)C)NC(C(=O)OC)OC N1(C(c2ccc(N3CCOCC3)nc2)=O)CC2CC(C1)N2C(=O)COCC(F)F CCC(C(=O)NCc1nc(C(=O)Nc2ccc(C)c(Cl)c2)c(C)o1)C(C)C c1(OC)ccnc(-c2nc(C3CC34CC4)nn2Cc2ccc(C(F)(F)F)cn2)c1 Cc1ccc(C(=O)NC(C2CCN(C(C3CCCC3O)=O)CC2)C)cc1O N1(C(C(CCC)CC)=O)CCC2CN(C(=O)C(c3cscc3Br)=O)CC12 Cc1cccc(C(=O)NC2(CF)CN(C(=O)CSC3CC3)C2)c1C#N C1(C(=O)NC(CNC(c2cnc(C(C)(C)C)o2)=O)(C)C)CCc2c[nH]nc2C1 C(=O)(CC(O)CC(C)(C)C)N(C(C(N1CC(OCCCCC)C1)=O)C)CC C(CCCC(=O)NCC1CCN1C(C)C(=O)NCc1ccccc1F)SC C1CCOC1C(=O)N(CCN1CCOCC1)C1CC1.C1(C=O)(CC)COC1.N CC1=CCSC1C(=O)N(C1CC1)CC1CCCN1C(C1CCCN1C)=O N1(C(c2cc(C(C)(C)C)n[nH]2)=O)CC2C(C)C2C1.C1(CC(=O)N)CC12CC2 N1(C(CC(C)O)=O)CCN(C(C2CC2C(F)(F)F)=O)C(C2CC2)C1 C1(NC(C(C)C2CCC2)=O)C=CCN(C(C2(c3cccc(Cl)c3)CC2)=O)C1 S(=O)(=O)(c1ccc2ncsc2c1)N1CC(C#N)N(C(C2CC2(F)F)=O)CC1 C1(C(=O)NCC(CC)(CC)CO)CN(C(=O)CC(=O)NC(C)C)CCC1(C)C c1(OCC=C)ccccc1C(N1CCCC(C(C)(O)C)C1)=O.C(=O)CNC=O c1(C(=O)OC)ccc(C(N)CC(=O)NCC(C2CCCNC2)C)cc1 C1(NC(CSCCC(C)C)=O)CC2CCC(C1C)N2C(=O)CC1CCCCCC1 c1(C(C(=O)N(CCCNC(C(C)OC)=O)C(C)C)C)cc(C)cc(F)c1 c1(C(=O)NC2CN(C(CSCC)=O)CC23CC3)nc(Cl)c(=O)[nH]c1N N1(C(C2(C)COCCO2)=O)CCN(C(=O)CCn2ccnn2)CC12CCC2 C1(C(=O)N(C)OC)(CCC=C)CN(C(c2cc(C3CC3)[nH]n2)=O)C1 n1(CCCC)cc(C(=O)NCCN(C)C(C2CCCCC2)=O)c(C)n1.C(C)=O Cc1nc2sccn2c1C(=O)NCCN(CC(C)O)C(c1ccc[n+]([O-])c1)=O c1(CCC(=O)NCCC2CCN(C(=O)C#CC3CC3)C2)cc(Cl)cc(Cl)c1 CN=c1[nH]cc(C(=O)N(C)CC2(O)CN(C(=O)C(C)OCC(F)(F)F)C2)s1 C1(NC(C(C)=C2CC2)=O)CCC2CCN(C(C3CC4CC4C3)=O)C1C2 CC(C)(F)C(C)(F)C(=O)N1CCN(C(C2COC2)=O)C(C2CCC2)C1 Cc1cc(C(=O)NCC(C)(F)CNC(C2CC2(C)C(F)F)=O)co1 C(C)(C(=O)NN=c1sc2ccccc2n1C)SCCC(C)C N1(C(C(=O)NCCOCC)C(C)CC)CCOC2(CCOCC2)C1 c1(SC)cc(C(N2CCC(NC(c3cnc(C(F)(F)F)nc3)=O)C2)=O)ccn1 C(=O)(N=c1[nH][nH]c2ncc(Br)cc12)C1N(C(c2cc(C)c(F)nc2)=O)CCCC1 Cc1ccc(CCC(N2CC(NC(c3cccn3C)=O)CC(F)C2)=O)c(C)c1 N1(C(CCN(C(C)=O)C)=O)CCCOC(CNC(=O)CC2CCOCC2(C)C)C1 C1(C2N(C(C(C)C)=O)CCC2)CCCN(C(c2cccnc2O)=O)C1 c1(C(N(C(C(=O)NCC(=O)N(C)C)(C)C2CC2)C)=O)cc([N+](=O)[O-])c[nH]1 Nc1cc(NC(=O)Nc2cccc(CS(=O)(=O)Cc3ccccc3)c2)cc(Br)c1 Cc1cc2nccnc2cc1C(N1CCCC(CNC(=O)CC(C)O)C1)=O c1(CC(=O)N(CC)C2CC2)cccc(C2CC2)c1.CCC=O.C(C)(C)C.O c1(SCC)ccccc1CC(=O)NCC1CN(C(c2nc(C)oc2C)=O)CCO1 C=CC(C)(C)CC(=O)N1CCC(C)C(CNC(c2cc(C(C)=O)cnc2C)=O)C1 c1(C(N2CCC(NC(CC3(OC)CC3)=O)C(C)C2)=O)cn2ccc(C)cc2n1 O=C(CCCN=c1nccc[nH]1)NCCC1CCCN(C(C2CC2Br)=O)C1 N(C(=NCC1CC1)NCC1CCN(CC(F)(F)F)CC1)CC1(OC)CCSC1 c1(C(=O)NC2(C3N(C(C(CC)F)=O)CC=C3)CC2)ccc(S(N)(=O)=O)s1.O CCC(CC1CCCC1)C(=O)NC1CC1NC(c1c(C)cnn1C)=O Cc1ccc(S(=O)(=O)Nc2ncc(-c3ccc(C(F)(F)F)c(F)c3)cc2O)cn1 C1CCN(C(=O)CC2(O)CCCC2)C1.C#CC(C)(C1CCOC1)NC(=O)CO Cc1nnc(=NCC2CCC(NC(=O)C(F)Cc3ccccc3)CC2)[nH]c1C C1(NC(C2(CC#C)CCCC2)=O)C=CCN(C(=O)CC(C)n2ccc(C)n2)C1 c1(C(C(=O)OCCN(C)C)NC(=O)C(N)CO)ccccc1.c1ccccc1 N#Cc1ccc(NC(N2CCC(OCC(F)(F)CC3CC3)CC2)=O)cc1F N(C(=NCCC(=O)NCC)N1CCC(Sc2ccccn2)C1)CC1(C=C)CC1 C1(C(N(C2CCOC2)CC#C)=O)CCN(C(=O)c2cncc(OC)n2)O1 C1(NC(c2[nH]cc(C)c2)=O)CCC(NC(C23CCC(C2)C3)=O)CC1 c1(C(=O)NC(C2CCN(C(=O)CCC(=O)N)C2)C)cnc(N(C)C)cn1.CCO N1(C(c2ccc(C(=O)NCc3cc(C)[nH]c3C)cn2)=O)CCC2(C1)CC2(F)F N1(C(C2(C)ON=C(C)C2)=O)CCOC2(CCCN(c3cc(C)nc(CO)n3)C2)C1 CC(C)C(CC(=O)N(C(C)CCNC(=O)CNC(N)=O)C)c1ccccc1 Nc1cc2c(cc1C(N1C(CNC(=O)C(O)C(F)F)CC3CCCC13)=O)OCO2 n1(CCC(N2C(CNC(c3ccns3)=O)CC3CC32)=O)ccc2ccccc12 CC(C)(C)C(CNC(=O)CC1(C)CCOC1)NC(=O)Cn1cnnn1 N1(C(C(CC=CCC)C)=O)CCCC2CN(C(=O)CN(C)C)CCC12 C(CC(CNC(=O)CN1CSCC1=O)NC(C1CC(C)(C)C1)=O)OC C1(OCCC)CCCN(C(c2cn(CC3CC3)nn2)C(=O)NC2(C)CC2)C1 N1(CC=O)CCc2sccc2C1.N1(C(C=CC=CC)=O)CCC(C)(CC)C1.N c1(C(N(C2CCC(Nc3nccc(OC)n3)CC2)C)=O)ccc(F)c(OC)c1 N(C1COc2ccccc21)C(C1CC2CC2N1C(c1ccco1)=O)=O Cc1nc(C(N2CCCC2CN(C)C(C2(CC(F)F)CCC2)=O)=O)co1 C(N=c1cccc(S(=O)(=O)NCC(N2CC(C)OC(C)C2)C)[nH]1)C1(OC)CCC1 C1(C(=O)NCCC2CCO2)CC2CC1CN2C(C1C2C=CSC12)=O C(=O)(CC(CC)C1CC1)N(CC(CC)NC(c1ccccc1O)=O)C C(=O)C(C)S(N)(=O)=O.C(=O)(CCC1CCC1)N1CCC1.C(=O)(C)NC.O Cc1c(C(=O)NC2CC3CC2CN(C(=O)Cc2cc[nH]n2)C3)sc2ccccc12 N1(C(C(C=C)O)=O)CCC=C(C(=O)Nc2cccc(COC)c2)C1 Cc1nc(Cl)ccc1C(=O)NC1(CNC(=O)CC)CCCCC1C.CC(C)C.O C1(C(C(=O)NCCCN(C(=O)C(n2ccnc2C)C)CC)O)CC(F)(F)C1 c1(C(=O)NC(CNC(CC2C(C)(C)COC2)=O)(C)C)ccc(O)c2ncccc12 C1(CC(=O)NCCCCN(C(CC(C)OC)=O)C)CCC2(CCC2)CO1 N1(C(CN(CC)CC)=O)CCC2(CC(C(=O)NCCN3CC4CC4C3)C2)C1 C1(CC)CN(C(=O)C(F)(F)CC)CC1NC(c1nn[nH]c1Cl)=O N1(C(CC2(NC(C)=O)CCCCC2)=O)CCC(NC(=O)C(=O)CC(C)C)C(C)C1 c1(C=O)ccc(S(=O)(=O)CC(N)=O)cc1.C1(C(=O)NCCCC)CCOC1=O.N Cc1cc(Cl)c(C(N2CCCCC2Cn2cncn2)=O)cn1 Cc1cc(CNC(c2c(F)cccc2I)=O)ncc1CO C=CCC(CC)C(=O)N(C(C)C(=O)NCC(O)CC)C c1(N(C)C)ccncc1C(=O)NC(CC(N)=O)c1cn(Cc2cccnn2)nn1 C1(C(C(=O)NC(c2cccs2)CC)C)CCN(C(C2CCCN2CC)=O)CC1 N1(C(C2C(=C)C2)=O)CCN(C(=O)Cc2ccoc2C)CC1COC c1(C(N(CC(C=C)(C)O)CC)=O)cccc2c1OC(C)(C)C2 N1(C(C2C3N(C(c4c(C(C)C)occ4)=O)C(CC3)C2)=O)CC2(C1)OC(=O)NC2C c1(C(=O)NC2CCN(C(COC)=O)C23CCC3)cccc2c1ncn2C C1(O)(COC)CCCC1(C)C.C12(CCSC1)C(=O)N2.C1CCOC1C(=O)N N1(C(C(C2CC2)NC(=O)N(C2C3CCC23)C(C)(C)C)=O)CC=CC(O)C1 N1(C(CC(C)(C)NC(c2ccc(OC)s2)=O)=O)CCOC(C)(C)C1 C(CC(=O)NCCCOC1CC1)N(C(=O)Cc1cccs1)C C1(CC)CN(Cc2cccc(OC)c2)CCN1C(c1cccnc1OC(C)=O)=O C(=O)(CCCCC(C)(C)C)N1C(C)CN(C(c2nc(C)nn2C)=O)C(C)C1 C(C)(C(C(=O)N(C)CC1CCCCC1)C(C)C)NC(CCC(CC)OC)=O c1(OC)ccc(C(N2CC(NC(c3ncccn3)=O)CCC2C)=O)c2ccoc12 N1(C(CC(CC)N(C(=O)CN2CCCCC2C)C)=O)CCCC(O)C1C N1(C(C2CCC(O)C2)=O)CC2(CCC(NC(C3(F)CCCOC3)=O)CC2)C1 CC1CCc2nc(N3CCCC(C(F)(F)F)C3)[nH]c(=NCCCC3CC3)c2C1 N1(C(COC(C)=O)=O)CC2CCC1CN2C(=O)CCc1cccc(Cl)c1 c1(C(N2C(C(=O)Nc3c(C)ccnc3Cl)CSCC2)=O)ccc(F)c([N+](=O)[O-])c1 c1(C(N2CCN(c3ccc4nc[nH]c4c3)CC2)=O)cc(Cl)c2ccccc2n1 N1(CC)CC(NC)CCC1=O.c1(C(N2C3CCC(C3)C2=O)=O)ccc(C)nn1 Cc1noc(CNC(=O)CCn2cccn2)n1.c1(C(C(=O)N)=O)cnn(C)c1 C(=O)(C(F)C(F)(F)F)N(C)CC1CCN(C(c2ccc(CCC)[nH]2)=O)CC1 C(CCC(=O)NCCCN(C(=O)CCOC1CCOC1)CCO)C1C(C)C1 N1(CC(=O)NC)CCC(NC(=O)C(c2ccccc2Cl)N)C(O)C1.c1ccns1 CC1OCCOC1C(=O)NC(C1CCCN1C(c1cccc(N(C)C)n1)=O)(C)C C(=O)(CCCCCCNC(C1CC2(C1)CC21CC1)=O)N1CC(CCOC)C1 N1(C(c2ccc(NC(C)=O)o2)=O)CC(C2CC2)C1.C1(CC=O)CCCC(C)O1 C12(NC(C3C(C)C3)=O)CCC(CC1)N(C(=O)Cc1nc3cnccc3[nH]1)C2 c1(NC(CC(=O)NCCN(CCOC)CC)=O)ccccc1OC N1(C(Cc2c(C)cc(Cl)nc2)=O)CCCC2(CCC(NC(=O)CSC(C)C)C2)C1 C(CC(C(=O)O)c1ccc(F)cc1)NC(=O)NC(c1cccc(F)c1)CF C1(C(C)(C)C)CCCN(C(=O)Cc2cc(=N)[nH][nH]2)CC1.C1(C=O)C2CCCCC12 c1(OC)ccc2c(C(=O)NCCCCCCNC(C3(C)CC=CC3)=O)cnn2c1 N1(C(C(=O)OCC)=O)CC=CCC1.c1(C(=O)N)cc(C)n(-c2ccccc2Cl)n1 Cc1ccc(Br)c(NNC(=O)c2cccc(OCc3ccccc3C#N)c2)c1 C(=O)(C(C)(O)C(C)C)NC(C1CN(C(c2cc(C(C)C)nn2C)=O)C1)C C(=O)CCCCC#N.c1(C(C)C)nc(C(=O)NCCSCC2(C)CC2)cs1 C1(C(N2CC(O)(CNC(C)=O)C2)=O)Cn2c(C)nnc2CN1 C(C(C)(CCO)NC(c1oc(CNC(c2ccc(F)cc2)=O)nc1C)=O)OC c1(C(N(C2CCC(NC(c3c(C)nco3)=O)C2)C)=O)cc2ccccc2c(O)n1 c1(C(N2CCC3(CC3)C2)=O)cc([N+](=O)[O-])ccc1N.Cc1csc(C(=O)NC)c1 C(=O)(CC(O)C(Cl)(Cl)Cl)N(C1CN(C(c2coc(C(F)F)n2)=O)CC1O)C C1(C(=O)N)CCC2(CCC2)OC1.CC(C)C(O)CC(=O)NCCc1ocnc1C C1(NC(CNc2ncc(C)s2)=O)CCCN(C(=O)CCc2ccccc2)C1 C1(CC=C)(NC(=O)C(CC)CC)CCCN(C(=O)CC2C=CCCC2)C1 c1(C(N(CCNC(=O)NC)CCOCCOC)=O)ccc2n[nH]cc2n1 c1(C(N2CC(CCNC(CCCn3ncc(C)c3)=O)C2)=O)nc(C)ccc1F N#CCCCCC(=O)N1CCOCC(NC(=O)C(c2ccccc2F)(F)F)C1 S(=O)(=O)(CC(=O)N1CCCCC1)NCC.c1(CC(=O)N)cc(C2CC2)on1 Cc1ncc2c(n1)CN(C(=O)NC(c1cccc(Br)c1C)C)C2 CC1(C)Cc2nc[nH]c2C(NCC2(O)CCC(C(F)(F)F)CC2)C1 C1(CN(C(C2CN(C(C)C)C2)=O)C)CCCN(C(=O)Cn2cnnn2)C1 c1(C(C)NC(CC2(C#N)CC2)=O)cccc(Cl)c1Cl.C1(C=O)CCC2(CC2)C1.N C1(CNC(c2cnc[nH]2)=O)COCC1NC(=O)C(F)C1CCCC1 C1(C(=O)N)C2CCC1(c1cscn1)C2.C(C(=O)NCC=CC)N(C(C)C)C C#CC1CC2(CC(C(N3CCN(C(C4CCCN4C(C)=O)=O)CC3CC)=O)C2)C1 Cc1ncc(NC(C2(C)CCN2C(c2cccc(F)c2I)=O)=O)cc1Cl N1(C(c2n[nH]c(C)c2C)=O)CCC2(CCN(C(c3cnc(Br)s3)=O)C2)C1 N1(C(C(C=C)O)=O)CC(C2CCN(C(C3CCCCN3N=O)=O)CC2)C1 C#Cc1ccc(C(=O)NC(CC)C(=O)NC2CN(C3CCC3)C2)cc1 c1(C(N2C(CC(=O)OC)C3CCC2C3)=O)cnc2c(=O)[nH]ncc2c1 C(CC(=O)N1CCCC(CCNC(=O)CC2OCCC2C)CC1)(C(F)(F)F)OC C(=O)C(F)(F)C(F)(F)F.C1(CC(=O)N(C(C)C)CC)CS(=O)(=O)C1.N c1ccc2c(-c3nc(-c4nc5c(s4)CCC5)no3)coc2c1 C12(C(N3CCC(C#C)C3)=O)C(NC(c3ccon3)=O)C3CC1C2C3 c1(C(N(CCCN(C)C)CC)=O)cc(C)c(Cl)s1.C#CC1(C(=O)N)CCC1 C1(SC)CC2C(=O)N(c3cncc(F)c3)C(=O)N2C1 CC(C)(CCNC(=O)C(F)CC1CCOC1)C(=O)NC1CCCC(F)C1 Cc1c(C(=O)NCC(C)C(F)C(=O)N2CCC(CN(C)C)CC2)[nH]ccc1=O C(N=c1[nH]c(N2CC3CCC(CC3)C2)nc2c1CSC2)c1c(O)cccc1 C(=O)(C(C)C(C)O)NCC1(NC(COCCOC)=O)CCC1 CC1OCCC1(F)C(=O)N(C)CCN1CCN(C(=O)C=CCN(C)C)CC1 c1(C(=O)NCC(C(=O)NC2C=C(C)CCC2)OC)c(C)cccc1O CC(CC1CC1)N=c1nc2c(cnn2C)c(NCCOCC2CCOC2)[nH]1 CCC(CC(=O)NC1(CCO)CCCCC1)C1CC1.c12occc1C(=O)NC2 C1(C2CCC2)(C(=O)NC(C(C)NC(c2nc(C)oc2C)=O)C)CCC1 Cc1ccc(C(N2CCCCCC2CNC(C2CC2C)=O)=O)cc1Cl N1(C(C2CC(O)(CC)C2)=O)CC2CC(C1)CN(CC1(CCF)CCOCC1)C2 C1(CNC(c2c(C)sc(O)n2)=O)(CNC(=O)CCCC#N)CC2CCCC2C1 C1(CNC(CCCn2cc(CCCC(C)O)nn2)=O)CC2(CCCO2)C1 c1(C(N2CC3(C(C(=O)NC4CCNC4=O)C3)C2)=O)ccc(Br)nc1F C(C(=O)N)(C(C)C)OC.C1CN(C(c2cccc(C3(C#N)CC3)c2)=O)CCO1.C C12(C(N(CC(Cc3ccccc3)NC(CC=C)=O)C)=O)CCCC1C2(F)F C1(NC(C(C)Cn2ccnc2)=O)CCC2CC1CN2C(=O)CCN1CCOC1=O N1(C(c2c(C)cc(C)cc2C)=O)CCC2CCC(C1)N2c1nnc(C)c(C)n1 CS(=O)(=O)c1cnc(NC(N2CCC(CC(c3ccc(F)cc3)O)CC2)=O)nc1 C1(CC)CCCC(NC(=O)CONC(C2CC(F)CN2C)=O)CC1 N1(C(c2c(CC)noc2)=O)CC(CNC(C2(C)COCCO2)=O)C(O)C1 c1(C(=O)NCC2N(C(CCCOCC)=O)CC=C2)cc(COC)nn1C CN1CCN(C(=O)Cn2cnnc2O)C(CNC(C2CC2c2ccccc2)=O)C1 c1(OC)cccc(C(=O)NC2(CO)CN(C(c3cccc(Cl)c3C)=O)C2)c1Br N1(C(C(CC(=C)C)NC(C2CCC(C)O2)=O)=O)CC2C3CCC(C3)C12 c1(OC)ccc(O)c(C(=O)NCC(O)CNC(=O)CC2CCCC2C)c1 c1(C(=O)NC(CNC(CC(C=C)c2ccccc2)=O)(C)C)ccc2c[nH]nc2c1 C1(c2ccccc2)(C(=O)NCC(CC)NC(=O)COC(F)F)CC1(C)C O=C1CCCCC(C(N2CCC(F)(C(N3CCC(CCF)CC3)=O)C2)=O)C1 C(CNC(C1COCC1C(N)=O)=O)(C(=O)N(CCC(F)(F)F)C)OC C1(NC(CCCC)=O)CCCN(C(C2CC3(C2)CC(C)(C)C3)=O)CC1F C1(C(N2C(CNC(CNC=O)=O)CC2)=O)OCC2CCCC12 N1(C(CC(=C)C)=O)CC2(CCN(C(c3ccc(NC(=O)C(C)C)cc3)=O)C2)C1 Cc1nc(=NCc2cccc(C(N)=O)c2)[nH]cc1Br.C12CCC(C(=O)N)(CO1)C2.C c1(C(N2CC(C)C(O)CC2)C(=O)NC2CCOC2)cc(F)c(F)c(Cl)c1F C=C(C)C1OCCC1C(=O)NC(c1nc(C(=O)NCC2CCCC2)co1)C Cc1c(N(C(CCc2ccccn2)C(=O)NC2CCCC2)CCO)cccc1Cl c1(C(=O)NCC2CN(C(C3CCC(CC)C3)=O)C2)cncc(-n2ccnn2)c1 C(CCC(C(=O)NCC(C)(O)C1CC1)NC(c1ccc(C)nn1)=O)OC C1(NC(C(CCCCC)F)=O)CCC12CCCN(C(c1ncn(C)n1)=O)C2 c1(OC(C)C(N2CCC(C)C2)=O)ccc(Cl)cc1.C(=O)(C(F)(F)c1nccs1)N Cc1ccc(C)c(CC(N2CCOC(CCCNC(=O)C3=NOCC3)C2)=O)c1 CN1CCC(C2(C(=O)N(CC(O)CNC(=O)C=Cc3cn[nH]c3)C)CC2)CC1 c1(CC)cc(C)c(C(=O)NC(CCN(C)C)C=O)o1.c1(CC)cccc(O)n1 C(=O)(C#CC1(C)COC1)N1CCCC(N(C(=O)Cn2nc(O)ccc2=O)CC)C1 Cc1ccc(C23COC(C2)C3C(=O)NC2CC(C)OC2=O)cc1 CC1CN(C(c2ns[nH]c2=O)=O)CC(C)N1C(C1CCCOC1)=O C=CC(CCC)CC(=O)NC1CC2CC1CC2C(N1CCC1(C)CCC)=O N1(C(C(CCCC)C)=O)CCOC2CN(C(C3(c4ccccc4F)CC3)=O)CC12 c1(C(N2CCC(C)(CNC(c3cn[nH]c3)=O)C2)=O)cc(C(F)(F)F)cc(Br)c1 C1(N(CC#C)C(C2CC2C)=O)CCN(C(c2cnn(CCC)c2)=O)C1 C1(CNC(=O)CC2CCCCO2)CCN(C(=O)Cn2cc(C3CC3)nn2)C1.O CCC(CNC(=O)CC1CCOC1=O)(CC)C(=O)N1CCOC2(CC2)C1 CCC(CC)C(C)C(=O)NCCNC(=O)CC(C)CF c1(OC)cccc(OC)c1C(=O)NCC1CCCN(Cc2cnn(C)n2)C1 c1(C(=O)NCCC2N(C(C(C)SCC)=O)CCCC2)cc2c(Cl)cncc2s1 CCCC(C)CC(=O)NCCC1(C(=O)NCCNC(=O)CC)CCC1 C(=O)(CC(C(F)(F)F)P(C)(C)=O)N(C1CCN(C(CC=C)=O)C1)CC N1(C(C(Cc2ccccc2)N(C)C)=O)CCCC(C(N2CCSCC2)=O)C1 N1(C(c2c(OC)cccc2O)=O)CCN(C(=O)CC2(OC)CCC2)CC2(CC2)C1 C(CCCCCCC(=O)OCC)NC(C(=C)CC(=O)OC(C)(C)C)=O Cc1cccnc1C(F)(F)C(=O)NCC(c1ccccc1F)NC(C1CC1C)=O O(NC(=O)C1=CCN(C(C2CSCC(=O)N2)=O)C1)CC(=O)OCC C(=O)(C(C(=O)OC)C1CC1)N(CC(CNC(CCSCC)=O)(C)C)C CCCC(C)C(=O)NC1CCCC(NC(c2cc(Br)c(C)s2)=O)C1 N1(C(C2(CC)CC2(F)F)=O)C2CCC1CC(NC(=O)CCC(C)N(C)C)C2 C=C(C)CC(C)C(=O)N1CC(O)CC1CNC(=O)Cc1c(O)ncnc1O C=CCN=C(NC1CC1)N1CCN2C(=O)NCC2C1.c12ccc(cc1)S(=O)(=O)N2 N1(C(C2CC(C)C2(C)C)=O)CCOC2(C1)CN(C(=O)C=C1CCCCC1)C2 C(CC(C)C(=O)NCC1(C)CCCN1C(=O)Cc1cnccn1)OC c1(C2(C(=O)NCC(=C)CCNC(=O)Cc3ccoc3)CC2)ccccc1.O N1(C(CCC=CC)=O)CCC(C(C)(C)C)C1.C(=O)C(C)(C)C1(O)CCOC1.C c1(CNC(c2c(CC)c[nH]n2)=O)nc(C(=O)N)c(C)o1.C1CC(O)CN1C c1(C(=O)NCC(C2CCCC2)NC(C(C)=C2CCC2)=O)ccc(N)cc1C N1(C(=O)CCc2ccccn2)CCCC2(NC(C34CC(C3)C4)=O)CC2C1 c1(C(N2CCN(C(CCC)=O)C3C2C3)=O)cccc2c1OC(C)(C)C2 C1(C(=O)NCCN(C(c2nccnc2N)=O)CC)C2CCN1CC2 C1(C(=O)NCCCC(C)NC(c2ccc(CC)[nH]2)=O)CCc2nc(O)[nH]c2C1 CN1C(=O)C(F)CC1C(=O)NCCNC(=O)C(c1ncccc1F)(F)F C1(C(=O)NC(C2CCN(C(c3cncc(N(C)C)n3)=O)C2)C)COCCN1C C1(C(=O)NC2C(NC(C(F)=CC)=O)C2)CCN(CC(F)(F)F)CC1 N1(C(C=NOC)=O)CCCC2(C1)CN(C(=O)C1=CC3(CCOCC3)C1)CCO2 C1(C(=O)NCC2CC3CCC2N3C(C2CC3(C2)CC3F)=O)Cc2ccccc2O1 CCC(C)CCCCC(=O)N1CCC2(C1)CN(C(C1(C)CCCC1(F)F)=O)C2 C(C)(C(C(C)C)NC(c1ccncc1O)=O)NC(CCc1nnc(C(C)C)o1)=O Cc1nc(=O)n(C2CCN(C(=O)NCc3cccc(Cc4ncc[nH]4)c3)CC2)[nH]1 N1(C(C2N(C(CN3C(=N)NCC3)=O)CCOC2)=O)CC2CCCC2C1 CN1CCN(C(=O)CC2CCN2C(=O)C(F)C(C)(F)F)C(C2CC2)C1.CCS c1(OC)n[nH]cc1S(=O)(=O)NC1CS(=O)(=O)C1 c1(NCC2C(C)(C)COC2)ncc(S(=O)(=O)NC(CCO)c2cccs2)cc1Cl n1(CC)ccc(C(N2CC(OC)C(NC(C3CC(F)(CO)C3)=O)C2)=O)cc1=O c1(OCC)ccc(NC(=O)CC(C)(C)N(C(=O)CC2CCC(=O)C2)C)cn1 CC1(C)CC(C(=O)NCC(O)C)C1C(F)(F)F.C1(C=O)(C(F)F)CCC1 Cc1noc(C(c2ncc(-c3ccccc3)o2)NC(=O)CCc2nccn2C)n1 n1(CC(=O)N(CCC)CC)cc(F)ccc1=O.C1(CCC(=O)N)CCN(C)C1 C1(O)(CC(C)NC(C2CCCO2)=O)CCN(C(=O)COCCO)C1 c1(C(N2CC(O)(CNC(C3C(C#N)C3)=O)C2)=O)cc(Cl)c(Cl)[nH]1 C1(N(C(CCOCCCOC)=O)C)CCN(C(=O)CCCOC(C)C)CC1C N1(C(C(C(C)(C)C)NC(=O)CCN2CCCC2=O)=O)CCC2CC1C(=O)O2 c1(C(N2CCC(O)C2)=O)cc2c(cc1Cl)NC(=O)C2.[N-]=[N+]=NC1(C(=O)NC)CC1 c1(CNC(C(COCC)NC(=O)C(CC)NC(N)=O)=O)ccccn1 Cc1c(NC(C2CC(NC(c3nccc4cc[nH]c34)=O)C2)=O)ccc(Br)c1Br CC1OC(C)C(C(=O)NC2CC(CNC(c3sccc3Cl)=O)C2)C1C C(=O)(CC(O)C(C)(C)C)NCCCCCCN(C(C(F)OC)=O)C C1(CNC(Cc2cc(C(=O)OC)ncc2)=O)CC(C)CCN1C(=O)CC(C)CF N1(C(C=CCOCCOC)=O)CC2(CC)CCC1CC2.C(=O)CC.C(C)C c1(C(N2CCN(c3cc(-c4cscn4)ccn3)CC2)=O)ccc(C(F)(F)F)cn1 N1(C(c2c(CC)n(C)nc2)=O)CCCC1C1CCCCN1C(c1ccoc1Cl)=O c1(CNC(C(N2CCC(CC(=O)NC)C2)=O)=O)c(F)ccc(C)c1Br c1(OC)ccc(C(=O)N(C2CN(C(=O)C(O)CN(C)C)CC2(C)C)C)c(Cl)n1 c1(C(N2CCN(C(=O)CC3CCCOCC3)CC2CO)=O)cccc2nc[nH]c12 C1(C(=O)NC(C2CCOCC2)C)C2CCCC2CN1C(=O)CCC(C)(C)C#N C12(CO)CN(Cc3nc(-c4cccc(Cl)n4)no3)CC1(C(F)(F)F)C2 N1(C(C2(CC=C)CCC2)=O)CCN(C(c2ccoc2)=O)C(c2ccccc2)C1 C1(C(=O)NCC)CCCOC1C.C1(CCC(N2CC(COC)C2)=O)CCCCCC1 c1(C(C(=O)NC2CCOC2)N(C(C#C)C)C)sc(C(=O)OC)nc1C C12(NC(CCCC(=C)C)=O)CN(C(c3nc(Cl)sc3C)=O)CC1CS(=O)(=O)C2 c1(CC(=O)NCc2nc3c(s2)CCC3)cccc(Br)c1Cl c1(CN(CCN(C(c2ccnc(C(C)C)n2)=O)C(C)C)C)cccc(C#N)n1 C1(CNC(c2noc3c2COCC3)=O)CCC12CCN(C(C1CC1CF)=O)CC2 c1(OC)cc(C(=O)NC2CCCCC2NC(=O)C(F)(F)C(C)O)ccc1F N1(C(c2ccnc(C)n2)=O)CC(C)OC2(CCN(C(c3cc(N)ccn3)=O)C2)C1 c1(C(=O)NC(CCC)C(F)(F)F)cnc2c(Br)n[nH]c2c1 O=C(CS(=O)(=O)CCO)NCCCCC1CN(C(=O)C=Cc2cocn2)C1 C1(CC(=O)N(C(C)CO)CC)CN(C(=O)C(C2CCC2)OC)CCO1 O=C1CC(CC(=O)NC2CCCN(C(=O)COC3CC3)CC2)=NN1 CC1(C(=O)Nc2nnc(-c3cccc(C#N)c3)s2)OCCc2ccccc21 CN1CCOC(C(=O)NC(CC2CCCC2)C(=O)NCCc2cnccn2)C1 N1(C(=O)C2=CS(=O)(=O)CCC2)CCC2CCN(c3ncccc3C#N)CC2C1 CC1CCC(C(=O)NC2CC(CC(=O)NC3CCCCC3)C2)O1 C1(C(CNC(Cn2c(C)cnc2)=O)C)CCN(C(=O)CC2CCN(C)C2)CC1 C1(NC(C2N(C(C(C3CC3)OC)=O)CC3CC32)=O)CC2(CCCCO2)C1 C1(NC(C(COC)(C)OC)=O)CC2CC(C1)N(C(=O)CCCCC1CC1)C2 C12(C(=O)N)CC(CO1)N(C(=O)CC1CC(C)(C)CO1)C2.Cc1ncccc1C CC(C)(C)CC(O)CC(=O)N1CCN(C(=O)C=C2CCOCC2)C(CF)C1 CC(C)C(CN(C)C)C(=O)N1CC(N(C(=O)C(F)C2CCCC2)C)C2(CC2)C1 c1(C(=O)NC(CCN(C(CN2CC(SC)C2)=O)C)C)ccccc1N(C)C C1(C(=O)NCC(C)(C)C#N)CC=CCN1C(=O)CSCC(N)=O CCCC(C#N)C(=O)NC1CC2CC(NC(=O)C=C(C)C3CCCCC3)C1C2 C(=O)(C(O)C1=CCCCC1)NC1CC=C(C(=O)NCC(CO)C2CCC2)C1 c1(C(=O)OC)cc([N+](=O)[O-])c(C)cc1N.c1(C(N2CCC2)=O)ncc(F)cn1 CCCCCC(O)C(=O)NC1CC2CC(NC(=O)C(C)(C)OCC)CC2C1 C1(CNC(Cc2c(C)noc2C)=O)CC2(CCN(C(=O)CCC3CC3C)CC2)C1 C12(C=O)CCCC(C1)C(=O)N2.C(C)C(C)(C)C.c1(CC)ccc(C(=O)N)s1 C(c1ccc(OC)cc1)=CC(=O)N(CC(=O)NC1CC2(CNC2)C1)CC C1(NC(C2CC(CC)C2)=O)CN(C(=O)CCc2ccccc2)CC1C(F)F Cc1noc(C)c1C.C1(C#N)(CCC=O)CN(C(C)=O)C1.N1(C=O)CCC1 C=C(C)CC(C(=O)NC(Cn1cc(Cc2ccc(Cl)s2)nn1)CC(C)C)OC C1(NC(CS(CC)=O)=O)CCC2(CCCN(C(C34CC(C)(C3)OC4C)=O)C2)C1 C1(CNC(C(c2cccnc2)OC)=O)CCN(C(c2csc(Cl)c2Cl)=O)C12CC2 C(=O)(CCCC(=O)Nc1nccs1)NCC1CN(C(c2c(C)snc2)=O)CC1C CC1OCCN(C(=O)CC2CCN(C(=O)CC3NC(=O)NC3=O)CC2)C1CO c1(CC(=O)NC2C(NC(C(CC)c3ccccc3)=O)C2)nnc(C)n1C c1(C(C(=O)NC(c2ncnn2C)CC)NC(=O)COC)c(C)cccc1Br CON(CCC(=O)NC(C)CC(F)(F)F)C(=O)C1(C)CCOC1 CC12CC(C(=O)NC3CC4(C3)CC(NC(c3cscc3Br)=O)C4)(CCO1)C2 C(=O)(C(CC(F)F)NC(C1CCNC1=O)=O)NCCC1C(C)C1 Cn1nc(C(=O)NCC2(C(=O)N(CC(N)=O)C3CC3)CCC2)ccc1=O c1(-c2ccc(C)[nH]2)nc(Cc2ccc(F)cc2)nn1C1CCCSC1 N1(C(C(Br)=C(C)C)=O)CC(NC(C2(N3CCCC3)CCC2)=O)CCC1C c1(C(N2C3(CNC(C4CCCCCC4)=O)CCC3CC2)=O)cnc2ccccn12 N(C1CCCc2ccccc21)CC1C(CC)CN(C(C2CCC2)=O)CC1 C(=O)(C1=NN2CCCN=C2N1)NCC1CCCN(C(Cc2c(C)ccnc2)=O)C1 C12(CNC(C3CC(=O)NCC3)=O)CCCC1CCN2C(=O)C=C(Cl)Cl c1(C(N(CC)C)=O)ccccc1C(N)=O.CN1CCC(CC(=O)N(C)CC)C1.O O(NC(=O)C1(N(C(=O)C(C)N2CC(C)C2)C)CC1)CCC c1(CCNC(NC(c2ccccc2)C#C)=NC)c(F)cc(Br)cc1F N1(C(C=CC=CCC)=O)CCN(C(=O)Cc2cccs2)CC1c1cccc(Cl)c1 C(=O)(CC(CC(C)C)NC(=O)C(C(=O)OCC)OC)N(CCCC#C)C CCC(O)CC(=O)N1CCCC1(C)C(N1CC(O)(C(C)C)C1)=O c1(-c2nc(-c3ccsc3)nn2CCC2CC2)cccn2nncc12 S(=O)(=O)(c1cncc(Br)c1)N1CC2C(C(=O)Nc3c(Br)ccc(C)n3)(C2)C1 C=CCC(C)(CC)C(=O)NCC(CC)NC(c1ccc2c[nH]nc2n1)=O c1(C(=O)NC(CCCC)CNC(=O)C(CC)CCCC)coc2c1C(=O)NCC2 C1(C(=O)NC2CC(CNC(C(C)OC3CCOC3)=O)C2)CN(C)CCO1 Cc1cc(Br)c(N)cc1C(N1CC2CN(C(c3cc(Cl)ncc3Br)=O)C2C1)=O Cc1nc2cc(C(=O)NCC(C)N(C)C(C3CCC(=O)C3)=O)ccc2s1 c1(C(=O)NC2CC2NC(C2CC3CC3C2)=O)cccc2sccc12 N1(C(Cc2nc(C)[nH]n2)=O)CC(O)C(O)C1C.c1(C(=O)N)ccncc1N(C)C C1(NC(C(C)(C)OC)=O)CC(C)CC1O.C1(C=O)CCCN(c2nccs2)C1.N N1(C(CCCC(C)C)=O)CC2CCN(C(c3ccc(O)nn3)=O)C2C1 C1(COC)CN(C(c2cnc(Br)c(C)c2)=O)CCN1C(c1cccs1)=O C(=O)(CS(=O)(=O)C(C)(C)C)N1CCC(NC(C2CCCN(C(C)=O)C2)=O)C1 C1(NC(c2cnc(-n3cccn3)cn2)=O)CN(C(=O)CCc2nc[nH]n2)CC1O C(N=c1ccn2ccnc2[nH]1)C1(CNC(CC(CC)CC)=O)CCC1 C1(C(=O)NC(C)C(C)SC)(NC(C=CCOC)=O)CCN(C)C1 C12(NC(C(CC)C(C)C)=O)CCCN(C(c3sc(C)nc3C)=O)CC1C2 C1(CNC(CC(=C)C)=O)CN(C(c2cnc(N3CCOCC3)nc2)=O)CCO1 C12CCCN(C(c3ccc4c(c3)CC4)=O)C1C2.c1(OC)cncc(C(=O)NC)n1 C1(F)(CNC(C(CC#C)O)=O)CCN(C(C2(C)CC2C)=O)CC1 C1(COC)(NC(c2cccc(N)n2)=O)CCN(C(=O)C(c2cccn2C)=O)CC1 c1(CC)nocc1C(N1CCC1CNC(=O)CCCC1CCCO1)=O C(C)(CCC(=O)N1CC(O)(C(F)C(=O)NC2CC(C)(O)C2)C1)SC CC#CC1CCN(C(=O)C(O)CNC(C2CCCC(=O)CC2)=O)C1 c1(C(=O)NCC2(O)CCN(C(c3cc(C)n(C)c3)=O)CC2)cccc(C#N)c1F C1(NC(C(=O)N(C)C)=O)CCCCN(C(=O)CCc2ccncc2)C1 Cc1cccnc1C(=O)NC1C=CCC(C(=O)N(C)C(c2nccs2)C)C1 c1(-c2ccc(C(=O)NC3C(NC(COC)=O)C3)s2)ccccc1OC c1(-c2cccc(C(C)=O)c2)nc(OCCc2csc(C(F)(F)F)c2)ccc1F CC1CC(C(=O)NCC2(C(N3CCC3CC(C)(C)C)=O)CCC2)CC(=O)N1 C#CC1CCN(C(C2CC(C)CN2C(=O)CCc2nc[nH]n2)=O)C1 c1(OC)ccc(C2(C(N3CCCC(CC(=O)O)C3)=O)CCCC2)cc1 c1(OC)ncc(C(=O)NCCC2CCCN(C(=O)C3=CC(C)(C)C3)C2)c(C)n1 c1(C(N(C)CCNC(=O)Cn2ccc(C3CC3)n2)=O)ccc([N+](=O)[O-])o1 C=C(C)CCC(C)N=c1[nH]c(N(C)Cc2nnnn2C)nc2ccsc12 C1(NC(CC2CCN(C)C2=O)=O)CCN(C(c2ccsc2C(F)(F)F)=O)C1(C)C C1(CNC(C(C)O)=O)CN(C(c2ccc(=O)n(C)n2)=O)CC12CCOCC2 CC(C)(CNC(C1(NC(=O)C2CC2)CC1)=O)C1CCC1 C(=O)(CCC(C)C)NC(c1cn(C(C(=O)OCC)C)nn1)C CC(C)C(O)C(=O)NCC1CC1CC(=O)NC1(C)CCCC1O C1(CC(=O)N(C(=O)C)C)CCCCN1C(=O)C1CC1.n1(CCN)cccn1 CCC(C)(CC)C(=O)N1CCC(O)(Cn2cc(CC(O)C(C)C)nn2)CC1 n1(CC)nc(C)c(C(N2CCN(C(c3ccc(=O)n(C)n3)=O)CC2C)=O)c1Cl C#CCC(C(=O)OC)NC(=O)C(CC)N(C(=O)CCCOC)C c1(OC)ccc(C(C)C)c(C(=O)NC2CCC2)c1.c1(CC(=O)N)nncn1C Cc1cc(O)c(C(C)NC(=O)CCSc2nccn2C)cc1Cl c1(C(N2C(C(=O)NC3C4CCCC34)(COC)C=CC2)=O)cncc(C#N)c1 C1(C(N2CCC(Cn3cc(C(O)C4CC4)nn3)CC2)=O)Cc2cc(Br)ccc2O1 c1(C(=O)NCCC23C(CN(C(CS(N)(=O)=O)=O)C2)CC3)cc(N)c(O)c(F)c1 C=CC(C)(O)CC(=O)NCc1ccc(C(=O)NC23CC2COC3(C)C)nc1 N1(C(C(C)(C)N)=O)CCC(NC(C2(O)CCNCC2)=O)CC1 N1(C(C(=O)NCC)=O)CC2CN(C(c3cc(N)cnc3C)=O)CC2(C)C1 CC(C)C(CCC(=O)NCC(CC1CC1)CO)NC(=O)COC1CCCC1 C1(NC(CNC(=O)NC)=O)C(C)(C)CN(C(C2CC2OC)=O)CC1(C)C N1(CC)CCOCC1CC(N1CCCC1C1(NC(c2[nH]ccc2C)=O)CC1)=O C(CC(C)(C)C)NC(C(C)(C)OCC)=O.c1(C=O)cccnc1C1CC1.N c1(C(=O)NC(CNC(C2(C(=O)NC)CC2)=O)C2CC2)ccncc1.O C12(NC(CSCC)=O)COC(C1)C(NC(=O)C(C)(O)C1CC1)C2 C1(CCC)CN(C(=O)C(C)(O)C2CC2)CCN1C(=O)CC(C)N(C)C N1(C(C(C)Cc2ccccc2)=O)CCN(C(=O)CC2CCC(C)(C)C2)C(C)C1 Cc1ccc(C(N2CCC(C)(NC(=O)CC3CCC4CC34)C2)=O)c(C)n1 N1(C(c2c(CC)ccc(F)c2)=O)C2CCC1CN(C(C1(F)C3CCCC13)=O)C2 C1(N)(CNC(c2cccc(C)n2)C)CCCC(C)(C)C1 S(=O)(=O)(c1ccc(OC(F)F)cc1F)Nc1cc(C(C)(C)C)cc(C(C)(C)C)c1 N1(C(c2ccn(CCC)n2)=O)CC(CNC(c2cccnc2C)=O)CC(C)(C)C1 CC1CCC(CNC(C2CCCSC2)=O)CN1C(=O)CN1CCC(CO)CC1 c1(C(=O)NC2CC3CN(C(C(CC)O)=O)CC2C3)cc(S(N)(=O)=O)ccc1F c1(C(N2CC(CC(N3CC(=CC)C3)=O)C(C)CC2)=O)cccc(C#N)c1C N1(C(CCC(=C)Br)=O)CC2CC(C1)C2NC(=O)COc1cccc(C)c1 C(CN=c1[nH]c2ccccc2[nH]1)Cc1cn(CCCC(N2CCCOCC2)=O)nn1 N1(C(C2(CC)CCC2)=O)CCN(C)C(C(N2C3COCC2C3)=O)C1 CC1CC(C(=O)NCC2CCC(NC(=O)C(C)(C)CO)CC2)C1(C)C c1(-c2cc(NC(c3cnn(CC4CCCO4)c3)=O)ncc2)c(F)cc(F)cc1F Cc1cccc(C)c1C(O)C(=O)NC(CCNC(c1c(C)ccn1C)=O)C(C)C c1(C(=O)NCCCCCCNC(C2CCC(O)CC2)=O)cc(Cl)cc([N+](=O)[O-])c1 c1(C(C=O)N(C(COCC)CCC)C)ccc(Cl)c(F)c1.C1CC1.OCC N1(C(C2C(C)(C)C2)=O)CCCCC1C1CN(C(=O)Cn2[nH]cnc2=N)C1 c1(C(N(C)C)=O)ccc2[nH]ccc2n1.c1(C(N2CC(O)C2)=O)cc([N+](=O)[O-])n[nH]1 C1(CC(=O)N(C2CCN(C)C2)CC)CCCN(C(c2ns[nH]c2=O)=O)CC1 N1(C(c2c(OC)ccnc2OC)=O)CC(NC(=O)CC2CSCCS2)CC(F)C1 C(=O)(C(Cn1ccnn1)NC(=O)CC1CC1)NC(C)C(N)=O c1(NC(=O)N)ncc(I)cc1C(F)(F)F.c1cccc(F)n1.C1CC1C=O C(CC(C)(C)C)(C(=O)NC1(C(N2CCC3(CCSC3)C2)=O)CCCC1)OC c1(N2CC(CNCc3c(C)cc(O)cc3)OCC2)ncc2cccc(O)c2n1 S(=O)(=O)(c1ccc2c(c1)CCC2)N1CC2CCN(Cc3n(C)ccc3)C2C1 c1(CC)cc(C(=O)N)nn1C.c1(C=O)cn(C(F)F)nc1C(F)F.C(C)CC c1(C(=O)NCC(C2CCOC2)NC(CCCOCC)=O)n[nH]c2c(C)cccc12 Cc1nnc(CC2(C(=O)N)CC2)n1C.C1(F)(C=O)CC1C.C1(CC)CCCC1 C#CC1(O)CCN(C(=O)C(CC=C)NC(C23CC(CO)(C2)C3)=O)C1 c1(C(N2CCCC(CO)(OC)C2)C(=O)NCC=C)cccc(Cl)c1C c1(C(=O)NC(C2CCN(Cc3ccc(Cl)s3)C2)C)ccc(C(F)(F)F)[nH]1 C=C1CC2(C1)CC(C(=O)NCC1CCCN(C(c3cncc(O)c3)=O)C1)C2 c1(C(=O)NC(CN(C(C2C=CCC2)=O)CC)C)nn(C)c2ccc(F)cc12 C(=O)(C(CNC(C1CCSC1)=O)NC(=O)C(CN(C)C)N(C)C)OC c1(-c2nc(OC)c(C(=O)Nc3cc(Cl)ccc3CO)cc2)ncn2ccccc12 C1(NC(CC(CC)C)=O)CC2(C1)CC(C(N1CCC(C(=O)OC)CC1)=O)C2 N1(C(C(COCC)C)=O)CCCCC2(CCN(C(=O)C(=O)NCCC(N)=O)C2)C1 Cc1c(Br)cc(S(=O)(=O)N2CC(Nc3ccc(Br)cn3)C2)cc1[N+](=O)[O-] N1(C(C2N(CC)CC2)=O)CCCCC1CCC(=O)NCCOCCOC C12CCC(CC1)N2C(=O)CC1(C)CC1(Cl)Cl.Cc1cc(C(=O)N)nn1CCO N1(C(C(C)N(CC)CC)=O)CCCC(C(=O)NCC2(F)CCOC2)C1 c1(C(N(C)CCN(C)C(C2(C)CCCO2)=O)=O)ccc(-c2ccsc2)nc1 C(C(F)(F)Cn1cc(C(C)OCC)nn1)NC(CCOCC)=O c1(C=O)ccnc2cc[nH]c12.C1(OC)CC(CO)N(C(C2CN(C)C(=O)N2)=O)C1 Cc1ccc(OCC(=O)NCC(C)(O)CNC(=O)CNC=O)c(C)c1 c1(C(N2CCCCC2)C(=O)NCCOC)ncc2ccccn12.C(=O)(C(C)C)N c1(CC(N)C(=O)NCc2ccc(Br)c(Br)n2)cccc(Cl)c1F c1(CC)c(C(=O)N(CCC(C)NC(c2cn(CC(F)(F)F)cn2)=O)C)csc1C C1(CC(C)NC2CC(N3CCCCC3)C2)CCCOC1 N1(C(C(C(C)C)F)=O)CCN(C(=O)CN(C)Cc2ccc(Cl)s2)C(C)C1 N1(C(c2sc(C)c(C)c2C)=O)CC(O)(C2CCN(C(=O)CCC(C)C)CC2)C1 CCCC(C)(O)CC(=O)N1CCC(C)CC1C(N1CCC(NC(C)=O)CC1)=O C(c1ccccc1C#N)=CC(=O)NCCOCCCNC(CC(COC)C)=O C(=O)(CC(C)(C)C)NC1C(NC(C(C)OCCC#C)=O)C1 CC1C(C)N(C(=O)CCOCCN(C)C)CCN1C(c1cccc2c1CCC2)=O Cc1nc2c(o1)CCCC2CC(=O)NCC(C)NC(=O)CC1C=CS(=O)(=O)C1 C12(C(=O)NCC(CC=C)NC(=O)C(CC=C)OC)CC(C)(CCO1)C2 c1(C(=O)NCCCN(C(C#C)C)C)c(N)sc2c1CCSC2 c1(CC)nocc1C=O.C1CCN(C)C1.C(=O)CC1(C(F)(F)F)CC1.CC CCC(CC(=O)N1CC(CC(C)NC(c2ccc(CN(C)C)nc2)=O)C1)SC c1(C(N(C2(C(N(CCN(CC=C)C)C)=O)CC2)C)=O)c(NC)ncnc1Cl CCC(C)(C(=O)NC1CN(C(c2cn(C)c(=O)nc2O)=O)CC1O)C(F)F c1(C(N2C(CNC(Cc3c(C)n[nH]c3C)=O)COCC2)=O)cccc2ccoc12 CCCC(C(=O)NCc1cc(C(=O)NCC(CO)CC(C)C)cs1)C(C)C c1(C(N(CCCC(=O)NC(CC2CC2)CO)C)=O)cc(F)cnc1O CC(=O)CCCCC(=O)NCC1CC(C)(C)CN1C(c1c[nH]c2cnccc12)=O N1(C(c2c(C(=O)OC)cncc2)=O)CC2(CCN2C(=O)C(C)c2cccs2)C1 c1(-n2cc(-c3cn(C)c(=O)cc3)nn2)ccc(S(C)(=O)=O)c(Cl)c1 N1(C(C2N(C(C)=O)CC(O)C2)=O)CCN(C(C2CC2c2cc[nH]n2)=O)C(C)C1 c1(C(c2nnnn2CCCF)NCC(CC)(C)OC)nc(Cl)sc1Cl C1(CNC(c2cc(C)cc(C)n2)=O)CCCC12CCN(C(=O)CC(C)(C)C)CC2 c1(C(N(CCNC(CC(=O)OC)=O)C)=O)cnc2ccc(F)cc2c1 c1(OC)ccc(F)c(C(N2CC(CCCCNC(c3[nH]c(O)nc3C)=O)C2)=O)c1 N1(C(C2N(C(c3c(N)nccn3)=O)C3C(C2)C3)=O)CCc2ncccc2C1 CC(F)(C(=O)NCC(C1CCC1)NC(C1CC1)=O)C1CC1.C1CCC1.C N1(C(C2CC(n3cc(CC4CCC(C)C4)nn3)C2)=O)CCN(c2cnsn2)CC1 N1(C(c2cc(OC)c(O)cc2)=O)CCCC(C)(C)C1C.C(=O)C(C)C(F)(F)F.N CC1CCN(C(=O)CCNC(c2cccs2)=O)CCN1c1cc(O)ncn1 C1(C(=O)Nc2cc(CC)ncn2)CN(C(=O)CC2(CBr)CCC2)CCC1(F)F c1(C(=O)NCC2N(C(c3c(C)onc3)=O)CC(C)CC2)cnc2c(c1)COC2 c1(OC)cc(C)cc2c1OCCC2NC(=O)C(C)C c1(C(C(=O)NCC2(OC)CN(C(c3nonc3N)=O)C2)O)ccc(Cl)c(Cl)c1 C1(C(=O)NCC2N(C(C(N3CCCC(O)C3)C)=O)CCC2)CCCC(C)(C)O1 c1(CC(=O)NCC2CCN(C(c3ccn(CC(F)F)n3)=O)C2)cccc(Cl)c1F C=CCC(C)(CC)C(=O)NC1CC(C(=O)NC(C)(C)CC(=O)NC)CC1O c1(NC(C2CC2c2ccccc2C(F)(F)F)=O)cc(-n2cccn2)cc(F)c1 Cn1nc(CC(=O)N(CCNC(=O)CCc2ccnn2C)C2CC2)cc1Cl Cc1cc(CC(=O)N(CCCNC(=O)CCC)C2CC2)c(C)s1.C(N)(=O)N N(C(=NCCC1(OC)CCCC1)N(C)Cc1ccsc1)C(C=C)C N1(C(C2N(C(CCc3scc(C)c3)=O)CCSC2)=O)CCC(C)(CO)C(O)C1 C(=O)(CC(C)(C)C(C)(F)F)NC1CCCCCN(C(CC2N(C)C(=O)CC2)=O)C1 N1(C(C2N(C)C(=O)OC2)=O)CC(O)C(O)C1.c1(C=O)cn(C)nc1C1CC1.C N1(C(C(C)CC2CC2)=O)CCC2C(C(=O)NCc3cc(O)ns3)C2C1 C(=O)(C1=Cc2ccccc2C1O)NC(CCCCNC(C(CSC)(C)C)=O)C C1(C(N(C)CC2(C)CCCO2)=O)CCC(C)(C)N(C(=O)CCN2CCOCC2)C1 Cc1cc(N2CCOC(CN(C)C(C3(C)C=CCC3)=O)C2)cc(C#N)c1[N+](=O)[O-] N1(C(C(C)=C2CC2)=O)CCC(C2CN(C(C3CCc4cnc(C)n4C3)=O)C2)CC1 C12(C(=O)NC(CN(C(C=Cc3c(C)cccn3)=O)C)C)CCC(=O)N1CCS2 CC(C)(C)CC(O)CC(=O)NCC(C)(O)CNC(c1ccc(N)c(N)n1)=O CC1(C)CN(C(c2cccnc2C(F)(F)F)=O)C(Cc2ccc(N)cc2)CO1 C1(NC(C2CCc3ccnn3C2)=O)CC2CCC1N(C(=O)C(F)C1CCOC1)C2 C1(NC(CC2CC(=C)C2)=O)CC(O)CN(C(=O)C=C(C)Cl)C1 c1(C(=O)NC2C3CCN(C(C(N)=O)=O)C3CCC2)cnc2ccccc2n1 C(=O)(C(C)(CC)CCC(C)C)N(CCN(C(C(C1CCCCC1)OC)=O)C)C CP(C)(=O)c1cnc(C(N2CCCC3(C2)CN(C(C2CC4CC4C2)=O)C3)=O)cn1 c1(CC(N2CCC(CNC(C(CSC)C)=O)CC2)=O)ccc(O)c(Br)c1 Cc1oc(-c2ccccc2)nc1C(=O)NC1CC1C.c1(CC=O)nnc(O)s1 S(=O)(=O)(c1cc(C(N2CCC(O)C2)=O)co1)N(C)C.c1(C=O)cc(F)n[nH]1.C