SMILES N1(C(C(CNC(c2ccc(OC)nc2)=O)OC)=O)CC(=O)N(C)C(=O)C1 CC1CCC(C)(O)CCC1NCc1ccc(Cl)c(C(F)(F)F)c1 C1(n2ccnn2)CCCN(C(=O)C)C1.CC(C(=O)O)NC(=O)OC(C)(C)C C(CCC(C(=O)NC(C)Cc1nccn1C)NC(c1cc(Cl)no1)=O)OC C1(CNC(C(CC)OC)=O)CC2(CO1)CN(C(c1cccc(Br)c1)=O)C2 N1(c2ccnc(SC)n2)Cc2c(F)cccc2C(C)(C)C1 C(=O)(C=C1SCC(=O)N1C)N1CC(C=C)C(NC(C2CCCCS2)=O)C1 C1(O)(CC(=O)NC2CC(F)(CNC(c3ccc(=O)oc3)=O)C2)CCCOC1 c1(C(=O)NCCCNC(CCC#CC)=O)cc(C)c(CC)nc1O N1(C(C=C(CC)C)=O)CCC(NC(=O)CN2CCCS2(=O)=O)C(C)(C)C1 C(=O)(C#CC1CCCOC1)NCCCCCNC(C1(O)CCCN(C(C)=O)C1)=O CC1CCc2onc(C(=O)N(C3CN(C(=O)CCP(C)(C)=O)CC3O)C)c2C1 C(CCCCC(=O)NC(C)CNC(c1cccn1C(C)C)=O)=CC c1(NC(C2C(CNC(C3(OC)CCC3)=O)CC2)=O)cc(CO)cc(C)c1 c1(C(=O)NCC(C)NC(C2(C)CCC23CCC3)=O)cc2c(F)ccc(F)c2[nH]1 c1(OC)cnc(NC(C2CC(NCc3cccc(OC(F)F)c3)C2)=O)c(F)c1 c1(C(N2CCC(C)(CC)C2)C(=O)NCCC)cccc2ccc(Cl)cc12 N1(CC)CCCCC1CNC(=O)CCC1CCCN1C(c1ccc(CO)cc1)=O c1(C(=O)NC2CC3CN(C(C(C(C)(F)F)F)=O)C2C3)cn2c(n1)CCCC2 c1(C(=O)NC(c2ccccc2)C)cccn(C2CCC2)c1=O C12(C(=O)N)CC(C)(CO1)C2.C(=O)(CC(O)c1ccccc1)NCC(C)OC n1(CC=C)cc(C(=O)NC2(C)CN(C(C3CC=CCC3)=O)C2)c2ccccc12 C1(NC(CCC=C(C)C)=O)CC2CCCC(C1)C2NC(=O)CCCC(F)F N1(C(C(C)OCCC=C)=O)CC2CCN(C(C3CCC(N=[N+]=[N-])CC3)=O)C(C2)C1 c1(C(N2CC(C)C2C(N2CC=CC2CF)=O)=O)ccccc1F C1(NC(C2C(CC)CN(C(=O)CC(C)F)C2)=O)Cc2ccccc2C1 c1(CC)sc(C(=O)NC2CCC(F)(C)C2)cc1C.C(=O)CC(CC)C1CCC1.N c1nc2c(s1)CCN(C(C1(CCF)CCOCC1)=O)C2.C(C)(C(=O)N)OCC.C N1(C(C2=C(C)CC2)=O)CCC(C)C(CC(=O)NCCN2CCC(CO)C2)C1 C1(CC=O)CCC1O.C1(CC=O)CC2CC2C1.C(C(C)C)N(CC)CC.N Cc1c(CN2CCC(N3CCCCC3)CC2)cnn1CC(F)F N#CC1(C(=O)NC2C3CN(C(c4ccn5ccnc5c4)=O)CC23)CC2(CCC2)C1 c1(C(=O)NC(CCOC)CNC(=O)CCOC)sc2ccccc2c1CSC c1(SC)nc(Cl)cc(=NC2C(NC(C3CCC4(CCOCC4)O3)=O)C2(C)C)[nH]1 c1(C(N(CC(CN(C(=O)CCCC2CCCC(=O)N2)C)O)C)=O)cncc(Cl)c1 Cc1cc(C(=O)NC2CN(C(C3CCC(C)CC3)=O)CC2(C)C)cn(C)c1=O C1CC(C)N(C(c2cccc(-c3nc(C)cs3)c2)=O)C1.C(C(=O)N)=CCOC C1(C(C)C)(C(N2CC3CC2CO3)=O)CCN(C(=O)Cn2[nH]cnc2=N)C1 N1(C(C(C)NC=O)=O)CCc2[nH]nc(C(=O)Nc3ccccc3C(F)(F)F)c2C1 C1(CN(C(C(c2ccco2)NC(CCCSC)=O)=O)C)CCCN(C)C1 c1(CC(=O)NCCCC)cc(C)ccc1OC.C1(O)(C(=O)N)CC(F)(F)C1 N1(C(CCCc2n(C)cnn2)=O)CCCN(C(c2cccnc2O)=O)CCC1 N1(C(c2cccs2)=O)CCC2C(C1)CN2C(C1(CO)CCOC1)=O C(N=c1nc2ncn(C)c2c[nH]1)C1C(NC(C(C)CSC(F)(F)F)=O)CCC1 C1(CNC(C2COCCN2C(C2CC(CF)C2)=O)=O)CCC(F)(F)C1 N1(C(CCCC(=O)NC)=O)CCOC2(CCN(C(C3C=CCC3)=O)CC2)C1 [SH](=O)(=O)c1ccccc1.C1(O)(CC)CCN(C(c2ccns2)=O)C1.C(=O)(C)N CCCC(C)(O)C(=O)NCc1cc(C(=O)NCc2cc[nH]n2)no1 c1(C(=O)NC2CC(C)(NC(c3ccnn3CCF)=O)C2)cccc(OC(F)F)c1 C1(NC(c2ccc(C)nc2C)=O)C(C)CN(C(C23CCOC(C)(C2)C3)=O)CC1C N1(C(CCN(C)C)=O)CC(C(N)=O)CC(C)(C)C1.C1(C(=O)N)CC(F)C(=O)N1 Cn1ccnc1CCNC(=O)N(CCc1ncco1)CCc1ccccc1 C1(C(=O)NCCNC(C2(C)CC(F)C2)=O)CCc2ccccc2O1 c1(C(N2CCCC2c2cnn(C)c2C)C(=O)N)nc(C)c(C)o1.CCCC.C1CC1 Cc1noc2ncc(C(=O)NC3CCc4nc[nH]c4C3)cc12 C(=O)(CC(C(F)F)c1ccccc1)NCCSC(c1n(C)cnc1)CO Cc1cc([N+](=O)[O-])c(C)cc1C(N1CC2CC2(C)C1)=O.C(=O)CCc1cccs1 C#CCC(CC(F)F)C(=O)N(C(C)C(=O)NC1CC(CSC)C1)CCC C1(O)(C(=O)NC2C(NC(c3nccc(C)n3)=O)CCC2)CC2CCC1C2 c1(CC(=O)NC(CC2CN(C(C(C)OCC#C)=O)C2)C)ccc2ccccc2c1 c1(C(=O)NCC(C2CC2)NC(c2c(CC)non2)=O)cc2ccsc2s1 c1(OC)cc(C(=O)N)cc(C)n1.C1N(C(=O)CC2CC2(Cl)Cl)CCC1(C)C.C c1(C(C(=O)N)N(CCN(C)C=O)C)ncn(C)n1.C1CCOC1.C(C)(C)C C1(CNC(c2ncccc2Br)c2n(C3(C)CC3)nnn2)CCOC2(CCC2)C1 C(C(C)(C)C(=O)N1CCCCC1CNC(=O)Cc1n[nH]c(=N)s1)OC C1(NC(C(C(C)C)C)=O)CCOC12CCN(C(=O)C(C)(C)CCC#N)CC2 CC(=O)CCCC(=O)N1CC(C)CCC1C(N1CCC(C)(N(C)CC)C1)=O Cc1noc(C)c1C(C)NC(=O)NCC1(c2ccn(C)n2)CC1 C1(C(N(C)CCN2CCN(C(=O)C3CC3)CC2)=O)CCOCC12CCCC2 C1(C(C)C)CC(O)CN1C(=O)CC(CNC(=O)C=Cc1cccnc1)C1CCC1 CC1=CCC(C(=O)NC(c2cccc(F)c2)CNC(=O)Cc2cncn2C)CC1 c1(C(=O)NCCCC(C)NC(=O)C#CC2(C)COC2)cncc2c1CCNC2=O C(=O)(C(CC(C)C)NCc1cnn(C2CCC2)c1)OC c1(CC)nc(N2CC(NC(=O)CSCc3cccs3)CCC2C)c2ccsc2n1 CCCCCC(CC)C(=O)N1CCN(C(c2ccnn2CC2CC2)=O)C(CF)C1 C(=O)(CCCC(C)(C)C)N1CC(C(N(C(C)C(C)(C)O)C)=O)C(F)C1 CCCC(O)C(=O)N1CCN(CCNC(=O)C(c2ccc(F)cc2)(F)F)CC1 C(CC(C)C)(C(=O)O)NC(C1N(Cc2cnc(CCCC)[nH]2)C2C(C1)C2)=O N1(C(C2(C)C=CCN2C(C2C3CCC(F)C23)=O)=O)C2CCC1CC1(C2)N=N1 c1(CC(N2CCN(C(CCC(=C)Cl)=O)CC2C(C)C)=O)cccc([N+](=O)[O-])c1 Cc1ccn2cc(C(=O)NCC(C)CN(C)C(C3(CO)CC3(F)F)=O)nc2c1C n1(CC)ncc(Cl)c1C(=O)NC(C)(C)CCNC(C1CCOC1)=O c1(OCC)ccc(OCCC(=O)NCC2CCCN(C(=O)CC(O)CC)C2)cc1 C1(CNC(C(C(C)C)C)=O)CN(C(c2nocc2C2CC2)=O)CC12CC2 C(CCCCC)NC(CN(C1CC1)CC)=O.C1(C(=O)N)(C(F)F)CC(O)C1 C#CCC(C(=O)NC1CCCN(C(c2cnn(C)c2CC(C)C)=O)C1)C1CC1 CC1(C)CC(C(=O)Nc2ccc[n+]([O-])c2)N(C(=O)CC2CCC(=O)C2)C1 N1(C(COCCCC)=O)CCC(C)(C)CC1C(N1CC2CSCC2(C)C1)=O C12(CNC(=O)CCCCCF)CCC(CC1)N(C(C1(N3CCCC3)CC1)=O)C2 C1(C(CNC(c2c(CC)nns2)=O)=O)COCCN1C.C1CCC1.C(C)(C)C N1(C(CCC=CC)=O)CCN(C(c2nc(C)oc2OC)=O)CC(C)(F)C1 Cc1c(C(N2CCCC(F)(CNC(c3cnn(C)c3)=O)C2)=O)nn2c1CCCC2 C=CC(C)(CC)C(=O)NCCCCCNC(=O)Cc1ccsc1C CCCCS(=O)(=O)CC(=O)NC(CO)C(C)NC(=O)CCC(=O)N(C)C c1(C(=O)NC2CCCN(C(C3C(C(C)C)CCO3)=O)CC2)ccc(F)c(O)c1F c1(C(N(CCC(C)NC(C2CCOC2)=O)C)=O)c(Br)ccc2n[nH]cc12 C(=O)(C(C)(F)C(=O)N1CCCC(CC(=O)Nc2csnc2C)C1)OC C(=O)(C1=CCSC1)N(C(C)C(=O)NCC(c1ccccn1)O)CC C(C(C)(C)CC(=O)NCCC1CCCN1C(c1cccc(C2CC2)n1)=O)N(C)C C(C(C)NC(=O)C(C)(C)c1ccns1)(C(C)C)NC(CCc1cnc(C)s1)=O c1(OCC)ncc(C(C)NC(C2CCOC2)C)s1 CCC(C)(C)C(C)CC(=O)NCC1CCN(C(c2nccc3cccnc23)=O)C1 C(=O)(NNc1cc(Cl)ccn1)NC1CCC(C)NC1 c1(CC(N2CCCCC2)=O)ccc(C(F)(F)F)c(F)c1.C(C)(C)(C(=O)N)OC C1(C(=O)NC(CC)CN2CCCC2)CCN(C(=O)c2nccs2)O1 N1(C(=O)CCCc2cnn[nH]2)CC2COCCC2(NC(C23CCC2C3)=O)C1 N1(C(c2cnn(CC)c2Cl)=O)CCC(NC(=O)Cc2cc(C)cs2)C12CC2 N1(C(C2N(C(c3ccnc(C)c3N)=O)CC(=O)NC2)=O)CCC2(CC(F)C2)C1 Cc1cc(Br)cc(Cl)c1C(=O)NCC12CC1CN(C(=O)CC1CC1(C)C)C2 N1(C(C2CC(=O)N2)=O)CCCC2CN(C(c3c(Cl)n[nH]c3C3CC3)=O)CC12 C1(CC)CN(C(c2ccc(Cl)nc2OC)=O)CCN1C(=O)CCc1ccc(C)s1 Cc1c(C(=O)NC(C2CCCC2)CNC(C2CCC2OC(F)F)=O)cccc1Cl c1(C(=O)NCC(C)(CO)NC(CC2CC(C)(C)OC2)=O)cc2c(Cl)cncc2s1 C(C(C)(O)CC(=O)NCC1(CC)CC1)OC.c1(C(=O)N)cc(C)n(C)c1 C1(NC(CC(CC(C)C)O)=O)C2CC3CC(C2)CC1(CNC(c1cscn1)=O)C3 O=C1c2ccccc2C(=O)N1CC(O)CNC(c1ncc(Br)c(O)n1)=O C(=O)(C1CCc2nccn21)NCC1C(NC(C(COC)(C)C)=O)CCCC1 c1(C=O)cc(S(N)(=O)=O)n(C)c1.C1(OC)CN(C(c2cc(C)on2)=O)CC1 C1(NC(N2CC(=O)NCC2)=O)CC2CCC1(CO)C2.c12cncc(n1)N2 N1(C(C(C)N(C)C)=O)CC2CCN(C(=O)C(C)(C)NC(N)=O)CC2C1 CCCC(CC)CC(=O)N1CCN(C(c2cccc(C(F)(F)F)c2O)=O)C(C)C1 c1(NC(N2CC2)=S)c(C)cnn1CC1CCCCC1.c1ccc(C)cc1.CCN c1(CN(C)CCOc2ccccc2C(=O)O)ccc2c(c1)NC(=O)C(C)O2 CC1CCN(C(=O)CCCC2CCC2)CC1NC(=O)CC1(O)CCN(C)CC1 C1(CC(=O)NCC2CCC(CC)O2)CN(C(c2cccn(C)c2=O)=O)CCC1C c1(C(N2CC3C(CN(C)C(c4nnc(S)n4C)=O)C3C2)=O)ccc(F)c(O)c1 Cc1cc(C(=O)NCCNC(=O)Cn2cnccc2=O)c2cnn(C)c2n1 c1(NC)ccc(C(=O)NC(Cc2ccoc2)C(=O)N2CCC(OC)C2)[nH]1 N1(C(CC(CN(C)C)O)=O)CCC(C)CC1CNC(=O)CN1CCOC1=O CCCC(C)(O)C(=O)NCC(C)C.c12c(cccc1C)SC1CCN(CC1)C2=O C1(C(=O)N)CCCC2CC12.c1(CC)conc1C(=O)NCC(C)(C)OCC C1(NC(c2n(CCC)ccc2)=O)CN(C(c2cncc(NCC)c2)=O)C2CC12 C1(CC(=O)OC)CCCCC1NCC1(O)CCCCC1 C(=O)(C(O)CCCNC(=O)CCC(C)CN(C)C)N(CCn1ncc(C)c1)C c1(OC)cccc(SCC(=O)NCC2CCCCC2)c1.C1(F)(C(=O)N)CC1 c1(C(N(CCN(C(C(CC)N(C)C)=O)C)C)=O)ccc(F)nc1F N1(C(c2ccc(CC)[nH]2)=O)CCC(NC(c2cnc(C(F)F)s2)=O)C1C C=CCC(CC=C)C(=O)N1CCCCC(NC(c2ncccc2N(C)C)=O)CC1 CCC(COC)(CC)C(=O)N1CCC(CN(C(=O)CCC(C)OC)C)CC1 C(=O)C(CCC)S(N)(=O)=O.c1(COC)cc(C(=O)NC2(C)CCC2)no1 C1CCC(C)N(C(=O)CC)C1.c1(OC)nc(Cl)c(C(=O)N)s1.C(=O)C=CCl.C N1(C(C(C2CC2)NC(c2cc(C(N)=O)oc2)=O)=O)CC2(CCC2)C1 C(C1CN(C(C2(C)CCC2)=O)Cc2ccccc21)NC(C1N(C)CCCC1)=O CC1=C(C(=O)N2CCC2CNC(c2ccnc(C3CC3)n2)=O)CCC(C)(C)C1 C(=O)(C(CC(C)C)C(N)=O)N.C1(C(=O)NCCOCC=C)CCOC1C N1(C(C(C)(C)c2ccsc2)=O)CCC(F)(CNC(C2CSCC(=O)N2)=O)C1 N1(C(C(COCC)C)=O)C(C(=O)NC2CN(CC)C2)CCC12CC2 C1(C)(C(N2CC=C(CNC(c3cc(OC)ncc3)=O)CC2)=O)CCCCCCC1 C(CN=c1[nH]c(=NC(CCO)c2cccs2)c2c(ncn2C)[nH]1)N(C(CC)C)C c1(NC(c2cc(Br)cc3cn[nH]c23)=O)cccc2c1C1CCC2O1 C1CCCC2(CN(C(=O)C3=CCCO3)C2)O1.C1(C(=O)N)CCC2C(C1)C2(F)F.C CC(C)CC(CNC(C1CC2CCC1CC2)=O)C(=O)NCCCC1(O)CC1 c1(NC(c2ccc(-c3nnn(C)n3)cc2)=O)cc(=O)nc(-c2ccc(Cl)cc2)[nH]1 C1(C)(C(N2C(CCC)COCC2)=O)CN(C(=O)CCc2cnoc2)CC1C C1(=CC(=O)NC2CCCC(NC(CC3CC(C)C3)=O)C2)CN2CCC1CC2 C1(c2cc(COC)on2)CCN(C(=O)C=CC(=O)OC(C)=O)CC1 c1(OC)cc(C(=O)N(C)CCNC(=O)C(C)CS(C)=O)c(N)c(Br)c1 c1(C(N2CCN(C)CC2)=O)cc(F)cc2nn[nH]c12.C(C)(C(=O)N)OCC=C.C C(=O)(C(CCC1CC1)NC(C1CC1(F)Cl)=O)NCCC(C)(C)C c1(CC)cc(C(=O)NCCCC(C)NC(C2C(C)C2(F)F)=O)oc1CC N1(C(C2CC3(CC3)CN2c2ncc3ccsc3n2)=O)Cc2cncnc2C1 N1(C(c2cccc(=O)o2)=O)CCC2(C1)CN(C(C1CN(C(N)=O)C1)=O)C2.CC C#CC1CC2CCC1N(C(C1CC(C)(C)CCN1C(=O)C(CC=C)CC=C)=O)C2 CC1CC2CN(C(=O)C(C)(F)F)CC2N1C(=O)CNC(c1ccco1)=O N1(C(=O)C#CC2CCOC2)CCC2CCCC(C1)N2C(c1ncc(F)cc1F)=O C1CCC(F)C1.c1(CC=O)cc[nH]n1.C1(C(=O)N)(COCC)CC1.C Cc1ccc(-c2ccc(NS(=O)(=O)CC3CCOCC3)cc2)cc1 N1(C(C2(C)COCCO2)=O)CCCCC(NC(=O)CS(C)(=O)=O)C1 c1(N2CCC(C#N)C2)nc(N2CC3CCC2C3)nc2ccc(Cl)cc12 C1(C(=O)NC2(CF)COC2)Cc2ccc(Br)cc2NC1=O C(=O)(C#CC1(C)CC1)N(CCCN(C)C(c1cccc(SC(F)(F)F)c1)=O)C c1(OCC)ccc(CNC(=O)C)cc1.C1CCN1C(C)=O.CC(C)C.C c1(NC(C23CC2CN(Cc2cc(Cl)ccc2F)C3)=O)nc(Cl)ccc1F N(C1CCCc2c[nH]nc21)C(N1CCC(O)(C2(C(=O)O)CC2)CC1)=O CN1CCC(CC(=O)NC(Cc2ccco2)C(=O)NCC2CCCO2)CC1 c1(C(N(CCCNC(CCC)=O)Cc2ccccc2)=O)cc2c(Cl)ccnc2s1 c1(C(=O)NC(CNC(c2n[nH]c(CC)c2Cl)=O)CO)cc(C)c(Cl)c(N)c1 N1(C(C2N(CCC)C(=O)CC2)=O)C2CCC1CC2.C1(C=O)(C(N)=O)CCC1.C C1(CNC(C(CC)=CCCC)=O)CC(C)N(C(c2n[nH]c(COC)n2)=O)C1 c1(C(=O)NC(C(C)NC(=O)CC2CCCCCC2)CO)ccnc(F)c1N C#CC1(COC)CCN(C(=O)C(C)Cc2cccc(C(F)(F)F)c2)C1 N1(C(C(C)O)=O)CCCC(C2CC2NC(=O)CCc2cncs2)C1 C12(CN(C(c3cccc(F)c3)CO)C)CC(C1)NC(=O)O2 N1(C(C(C2CCCC2)OCC)=O)CC(C)(C)CC1C.c1(C(=O)N)cnnn1C C(CCC(=O)NC(C1CCN(C(c2nonc2N)=O)C1)(C)C)N(C)C c1(C(C)C)cc(C(=O)N(C2(CC(=O)NCC3CC3C3CC3)CC2)C)on1 C1(CNC(Cc2c(C)noc2C)=O)CCC2(CN(C(c3csnn3)C)C2)O1 C1(COC(=O)CCCCc2cccc(O)c2)CC2(CCCC2)CO1 N1(Cc2c(C)ccc(OC)n2)CC2(C1)SCCC2C(=O)O c1(C(=O)NC2CCC(C)N(C(c3coc(Cl)c3)=O)C2)cc2ccccc2o1 Cc1ccccc1C(C)CC(=O)N(C)C.C1C2CN(C(C3(C(F)F)CC3)=O)CC12 C1(C(N2C3CN(Cc4cc[nH]c4)CC23)=O)CNCC(F)(F)C1 CC(C)CC(C)CC(=O)N1CCC(CO)(CNC(c2cc(F)c(F)cc2N)=O)C1 Cc1cn2c(n1)CCC(C(=O)NCCCCNC(=O)CCc1cc(C)n(C)n1)C2 c1(OC)cccc(SCC(N2CCC(N(C(C3CCC(=O)N3C)=O)C)C2)=O)c1 CCCCCC=CCC(=O)N1CC(CC(F)C(=O)NC(C)CSC)C1 CC1CN(C(c2cnccc2N(C)C)=O)CCN1C(C1CNC(=O)C1)=O C12(C(N3CCC3)=O)CC3CC(C1)C(=O)C(C3)C2.[nH]1cc(C=O)cn1.CCS C#Cc1cn(C)nc1C(=O)NC1(COC)CCC1.C1(C(=O)N)CCC(F)C1 N1(C(CC(C)(C)NC(C2C(CC)CCCC2)=O)=O)CCCC2(CC(O)C2)C1 N1(C(C2N(C(CC)=O)CSC2)=O)CC2CC(NC(=O)C)C2C1.c1cnn(C)c1.S N1(C(C(C)CO)=O)CC(CO)C2(C1)CN(C(c1cccc3c1C(=O)CC3)=O)C2 C1(C(=O)NCCCN(C)CC2CCOC(C)C2)CC2CCC1CC2 CSC1=C(C(=O)NC(CN(C)C(c2nnc(Cl)cc2N)=O)(CO)CO)CCCC1 c1(N(C(CC)C(N)=O)C(=O)OC(C)(C)CC(=O)N2CCCC2)cncc(C)c1 N1(C(CC(c2ccc(C)cc2)C)=O)CC2CC(C1)CN(C(=O)Cc1ccno1)C2 C=CCC(CC=C)C(=O)NC1CN(C(=O)C2=CCCSC2)CC1CC(C)(C)C N1(C(C(C)NC(C)=O)=O)CCCN(C(=O)Cn2ccc(Br)n2)C(C)C1 C=CC(C)CC(=O)N1CCCC1c1nnc(C(=O)NCC2CCN(CC)CC2)s1 C=CC(C)(CC)C(=O)NC(=O)C(C1(O)CCCCC1)(F)F.C(C)(C)C.C=O.N c1(C(N2CCC(N(C)C(C3CCC(C)(C)CC3)=O)C2)=O)cc2c(=O)[nH]ccn2n1 C1(C(N2CCC=C(CNC(c3nc(C)nn3C)=O)C2)=O)CCC2CC1C2(C)C C1(N(C(=O)CSC)C)CCN(C(C2CCOC2)=O)CC12CC2.c1ccc(O)cc1 CC1CCC(CC(N2CCC(N(CCO)C(c3ncccc3Cl)=O)C2)=O)CC1 C#Cc1ccc(C(=O)NC(CC=C)C(=O)NC2COC(C(F)F)C2)cc1C c1(C(=O)NCC2C(NC(CC3CCC(C)(O)CC3)=O)CC2)cnn2c1OCCC2 C#CC1CN(C(C2CC(=C)CCN2C(=O)C(F)C(F)(F)F)=O)CCN1C c1(C(N2CCC(CCNC(C3CCOC3)=O)CC2)=O)cc(=O)cc(Cl)[nH]1 C1(CC(=O)N)CCCCC1(F)F.c1(CCCC)nc(C(=O)NCC2CC2)cs1 N1(C(c2c(OCC)cnnc2)=O)CCC(NC(c2ccc([N+](=O)[O-])s2)=O)CC1C N1(C(C(C)OCCOC)=O)CCCC12CCC2.C1(CC=O)CC2(CCC2)C1.C C1(C(=O)NCC2N(C(c3scc(C)c3)=O)CC2)CCC(F)(CO)C1 Cn1cc(C(=O)NCC2C=CCN2C(C2CC(F)C2)=O)c(C2CCC2)n1.C c1(NC)ccc(Cl)cc1C(=O)NCCCNC(=O)C(C)P(C)(C)=O c1(OC)ccsc1C(=O)NCc1cc(C(=O)NC2CCC2)cs1.C1CC1 c1ncc(C=O)cn1.c1(C(N(CC(C)C)C)=O)sc(N(C)C)nc1C.CCO N(C(=NCCCCl)NCc1nc2c(s1)CCCC2)Cc1ccc(OCC#C)cc1 n1(CC)cnc2c(N3CCC(CCF)CC3)nc(=NCCC3CCCC3O)[nH]c12 Cn1nc(C(N2CC(NC(=O)CC3CCOC(C(C)C)C3)C2)=O)cc1Cl c1(C(N2CC(NC(C3C(c4cn(C(C)C)nc4)C3)=O)C2)=O)nn(C)nc1Br Cc1nc(Br)sc1C(c1nnnn1C1COC1)NCCCS(C)=O C1(OC)CCCCC1C(=O)NC1(C)CC(NC(=O)C(=O)N(C)C)C1 C1(C(=O)N)CCC12CCC2.C(=O)(C(C)(C)C)OC.c1(CC=O)coc(C)n1 CCCCC(C(=O)Nc1ccc(F)nc1C)NC(=O)C(O)C1CCC1 C(=O)(C1=CCCC1(C)C)NCCCCC(C)NC(c1cnn2c1NCCC2)=O C(C1=NOC2CCCC12)NC(C(C)(CSC)NC(CCCOC)=O)=O c1(C(c2nnnn2C)NC(C=C)(C)C)cc(C(C2CC2)C)[nH]n1.c1ccccc1 C(=O)(C1=C(C)OCCC1)N.C(=O)(C(O)CC)NC(C(=O)OC)C1(C)CC1 C1(C(=O)NC(C(C(=O)NCC(C(=O)OC)(C)O)C)C)OCCCC1(C)C C=CC1CN(C(=O)C=CC(C)(C)SC)CC1NC(=O)C(C)(C)C1CC1 c1c(Cl)c(C(=O)O)nc(Cl)c1Cl.C1(c2cn(CC(=O)N)nn2)CCS(=O)(=O)C1 