C#CC#CC(C)(C)NC(=O)CC1CCCC(NC(C2(C)CCCCC2)=O)C1 C(CN=c1[nH]cnc2cccnc12)C1CCC(NC(=O)C(C2CC2)C2CC2)C1 c1(C(N2CC(NC(c3ccccc3)=O)C(CO)CC2)=O)nccc2ncncc12 C(CC(N)=O)(C(=O)NCC1CC[Si](C)(C)C1)NC(CC1CCC(C)O1)=O c1(CCC(=O)NCCOC2CCN(c3nnc(C4CC4)s3)CC2)ccnc(Cl)c1 C(CC(C)(C)CC(=O)NCCC(C)N(C)C(C1CC12CC(F)(F)C2)=O)OC CC1(C)CN(C(C2CC2C(C)(C)O)=O)CC(CNC(=O)CC2=CCCC2)O1 CCN=C(NCCc1ccccc1C(N1CCCC1)=O)N1CCC(COC)C1 C1(NC(c2ccc(OC)o2)=O)CC(CNC(C2CC2C(C)C)=O)CC1O c1(NCCN(CCCO)C)ccc(Cl)c2c1CCNC2 c1(CCN(C(=O)C=CBr)CCCN(C)C)ccccc1.C(=O)CCN1CCCC1 c1(-n2c(CCCNC(C)=O)nc(-c3ccc(Cl)cc3)n2)ccc(Cl)cc1Cl N(C1CCC(NC(=O)CC(F)(F)Cl)c2ccccc21)C(C=C(CCC)C)=O c1(CC(C)C)ccc(C(=O)N(CC(O)CN(C)C(c2ccncc2)=O)C)cn1 C(=O)(CC(C)CC(F)(F)F)N(C1CCN(Cc2ccccc2Cl)C1)CCC C(=O)(C#CC1CCCCC1)N(C)CC1(CNC(=O)C2=C(C#N)CCC2)CC1 C12(CC(=O)NC3CC(C)N(C(C4CC=CC4)=O)C3)CCC(CC1)OC2 C(=O)(CC(C(F)F)C(C)(C)C)NCC(C)NC(c1cc2n(c1)CCC2)=O C12(C(=O)NC(COCCCC)C)CCCC1CN(C(c1ccc(C)c(C)n1)=O)C2 Cc1cnc(N2CCC(NC(c3ccccc3F)=O)C2)nc1O C1(NC(CC2C(C)CCC2)=O)CC2CCC1CC2NC(=O)Cn1cnc(C#N)n1 c1(C(=O)NCCCCCN(C)C(c2scnc2Cl)=O)cnc2n1CCS2 CCCCCCCCC(=O)NCC(CCC)C(O)C(=O)NC(c1nncn1C)C C1(C2(O)CCOC2)(C(=O)OCCOC(CCCCCCC)=O)CCC1 N1(C(C(CC)NC(c2ccco2)=O)=O)CCCC1C.n1(CC=O)ncn(C)c1=O.N N1(C(C(CC)SC)=O)CCC(CNC(C2CCC(=O)N(C)C2)=O)C(O)C1 C1(C(=O)NCCC2CCN(C(c3cccc(NC)n3)=O)C2)CCC(F)(F)CC1 C1(C(=O)NC2(C(=O)OC)CCC23CCC3)COCCC1C1CC1 C(=O)(CCCCC(C)(C)C)NC1CC(C)N(C(C2CC(N(C)C)C2)=O)CC1 C1(C2CCN(C(=O)C3=CCC3)C2)(NC(=O)CCc2n[nH]c3ccccc23)CC1 c1(C(=O)OC)cccc(CC(=O)N(c2ncccn2)C2CNC2)c1 O=C(CCC1=CCc2ccccc21)NCC1(C)CCC1.C1(C2CC2)(C=O)CC1.N N1(C(CC2ON=C(C)C2)=O)CCN(C(=O)CSc2cn[nH]c2)C2COCC12 C12(NC(C(F)=CCC)=O)CC1CN(C(=O)CCOCCCOC)C2 Cc1cccc(C(CNC(C2(c3ccsc3)CC2)=O)NC(=O)C=CS(C)=O)c1 O=C1CCC(C(=O)NC2CC3(C2)CC3)=NN1.c1(C=O)ccccc1OC(F)F.N Cc1cc(C(=O)NC2(c3ccc(Cl)cc3)CCOCC2)c(F)cc1F N1(C(c2cncc(C(=O)OCC)c2)=O)CCN(C(=O)C(C(C)C)SC)C(C)C1 c1(N2CCC(NC(CCC=C)=O)C(C)C2)ncnc2cc(Br)sc12 c1(-c2cc(C(C)C)ncc2F)c(F)ccc(F)c1F c1(C(N2CCN(C(c3cc(Cl)c(Cl)s3)=O)C3(CC3)C2)=O)cc(F)cc(Br)c1F c1(C(N2CC3(N(C(c4cnc(CC)s4)=O)CC3)C2)=O)cc(C)cc([N+](=O)[O-])c1 N1(C(C2(OC)CCCOC2)=O)CC2(CC(NC(=O)C3=C(C)CC3)C2)C1 C1(COC)CN(C(C2C3COCC23)=O)CCN1C(c1ccc(O)c(I)c1)=O N1(C(C(CCSC)O)=O)CCC2(CCCC2NC(c2ccnnc2O)=O)CC1 C1(SCC(=O)OC2CC(CCS(C)(=O)=O)C2)CCCNC1=O C1(C(N(CCOCCNC(c2cc(C)sc2)=O)C)=O)CN(C)CCN(C)C1 C1(C(=O)NCC(CNC(c2cc(C(C)C)no2)=O)C)CCOC(C)C1 C1(=CC(N2CC(CC)C2)=O)CN2CCC1CC2.CC1(C=O)CC1C(F)(F)F Cc1ccc(Cl)c(CSCC(=O)Nc2cc(Br)ccc2F)c1 C(=O)(C1=C(Cl)CCOC1)NC12CC(CNC(CC(CC)SC)=O)(OC1)C2 CN1CCn2nc(C(=O)N(CCCCNC(=O)CC(=O)OC(C)(C)C)C)cc2C1 C1(C(N2CC(C(=O)NCCS(N)(=O)=O)(CC)C2)=O)CCCCC1(C)C c1(C(=O)NC2CN(C(CCCCC=C)=O)C(C)(CC)C2)cncc2cnccc12 C1(C(=O)NCC(C)CNC(=O)C(c2ccc(O)cc2)(C)C)CCSC(C)C1 c1(C(N2C3C(CNC(=O)C(c4ccccc4)F)C(C3)C2)=O)c[nH]c2ccncc12 C1(CNC(c2cc(C)on2)=O)CCCN(C(=O)C(C)NC2CCCC2)C1 C1(C(=O)OC)C2C=CC(CC2)C1C(N1CCCNCC1)=O c1(C(=O)OC)cc(S(N)(=O)=O)ccc1NC(c1cn2ccc(Cl)cc2n1)=O C(=O)(C1CCc2c[nH]nc21)N1CC(C(N2CC=CCC2)=O)CC(C)(C)C1 N1(C(=O)N)CC(C=O)OC2(CCC2)C1.C(=O)(Cc1ccsc1)OC(C)(C)C CCC(CC(=O)NC(C1CCCC1)CO)N(C(=O)CSc1n[nH]c(C)n1)C CCC(C(c1nnnn1C)OC(=O)NC)NC(=O)CCCNC(C)=O CC1CN(C(=O)CN2CCC(C)C2)CCN1C(=O)Cn1cccnc1=O C1(=O)CC(O)CO1.c1(COC(C(=O)NCC=C)C)ccccc1 c1(CN2C(C(=O)NCCC(N)=O)CSCC2)cccc2[nH]ccc12 N1(C(c2cn(CC)nn2)=O)CCC(C=CC(=O)N)CC1.C1CC(=C2CC2)C1 C1(CC)CCCCCN1C.c1(C=O)c(C)nn(C2CCS(=O)(=O)C2)c1Cl.C1CC1 N1(C(C2CCC(CC)O2)=O)CC(F)CC1CNC(=O)CCn1cnnn1 N1(C(c2cn(CC)nc2)=O)CCC2(CCN(C(C3CC3c3ccc(Cl)s3)=O)C2)C1 c1(C(=O)Nc2cc(C)cc(F)c2)c[nH]c2ncc(-c3nccs3)cc12 Cc1cc(NC(C2CCN(C(=O)CCCCCl)CC2O)=O)nc(C)c1 C1COC(C)(C)CN1C(C1CCS(=O)(=O)N1C)=O.C(C(=O)NC)OC(C)C N=c1nc(C(N2CCCCC2C(=O)NCCCN2CCCCC2)=O)cc[nH]1 C(=O)(NNc1cccc(COc2ccc(F)cc2)n1)NCC(CC=C)C c1(C=O)cc(C)nn1C.C(=O)(CC1CCCC1)NCCCOC(=O)NC.N CCC1(CC)CN(C(N2CCC(C)C(C)C2)=O)c2ccccc21 c1(C(C(=O)N2CC(CCCCOC)C2)CO)ccc(F)cc1 C(=O)(C(C)(C)CS(N)(=O)=O)NC(CCC)CC(=O)NCC.C(C)(C)C.C=O N1(C(CN2CCN(C(C)=O)CC2)=O)CC2(CCC2)CCC1C.[nH]1cc(Br)cn1 CC1CN2CCN1CC2C(=O)NC1CCC(NC(C2(F)CC=CCC2)=O)CC1 c1(CNC2C(C(=O)NCC(C)(C)O)C2)cc(F)cc(Cl)c1 Cc1nccnc1C(C)NC(C1(NC(=O)CCN(C)CCO)CC1(C)C)=O N1(C(CCC(C)(C)C#N)=O)CCC(C2(C(N3CC4CC3C4)=O)CCOCC2)CC1 N1(c2c(C#N)ccnn2)CCC2(COC(CNC(C3CC4(CCC4)C3)=O)C2)C1 Cc1nn(C)nc1C(=O)N(C1CCN(C(=O)CC2(CO)CC2)C1)C C(=O)(CCCCCCCN)N(c1ccc(Cl)nc1)CCOC CC1CN(C(=O)COCC2CCOCC2)CCN1C(C1CC2(C1)CC2F)=O CC(O)CCN=c1ccnc(NCc2ccccc2[N+](=O)[O-])[nH]1 C12CCC(CC1)C2.Cc1cnc(C=CC(=O)N)[nH]1.C(=O)C=CCN(C)C N1(CC)CC2CCC(C1)C2NS(=O)(=O)CC1CC=CC1 N1(C(=O)Cc2ccc(O)cn2)CCN(C(=O)CC2CCCCCO2)C(CCO)C1 C1(C2CCN(CC#C)C2)CCCCN1C(=O)C(C)OCOC CCC(CC)C(C)C(=O)N1CCCC(CC(=O)NC(C)C)CC1 c1(CC(=O)NC(CC=C)CNC(=O)CCOCCC)cccc(OC)c1F c1(C(=O)NC2CCCN(C(C(F)=C(C)C)=O)C2C)ccc(C)c(Cl)c1N CN1CCOC(C(=O)NCC(CO)NC(=O)C(C2(O)CCOCC2)(F)F)C1 C(=O)(CC(C)(C)C(F)F)NC1CN(C(c2c(C)cc(F)cn2)=O)C(C)CC1 N1(C(C(CC)(C)O)=O)C2CCCC1CN(C(=O)Cc1ccc(OC)nc1)C2 N1(C(COCCOC)=O)CCCCCCC1C(=O)N(C(C)C)CC1CCC1 N1(C(=O)Nc2ccc(C)cc2F)CC2CCN(C(c3ccncc3)=O)C2C1 c1(C(=O)NCCC2N(C(c3cnn(C)n3)=O)CCOC2)cc2c(s1)CCOC2 N1(CCc2ccc(C)cc2C)CCC2(CC1)CC2F C1(O)(C(N2CC(C(C)NC(C(C=CC)O)=O)OCC2)=O)CCCC(C)CC1 c1(OC)ccc2c(C(=O)N)n[nH]c2c1.C12CC(C1)C2.C(=O)CN(C)C1CC1 N1(C(C=CC(C)(C)SC)=O)CCC(C(CO)NC(C2CCC(C)O2)=O)CC1 c1(OCC(C(=O)NCc2ccccc2)c2nn[nH]n2)ccn2ccnc2c1 C(=O)(CCCCCC(C)(C)C)NCC1(NC(C2C(C)CC(=O)NC2)=O)CCCC1 c1(C(=O)NC(C)CNC(=O)CC2COCCOC2)ccc(C2CC2)cc1Cl C(CCCC)(CN=c1[nH]c2cc(F)ccc2o1)NC(CC1(C=C)CCOCC1)=O C=C=C(C)CC(=O)N(C(C)CCNC(c1cc(C)n(-c2ccccc2Cl)n1)=O)C N1(C(C(C)C(C)(F)F)=O)CCC2(CCCCN(C(=O)CCc3cccnc3)C2)C1 N1(C(C2(CC3CCOC3)CC2)=O)CC2CCC(C1)N2CCc1ccc(F)cc1 C(=O)(C1=CCCOCC1)N1CCC(=C)CC1C(=O)NCCc1nnc(O)o1 N1(C(c2cc(F)nc(F)c2F)C(=O)NCCCSC)CCC(C)c2ccccc21 C(=O)(C1=NOC(C2(O)COC2)C1)NCC1C(C)(C)C(Nc2ncccc2N)C1 C(=O)(C1=C(C)CCOC1)N1CC(CNC(C(CCCC)F)=O)C(CC)C1 C1(C(=O)NCCCN(C(=O)Cc2cnn(C)c2)CCC)CC2CCC1NC2=O C(N=C(NC1CN(C(C)=O)C1)N1CCC(n2cc(C)cn2)C1)C1C(C=O)C1.CO CC1=C(C(=O)N2CCCC2CNC(=O)C(C)c2cccs2)SCCO1 Cc1cc(O)cc(=O)n1CCC(=O)NC(C)C1CC1.C(=O)C(C)SC(F)(F)F N1(C(c2cc(C)n(C(C)(C)C)n2)=O)CC2(C1)CN(C(C1(F)CCOC1)=O)C2 C(=O)(CCCN=C(NCC(c1cccc(Br)c1)O)N1CCC(C)C1)NC c12sc3c(c1C(=O)N2CC(=O)N(C)C)CCC3.Cc1cnc(C(=O)O)cn1 Cc1scc(C(=O)NC2CCCC2NC(=O)CSCC2CCCO2)c1N N1(C(C2CCC(=C)CC2)=O)CC(CN=c2nc(OC)[nH]c(OC)n2)C2(CCC2)C1 C(C(O)(C(=O)N1CC(CCCC)C1)C(F)(F)F)N(C)C.C1(C(=O)N)CNC(=O)C1 CC1(C)COCC(C(=O)NC2CCN(C(c3cc(C(F)F)cs3)=O)C2)O1 C(CCNC(c1n[nH]c2c1CCC2)=O)(C(=O)NOCCC(F)F)OC C1(CNC(CCC=C)=O)CN(C(C23CCC(C(F)F)(CC2)C3)=O)CCC12CCC2 c1(C(N2CCN(CC(C)(C)NC(C=CSC)=O)CC2)=O)cc2cccnn2n1 c1(OCC(=O)N(CC(C)NC(=O)C=Cc2cncn2C)C)cccc(Br)c1 c1(C(=O)NCCC2(NC(C(CC)OCC)=O)CCCC2)cccc(Br)c1F C(C)(C(C)(C)C)=CC=O.c1(CC)ccccc1.C(=O)C=CC=O.CC N1(C(C(C)NC2CCCCC2)=O)CCC(C)(NC(=O)CCSC(F)(F)F)CC1 CN1CCC(CN)C1=O.n12nc(-c3ccccc3)cc1C(=O)N1CCC2C1 c1(C(N2CC(O)C2)=O)ccc(F)cc1C#N.c1(OC)cccc(F)c1C(=O)N.C c1(N2CCC(NC(c3c(C)noc3)=O)(CF)C2)nc(Cl)nc2cnn(C)c12 CCC(C)(C)C(=O)N1CCC(Cc2cn(Cc3ccc(Cl)s3)nn2)C1 CC(=O)CCC(=O)NC(C1CC1C(=O)N(C1CC1)C)C.C1CCN(C)CC1 c1(CC)cc(C(N2CC3C(C(=O)NC(C)CS(N)(=O)=O)C3C2)=O)n(C)n1 C1(C)(C(N2CCCC2)=O)CC2(CC2)C1.C(C(C(=O)N)NC(C)=O)OC.C N1(C(C2(C#C)CCCC2)=O)C2CCC1CC(N(C)C(c1ccnc(C)c1O)=O)C2 C1(C(=O)NC(C)CCNC(=O)CC(C)(C)O)C2CCN(CC2)S1(=O)=O c1(OCC(=O)NC(CC)(C)C)cccc(COC(=O)C(C)O)c1 N1(C(c2cc(CCCCC)[nH]n2)=O)CCOC2CCN(C(=O)C(CC)CC)CC12 Cc1ncnc(C(N2CCCC(NC(C3(C4CCCCO4)CC3)=O)C2)=O)c1C c1(C(=O)OC)cncc(NC(C2CC(F)CN2C(C2CNC(=O)C2)=O)=O)c1 CCC(C)C(C(=O)O)NC(=O)CN(C)C(c1nc2c(s1)CCC2)C C(=O)(CC(CC)N(C)C(c1ccc(C)nc1)=O)NCC(CCC)OC C(=O)CC(C)(C)C(C)(F)F.C(=O)(C(C)C)NCC(C)C.C(=O)C(F)(F)F C1(F)(CNC(C2C(C)SCCC2)=O)CCCN(C(=O)Cc2ccsn2)CC1 c1(CC(=O)N(CC)C2CC2)ccc2nc[nH]c2c1.CC(C(C)(C)C)=CC=O.N CS(=O)(=O)c1ccc(C(N2C3CN(C(c4cc(C(F)F)no4)=O)CC23)=O)cc1 N1(C(CCc2nnc(C)o2)=O)CCC2(NC(=O)C(C)(C)CC3CC3)CCCC12 C(=O)(C1=CCCCO1)N(CC(C)O)CCNC(=O)C(C)(C)c1cccs1 c1(C(=O)NC2CCC(N(C(=O)CCC3CC3)C)C2)ccc(-c2ccsc2)nc1 c1(C(=O)NC2(CF)CCN(C(=O)CC3CCOC3)C2)cc(Cl)c(F)c(Cl)c1 O=C1COc2ccc(NC(c3cccc(-c4nn[nH]n4)n3)=O)cc2N1 N1(C(C2(F)CC(C=O)C2)=O)CCN(C(=O)CCC(C)CC)C(C(C)C)C1.CC.O c1(C(=O)NCCC(CC)(CC)NC(=O)CCF)cccn2cc(C(F)(F)F)nc12 N1(C(CC(CCC)C)=O)CC(NC(=O)CSC)C(S(C)(=O)=O)C1.c1ncc[nH]1 CC1=C(C(=O)N2CCC(NC(=O)C(C)(C)Cc3ccccc3)C(O)C2)SCCO1 c1(C(N2CCC(C)(CCNC(C(C)n3cccn3)=O)C2)=O)cc2nnn(C)c2s1 c1(C(=O)N)ccc2c(c1)OCCO2.c1(C(N(C)CC2CC2)=O)nnc(O)cc1O C1(NC(c2cc(CC)[nH]n2)=O)C2CN(C(=O)C(F)(Cl)c3ccccc3)CC12 N1(C(C(C)O)=O)C2CCC1CC(O)(CNC(c1sc3nccnc3c1N)=O)C2 CCCC(CC(C)C)C(=O)NCCC(C)(C)CNC(=O)CC(C)C(F)(F)F C1(CNC(=O)CCc2cnc[nH]2)CC2CCCC(C1)N2C(c1cnsn1)=O C(C)(CCCCNC(=O)C(c1ccccc1)SC)NC(c1c(OC)ccs1)=O N1(C(CC(CC)(F)F)=O)CC2CCC(N(C)C(c3ccc(C(F)F)o3)=O)C2C1 c1(CC(=O)OCc2c(C)cccc2)nsc2ccccc12 C1(NC(c2c(CNC(CC3(C)OCCO3)=O)ccs2)=O)CCCCC1(F)F C(=O)(N=c1[nH]oc2cccnc12)NCCc1c(Br)ccc(C)n1 C(=O)(C1=CC2CCCC12)NCC(C)NC(c1cnn(C(C)C)c1C1CC1)=O C(=O)(C(CC(C)C)C(C)C)NCC(C)=CC(=O)NCCCCC(C)(C)C Cc1nc(C)c(C(=O)NCC2COCC2NC(=O)C(C)O)[nH]1 N1(C(CC(CC)SC)=O)C2CCC1CC(CC(C)NC(=O)Cc1ccccn1)C2 N1(C(N)=O)CCOCC1CC(=O)NCC(N1CCCC1)C CCCC(C)(O)CC(=O)NCCCCNC(=O)C(c1ccc(Cl)cc1)C C1(CNC(C2C=CCN(C(=O)C(Cl)Cl)C2)=O)C2CCCCCC12 c1(CCC)nc(C)c(C(N2CC3C(CNC(C4(O)CCOC4)=O)C3C2)=O)s1 CC1C(C(=O)NCC2(C)CN(C(c3cnc(C(C)O)s3)=O)CCO2)=NOC1C C1(NC(C=C(C)CNC(c2cc(O)nc(C)n2)=O)=O)(CO)CC2CCC1C2 C1(C(=O)N)CN(C(c2ccc(O)nc2)=O)CCC1(C)C.C(=O)(C(C)C)OCC C1(CCC(=O)NC2CC2NC(=O)CCC2CCOCC2)CCCOC1 c1(C(=O)N)cc(Cl)cnc1.C1(NC(CN(C2CC2)CC)=O)CCCC1C CCC(C)(CC)C(=O)N1CC(O)(C(C)(C)CNC(c2cc(Cl)cnc2O)=O)C1 N1(C(COC(C)C)=O)CCN(C(C2CC3(CCC3)CO2)=O)CC12CC2 C1(C=O)CNC(=O)C(C)(C)C1.C1(CN(CC(C)C)C)CC2(COC(=O)N2)C1 CC1(NC(C2OCCC2NC(C2CCCS2)=O)=O)CCOCC1 c1(C(N)=O)cc(NCc2ncc(-c3cccc(C(=O)O)c3)[nH]2)cc(Br)c1 CS(C)(=O)=NCC(=O)NCc1cc(C2CCN(C(c3cc(O)cs3)=O)CC2)no1 c1(C(=O)NC2C(CNC(C(F)=CC)=O)C2)cc(C)c(Cl)cc1Cl CN=C(NCC1(O)CCC1CO)N1CCN(c2ccccn2)CC1 c1(CC)nc(C)cc(=NCC(C)CNC23CC(CN2C2CC2)C3)[nH]1 C1(NC(c2ccc(CC)cn2)=O)CN(C(=O)C(c2cccn2C)=O)C2(CCC2)C1 Cc1cc(NC(C2CCCN(C(C3CCC3C#N)=O)C2)=O)ccc1Cl C1(S(C)(=O)=O)(C=O)CCCC1.C1(C(F)(F)F)(OC)CC(C=O)C1.CCCC CP(C)(=O)C(O)C(=O)NCCOc1cnc(-c2cncnc2)nc1 C(C(C(C)C)NC(=O)C(O)C1CC1)NC(COCC#C)=O CC(C)CCC.C(=O)(C(C)(C)C=O)N.C(C1CCOC1)=CC=O.C(C)(C)C C(N=c1[nH]nc(C(N)=O)s1)C1C(NC(C(Cc2ccc(OC)cc2)C)=O)CCC1 c1(C(=O)NC(CSCC=C)C(=O)OC)cccc2c1CCCC2N C(C(C)(C)C(=O)NC1C2CCN(C(=O)C=Cc3ccco3)C12)OCC C=C1CC(C)(C(=O)NCCOCC(=O)Nc2conc2C)C1 N(C)(C1CCCc2ccccc21)CC(N1CCC(OC)CC1)=O N1(C(C2(C)CCC2)=O)CCC2(CC1)CC2NC(c1[nH]cc2c1CCCC2)=O c1(OC)ccc2[nH]c(C(N3CCC(C(C)(C)NC(c4cncs4)=O)C3)=O)cc2n1 N1(C(C2N(C(=O)NCc3ncc(C)s3)CCC2)=O)CCc2ccsc2C1 C(=O)(NNC(=O)C1(OC)CCOC1)NCC(C#C)CC1CCCCC1 c1(NC2CC(NC(CC3C(C)(C)CCO3)=O)C23CCC3)ccc([N+](=O)[O-])cc1Br N1(C(C2C(c3ccc(-c4c(C)cc(O)cc4)cc3)C2)=O)CCn2nccc2C1 C1(O)(CC(N2CCC(OCC#C)CC2)=O)CCN(Cc2cccc(O)c2O)CC1 CCC(C)(C#N)C(=O)NCC1(NC(=O)C)CCOCC1.C1(C=O)CCCCC1 Cc1cc(=O)n(C)cc1C(N1CCCN(C(=O)CCC2CCCN(C)C2)CC1)=O c1(OCC=C)ccccc1C(=O)NC1CCN(C(=O)COCCF)C1 c1(C(=O)OC)c(Cl)ccc(CN2CCCC(C3(C)OCCO3)C2)c1Cl C1(NC(C2CCCN(C(C)=O)C2)=O)CCCN(C(C2CC(=O)NC2(C)C)=O)C1C c1ccccc1O.n1(C)ccnn1.C1(C(=O)OC)CC1C(=O)NCC1CC1 c1(C(=O)NCC(C)OC)c(F)ccc2ccncc12.C(=O)(C(C)C(F)(F)F)N Cc1cc(CN2CCCC(NC(=O)Nc3ccc(Br)c(C)c3)CC2)cc(C)c1 C1(NC(c2cncc(OC(C)C)c2)=O)CCN(C(c2cnc(Cl)n2C)=O)CC1F C1(C(=O)Nc2c(C)ncc(C)n2)Cc2nccnc2CN1C(c1ccc(Br)s1)=O C1(C(=O)NCC(CC(C)C)NC(CCC=C)=O)COc2c(OC)cccc2C1 c1(CC(=O)NCC2CN(C(=O)CC3(C)CC3)C3CC23)cnc2ccccc2c1 CN1CC23CCCC2(C1)CN(N(C)C1CCCC1NC(=O)OC(C)(C)C)C3 C(=O)(CCC(C)CN(C)C)N(CCCCCNC(C1N(CC)CCC1)=O)CC c1(C(N2CCC(CCNC(=O)CC3CC34CC4)C2)=O)c[nH]c2ncnc(O)c12 N1(C(C(C(C)C)OC)=O)CC=C(CC(=O)NCCc2cnn[nH]2)CC1 CC1(C)CCCCC1C(N1CCC(CCNC(c2nccs2)=O)CC1)=O Cc1cc(C)c(NC(=O)C(N2C3CCC2CC(O)C3)C2CC3C=CC2C3)c(C)c1 c1(C(=O)NC2CN(C(C3CCC(=O)OCC3)=O)C2)coc2c1CS(=O)(=O)C2 C1(O)(CN(C)C(c2sccc2C)=O)CCCCC1.c1(C(=O)N)cc(O)ncn1 C1(NC(=O)C(O)C(F)(F)F)(C)CCC(F)(F)CC1.C1CCCOC1.C(=O)(C)N c1(OCC(N2CC(CC(C)NC(=O)C3=CCCCC3)C2)=O)ccc(Cl)c(F)c1 C12(CNC(c3c(C)nsc3)=O)CCCC1CN(C(c1n[nH]c3cccnc13)=O)C2 N1(C(CC2CN(C)C2)=O)CCC(C2CC(NC(=O)CSCc3cccs3)C2)C1 c1(C(=O)NC2C(C)CN(C(=O)C(=Cc3c[nH]cn3)F)C2)ccc([N+](=O)[O-])nc1 N1(C(CN(C)C2CC2)=O)CC2CC2(CNC(=O)CCCCC2CC2)C1 C(=O)C(CCS(C)=O)N(C)C.c1(CC)ccc(F)cc1.C1(C(=O)N)(CC)CC1 N1(C(c2cc(C(CC)C)no2)=O)CC2CCN(C(c3cccn(C)c3=O)=O)CC12 N1(C(CN(C2CCC2)C(c2c(C)ncnc2)=O)=O)CCC12CCCSC2 Cc1cccc(Oc2nc(-c3nc(CO)cs3)nn2-c2ccc(C3CC3)cc2)c1 N1(C(c2cnn(C)n2)=O)CCOC(Cc2cn(CCCSC)nn2)C1 C(=O)(CCCCC(F)(F)F)N(C)CC1(O)CCCN(C(c2csnc2Cl)=O)C1 S(=O)(=O)(c1c[nH]c(C(=O)N)c1)N(C)C.C12CCCN(C(C3CCC3)=O)C1C2.C C(=O)(C(CC(F)(F)F)c1ccccc1)NC(CNC(C(C)(C)O)=O)CO N1(C(c2cnc(CC(C)C)[nH]2)=O)CC2=C(C1)CN(C(C1CC3C=CC1C3)=O)C2 C(CNC(C1C(C)C1(F)F)=O)(CC(C)C)NC(c1n(CC)ccn1)=O C(=O)(C1=Cc2ccc(Cl)cc2OC1)NCCC1N(C(C(C)C2CC2)=O)CCCC1 Cc1cc(F)ccc1CC(=O)N(CCC(C)NC(=O)CCSC1CCCC1)C c1(C(=O)NC(CCCC)CNC(=O)C(C)S(C)(=O)=O)cc(C)c(F)cc1F CC(C)(C(=O)N1CCC(CC(=O)NCC2CC(F)(F)C2)C1)N1CCCC1 C(CCC1CC1C)(C(=O)NCCCSC)N(CCS(CC)=O)C N1(C(C(=O)NC(c2ccc(F)c(Br)c2)CC)=O)CCOc2ccc(C)cc2C1 CN1CC(C)(C)CC1C(N1CC(CC)C1)=O.c1(C(=O)N)ncoc1C1CCCO1 Cc1c(C(N2CCC(O)(CNC(C3CCCC(C)C3)=O)C2)=O)cnn1CCC#N c1(CC)cc(C)c(C(N2CCC(N(C(=O)CCSc3nccn3C)C)C2)=O)o1 C1(COC(C)=O)CN(C(=O)CCN(C(=O)C(C)=C2CC2)C)C1 N1(C(C(c2cc(C)cc(F)c2)C)=O)CCCC(C)(C)C1CNC(=O)C(C)C Cc1ccc(NC(C2CC(O)CN2C(=O)C(C)(C)CO)=O)c(C)n1 C1(NC(C=CC)=O)CCCCN(CCSC)C1 N1(C(CCCCNC(=O)OC)=O)CC=C(CNC(=O)C(F)C(C)(C)O)CC1 Cc1cc(C(N2CCC(O)(C(C)NC(=O)CCc3cnc[nH]3)C2)=O)cc(C)c1C c1(C(=O)NC(C)CCN(C)Cc2nccs2)cnc2n1CCOC2 c1(OC)ncc(C(=O)NC2(C)CC(NC(=O)CC3CC(SC)C3)C2)cc1Cl Cc1ccc(N2CCCC2NC(N2CCC(Oc3ccccc3Br)C2)=O)cc1 CCCCCC(O)C(=O)N1CC2(CCN(C(=O)CC3CCC3(C)C)C2)C1 C1(C=O)CC2CCCC(C1)C2.C(O)(C(F)(F)F)C1(C(N(C)CC)=O)CCC1.N c1(C(N2CCC(NC(CC(COC)(C)C)=O)C(C)C2)=O)nccc2ncccc12 N1(C(CC2OCCN(Cc3c(C)n(C)nc3)C2)=O)CC(C)OCC1C N1(C(C2C(COC)C2)=O)CC2OCCC2C1.c1(C=O)ccccc1OC(F)F.N C(=O)(CC(O)C(C)CC)N1CC(C(=O)NCC=CC)(CC)C1 c1(C(N2CCN(Cc3nn(CC)nc3C)CC2C)=O)cn(C)c2ccccc12 CC1CN(C(=O)C=CCN(C)C(C2CC(C)(C)C2)=O)c2ccccc21 N1(C(COCCC=C)=O)CCN(C2CCN(C(=O)CSc3ccccc3)C2)CC1 C(=O)(CS(=O)(=O)C1CC1)N(CC(C)(C)NC(C1CC(C)CC(C)C1)=O)C c1(C(c2n(CCC)nnn2)NC(C)C(C2CC2)OCC)ccc(F)c(I)c1 Cc1cccc(Cl)c1C(N1CC2(CCC2NC(=O)C(C)C(F)(F)F)C1)=O N1(C(CN(C(C)=O)C)=O)CC2(CCN2C(=O)C(C(C)C)N2CCCCC2)C1 C1(NC(C2C(C)(C)C2(C)C)=O)CC(C2CCN(C(c3occc3Br)=O)C2)C1 c1(C(=O)NC(C2CCCN2C(=O)CC(Cl)Cl)C)ccnc(-c2ccco2)c1 c1(NC2C3CN(C(C(=C(C)C4CC4)F)=O)CC32)nc2c(C)c(C)ccc2s1 C1CCN(C(=O)C=Cc2cnn(C)c2)CC1C(C)C.CC(C(C)C)=CC(=O)N O=C(CCOCC1CC1)NC1(C2CCCO2)CC1.C12CC(C1)NC2=O C1(C(N(CCN2CCCC2)CC)=O)CSCCN1C(c1cncc(O)c1)=O c1(C=O)n[nH]c2nccc(Cl)c12.N1(C(C=C(C)C2CC2)=O)CCC(C)(C)C1C.N N1(C(C2(NC(c3cc(OC)nn3C)=O)CC(F)C2)=O)CC2CCC2(C)C1 CC(C)CC(C)(O)C(=O)N1CC(C2CN(C(c3cccc(F)c3C(F)F)=O)C2)C1 c1(C(=O)NCC(C)NC(C2CC3OC(=O)OC3C2)=O)ccc2nc(S)[nH]c2c1 Brc1ccc2cc(OC3CCCN(CCCNCc4ccccc4)C3)ccc2c1 c1(NC2CC(C)n3c2ncn3)nc(NCC2=CCCC2)c2cnn(C)c2n1 c1(C(=O)NCCC(C)CCNC(=O)C=Cc2ccco2)c2c(nn1C)CCC2 C1(C(=O)NCCCCOCC)CN(C(=O)CCC2OCCO2)CC1F C(CCC(=O)NCC1CC(OC)C1)(C(C)C)NC(C(C(C)OC)N(C)C)=O C12(NC(C(CC(C)C)n3ccnc3)=O)CCCC1CN(C(c1ccsc1)=O)C2 C1(C(=O)NC)CC=CC(n2cc(C3(O)CCOC3)nn2)C1.c1n[nH]c(C(F)F)n1 C1(C(N2CCC(CCN(C)C(C3CCC3(C)C)=O)CC2)=O)CC2C(C1)C2(C)C CCC(CCCO)NC(C1CCCCN1C(C1(C#N)CC(=O)C1)=O)=O c1(C(=O)N)ccc2c(c1)CCNC2=O.Cc1cn(C)cc1C(=O)NC(C)C(C)C CS(=O)(=O)C1CCCC1C(=O)NC1CC(C)C1.c1(C=O)cc2cccn2cn1.N C1(C2(O)CCCOC2)(Cn2cc(C(C(C)C)O)nn2)CC1 C1(c2n(CC)nnn2)(NC2C(C)C2(C)C)CCN(CC(F)F)CC1 c1(C(N(C)CC2CC(=C)C2)=O)nc(C)oc1C.C(=O)(C(C)C1(O)CCC1)N Cc1cc(C(=O)NC2CCN(C(c3cc(F)c[nH]3)=O)C(C)C2)nc(C)c1 Cc1cc(C(=O)NC2C3CN(C(=O)COC4CCCC(C)C4)CC23)ncc1C C=C(F)C1(CC(=O)NC2CC(C(F)C(N3CCC(SC)C3)=O)C2)CCC1 Cn1cc(Cl)c(C(=O)NCC2(CCNC(C3(CF)CC3)=O)CC2)n1 c1(CNC(c2nncc(OC)c2)=O)cc(O)ncn1.C(=O)CC.C(N)=O.C C=CCCC(=O)NC(C(=O)NCC(C)CO)C1CCCC1 c1(C(=O)NCC2CC(CNC(CSC)=O)OC2)ccccn1.CC(F)F.O c1(CCNC(c2cc(COC)on2)c2nnnn2C2CCC2)cccc(Br)c1C O(NC(=O)C1=CCC(C)(C)CC1)C(C(=O)N(C(CC)C1CC1)C)CC(C)C N1(CC)CC(C(=O)NC2CCN(C(C3CCC(C)CC3)=O)C2C)c2ccccc21 CCC(C)(C(=O)NCC(N1CCCC1c1cnc(OC)c(C)c1)=O)C(=O)O c1nnc2c(c1C=O)CCC2.C(C(C)CC(=O)NCC(C1CC1)N)OCC c1(C(C)C)nc2n(n1)CCCC2NC(c1c[nH]nc1-c1ccc(I)cc1)=O N1(C(C(C)(C)OCC)=O)CCC2CN(C(C3CCC=CCCC3)=O)CC2C1 CC1(C(=O)NCc2cn[nH]c2)CCCN1Cc1ccc(Br)o1 C1(C(=O)NCC(CO)NC(C(n2c(C)ccn2)C)=O)COC(=O)N1C C(N=c1nnn(C)[nH]1)C1OCCN(C(c2c(C)nc(O)[nH]2)=O)C1 C1(CCNC(C2ON=C(CC)C2)=O)CN(C(c2c(N)sc(C)c2C)=O)CCCO1 N1(C(c2c(C)nns2)=O)CC2CCN(C(c3cnn(C(F)F)c3)=O)CC12 S(=O)(=O)(c1ccccc1C#N)N1CCOCC(NC(C(C)C)=O)C1 C1(NC(C#CC(C)(C)C)=O)CCN(C(C2CC2C2CCCC2)=O)CC1(C)C N1CCCC2(CCN(C(=O)CS(C)(=O)=O)C2)C1.c1(NC(=O)OC)ccccc1.C N1(C(C2(CCC)CC2)=O)CC2CCCC(C1)N2C(=O)CCC=Cc1ccccc1 c1(C(=O)NCc2c(F)ccc(C)c2)ccc2nnn(C)c2c1 C12(C(N3CCC(OCCNC(=O)C=Cc4cnc[nH]4)C3)=O)CCOCC1C2 C1(NC(c2nc(C)[nH]n2)=O)CC2CCC(C1)N2C(C1(F)CC12CCCCC2)=O c1(OC)cnc(Cl)[nH]c1=NCCCC(C)NC(c1ccc(F)cn1)=O CC1(CNC(=O)C=Cc2cccs2)CCCC1.C(=O)(CCCCn1ccnn1)N c1(C(N(CCCCN(C(C2(CCC)CCC2)=O)C)C)=O)cc[nH]c1C1CCC1 C1(C)(CCC(=O)N(CCC)C)CCC(=O)N1.c1(C(=O)N)cccnc1.N(C)C C(C(CC(C)C)C(=O)NCc1cc(F)ccc1F)NC(C1(C(C)=O)CC1)=O c1(C(=O)NCC2(C)CN(C(C(C(=O)OC)C)=O)C2)scc2c1CCCC2.O Cc1ccnnc1C(=O)N(C1CCC(NC(C2CC2(F)Cl)=O)CC1)C C1(C(=O)NCC(CC)NC(=O)CCC=CBr)CCn2c(cnc2C)C1 Cc1ccn(C)c1C(=O)NC1CN(C(=O)C(C)(F)F)C1.N12CC(CC1=O)C2 c1(C(N2CC3(C(NC(c4ccsc4Cl)=O)CCC3)C2)=O)cc2c(cc1Cl)NCC2 C(CN=c1[nH]c(=NCC=CBr)[nH]c2c1CSC2)(C1CCOC1)OCC C(=O)(C(CCCSCCNc1nc(C)cc(C)n1)C(=O)OC)OCC N1(C(C2CCCNS2(=O)=O)=O)CCC2(CNC(C3(O)CCSC3)=O)CCCCC12 c1(CN(CC(c2nc(Br)ns2)O)Cc2ccccc2)ccc(Br)cc1 c1(CC#N)ccccc1C(N1CCC(CNC(=O)C(F)CC2CCOC2)CC1)=O CN1CCOC(C(N2CC(C)(CCC(=O)NCCc3cn(C)cn3)C2)=O)C1 N1(C(c2nc(C(C)(C)C)[nH]n2)=O)CCN(C(=O)C(C)(C)CC#N)CC1C1CC1 C(=O)(C1CCc2ccc(O)cc21)N1C(CNC(C2(OC)CCC2)=O)CC(F)C1 c1(C(N2CC3C(CNC(C(C)C4CC4)=O)C3C2)=O)ccc2ncnc(O)c2c1 CC(C)C(O)C(C)C(=O)NCc1cccc(C(N2CCOCC2C2CC2)=O)n1 c1(OC)ccc(CNC)cc1O.c1cc(C(N2CCC(C(C)(C)O)C2)=O)ccn1 c1(CCN(c2cc(-c3c[nH]nc3C(C)(C)C)[nH]n2)C)ccccc1Br C(C(C)(C)C(=O)N(C1CCOC1)C1CC1)SC c1(C(=O)NC(C)(C)CCS(C)(=O)=O)ccc2ccc3ccccc3c2n1 N1(C(Cc2nc(C)sc2C)=O)CC2(C1)SCCC2NC(=O)CC1COCCO1 C1(C(=O)N)CCC(=C(F)F)CC1.C1(CC(=O)NCC(O)CC)(CC=C)CCCC1 c1(C=O)cc(C)nn1CCC.C(C)(C(=O)NC(C)(C)C1CC1)OCCCC O=C1CCC(CCC(=O)N2CCN(C(=O)CCOC3CC3)C(CCO)C2)=NN1 C(=O)(CCCCN=[N+]=[N-])NC(CC#C)(C)C(=O)NCC1(C)NC(=O)NC1=O N1(C(=O)NC2OCCN(C(C)=O)C2)CCCC12CCCS(=N)(=O)C2 N1(C(c2cc(OC)ncn2)=O)CCCC(C)(C)C1C(=O)NCC(F)CO C1(C(N(CC(C)(C)NC(=O)Cc2ccc(O)nc2)C)=O)CCc2ccccc2O1 N1(C(CC(C)C(F)F)=O)CCCC12CCN(C(C1(c3cccnc3)CCC1)=O)C2 C1(NC(CC(=C)C)=O)CCN(C(C2CCCCN2C(C)=O)=O)C1(C)C C(C(C)(C)C(=O)NCCCO)OC(C)C.C(=O)C(O)Cc1ccccc1.CC N1(C(c2c(C)ncs2)=O)CC=C(CNC(C2CCC(=O)N(C3CC3)C2)=O)CC1 O(C=CC(O)(CNCCCC1CCCCO1)C(F)(F)F)CC C1CN(C(=O)CC2(O)CCOC2)CCC1(F)F.N1(CC)CCCCC1C(=O)NC N#Cc1ccc(C(=O)NC2CCCCC2CNC(=O)C(=Cc2c[nH]cn2)F)s1 N1(C(C2CC(C)(C)C2)=O)CCCOC(CNC(=O)C=O)C1.c1ccc(Cl)cc1.N N1(C(CCCC#C)=O)CC2(C)CN(C(c3nnc(S)n3C)=O)CC2(C)C1 C#CCCCC(=O)N1CCCC(N(C(C2C3CCC2(c2cnco2)C3)=O)CC)C1 C12(NC(c3ccc(F)cc3)=O)CCCN(C(c3ccc(Cl)cc3Cl)=O)CC1C2 C1(COCC)COC(C)(C)CN1C(c1ccc(C=O)cc1)C(=O)N.C1CC1 CC1CN(C(C2C=CC(NC(=O)CC(C3CC3)C3CC3)C2)=O)C12CCOCC2 c1(C(N(CCCN(C(Cc2c(C)ocn2)=O)C)C)=O)cc(F)cc(Cl)c1N N1(C(C(N2CCC(C)(C(=O)OC)CC2)=O)=O)CCC(F)(F)C(CO)C1 C12(CNC(C=CCOC)=O)CC1CN(C(=O)CCC(=O)c1ccccc1N)C2 C1(CC(=O)NC2(C)CC(NC(C=CC=CC)=O)C2)CCC1C1CC1 C1(C(N2CC3(NC(C4CCN(C5CCSC5)CC4)=O)CC2C3)=O)CC12CC2(F)F C(=O)(C1=CCC(C)(C)CC1)NCCNC(C1N(C(C)=O)CC(O)C1)=O C(=O)(C(C(C)(C)C)n1ccnn1)NC1CC(NC(c2n(C)nnc2Br)=O)C1 CCCCCCC(C(=O)NCC1CCOCC1)N(CC)CC1CCC1 c1(CC=O)ccncc1F.C(C(=O)N)=CCN(C)CC.C1CC1C(N)=O CC(C)(C#N)CCC(=O)N1CCCC(CO)(NC(C2CCC(C(N)=O)CC2)=O)C1 c1(C(=O)NCC2N(C(C=C)=O)CCC2C)ccc([N+](=O)[O-])cc1F N1(C(c2cccc(CC)n2)=O)CC=C(C(=O)N2CCC(CC3CC3)C2)CC1 C1(C(=O)NCC(C2CCCCC2)NC(CCC(C)(C)C)=O)CC2CCCCN2C1 C12(NC(CC(CCC)C)=O)CCC(CN(C(=O)CCSc3ccc(C)cc3)C1)C2 N12CCN(CC1=O)CC2.Cc1onc(C2CC2)c1C(=O)OCC(C)(C)C C(=O)(C(CC)CCCCCC)NC(CC=C)CNC(=O)C(COC)CC(C)C N1(C(c2c(C)cc(C(=O)OC)o2)=O)CCC2CN(C(=O)Cc3cnoc3)CC2C1 c1(C(=O)NCC2CC2)cc(F)c(F)cc1O.c1(C2C(C=O)C2)ccccc1Cl C1(C(N2CC(CNC(COCCOCC)=O)C(O)C2)=O)CCn2ncnc2C1 c1(OC)cc(C(N2CCC3CCN(C(=O)C(C)C)CC3C2)=O)cc2c1OCCO2 c1(CC(=O)NC2(CCNC(CS(CC)=O)=O)CCCC2)ccccc1[N+](=O)[O-] C1(C(=O)NCCC2N(C(c3c(CC)c[nH]c3)=O)CCSC2)CCC(C)NC1=O c1(OC)cnc[nH]c1=NCC1(NC(c2cnn(C)c2C)=O)CCCCC1C C(=O)(CCCCCSC)NC1(CNC(CC(COC)C)=O)CC1 C=CCC(C)(C)CC=O.C(=O)(C(=O)N=S(C)(C)=O)N1CC2C(C(F)(F)F)(C1)C2 c1(C(N(CCN(C(C(CCC#C)O)=O)C)C)=O)cccn2c(Br)cnc12 c1(-n2c(C)nnc2)ccc(C(=O)N(C2CCC(NC(=O)C=C3CC3)C2)C)cc1 C1CC2CCC(C1)N2C(c1cc(C)ccc1O)=O.S(=O)(=O)(CCC(=O)N)NC.C C(=O)(C1CCCc2c1ncn2C)NC(C1N(C(CNC(CCC)=O)=O)CCC1)C c1(C(=O)NCC(CNC(C(CC)OCC)=O)O)ccc2c(c1)OCCN2 CC1C2CC(C2)N1C(c1cc(C2CC2)no1)=O.C1(N(CC=O)C)CCSC1.N c1(OCC)cc(Br)cc(C(N2CCC23CN(C(=O)C(C)SC)C3)=O)c1N c1(C(=O)NC(CNC(C(CC)N(C)C)=O)(C)C2CC2)cc(F)cc2ccccc12 C=C(Br)CC(C)(C)C(=O)NCC1CC(NC(=O)C(CCC)OCC)CC1O c1(C(C)C(N2CCC(CNC(=O)C3=NOCC3)C23CC3)=O)cc(F)c(F)c(F)c1 c1(CCC(N2CC(Nc3ccnc(Br)n3)CC(F)C2)=O)ccc(Br)c(F)c1 N1(C(c2cncc(SCC)n2)=O)CC(NC(c2ccc(N)cc2C)=O)CC(C)C1 CC(C(C)C(=O)N1CCC(S(=O)(=O)NC(C)(C)C)CC1)S(C)(=O)=O CCC(C)C(O)CC(=O)N1CC(F)(F)CC1C(N1CCCC(CN=[N+]=[N-])C1)=O C1(NC(N2CC(C(=O)NC)C(C3CC3)C2)=O)Cc2ccccc2N(C)C1=O C1(NC(C(C)n2ccnc2)=O)CC(C(N2CCC(C(C)(C)O)C2)=O)CC1O Cc1cc(C)c(CNC(=O)NCC2CNC(=O)C2)cn1 c1(C(=O)NCC2N(C(C(C3CCC3)OC)=O)CC2)ccc2c(c1)CCO2 C(=O)(C(CC1(C#N)CCC1)N(C)Cc1cnc(-n2cccn2)s1)NCCC C1(NC(c2cn(C)nc2)=O)CN(C(=O)C2=COCCO2)CC2(CC2)C1 N1(C(c2cncc(SC)c2)=O)C(CNC(=O)Cc2nonc2C)CC2CCCC12 CN1CCC(O)(CNC(C2(C)CC2)=O)CC1.C1(CC=O)CCCC(O)C1.N CC(C)CS(=O)(=O)CCC(=O)N.n1(CC(=O)NC)cnc([N+](=O)[O-])c1.C1CC1 C(=O)(C(C(C)(C)CC)OC)NC1(CNC(C=CC)=O)CC1 CCCC(CCC)CC(=O)NCC(c1ccccc1)CNC(=O)CC(=O)N(C)C N1(C(CNC(=O)OCC=C)=O)CC2(NC(c3nc(Cl)sc3Cl)=O)CCC1C2 C(=O)(C(=O)N=c1cc(C)n(Cc2ccccc2)[nH]1)NC1C(CC)CN(C)C1 N1(C(C(C)(Cl)CCl)=O)CCCC2(CCCN2C(c2ccc3ncoc3c2)=O)C1 C1(C(N2CCC(c3ncno3)C2)=O)CC(=O)N(Cc2ccccc2)C1 c1(C(N2C(CCCNC(C(C(C)C)SCC)=O)CCCC2)=O)ccc(Cl)nc1O C=C=C(C)CC(=O)NC1CC(C)CC1O.N1(C(C=CC(=O)N)=O)CCOCC1 c1(C(=O)NCC(CN(C(c2cc(COC)no2)=O)C)O)sc(F)cc1Cl C1(C(=O)OCC)OCCNCC1N(C(C1(C#N)CC1)=O)Cc1ccncn1 c12ccc([N+](=O)[O-])c(c1)CN2C(C)=O.N1(CC)CCNC(c2nn[nH]n2)C1 c1(OCC)ccc(C(=O)NC2CCCN(C(=O)C(C)C#N)C2)cc1Br N1(C(C(C=C)O)=O)CCC(C2N(C(C3CCC(C(=O)OC)C3)=O)CC2(C)C)CC1 N1(C(=O)Cc2csnn2)CCCC(C2CC2NC(=O)C(F)(F)C(F)(F)F)C1 N1(C(C(C)OC)=O)CCC2(CC1)CC(C)N(C(=O)Cc1ccnc(F)c1F)C2 CC1CCC(O)(C(N2CC(NC(=O)CSCC(F)(F)F)C(C)C2)=O)CC1 C1(C(N2C(C(C)C)CCC2)=O)CC2C(C1)C2(F)F.N1(CC=O)CCC(F)CC1.N C1(CC=C)(NC(c2cc(Cl)no2)=O)CCCN(C(=O)C(C)C2CCCO2)C1 C1(NC(c2cc3cscc3s2)=O)CCN(C(c2cnn3cc[nH]c23)=O)C12CCC2 CCCCCCC(C)C(=O)NCC1(CNC(=O)C(C)SC(C)C)CC1 C1(C(=O)OCC)CCC(CC=O)CC1.C1CCCCN1C(=O)CN(C)C(C)C c1(C(=O)NC2C(c3n(C(C)C)ccn3)OCC2)cc(Br)cc(C(=O)O)c1F C=C(C)CCC(=O)NCC(C)(CO)NC(=O)Cc1ccc(Cl)cc1 c1(C(=O)NC2CCC(C)N(C(c3cnns3)=O)C2)n[nH]c2ccccc12 c1(C(=O)NC2(C3CCCC(C)(C)O3)CC2)cc(S(N)(=O)=O)c(F)c(F)c1F C1(CCC)CN(C(=O)CCn2cc(Cl)cn2)CC1C(=O)NCCOCC C1(NC(=O)C2=COCCO2)CCS(=O)(=O)C12CN(C(c1ccc(O)c(F)c1)=O)C2 N1(C(c2c(C)cn(C)n2)=O)CCCC(C2CC2NC(c2nc(Cl)cs2)=O)C1 c1(C(=O)N)ccc(C(F)(F)F)c(C)c1N.C1(C)(C(=O)NCCCC)SCCCS1 CC1CN(C(=O)Cc2csc(C(C)(C)C)n2)CCC1NC(c1cnc(O)n1C)=O c1(N(CC(C)C)Cc2n(CC)c(O)nn2)ccc(Br)cc1Cl c1(OC)cncc(NC(=O)C(CCN(C)C)NC(C2CN(C)CCO2)=O)c1 CC1CCOCCN1C(=O)CC1CN(C(c2ccccc2CC#N)=O)CC1C Cc1ccc(C2(NC(C3COC(CNC(c4ccncc4)=O)C3)=O)CC2)cc1 Cc1cnc(C#N)nc1N(CCNC(c1cnc2n1CCCC2)=O)C1CC1 C1(C(N2CCC(NC(CC(COC)C)=O)C(F)C2)=O)CCN(S(N)(=O)=O)CC1 C1(NC(C(=O)NCC)=O)CCC2(CC1)CCN(C(C1CCCCC1F)=O)C2 N1(CC(=O)NC2(CC)CCCN(C(c3cnc(Cl)s3)=O)C2)Cc2ccccc2C1 c1(CC)cc(C(=O)NC2CC(F)CN(C(c3ncccc3F)=O)C2)ccc1F c1(C(=O)NCC(CC)NC(=O)C#CC2(CC)CC2)ccc2c(c1)OCO2 N1(C(c2ccc(C)s2)=O)CCCC(C(C)(C)C(=O)N(C)CCc2ccncc2)C1 Cc1c(C(=O)N(C(C)CNC(=O)Cc2csc(Br)c2)C)cnn1C(C)C c1(C=O)ccnc(S)c1.C(CCCNC(C1CC(C(F)(F)F)(O)C1)=O)OC CC1c2cccn2CCN1C(=O)C(N1CCC(C)(O)CC1)=O C1(C(=O)NC2CN(C(c3cc(CC)on3)=O)CC2C)CC2CCCCCC12 c1(C(C)NC(N(C2C(C)CN(C)CC2)C)=O)ccc2ccn(C)c2c1 C1(C(=O)NC(C)CNC(c2cc(-c3ccccc3)no2)=O)CCC12CCOCC2 c1(C(=O)NC23CC(NC(C(C(C=C)C)C)=O)(C2)C3)n[nH]c2nccc(Cl)c12 c1(OC)cc(CN2CCC(=CC(=O)N(C3CC3)CC#N)CC2)ccc1F c1(CC)c(N2CCCC(CCNC(C3CCCC(OC)C3)=O)CC2)ncnc1Cl C(=O)(CC(CC)C(C)C)N1CCN(C(c2cc(CC)c(F)cc2)=O)C(CCO)C1 C1(NC(CC(CC)N(C(CCC#CC)=O)C)=O)CCC(C2CC2)C1 CC(C)(C)C(=O)CCC(=O)N1CC=C(C(=O)Nc2cccc(F)c2)CC1 c1(OC)cnc(CNC(C2CN(C(=O)C)CC2C)=O)cn1.C(=O)C(C)(C)C CC1CCN(C(=O)NC(C(F)(F)F)C2CCOC2)CC(C)O1 CC1(C)C(NC(=O)C(F)(F)C(O)C2CC2)CCN1C(c1cc2cscc2s1)=O CC1(C)C(O)CC1(CO)NC(=O)C(c1ccccc1I)F N1(C(CC2C(C)(C)OCC2)=O)CCN(C(c2[nH]cc3c2CCC3)=O)CC1C1CC1 C1(C(N2CC(C(C)NC(C3CC(F)(F)C3)=O)C2)=O)CCCN(C(N)=O)C1 c1(OC)ccc(C(C)C)cc1C.N1(C(C2(C=O)COC2)=O)CCCC(C)(O)C1 c1(C(=O)NCC2(O)CCN(C(c3cnc(C)o3)=O)C2)ccc([N+](=O)[O-])s1 c1(C(=O)NC23CC(NC(CSC)=O)(C2)C3)ccc(-n2cccn2)nc1 c1(NC(c2c(C(C)NC(CC(=C=C)C)=O)noc2)=O)cc(C)c(F)c(C)c1 CC(C)CC(C(=O)NC1CCN(C(C2C3COCC23)=O)CC1O)N(C)C c1(C(C(=O)NCC(CC=C)NC(c2cc(Cl)cnn2)=O)C)cc2ccccc2o1 c1(C(=O)NC2(C3N(C(Cc4ncc(C)o4)=O)CCC3)CC2)cccc(N(C)C)c1 O=S(=O)(c1cc(Cl)c(Br)cc1F)NCC1CCN(Cc2c[nH]ccc2=N)CC1 C1(CC)(NC(C2CCOC(C(C)C)C2)=O)CCN(C(=O)C(C)=C2CCC2)CC1 c1(C(N2C3CCC(C3)C2)=O)ccc(S(C)(=O)=O)s1.CC1(C)CC1C(=O)N c1(C(=O)NCCC(C)C)ccc(OC(F)F)c(F)c1.C12(C(=O)N)CCOCC1C2 C(=O)(C(F)(F)C(F)(F)F)N1CC(C)(C)CC1.C(c1ccc(F)c(F)c1)=CC=O N1(C(c2c(C)snc2)=O)CC(NC(=O)C(N2CCCC2)C2CC2)C(O)C1 N1(C(c2cc(C(=O)OC)no2)=O)CCC(F)CC1.C1(CC=O)CCN(C)CC1.N N1(C(C=CC)=O)CCN(C(=O)Cc2cc(Cl)ccc2Cl)C2CC12 CCC(CNC(c1oc(CNC(c2cccc(F)c2)=O)nc1C)=O)CCO c1(CC)ccccc1OCC(=O)NCC(C)CNC(=O)Cc1cnnn1C c1(NC(C2(C)CN(Cc3sccc3Br)C2)=O)ccc(Br)nc1Cl C1(NC(c2ccc([N+](=O)[O-])o2)=O)CCN(C(=O)CCCc2ccncc2)C12CC2 CC1CCN(C(c2ccc(Cl)nc2Cl)=O)CCN1C(=O)CC1CCC2CC2C1 C1(C(=O)NCC2C(NC(=O)CCn3cncn3)CCC2)CC2COCC2C1 c1(C(N2CCC(COC)(NC(c3ccc(O)nc3)=O)C2)=O)ccc(F)cc1O c1(C(C(=O)NC2COC2)N(C(CC)C)CC)ccc(C2CCCC2)cc1 CC1CN(C(=O)Cc2cncs2)CCC1NC(=O)C(c1cscn1)N(C)C N1(C(CCN(C)CC)=O)CCCC(C)(CNC(=O)Cc2cc(C)cs2)C1 N1(C(C=CCOC)=O)CCC2(CC1)CN(C(=O)C=CS(C)=O)C2C(C)C C(=O)(C(C)(C)c1ccn(C)n1)N(C1CCN(C(=O)CCOCC(F)F)C1)C C1(NC(CC2N(C)CCC2)=O)CC2(C1)CC(C(N1CC3CC3C1)=O)C2 C1(NC(N(C(C)(C)C)C2CC2)=O)CCCC(C(=O)OC(C)(C)C)CC1 c1(CO)ccc(NCc2cc(OC)nc(-c3ccncc3)n2)cc1C#N C(CCN=C(NCC1(CSC)CC1)NCC1CC1(F)F)SC C1(NC(C(C2CC2)SC)=O)COCC1C(=O)NCc1cn(C2CC2)nn1 C1(NC(C(COC)(C)OC)=O)CCC(O)CN(C(=O)C2=NOCC2)C1 c1(NC(C(=O)OC)=O)cc(C(NC(=S)Nc2ccccc2)=O)cn1C N1(C(COC(C)C)=O)CC(C(F)(F)F)CC1C.c1ccccc1.C(=O)(CC)N C1(OC)(C)CCN(C(c2cccc(Cl)n2)=O)CC1.c1(CCC(=O)N)ncc(C)[nH]1 c1(CC)ccc(C(N2CC3(CNC(C4CC=CCC4C)=O)CC2CO3)=O)cc1F c1(C2C(C)C2)cc(NC(N2CC(C)(CC(F)F)C2)=O)no1 c1(C(N2CCC(C)(C(=O)O)CC2)=O)cc2nc[nH]c2cn1 C1(C(N2CCCC(Nc3nc(C)nc(C)c3F)CC2)=O)CCn2c(cnc2C)C1 C(=O)(C1=NNC(=O)CC1)N1CCN(C(C)C(=O)O)CC1 Cc1cc(Cl)cc2c1N(C(N1CCC3(O)CCCCC3C1)=O)CCC2 C1(CNC(=O)C(F)=CC2CC2)CN(C(C23COCC2C3(F)F)=O)CC1(F)F N1(C(CC(=C)Br)=O)CC(n2cc(-c3cncc(C(=O)OCC)c3)nn2)C(SC)C1 c1(NC2CC(F)(CNC(C(CC(C)C)C)=O)C2)ncnc2cnn(C)c12 C1(NC(=O)C=Cc2cnc[nH]2)CN(C(c2cc3n(c2)CCCC3)=O)C2(CCC2)C1 C1(C(C(=O)NC(C)(C)C)N(C)CCF)CCC(C)CC1 C1(C(NOC(C(C)C)CO)=O)CNC(=O)CN1C(=O)CC1C=CCCC1 C1(CCCC)CN(C(c2nc(C)c(C)s2)=O)CCN1C(=O)C1=CCCOC1 c1(N2CC(CC(C)NC(CN(CCOC)C)=O)C2)ncc2ccnc-2[nH]1 N1(C(C(C)c2ccsn2)=O)CCCC(O)(CCNC(c2ccncc2F)=O)C1 c1(NC(C2CC(O)CCN2C(C2C3COCC23)=O)=O)c(Cl)c(F)nc(F)c1Cl C1(NC(C(CC)(C)CC)=O)CN(C(c2ccc(F)c(C#N)c2)=O)CC(F)(F)C1 C(=O)(CCCS(C)(=O)=O)NC(C1(O)CN(C(C2OCC3CCCCC23)=O)C1)C c1(N2C3(CN(C(c4cc(=O)cco4)=O)C3)CC2)nc2ccccc2s1 Cc1cc(CNC(C2(CCNC(=O)CCC)CCC2)=O)co1.C(N)(=O)N Cc1[nH]nc(C(=O)NC(Cc2cnc[nH]2)C(=O)NC23CC2CN(C)C3)c1O CC(C)CC(C(=O)N1CC(CO)C1)NC(C1CC(=O)C12CCC2)=O N1(C(C2C(C(=O)OC)CCCC2)=O)CCN(C(=O)CCC2CCC2)C(CO)C1 n1(CC(=O)N(CCC(=O)NC(CCC)C2CCC2)CCO)ncn(C)c1=O C(CC)(CCC(=O)NC1CCCN(O)C1=O)NC(C(CCC)N(C)C)=O C(=O)(C1=C(F)CN(C(c2ccc(F)cn2)=O)CC1)Nc1cc(C)cc(F)c1 c1(OC)nn(C)cc1C(N1CCC(C(F)C(=O)NC)C1)=O.c1ccc(C#N)s1 Cc1cc(C(CO)NC(=O)COC(c2conc2-c2ccc(Cl)cc2)=O)ccc1Br c1(C(N(CCCNC(C2(C#N)CC2)=O)C)=O)nc(Br)[nH]c1C(F)(F)F C(=O)(C(N=[N+]=[N-])C(C)C)NCCC1CCN(C(C2CC(CC)C2)=O)C1 c1(CC)sc(C(N2CC(OC)C(NC(=O)CC3(C)OCCO3)C2)=O)cc1C N1(c2c(C)c(NC3CCCC(CO)C3)ncn2)CCOC2(CCOCC2)C1 N1(C(CSCC(N)=O)=O)CC2CC(NC(C3CCCCNC3=O)=O)CC1C2 CCCC(C(=O)N1CCCC1C(C)(C)CNC(c1cccc(F)c1)=O)OCC Cc1cc(C)c(C(=O)NC(C(=O)NCC(c2ccncc2)C)C2CC2)cn1 N1(C(c2c(OC)c(F)ncc2)=O)CCC2CCC(NC(=O)C(C)C3CC3)C1C2 CC(C)(C(F)(F)F)c1ccc(CNC(c2ncn(-c3ncccc3F)n2)=O)cc1 C(=O)(C1=CS(=O)CCC1)N(CC(C)(C)C)C.C1(C=O)CCCN(C(N)=O)C1.N [SH](=O)(=O)c1cccc(C(=O)N)c1.C(=O)CC(C)(C)C.CC(C(N)=O)N1CCC1 Cc1nn(C)c(N)c1C(N1CC(NC(C2CC2Br)=O)C(C)(C)C1)=O CCC(C(=O)NCC(C1CCCC1)NC(=O)C(=O)NC(C)C)C(C)C C1(CNC(Cc2c(C)cco2)=O)CCCCCN1C(c1cnc(Cl)s1)=O C(=O)(C(C)CC(F)(F)F)NC1CC(C)(NC(CCCc2ncc(C)o2)=O)C1 c1(C(=O)NCC=CCNC(c2ncc(C)cc2C)=O)c[nH]c2nc(F)ccc12 c1(CC)noc2ncc(C(=O)NC3CCN(C(c4cn(CCF)nn4)=O)C3)cc12 c1(OC)ccc2sc(C(=O)NC3CC3NC(=O)Cn3cnnc3)c(C)c2c1 N1(C(c2c(C)non2)=O)CCOCC1C(=O)NCC(C)(O)C(C)C C1(C(N2CCC(C(C)(C)NC(=O)C(F)CC3CC3)CC2)=O)CCC2CCCCN12 CC(C)C1=NOC(C(=O)NC2CC(CNC(C3CNC(=O)CC3C)=O)C2)C1 N1(C(C2(N(C)C(C3CC3[N+](=O)[O-])=O)CC2)=O)CCC2(COC(=O)N2)C1 CN=c1nc(N2CCC(OC(C)(C)C)C2)[nH]c(=NCC2(F)CC2)[nH]1 C1(OC)CC2(C1)CC(C(=O)NC(C)C1CC1)C2.C(=O)C=CC(C)C.N c1(C(=O)NC2C(C)N(C(=O)Cc3cncs3)CC2)ccnc2ccnn12 c1(OCC(N2C(C(=O)NCC(=O)N)C=CC2)=O)cncc(Cl)n1.C1CC1 C(=O)(CCS(C)(=O)=O)NCC(C(C)C)NC(=O)CCC(=O)c1cccnc1 N1(C(c2ccc(C)c(C)c2)=O)CCOC2(C1)CN(CC(=O)NCC1CCC1)C2 c1(N2CCCC(COC)C2)nc(NC2CCC=CCC2)nc2scnc12 N1(C(CSc2n(C)ccn2)=O)CC2CCN(C(C3Cc4nccn4C3)=O)C2C1 c1(C=O)ccc(Br)c(C)c1C.c1(OCC)cccnc1C(N1CC(CO)C1)=O.N C1(CC(NOCC)=O)CN(C(c2nocc2C)=O)CCO1 c1(OCCC)cccc(N(C(=O)C(O)C(C)OCc2ccccc2)CC)c1 c1(OCCOC)ccc(C(=O)OCC(=O)Nc2nc(Br)ccc2Br)c(F)c1F CC(C)CC(C)C(=O)N1CCC(CNC(c2ccc(NC=O)cc2)=O)C12CC2 c1(C(C)CC(=O)NCC2CCC(NC(C3(F)CCC3)=O)C2)ccccc1Br N1(C(C=CCN(C)CC)=O)CCN(C(c2ccnnc2C)=O)CC2(C)CCCC12 C1(NC(c2cc(C)n(C(C)(C)C)n2)=O)C(C)CCN(C(=O)C2=CCCC2)C1C N1(C(c2cc(C)n(C)c2C)=O)CCC(C2CCN(C(=O)CC3CCCO3)CC2)C1 O=C(C1CCCc2nccn21)NCCCCCCn1cc(CCCO)nn1 C1(CC(=O)NCC(=O)NC(C)C)CCCN1C(c1cnc(O)o1)=O N1(C2CC(CC(=O)NCCC3CC(CN)CO3)C2)CCOCC1.c1cn[nH]c1.C c1(C(=O)NCC(C)(C(C)C)NC(CC(=C)C)=O)cc(Cl)ccc1Br C(C(C)(C)CC(F)F)NC(C1OCCC(NC(CC=CCC)=O)C1)=O c1(OC)cccc(-c2noc(CNC(=O)C(=O)N)n2)c1.C1(O)(CC)CCCC1 C1(CC(=O)NCC(c2ccccc2C(F)(F)F)N)CC2(CNC2)CO1 c1(C(=O)NCC(C)CNC(C2CCCC2C2CC2)=O)coc2c1C(=O)NCCC2 c1(OC)ccc(OC)c(C(=O)NCCC2CCCN(C(c3sccc3C)=O)C2)c1 c1(C(=O)NC(C)C(C)(C)NC(=O)C=CC2CCOC2)cccc2ccn(C)c12 C1(C=O)CC2(CCOCC2)CO1.C(c1ccoc1)=CC(=O)NCC1(CC)CC1 C(CCC(C(=O)NCC(c1cccnc1)O)NC(=O)C(O)C1CCC1)OC N1(C(=O)CCCC2CC2)CCC2(CCCN(C(=O)CCc3cccs3)C2)C1 C1CN(C(=O)C=CC(C)C)CC12CCCC2.c1(OC)cc(C=CC(=O)N)sn1 C1(NC(c2ccc(Cl)c(O)c2)=O)CC2CN(C(=O)Cn3nccn3)CC12 C(=O)(C(O)CC(F)(F)F)NCC1(CO)CCN(C(c2cn(C)c(=O)cc2)=O)C1 c1(C(N(CCC(=O)NCC2CC(=C)C2)CCO)=O)cnn(C2CC2)c1 c1(C(=O)NC(CC)(C)C(=O)O)cnc(C)c(C(C)=O)c1 C(C(CO)(CO)NC(=O)CC1CC(=O)NC1=O)N(C(C(C)OCC)=O)C C(c1ccc2[nH]ccc2c1)=CC(N1CC(C)CCC1)=O.C1(CC#C)(C(=O)N)CC1 C(c1cc[nH]c1)=CC(=O)NCCN(C(c1cccn1C)=O)CC C(=O)(CCCCC#N)N1CC=CC(C(N(CC(C)O)CC(F)F)=O)C1 N1(C(C2CC(NC(C3(CCN(C)C)CC3)=O)C(O)C2)=O)CCC(C2CC2)C1 C(CC(C)C)(C=O)NC(CC1(CS)CC1)=O.C1(C#N)CC12CCC2.CCC CC1(C)CCC(CNC(=O)CC2(C)CC2)N(C(C2CCC(=O)O2)=O)C1 N1(C(C23CC(C)C2C3)=O)CCC2(C1)CN(C(c1cc3sccc3[nH]1)=O)CC(C)O2 c1(C(C)=O)c[nH]c(C(=O)NC2CC(NC(=O)CSc3nccn3C)C2)c1 c1(C=O)ccc(F)c(S(N)(=O)=O)c1.C(C)(C)(CC(=O)N1CCC(CC)C1)OC CCC(=O)CCC(=O)N(C(C)C(=O)NC(CCOC)C(C)C)CCC N1(C(C2C(NC(c3ccn(C)n3)=O)CCC2)=O)CCC2(CC1)CC(C)(O)C2 C1(CNC(C(C)NC(c2ccccc2Cl)=O)=O)CC2CCC(C1)C2 C12(C(=O)NCCCN(C(c3ccccc3F)=O)CC)CCCN1CC(OC)C2 Cc1cc(C(F)(F)F)ccc1C(N1CCC(CC)C1)=O.C(=O)(C=O)N.C(C)C C1(C2N(CC)CCC2)CCCNC(=O)C1.C1CCS1.C1CO1 c1(CCC(N2CC(NC(C(CC=C)C)=O)C2)=O)ccc2c(c1)COCC2 C(=O)(C(O)CC(F)(F)F)NC(CCC)C(N1CC2(CCN2C)C1)=O c1(C(=O)NCCC2(O)CCN(C(C(C)OC)=O)C2)cc2c[nH]cnc-2n1 C12(NC(c3c(C)c(N)cnc3)=O)CCOCC1CN(C(C1(CO)CC1)=O)C2 N1(C(c2cc(CNC(c3c(C)ccs3)=O)sc2)=O)CCC(C)C(F)(F)C1 CC1CN(C(=O)CC2CC(F)C2)CC1.C(=O)CC(O)CC1CC1.C(=O)(C)N C1(C(=O)NCCN2CCC(NC(C(CC#C)C)=O)CC2)OC2CCC1CC2 c1(-c2cc(OCC)ncc2)ccc2[nH]c(C(=O)NCC3CCC(F)C3)cc2c1 CC1(C)CC(C(=O)NC2CCCCCC2O)CN(C(C2CCSC2)=O)C1 CN1CC(C(=O)NC2CCC(NC(=O)CC(c3cccc(F)c3)O)CC2)NC1=O O=C(CC=C(Cl)Cl)NCCOC1CN(c2cccc(-c3nn[nH]n3)c2)C1 CC1CN(C(=O)CCC(C)(F)F)CC(C)C1NC(C12COCC(C1)C2)=O C(=O)(CCCc1ccncc1)NCC1N(C(C(C)C2CCCO2)=O)CC1 CC1Cc2c[nH]nc2C(C(=O)NCCCOCCNC(=O)Cc2ccoc2)C1 N1(C(CC(COC)C)=O)CC(NC(c2cnsc2C)=O)C2(CCOCC2)C1 C(c1ccc(F)cc1)=CC(=O)NCC1(C)CCC1.c1(CC=O)cc[nH]n1.N N1(C(C(C)CC(N)=O)=O)CCCCC2(CCN(CCCC(C)(C)C)C2)C1 c1(C(=O)NCC(CC)(C)NC(c2cnnn2C)=O)cn2c(C)cccc2n1 c1(C(N2CCC(N(C)C(=O)O)C2)C(=O)NCC=C)cc(C(C)C)on1.C C1(C(=O)NCC(C)C)C2CCC1(c1ccncc1)C2.C1(C(=O)N)CCC(=O)N1 N1(CC=O)CCN(c2cnn(C)c2)C(=O)C1.c1(NC(CC)=O)cccc(C)c1.N C1(C(N(C2CCN(C(c3ocnc3COC)=O)C2)CC)=O)CC(=O)CCO1 N1(C(C(C2CCN(C(c3cc(C)n(C)c3C)=O)CC2)CC)=O)CCCC(O)CC1 N1(C(c2c(CC)ncs2)=O)CC=CC1(C)C(=O)NCc1sc(C)cc1C CC(C)(C#N)CCCC(=O)N1CCCC(NC(=O)C(C)(C)c2ccccn2)C1 N1(C(c2c(F)ccc(C(=O)OCC)c2C)=O)CCC2(CCN(C(=O)C)C2)C1.O CC1CN2CCN1CC2C(N1CCCCC1CCNC(C1CN(C(N)=O)C1)=O)=O Cc1cccc(-c2ncccc2C(=O)NC2(C)CCN(C(=O)C(C)(C)Br)C2)n1 N1(CCCC(=O)NC2CCN(Cc3ccccc3)C2)C(=O)CCC1=O CC1COC2(C1)CN(C(=O)C(C)(C)C1CCN(C(c3cnc(N)cn3)=O)C1)C2 S(=O)(=O)(c1cccc(Br)n1)N1CC(C(=O)NC2CN(C)C2)C(F)(F)CC1 C(=O)(C(O)C(C)(C)CC)NCC(CC(=O)NC(C(CC)CC)C)OC Cn1cc(N(C(=O)CONC(=O)CC2CCC(=O)C2)CC2CC2)cn1 c1(C(N(CC(CC)NC(C2CCCCN2C)=O)C)=O)cc2sc(C)cc2[nH]1 C1(NC(C(CC)c2ccccc2)=O)CCN(C(c2cc(C)cs2)=O)C1CC N1(C(C(C)C2CCCO2)=O)CCC2(CC1)CN(C(=O)CCCC1OCCO1)C2 C1(C(=O)N(c2ccnn2C)C)(CC)CCCN(C(C2CCOCC2)=O)C1 Cc1cc(C2(C(=O)NC(C)CC(C)NC(=O)CCCN(C)C)CCC2)no1 N1(C(C=C(C)C)=O)CCC2CCN(C(=O)C(N3CCC(C)CC3)=O)CC2C1 C1(CC#C)(C(=O)NCCC2(C)CC2)CCCC1.C1(CC=O)CCOC1=O.N CCC(O)CC(=O)N1CCCC1C(C)(C)CNC(=O)COC(C)=O Cc1cc(C(=O)NCC2CCC2)c2cccc(C)c2n1.C(=O)C(F)S(C)(=O)=O N1(C(C(CCC)C(=O)OC)=O)CCCC(C2CC2NC(C2CCC(=O)N2)=O)C1 Cc1c(C(=O)NCCC2CC(NC3(c4cn(C)nn4)CC3)C2)cccc1F C1(NC(c2nnc(CC)s2)=O)CC(C)N(C(=O)CC2(CO)CCC2)C1 N1(C(C2CCC(=O)OCC2)=O)CC2CCCC(CNC(c3coc(Cl)n3)=O)(C2)C1 n1(CC)cnc2nc(=NCc3cc(Br)no3)[nH]c(NCC3(COC)CCCC3)c12 C1(C(=O)OC)CCC(C(=O)O)N(C(=O)NC2(CN3CCCC3)CCCCC2)C1 c1(C(c2csc(C)n2)CC)ccc(C(N)=O)cc1.C1(C(=O)O)(C(C)C)CC1 N1(C(C2C3(C)CCN(CC3)C2)=O)CCCC(C2CCN(C(=O)C3=NOCC3)C2)C1 c1(CNC(N2C(Cc3c(OC)cc(Cl)cc3)CCC2)=O)cnn2c1CCCC2 C1(C(N(CCC(=O)N(C2CCCC2)CC)C)=O)CN2CCN1CC2 Cc1cc(Cl)cc(C)c1C(=O)NC1CC2CC1CN2C(=O)CCCn1ccnc1 c1(C(N2CCN(C(C3C(CC)OCC3)=O)C(CO)C2)=O)sc2cccnc2c1Cl C1(NC(CSCC(N)=O)=O)CCOCC1.c1(C=O)ncccc1C(F)(F)F.N C(=O)(CC(C)CCC)NC(CC#C)C(N1CCOC(C#N)C1)=O c1(C(N2C(CN(C(C3CC(C#C)(O)C3)=O)C)CCC2)=O)ccc(C2CC2)cc1F Nc1cnc(Cl)cc1C(=O)N(C1CCN(C(=O)CCC(F)F)C1)CCO N1(C(C(c2cccc(Cl)c2)C)=O)CC23CCCC2(C1)CN(C(=O)C(N)=O)C3 N1(C(C(c2cn(C)nn2)NC(Cn2ccc(C)c2)=O)=O)C2CCCC1COC2 CCCCCC(O)C(C)C(=O)NCCCC(C)(C)NC(C1CCCC1CCC)=O C(=O)(C#CC1CCOCC1)N1CCCC(CC(=O)NC(CCC)C(C)(C)C)C1 c1(NC(=O)NCC2N(CCC(C)C)CCC2)ccc(CN(C)C)nc1 N1(C(C(C2CC2)OC)=O)CCN(C2CCCN(C(c3ccncn3)=O)C2)C(=O)C1 C1(CNC(C2CC(OC)C2)=O)CCCN(C(c2ccc(O)cc2)=O)CC1 CCC(C)(C#N)C(=O)N1CC(CC(=O)NCC=C(C)C)C(C)C1 n1(CCNC2C(OC)C(C)(C)C2)cnc2c(oc3ccccc23)c1=O c1(C(N2CC3C(C(=O)Nc4c(OC)ncnc4)(C3)C2)=O)c(Cl)cccc1Br C1(NC(c2cncc(Cl)c2)=O)CN(C(c2nccc3n[nH]cc23)=O)C2(CCC2)C1 C1(C)(CNC(C2(CC#C)CCOC2)=O)CCCN1C(c1ccns1)=O c1(C(N(CC(C)C)C)=O)cccnc1-n1cccn1.C(C1CCOC1)=CC(=O)N N1(C(Cc2cn(CC)nn2)=O)CC(CO)C2(C1)CN(C(=O)C(C#N)C(C)(C)C)C2 CCCCCCCCC(=O)N(C)CC1CCCCN1C(=O)CC1COCCN1C c1(C(=O)NC(CC)CN(C(=O)CCSCc2ccccc2)C)cc(O)ccc1C N1(C(C=C(C)Cl)=O)CC2(COC(CNC(c3cnc4n3CCCC4)=O)C2)C1 c1(C(=O)NC2(CN(C(=O)CCC3CCOCC3)C)CC2)ncoc1C1CC1 C(CC)(CC)(CCNC(=O)Cc1c[nH]nc1O)NC(CCCOCC)=O C12(NC(C(c3cc(C)sc3)(C)C)=O)CCC(CC1)N(C(C1C3COCC13)=O)C2 Cn1nnc2c1CC(C(N1CCC3CN(C(c4cnsn4)=O)C3C1)=O)CC2 N1(C(C(CN(C(c2c(C)cccc2F)=O)C)C)=O)CC(O)C(C2CC2)C1 c1(C(=O)NC2CCN(C(=O)CC3CC=CCC3)C2)cc2nn[nH]c2cc1F C1(C(CNC(C(C=C)O)=O)C)CCN(C(c2c[nH]nc2C2CC2)=O)CC1 Cc1ncn(C)c(=O)c1C(=O)NCC1CC1.C(=O)C(F)CC1CCC1.C Cc1sc2ccccc2c1C(N1CCC(NC(=O)CC2CCCN2C)CC1)=O N1(C(Cc2c(C)cccc2)=O)CCC2(CC1)CN(C(c1cccc(=O)o1)=O)C2 N(C)(S(=O)(=O)N(C)C)CC=O.C1(O)CCN(C(=O)C=CC2CCC2)C1.C CC(CCNC(c1ccnnc1)=O)CCNC(=O)C(O)Cn1cncn1 C1(NC(Cc2c(C(C)C)cccc2)=O)CCCN(C(C2(O)CC(CF)C2)=O)CC1 Cn1cc2cc(CN3CCCC(CNC(c4cc(F)cc(Cl)c4)=O)C3)ccc2n1 N1(C(C(CC#C)C)=O)CCOC2(CCN(C(c3ccc(Br)cc3Cl)=O)C2)C1 C(C1CCCC1)=C(C)CNC(=O)CC1CCN(C(=O)C(=Cc2cnc[nH]2)C)C1 Cc1cc(O)cc(O)c1CNC(N1CC(O)C1)=O.c1cccc(C(F)(F)F)c1 C(=O)(C(C)(C)c1ccn(C)n1)N.C(C)C=O.CCC.C1(CC=C(C)C)CCC1 C1(NC(C2CN(C(C)=O)C2)=O)CC2(CCCN(C(c3cccnc3N)=O)C2)C1 c1(C(=O)NC(CC)CNC(c2cc(C)on2)=O)cc(OC)nn1C N1(C(C2CC(C)OC2)=O)CCC(C)(CNC(c2cc(C3CC3)no2)=O)CC1 N1(C(C=CC=CC)=O)CC2CCC(C(=O)NC(C)C(C)(C)OC)(C2)C1 C1(C(=O)NCC=CCSC)CN(C(=O)C=C(C)C2CC2)CC1C C(=O)C(C)S(C)(=O)=O.c1(OCC)ncccc1C(=O)NCC1CCCC1 N(C1CCCNc2ccccc21)C(c1ccc2c(c1)CCOC2)=O C(=O)(C(C(C)C)NC(c1c(C)nsc1C)=O)NCCOCCOCC C1(NC(CC(C=C)C)=O)CC2(C1)CC(NC(=O)C(C)(C)c1ccno1)C2 C1(NCCCc2cn(-c3cccc(COC)c3)nn2)COCC1C1CC1 Cc1c(C(=O)NCC2CCN2C(C2(Cl)CC2)=O)sc2cncn12 C(=O)(C=CS(C)=O)N1CCC(N(C(c2c(C(C)C)ncs2)=O)CCO)C1 C1(CNC(c2c(C)ccs2)=O)CCCCC1C(=O)NC1CCSCC1 O=C(CCC(F)(F)F)NC1(C(N2CCC(O)(C(F)F)C2)=O)CCOCC1 C1(CNC(=O)NCC2OC(=O)CC23CCC3)CCCC2(C1)OCCO2 C12(CC)CN(C(=O)CC3(C(F)F)CC3)C(C1)C2.c1(C=O)cnc(O)cc1C C1(C(CO)NC(=O)CN2CCCC2CO)CCN(C(C2CC(O)C2)=O)CC1 c1(C(N2CC(O)(CCNC(CC(CC)OC)=O)C2)=O)nn2c(c1C)OCCC2 C12(CNC(C(C)Cc3ccco3)=O)CC1CN(C(=O)CCc1cccnc1Cl)C2 N1(C(COC)=O)CCN(C2CN(Cc3ncn(-c4ccccc4)n3)C2)CC1 C1(CC)CCCCO1.n1(CCC)nccc1C(C(=O)NC)N(C1CCC1)C CS(=O)(=O)C1CN(C(C2CSCN2C(=O)CC2CCCCCC2)=O)C1 CC(C)C(CNC(c1cnn2c1CCC2)=O)C(=O)NCCC1C=CCC1 N1(C(C(COCC)C)=O)CC2CC(NC(=O)CN3CCCCS3(=O)=O)C1C2 Cc1nc2cnn(C)c2cc1C(=O)NC1CCCC1NC(C1(ON)CCCC1)=O C1(C)CCCN(c2cc(C(=O)N(C)C)ncn2)C1.c1(OC)noc(C)c1C(=O)N C(C=O)(C(C)C)OCC.C1CC2(C1)CC2.c1(C=O)sc(CC(C)C)nc1C.N N(C1c2cc(Br)ccc2SCC1C)NC(C(C1(O)CN(C(=O)NC(C)C)C1)F)=O N1(c2cccc(C(C)O)n2)CCC(O)c2cc(Cl)ccc21 C1(C(C)C)CN(C(=O)Cn2nccn2)CCC1NC(C1CCC(C)(F)CC1)=O C1CC2(CCC2)CN1C(=O)Cc1ccc(Cl)nc1.CC1(C)CCC(C(=O)N)O1.C c1(C(C)C)cc(C(=O)OCc2ccc(CN(C)C)cc2)nn1-c1ccncc1 c1(C(N(CC(O)CNC(=O)CC2CNC(=O)C2)C)=O)cc(O)ncc1F N1(C(CN2CC(=O)NC2=O)=O)CCc2ccccc2C1CCCNC(=O)CO c1(OC)cccc(C(=O)NC2CN(C(=O)CC(C)(C)C3CC3)CC2OC)c1F CC(C)C(CCN(C)C(C1CC(C)(C)CO1)=O)NC(c1ccoc1Cl)=O c1(NC(C2CCC(OC(F)F)C2)=O)cc(Cl)c2ccccc2n1 C1(CCC=C)(C(=O)O)CCN(C(=O)Nc2cccc(C3CCC34CCC4)c2)CC1 c1(NC(C2CCC(NCc3ccccn3)C2)=O)ccnc2c(Br)cccc12 c1(C(=O)NCC(CNC(C(C2CCCCC2)OC)=O)CO)ccc2cncn2c1 c1ccccc1.C1(C(=O)OC)CC(C(=O)NCC2CC2)C1.C(=O)C1CC1 c1(OC)ccccc1C(C(=O)NCC1CCCO1)N(C)CC1CC1 Cc1cc(C=O)nc(C)c1.C1(C)(CC=O)CCS(=O)(=O)N1.C(C)C1CC1.N Cc1sc(S(N)(=O)=O)cc1C(N1CC(NC(C23CCC2C3)=O)CC12CCC2)=O c1(C(N2CC(C)(NC(C3C(=C)C3)=O)C2)=O)nc(C)oc1-c1ccccc1 N1(c2ccc(S(=O)(=O)NC(c3nnc(C)o3)C)cn2)CCc2ccc(F)cc2C1 N1(C(c2ccc(O)nc2Cl)=O)CCC2(CCN(Cc3c(Cl)cncc3Cl)CC2)C1 Cc1nc(C(=O)NCC2CCCC(NC(C3(C)CC(C)(C)C3)=O)C2)cn1C C12(NC(Cc3n(C(C)C)cnn3)=O)CCCC1N(C(c1nccnc1N)=O)CC2 C12CN(CC1c1ccccc1F)C(=O)COCCC(=O)N2.C(C(=O)OC)OC C(C(=O)NCC1CCCCN1C(C1CCCOC1C)=O)(C(C)C)OCC N1(CC(=O)NC(C)C(C)(C)NC(C2CCC=CCC2)=O)CCC(F)(CO)C1 C1(NC(=O)CCc2cnoc2)CN(c2ccnc(C3CC3)n2)CC12CCOCC2 c1(CNC(c2ccnc(O)c2)=O)cccc2c1CCN(C(c1coc(Br)c1)=O)C2 C(=O)(C(C#N)CCC)N.N1(C(C2(CC#C)CC2)=O)CCC1CN=[N+]=[N-] Cc1ccc(CCC(=O)NC2CCCC2NC(=O)C(O)C(F)(F)F)c(C)c1 C1(NC(C(CCC(C)C)O)=O)CCS(=O)(=O)C12CN(C(=O)CC1CC1)C2 C(c1cccc(Br)c1)=CC(=O)NCC1N(C(COc2cc(C)on2)=O)CC1 c1(SCC)cncc(C(=O)NCC(C)CN(C)C(c2cnn(C)c2)=O)n1.O c1(C(N2CC3(C(C(=O)Nc4ccc(OC)nn4)C3)C2)=O)cccc(C#N)c1OC c1(C(=O)NC2C(C)CCN(C(c3c(C)nsc3N)=O)C2)ccc2nncn2c1 C12(NC(Cc3c(C)nn(C)c3)=O)COCCC1CN(C(c1cc(Cl)cs1)=O)C2 c1(CC)nc(C)c(C(=O)NCc2ccc(C(=O)NCC(C)CC)cn2)o1.O N1(C(CCN(C)CC)=O)CC(CCNC(c2cc(C)c(Br)s2)=O)C(C)C1 Cc1nc(NC2CN(C(c3ccc(=O)n(O)c3)=O)CC2(C)C)cc(C#N)n1 Cc1cnc(C(N2CCOC(C(C)NC(C3(CCO)CC3)=O)C2)=O)cc1C NS(=O)(=O)C1(C(N2CCN(C3CN(C(c4cnc(OC)cn4)=O)C3)CC2)=O)CC1 C(=O)(CCCCCCCN)N1CC(CCC)C1 C1(C(=O)Nc2ccc[n+]([O-])c2)CN(c2ccnc(N3CCCC3)n2)CCC1O C1(NC(C2CC(C)C2)=O)CCC(NC(C2CCCC(CC(F)(F)F)C2)=O)CC1 C(=O)C(C)CC(C)(C)C.C12(CNC(c3ccc(C(C)C)o3)=O)CC(CO1)C2 C#Cc1cc(NC(C2CCCN3CCCC23)=O)ccc1Cl N1(C(C(C2COCC2(C)C)C)=O)CCN(C(c2cn3ccnc3s2)=O)C(CO)C1 c1(OC)cc(CNC2CC2C(=O)Nc2cnc(I)c(Cl)n2)cc(C)c1 C1(NC(C(=CC2CCCC2)C)=O)CC2CCC1CN2C(C1(C)CC2CCC1C2)=O O=C(CC(C(F)F)NC(c1ccc(F)cc1)=O)NCC(Cl)=CCl C1(C)(C(N(CCCCN(C)C)C)=O)CN(C(C2CCOC2CCC)=O)C(C)(C)C1 N1(C(C=CCCC)=O)C2CCC1CC(CC(C)NC(c1cncn1C(C)C)=O)C2 C1(NC(c2c(CC)ccs2)=O)CCCCC12CCN(C(=O)C(C)(F)F)C2 Cn1ccc2c(c1=O)CN(S(=O)(=O)c1cccc(N3CCOCC3)c1)CC2 N1(C(c2cn(CCC=C)nn2)=O)CCCC(CO)(NC(=O)C(F)CCC)C1 CCC(CC)(CC)C(=O)NC(C)CCCNC(=O)COc1cccc(Cl)c1 c1(N2CC(C)C(F)C2)[nH]c(=NCCC2CCCS2(=O)=O)nc2c1cnn2C CCC(C)CCC(O)CC(=O)NCC(CNC(c1cccc(NCC)c1)=O)OC N1(C(C=CCCC)=O)C2CCC(C2)C1CC(=O)NC(CCOC)C(N)=O C1(NC(C=CCCC)=O)COC2(CCN(C(=O)CC3CCC(OC)CC3)C2)C1 C=C(Cl)C(C)(C)C(=O)N(CCCNC(=O)CCC1(C)CCC(=O)N1)CC c1(C(N(CC(C)(C)NC(C(C)O)=O)C)=O)cc(F)cc([N+](=O)[O-])c1Br C12(CO)CCCC1CN(C(=S)NCc1ccc(F)cc1)C2 N1(C(CC(C)(O)C2CC2)=O)CC2(CCCN(C(C3COCCO3)=O)C2)C1 C1(C(=O)NCc2n(CC)cnn2)C2CC1N(C(=O)CCCNC=O)C2.O C1(NC(c2nnn(CC)c2C)=O)CN(C(=O)C(C)(O)CC(C)C)CC2CCCC12 c1(N2C(C)CN(C(=O)C(c3cncn3C)O)CC2)ncnc2c1cnn2C CC1(C)CCOC1CNC(=O)CCN(C(c1ccc[n+]([O-])c1)=O)C1CC1 N1(C(c2c(COC)cco2)=O)CCN2CCN(C(C3CCCSC3C)=O)CC2C1 C1(C(=O)OC)CN(N2CCC(c3nccn3C)C2)CC1C1CCCC1 c1(CN(C(C(N2CCOC2=O)C)=O)CC(O)CO)ccccc1 c1(C(=O)NCCNC(CCCc2ccc(C)cc2)=O)ccc(O)c(C)c1C c1(C(=O)OC)cccnc1NC(C1(F)CN(C(=O)C)C1)=O.c1cc(C)on1 C(=O)(CC(C)(C)C(=O)OC)N1C2(CNC(C=COCC)=O)CCC2CC1 C1(NC(c2c(C)coc2)=O)CCCCC1CNC1CCN(CC(F)(F)F)C1=O CC(C)(C)C(CC(=O)NCCN(C(=O)C)C1CC1)C(F)F.c1ccncc1.O N1(C(c2n(C)nnc2)=O)CC(NC(c2occ3c2CCC3)=O)C(C)(C)C1 CCCC(C(=O)OC)C(=O)NC(c1cn(C)nn1)C(=O)NCC=C(Cl)Cl C1(C(C)C)CCOC1C(N1CC(C(O)C(=O)N)C1)=O.C1(CC2CCC2)CCC1 c1(OC)ccn2ccnc2c1C(=O)NC1CC(CO)N(C(c2cnsc2C)=O)C1 C#CCC(C)(CC)C(=O)N1Cc2occ(C(=O)NC(c3nncn3C)C)c2C1 C1(C)(CNC(C(C)N(C)C)=O)CCCN1C(=O)CN1CCCNC1=O c1(OCC(N2C(CNC(=O)CCCCC3CC3)CC2)=O)ccc(F)cc1Cl N1(C(CCOCC)=O)CCC(C(=O)NCC(C)(O)C(=O)OC)C(O)C1 N(C(=NCC(C)N1CCOC1=O)N(C)Cc1ccc[nH]1)C(CC)C c1(C(C(=O)NC(CCC)CNC(c2cc(C(C)=O)c[nH]2)=O)C)cc(C)oc1C CC1CC(C(=O)NC)CCC1C.C(=O)(C1=NNC(C(F)(F)F)C1)N1CCC(O)C1 CCCCCC(C)(CC)C(=O)NC1CN(C(=O)Cc2cccc(C)c2F)CC1C Cc1ccnc(C)c1-n1cc(C2CCCCN2C(=O)CC2CC3(CCC3)C2)nn1 Brc1cc2c(C(c3nnnn3CC3CC3)NCC3CSC3)ccnc2[nH]1 c1(C(=O)NC2C(CNC(CCC3N(C)CCC3)=O)C2)cccc(CO)n1 C1(N(C(=O)CN(C(c2cc[nH]n2)=O)C2CC2)CC)CCNCC1.C1CC1 N1(C(C(CCCC)O)=O)CCC2CCC(C1)N2C(c1scc(Cl)c1Cl)=O N1(C(C(C=C)C)=O)CCN(C(c2ccc(Cl)o2)=O)C(c2cn[nH]c2)C1 C1(C=O)CCS(=O)(=O)N1.C1(C(=O)N)CCCN(CC)C1.C1(=CC)CCCC1 C1(CCN(C(C(C)Cn2ccnc2)=O)C)CCCCN1C(c1cccc(O)n1)=O c1(C(=O)OCCCOC(C)C2CC2)ncoc1C1CCCO1 Nc1c(C(N2CC3CC3(NC(C3CCCC(F)(F)CC3)=O)C2)=O)ccc(F)c1F CCC(CC)C(C)NC(N1CCCC1(CC)COC)=O c1(C(=O)N)cc(Cl)c(F)cc1O.c1(C(C(=O)NCCC)C)ccc(C(F)F)cc1 C(C(C(C)C(C)C)NC(=O)C1=CC(C)(C)C1)NC(CCC(=O)NCC)=O c1(C(N(CCC)CC)=O)csc(N=S(C)(C)=O)n1.C(=O)C(C)n1cnnn1.N C(=O)(C1=CNS(=O)(=O)N=C1C)N.N1(C(CCC(C)=O)=O)CCC2(COC(C)C2)C1 c1(COC(C(c2c(C)nc(CC)s2)(C)C)=O)ccc(OC)cc1S(C)(=O)=O N(C1CCc2cccnc21)C(C1(C)CC(NC(=O)CCOC2CC2)C1)=O c1(C(=O)N)cn2c(C)cccc2n1.C1(NC(CCC2CC(OC)C2)=O)CC(C)C1 C(=O)(CCC(O)C(C)(C)C)N1C(CC)CN(C(c2cc(F)c(N)cc2F)=O)CC1 c1(C(=O)NCCN(C(=O)C(C)(CC)CCC)CCC)cn2cccc(C)c2n1 Cc1nc(C2CCCO2)sc1C(N1CC(C)C1)=O.c1(C=O)cc(C(N)=O)no1.N C(CC(C(=O)NC12CCN(CC1)C2)NC(=O)CSc1ccccn1)OC N1(C(c2cnn(CC)c2Br)=O)CCN(C(c2cc(C)on2)=O)C(CO)C1 c1(C(=O)NC2CCC(CCNC(c3cnn(C)n3)=O)C2)cc(C(F)F)ccn1 n1(C2CC(NC(=O)C(Cl)Cl)C2)cc(CN2CC3CC3C2)nn1 c1(N(C2CCC2)C=O)cc2c(cc1Br)CCN2.Cc1cc(C)n(C)n1.C(C)(C)C N1(Cc2scc(-c3cn(C(c4c(C)cccc4)C)nn3)n2)CCc2ccccc21 Cc1cccc(C(N2CCCC(O)(CNC(C3(C)CC(O)CN3C)=O)C2)=O)c1O c1(NC(=O)C(Cl)Cl)nc(C(F)(F)F)ccc1C(=O)N(CCO)C1CC1 c1(C(C)OC)ncc(C(=O)NCC2CCC2)s1.c1(CC(=O)N)c[nH]nc1C CC1CN(C(=O)CCc2ccc(Br)cc2Cl)CCC1CO c1(C(N2CC(OC)C(NC(c3cc(C)n(C)n3)=O)C2)=O)ccc(Cl)cc1I c1(C(=O)NC2CCC2NC(C2Cc3cscc3C2)=O)ccc(F)c(Cl)c1F c1(C(=O)NC2CC3CN(C(C(C)(Cl)Cl)=O)CC2C3)ccnc2ccncc12 c1(C(N2CCC(c3nnc(C(=O)OCC)s3)C2)=O)c(Cl)ccc(Br)c1F CC(CC(=O)N1CC(N(C(=O)Cc2c[nH]c3cccc(F)c23)C)C1)CC(F)(F)F C=CCN=c1[nH]cc(C(N2CC(c3ccccc3)C(O)C2)=O)s1 N1(C(C=CC=CCC)=O)CCC(N(C)C(c2cncc(C)n2)=O)C(C)C1 c1(OC)cc(C(=O)NC)cnc1C.C1CC(O)CN1C(=O)C=CC(C)(C)C N1(C(CC2(C)CCN(C(c3c(C)scc3)=O)C2)=O)CC2(CCOCC2)C1 c1(CN(CC(=O)NC(CC)COC)C)ccc(Cl)c(Cl)c1 c1(C(=O)NCC(=O)N)csc(CC(F)(F)F)n1.c1(C2CC2)cn(CCO)nn1 Cc1nc(N2CCCC2C(=O)Nc2cc(Br)ccc2CO)nc(C)c1Br C1(OC)CC(NC(=O)CC2CCCCN2C)CN(C(c2ccc(C#N)cn2)=O)C1 C1(CC(=O)NC2CN(C(=O)COC)C2)CNC(=O)O1.C1(CCO)CCCC1 c1(C(=O)NC2CN(C(C3CC(C#C)(O)C3)=O)CC2C)ccc2n[nH]cc2c1Cl C=CCC(C(=O)N1CCC(=CCNC(=O)CCSc2ccccn2)CC1)N(C)C n1(CCNC(C(C)C2CCCC2)=O)cc(CNC(=O)OC)nn1.c1cncnc1 C1(NC(C2CC(OCC)C2)=O)CC(C(=O)NC2COCCOC2)C12CCC2 C1(NC(c2csc(=N)[nH]2)=O)CN(C(=O)CO)C2(CCOCC2)C1.c1ccccc1 c1(C(N2CCCCC(N(C)C)C2)C(=O)OCC)ccc2nc(C)[nH]c2c1.C1CN1 c1(C2CC(=C)C2)cn(CC(C)NC(=O)C(C)(C)C2CCCO2)nn1 C1(NC(C(C)OCCCCCC)=O)CC2CCC(C1)N2C(c1cc(CC)[nH]n1)=O c1(OC)cc(C(=O)NC2CC(CO)N(C(c3cc(C)ns3)=O)C2)cc(F)c1C#N C1(NC(c2cc(C)sn2)=O)CC(C)CN(C(=O)C(C)Oc2cccnc2)C1 C(=O)(C1=CCCC1C)N1CCC(O)(C(C)NC(c2ccno2)=O)C1.C1CC1.N c1(C(c2nnnn2C(C)C=O)NCc2cn(CC)nn2)cn(C)c(=O)n1C N1(C(Cc2c(C)n(C)cn2)=O)CCN(C(c2cnc(C(C)C)[nH]2)=O)C(C)CC1C S(=O)(=O)(c1ccc2sc(Cl)nc2c1)NC(C(CC(C)C)OC)=O C(C(=O)N1CCC(C(N2CC=C(C(C)(C)C)CC2)=O)O1)(C1CC1)OC C1(NC(c2cccc(OC)c2)=O)CCN(C(=O)C(=O)NC2CC2)CCC1CO CC(C)C(C)C(=O)NCc1ccc(CN(C)C(C2CNC(=O)N2)=O)cc1 c1(OC)cc(C=CC(N2CC3CC2CC3NC(c2cncs2)=O)=O)ccc1F c1(OCC)cnc(C(=O)Nc2ccncc2F)c(Cl)c1 C(=O)(C(C)S(N)(=O)=O)NCCC(C)NC(CCC(C)N(C)C)=O CCCCC(C(=O)NC1CC(OCC(=O)N)C1)C(C)C.C1OC(=O)NC1(C)C.C c1(N(CC(COC)(F)F)C)nc(=NC2CCS(=O)(=O)C(C)C2)[nH]c2c1CSC2 N1(C(C)=O)CC2CCC1CN(C(=O)Cc1ccnc(Br)c1)C2.C1CO1 Cc1cc(Cl)cc([N+](=O)[O-])c1C(=O)NC(=O)CCCCCO C1(C(N(C2CCCC2)CCC)=O)CCCC(C)(C)O1.C#CCCN(CC(=O)N)C CC(CN(C)C)CCC(=O)N1CCC(CO)(NC(c2cc(C(N)=O)[nH]n2)=O)C1 c1(C(C)(F)F)ccc(C(N2CCC(CCNC(=O)CC3CC3)C2)=O)nc1 N1(C(CN(c2ccccc2)C)=O)C2CCC1CN(C(c1cccn(C)c1=O)=O)C2 C(=O)(C(F)C(F)(F)F)N1CCC(CN(C(C2C(C(=O)OC)C2)=O)C)C1 c1(C2(C(N3CC(NC(C(C)n4ccnc4)=O)C3)=O)CC2)cccnc1 C1(C(N2CC(OC)(C)C2)=O)CCCC2(CCOC2)O1.c1(C=O)cc(C#N)c[nH]1.N n1(N(C)C)cnc2cc(NC(c3nnnn3C3COC3)C3CCC3)ccc12 C1(C(=O)NC(CCSC)CO)CNCCC12CCC2 C1(CC=O)CN(C(c2ccc(C#N)s2)=O)CC1O.C1(C(=O)OC)(C)CC1.N N1(C(c2nc(CC)oc2C)=O)CC(NC(=O)C=CC2CCCCC2)CCC(O)C1 C1(NC(C(N2C3(CC(C(=O)OC)C3)CC2)=O)=O)CCCC2(CCOCC2)O1 c1(OC)cccc(N2CCN(C(=O)C(=O)NCC3COCC3N(C)C)CC2)c1 c1(CCNC(=O)NC(CSC)C(=O)O)cccc(Br)c1O CC1(C)CC(C(=O)NCC(C2CCCCC2)NC(c2cnns2)=O)C1 CC(CC(=O)N(CCC(c1cccs1)NC(=O)C(O)C1CC1)C)n1cccn1 CC1CC(NC(=O)CC2CCSCC2)CN1C(=O)CCOCC(C)(C)C C(c1ccc(S(C)(=O)=O)o1)=CC(=O)NC1CN(C(CC(CCC)O)=O)CC(O)C1 N1(Cc2c(C)cccn2)CC2CN(C(=O)Cc3cccc(F)c3I)CC2C1 C(=O)(CN=S(C)(C)=O)N(C)CCn1cc(COC(=N)O)nn1 C1(CNC(C2=NOC(C)C2)=O)CC2(CCC2)CN1C(=O)C=Cc1cncnc1O O=C(C(F)(F)c1ccncc1)N1CC2(CC2)C1 c1(CNC(CCC2(C)CN(C(C3CCC(CC)O3)=O)C2)=O)ccc(C)c(F)c1 C(=O)(C#CC1CCOCC1)N(C1C(C)CN(C(c2cnc(Cl)s2)=O)CC1)C c1(SC)ccc(C(=O)NC(C)C(CO)NC(C2CCC23CCC3)=O)c(Cl)c1 Cc1cc(F)ccc1CC(N1CC(OCCNC(=O)C(O)c2ccsc2)C1)=O c1(C(N(CCNC(CSc2ccc(C)cc2)=O)C)=O)noc2c1CCCC2 C(=O)(C(O)C(F)(F)F)N.C1(C=O)CCCCN1C(=O)C(C)(C)C.CC1CCC1 C1(CC)CCCC(N=c2ccnc(NC3CC(C)n4ncnc43)[nH]2)C1 c1(C(C=C)OC)ccc(NC(c2ccccc2Nc2ccccc2)CO)cc1 C(C(N=c1nc[nH]n2c(Br)ccc12)c1ccncc1)NC(=O)OC(C)(C)C C(=O)(C1=CNC2=NCCCC2=C1)N(C)CC.c1(C(=O)N)cc(OC(F)F)n(C)n1 c1(NC(C2CC(CCNC(CN(CC(C)(C)C)C)=O)C2)=O)cccc(Cl)c1 S(=O)(=O)(c1cccc2nc(O)oc12)NC1(CO)C(C)(C)OCC1 n1(C2(CNC(N3CC(O)CC(C)C3)=O)CCOCC2)cnc2ccccc12 C1(C(=O)NC(c2nc(C(=O)NCC#CCCO)co2)C)CCCC(C)CC1 CCC(CCCC(=O)NC1CCOCC1)NC(C1CC(C2CC2)C1)=O N1(C(C23N(C(c4ccc(=N)[nH]n4)=O)CCC2C3)=O)CC2CCCC1C2CO Cc1c(C(C(=O)O)NC(=O)NCCC2CCCOC2)sc2ccccc12 C1(C(=O)NCCC2(C(=O)NCC(CC)n3cccn3)CCC2)CC2CC2C1 N1(C(c2ccccc2-c2ncc[nH]2)=O)CCN(C(C2(Br)CC2)=O)CC(O)C1 C1(C(N2C(C3(NC(CC(CC)O)=O)CC3)CCC2)=O)CCC(=O)N(CC)C1 C(=O)(C(O)CC[S+](C)C)N1CCC(N(C)C(C2CC2c2ccoc2)=O)CC1 C1(NC(C2C(C(C)(C)C)CC2)=O)COC2CN(C(c3snc(Cl)c3Cl)=O)CC12 c1(OC(C(=O)NCC(CC)NC(=O)C)C)ccc(OC)cc1.CC(C)(C)C c1(C(=O)NC2CCN(C(C3CC34CCCC4)=O)C2)cnc2cc[nH]c2c1 N1(C(c2cc(COC)ncc2)=O)CCC(C)C(C)C1.c1(CC=O)cc(C)no1 c1(N2CC(C)OC(C(N)=O)C2)ccc(S(=O)(=O)NCC(C)(C)F)c(Br)c1 CC1CCc2c(C(=O)NC(C3CN(C(=O)CC(O)C4CC4)C3)C)csc2C1 N1(C(C2CN(C(C#CC(C)(C)C)=O)CC(C)(C)C2)=O)CCc2ccc(F)cc21 N1(C(C2(NC(CCC(C)(C)F)=O)CC(F)C2)=O)CCCC2(CC1)CC2 N1(C(CC(=O)NCC#C)=O)CCC2(C1)CN(C(c1cccc(F)n1)=O)CC(C)O2 c1(C(N2C(CNC(C3(CF)CC3)=O)CC(OC)C2)=O)onc2c1CCCC2 N1(C(C2CCC(=O)C2)=O)CCC2CN(C(c3cccc([N+](=O)[O-])c3)=O)CCC2C1 C(c1ccccn1)=C(C)C(=O)NC1CCC1C.C(=O)(C(C)(O)c1ccccc1)N CC1C2CC(C2NC(=O)COC2CCCCC2)N1C(=O)CCC#N C1C2CN(C(=O)C)CC12.c1(CC=O)cccc(F)c1.C(=O)C=CC=O.C C12(CCNC(C(C)(C)C)=O)CCC1CN(C(=O)Cc1ccccc1F)C2 C1(CCNC(CCC2CCC(C)O2)=O)CCN(C(=O)CCC2CC2)CCC1(F)F N1(C(C(C)Sc2ccc(Cl)cc2)=O)CCC2(CC2)C1.C(=O)(C(F)=CC1CC1)N N1(Cc2c(S(C)(=O)=O)ccs2)CCC2CCC(C1)N2C(=O)CCc1ccccc1 c1(C(=O)NCC2N(C(C(C(C)C)SC)=O)CCCCC2)cncc2[nH]ccc12 N1(C(=O)NCc2c(OC)ccc(Cl)c2)CCc2ccc(C#N)cc21 N1(C(c2cc(C)n(C)n2)=O)CCCC(F)(C(=O)N(C)Cc2nccs2)C1 N1(C(C(CC(C)C)C)=O)CCCN(C(=O)CCc2nc[nH]n2)CC1C C1(C(=O)NC)(CCNC(COCC#C)=O)CCC1.C(CC)NC=O.O CN=c1[nH]c(=NCCCOC)[nH]c(=NC2CCOC3(CCOC3)C2)[nH]1 CC1CC(=O)CCC1C(N1CCC(F)(C(=O)NCC2CC3C=CC2O3)CC1)=O c1(C(=O)NCCC2CC(OC)CN2C(=O)CC)ccn2c1CSCC2.C(C)C.O C1(N(C(C(C2CN(C(CCn3c(C)ncc3)=O)C2)O)=O)C)CCCC1(F)F C1CN(C(=O)Cc2cnn(C(C)C)c2)CC12CC2.Cc1ccsc1CC(=O)NC C(CN=c1[nH]c2ccc(O)cc2s1)(C(C)(C)C)NC(CC1(C)CC1(Cl)Cl)=O C(C(C)C(C)C(=O)NC1C=CCN(C(C23CCC(F)(CC2)C3)=O)C1)OC N1(C(c2cn(CCC)nn2)=O)CCN(C(c2cc(C)cc(O)n2)=O)CC(C)(C)C1 C(=O)(C1=C(Cl)CCC(C)C1)NCC(N(C(Cc1c(C)noc1C)=O)C)C1CC1 C1(CC(=O)NCC2(OC)CC2)CCCC1.C(=O)(C(C)(O)C1CCCC1)N N1(C(c2cc(CSCC)on2)=O)C2CCC1CC2.c1(C=O)cnn(C)c1C.C C1(C(N(CCCNC(=O)CC2CCOC2)CCO)=O)CCn2c(O)nnc2C1 C(N=c1[nH]cnc(Cl)c1OC)C1(C)CCN(C(CC2CC(OCC)C2)=O)C1 CCC(C(=O)OC)C(=O)NCC1(C(=O)NCC(C)CC2CC2)CCC1 c1(C(N2CCCC(CCNC(c3cscn3)=O)C2)=O)cc2ccccc2o1 N1(C(C(CC=C)NC(C)=O)=O)CC2(CCC(NC(=O)C(C)CC(F)F)CC2)C1 C1(N(C(CC2(C=C)CC2)=O)CCO)CCN(C(=O)CCCc2nncn2C)C1 CCCCC(=O)C(=O)N(CCC(C)NC(=O)C1=C(C)OCC1)C N1(C(CC)=O)CCCC(C(=O)NCC2CCCCN2C(=O)Cc2cnc(C)[nH]2)C1 C=C1CCC(CNC(=O)CCN(C(C2CCCOC2)=O)CC)CC1 Cc1nnc2c(C(=O)NCC(O)CNC(=O)CC)cccn12.C(=O)CC(C)C.N c1(C(N2C(C(=O)Nc3nccc(C)c3F)CCC2)=O)cccc2c1OCC(=O)N2 Cc1cccc(Cl)c1CC(=O)Nc1nnn(C)n1 