C=CCC(C(=O)N1CCCC1C1(O)CN(C(=O)C(O)C(C)C)C1)NC(C)=O CCCCC(C(=O)N1C2CC1CN(C(C1(C)CC3CC3C1)=O)C2)NC(N)=O c1(-c2c(C)nn(C)c2)ccc2cc(C(=O)Nc3ccccc3N(C)C)[nH]c2c1 C1(NC(C2CCC(C)(C)CO2)=O)CCCC2CN(C(C3(C)COC3)=O)CC12 Cc1c(F)cc(-c2nc(C(=O)NCCc3cccc(Cl)c3)cs2)cc1F C1(N(C)C(c2csc(C3CC3)n2)=O)C2CN(C(=O)CS)CC12.c1ccccn1 C1(NC(C2(C)CCN(C)C2=O)=O)CC2CCC(C1)N2C(c1nc(=O)n(C)[nH]1)=O C#CCCCCCCNC(C1CN(C(C2(CO)CCCO2)=O)CC1OC)=O C1(NC(COCCOC)=O)CCC2CC1CN2C(=O)CCC(C)c1ccccc1 N1(C(CC(C)C)=O)CCC(N=[N+]=[N-])(C(N2CC(N(C)C)C(C)(C)C2)=O)C1.CC C1(C)(NC(Cc2n(C(C)C)cnn2)=O)CCCN(C(c2ccc(O)nc2Cl)=O)C1 C1(CC(=O)NC(C2(O)CN(C(=O)CCCCC(F)F)C2)C)Cc2ccccc2O1 c1(CN2CCC(CCCC)C2)ccc(-n2cc(CN(C3CCC3)C)cn2)cc1 c1(CC)ccc2nc(-c3nc(-c4ccnc(SC)c4)no3)sc2c1 n1(CCC#C)c(N(C)Cc2cccc(Br)c2)nnc1C1CCCN(C)C1 CCC(C)(C#N)C(=O)NCCCOCCN(C)C(C1CCSC1)=O C1(C(=O)NC(c2ccc(Br)s2)C(=O)O)CCCC(C(F)F)CC1 CCC(CCC(=O)NC1(C2CCCN2C(c2ccc(NC)cc2C)=O)CC1)OC CC(CC(C)NC(=O)CC1(O)CCCCC1)C(F)F.C1(C=O)CCCCC(=O)N1.N c1(C(C)=O)ncccc1C(=O)NCC(O)CCNC(C1CCC1(F)F)=O C1(C)(CC)CC(NC(=O)Cc2ccc(CO)cc2)CN1C(=O)CSC(F)F C1CC(C)N(C(=O)Cc2nn(C)cc2Cl)C1.C(=O)(CC(=O)NC)NCC#C c1(SC)cc(C)ccc1NC(c1nc(-c2ccc(Cl)cc2)no1)=O C1CCN(C(=O)CC)C(C)C1.c1ccccn1.C1(C)(C(=O)OC)CC1C(=O)N C12(CNC(COCCCCCC)=O)CCC(CC1)N(C(C1(C)CCC1)=O)C2 C(=O)(C(O)CCC(F)(F)F)N(CC)CC1CCN(C(c2nccn2C)=O)CC1 C1(C(=O)NCc2ccccc2)(OC)CCCOC1.C(=O)CN(C)C(C)=O.C C1(NC(=O)CC2NC(=O)NC2=O)CN(C(c2cc(Br)ccc2O)=O)CCC1F c1(C2(NC(=O)CC3COCCN3C(=O)C(F)(F)F)CC2)ncc(F)cc1F C1(C(N2CCC(O)(C)C2)=O)(OC)CCC(C)(C)CC1.C(=O)CCC=C(C)C c1(C(=O)NC2CN(C(c3c(C)ncnc3)=O)CC2C)cc2occc2s1 C1(CC=C)(NC(=O)CN(C)C(N)=O)CCCN(C(C2CC(CC)=NO2)=O)C1 N1(C(c2nc(C)oc2)=O)CC2(C(=O)NCC(c3ccccc3)O)CC1CCO2 CC(C(C)(C)C(=O)NCc1ccc(C#N)cc1)NC(=O)C=CCF C1(NC(C(C2(O)CN(C(c3c(C)cco3)=O)C2)F)=O)CN2CCC1CC2 c1(CNC(CSC)=O)ccc(CCNC(C2CC23CC3)=O)cc1 C=C(C)C(C)(C)C(=O)NC(CNC(=O)Cn1ccc(C=O)n1)C1CC1 c1(C(=O)NC2CN(C(c3n(CC)ccn3)=O)CC2C)ccc2cc[nH]c2c1 Cc1cc(C(C)C)nc(C2CN(CC3(C(=O)Sc4ccccc4)COC3)C2)n1 c1(CNC(C23CC2CN(S(=O)(=O)CC2CCC2)C3)=O)ccc(F)cc1 C(c1cnccc1C)=CC(=O)N(CCCNC(C(C(=O)OC)OC)=O)CCO N1(C(C=CC(C)C)=O)CC2=C(C1)CN(C(C1(C#N)CCC1)=O)C2 CCCCCCCC(=O)NCCCN(C(c1cnc(OC)cn1)=O)C1CC1 C1(CS(=O)(=O)NC)CC2(CCN(C(c3ccccn3)COC)CC2)CN1 C1(C2CC2)(CNC(C(C)=Cn2ccnn2)=O)CCN(C(=O)CCCCC(C)C)C1 C(CC(C)C)(C(=O)N1CCC(N=[N+]=[N-])C1)NC(CC1(NC(C)=O)CC1)=O Cc1cnc(Cl)nc1NCC1(CCNC(=O)Cc2cscn2)CC1 c1(OC)c(C2CCCN2CCc2cccc(Br)c2)cnn1C CC1=C(C(=O)N2CCCCC2CCNC(=O)Cc2[nH]cnc2C)CCC(C)(C)C1 C1(C(N2C(C#C)CCC2)=O)CCOCCN1C(=O)C(C)C(=O)OC Cc1sc(C(N2CC(NC(=O)Cc3cccc(F)c3)C(C)C2)=O)nc1O CCC(CC(=O)NCc1ccc(C(=O)NCC2CCC(=O)O2)o1)CC(C)C CC(C)C(CCNC(=O)CC1CCCCN1C(C)C)NC(=O)C1CC1 C1(CNC(c2ccccc2Br)=O)CCCC2CN(C(=O)C(F)Cl)CC12 N1(C(CCNC(C)=O)=O)CCCC(C)(C)C1CNC(C1CCCC(=O)O1)=O c1(NC(C2CCCN(Cc3cc(C)cc(Br)c3)C2)=O)c(Br)cc(Cl)cc1[N+](=O)[O-] c1(NC(=O)Nc2c(OC)ncnc2OC)ccc2c(c1)C(=O)N(C)C2 N1(C(=O)OC(C)(C)C)CCN(C(=O)CCCc2nn[nH]n2)C(CC2CC2)C1 c1(C(=O)NC2(C)CC(NC(c3c(C)cc(O)cc3)=O)C2)cnc2occc2c1 C(CNC(=O)Cc1sccc1C)(CC(F)(F)F)NC(CCc1cnc(C)o1)=O c1(C(C(C)C)C(=O)NCC2CC(NC(C3CC3)=O)C2)cccc(C#N)c1.C C1(NC(CC(C)c2cnn(C)c2)=O)CN(C(C2(Br)CC2)=O)CC1O C1(C=O)CS(=O)(=O)CC(=O)N1.N1(C(C2(OC)CCC2)=O)CCCN(CC)CC1 c1(C(N2CCCC(O)(CNC(C3CCN(C)CC3)=O)C2)=O)ccc(C#N)cc1Cl C1(F)(C(=O)NC(C)CC2CCOCC2)CCN(C(C2(C)CC(O)CN2C)=O)CC1 CC1(CC(N2CCC(Cc3ccccc3)C2)=O)CCN1Cc1ccc(CO)o1 C1(C(=O)NCCC(C(C)C)NC(c2c[nH]nc2C2CC2)=O)CCC(C)(C)OC1 c1(C(CC(=O)NCCC(C)N(C(CCOCC)=O)C)C)ccccc1F CC1CCCCC1C(=O)NCCNC(c1cnc(O)o1)=O.c1ccc(Cl)nc1.C CC(CC(=O)N1CCC(C)(C)CC1)CC(F)(F)F.C1(CC=O)CS(=O)(=O)C1.N C(c1ccc(-n2ccnc2)cc1)=CC(=O)NCC.C1(C=O)CS(=O)(=O)C1 C1(N(C(=O)CSS(C)(=O)=O)CCC)CCN(C(c2nccnc2N)=O)CC1 N1(C(c2c(CNC(C3(C(CC)=O)CC3)=O)noc2)=O)CCCC(N(C)C)CC1 c1(CNC(c2c(OC)csc2)=O)ccc2c(c1)CN(C(=O)C=CSC)C2 CC1(C)CN(C(C2CCC(C(F)F)CC2)=O)CC(C)O1.c1(CC(=O)N)cc[nH]c1 Cc1[nH]nc2ncc(C(N3CCCC3CCCNC(=O)CC3(O)CC3)=O)cc12 C(=O)(C(CC(F)F)C1CCC1)NCCN(C(=O)C(CC)C=O)CCOC.O C(CN=c1ccc(Br)c(S(=O)(=O)N2CCCC(F)C2)[nH]1)(c1ccccc1)N(C)C c1(CC)noc(C(=O)NC(C2CN(C(=O)C(C)C)C2)C)c1C N1(C(C(=O)NCCCC(=O)OCC)C2(CC)CC2)CC(OC)C(F)C1 C1(CC)CN(C(c2cc(C)nnc2O)=O)CCC1NC(=O)CCNC(C)=O C1(C(=O)NCCC2N(C(CN3C(=O)CSC3)=O)CCCC2)CC12CCSCC2 N1(C(c2n(CC)ccc2)=O)Cc2[nH]nc(C(=O)NOCC(O)CO)c2C1 Cc1cc(C(N2CCC(NC(=O)CCCCC#N)C(C(C)C)C2)=O)cc(=O)n1C CCC(C)C(=O)C(=O)NC1CCC1c1cn(-c2ccc(F)cc2F)nn1 c1(OC)cccc2c1OCCC2NC(c1cc(C)c(Br)s1)c1nnnn1C(C)C c1(C(N2CC3C(NC(c4c(C)scc4)=O)C3C2)=O)ccc(C#N)c(Cl)c1 n1(CCC)ccc(C(=O)N(C(C)CNC(=O)CC(=O)N(C)C)C)n1 C1(NC(c2ccc(C)cc2O)=O)CCCCCN(C(c2coc(O)n2)=O)C1 C1(CC(=O)NC(c2ncc(C)o2)C)(OC)CN(C(=O)CCc2ncc(C)[nH]2)C1 C1(c2ncnn2C)(NC)CN(C(C2(C)CC2)=O)C1 c1(C=O)c(F)c(F)c(F)c(F)c1F.C=CCC(CC=C)C(=O)NCC1CCC1.N C1(NC(c2c(C)nc(O)[nH]2)=O)CCCC2CN(C(c3cnn(C)c3)=O)CC12 C(C)(N=c1[nH]c(N2CCC(C)=C(C)C2)nc2c1CSC2)c1c(OC)cccc1F CC(C)(C)CCCC(=O)NCC(=O)NC12CC(C)(C1)OC2C(=O)O C(=O)(C(CCC(C)C)NC(=O)CC1CC2(CC2)CO1)NCc1c(C)scc1 N1(C(Cc2cn(C)nc2)=O)CC2CCCC2(CNC(c2ncc[nH]c2=O)=O)C1 C=CC1CN(C(C2CCN(C(=O)C(C)c3cccs3)C(CC)C2)=O)CC1O Cc1cc(C(=O)NCC2CCN(C(=O)Cn3nnc(=O)[nH]3)C2)cc(O)n1 Cc1cc(NC2CCCCC2NC(C2(N(C)C)CCCC2)=O)ncc1[N+](=O)[O-] N1(C(c2nccc(C)n2)=O)CCC(NC(=O)Cc2ccc(C)nc2Cl)CC(C)(C)C1 N1(C(C)C)CCCC(CC(N2CC(N(C)C(c3nncs3)=O)C2)=O)C1 c1(N2CCC(OCC)C(C)C2)nc(=NCc2cc(Br)cs2)[nH]c2ncn(C)c12 c1(OC)ccc(C(N2CCCC(NC(=O)C(c3ncccc3C)(F)F)C2)=O)nc1 CCCC(C)(O)C(=O)NC1CCCCC1NC(c1cc(F)c[nH]1)=O c1(CN2C(COC)CN(C(C3CC=CCC3)=O)CC2)ccc(Br)cc1C#N Cc1oc(C2CCOCC2)nc1C(=O)NC1CC1C.n1(CC=O)nnnc1C.N C12(NC(c3cc4ccccn4c3)=O)CCN(C(c3ccc(F)cc3)=O)CCC1C2 Cc1nc(CC(=O)NC2CCCC2C(=O)NC(c2cnc[nH]2)C)n[nH]1 CCC(CC(=O)N1CCCC1C(C)NC(c1cc(C)no1)=O)C1CCC1 C(=O)(CCC(=O)NC(C)CN(C)C(C1CC2CC2C1)=O)NC C=Cc1cc(C(N2CCN(C(c3nccc(OC)n3)=O)C(CC)C2)=O)cc(F)c1 Cc1cc(Cl)ccc1CC(=O)NCC1CCC1.C1(CC(=O)N)OCCOC1(C)C N1(C(=O)Nc2sc(C)c(-c3cc(O)nc(=N)[nH]3)n2)CCc2cncc(Br)c21 N1(C(C2(NC(=O)CCC3CCCO3)C(C)C2)=O)CCC(C)(OCCO)CC1 C(C(CC(C)C)NC(CCC(C)(C)F)=O)NC(COCC=C)=O c1(OC)c(C(=O)NC(C)C2=CCN(C)CC2)cc(C)cc1C c1(OC)cc(CCCNC(N2CCOCC23CC3)=O)cc(OC)c1O C1(C)(C(N2CCC(CC(C)NC=O)CC2)=O)CCC(F)(F)CC1.C(C)(C)C.O C1(CNC(C2C(CC)C2)=O)CCCN(C(c2ccn(C)n2)=O)CC1 N1(C(=O)N=c2[nH]nc(-c3ccc([N+](=O)[O-])cc3)s2)CCc2cccc(Br)c2C1 N1(C(CSCc2nc(C)sc2)=O)CCC2(CC1)CC(N1CCCC1C#N)CCO2 N1(C(c2cc(OC)ns2)=O)CCC2OCCN(C(c3ccc(O)nc3C)=O)C2C1 C1(CNC(CC(=O)NCC#C)=O)CC(C)N(C(=O)CC2(C#N)CC2)C1 C(=O)(CC(C)(C)C(F)F)NCC(C1(O)CCN(C(C2CC3(CSC3)C2)=O)C1)C c1(N(C)CC2CC2(F)F)nc(N2CCC(C(F)F)(CO)C2)c2c(n1)COC2 C=CC(CC)C(=O)N(C)CC1CCCC1NC(=O)C(C)O N1(C(COCCC)=O)CC2CC1CCC2NC(=O)Cc1cnoc1 C1(Cn2ccnn2)CCC(c2ccccc2)=NO1.CC(=O)CCCCC(=O)NC CC(F)CC(=O)N(CCC(=O)NC(C(CO)C1CC1)C1CC1)C1CC1 C(=O)(C(F)(F)C(O)C(C)C)NCC1CC(CNC(CC(CC)C)=O)C1 C1(OC)CN(C(=O)CCCC2CC2)CC1NC(=O)CC1(CO)CCCCC1 c1(C(N2C(C)C(NC(C3CCCN3C=O)=O)CC2)=O)cccc2nncn12 N1(C(CN(C)C(C2(C#N)CCOC2)=O)=O)CC(S(N)(=O)=O)C1 C1(CNC(c2ccc(CC)cc2F)=O)CN(C(c2cccnc2S)=O)CCC1C CC1(C)CN(C(=O)C#CC2CC2)CC1CNC(C1CC(=O)C12CCC2)=O CCC(C)(CCNC(c1cc(=O)cc[nH]1)=O)NC(=O)Cn1cnnn1 N1(C(c2c(NC)nccc2)=O)C2CCC(C2)C1CNC(=O)CC(C)(C)C.S C1(C(N(C)CCNC(C2(O)CCOC2)=O)=O)CCC2(CCC2)CO1 C1(NC(C=CC)=O)CN(C(C2(CC3CC3)CCCO2)=O)CC(C)(C)C1 C1(C(=O)NCc2cccc(NC(C(COC)OC)=O)c2)CCS(=O)(=O)N1C Cc1cc(CNCC2COc3cscc3O2)nc(Cl)c1Br C(CC1CCC1)(C(=O)N(CC(C)N(C(=O)C(C)C1CC1)C)C)OC C(=O)(CCCC(F)(F)F)NC1C2OCC(NC(Cc3ncc(C)s3)=O)(C2)C1 C1(CNC(C(C=C)OC)=O)CC2(CO1)CN(C(c1c(C)csc1C)=O)C2 c1(OCCOC)ccc(Cl)nc1C(=O)NCc1cnsc1 N1(C(CSCCC(C)C)=O)CCC(N(C)C(c2cnn(C3CC3)c2)=O)C1 CC(C)C(O)C(F)(F)C(=O)N1CC2CC(C1)N2C(=O)COCC(F)F C=Cc1ccc(C(=O)NC2(C)CCC2)cc1.C1(C=O)CCC(=O)N1C1CC1.N C(C)(CCC(=O)N1CC(=O)CC1C(N1CCC(N2CCCC2)C1)=O)OCC CC(C)C(C(=O)NCC(C)CNC(=O)C)N(C)C.C(C)(C)C.C(=O)N C1(N(C)C(c2cc(Br)co2)=O)CN(C(c2ccnc(O)c2)=O)CC1F C(=O)(C(CC)CC(C)C)NC1CC2CC(NC(CCC=C)=O)C2C1 N1(C(Cc2ccn(CC)n2)=O)CC2C(CN(C(=O)C(C)OC)C)C2C1 C(=O)(C1CCCn2ccnc21)NC1C(OC)CN(C(C=CC=CC)=O)C1 CC1(C)C(CNC(=O)CC23CCCC2C3)CCN1C(=O)CCc1ccc[nH]1 c1(C(=O)NCCC(C)N(C)C(C23CCCC2C3(F)F)=O)cccc2scnc12 N#Cc1ccc(=NC2C3CC2CN(C(c2cscn2)=O)C3)[nH]c1 C1(OC)CCC2(C(=O)NCc3ccc(C(=O)NC4C=CCCC4)cn3)CC12 N1(C(C(c2cn(C)nc2)O)=O)CC=C(CC(=O)NOCC(O)C(C)(C)C)CC1 c1cc(C(N2CCCC(C)C2CC)=O)oc(=O)c1.C(=O)C=C(C)C.CC.O C1(CNC(C(C)C)CN(C)C)CCCC2(CC2)C1 c1(C(N(C(c2cn(Cc3ccnc(F)c3F)nn2)C)C)=O)nnc2n1CCCC2 Cn1c(C(=O)NCCC(O)CNC(c2coc(C3CCOCC3)n2)=O)cnc1O Cc1cccc(C(N2CC3CC3(CNCc3cnn(CC(C)C)c3)C2)=O)c1Cl CC1(C)CCC(CC(=O)NC2CC(NC(=O)Cc3csc(S)n3)C2)C1 CN1N=C(C(=O)N2CCC=CC2C(N2CCCCCCCC2)=O)CCC1=O N1(C(C(C)=C(CC)C)=O)CC=C(CC(=O)NCCCCC(N)=O)CC1 c1(C(CC)NCCSCCOC)nnc2ccccn12 c1(C(=O)NC(CNC(CCS(=O)(=O)NC)=O)C(C)C)nnc2n1CCCC2 N1(C(c2c(C)csc2)=O)CC(C2CCCN(C(c3ccc([N+](=O)[O-])cn3)=O)C2)C1 c1(CNC(=O)NCc2noc3c2COCC3)ccc([N+](=O)[O-])c2cccnc12 N1(C(c2c(OC)cc(C)s2)=O)CCN(C(=O)CCC(C)(F)F)C(CO)C1 C1(NC(c2nc(OC)oc2)=O)CC(NC(=O)C2=CCCC2(C)C)C12CCOCC2 C(=O)(CCCC(=O)NC1CN(C(c2ccc(Cl)cc2O)=O)C1)NCCC N1(C(=O)C=CCO)CCC2C1CCCN2C(C1CC12CCSCC2)=O c1(CCC)nc(C)c(C(=O)N(CCCCNC(=O)CCC2CC2(Cl)Cl)C)o1 C1(NC(C(CC)OC)=O)CCC(CC(=O)NCc2cnc(C)[nH]2)CC1 c1(OC)ccnc(O)c1C(=O)NC.C1CCCC1.C1(C#N)(CCC=O)CCC1 C=C=C(C)CC(=O)N1CC(CNC(c2cnn(C)c2C)=O)C(c2ccccc2)C1 CCC(C)(C#N)C(=O)NC1CCCN(C(c2c(C)nn(C(C)C)c2C)=O)CC1 c1(CC(C)NC(=O)Nc2cccnc2Cl)cn(C)c2ccc(F)cc12 Cc1cnn(C)c1C(=O)NC1CCCN(C(c2ccc(-n3cncn3)cn2)=O)C1 N1(C(C2(C#C)CCC2)=O)CCC(CNC(=O)Cc2sccc2Br)C(C)C1 C(=O)(CCC(C)OCC)N(C1CC(NC(C2(CCC=C)CCCC2)=O)C1)C CC(C)CCC(=O)C(=O)N1CCC(C(CO)NC(C2CC2C(F)F)=O)CC1 c1(C(=O)NCCC2(O)CN(C(CCC(C)C)=O)C2)cc(O)c2ccccc2c1 N1(C(c2ccn(C)c(=O)c2)=O)CC(NC(c2cnc(S)[nH]2)=O)CCC(O)C1 CC(CCO)C(=O)NCC1CCC(CNC(C2CCCC2C(C)O)=O)CC1 CC(C)CCC(C(=O)N(CCC(=O)OC)C)NC(=O)C(C)OCC1CC1 CN=c1ncc(-c2nn[nH]n2)c[nH]1.c12ccc(cc1Cl)C(=O)NC(=O)CO2 C(=O)(CC(O)C(C)CC)NCCN(CCC)C(c1csc(C#N)c1)=O c1(C(N2CCCC2CCc2ccncc2)=O)ccc(C2CCOCC2)cc1 c1(C(NCCN(C(=O)C=CS(C)=O)CC)=O)ccccc1C(F)(F)F.C c1(C(=O)NCC(CC)(C)COC)cc(S(=O)(=O)N(C)C)cn1C c1(OC(C)C)cc(NC(C)CCNC(C2CCC(C)CC2)=O)ncn1 C1(C(N(CC(N2CCC(c3ccon3)C2)=O)CC)=O)CN2CCN1CC2 Cc1nnc2cc(NCC3CC(NC(c4cncn4C)=O)C3)ncn12 c1(C(=O)NCC(CCOC)NC(c2n[nH]c(C)c2F)=O)ccc(F)cc1 CC(C)CC(C)(CNC(C1CC1c1cccnc1)=O)NC(=O)CC(C)(C)F c1(NC(=O)C#CCNC(=O)CC2CC(F)(F)C2)ccc(F)c(F)c1 c1(NC2CC2NC(C2CCN(CC)CC2)=O)cccc(F)c1C#N Cc1ccc(C(=O)N(CC(=O)Nc2cnn(C)c2)C2CC2)cc1C#N C(C(=O)NC1CCOC1)(C1=NOCC1)N(CCOC)C1CC1 C(=O)(C1=CCN(C)C1)N(CCC(C(C)C)NC(c1nc(Cl)ccc1N)=O)C CCC(C)C(C(=O)NCC12CC(NC(=O)C=C3CCCCC3)(C1)C2)OC Cc1cc(C(=O)NS(=O)(=O)CCNc2ccccc2)cc(C)c1F N1(C(CCC#CC)=O)CCCCC12CC(NC(C1C(C(F)F)C1(C)C)=O)C2 C1(SC)CN(C(C2(CC(C)C)CC2)=O)CC1NC(=O)C(O)c1ccco1 n1(C(C)C)nc(Br)c2c(N3CCC(Oc4ccccc4[N+](=O)[O-])C3)ncnc12 Cc1ccc(F)cc1CC(=O)NC1CN(C(=O)CO)CC1C(F)F.c1ccon1 c1(C(=O)Nc2ccc(C(N3C(C(N)=O)CCC3)=O)nc2)cn2ncccc2n1 CC1CN(C(=O)COC2CCOCC2)CC(C)N1C(=O)C=CC=C(Cl)Cl Cc1c(Cl)ccc(C(N2CC(NC(C3(n4cncn4)CC3)=O)C(C)C2)=O)c1O c1(C(N2CC3C(CNC(C(N4C(=O)CCC4=O)C)=O)(C3)C2)=O)cn2ccnc2s1 N1(C(C(CC)(C)O)=O)CC2CCN(C(=O)C=Cc3cc(F)cc(F)c3)C2C1 C(=O)(C1=NOC(C)C1C)N1CC(COC)C1.c1(C=O)cc(C(C)=O)cn1C.N C1(OCC(N2C(CNC(c3cc(C)sn3)=O)C=CC2)=O)CCC(F)(F)CC1 c1(CCC)cc(C(=O)N(CC(O)CNC(C2CC(O)C2)=O)C)n[nH]1 c1(C(=O)Nc2ccc(Br)nc2)cc(-c2ccc(F)cc2F)cnc1F C(=O)(C1=Cc2ccccc2OC1)NCCCN1CCN(C(C2C(C)CC2)=O)CC1 C=CC1(C(=O)NCc2cc(C(N3CC(O)C(C)(C)C3)=O)co2)CCOCC1 C1(SCC)CCC(C(N2CCCC2(C)CNC(=O)CC(F)F)=O)CC1 c1(CCCCC)nc(C)c(C(=O)NCC2CN(C(C3CC4CC4C3)=O)CC2C)s1 C1(OC)CC(C)N(C(=O)C(c2ccccc2)C)C1.n1(CCC(=O)N)cc(N)cn1 c1(C(=O)NC2(CC=C)CN(C(=O)C(O)C(C)(C)C)C2)cc(N)cc(O)c1 N1(C(C(CC=CCC)C)=O)CCOCC(C(N2CCCC(CCF)C2)=O)C1 c1(C(N(C)CC2(O)CCCN(C(CSC)=O)C2)=O)ccc2nccc(C)c2c1 C1(NC(CCCC=C)=O)CCN(C(=O)CC2(CSC)CC2)CC1C c1(C(=O)NCCCC(C)NC(CS(CC)=O)=O)cc2cccn2cn1 C1(NC(C2(CC)CCN(C(c3ccc(C#N)cc3)=O)C2)=O)COC2(CCCC2)C1 N1(C(C(=O)NCc2n(C)ccn2)=O)CCCC(O)(Cc2ccncc2)C1 c1(C(=O)NCC2N(C(C=CC=CCC)=O)CCC2)cc(O)nc(O)n1.C C(C)(CO)(C(=O)NC1CCCC(NC(=O)CCc2scnc2C)C1)OC Cc1cc(C(N2CC(NC(c3n[nH]cc3C(C)C)=O)CC2C)=O)ncc1C(N)=O C1(C2(O)CN(C(C3CC3F)=O)C2)(CNC(=O)C=Cc2cccc(Br)c2)CC1 Cc1cc(Cl)cc2cc(C(N3CCC(NC(=O)C(C)CS(C)(=O)=O)CC3)=O)[nH]c12 C1(CCNC(C(C)OC(C)(C)C)=O)CCN(C(=O)COC2CCCC2)C1 N(C1CCCc2ccoc21)C(CC(CCC)NC(C(CCCC#C)C)=O)=O C1(CC)CCN(C(C2CC2c2ccco2)=O)CC1.c1(C(=O)N)cnc(O)c(C)c1 c1(C(=O)Nc2cc(NC)c(OC(C)C)cc2)cnn2c(O)cc(C)nc12 CON(CCC(=O)N1CCC(CO)C(C)C1)C(=O)C1CCC(C)O1 C1(CCC)CCC(O)(C(=O)NC2CCC(C)C2)CC1.c1(C(=O)N)nnc(C)s1 C=CCC(C)C(=O)NC1CCN(CCNC(C2(F)CC=CC2)=O)CC1 C1(CC)C(=O)N(C)CCN1C(=O)CNC(=O)C(C(C)C)C(C)C