N1(C(C2(COC)CCCO2)=O)CCC2(CC1)CC2.C1(CC=O)C=CCCC1.C C(=O)(C(CCCC(C)(F)F)N1CCC(C)C1C)NCCCCCC C1(C(N(C)CC)=O)CCC2(CC2)N1C(=O)CCCC(OC)OC c1(N2CCC(N(CC#C)C(c3cnnn3C)=O)CC2)cc(O)nc(O)n1 c1(CC(N2CCC2)=O)cn2c(n1)CCCC2.C1(C(=O)N)CC2(CCOCC2)C1.C O=C(CCCN1CCCC1)NCCCC1CCCN1C(=O)NC12CC3CC1C2C3 C1(C(=O)NC2CCC(CNC(C(CSC)C)=O)C2)CC2CC1C1CC21 C=CC(C)(CC)C(=O)NCc1cc(O)nc(CNC(C2CC=CCC2C)=O)n1 C1(C)(NC(C2(C(C)C)CCC2)=O)CCCN(Cc2ccsc2)C1 CCS(=O)CC(=O)NC1(C)CCN(C(=O)CNc2ccc(C(N)=O)cc2)C1 C(=O)(CC(C)(C)C)N1CCC(N(C(C(C2(O)CCCCC2)C)=O)CC2CC2)C1 C1(CNC(Cc2cc(C)on2)=O)CCN(C(=O)CS(N)(=O)=O)CC1C1CC1 CC1CN(C(=O)C(O)C2CC2)CC1n1cc(CNC(N)=O)nn1 CC1(c2ccccc2)CN(CC(c2ccccc2)O)CCO1.c1(C=O)cccs1 C(=O)(C1c2ccccc2CCN1C(c1cc(Br)co1)=O)N(C)C C1(C(N2CC(OCC#C)C2)=O)CC2(CCN1C(=O)CC13CCCC1C3)CC2 CC1CN(C)CC(C(=O)NC2(C)CCCC2)O1.c1(C=O)cn(C2CCC2)nn1.N C1(NC(CC(C=C)(C)C)=O)C(CNC(=O)C)CCC12CCC2.C1CC=CC1.O CC(CC(=O)NC1CC(N(C)C(c2cc(F)c[nH]2)=O)C1)c1cccnc1 C=CCC(CNC(=O)C=Cc1cncs1)C(=O)Nc1cnsc1 N1(C(Cc2cc(CC)no2)=O)CCCC(O)C1.c1(CC(=O)N)cc(C(C)C)no1 c1(NC(C)=O)cccc(CNC)c1.C1(CC(=O)NC)CNC(C(F)(F)F)CO1 C1(N(C(C2CC(SC)C2)=O)C)CCCN(C(=O)CCC(C)c2ccccc2)C1 c1(OC)ccncc1CNC(C1CN(C(=O)C(C)C2CC2)CC1C)=O c1(C(=O)N)c[nH]c2ncccc12.C1(C(N)=O)CCC(C(=O)NC2CC(CC)C2)C1 C(=O)CN=c1ccc(Cl)n[nH]1.N1(C(C2(C)CC(C(F)(F)F)C2)=O)CC(C)C(O)C1 c1(C(C)C)cccc(S(=O)(=O)NC2CCN(C(c3cc[nH]c3)=O)CC2O)c1 c1(C(N(C2CCN(C(C3CCSC(C)C3)=O)CC2)CC#C)=O)ccc(C)nc1 Cc1c(CNC2CC2C(=O)Nc2cc(Cl)nc(Cl)c2)cccc1F Cc1c(C(=O)NCC2CCN(C(=O)C(C)O)CCC2(F)F)sc2cccc(F)c12 C(CCC1CC1)(C(=O)N1CCCCC1CF)NC(C=CC1(C)COC1)=O c1(C(=O)NC(CNC(c2c(C(C)C)ccc(C)c2)=O)C)c[nH]c2nc(F)ccc12 c1(OC)cc(Cl)c(C)cc1C(=O)NC1CC(C)CN(C(=O)CC2CCCOC2)C1 Cc1c(C(=O)N(CC(C)NC(C2(C)CCC(=O)C2)=O)C)cccc1[N+](=O)[O-] N1(C(CCCCC)=O)CC(C2CCCCN(C(C3CS(=O)(=O)C3)=O)C2)C1.C(N)(=O)N C(c1cccc2cccnc12)=CC(=O)NC1C(NC(C(CCC)CC)=O)COC1 N1(C(C(CCC)OC)=O)CCCC(C)(C)C1CNC(c1cc(O)nc(NC)n1)=O CCC(CC)C(=O)NCC(=O)NC1CCN(C(c2cc(C(F)F)nn2C)=O)C1 N=c1[nH]cncc1C(N1CC2C(C(=O)NCC34CC(CO)(CO3)C4)C2C1)=O C(C1=CCC2CC1C2(C)C)NC(c1cc(OC(C)C)nc(Cl)c1)=O N1(C(c2cc(C)c3c(c2)CCCN3)=O)CC2C3CCC(CC3)C2C1 c1(C(=O)NCC2N(C(CS(CCC)(=O)=O)=O)CCC2C)cccc2nc(C)nn12 C1(NC(c2ccc(C#N)s2)=O)CCCCCC1NC(c1ccc[nH]1)=O c1(C(N2C3CC(NC(c4c(C)ccs4)=O)C(C3)C2)=O)cccc2c1NC(=O)C2=O c1(C(=O)NC2CC3(CN(C(CC(CC)SC)=O)C3)C2)ccc2c(c1)C(=O)NC2=O N1(CCn2c(CC)ncc2)CC2CC1CN2CC(C)O C1(C(=O)NC2CCCCC2)C=CCN1C(c1ccc(-c2nn[nH]n2)s1)=O N1(C(c2c(SCC)nccn2)=O)CCN(C(c2c(Cl)ccnc2C)=O)CC1C C(=O)(C1=NOCC1)N(CCCNC(CCCN(C)C)=O)C1CC1 C12(C(=O)NC(CC)C(C)(F)F)CC(C)(CN1C(=O)CN1CC3CC3C1)C2 c1(CCC)ccc(S(=O)(=O)N2CC(F)(C(=O)Nc3cc4nccn4cn3)C2)cc1 C=C(F)C1(CC(=O)NC(C)(CNC(C2CC(C)(CC)C2)=O)CC)CCC1 C1(CC(=O)NC2(CCF)CCC2)CC2(CCC2)CN1C(C1CCOC1)=O C1(C(N2CCC(N(C(c3ccc(CC)cc3N)=O)C)C2)=O)CC2CCC(C1)C2O CCC(O)C(C)NC(=O)C(N1CCC(C(=O)O)C1)=O c1(C(=O)NCCC(C)NC(c2cccnc2C(F)F)=O)sc2ncccc2c1Cl Cc1cc(C(N2CCCC(N3CCCC3=O)CC2)C(=O)NC(C)(C)C)nnc1C C(=O)(C1=C(Cl)CCC1)NC1C(C)N(C(=O)CCSC(F)(F)F)CC1 CC(C)C(C)CC(=O)N1CCC(CN(C)C(c2cnc[nH]2)=O)C1 C(=O)(C1COc2ccc(F)cc21)N(C)CCNC(C1CCC1(C)C)=O Cc1cnc(NC(CNC(c2ccccc2)=O)C(C)C(C)C)nc1C Cc1cc(C(N2CCC(=CC)CC2)=O)c[nH]c1=N.N1(CC=CC=O)CCCC1.N N1(C(c2ccn(CCNC(C(CCOC)C)=O)c2)=O)CC2CC(C)(C)C2C1 C1(C(C)(C)C)(CNC(c2cc(O)no2)=O)CCN(C(C2CC3CCCC23)=O)C1 Cc1csc(C=O)c1.CC(F)(F)F.C(CCN(C)C)N(C(=O)C=C)CC N1(C(CSc2nc(C)[nH]n2)=O)CCC2(CCN(C(=O)C(C)(C)CC3CC3)C2)C1 c1(C(C(N2C(C)CC(OC)C2)=O)C)ccc(C#N)cc1.c1(C=O)ccc(F)s1.N C(C)(c1ccccc1F)=CC(=O)N.C1(OC)CCCN(C(=O)CC(=O)N(C)C)C1 C1(CC=C)CCCCC1NC(=O)CCOC1CN(C(c2ccns2)=O)C1 NS(=O)(=O)c1cc(C(N2CCCCCC2CNC(c2cc(C)on2)=O)=O)co1 C(=O)(CC(C(F)(F)F)OC)N1CC(C2OCCN(C(C(C(CC)C)O)=O)C2)C1 CC1N(C(=O)CCCn2cc(CCCC(C)O)nn2)CCC1(C)C C12(CNC(c3cnn(CC)c3)=O)CCC(CO1)C2.C1(F)(C=O)CC=CCC1 N1(C(C2C(OC)CC2)=O)CCN(C(=O)Cn2nc(C)oc2=O)CC(CO)C1 c1(C(=O)O)cccc(N2CCN(C(=O)CC3COC3)CC2)n1 c1(N(CCCOC)C)nc2cc[nH]c2c(=NC2CC2c2cccc(C)c2)[nH]1 n1(CC)nc(C)cc1C(N1CCC1c1ccccc1)C C1(C(N(C2CCN(C(=O)C(C)C)CC2)CC)=O)CC(=O)NC1(C)C.CCO C1(C(N(C)CC2(NC(CCNC(COC)=O)=O)CC2)=O)CC2CCC1C2 c1(OC)ccc(C(=O)NCC(n2cc(-c3cccnc3)nn2)C)c(F)c1F C1(NC(c2nc(CCC)oc2)=O)CN(C(c2cnc(S)nc2)=O)CC1(C)C N1(C(C2(C)CC=CC2)=O)CCC(C2CCN(C(=O)CCc3ccon3)CC2)C1 N1(C(C=C(CCC)C)=O)CCN(C(c2scc3c2OCCO3)=O)C(C)CC1C C1(CNC(CC#N)=O)CC(NC(=O)CC2CCCC2O)C12CCC2 C(CC(=O)NNC(=O)Cc1ccc(Cl)cc1)SCC(=O)NC1CCCC2(CNC2)O1 C(=O)CCP(C)(C)=O.c1(CCNC(c2c(CCC)nco2)=O)ccc(F)cc1.N CC1CC2(CCC2)CN1Cc1ccc(Oc2ccccc2)c(Cl)c1 C1(N(C)C)(C(N2CCC(C)C2)=O)CCCCC1.c1(C=O)ncoc1C(F)(F)F.N N1(C(C(c2ccc(C)cc2)C(C)C)=O)CCC(CO)(NC(C2CCCO2)=O)CC1 N1(C(C(C(C)O)C)=O)CC2CCC(NC(=O)C(c3cnccn3)C)CC2C1 CC1SCCCC1C(=O)NC(C)(C)CN(C)C(c1nccn1C)=O c1(C(N2C(C)CC(NC(CN3C(C)CCC3)=O)C2)=O)cc(F)c(F)c(F)c1 c1(C(=O)NC(c2ccc(S(N)(=O)=O)cc2)C)nccc2ccccc12 C(=O)(CN=c1ccc(Cl)n[nH]1)N1CCC(C(C)NC(CNS(NC)(=O)=O)=O)C1 C1(O)(CN(C(=O)C(C)(C)C)C)CN(C(=O)Cc2coc(C(F)F)n2)C1 N1(C(C23CC(CSC)(OC2)C3)=O)CC2(CCN(C(=O)C(C)C(C)C)CC2)C1 Cc1nc(C(=O)NC2CC(F)CN(C(=O)CC(C)C)C2)cc(O)n1 N1(C(C(=O)NCC(=C)C)CCC=C(C)C)CCC(SC)CC12CC2 N1(C(C(CC=C)CC)=O)C(C)CC2CN(C(=O)C(CC3CC3)CC3CC3)CC12 C(=O)(C(CO)C(C)C)NCCC(C(C)C)NC(C1(O)CC1)=O CCCC(C(=O)NC1CCN(C(=O)CN2CC(C)(C)C2)CC1CO)S(N)(=O)=O N1(CCC(=O)OC)CCC(C)(CNC(C2CCC(CN(C)C)CC2)=O)CC1 N1(C(c2csc(Cl)n2)=O)CCC(CNC(C2(c3cncs3)CC2)=O)C12CC2 C1(S(C)(=O)=O)(C(=O)NCC=CCNC(C2C(C)OCC2)=O)CCOCC1 Cc1cccc(C(=O)NC(C(=O)NCc2ncoc2C)c2ccoc2)c1C#N N1(C(c2cc(C)[nH]c2)=O)CCC(C(=O)NCC2CCC(F)(F)CC2)C(O)C1 C1(NC(CNC(=O)NC)=O)CCCN(C(=O)C(C)CCc2ccc(F)cc2)C1C c1(C(N(CCCN(C(C2CCC(C#C)CC2)=O)C)C)=O)c(F)cc(C)cc1Cl c1(OC)ncc(C(=O)NC2CCN(C(c3cc(C(C)=O)[nH]n3)=O)CC2F)cc1F c1(C(=O)NC2(C(N(CC(COC)O)C)=O)CSC2)cc(O)ncn1 CCCCC(=O)N(C(C)CN(C)C(c1ccc(Cl)s1)=O)C.C=CCOC=O.N C1(CNC(c2ccc(OC)cn2)=O)CN(C)CCN1C(C1CN2CCN1CC2)=O C(CC(=O)NCC1CCC1)OCCOC.C1(C)C=CC(=O)N1 N1(C(CSCC)=O)CCC2(CCN(Cc3cc(Cl)c(Cl)cc3F)CC2)C1 N1(C(c2nccc(OC)c2)=O)CC(CNC(=O)CCn2ccnc2)CC(C)C1 N1(C(=O)Nc2ccc3c(c2)C(=O)CCO3)CCCc2c(Br)cccc21 c1(C(N(CCN(C(c2c(C)nco2)=O)C)C(C)C)=O)nc2c(Br)cccn2n1 c1(C(CNC(=O)CCc2ccc(Cl)s2)CO)ccccc1F N1(C(=O)OC)CC2C3CCC(C2C1)N(C(=O)C(F)(F)c1nccn1C(C)C)C3 C1(CC)CCN(C(c2cc(C(N)=O)[nH]n2)=O)C1C(=O)NCCC(C)(C)F C1(N(CC(=O)N(CC)C)C)CCS(=O)(=O)C1.C1(CC=O)(COC)CC1 C12(C(=O)NC3CCN(C(COC(C)=O)=O)CC3)CC3CC(C(=O)N1)C2C3 CC(C)(C(=O)N1CC(OCCNC(=O)CO)C1)c1cccnc1.C1CCC1 C1(C(=O)NCC2C(C)(C)CCO2)CN(C(=O)CC2CCC2)CC12CCC2 CC1(C)C(C(N2CCCC(CNC(C3(C)CCCC3(F)F)=O)CC2)=O)CC1(F)F c1(C2C(C(=O)NCC(C)N(C)C)C2)nccn1C.C12(CC1)CC(=O)N2 N1(CCCCNC(c2c(NC(C)=O)cc(Cl)cc2)=O)CCCc2ccccc21 C(C1CCCCCC1)=CC(=O)N(C)CC1CCCN(C(c2c(C)nn(C)c2)=O)C1 CCC(C(O)C(C)C)NC(=O)CC1(OC)CN(C(C2CCCCC(=O)N2)=O)C1 c1(C(N2CCCC(N(C(=O)CCc3ccc[nH]3)CCO)C2)=O)cnc2ccccn12 C1COCCN1C(=O)C=Cc1ccc(CN)o1.C1(=CC(=O)NC)CCCC1 C1(C(=O)NCCC(CNC(C2(C)CC(F)(F)C2)=O)OC)CCC=CCC1 c1(N(C)CC2CCCN(C)C2)ccc(S(=O)(=O)NCC(Cl)Cl)cc1Cl c1(C(=O)NC(CNC(c2ccnc(C)n2)=O)C)ccc(Cl)c2ccccc12 C1(C(N(C)CC2CCC(C)CC2)=O)CN(C(=O)CN2CCCC2=O)CC1(C)C CCCCC(CNC1CCCC(C(=O)O)CC1)CCC c1(COC)cc(C(N2CC(F)CC2)=O)n(C)c1.C(C(C)(C)C)=CC=O.C Cc1c(O)c(=O)ccn1CC(N1CCC(NC(C23CC(C2)C(C)O3)=O)C1)=O C(=O)(CCCCCCC(=O)N1CC(NC(c2cc(F)c[nH]2)=O)C1)OC CP(C)(=O)C(O)C(=O)NC1(CCNC(=O)COCC(F)F)CCCC1 C1(CNC(c2c(CC)cns2)=O)CCC2CN(C(=O)Cc3ccc(C)s3)CC12 C1(C(=O)N)CCn2cncc2C1.C1(OC)(C)CCN(C(=O)Cc2csc(Cl)c2)C1 N1(C(c2c(CC)n[nH]c2)=O)CC=CC(NC(=O)C(O)Cc2cnc[nH]2)C1 c1ccc(Cl)cc1.c1(OC)nc(C(=O)NCC)ns1.C(=O)(CC)N(CC)C.O C1(C(N(CCSC)C)=O)CCN(C(=O)Cc2cnns2)C1C c1(C(C2CC2)OC)cn(CCN2CCC(Oc3cccnc3)C2)nn1 C1(C(=O)NC(C(=O)OCCC)C)CC2(CCN1C(=O)COCC)CC2 c1(C(N2CCC(NC(C3(C)CCC3)=O)CC(O)C2)=O)nnc2ccccc2c1N c1(C(N(CCNC(CC(C(C(C)C)C)C)=O)C)=O)ccc2cc(F)c(F)cc2n1 C1(NC(c2ccc(F)c(C(F)F)c2)=O)COCCN(S(=O)(=O)C2CC2)C1 c1(CC(=O)N)csc(-c2ccoc2)n1.C(C)(C)(C1CCC1)NC(CN(C)C)=O C(CN=c1cccc(S(=O)(=O)NCCC(F)(F)F)[nH]1)c1c(C)nns1 c1(OC(C)C)ccsc1C(=O)NC1CCC1NC(=O)C(C)n1cccc1 c1(OC)cccc(C(=O)NC(C)CNC(C2CCOCC2(C)C)=O)c1C c1(-c2nc(-c3cccc(C)c3)nn2CC2(C)CCCC2)n[nH]c2c1CCCC2 c1(N(C2CC2C2CC=CC2)C)ccc(S(=O)(=O)N2C3CCCC2CC(O)C3)cc1F C1(N(C(CC)=O)C2CC2)CCN(C(=O)C(F)CC2CCCCC2)CC1.CC(C)C C1(NC(C2(CC=C)CC2)=O)CCN(C(=O)CCSc2ccccc2)C1(C)C C1(C(N2CCCC(CN(C(Cc3nc(C)oc3)=O)C)C2)=O)CCCC(F)(F)CC1 C(C1CN(C(=O)C(O)CN2CCCC2)CC1C(=O)N(CC(C)SC)C)=CC C1(NC(C2CCC3(CCC3)C2)=O)CC(O)CN(C(=O)COC2CCOCC2)C1 N1(C(C2CC3(C(OC)CC3)C2)=O)CCC2(CC1)CC2NC(C1CN(C)C1)=O N1(C(c2cc(CCC)ncc2)=O)C2CCC1CN(C(c1cc(Cl)no1)=O)C2 Cc1cc(Br)ccc1CC(N1CCCC(C)(C(N2CCSCC2)=O)C1)=O c1ccc(F)cc1F.C1(NC(C=C(C)C2CC2)=O)CCCC(NC(=O)C=O)C1.N c1(C(=O)NCCN(C(C(CCCC)O)=O)C)ccc2c(c1)C(=O)CCN2 CN=c1nc(N2CCCC(C)(CO)C2)[nH]c(N2Cc3ccccc3C2)n1 C1(C(=O)NC2CCC(F)CC2)(NC(CN(C(C(C)C)=O)C)=O)CCN(C)C1 C=C1Cn2c(C(=O)NC3(C)CCC(NC(=O)CC(CC)CC)CC3)nnc2S1 Cn1nnc2cc(CN3CCCC(C(O)C(F)(F)F)C3)ccc12 C=CCC(C)(CC)C(=O)N1CC(CC(C)NC(=O)COc2ccc(Cl)cn2)C1 C(=O)(C(F)C(C)(F)F)N(C)CC1N(C(c2ccn(CCC)n2)=O)CCC1 CC1Cc2cc(F)ccc2CN1C(=O)C(C1COC(C)(C)O1)O N1(C(C2C(C)CC2)=O)CC2(CC(NC(=O)CC3CCC4CC34)C2)C1 C1(CNC(c2c(C)c(Br)no2)=O)CC(F)(F)CN1C(C1CC1)=O.N(C)C C(CC(CC)C(=O)NC1CC1CNC(C1(C(N)=O)CC1)=O)=CC c1(Nc2c(C(=O)NCc3ccc(OCCBr)cc3)scc2)cccc(Cl)c1I.O C1(C2(O)CN(C(=O)C(C)C3CCCC3)C2)(CNC(CC(=C)Br)=O)CC1 c1(C(=O)NC2C3(CC(NC(CC(C)SC)=O)C3)C2)ccc(C)c(O)c1 C1(NC(c2cc(C)[nH]c2C)=O)CCN(C(c2sc(C)c(C)c2C)=O)C(C)C1 C(C)(CO)(C(=O)NCCCCN(C)C(c1coc(C2CCC2)n1)=O)NC(C)=O C1(N(C)C(c2cccs2)=O)CCCN(C(C2CS(=O)(=O)C2)=O)C1.C1CC1.C N1(C(CC2CC(=C)C2)=O)CCC(NC(c2scc(C)c2Br)=O)C1C1CC1 N1(C(CCOc2ccc(C)cc2)=O)CCC(NC(=O)CC(O)C(C)C)C(C)(C)C1 C1(OC)CCC2(C(N3CCCC3CNC(=O)C(C3CCC(=O)N3)C)=O)CC12 CCCCC(C)C(=O)NCC(F)(F)Cn1cc(C(C)(C)NC(N)=O)nn1 c1(C(=O)NCC(CN(C(C(C)NC(C)(C)C)=O)C)O)cnc2ccccn2c1=O C(=O)(C(C)C(O)CC(C)C)NC(CC)C(=O)NC(C)CNC(=O)C(C)C c1(CC)nnc(C)cc1C(N1CCC(C)C(CNC(C2CCCC2)=O)C1)=O.C C(=O)C1=CS(=O)(=O)CCC1.CC1CN(C(=O)Cc2cccc(Cl)c2)CCC1C.N C1(C(=O)NCC2C(NC(C(C)OC)=O)CC2)CCc2cc(C)ccc2O1 C#CCC(C(=O)NC(c1cn[nH]c1)C)NC(C1CN(C)CCO1)=O C(CCCCCNC(c1[nH]nnc1C)=O)N(C(COCCSC)=O)C N1(C(c2ccc(C(=O)OC)cn2)C(=O)NC)CCC(O)(C(N)=O)CC1 c1(C(N2CC3CCC3(C(=O)NCC3CCC3)C2)=O)c[nH]c2cc(F)ccc12 Cc1cc(Cl)cc(CN2CCCC2CCC(=O)NCc2c(F)cccc2Cl)c1O N1(C(CC(C=C)(C)O)=O)CC2CCC1CC2NC(C1(Cl)CC1C(C)=O)=O C1(COC)CCCN1C(=O)C(CC1CCCCC1)CC.C(=O)C=C(C)Cl.C C1(C)(C)C(=O)NOCC(=O)N2CCC1C2.C1(O)(CCC)CCCOC1 C(CSC)(C(=O)NCC(C)(C1CC1)NC(=O)CCC1CCOCC1)OC C1(NC(Cn2cc(-c3n(CC)ccn3)nn2)=O)CC2(CC(C)=NO2)C1 c1(NC(c2c(C)cc(C)cc2C)C)[nH]c(=NCC2CC(F)(F)C2)nc2sccc12 C12(C(N(CCC)CCNC(C3(OC)CCSC3)=O)=O)COC(CF)(C1)C2 C1(C=O)CCOC(=O)CC1.C(CCCNC(=O)C)OC.c1(C(=O)N)ccco1 N1(C(c2cnc(OC)s2)=O)CC2CCN(C(C34CCCC3C4(F)F)=O)C2C1 C(CCCCC(=O)NC(C1CCCC1)CNC(C1CCOCC1)=O)OCC C(C1=CCN(C(=O)CSCc2ccccc2F)CC1)NC(C(C)C1CCC1)=O N1(CCC=O)C(=O)NC(C)(C)C1=O.C1(C=O)CC2C(C1)C2(F)F.CCCC.N c1(CNC(C2CCCN(C(c3ccncc3)=O)C2)=O)cc(Cl)cc(F)c1Cl C1(NC(C2C(CC)N(C)CC2)=O)C2CC3C(C2)C13C(=O)N(C)CCOC Cc1c(CCC(=O)NC(C)CCNC(=O)C(C)Cn2ccnc2)cnn1C C1(C(=O)OCC)(NC(=O)C(O)CNc2nc(C)no2)CCOC1.CC.O Cc1cc(C(=O)NCCN(C(=O)C(C)C(C)O)C2CCCCC2)nn1C CCCC(C)(O)CC(=O)N1CC(CC(F)C(=O)N2CC(O)(C(F)(F)F)C2)C1 C1(NC(C2C(C)CCO2)=O)CCN(C(=O)Cc2ccc3c(c2)CC3)CC1O CC1(C)CC(N=c2nc(N3CC45CCC4(COC5)C3)c3c([nH]2)COC3)CO1 N1(C(CN2CCN(C)CC2)=O)CCC(F)C(NC(C2C(C)(C)C2(C)C)=O)C1 Cc1nc(O)[nH]c1C(N1CCN(CCNC(C2(C)CC2C)=O)CC1)=O C1(OC)CCN(C(C2(C(N)=O)CC2)=O)C1.N1(C(C=O)C)C(=O)CCC1=O.C C(C(C)(C)CS(N)(=O)=O)N(c1ccnc(NCc2scc(N(C)C)n2)n1)C CCCN=C(NCc1ccc(NC(=O)CCC)cc1)NCC1CC12CCSCC2 CCC(C)CC.C1(CC=O)CCC(=O)O1.C1(CS(N)(=O)=O)(C(=O)N)COC1 N1(CC(c2cccnc2)C)CCC(C(CO)NC(=O)CN)CC1 c1(C(N2CC(CC(C)NC(C(CCSC)O)=O)C2)=O)ccc(C)c(Cl)c1Cl N1(C(c2cnc(C)o2)=O)CCC(N(C(=O)CC(C)c2ccncc2)CCO)CC1 C(CC(CC)(CC)NC(c1cc[n+]([O-])cc1)=O)NC(c1[nH]cc(CC)c1)=O C1(C(=O)NC(C)CCNC(C2CC(N3CCCC3)C2)=O)COCCC1(F)F c1(OC)ccnc(C(=O)NC(C)(C)CNC(C2CC3CC2CC3O)=O)c1C c1(C(C(N2CCCC(=C)C2)=O)C)ccc(C(=O)NCC2CCCO2)c(C)c1 CCCCCCCCN.C1C2CC3C1C3C2CN.C1(NC(=O)NCC)CCC1 N1(C(c2cc(CC(C)C)on2)=O)CCN(C(c2c[nH][nH]c2=N)=O)CC(O)C1 C1(C(N2CCN(C(c3cc(C)oc3)=O)CC2)=O)C2CCC1(C)C2(C)C c1(CC)nc(C(=O)NCC2CC2)c(N)s1.c1(CCC=O)ccc(Cl)nc1.C c1(C(=O)NC(CN(C(=O)Cc2ccsc2)CC)C)c[nH]c2cccc(Cl)c12 C1(NC(c2cncc(C(C)=O)c2)=O)CCN(C(=O)C=C(C)c2ccsc2)CC1C Cc1c(C(=O)OCC(C)C)c(O)nc2ccccc12.C1(C)(C)C(=O)N1 C(C(C(=O)NCC1CCN1C(c1cnsc1C)=O)NC(C)=O)OC Cc1ccnc(CNC(c2nc(CNC(=O)C(C)(C)N(C)C)oc2C)=O)n1 CC(C#N)CCC(=O)N(C1CCN(C(=O)CCOC2CC2)CC1)CC(C)C C(=O)C1=NNC(=O)C1.c1(C(=O)OC)ccc(CC(=O)NC(C)(C)C)cc1.N CC(C(=O)N1CC(CC(F)C(=O)NCc2ccccc2)C1)C1=CCCC1 Cc1ncc(C(N2CCC(O)(CNC(=O)CCN3CCCC3)CC2)=O)cc1N C(C(CN=c1[nH]c2c(c(=NCCc3cn[nH]c3)[nH]1)COC2)C(C)C)OC c1(C(N2CC(CN(C)C(C3CCC(C)CC3)=O)C2)=O)ccc2cccnc2c1 C1(C(N2CCC(CNC(=O)CC(F)F)C2)=O)CCC2(CCOCC2)O1 c1(OC)ncc(F)c(N(C)CCN(C(=O)COc2ccccc2)C)n1 N1(C(c2n(CCC)ncc2)=O)CCC(COC)(NC(c2nncn2C)=O)CC1 C1(CNC(C(COC)OC)=O)CCCC2(CN(C(=O)C(C)(C)C(N)=O)C2)O1 c1(C(=O)OC)cnn2c1OCC(NC(=O)NCC1(F)CC3CCC(C1)S3)C2 C(=O)(C(C)(C)C1=CCSCC1)NC1C(C)CN(C(=O)CC2(CO)CCCC2)CC1 c1(C(=O)NC(CNC(C2(CCC)CC2)=O)CO)cc(O)c(F)cc1N CC(C)C(O)CC(=O)NCCN(C(=O)CCCc1ccsc1)CC(C)O C12(C(=O)N)CCC(C1)C2(C)C.N1(CCC)CCCCC1C(=O)NC1CCCCC1 C1(C(N2C3CN(C(=O)Cc4ccno4)C(CC3)C2)=O)CCC2CCC(=O)N12 CCC(C)C(O)C(=O)N(CCC(=O)N(C)Cc1cn[nH]c1)C CCC(CNC(c1c(Cl)ncn1CCSC)c1nnnn1CCCOC)CCO c1(C(N2CCCCC(CNC(c3c(C)cno3)=O)C2)=O)c2c(c[nH]c1=N)CCC2 C1(CNC(COCCOC)=O)CCCN1C(C1CC1c1ccnn1C)=O N1(C(c2c(C)nc[nH]2)=O)CCCC1(C)CNC(=O)CCn1cncn1 c1(OC)cccc(C(O)C(=O)NCC(O)CNC(c2cn(C)c(O)n2)=O)c1 n1(CC)cnc2[nH]c(=NCc3ncccn3)[nH]c(=NC3CN4CCC3C4)c12 c1(C(=O)NCC(CNC(CCSC)=O)F)c(Cl)ccc2c[nH]nc12 c1(C(=O)NC2(C)CN(C(C(C)c3ccsc3)=O)C2)cc(Cl)c(Cl)s1 C1(NC(=O)C=CCN2CCCC2)CN(C(C23CC(F)(C2)C3)=O)C2CCCC12 c1(CC(=O)NCC(CC=C)NC(=O)CCSCC(C)C)cncnc1O CCCCC(F)(F)C(=O)NC1C2CC3C1C3C2C(=O)NC(CC)CC(C)CO c1(C(=O)NC2(CC=C)CCN(C(C3CNC(=O)C3)=O)C2)ccc2oc(O)nc2n1 C12(C(N(CCNC(C3CC(=O)NC3)=O)CC3CC3)=O)CCCC1C2(F)F CC1(CS(N2CCN(c3nc[nH]n3)CC2)(=O)=O)CC(F)(F)C1 C(C(C)C)C(C)(C)O.c1(CC)oc(C)cc1C(=O)NC.c1ccsc1C=O C1(C(=O)NCC2(C)COCCN(C(CSC)=O)C2)CNC(=O)CC12CCC2 c1(NC(C2C3(CN(C(c4ncc(C)s4)=O)C3)C2)=O)cc(Cl)c([N+](=O)[O-])cc1O Cc1ccc(C2CC2)c(C(=O)NC2CN(C(C3CC3C3CCC3)=O)CC2C)c1 c1(SCC)ccc(CC(=O)NCCO)cc1.CC(F)F.CCN(C)C(C)=O C1(C(=O)NCC(C)N=[N+]=[N-])CN(C(=O)Cc2ccn(C)n2)CC12CCC2 N#Cc1ccc(C2CN(C(=O)NCc3ccc(I)cc3Cl)CCO2)cc1 n1(CC(=O)NCC23CC2CN(C(C2CC(n4ccnn4)C2)=O)C3)cccnc1=O c1(OC)cc(Cl)c(C)cc1C(=O)NC(CNC(c1ccsn1)=O)CC(C)C N1(C(C2C(C=C)CC2)=O)CCOC2CCN(C(=O)CN(CC)CC)CC12 CC1CC(CNC(=O)CC2CCN(C)C2=O)CN1C(=O)CC.c1ncccn1.S C1(CNC(c2n(CCCOC)nnn2)c2nccs2)CCCCCCC1 C1(CCC)CN(C(c2cnc(C)s2)=O)CCN1C(c1cc(CC2CC2)on1)=O C1(C=O)CC2(CCC2O)C1.c1(SCC)ccc(C(N2CCOC(C)C2)=O)cn1.N C(c1cccc(Cl)c1)=CC(N1CC=CC(NC(c2ccc(NC=O)cc2)=O)C1)=O CC1(C)COCC(NC(C2(NC(C3CCSC3)=O)CCCCC2)=O)C1 c1(OCC=C)ccc(CC(=O)NCC#CCNC(=O)Cc2csnc2C)cc1 C1(C(N2CCCC(Br)C2)=O)CCCC12CCN(c1nccc(Br)n1)C2 N1(C(C(CC(CC)C)=O)=O)CCC2C(CCCN2C(=O)CCS(C)=O)C1 N1(C(C2CC(C#C)(O)C2)=O)CC2CCCC(C1)N2C(=O)C(C)C(C)n1cccn1 c1(N2C3(CCN(C(Cc4n(C)cnc4)=O)C3)CCC2)ncnc2c(Br)nn(C)c12 C1(CCNC(C2CCSC2)=O)CCN(C(c2cc(C3CC3)[nH]n2)=O)CC1 C(CN=C(NCC1CC2(C1)CC2(F)F)N1CCC(S(=O)(=O)N2CCCC2)C1)OC N1(C(C(C)ONC=O)=O)CCCC1CC.C(C)(C)C.C1(C=O)(N(C)C)CC1.O CCC(C)(C)C(C)CC(=O)NCC(O)CN(C(=O)CO)C.c1(CC)nccn1C C(=O)(C(F)(F)C(F)(F)F)NCC1(F)CCN(C(c2ccnc3ncnn23)=O)C1 C1(NC(C2C(C)SCCC2)=O)CC2CC1CC2C(N1CCC(C(N)=O)C1)=O C(c1ccco1)=CC(=O)NCC(c1cccnc1)NC(=O)CC.C1CCCC1.O c1ccc(F)cc1.C(=O)(C(F)CC1CCC1)OCCCOC(=O)Cn1nccn1 C(N1C(=O)Cc2ccccc21)c1n(C)c(NC2CCCC3(CC3)C2)nn1 C1(C(=O)OCc2cc(C(=O)OC)no2)CC2CSCC(C1)C2(F)F Cc1ccc(CC(=O)NC2CCN(CCC3CCOC3)C2)cn1 c1(C(=O)NCC(CC)NC(c2ccc(N)cc2O)=O)cc(Cl)cc(Cl)c1O N1(C(CC2(C(=O)OCC)CC2)=O)CCC(OC2CCCC2)C(O)C1 N1(C(C2(SC)CCC2)=O)CC(NC(c2cc(C3CCC3)on2)=O)C2(CCC2)C1 C(C(=O)NC1(C)CN(C(=O)CC(C)F)C1)(c1ccccc1)=Cc1ccc(C)cc1 c1(OC)ccc([N+](=O)[O-])c(CN2CC3CN(C(=O)Nc4ccccn4)CC23)c1 N1(C(C2C(C)N(C(C3CC4(C3)CC(O)C4)=O)CC2)=O)CCC(C)(O)CC1 C(=O)(C1CCCc2nn(C)cc21)N1CCC(CCCNC(CC=C=C)=O)CC1 C1(CC=C)CC2CCC(C1)N2C(=O)C=CC1CCC1.c1(C)ccc2c(c1)CC2 c1(N2CCC3(C(C(=O)Nc4c(C)cnc(Br)c4)C3)CC2)ncnc2c(F)cccc12 c1(C=O)ccc([N+](=O)[O-])cn1.C1(C(=O)NCCOCC)(SC)CCC1.N CC(C)CC(=O)C(=O)N1CCOC(C)(CNC(c2cn(CCO)nn2)=O)C1 N1(C(c2c(C)nn(C)c2N)=O)CC2CC(C)N(C(=O)C(C)n3cnnn3)C2C1 c1(OC)nccc(C)c1-c1cncc(C(=O)Nc2cc(OC(C)C)no2)c1 C1(NC(C(CCOC)C)=O)CN(C(c2csc(-c3nc[nH]n3)n2)=O)CC1C1CC1 N1(C(C(CNC(C(CCCC)F)=O)CCC)=O)CC2CC(O)CC1C2 CC1CN(C(c2cc[nH]n2)=O)CC2(CCN(C(=O)C(C)(Cl)Cl)C2)O1 c1(C(=O)NCC2C(NC(C(CC)C)=O)COC2)onc2c1CCCC2 c1(C(=O)NCC2N(C(COCC(=C)C)=O)CCCC2)cc(C)cc2cccnc12 C1(C#N)(CCCN(C(CC)C(c2ccc(F)cc2)=O)C(C)=O)CCOCC1 c1(OC)ccc(C)cc1CCNC(=O)N(C)CCOc1ccc(Cl)cc1C c1(C(N2CCC(O)CC2)=O)ccc2c(c1)CCC2.C(=O)(CCS(C)(=O)=O)N(C)C c1(CN2CC3(CC(C(=O)NCc4c(C)cno4)C3)C2)ccc2occc2c1 N1(C(C(CC)(C)C)=O)CC2CCC1CC2NC(=O)CCn1cccn1 c1(C(N2CCCN(C(C3CCS(=O)(=O)C3)=O)C(CO)C2)=O)ccc2sccc2c1 c1(OC)ccnc(C(=O)NCC(C2CCN(C(=O)C(C)S(N)(=O)=O)CC2)C)c1F c1(C(N2CCC(O)(C(CNC(C(C)(C)SC)=O)C)C2)=O)cc2ccncc2[nH]1 CCC(C)(C#N)C(=O)NC1CCCCN(C(=O)C(C)(C)C2CCCO2)C1 N1(c2c(C(=O)OC)cc(C)cn2)CCCC12CCC2.C(=O)C=CC(=O)N(C)C C1(CC=C)(C(=O)NCCc2ccncc2)CN(C(C2CC23CC3)=O)C1 c1(C(=O)NCCC(C)NC(C(CC(C)C)NC(C)=O)=O)ccn2ncccc12 n1(CC)ccc(C(N2CCC(N(C(=O)CC3CC(F)C3)CCO)C2)=O)c1C S(=O)(=O)(c1ccc(Cl)c(CO)c1)N1CCN(C(=O)Nc2cc(C)cc(Br)n2)CC1 CCC(C)C(C(=O)NCC(C)(C)CNC(C1CC(F)CN1C)=O)N(C)C CCC(CC)CCNC(c1ccc(COC)cc1)=O.C1(CC=O)CC(F)(F)C1 CCCC(C(=O)N1CC(NC(=O)CCc2sccc2Br)C(O)C1)OC CCCC(CCC)CC(=O)NC(c1cnn(C)c1)C(=O)NC(CC)CC(F)(F)F N1(C(c2n(C)c(=O)ccc2)=O)CC(NC(C23CCC(C)(CO2)C3)=O)CCC(O)C1 C1(C(N2CCC2)C)CCN(C(=NCCC2OCCC2(C)C)NCC2CCCCO2)C1 c1(C(=O)OC)cc(NC2CCCCC23CC3)cc(F)c1 N1(C(CCC(=O)NCC)=O)CCC2(C1)CN(C(=O)CCc1cscn1)C2 Cc1ccc(C(N2CCN(C(=O)COc3ccccc3C(N)=O)CC2)=O)c(N)n1 c1(NC(CC(CNC(=O)C(C(C)C)SC)OC)=O)ccc(OC)nc1C c1(C(=O)N)cccn2nnnc12.N1(C(c2nc(CC)sc2)=O)CC(C)C2(CC2)C1 c1(C(N2CCC2)=O)ccc([N+](=O)[O-])c(Cl)c1.c1(N(C)C)ccc(C(=O)N)nn1.C C1(N(CCOC)C(c2cnoc2C)=O)CCN(C(=O)CC2CCC(=O)N2C)CC1 C1(C(=O)NCC(=O)OCC=C)CN(C(=O)CC2COC(=O)C2)CCO1 c1(CC)nc(N2CC(CO)(NC(C3(C)CNC(=O)C3)=O)C2)cc(C)n1 S(=O)(=O)(c1ccc(NCc2conc2C(C)C)c(C#N)c1)NC(CCCCC)C CC(C)(C)C(=O)NCC(=O)NCC1(CC)CC1.c1(C(=O)N)nocc1Br c1(C(c2nnnn2C)NCc2cc(C)c(O)nc2)csc(S(N)(=O)=O)c1 N1(C(Cc2c(C)nc[nH]2)=O)CC2CCCC(C1)N2C(C1CC(=O)NC(C)C1)=O N1(c2snc(C(C)=O)n2)CCS(=O)(=O)C(CC)C1.c1(C=O)c(C)nn(C)c1C.N N12CC(CC1=O)C2.C=C(C)CN(CC(=O)N1CCC1)C(=O)CSC(F)F C1C2CCC1CN(C(C1CCSC1)=O)C2.c1(OCC=C)ccccc1C(=O)NC c1(C(=O)NC2C(NC(c3c(CCC)n[nH]c3)=O)COC2)cc(O)nc(Cl)c1 c1(C(=O)NC2CC(CCNC(c3cccc[n+]3[O-])=O)C2)n[nH]c2c1CC1CC21 C1(NC(c2cnco2)=O)CCCN(C(=O)CC2(O)CCCOC2)CC1.C1(C)CC1 c1(SC(N)CC(=O)NC2CCCCC2O)c(O)cccc1F Cc1nc(NC(C2CCN2C(c2cnc(Cl)c(I)c2)=O)=O)cnc1C#N CN1CCOC(C(=O)NC)C1=O.C1(O)CCN(C(=O)CN2CC(=O)NC2=O)CC1 C12(C(=O)O)CCCC1(C(=O)NC1(c3cn(CCN(C)C)nn3)CCCOC1)C2 N(C1CCOc2ccc(C(=O)O)cc21)C(C(=O)N(C1CCN(C)C1)C)=O c1(OC)ccc(OC(F)(F)F)cc1CNC1CC(NC(c2[nH]ccc2C)=O)C1 Cc1cc(C(=O)NCCC2CN(C(=O)C(F)CC(C)C)C2)c(N)c(Cl)c1 C1(C(=O)NC2(CC=C)CC=CC2)CC(=C)CCN1C(=O)CCCCCSC C=CCCCCC(=O)NCCN(C(C1CC1c1cc(C)oc1C)=O)C(C)C C(=O)(CC1OCc2ccccc21)N1CCC(CNC(CN(CCC#C)C)=O)CC1 C1(CCC)(NC(C2CCCC2(F)F)=O)CCCN(C(c2cnsc2C)=O)C1 N1(C(Cn2nc(C)oc2=O)=O)C2CCC(C2)C1CC(=O)NC(C)CSC(F)F N1(C(C(C(C)O)NC(=O)C#CC(C)(C)C)=O)CCC2CCCC2CC1 c1(NC(CCCC=C)C)[nH]c(=NC2CC2c2ccccc2)nc2c1cnn2CC C1(CCC)CN(C(c2cc(CC)ccn2)=O)CCN1C(c1ccccn1)=O c1(C(N(CCCCN(C(C(CC=CC)CC)=O)C)C)=O)cn2cnnc2cn1 N1(C(C2(N(C(=O)CCCC3CCCC3)C)CC2)=O)CCNC(=O)C12CC2 c1(N2C(C)C(NC(c3cc(Cl)c[nH]3)=O)C(C)CC2)ncc([N+](=O)[O-])c(=N)[nH]1 C1(NC(c2cc(O)nc(O)c2)=O)CC2CCC(C1)N2C(C1CC=CCO1)=O C1(O)(C(=O)NCC2C3CN(C(C4CC45CCSCC5)=O)CC23)CCCCCC1 c1(C(C)C)nc(C(=O)N(CC(C)CNC(=O)CC2CC=CC2)C)co1 C1(CCCNCC2CCC(=O)N2)CCCCN1CCO N1(C(C(CC)n2cccn2)=O)CC2CC1CN(C(c1ccnnc1Cl)=O)C2 S(=O)(=O)(C1(Cl)CC1(C)C)N(CCCc1nc(-c2cccnc2)no1)C(C)C N1(C(C(N2CCN(c3n(C)c(Br)cn3)CC2)=O)=O)CCCC(O)C1C(F)(F)F.CC c1(C(=O)NC2C3(CC(NC(C(CCC)C)=O)C3)C2)cc2cccnc2[nH]1 C(CCC(=O)N1CCC(CN(C)C(c2csc(Cl)c2)=O)C1)NC(=O)OC c1(-c2ccc(S(=O)(=O)NC(C3CC3)=O)cc2)c(O)cc(=O)n2c1CCCCC2.C C=C1CCN(C(=O)CN2CCC(C)C2)C(C(=O)NCC2Cc3nccn3C2)C1 C(=O)(C1=C(Cl)CCCC1)N(C(C)C(=O)NC1(CCCF)CC1)CCC C1(C(=O)NC2(CO)CCN(C(CC(C)O)=O)C2)CCCC(C#N)C1 C1(C(=O)NCC2(C)CCN(C(C3(O)CCOC3)=O)CC2)CCCC1S(C)(=O)=O c1(C(=O)NCC2OCC(CNC(CCCC=C)=O)C2)c(C)nn(C)c1Br CCC(C)(C)C(C(=O)N1CCCC1CN(C(=O)CC1(OC)CCCC1)C)OC C1(NC(C(C)C)=O)CCN(C(=O)Cc2c(F)cncc2Cl)CCC1(F)F c1(C(=O)NCC(C)(CO)NC(c2nncc(CCC)c2)=O)cccc2[nH]ncc12 O=C(CCCCc1ccc(OC(F)(F)F)cc1)NCCc1ccc(O)cc1 c1(OCC)cncc(NC(C2CC(O)CN2C(c2ncc(C)s2)=O)=O)n1 N1(C(C23OCC(COC)(C2)C3)=O)CCC2CN(C(C3CCC3O)=O)CC2CC1 C1(C(N(CCNC(c2ccc(O)cc2Cl)=O)CC)=O)CN2CCN1CC2C Nc1cncnc1C(=O)NC(C)C1CCC1.C1(CC(=O)N)CCS(=O)(=O)C1 O=C(C(C1=CCSC1)N1CCC2(CCCO2)C1)Nc1ccccc1 C1(NC(C(CNC(CNC(=O)OC)=O)C(C)C)=O)CN(C)C2(CCC2)C1 N1(C(c2nc(COC)[nH]n2)=O)CCN(C(=O)COC2CCCCC2C)CC(O)C1 C1(NC(C2OCC(C)(C)C2)=O)CN(C(=O)CCNC(N)=O)CC2(CC2)C1 N1(C(Cn2c(C)cnc2)=O)CCCC(N(C)C(c2scnc2C(C)(C)C)=O)CC1 c1(NC(C(C)=C2CC2)=O)ccc2c(c1)CCO2 c1(N(C2CCN(C(c3c(OCC)cccn3)=O)C2)C)ccnc(C#N)n1 N1(C(C(CC)n2cccn2)=O)CC2CCN(C(C34CCC(CO)(CC3)C4)=O)C2C1 C(CCCC)(C(=O)N1CCC(O)C(O)C1)NC(CC1CC(CC)C1)=O c1(C(C(=O)NCCCN(C(C(F)=CCC)=O)CC)CO)ccc(Cl)cc1 c1(C=O)ccc2[nH]nc(O)c2c1.C(c1cn[nH]c1)=CC(=O)NCC1(C)CCC1 c1(C(=O)OC)cccc(C(=O)NCC(C)(C(C)C)NC(c2nocc2Cl)=O)c1 c1(C(=O)NC23CCCC(NC(C(C)SC)=O)(C2)C3)nccc2c(F)cccc12 N(C1CCCn2ccnc21)C(CC(CNC(c1cncc(NC)c1)=O)OC)=O c1(C(=O)NC(CC)CN2CCCC2)cn(C2CCNCC2)nc1C(F)(F)F C(C)(C)(C(=O)NC1CC(CCC(=O)NCc2ncn(C)n2)C1)NC(C)=O CCC(CC)C(C)C(=O)NCCCN1CCC(NC(C23COCC2C3)=O)C1 c1(C(N(CCN(C(C2CC2F)=O)CC)CC)=O)ccc(OC)cc1N N1(C(c2c(C)ncn2O)=O)CCCC(CO)(NC(=O)CSC2CCCCO2)C1 Cc1c(C(N2CC3(COC(C)C3)C2)=O)sc2cncn12.C(=O)C(F)(F)C1CC1.N C1(NC(C2C(CNC(CCc3cn(C)nc3)=O)OCC2)=O)CCCN2CCCC12 C1(O)(C(N2CCC(CNC(c3cn(C)nc3O)=O)C2)=O)CCCCCC1 c1(C(N2CCC(N(C(=O)C(CC)N(C)C)CCC)C2)=O)cccc2nc(C)nn12 c1(SCC(=O)NCC2(CCNC(C3CCCSC3)=O)CC2)ccccc1 c1(NC(c2cccc(NC(=O)Nc3ccc(OC)nc3)c2)=O)ccccc1C#N N1(C(CC=C)=O)CCCC(C(N2CCC(CO)C(O)C2)=O)(CC)C1 C(=O)C1=C(Cl)CCC1.C(=O)(CC(F)(F)F)NCC(=O)NCCC1CCCC1 N1(C(c2ccnn2C)C=O)CCN(CC(N)=O)CC1.CC.CCC1CC1.CCO C12(NC(C(CC)N(CC)CC)=O)CC1CN(C(=O)CCC1(C)N=N1)C2 Cc1nc(C2CC2)sc1CC(=O)N.c1(C=O)[nH]nnc1C1CC1.C1(CC)CC1 CCCCC(=O)NC1CC(C)C1.C1(CS(C)(=O)=O)(C(=O)N)CC(F)(F)C1 CC1C2CCC(C2)C1C(=O)NC1C=CC(C(N2CCC(CC(N)=O)CC2)=O)C1 C1(OC)(C)CCN(C(=O)Cc2csnn2)CC1.C1(C=O)CN(C2CCOC2)C1.N n1(CC#C)c(C)cc(C(N2CCCC2(CNC(=O)CSC)C)=O)c1C.O N1(C(C(C=CCCC)O)=O)CC2(CC(NC(=O)C(C)(C)c3cncs3)CO2)C1 CCCC(CO)NC(C1(CCNC(c2ccn(C(F)F)n2)=O)CCC1)=O CC1CC(=O)CCC1C(=O)NCCCOCCNC(=O)C(c1ccccc1)F c1(C(C)C)ccc(C(N2CC3C(NC(c4cn(CCO)nn4)=O)C3C2)=O)c(O)n1 C1(C(=O)NC2CC(O)(CO)C2)C(O)CCN1C(=O)C=Cc1nccs1 N#Cc1c(CNC(C2CC23CCN(C(=O)C2=COCCC2)C3)=O)cccc1F c1(C(=O)NC2C(CCC)CN(C(=O)CC(O)C(C)C)C2)cc(O)c(C)cc1C Cc1nc(-c2ccccc2)oc1C.N1(CC(=O)NCc2cccs2)CC(O)CC1CO CCC(CC(C)C)C(=O)N1CCN(C(=O)CSCCNC)C(CC=O)C1.C1CC1 N1(C(COC(CC)C)=O)CCN(C)CC1C(=O)NC(C)C(C)n1cccn1 N1(C(C(C)=O)=O)CCCC(CC(=O)NCC2CCCCCC2)C1 Cc1noc(Cl)c1CCC(=O)N(C)CC1CCCN1C(C1CC(CC(F)F)C1)=O C(=O)(C1=Cc2ccccc2OC1C(F)F)N.CC(C)C(F)C(=O)NC1CC(C)C1 N1(C(C)=O)CCN(C(=O)C(CN(C)C)NC(C2CC(C3CC3)C2)=O)C(C)C1 N1(C(CNC(Cn2ncc(C)c2)=O)=O)CC(C)OC(C)C1.c12ccnc(c1)NC2 CCC(C)C(O)C(=O)NCCC(C(C)C)NC(c1nn(C)c(Br)c1C)=O CCCCCCN(C(=O)CC1CC1)CCN(c1nnc(C)s1)C.CCC N1(C(C(CC)(F)F)=O)CCC(C(N2CC3C(C2)C3(C)C)=O)C(O)C1 Cc1cc(N2CC3CC3(CO)C2)ncc1S(=O)(=O)NC1CCn2ccnc2C1 c1(C2(CC(N3C(CNC(CN(C(C)C)C)=O)CC3)=O)CCC2)ccccc1 c1(C(=O)NC2C3(CCC(NC(CC(CC)C)=O)CC3)C2)cc(Cl)c2n[nH]cc2c1 Cc1cc(C(=O)NCC2CCCCN2Cc2sc(Br)nc2Br)cc(Cl)n1 C(=O)(C1CCSc2ccccc21)N1C(C)(CNC(c2nc(C)oc2C)=O)CCC1 C(C)(C)(CC(=O)NOCc1nc[nH]n1)N(C(c1c(F)ccc(C)c1)=O)C N1(C(CN(C(C)=O)C)=O)CC(C(=O)N(CCCCC(C)C)C)C(C(C)C)C1 CCC(O)(C(=O)NCC=CC)c1ccccc1.C1(C(=O)N)CCOC1.C(C)C n1(CC)ccc(C(N2CCC(CN(C(=O)Cc3cnsc3)C)C2)=O)n1 C1(C(=O)NC2(CC=C)COC2)CCCCC1c1cccc(F)c1 CN1C(=O)CCC1CC(=O)NCC(CNC(c1cccnc1N(C)C)=O)CO N1(C(c2cn(C)nc2)=O)CC(C(=O)NC(c2cncn2C)CO)C(F)(F)C1 C(=O)(CCN(OC)C(=O)c1cncnc1)N1CCN(CC)C(=O)C1C c1(OC)cc(CN(CC(N2CC(c3ccc(OC)cc3)CC2C)=O)C)ccc1O C1(CCCC)NC(=O)N(CC(c2ccccc2)OCCN2CCCC2)C1=O C(=O)(C(C(C)O)N(C)C)N.c1(C(=O)NCC(C)(C)OC)cc(CC)on1 Cc1nc(C2CCC2)oc1C(N1CCCCC1C1CC1)=O.C(=O)(C(O)C1CC1)N N1(C(CN(C)Cc2c(C)nc(CC)o2)=O)CCC(C2CCCN(CCOC)C2)C1 C1(NC(C2CCN(C(C=CC(C)(C)SC)=O)CC2)=O)CC(=O)NC(=O)C1 CC(C)C(C)(O)C(=O)NCC1CCC(C(=O)NC2(C3CC3)CC2)O1 N1(C(c2cncc(NC)c2)=O)CCN(C(=O)Cc2cccc(F)c2)C(C)CC1C C1(CNC(C=Cc2occ(C)n2)=O)CCCN(C(C2CC(C(C)C)C2)=O)CC1 N1(C(CCOCC)=O)CC2COCC2(C(=O)N(C2CCCC2C)C)C1 c1(OC)ccc(NCC(O)CC2CCCC2)cc1NC(C)=O CC(C)CCCCCN=c1[nH]c(=N)[nH]c(=NCC2CCC3(CCCC3)O2)[nH]1 c1(CCC(N2CCC(C)(CNC(C3C(C)CCCC3)=O)C2)=O)c(F)cccc1F Cc1ccc2nnc(CNC(c3cnn(CC4CCOC4)c3)=O)n2c1 N1(C(Cc2cc(C)nn2C)=O)CC(NC(C2CC(C)(C)CN2C)=O)CC1(C)C N1(C(CCCOCC)=O)CCN(C(C2CC(O)CN2C)=O)CC(C)(C)C1 C1(CC(C)C)(NCCNS(=O)(=O)C2CC2)CC(=O)C1 c1(CCC(=O)NC2C(C(=O)NC(c3ccncc3)CC)C2)ccc(O)cc1 c1(C(=O)OCC)c2c(nn1C)CN(c1nnc(-c3cc(C)[nH]n3)n1C)C2 CC1CCC(S(C)(=O)=O)CN1C(=O)CSC(c1cccc(F)c1)=O Cc1cc(CC(=O)NCC(C)NC(=O)CCCc2ccccc2Br)ccc1O C1(CC=C)(NC(=O)C(c2ccn(C)n2)C)CCCN(C(c2coc(CO)c2)=O)C1 C(=O)(C(C(C)CC)NC(=O)CSC(F)(F)F)NC1CC(C=C)C1 c1(OC)ccc(C(N2CC(NC(C3CC3F)=O)CC2(C)C)=O)c2ccoc12 C(CC(=O)N1CCC(CC(C)O)CC1)(C(F)F)NC(C(COC(C)C)(C)C)=O c1(NC(C)=O)cc(C(N2CCC(NCc3nnsc3Cl)C(C)C2)=O)ccc1C c1(C(=O)NCC2(O)CN(C(C(C)C)=O)C2)cccc(-n2cccc2)c1 CC(CNC(=O)C(CO)NC(=O)COCC1CC1)C(F)F Cc1nc(C(=O)N)c(C)s1.c1(CC=O)cn(C)nn1.C1CN(C(=O)C2CC2)C1 CN1CCN(CCNc2c(Cl)cc(Cl)nc2N)CC1(C)C C12(C(=O)NC(C3(O)CN(C(c4cc(C)c(O)nc4)=O)C3)C)CCC(C)(CC1)OC2 C1(CNC(C(CCC)CC)=O)CN(C(=O)C(c2cccc(C)c2)F)CC12CCC2 c1(NC(c2ccccc2F)CO)cccc(-c2ccc(Cl)cc2)c1 N1(C(c2cc(C)c(C)[nH]2)=O)CCC(C)CC1C(N1CC2C(C1)C2(C)C)=O Cc1cc(OCC2CN(Cc3ccccc3)CCO2)cc(C)c1O C1(C(N(C)CC2CCCN(CC)C2)=O)CC(C)CN(C(C2(CF)CC2)=O)C1 c12ccccc1NC2C.C1(C(CSC)O)CCN(C(=O)OC(C)(C)C)CC1 C1(NC(CCOCCOC)=O)CCCN(C(c2ccc(Cl)cc2)COC)C1 c1(CC)nc2c(C)csc2c(=NCC2CN(C(=O)Cc3csnn3)CCO2)[nH]1 C12(CNC(COCC(C)C)=O)CCCC1N(C(c1cc(Cl)nnc1Cl)=O)CCC2 N1(C(C(C(C)C)SC)=O)CCn2c(CNC(=O)Cn3ncnn3)nnc2C1 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O=C(C(O)CC(F)(F)F)N1CCC2(CC1)CC2C.C12(C(=O)N)CCC(C1)OC2C N1(C(c2c(CC)ccs2)=O)CC(N(C)C(c2cncc(Cl)c2)=O)C(F)C1 c1(C(=O)NCC(CC(C)C)NC(=O)CN(C2CCSC2)C)cc(N)ccc1O C1(NC(CC2(OC)CCC2)=O)CCN(C(=O)CCc2cnoc2)CCC1(F)F c1(C(=O)NC2C(C=C)CN(C(c3cnc(C)s3)=O)C2)cccc2c(C)c(C)[nH]c12 N1(C(c2cc(OC)no2)=O)CC2(CCC2)C1.c1(C=O)ccc(C(C)(C)C)s1.N C(=O)C(F)CC(C)(C)C.C1(C(=O)NCCC(C)N(C)C)C2CC3C(C2)C13.N c1(OC)cc(C)sc1C(=O)NC1CN(C(c2c(C)nsc2)=O)C1.C1CC1.N Cc1cc(Cl)c(C(=O)NCC2CCC3(CN(C(=O)C(O)C4CCC4)C3)O2)cc1F C1(OC)(CN2CCCC(C(=O)N(CCCO)C)C2)CCCC(C)(C)CC1 N1(C(c2ccc(C)cn2)=O)CCC2(C1)CN(C(c1cc3ncsc3[nH]1)=O)C2 c1(C(=O)NC2CC(C)N(C(c3csc(Cl)c3)=O)C2)c(C(F)F)cccc1N c1(C(N2CCCC(N(C(C3(CC)COC3)=O)C)C2)=O)cccc2nc(CO)[nH]c12 c1(CC(=O)NC2CN(C(C34COCC3C4)=O)CC2C(F)F)ccc2c(c1)OCO2 C1(CNC(c2ccn(-c3ccccc3)n2)=O)CCCCN(C(=O)C=C(Cl)Cl)C1 c1(SC)nc(CN2CCN(C3CN(c4cnc(C(F)(F)F)s4)C3)CC2)cc(C)n1 c1(C(=O)NC2CC2C(=O)Nc2ccnc(O)c2)nc2ccccc2[nH]1 C1(c2c(C(N3CCC3)=O)c[nH]n2)CCCCN1C(C1CCCS1)=O O=C(N=c1cnn(-c2ccc(Cl)cc2)[nH]1)c1ccc(CCC(F)(F)F)cc1 c1(CNC(c2cn(C)cn2)C)nc(C(C)S(C)(=O)=O)no1 N1(C(C(C=C)O)=O)CCN(C)C(C(=O)NCC(C)C(=O)NC)C1 c1(OC)ccc(COCC(N2CC(C)CC2C(=O)NC2CC(F)C2)=O)cc1 N1(C(C(F)OC)=O)CCCC2(C1)CN(C(C1(CCF)CCOCC1)=O)CCO2 CCC1=C(C(=O)NCCOC(C)(C)C)CCCO1.C1(C=O)CSCC(=O)N1.N C(=O)(C(C)(C)C(F)F)N1CCC1.N1(C(C=CCCC)=O)CSCC1NCC.O CCC(COC(N1C(C(C)C)CCC1C(C)C)=O)(CC)OC C(=O)(CCC(C(C)C)NC(=O)C1=C(C#N)CCC1)N(C1CCCC1)CCC C1(CNC(c2ccsn2)=O)CCN(C(c2ncnc3cc[nH]c23)=O)CC1C1CC1 c1(C(N2C(c3cn(CCC=C=C)nn3)C(C)CC2)=O)ccc2[nH]ccc2n1 c1(OC)nc(N(C2CCC(N)C2)C(c2cnc(F)c(C)c2)=O)ncc1Br c1(C(=O)NC(CN(C(C2CC(Cl)(Cl)C2)=O)CC)C)cc2ccccc2nn1 C1(NC(c2c(COC)cco2)=O)CCOCC1C(=O)NOCC=C(C)C C1(N(c2cc(CCC)no2)C(=O)C(Cl)(Cl)Cl)CC2CNC1C2 C(=O)(C1Cc2ccccc21)NC(C(N1CCS(=N)(=O)CC1)=O)Cn1cncn1 c1(C(=O)NC2(C)CCN(CC3CC3)C2)n[nH]c2ccc(Cl)cc12 N1(C(c2c(C)ccnc2F)=O)CCC2(CCCN2C(=O)CCCCN(C)C)CC1 c1(C(N2CC(C)(NC(C3N(CC)C(=O)CC3)=O)C2)=O)cn2nc(C)sc2n1 C(=O)(C(C)C(F)(F)F)N1CC(O)(CNC(c2ccn(CC)c2C)=O)C1 CC(C)C(C(=O)N(CC(O)CNC(=O)C(C)(Cl)Cl)C)c1cccc(Cl)c1 c1(C(N(C2CCCCN(C(C(C)SC)=O)C2)C)=O)cnc(O)n(C2CC2)c1=O C=CCC(C(=O)N1CC2CC1CN2C(c1ccc(C#N)cn1)=O)C(C)(C)C C1(NC(C(C)CC(F)F)=O)CN(C(=O)CCc2cc(Cl)no2)C2(CCC2)C1 c1(CC(=O)NCC(CNC(C(c2ccc(Cl)s2)C)=O)F)sccc1Cl C1(C(N2CCN(C(=O)OC)CC2)=O)CCC(C)N(C(=O)CCCC2CCC2)C1 C(=O)(N=c1cc[nH]cc1Cl)C1N(C(c2ccc(C(C)(C)C)s2)=O)CC(F)C1 c1(C(N(CC(Cc2ccccc2)NC(C(CC)O)=O)C)=O)cc(F)c(F)cc1Cl C1(CNC(C(C(CC)C)O)=O)CCC2(CN(C(c3ccoc3Br)=O)C2)O1 Cc1nc(N(C2CN(C(=O)C(C(C)C)c3ccccc3)C2)C)cc(S(C)(=O)=O)n1 O=C(CC(O)(C(F)(F)F)c1ncc[nH]1)NC1CCC(C)CC1.C(=O)(C1=CCC1)N C(=O)(C1=CCN(C(C2CC(C)N(C)C2)=O)C1)NC(c1c(C)ccnc1)C N1(C(CSC(C)(C)C)=O)CC(C2CCCCN(C(C3CCCN3N=O)=O)C2)C1 c1(C(=O)NCC2N(C(CS(CCC)(=O)=O)=O)CC2)ccc2c(c1)C(=O)NCC2 c1(C(N2CCC(NC(c3c(CCC)nco3)=O)C(C)C2)=O)ccccc1[N+](=O)[O-] N1(C(C(C(=C)C)(C)C)=O)CCC2(C1)CN(C(=O)C(C)(C)C1CC1)CCO2 O=C(N=c1ncnc2[nH][nH]cc1-2)c1ccc(NCc2cc(F)c(O)c(F)c2)nc1 C(CC(F)CN=[N+]=[N-])NC(C(Cc1cnc[nH]1)NC(CC(C)n1cccc1)=O)=O C#Cc1cccc(C(C)(C)NC(c2nccc(Cl)c2O)=O)c1 c1(C=O)cc2c(cc1)OCO2.C(C)(CC)NC(C1C(CC)C1)=O.C1CC1.N C(C)(C)(C(=O)NC(c1ccccc1)CNC(C12CC(F)(C1)C2)=O)OC N1(C(c2cc(CO)[nH]n2)=O)CC(C)CC12CCC2.C1(C=O)(C(F)F)CCCO1.N CC1SCCCC1C(=O)NCC1(F)CC(NC(c2cnco2)=O)C1 C(C(C=O)NC(c1cc(C2CC2)no1)=O)OCC.C1CC(n2ccnc2)C1.N C(CC(=O)NCC1C2CCCOC12)(C(C)C)NC(CC(CC)SC)=O C1(C(=O)NCc2n(CC)ncc2)CN(C(=O)CS(C)(=O)=O)CCC1C C1(CNC(C2C3CCC(F)C23)=O)C2CC1N(C(=O)CCn1cnnn1)C2 C1(NC(C(N)=O)=O)CCC(F)(C)C1.c1(-c2c(C(=O)N)c[nH]n2)ccc(Cl)cc1 N1(C(CNS(CC)(=O)=O)=O)CCC(NC(=O)COc2ccccn2)C(F)C1 Cc1ncc(C(=O)NCC2CCN2C(=O)C(C)C(F)F)c(Cl)c1Br NCCCCCCCCNC(=O)C(=O)NCCC1CCCOC1 C1(O)(Cn2cc(CN)nn2)CCCN(C(c2ccc(Cl)cc2Cl)=O)C1 C1(CC=C)(C(=O)NCC)CCN(C(=O)C(O)CC2CCCC2)C1.C(N)=O.N C(=O)(CC(C)(C)CC(=O)NCC1CN(C(=O)C(C)CSC)CC1)OCC CC1(C(=O)NOCc2cn(-c3ccc(F)c(Cl)c3)nn2)CCCC(F)(F)C1 CCCC(C(=O)NC(C)C(CO)NC(C1CN(C)C1)=O)N(C)C C(C)(C)(C(C)C)NC(c1cc(CCOC)on1)=O.C1CCOC1=O.C(=O)C c1(-c2cc(CC)c(F)cc2)cnc2ccc(C(=O)Nc3ccc(CO)nc3)cn12 N1(C(C2C(C(=C)C)OCCC2)=O)CCC2CN(C(c3cnccc3C)=O)CC2C1 Cc1c(NCC(c2ccccc2)N2CCCC2)cccc1N1C(=O)NC(C)C1=O Cc1c(C(=O)N(CCC(C)NC(c2ccccn2)=O)C)cccc1CO C1CCCC1.C1(C#N)(C=O)CCC1.CS(=O)(=O)CC1(CC(=O)NC)CC1 CCCCCCCCCC(=O)NCCCc1cn(CC2CCC2)nn1 Cc1ccc(=NCCC(=O)NC(C)CCCNC(=O)CC2C=CCC2)[nH]c1 C1(C)(CNC(C2(F)CN(C(CC=CCCCCC)=O)C2)=O)CCCC1O N1(C(C2C(C)OC(C)C2)=O)CCCCC(C2CN(C(=O)COCCO)C2)C1 C1(NC(C(c2n(C)ncc2)(C)C)=O)CN(C(=O)C(O)C(C)(C)C)CCC1O c1(C(N(CCN(C(C2C(C(C)C)C2)=O)C)C)=O)cc(Br)c2[nH]nnc2c1.CC Cn1cc(Br)c(CNC(N2CCSCC2c2ccc(C(F)(F)F)cc2)=O)n1 C1(NC(=O)C=CCO)CCCCC1NC(C1(n2cccc2)CCCC1)=O c1(COC)ccccc1OCC(O)CN(C=O)Cc1cccnc1 CC1CN(C(=O)C2=NNC(=O)CC2)CC2(CCN(C(c3csc(C#N)c3)=O)C2)O1 C(=O)(C(C)(CC)CO)NCC1C2CN(C(C=COCC)=O)CC21 C(CC(=O)N1CC(CO)C2(CC2)C1)(C(C)(C)C)NC(C(CSC)OC)=O C=CC1(C(=O)NC2CC(NC(=O)CC3CC3(C)C)C(O)C2)CCOCC1 C1(CCNC(C2CCCOC2)=O)CCCN(C(c2coc(C(F)(F)F)c2)=O)C1 Cc1c(Br)cc(C(=O)O)cc1S(=O)(=O)N(C)Cc1ccc(CC(C)C)cc1 c1(C(=O)N)cc2ccc(Cl)nc2s1.n1(CC)ccnc1C(=O)NC1CC(C)C1 C(=O)(C(C)N=c1cc[nH]cc1)NC1(C2C(C)OC(C)(C)N2)CC1 N1(C(c2cnn(Cc3ccccc3)c2)C(=O)NCCSC)CCc2ncccc21 N1(C(C(c2ccnn2C)N(C)C(c2cc(Cl)c[nH]2)=O)=O)CCC(c2nn[nH]n2)C1 C1(C(=O)NCCC2N(C(C=CC)=O)CCSC2)CC2(CCC2O)C1 c1(C(=O)NC2CC(CNC(c3ccncn3)=O)C2)n[nH]c2cc(Cl)ccc12 C(N=c1[nH]c2ccc(Br)cc2o1)C1C(C)CCN(C(CC2C(C)CCC2)=O)C1 N1(C(c2c(OC)c(F)ccc2)=O)CC(C)CN(C(=O)C=C2CCCCC2)CC1C Cc1nn(C)c2c(N(C)CC3CC(F)(F)C3)nc(=NCC(C)c3cccs3)[nH]c12 C1(C(NOC(C(=O)OC)C)=O)N(C(=O)CC2(N(C)C)CCC2)CCC1(C)C c1(C(C(=O)NCCC2CC2)N(C(CC)C#N)C)ccc2c(c1)OCC2 Cc1cc(CNC(C2CSCN2C(C2CC(C)N(C)C2)=O)=O)nnc1C CCCC(CC)C(=O)N1CCN(C(C)CNC(=O)CC2CCC2)CC1 c1(C(=O)NC(C(=O)NCc2onc(CC)n2)COC)oc(C)nc1CC C1(NC(c2nc(C(C)(C)C)sc2)=O)(CO)CCCN(C(C2CCC(=O)N2)=O)C1 c1(-c2ccc(C(=O)NS(=O)(=O)CCCCl)o2)ccc(Cl)cc1 N1(C(c2nc(C)[nH]n2)=O)CCC2(C1)CN(C(C1(CC(F)F)CCC1)=O)CCO2 N1(CCOC)C(=O)NC(c2cc(OC)ccc2F)C2=C1C(C)N(C)C2=O C1(C(=O)NC2CCC(CNC(=O)C(O)C3CCCC3)C2)CC2(CCOCC2)C1 C1(N(C(c2ccccc2)=O)C)CC2CCC(C1)N2C(=O)C(C)(C)C=C.C#CC.N N1(C(c2c(CC)cncc2)=O)CCC2CC2(NC(=O)CCc2nc(C)cs2)CC1 C12(NC(C3COC3)=O)CCCCC1CN(C(c1cccc3nsnc13)=O)C2 C#Cc1ccc(CC(=O)NCCCOCCCNC(=O)CCCCCF)cc1 Cc1[nH]nc(C(=O)N(C2CC(NC(=O)CC3CCC(C(F)(F)F)O3)C2)C)c1C N1(C(Cc2cc(C)no2)=O)CC(C(=O)NC2COCC2CO)CC(C)C1 CC(C)(O)COC(=O)CCNC(=O)COCCOCC1CCOC1 C(=O)(C(O)CC[S+](C)C)NC1C(CO)CCN(C(c2c(C)cn(C)c2)=O)C1 C(=O)(C(C)(O)CC(C)C)N(CCC(C)NC(C=Cc1cncc(C)c1)=O)C N1(C(c2cccc(CC)n2)=O)CC(CNC(C2CCNC2=O)=O)OC2(CCC2)C1 C1(C)(C(N(C2CCN(C(C(C)(C)OC(C)=O)=O)CC2)C)=O)CCC(C)CC1 c1(C(=O)NCC(CO)NC(C=C(CC)C)=O)cc(CC)oc1C CC1(F)CN(C(=O)CC2CCCC2)CCN(C(c2ccc(Cl)c3occc23)=O)C1 Cn1ccc2nc(N(Cc3[nH]cnc3C#N)CC3CCNCC3(F)F)nc(Cl)c12 c1(OC)ccc(C(C)NCc2ccc(I)c(Br)c2)cc1F N1(C(=O)OC(C)(C)C)CCCC(CC(=O)NC2CC(O)CC2O)C1 Cc1cc(C)c(C(=O)NCC2CCCN(S(=O)(=O)c3cccnc3)C2)c(C)c1 CCCCCCCC(=O)NC1CC(CNC(=O)C(C#N)(CC)CC)C1 C1(NC(CN(CCOC)C)C)CCN(C(=O)CC(C)n2cccn2)C1 c1(OC)cn(C)c(C(=O)NC2CCN(C(c3cnn(C)n3)=O)C2)cc1=O C(CC(C)C)(C=O)NC(C)=O.C12CN(C(C3(C4CCC4)CC3)=O)C(C1)C2.N N1(C(C)C)Cc2c([nH][nH]c2=NC(=O)OCC(N2CC(C)OC(C)C2)=O)C1(C)C C1(C(=O)NCC2(CC)CCCO2)C2CCCC2CN1C(=O)C.C1(C)CCCC1 c1(C(N(C(C)C(N)=O)C)=O)ccc2c(c1)CCC2.C12CCN(C1)C2 C(=O)(C(C)(C)CCNC(=O)C(C)c1cc[nH]n1)NC(c1cccnc1)C N1(C(C2C(C)=C2)=O)CCC2(C1)CN(C(=O)CC1(C)CC1(F)Cl)C2 C1(C(N2C(C)(C(=O)NCC(c3cccs3)O)C=CC2)=O)CC2CC1CC2O C1(C(NCC(C)C=O)=O)CC(O)C(O)CC1.C1(CC=O)CC(C)=NO1.CC CC(Cc1ccco1)C(=O)NCC(O)(Cc1ccccc1)c1nn[nH]n1 C12(C(=O)NCC3CC(C)N(C(c4ccn(C)c4)=O)C3)CC3CC1C2C3(F)F C1(C(=O)NC(CC#C)CC#C)CC2(CCN(C(C3(C)CC4C=CC3C4)=O)C2)C1 N1(C(c2cccc(CC)n2)=O)CCC2(CCCN2C(c2ncoc2CC)=O)C1 N1(CC)CCCC(N=c2c(Br)c[nH]cc2Br)C1=O N1(Cc2ccc(OC)c(Br)c2)CCC2CN(C(c3cnc(O)cc3O)=O)CCC12 C1(CC(=O)NC2NC(=O)N(c3cccc(C)c3C)C2=O)COc2ccccc2O1 Cc1ccc2oc(C(=O)NCC(C)(C)NC(c3cnc(C(C)O)s3)=O)cc2c1 C1(O)(C(N(CC(C)C(=O)NC(c2nccn2C)CO)C)=O)CCSCC1 N1(C(c2nn(C)c(C3CC3)c2)=O)CC(NC(c2ccoc2)=O)C(C)(C)C1 c1(C(N2C(C)CCC2C(=O)Nc2cc(Br)cnc2I)=O)ccc2nc(Br)sc2c1 C(C(N=c1[nH]nc(C(F)F)o1)C1CCC1)NC(c1ccc(=O)n(C2CC2)c1)=O C12COCCN1C(=O)COC2.C1(O)(CCNC(=O)OC(C)(C)C)CCN(C)CC1 C1CCN(C(c2nn(C)c(C3CC3)c2C)=O)C(C)C1.n1(CC)nncc1C(=O)N C(CN=c1[nH]c(=N)[nH]c(=NC(C)CC(=O)N(C)C)[nH]1)OCc1c(C)cccc1 CC(C)(C(=O)N1CCCC1(C)C(=O)NC1CC1)C(O)c1ccccc1.C1(C)CC1 c1(C(N2CC(CC(N3CCC(C)CC3)=O)C2)=O)cc(F)c(Cl)nc1Cl C=CCCCCCC(=O)NC(C)(CNC(=O)C=CCO)C1CC1 C=CC1CN(C(=O)CCc2cccnc2C)CC1NC(c1c(C)ccn1C)=O c1(C(=O)NCCC2CC(NC(C(CCC)(C)CC)=O)C2)cc2c(cn1)CCCC2 N#Cc1ccc(S(=O)(=O)Nc2ccc3c(c2)CCN3)c(Cl)c1 C1(C)(C(=O)NCCN(C(C(C)(C)OCC)=O)C2CC2)CC=CCO1 Cc1cc(C(=O)NC2(C)CCN(C(=O)CC3CC4CC4C3)C2)c(C)nc1C N1(C(C2CC(C)CC(C)C2)=O)CC(NC(=O)C(F)C(C)(C)O)C2CCCCC12 C1(C(N2CCC(N(CCC)C(c3cnc(O)s3)=O)C2)=O)CCCCC1O c1(-n2cc(CN(C(=O)C3=COCCO3)C)nn2)c(F)cncc1F c1(COC(C(=O)NC2CCN(Cc3onc(C(C)C)n3)C2)C)ccccc1F CCC(CC)CC(F)C(=O)NC(C)(CC)CO N1(C(C(CC2CC2)OC)=O)CC2C(NC(=O)CC(C)C)CS(=O)(=O)C2C1 C1(CCC)CN(C(=O)Cc2ccc(C)nc2)CC1C(=O)N(C)CC1CCCN1C Nc1cc(C(=O)NC23CC(C2)C3)cnc1Cl.C(=O)C(Cc1ccsc1)NC=O.N N1(C(C2C(C)(C)C2(C)C)=O)CC(F)(F)CC1(C)C.c1(C=O)cnc2n1CCC2.N c1(CN2CC3C(NC(CC4CCC(OC)CC4)=O)C3C2)ccc2c(c1)OCO2 C1(C(=O)NCc2cn(C)nc2)CCC(O)CN1C(c1cnn(CCO)c1)=O c1(C(N2CCCC(N(C(=O)CSC(C)(C)C)C)C2)=O)ccc(Cl)c(F)c1O Cc1c(C(=O)NCCOCCCN(C(=O)CCC(F)F)C)cnn1C N1(CC)CCN(CCN(C)C(=O)NCCC2COC2)CC1 c1(C(=O)NCCN(C(C2CCCCC(=O)N2)=O)CC)ccc2cc(Cl)ccc2c1 C1(C(N2CCC(C(=O)OCC)C2)=O)CCCN(C(=O)C(CC)(CC)OC)CC1 CCC(C)C(O)C(=O)NCC(CNC(=O)C(=O)Nc1ncc[nH]1)C(F)(F)F c1(OC)cccc2c(C(=O)NCC(C)(O)CNC(=O)C=O)csc12.C1CC1 N1(S(Cc2ccc(C)cc2)(=O)=O)CC2CCN(C(c3oc(C)nc3C)=O)C2C1 CCC(C(=O)N(CCNC(c1cc(CF)on1)=O)CC)C1CCC(=O)N1 C1(C(N(CC(O)C(C)(C)C)C)=O)C2CC3C(C2)C13.C12(C=O)CC1CNC2=O O=C(CCCCCCNC(=O)CC1CCSC1)NCC(F)F C1(NC(CC2(NC(C(C)OCC)=O)CCCCC2)=O)CC(O)C12CCC2 C12(C(=O)NCC(CC)(C)C)CCN(C(=O)C=Cc3cnccn3)CCC1C2 C1(CNC(C(C)Cc2ccsc2)=O)CN(C(=O)Cc2cnc[nH]2)CC1O CCCCCCCCCC(=O)NC1CN(C(=O)C(C)CCO)Cc2nccn2C1 C(=O)(CCC(=O)NC1(C)CC(NCc2ccsn2)C1)NCC CC(C)(CC(=O)NC1(CC(N2CC(O)C(O)C2CO)=O)CCC1)C(F)F Nc1cc(Cl)c(Cl)cc1C(N1CC2OCC(NC(C3(F)CCOCC3)=O)C2C1)=O C1(CC(N2CCC(C)C2)=O)C2CCC(C2)N1C(C1CCC(=O)N(C)C1)=O.CC c1(N2CCC(NC(c3cccc(OCCC)c3)=O)(CF)C2)cc(=O)n(C)cn1 N1(C(C(C(C)(C)O)F)=O)CCC(CNC(=O)COc2ccsn2)C12CCC2 C1(C(N2CCC(N(C)C(c3c[nH]c(-c4ccncc4)n3)=O)C2)=O)CC2(CC2)CO1 C1(C)CCCC1.C1(CC=O)CSCCS1.C1(C(N(C)C)=O)(C(=O)NC)CC1 CC(C)(O)CCCNC(=O)CNC(C1CCS(=O)CC1)=O CCCC#CC(C)(C)NC(C1OCCC1CNC(=O)C(O)C(C)(C)C)=O C1(C(N2CC3CC3(CNC(c3cccnn3)=O)C2)=O)(COC)CCCCO1 C1(N(C(CCC(=C)C)=O)C)CN(C(=O)Cn2nnnc2C2CC2)CCC1O c1(CNC(c2ccncc2Cl)C)cccc(-c2cccc(Br)c2)c1 C(=O)(CCCCCC(C)C)NCC(CNC(C(CC)CC1CCCC1)=O)F C1(OC)C2CC1CN(C(C1CC3(CCOC3)C1)=O)C2 N1(C(c2ncn(C)n2)C(=O)NCCOCC)CCC(C)CC1C(C)O C1(=CC(N2CCC(NC(CC(C=C)CC)=O)C2(C)C)=O)CCCCCC1(F)F C(C(C)CN=C(NC(C)C)N1CCN(C)C(=O)C1)Oc1c(OCC)cccc1 c1(C(=O)N)ccc(=O)n(C)n1.Cn1nnc(CNC(c2coc(C)c2)=O)n1 CN=c1[nH]c(C(=O)NCCCC(C)NC(C2(S(N)(=O)=O)CC2)=O)cs1 C12CC1CN(C(c1cc(C)n(C3CC3)n1)=O)C2.C(C)(C)(C(=O)N)OCC CC(c1ccccc1F)=CC(=O)NC12CCN(C(=O)CS(N)(=O)=O)CCC1C2 N1(C(c2nnc(C)s2)C)CC(NC(c2csnn2)=O)CC2(CCOCC2)C1 C(=O)(CC(C)(C)C)N(CC(C)NC(CN(C)CC)=O)CC N1(C(CC2(OC)CC2)=O)CCC2CN(C(=O)C=Cc3cccs3)CCC12 CC(C)(C#N)CCCC(=O)NC(CC(F)F)C(=O)NCC(O)CC(F)(F)F N1(C(CC2C(CNC(c3ccc(C)cn3)=O)C2)=O)CC2(CCC(O)CC2)C1 CCCC(C)(CC)C(=O)NC1CC2CN(C(=O)CCC3CC(OC)C3)CC2C1 N1(C(C=CC(C)C)=O)CCC2(CCN(C(C3CCCC(=O)N3C)=O)C2)C1 N1(C(Cc2cc(CC)no2)=O)CC2C(NC(=O)C(=Cc3ccco3)C)C2C1 Cc1ccc(C(C)C(N2CC3CC2(CNC(=O)C=Cc2ccsc2)C3)=O)cc1 CCCN=C(NN1C(C)CC1)NC1CCN(c2ccccc2)C1.c1ccccc1 c1(OC)cc(C(=O)NCCC(C)NC(=O)CCc2ccc(Br)cn2)nn1C C(=O)(C(C)(CO)NC(c1ccc[n+]([O-])c1)=O)NC(C)CC1CCCCC1 N1(C(CCC(C)NC(C2CCO2)=O)=O)CC(S(C)(=N)=O)C1 c1(Cc2cnc(C(=O)NCC3(C)COC3)s2)ccc(I)c(O)c1 c1(CCC(=O)NC(C(=O)NC(C)C(=O)NCCF)C)nc(O)n[nH]1 CCC(CNC(c1c(C)nn(CCO)c1C(F)(F)Cl)=O)(CC)CC c1(N2CCC(CC(=O)N(CC)CC)C2)ccnc2c(F)cccc12 C1(C(=O)NCCN(C(=O)Cc2cnns2)CCC)CC1C1CC(F)(F)C1 c1(C(CO)NCC(C)CC2CCCC2)ccc(Cl)cc1Br N1(C(c2ccc(C)c(F)c2)=O)CCCC2(C1)CN(C(C1(n3cncn3)CC1)=O)C2 C(=O)(C#CC1CCOCC1)NC(C=CC(N1CCCC(OC)C1)=O)C C1(O)(CC)CCCN(C(=O)CC2(O)CCC2)C1.C1(C(=O)N)CCCC2(CC2)C1 c1(C(=O)NC(C2(C)CC2)C)cnc2cccnn12.C1CCCOC1.C(=O)(C)N Cc1cccc(C)c1C(=O)NCC1CC(NC(=O)C(C2CCCCC2)O)CCO1 CN1C(=O)OC2CN(C(=O)C)CC12.C1(C#N)(C=O)CC(F)(F)C1.C1CCC1.O C#CCC(CC#C)C(=O)NCC(CNC(c1ccc(C)c(C#N)c1)=O)OC C(=O)(CCCCC)N1C(CNC(C(C)OCCC#C)=O)CC1 Cc1sc(C)c(C(=O)NC(C)CN(C)C(c2cn(C)cn2)=O)c1C#N c1(C2C(C(=O)NCC(CO)NC(CC(C)C)=O)C2)ccccc1F c1(C(=O)Nc2cc(OC)cc(OC)c2)ccc2ccn(C(C)C)c2c1 Cc1cc2[nH]c(C(=O)NC34CC3CN(C(=O)Cc3ccc(Cl)c(Cl)c3)C4)cc2s1 Cc1cccc(C(=O)NC(C)C(=O)N(C(CO)C2CC2)C)c1C N1(C(c2cc(C)c(C)nc2)=O)CC2CCC(C1)N2C(=O)C(c1cccc(Br)c1)O C(=O)(C(CNC(c1sccc1CO)=O)C(C)(C)C)NCCC(C)N1CCC1 N1(C(C=CCOC)=O)CCN(C(C2CCCC(=O)O2)=O)C(C(C)C)C1 C12(C(=O)NCC(C)OC)CC(C)(CN1C(=O)C(C)(C)c1ccno1)C2 Cc1noc(C(c2nnnn2CC2CCCO2)NC2CC(CCO)C2)n1 CCC(COC)C(=O)N1CCCCC1C(=O)NC(c1nccc(O)n1)C Cc1c(CC(N2CCCC2CNC(c2cc(Cl)ns2)=O)=O)cccc1Br C(CC1=CCN(C(c2cccnc2C(F)F)=O)CC1)NC(C1(F)C(C)OCC1)=O C(C(C)(C)C(=O)NC(C1(O)CCCCC1)C)N(C(CC1C(CC)C1)=O)C C(=O)(C(O)CC(C)(C)C)N(CCCCCC(=O)N1CCCC(C)(CO)C1)C C(=O)(C1=C(C#N)CCC1)N1CC(NC(COC(CC)C)=O)C(SC)C1 c1(C(=O)NC2CC(O)CN(C(=O)CCC3CCC3)C2)cc2c(F)ccc(F)c2[nH]1 C(C(C(=O)NC(C1CCCN1C(=O)CCC1CCC(=O)C1)C)OC)OC C(C(=O)NCc1ccccc1)(C(C)(C)C)OC(C(Cc1c(C)cccc1)C)=O N1(C(C2C(CC)C2)=O)CCC2(C1)CN(C(c1sc3nccn3c1C)=O)C2 C(CCNC(=O)CCc1cnccn1)(C(=O)NC(C)CC(C)C)OC N1(C(c2ccc(N(CC(C)C)C)cc2)=O)CC(NC(=O)CCC(F)F)C2(CC2)C1 C1(NC(c2c(C)ncnc2C)=O)COC2(CCN(C(=O)Cn3cnnc3)C2)C1 c1(NC(C)(C)C)ccccc1NS(=O)(=O)CCc1cccc(Cl)c1 N1(C(c2c(C)cc(F)cc2)=O)CC(NC(=O)CCSCC(N)=O)CC(F)(F)C1 c1(C(N2C(C(C)C)CN(C(C3CCC(=O)C3)=O)CC2)=O)cnc2c(n1)CCCC2 c1(C(N(CC(CNC(COC)=O)(C)C)C)=O)ccc([N+](=O)[O-])c(C)n1 C(=O)(CCC(F)F)NC1CCC(NC(CC=CC(C)(C)C)=O)C1 C1(CNC(c2c(CC)c[nH]n2)=O)CC(NC(=O)CCc2scnc2C)CC1O C1(NC(c2nc(C)sc2)=O)CCN(C(=O)CCn2c(C)ccc2C)C1C C1(C(=O)NCC(CCNC(c2c(CC)n(C)nn2)=O)O)COCCC1(F)F N1(C(C(C)(C)C2(O)CCC2)=O)CC(NC(c2ccc(F)c(O)c2)=O)C(C)(C)C1 C1(CC=C)(NC(=O)C(CNC(C2C3CCC(F)C23)=O)N(C)C)CCCCC1 C1(NC(C(C)OC2CCCC2)=O)CCCN(C(=O)CCc2cccs2)CCC1 CCCC(CNC(=O)CSCC)C(=O)NCC1(C#N)CCCCC1 c1(C(=O)NCCC(=O)NCCCC2C(C)C2)cccc2c[nH]nc12 CC(CC(C)NC(=O)COCc1ccccn1)NC(=O)Cn1ccnn1.C c1(C(N(C(CCNC(C2(CC=C)CCCC2)=O)C)CC)=O)cccn2nncc12 c1(NC(=O)C(N2CCN(Cc3cccc(C4CC4)c3)CC2)=O)cc(Cl)nc(Cl)c1 N1(C(CCC2CCCCN(C(C(CC)(C)OC)=O)C2)=O)CCC2(CCCC2)C1 N1(C(C2(C(N)=O)CCC2)=O)CCC2(CC1)CC(NC(=O)C1=C(Cl)CC1)C2 N1(C(C)C)CCCC(C(=O)N(C(C)CCNC(c2cccc(C(F)F)n2)=O)C)C1 C(=O)(C#CC1CCCCC1)N1CCC(N(C(C(C2CC2)OCC)=O)CCO)C1 C(=O)(C(CC(F)(F)F)c1ccccc1)NCCCN(C(C(CC)NC(N)=O)=O)C c1(OC)ccc(C(C)C(=O)NCC=CC)cc1.C1(C(=O)N)CC1C1CCC1 c1(CC(=O)NC2CC(NC(c3ccoc3)=O)C(O)C2)cccc2nonc12 C(=O)(C1SCCc2ccccc21)N1CCC(C)N(C(=O)Cc2cccs2)CC1 CC(O)C.C1(C=O)CCC1.C1CC(C(F)(F)F)C1.CC(C)(C)OC(=O)N C1(C(N(CCOC)CC)=O)CNC(=O)CC1(C)C.c1(C=O)cccc(C)n1.N CC1(C(=O)NC2CCCC2CCO)CCCN1C(c1csc(CO)n1)=O C1(NC(c2cncc(C)c2Cl)=O)C(C)CCN(C(c2csc(Cl)c2)=O)C1C c1(C(C(=O)NC)N(CC(C)C#N)C)cc(COC)ccc1F c1(C(N2CCCC(N(C(C(C)NC(CC)=O)=O)C)C2)=O)cc(Cl)cnc1O N1(C(C=C(CC)CC)=O)Cc2ccccc2CC1CNC(C1CCOC1)=O c1(C(=O)NCCCN(C(CC(C)CF)=O)CCO)cc(F)cc2c1CCC2 c1(C(=O)NCC(CO)NC(c2csc(C)c2N)=O)cccc2ccn(C)c12 c1(C(N2C(C)CC(NC(c3nc(C(C)C)oc3)=O)C2)=O)ccc(F)c(Cl)c1 C(C(C)C(F)C(=O)N(CCCOC(C)C)C)NC(CCOCC)=O N1(C(C=C(C)C)=O)CCCC2(C1)CN(C(C1(O)CN3CCC1CC3)=O)CCO2 C1(C(N2CC(CN(C)C(C3CC4CCC(C3)O4)=O)OCC2)=O)CN2CCC1CC2 c1(C(=O)NCCCNC(CC(N2CCCCC2=O)C)=O)ccnc(C(N)=O)c1 C(C)(CO)(C(=O)NCCOCCNC(C1(C#N)CCCC1)=O)N(C)C N1(C(c2ccc3c(c2)CNC3)=O)CCC2(CC1)OCC1CC21 C1(NC(c2ccc(C)c(C)n2)=O)COC2CN(C(C3CCC(C)(O)CC3)=O)CC12 N1(C(C2(CC#C)CCCO2)=O)CCC(CC(C)NC(=O)C(C)CO)CC1 C1(C(=O)NCc2cc(C)on2)CCC(CNC(=O)Cc2cccnc2F)CC1 O=C1CC(C(N2CCC=CC2C(=O)NCCCN2CCC2)=O)C(=O)N1 C1(CC)(NC(c2cc(C3CC3)cs2)=O)CCN(C(=O)CCOC2CC2)CC1 CC1CN(C(c2cc3ccsc3[nH]2)=O)CC2(CCN(Cc3ccccc3F)C2)O1 CC(N=[N+]=[N-])C(=O)NCc1cc(C(=O)NC(C)CCO)no1 Cc1nc(C(N2CCCC(C(C)NC(=O)CS(N)(=O)=O)C2)=O)n(C)n1 CC1CN(C(=O)CCCN=[N+]=[N-])CC(C)N(C(c2cnn(C)c2F)=O)C1 c1(N(C(c2nc(O)c(C)s2)=O)CC2COCC2)ccc(O)c(F)c1F.CC=CC [N-]=[N+]=Nc1cncc(C(=O)NC2CCCC2C)c1.C12(C(=O)N)CCCC(CO1)C2 c1(C(=O)NC2C(NC(c3c(OC)cccn3)=O)CC2)ccc2cc(Cl)ccc2c1 CCC1=C(C(=O)NC2(C3CN(C(c4c(C)ccc(C)c4C)=O)C3)CC2)CCCO1 N1(C(C(CNC(c2c(C)cccn2)=O)CC2CCCC2)=O)CC2C(C1)C2(F)F N1(CCC)CCC(C(=O)N(C2CC(NC(C3(C(=O)O)CCC3)=O)C2)C)CC1 Cc1ccc(F)cc1NC(=O)Nc1ccc(Cl)cc1.C1(C(=O)N)CNC(=O)C1 S(=O)(=O)(c1ccc(N2CCCC(c3ncco3)C2)c(Br)c1)N1CCCC(C)(F)C1 c1(N(C(C)=O)C)ccccc1C(N1CC(F)(CNC(C2CCC2C)=O)C1)=O CC(C(=O)N(CCCNC(=O)C(C)=C1CC1)C(C)C)=C1CC1 N1(C(=O)COCc2cccnc2)CCN(C(C2COCCN2CCO)=O)C2CCC12 CC(C)(O)C(C)(C)C(=O)NCc1ccc(C)cc1.C(=O)CS(=O)C(F)(F)F C1(C(=O)NC2C3CN(C(C4NC(=O)OCC4)=O)C2C3)CCOCC12CCC2 N1(C(CSCCC#N)=O)CC(NC(C2CCCCO2)=O)C(F)C1 C1(CC)CN(C(=O)CCc2cnccn2)CCC1NC(c1n[nH]c2c1COC2)=O CCC(C#N)C(=O)NC(CCNC(c1sc(Br)cc1Cl)=O)C(C)C c1(C(=O)NC2C3CN(C(C=CSC)=O)C(C3)C2)cn(C)c2ccccc12 N1(C(c2ccoc2)=O)CC2(CNC(C34CCCCC3C4)=O)CCC1CC2 N1(C(C(COC)OC)=O)CC(NC(=O)CN2CCCCC2C)C2(CCOCC2)C1 C1(C(=O)NC2C(CC)CN(C(=O)C3=CCCCO3)CC2)CC(C)(C)OC(C)(C)C1 CC(C)C(CCNC(=O)Cc1cc[nH]n1)NC(c1ccncc1N1CCCC1)=O c1(C(=O)NC(CO)CCCNC(=O)C(O)c2ccsc2)cn2ccccc2n1 c1(C(N2CCN(C)C(=O)C2c2ccccc2)=O)cc2cc([N+](=O)[O-])ccc2n1C c1(C(=O)NCC(C)NC(c2cnn3c2CC(F)(F)C3)=O)cccc2c1ccn2C CCCCCC(O)C(=O)NC1C(C)CCN(C(C23CC(CO2)C3)=O)C1C C1(CN(C2C=C2C)CCC)CCCC1 CCC(COC)C(=O)NCCN(C(=O)CCC1CCCN(C)C1)C1CC1 Cc1ccc(NC(C2CC(C)CN2C(c2ccc(C(F)F)o2)=O)=O)cc1C C(C(=O)N=c1nc(C)[nH]s1)NCc1ncc(OCC)nc1 N1(C(CSCC)=O)CCC=C(C(=O)N2CCCCC2CC(=O)OC)C1 C(=O)(CC(C)C)N1CC(CC)(NC(C2CN(C=O)C2)=O)C1.C(C)=O.O Cc1noc(-c2cn(CC(N3CC(C)(NC(=O)C(O)C4CCCC4)C3)=O)cn2)n1 c1(CC2(C(=O)O)CN(C(C3(c4ccccc4)CC(=O)C3)=O)C2)ccccc1F c1ccc(F)cc1.C1(CC(=O)NCC2CC2NC(=O)CCO)CC1(Cl)Cl c1(N(C)C)ccc(CCC(=O)NCC2CCN(C(=O)C=Cc3cncs3)C2)cc1 N1(C(c2scc(C(=O)OC)n2)=O)CCCC(CN(C)C(c2ccn(C)c2)=O)C1 N1(C(N(CC(CC)O)C)=O)CCN(C(c2nc(=N)[nH][nH]2)=O)CC1 Cc1[nH]c(=NCC(O)C2(C(=O)O)CCC2)ccc1C(F)(F)F C(=O)(C1CCCc2c(O)cccc21)NC1CN(C(c2cc(C)c(Cl)cc2C)=O)C1 Cc1noc(C(N2CCCCC2CN(C)C(C2OCC2(C)C)=O)=O)c1C c1(CCC)nc(C)c(C(=O)NCC(C)CNC(=O)CC2CCC(C)C2)o1 CCCCCC(C)(C)C(=O)NCCC1CCN(C(=O)C(F)C(C)(F)F)C1 C1(C)(C(N(CC(C)(C)C)CCCO)=O)CC(O)CN1C(=O)CSC1CC1 c1(C(N(CCCN(C(C(CC#C)O)=O)C)C)=O)cc2c(cc1Cl)OCO2 c1(CC2N(C(CC(C)=C(C)C)=O)CCC2)ccccn1.C1(CC(=O)N)CCC1 CC(c1ccccc1F)=CC(N1CCC(NC(=O)C(C)O)C12CC2)=O C1(NC(c2cn(CC=C)nn2)=O)CC12CCN(C(c1c[nH]c(=N)nc1C)=O)CC2 C1(C2(O)CCC2)(C(=O)NCC(C(=O)NCCC(C)C(F)F)O)CC1 Cc1cc(C)c(C#N)c(NC23CCCC2CN(C(=O)CCOC(C)C)C3)n1 C1(C2CCN(N3CC(C(C)(C)C)(CO)C3)CC2)(C(=O)OCC)CCOCC1 C1(C(=O)NCC2CCCCN2C(c2cnc(S)nc2)=O)CCn2c(O)nnc2C1 N1(C(c2c(CC)con2)=O)CCC(C(=O)NC2CC(C)(C)OC2(C)C)=C(F)C1 c1(C(N2CCC(C(C)NC(C(C)C(F)(F)F)=O)CC2)=O)ccnc2c1cnn2C CCCCS(=O)(=O)CC(=O)NC1CC1C.c1(C(=O)N)nc(-c2nc[nH]n2)sc1C C(=O)(C1CNC(=O)c2ccnn21)N1CCN(C(c2c(C)scc2)=O)CC12CCC2 c1(CNC(N2C(CC#C)CCC2)=O)c(F)cccc1F.c12ccccc1OC2 C1(C2CCN(C(c3cc(Cl)on3)=O)CC2)(NC(C=C(CC)CC)=O)CC1 c1(C(=O)NC(CC)CN(C)C(C23CCC(F)(CC2)C3)=O)cc2c(s1)CCCC2 N1(C(C2(C#N)CC2)=O)CCC(NC(c2conc2C(F)(F)F)=O)C(O)C1 C(=O)(CCCN=[N+]=[N-])N(C1CCN(Cc2cc(C(F)(F)F)n(C)n2)C1)C C1(O)(C(C)NC(c2ccc(C)nc2)=O)CCN(C(=O)C(O)Cn2cncn2)CC1 N1(C(CN)=O)CC2CCCC(Nc3ccc(NC(N4CCCC4)=O)cc3)C2C1 C1(C(N2C(CN(C)C(c3ccc(O)nc3)=O)COCC2)=O)CCCC(C)(C)C1 C(=O)(C(C)C(C)(C)C)NC1(CO)CN(C(C2(C)CC(C)C2)=O)C1 c1(CC(=O)NCC(C)NC(C2CCCN2c2nccs2)=O)ccnn1C N1(C(=O)C(F)C2CCOC2)CC2(CCCN(C(C3CC(O)C3)=O)C2)C1 C1(C(N(CC(C)(C)NC(C2CC(C)(C)CO2)=O)C)=O)CC2CC1CC2O CC1OC2(C(=O)N(CCCNC(C3OCCOC34CCC4)=O)C)CCC1CC2 c1(CCC(=O)N)nc2ccccc2[nH]1.C=C(C)CCNC(=O)Cn1cc(C)cn1 c1(CNC(C2NC[Si](C)(C)C2)=O)ccc2c(c1)CCCC2=O c1(CCC(N2C(CN(C(C)=O)C)CCC2)=O)cncc(F)c1 N1(C(C(CC)(CO)OC)=O)CC2CCC1CN2C(c1cc[nH]c(=N)c1Cl)=O c1(C(c2nnnn2CC2CCOC2)NC2(CC)CC2)conc1C(C)(C)C C#CC1CCC(C(=O)N(C2CN(C(c3ccc(OC)cc3OC)=O)C2)C)CC1 O=C1CC(C(N2CC(F)CC2CNC(C2CC2CF)=O)=O)NC(=O)N1 C1(NC(CCC=C)=O)CN(C(C2CC2c2ccncc2F)=O)CC1CC1CC1 N1(C(CC(CC)CC)=O)CCCC12CCN(C(C1CC3COCCN3C1)=O)CC2 c1(C2(C(N3CCC3CNC(C3(C(F)F)CCC3)=O)=O)CC2)ccncc1 N1(C(CC(c2cccc(Br)c2)C)=O)CC(NC(=O)CC2CCC2)CC1(C)C C1(C(N2C(C)CC2C(=O)NCc2ccsc2)=O)CC2(CSC2)C1 C1(C(N2CCC(C#CC)C2)=O)Cc2ncccc2N1 C1(O)(CCNC(C2CC23CC3)=O)CCCN(C(c2cnc3sccn23)=O)C1 C1(O)(CCNC(c2ccn(CC)n2)=O)CCN(C(C2C3CCCC23)=O)CC1 c1(C(=O)NC2CN(C(c3c(CC)csc3)=O)CC2C)ccc(OC)c(F)c1N C1(C(F)(F)F)(C(=O)NCCC(C)NC(C2(C)COC2)=O)CCCCO1 c1(C(=O)NCC(CC)NC(=O)C(C)C2CCOCC2)cnnc(O)c1.C1CC1.O C1=CCOc2c(OC)ccc1c2.C=C=C1CCC(CC)CC1 C1(C(N2CC(n3cc(-c4ccc(C)nn4)nn3)C2)=O)(CC)CCCS1(=O)=O c1(NCCC(=O)N(C)C)nc(N2CC3C4C=CC(O4)C3C2)nc2scnc12 C1(C(=O)NC(C(C)O)(C)C)CN(C(c2ccc(C#N)o2)=O)CCN1C c1(C(=O)NCC(CO)NC(C=C(C)C2CCCCC2)=O)cc(Cl)cc(C)c1N Nc1cc(Cl)nc(Cl)c1C(N1CC=CC(NC(C2CC3(C2)CC3F)=O)C1)=O C1(C)(C(=O)NC2C(C)(NC(c3cccc(C)c3)=O)CCC2)CCCCCC1 C1(C(=O)NCC(C)NC(=O)CCC(=O)N(C)C)CCCN1S(=N)(=O)N(C)C C1(CNC(C(SC)SC)=O)CN(C(C2CC=CCC2)=O)CC1C c1(C(=O)NC(C2CCN(C(C3(OC)CC3)=O)CC2)C)cccc2c1OCCCO2 C1(CNC(c2n(CC#C)ccc2)=O)CN(C(=O)C(CC)CC)CC(C)(C)O1 C(=O)(C1=C(Cl)CCCC1)N1CCCC(COC)(NC(c2ccc(OC)cn2)=O)C1 N1(C(C2C(C)(CC)C2)=O)CCC2(CCCCC2NC(c2cccc(C)c2)=O)C1 Cc1cc(C(=O)N(C)CCN(C(=O)C(O)Cc2cc(Cl)cc(Cl)c2)C)cc(C)c1 N1(C(CC2CC(C)C2)=O)CCCC(NC(=O)C=C2CCSCC2)C1 C1(NC(c2ccc(C3CCCC3)o2)=O)CC2CCC(C1)N2C(C1SCCS1)=O c1(-c2nccc(-c3scc(C(=O)Nc4cc(CC)on4)n3)c2)ccc2c(c1)CCO2 N1CCC2(CCC(N(c3ncnc4[nH]ccc34)CCC)CC2)CC1.SC CCC(=O)CCC(=O)N1CC(C)(C)CC1C(=O)NCc1cn(C(C)C)nn1 c1(C=O)cc(S(N)(=O)=O)cn1C.C(C(C)(O)CC(=O)NCC(C)C(C)C)OC c1(CC)ccc(C(=O)NCC2CCC2)cn1.n1(CC=O)cc(C2CC2)cn1 c1(CC2N(C(=O)NC3CCC(OC(F)F)CC3)CCC2)ccc(F)cc1F N1(C(C=C(C)CN2CCOCC2)=O)CC(C2CC2)C1.C1(C=O)CCC(C)=C(C)C1 N1(C(C(F)OC)=O)CC2CN(C(=O)CC3(C)CC(F)(F)C3)CC2(C)C1 N1(C(CC(CCSC)O)=O)CCN(C(=O)CSC(C)(C)C)CC(C)(C)C1 c1(C(c2nnnn2Cc2ccco2)NCC(=C)Br)ccc2c(c1)CCC(=O)N2C N1(C(CCn2ccc(C)n2)=O)CC(CC(N2CC(S(C)=O)C2)=O)C(C)C1 C(=O)(C(CCC1CCC1)NC(=O)CC1C=CCC1)NCCc1ncn(C)c1 c1(OC)cc(C)ccc1-c1cnc(CNCc2cncnc2)nc1 c1(C(=O)NC(CN(C(C(C2CCCC2)OC)=O)C)C)cc(Cl)c(N)c(Cl)c1 N1(C(CCCCCNC(C)=O)=O)CC2(CC(C(=O)NCC(C)(C)CO)CO2)C1 c1(C(=O)NC2C(NC(C(OC)OC)=O)COC2)cccc(C2CC2(F)F)c1 CC1=NS(=O)(=O)NC(C)=C1CC(=O)NCCCC(C)NC(=O)C(C)CF n1(CC)cc(NC(C2CCCCN(C(c3cc(C)nnc3C)=O)C2)=O)c(C#N)n1 Cc1cc(Cl)ccc1C(N1C2CCC1(CNC(C1CCCC(F)(F)C1)=O)CC2)=O CC1(C)C(NC(C2SCCCS2)=O)CC1CNC(=O)C1=NOCC1 c1(CC)onc(C(N2CC=CC2C(=O)NC(CN2CCCC2)CO)=O)c1C N1(C(C(=O)N(C)Cc2nc(Br)cn2C)=O)CCC2(CC1)CS(=O)(=O)C2 c1(C(=O)NC2C(CNC(c3c(CC)noc3)=O)C2)ccc(F)c(C)c1N C1(NC(CC(C)NC(N)=O)=O)CCN(C(=O)C=Cc2ccc(O)cc2)C12CC2 CC1(C(N2CCC(C)(NC(c3csc(F)c3)=O)C2)=O)CCSCC1 n1(-c2ccn(C(C)C)n2)nc(-c2ccc(Cl)s2)nc1C(O)Cn1cncn1 N1(C(CC(C)n2ccnc2)=O)CCC2CN(C(c3ccnc(CO)c3)=O)CCC12 C1(CC=C)CCCN(C(=O)C(=O)N(C)Cc2cncnc2)C1 c1(C(N2CCC(CCN(C(=O)Cc3cncs3)C)CC2)=O)cc(C#N)ccc1N c1(C(N2CCCC(C)(CNC(CCOC(C)C)=O)C2)=O)ccc2nc[nH]c2c1F C1(C(N(CC)CC)=O)CCc2nccn2C1.c12cccc(c1)SC2 c1(OC)c(C)csc1C(=O)NC1CCC(CC)C1.c1(C(=O)N)ccc(C)nn1 C1(NC(=O)CCc2ccc(F)nc2)CC2CN(C(C3CCCO3)=O)CC2C1 CN1CCC(OCC(N2CC(N(C)C(C3(C)CC4CC4C3)=O)C2)=O)CC1 C1(NC(C(C)NC(c2ccco2)=O)=O)C2CN(C(C3CC=CC3)=O)CC12 c1(C(N2CC(CC)C2)=O)cn(C)c(=O)n(C)c1=O.CC(CC1CCC1)C(=O)N C1(C(N)=O)(CNC(C2CCC2)=O)CCCC1.c1(C=O)coc(C(F)F)n1.N C(=O)(C(O)CCC#C)N1CCC(CC#C)(NC(=O)C=CSC)C1.C(=O)CCCC c1(OC)cccc2c1CCCC2NC(=O)C(c1ccc(=O)n(C)c1)(F)F C(=O)(C1=Cc2cccc(Br)c2OC1)NC(C(C)NC(C(COC)C)=O)(C)C CC1=CCC(NC(C2(CCNC(=O)CC3(O)CCOC3)CCCC2)=O)CC1 C1(N(C)C(c2cnc(C(F)F)s2)=O)CCC(NC(=O)CO)C1.C1CC1.C C1(COC)(NC(=O)C(C)CN2CCCCC2)CCN(C(c2cnc(C)[nH]2)=O)C1 c1(C(=O)NC2CC(C)N(C(c3ccnn3CCF)=O)C2)ccc2c(O)n[nH]c2c1 N1(C(=O)NCC2CN(CC)C(=O)O2)CC2(C)CS(=N)(=O)CC2(C)C1 c1(C(N2CC(C)(NC(C3OCC(C)C3)=O)C2)=O)cc2c(cc1N)CCCC2 c1(CCC(=O)NC2C(C)CN(C(C3CC3(C)C)=O)CC2)cncc2ccccc12 C1(NC(CCC(=C)Cl)=O)CCN(C(c2cn(C3CCOC3)nn2)=O)CC1O N1(C(C2CC(OC)C2)=O)CC(NC(C2CC3CCC2C3)=O)CCC1C C(=O)(C1Cc2ccccc21)NCC1CCCN(C(C=C(C)Cl)=O)C1 C1(C(N2CCCC(C#C)C2)=O)CC(C)(C)CC(C)(C)C1 CCC(CC)CCCC(=O)NC1(C(=O)NOCC2CCCO2)CSC1 n1(CCC(=O)NC2CCCCC2NC(C2CC3CC2C3)=O)cnc2ccccc12 CC(F)(F)CCC(=O)NC1CC2CC1CN2C(c1cc(F)ccc1C(F)(F)F)=O C1(C(=O)NC2C(C=C)CN(C(=O)C=C3CCCC3)C2)CCn2nnnc2C1 c1(OC)cc(O)ncc1C(=O)N.C1CC(C)N(C(=O)C=C(C)c2ccco2)C1 C1(C(=O)NCC(CNC(c2n(C)cnc2Br)=O)O)CC12CC(C)(C)C2 C12(NC(c3cn(CCCC)nn3)=O)CN(C(=O)CC(C)C)CC1CS(=O)(=O)C2 c1(CC(=O)NCC2C(C)CN(C(=O)C3=C(Cl)CC3)CC2)c[nH]c2ccccc12 N1(C(C(C(C)C)O)=O)CCC(C2CC2)(CNC(=O)C(C2CCOCC2)O)C1 N1(C(CN(C(c2ccc(CC)cc2)=O)C2CC2)=O)CC2(COC(=O)N2C)C1 c1(C(C)(CC2C=CCC2)NCCC(=O)NC(N)=O)nnnn1CC1CC1 Cc1cc(=O)n(C)cc1NC(=O)CC1(NC(c2ccccn2)=O)CC1 CCC1=C(C(=O)N2CC=CC2(C)C(=O)NCC2SCCS2)CCCO1 C(=O)(CC(F)(F)C(F)(F)F)N1C(CNC(CCCC(C)=O)=O)CC1 