c1(C(=O)NCC2(NC(C3N(C)CCC3)=O)CCOC2)ccc(CN=[N+]=[N-])cc1 C=CC(C)CC(=O)NCC1(C(=O)NC(C(N)=O)C2CCCC2)CC=CC1 C(=O)C#CC1(C)CC1.C12CCN(C1)C(=O)C=CC2.C1CCC1.NC.C=O N1(C(C(C=C)(C)C)=O)CCC2CCCC(C1)N2c1nc2cc(C)ccc2s1 N1(C(C2C(CCC)C2)=O)CCCC1C(C)(C)NC(=O)C=CSc1nc[nH]n1 C(=O)CS(=O)(=O)c1ccc(Cl)cc1.C(C=O)NC(C)=O.CC(=O)N(C)CC.N CCC(C)(CO)C(=O)NC1CCC(CCNC(c2cc3n(n2)CCC3)=O)C1 CC1(C(=O)Nc2c(Cl)cccc2Br)CCCN(Cc2ccc(Br)o2)C1 CCC(C)(CNC(=O)C(C)Cn1cccn1)NC(c1ccncc1)=O N1(C(c2cn(-c3ccccc3)nn2)C)CCCN(C(C2CCCCS2)=O)CC1 C1(NC(c2cn(CC)nn2)=O)CC2CCC1CN2C(=O)CC1COCCO1 C1(O)(CN(C)C(c2cn(C3CC3)cn2)=O)CCN(C(C2(C)SCCCS2)=O)C1 C1(C)(NC(=O)OC(C)(C)C)CN(C(c2cnc3nccn3c2)=O)C(C)(C)C1 FC1CCN(N2CC(n3cc4ccccc4n3)C2)CC1 c1(C(=O)NCC(CCNC(=O)Cc2nnc(O)s2)O)ccc(F)cc1Br c1(-n2cc(C(C3CCCOC3)OC)nn2)ncccc1C(=O)O C1(NC(C2C3CCN(C(C4CN(C)CC(C)O4)=O)CC32)=O)CCn2cnnc2C1 C(CCCCC(=O)NC1CC(OC(C)(C)C)C1(C)C)OCCN(C)C C1(C(=O)NC(C2CN(C(=O)C3=CS(=O)CCC3)C2)C)CCN2CCOCC12 c1(C(=O)NC(C2CCCN2C(=O)C=Cc2cnn(C)c2)C)cn2ccnc2cn1 S(=O)(=O)(c1cccc(Br)c1)NC(C(CC)C)c1nn[nH]n1 C1(NC(CCCC#C)=O)CC2CC1CN2C(=O)C1=CCCCO1 c1(C(=O)OCC)cc([SH](=O)=O)cc([N+](=O)[O-])c1C.C(CC1CCOC1)(CO)N N1(C(C(N2C(CC)CCC2)=O)=O)CCC(O)C(NC(=O)CCc2cncn2C)C1 c1(C2(C(=O)NCC(CCOC)NC(c3cncnc3)=O)CCC2)cccc(F)c1 c1(C(N2C3C(NC(c4cc(C)n(C)n4)=O)C(C3)C2)=O)cc2cccc(C)c2[nH]1 C1(NC(C2(OC)CC2)=O)CCC(NC(c2ccnn2C2CCC2)=O)CC1 C=CCCCCC(=O)NC(c1nocc1C(=O)Nc1cn(C)nc1C)C N1(C(CC(=O)NCC#C)=O)CC(NC(=O)CC(O)CCSC)CC2(CCC2)C1 N1(C(c2c(C(C)C)ccs2)=O)CCCC(CCNC(C2CC3(C2)CC3F)=O)C1 c1(CNC(CCN(CC=C)C(C2CCCN2C2CC2)=O)=O)cc(C)ncn1 Cc1cc(C(N2C3CCC2C(CNC(C2COCCOC2)=O)C3)=O)c(C)c(C)c1 c1(OC)cc(C(=O)NC2CCCC2)cnc1C(F)(F)F.C(=O)C#CC1CC1.C c1(C(C(=O)N(CC(N)=O)CC)C)cccc([N+](=O)[O-])c1 N1(C(CC)=O)CCOCC(NC(=O)CONC(=O)OC(C)(C)C)C1 c1(NC(C2CCN(Cc3nc(Cl)ccc3F)C2)=O)c(F)cc(I)cc1[N+](=O)[O-] C(=O)(C1CCCc2nnn(C)c21)NCC(CC=C)NC(=O)C(F)(F)C(C)(C)O N1(C(CC(=O)NCC)=O)CC(NC(C2(OCC)CCOCC2)=O)CC(C)C1 N1(C(C(C)c2ncco2)=O)C2CCC1CC(NC(=O)C=Cc1cocn1)C2 C(=O)(C1=Cc2ccccc2OC=C1)NCCCCN(C)C(c1cnc(O)o1)=O c1(C(C(=O)N(C(C)CC)C)=O)ccc(F)c(F)c1.C(=O)(C(C)(C)N1CCCC1)N C1(NC(c2cc(CC(C)C)[nH]n2)=O)CCC12CCOCC2.C(=O)(COC(F)F)N c1(OCC=C)ccccc1NC(=O)Nc1ccc(C(N2CCCCCC2)=O)cc1 C=C=CC(C)C(=O)NC(CCC1CCC1)C(=O)N1CC2CC1CS2 C(C1Cc2ccccc21)NC(C(Cn1cncn1)NC(=O)C=Cc1ccco1)=O C(C(C)(C(C)C)NC(C1CC2C=CC1O2)=O)NC(C(COC)OC)=O C12(C(N3CCC4(C3)CC4)=O)CC(C1)Oc1ccccc12.O=C(C=C1CCC1)N.C C(=O)(C(C)(C)CC(=O)NC1(C(=O)NC2C(O)CC2O)CCCC1C)OC N1(S(CC2(C)NC(=O)NC2=O)(=O)=O)CCC2(CC1)CC(C(=O)O)S2(=O)=O N1(C(C(Cc2ccco2)NC(=O)CCCn2cncn2)=O)CCSC2(CCC2)C1 C1(OC)CCC(C(=O)NC2CCN(C(C3(CC4CCCC4)CCOC3)=O)C2)CC1 CCC(C)(C#N)C(=O)NCc1cc(C(N2CCCCC(CO)C2)=O)no1 C(=O)(CCC(=O)NC1CCCCC1NC(=O)CCc1cc(Cl)no1)OC N1(C(c2c(SC)n(C)nc2)=O)CCN(C(C2CCC2S)=O)CC1CS(C)(=O)=O CC(=O)CCC(=O)NC(C1CCCN(C(=O)C(C2CCOCC2)O)C1)C c1(CC(N2C(CNC(c3nn(C)c(Cl)c3)=O)C=CC2)=O)ccc(O)cc1Cl C(C)(CNC(=O)C(F)OC(F)(F)F)(C(C)C)NC(CC=CC)=O C1(CC)(NC(c2cncs2)=O)CCN(C(C2(C#N)CCOC2)=O)CC1 Cc1cc(C(N2CC=CC2C(N2CC(O)(c3nn[nH]n3)C2)=O)=O)c(C)[nH]1 N1(C(c2cnc(OCC)s2)=O)CC2(C1)CN(C(C1CCCS1)=O)CC(C)(C)O2 c1(OC)ccc(Br)cc1CN(C(c1scnc1C)C(=O)NC1COC1)C CC#CCC(C(=O)NCCNS(N)(=O)=O)NC(=O)Cn1cc(C)cn1 CCC(C)CC(C(=O)NCC(C)(C)C(=O)OC)NC(c1cc2cc[nH]c2cn1)=O C1(CC(NOC(C=C)C)=O)CCC(NC(c2ncccc2O)=O)CC1 C1(CC(=O)NC(C#C)CC2CCCC2)CCCN(C(C2CCCCO2)=O)CC1 C12(C(=O)NCC(CC)NC(=O)C=Cc3ccnn3C)CC(CO)(C1)OC2C N1(C(c2c(N)nccn2)=O)CCC(CNC(=O)COc2ccccc2F)C12CC2 C1(CNC(CNC(CCC)=O)=O)CCC(NC(=O)CC2COCCO2)CC1 Cc1nc(SC(F)(F)F)[nH]c(=NCC2CCCN2C(C2CN(C(C)C)C2)=O)c1C c1(CC(C)C)cc(C(=O)N(C2CCCN(C(=O)C3=CCCS3)C2)C)n(C)n1 c1(OCC)ccccc1C(=O)NCCCCC(C)NC(=O)Cn1nnnc1C N(C(=NCc1cncnc1)NC1CCCN(CC2CC2)C1)C(COC)C c1(CC=O)ccc2c(c1)CCN2C.C1(C(=O)NC(C)C(C)C)CC(C)(C)CO1.N c1(C(=O)NCC(C)OC)cnn2cc(C#N)cnc12.C(=O)C(C)(O)C1CCC1 c1(C(N2CCCC(N(C(CCC(=O)NC)=O)C)C2)=O)cn2c(n1)CCC(C)C2 c1(C(=O)N)cc(O)cc(C#N)c1.N1(CCOC)CC(C(N2CCCC2)=O)CC1=O CC(C)=C=CC(=O)N(C)CCOCCC(=O)N1CC(n2cnnn2)C1 N1(C(C2(C)CCC(=O)N2)=O)CC=C(CCNC(=O)CC2C=CCCC2)CC1 C1(NC(C=CCOC)=O)C2CC(CN(C(=O)C3=C(Cl)CCCC3)C2)C1CO C1(C(=O)NCC(CC(C)C)(C)O)C(C2CC2)CCN1C(c1cn(C)cn1)=O C1(C(C)C)CN(C(=O)C(F)n2cccn2)CCCN1Cc1ccccc1 n1(CC)cc(C(=O)NC2(CF)CCN(C(=O)Cc3cnc(C)s3)C2)c(C)n1 CCCC(C)(O)CC(=O)NCC(Cc1ccccc1)NC(c1nc(Cl)oc1C)=O c1(C(=O)NCC(CC)NC(C2(C)COC2)=O)cc(C(C)=O)c(C)o1 CC1=C(C(=O)NCC2(CO)CCN(C(c3csc4nnsc34)=O)CC2)CCO1 c1(CNC(c2c(F)cccc2I)C)ccn2nccc2n1 C(=O)(C(C)C1=CCCC1)NCCC1CN(C(c2c(C)cns2)=O)C1 C1(NC(C(CO)N(C)C)=O)CCN(C(C2CCC2C(F)(F)F)=O)CC1 C1(CNC(COCCCC)=O)(CO)CCCN(C(=O)CSC(C)(C)C)C1 n1(CC=O)cccc(C)c1=O.c1(OC)cccc(CC(=O)NC(C)C(C)C)n1.N Cc1nc2cc(C(N3CCC(N(C)C(c4cc(Cl)c[nH]4)=O)C(C)C3)=O)ccc2o1 C(C1CCCC1)=C(C)C(=O)NCCCO.C1(CC(=O)N(CC)C)CCC1(F)F N1(C(C2CC2CNC(C23CCCC2C3)=O)=O)CCC2(CC1)CC2CO c1(C(N(CCCNC(C(CCSC)OC)=O)C(C)C)=O)ccc(O)c(N)n1 c1(C=O)cc(S(N)(=O)=O)oc1Cl.C1(CC)CCN(C(=O)C(C2CC2)C)C1 C1CCCCN(C)C1=O.c1(CC)cc(C)c(C(N2CC(C)(OCC=O)C2)=O)o1.N N1(C(C(C)(CSC)NC(C(CC)C)=O)=O)CC2(C1)CC(C)(C)C2 C(=O)(C1CCc2cccnc21)NCC1CC(NC(CCCC#C)=O)C1 C(=O)(C(C)(C)S(=O)(=O)c1ccccc1)N.N1(C(C2(F)C(C)C2)=O)CCCC(C)C1 C12(C(=O)NCC(CN(C(c3cnc(C)nc3C)=O)C)C)CCCCC(F)(C1)C2 CCCCS(=O)(=O)CC(=O)NC1CCCCCC1NC(C1(O)CCCC1)=O Cc1ccccc1C(=O)N(C(=O)CC1CCC(N)CC1)CC1CC1 c1(SC)cn(C)nc1C(=O)NCC(O)C.c1(C=O)nc(C(C)(F)F)cs1.N C1(NC(C=NOC)=O)CCCCC12CCN(C(=O)CC1(OC)CCC1)CC2 N1(C(C2CCC(C(=O)OC)O2)=O)CCN(C(=O)C)C2(CC2)C1.CCN(C)C C12CC(C(F)(F)F)(CO1)C2.c1(-n2nccn2)ccc(Cl)cc1.O=C(C=O)NC N1(C(CONC(=O)OC(C)(C)C)=O)CCCC(NC(C2CSCCS2)=O)CC1 CC1CCC(NC(c2ccc(-n3cncn3)cc2)=O)CN1C(C1CCS1(=O)=O)=O N1(C(C2(C#C)CCN(C(=O)C(C3CCOCC3)O)C2)=O)CCCC(F)(F)CC1 Cc1cccc(C(c2cnnn2C)NC(C2CC2(C)C)C)c1 Cc1ccc(N2CCN(Cc3ccnn3C3CCS(=O)(=O)C3)C(C)C2)cc1C c1(C(=O)NCC2CCCCC2NC(C2CCS(=O)CC2)=O)ccnc(Cl)c1O c1(C(N2CC(C(C)NC(c3cc(C(C)C)no3)=O)OCC2)=O)ccc(O)c(O)c1 C1(NC(c2cc(C)sc2C)=O)CN(C(c2cc(C(C)C)on2)=O)CCC1C C(=O)C1=CS(=O)(=O)CCC1.c1(NC(C)C)ccc(C(N2CC(CC)C2)=O)cn1 C1(C(C)C)CN(C(C2CC3(F)CC2C3)=O)CCN1C(=O)CC1CCCC1 Cc1ccn2cnc(C(=O)NC(C)(C)CCNC(c3ccc(C)s3)=O)c2c1 CCCCCC(CC)C(=O)N1CCC(C(N2CCCC2C)=O)(CC)CC1 c1(OC)ccc(O)cc1C(=O)NC1CC(C)C1.C1(C=O)CCCC(C2CC2)O1 CN=c1[nH]c(=NCc2c(Cl)cccc2Br)[nH]c(=NC(C)Cc2ccccc2C)[nH]1 C(C(C(=O)NCC#CC(F)(F)F)C(C)C)NC(CC(CC)OC)=O c1(OC)cc(O)ncc1C(=O)N.C1(CC=O)OC(C)(C)OC1=O.C1CC1.C c1(OC)cc(C)c(Br)cc1C(N1CCN(C(c2cnc(=N)[nH]c2)=O)C(C)C1)=O C1(NC(C(C)c2ccsc2)=O)(CO)CCCN(C(=O)CCS(N)(=O)=O)C1 c1(N2CCN(c3nc(NC(C)=O)sc3C#N)CC2)cc(C)nc2cc(C)nn12 C1(C)(C(N(CC)CC)=O)CC(C(F)(F)F)=NO1.Cc1ccsc1C=CC=O C(C)(C)(CC(F)C(=O)NCCn1ncnn1)NC(c1c(OC)nccc1)=O c1(C(N(CCCCN(C(=O)CC2CCCC2)C)C)=O)cc(N)ccc1Cl CC1CN(C(=O)CC2CC3CC(=O)C2C3)CCN(C(c2ncn(C)n2)=O)C1 c1(C2C(CC)C2)nc(CCOC)nn1C12CC(C)(C1)C2 c12cc(Cl)ccc1C(=O)N1CCC(C1C)NC(=O)CS2.CC=CC C1(C(=O)N)CC2CCCC(C1)C2.N1(C(c2c(CC)occ2)=O)CCC(C)C1(C)C Cc1cc(C(=O)NCC23CC(CO2)N(C(=O)COCCCF)C3)c(C)nc1C n1(CC)ncn(NC(=O)C2CN(C(=O)CC3COCC(C)O3)C3(CCC3)C2)c1=O N(C(=NCC1CCCN1C(=O)OC)N1CCC2(C1)C(=O)Nc1ccccc12)CC CC1(C)C=C(C(=O)N2C(C(=O)Nc3cccc(Cl)c3)CCC23CC3)C1 C1(CNC(C2CN(c3nncs3)C2)=O)COCCN(C(=O)CCn2cnnn2)C1 CC(C)(CC(=O)NC1CC2CC1CC2C(N1CCCC1)=O)C(F)F CC(F)(F)CC(=O)N1CC=CC1C(N1CCC(N2CCC2)C1)=O C=C1CC(C(=O)NCCc2ncon2)(CNC(=O)CCc2cnn[nH]2)C1 C1(NC(c2n(CC(C)C)ncc2)=O)CCN(CC)CC1.n1(CC=O)cccn1.N N1(C(CCc2onc(CC)n2)=O)CCC2(CCC2)C(NC(=O)CC(O)C2CC2)C1 C1(CCC)CN(C(c2ccnc(CC)c2)=O)CCN1C(=O)C(C)CC(F)F c1(C(=O)NC2CCN(C(c3c(C)nc(CC)s3)=O)C(C)C2)cc2c(s1)CCOC2 C(=O)(Nn1ccccc1=O)C1(CC)CN(C(=O)CCc2cnco2)C1 CC(C)(C)C#CC(=O)N.C1(C(N2CC(O)C2)=O)CC(=O)N(c2ccccc2)C1.C C12(Nc3cc(C(N)=O)ncn3)CCC(CC1NC(c1ccnnc1Cl)=O)C2 c1(C(=O)NC2CC(CCNC(C(COC)C)=O)C2)scc(C)c1Cl N1(C(CONC(c2cn(CC)nc2)=O)=O)CC2CCC2(CC2CCCO2)C1 C(=O)(C1=NOC(C)C1C)N1CCC(O)(CC)C1.c1(OC)nc(C)cnc1C(=O)N N1(C(c2cc(OCC)no2)=O)CCC2(C=C(C(=O)N3CCCNC(=O)C3C)C2)C1 N1(C(C(C)SCC)=O)CCC(=CCNC(C2(CO)CCOCC2)=O)CC1 c1(C(N2CCCCC2C2(C(=O)O)CC2)C)cc2ccccc2cn1 C1(CC=C)(C(=O)Nc2c(F)ccnc2F)CCN(C(=O)C(C)OCCO)CC1 C1(C=O)CCCC(C)(C)C1.Cc1ccc(COC(C)C(=O)N(C(C)C)C)cc1 N1(C(c2c(CC)ncs2)=O)CC=C(C)CC1.c1(C(C(=O)N)O)cc(F)cc(F)c1 C(=O)(CC(F)(F)CC(=O)N1CC(CO)(NC(c2cc(OC)ccc2F)=O)C1)OC N1(C(CCC=C)=O)CCC2(CCC(NC(c3ccc(F)cc3F)=O)C2)C1 N(C)(S(C)(=O)=NC(=O)c1ccc(C(c2nccs2)=O)c(Cl)c1)C(C#C)(C)C N1(C(C2(O)C(C)(C)C2)=O)CC2(NC(=O)Cc3csc(Br)n3)CCC1C2 N1(C(CCN(C)CCO)=O)Cc2nccn2CC(NC(=O)COC2CC2)C1 Cc1oc(C)c(C(=O)NC(C)CCNC(c2cnn(C)c2C2CC2)=O)c1C CC1C(NC(=O)C(F)OC(F)(F)F)CCCN1C(c1cc2cscc2s1)=O c1(C2CCN(C(C3C(C)C3(C)C)=O)C2)ccccc1O N1(C(CCOC)=O)CCCC(C)C1CCNC(=O)CNC(c1ccco1)=O c1(CN(C(C(=O)NCCSC)C2COC2)C)nnc2n1CCNC2=O C(=O)(C(O)P(C)(C)=O)NC(C1CN(C(c2coc(O)n2)=O)C1)C C1(C2CCCOC2)(NC(C2CSCN2C(=O)C#CC2CCC2)=O)CC1 C12(NC(CCC(C)CN(C)C)=O)CCCC1(F)CN(C(c1nonc1N)=O)C2 c1(NC2C(C)CN(C(=O)CCc3nc4cccnc4[nH]3)C2)ccnc2ncnn12 C1(C(=O)NC(C2CCN(C(C(CSC)(C)C)=O)C2)C)COC2COCC12 N1(C(CC(=C)C)=O)CCC2(CCCCC2NC(C2CSCCS2)=O)CC1 C=C(C)C1OCCC1C(=O)NCCC(C)N(C)C(c1cc(N)cc(O)n1)=O C(=O)(C1=CNC2=NCCCC2=C1)N1CC(CNC(c2cc(Cl)cs2)=O)OCC1 Cc1cccc(C(O)C(=O)NC2CCC2CNC(c2c(C)cnnc2O)=O)c1F c1(C(=O)NC(C2(C)CC2)C)cc(Cl)c(C#N)c(Cl)c1 Cc1ccc(CC(O)CNC(=O)C(C)C2(O)CCC2)cc1F Cc1ccn(C)c1C(=O)NC1C2CC(NC(=O)CC(O)CN(C)C)CC12 c1(CCC(=O)NC(CCCNC(C(C)CN(C)C)=O)C)ccc(F)cc1Br C12(C(=O)NCCn3cc(C(C)(O)CCO)nn3)CCC(CC1)OC2.c1cncn1C CC(CC(=O)NC1CCN(C2CC2)C1=O)C(C)(C)NC(C1CCC(=O)CC1)=O C#CC1(NC(=O)COC(C)(C)CNC(=O)C=C=C(C)C)CCCOC1 S(C1CCc2c(F)cccc21)CC(=O)NC1C(C)(C)CCCC1 C1(C(=O)NC(Cc2ccc(C(=O)OC)cc2)C)CNc2ccccc2C1 Cc1nc(N2C3CN(C(=O)CC(C)C)CC23)cc(C(F)(F)F)n1 N1(C(c2ccc(CC)o2)=O)CCCC12CCN(C(C1CCN(C)S1(=O)=O)=O)C2 C1(C)(CC)CCC(C(N2CCC(C)C2CNC(C2CCC(=O)N2C)=O)=O)O1 CCC(C)C(C(=O)NC1CC(NC(c2cncc(N)n2)=O)C1)NC(C)=O C(=O)(C(C)CC(=O)NC(CCN(C)C(C1CN(C)C1)=O)C(C)C)OC c1(C(=O)NCCC(C)(C)NC(CCOCCOC)=O)cccc(Br)c1 N1(C(c2nn(CC)c(O)c2)=O)CCC(CO)(NC(=O)C(C)=C2CCC2)CC1 c1(C2(C(=O)Oc3c(C)scc3)CCCO2)ccccc1Br c1(SC)ccc(O)cc1Cl.c12ccc(cc1)NC(=O)Nc1c[nH]nc1C(=O)N2 c1(OCC(=O)NCC2CCN(C(C3(O)CCCC3)=O)C2)ccc(Cl)c(F)c1 c1(C(N2C(CNC(Cn3c(C)ccc3C)=O)CC2)=O)cc(F)c(O)c(Cl)c1 CC1C(NC(c2cncc(Cl)c2)=O)CCN1C(c1cc(CN(C)C)on1)=O CC(C)(C)C(=O)C(=O)N1CCSCC1CCNC(=O)CC1CC(O)C12CCC2 c1(C(=O)OC)ccc(C(N2CCCC(NC(c3coc(Cl)c3)=O)CC2)=O)c(C)c1 CC(C)(C)C(=O)C(=O)NCC1(NC(C2(CC(F)F)CCC2)=O)CCC1 c1(C(=O)NCCCCN(C)C(c2cc(=O)cc(Cl)[nH]2)=O)cnc2sccc2c1 N1(C(c2n(CCC)ncc2)=O)CC(C(F)F)C2(CCC2)C1 c1(CCC)nccn1CC(=O)NC(C)(C)CC.c1(C(=O)N)ocnc1C1CC1 C1(CN(C)C(c2cnc(S)nc2)=O)CCCCN1C(=O)CCCc1n[nH]c(=N)s1 N(C1c2ccccc2CC1NC(=O)C(n1nccc1C)C)C(CSC)=O N1(C(C(C)=CC)=O)CCCCCC(NC(c2cc(C(C)C)sn2)=O)C1 c1(C(=O)NC2(C3N(C(COC)=O)CCCC3)CC2)ccc(N(C)C)cc1F c1(OC)ccc(NC(=O)C(F)C(=O)N2CCCC(CN3CCN(C)CC3)C2)cc1 c1(C(=O)NC2(CCC(=O)NC(C(C)CO)C)CCC2)cc(O)ccc1F c1(OCC)cc[nH]c(=NCCCCC(C)NC(c2cnn(C3CC3)c2)=O)n1 c1(NCc2nc(CCC)sc2)ccc([Si](C)(C)C)cn1 c1(N(CCCF)CCO)cc(CO)ncn1.c1ccccc1 C1(C(=O)NCC(=C)C)CC(F)CN1Cc1ncccc1F n1(CC(=O)NC2C=CCN(C(CCCC=C)=O)C2)c(C(F)F)nc2ccccc12 Cn1nc(C(N2C(CNC(C3(C)SCCCS3)=O)CC3CC23)=O)cc1F N1(C(C2CC(C)C2)=O)CCC2(C(=O)NC3C(O)C4CCOC34)CCCC12 c1(OC2(c3nnnn3CCO)C(OCC)CCC2)nc2sccn2c1C.CSC Cc1cc(Cl)c(C(N2CCN(C(C3CCCOC3C)=O)CC2CO)=O)cc1C N1(C(CCC(CC)OC)=O)CC(C(=O)N(C2CCC2)C2CC2)CCC1(C)C C1(C(N(CCCCNC(=O)CSCCC#N)C)=O)CC12CCOc1ccccc12 CC1(C)OCC(C=CC(=O)NCC2NCCC2C2CC2)O1 C=CCCC(F)(F)C(=O)N1CCCC1CN(C(=O)C(CCC)C(C)C)C n1(C(CC)C)nnnc1C(c1ccc(C)o1)NCCn1ncnn1 C1(NC(c2nc(CC)sc2)=O)CC(F)CN(C(=O)C(O)CC(N)=O)C1 C1(CC(=O)NC(C)CCCCNC(=O)C(F)C2CCCC2)(OC)CCCCC1 c1(OC)cc(Cl)ccc1CCN(C=O)Cc1ccc(C(C)C)cc1F CS(=O)(=O)C1CN(C(C23CCC(F)(CC2)C3)=O)CC1.C1(C2CC2)(C=O)CC1 c1(OC)cc(C(N2CCC(NC(c3ncn(C)n3)=O)C(F)C2)=O)cc(F)c1F C(=O)(C(F)C(F)(F)F)N(CC)C.C1CCCN1C(C1CN(C2CCC2)C1)=O O=C1CN(CC2CCC(F)C2)C(=O)N1CC(Cl)Cl C=CC(C)(C)C(=O)NCc1cc(C(N2CC(C)CC2CC)=O)n[nH]1 CS(=O)(=O)c1ccc(C(N2CCC(CO)CC2)=O)[nH]1.C1(CC(=O)N)CC1(Cl)Cl CC(CC(=O)NCCC1(O)CCC1)C(C)(C)NC(=O)NC1CC1 c1(N(CC(C)C(C)(C)C)C)ccc(S(=O)(=O)NC2(CO)CCSC2)cn1 CC1CN(C(C2(Cl)CC2)=O)CC1CNC(=O)CC1CC(=O)C1 C(=O)(N=c1[nH]oc2cc(Br)ccc12)C1N(C(CCNC(C)=O)=O)C2C(C1)C2 CC(C)C1=NOC(C(=O)NCC2CN(C)CCN2C(=O)Cc2ccsc2Cl)C1 n1(C(C)C)ncc(C(=O)NCC(CO)NC(=O)CN2CCCC(N(C)C)C2)c1F N1(C(C(CC)NC(C)=O)=O)CCC2(CC1)COCC(CNC(=O)CCF)O2 C(CCCC(=O)NC1CCOC(C(=O)NCCn2cnnn2)C1)OCC CC(C)CCC(C(C)(C)C)NCCOC(=O)CN1CCCC1C C(=O)C1=CC2C=CC(C1)C2.Cc1cccc(C)c1OCC(=O)N(CC(O)C)C.N C(=O)(CCC(N)CO)N1C(c2ccc(C)cc2)C(C)C1 C#Cc1ccc(C(=O)NC2CC(CNC(c3cccnc3S)=O)C2)c(C)c1 N1(C(Cc2ccc(C)c(C)c2)=O)CC2CC1CCC2NC(=O)C(C)n1cnnn1 C1(NC(CCCC#C)=O)CC2(C1)CN(C(c1cccc(C#N)c1)=O)C2 C(=O)(C(C(C)C)C(C)C)N1CCC(NC(C(CC(C)C)ON)=O)CC1 N1(C(C(C(C)O)NC(=O)C2CC2)=O)CCC(C2(O)CN(C(=O)CO)C2)CC1 CCC(O)C(F)(F)C(=O)NCc1cncnc1 C1(F)(CNC(C2CCCCC2(F)F)=O)CCCN(C(=O)Cc2cn[nH]c2)CC1 n1(CC(=O)NCCC2CCC(NC(c3ccn(CC)n3)=O)C2)cnccc1=O N1(C(CCC=C)=O)CCC2(CCC2NC(=O)C=Cc2c[nH]c(=N)c(C)c2)CC1 N1(C(c2c(C)cc(C)o2)=O)CCN(C(c2sncc2Br)=O)CC12CCC2 C1(CN(C(=O)C)CC)CCCN1C(=O)C(C)O.C1CCOCC1.CCC(C)C Cc1nccc(C(N2CCN(C(=O)CCc3c(F)cccc3F)CC2C)=O)c1Cl c1(N(C(=O)CC(Cl)Cl)CC(=O)OCCSC)ccc(C#N)cc1F C=CCC(CC(C)C)C(=O)N1CC2CCC1C(CNC(=O)C(C)(C#N)CC)C2 C1(C(=O)NC)(COC)C=CCN1C(=O)CCn1ccnn1.c1ncc(C)o1 C1(NC(C2CC(=O)N2)=O)CCCNC12CCN(c1ncncc1Br)CC2 c1(C(=O)NC2CC3C=CC2O3)ccc2nccn2c1 C1(NC(c2c(CC)ncs2)=O)CC2CCC1N2C(=O)C(C(C)C)N1CCCCC1 c1(NC(C2C(NC(CCNC(C)=O)=O)C2)=O)cnnn1C c1(CN(C(=O)C(C)(C)NC(=O)Cc2cnn(C)c2)C)cnnn1C C(=O)(C#CC1CCCCC1)N1CCOCC(NC(C(C)CF)=O)C1 c1(CNC(C2C(C(=O)OCC)C2)=O)cc(C(=O)OC)cc(I)c1 C1(NC(CCc2cc(C)[nH]n2)=O)CCCCN(CCOc2cccc(F)c2)C1 N1(CC(C)C)N=C(C(=O)NC2CC2NC(c2ccc3ccsc3c2)=O)CCC1=O C(C(CC1CC1)C(=O)N)SC.C1CCCCO1.C1(C(N2CC(O)C2)=O)CCC1 C(=O)(C(C)(C)C(C)(C)C)N.C#CCCN(CC(=O)NCC1CC1C)C C(=O)(CCCCC(=O)NCCCNC(c1ccc(OC2CC2)cc1)=O)NC.O C(=O)(CC(C)(C)C(C)(F)F)N1CC2CN(C(COC)=O)C2CC1 c1(C(C)=O)ccc(C(=O)NCCN(C(=O)C(O)C(C)C)C)cc1C C1(CNC(c2cn(C(C)C)nn2)=O)COCCC1(F)F C1(C(N2CCC(O)(CCNC(C(C=C)(C)C)=O)C2)=O)CCC(C)(C)CO1 C1(C(=O)N)CCCCC1.C1(C=O)CC12CCC2.N(CC)(CC)CC.C(C)C C1(C2CN(C(c3cc(C)[nH]c3)=O)C2)CN(C(=O)CCn2c(C)ccc2C)CCO1 C1(NC(CC=CC)=O)C2CC(O)C1N(C(c1cnn3ccncc13)=O)C2 CC(C)(C)C(C)(O)C(=O)NCC12CCC(CC1)CO2.C(=O)C=CCF.C Cc1nc2ccccc2c(=O)n1CC(=O)NC(CNC(=O)C1=CCC1)CC(C)C c1(CC(=O)NC2CCN(C(C(CC)(C)F)=O)CC2F)ccc(OC)c(OC)c1Cl CCC(C)(COC)C(=O)NC1CN(C(c2cc[nH]c(=NC)c2)=O)CC1F C(=O)(C(O)CC(F)(F)F)N1CC(C(C(=O)OCC)F)C1 c1(C(N2CCC3(NC(c4cccs4)=O)C(CC2)C3)=O)cc2c(cc1F)NCCC2 CC(C)CN=C(NCCc1cc(C)cnc1O)N1CCCC(C(=O)OC)(CO)C1 C1(NC(C(C)O)=O)CCC12CN(C(c1ccc3c(c1)CC3)=O)C2 C12(C(=O)NC(CNC(CSCC(C)=O)=O)C3CC3)CC1COC2(C)C C1(CC(=O)NCC(C)N(C)C(C2CCCOC2)=O)Cc2ccc(Cl)cc2C1=O C1(NC(C(COC)O)=O)CC2CC(NC(C3CC4(CC(OC)C4)C3)=O)C1C2 CC1(C(F)F)CC1C(=O)NC(C(=O)NCCOC1CC1)c1cccs1 C1(C(=O)NC2C(C)COC2)CN(C(c2ccccc2)=O)C(C)(C)C1 N1(C(C2=C(C)OCCS2)=O)CCN2C(=O)C(NC(=O)C=CC(F)(F)F)CC2C1 C12(CNC(c3ccns3)=O)CCC1CCN2C(=O)C.c1ccc(Cl)c(Cl)c1.O N1(C(C23CN(C(CC4(OC)CCC4)=O)C(C2)CO3)=O)Cc2ccccc2C1 c1(CN2CC3N(C(C4CCC(C(F)(F)F)CC4)=O)C3C2)cc(F)ccc1Br CC1=C(C(=O)N2CCCN(C(c3cnn(C)c3C)=O)C(CO)C2)S(=O)(=O)CCO1 c1(OC)ccc(C(N2CCN(CCNC(C3C(Cl)(Cl)C34CC4)=O)CC2)=O)nc1 N1(C(=O)C2=COCCO2)CC2OCCN(C(C3CC4(C3)CC4F)=O)C2C1 C(CNC(=O)CN1CCN(C)CC1)(CC(=O)NC1(CF)CCCC1)OC N(C)(C(=NCC(C)(CC)OC)NCc1cccs1)Cc1ccn(CC)c1 C(=O)(C(C(C)NC(=O)C(O)CN1CCCC1)C(C)C)NCC=CCCC C1(N(c2ccnc(OC)n2)C(c2ccnc(Cl)c2Cl)=O)C2CCC1CNC2 C12(NC(CC(C=C)(C)C)=O)CCCC1N(C(=O)C1=CCC(C)(C)CC1)CCC2 c1(NC(=O)C(O)Cc2cnc[nH]2)ccccc1.C1(C=O)CC(=O)N(C2CC2)C1.N C1(NC(C(C)NC(CC)=O)=O)CCCC1NC(=O)CCO.CCN(C)C c1(C(N2CCN(C(c3ccc(OCC)nc3)=O)CC2)=O)cccc(Cl)c1O C(=O)(C(F)C(F)(F)F)N1CC(C)C(CNC(c2ccc(Cl)c(C=O)c2)=O)C1 CCCS(=O)(=O)C1CCN(c2cnc(SC)cn2)CC1 c1(OC)ccc(NC(=O)C(=O)NCCc2[nH]cnc2C)cn1 c1(NC(c2ccc(Br)o2)C)ccc(S(=O)(=O)NC2CC(C)(C)C2)c(Br)c1 Cc1ccc(C(N2CC3CC(NC(c4ccc(C(N)=O)[nH]4)=O)C2C3)=O)c(F)c1Cl c1(C(=O)NCC(CC)NC(=O)CS(C)(=O)=O)nc(C2CC2)n2ccccc12 C1(C(=O)NCC=CC)CN(C(C2CCCCC2(C)C)=O)CCN1C C1(CC)C(NC(c2nn(C)nc2C)=O)CCCN1C(=O)C(C1CCOCC1)O N1(C(C2C(C)(C)OCCO2)=O)CC(CO)C2(C1)CN(C(c1ccc[nH]1)=O)C2 c1(C(=O)NC(C)C(C)(C)NC(C2CC2[N+](=O)[O-])=O)coc2c(F)cc(Cl)cc12 c1(C(N(C2CCN(C(CCCNC(C)=O)=O)CC2)CCO)=O)nn(C)c(C)c1Cl CC1CN(C(=O)C(F)(F)c2ncc[nH]2)CCC1N(C)C(c1ccc(Cl)s1)=O c1(C(N(C2CCNC2)CC)=O)ccc(C2CC2)o1 C12(CNC(CCCC(C)=O)=O)CCCC1N(C(=O)Cn1cccnc1=O)CCC2 Cc1nc(C(=O)NCC2CC(F)CN2C(=O)CNS(=O)(=O)N(C)C)cn1C c1(CC)nc(C(=O)N)c(C)o1.C1CCCC(C)C1.C(C)(C)CN(C(=O)C)C C(C1CCCCCC1)=CC(=O)NCC1(C(N)=O)CCCO1 N1(C(C(CC)(C)C)=O)CCCC(C2CC2NC(c2cc(OC(F)F)n(C)n2)=O)C1 c1(OC)ccc(C(=O)NC2CCN(C(c3c(Cl)cnn3C)=O)C(C)C2)c(OC)c1 Cc1ccc(C(=O)NCCn2cc(Cn3nc(C)cc3C)nn2)c(F)c1 c1(C2CC(OC)C2)nc(-c2ccc(F)cc2)nn1C1CCOCC1 C1(C2CC2)(OC)CN(C(=O)C(F)C2CC(NC(C3CCNC(=O)C3)=O)C2)C1 Cc1nc(C(=O)NCC2CCC(C)N(C(=O)C#CC3CCC3)C2)c(=O)[nH]c1C C=CCC(C(=O)OC)NC(C1(SC)CN(C(=O)Cc2ccnn2C)C1)=O Cc1nc(Cl)nc(N2CCCC(CNC(c3ccccc3N=[N+]=[N-])=O)C2)c1C#N c1(CC(N2CCN(C(C(CC)C)=O)C3C2CC3)=O)ccc2ccccc2c1 C(=O)(C(CCC(C)C)NC(c1nonc1CC)=O)NCC=CCCC CC(C)C(CNC(c1cnc2n1CCC2)=O)C(=O)N(C1(CO)CC1)C N1(C(CC(C)(C)F)=O)CCN(C(C2(c3cc(N(C)C)cc(F)c3)CC2)=O)C2CC12 CC1=NOC(C(=O)NCCOC2CN(C(c3cn(C4CC4)nn3)=O)C2)C1C N1(C(CC(C)n2ccnc2)=O)CCN(C(=O)COc2ccc(Cl)nn2)CC1CO C(=O)(C(C)N(C(=O)C(C)N(C(=O)Cn1ccnn1)CC)C)OCC c1(C(c2nnnn2C2CCC2)Nc2ccc(C(F)(F)F)nc2)cc(Cl)ccc1Br N1(C(CC2(COC)CC2)=O)CCOC(C(=O)NCC2=CCCCC2)C1 c1(SC(C)C(=O)NC2C3CC2N(C(=O)CCc2nncs2)C3)ccc(F)cc1 C1CC2(C1)CCC2.C1(C=O)CCCN1CC(F)(F)F.C(C=O)(C1CC1)OC.N N1(C(CC(=C=C)C)=O)CCC2CCC(NC(=O)C(CCC(=O)OC)N(C)C)C12 c1(C(=O)N)cn2c(n1)COCC2.CCC(CCOC)C(=O)NC1CCC(F)(C)C1 CC(CC(F)(F)F)C(=O)NC1(C(=O)NC(c2ccncc2F)C)CC(O)C1 C1(NC(=O)COC2CC2)CCOCC1NC(=O)C(F)CC1CC1 C#Cc1cn(C)nc1C(=O)NC(C)(CNC(c1cccs1)=O)C1CCC1.C N1(C(CCC=C(C)C)C)CCOCC(C(=O)NCCCc2nc(C)cs2)C1 CC1CC2(CC2)CN1C(C1CC(O)CCN1C(=O)CCc1ccccn1)=O c1(NC(c2c(CC)ncs2)c2nnnn2C)ccc2c(c1)nnn2C N1(C2CCN(C(CCCC)=O)C2)CCN(C(c2cc(OC)n[nH]2)=O)CC1 CN1CC(O)CC1C(=O)NCCOCCC(=O)NCc1ccc(O)cc1 c1(OC)cc(OC)nc(N2CCCC(C)(C(N3CCC(O)C3)=O)C2)n1 N1(C(Cc2c(C)noc2Cl)=O)CC2(CCC(NC(=O)C(O)C3CCCC3)CC2)C1 C1(NC(c2coc(Br)c2)=O)CN(C(C2(C3CCCO3)CC2)=O)CC1F N1(C(c2c(C)cnc(F)c2)=O)CCN(C(=O)C2=CCCS2)CCC1C C1(CC(=O)NC(CC2CN(C(C3(OC)CCSC3)=O)C2)C)C(=O)ON=C1C C(=O)(CCCCNC(=O)C(F)C1CCOC1)N1CC(OCC)C1 N1(C(CC2C(C)=NN(C)C2=O)=O)CC2CCC1CN2C(=O)C=Cc1cccnc1 Cc1ccc(C(=O)NCCCN2CCN(c3snc(C)c3C#N)CC2)c(Cl)c1 C1(F)(C(N2CCCC(C(C)(C)O)C2)=O)C(C)(C)C1(C)C.CC1CC1(F)C(=O)N N1(C(C2C(CC)C2)=O)CCCC(C2CN(C(C3(c4ccncc4)CCC3)=O)C2)C1 C1(CNC(CSC)=O)CCCC1NC(C1CC(n2cnnc2)C1)=O N1(CC(C)C)CCN(C(=NCc2ccnn2C)NC2CCCC2(F)F)CC1 C1(CC(=O)NCCCC(=O)NCc2ccn(CC)n2)CCOC1(C)C C1(CC=C)(C(=O)NCC2(C)CCCCC2)CCN(C(=O)CC(C)(C)O)C1.O C1(CNC(C(COC)OC)=O)N(C(c2cn3ccnc3cn2)=O)CCCC1(C)C C1(C)(CNC(C(CC)OC2CCCC2)=O)CN(C(=O)C(CC)(CO)OC)CCO1 c1(C(N2CCCC(N(C)C(C3CCS(=O)(=O)C3)=O)C2)=O)cc2c([nH]1)CCCC2=O c1(C(N2C(C(N(C)CC3C(C)C3)=O)CNC(=O)C2)=O)coc2ccccc12 C1(C(N(C)CCC2CCCN2C)=O)CC(O)CN1C(C1(C)CC(C)(C)C1)=O C1(CNC(C(c2ccc(C)s2)C)=O)CC(F)CN1C(C1C(C)C1C)=O C1(C(C)(C)O)CCN(C(C2(NC(=O)CC3CCC(=O)O3)CCC2)=O)C1 C1(CN(C(=O)CCn2ccnn2)C)CN(C(C2CC(CF)C2)=O)CCO1 C1CCN(C(c2ccc(C(F)(F)F)nc2)=O)CC1(F)F.c1(C(=O)NC)cnn[nH]1 C1(NC(c2ccncc2O)=O)CCCCCC1C(=O)NCC1(Cl)CCC1 CC1CN(C(C2CC(Cl)(Cl)C2)=O)CCCN1C(C1CC1(C)C)=O C1(C(C(=O)NC2CC(C)(NC(COC)=O)C2)C)CCC(C)(C)CC1 C#CC1(C(=O)NOCC2CCCC2)CN(C(=O)CCOCC)C1 N1(CC(=O)NC)CC2CC1CN2C(=O)NC1CC1.C1CCN(CC(F)F)CC1 C1(N=[N+]=[N-])(C(N2CCCC(C)(O)C2)=O)CCN(C(c2csc(O)n2)=O)C1 N1(C(C=CC(CC)C)=O)CCC(CCCCNC(c2ccc(OC)nn2)=O)CC1 N1(C(C(CSC)(C)C)=O)CC2(C1)CN(CC1CCCC1)C2 C(=O)(C(C)(C)CCNC)N1CCC(CC(C)NC(=O)C=CC2CCOCC2)CC1 c1(-n2cc(CCCC)nn2)cc(C)ccc1C(=O)NCCSC.c1ncc(C)o1 [N-]=[N+]=Nc1ccccc1C(=O)N(CCCNC(c1cnsc1)=O)CCO N1(CC)N=C(C(=O)N2CCN(C(C3CCN(CC)CC3)=O)C3CC23)CCC1=O Cc1c(C(N2CCC(F)(CNC(c3cnsc3)=O)C2)=O)ccc(F)c1F N1(C(CCC(CC)C)=O)CC2CC(C1)CN(C(c1ncnc(C)c1OC)=O)C2 C12CCN(CC1)CCCN2.C1(c2cccc(Cl)c2)(C(=O)OCC)CC(F)(F)C1 CC(C)CCCCC(=O)NC1CCC(CCNC(c2ccc(F)c(O)c2)=O)C1 Cc1nc(C(=O)N(C)CCN2CCN(C)CC2)nc2ccccc12 c1(C(=O)N)ccc(C2CC2(Cl)Cl)cc1.C1(C=O)CC=CCO1.C1(CC)CC1.C Cc1nc2n(c1CC(N1CCC(CF)(NC(=O)CC)C1)=O)CCCC2.C(N)=O.N CN=S1(=O)CCC2(CC1)CN(C(=O)NCC(c1cc(C)nn1C)=O)CCO2 C1(C(N2CCC(CSC)C2)=O)CN(C(=O)Cc2ccnn2C)CC1F N1(C(CCN(CC(F)(F)F)C)=O)CCN(C(C2CCCN2C=O)=O)CC1C(F)F C1(C#CC(=O)N2CCCC(C3CCCN3C(=O)CCCN=[N+]=[N-])C2)(CC)COC1 Cc1ccc(S(=O)(=O)Nc2cccc(CNC(c3ncc(C)cc3O)=O)c2)cc1 C1(CC)CC(C)CN1C(c1snnc1C(F)F)=O n1(CC)c(C(=O)C2CC2)cnc1O.C(=O)(CC)NCCN.[SH](C)(=O)=O n1(CC(N2CCN(C(=O)CNc3ncccn3)CC2)=O)c(=O)oc2ccccc12 Cn1cnc2c(C(=O)NCC34CC3CN(C(C3CC(C)(O)C3)=O)C4)ccnc12 C(=O)C1Cc2c(Cl)cccc21.c1(CC)[nH]c(=N)sc1C(=O)NC1CCCC1C N1(C(C(c2cnn(C)c2)C)=O)CCC(CNC(=O)CCCC2CC2)CC1C c1(C(C)=O)cnc(N2CC3(CC3C(=O)NC(c3cc(Cl)cnc3Cl)=O)C2)nc1C c1(OCC)ccc(-c2cn(CCC(=O)N(C(C)CS(C)=O)C)nn2)cc1OC c1(C(=O)NC2CC(C)N(C(=O)C3=CS(=O)CCC3)CC2)cc2ccccc2o1 C(CCCN=c1[nH]c(N2CCC3(CCC3)C(CO)C2)nc2cc[nH]c12)OC n1(CC2C(C)C2)nc(CS(C)(=O)=O)nc1-c1csc(C(F)(F)F)c1 C1(CC(=O)NC(C)Cc2cn[nH]c2)CCCC1NC(c1ccc[nH]1)=O CC1CN(C(C2CCC(F)CC2)=O)CCC1NC(c1cnc(N)c(O)c1)=O N1(CC(=O)NCCCC2(CNC(C(C)CO)=O)CCCC2)CC2CCC1C2 C12(CNC(CCC3(C)CCC(=O)N3)=O)CCC(C1)N(C(c1cn[nH]c1)=O)C2.C CCC(CC)C(=O)N(CC(O)CN(C)C(c1ncsc1NC)=O)C Cn1nnc2c1CC(C(=O)NCC1(O)CN(C(C3(C4CCC4)CC3)=O)C1)CC2 C1(NC(C2CC3C(C2)C3(F)F)=O)CN(C(C2SCCCS2)=O)C2CCCC12 c1(CCC(=O)NCCC(C)NC(C=Cc2c(C)ncs2)=O)ccc2[nH]ccc2c1 c1(C(C(=O)NCCCSC)OC)nc(C2CC2)n(-c2ccn(C(C)C)n2)n1 c1(NC(C=C2CCN(Cc3n(C)ccn3)CC2)=O)c(F)ccc(Cl)c1F CC(C)CCCC(=O)NCC(O)CC(=O)N1CCN(C(C)(C)C)CC1 C1(NC(Cc2cccc(C(=O)OC)c2)=O)CC(=O)N(C2CC2)C1C N1(C(CSCCC)=O)CCCC1CCCNC(=O)COC1CCOC1 N1(C(CC(CC)C)=O)CCCC12CCN(C(c1cncc(O)c1)=O)CC2 CC1CCCCC1OCC(=O)NCC1(NC(C2CCC2C#N)=O)CCCC1 N1(C(C2N(C(C)=O)CSC2)=O)CCC(C)C(N(C(=O)CC2CNC(=O)O2)C)C1 CC1(C(=O)NC2CC(F)(CNC(=O)CCCn3ccnc3)C2)CCCCCCC1 N1(C(Cc2scc(C)c2)=O)CC2(CCCN(C(C3CC3C3CC(F)(F)C3)=O)C2)C1 c1(N2C(CCNC(Cc3cnc(C)o3)=O)CSCC2)cnc(C#N)c(C#N)n1 c1(CC)c(C(=O)NCC2CCN2C(C2CC2CC)=O)nnn1CC CCCC(C)(CCC)C(=O)N1CC(NC(C2CCN(C3CC3)C2=O)=O)C(C)C1 Cc1ccc2nc(NCc3c[nH]c4cc(OC(F)(F)F)ccc34)ccc2c1 C(=O)(C1CCCn2nccc21)N1CC(NC(c2cc(F)ccc2F)=O)C1 N1(C(c2csc(C)c2C)=O)CCC2CCCC12C(N1CCSC(C)C1C)=O C#Cc1cnn(C)c1C(N1CC2CC1CN2C(=O)Cn1nnc(C2CC2)n1)=O c1(C(N2CC(OC)(CNC(=O)CSC)C2)=O)sc(C2CC2)nc1C C1(O)(CC)CN(C(=O)C=CC(c2ccccc2)=O)C1.C(CC=O)N(CC=C)C C1(C)(C(=O)NC2CC(NC(CC=CC(C)(C)C)=O)C2)Cc2ccccc2C1 c1(CC)nc(Cl)c(C(C)C)c(=NC(C2CCN(C(=O)C(O)COC)CC2)CC)[nH]1 c1(C(C)(F)F)ccc(C(=O)NCCN(C(=O)C(C)(C)C2CC2)CC)cc1 N1(C(CC=CC=C)=O)CCCC(CO)(NC(=O)C=C2CCC2)C1 C1(C(=O)NC2CN(C(CC(C)(C)F)=O)CC23CC3)CCc2nccn2C1 CCC(C)(CNC(=O)CC(C)(C)C#N)C(=O)N(C)CCC1CCCO1 c1(N(CC)CC2CCN(C(c3cnco3)=O)CC2)ncc(Br)c(C)n1 c1(C(=O)NC2C(CNC(=O)CC3CCCOC3)C2)ccc(N2CCCCC2)cc1 c1(CC)ncc(C(=O)NCC(C)CNC(C2(C)COC(=O)C2)=O)c(C)n1 C=CC(CCC)CC(=O)N1CCCC(CCNC(=O)CCOCC(F)(F)F)C1 c1(CC)ccc(C(=O)NCC2CC2)c(Cl)c1.n1(CC=O)cc(Br)c(C)n1 Cc1cc(C(=O)N)c(O)nn1.C1(C)(C(N2CC(O)(C(C)(C)C)C2)=O)CC=CCC1 C1(C(=O)NC2CCN(c3cc(C(F)F)ncn3)CC2O)CCC(C2CCCO2)O1 N1(C(C(C(C)NC(c2ncccn2)=O)C)=O)CCOc2ccccc21 c1(C(=O)OC(C)(C)C)ccc(-c2cncc(CO)c2)cn1 c1(C(N2CCC(C)(CNC(CN(CCOC)C)=O)C2)=O)ccnn1C1CCCC1 c1(OC)ccc([N+](=O)[O-])c(-c2noc(C(C)OC(c3ccccc3)=O)n2)n1 CC(C)(O)CCC(=O)N1CC(c2cn(C3CCCC3)nn2)C1 C(CC(C(C)(C)C)NC(=O)C(C)n1cncn1)N(C(Cc1cnc(C)[nH]1)=O)C c1(C(=O)NCCNC(Cc2n(C(C)C)cnn2)=O)cc([N+](=O)[O-])ncc1Br c1(C(=O)OC)cccc(C(N2CC3CC3(CNC)C2)=O)c1.c1cc(C)nn1C Cn1c(C(N2CC3CC2C3NC(c2csc(O)n2)=O)=O)cc(Cl)c1Cl N#CC1CCN(C(=O)CNC(=O)CCc2ccncn2)C1.C1(C(N)=O)CCCCC1 Cc1c(-c2ccccc2)nn(C)c1NC(=O)CC1C(N)CC1O N1(C(C(C)CC2CC2)=O)CC(NC(c2cccc(-c3cscn3)c2)=O)C(O)C1 Cc1cc(=NCC23CC(NC(C4CC(F)C4)=O)(C2)C(C)O3)[nH]c(C2CC2)n1 C(N=c1[nH]cnc2ccc(Cl)cc12)c1cn(CC(COC)O)nn1 N1(CC(=O)NC2(CCC)CCN(C(=O)CCCSC)CC2)CCn2ccnc2C1 Cc1cc(F)c(NC(=O)NC(C(F)(F)F)C2CCCOC2)cc1I Cc1[nH]c(C#N)cc1C(=O)NCC1CC(F)C1.C1(C=O)CC1C1CCCC1.C C(=O)(CCS(N)(=O)=O)NC1C(C(=O)NCC2(S(C)=O)CC2)CC1 C1(C(=O)OC)(CN(C)C(C2CCS(=O)CC2)=O)CCCCO1 C1(N(C(C2N(C(C)C)CCC2)=O)C)CCN(C(c2coc(C(F)(F)F)c2)=O)CC1 C(=O)(C(C)(CC)CO)NC(C(=O)NCc1c(CC)ocn1)Cc1cnc[nH]1 Cc1ncccc1CCC(=O)NC(C1CCCN1C(=O)CCCc1cc[nH]n1)C Cc1cnn(C)c1CC(=O)NC1CCN(C(c2ncccn2)=O)CC1 C1(CCC)CN(C(C2CN(CC)CCO2)=O)CCN1C(=O)CN(C)CCOC c1(OC)c(C(=O)NC2C3CCN(C(=O)C(CO)N(C)C)C23)sc(Cl)c1Cl C1(C(N(C2CC(C(=O)NCC(C)OC)C2)C)=O)CC2C=CC1O2 CCC(CCCC(=O)NCC1(C)CCCS1)NC(c1ncn(CC)n1)=O N1(C(C(COCC)n2cc(-c3csnc3C)nn2)=O)CCC2(CCC2)C1 c1(CN(C)CC2CCN(C(c3ccc(Cl)s3)=O)C2)ccc(Cl)s1 C1(C(N2C(C(C)(C)NC(C3CC=C(C)CC3)=O)CCC2)=O)CNC(=O)CC1(C)C N1(C(c2cn(C)c(Br)c2)=O)CC(NC(=O)CNC=O)C(N=[N+]=[N-])C1 c1(C(=O)NCCCN(C(C2(C(C)C)CC2)=O)C)cnc(Br)s1 c1(CN(CC)CC)cccc(C(=O)N(C)Cc2ncc[nH]2)c1 C1(NC(=O)CCCn2cncn2)(CF)CCN(C(=O)CC2(C3CC3)CC2)C1 C1(C(N2CC3C(CNC(C(=O)N(C)C)=O)(C3)C2)=O)CCCCC(C)(C)C1 Cc1nc(-c2cccs2)sc1C(=O)NC(C)(C)CCCNC(=O)C(F)C(C)C N1(C(C(N2CCSCC2)C)=O)CCC(CO)C(NC(C2CCC(F)(F)CC2)=O)C1 c1(C(N2CC(C(C)C)N(C(C3CCCS3)=O)CC2)=O)cccc2c1OCCO2 CC(CCC(=O)NC(C)C(O)C(F)F)NC(c1[nH]ccc1C1CC1)=O CC1C(NC(=O)NCC2CCCN2c2ccccc2)CC1(F)F