N1(C(C)=O)CCN(C(C2(c3ccc(Cl)cc3)CCOCC2)=O)CC1C(=O)O c1(-n2c(NC(C3C(C)CCO3)=O)ccn2)ccc(Cl)c(Cl)c1 Cc1c(C(=O)NC2COC3C(NC(=O)CN(C)C)COC23)oc2c(Cl)cccc12 c1(CN2CC3N(C(c4c(F)cncc4F)=O)C3C2)c(Cl)cnc(Cl)c1Cl c1(C2(C(=O)NC(C)CCNC(=O)C3CC3)CC2)ccc(F)c(Br)c1 Cc1[nH]c(=N)sc1C(N1CC2CC2(C)C1)=O.c1(C=O)cscn1.C(=O)(C)N C#CC1(C(=O)NC(CNC(=O)C(c2cnn(C)c2)C)C2CC2)CCC1 C(=O)(C(C)(C)CC(F)(F)F)N1CC(CC)N(C(=O)CSCCC(F)(F)F)CC1 c1cccc(C(C)=O)c1.C=CC(C(=O)N1CC(NC(=O)CO)C1)c1ccccc1 C1(C(=O)NC(CC)CNC(c2cncc(C)c2Cl)=O)CCc2ccnn2C1 CC(=O)C(C)(C)CC(=O)NC(CO)C(=O)N(C)Cc1cnccn1 Cc1cc(C(N2CSCC2C(=O)NCCOCC2CC2)=O)ncn1 C(C(=O)NCC(C)(C)C1CCCO1)(C(C)O)NC(C(COC)N(C)C)=O c1(C(N2CCCC2)=O)cc(F)c(F)c(Cl)c1F.C(C(=O)N)(C(C)C)SCC.C c1(CC)c(C(=O)NCCC2CCCN(C(=O)Cc3ccsc3Cl)C2)cnn1CC CC1CN(C(C23CC(C2)C3)=O)CC(C)N(C(=O)Cc2cccc3cccnc23)C1 CC1CC(NC(c2ccc(Cl)nc2N(C)C)=O)CCN1C(=O)CCc1ccco1 c1(OCCNC(C(=O)N(CC)CC2CC(O)C2)=O)ccc(F)cc1 C1(NC(CCc2n(C)ncc2)=O)COC2CN(C(=O)COC3CCCOC3)CC12 C(CCCCCNC(=O)CCc1cnc(O)[nH]1)N(C)C(C1(C(F)F)CCCC1)=O Cc1cc(=O)c(C(N2CC(N(C(=O)CNC=O)C)C(C)(C)C2)=O)cn1C CCCC(O)CCN=c1nc2c(ncn2C)c(NCCC2CC2(Cl)Cl)[nH]1 C(=O)(C(C(C)C)C(C)C)NC(CC)(C)CCNC(=O)C(O)C(F)(F)F Cc1cc(Cl)ccc1C(=O)NC1CCC1NC(=O)Cc1nc[nH]n1 C1(CC(=O)NCCN(C(=O)CCC2(C)CC2)C)CCOC(C)(C)C1 C1CCN(C(=O)CC2CCCS2(=O)=O)CC1.c1(CC)oncc1C(=O)NCC C1(CCOC)CCOCC1(c1nnnn1C1(C)CC1)NCc1cnc(C)n1C C12(CNC(C(CC)C)=O)CCC(CC1)N2C(c1snc(C)c1N)=O c1(N(C)C)cc(C(=O)NCCCCNC(c2ccnc(Cl)n2)=O)ccc1[N+](=O)[O-] CC(C)(C)CC(O)C(=O)NC1(CC(=O)NC2CCC2CO)CC1 c1(C(=O)Nc2ccc(C#C)cc2)cc(S(=O)(=O)C(C)C)ccc1OC N1(C(C(C(CC)C)O)=O)CCCC2(NC(=O)C#CC(=O)N(C)C)CC2C1 c1(C(=O)NC2CCN(C(C(N3CCOCC3)C)=O)C23CC3)cc2ccccc2o1 N1(CC)CC(NC(=O)CC(O)CNC(c2c[nH]cc2C)=O)C(C)C1 c1(CC=O)cc(F)cc(Cl)c1.n1(CCOC)cc(C(=O)NC2CC2)nn1.N c1(SC)ccccc1NC(=O)CC1CCN(C(=O)C)C1.c1(C=O)cccs1.N C1CN(C(C2CC2(C)C(F)(F)F)=O)CCC1C.c1(CCC)occc1C(=O)N.C N1(C(c2ccc(C)cn2)=O)CC2CC3CC2C1C3NC(C1C2CC3C(C2)C13)=O C1(C=O)CC2(C1)CC(C(F)(F)F)C2.C(CC)(C(=O)N)OCC.CC(C)C C1(NC(C(C)N(C)C)=O)CCCN(C(=O)CC2(CS(C)(=O)=O)CC2)C1C C1(OC)COCCC1CC(N1CCCC1)=O.C1(CC(=O)N(C)C)CCC(F)(F)C1 O(CP(C)(C)=O)CC(=O)N(C1CC(NC(=O)C=Cc2cscn2)C1)C Cc1cc(O)ccc1C(N1CCOCC(NC(C2CCN(C)C2=O)=O)C1)=O C1(n2cc(CCCSC)nn2)CCC(C)(C)N(C(=O)C(O)C(C(C)C)OC)C1 C1(C(N(C(=O)CCC2CCC2)C2CC2)=O)CC(CC)C1.C(C(=O)N)OC C1(N(C(c2c(CC)[nH]cc2)=O)C)CCN(C(c2nccc(OC)c2N)=O)CC1C N1(C(C2(CC#C)CCOC2)=O)C2CCC1(CNC(c1c(C)noc1C)=O)CC2 C1(NC(C2CCC2)=O)(CF)CCN(C(=O)Cc2c[nH]ccc2=O)C1.C1CC1.C N1(C(CS(CC)=O)=O)CC2CCC1C(CNC(C1CCC(=O)C1)=O)C2 c1(C(=O)NC(C)(CNC(c2ncccn2)=O)C2CC2)c(Cl)nsc1Cl Cc1nnn2c1CN(c1nc(NC3CCC(O)C3)c3ccsc3n1)CC2 c1(CC)ccsc1C(=O)NC(CNC(=O)C(C1CCCC1)OC)CO c1(C(=O)N)cccc(Cl)c1C(F)(F)F.C1(O)CN(C(=O)CCc2cnco2)C1 C1(NC(C(C)NC(N)=O)=O)COCC1CNC(c1cncs1)=O C(C1=NOC2CN(C(C3CCC3)=O)CC12)NC(C1=C(C)CCCC1)=O C=CC1(C(=O)NC(CNC(c2cccnc2S)=O)CC(F)(F)F)CCOCC1 Cc1cc(=NC2CCCCN(C(c3nc(Cl)sc3Cl)=O)C2)[nH]c(C(F)(F)F)n1 C#CCC(O)C(=O)NCC(O)C(=O)Nc1cccc(C(C)F)c1 C1(NC(c2cc(OC)c(F)cc2)=O)COC2CN(C(C3CCC3C(F)F)=O)CC12 n1(CC(N2CC(NC(C(C)C(F)(F)F)=O)C(F)C2)=O)sc2ccccc2c1=O C1(C2N(C(C3CCC=CO3)C(=O)NCC(=C)C)CCC2)CCCCCC1 CCC(CNC(=O)C(C)CN(C)C(c1ccnn1COC)=O)CCO C=CCCCC(=O)NCC1CCN1C(=O)CNc1cnn(C)c1 CC1CN(C(=O)C#CC2(C)CC2)CC2(CCN(C3CCN(C(C)C)C3=O)C2)O1 C(=O)(C(CC(=O)O)N1CCCCCC1)NCC(CCC)O c1(C(N2C(C)(C(=O)NC(CCO)C3CCCC3)C=CC2)=O)cc2ccccc2[nH]1 c1(CC(=O)NCCC2CN(C(=O)COC(F)F)CCCO2)cc(F)ccc1F C1(NC(C(=O)NCC(C)(C)O)=O)CCN(c2cnccn2)CC1 C12(C(NCC)=O)CCCC1C2(F)F.c1(C=O)c[nH]nc1C=O.C1CC1.CO C12(NC(C(CO)OC)=O)CCCC1CN(C(c1c[nH]cc(C)c1=O)=O)C2 CCCC(C(=O)NC1(C)CN(C(C2CCC(=O)NC2)=O)C1)OC S(=O)(=O)(CC(=O)NCCCCCC)NCC.c1(C2(C=O)CCC2)cc(C)on1 C1(CCNC(C(CCO)N(C)C)=O)CC(F)(F)CN1C(C1CC(F)(F)C1)=O C1(NC(c2n(C)cnc2)=O)CN(C(c2cc(Cl)ncn2)=O)CC1C#N C1(CC(=O)NCCC)CC(NC(=O)CCCCSC)C1(C)C C1(C(F)(F)F)(CNC(=O)NC(c2cc(F)ccc2Cl)C)CC2(CCC2)C1 N1(C(CNC(=O)NC)=O)CCC2(CCCN2C(=O)CCCCc2cnc[nH]2)C1 C(=O)(CCCC(C)(C)C)NC(C(=O)NC(CCC=C)C)C1(C)CC1 c1(CC)cncc(NC2CCCC(CN(C)Cc3cscn3)C2)n1 CN1CCN(C(c2ccc(NC3CCC3)cc2)=O)CC1C.C1(C=O)CC1(F)F.N c1(OC)ccc(CC(=O)NCC2CN(C(=O)COC(F)F)CCO2)cc1O CC(C)C(C)CC(=O)NC1CN(C(=O)C(c2ccc(Br)s2)=O)CC1O c1(C(N2CCC(n3cc(-c4ncc(C)cc4C)nn3)C2)=O)cc(C)c(Cl)cc1C CC1CCN(CCC(=O)NC(C)CCNC(=O)Cc2cncc(Br)c2)CC1 C(=O)CCCCC(C)(C)C.c1(SCC)cccc(C(=O)NC23CC(C2)C3)c1.C C1(NC(CSc2cn(C)nc2)=O)CCCCC1NC(=O)C=C1CCSCC1 N1(C(CCC2CC2)=O)CCN(CCO)C(C)C1.c1(COC)cc(C(=O)N)co1 C(=O)(CC(O)CC(C)(C)C)NCC(C(C)C)NC(c1ncc(C)cn1)=O N1(C(C(c2cn(C)nn2)NC(c2c(C)c(=O)cc[nH]2)=O)=O)CC2CC(C)(C)C2C1 Nc1cc(C(=O)NC2CCC(NC(c3ccc(Br)cn3)=O)C2)cc(F)c1O N(C1CCCn2ccnc21)C(C(C1(O)CCCCC1)NC(C(CC(N)=O)O)=O)=O N1(C(c2c(C)onc2)=O)CCN(C(c2ccnn2C(F)F)=O)C2CC12 C1CC2CCCC(C1)N2C(=O)CC.C1(OC(C)(C)C)CC(C=O)C1.C1CC1.N N1(C(c2c(C)snn2)=O)CC2CCC2(CC(=O)NC(C2CCCCC2)(C)C)C1 N1(C(CC(CC)C)=O)CCCC(CO)(NC(c2ccccc2NC(=O)CC)=O)C1 N1(CCOCc2nnc(-c3ccc(OCC)cc3)o2)CCOc2ccccc21 c1(CSC=CC(=O)N2CC(F)(c3ccncc3)C2)cccnc1Cl c1(N(CCC)CC)ccc(C(=O)N(CCCC)C)cn1.C1(C=O)(N(C)C)CC1 c1(C(=O)NC2CCC(C)N(CC=CCl)C2)cccc2ccccc12 c1(-c2cc(C)sc2C)ccc(C2(C(=O)Nc3nccc(Br)n3)CC2)cc1F C12(CNC(CCC#C)=O)CC(CN1C(=O)CC(c1ccc(C(C)=O)cc1)C)C2 C1C(O)C(O)CN1C(c1ccccc1)=O.C(=O)(CC(=O)NC)OC.CC(F)F Cc1cc(C(=O)NCC2CCCN2C)cc(C)n1 c1(-c2nc(C(C)OC)nn2C2CCOC2)cc2cccnc2s1 c1(C(N(C2CCN(c3c(C(C)=O)c(Cl)ncn3)C2)C)=O)cnc2c(c1)COCC2 c1(C(N(C2CCN(Cc3cccc4sccc34)C2)C)=O)cc2cc(F)ccc2[nH]1 C(=O)(C(=O)NNc1ncnc2ccsc12)Nc1c(N(C)C)cccc1 c1(C(N2CCC(COC)(NC(C34CCC3CC4)=O)C2)=O)cc2ccccc2cn1 c1(CNC(=O)CC2COCCN2C(c2nccs2)=O)ccc(F)c2ccccc12 C1(NC(C(c2ccccc2)SC)=O)CCN(C(=O)CN2CCC2C)CC1CO N1(C(C2C(C(=O)OC)C2)=O)CCC(NC(=O)CC2(C)CCCO2)C(C)C1 N1(C(C(c2cccc(Cl)c2)OC)=O)CC2(CCC2)CC1CNC(=O)C(C)C c1(C(=O)NC(C(C)NC(c2cnc(C)c(C#N)c2)=O)C)cnn2c(C)cccc12 C1(C=O)(COC)C=CCN1C(C1COCC(C)O1)=O.C1COC(C(C)C)C1.N CC1(CC(N2CCC(CCNC(c3ccc(Cl)s3)=O)C2)=O)CCS(=O)(=O)N1 C1(NC(C2C(C=C)C2)=O)CCSC12CN(C(C1(CN(C)C)CCCC1)=O)C2 C1(C=O)(C=O)CCCO1.CC(C(=O)N)N(C)C.C1(CC)CCC1.C(C)(C)C C1(CNC(CCCCCC)=O)CN(C(c2ccnc(F)c2)=O)CCC12CCOC2 C1(NC(c2c(C)nn(CCO)c2)=O)CN(C(C2CC(F)(F)C2)=O)C2(CCC2)C1 Cc1nc(Br)ccc1C(=O)OCCCN1CCN(c2ccc(Cl)cc2)CC1 C1(CC(=O)N(C2CCCN(C(c3ccc(OC)s3)=O)C2)CC)OCCOC1(C)C C(=O)(CCCS(N)(=O)=O)N1CCN(C(c2ccc(C)c(O)n2)=O)CC1CC(F)F c1(C=O)cc2n(n1)CCOC2.CC(C)(C)COCC(=O)NCCOCCC N1(CCC(=O)NC(CNC(C(C)(C)CF)=O)CO)C(=O)c2ccccc2S1(=O)=O c1(C(=O)NC(CNC(C(n2ccc(C)n2)C)=O)C)coc2cc(O)ccc12 N1(C(C2C(=C)C2)=O)CC2CCC(NC(=O)Cc3coc(C(F)F)n3)CC2C1 c1(-c2cc(C)c(F)nc2)cnn2c1CN(Cc1cccc(OC(C)C)c1)CC2 O=C(CCCCCCCBr)N1CC2(CC2C(N2CC3OCCOC3C2)=O)C1 C(=O)(CC=CCNC(c1cc[nH]c1)=O)NC1(C(COC)O)CC1 CCCC(C(=O)NC1CCN(C(=O)CCc2cnc(C)s2)C(C)C1)S(N)(=O)=O c1(NC2(CNC(=O)Cc3ccc(Cl)cn3)COC2)ncnc2occc12 C(=O)(CC(C)(C)CC(F)F)N1CC(CCC)N(C(c2cc(OC)n(C)n2)=O)CC1 N1(C(CCCOC(C)=O)=O)CCC2CCC12CNC(c1cc(C)nc(C)c1)=O CCCCC(CC)N1CCC(C(=O)NCCCOC(C)=O)CC1 C1(C)(NC(c2c(CC)nns2)=O)CCN(C(c2cncc(Cl)n2)=O)C1 c1(C(=O)NC2CCN(C(c3ccc[nH]3)=O)CC2CO)cnc2c(c1)CCCO2 c1(N2CC(C#N)C(NC(c3ccc(C(F)F)nc3Cl)=O)C2)ncc2c(n1)CCC2 C(=O)(C1=C(Cl)CCCC1)NCCN(C(Cn1nc(C)c(Cl)c1C)=O)C1CC1 N1(C(c2sc(C)c(O)n2)=O)CCC2(NC(c3cn(CCC4CC4)nn3)=O)CC2C1 CC1(C)CC1(C#N)C(=O)NCC#CC(=O)N1CC(OC(F)F)C1 S(=O)(=O)(CCC(=O)N1CCCC(N(C(=O)C2=CCOC2)C)CC1)NC c1(C(=O)NC(CNC(C(CC)O)=O)(C)C2CC2)ccc(F)cn1 C1(C(=O)OC)CCN(C(c2cccn2C(F)F)C(=O)NCC(C)C)C1 C1(NC(c2cccc(C)c2O)=O)CCN(C(=O)CCC(C)N(C)C)CC12CCC2 c1(C(=O)NCC2(O)CCCN(C(CC(C)N(C)C)=O)C2)cc(C#N)ccc1F C1(NC(C2(CCC=C)CN(C(=O)C(O)C3CC3)C2)=O)COCC1(C)C c1(C(=O)NCC2CCN(C(c3c(CC)occ3)=O)C(C)C2)c(F)ccc(Cl)c1F CC1(C)CC(C)(C(N2CC(CCNC(=O)CC3(C)CC3(F)Cl)C2)=O)C1 c1(CN2CCC(C(C)NC(C3CCN(C)CC3)=O)CC2)csc2ccccc12 N1(CN2CC(OC)(Cc3ccnc(O)c3)C2)CCCC(C)C1 c1(NC)ccc(CCC(=O)NCC2(F)CN(C(=O)CC(C)F)C2)cc1 c1(C(N2CCC(C(C)(C)NC(CCCCOC)=O)C2)=O)ccc(F)c2c1OCC2 C1(C(N2C(CC(=O)NCc3ccn(CCC)n3)CC2)=O)CC2CCCC2C1 C(=O)(C1CCCc2sc(=N)[nH]c21)NC1C(NC(CCc2cn(C)nn2)=O)CC1 C#Cc1ccc(C(=O)NC2CN(C(=O)CCP(C)(C)=O)CCC2O)nc1 c1(C(=O)NC(CC)(CNC(c2csc(CO)n2)=O)CC)cnc2[nH]ncc2c1 C(C(CC(C)C)C(=O)NCC1COCCN1C(=O)CN1C(=O)CCC1=O)OC c1(OC)c(C(N2CCS(=O)CC2)=O)ccc2c1CCC2 c1(CCC(=O)NCC23CC2CN(C(C24CCC2CC4)=O)C3)cccc(F)c1 c1(NC(CN(C(CC=Cc2ccc(C)cc2)=O)C)C)ccn2nccc2n1 c1(C(=O)NCCCNC(c2c(C)nc(Br)s2)=O)sc2cncn2c1C N1(C(CCN(CCC)C)=O)CC2CCC(C1)N(C(=O)CCN1CCC1)C2 C(=O)(C1c2ccccc2CN1C(=O)CCC(N)C(N)=O)NC(C)CC#N c1(C(N(C2CN(C(Cc3nnc(C)s3)=O)CC2F)C)=O)cnc(O)cc1O c1(OC)ccc(Cl)cc1C(=O)N.C1(C(N2CCC(CC)C2)=O)CC2(CCCC2)C1 C(CC(=O)N1CC=CC(NC(=O)CC2CCC(C)CC2)C1)(C(N)=O)NC(C)=O C(CCCCCC(=O)O)N(C(C)=O)C(c1ccc(SS(C)(=O)=O)cc1Cl)=O CCC(C)CC(C)C(=O)NCC1(C)CN(c2cc(Cl)nc(C(C)C)n2)CCO1 N1(C(C(CC)CN(C)C)=O)CC(NC(c2ccoc2)=O)C2(CCCC2)C1 C1(C(N2C(CNC(c3ncc(OC)cn3)=O)CCC2)=O)CCn2c(C)nnc2C1 c1(C(=O)NCC(=O)NCCC(C)NC(CC(=C)C)=O)cc(C)cc(C)c1 N1(C(C2CN(C(C(CC)SC)=O)CC2C)=O)CC(=O)NC2(CC2)C1 N(C(=NCCCn1nccc1C)NCc1cccc2c1OCO2)CC(=C)C c1(C(N2CCN(C(c3c(S(C)=O)cccc3)=O)CC2)=O)ccc2ncncc2c1 C1(c2nnnn2C)(Nc2ccc(OC)c(OC(C)C)c2)CCCC(C)(C)CC1 C(CCCCC(=O)N1CCCOC(c2ccc(Br)cc2)C1)N(CCC=C)C(=O)CC Cc1c(Br)ccnc1C(=O)NC(CNC(=O)C=Cc1ccco1)C(C)(C)C C=C1CC(C(=O)NC2CCCCC2CO)N(C(=O)C(c2ccc(O)cc2)C)C1 C1(NC(C)=O)CCN(C(=O)C(=O)NC2CC2)CC1.N12CCC1(C)C2=O C1(O)(C(CNC(C2(CCC)CCC2)=O)C)CCN(C(c2nnc(C)s2)=O)C1 c1(C(c2cn(CCCC)nn2)n2cncn2)cccc(OC(F)F)c1OC c1(C(N2CC(CNC(C(C)C3CCCO3)=O)C2)=O)ccnc2c1CC(=O)N2 Cc1oc(CCC)nc1C=O.C(CCN(C(=O)CC=CC(C)(C)C)C)C(C)C CCC(CC)C(=O)NCC12CC1CN(C(=O)C(c1cccc(Cl)c1)OC)C2 N#Cc1ccc(Cl)c(C(N2CCC(C#N)(NC(=O)CCC(N)=O)C2)=O)c1 C(=O)(C(C(C)C)c1ccn(C)n1)N1CCC(CCNC(c2c(C)nco2)=O)C1 N1(C(C2CC(OC)C23CCC3)=O)CCC2CN(C(c3cnc(C4CC4)o3)=O)C2C1 C1(OCC=C)CCN(C(C2(C)CC(NC(=O)CCOCC(C)C)C2)=O)C1 C12(C(N3CC4C(NC(Cn5c(C)cc(C)n5)=O)C4C3)=O)CC(CO)(C1)OC2C C1(NC)CCCN(Cc2cn(CC(N3CCOCC3)=O)nn2)C1.c1(S)ccccc1 c1(OC)cc(CCNC(=O)C(=O)CC(C)C)ccc1C C1(C(=O)NCCc2ncon2)CCN(C(=O)CCc2cn[nH]c2)O1 C=C(C)CCCC(=O)NCC1(CNC(C2(Br)CC2(C)C)=O)CCC1 C(=O)(CCCn1cc(C)nn1)N(C)C.C(=O)(CCOC1CC1)NC n1(CC(=O)NCCC2COCCN2C(=O)CC2CSC2)cccnc1=O CC1=NOC(C)(C(=O)NC2CCC2NC(=O)CCOc2cccnc2)C1 c1(C(N=S(Cc2cccc(C)c2)(C)=O)=O)cccc2c(O)cccc12 c1(N(C)C)cccc(N(C2CCC2)C(c2cc(C3CCCN3)nn2C)=O)c1 C1(CC=O)COCCN1C=O.C(CCCC)N(C)C.C1CC(=O)N1.C(C)(C)C c1(C=O)cc(O)cc(O)n1.C(C)(C)C(C)C.c1(COC)nocc1C(=O)N C1(C(=O)NC2CN(C(C3(CC#C)CCC3)=O)CC2O)CC2(CCC2)CCO1 C1(CC(=O)N(C)Cc2cc[nH]c2)CN(C(C2CC2(C)C(F)F)=O)CC12CC2 N(C1CCCOc2cccc(F)c21)C(C)C(=O)Nc1ccc(I)cc1 CN1CCC(C(=O)NC2CCCC2CNC(=O)C=Cc2cc[nH]n2)CC1 C1(CNC(COC(C)=O)=O)CCCCC1OCC=C1CCSCC1 CCCC(CC)C(=O)N1CCCC1C=CC(=O)NCCCNC(N)=O C1(C(NOCCC)=O)C(C(=O)N(CC(=O)OC)C)C1(C)C c1(C(N2CCC(N(C(C3=CCN(C)C3)=O)C)C2)=O)cc(F)cc(F)c1O Cc1cccc2oc(C(=O)NC3CC(NC(c4ncncc4Br)=O)C3)cc12 C=CCC(F)(F)C(=O)NCCC1(C)CCN(C(C2CC2(C)C(F)(F)F)=O)C1 CCCC(C)CC(=O)NCC(C)C(F)C(=O)NCC12CCC(CO1)C2 CC(c1ccccc1F)=CC(N1CCN(C(=O)C(F)C(C)(F)F)C2CC12)=O C(CCCCC(=O)N1CC(NC(=O)Cn2cc[n+](C)c2)CC1C)SC n1(CC)cnc2nc(=NCC3(CO)CC3)[nH]c(NCc3ccc(Cl)c(F)c3)c12 C1(NC(C(C)NC(C2CCCOCC2)=O)=O)C(O)C2CCOC12 N1(C(c2cc3cccc(C)c3nc2)=O)CCCc2c1cc(F)c(F)c2F N1(C(c2ncc(CN(C)C)s2)C=O)CCC(S(=O)(=O)C(C)(C)C)C1.C1CC1.N C1(C(=O)NC(CCC=C)C)CCN(C(C2(C)CCC(=O)C2)=O)CC1C N1(C(C(C)=C2CC2)=O)C2CCC1C(C)C(NC(c1nn(C)cc1[N+](=O)[O-])=O)C2 C1(OCC)CC(NC(C2CCC(C(=O)O)N2)=O)C1(CC)CC c1(N(C)C)noc(CCC(=O)NCC2CNC(=O)C2)n1.C12C=CCN1C2=O c1(OCCC(N2CCC(NC(CC(C)c3cnn(C)c3)=O)C2)=O)ccccc1F N1(C(C2C(C)C2C)=O)CC(C)N(C(=O)CCC(C)(C)C)CC1C c1(C=O)ccc(F)c(O)c1F.N1(C(C(CC)NC(C)=O)=O)CCC(C)C(C)C1.N FC1(F)CCC(c2ccccc2)C(NC2CN(C3CCCNC3)C2)C1 C1(CNC(c2nc(CC)sc2)=O)CCN(C(=O)C=Cc2cncs2)C12CC2 c1(CNC(C2C(C)CC(C)O2)=O)ccc(C)cc1F.C(=O)C(C)C(C)(C)C.N c1(C(N(CCCCCCNC(=O)CSC(F)F)C)=O)cccc2nn[nH]c12 c1(CC)nc(C#N)cc(=NC(C)C2CCCN(C(=O)C=Cc3cncn3C)C2)[nH]1 CC1(C(=O)NCCCC(=O)NC2CCCNC2=O)CC=CCC1 N1(C(c2ccc(COC)cc2)=O)CCC(C(=O)N)C(O)C1.C1(N(C)C)CCC1 C1(CC(C)C)(C(=O)NC2CCC(C)C2)CCNC1=O.c1(C=O)cnc(O)o1.N c1(C(C)O)ncc(C(N2CCC2CC2CCC2)=O)s1 C1(CCC)(C(=O)NCC)CCNC1=O.C(=O)(C(C)CC=C(C)C)N1CCC1 C1(O)(CNC(CC2(O)CC(C)(C)OC2)=O)CCCN(C(=O)Cc2ccon2)CC1 CC(CCNC(c1cc(CNC(C2(C)CCCOC2)=O)cs1)=O)C(F)(F)F C12(NC(c3ccnc(OC)n3)=O)CCC(CN(C(c3cc(Br)oc3C)=O)C1)C2 C(N=c1[nH]c(=NCC2(CSC)CC2)[nH]c2c1SCC2)C1CC(CC)OCC1 N1(C(C(C)NC(=O)NCCS(C)(=N)=O)=O)CCc2ccccc2C1 c1(N2CCC(c3nc[nH]n3)C2)nc(N2CCCC3(CCCO3)C2)c2[nH]ccc2n1 C(=O)(CC(C)(C)CCC)N1CC(C=C)(CC(=O)NCCOCCCO)C1 C(=O)(C1(C)COc2c(Br)cccc21)NS(CC(C#C)(C)C)(=O)=O Nc1ccc(C(=O)NCC2CN(C(=O)CCn3ccnn3)CCCO2)nc1N C#CCC(C)C(=O)NCCCC1(CNC(C2CCN(C)C2=O)=O)CCCC1 c1(N2C(C)CC(NC(c3cn(CCO)nn3)=O)C2)nccc2c1C(=O)OC2(C)C C=CCCC(CO)NC(=O)CC=CCNC(=O)C(CCC)SCC C(=O)(C(C)CC(F)(F)F)NCC1N(C(CC=CC)=O)CCC(C(F)(F)F)C1 N1(C(c2cc(C3CC3)nn2C)C(=O)NCC(=C)C)CC=CCC2(CCOCC2)C1 N1(C(C2(CC#C)CC2)=O)C2CC=C(C(=O)NC(c3ccc(C)cc3)C)C1CC2 c1(C(=O)NC2C(CC)N(C(=O)C(O)CN(C)C)CC2)ncc(F)cc1F N1(C(C2C=C(C)CS2)=O)CCN(C)CC1C(=O)Nc1cn(C)nc1O c1(CC)cc(CS(=O)(=O)Cc2ccccc2)on1 c1(C(N2CCC(N(C(c3c(C)c(Cl)ccc3)=O)C)C2)=O)scc2c1CCCC2 N1(C(=O)OC(C)C)CCOCC1C(=O)NC1CN(C(c2ccncc2)=O)C1.C c1(COC)cc(-c2cncc(NC(=O)CCc3ccccc3Cl)c2)ccc1F N1(C(CSCCC#N)=O)CCCC(CC(N2CCN(CCO)CC2)=O)C1 N1(C(c2nccc(CC)c2)=O)CC(=O)NCC1C(=O)NCCCSCCO N1(C(C=Cc2c(C)nn(CC(C)C)c2Cl)=O)CCOC2(C1)CN(C(=O)CNF)C2 C1(C(N(CC)C)=O)CC2(CC2)CN1C(C1CC2(CC2)C1)=O.c1ccccc1 CC#CCCCC(=O)N(C)CC1CCCCN1C(=O)Cc1csc(CC)n1 C1(CCCC)CN(C(C2(O)CC(C)(C)C2)=O)CCN1C(=O)CN(C)C(=O)O CP(C)(=O)C(O)C(=O)N1CCN(C(=O)CC2CCOCC2)C(CCO)C1 C(=O)(C(C)(CC)OC)NCCC(C)(C)NC(C1CC(=C)C1)=O c1(CCC=O)cccc(C=O)c1.c1(C(=O)OCC)cnc(C(C)C(=O)O)s1 NS(=O)(=O)CCCC(=O)N1CCC2(CC(NC(=O)CSc3ccccc3)C2)C1 C1(CC)(CNC(C2CC2C(C)NC(c2csc(Cl)c2)=O)=O)CCCO1 C(=O)(CC(C)P(C)(C)=O)NCC(C)N(C(C1CCN(CC(C)C)CC1)=O)C Cc1ccc2c(N3CCOC(C4CCC4)C3)nc(N3CCC(CC#N)C3)nc2c1 c1(C(C(=O)NCCC2CC2)N(C2CC2)CC)cn(Cc2ccco2)nn1 C=CCCCCC(C(=O)NCCCCCC)N1CCC1(C)C(=O)NC CC12CC(C1)N(C(C1CC1[N+](=O)[O-])=O)C2.c1(C(=O)N)ccc(-n2cncn2)nc1 N1(C(CSC(C)C)=O)CCCC2(NC(c3ccc4cn(C)nc4c3)=O)CCCC12 c1(C(N2CC3CN(Cc4c(F)cc(C)c(Br)c4)C3C2)=O)cc2cccc(Br)c2[nH]1 c1(C(=O)NC(C(C)NC(C(C)OCC=C)=O)CO)nnc(O)c2c1CCCC2 C1(COC)(NC(=O)Cc2cccc(Cl)c2)CCN(C(C2(C)C=CCC2)=O)C1 Cc1ccc(CCC(=O)NC2CC(=O)N(C3CN(C(=O)C(C)CF)C3)C2)cn1 C(=O)(CCCCCCN=[N+]=[N-])NCC1OCC2(CN(C(C3(OC)CCC3)=O)C2)C1 N1(C(Cn2c(C)ccc2C)=O)CCCCC(N(C(=O)COc2ccccc2)C)C1 C(=O)(C1(C)CCn2ccnc21)N.C(C)(CC)NC(COCCOCC#C)=O c1(C(=O)NC2C(CNC(=O)CC3CCCSC3)C2)cc(=O)cc[nH]1 c1(NC(C2C(C(N3CC(OC)C3)=O)C2)=O)cccc(OC(F)F)c1Br C(=O)(C(C)C(C)(F)F)N1CCN(C(Cc2ccc(OCC#C)cc2)=O)CC1 C=CCC(C)(C(F)F)NC(=O)CN(C(=O)C(C)CC(=O)OCC)C CC1(C)CCCCN(C(=O)C(CNC(=O)C(C2(O)CCCC2)F)CC2CC2)C1 c1(C(N2CC(C=C)C(NC(C3CCNC3=O)=O)C2)=O)cc2c(C)cccn2n1 Cc1ccc(Cl)cc1-c1cn(CC2CCCN2C(=O)Cc2cccc(Cl)c2)nn1 C(C(CC(=O)NCC(CC)CC)C1CCC1)NC(C(C=C)OC)=O Cc1ccc(C(=O)N(CC)C(C)C)c(C)n1.c1(C=O)cnc(-c2ccsc2)s1.N N1(C(C(C(C)O)(C)C)=O)CC2(CC(C(N3CCOCC3)=O)CO2)C1 N1(C(C(C)N(C(C)=O)C)=O)CCC2(CC1)CC2C(=O)N.c1nncn1C(C)C CC1(C)CCC(CNC(c2ccc(C#N)o2)=O)CC1.C(=O)C(F)OC(F)(F)F N1(CC(N2CCOC(C)C2CO)=O)C2CCC1CC(NC(=O)OC(C)(C)C)C2 CC(C)CCCCC(=O)N1CCC(CN(C(=O)C(C)(C)N(C)C)C)C1 C(CC1=CCN(C(=O)CCC=CBr)CC1)NC(CCCC(N)=O)=O c1(NC)ccc(C(N2C(C(=O)NC(C)CO)CC3CC23)=O)cc1 C(C)(CCC)NC(CN(CCC)C=O)=O.C1(C=O)CCC1.C(C)(C)C.N Cc1cc(=NC(C)c2ccc(C(F)(F)F)nc2)[nH]c(=NCC2(C)COCCO2)[nH]1 c1(OC)ncc(Br)cc1CN1CCC(O)C(C(=O)Nc2nc(Cl)nc(Cl)n2)C1 C1(CCC)(NC(=O)CSc2ccc(Cl)cc2)CCN(C(=O)CCSC)CC1 N1(C(C=Cc2ccc(OC)cc2)=O)CCCC2C(NC(=O)C(C)C)C(C)(C)C12 N1(C(C(OC)OC)=O)CCN(C(=O)CN(C(=O)CCc2cc(Cl)no2)C)CC1 C1CN(C(C2(C)CCCNC2=O)=O)CC12CCC2.n1(CC)cc(CC(=O)NC)cn1 N1(C(C(C2CCOC2)NC(c2cc(Cl)no2)=O)=O)CC2CSCC(C2)C1 c1(C(=O)Nc2c(C(C)C)nn(C)c2)ccc(C#N)c(-c2c[nH]c3ncccc23)c1 CCCC(CCC)C(=O)NCC1CC(OC)CN1C(=O)CCP(C)(C)=O c1(-n2ncc(C(N3CCC(CN4CCOCC4)C3)=O)c2)ccc(Cl)cc1 Cn1cc(CC(O)C(=O)N(Cc2ccccc2)Cc2cnc[nH]2)cn1 N1(C(c2cn(C)nn2)=O)C(C(=O)NCC(C)(F)F)CC2CC12 N1(C(C(CCC)=CCC)=O)CC2(CCCC2NC(=O)C(c2ccccc2)=O)C1 C1(NC(Cn2nnc(C)n2)=O)CN(C(=O)C(F)=CC2CC2)CC1CC1CC1 c1(C(=O)NCCC2CCN(C(CC)=O)C2)c(N)cccc1[N+](=O)[O-] C(N=c1nc[nH]cc1C#N)C1C(NC(Cn2c(C)ncc2)=O)CCCC1 c1(CN2CC3N(C(c4nn(C)c(O)c4)=O)C(C3)C2)ccc2ccsc2c1 N1(C(C(c2ccc(OC)cc2)OC)=O)CC2CC(NC(=O)C(Cl)=CCl)CC2C1 c1(-c2onc(-c3c(Cl)cn(C)n3)n2)cc2cccnc2nc1O C1(CC)CN(C(=O)CP(C)(C)=O)CCC1NC(=O)C.c1ccccc1.C=O.N c1(-c2cn(CCC(=O)NCc3nnc(C(N)=O)s3)nn2)ccc2ncsc2c1 CCCC(CC)C(=O)NCC1(F)CC(CNC(=O)CCC2CC2(Cl)Cl)C1 C1(C(=O)NCC2N(C(Cn3nnc(C)n3)=O)CCCC2)C2CC3C(C2=O)C13 N1(C(c2c(C)nc(C)o2)=O)CCC2(CCCN2S(=O)(=O)c2cnn(C)c2)CC1 N1(C(C2N(C(C)C)CCS2)=O)CC(=O)N(C)c2cc(C(=O)N(C)C)ccc21 Cc1ncsc1CC(=O)NC(Cn1ccnn1)C(=O)NC(CO)CCO C(=O)(CC(O)C(C)CC)N1CC(c2c[nH]nn2)C1.C1(CC=O)CCC(C)(C)O1.C N1(C(c2cc(C)nn2C)=O)CCC(C)N(c2ccc([N+](=O)[O-])cc2)CC1 CC1CC(C(=O)O)N1C(=O)CCc1nnc(-c2ccsc2)o1 C(=O)(CCC(=O)NC1(c2ccccc2)CN(C(c2coc(C)c2)=O)C1)NCCC C1(NC(c2cncs2)=O)CC(=O)N(C2CN(C(=O)C=C3CCOCC3)C2)C1 Cc1cccc(C2(C(=O)NC3CCC3NC(=O)CCCC#N)CCCC2)c1 C1(NC(Cc2cc(C)on2)=O)CN(C(=O)C(C)CF)CC2(CCC2)C1 N1(C(C=C(CCC)C)=O)CCCC1CCNC(=O)C(C)NC(=O)CC C(=O)(C(C)(C)COCC(F)F)NCC(CNC(c1c(C)cno1)=O)(C)O N1(C(C(C)Br)=O)CCCC12CCCN(C(=O)C(C)(C)C(C)(F)F)CC2 c1(C=O)ccc(S(N)(=O)=O)cc1N.CC1(C)C(C(=O)NCC(O)CC)C1(C)C C1(C#CC(=O)N2CCC(NC(=O)C(O)C3CCC3)CC2)(CC)COC1.C1CC1.C N1(C(CCCOCC)=O)CCC2CCC(C1)N2C(C1CCCCC1C)=O N1(C(c2c(CC)csc2)=O)CCC2CN(C(=O)C(F)C(C)C)C2C1 CCCC(CCC)=CC(=O)NCC1CCN(Cc2nnc(CC)s2)C1 CC1CN(C(C2CCCN2N=O)=O)CC1CNC(c1ccn(CC(F)F)n1)=O C1(NC(c2cc(C)n(C)n2)=O)CCCN(C(=O)COc2ccc(O)cc2)CC1F C1(CNC(=O)CC2CCCC2NC(=O)C(O)C2CCC2)CCCO1.C1CC1 CCC(C)CCCC(=O)NC12CC(C(N3CCCC(C)CC3)=O)(C1)C2 c1(C(C)C(=O)NCCCC2CCCN2C(=O)CCc2cn[nH]c2)cccc(Cl)c1 C1(C=O)CCC(F)(F)CC1(C)C.n1(CC(=O)OC)cnc(C(=O)N)c1.CCC c1(C=O)ccc([N+](=O)[O-])cc1Cl.c1(CC)cc(N)c(C(=O)NCCC)c(F)c1.N C#Cc1ccc(OCC(=O)NC2CC(NC(=O)CN=S(C)(C)=O)CC2O)cc1 c1(C(=O)NC23C(CCN(C(C=CSC)=O)CC2)C3)ccc2cc(Cl)ccc2c1 N1(C(C(C=C)(C)CC)=O)CC2CC(O)C1C2NC(c1ccc(C(=O)NC)cc1)=O c1(C(=O)NC2CCS(=O)CC2)cccc2nn[nH]c12 c1(C(=O)NCC2C3CN(C(=O)CC4OCCO4)CC23)cccc2occ(Br)c12 CCC(CN(C(=O)C(C)OCC(C)C)C)NC(C1(c2ccon2)CC1)=O c1(SCCNC(=O)NCc2cccc(C(F)(F)F)c2)ccc(O)cc1O N1(C(C(=O)NCCOC)=O)CCC(CNC(c2cnnn2C)=O)C12CCC2 c1(C=O)cccc(C(N)=O)c1N.N1(CC(=O)NCCC)CCCC(C(N)=O)C1 C1(C(=O)NC2C(c3c(C)n(C)nc3)C2)CCCCC(F)(F)C1 c1(NC(C)=O)ccc2[nH]c(=NC3CCN(C(=O)CCC4(C)CC4)C3)sc2c1 C1(NC(C(C)O)=O)CCN(C(c2ncncc2Cl)=O)CC(C)(C)C1 C=C(C)C(CC(=O)NC1CC(NC(c2c(Cl)n[nH]c2C2CC2)=O)C1)OC C1(NC(C(CCCNC(CCCOCCOC)=O)O)=O)CCn2cnnc2C1 c1(OC)nc(N2CCCC3(CNC(=O)C(C)OC)CCCC23)nc2[nH]cnc12 N1(c2nnc(COC)s2)CCSCC1CCNC(=O)C(O)C1CCC1 C1(NC(Cc2nc(CC)sc2)=O)CCC(Cn2cc(C3CCN(C)C3)nn2)CC1 O=C(NNc1ncncc1F)C(=O)NCc1cc2sc(Cl)cc2[nH]1 c1(C=O)cccc(SC(F)(F)F)c1.c1(C(=O)NC(C2(C)CC2)C)cccs1 N1(C(COCCCOC)=O)C2CCC1CC(NC(=O)CC)C2.C1(C=O)CCC1 CCC(CC(=O)N(CC(C)NC(=O)CC1CCC1(C)C)C)C(F)F CCC(C)(COC(C)(C)C)CN=c1cccc(S(=O)(=O)N2CCCC2COC)[nH]1 C1(C(=O)OC)CN(C(=O)NCc2cnc(C(C)C)s2)CC1(C)C C1(CNC(=O)CCN2CCOC2=O)CC(C=O)=NO1.C1CC2(CC2)C(=O)O1.N CC(C)C(CNC(=O)C(=O)C(C)(C)C)C(=O)NCC(C)CO S(=O)(=O)(c1ccc(Cl)cc1)N1C(C(N2CC(C)(C)OCC2)=O)CC1 c1(NC(C(CCCC)N2CCCS2(=O)=O)=O)cc(Br)c(Cl)nc1C c1(CC)cc(Nc2cc(NCC)ncn2)cc(NC(c2ccc(Br)c(F)c2)C)c1 C(=O)(C#CC1CCCO1)N1CCC(O)(CNC(C2C3COCC23)=O)C1 C1(NC(CN(CC)CC)=O)CCC2CN(c3nccc(CO)n3)CC2C1 CC1CN(C(=O)CN(c2ccncc2)C)CC1CNC(=O)COC1CCC1 C1(NC(C(C)C2CC2)=O)CC2CC1CN(C(c1coc3ccccc13)=O)C2 N1(C(C2(CC=C)CCNCC2)=O)CCCN(C(c2ccc(Cl)cc2)=O)CC1 C1(NC(c2nn(C)c(C3CCCO3)c2)=O)CCN(C(=O)C2=C(Cl)CCC2)C1(C)C c1(C(=O)CO)ccc(C=Cc2nnc(-c3ccco3)o2)cc1C(c1ccsc1)=O c1(C(C)C)ccc(C(=O)N(C)CC2COCCN2C(=O)CCC(C)N(C)C)cn1 Cc1nc(C)n(O)c1C(N1CCCCC1C)=O.C1(=CC(=O)N)CCN(C)CC1 C1(S(C)(=O)=O)(C(=O)NC(CC)CNC(C2COC(=O)N2C)=O)CCC1 C12(C(N3C(C(N4C(C)(COC)CCC4)=O)CCC3)=O)CCCC1OCC2 N1(C(CNC(N)=O)=O)CCC2CCN(C(=O)Cc3c[nH]ccc3=O)C2C1 Cc1ccc(S(=O)CN2CCC(c3cnn(C)c3)C2)cc1 C=CCC(Cc1ccccc1)C(=O)NCC#CCNC(C12CC(C)(C1)C2)=O N1(C(c2cc(C(F)F)cs2)C(=O)NCCCC2CC2)CCC2CCNC(=O)C12 N1(CCNC(CCC=CCC=C)=O)CCCN(C(=O)C#CC2(CC)CC2)CC1 C(=O)(C1CCC(=O)c2cccn21)NCC(CC)NC(c1coc(C)c1)=O C1(C)(OCC)CCN(C(=O)C(O)C2CN(C(=O)CCC(C)CN(C)C)C2)CC1 C1(CNC(c2nccc(CC)c2)=O)C(C)CCCN1C(c1ccnnc1O)=O CC1(C)OC2C3CCC(Nc4ccccc4NS(=O)(=O)C(F)(F)F)(C3)C2O1 C1(CS(=O)(=O)NC(CC#C)COC)CCC2(CCOCC2)CO1.C(C)=O C(C(C)(C)NC(=O)C(C)c1ccco1)N(C(CNC(=O)OCC)=O)C c1(C(=O)NC2C(SC)CN(C(C3CC(C)CCO3)=O)C2)ccc2nc[nH]c2c1 CCC(C)CCC(=O)N1CC2CC1CN2C(=O)Cc1cc(C)ccc1Br C=CC1(C(=O)NC2CCN(CC)CC2)CCN(C(c2cc(C)c[nH]2)=O)CC1 CC1CC(CNC(=O)COc2ccsn2)CN(C(=O)CC)C1.c1ncccn1.N c1(C(=O)NC2(CC=C)CCN(C(=O)C3=CCCC3)C2)cc2nc(OC)ccc2[nH]1 CCC(CCOC)C(=O)N1CCC(COC)(NC(=O)C(C)(C)CSCC)C1 CCCCC(CC)C(=O)N1CCOC(C)(CNC(c2scc3c2CCCC3)=O)C1 c1(CNC(C(C2CCOC2)OC)=O)ccc(CC)cc1.c1(C(=O)N)nocc1C N1(C(C2CC(C)C2)=O)CC2(C1)OC1(C)CC2C1.C1(C=O)CC(=O)N(CC)C1 c1(OC)ccc(CN2CCN(C(c3cnc(O)cc3O)=O)C3CC23)c(Cl)c1 N1(C(CN(CCC)CCC)=O)CCN(C)C(C)(C)C1.c1(C=O)ccc(F)s1 CCCCCC(F)C(=O)N1CCCC(O)(CN(C(=O)CSCCSC)C)C1 c1(NC2(CNC(CC3N(C)CC=CC3)=O)CCCC2)nc2c(F)cc(Cl)cc2s1 CCC(O)C(C)(C)C(=O)NCCSCC(N1CCOCC1CCO)=O Cc1nc(CNCc2ccc3c(Br)csc3c2)c2ccccn12 N1(C(=O)OC(C)(C)C)CCC2(CSC2)C1.C12CC(C1(C)C)NC2 c1(N2CCC(N(C(=O)C(O)C3CC3)CC#C)CC2)nccc(C(F)(F)F)n1 Cc1cc(C(=O)NCC(C2CC2)NC(=O)CCn2cccn2)ns1 N1(C(CCCCC(C)C)=O)CC(C2CCN(C(c3snnc3C(C)C)=O)CC2)C1 C12(C(=O)NCCC(=C)C)CCC(CO)(CC1)CC2.C1(C)(C(=O)N)C=CCC1 CC1(C(=O)NC2CCC(NC(=O)C(c3cccc(F)c3)O)CC2)CC2CCC1O2 Cc1cc2[nH]c(C(N3CCC(NC(=O)Cn4cnnc4)C(CO)CC3)=O)cc2o1 C1(CC)CCN(C(=O)C(O)Cc2ccc(Cl)cc2)C1C C(=O)(CCCCCC#N)N1CCC(C)(NC(C(C=C)c2ccccc2)=O)C1 CN1C2CCC1CC(C(=O)NCC1CC3CCC(C1)N3C(C1CC3CC3C1)=O)C2 C1(O)CCN(C(C2OCCCO2)=O)C1.Cc1csc(C2C(C(=O)NC)C2(C)C)n1 Cc1ccc(-c2cn(CC(=O)NCCSCC3CN(C)CCO3)nn2)nc1 C1(C(N2CCC(NC(Cn3c(C)nc(C)n3)=O)C2)=O)C2CCC3(COC(=O)C13)O2 C1(C(N(C)C)=O)C2CCC(C2)N1C(c1ccon1)=O.N1(C)CCC(N(C)C)CC1 C12(C(=O)NCCc3ccn(CC)n3)CC1CCN2C(=O)CCCOC C1(C2CN(C(c3ccnn3C)=O)C2)(NC(CC(C)C2CCCO2)=O)CC1 c1(OC)noc(C(C)C)c1.C(=O)CC(=O)N1CCC1.C1CC1.C1(C=O)CC1 N1(C(C2CCCC(C(=O)OC)C2)C(=O)NCCOC)CC(=O)Nc2ccccc21 C1(NC(c2ccc(Cl)o2)=O)CCCCC1NC(c1ccnn1C1CC1(F)F)=O C1(O)CCN(C(c2ccc(F)c(O)c2)=O)CC1.CC1C(=O)CCC1CC(=O)NC c1(C(CNCC=CC(CC)C)NC(C)=O)ccc(F)cc1 C1(C(N2CCC(C)(C(=O)NC3(CC#C)CCCCC3)C2)=O)OCCCC1(C)C c1(C(=O)NC2C(C)CN(C(=O)Cn3cc(Br)cn3)C2)occ2c1CCCC2 N1(C(C(C2CCC2)NC(C2N(C)CCN(C)C2)=O)=O)CC2(C1)CC(C)(O)C2 N1(C(C(C=C)C)=O)CC2(CCOCC2)CC1CNC(C1(CCF)CCOCC1)=O C1(NC(C=CCCC(C)C)=O)CCC2CN(C(C3CCC4(CCCC4)C3)=O)CC12 C(=O)(CC(C)(O)C(F)(F)F)NC1C(C)CCN(C(CCC(C)O)=O)C1 c1(C(=O)NC2C=CCN(C(COCC(=O)OC)=O)C2)cnn2c1CCCC2C C1(NC(CCCCCNC(C)=O)=O)CCCCCN(C(=O)C(C(C)C)NC=O)C1 C1(CNC(CC=C)=O)CC2(CO1)CN(C(=O)CCC1CC1(F)F)C2 c1(OC)cccc(CN(C2CCC2)C(=O)NCc2ccn(C(C)C)c2C)c1 CS(=O)(=O)c1cc(C(=O)NCC2CCN(c3ccncn3)CC2)ccc1Cl c1(Cc2cccc(COC3C(C)CCCC3)c2)nc2ccccc2c(=O)n1C C1(C)(C(=O)NC(CN(C(=O)CCc2cncc(F)c2)C)CO)CC2(CCC2)C1 c1(C(N(CCC)CC)=O)cccnc1SC(F)F.C(=O)C(C)(C)n1cnnn1.N c1(C(N2CCOCC(C(=O)NCCN(CCC)C)C2)=O)cnn2ccn(C)c12 N1(C(C)=O)CC2(C1)CN(N1CC(C)(C(=O)N(C(C)(C)C)CCO)C1)C2 N1(C(c2c(CC)nn(C)c2)=O)CCN(C(=O)CNC(=O)C(C)CC)CC1.C N1(C(C(F)=C(C)C)=O)CC2(CCC(NC(=O)C(C)CS(C)(=O)=O)CC2)C1 O=C(Nn1cccc1C(F)(F)F)c1ccc(Cl)c(F)c1O c1(C(C(=O)NCCCNC(c2cnsc2)=O)N(C)C)c(F)cccc1F C1(C(=O)NN(CCNC(CCSCCCC)=O)C2CC2)(C)CC1(C)C Cc1cc(Cl)cc(C(N2C3CCC2CC(NC(=O)C(C)S(C)(=O)=O)C3)=O)c1N c1(CNCC(Cc2ccc(OC)c(OC)c2)C)cccc2[nH]ccc12 C1(N(C(=O)CC2CCOC2)C)CCN(C(C2CCC(CCO)CC2)=O)CC1 C1(NC(COC2CN(C(c3c(C)cco3)=O)C2)=O)CCCNC1=O Cc1cc(NC(N2CCN(c3ccc(N)cc3C)CC2)=O)c(C)cn1 N12CCC=C(C(=O)NC(C)C1=O)C2.C1(C)(COCC(C)C)CC2(CC2)C1 CC(C(C)C(=O)N1CC(N(C)C(C2CCC(C(F)(F)F)CC2)=O)C1)S(C)(=O)=O N1(C(C2CCC(CC)O2)=O)CCCCC(C(N2CCC(CO)C(C)C2)=O)C1 N1(C(=O)C(O)CN2CCOCC2)CC2(CCN(C(=O)C(O)CN3CCCC3)C2)C1 c1(C(CCOC)OC(CC(CC)OC)=O)nc(O)c2ccccc2n1 C1(CC)CCN(C(c2csc(F)c2)=O)C1C(=O)N(CC1CCCCC1)OC Cc1occ(C(F)(F)F)c1Cn1nnnc1C1(NCCF)CCC1.C(C)(C)C C1(C(=O)NC(C2CN(C(c3cc(-c4ccco4)no3)=O)C2)C)CC1C1CC1C N1(C(C(C)n2cccc2)=O)CCC(C(N2CCN(C)C(=O)C2)=O)C12CC2 N1(C(C(C=C)O)=O)CCCC(CCC(=O)NCCc2ccon2)C1 c1(C(=O)NC(C)(CNC(C2CNC(=O)N2)=O)CO)cc(Cl)ccc1Br CCCCC(CCCC)N=c1cc[nH]cc1S(=O)(=O)NCC1(C)OCCc2sccc21 N1(C(Cc2c(C)ccs2)=O)CC2CC(C(=O)NCCc3ccc(F)cc3)(C2)C1 C1(CNC(CC(=O)OCC)=O)CN(C(c2coc(OC)n2)=O)CC1C C1(OC)CCC(C(N2CC(CO)(NC(=O)CCC3CCCOC3)C2)=O)CC1 N1(C(C(C2CCCC2)OC)=O)CCCC1(C)C(=O)NCCc1nc[nH]n1 N1(C(CCC(CC)C)=O)CC2(CCCC2NC(=O)Cc2cc[nH]c2)C1 C1(CC(=O)NC)CC(C)(C)OC(C)(C)C1.C1CCCN1C(=O)C.C=O.C C1(NC(C(c2cnn(C)c2)OC)=O)CCCC1NC(c1cn(C)nn1)=O C1(CNC(CCN(CC#C)C(C2CC3(CCO2)CC3)=O)=O)C2CCCCCC12 C1(CNC(C(CC#C)C2CC2)=O)CCCC12CCN(C(=O)CS)CC2.CC(N)=O C#CCC(CC#C)C(=O)NC1(CNC(=O)CCc2cc(F)cc(F)c2)CCOC1 N#CC1(C(=O)NC2CC=CCC2C(=O)NC2CC(O)CC2O)CC(=O)C1 N1(C(CSCCCC)=O)CCC2(CC1)CN(C(=O)CSC(F)F)CC(C)O2 C(C)(N=c1ccnc(NCC(=O)NC(C2CCCCC2)C)[nH]1)c1c(C)nn(C)c1 CC(F)(F)C(C)(C)C(=O)N1CC2CC(NC(=O)CCC3CCOC3)C2C1 C(CCCCCCCCSc1ccccc1)NC(CN(C)C)CCO CCCCCC(CC)C(=O)NC1CCOC(CNC(=O)CCC(C)CN(C)C)C1 N1(Cc2ccc(C(C)(C)C)cc2)CCOC(C)CC1.C1(C2C(=O)N2)CCOCC1 N1(C(c2c(Cl)ncn2C)C(=O)Nc2c(C)cccc2C)CCOCN(C)CC1 C1(Nc2c(CO)ccc(OC)c2Cl)CC(C)(N=c2[nH]cnc3cnccc23)C1 c1(OCCCC)ccc(C(N2CCC(N(C(=O)CC3CCC4CC34)C)C2)=O)cc1 c1(NC2C(C)CN(C)CC2)cc([N+](=O)[O-])ccc1NC(C)C.C(=O)C1CC1.N c1(CC(N2C(c3nc(COC)on3)CCC2)=O)ccc(C2CCC2)cc1 C12(C(=O)NC3C=CC(C(N4CCC(N5CCC5)C4)=O)C3)CCC(C)(CC1)C2 C(C(=O)NCC(C1CC1)N(C)C(c1ccccc1Cl)=O)(C(C)(C)C)OC N1(C(CNC(C2(CC#C)CCC2)=O)=O)CCN(C(=O)CC(C)NC=O)CC1 Cc1c(C(=O)OCC2OC(=O)CC23CCOCC3)sc2ncncc12 C1(NC(COCC(=C)C)=O)CC(C(N2CC(CC(C)C)C2)=O)C1(C)C c1(-n2c(C(C3=CCCCC3)NC(C)C(C)F)nnn2)ccc2c(c1)OCO2 C1CC2CC(C1)N(C(C1(C3CC3)CC1)=O)C2.c1(OCC)cc(C(=O)N)[nH]n1 