C(C)CC(F)(F)F.C(=O)C(C)Cn1ccc(C)n1.C1(CC=O)CC1.CC=O.N CC(C)CC(F)C(=O)N1CCN(C(C2CC(n3cnnc3)C2)=O)C(C)C1 C(=O)(C1NCCc2c(C)cccc21)NCc1cc(CC)on1 c1(C(=O)NCCC(CNC(CN(CC)CC)=O)O)cc(Cl)ncc1NC Cc1cc(Cl)c(C(=O)NC2CCCC2NC(=O)Cn2nc(C)c(Cl)c2C)cc1C C(=O)(CS(=O)(=O)C1CC1)NCCN(C(=O)CCc1cccc(O)c1)C N#Cc1cncc(CNC(=O)C(=O)NC2CCN(c3ccc(F)c(Cl)c3)C2=O)c1 C1(C=O)CCCCC(=O)C1.c1(OC)cncc(CNC(=O)C)c1.C(C)(C)C c1(CC)cccc2c(C(N3CCC(CN(C)C(c4cnc[nH]4)=O)C3)=O)c[nH]c12 c1(OC(C)C)ccccc1.C12CC1CN(C(=O)CN(C)C(N)=O)C2.CC=O.O C1(CNC(=O)COCCF)C2CN(C(c3csc(Cl)n3)=O)CC12 C1(CNC(C(C)C2CC2)=O)CC(F)CN1C(=O)COCc1cccnc1 C1(CNC(CCNC(c2nc(CCC)oc2)=O)=O)OC(=O)CC1(C)C C(=O)(CCCCCNC(c1cc(F)ccn1)CO)OCC N1(C(Cn2cnc(=N)[nH]2)=O)CCC(C(=O)NCCn2cnccc2=O)=C(F)C1 c1(S(C)(=O)=O)ccc(N(C(=O)NCCO[Si](C)(C)C)C2CC2)cc1 C(=O)(CC(C(=O)NC1CC(C)C1)c1ccccc1)NC.C(=O)(C)N.C(C)=O Cc1csc2cccc(C(=O)N(C(C)CCNC(c3csc(O)n3)=O)C)c12 c1(C(N(CC(C)NC(CC(n2c(C)cc(C)n2)C)=O)C)=O)ccc2c(c1)CCC2 N1(C(C2C(C(=O)OCC)C2(C)C)=O)CC2CCC1CN2C(=O)CCC(C)CC C12(C(=O)NCCN3CCC(OC)C3)CC(CN(C(c3nc[nH]n3)=O)C1)C2 N1(CC2(C(=O)NC3CCC(n4cc(-c5ccns5)nn4)C3)CC2)CCCOCC1 c1(CC(C2CC2)NCCCC(=C)C)cccc(OC)c1 C1(NC(c2c(C)ncn2O)=O)CC2CCC1CN2C(=O)C1=CC(C)(C)C1 C1(CNC(CCC)=O)CCCC2(CN(C(c3nc[nH]c4ncc(Br)c3-4)=O)C2)O1 CCCCCCN(C)C(C1CCOC1CNC(=O)CC1CCSC1)=O c1(C(=O)NC2CN(C(C(CCCC)N(C)C)=O)C2)oc2ccccc2c1CO N1(C(C(C=C)O)=O)CC2CCC1C(NC(=O)CN=S(C)(C)=O)C2 C(=O)(C1=CC(C)(C)C1)NC(CC#C)C(=O)NC(C)Cc1nc[nH]n1 C1(C(=O)NCC(C)(CNC(C2CCCOC2)=O)OC)(COC)CCOCC1 CC1CC(CNC(c2nc(=N)cc[nH]2)=O)CCN1C(=O)CCS(C)(=O)=O CC1(C)CC(CO)N(C(C2CCN2C(c2cncc(O)c2)=O)=O)C1 N1(C(C(C2CCC2)OCC)=O)CCC(F)(CNC(c2ccccc2)=O)C1.C Cc1cn2cccc(NC(C3CC34CCN(Cc3sccc3C)CC4)=O)c2n1 c1(C(=O)N)ccc2c(c1)CCO2.Cc1coc(C2CC2)c1C(=O)NC(C)CCC C1(OC)COC2CN(C(=O)Cc3ccnc(OC4CCOC4)c3)CC12 N#Cc1ccc(C(=O)NC(C)C2CCC2)o1.C1CCCCC1.C(=O)C=CC.N C1(C(=O)NC(C(C)C)CNC(=O)C=Cc2cscn2)CC1C1CCC1 CC(CC(C(=O)NCc1ccccc1)N1CCOC(C(N)=O)C1)c1ccccc1 c1(CC(=O)NCC2CC(C(=O)Nc3ccccc3O)C2)c(F)cccc1F c1(C(=O)NC2C3CCN(C(C=Cc4scc(C)n4)=O)C32)ccc2c(c1)nnn2C C1(NC(COC2(C)CN(C(c3ccc(C#C)cn3)=O)C2)=O)C(=O)OC2CCCC12 C1(COC)CCN(C(=O)Cn2cc(C3CC3)nn2)CC1.C(=O)CC=C(Cl)Cl.C C1(NC(c2nnn(C(C)(C)C)n2)=O)CCOCC1.c1(C2(C=O)CC2)ccno1.C C=CC1(C(=O)NCC2CCCC2)CCN(C(=O)C=Cc2cc(C)no2)CC1.O C(c1cncc(O)c1)=CC(=O)N(CCNC(Cc1nc(C)sc1)=O)C1CC1 C1(CC)CN(C(=O)CC2CCN(C(C3CC3c3ccco3)=O)CC2)CC(=O)N1 CCCCCCCC(=O)NCCN(C)C(c1cnc(OCC(C)C)c(Cl)c1)=O C1(CCNC(c2cscc2Cl)=O)CCCN(C(=O)Cn2ncnn2)C1 N1(CCC)CCC(O)(NC(C)C(=O)N(c2ccc(O)nc2)C)C1 N(C(=NCCCC(C)(C)C)NC(C1CCOC1)C)Cc1c(C)nns1 C1(C(=O)NC2(CNC(=O)CCC3CC(F)(F)C3)CC2)CC12CCSCC2 C1(C(=O)N)OC(C)(C)OC1(C)C.c1(C(C)C)ncc(C(=O)NCC(C)CO)n1C C1(C2CCN(C(c3cn(C)c(O)n3)=O)CC2)(NC(c2n(C)nc(C)c2Cl)=O)CC1 C1(NC(C(C2CCOC2)OC)=O)CCN(C(=O)C(F)(F)CC2CC2)CC1C N1(C(c2c(C)cccn2)=O)CCC(F)C(NC(=O)CN(C)C(c2cccs2)=O)C1 c1(C(=O)NCC(=O)NCC(N2C(C(CC)C)CCC2)=O)ncncc1Cl Cc1cc(=O)n(C)cc1C(=O)NC(C)CCCc1cccnc1 C(C)(C(=O)N(Cc1ccc(C)o1)OC)C1CC(NC(C(C)OCC=C)=O)C1 c1(SC(C)C(=O)N(C)CCN(C(c2cnc[nH]2)=O)C(C)C)ccccc1 Cn1c(C(=O)NC2CC(F)(C)C2)cccc1=O.C1(O)(C(C(=O)N)F)CCCC1 CC(C(=O)N1CCCC(C(C)(C)NC(=O)COCc2ccncc2)C1)C(C)O n1(CC)cc(NC(C2(C)CCN(C(c3ccsc3OC)=O)CC2)=O)ccc1=O C1(C)(CNC(CC2C(C)(C)C2)=O)CCCN(C(C2(N3CCCC3)CCC2)=O)C1 N1(C(C2CCC(OC)C2)=O)CCC(C(CO)NC(=O)CCc2ccncc2)CC1 C1(CNC(CC=CC)=O)CN(C(=O)C(C)n2ccnc2)CC(C)(C)C1 C(CC(C)(C)C(=O)NCCC1(C)CCCO1)NC(c1n(CC)ccc1)=O N1(C(c2c(CC)non2)=O)CC2CC1C2NC(=O)CC(C)C1CCCC1 N1(C(C#CCNC(c2ccc(C)cc2O)=O)=O)CCCC2CCCC12 c1(OC)c[nH]c(C(=O)N(C)CC2CCCN2C(=O)C(C)NC(C)=O)cc1=O CC1(C)CCCN(c2ccnc(NCc3ccc(O)c(F)c3)n2)C1 C1(C)(C(C)NC(CNC(=O)OC(C)(C)C)C2CCC2)CCCO1 c1(C(=O)NCC2C=CC(NC(=O)C#CC3CCCO3)C2)cc2cc(F)ccc2[nH]1 CC(C(CO)NC(=O)CCc1cnc(O)[nH]1)NC(=O)CC1COCCO1 C1(CNC(CCC=C)=O)(CNC(=O)CC2CNC(=O)C2)CC12CCC2 N1(C(COc2ccc(OC)cc2)=O)CCC(F)CC1.C1(CC(=O)N)CC2CC2C1 C(=O)(CCC1CCC1)NC1C(CC(=O)OC)C1.C1(C(=O)N)CN(C)C1 C1(C)(C(N(CCCC)CCCC)=O)CC(OC)CN1C(=O)CCNC(=O)N C=CCN=C(NCCC1CCOC1C)NCC1COCCOC1 CCC(CN=c1[nH]c2c(c(=NC3CCOCC3F)[nH]1)COC2)N(C)C c1(CC)cc(C(N2CCCC(C)(NC(c3cnc(C4CC4)o3)=O)C2)=O)ccc1O C(C(C(=O)NC(C)Cc1cccnc1)n1cc(CC2CCC2)nn1)OCC C=CCC(F)(F)C(=O)N(C)CCN1CCN(C(C2(SC)CC(O)C2)=O)CC1 c1(C(C)C(=O)N(C(C)CNC(=O)C=Cc2ccsc2)C)cccc(F)c1 c1(C(C(=O)NC2C(NC(C3CC3(F)F)=O)COCC2)(F)F)cc(F)ccc1F NS(=O)(=O)CCCC(=O)NCCC1CSCCN1C(c1cncc(C(N)=O)c1)=O C1CCN(C(=O)C=CCN2CCCC2)CC1(C)C.CN1CC(C)(C)CC1C=O.N c1(C2CC(=O)NC2)nnc(CC2CCCO2)n1CCCOCC1CC1 c1(C(N(CCCNC(=O)C(C)(F)CC)CC)=O)cnc(C)cc1Cl n1(C(C)C)ncc2c(NCc3ccnc(Br)c3)[nH]c(=NCCCCCF)nc12 c1(OC)ccc(NC(C2CC2NC(c2ncc(Cl)cc2F)=O)=O)cc1O c1(C(N(CCCN(C(=O)Cc2csc(=N)[nH]2)C)C)=O)cnc2[nH]cnc2c1 c1(CC)ccc(F)c(C(=O)N(CC(C)NC(C2CCC(C)(C)O2)=O)C)c1 N1(C(C2(CO)COC2)=O)CC2CN(C(=O)Cn3cc(OC)nn3)CCC2(CO)C1 c1(CC(C)N(C)CC2CCNC(C)(C)C2)cc2ccccc2o1 N1(C(C(c2cnccn2)C)=O)CC(C)(NC(c2cc(Br)c[nH]2)=O)C1 CC1(C)C2CCC(C2)C1C(N1CCN(c2ccc(F)cc2C#N)CC1)=O c1(C(CF)NC(CONC(C2C(C(C)(C)C)CC2)=O)=O)ccccc1 Cc1cc(F)c(C(=O)NCC(n2cc(-c3c[nH]nc3C(=O)O)nn2)C)cc1C C1(C(N2CC(C(C)(C)O)(CNC(C)=O)C2)=O)CC2CCC1O2 C1(NC(CNC(CNC(C2(C)C(C)OCC2)=O)=O)=O)CN2CCC1(C)CC2 C1(C(C)NC(=O)CCCN2CCCC2)CCCN(C(C2CC(N(C)C)C2)=O)C1 C1(F)(CNC(CCCN(C(C)=O)C)=O)CCCN(C(=O)COCCCF)C1 c1(C(N2CCC(C)N(C(c3ccc(O)nn3)=O)CC2)=O)cccc2nc(Cl)cn12 C12(C(=O)NC3CC(CNC(=O)Cc4ccco4)C3)CCCN(CC1)C2 C1(CNC(c2ccc(N(C)C)nn2)=O)CN(C(=O)CCC(C)(F)F)CCC1(C)C n1(CC)cc(NC(C2CN(C(=O)C(C)C)CCO2)=O)ccc1=O O=S(=O)(CC1(CCl)CCC1)NCCc1nccs1 c1(C(N(CCC(=O)NC2CC(C)(OC)C2)CCC)=O)sc2nnc(S)n2c1C C(=O)(CCCC(F)(F)F)NCCC(C)NC(c1cc(-c2ccco2)no1)=O C1(NC(=O)NCC(C2CCCC2)OCC)CC2CCC(C1)N2CC C12(C(=O)NC3(C)CCC3)CCN(C(=O)CCC3OCCO3)CCC1C2 C12(COC)CC(CN1C(=O)CCC1CC1(Cl)Cl)C2.C(=O)CCC1CC1.N c1(N(CCNC(C)=O)C)cc(C)c(S(=O)(=O)N=c2[nH]ccnc2Cl)cc1O CCC(C)C(O)CC(=O)NC1CC2CC(C1)N(C(=O)C(F)C(C)(F)F)C2 N1(C(c2cnc(C#N)s2)=O)CCCC(CNC(=O)C(C2CCCO2)C2CC2)CC1 CC1C(NC(=O)Cn2cc(C)nn2)C(C)CCN1C(c1cc(=O)cc(Cl)[nH]1)=O c1(OC)cccc(F)c1C(=O)NC12COC(C1)C2.C1(CC=O)CCCN1C.C N1(C(C2(C)CSC2)=O)CCCC(C)(CNC(c2ncn(-c3ccccc3)n2)=O)C1 C1(CC)C(NC(c2cccn2C)=O)CCN1C(=O)CC1CSCCS1 C1(CNC(CCn2c(C)ncc2)=O)CCCC(NC(c2ccn(C(C)C)n2)=O)C1 C12(C(N(CCCO)CC#C)=O)CCN(C(c3cc4occc4[nH]3)=O)CCC1C2 c1(NC(CN(C)C)CCO)ccnc(N(C)CC2(C(F)(F)F)CCC2)n1 Cc1nocc1CC(=O)N(CCCN(C)C)CC.C(=O)(CCC)N.C(C)(C)C C1(OC)CC(CNC(=O)CC(C)O)N(C(c2cc(CF)on2)=O)C1 C1(C(=O)NCCCN(C(=O)CCCCN2CCCC2)C)CCCC2(C1)CC2(F)F c1(OC)ccc(O)c(OCC(=O)OCC(c2ncon2)C)c1 N1(C(C2CCCOC2)=O)CC2CCCC(C1)N2C(c1cc(O)cc(O)n1)=O C(c1ccccc1)=C(C(=O)NCC(C)N(C(CN(C1CC1)CC)=O)C)OC CCC(C)C(O)CC(=O)N1CCCC(CC(N2CC3CC3(C(N)=O)C2)=O)C1 C1(CNC(C2CCC(NC(C3(SC)CCC3)=O)C2)=O)CCCCCCC1 N=c1[nH]cc(CNCC(O)Cc2ccccc2Br)c(=N)[nH]1 c1(NC(CC(C)(C)OC)=O)cc(C(F)(F)F)ncc1I C1(C(N2C(CCNC(C(CC#C)(C)C)=O)CCCC2)=O)CCc2cn(C)nc2C1 N#Cc1cc(NC(C2CCN(Cc3cccc4c3CCC4)CC2O)=O)cc(F)c1 N1(C(CC2CC(OC)C2)=O)CCC(C2CC(NC(=O)Cc3nn(C)cc3Cl)C2)C1 N1(C(CCc2cc(C)on2)=O)CC(CNC(=O)CC(C)(C)O)C2(CC2)C1 CCCCN=C(NCC1CCC(C(N)=O)CC1)NCC1(SC)CCN(C)CC1 N1(C(C2N(C(C)=O)CSC2)=O)CCC(CNC(C2CC2F)=O)C(F)(F)CC1 C1(N(C)C)CCCCC1C(=O)NCC1CC1NC(=O)Cc1ccccc1.C C1(CNC(C2N(CCC)CCCC2)=O)(NC(c2ccccc2)=O)CCCCC1C C1(NC(C2(n3cc(C4N(C(C)=O)CC4)nn3)CC2)=O)CCN(C)C(=O)C1 N1(C(=O)NC(C2CCOC2)C#C)CCC(COC(C)=O)CC1 CC(C)CCCC(=O)N1CC2C(CNC(C3CCCC3C(F)(F)F)=O)C2C1 S(=O)(=O)(c1cccc(Br)c1Cl)NC(=O)CCc1cc(Br)c(F)cc1F c1(OCC)ccc2cc(NCCCCOC(C)C)oc2c1 CCCC(C(=O)OC)C(=O)N1CCCC(CNC(=O)CC2OCCC2(C)C)C1 c1(NC(C2C(C)(C)CN(C(=O)CN3CC4CC4C3)C2)=O)ccc2nccn2c1 N1(C(C(N2CCCCCC2)C)=O)CCC(CO)(CNC(C2CCCN2C)=O)CC1 c1(C(N(CCC(C)NC(c2occ(C)c2C)=O)C)=O)ccn2nccc2n1 C1(C(CC)C)CCN(C(=O)CN2CCC(C)(c3ccc(OC)cc3)C2)CC1 C1(NC(C(N(C)C)C2CC2)=O)CCC2(CC1)CN(C(c1cnn[nH]1)=O)CCO2 N1(C(c2cc(CC)nc(O)c2)=O)CCC2(CCN(C(=O)C(C)(C)OC)CC2)C1 CCCC(C(=O)NC1CC2(C1)CC2NC(=O)CC1CCC2(CC1)CC2)C(C)C CCCC(CCCNC(=O)Cc1cc(Cl)cc(Cl)c1)NC(=O)Cc1cnn(C)c1 N(C1CCc2ccc(Cl)nc21)C(C(C(C)C)OC)c1n(CC(=C)C)nnn1 CCCC(C)NC(=O)CSCc1ccccn1.C(=O)(C(C)Cc1cnc[nH]1)N c1(C(=O)NCC2N(C(CCSCC)=O)CCC(C)C2)ccc2c(O)nccc2n1 c1(NC2CC(CNC(C3CCN(CC(C)C)CC3)=O)C2)cnc(C#N)cn1 N1(C(C(C)(CO)OC)=O)CC2CCCCC2(NC(c2cc3cccnc3s2)=O)C1 c1(-n2cc(CC3(NC(c4coc(Cl)c4)=O)CCC3)nn2)cc(F)cc(Br)c1 N1(C(Cn2ccc(C)n2)=O)CCC2CCN(C(C3(S(C)(=O)=O)CCC3)=O)CC2C1 C1(CC)(CC)CC(NC(=O)C2=CCCS2)CN1C(C1CCC(=O)NC1)=O c12cccc(c1C)NC2C1CC1.n1(CCOC)cccn1.C1CCCC1C.N C(C(=O)NC)C(C)C.C1CCN(C(=O)Cn2cnnc2)C1.C(=O)(OCC)N C12(CNC(CC(=O)OC)=O)CC(C1)C(NC(=O)CCCN=[N+]=[N-])CO2 N1(C(CNS(N)(=O)=O)=O)C2CCC1CC(F)(C)C2.C(=O)(C(F)n1cccn1)N CC(C)CC(C)(O)C(=O)N1CCC(CNC(c2cnc(C(F)F)nc2)=O)C1 CCCCC(CC)CC(=O)NCC1(NC(C2CC(=O)C2C)=O)CCCCCC1 N1(C(c2c(CC)ncs2)=O)C(C(=O)NCC(C)OCCO)CC2CCCC12 CC1(C)CCC(C)(NC(C2(CO)CCN(C(C3CCCS3)=O)C2)=O)C1 CCCC(CCC)C(=O)NC1CCCC1NC(c1ccc(N)c(Cl)n1)=O N1(C(c2cc(OCC)ncc2)=O)CCC2CCCC(C1)N2C(c1cc(Cl)c[nH]1)=O c1(C(=O)NCCCN(C)C(C2CC2c2cccc(O)c2)=O)cccc2scnc12 C1(C(CNC(c2n(C)ccn2)=O)(C)O)CCCN(C(c2cccs2)=O)C1 N1(C(c2cnc(OC)nc2)=O)CCOCCC1C(=O)N(C1CCC(F)(F)C1)C c1(SC)cccc(CC(=O)NC)c1.c1(C=O)cn(C(C)(C)C)cn1.C1CCC1 N1(C(C2(CC#C)CC2)=O)CCC2C(C(N3CCSCC3)=O)C2C1 CC(C)C(C(=O)N1CCC(C)C1CNC(c1cnco1)=O)N1CCCCC1 C=CC1OCCCC1C(=O)NCC1CCCN(C(c2cc(CCOC)on2)=O)C1 c1(NC(C2C(C(N(CCCCO)CC)=O)C2)=O)nnc(Cl)s1 N1(C(CS(CC)(=O)=O)=O)CC2CC(N=c3c(C)c[nH]cc3[N+](=O)[O-])C2C1 C#CCCCCCCCC(=O)N1C(CNC(=O)CCC2CC2C)CC1C c1(C(=O)NC2C(C)CSC2)ccc2c(c1)oc1ccccc21 N1(C(C(=O)N(C)C)=O)CCN(C(=O)COc2ccccc2)C(CCN(C)C)C1 C1(C(=O)NCC(C)C)CN(C(=O)C(C)(C)C2CCOC2)CCN1C c1(OC)cccc2c1OC(C(=O)NCCNC(c1csc3cncn13)=O)C2 C(=O)(CCS(C)(=O)=O)OC.C1(n2cc(C34CN(C3)C4=O)nn2)CN(C)CCC1O c1(OC)c[nH]c(C(=O)NC2(C)CCCN(C(=O)C(C)(CO)OC)C2)cc1=O N1(C(CN(C(CC2CCN(C)C2=O)=O)C2CCC2)=O)CC2CCC(CC2)C1 Cc1occc1C(N1CC(CNC(=O)C(C)(C)C2(O)CCOC2)C1)=O C1(CC(=O)NC2CC(CNC(=O)C(Cl)=CCl)C2)CCCC(C(F)(F)F)O1 N1(C(Cn2c(C)nc(C)n2)=O)CC(NC(C2CCCNC2=O)=O)CC1(C)C C12(CNC(c3ccoc3Br)=O)CCCCC1N(C(=O)CN1CSCCSC1)CC2 c1(CC)ccc(C(N2CCC(C)(CNC(C3CC3C)=O)C2)=O)cc1Cl c1(CCC(=O)NC(CCCCNC(C=CC=CCC)=O)C)n[nH]c2c1CCCC2 Cc1cc(C(=O)NC2CC2CNC(=O)C(C)Oc2cccnc2)n[nH]1 c1(OC)cc(C)sc1C(=O)NCCCCC(C)NC(=O)C(c1ccccc1)C N12CCC(F)(CC1)C2=O.N1(C(C2CCCCC2O)=O)CCCN(CCO)CC1 C12(C(NC3CCN(C(=O)C(O)CC)C3)=O)CCC(F)(CC1)CC2.C(C)=O.C N1(C(c2c(C)nc(CCC)o2)=O)CCN(C(C2(O)CCCCC2)=O)CC(C)(F)C1 c1(CC)c(C(=O)NCC(CC(=O)NC(C)C(=O)OC)OC)ccn1C c1(C=O)cc(O)c2c(cnn2C)c1.C(CCC(=O)NC12CC(C)(C1)C2)SC.N N1(C(C2CCC(CNC(C(C)CN(C)C)=O)CC2)=O)CCCCCCC1 C1(C(N2C3(CNC(C(CC)C(C)C)=O)CC(C2)C3)=O)CC(c2ccncc2)=NO1 C1(NC(C2ON=C(CC)C2)=O)CCCCCN(C(=O)C(CO)C(F)(F)F)C1 C1(NC(C(C)N(C(C)=O)C)=O)COCCN(C(C2CC(S(C)(=O)=O)C2)=O)C1 C1(C=O)CCCC12OCCO2.Cc1cc(C)n(CCC(=O)NCC2CC2C)n1.N C=CC(C)CC(=O)NCC(CC)(CC)NC(c1cn(CC)nc1C1CC1)=O C1(NC(c2ccc(CC)s2)=O)CN(C(C2CCCCC2O)=O)CC1C C1(NC(CC(CC)(C)C)=O)CN(C(=O)Cn2cnccc2=O)C2(CCC2)C1 N1(C(CC(C(C)C)O)=O)CCC2CN(C(=O)CNC=O)CC12 N1(C(c2cc(C)n(C)c2C)=O)CC2OCC(NC(=O)CC(C)C(C)C)C2C1 C1(CNC(CN(C)C2CC2)=O)CCC(NC(c2cccnn2)=O)C1 N(C1CCOc2cc(Br)ccc21)C(c1cc(Cl)c(F)c(Cl)c1)C N1(C(CCN(C(C(CC)NC(C)=O)=O)CC(C)C)=O)CCN(C(C)=O)CC1 c1(C(=O)NC2C(NC(C(CCCCC)(C)C)=O)CC2)cc(C)nc2c1CCCC2 N1(C(C2(C)CSC2)=O)CCC(O)(CNC(c2c[nH]nc2C2CC2)=O)CC1 C1(OC)CC(NC(C2(F)CC2)=O)CN(C(c2ccc(Br)c(N)n2)=O)C1 C(=O)(CCC(=O)N(C)C)N(CC(C)CNC(=O)CC=O)CCC.C1CC1.N n1(CC)ccnc1C1OCCC1CN=C(NCc1cnn(CC)c1)NCC(F)F c1(C(=O)NCCC2OCCN(C(C(CC)O)=O)C2)nccc2n[nH]cc12 C1(C(F)(F)F)(C=O)CCCCO1.Cc1ccoc1CC(=O)N(CCC)C1CC1.N N1(C(c2c(C)nn(C)c2N)=O)CC2(CCC(NC(=O)C(O)CC[S+](C)C)CC2)C1 CCC(C)C(C)C(=O)NCC1CCCC1NC(C1CC2CCC(C1)C2)=O C(C(=O)NCCCNC(c1cc[nH]n1)=O)(C1CCCC1)OCC.C1CCCC1 N1(C(C(C)(C(F)(F)F)c2ccccc2)=O)CCN2CC3(CC3)CC2C1 N(C1CCCn2ncnc21)C(C1CN(C(c2c(C)noc2N)=O)CC1C1CC1)=O C12(NC(=O)CC3CCCCO3)CC1CN(C(c1[nH]ccc1-c1ccccc1)=O)C2 N1(C(C(n2ncc(C)c2)C)=O)CCCCC1CC(N1CCC(F)(CN(C)C)C1)=O Nc1ccc(F)c(C(=O)NC2CCN(C(c3cc(Cl)c[nH]3)=O)C2)c1 C(=O)(CC(C(F)(F)F)n1cccn1)N(C)CC1CCN(C(=O)Cn2cccc2)C1 C1(C(N(C)CCC2CCCO2)=O)CC1C1CN(C(c2cc(C#N)c[nH]2)=O)C1 N1(C(c2c(CC)n(-c3cccc(Cl)c3)nn2)=O)CCC(OC)C12CCC2 C1(NC(C2CC(C)(CC)C2)=O)CCCCC1.C(=O)(CC)N.C1(C=O)CCC1 C(=O)CCCC(C)(C)C.Cc1nn(CC2CC2)c(C)c1CC(=O)N.C1CC1.C C1(CCNC(c2cc(C)ncc2)=O)CN(C(=O)CCc2cnoc2)CC(C)O1 N1(C(CCC=CCC=C)=O)CCN(C(=O)CCC(=C)Cl)C(c2cccnc2)C1 C(=O)(C1=CCC(C)(C)CC1)NC1(CCOC)CCN(C(=O)Cn2cnnn2)C1 C1(NC(=O)C(C2CCOCC2)O)CC2CCC1CN2C(=O)CCc1cocn1 C1(OC(C)C(=O)N2CC(N(C)C(C3CNC(=O)C3)=O)C2)CCCCC1 C(C(C)(O)CC(=O)NCC(O)CC(=O)NCC(N1CCCC1)C)OC Cc1cnc2ccc(C(N3CC4CC3C4NC(=O)CC3CC(C)C3)=O)cn12 C(=O)(C(C)(C)S(C)(=O)=O)N1C(CNC(c2c(C)sc(Cl)n2)=O)CC1 c1(OC(C)=O)ccccc1C(=O)NC(C)(C)C.C12CC(C1)NC(=O)C2 N1(C(c2c(C)oc(CO)c2)=O)CC2CCCC2(NC(c2cc(=N)[nH]c(Cl)n2)=O)C1 C1(NC(COCCOCC)=O)CCCC1C(=O)N.CCC(C)N(C)CCO C(N=c1[nH]cncc1OC)C1CCC(NC(CS(CCOC)(=O)=O)=O)C1 c1(C(=O)NC2C(CNc3ncc(C)c(O)n3)CCC2)cccc2cc(O)ncc12 C1(C(=O)NC2CCCC(SCC)C2)CC12CCOc1ccccc12 C1(CC(=O)NC2CN(C(c3cc(OC)no3)=O)C2)CCC(=O)NC1=O CC1CC(NC(=O)CC2CC(=O)NC2=O)CCN1C(=O)CCc1cncnc1 CC1CC(C)CN(C(C2CC3CCCC3C2)=O)C1.C1(C)(C=O)C(C)(C)C1(C)C.N C=CCCCCC(=O)NC(CNC(C1CN(C2COC2)C1)=O)C1CCC1 C1(C(N(CC(CC)(O)CC)C)=O)N(C(c2ccc(C)nc2C)=O)CCCC1(C)C C1(C=O)CCC2(C1)CC2(F)F.C(=O)(C(C)(C)C(=O)N1CCC1)O.CC.CC N1(C(c2ccc(CCC)s2)=O)CCC(NC(=O)CCc2cn[nH]c2)C1C C1(NC(=O)Cc2cnsc2)CC2CCCC(C1)N2C(C12CCC(F)C1CC2)=O C(=O)(C(O)CCC(C)C)NCCN(C(C1CCCCS1)=O)CC c1(C(=O)NC2CN(C(C=Cc3cccc(Cl)c3)=O)CC2O)cn2ccccc2n1 c1(OCCOC)ccccc1C(=O)N.C(C1CCOCC1)=CC=O.CC(C)C C1(NC(c2c(C)nn(CC)c2Cl)=O)CC2CC(C1)N(C(c1cc(O)no1)=O)C2 c1(C(=O)NC(CC)CN(C)C(c2cnc(O)s2)=O)ccncc1C(=O)OC Cc1nc(Cl)ccc1C(=O)NC(C)CC1CCN(C(=O)CSC(=N)N)CC1 c1(NC(CC(CC)O)=O)n[nH]c2ccc(-c3cnn(-c4cccnc4)c3)cc12 N1(C(C=CC=CC)=O)CCCCC(C2CN(C(=O)C(CO)C(C)(C)C)C2)C1 C1(NC(CC)=O)COC2(C1)CN(C(=O)CC(C)C1CCCO1)C2 C12(CNCC3N(C(C4(O)CCCCC4)=O)CCC3)CC3CC(CC(C3)C1)C2 c1(C(=O)NCCNC(C(c2ccc(OC)cc2)CC)=O)cc2ccncc2s1 C1(NC(c2ccc(CO)s2)=O)CCC2(CCCN2C(=O)C=CBr)CC1 C1(C(=O)NC2C(CNC(C(C=C)O)=O)CC2)(CC2CCCC2)CCOCC1 N1(CC)CCCN(C(=O)C(CC(C)C)NC(c2cscc2NC)=O)CC1=O C1(CN(C)C(C2(F)CCOC2)=O)C2CN(C(c3cc(Cl)c(Br)[nH]3)=O)CC12 C(c1csc(C)n1)=CC=O.C1(CNC(C2C(C=C)C2)=O)CC(F)(C)C1 C=CCCCCC(=O)NCC(C(N1CCCC(CC(C)C)C1)=O)N(C)C C1(C)(C(N2CC(C(C)(C)O)(CNC(=O)C(C)n3ccnc3)C2)=O)CCCN1C n1(CCC)nc(C)c(C(=O)NCC(C)N(C)C(C2CCCC(C)(C)C2)=O)c1C C1(NC(CCC=C=C)=O)CCCCCN(C(c2ccnnc2)=O)C1 N1(C(c2cccc3sccc23)C(=O)NCCC)CCS(=O)(=O)C2CCCC12 c1(CC(=O)N(CC)CC)ccccc1.C(=O)C(F)=C1CCC1.C1CC1.C c1(C(C(=O)N)N(CCC)C)ccc(S(C)=O)cc1.C1(C(=O)OC)(C)CC1 c1(C(N(CCCN(C(C(C(C)O)(C)C)=O)C)C)=O)cccc2cccnc12 Cc1cnccc1C(=O)NC(C1CCN(C(=O)C(O)CCn2cncn2)C1)(C)C N1(C(C2C(C=C)OCC2)=O)CCOCC(NC(c2ccnc(CC)c2)=O)C1 N1(C(C)C)C(=O)COCC1C(=O)N(CCCCCNC(c1ccnc(O)c1)=O)C C(=O)(C(F)(F)C(F)(F)C(F)(F)F)NC1CCCN(C(C(C(C)(C)C)O)=O)C1 C(C(C(C)C)NC(C12CC(C1)C2)=O)OCC.C1(C=O)CC(F)(F)C1.N c1(OC)cccc(C(C)(C)CNC(=O)NC(c2cnn(C)c2C)C)n1 N1(C(C2CCC(=O)N2)=O)CCC(O)(CNC(=O)C(C2CCCCCC2)O)C1 C12(C(N(C3CN(C(C4CCSC4)=O)CC3F)C)=O)CCC(CC1)C2 C(=O)(N=c1[nH]oc2cccc(Cl)c12)N(CCn1ncc(C)c1)C C=CC1CCCN(C(=O)C(C2(C)CC2)NC(=O)CCOC2CCCC2)C1 CC1CN(C(C2CCCN2C=O)=O)CCC1NC(c1cn(CC(N)=O)nn1)=O C1(C(=O)OC)C2CCC1(C(=O)N(CC(C)NC(c1sccc1C)=O)C)C2 C1(COCCOC)CCN(C(=O)NCC2(CN=[N+]=[N-])CC2)C1 c1(C(N2CCCC(N(C(CC)=O)CC3CC3)C2)=O)ccc2c(c1)CCC=C2 c1(OC)cc(F)c(F)cc1C(N1CC(NC(c2[nH]cc(C)c2C)=O)C(O)C1)=O c1(NC(C(CCOCCO)NC(C(C(CC)C)O)=O)=O)cc(C)c(F)cc1O c1(C(=O)NC2(C(=O)NCCC3C(C)C3)CCCC2)ncccc1O N1(C(c2nc(SC)sc2)=O)CC2OCCN(C(C3C(C)(C)C3(C)C)=O)C2C1 C1C2CCC(C2)N1C(=O)O.Cn1cc(SCC(=O)OC(C)(C)C)c(=N)[nH]1 N1(C(C2(CC)CC2(F)F)=O)C2CCC1CC(N(C)C(C1C3COCC13)=O)C2 c1(CC)ccc(NC(=O)CC(C)(C)N(CC(O)CNC(=O)C2CC2)C)cc1 C(=O)(C1=CCCCC1)NC1(CC=C)CCN(C(c2ccccc2)=O)C1 OCCC(N=c1ccnc(N2CCC(NC3CCC3)CC2)[nH]1)C1CCOCC1 S(=O)(=O)(c1ccc2[nH]c(=NCc3csnn3)sc2c1)NCC#CC N1(CC)CCC(NC(=NCc2ccc(Cl)cc2)NC(C2CCCO2)C)CC1 C1(CCC)(C(=O)NCC(C)C(=O)NC2CC(CCC(N)=O)C2)CC(=O)C1 c1(C(N2C(C(N3CCC(SC)CC3)=O)C(C)CC2)=O)cccc2c[nH]nc12 N1(C(=O)CCC2CC2)CCN(C2CCN(C(c3cnccc3Cl)=O)CC2)CC1 N1(C(=O)COCCF)CCC2CN(C(c3cnc4c(c3)CCC4)=O)CCC2C1 c1(C(C)(C)SC)nnnn1C(c1ccccc1)C1CC1.C1CCN1.C(C)C.O c1(OCC=C)ccc(C(=O)NC2CCC2CNC(=O)C(C)SC)cc1 C(CC(CC)C(=O)NCCC(=O)N(C(C)C(=O)N(C)C)C)=CC c1(C(C(=O)NCC(=C)C)N(CC=C)CC#N)cn(-c2ccccc2Cl)nc1C c1(OCC)cnc(C(=O)NCC2CCCCN2C(=O)CC2COCCN2C)cn1 C1COCCC1.c1(N(CC=O)C)ccc(Cl)nn1.C(C)(C)(C=CC=O)SC.N C1(NC(CCC(N)=O)=O)CCCC12CN(C(=O)Cc1ccc(Br)cc1)C2 C1(CC(N2C(CC(=O)NCCNS(N)(=O)=O)CC2)=O)C=CCCC1 C(=O)(CC1OC(=O)c2ccccc21)NCC(CCNC(CN(C(C)=O)C)=O)(C)C CC1OCCC1CC(=O)NCCCN(C)C(c1cc(C2CCC2)[nH]n1)=O c1(NC)scnc1C(=O)NCC=CCNC(=O)CC(C)NC(N)=O N1(C(CSC(C)C)=O)CCC2CN(C(=O)CC3C=NN(C)C3=O)CC2C1 c1(C(C)C)cn2c(n1)CN(C(c1nnc3n1CCC3)C(=O)NC1CCC1)CC2 c1(SC)ncc(C(=O)N(C(C)CNC(C2(c3cc[nH]n3)CC2)=O)C)s1 CC1CC(C(=O)NCC(C)(C)NC(=O)C=Cc2cn[nH]c2)CCO1 C#CC1(C(N2CC(F)(CNC(C3CCOC3CC)=O)C2)=O)CCOCC1 N1(C(CCN(CC)CC)=O)CCCC(C)(C)C1C(=O)NC1CCC(C)(C)CC1 CC1CN(C(c2ccc(CC(F)(F)F)cc2)=O)CCCN1C(=O)CCF N1(C(c2cccc(C)c2Br)=O)CCCC12CCN(C(C13CCCC1C3)=O)CC2 CC1C(NC(C2(C)CC=CCC2)=O)CCCN1C(c1c[nH]cc1Br)=O O=C1NC(=O)C2(CC3CCC2(C(N2CCC(O)C2c2ccc(Cl)cc2)=O)C3)N1 c1(C(=O)NC2CCC23CN(C(C2(CO)CCCO2)=O)C3)ccc2ncccc2n1 C1(C)(NC(C(C)CC2CC2)=O)CCCCC1C(=O)N(C)CC1CC1 CC1(C)COC(C(N2CCSCC2C(N2CCCC(OC3CC3)C2)=O)=O)C1 Cc1noc(C)c1CC(=O)NCC1CCCC1NC(=O)C(C)Cc1cnc[nH]1 C12(C(=O)NC3CCCCC3CNCc3c(C)cnn3C)CCC(CC1)C2.C C(=O)(CCC(C)(C)[N+](=O)[O-])NCCCC(C)NC(c1cnn(C)c1C(F)F)=O C1(NC(CCc2cnc(C)s2)=O)CN(C(=O)CSCCC(F)(F)F)CC1C1CC1 N1(C(CCSC)=O)CC2CCC(C1)C(NC(c1cccc3ncccc13)=O)C2 C(=O)(C1=CC2CCCC12)NCC(CC)(CC)NC(c1c(O)ccc(CC)c1)=O N1(C(C(C)(C)c2ccno2)=O)CC=C(CC(=O)NOCC2CCC2)CC1 c1(C(N(CC(CN(C(C(CC=C)(C)NC)=O)C)O)C)=O)cc(C)c(Cl)c(N)c1 c1(C(N(C2CCCCN(C(=O)CC3CC3)C2)C)=O)cnc2ccc(Cl)cn2c1=O O=C1OC2(CCCCC2)CN1CN1CCc2nc(-c3ccccc3)[nH]c2C1 c1(NCC2C(C)(C)CCC2)ccc(S(=O)(=O)NCCCN2CCCC2)cc1Br C(=O)C(C)C(C)(C)C.C1(C=O)CCC(C)=C(C)C1.C(C)C.C(=O)(OC)N C1(NC(c2cnsc2)=O)CC2CC1CN2C(c1ccc(N2CCCC2)cc1Cl)=O C1(NC(COCCCOC)=O)CCCCC1.C1(C(C=O)(C)C)CCC(O)CC1.N c1(C(N2C(C)CCC(NC(c3cc(F)c[nH]3)=O)C2)=O)cc2cccnn2c1 CCC(CC(=O)N1CCC(NC(=O)CC2CN(C)C2)C(C)C1)CC(F)(F)F C1(C(N(C2CCN(C(=O)C=CC(C)C)C2)CC#C)=O)C2CCC1CC2 C1(CC(N2CC(N(C3CCOC3)C)C2)=O)COCCN1CC(F)(F)F N1(C(C(CCCC)C)=O)CCCC2(CCN(C(=O)C3=CCS(=O)(=O)C3)C2)C1 c1(CC(C)(C)C)ccccc1-c1cccnc1C(=O)NC1CN(S(C)(=O)=O)C1 N1(C(C(C2CN(C(=O)C(C)N3CCCC3)C2)OC)=O)CC2CC2C2CC12 Cc1nc2c(s1)CC(C(=O)NC1(C)CCN(C(C3CSC3)=O)CC1)CC2 C1(NC(c2ccnn2C2CC2)=O)CC1C1CCCN(CC2(CO)CCCCC2)C1 C1(C(=O)NC2CC(O)(C(=O)N(C)C)C2)CCCC1(F)F.C1CO1 N1(C(CN(CC(C)(C)C)C)=O)CC2(C)CCC1CC2.C12(C(=O)N)CCCCC1C2 Cc1cc(O)c(C(N2CCCC(N(C)C(c3cc(O)ccc3F)=O)CC2)=O)nn1 O=C(C#CC1CCC1)NC1CCN(C(c2csc(Br)n2)=O)C(C2CC2)C1 N1(CC=O)CCP(C)(=O)CC1.c1(C(=O)OC)ccc(C(=O)N(CCC)C)nc1 N1(C(C(CC#C)C)=O)CCOCC(NC(=O)Cc2cccc(-n3cnnn3)c2)C1 N1(C(=O)CC2CCC(O)C2)CC2CC1(C(=O)N(CCO)CCO)C2 C1(C(N(CCC(=O)NC2CN(CC(F)F)C2)CC=C)=O)CCN(OC)CC1 Cn1cc(C(N2CCN(C(=O)CC3CCCSC3)CC2)=O)n(C)c1=O CC1(C)OC(=O)CC1C(N1C(C(=O)NC2CC3(CC3)C2)CC2CC12)=O c1(NC(N(C2CC2)CC2N(C(C)(C)C)CC2)=O)cn(C)nn1.C1CCC1 CC(C)(CC(=O)NCC1CCCC2CN(C(=O)C=C(Cl)Cl)CC12)C(F)(F)F c1(OC)cc(Cl)c(C)cc1C(=O)NC1CCC1.c1(C(=O)N)cc2ncccc2[nH]1 N#CC1(C(=O)NCC2CCN(C(=O)C=CSCc3ccco3)CC2)CCSCC1 C12(CC=O)COCC(C1)C2.c1(CC)nccn1C(C)CC(=O)NC1CC1.C C(=O)(CCC(C)C)NCC.c1(C(C(=O)N)O)ccccc1Br.C(C)(C)(C)C=O C1(CC)C(O)CCN1C(c1ccc(N2CCN(Cc3cc[nH]c3)CC2)cc1)=O C(=O)(C1=CC2C=CC1C2)Nc1c(OC)cc(F)cc1.C12(CC1)C(=O)N2 c1(C(N(CCN(C(C)C)C(c2scnc2Cl)=O)C)=O)nccc2c[nH]nc12 Cc1cccc(CC(=O)NCC2CN(C(=O)CN(C)C(N)=O)CC2C)c1Cl N1(C(c2cn(CC=C)nc2)=O)CC(C)C(NC(=O)C=CCCC)C(C)C1 c1(CC)nc(C)[nH]c1C(=O)NCCC1(NC(=O)CC(=O)N(C)C)CCC1 C1(NC(c2ccsc2)=O)CC2CC1CN(C(C1CC(C3CCCC3)C1)=O)C2 C1(CNC(C(C)N(C)C(c2cc(CO)on2)=O)=O)CCCNC1=O Cc1c(C(=O)NC2CN(C(=O)C(F)C(C)C(F)(F)F)CC2C)ccc2n[nH]cc12 CC(C)C(O)CC(=O)NCCC1CN(C(C2CCS(=O)(=O)CC2)=O)C1 c1(CC)cccc(CC)c1CC(=O)NC1CC1NC(C12CCC(CC1)C2)=O c1(C(N2CC(O)C2)=O)cccc(N2CC=CC2)c1.C1(CC(=O)NC)CCCO1.C Cc1cc(O)cc(C)c1CC(N1CCC(NC(C2(F)CC3(CCC3)C2)=O)C1)=O N1(C(C(SC)SC)=O)CC2C(CC(=O)NCC=C(C)C)C2C1 c1(CC)cc(C(=O)NC(CNC(=O)CCC2CCCC2)C2CCC2)ccn1 C(=O)(C(CO)N(C)C)NCCN(C(=O)C(C)CN1CCCCC1)CCC N1(CC)CC(C(N2CC(O)(CNC(=O)CCC3CC3(Cl)Cl)C2)=O)CC1=O Cc1cc(C(N2CCN(C(=O)C3CC3)CC2Cc2ccccc2)=O)cc(O)n1 C12CC1CN(C(=O)CCN1C(=O)CCC1=O)C2.CC(C)(C)C.C(C(=O)N)NC CCC(F)(F)CC(=O)NCC1CCC(N(C)C(C2CCC(C)S2)=O)CC1 c1(CC)ccccc1.C1CCCC1(F)F.CC(C)(C)S.C1(C(=O)N)CC1C=O N1(C(C=C(C)C2CC2)=O)CCC2CN(C(c3ccn(C4CC4(F)F)n3)=O)CC12 C1(NC(CC=CCC)=O)CCCOC1C1CCN(C(=O)Cc2coc(C)n2)CC1 c1(OC)ccc(CC(=O)NCCC2CCCN2C(C2C(C)C2C)=O)cc1Cl C1(NC(c2nc(C)oc2)=O)(CO)CCN(C(=O)C(c2ccccc2)C2CC2)C1 c1(C(N(CCCC)C)=O)ccc2c(c1)N(C)CC2.C(=O)(CCC(=O)N)OCC CC(C)C(C(O)c1ccc(Cl)cc1)Nc1nccc(N2CCC(C(F)F)CC2)n1 C1(C)(CC)CC(C(=O)NCc2csc(C)n2)CCO1.C(=O)CC.C(N)=O N1(C(C2N(C(c3c(OC)n[nH]c3)=O)C(C)C2)=O)CC=CC(O)C1 c1(CC)ccc(F)cc1C(=O)N(C)CC1(C)CC1.C1(F)(C=O)CCOC1C C1(CNC(CCOCCC)=O)CN(C(c2cccc(SCC)c2)=O)CC1(F)F C1(C(=O)NC(C2CC(NC(c3cscn3)=O)C2)C)(COC)CCOC1 N1(C(CC(c2ccc(C)cc2)C)=O)CCC(NC(C2(C#N)CC(=O)C2)=O)C(C)C1 c1(NC(=O)Nc2cn(C)nc2C2CCOC2)ccc(Cl)c(Cl)c1 C1CN(C(=O)C(F)CC2CC2)C(C)(C)C1.c1(COC)cccc(C(=O)N)c1 c1(-n2cc(-c3cc(C(C)=O)cc(Cl)c3)nn2)ccc2nn[nH]c2c1 C12(CN3C(=O)CN(Cc4cn(CCCOC)nn4)C3=O)CCC(C)(CC1)OC2 N1(C(C2C(C)OCC2)=O)CCOC(Cn2cc(C(N3CCOC3=O)C)nn2)C1 N1(C(C(COC)(C)OC)=O)CCC(NC(c2c(C)oc(C)c2C)=O)CC(C)(C)C1 N1(C(C2(COC)CCCCC2)=O)CCC=C(C(=O)NCC(C)C(=O)OC)C1 c1(C(=O)N)cc(F)cc(F)c1N.C(=O)(C(C)(C)C(=O)NCCCC(C)C)N(C)C C=CC1(C(=O)N(CC2CC2)OC)CCN(C(C2CC(OC)C2)=O)CC1 C(=O)(C1CCCc2sc(C)nc21)N(CC(C)NC(c1cc(C)nc(O)n1)=O)C CCC(C)(C)CNC(=O)C(CO)NC(=O)COc1ccn(C)n1 Cc1cc(C)c(C(N2CC3CC3(NC(c3cc(Cl)c[nH]3)=O)C2)=O)[nH]1 c1(CNC(c2ncncc2F)=O)ccc(CNC(C2CC3CCC3C2)=O)cc1 C12(NC(CCCC)=O)CCOCC1CN(C(c1nc(C)ccc1F)=O)C2 c1(COC(c2c(C(C)C)sc(Cl)n2)=O)cc(=O)n2ccccc2n1 Cn1nnc2c1CCC(NC(=NCCC1COC1)NCc1ccoc1)C2 Cn1cnc2nc(=NCCC3CCCO3)[nH]c(NCC3(F)CCC3)c12 C(=O)(C(C)(C1CC1)N(C)C(c1cncn1C)=O)NC(c1ccco1)COC c1(C(C)=O)ccc(C(=O)NCc2cc(C(=O)N)co2)[nH]1.c1(CCO)cccs1 CCCCCC(CC)C(=O)NC(C)CCCCNC(=O)CCC(=O)NN(C)C C1(CC(=O)N(C)Cc2cc[nH]n2)CN(C(=O)CSc2nc[nH]n2)CC12CC2 N1(C(CSCC#C)=O)CC2(CCCN(C(=O)C(c3ccc(F)cc3)CC)C2)C1 C1(CNC(CN(CC#C)C(C2CC(C)=NO2)=O)=O)CCCCC1C C(C)(C(=O)NCC=CC(=O)NCc1nncs1)NC(=O)NC c1(C(=O)NCC(CC)Nc2cccnn2)ccccc1C.c12cc(c(C)s1)C2 C(N=c1[nH]cnc2[nH]ccc12)c1c(CNC(=O)CC23CCC(CC2)C3)cccc1 C(=O)(CCCc1nc(C(C)(C)C)no1)N(CCN(C)CCF)C(=O)C1CC1 C(c1ccc(N2CCCC2=O)cc1)=CC=O.C(CC)(C(=O)NCC(F)C)=CC C1(NC(CCNS(CC)(=O)=O)=O)CCCC(C)C1.C12(C=O)CC(F)(C1)C2 C(c1ccc(F)cc1)=C(C)C(=O)NCC1CCCC1NC(=O)CCP(C)(C)=O c1(C(=O)NCC2(CNC(=O)C(F)C3CCOC3)CC2)ccc(Cl)cn1 N1(c2n(CC)c(C(C)[N+](=O)[O-])nn2)CC(C(=O)OC)C2(CCCCC2)C1 CCCC(CCCNC(c1cnn(C)c1C)=O)NC(C1CC1C(C)(F)F)=O C(c1ccc(F)c(Cl)c1)=CC=O.C(=O)(CCCn1cccc1)N(CC(O)C)C.N C(=O)(CCCO)N1C(CNC(C2(CN(C)C)CC2)=O)CC1.c1ccccc1 Cc1ccc(C(=O)NC2CCC(C(=O)NC3CC4CCC3C4)CC2)cn1 c1(C(=O)NCC(C2CCCCC2)NC(c2nc(C)[nH]n2)=O)cccc2ccsc12 C1(C(=O)OC)CCCC(NC(C2CCCC2NC(=O)CC2CCCC2)=O)CC1 n1(CC2C(C)C2)nc(-c2ccc(OC)nc2)nc1-c1ccc(-n2cccn2)cc1 CN=c1nc(N2CC3CCCC3C2)[nH]c(=NC2C=C(C)CCC2)[nH]1 C(=O)(C1=CCN(C)C1)N1c2ccc(cc2)CC1.c1ccc(N(C)C)nc1.CCS C1(C(=O)NC(COC)CO)CCN(C(c2cnn[nH]2)=O)C1 c1(CCCC)c[nH]c(=O)c2c1cnn2-c1ccc(C)cc1 Cc1cccc(Br)c1CNC(N1CCC(CCn2cc(Br)cn2)CC1)=O N1(C(COC)=O)CCC2(NC(=O)C=CCO)CCCCC12 CC1(C)CN(C(=O)C(O)C2CN(C(=O)CC3CC=CCC3)C2)C1 c1(CC(C)NC(c2conc2CNC(c2cn[nH]c2)=O)=O)nccn1C C1(CC)(NC(=O)COC2CCN(C(C3CC(SC)C3)=O)C2)CNC(=O)C1 C1(CNC(C)CN2CCOCC2)CC(c2ccccc2)=NO1 C1(C(=O)NCCC2(OC)CN(C(C3CCN(C)CC3)=O)C2)CC2C=CC1C2 c1(CC=O)cc(C)nn1C.N1(C(C2(C)CC(=C)C2)=O)CCN(C(C)(C)C)CC1 c1(-c2cc(OCC)c(F)nc2)ccc2nc(C(=O)N=c3cc[nH]cc3F)cn2c1 Cc1ccncc1C=CC(=O)NCC1CCC1NC(c1ncc(Br)cc1O)=O CCC(C)C(C)C(=O)NCC1(C)CC1.c1(-c2cc(C=O)on2)cccc(Cl)c1 C1(NC(C(C)O)=O)CCC(NC(c2csc(-c3ccco3)n2)=O)C1 C(N=c1[nH]c2c(c(=NCC3CC(O)C3)[nH]1)CCC2)C1(C)CC1(Cl)Cl NS(=O)(=O)C(C(=O)N1CC2CC(C1)C2NC(C1CC1C)=O)c1ccccc1 Cc1nc(C(C)(C)C)sc1C(N1CCOC(C(C)NC(C2CSCN2C)=O)C1)=O Cc1ccc(NC(=O)NC(C)CCN(C)C)c(SCC2CC2C)c1 N1(C(=O)CC(O)c2ccccc2)CC2CC1CN2C(C1COCCC1(F)F)=O c1(CC(=O)NCCCN(C(=O)C(O)CC2CCOCC2)C2CC2)cc(Cl)cs1 c1(C(N2CCN(C(CNS(CC)(=O)=O)=O)CC2CO)=O)cn2cc(Cl)cnc2n1 N1(C(CN(C)C)=O)CCN(C2CCN(C(c3ccn(C(C)(C)C)n3)=O)CC2)CC1 C1(NC(C2C(NC(=O)CCc3csnn3)CCO2)=O)CC(O)C(F)C1 C1(CNC(C(C)(C)OC)=O)CC2(CCC2)CN1C(=O)CCC(C)SC CC1CCCC(C(=O)N(CCCOCCNC(=O)CCS)C)C1.c1nccn1C C(=O)(C(CC1CC1)NC(=O)CN1CCSCC1)N1C(COC)CC1 c1(C(N(C2CCC(NC(c3c(O)cccc3Cl)=O)C2)C)=O)cc(F)ccc1Cl c1(CN2C(C(=O)OCC)CCCC2)cc(C)ccc1C(C)C c1(NC(C2N(CCC(=O)OCC)CCCC2)=O)cccc(Cl)c1.CCC(C)C.O c1(C2C(C(=O)NC(C3(O)CN(C(=O)Cc4ccsc4)C3)C)C2)ccncc1Cl CC1(C)CCC(CC(N2CC(F)(CNC(C3CCN(CCF)CC3)=O)C2)=O)C1 N1(C(C(C)Sc2ccccn2)=O)CC2CC2(C(=O)NCCc2csc(=N)[nH]2)C1 CC1COc2c(C(=O)NC3CCN(c4ccc(F)cc4)CC3)cccc21 CC1(C#CC(=O)NCCOC2CCN(C(=O)C(F)F)C2)CCCO1 C1(CNC(c2ccc(C)cn2)=O)C2CCCCCC12.C12(C=O)CCN(CC1)C2 C(=O)(C1=CCN(C(c2cnn(C)c2Cl)=O)CC1)N(c1cccc(Cl)c1)C C12CC3CC(C1)CC(F)(C3)C2.C1(O)(CC=O)CCC1.C1(CC)(C=O)CC1 c1(-c2cc(-c3n(C(CC)C(F)(F)F)ccn3)c(F)nc2)ccc(F)c(OC)c1F