N1(C(c2nc(Br)cs2)C(=O)NCC)CC(C(=O)O)C2(C1)CS(=O)(=O)C2 C1(C=O)(C(C)C)CCN(C(C2CCCNC2=O)=O)C1.C(CC)NC(C)=O.CC N1(C(c2ccn(CCC)n2)=O)CCCC(O)(CN(C)C(C2CCCC(=O)C2)=O)C1 C=CCC(CC(=O)Nc1cccc(C2CC2)c1)NC(=O)CC1CCCO1 N1(C(C)C)CCCC1C(=O)N(C)CCOCC.c1(C=O)ccc(Cl)[nH]1.CC.N C1(C(N2CC3C(NC(c4c(C)nc(C5CC5)s4)=O)(C3)C2)=O)CC(=O)OC1(C)C c1(C(N2CC(CC(C)NC(C=C(C)C(C)C)=O)C2)=O)cc(C(N)=O)ccn1 N1(C(c2c(OC)cnc(F)c2)=O)CCCN(C(=O)C(C)C(F)(F)F)C(CO)C1 CC1CC(NC(=O)CCc2ccc(Cl)s2)CN1C(=O)Cn1cc(Br)cn1 c1(C=O)cccc(C#N)c1.C(C)(CCC)NC(CCOCCC)=O.C(=O)(C)N c1(C(=O)NC(CC)Cc2ccncc2)nc2cc(Br)ccc2n1C CCCCC(CNC(c1cccc(F)n1)=O)NC(C1(CSC)CC1)=O CCCC(C(=O)OC)C(=O)N1CC=CC1C(=O)NCCc1cnco1 C12(CNC(CC(C)C)=O)CCCC1N(C(=O)CSCc1cscn1)CCC2 CC1CCc2nc(CNC(=O)C(=O)NCC3CC4CC3C3CC43)sc2C1 Cc1cc(C(F)F)n2ncc(C(N3CCCC(C)(C(F)F)C3)=O)c2n1 c1(CNC(C(=O)NCC2CCC(N)C2)=O)nc2c(s1)CNCC2 N1(C(c2n(C)cnc2)=O)CCC2(CC1)CN(C(=O)Cc1ccc(Br)nc1)C2 Cc1cccn2cc(CC(=O)Nc3ccccc3OCc3cnn(C)c3)nc12 c1(C(=O)Nc2c(C)c(Br)cnc2)ccc2nc(NC(=O)C(C)(C)CCl)sc2c1 c1(C(C(=O)N2CC(=CC(=O)OC)C2)(C)C)ccc(F)c(C)c1 Cc1ccc(C(=O)NC2CCN(Cc3ccc(CC(=O)O)cc3)CC2F)c(I)c1 C(N=c1ncc(O)c[nH]1)C1(O)CN(C(c2ccccc2C2CC2(F)F)=O)C1 C(=O)(C(C)C(C)COC)NCCCCCN(C(c1cn(CCC)nc1)=O)C N1(CC(=O)N)CCCCCC1=O.n1(CC(C)C)cc(CN(CC)C2CC2)cn1 c1(C(=O)NCCC(C)N(C)C(c2cc(=N)[nH]c(Cl)n2)=O)ccn2c(O)nnc2c1 N1(C(C2CCC(CNC(C(COC)OC)=O)C2)=O)CC=C(C)CC1 C(=O)(CC(C)CC(C)(C)C)NC1N(C(c2nc(N(C)C)no2)CC)CCCC1 N1(CCOC)CC(C(N2CCOCC2CN(C(=O)C(C)C(C)O)C)=O)CC1=O c1(C(N2CCOCC(NC(CC(CCC)O)=O)C2)=O)ccc2c(c1)CCN2C C1CCN(C(=O)C(=Cc2cnc[nH]2)C)CC1.C(=O)(CCc1cn[nH]c1)N(CC)C c1(CC(c2ccncc2)NC(=O)CNC2CCCC2)nnnn1C1CCOCC1 C1(C(N2CCC(CCNC(c3n(C)cnc3)=O)C2)=O)CCCC1P(C)(C)=O c1(C(N2CCCC2C2CCC2)C)cccc(C(C)(F)F)n1 C1(CNC(c2c(C)nns2)=O)CN(C(=O)CCc2cccnc2Cl)CC12CC2 c1(SC)nn(C)c(NC(=O)NCC2CCC3SCCSC23)c1C#N CCC(C)CCCC(=O)NCC(CC(=O)NC1CCC(CO)CC1)OC c1(OC)ccc(Cl)cc1NNC(=O)NCC(c1ccc(C)o1)N(C)C N1(C(c2c(SC)nccn2)=O)CC2(C1)CN(C(=O)CCCCC(N)=O)CC2CO c1(CC)ccccc1C(N)CNC(C1OCCC1C)=O C1(S(N)(=O)=O)(C(=O)N)CC1.c1(SC)cc(C(=O)N(CCC)CCO)co1 c1(C(C)=O)cnc(NC(C2C3CN(C(=O)C=Cc4cccs4)CC23)=O)nc1C C(=O)(C1=NNC(=O)CC1)N1CCN(C(c2cnc(C(C)C)[nH]2)=O)CC1C1CC1 N1(C(CC(CCC)C)=O)CCCN(C(=O)C(F)=CC2CC2)C(C(C)C)C1 C1(CC(=O)NC(C(=O)N(CCC(N)=O)C)CC2CCC2)CCCC2CC12 c1(C(N2CC3N(C(C(C(C)C)(C)C)=O)C(CC3)C2)=O)cnn2c1OCC(F)C2 CCS(=O)(=O)CCC(C=O)NC(=O)NC(C)(C)C.c1(C(C)C)ccncc1.N Cc1cccc2c1CCN(C(c1cncc(NCc3c(F)cccc3I)c1)=O)C2 C1CC2CCC(C1)N2C(=O)CC1CCCC(C#N)C1.Cc1nscc1C(=O)NC c1(C(=O)NC2C=CC(C(=O)NCCCC)C2)cc(Cl)cc([N+](=O)[O-])c1Cl c1(CNC(C)=O)n[nH]c2c1CN(C(c1ccc3c(ccn3C)c1)=O)CC2 CN1N=CC(CC(=O)NCCN(C(c2ccns2)=O)Cc2ccccc2)C1=O c1(OC)cncnc1NCC(Cc1ccc(OC(F)(F)F)cc1)CO Cc1ccc(CC(N2CC3CCC3(CNC(C3(C)CC3)=O)C2)=O)c(C)c1 c1(C(C)C)ccc(C(CNC(=O)CCC(C)SC)NC(c2ccoc2C)=O)cc1 c1(C(=O)O)cnc(N(C2CCC2)C2CNCC2)c(Br)c1 Cn1cnn(CCC2CC=CC2)c1=O.C1(O)(C(C=O)(C)C)CCN(C(=O)C)C1.N C1(C(N2CC(CC(C)NC(=O)C=CBr)C2)=O)CCCC2(C1)CC2(F)F C(=O)(C1=Cc2ccccc2OC1)N1CCC(NC(C2N(CC)CC2)=O)C12CCC2 CC(C)C(CCNC(C1(C(C)C)CC1)=O)N=c1[nH]c2c(F)cccc2o1 Cc1cc(F)cc(C(N2CC3C(C(=O)N(C4CCOC(C)(C)C4)C)C3C2)=O)c1N C(=O)(C1=CCc2ccccc21)NCCn1cc(C(C)(C)OC)nn1 O=C(CCCC(F)(F)CO)NCCc1ccc(CNC(=O)C(Cl)=CCl)cc1 c1(N(CC(=C)C)C)nc(-c2ccccc2)nc(=NCC2CCCCS2(=O)=O)[nH]1 CCCC(C)C(=O)NCC1OCCC1C(=O)Nc1cnc(C(C)C)nc1 N1(C(C(CC)N(C)C)=O)CCN(C(c2cc(C3CC3)cc(F)c2)=O)CC1C(F)F N1(C(C2CCCC(=O)O2)=O)CCCOC(CNC(=O)Cc2nc(C3CC3)cs2)C1 Cc1cc(O)nc(C)c1C(=O)NC1CN(C(C2CC2C2CCCC2)=O)CC1C N1(C(C2CCC(=C)CC2)=O)CCC(NC(c2cccc(C3(C)CC3)c2)=O)C(F)C1 c1(C(N2CC(CCNC(=O)C3=CCCOC3)(OC)C2)=O)cc2c(s1)COCC2 CCCC(CCCNC(C1CCN(c2nc(=N)[nH][nH]2)C1)=O)NC1CSC1 CCCC(CC)C(=O)N1CCC(N(CCO)C(c2nc(CC3CC3)cs2)=O)C1 C1(C(=O)N)CC2(C1)CC21CC1.O=C1CC(C(=O)NCCc2ccccc2)CN1 C1(OCC)CCC(NC=O)CC1.C(C)CC.C1(n2cccn2)(C=O)CCC1.N C1(C(=O)NC(C2CN(C(c3c(C)ccs3)=O)C2)C)NC(=O)CC1C(F)(F)F C(=O)(CC1=CCCC1)N(C(CNC(CC1(OCC)CCC1)=O)C)C c1(OC)ccc(C(=O)C(=O)NC(CNC(=O)C=CC(C)C)CO)cc1Cl c1(C(C(=O)NCC=CCNC(C(c2ccccc2)C)=O)O)cccnc1 CCCC(CC)CCC(=O)NCC1(C(=O)N(C)CCc2cnc[nH]2)CC12CCC2 CC1CN(C(c2cc(O)nn2C)=O)C(C)CN1C(c1ccc(CO)o1)=O Cc1c(C(=O)N)nc2sccn12.C1(O)CCCN(C(C2CC2C(N)=O)=O)CC1.C C(=O)(C1=CCCN(c2ncncc2Br)C1)NCCCCCNC(C)=O C1(C(C)NC(=O)Cc2cn[nH]c2)CCN(C(=O)CC2CCC(=O)NC2)CC1 CC(O)C(C(=O)NCCCCNC(c1csc(C(F)F)n1)=O)NC(N)=O c1(C(N2CCOCC(CNC(C(C)SC(C)C)=O)C2)=O)nn(C)c2c1CCCC2 CC(=O)CCN=C(NCCN1CCCC1)N(C)C1CC1c1ccco1 N1(C(c2cc(C)oc2)=O)CCN(C(=O)C=Cc2cnn(C)c2C)C(CC(F)F)C1 C1(NC(c2cc(C)[nH]c2C)=O)CC2CC(NC(c3ccccc3F)=O)CC12 c1(C(=O)NCC2C(C)CN(C(C3CCC(C)S3)=O)C2)c(Cl)nc2ccccn12 C(=O)(C(F)(F)C(C)O)N(CCC(C(C)C)NC(COCC=C)=O)C c1(CCC(=O)NC2CN(C(C#CC(C)C)=O)C(C)C2)cccc2cnccc12 CCCCC(C)C(=O)N1CCC(C)(CC(=O)NCCn2cc(CC)cn2)C1 Cn1cc(Cl)c(C(=O)NC2C3CN(C(C4(C5CCC5)CCCO4)=O)CC23)n1 C(=O)(C(O)CCC(C)C)N(CCC)CCNC(=O)CSC c1(C(N(CCCNC(C(C(C)O)(F)F)=O)C)=O)cnc2c(n1)CCCC2 c1(Cc2nc(CC)nn2-c2ccc(OC)cc2)ccccc1S(C)(=O)=O S(=O)(=O)(c1ccc(Br)cc1NCCSC)N(C)Cc1ccn(CC)n1 C1(C(=O)NCc2cccc(C)c2)C2C3CC4C1C2C34C=O.C1(F)CCC1 c1(SC)ccc(O)c(C(=O)NC2CCCCN(C(C3CN(C(N)=O)C3)=O)C2)c1 c1(NC2CC(C)(C)OC2)ncccc1S(=O)(=O)NC1CC=CCC1 c1(C(=O)NCC(CNC(=O)C=Cc2ccsc2)O)cnc2c(Cl)cccn12 C1(CC)CN(C(=O)CN2CCC(=O)NC2=O)CCN1C(=O)CCCCC1CC1 c1(CC)nc(C)c(CC(=O)N)c(C)n1.C(=O)C(C)(O)C1CCOC1.C1CC1.C C1(NC(CC(CCCC)O)=O)CCOC2(CCN(C(=O)C(C)(C)F)CC2)C1 c1(C(=O)NC(C(C(C)C)NC(=O)CC2CC2)C)cc2cccn2cn1 S(=O)(=O)(c1cn(C(C)C)nc1C)NCC(CC)C(C)C c1(OC)cc(C(=O)NC2CC2CNC(=O)C(C)C)cc2cn(C)nc12.S C#CC1CC2(CC2)CN1C(=O)CC1(C)CCN1C(C1(CC=C)CC=CC1)=O C1(NC(C(c2c(C)cccc2)C)=O)CCN(C(c2cnoc2C)=O)CC1O Cc1c(CC(=O)NCCC2(CN)CCOC2)cnn1C c1(OC)nc(=NC(C)CC(C)NC(=O)C2=CC(C)(C)C2)nc(SC)[nH]1 N1(C(C=CC2N(C)CCC2)=O)CC2CC(C1)CN(C(=O)CC1(C)CCCO1)C2 C1(C(N2CC(C(=O)NC3(C#C)CC3)C(C)(C)C2)=O)(OC)CCC(C)(C)C1 c1(C(=O)NC2CC(NC(C=C(C)C3CC3)=O)C2)cnc2c(c1)CCCO2 Cn1nnc(C(=O)NC2CC(CC(N3CCC(CNC=O)CC3)=O)C2)c1N C1(CNC(c2ccc(F)s2)=O)CN(C(=O)CO)CC12CCC2.c1ccccc1F c1occc1C(=O)N.C(=O)(CC)N(CC(C)O)CCOCC.C=O.N CC(C(C)(C)C#N)NC(=O)C(O)CNC(=O)CCCC1CC1C C(C(C)C(F)C(=O)NCCc1ccn(C)n1)NC(CN(C1CC1)CC)=O C1(CC(C)C(=O)N)CCN(C(C2CC2c2ccco2)=O)CC1.C12CCC(C1)C2 CC(C)C(C)CNC(=O)C=Cc1cncn1C.C(=O)(CC)N.CCN(C)C Cc1ccc(C(=O)NC2CCC2NC(c2cc3sccc3[nH]2)=O)c(Cl)c1 CCCC(CC(C)C)C(=O)N1CC2CCCN(C(=O)C(F)C(C)C)C2C1 c1(C(=O)NCC2C(NC(c3c(Cl)cc(C)s3)=O)CCC2)ccn2nccc2c1 c1(CNc2ccnc(C3(C)CC3)n2)cccc([N+](=O)[O-])c1 Cc1nc(C)c(C(=O)NCC2(C(=O)N(C3CCN(C)CC3)C)CC23CCC3)s1 N1(C(c2cn(C)nc2O)=O)CCC(O)C(NC(c2cccn(C)c2=O)=O)C1 C(CN=c1ccnc[nH]1)C1CCN(C(c2c(CC)nc[nH]2)=O)CC1 C1(C2CC2)(C=O)CC=CC1.C(CC)(C(=O)NCC(C)(C)OCC)OCC C1(O)(CN(C(COCCCCCC)=O)C)CCCN(C(=O)CSC2CC2)C1 N1(C(C(CC)CC)=O)CC=C(C(=O)NC2CCCCC2O)CC1 C1(C(N2C3CC(NC(C4CC45CCOCC5)=O)(C3)C2)=O)CCCC1C1CC1 c1(OC)cc(C(=O)NC2CCN(C(C34CC(C3)C4)=O)CC2F)c(C)cc1Br c1(C(C(=O)N(CCCNC(C(C)C2CC2)=O)C2CC2)C)ccc(Br)s1 CCCCC(C(=O)N1CCC(O)C(O)C1)NC(=O)CCc1cnn[nH]1 Cc1nccc(C(=O)NCC(CNC(C2CCN(C)C2)=O)C(F)(F)F)c1C N1(C(CC(c2cccs2)NC(C)=O)=O)CCC(NC(c2cscn2)=O)C(C)(C)C1 C1(C(N2CC(C)(NC(C(C)OC)=O)C2)=O)CC12CCCCCC2 c1(OC)ccc(C2CC2)c(C(=O)NCC2(C)CCN(C(=O)CCC(C)C)C2)c1 N1(CCOC)CCCC(NC(=O)CCc2ccn(C)n2)C1 c1(C(=O)NC2CCC(C(N3CCCCC(C)C3)=O)C2)cc2cc(Br)ccc2s1 N1(C(CC2CN(C)CC2O)=O)CC(C)(C)OC2(C1)CN(C(=O)CCO)C2.C1CC1 N1(C(c2ccc(SC)o2)=O)CCCC(O)(CC)C1.C(=O)(C(F)CC1CCOC1)N CC1CCC(C(=O)NCc2cncn2C2CC2)N(C(c2cnc(O)o2)=O)C1 N1(C(COc2cc(C)c(Cl)cc2)=O)CCC(C)N(C(=O)CCCCC(C)C)CC1 C1(CC=C)(NC(c2ncoc2C)=O)CN(C(C2CCC(CN(C)C)O2)=O)C1 N1(C(c2cn(CC)nc2)=O)CCC2CN(C(=O)C(F)(F)C(O)C3CC3)CCC12 C1(CCOC)CN(C(=O)C(c2cc(F)cc(F)c2)O)CCN1C(=O)CN(C)C N1(C(c2cc(C)nn2C)C(=O)NCCC2(C)CC2)CC(CO)OC2(CCC2)C1 CC(C)(C#N)CCC(=O)NC1CCCC(CNC(C2CCC3CC2CO3)=O)C1 O=C(C(O)CCCNC(=O)C(C1CC1)C1CC1)NC1CCC=CCCC1 c1(OC)ccc(NC(=O)C(=O)N(C(C)CCNC(=O)C=C(Cl)Cl)C)cc1 CC(C)C(C#N)C(=O)NCC1(C(C)(C)C)CCN(C(=O)C2=COCCO2)C1 c1(C(=O)NC2C(NC(C(CC)C3CCOCC3)=O)CCC2)ccncc1F Cc1cnc2cc(C(=O)NC3CN(C(c4nc(=N)cc[nH]4)=O)CC3(C)C)ccn12 N1(CC)C(=O)CCC1CC(=O)NCCC(C)(C)C.C(=O)(CCC1CCCC1)N CC1CN2CCN1CC2C(=O)NC1CC1.C1(C(NC)=O)CCC(N(C)C)CC1.C C(=O)(C1=CCC(F)(F)CC1)NC(CCC)CCCNC(=O)CN1CCCC1C C12(CNC(c3ccc(CCC)s3)=O)CCC1CN(C(C1CCN(OC)CC1)=O)C2 N1(C(C(C)O)=O)CC2CC(C(N3CCN(c4ncccc4C#N)CC3)=O)CC1C2 C=CC(C(=O)NC(C1CCCN1C(c1cn(C2CC2)nn1)=O)C)OC N1(C(c2cccc(CC#N)c2)=O)CCCC(NC(c2nc(Br)c[nH]2)=O)CC1 Cc1nn(CCNC(CCCC#N)c2nnnn2Cc2ccco2)c(C)c1Cl c1(C(N(CC(c2ccccc2)C)Cc2ccccc2)=O)ccnc(OCCO)c1 C1(N(C(c2cncc(-n3ccnc3)n2)=O)CC)CCCN(C(C2(SC)CC2)=O)C1 CC(C(=O)NC1CC(C)C1)S(=O)(=O)c1ccc(F)cc1.C1(C(=O)N)C=CCC1 Cc1cn(C)nc1C(=O)NC1CCOC1C(=O)Nc1cncc(CO)c1 CCC(C)CC(=O)N1CCCC1C(C)(C)NC(C1CC1)=O.N1(C)CCC(C)CC1 Cc1c(C(=O)N(CCNC(C2CC3CC3C2)=O)C2CC2)sc(Cl)c1Cl c1(-c2c(N)ccc(C3CCCN3)n2)cccc2occc12 CC1(CNC(=O)C=Cc2ccco2)CCN(C(=O)C=CCF)C1 c1(C(c2nnnn2C(C)C)OC)cnccc1N(C)C.c12ccccc1NC2 N(C1CCCc2cc(CNC(=O)CC3COC(=O)C3)ccc21)C(CCOCC)=O C(=O)(C(C)(O)C=C)N(CCCNC(CC=C=C)=O)C N1(CC)CC2CC1CN2C(C1OCCC1NC(c1cn(C)c(=O)n1C)=O)=O N1(C(C(C)=C2CCCC2)=O)CCC(C)C(NC(c2cccnc2)=O)C1.N(C)(C)C Cn1cc(CC(N2CCOC(C3CCNCC3)C2)=O)c(Cl)n1 CN1CCCC2CN(c3ccnc(N4CCCC(n5nccn5)C4)n3)CCC12 N1(C(CC2C(NC(C3CCC(C)(C)OC3)=O)CCC2)=O)CC2C(=O)NC(=O)C2C1 C1(NC(CCCN)=O)COc2c(C(=O)O)cnn2C1 N1(C(c2n(CC)ccc2)=O)CCCCC(NC(=O)C=Cc2cccn2C)C1 C1(CC(NOC(CC)C)=O)N(C(c2ccns2)=O)CCC1(C)C O=C(CCC(=O)c1ccc(Cl)s1)NCC(CO)NC(C1CCCOCC1)=O N1(C(C(=O)N(C)Cc2ccc(C)c(F)c2)=O)CCOc2ccc(O)cc2C1 C1(C(N2C3C(NC(C4(SC)CCC4)=O)C(CC3)C2)=O)(O)CCS(=O)(=O)C1 c1(C(N2CCC(N(CC#C)C(c3[nH]c(C)nc3C)=O)CC2)=O)ccc(N)cc1O N1(C(C=CSC)=O)CCC(C(C)NC(c2csc(C)c2N)=O)CC1 C#CC1CN(C(=O)C(c2ccnn2C)NC(=O)Cc2cncs2)CCO1 O=C(C1=Cc2cc(Cl)ccc2OC1)N1CC2(CCN(C(=O)C(O)C(F)F)C2)C1 c1(C(C(N2CC(C)(NC(CC3CCC(C)CO3)=O)C2)=O)=O)cc(F)ccc1F N1(C(CN(C(C(CC)OC)=O)C2CC2)=O)CC=C(C)CC1 N1(C(CCN(CCCCC)C)=O)CC(CNC(=O)Cc2cscn2)C2(CC2)C1 c1(CN(C(=O)COC2CCN(C(C3CCCC3)=O)C2)CC)cccnc1.O CCCC(C(=O)NCc1nccnc1C)NC(=O)CCC(C)N(C)C c1(C(N2C(CC)CN(C(c3cc(C)oc3C)=O)CC2)=O)cc(Cl)c(O)c(Cl)c1 C1(NC(c2c(C)n(C(C)C)cc2)=O)CN(CC(c2ccc(F)cc2)O)CCC1O c1(CNC(CCSCCCC)=O)ncccc1C(=O)NC(C)C(C)CO c1(CC2CCCOC2)ccc(-n2nc(C3CCC3)nc2Cc2ccccc2)cn1 CC1(C)COC(CC(=O)NC2CC(=O)N(C3CN(CC4CC4)C3)C2)C1 C1(CC(=O)NCc2c(C)nn(C)c2Cl)CCCC12CN(C(=O)CO)C2 c1(CC(=O)N(CCC(C)NC(C2(O)CC(C)(C)C2)=O)C)ccc(Br)cn1 N1(C(C2(C(N(C)C)=O)CC2)=O)CC(CO)(NC(c2cc(O)no2)=O)C1 c1(C(C(=O)N(CC)C)(F)F)ccc(=O)n(C)c1.CC1OC(=O)NC1C=O c1(N(C)Cc2ccc(C)o2)ccc(S(=O)(=O)N(C2CCOC2)C2CC2)cc1F C1(NC(C(=O)NC2C3CC3C3CC23)=O)CCCCC1O C(=O)(n1ccc(C)n1)NCC.c1(OC(=O)NC(=O)C)cnn(C)c1.N c1(CC(=O)OCC(=O)NCC(=O)OC(C)(C)C)ccc(I)c(Br)c1 c1(OC)cc(OC)c(C(=O)NC2(C)CCCN(C(=O)CC3CCC3)C2)cc1.O c1(C(N2CCC(C(=O)O)CC2)=O)cc(-c2c[nH]nc2C(F)(F)F)cc2[nH]ncc12 c1(C(=O)NC2CN(C(c3c(C)cc(C)s3)=O)CC2O)cccc(C)c1[N+](=O)[O-] Cc1cccc(OCC(=O)NCCC2(CNC(C3(O)CC3)=O)CC2)c1C CC1CCC(C)(C(=O)N(CCC(=O)NC(C2CCOC2)C)CCCO)CC1 C1(C(N(C)CCC2CCCO2)=O)CCN(C(=O)CC2CSCCO2)O1 c1(OC)ccc(C(=O)NC2CCC(C)N(C(=O)Cc3conc3C)C2)cc1OC c1ccccc1C(=O)N(C)CC.c1(C=O)ccco1.CCCSCC.C(C)=O C(=O)(C(C)C(=O)NC1CCC(C(=O)N(C(C)C)C2CC2)CC1)OC CCC(C)C(C(=O)N(C)Cc1ncc(C)o1)NC(C1CCC(=O)N1)=O C(=O)(C1CCCc2nn[nH]c21)N1CC(CNC(=O)CC=C(Cl)Cl)C1 c1(C=O)cc(S(N)(=O)=O)c(Cl)o1.c1(C(N(CCC)C)=O)ccc(F)c(N)c1F N1(C(C(C)NC(CC)=O)=O)CCC(CC(N2CC(C(C)CC)C2)=O)C1(C)C c1(N(C(c2cn(C)nn2)C(=O)NCCC)CC(C)C)ccccc1OCC CCCCCC#CCONC(=O)C(N)Cc1ccccn1 C1(NC(c2c(Cl)nsc2Cl)=O)CCCCC1.C12(C=O)CC(CN1C1CC1)C2.C c1(CC)cnn(CC(=O)NC2CC2)c1.c1ccccc1.C12(CCC1)C(=O)N2.C N#Cc1cc(C(=O)NCCOC2CCN(C(=O)C(c3cccnc3)O)C2)no1 C(=O)(C#CC1(C)COC1)N1C(CC(=O)NCCOCCC#C)CC(C)(C)C1 c1(C(=O)NCCCN(C(C)C)C(C2CNC(=O)C2)=O)ncnc(O)c1Br CCC(CCC(=O)NCC(C)(COC)CO)NC(c1ccc(Cl)s1)=O CC(C)C(CCNC(C1CCC(C)CC1)=O)NCc1ncncc1Cl N1(C(C(C)N(C)C)=O)CCN(C(c2c(Br)ncn2C)=O)CC1CO Cc1c(NC(N2CCOCC2c2ccccc2)=O)cnn1C1CCCCC1 C(CNC(c1ccc(Cl)c(F)c1)=O)(C(C)C(C)C)NC(Cc1nnc(C)o1)=O CCCC#CC(C)(C)NC(=O)C(C)(C)NC(=O)CCC(C)(F)F C(=O)(CC(CC#N)c1ccccc1)NCC(CN(C(C1C(C)OC(C)C1)=O)C)O N1(C(CNC(COC)=O)=O)CC2(C1)CN(C(=O)CC(C(F)F)C1CC1)C2 n1(CC)cc(C(=O)N(C)CCNC(c2cncnc2C)=O)c(C2CCOCC2)n1 C1(C(N2CC(C(C)NC(c3cc(N)cc(N)c3)=O)C2)=O)CCCCC1C1CC1 CC1(C)CCC(C(N2CCCC2c2ccco2)=O)CN1C(=O)OC(C)(C)C C(C)(C(C(=O)NOCCC(F)(F)F)NC(=O)CC1CC=CC1)OC c1(N2CCC(C)(CC)C2)nc(N2Cc3ccc(Cl)nc3C2)nc2c1CCC2 C(CN=c1nc2sccc2c(N2CC3CC2CN3C(=O)OC)[nH]1)(OCC)OC C1(NC(c2nc[nH]n2)=O)CCCCCC1C(=O)NC1(CCCF)CC1 C1(CC(=O)NCC2(F)CN(C(c3ccc(C(C)=O)cn3)=O)C2)CCCCCCC1 C(=O)(C(C)CC(=O)N1CCCC(O)C1)OC.c1(C(=O)N)c(C)nn(C(C)C)c1C C1(NC(C(C)(C)F)=O)CCCCC1NC(=O)CCc1nnc(C2CC2)o1 c1(C(N2CCC(F)C2)=O)ccc(O)c(Cl)c1.CC(C(=O)N)NC(C1CCC1)=O S(=O)(=O)(c1ccc(NC(C)CC(C)(C)CO)c(F)c1)NCC(CC)OC c1(-c2c(OC)ccnc2)cc(C(=O)NCc2ccccc2C#N)cc2c[nH]nc12 CC1CCN(CCC(=O)NCc2ccc(C(C)NC(c3cn[nH]c3)=O)cc2)CC1 c1(CC)nc2ccccc2c(C(=O)NCC(CO)NC(=O)COCCCF)c1C C1(NC(C(COC)O)=O)CC2CCC(C1)N2C(=O)Cc1cc(C)ccc1Br c1(CN(C(c2csc3c2CCCC3)=O)C2CC2)ccc2ccccc2c1 CC(C)CC(CNC(=O)CCF)NC(=O)CCc1ccc(O)cc1.C(N)(=O)N C1(NC(c2nc(CCC)sc2)=O)CC2CCC1N(C(=O)C(CC)n1cccn1)C2 N1(C(C2(C(C)(C)C)CCC2)=O)CCCC(NC(=O)CNS(N)(=O)=O)C1 N1(C(C(=O)NCC=C)C2=CCCCC2)CCc2c(Br)ccc(F)c2C1 N1(C(C(C)=C2CCC2)=O)CCC(CNC(C2CN3CCN2CC3C)=O)C(F)(F)C1 c1(C(=O)NCC(CN(C(C(CC(C)C)O)=O)C)O)ccc2scnc2c1 C1(CC=C)(NC(=O)C=COCC)CN(C(=O)C(C2CCOCC2)OCC)C1 C(=O)(CCCCCc1ccccc1)N(CCNC(c1ccns1)=O)C1CC1 N#Cc1cc(C(=O)NC2CC(C)(NC(c3ccccc3)=O)C2)c(O)cc1N c1(C(=O)NCC2CC3CC3N2C(c2cccnn2)=O)ccc2cccc(F)c2n1 Cc1cnn(CC(=O)NC(Cc2cn[nH]c2)C(=O)NCCc2ncccn2)c1 C(=O)(CCC(=O)NCC1(CCNC(c2cc(C)oc2C)=O)CC1)NC c1(OC)cc(C(=O)N)cc(Cl)n1.C1CCN(C(c2csc(C(F)F)n2)=O)C12CC2 C=CCC(F)(F)C(=O)NC(CNC(=O)CC1(OCC)CCC1)CC C1(C(N2CCN(C(=O)CN3CC4CC4C3)C(CCO)C2)=O)Cc2cccnc2C1 C12(C(=O)NC34CCCC(NC(CN(CCC)C)=O)(C3)C4)CCCCC1CCC2 c1(C(=O)NC2(CO)CCCN(C(C3C(C)=C3)=O)C2)cnc2c(c1)NC(=O)CO2 c1(OCC(=O)NC(CC)(C)CO)c(Cl)cccc1Cl CCC(CC)(CCC(=O)NC12CC(C1)C2)[N+](=O)[O-].C1(C)(CC(=O)N)CCCO1 C(=O)(C(CC(F)F)c1ccccc1)NCC(=C)C C1(C(=O)Nc2c(CC)cccc2)CCCC12CCN(Cc1cc(F)ccc1Br)C2 c1(C(=O)NCC2CCCC(CNC(=O)C(F)C3CCC3)C2)ccc2occc2c1 CCC(C(=O)NCc1ncc(C(=O)Nc2cn(C)nc2S)cn1)C(C)(C)CC c1(CN(C)C)c(N2CCN(C3CCN(C(=O)CP(C)(C)=O)C3)CC2)ncnc1Cl N1(C(CCN(C(CC=CCC)=O)CCO)=O)CCC(N=[N+]=[N-])C(O)C1 CCCC(C)C(=O)NC(CCC1CCC1)C(=O)N(C1CN(C)C1)C C1(C(=O)NCCS(CC=C)(=O)=O)CN(C(=O)C(C)C)CCC1(C)C c1(OC)ccccc1C(N1CCN(C(=O)C(C(C)O)NC(C2COC2)=O)CC1)=O c1(C(=O)NC2C(NC(CC(C)F)=O)CCC2)cc(C2(Cl)CC2)n(C)n1 N1(C(=O)NCC2(CO)N(C)CCOC2)CC2(CC1CO)OCCO2 Cc1nn(C)cc1C(C)NC(C1(NC(C2CCC(=O)N2C)=O)CCCC1)=O C1(C2CN(C(=O)CC34CCC(CC3)CC4)C2)CC1.C1C(F)(F)C12CCC2.O=C C1(NC(CS(C)(=O)=O)=O)CC(C(=O)NC2CCC=CCC2)C12CCC2 Cc1cc(C(=O)N)c(O)nc1C.C1CCC(O)C1.C1(C=O)CC1C(C)(F)F.C CC(C)CC(C(=O)NC1CC(C(=O)NCc2c(F)cncc2Br)C1)N(C)C c1(CC(=O)NC23CC2CN(C(=O)COc2cccnc2)C3)cc(F)cc(Br)c1 C1(CNC(c2ncsc2C2CC2)=O)CCCCC1.C(=O)(CCc1cncs1)N N1(CC)CCN(c2cnc(OCC)cn2)C(C)C1.c12ccnc(n1)OCCO2 C1(C)(CC)C=C(C(=O)N2CCC3(CC3C(N3CCS(=O)C(C)C3)=O)C2)C1 C1(C(=O)NCC(CC)NC(c2ccc(C(C)(C)C)o2)=O)CCC(F)(F)C1 c1(C(C(=O)NCC(CC)NC(=O)CN(C)C2CC2)(F)F)cc(Cl)sc1Cl C1(CC(=O)NCCC2(C(N(CCCCC)C(C)C)=O)CC2)CCC(C)C1 c1(C(=O)NC2CCC(NC(CCC=CCC=C)=O)CC2)ccn2c1CCCC2 CCC(C)C(C(=O)NCC1CN(C(c2csc(CO)n2)=O)C1)OC N1(C(=O)NCCc2cccc(C)n2)CCC2C(=O)NCC2C1 CCC(C)CCC(=O)N1CCN(C(=O)CC(O)C(C)C)C(c2ncc[nH]2)C1 N1(C(C(CCC)OC)=O)Cc2ccccc2CC1CNC(=O)C(C)(CC)CCC N1(c2ncnc3onc(C)c32)CCC2(CC1)C(NC(=O)C(C)N(C)C)CS2(=O)=O c1(C=O)c(Cl)cc(C(F)F)cc1Cl.C(CC(C)(C)C)NC(C(=O)NCC)=O c1(C(C)=O)c(N2CCN(C(=O)CCCC3CCCC(=O)N3)CC2)ncnc1Cl Cc1cn2c(CC(N3CC(NC(=O)C(O)CN(C)C)CC(F)(F)C3)=O)csc2n1 N1(C(CC2ON=C(C)C2)=O)CCN(CC(N2CCCC2C2(C)CC2)=O)CC1 N1(Cc2c(N(C)C)nccc2)CCC12CCSCC2 N1(Cc2c(OCC)ccs2)CC2CC1CN2C(=O)CCCC(=O)OC N1(C(C(CSC)C)=O)CC2(CCCC2)C1C(=O)NCCC1CCC1 CC1CC2(CC(C(N3CCC(C(=O)NCC(O)CF)(CO)C3)=O)C2)C1 c1(C(=O)NC2CCC(F)(CNC(c3nccc(C)n3)=O)C2)cnc2ccoc2c1 C1CC2COCC2N1C(=O)C=C(C)C(C)C.C1(C(=O)NC)(SC)CCCC1 c1(NCCOCC)nc2ccc(OC)cc2c(=NCCn2ccc(O)nc2=O)[nH]1 c1(C(=O)Nc2cccc(CNC(CC3(OC)CC3)=O)c2)nc2ccccc2[nH]1 CS(=O)(=O)c1ccc(C(=O)NCCCNC(c2ccc(O)nc2)=O)nc1 C(=O)(CC(C)(C)C(C)(F)F)N1C(CNC(c2c(CC)[nH]cc2)=O)CC(O)C1 Cc1sncc1C(=O)N(C1(CC(N2CC(CO)(CO)C2)=O)CC1)C C1(C(F)(F)F)(C(N(CCCC)C)=O)CCN(C)C1.C(C1CCCC1)=CC=O.N c1(NC(=O)Nc2ccccc2-n2ccnn2)cc(Br)c(F)cc1Br C1(C(=O)NCCN(C(=O)Cn2cnnc2)CCC)C(C)CC1C C(=O)(C(O)C=CCC)N(C(C)C(=O)N1CC(CC(N)=O)C1)CCC C(=O)(CN1C(=O)CCc2ccccc21)NC(CNC(C1(C)ON=C(C)C1)=O)CO C1(CC2(OCC)CCCC2)CN(c2ncnc(C(=O)OC)c2F)CCC1C c1(OC)cc(OC)c(NC2CCN(c3ncc(C4CC4)cn3)CC2O)c(OC)c1 N1(C(CCSC(CC(C)C)C)=O)CCC2(CC1)CC2NC(=O)C(F)OC(F)(F)F C(C(C)(O)C(=O)N1CC(O)(C(C)NC(=O)C(C)O)C1)OC c1(COC)ccnc(NCC(C)N(C)C(c2cn(C(C)C)nc2C)=O)n1 c1(C(=O)NCCCOCCC(=O)NCCc2nc(C)on2)ccc(C#N)[nH]1 C(C(O)CNC(=O)C1CC1)NC(=O)CNC(C1(CCF)CC1)=O c1(OC)ccc(OCCO)c(C(CC(C)C)NC(=O)CC2CC(N)C2)c1 c1(NC(C=C(C)CNC(c2cncn2C2CC2)=O)=O)cncnc1O c1(-c2cc(C(N3CCCC3c3cccnc3)C(=O)NC)on2)cccc(Br)c1 C1(CNC(CC2C(C)(C)CCO2)=O)CC2CCC1N2C(C12CCC(CC1)C2)=O C(c1ccc(Cl)c(Cl)c1)=CC(=O)NCCC(C)C.C1(CC(=O)N)COCC1O c1(OC)cc(CC(N2CCC(C(C)NC(C3COCCN3C)=O)CC2)=O)ncn1 C1(CNC(C(CC)OC)=O)CN(C(C2CC(=O)C23CCC3)=O)CC1(C)C Cc1nn(C)cc1C(N1CCOC(C(=O)N(C)CCc2cccs2)C1)=O c1(NC(C2C=CCN2C(C2CCN(CCF)C2)=O)=O)cccc(C2CC2)n1 C1(C(=O)NC(C)(C)CN2CCN(C(C3CCCS3)=O)CC2)CC(C2CC2)=NO1 O=C(CC1=CCN(C(=O)Cn2cncn2)CC1)NCC1CC2(CCC2)CO1 c1(C(N2CCC(CC=C)(NC(=O)CN3CC4CC4C3)C2)=O)cnc(C)nc1C C1(C)(C(=O)NC(c2c(C(N(CC(C)C#N)C)=O)con2)C)CCNC1=O N1(C(C(Cc2cn(-c3cccc(N)c3)nn2)OCC)=O)CCC(C)(C)CC1CC Cn1cc2c(n1)CCC(N(C(=O)Cn1cc(-c3ccc(Cl)nc3)nn1)C1CC1)C2 Cc1ccc(OCCCC(=O)NC(C)(CNC(c2nn[nH]c2Cl)=O)C2CC2)cc1 c1(NC(C2CCN2C(c2ccns2)=O)=O)ccc(Cl)cc1O C1(=CC(N2CCC(c3cn(CCOC4CCOC4)nn3)C2)=O)CCCCC1 C1(CNC(c2cc(C)n(C)c2)=O)CCC(C)N(C(c2ccc(N(C)C)nn2)=O)C1 CC(=O)CCCC(=O)NC1C2CCN(C(c3ccn(C(F)F)n3)=O)C12 C1(N(C)C(C2CC2(F)F)=O)CN(C(=O)CN2CC=CC2)CC1O C(CC=O)C1C(C(=O)OC)C1.C(CC1CC1)N(CC(=O)N)C.C1CC1 C(=O)(C(CO)C(C)C)NC(CCCC)CNC(c1ccc(C(C)(C)C)s1)=O C1(CN(C(C(C)N(C)C)=O)C)CCCCN1CC(=O)NC1CC1.c1ccccc1 CC1(C)CC(CNC(c2ccc(Cl)[nH]2)=O)CN(C(c2cc(CCO)on2)=O)C1 C1(C2CCCN(C(=O)C=Cc3ccc(C)cc3)C2)(NC(C2(C#C)CCC2)=O)CC1 C1(O)(CC(CC(O)C(F)(F)F)=O)CCN(C(c2cn(CCO)nn2)=O)CC1 N1(C(CC)=O)CC2CC(NC(c3n[nH]c(C4CC4)c3Br)=O)C1C2 c1(CCC)ccccc1NC(C12CC(NC(=O)CCC(=O)OC)(C1)C2)=O C1(C)CCCN1C(c1cc(N(C)C)nc(Cl)c1)=O.C(=O)C(F)=C1CCC1.CC CC1(C(=O)NCCC2(C)CCN(C(c3cc(C#N)cs3)=O)C2)CC2(CC2)C1 C#CCC(C)(CC)C(=O)NCC1CC(NC(=O)Cc2cc(O)nc(O)n2)C1 c1(C(C(=O)NCCN(C(=O)CCCCSC)CCC)(C)C)ccccc1Br CC1(C)OC(=O)CC1C(=O)NCCN1CCN(C(c2cncs2)=O)CC1 N1(C(c2c(C)nns2)=O)CC(NC(C2CC(NC3CC3)C2)=O)CC1C C(=O)(CCC(O)C(C)(C)C)N1CC(C)C(NC(c2cccc(N(C)C)n2)=O)C(C)C1 C(C(C(=O)N1CCC(NS(C)(=O)=O)C1)NC(=O)CCSC)OCC c1(OC)nscc1C(=O)NC(C1CC(NC(c2cc(Cl)no2)=O)C1)C CC1CC(O)CCN(C(=O)CCC2CCN(C(=O)C(C)(C)C3(O)CCC3)C2)C1 Cc1c(C(N2CC(NC(=O)CC3C=NN(C)C3=O)C2)=O)oc2c(C)cccc12 N1(C(c2c(NCC)scn2)=O)CCCCC(NC(C2(C)CCCC2C)=O)C1 C1(OC)CC(NC(=O)Cc2cscn2)CN(C(=O)CCc2ccc(O)nn2)C1 CN=c1ccc(C(=O)NCC2CCCN2C(=O)CC2CCCNC(=O)C2)c[nH]1.C C(=O)(C(F)(F)C(F)F)NC(C1CCCN1C(=O)C=Cc1cn[nH]c1)C C1(CC(=O)NC(C2CCN(C(c3scnc3Cl)=O)C2)(C)C)CCCNC(=O)C1 c1(NC(C)=O)cccc(C(=O)NC2CC(F)C2)n1.C(=O)CCCC1CC1.C N1(C(=O)OC(C)(C)C)CCOC(c2nc(C(C)(C)C)n[nH]2)C1.C(CCO)C=O.O c1(CC(=O)NC2CN(C)C2c2ccccc2)cc(Br)ccc1F C1(NC(C2(CC)CC(F)(F)C2)=O)CCCN(C(=O)CC2CC2(C)C)CC1 C1(C(N(C2CN(C(C)=O)C2)Cc2cccn2C)=O)OCCOC12CCC2 N1(C(C(CC)OC)=O)CCC2(CCC2NC(=O)C(C)C)CC1 Cc1[nH]ccc(=NC(=O)C2CCN(C(=O)C(C)(C)CCl)CC2O)c1C N1(C(C=CCC)=O)CC(F)(F)CC1CCNC(=O)C(C)(CC)CC C(=O)(C(CC#N)c1ccccc1)N1CC(O)(CCNC(CC2CN(C)C2)=O)C1 C1(C(=O)NC(CC)CNC(=O)CC2C(C)C2(F)F)CN2CCCN1CC2 C1(CC)CCCCN1C(C1C(C)(C)C1(C)C)=O.N1(C(C)=O)CCC(C(=O)N)C1 c1(C(CNC(=O)Nc2cccc(OC)c2C)O)ccc(S(C)(=O)=O)cc1 C=CC(O)(C(=O)N1CCCC(CNC(=O)CN(CCCCC)C)CC1)C(F)(F)F n1(CCC(=O)NC2(c3ccccc3)CC(F)C2)c(O)nnc1O.C1(=O)CCCN1 C1(C)(C(=O)NC(CN(C(c2cc(SC)oc2)=O)C)C)CCCCC1(F)F c1(C=O)cc(C)c(C)c(C)c1.CC1=NOC(CC(=O)NCCCOCC)C1.N C(=O)(C(F)C(=O)N1CCC1)OCC.c1(C=O)cccc(-n2cc(C)cn2)c1.C N1(C(c2c(CC)ccs2)=O)CCCC(CCNC(c2cnn(C3CC3)c2C)=O)C1 C1(NC(=O)C=CC2CCCCC2)CCC2CN(C(c3cc(F)cs3)=O)CC12 C1(NC(Cn2cc(-c3ccc(OC)c(Cl)c3)nn2)=O)CC(O)C12CCOCC2 N1(C(C(F)=CCC)=O)CCC(F)CC1C(=O)NCc1cncc(Cl)c1 c1(C(=O)OC)nc(Cl)[nH]c(=NCC2CCCN2C(=O)C(O)C2CC2)c1OC C1(NC(C(CC)C(C)C)=O)CCN(C(=O)Cn2cncc2C)CCC1CO CCC(CO)C(=O)N(CC(O)CN(C)C(c1cnc(-n2cccn2)cn1)=O)C C1(C(N(CCCF)CC)=O)COCCC1NC(=O)CC1CCC(C)(C)O1 CCC(C)(CNC(=O)CC1(NC(=O)CN2CCN(C)CC2)CC1)CC C1(N(C(c2c(Cl)n[nH]c2C)=O)CC)CCCN(C(C2(C)CCCS2(=O)=O)=O)CC1 C1(NC(C2=C(C)OCC2)=O)CC2CCC1CC2NC(=O)C(C1CCCCC1)O N1(C(CCC=CC)=O)CCC(C)C1C(=O)NOCCC(C)C C1(C(=O)NCCOC)CC2CCC(C1)N2C(C1(O)CC1)=O.Cc1ccccc1 C(=O)(C1CCCc2n[nH]cc21)N(C1CC2CCC(C1)N2C(=O)C(=O)C(F)(F)F)C c1(NC(C(COC)OC)=O)ccc(NC(=O)CC2(NCC)CCC2)cc1C N1(C(CC(COC)(C)C)=O)CC=C(C(C)(C)C(=O)NC2CCCC2(C)O)C1 C1CN(C(C2C3COCC23)=O)CCC1(F)F.N1(CC(=O)N)CCS(=O)(=O)CC1.C C=CC(CCC)CC(=O)NCC(C(=O)NC1(C(C)C)CC1)C(C)(C)C N1(C(c2scc(CC)n2)=O)CCN(C(C2CCOC2)=O)CC1C c1(C(C(=O)NCCCC)N(C)CC2CCCN2CC)cc(OC)ccc1Cl CN1CCN(S(=O)(=O)CC(=O)NC2(C)CCC2)CC1.c1(C(=O)N)ccnnc1S c1(C(=O)NC2CCCC2C)ccc(C(F)(F)F)cc1.C1(O)(C=O)COC1.N N1(C(C=C(C)Cl)=O)CC2CC(NC(=O)CCc3cnc(C)s3)C1C2 C(c1ccc(C(N)=O)o1)=CC(=O)N.CC1CCC(=CC(=O)NC(C)C)C1 CCC(C)C(O)C(=O)NC1CCCN(C(=O)COc2ccccc2)C1C Cn1c(C(N2CCCC2C2CCN(C(C3CNC(=O)O3)=O)C2)=O)cccc1=O C1(COC)(NC(=O)C(C)NC(=O)CSC)CCCCC1 c1(CCCSCC(C)C)nc(C2CCCO2)nn1C1COC(C)(C)C1 N1(C(CC=CCC)=O)CCC(NC(c2cc3n(c2)CCC3)=O)C(CC)C1 N1(C(c2c(COC)scc2)=O)CC2CC2(NC(c2nc(=O)n(C)[nH]2)=O)C1 C1(NC(CCC2CCCN(C(COCC#C)=O)C2)=O)CCCC2(CCC2)C1 C[Si](C)(C)c1ccc(CNC(=O)NCc2ccc(C(F)F)nc2)s1 c1(C(=O)NCC(CN(C(COCC)=O)CC)C)ccc(F)cc1C1CC1 N1(C(C=C(C)Cl)=O)CC2CC(NC(=O)C3=C(Cl)CC3)CC2C1 C1(CC)C(C(=O)N(CCCC(O)CO)C)CCCN1C(=O)CC(C)O C1(CC)CCC(C)N(C(c2ccc(Cn3cccn3)o2)=O)C1.C12CCN(CC1)C2 c1(C(N2CCN(C(CC)C)CC2)C(=O)NCCC#N)ccc(O)cc1OC(C)=O C12(C(NC)=O)CC(C)(C1)OC2(C)C.C1CCCN1C(=O)CC1(O)CCC1.C c1(C=O)cc(S(N)(=O)=O)c(C)o1.N1(C(CN(CCC)C)=O)CC2(CCCO2)C1 N1(C(C(N2CC(OC)CC23CCCC3)=O)=O)CCOc2c(C)cc(F)cc2C1 CCC(O)C(=O)NC(C(=O)NCc1cn(C)cn1)C1(C)CC1 N1(C(C2CCC(F)CC2)=O)CCC2CCN(C(=O)C(C3CCCCC3)O)CC2C1 C(C(CC1CCCC1)C(=O)NOC)NC(c1c(CCC)[nH]cc1)=O.C1(C)CCC1 N1(C(C(CCC)C(=O)OC)=O)CCOC2(C1)CN(C(c1cccc(C)c1)=O)C2 N1(C(CC(CC)C(C)C)=O)CCC2(C1)CN(C(=O)CCN1CCOCC1)CCO2 C1(C(=O)NCCc2c(C)cccc2)CC(C)(C)CN1C(=O)CC1CCSC1 C#CC1CC2(CC2)CN1C(=O)C1CC1.c1(C=O)ccccc1.C(C)(C)C.C=O c1(C(N2CC(F)(C(N(CCC(N)=O)CC)=O)C2)=O)cncc(C#N)c1 NC1CCCC1CNC(=O)N(CC(F)(F)F)CC1CCC1 C1(C2CCS(=O)(=O)CC2)(OC(CC(=O)OC)CNC(=O)NC)CC1 c1(C(=O)N)cc(F)c(Cl)cc1Cl.N1(C(C2(OC(C)=O)CC2)=O)CCCC(C)C1 C=CCCC(C(=O)N1CCC(CF)C1)NC(=O)CN1CC(OC)C1 C(=O)C1=CNS(=O)(=O)N=C1C.C1(CC)CN(C(=O)COCCOC)CCC1 c1(-c2nc(Cc3ccc(F)cc3)nn2-c2cccc(Br)c2)ccc2ncnn2c1 Cc1nccc(C(=O)NCC(O)C(=O)NC23CCN(CC2)C3)c1N N1(C(CCC(=C)Cl)=O)CC2CC(C1)CN(C(c1ccc(F)c(C(F)F)n1)=O)C2 N1(C(c2cc(CC)oc2)=O)CCCC(N(C(=O)CC2C(=O)N(C)N=C2C)C)CC1 CN1CC2(CCN(C(=O)COC3CN(C(C4CC(CCO)C4)=O)C3)CC2)C1 c1(OC)ncc(C(=O)NC2CCCCC2)c(C)n1.C(=O)(C(C)Cc1ccco1)N N1(C(C2CC(CC)OCC2)=O)CCOC2(C1)CN(C(C1(OC)CCC1)=O)C2 Cc1c(CC(=O)NCC(C)N(C)C(C2COC(C)(C)CO2)=O)cccc1[N+](=O)[O-] c1(C(=O)NC2CC(CNC(CC3CCCC(C)C3)=O)C2)ccc(F)c(C#N)c1 CN1C2CCC1CC(=CC(=O)NC1CCCC1NC(c1n[nH]c3c1CCC3)=O)C2 c1(C(=O)NC2CCN(C(CC(C(=C)C)O)=O)CC2)ccc(C2=NOC(=O)C2)cc1 N1(C(Cc2n(C)ncc2Cl)=O)CCCC(NC(c2cnn(CCO)c2)=O)CC1 CC(N=c1ccn(C(F)F)[nH]1)c1nnnn1-c1ccc(Cl)cc1 c1(C(=O)NC(C(C)(C)C)CNC(c2ccccc2CO)=O)ccnc(F)c1N Cc1cc(NCCC(C)C(C)C)c(F)cc1Br N1(C(C(c2ccc(C)cc2)(C)C)=O)CC2(C1)CN(C(=O)COC1CCCOC1)C2 C(=O)C(C#N)CC1CC1.c1(NC(=O)OC(C)(C)C)scnc1.