C(=O)(CCCC1CCC1)N1CC(OCC#C)C1.N1(CC=O)CCNC(=O)C1.N C1(C(=O)NC(CCC=C)C2CC2)CC2CCC1N2C(C1CSCC(=O)N1)=O C1(NC(=NCCc2scc(C)n2)NC(C)C2CC2)CC(C)(C)OC1(C)C c1(C(N2CC(C(=O)Nc3c(OC)ncnc3)SCC2)=O)ccc(OC)c(C)c1 c1(C(=O)NCC2CC(CN)OC2)ccc(C2=CCCC2)cc1 O=C(NNc1ccc(C(F)(F)F)cn1)N1CC(c2ccccn2)C1 c1(C(=O)NC2(C)CC(NC(C3(OC)CCOC3)=O)C2)ccc2ncn(C)c2n1 CC(CCCNC(c1cc(C(N)=O)cs1)=O)NC(=O)CC1CNC(=O)C1 C1(C(N(C2CCN(C(=O)CN3CCC(=O)NC3=O)C2)C)=O)CC2(CCC2)C1.C C1(C(=O)Nc2ccc(SC)nc2)(CC)CCCN1C(c1c[nH]c(=S)cn1)=O c1(NC)ccc(C(=O)NCCC2CCC(=O)N2CCc2ccccc2C)cc1C N1(C(C2C(C=C)C2)=O)CCC(CN(C(=O)CC(=O)N)CC)CC1.c1nccs1 n1(CC(N2CC(NC(CCCC=C)=O)C(C)C2)=O)ccc2ccccc12 C(=O)(C1=CC2CCC(C1)C2)NCC1C(NC(c2cnc(OC)s2)=O)CCC1 c1(C(N2CC(NC(c3n(C)c([N+](=O)[O-])cc3)=O)C2)=O)ccc2c(Cl)nccc2c1 CN1CCOCC(NC(C2CC(O)CN2C(=O)CC2CCC(=O)C2)=O)C1 c1(C(N2C3CC2CN(Cc2cc(O)ccc2Br)C3)=O)c[nH]c2ncccc12 N1(C(C(CC(C)C)C)=O)CC(NC(c2cc3ncccc3s2)=O)C2CCCCC12 C1(C(N)=O)CCN(C(=O)CCc2nccs2)CC1.CC(C(=O)N)SC(F)(F)F.C N1(C(C2(C(=O)OC)C(=C)CC2)=O)CCCC(N(CCF)C(c2ccsc2)=O)C1 Cc1cccc(O)c1C(=O)NCC(C)(C)NC(=O)Cc1cc(Cl)sc1Cl N1(C(C(c2ccccc2)C)=O)CCCC(N(C(=O)COC(F)(F)F)CCF)C1 CCC(CC)N=c1[nH]c2cc(Cl)c(S(=O)(=O)N3CC(C)CC3C)cc2s1 C1(C(N2CCCC(CC=C)C2)=O)CC(O)CCN1C(=O)C(C)N(C)C Nc1c(F)c(F)c(CNC2CCc3ccccc3C23CC3)c(F)c1F C1(CC(=O)N(C2CN(C(=O)CSC(F)(F)F)C2)C)CCCC(C2CC2)O1 C1(CC)CN(C(=O)CCc2cn(C)cn2)CC1C.C1(CCOC)CC1C(=O)N C1(CNC(C(CC)n2cncn2)=O)CC(F)(F)CO1.C12CC(C1)CCC(=O)N2 c1(C(=O)NCC2N(C(C(C)NC(=O)NC)=O)CC2)n[nH]c(C(C)C)n1 C1(C(N2CCC2)=O)CC(=O)N(CCN(C)C)C1.Cc1nc[nH]c1CC(O)C=O.N C12(C(N3CC(O)(CC)C3)=O)COC(CCO1)C2.CC1CC1C(=O)NCC=O CC(C)CC(CNC(C1CCCN(CC(C)C)C1)=O)NC(C1(C)CC(F)C1)=O c1(C(=O)NCc2nn(C)c(C(=O)NC3CC(F)(F)C3)c2)cccc(F)c1N C(=O)(CCCC(=O)NC1CN(C(=O)Cn2cccn2)C2CC12)NCCC C1(NC(C(C)(C)N2CCOCC2)=O)CN(C(C2CC23CC3)=O)CCC1C(F)(F)F C(C(O)C(=O)NCC(O)Cn1cccn1)NC(c1cc(C(N)=O)c[nH]1)=O C1(CCC)CN(C(=O)CCc2ccc(C)o2)CCN1C(=O)C=C1CCOCC1 c1(C(C(=O)NC2CC(F)(F)C2)N(C(CC)C)CC(=O)OC)ccc(Cl)cc1Br C1(CNC(c2c(NCC)cccc2)=O)C2CCC1CN(C(C1CCOC1)=O)C2 c1(NC(C2C(NC(c3cnn(CCF)c3)=O)CCCC2)=O)ncnc(Cl)c1Br CC(C)(C)C#CC(=O)NCC1C2CN(C(=O)CCc3ccncn3)CC12 C1(C(=O)NCCCCNC(C(C)C2CC2)=O)CCNC(=O)C1 Cc1ccn(CC(C)C(=O)NCCC(O)CNC(=O)CO)n1.c1nccn1C.C C1(CNC(=O)CO)CC2(CCOCC2)CN1C(c1ncnc2sccc12)=O C=CCC(C)(C(=O)N1CC(N2CCN(C(C3CCC(=O)N3)=O)CC2)C1)N(C)C c1(SCCC2CCN(Cc3nc(CC)on3)C2)c(C)noc1Cl.C(C)=O CC1(C)COC(C(N2CCC(CNC(C3CNC(=O)N3)=O)CC2)=O)CO1 c1(CC(=O)NC2(CO)CCN(C(C)=O)C2)cc(OCCN(C)C)cc(F)c1 c1(CN2CCC(O)(C(=O)NCc3cscn3)C2)cc(O)cc(F)c1 C1(CNC(C(C)N(C)C)=O)CC2(CC2)CN1C(=O)CC1CCOC(C)(C)C1 c1(C(N2CC(CCC)CC2)=O)ccc(=O)n(C)n1.c1(C=O)nncn1C1CC1.N c1(SC)cc(C(N2CCC(CNC(=O)C(C)n3cnnn3)C2)=O)c(Cl)cc1Cl c1(C(=O)NC2C(NC(c3cnc(C4CC4)o3)=O)CC2)cn2ccnc2cn1 C(=O)(C1=CCCN(C(c2csc(=N)[nH]2)=O)C1)NC(C(C)(C)CO)(C)C c1(C(=O)NC(C(C)NC(=O)CCn2cccn2)CO)cc(O)nc(N(C)C)n1 C1(O)(C(CNC(N(CC(O)CF)CC)=O)(C)C)CCCOC1 CC(CS(C)=O)C(=O)N1CCCN(C2CN(C(=O)Cc3ccccc3)C2)CC1 C(=O)(C1CCc2ccccc21)N1C(C(=O)N=c2ccnc(C(F)(F)F)[nH]2)(C)CC1 N1(C(C(C2CCCCC2)OCC)C(=O)NC(C)C)CC2(CNC(=O)OC2)C1 N1(C(c2cn(C)c(Br)c2)=O)CCC2C(NC(=O)CCS(C)=O)CC12 CC(C)S(=O)(=O)C(C)C(=O)N1CCC1CNC(c1cc2scnc2[nH]1)=O S(=O)(=O)(c1cc(Cl)cc(Cl)c1)N1CCC2(N(Cc3ccc(C#N)cc3)CCC2)C1 c1(C(=O)NC(CN(C(=O)CCC(C)C)CC)C)ccc(OC)nc1F.C(C)=O c1ccc(F)c(C(N2CCN(C(C3CCS(=O)(=O)C3)=O)C(C3CC3)C2)=O)c1.C C1(NC(C(C)C2CCCC2)=O)CN(C(=O)CC2CC(F)(F)C2)CC2(CC2)C1 C#Cc1cnn(C)c1C(N1CC(CCNC(C2CCC2C(F)F)=O)C1)=O C1(C(=O)Nc2cnn(CC)c2C)CN(C(=O)Cc2ccsn2)CC(C)O1 C12(C(=O)NCC(C)NC(c3cc4nc[nH]c4cc3F)=O)CCCC(=O)N1CCC2 C1(CN(C)C(=NCC2CC=CCC2)NCc2ccnn2C)CC2(CCOCC2)O1 c1(C(=O)OCC2N(C(C(C)C)=O)CCCC2)ccc(C(F)(F)F)nc1O N1(C(c2nc(COC)oc2)=O)CCC2CC(C1)CN(C(=O)CC1CCOC1)C2 N1(C(C(CCCC)O)=O)CC2CCCC2(NC(=O)COCCOCCO)C1 C1(CCC)CN(C(=O)C(C)Sc2ccc(F)c(F)c2)CCN1C(c1ccsn1)=O C=CCCC(O)CNC(=O)C(CCC1CC1)NC(=O)COC(CC)CC N1(c2nc(C#C)c(F)cn2)CCC(C2CCCC2C(=O)O)CC1 c1(N2CC(C)OCCC2)nc(N2CCC(OCc3nccs3)C2)nc2c1SCC2 N1(C(c2ccc(C(C)=O)cc2)=O)CC(NC(=O)C(C)CC(N)=O)C2CCCCC12 C1(O)(C(C)NC(CN(C(=O)CCC2(C)CC2)CC#C)=O)CCCCC1 c1(OC)ccc(C(C)=CC(=O)N)cc1.C(C)CC(C)C.C1(Cl)(C=O)CC1(C)C c1(CN(C(C)CO)C2CC2)ccncc1.C1(=O)CCO1 C1(C(N(CC(C(=O)NC)C)C)=O)CCCN(C(=O)CCc2nncs2)C1C c1(CC)cnccc1C(=O)NC1CCCCC1C(=O)N(C)CC1OCCC1(C)C c1(C(N2CCC(C)C2C(N2CCCC(C)CC2)=O)=O)cc2cnccc2[nH]1 c1(C(N2CC(F)C2)=O)ccc(C#N)c(C)c1.n1(CCC)cc(Cl)c(C(=O)N)n1 CC1N(C(=O)C(C)(C2CC2)N(C)C(C2CCCOCC2)=O)CCCC12CCC2 Cc1ccc(C(C)NC(C2CC(NC(C3CCCN3C(C)C)=O)C2)=O)s1 Cc1nnn2cc(C(=O)N(C(C)C)Cc3cccc(Br)c3)ccc12 C1(NC(C(CC#C)O)=O)CC2(C1)CN(C(c1ncccc1NC(C)=O)=O)C2 c1(C(=O)NC2C(C)N(C(c3ccn(C)c3)=O)CC2)cc2c(F)cc(F)cc2[nH]1 n1(C(C)C(=O)NCC2CCN(C(=O)C(C)(C)C#N)C2)cnc2ccccc12 c1(C(N2C(CNC(C3CCCCC3O)=O)CCCC2)=O)ccc([N+](=O)[O-])c(Cl)c1 Cc1nc(NCC(N2CCCC2)C)cc(NC(C)CCCO)n1 Cc1cc(C(=O)NCC(C)NC(=O)CC2CNC(=O)C2)cc2cccnc12 CCCCCCC(C)CC(=O)NCCC(Cc1ccccc1)NC(=O)C=CCF Cc1ccc(OC(F)(F)F)c(C(=O)NC2CCC(S(C)=O)C2)c1 c1(C(N(CCCNC(C2CN(C)CC2C)=O)CC)=O)cc2nc(O)[nH]c2cc1N c1(C=O)cnc2n1CCC2.Cc1nc(NC2CC2)sc1C(=O)NCC(C)(C)C C(C(C)N=c1nc(Cl)[nH]c(CC)c1C#N)N(C(CCCC)=O)C c1(CN(C2CN(C(c3ccc(N(C)C)cc3)=O)C2)C)c(F)cccc1Br C(CC1=CCN(C(=O)C=C2CCOCC2)CC1)NC(=O)CSc1cccnc1 C1(NCC(=O)NCc2ccc(-n3cncn3)cc2)CCC2C3C=CC(C3)C12 c1(C=O)ccc(F)c(I)c1.C1(NC(=O)OC(C)(C)C)(CF)CCOC1 N1(C(C(=O)NC)c2cscn2)CCN(S(=O)(=O)N(C)C2CCCCC2)CC1 C1(C(N2CCC(CCOC)(NC(=O)CC(C)C)C2)=O)CCCCC(=O)N1 N1(C(c2ccn(C3CC3)n2)=O)C2CCC1(C)CC2.C1(C=O)CC1.C1CC1.N c1(C(N(C)CCN(C)C(C2Cc3ccccc3O2)=O)=O)nccc2c1CNC2=O N1(C(C(C(C)C)F)=O)CC2C3CCC(C2C1)N(C(C1CCOC(C)C1)=O)C3 N(C(=NCCF)NCC(N1CCC(OC)CC1)(C)C)C1CCC(COC)CC1 C1CS(=O)(=O)CC1C=O.c1ncc(F)cn1.C(C(=O)N)OCCOCC C1(CCC)CN(C(c2ccon2)=O)CC1C(=O)N(CCCC)C(C)C C1(C)(C(=O)N)CCC(=O)NC1.c1(OCCOC)ccnc(N(CC(C)C)C)n1 C=C(C)CC(C(=O)NC1CN(C(C)=O)C1)NC(=O)C(C)NC(N)=O S(=O)(=O)(c1ccc(Br)c(F)c1)N1CC(COC)N(C(=O)C(C)C)CC1 C1(CNC(=O)C(O)Cn2cncn2)CC(F)CN1C(C12CCC(C1)C2)=O Cc1ncc2c(n1)CCC(C(N1CC(NC(c3cscc3Cl)=O)CC(C)C1)=O)C2 c1(C(N(CC(CN(C(C2C(CCC)CCC2)=O)C)O)C)=O)cc(Cl)nc(Cl)c1 CC1CN(C(C2CCC=CC2NC(=O)CC2CCCC23CC3)=O)CC1CO C1(C(N2CCCC2)=O)CCCCC(F)(F)C1.C1(C(N)=O)(C(=O)N)CC1.C1CC1 Cc1cc(C(=O)Nc2cnn(C3CN(Cc4ccc(Cl)nc4F)C3)c2)cc(Br)c1 C1(C(C(=O)NCCC(C)(C)NC(=O)CCC2CCCO2)O)CCCCCC1 C1(C=O)CCN(S(=O)(=O)CC)CC1.C1(C(C(=O)NCCCC)C)CCC(=O)N1 N1(C(C2(C=C)CC2)=O)CC2C(NC(C3CC34CCC4)=O)C2C1.C(C)(C)C.O c1(C(=O)NC(C)CN(C)C(c2coc(-c3cccnc3)n2)=O)cc(Cl)ccc1F c1(N(C)CC2(CO)CC2)nc(N2CCC(C(F)F)C2)c2c(F)cccc2n1 CC1C(NC(=O)CC(C)(C)CNC(c2ncn3c2CCC3)=O)CCCN1C N1(c2ccnc(Nc3ccc(N4CCC(Br)C4)cc3)n2)CCCC2(C=CCO2)C1 CC(C)C(C#N)C(=O)NC(C)(C)CC(C)C.C(=O)CN(S(C)(=O)=O)C.N C(=O)(C1c2c[nH]nc2CN1C(=O)CCc1cnn[nH]1)NC1C(C2C(C)C2)C1 C(=O)(N=c1c(C)c[nH]cc1Br)C1CCC(NC(C=CC=CC)=O)CC1 c1(C(=O)NCC2CCN(C(C3Cc4cscc4C3)=O)CC2)cnc2occc2c1 C(CNC(C1C2CCC(F)C12)=O)(CC(=O)NC1CC(N(C)C)C1)OC CCC(C#N)C(=O)N1CCC(C2CCCN2C(c2scnc2C(F)F)=O)C1 n1(CC(N2C(C(C)(C)C)CCC2)=O)c(C)c(C)sc1=O.Cc1c[nH]nc1C(=O)N C1(C(C)C)CCCCC1NCc1cc(C2CC2)no1 C(=O)(CC(C)P(C)(C)=O)NC(C1CCCC1)CNC(c1c(C)n(C)nc1Cl)=O c1(OC)ccc(OC)c(CC(N2CCN(C(C3(OC)CCSC3)=O)C(C)C2)=O)c1 Cc1ccc(N(C)CCN(C(c2sccc2Br)C(=O)NC(C)C)C(C)C)cc1C C1(CC(=O)NC(CNC(CCOC(C)=O)=O)(C)C(C)C)COc2ccccc2O1 c1cncc(Br)c1.C1(CNC(=O)OC(C)(C)C)OCCC1NC(=O)C.O N1(C(C(=O)Nc2ccc(CCCC)cc2)=O)CCc2cc(F)c(F)cc2C1C C12(NC(CS(C)(=O)=O)=O)CCN(C(=O)CCc3nc[nH]n3)CC1C2 Cn1c(C(=O)NCC2CCN(C(C3C(C)(C)C3(C)C)=O)CC2)cc2ccccc12 c1(CCCC(N2CCC(C(C)NC(c3c(C)ccs3)=O)C2)=O)ccc(F)cc1 c1(CCC(=O)NC(CCCNC(C2(OC)CC2)=O)C)ccc(N)c(F)c1 c1(C(=O)OC)cccc(Oc2ccc(NC(=O)CCNC(=O)NC)cc2)c1 C1(NC(C=C(C)CNC(C2CC=CCC2)=O)=O)CC2(C1)CC21CCC1 C1(OC)CC2(CCC(C(=O)NCC(F)CNC(=O)C(N)=O)CC2)C1 N1(C(Cc2ccc(C)s2)=O)CCCC(CC(=O)NC2CCN(C3CC3)C2)C1 C1(NC(c2cc(C)oc2C)=O)CC2CC(C1)CN(C(=O)CCC1CCC(=O)C1)C2 C1(C(=O)NCC(CC)NC(c2ncnn2C)=O)CCCNS1(=O)=O C(=O)(CCC(=O)N1CCOCC1)NC(CCNC(CN1C(C)CC1)=O)C c1(CN2CC(CNC(=O)Cc3cc[nH]n3)OCC2)cnc2ccccn12 N1(C(CC(C)(O)C2CC2)=O)CCCCC(NC(=O)Cc2cnns2)C1 CC1COC2(C1)CN(C(C1(C3CC3)CN(C(c3sccc3Cl)=O)C1)=O)C2 N1(C(c2c(CC)nco2)=O)CCCC2(CNC(C3(C)CCCS3)=O)CCCCC12 c1(C(=O)NC2(c3c(C)non3)CC2)cccc(OCC(C)C)c1 c1(C(N(CC)CC)=O)cnc(O)c(C)c1.c1(C=O)c[nH]c(C(F)(F)F)c1.N C1(CNC(c2cccnc2Cl)=O)CC(F)(F)CN1C(=O)CC1CC1 c1(CC(=O)N(CC(C)O)CCNC(C2CC2C#N)=O)nc(F)c(F)cc1F C1(C)(CC)Oc2ccc(NC(=O)NC(C)CN3CCNC3=O)cc2O1 C1(NC(c2ccccc2Cl)=O)CC1C1CCN(C(c2cnn(CCF)c2)=O)CC1 C=CC1(CC(=O)N(C2CCC2C)C)CN(C(=O)CCc2cn(C)cn2)C1 N1(S(=O)(=O)Cc2ccc(Cl)cc2)CC2CCN(C(c3ccc(I)cc3F)=O)C2C1 c1(C=O)ccc(C(F)(F)F)cc1Cl.c1(CC(=O)N(CC)CC)cnns1.CO C1(CNC(c2c(CC)nc(C)o2)=O)CN(C(=O)C(C)C2CCC2)CC1(C)C CCCC(CCO)N=c1[nH]c(=NCCc2cccc(Cl)c2Cl)[nH]c2c1CSC2 CN1CC(C(=O)Nc2cccc(-n3cc(-c4cccc(F)c4)nn3)c2)C(C)(C)C1 CS(=O)(=O)C1(C(N2CCN(C(C3CCC=CCC3)=O)C(C3CC3)C2)=O)CCC1 C1(NC(C(COC)O)=O)CCCN(C(c2cc(C#N)cn2C)=O)C1C N1(C(=O)NC(c2ccc(F)c(Cl)c2)C)CCC2C(F)(F)C2(C)C1 N1(C(CCCCNC)=O)CCCc2c1cc(Cl)c(C)c2Cl c1(CN(C)CC2(CO)CCOCC2)cc2c(cc1Br)OCO2.c1(C=O)n[nH]cc1Br C1CCS(=O)(=O)C12CN(C(=O)CC13CCC(CC1)CC3)C2.C(C)C=O.CC.O c1(CC)nnc(N2CCC(OCC(C)C)C2)n1CC(C)(C)O N1(C(C2CN(C)C(=O)CC2)=O)CC(NC(=O)C(F)=C2CCCC2)CC12CCC2 C1(C(N(C2CCN(C(c3c[nH]c(C(N)=O)c3)=O)C2)C)=O)CCc2[nH]nc(O)c2C1 Cn1cc(CC(=O)NCCCCCCNC(C2COC(=O)N2)=O)c(C(F)(F)F)n1 c1(C(N2CC(C#C)C2)=O)nc(CNC(C2(Cl)CC2(F)F)=O)oc1C N1(C(C(CC2CCC2)OC)=O)CC=C(C(=O)NCC2(C)CCCO2)CC1 c1(C(N(C(C)C)CCN(C)C(C2CCC3CCC23)=O)=O)ccn2cncc2c1 N1(C(C(COCC)C)=O)CCN(C(c2cccc(C(C)C)c2)=O)CC1C1CC1 c1(C(N2CCCC2)=O)c(C)nn(C(C)C)c1Cl.C1(C=O)(OC(C)=O)CC1.N c1(COC)ccccc1.C(CCCCS)NC(CC1CN(C=O)C1)=O.C1CC1 C1(NC(C2C(C)CC(C)O2)=O)COC2(C1)CN(C(C1(C3CCCO3)CC1)=O)C2 C(=O)(C1=CCCCC1C)NC1(C2N(C(c3c(C)nc(CO)o3)=O)CCCC2)CC1 N1(C(C(S(C(C)C)(=O)=O)C)=O)Cc2nccn2CC(NC(=O)C2=CCOC2)C1 c1(CC)noc(C(=O)NCC2CCC(C)CC2)c1C.c1(C=O)ccc(C#N)s1 C(=O)(CC(C)C(F)(F)F)N1C(C)C(NC(c2ccc(Cl)nn2)=O)CCC1 CC1(C)COC(CC(=O)NCCc2ccccc2N2CCOCC2)CN1 N1(C(c2ccc(C)cc2)=O)CC(NC(c2cnc(S)nc2)=O)CC(O)C1 C(CCCC(CO)NC(C1CC2CC2C1)=O)NC(c1n(C)ncc1Cl)=O c1(C(=O)Nc2c(C)cc(F)c(F)c2)c(Br)cccc1[N+](=O)[O-] C(=O)(C(C)(F)CCCC)N1CC(C=C)(CC(=O)NCC(CC(C)C)OC)C1 c1(CN(CC(C)(C)C)C(=O)NCCC(F)(F)F)ccc(C(C)(C)C)cc1 n1(CC(=O)NCC2CN(C(C(C)C3CCOC3)=O)CC2C)ccc2ccccc12 N1(CC(C2CC3CCC2C3)=O)CC(C2CC2)OC(c2ccccc2)C1 c1(CN2CC3(C(=O)OC)C(C2)CCCO3)ccc2c(c1)OCCCO2 C1(NC(C(C=C)O)=O)CC2CC(C1)N(C(c1cnn(CC(C)C)c1C)=O)C2 c1(NC(CC2CCN(Cc3ccn(C)n3)C2)=O)ccc(F)cc1I N1(C(C(C(CC)O)(C)C)=O)CCC2CCC(C1)N2C(=O)Cc1cnn(C)c1C n1(CC(C)C)cc(CO)nn1.c1ccccc1.C(C)C(F)F.C(=O)CC1CC1 N1(C(C2CC(C(=O)OC(C)(C)C)C2)=O)CCCC(CC)C1.c1(C=O)ccco1 N1(CCC(=O)NC(CC(C)NC(c2cnc(C)o2)=O)C)CCNC(=O)C1 Cc1cc(CCC(N2CCCC2CN(C)C(c2ncn(C(C)C)n2)=O)=O)no1 C(C)(C)(CCC(=O)NC(C1CCCN1C(=O)C(c1ccccc1C)C)C)OC c1(CC)nn(C)cc1C(=O)NCC1CCN(C(C2CCOC2)=O)C1 C(=O)(CCS(C)(=O)=O)NC(C1(O)CN(C(c2cccc(CO)c2)=O)C1)C N(C1CCCc2sccc21)OCC.N12CCC(CC1)Cc1cn(nn1)CCC2=O CN1CC(C(N2CCC(N(CCO)C(c3cc(Br)co3)=O)C2)=O)CC1=O Cc1ccc(C2(C(=O)NC(C)C(C)C)CCC2)cc1.c1(C(=O)N)scc(C)c1Cl Cc1ccc(-n2cc(CN(O)C(C3CCN(c4ccncc4)CC3)=O)nn2)cc1 CC1OCCCC1C(=O)N(C)CCOCCCNC(c1ccnn1C(F)F)=O N1(C(c2cc(CSCC)on2)=O)CCCC(C(=O)N(C)CCOC)CC1 C1(NC(c2c(C)c[nH]n2)=O)CCN(C(=O)Cc2c(C)n[nH]c2C)C(C)C1 c1(N(C2CCN(C(C3CC(=C)C3)=O)C2)C(=O)C=O)scc(C)c1C.C1CC1.S n1(CC)nc(C)c2cc(C(=O)NC(C)(C)CNC(=O)C3=COCC3)sc12 CCCC(C#N)C(=O)N(CC(N1CCCC1CCCO)=O)CC1CC1 C1(C(N2CCCC(c3onc(-c4c(C)con4)n3)C2)=O)CN2CCC1CC2 C1(C(=O)NCC(CCNC(c2c(CC)[nH]c(=N)s2)=O)O)COCC(C)(C)O1 Cc1ccc(C(=O)C(N2CCC(N(C(=O)Cc3conc3C)CCO)C2)=O)cc1 CC1(C)C2COC1(C(N1CCN(C(c3sccc3Cl)=O)C(CC(F)F)C1)=O)C2 C(C)(C(=O)NC(C)CCCC)(C(C)C)NC(C)=O.C(=O)CCCn1ccnc1.N c1(C(N2CCC(C(=O)OC)C2)=O)cc2ccc(-c3cccc4[nH]ncc34)cn2c1 C1(C2CCCOC2)(NC(C(c2cc(Br)ccc2F)N)=O)CC1 C1(C(=O)NCC2CCN(C(CCC(C)CN(C)C)=O)CC2)CC(C)(C)OC1(C)C C=CCC(CC)C(=O)N1CCC(c2ccncc2)CC1 c1(C(=O)Nc2c(SC)cccc2)ccc2nc(-c3cccc4c3OCC4)sc2c1 C(c1ccccc1)=CC(=O)NC(=O)COC(=O)COc1cccnc1 O=S(=O)(c1ccc(NC2C3CCCCCC23)c(F)c1)NCCN1CCSCC1 N1(C(Cc2cccc(OC)c2)=O)CCN(C(c2cccc(C3CC3)c2)=O)C2CC12 C(=O)(C(CC(N)=O)NC(=O)C(c1cncnc1)C)NCc1c(C)nc(C)s1 c1(CC(C)C)n[nH]c(=NC2CC(NC(C3CNC(=O)N3C)=O)C23CCC3)s1 N1(C(=O)CC2CC(F)C2)CCC2CN(C(C34CSCC3C4)=O)CC2C1 CCCC(C(=O)N1CC2CCN(C(=O)CC(=O)OC(C)(C)C)CC12)S(N)(=O)=O C(CC(C)(c1nnnn1CCCF)NCc1ccc(Br)s1)(OC)OC1CC1 N1(C(C2CC2C2CC2)=O)CC2CCCN(C(c3ccccc3Br)=O)C2C1 N1(C(C=CCN(C(C2(OCC)CCC2)=O)C)=O)CC(=O)NCC1C C#CCC(CC(F)F)C(=O)NCC(O)CCNC(c1ccc(C#N)c(C)c1)=O C1(C(=O)NC2COCC2CO)(NC(c2cc(C)oc2)=O)CCC(C)(C)C1 