[nH]1ccnn1 N1(C(C2(CC#C)CCCO2)=O)CCC(C(=O)Nn2cnnc2)C(C)(C)C1 C(N=c1[nH]c2cc(Cl)ccc2s1)C1(F)CC(NC(c2c(C)cccc2)=O)C1 C12(C(=O)OC)CCC(C(=O)NC3CCC3NC(=O)CNC=O)(C1)C2 N1(C(CCc2c(C)noc2Cl)=O)CCCC(C)C1CNC(=O)C1=C(Cl)CCC1 CCCCCC(O)CNC(=O)CC1(N(C)C(C2(O)CCCC2)=O)CC1 Cc1csc(C)c1NC(=O)NC1(n2nccn2)CC1 N1(C(c2cncc(C)c2)=O)CCN(C(c2ccc(C)s2)=O)CC1c1ncc[nH]1 C12(NC(C3C(C)OCCC3)=O)CC(C)(C1)OC21CN(C(=O)C2=CC(C)(C)C2)C1 c1(CC(=O)NCC(C)NC(C(C)=C(CC)C)=O)ccc(Cl)nc1F c1(C(=O)NCc2cccc(C(=O)NC(C(CC)O)CC)c2)nc2ccccc2[nH]1 c1(OC)c(Cl)ccc(C(=O)NCC2CC2)c1N.C1(C)(CC=O)CC1(F)Cl c1(C(C)=O)ccccc1S(=O)(=O)N1C(CC(=O)NCc2ccon2)CCC1 c1(C(=O)NCC2C(NC(CCN(C(CCC)C)C)=O)CC2)csnc1Cl S(=O)(=O)(c1cccc(Br)c1)NC1CCN(C(c2cccc(NC(C)=O)n2)=O)C1 C(CN=C(NCC(=O)NS(C)(=O)=O)NCCS)C1C(C)(C)CCC1.C1CC1 O=C(CCC1=CCCCC1)N1CCC2(CC2C(N2CCc3ccncc3C2)=O)C1 CC1(C)CC1(C)C(=O)NCC1CCCC1.n1(CC=O)cc(C2CC2)nn1.N C1(CNC(C(CCC)NC(N)=O)=O)CC2CCC1N2C(=O)CC1CCCCC1 c1(CC(C)NC(=O)Cn2ccnn2)cnn(C)c1.C1(C=O)CC1.C1CC1.C Cn1cnc2ccc(C(=O)NCCNC(c3ccc(O)c([N+](=O)[O-])c3)=O)cc12 C1(C(=O)NC2(C)CCN(C(c3n(C)ncc3)=O)C2)CCCN(CP(C)(C)=O)C1 C(=O)(C(C)(C)F)NCC1C(CC(=O)NC2CC(C(C)O)C2)C1 Cc1cc(NC(=O)CC(C)CNC(=O)CC2CNC(=O)O2)c(=O)n(C)c1 N1(C(c2c(COC)ncs2)=O)CCN(C(=O)CC(O)C(C)C)C(C(C)(C)C)C1 C1(CNC(C(C)c2cc[nH]n2)=O)CCC(C)CN1C(=O)OC(C)(C)C N1(C(C2CCCN2S(=O)(=O)C2CC2)=O)C2CCC1CC1(C2)OCCO1 c1(OCCCNC(C2(C=C)CCC2)=O)ccc(N)cc1 CCC(C)(C(=O)NCCC1(NC(c2cnc3[nH]cncc2-3)=O)CC1)C(F)F C(=O)(CCCC(=O)N1CCC2CC12)NCCC.c1(C(=O)N)ccc(C(N)=O)cn1 N1(C(C2N(C(c3n(CC)ncc3)=O)C3C(C2)C3)=O)CCC2C(=O)NCC2C1 N1(C(C(CC)C)=O)C(C(=O)NC2CC(OC(C)C)C2)CCC1C1CC1 c1(OC)ccc(F)cc1C(=O)NCCOCC.c1(CC(=O)N)ccccn1 C1(NC(c2cn(CC(=O)NCCO)nc2)=O)CCN(c2ccncn2)CC1 N1(C(CCSCCC)=O)CC2(CCCC(C)O2)C1.c1(C=O)ncoc1C1CC1.N CC(C)C(C(=O)N(c1cccc(Cl)n1)C)N1CCCC1 N1(C(C(CC)(CC)CC)=O)CC2(CCC(NC(=O)C3=CCCS3)CC2)C1 N1(C(CC(CC)(C)C)=O)C2CCC1C(C)CC2.C1(C(=O)N)CN(C(=O)N(C)C)C1 c1(C(N2CC(CC(C)NC(C3(F)CCOC3)=O)C2)=O)ccc(Cl)c(F)c1F c1(C(=O)N)c(Cl)csc1Cl.C1(C(F)(F)F)(C(N2CC(O)C2)=O)CCCCO1.C C(=O)(C(C)CCC(C)(C)C)N1CCCC(NC(c2c(C)cc(O)cc2C)=O)C1 N1(C)CCN(CC=O)CC1.c1(C(=O)OCC)cccs1.C(C(F)(F)F)C1CC1 N1(C(CC2C(=O)N(C)C(=S)S2)=O)CC(S(C)(=O)=O)CC12CCC2 C1(CNC(=O)C(C2(O)CCCCCC2)(F)F)CCC2CNCC2O1 c1(C2CCN(C(C(=O)NC(C3(C)CC3)=O)=O)CC2)ccc([N+](=O)[O-])cc1 c1(C(=O)NCC(CC)NC(=O)C(C)OCC(C)C)cn(C(C)C)cn1 C(CCN=c1[nH]c2c(c(=NCC(=O)NC3CCS(=O)(=O)C3)[nH]1)CSC2)SCC C1(OC)CC(NC(=O)C(=Cc2ccco2)C)CN(C(c2cc(C)ccn2)=O)C1 N1(C(C)=O)CCCC(C(=O)N)C1.C1(c2nc[nH]n2)CCN(CC=C(C)C)CC1 N1(C(Cn2cc(-c3c(CC=C(C)C)csc3)nn2)=O)CC(C)CCC1C1OCCO1 c1(NC2CC(CNC(CC3CCC(C)C3)=O)C2)ncc(Br)cc1C#N CCC(C)C(C(=O)N1CC2CC1C2)N(C)C(c1cn(C)nc1OC)=O c1(C2N(S(CC)(=O)=O)CCC2)ccc(Cl)c(Cl)c1 C#Cc1ccc(CC(=O)N(CC(C)(C)NC(c2nc(Cl)sc2Cl)=O)C)cc1 c1(C(=O)NC2(CNC(CC3ON=C(CC)C3)=O)CCC2)ccnc2ncccc12 c1(NC)ccc(C(N2CC(O)(C)C2)=O)c(Cl)c1.C1(C=O)NC(=O)C2CC12.N c1(CNC(C2=CC(C)(CC)C2)=O)cn2ccc(C(=O)O)cc2n1 C1(CNC(C(C)SCC)=O)CN(C(=O)CCC2CCCN2C)CC(C)(C)O1 C1(CNC(c2cocn2)=O)CN(C(=O)CCC2CCCCO2)CC2(CCC2)O1 C1(NC(C2CCc3nccn3C2)=O)CCCC12CCN(C(C1(F)CC1)=O)CC2 c1(C(=O)NCCCCCN(C)C(c2nn(C)cc2Cl)=O)ccc(O)c(F)c1 CC(C)CCNC(c1ccnn1CC(F)(F)F)=O.c1(C=O)nccn1C(C)C C1(C(C)C)CCC(C(=O)NCCC2(O)CCCN(C(=O)C(C)(C)C)C2)C(=O)N1 c1(C(=O)OCC)cc2c([nH]1)CCN(Cc1nnc(C3CNC3)s1)C2 N1(C(c2cnc(CCCC)s2)=O)CCC(O)(CN(C(=O)Cc2ccns2)C)C1 N1(C(CC(=O)NC)=O)CCc2nn(C)c(C(=O)Nc3cccc(C#N)c3F)c2C1 C(CCCC(C(=O)NC1CCC1)N(C)Cc1ccc(Cl)cc1)OC C1(NC(=O)NCC2=C(C)CCC2)CC1C1CCCN(C(=O)OC(C)(C)C)C1 CC1CN(C(C2CC3COCC3C2)=O)CCC1C(=O)NCC=CC1CC1 C12(CC=O)CCCN1CCC2.C1(NC(CN(C(=O)OC)C)=O)CCC(CC)C1 C=C(CNC(=O)C(C)CNC(C1CC(OC)C1)=O)c1ccccc1 N1(C(c2cc(=N)[nH]cc2)=O)CCC(NC(=O)Cn2cc(CO)nn2)C(CO)C1 Cc1ccc(I)cc1NC(=O)C(C1CCN(C(=O)CC(C)(C)C)CC1)C C(=O)(C(=O)CCC(C)C)NCCC1CCCN(C(C2CCN(CC#C)CC2)=O)C1 C(CO)(C(=O)NCC1CCCCO1)NC(C(C)c1cc[nH]n1)=O C1(C(=O)NC2CN(CC)C2)CCC(C)(C)N(C(=O)CC2(C)CCOC2)C1 Cc1nc(C)c(CC(N2CCC(NC(C3CC34CCOC4)=O)CC2)=O)s1 C(c1ccncc1C)=CC(N1CCC(N(C(=O)CC(C)CC)CCCC)CC1)=O Cc1ccsc1C=CC(=O)N(CC(N1CCC1(C)C)=O)CC(C)C Cc1c(N2CCC(c3cc(C(=O)O)on3)CC2)ncnc1N1CC(=O)NC(=O)C1 C1(N(C(CCOCCOC)=O)C)CN(C(=O)C=Cc2ccc(C)o2)CC1O Cc1ccc(O)c(C(N2CC(NC(C3CCCCS3)=O)C(F)C2)=O)n1 C1(CC(=O)NCCC2N(C(C=C(C)Cl)=O)CCCC2)Cc2ccccc2N1 CC1CC(C)CN(C(=O)CCN(C(=O)C(c2ccccc2)F)CCCO)C1 N1(C(c2cncc(O)c2)=O)CC2CCN(C(c3cnn(C4CCC4)c3)=O)CC2C1 C(CCCC(=O)N1CCCC1C=CC(N1CCCC(CCO)C1)=O)N(C)C c1(C(=O)NCC2N(C)CCN(C(C(CCC)O)=O)C2)cc2cc(F)ccc2cn1 CC1(C)CN(C(C2(C)CC3CC3C2)=O)CC1NC(=O)C.c1(C=O)ccncc1 N1(C(C=CCC)=O)CCN(C(=O)CC2CCCC2)C(c2cccc(F)c2)C1 N1(C(Cc2c(C)n[nH]c2)=O)CC(NC(c2n[nH]c3c2COCC3)=O)CC(C)(C)C1 c1(CNC(C(CCC)CNC(=O)OC(C)(C)C)=O)cc2ccccc2o1 CCC(C)CCCCC(=O)N1CCN(C(c2cccn(C)c2=O)=O)CC(O)C1 c1(CC)ccc(C(=O)N(CCCCCNC(=O)Cn2c(C)ccc2C)C)c(C)n1 CCC(CCCO)NC(C1C2CC2CN1C(c1nonc1C)=O)=O O(NC(=O)CC1CN(C(=O)CNC(C)=O)C1)CCCCC c1(C(N2CCC(NC(C3CCN(C)CC3)=O)(CF)C2)=O)ccnc(Cl)c1O c1(C(N(CCC(=O)NCCCCCN(C)C)C)=O)ccc2c(c1)CCC2 CC1CCC(F)(F)CN1C(=O)C(C)(C)NC(C1CC1(F)F)=O N1(C(c2c(C)nccc2Cl)=O)C2CCC1CN(C(=O)Cc1ccsn1)C2 c1(OC)ccc(C(=O)NCC(C)N(CCC(=O)NC(C)C)C)cc1OC C1(NC(c2c(C)c(N)ccc2)=O)CCN(C(=O)C(C)(C)C2CCCO2)CC1(C)C Cc1oc(Cl)nc1C(=O)N(C(CNC(=O)C=Cc1ncco1)C1CC1)C n1(CC(=O)NCC(C(C)O)(C)C)cc(S(N)(=O)=O)cn1 C(=O)C=CS(C)(=O)=O.CC1(NC(=O)CNC(=O)C(F)(F)F)CCC1.N C(=O)(CCC(=O)NCC1CCC(C(=O)NCC(C)(Cl)CC)C1)NC c1(OC)ccc(S(=O)(=O)N2CCCC2(C)COc2cc(Cl)cnc2Cl)c(OC)c1 N1(C(CCCOC)=O)CC2CC(C(=O)NCc3ccccc3CO)(C2)C1 c1(C(=O)NCCC2N(C(C(C=CC)O)=O)CCCC2)ncn2cccnc12 c1(OC)cc(OC)c(C(=O)OCc2nnn(-c3ccc(Br)cc3)c2C)cc1Cl CCC(CC(=O)NCc1nn[nH]c1CO)NC(C1CCCOC1)=O CCC(C(=O)N)C(C)(C)CC.C1(S(C)(=O)=O)(C(N(CC(C)C)C)=O)CCOCC1 C(CC(CO)NC(=O)CN(C(=O)CC1CC(=O)C1)C)OCC.CCOC CCCC(C)(CC)C(=O)NC1C=CC(CNC(c2ccc(C)n2C)=O)C1 C1(NC(c2oc(C)c(CO)c2)=O)CC(O)CN(C(=O)Cn2cnnn2)C1 N1(C(CN(C(C=C(C)C(F)F)=O)CC2CC2)=O)CC2(CC=CC2)C1 C1(C(N2C3CN(C(C=Cc4c(C)ccs4)=O)C(C3)C2)=O)CCCC12CCOCC2 c1(CC(N2CC(C)(C)C(NC(=O)C3=CC4CCCC34)C2)=O)ccc2occc2c1 N1(C(CN2CCC(C)(O)C2)=O)CCN(C(C2COC(=O)O2)=O)C2(CC2)C1 CCC(C)C(O)CC(=O)NCCCN(C)C(C12CC3CC1(CO)CC3C2)=O C(C(O)(CNC(=O)NCCSCCO)CO)=CC CCC(C)CCNC(C1CC1C(F)(F)F)=O.C(C(C)(C)C)=CC(=O)N c1(COCCOC(C(C)N2CCCC2)=O)cccc(F)c1 C1N(C(=O)CN(C)C(C)=O)CCCC1(C)C.C(CCSC)(C(=O)NC)OC c1(CNC(c2ncsn2)C)ccc2c(c1)C(=O)NCCO2 N1(C(C(N2CCCC2)=O)=O)CCOC2(CCN(C(C3(N(C)C)CC3)=O)C2)C1.CC C1(OC)CCC2(C(=O)N(C)CCN(C(=O)CCn3ccnn3)C)CCC12 S(=O)(=O)(CC(=O)N(CC(O)CNC(c1cc[nH]c1C)=O)C)NC Cc1ccc(NCC2C(C)CCCN2C(=O)CCC2CCCOC2)c([N+](=O)[O-])c1 C1(CC(=O)N(CC#C)CCC)CCN(C(=O)C=Cc2cnc[nH]2)C1 N1(C(c2c(C)n(C3CCC3)nc2)=O)CC2CCC1CN2C(=O)C(C)CC(C)(C)C N1(C(C=CSC)=O)CC(NC(=O)Cc2ccc3c(c2)CCC3)CC2(CC2)C1 c1(C(=O)NC(CC(=O)N(C2CC=CC2)CC)C(C)C)c[nH]c2ccncc12 c1(C(N2CC(F)(CNC(COCCCC#C)=O)C2)=O)nc2ncc(C)cn2n1 N1(C(C2(C)CC2(F)F)=O)CC2(CCC2)CC1CNC(c1cc2ccccc2s1)=O C(=O)(CCCC(=O)C(C)(C)C)N1CC(CC(=O)Nc2c(CC)cccc2)C(C)C1 CC(C)(C(=O)NCC1CCCC1)C1CCCCO1.c1(C=O)coc(C(F)F)c1.N c1(C(=O)NCCC(CNC(=O)C=Cc2cocn2)O)ccc(=O)n2c1CCC2 N1(C(CSCC)=O)CCC(C)N(C(C2CCCN(c3ccc(C)cn3)C2)=O)CC1 C12(NC(C3CN(c4cccc(C)c4)C(=O)C3)=O)CCCC1N(CCOC=O)CC2 c1(C(C(N2C(CNC(C3CC3F)=O)CCC2)=O)O)cc(F)c(F)c(F)c1 N1(C(C(C=C)O)=O)CCc2sc(CNC(c3nnn4ccccc34)=O)nc2C1 c1(C(N2CCC(CC(=O)Nc3cnc(Cl)cn3)C2)=O)cccc(Cl)c1Br C1CCOC1.CC(C)(C1CCC1)C(C)=O.C(C)(C)C.N(C)C=O.CC.C=O.N C(C)(C(=O)N(C(C)CNC(C1CC(OC)C1)=O)C)SCC c1(C(C)=O)cnc(Cl)[nH]c1=NCC1CN(C(=O)Cn2cc(Cl)cn2)CCO1 C1(C)(C(=O)NCCC(C)NC(c2c(CC)non2)=O)CC2(CCC2)C1 n1(CCC=O)ccc(O)nc1=O.C(C)(CC(C)C)NC(c1cc(CC)[nH]n1)=O.N C1(NC(C(CCOC)NC(C(CCCC)F)=O)=O)CCc2nn[nH]c2C1 C(C1CN(C(C2CCC3(CCC3)O2)=O)CC1C(=O)N)=CC.C1CC(C)(C)CO1 C1(c2nnn[nH]2)CCCC1C=O.c1(COCC)cc(NCC2CC2)no1 N1(C(C2C(C)C2)=O)CCC(C=CC(=O)N(C)C(c2ccccn2)C)CC1 C1(CC(=O)NCC(CCCC)NC(=O)C(F)=CCCF)Cc2ccccc2O1.OC c1(N2CCCC(C)(CO)C2)ncc(S(=O)(=O)NCC2CC2(Cl)Cl)cc1Cl CC1CC(=O)NCC1C(=O)NCC(O)CNC(C1(n2cnnn2)CC1)=O c1(C(C)OC(c2nc3ccccc3n2C)=O)ccc2c(c1)OCCO2 CCC(C)CC(=O)NC(C)CCNC(c1cc(C2CC2)oc1C1CC1)=O N1(C(CCCOCC)=O)CCC(NC(c2cn(C)c(=O)cn2)=O)C(O)C1 c1(-c2cn(-c3c(CO)cccc3)nn2)c(Cl)cncc1Cl c1(C(N2CC3CCC(C2)N3Cc2cccc(O)c2)=O)cccc2c1OCO2 N1(C(C2CC(CC)C2)=O)CC2CCN(C(c3cc(C(N)=O)ccc3OC)=O)C2C1 N1(C(C(C)SCC)=O)CCN(C(=O)CCC=Cc2ccccc2)CC1CCOC C1CN(C(=O)C(C)n2ccnc2)CC1(C)C.C1(C(=O)NC)(C(=O)N)CCC1.C C(CSC)(C(=O)OCC1CCCO1)OC.C1CCCSC1 n1(CC)nc(C)c(CNC(c2cc(CCOC)on2)C)c1C C(=O)(C#CC1CCC(=O)CC1)NCC1C(C)CCCN1C(=O)CCC1CC1(C)C c1(C(=O)OC)cc(NC(CCC)=O)ncc1Cl.c12ccc(cc1)C(=O)COC2=O C1(C(=O)NC2(C)CCCN(C(c3c(C)noc3)=O)C2)CC2(CCC2)CCO1 CC(C(=O)N1CC(O)CCO1)N(C(=O)CC(=O)OC(C)(C)C)C CCC(C)CC(CO)NC(=O)CC1CC(NC(C2(C#N)CC=CC2)=O)C1 c1(N2CC(C)OC3(C2)CCCOC3)nc2ccsc2c(=NCC2CC3(CC3)C2)[nH]1 C(CC(C)C)(C(=O)N(C1CCN(C(=O)C(=Cc2c[nH]cn2)F)CC1)C)OC c1(C(=O)NC2C3(CCN(C(C(C)=CC)=O)C3)CCC2)cc(F)cc2nccnc12 CS(=O)(=O)CC(=O)NCC1CC(C(=O)NC(CO)CCC2CC2)C1 CC1COCCC1C(=O)NCCCCCn1cc(-c2cccc(N)c2)nn1 c1(C(=O)N(C2CCCCC2)Cc2ccc(C(F)F)cc2)ccc(Br)cc1[N+](=O)[O-] C(CC(C)(C)CC(=O)NC1CCC(CNC(=O)CC2CSCCS2)C1)OC Cc1ccc(CN2CCCC2C(F)(F)F)cc1.CC(=O)C1CC1.C(=O)N.CC C1(NC(C2C(NC(CCSC)=O)C2(C)C)=O)CCCC1(C)C Cc1ccc(NC(C2CN(C(=O)CCCCNC(N)=O)CCO2)=O)c(Br)c1 c1(OC)ccccc1OCCC(N1CC=CC1C)=O.C1(C=O)CC(F)(F)C1.N CC1CCc2c(C(=O)NCc3csc(C)n3)csc2C1.C(=O)CCP(C)(C)=O.N c1(C(=O)NCCN(C(=O)CCC(=O)c2ccc[nH]2)C)cc2c(=O)[nH]ccn2n1 N1(C(C(C)Oc2cccc(C)c2)=O)CC2CC(NC(=O)C(C)(C)C3CC3)C2C1 C(=O)(C(C)CC(N)=O)NC1(C)CN(C(c2c(C)nn(-c3cnn(C)c3)n2)=O)C1 CC1(C)CCN(C(C2CC(O)C2)=O)C1C(=O)NCC1CCN(C2CC2)C1 CC(C(=O)NC(C)(C)CCNC(c1cnn2c1CCC2)=O)S(N)(=O)=O C12(C(N3CCC(CC)C3)=O)CC1CN(C(C)=O)C2.CCCCC1(C=O)CC1.N C12CCC(CC1)CN2C(=O)C(C)(F)C(C)(C)F.Cc1cc(C(=O)NC)ccc1F N1(C(C(c2n(C)ccc2)=O)=O)CCC2(CC1)CCN(Cc1cc(Cl)ccc1Cl)C2 c1(C(N2CCC(CCNC(=O)Cc3cccc(O)c3)C2)=O)cccn2nccc12 C1(C(=O)NC(CNC(CCn2ncc(C)c2)=O)(C)C)CCCCCS1(=O)=O c1(C(c2nnnn2Cc2ccco2)NC(C2CC(OC)C2)C)cc(SC)sn1 C=CC(O)C(=O)NCC(CNC(=O)C(C)(C1CCOCC1)OC)OC CCS(=O)(=O)C=CC(=O)NCC1CCCN1C(C1(CC(C)C)COC1)=O Cc1nc(C)c(C(N2C(C(=O)NC3CC3)CC3CC23)=O)s1 S(=O)(=O)(c1ccc(N2CCC(C3CCC3)C2)cc1Br)N(CC)Cc1cccs1 CS(=O)(=O)c1ccc(CC(=O)N(C2CC2)C2CC2)cc1 c1(OCC)ccc(CN2CCOC(C(N3CCCC(CCOC)C3)=O)C2)cc1Br C1(CC)CN(C(=O)CS(C)(=O)=O)CCC1NC(c1c(C(C)=O)cccc1F)=O O=C1CC(C(N2CCCC(NC(C3(CO)CC3(F)F)=O)CC2)=O)CC(=O)N1 c1(C(N(CCCOC)C)C)cnc2ccc(OC(C)C)cc2c1 N1(C(CCN(C)C(c2csc(CO)n2)=O)=O)CCC2(CCO2)C1 C1(CNC(=O)C(N2CCC3(C2)CC(F)(F)C3)=O)COc2ccccc2C1 Cc1ncc(C(=O)N(CCCOCCNC(=O)C(C(C)C)NC=O)C)cc1C#N N1(C(C2(CNC(C=Cc3c(C)cccc3)=O)CCC2)=O)CC2CC(C1)C2(C)C C1(O)(C(C)NC(C(C)=CC)=O)CCN(C(=O)CC(F)(F)c2ccccc2)C1 c1(C(=O)NCC2(C)CCC2)cc(-c2cnc3cccnc3c2)c2cc[nH]c2c1 N1(C(C2(C)COC2)=O)CCC(C2CCN(C(=O)Cc3csc(S)n3)CC2)C1 c1(OC)cccc(F)c1C(=O)NCC1(F)CCN(C(c2ccoc2C)=O)CC1 C(=O)(C(C)CC1CCC1)N(CCNC(CCC)=O)Cc1ccccc1 N1(N(C(C)C)C(C2CCN2C)=O)CCC(CC(=O)NO)C1 c1(C(=O)NCCN(C(C(COC)O)=O)C)cnc2c(C)cccc2c1 C(N=c1[nH]c(=NCC23CCCC2C3)c2ccccc2[nH]1)C1CCS(=O)(=O)C1 C(CC(=O)N1CCCC1CC1CC1)(C(F)(F)F)NC(=O)C=Cc1ccco1 NS(=O)(=O)c1cccc(NCCC(c2ccccc2)NCc2cncc(F)c2)c1 CC(C)(C)C(C)(C)C(=O)NCC1CCN1C(=O)C(c1cccc(Cl)c1F)(F)F CCC(CC)C(F)C(=O)NCCOC1CCN(C(C2CCCC2(F)F)=O)CC1 N1(N(C)Cc2c(C(=O)OC)cccc2)CC(C2CC2)C(F)(C(=O)O)C1 N1(S(=O)(=O)C2CC2)CCc2cc(-c3ccc(F)c(Br)c3)ccc2C1 C=CCCCCCCCCCNC(c1nc(C)no1)c1nnnn1CC C1(C(=O)NCC2C(C)OCC2)CNC(=O)CN1C(C1CN2CCN1CC2)=O C(C(C)(C)C(=O)N1CCCC1C(=O)NC1CN(C(C)C)CC1C)OC N1(C(CC#N)=O)CC2C(CNC(c3ccnc(NCCO)c3)=O)C2C1 C1(C(=O)Nc2ccccc2)CCC2(CC2)N1C(C1CCO1)=O.c1(O)ccccn1 C(C1=CCCN(C(=O)CCOC2COC2)C1)NC(C1CCS(=O)(=O)C1)=O C1(O)(CC)CCN(C(c2ccc(CNC(=O)CCC(=O)C3CC3)o2)=O)C1 C(C(N=[N+]=[N-])C(=O)NCc1ccc(C(N2CCC2C)=O)cc1)OCC C1(CNC(C2(OC)CCOC2)=O)CN(C(c2c(C)cccc2F)=O)CC12CCC2 N1(C(=O)C2CC2)CCN(C(c2ccc(C3CCOC3)s2)=O)C(C(F)F)C1 CC1CN(C(c2ccccc2Cl)=O)CC1CNC(c1ncccc1CN(C)C)=O Cn1nc(C(=O)NCC(C2CCN(C(C3CC4CC4C3)=O)CC2)O)cc1O N1(CC(N2CC(C)(OCC(=O)N(CCCC)CCO)C2)=O)CCOCC1=O c1(CC)ccc(C(=O)NCCCCCn2cc(-c3cnc(C(=O)O)s3)nn2)nc1 c1(C(=O)Nc2n(C3CCN(C)CC3)ncc2)cc(N)c2ncccc2c1 n1(Cc2c(OC)ccc(-c3ccncc3)c2)cnc2sccc2c1=O C1(NC(C)=O)CCN(C(c2coc(CNC(=O)C(F)C3CCC3)c2)=O)C1 N1(C(c2c(CC)onc2)=O)CC(C2CN(C(=O)C(F)(F)C(O)C3CC3)C2)C1 CC(c1ccco1)=CC(=O)NC(C1CC(NC(=O)CC2CCC(C)C2)C1)C N1(C(C(C)SC)=O)CC(C)C(C)(CNC(c2c(SC)cccc2F)=O)C1 c1(CC(C)NCc2cc(-c3ccccc3)cs2)c(Cl)cccc1Cl c1(C(N2CCC(CC(NOCC(=C)C)=O)CC2)=O)cccc(C)c1N.CCC c1(OC)cccc(C(=O)NCC2(Nc3cc(Cl)c(O)nn3)COC2)c1[N+](=O)[O-] N1(CC2CCN(C(c3scc(CC)c3)=O)C2)CCCN(C(=O)C2=CCOC2)CC1 Cc1cc2ncnc(N3CC(O)(CCNC(=O)CS(C)(=O)=O)C3)c2[nH]1 CC1(C)CN(C(c2nnc(O)nc2O)=O)CC1C(=O)NC1(CCF)CC1 N1(c2n(C(CC#N)C(F)F)nnn2)CCc2[nH]cnc(=N)c2C1 C(CCN=c1ccnc(NCC(C)Oc2cccc(C)c2)[nH]1)=CCC c1(C(=O)NCC(CN(C(Cc2cc(C)on2)=O)C)O)cc(Cl)nnc1O c1(CNC(CCOCCNC(C(C2CCOCC2)C)=O)=O)c(F)cccc1F c1(OC)cc(CNc2nc(Cl)ccc2C(=O)Nc2ncc(F)cc2I)ccc1Cl C1(CC)CCC(C(=O)N(CCC(C)NC(=O)CCc2conc2C)CC)O1 C(C(=O)N1CCC(C(C)(O)C)CC1)(C(C)C)SCC.[nH]1ccnn1.C(C)=O.C CCC(C(=O)NC12CC(C(=O)N(CC(F)(F)Cl)C)(C1)C2)N(C)C C1(NC(C(C)=C2CCCC2)=O)CCN(C(c2cccc3c2CCO3)=O)C12CCC2 c1(N2CCC(COC(C3CC4(CCC4O)C3)=O)C2)ncnc2[nH]ccc12 C1(C)(CC(=O)OC)CCN(C(C(=O)NC2COC2)C(C)C2CC(F)(F)C2)C1 C1(C(N2CCN(CCN(C(=O)C(O)C)CCO)CC2)=O)CC2(C1)CC2(F)F N(C(=NCC(C)C#N)N1CCN(CCO)C(=O)C1)C1CC(OC(C)C)C1 c1(C(=O)NC2(C)CCN(C(=O)CNC(N)=O)CC2)nccc2[nH]ccc12 Cc1nccc(C(=O)NC2CCC(C)N(C(=O)Cc3cccnc3)C2)c1Cl c1(C(=O)NCC2CC(OC)CN2C(c2c[nH]nc2[N+](=O)[O-])=O)ncc(Cl)cc1F c1(C=O)csc(S(N)(=O)=O)c1.Cc1sc(O)nc1C(=O)NC.C1CCCCC1 Cn1cnn(CC(=O)NCC2CC(O)CN2C(=O)C(c2ccccc2)F)c1=O CCC(C)(C)CCCC(=O)N1CCC(C2(NC(=O)COC(F)(F)F)CC2)CC1 CCC(CC(=O)N1CCC2(CCCN2C(C2OCCC2C(C)C)=O)C1)CC(C)C C(=O)(C#CC1CCOC1)NCC(C)(C)C(=O)NCC1CC1[N+](=O)[O-] Cn1ncc(C(=O)NCC#CC(=O)NCC2CC3C=CC2C3)cc1=O c1(C(N(CC(CNC(C2(C)CC(C)C2)=O)O)C)=O)cnc2sccn2c1=O c1(C(N2CC3C(CNC(c4c(SC)ccs4)=O)C3C2)=O)c(F)ccc(Cl)c1N C#Cc1ccc(C(=O)NCCN(CCOC)C(c2ccncc2)C)c(Cl)c1 CC1C(NC(C2CC=CC2)=O)C(C)CCN1c1nnc(C2CC2)s1 N1(C(C2N(C(c3cnc(C)nc3)=O)CC(O)C2)=O)CC2(CCC2)OCC1C Cc1cc(C(=O)NC(C)C(C(C)C)NC(c2ncccc2F)=O)c(C)o1 c1(C(=O)NC(CC)(C)CNC(=O)C(C)N(C)C(C)=O)ccc2nn[nH]c2c1O C(=O)(CC1=NNC(=O)C1)N1CCC(N(C(C=Cc2n(C)cnc2)=O)CC)C(O)C1 c1(C(N(C2C3CN(C(CC(CC)C)=O)CC32)C)=O)cc2cc(Cl)ccc2nc1C c1(N(CC(=O)OC)C(N2CCC3(CCOCC3)C2)=O)cc2c(cc1Cl)NC(=O)C2 c1(CC(N2C(C(C)NC(c3nc(CCOC)oc3)=O)CCC2)=O)ccccc1O c1(NC2CCCC(NC(c3cc(C4CC4)no3)=O)C2)ccc([N+](=O)[O-])cn1 N1(C(C2CN(C)C2)=O)CCCC12CCN(C(=O)CCc1cnc[nH]1)C2 c1(CN2CCC(C)(C(=O)NCC(F)(F)CO)C2)c(O)cc(Cl)cc1Cl CC(C)CC(C(=O)NCCCC1CCCN1C(=O)C(O)C(C)(C)C)N(C)C c1(N2CCCC(CC(N3CC(=O)NCC3)=O)C2)ncnc2ccc(Br)cc12 C1(NC(C(=O)NC(C2CC3CCC2O3)C)=O)CC2CCC1O2 c1(CCC)nc(C)c(C(N2CCOCC2CNC(=O)C(n2ccnc2C)C)=O)s1 CC(C)(C(=O)NC1CN(C(=O)C=CC=C(Cl)Cl)C2(CCC2)C1)S(C)(=O)=O C(=O)(CCCC(F)(F)Br)NCC=CCNC(c1cc(C(C)=O)oc1C)=O C1(C(=O)N)CC2CN(C(=O)C=CCN3CCC3)CC2C1.CC1(C(F)F)CC1 CCC(C)(CC)C(=O)N1CC2(C1)CC(C)(O)C2.C1(CC(=O)N)NC(=O)NC1=O C(=O)(C(C(C)O)NC(=O)NCC(c1ccc(C(C)(C)C)cc1)C)OCC c1(CC(N2C(C3(C(N4C(COC)CCC4)=O)CC3)CCC2)=O)ccc(O)cc1 CS(=O)(=O)c1cccc(CN2CCC(C(=O)Nc3nccc(I)n3)C2)c1 c1(NC(CCC2CCC(NC(CC3N(C)CCC3)=O)C2)=O)ccc(CCO)cc1 N1(C(C=CSC)=O)CCC(C2CCC2)(CNC(C2CC(OC3CC3)C2)=O)CC1 n1(CC)ccc(C(=O)N(C2CCN(C(=O)CC3CCC(C)C3)CC2)C)cc1=O CCCC(C)CC(=O)NCC=CCC(=O)NOC(CC)CC c1(CNC(c2ncccc2Cl)=O)ccnc(N2CCCC(O)C2)c1 C1(C(N2CC(C#CC)C2)=O)CC2CCC1N2C(=O)C(CC)(CO)OC c1(NC(CCC)C)ccc(S(=O)(=O)NC)cc1Br.C(C(F)(F)F)NCCOC.O c1(C(=O)NC2CC(NC(c3nocc3Cl)=O)C23CCC3)cc2c(cc1Cl)OCO2 c1(CC)cccc(C(N2CCC(C)(NC(C3CCCCO3)=O)C2)=O)c1 c1(C(N2C(C)CC(NC(CCCCCOC)=O)C2)=O)cnn2c(=O)cc[nH]c12 C1(NC(CCCC)=O)CC2CN(C(=O)CC3SC4=NCCN4C3=O)CC2C1 N1(C(C)=O)CCCC(CC(N2CC(C(C)NC(c3cccc(=O)o3)=O)C2)=O)C1 N#Cc1cc(F)cc(F)c1NC(c1cc(NC(=O)N)ccc1F)=O.C1CC1.C c1(NC(C(C)(C)N)=O)cc(OC(F)(F)F)c(Cl)cc1Br c1(NC(CCC2N(C(c3cncnc3)=O)CCC2)=O)c[nH]ccc1=O C#Cc1ccc(C(=O)NC(C)(CNC(c2ccc(C#N)s2)=O)C(C)C)nc1 C(=O)(C1CCCn2ccnc21)NC(N1CC(N2CCC(N=[N+]=[N-])CC2)C1)=O CC(C)(CC(=O)NC12CC1CN(C(=O)C(F)OC(F)(F)F)C2)C(F)(F)F C(=O)(C(C)(CO)CC)NC(CN(C(=O)C(=Cc1cnn(C)c1)C)CC)C C(=O)(C1Cc2ccc(Cl)cc21)N(C1CCCCN(C(c2c(Cl)cnn2C)=O)C1)C C1(CC)CCCC1(C)C(=O)NC1CC(F)C1.C1(S(C)(=O)=O)(C=O)CC1.C N1(C(c2c(C)cns2)C(=O)NCCCF)CCC(c2cccc(F)c2)C1(C)C c1(C(=O)NCC2(O)CN(Cc3c(C)nc(C)[nH]3)C2)cc2ccncc2[nH]1 Cc1nc(CC(F)(F)F)sc1C(=O)N(C)CC1(C)CC1.C(=O)CC.CCF Cc1c(CN2CC(C)(C(=O)N(C)CCc3ccccc3)C2)oc2ccccc12 C1(C(=O)NC2C(C(N(CC(C)C)CC)=O)C2)CCCS1 C(=O)(C(C(C)CC)NC(C1CC2CCCC2C1)=O)N(CCCCC)CCO N1(C(N)=O)CCCC1C(=O)NCC(c1ccccc1)CNC(c1nocc1Cl)=O C1(CNC(C2CCN(CC(F)F)CC2)=O)CCCN(C(=O)C(O)C2CCC2)CC1 C1(CNC(NC2(C)CCC2)=NCCc2ccccn2)Cc2ccccc2CO1 C1(CCC)CN(C(=O)CCCN(C)C(C)C)CCN1C(c1cc(F)ccc1N)=O C1(NC(C)=O)CCC(C=O)CC1.C(c1ncc[nH]1)=CC(N1CC(CC)C1)=O.N Cc1cc(C)n(CCNC(=O)COC2CCOCC2)n1.C12CCN(C1)C2=O Cc1ccnnc1C1(CNc2csc(Br)c2)CC1 C(=O)(C1CCCc2nn[nH]c21)N1CCC2CN(C(C3(COC)CCC3)=O)CC2C1 O=C1CCC(C(=O)N2CCN(C(C3CC3F)=O)C(c3cc(F)cc(F)c3)C2)=NN1 c1cc(Cl)cc(Cl)c1.C1(NC(C2CC(CC)C2)=O)CCCCC1NC(=O)CC C#Cc1cc(C(N2CCN(C(c3c[nH]cc3Br)=O)C(CO)C2)=O)cc(F)c1 C1(F)(C(N(C2CCCC2)C(CC)C)=O)CCN(C(C2CN(C(C)C)C2)=O)C1 c1(C(=O)NCC(C)NC(C(n2cc(C)nc2)(C)C)=O)c(Cl)ccc(F)c1C C1(NC(=O)C(O)CC2CC2)CCN(C(c2cccc(Cl)c2F)=O)CC1O N1(C(CC(C)n2cccc2)=O)CC2CCC1C(NC(C1(C)CCCCC1)=O)C2 c1(NC(C)=O)sc(Cl)cc1C=O.C1CCN1C(C1CC1C(C)(F)F)=O.N C1(C(N2CCC(N(C)C)C2)=O)CC2(CCN(C(=O)C(Cl)(Cl)Cl)CC2)CO1 c1(OC)cc(C(=O)NC2COCCC2NC(C2COC(=O)N2C)=O)ccc1Cl N1(C(c2cnc(C(=O)OC)s2)=O)CC2CCC1(CNC(=O)CCCC(C)C)CC2 c1(C(N(C2CCN(C(C3(C=C)CC3)=O)CC2)CCO)=O)ncc(F)cc1C Cc1cc(NC(C2(C)CCCN2Cc2cccc(C)c2Br)=O)c(O)c(C)c1 C(CCC(=O)N1CC(CCCCNC(C2(C)CC2F)=O)C1)NC(C)=O C1(NC(C(C(C)C)SC)=O)CC(C(=O)NCc2nnn(CC)n2)=CC1O N1(C(C2(COC)CCC2)=O)CC(NC(=O)CCC2CC2(Cl)Cl)CC12CCC2 c1(C(N2CCCC2)=O)cc(S(N)(=O)=O)co1.c1(SC)cn(C)nc1C(=O)N C1(NC(C2(Cl)C(C(C)=O)C2)=O)CCCC1CC(=O)NCc1ccon1 C(C1CCN(C(C2CC3(CC(=O)C3)C2)=O)CC1)=CC(=O)NCCC=O.CC Cc1ccc(NC(C2(NC(=O)C(CN(C)C)C(C)C)CCN(C)C2)=O)cc1O c1(C(=O)NC2C(CC)C2)coc2c1CN(C(=O)C(C)(F)F)C2 c1(C(N2CCC(C)(NC(C=C(C)c3cccs3)=O)C2)=O)cnn2cccnc12 C1(CN(C(c2nc(COC)oc2)=O)C)COCCN1C(=O)C(CCO)N(C)C CCC(C)(C)C(C)CC(=O)NC1(C)CN(C(=O)C(O)C(C)C)C1 Cc1[nH]c(C)c(C(N2CCCC2C(=O)NCc2nnn(C)c2C)=O)c1C C1(CC(=O)N(C)Cc2nc(C)on2)CC(C)N(C(c2cn(C)nc2C)=O)C1 n1(CC(CC)O)cc(C(C)N(C(=O)CCc2ncco2)C)nn1 N1(C(Cc2nc(COC)sc2)=O)C(C(N2CCCC2)=O)C2CC(O)C1C2 c1(C=O)nc(C(C)C)oc1C.C1(C(=O)OC)CC(C(=O)NCC(C)C)C1.N c1(C(=O)NC(Cn2cc(CCOC)nn2)CC(C)C)ccnc2cc(C)ccc12 Cc1ccnc(C(=O)NCCC2(CNC(=O)CCn3ccccc3=O)CC2)c1 C1CC(C)(C)CN1C(=O)C(n1ccnc1C)C.N1(C(C)=O)CCCC1C(=O)N.C N1(C(C(CC=C)OC)=O)CC(C)N(C(C2(COC)CCOCC2)=O)C(C)C1 N1(C(c2nccc(C)c2)=O)CC23CCCCC2(C1)CN(C(c1c[nH][nH]c1=N)=O)C3 N1(C2CN(Cc3c(C(C)C)n[nH]c3)C2)CCN(CCc2cccnc2O)CC1 C1(C(=O)NC(CC)CSC)C=CCN1C(=O)CCN1CCCC1=O c1(C=O)cnc(O)n(C)c1=O.C=CCC(C(=O)N)NC(C)=O.C1CC(CC)C1 c1(C(=O)NCC2N(C(c3c(C)snc3)=O)CC(C)(C)C2)cccc2nnn(C)c12 C1(NC(C(CC=C)CC)=O)CC2CC(C1)N(C(=O)Cc1cscc1Br)C2 c1(C(C(=O)NC2(CC=C)CN(C(=O)CCOC3CC3)C2)C)ccc(C)cc1 C12(NC(c3c(C)nsc3)=O)CCCC1N(C(c1cc(C(C)C)no1)=O)CC2 c1(OC)cc(C(=O)NCCN(C(=O)CN2CCCCCC2)C)cnc1Br Cc1nc2ccc(C(=O)NCC3(F)CN(C(c4cc(Cl)cnn4)=O)C3)cc2[nH]1 C1(OCC)(CNC(=O)Cc2ccsc2C)CN(C(=O)C(C)C2CCOC2)C1 N1(C(C(c2ccc(C)cc2)=O)=O)CCC2(NC(c3ccc(Cl)cc3Cl)=O)CC2C1 N1(C(c2cncc(C#N)n2)=O)Cc2[nH]nc(-c3ccccc3OC3CC3)c2C1 CC(C)(C)CC(F)C(=O)N1CC(OCC(=O)Nn2ccnn2)C1 c1(C(=O)NCC2CN(C(=O)C(O)C3CCC3)C2)sccc1C1CC1 CC1CC(NC(=O)C=Cc2cncs2)CN(C(=O)CN(CC(C)(C)C)C)C1 c1(CC(C)NC(=O)OC(F)(F)C(F)(F)F)ccc(OC(C)(C)C)cn1 c1(C(C=O)(F)F)ccc(=O)n(C)c1.C1(C(=O)NCCCC)CCC(C)(C)O1.N C1(F)(CNC(c2c(C)nc(CC)o2)=O)CCCN(C(=O)C)CC1.c1cccs1 C12(NC(C3OCCN(C(CN4CCC(C)C4)=O)CC3)=O)CCC(O)(CC1)CC2 N1(C(C2(C(=O)O)CC2)=O)CCCC2(C1)CN(C(=O)CC1CCOC1)C2.CC C1(CC)CCCCCCN1C(=O)NCC(C(C)(C)C)SC Cc1c(C(=O)N(CC(C)NC(c2c(C(F)(F)F)cnn2C)=O)C)sc2cncn12 C(=O)(C#CC1CCCCC1)NC1C(CNC(C(C)(Cl)Cl)=O)CCCC1 N1(C(COCCOCC#C)=O)C2CCC1CCC2.c1(C(=O)N)cc(C)ccc1F CC1(C)OCC(NC(=O)Cc2csc(-c3cc(Br)cs3)n2)C1O N1(C(CCC#C)=O)CCc2cc(NC(c3ccccc3COC)=O)ccc2C1 C1(NC(C(=O)NC(C#C)CC2CC2)=O)CCCC(c2ccc(F)cc2)C1 C(C(CC(=O)NCCCC(C)(C)NC(c1cccn1C)=O)C(F)F)N(C)C N1(C(c2n(CCC)ncc2)=O)CCCC(N(C)Cc2ncnn2CC)C1 Cc1[nH]c(=N)sc1C(=O)Nc1cccc(NC(c2n[nH]cc2Cl)=O)c1 c1(CC(OCC)OCC)nc(C)c(C(=O)NC2CCCC(O)C2)s1 C(=O)(C(CC(C)C)OC)N1CC(CC(=O)NCc2cnc(OC)nc2)OCC1 N1(C(C2C(C)(C)CCCC2)=O)C2CCC1CN(C(=O)C=CI)C2 c1(C(c2n(CC=C)nnn2)NC(COC2CC2)CC)cccc(F)c1Br c1(C(=O)NCCC2C(C)CN(C(=O)C(=O)N(C)C)C2)cnc2[nH]nc(O)c2c1 N1(C(C=CC)=O)CCCC(O)(CCNC(=O)C=Cc2sccc2Br)C1 N1(Cc2c(C)c[nH]n2)CC2(CC(NC(=O)CN(C)S(N)(=O)=O)c3nccn32)C1 C(C(=O)N=c1ccn(CCO)[nH]1)N(C(Cn1ncc(C#C)c1)=O)CC(C)C C1(CC)CN(C(C2CCN(C(C)=O)CC2)=O)CCC1.C1(C(=O)N)CCCCC1(F)F N1(C(=O)C=CC(F)(F)F)CC(F)(C(=O)NC2CC2C2CC2)C1 CN1CCC(C(N2CCC3(C2)CN(C(=O)CCCOC2CCCC2)C3)=O)S1(=O)=O c1(CC(C(=O)NCCCCC)NC(C2CN(C(=O)O)C2)=O)ccnc(O)c1 CC1(C(=O)NCC2CC3CN(C(=O)Cn4nccn4)CC23)CCCCCCC1 CC1CC(CNC(C2CC(CF)C2)=O)CN(C(c2ccnc(Cl)c2N)=O)C1 C1(C)(C(=O)NCC(n2cc(-c3cccc(C(C)(C)O)c3)nn2)C)CNC(=O)C1 c1(C(N2CCCN(C(CC(CCC)(C)O)=O)CC2)=O)cccc2occ(Br)c12 C1(NC(Cc2c(C)non2)=O)CN(C(=O)C(C)C=O)CC2(CCC2)C1.C(C)(C)C c1(C(C)C)ncccc1NC(C1CCCN(C(C2CC=CCO2)=O)C1)=O N1(C(c2c(C)nc(CC)o2)=O)CCC(NC(c2cc(Cl)c(Cl)n2C)=O)C(F)C1 N1(C(c2cc(C)nn2C2CC2)=O)CCN(C(=O)C(C)C(C)C)C2(CC2)C1 C(C(=O)N(CCCSc1c[nH]nc1C(=O)OC)C)(C(CC)CCCC)N(CCC)C CC1CCCC(C(N2CC3CC2C3C(=O)NC2(CCF)CCC2)=O)C1 C1(C)(CNC(COCC#C)=O)CCN(C(C23CC2CNC3=O)=O)C1 N1(C(Cc2c(C)cc(C(F)(F)F)cc2)=O)CC=C(CCNC(C2CC2C)=O)CC1 CC(C)CC(C)OCC(=O)N(CCC(C)NC(c1cn(C(C)(C)C)nn1)=O)C c1(C(N2CC(NC(c3c(C)n(C(C)C)nn3)=O)C(O)C2)=O)cccc2oncc12 C1(N(CCC(=O)NC(c2nc(CC)[nH]n2)C)CCCN(C)C)CCCCC1C C(=O)(CC(C)CC(=O)O)NC1CCC(Cn2cc(CCC(=O)NC)nn2)CC1 c1(C(=O)NC2CN(C(=O)C(F)C3CCC3)CC23CC3)ccc2ccsc2c1 N1(C(c2ccc(CNC(C3CC(C)(O)C3)=O)cn2)=O)CC2CCC(C1)C(=O)N2 C(=O)(C#CC1CCOC1)NCC1COCCN(C(c2ccc(OC)c(N)c2)=O)C1 C12SC(=Nc3c[nH]nc3NC(=O)C1)N(CC)C2=O.c1(CC)cc2cc(F)ccc2[nH]1 c1(C(N2C(C)CC(NC(c3cc(C#N)cs3)=O)C2)=O)cnn2c(=O)cc[nH]c12 c1(C(=O)NC(CC(C)NC(C2C(C#C)C2)=O)C)cc(OC)c(F)c(F)c1 C1(C(N(CCCNC(CC(C)C)=O)Cc2ccccc2)=O)CCC2C1C2(F)F C1(CC(=O)NC)CN(C(C2CCC(=O)N(C)C2)=O)C(C)(C)C1.C1CCCS1.C C(=O)(CCS(=O)(=O)c1ccccc1)N1CC2OCC(C(=O)NC3CCOC3)C2C1 c1(CCC(N2C(CNC(=O)COc3cn[nH]c3)CC2)=O)ccccc1[N+](=O)[O-] C(=O)(CC(C)C(F)F)N(CC(C)NC(=O)CCc1conc1C)CC c1(NCC2CCC(N(C(C(C)SC)=O)C)CC2)ccc(C)cc1[N+](=O)[O-] C(=O)C1=C(C)OCC1.N1(C(C2(OC)CC(C(F)F)C2)=O)CCN(CCC)CC1.N C1(CC=C)(C(N2CCCC(CNC(=O)CC3CC(O)C3)C2)=O)CCCCC1 C=Cc1cc(C(N2CC(CC(C)NC(c3ncoc3CC)=O)C2)=O)cc(F)c1 c1(C(=O)N)cc(Cl)c(F)cc1F.C(C(C)(O)C)NC(C1C(C(C)(F)F)C1)=O CCC(CC)C(C(=O)N1CC(O)(CCNC(C2(Br)CC2(C)C)=O)C1)OC N1(C(C2(SC)CN(C(C3CCC(C4CC4)C3)=O)C2)=O)CCC(N=[N+]=[N-])CC1 N1(C(=O)Nc2c(C)nn(CCF)c2)CCOC(C)C1(C)C C1(NC(C(CC)CC(F)F)=O)CC2CCC(C1C)N2C(c1c[nH]nc1C(C)C)=O CC(F)(F)CCCCNC(C1CC=CCN1C(C1CN(C2CCC2)C1)=O)=O c1ccc(F)cc1Cl.C1CCOC1.N1(S(C)(=O)=O)CCC1C(=O)N.C(=O)C.C C(CC(=O)N1CCC(c2cnn[nH]2)C1)(C(F)F)NC(Cc1c(C)con1)=O c1(C(=O)NCCCCCCNC(C(OC)OC)=O)c(C)sc(C)c1Br N1(C(C(OC)OC)=O)C2COCC1CN(C(=O)CCc1ccc3cc[nH]c3c1)C2 C=CCC(C)(CC=C)NC(=O)CC1CCCC(NC(=O)C2=CCCC2C)C1 N1(C(c2ccncc2)=O)CCC(C=CC(N2CC3CSCC3C2)=O)CC1 c1(C(N2CC3CC(NC(c4cn(C)nc4)=O)C3C2)=O)ccn2ncnc2c1 N1(C(C2COCCN(C(c3c(C)ncnc3)=O)C2)=O)CCOC(C)(C)C1C N1(C(CSC(C)C)=O)CCCC1CNC(c1cn(C2CCC2)nn1)=O N1(C(C2(COC)COC2)=O)CCC(CF)(NC(=O)CCc2cnc(C)s2)C1 C#CCC(C)(C(=O)NCCC1OCCC1C)NC(=O)CCC1(C)N=N1 C1(NC(C2(F)CCCCC2)=O)CCC(C(N2CCC3CC23)=O)CC1 N1(C(COC(c2cccc(F)c2)C)=O)CCC2CN(C(c3nccn3C)=O)CC12 C(=O)(CC1C(=O)Nc2ccc(Cl)cc21)NCCN(C(C(CC)SC)=O)CCOC c1(CN2CC(F)(C(N3CCC(C)C(O)CC3)=O)C2)ccc([N+](=O)[O-])c(N(C)C)c1 c1(C=O)c(C=O)sc2ccccc12.C1(CC(=O)OCC)CS(=O)(=O)C1.N c1(C(N2CCC(C(=O)NCCNC(CC(C)C)=O)C2)=O)ccnc(F)c1Br c1(CN2CC(C)(C(N3Cc4cncnc4C3)=O)C2)ccnc2ccccc12 c1(C(=O)N)cnc2[nH]cncc1-2.n1(C(C)C)cccc1C(=O)NC1CCC(C)C1 C(C1CCN(C(c2ccc(O)c(F)c2)=O)CC1)=CC(=O)NC(C(C)C)C C(CCCC(=O)N(C)Cc1ncc[nH]1)N(C(C(CN(C)C)O)=O)C CC1(C(N2CCC(n3cc(CCCN4CCOCC4)nn3)C2)=O)CC1(F)Cl CC1(c2cn(-c3ccc(Cl)cc3F)nn2)COCCN1C(C1CCCO1)=O c1(C(=O)NC2CN(C(c3c(OC)csc3)=O)CC2C(F)F)cnn2c1CCC2 C(=O)(CCCCCF)NCC(CCC)NC(=O)COC1CCC1 c1(C(N2C(CCNC(c3nccc(CC)c3)=O)CCCC2)=O)ncc(N)cc1C c1(C(=O)NC2(C)CN(C(C(CCCC)CC)=O)C2)cc(S(=O)(=O)N(C)C)cn1C c1(OC)ccc2cc(C(=O)NC(C)CN(C(=O)Cc3cccnc3)C)ccc2c1 C1(CCNC(CC=CC)=O)CCCCN1C(=O)C(c1ccc(C)o1)C N1(C(CC(CCC)C)=O)CCC(N=c2[nH]c(Cl)ncc2Cl)C(F)(F)CC1 C1(NC(Cc2scc(C)c2)=O)CC(C)N(C(c2cccc(C(N)=O)n2)=O)C1 C=C(CNC(c1cc(C)[nH]n1)=O)CCNC(c1cn(CCCC#N)nn1)=O C(CC(=O)N(C(C)C(=O)N1CC(OC(F)F)C1)C)N(C(C)=O)CC1CC1 CC1(CC(=O)NC2CC(F)(CNC(=O)Cc3ccsc3)C2)CC1(F)F CN=c1[nH]cc(C(N2CCC(C)(CC(=O)NCCC3=CCOCC3)C2)=O)o1 c1(OC)c(CCC(n2cc(-c3ccc(C4CC4CO)cc3)nn2)C)cccc1F N1(C(C2C3CCN(C(C(CC)NC(N)=O)=O)CC32)=O)CCC2CN(C)CCC12 CN1CCN(CCC(=O)NC2CC(c3cn(-c4cccc(Cl)c4)nn3)C2)CC1 c1(OC)ccnc(C(=O)NCC(C)NC(=O)C(C)C)c1Br c1(CC)[nH]ccc1C(=O)NCCCCCNC(C1CC12CCC2)=O N1(C(CC(=C)Br)=O)CCC2(CCC2CNC(C2C=CCC2)=O)CC1 N1(C(Cc2c(C)occ2C(F)(F)F)=O)CCC2(CCCN2C(c2cc[nH]c2)=O)C1 N1(C(c2ccc(-n3cncn3)c(F)c2)=O)CCCC12CCOC2 c1(CNC(C(CC(=C)C)C)=O)nnc2n1CCN(C(c1cc(N)ccc1C)=O)C2 c1(C(N2CCC(O)(C(C)NC(c3n[nH]c(C)c3C)=O)C2)=O)ccc(Br)cc1N c1(C(=O)NCC2CCCN(C(C3C(C)CC3)=O)C2)ccc(=O)n2c1CCCC2 c1(C(C)=O)cc(NC2(CNC(=O)C(F)(F)CC(C)C)COC2)ccc1[N+](=O)[O-] Cc1cc(NC(=O)Cn2cc(-c3ccc(C)c(Cl)c3)nn2)cc(Cl)c1F C1(CNC(=O)CC2(CO)CCC2)CN(C(c2cnc(Cl)s2)=O)CCC12CCC2 C1(NC(=NCC(=C)Br)NCC(C)(C)C(=O)OC)C2CCc3ccccc3C12 CC(C)CCCC(C(=O)NCC(C)C)N1CCCC(c2ncccn2)C1 C1(NC(CSCCC(C)C)=O)CCN(c2nc(-c3ccccc3)ns2)CC1C Cc1ccc2c(c1)C(=O)N(C(CC(C)C)C(=O)NCCN(C)C)C2=O Cc1c(C(=O)NCCN(C)C)cnn1CC(C)(C)O.C1(=O)CN1 N1(C(c2c(Cl)cc(C)s2)=O)CCN(C(=O)CCn2nc(C)nc2C)C(C)CC1C c1(CC)ccc(CC(=O)N)cc1.C1CCC1.C(=O)C=CCN(C(=O)CC)C C(C(C)(C(=O)NCCn1cc(-c2nc(C3CC3)cs2)nn1)OC)OC c1(N(C)CC)ccc(C(=O)NC2(C(=O)NCCCSC)CCCC2)cc1.O N1(C(C2(NC(C)=O)CCCC2)=O)CCCC(C)(NC(=O)C(F)C(C)(C)O)C1 c1(C(=O)NC(CCN(C(CCCC(=C)C)=O)C)C)ccc(C)c(Cl)c1F C1(NC(c2nc(CCCC)sc2)=O)CCN(C(c2cc(C)sn2)=O)CCC1(F)F N1(C(COCC(CC)C)=O)CCCC(c2ccoc2)CC1 CN1CC=C(CC(=O)N2CC(NC(c3ccoc3C(F)(F)F)=O)CC(O)C2)CC1 C(CCC(=O)N1CCC1C1CCCOC1)SC.C12(CCCC1)CNC2 C1(C(N2C(CC)CC(O)C2)=O)CN(C(c2ccn(CC)n2)=O)CC(C)O1 C(=O)(CCC=O)N1C(C)(CC(=O)NCC(COC)(C)C)CC1.C1CCC1.N CC1(C(=O)NCCCCCCNC(=O)CCCC(F)(F)F)CCC(F)(F)CC1 c1(C(N2CCCC(CNC(C(CC)OC)=O)C2)=O)ccc(N(C)C)cc1C N1(C(CCC(=O)C2CCNCC2)=O)CCCC2CCNC(=O)C12 C1(CN(C(=O)CCc2nc(O)n[nH]2)C)CCCN1C(C1CC2CC1C2)=O C(=O)(C#CC1CCOCC1)N1CC(OCC)(CNC(C2CCNC2=O)=O)C1 CCCC(O)C(=O)NC1CCCCC1NC(=O)C(C)(C)OC C1(C(C)C)CN(C(c2sccc2CNC(c2ccccn2)=O)=O)CCO1 N1(C(C2N(C(C(n3c(C)ccn3)C)=O)CCC2)=O)CCOC(C)CC1 N1(C(c2nc(CC)oc2)=O)CC2N(C(=O)C#CC3CCOC3)CCC2(C)C1 C1(C)(CC(=O)NC(CNC(C(C=C)O)=O)C(C)C)CCS(=O)(=O)N1 CCC1=C(C(=O)N2CC(C)(NC(=O)Cc3conc3C)C2)CCCO1 N1(C(c2cc(C)nc(C)n2)=O)C2CCC(C(=O)N(CCC3CC3)CCC)C1CC2 c1(CN(CCOC)C)ccc(OC2CCN(C(=O)C(C)C)CC2)nc1 c1(CC(N2CCC(NC(C(C)=C3CC3)=O)C(C)C2)=O)ccc2ccoc2c1 C1(NC(=O)CC2CCCO2)CC12CCN(C(c1ccn3cccc3c1)=O)CC2 c1(CC(N2C(CCNC(CSCC)=O)COCC2)=O)n[nH]c2ccccc12 N1(C(c2c(CC)c[nH]c2)=O)CCCC(CCNC(=O)C(COC)COC)CC1 CC1(C)OCCC1c1noc(Cc2ccc(C(N)=O)cc2)n1 n1(CC)nc(C(N2CCCC2)=O)c(C)n1.c1(C=O)c[nH]nc1C(C)C.C(C)O c1(CC(=O)N(C(C)C)CCN(C)C(C2(C3CC3)CC2)=O)cccc(Cl)c1Cl C1CC2CS(=O)(=O)CC2C1.c1(CN(C(=O)C(=O)NC)C)cnc2[nH]ccc2c1 N1(C(C(CCOC)C)=O)CC(NC(=O)CCCCC2CC2)CC12CCC2 c1(C(=O)Nc2csc(C3CC3)n2)ccc(C2CCOC2)cc1 N1(C(CCC(C)OC)=O)C2CCC1CN(C(=O)COCC1CCCO1)CC2 C(C(CC(=O)N(C1CCCC1)CCC)OC)NC(c1c(CCC)nco1)=O N1(C(c2ccn(C)c2)=O)CCC(C)(CCNC(=O)CCN2CCC2)CC1 C(=O)(CC1OCCc2sccc21)N1CCOCC1.C(=O)(C=CC(=O)N)OCC.C