C1(C)(NC(c2cc(CC)oc2C)=O)CCCN(C(=O)C=Cc2ccsc2)C1 C(=O)(C1=C2CCCN=C2NN1)N(CCN(C(c1c(F)cc(C)cc1Cl)=O)C)C N1(C(c2ncn(CC)n2)=O)CCC(COC)(NC(c2cnc[nH]2)=O)C1 C1(C2CCN(C(=O)C(O)CCS(C)=O)CC2)(NC(c2ccc(C)cn2)=O)CC1 c1(C(NC)=O)ccoc1C(F)(F)F.C1(OCC)CC1C(=O)N.C1CC1 N1(C(CCCNC(C)=O)=O)CC(NC(=O)C(C)(C)c2cnsc2)C(CO)C1 c1(C(=O)NCCC(C)N(C(c2cc(C)n(C)n2)=O)C)cc(C(C)C)ccc1F CC(CC1CC1)C(=O)NCCC(C)(C)NC(C1CC(OC(F)(F)F)C1)=O C12(C(N3C(C)(COC)CCC3)=O)CCCC1CN(C(=O)CC1COC(=O)C1)C2 c1(CCOCC(N2CCC(O)(CCO)CC2)=O)ccc(Cl)cc1F c1(C(=O)NCC(C(N2C(CC)CC(O)C2)=O)OC)ncnc(O)c1F c1(CSCCN2CCC(C(=O)NC)C2)cccc(C)c1 N1(C(C(CC)c2ccccc2)=O)CCCN(Cc2nc(C)no2)CC1 c12ccc(cn1)[nH]2.N1(C(=O)OC(C)(C)C)CCC(C(=O)NO)CC1.C1CCC1.C c1(C(N(CC(CC)NC(C2(CCF)CC2)=O)CCC)=O)ccn(C(F)F)n1 c1(NC(C2CSCCN2C(c2cnc(C3CC3)nc2)=O)=O)cc(Cl)ncc1F c1(C(=O)NC(CCCNC(C(C)C)=O)C)sccc1S(C)(=O)=O C#CCCN=C(NCC(C(F)(F)F)OC)N1CCC(c2cnccc2C)C1 c1(C(=O)NCC2C3CN(C(c4ccc(C(C)=O)[nH]4)=O)CC32)cnc(C)cc1Cl C12(CC)CCC(C(=O)N(C)CCNC(C3CC4CC4C3)=O)(CO1)C2 C(C(=O)NC1CC1)(CC=O)N(CCC#C)C.C(C)(C)C.C(=O)NCC.S N1(C(Cn2c(C)ccn2)=O)CCCN(C(=O)C(S(C)(=O)=O)C2CC2)CC1C(C)C C(=O)(CC(C)C(F)(F)F)N(C(C(=O)NC(CC(C)C)CN(C)C)C)C1CC1 C(=O)(CCC(F)(F)F)NC(C)(CNC(C1CC1c1ccccn1)=O)CO N1(C(CNC(c2cccnc2)=O)=O)CCC2C1CCN2C(C1(F)CCCCC1)=O Cc1cc(F)c([N+](=O)[O-])cc1C(N1CC2CC1CCC2O)=O Cc1ccc2c(ccn2CCC(=O)NCC#CCNC(=O)C=Cc2ncc[nH]2)c1 CC1OCCC1(C)C(=O)NCC=C1CCN(C(=O)C=Cc2cc[nH]n2)CC1 N1(C(C(CCCC)ON=C(C)C)=O)CC2CC1CN(C(c1cc[nH]c1CC)=O)C2 C12(C(=O)NCC3CCC(C)(C)O3)CCC(CC1)N(C(C1(C)C=CCC1)=O)C2 n1(CC(=O)NC2(C)CC(NC(c3cnc[nH]c3=N)=O)C2)nc(Cl)ccc1=O c1(SC(C)(C)C)ncc(NC(N2CCCC2CC(=O)NCCO)=O)cn1 C(=O)(C(O)C(C)C)N1C(CNC(CC(=C)C)=O)CCC1 C1(NC(c2c(CCC)occ2)=O)CCN(C(c2cc(C)c(Cl)s2)=O)CC1C C=CC1(CC(=O)NCC(C)(C)CO)CN(C(=O)C(CO)NC(=O)OC)C1 N1(C(Cc2c(C)nc[nH]2)=O)CCC(CNC(c2cccnc2S)=O)C1(C)C c1(COC)nnc2n1C(C)CN(C(=O)CC1CCN(C(C3CCCC3)=O)C1)C2 C1(NC(c2onc(C)n2)=O)CCCC12CN(C(c1ncc(Cl)nc1Cl)=O)C2 N1(C(C2OCCN(C(C)C)C2)=O)CC(NC(=O)CCCS(N)(=O)=O)C(C2CC2)C1 Cc1cccc(NC(N2CC(C(N3CCN(CC(C)CC(C)C)CC3)=O)C2)=O)c1 N1(C(c2n(C)nc(CC)c2I)=O)CCC2(CC(NC(=O)CC3CCC3)CO2)C1 C(=O)(CN1C(=O)Cc2cc(F)ccc21)N1CC2C(CNC(C3(C)CC3)=O)(C2)C1 n1(CC)ccc(CC(=O)NCCC(O)CNC(=O)CCNC(N)=O)n1 C(c1cc(F)c(F)c(F)c1)=CC=O.CCCCCOCC=O.C(C)C1CC1.N c1(C(=O)NCCC(=O)NCc2onc(C)n2)c(F)ccc(C(F)(F)F)c1F C1(C(=O)OC)CN(C(=O)Nc2ccc(N3CCCC3)nn2)CCN1C N1(C(CCNS(CC)(=O)=O)=O)CCN(C(c2cnn(C(F)F)c2)=O)C2CC12 N1(C(C(C(C)O)(C)C)=O)CCN(C(=O)CN2CCCNC2=O)C2(CC2)C1 C(C(CNC(=O)CCc1ccnc(Cl)c1)C(F)(F)F)NC(CSC)=O C1(C(N2CCC(N(C(=O)C=Cc3cc[nH]c3)CCO)C2)=O)CC12CCCC2 N1(C(CN(CCC#C)C)=O)CC2CCCC2(NC(=O)C(CC)CC)C1 C=CC(C)(CC)NC(=O)C=CC(C)NC(C1(C(=O)OC)CC1)=O Cc1coc(C(=O)NC2CCCCC2NC(C2(C)CC=CCO2)=O)c1C c1(N(C(C(N2CC(CC(=O)OC)C2)=O)=O)C)cc(C#N)cnc1C.C1CC1 N1(C(c2c(CC)n(C)cc2)=O)CC(C(=O)NC(C)C(=O)NC2CC2)CCC1C C1(NC(c2[nH]nc(OC)c2Cl)=O)CC2CC(NC(=O)C(=O)C(C)(C)C)C1C2 C1(OC)CN(C(c2conc2CNC(C2CC23CCCC3)=O)=O)C2(CCC2)C1 Cc1ccc(Br)cc1CC(N1CCCOC(CNC(C2OCCO2)=O)C1)=O c1(NC(=O)CCN2CCC(OC3CCCC3)C2=O)cc(O)nc(C(F)(F)F)n1 c1(C(=O)NCC2(NC(CCCSC)=O)CCCCC2C)cc2cc(Cl)ccc2[nH]1 C1(CNC(Cc2n(C(C)C)ncc2)=O)CC(C(F)(F)F)CN1C(=O)C1CC1 C1(NC(C2CCCOC2)=O)CC2(CCCN(C(=O)Cc3cncnc3)C2)C1 c1(C(=O)NC2CN(C(Cc3c(OC)ccc(F)c3)=O)C2)ccc2occc2c1 C(CC(=O)NCc1nccnc1C)(C(C)(C)C)NC(CCCC(=C)C)=O C(c1ccc(N(C)C)cc1)=CCNC(CCn1cc(CC(=O)OC)nn1)=O N1(C(C(CCCC(C)C)C)=O)CCc2ccc(C(N3CC(N4CCC4)C3)=O)nc2C1 C1(C(=O)NCCCc2cn(CCCC(=O)N(C)C)nn2)OC(C)(C)OC1(C)C C1(NC(c2ncc(C)nc2)=O)CCC2CCN(C(c3csc(C(F)F)c3)=O)C1C2 c1(C(=O)NC2(CCNC(COCCOCC)=O)CCC2)ncoc1.C C1(COC)CC(O)(CNC(c2cc(C(N)=O)no2)=O)C1 C1(CC(=O)NCCCN(C(CC2(OC)CC2)=O)C2CC2)CCC(=O)N1 c1(OC)cc(O)ncc1C(=O)N.C(=O)(CC=O)NC(C)C.C1CC1.C1CC1 c1(SCC)ccc(C=O)cn1.N12CCCC1C(=O)NCC(O)CNC2=O CCC(CC(F)F)C(=O)NCC1CC2CCC(C1)N2C(C1CCSCC1)=O c1(N(C)CC2CCN(C(c3c(C)cc(F)cc3C)=O)C2)ncnc2cnccc12 N1(C(C2CCN(C(c3c(CC)occ3)=O)C2)=O)CC=CC12CCOCC2 N1(C(C)C)CCCC(Nc2nnc(CN3CCCC(C(N)=O)C3)s2)C1 C(c1cscn1)=CC(=O)N(CC(C)N(C)C(c1cocc1Br)=O)C C1(C(N(CC(C(=O)NC(C#CC)(C)C)C)C)=O)COCC1(C)C C(CCSC)(C(=O)N(CCC(C(C)C)NC(C1(CCOC)CC1)=O)C)OC c1(CN2CC(CNC(c3ccnc(Cl)c3Br)=O)OCC2)ccc(Br)c(F)c1F N1(C(c2c(CNC(C(CC#C)(C)C)=O)ocn2)=O)CCn2c(O)nnc2C1 c1(CC)noc2ncc(C(=O)NC3CC3C)cc12.C1(C=O)CCCC(C)(C)C1 Cc1cnc(C(=O)NC2CCC(NC(=O)C(=Cc3c[nH]cn3)F)CC2)c(Br)c1 CC(CCCC(=O)N1CCC(O)C(C)C1)NC(c1cnn(CCF)c1)=O c1(NC(CN2C(COC)CCC2)=O)sc(-c2ccc(F)cc2)nc1C Cc1ncc(C(=O)NC2CCN(c3ncccc3C(N)=O)C2)c(C)n1 c1(C(N2CCN(C(C(C)OCC=C)=O)C(C)C2)=O)cc2c(ccn2C)[nH]1 N1(C(C=CSC)=O)CCC(NC(=O)C=CCOc2ccccc2)CC1C N1(C(C(CC)OCC)=O)CCC(C)(C)C1CC(=O)NOCC1CCOCC1 N1(C(=O)NCc2cc(O)nc(O)n2)CC2C3CCC(CC3)C2C1 C1(CC)(NC(=O)C(c2ccoc2)NC(=O)CCOC)CC(C)(C)C1 Cc1cc(O)cc(C)c1C(=O)NC1CN(Cc2cccc(O)c2O)CC1F C1(C(=O)NC(CC(=O)OC)C)CCCN(C(C2OCCC2C(C)C)=O)CC1 c1(-c2cn(CC(=O)N(C)CCO)nn2)cc(N)n(C)n1 CC1(C)CC(NC(C2CCC(O)CN2C(c2ccnnc2O)=O)=O)C(=O)O1 C1(NC(CCSCCCC)=O)CN(C(=O)C=Cc2scnc2C)CC2CCCC12 c1(C(=O)NC(C2CCN(C(C=C(C)C)=O)CC2)C(C)C)c[nH]c2cccnc12 CC1(C)Cc2ccc(C(N3CC4(C3)CN(C(C3CCCCS3)=O)C4)=O)cc2C1 CN1C(=O)C(=O)N(CCN2CCC3(C2)CN(C(=O)C(C)(F)C(F)(F)F)C3)C1=O N1(C(CC2CCC(=O)O2)=O)CC2CC2(NC(c2ccncc2Cl)=O)C1 c1(C(N(CCC)CCOc2cc(C)cc(C)c2)=O)cc2c(s1)CCN(CC)C2 C=CC1(C(=O)NCC2(C)CCC(O)CC2)CCN(C(=O)CCc2cccn2C)C1 c1(N2C(C(N3CC(C)C(O)C3)=O)CC3CC32)ncnc2c(Br)c[nH]c12 c1(C(=O)NCC(CC)NC(c2cc(C)n(C)c2)=O)cn2cc(C)sc2n1 c1(C(=O)NCCNC(=O)Cc2cccc(OC(F)F)c2)ccc2n[nH]cc2c1 Cc1sc(C(N2CCC2C(N2CCCC2c2cccc(F)c2)=O)=O)cc1Br c1(C(=O)NC2CN(c3ccnc(OC)n3)C(C)C2)ccc2nccnc2n1 C#Cc1cccc(CC(=O)NC2CC3CC2CC3C(=O)NC(C#C)CCC)c1 N1(C(C2(CCC)CCC2)=O)CC2CC1CN(CC1CC(C)(C)C1C(F)(F)F)C2 C=CCCCCCC(=O)N1CC=CC1(C(=O)NC(c1ccoc1)C)COC C1(C)(CC)C=C(C(=O)NCC2CCCCC2)C1.C1(C(=O)N)CC2CCC2C1 Cc1cc(C(=O)N(C)CC2COCCN2C(C23COCC2C3)=O)n(C2CC2)n1 C(C)(CCBr)(c1nnnn1C1(C)CC1)NC(c1ccccn1)COC N1(C(CC2N(CC)CCC2)=O)CCCC(F)(CNC(c2ccccc2C)=O)C1 N1(C(C(OC)OC)=O)CCOCC(NC(c2sccc2-n2cnnn2)=O)C1 c1(C(=O)NC2(CC=C)CCN(C(=O)CCO)C2)cc2scnc2[nH]1.C1CC1.C CCC(C(=O)NC(c1ccccc1)CNC(c1ccc(F)o1)=O)N(CC)CC c1(C(=O)NC(CNC(c2scnc2C2CC2)=O)C2CC2)cccc(Cl)c1F N12CC(C(F)(F)F)OCC1C2=O.c1cnn(C)c1C(F)F.C(CO)OCC C(=O)(C#CC1CCCC1)N1CC(CCNC(Cc2n[nH]c(=NC)s2)=O)OC(C)C1 N1(C(C(CC)CC)=O)CCC(CNC(c2ccnn2CC(C)C)=O)(OC)CC1 N1(C(C(C)n2ccnn2)=O)CC(O)CCC1C(N1CCC2(CCC2)C1)=O N1(C(c2nc(CCC)sc2)=O)CCN(C(C2CNC(=O)CC2C)=O)C(C(C)C)C1 C(=O)(CCC(C)NC(=O)C=C(C)C(C)(C)C)N(C(CC)COC)C N1(C(CSCCCC)=O)CC2(CCN2C(=O)C(COC)Oc2ccccc2F)C1 c1(C(N(CCC(C)NC(C(CC)C(C)C)=O)C)=O)cnn2c(C)ccnc12 CCS(=O)(=O)CC(=O)NC1(CC)CCCN(C(=O)C2=CC(C)(C)C2)C1 c1(C(=O)NC2CC(Nc3cc(O)ncn3)C23CCC3)cc2nn[nH]c2cc1F N1(C(C(c2ccc(CC)cc2)C)=O)CCC(NC(=O)C=Cc2ccsc2)C12CC2 N#Cc1ccc(C(N2CC=CC2Cn2cc(C(N3CCCC3)C3CC3)nn2)=O)s1 n1(C(C)C)ncc(C(N2CCCC(NC(=O)C(C)CN(C)C)C2)=O)c1Br c1(NC(C2CCN(C(c3ccc(C)o3)=O)CC2O)=O)ccc(Cl)c(C#N)c1 Cc1ncnc(C)c1CC(=O)NC1CCC(NC(=O)CC2CCCC2(F)F)C1 N1(C(CCC2CCC(NC(C=C(C)C(C)C)=O)C2)=O)CC2(COC(C)C2)C1 CC1COCC(C(=O)NCc2ccc(C(=O)N(C3CCC(CO)CC3)C)o2)O1 C1(C(N2CC(CN(C(COC)=O)C)C2)=O)(COC)C=CCC1 C=CC1(O)CCN(C(c2cnc(N(C)C)c(C)c2)C(=O)NC2CCCC2)C1 Cc1cnc(C(=O)OCC(C2CC23CCCC3)=O)cc1C C1(NC(C)=O)CN(C(=O)C2CC2)CC12CC2 C(CC(C(C)(C)C)NC(c1nsnc1O)=O)N(C(=O)Cc1ncc(Cl)s1)C c1(CC)c(C)cc(C(N2CCCC(NC(=O)C(C)(C)C)C2)=O)c(=O)n1C c1(CC)c(C(N2CC(NC(c3nn[nH]c3Cl)=O)C(C)C2)=O)ccn1C N1(C(C2N(C(C3C(CC)C3)=O)CSC2)=O)CC(C)(C)C12CCC2 c1(OC(C)C(=O)N(C2CCN(c3ccccc3)C2=O)C)ccc2c(c1)CCC2 N1(C(C(C)=C2CC2)=O)CCC(C)(C)C(NC(=O)COC2CCCOC2)C1 CON(CCC(=O)NCC1(C)C=CCCC1)C(=O)COC1CC1 C1(CNC(c2c(CNC(c3cc(C)sc3)=O)n[nH]c2)=O)CC2(CCC2O)C1 C1(NC(C(C)=CC2CC2)=O)CCCCC1CC(=O)NC(c1nncn1C)C Cc1cccc(C)c1CC(=O)NC1(C(=O)NOCCC2CC2)CC1 N1(C(C2C(C(N)=O)C2)=O)CCC(CCCNC(=O)Cc2cc[nH]n2)CC1 CS(=O)(=O)c1ccc(C(=O)NCCn2ccnn2)o1.[SH](=O)(=O)c1cccs1.C c1(CC)ccc(C)c(NC(c2c[nH]nc2CCNC(C2CCCSC2C)=O)=O)c1 Cc1ccc(C(N2CCC(F)(CNC(=O)Cc3ncc(Cl)s3)C2)=O)c(C)n1 C1(OC)CC2COCC(C1)N2C(=O)NC(C1CCCCC1)C CCCC(O)C(=O)NCCCCCCNC(C1CCC1C(C)(C)C)=O N1(C(N(CC(C)C)CCCN2CCC(C)CC2)=O)CCCN2CCCC2C1 C1(C(=O)NCc2cccc(N)c2O)CCc2n[nH]cc2C1 CCC(C)C(O)C(C)C(=O)NCC1CC(C(=O)NC2CCOCC2(C)C)C1 N1(C(c2c(NCC)cccn2)=O)CC(NC(c2snnc2CC)=O)CCC1C CC12CN(C(=O)CCc3ccc(Cl)cc3)CC1CN(C(c1cc(=O)cc[nH]1)=O)C2 N1(C(Cc2nc(C)sc2)=O)CCN(C(C2CCCOCC2)=O)CC1 C(CCCC(=O)NC(CNC(=O)CCC1CCCO1)C1CCC1)N(C(C)C)C C1(OC)CCC(CNC(=O)NCC2CC(C)(O)C2)CC1 C1(C(C)C)CN(C(C2CC(C)CC(=O)N2)=O)CCCN1C(=O)Cc1cnccn1 CC1CN(C(c2cc(CNC(c3ccoc3Cl)=O)ccn2)=O)CC(CO)O1 C(=O)(CC(C)(C)CC)N1C2(C(N3CCC(C=C)C3)=O)CC2CC1 N1(C(c2cc(CC)ccn2)C(=O)NCCC)CCN(CC2CC2)C(=O)C1 C1(OC(C)C(=O)NCCC2CCCN(C(=O)CCC3(C)CC3)C2)CCCCCC1 C(CC(C(C)(C)C)NC(=O)Cc1ccsc1)N(C)C(c1nccc(N)c1Cl)=O c1(N2CC(CNC(CC(COC)(C)O)=O)OCCC2)ncc2c(n1)COC2 c1(COC)ncc(CNC(=O)CC2(C)CN(C(=O)C(C)OC)C2)[nH]1 c1(C(N2CCOCC(C)(CNC(CCCC#C)=O)C2)=O)cc(C)c2c(c1)CCC2 c1(C(N(CCC(=O)NC2CCN(CCC)C2)CCO)=O)ccc(=O)n(C)n1 CC(=O)CCCCC(=O)N(CC(=O)NC(CO)CCCO)C N1(C(CN(CCOC)C)=O)CCCC(F)(C(=O)NCc2cn(C)nn2)C1 C1(NC(C(COC)OC)=O)CCCCC12CCCN(c1cc(Cl)c(O)nn1)C2 Cc1csc2c(=NCCCNC(=O)CSCc3ccccn3)[nH]cnc12 CCCC(C)(O)CNC(C1CCN(C(c2cscc2OC)=O)C1)=O N1(C(C2N(C)CCC2)=O)CCC2(CC1)CC2NC(=O)CCN1CCCC1=O C(=O)(CCS(C)(=O)=O)NCc1c(C(=O)NC(C#C)C)n[nH]c1 C1(C(N2CC(C)C(NC(c3ncccn3)=O)CC2)=O)CCC2(CCC2)CC1 C(=O)(C1=CCCC1)NCC(C)NC(=O)COc1ccc(Br)cc1 C1(CC(=O)N(C2CCCN(C(=O)Cn3c(C)ccc3C)C2)CC)CC2CCC1O2 C1(C(N(CCNC(C2CC2(F)F)=O)CC)=O)CC1C1CCCCC1.CCO.O Cc1nn(C)c(CNC(=NCCc2cccc(Br)c2)NC2CCC2)c1Br Cc1ccnc(C(F)(F)C(=O)N2CCC(N(c3nc(C(C)=O)cs3)C)C2)c1 N1(C(C#C)=O)CCC2(CC1)CC2CNC(=O)C(C)Nc1nc(C)cs1 C1(C(=O)NCc2c(C)coc2C)CC2CC1CN(C(C1C3CCCC13)=O)C2 c1(C(=O)NCc2c(CNC(c3ccncn3)=O)cccc2)nsc2ccccc12 Cc1nc(C(=O)NC2CCN(C(=O)CCc3cncs3)C2C)c2n1CCCC2 C1(NC(c2c(C)ccs2)=O)CCN(C(=O)Cc2conc2C)C1C1CC1 C1(O)(C(N2CCC2)C(=O)OC)CCN(C=O)C1.c1ccccc1.C(C)(C)C.C Cc1cc(C(F)(F)F)ncc1NC(C1(CC(N)=O)CCCCC1)=O c1(C(=O)NC2(CNC(C3CCCN(C)C3)=O)CCCCC2)ccc(Cl)cc1N c1(COCC(=O)NCC2CCN(CC=CCl)C2)cccc(Cl)c1 C#CC1(C(N2CCC(F)C(F)C2)=O)CCN(C(c2ccc(C)c(O)c2)=O)C1 N1(C(C(C)Sc2ccccc2)=O)CCCC(S(C)(=O)=O)CC1 C1(CC(=O)OC)CCC(S(=O)(=O)NCCCCc2cccc(OC)c2)C1 C1(C(CC)NC(C2CCOC2CNC(c2ccc(C)s2)=O)=O)CCOCC1 C1(NC(CC2(CC(=O)OC)CC2)=O)CC(O)C1.C(=O)CC.C(C)=O.C c1(C(=O)NCC2(C)CCCN(C(C3CC34CCCC4)=O)C2)ncn2ccccc12 C1(C(=O)NC(CNC(c2c(Br)cn(CC)n2)=O)(C)CO)CCC2(CCC2)C1 CC(CCC(=O)NC1CC(n2ccnn2)C1)NC(C1CCC(C)(C)C1)=O C1(CC(=O)NC(C)CN(C(=O)CC(c2cccc(F)c2)O)C)OCCCC1(C)C c1(N(C)C)ccc(C(N2CCCC3(NC(c4cccnc4)=O)CC23)=O)cc1F C1(F)(C(N2CCC(C)(CNC(C3CCC(CC)CC3)=O)C2)=O)CCCCCC1 CC1(C2CC2)NC(=O)N(CC(=O)NC23CC(c4nn[nH]n4)(C2)C3)C1=O CC1(C)CCC(C(=O)NCCN2CCCC2)(NC(c2cnc(N)cn2)=O)C1.C N1(c2cn(C)cc(Br)c2=O)CCC2(CC=CCO2)CC1 CC1=C(C(=O)N2CCC(N(C)C(c3cc(Cl)c[nH]3)=O)C(C)C2)CCS1(=O)=O Cc1cc2ccccc2n1CC(=O)NCC(C)CNC(=O)C1CCc2c[nH]nc21 N1(C(c2cc(C)oc2)=O)CCC2(CC1)CCN(C(c1n[nH]c(C(C)(C)C)n1)=O)C2 C12(C(=O)NC3(CNC(c4cc(C)ncn4)=O)CC3)CCOC1CCOC2 c1(CN2CCN(C(Cn3c(C)ncc3)=O)C(C(F)(F)F)C2)cnn2ccccc12 c1(C(N2CCOCC(CC(=O)OC)C2)=O)cn(CCC#N)c2ccccc12 N1(C(C(C=C)(C)C)=O)CCC(CO)C(NC(=O)CC(C(F)F)c2ccccc2)C1 C(c1cccnc1C)=CC(=O)NC(C1(O)CCN(C(c2c(C)cnnc2)=O)C1)C C1(C(=O)NCCCNC(CCc2cc(C)[nH]n2)=O)CCC(C(F)(F)F)CC1 c1(C(N(C2CCN(C(C3CC(S(C)(=O)=O)C3)=O)C2)C)=O)ccc2nccn2n1 N1(C(c2cnc(C(C)C)[nH]2)=O)CC(O)C(O)C1CNC(c1ccncc1)=O c1(C(=O)NC(CN(C(CC(=C)C)=O)C)CC)cccnc1C(C)=O CC1(O)CCC(CC(N2CCC(NC(=O)Cn3ncccc3=O)C2(C)C)=O)CC1 C(=O)(C(C(C)(C)C)NC(=O)Cc1ccccc1F)N(C)Cc1cnco1 c1(NC(CC(C)C)CS(C)(=O)=O)ncc(S(=O)(=O)NC)cc1Cl.C1(C)CCCO1 Cc1c(Cl)c(C(=O)NCC2CC(NC(c3ccnc(S)c3)=O)C2)nn1C C(=O)(C(C)(C)CC1CC1)NC(C)CCNC(=O)C=CCN1CCOCC1 C(C)(CN=c1[nH]c(=NCc2cc(Cl)c(F)cc2F)[nH]c2cc[nH]c12)OC c1(C(=O)NCCOCCCN(C(=O)C(F)C2CCC2)C)cccc2c1NCCC2 C1(CC(=O)N(CCC)C(c2cnn(C)c2)C)CCN(Cc2ccccc2)C1 N1(C(Cn2c(C)c(Cl)cn2)=O)CCC(F)(CNC(C23CCCC(CO2)C3)=O)CC1 Cc1n[nH]c2cc(C(=O)NC3(C)CCCN(C(=O)CCCOC(C)=O)C3)ncc12 c1(C(=O)NCC2CC(F)CN2C(C2CCCOCC2)=O)cc(F)ccc1F C1(NC(c2ccc(C3CCCO3)nn2)=O)CN(C(c2cccnn2)=O)CC1F C1(C(=O)NCCCC(C)(C)NC(c2n(C)c(Cl)c(Cl)c2)=O)CC2CC1CC2(F)F N1(C(c2cnc(CC)[nH]2)=O)CC2(CCCC2NC(=O)C(C)C(C)CC)C1 CCC(CC(=O)N1CC(NC(c2cc(C(=O)OC)cc(C)c2)=O)C(C)C1)C(C)C C=C(Cl)CCC(=O)NCC(C)N(C(=O)CCC1(C)CCC(=O)N1)CC c1(C2(C)CC2)ccc(C(=O)NCCCCNC(C2(O)CCSCC2)=O)cc1 N1(C(Cc2cc(C)on2)=O)C2CC(F)C(C2)C1C(N1CCNC(=O)C1C)=O Nc1cc(C(N2CCCC(N(C(=O)CCc3ccncc3)CF)C2)=O)cnc1N c1(C(N(C2CC(NC(=O)CCO)C2(C)C)C)=O)cc(C)ccc1O.C(N)(=O)N N1(C(=O)NC2C(OCC)CC2)C(C)CN(c2cccc(C)c2C)CC1C C#CCC(CC)NC(=O)CC1(NC(=O)C(C)Cn2ccnc2)CC1 N1(C(C=CC(C)(C)SC)=O)CCC(O)CC1.C1(C=O)CCCC(C2CC2)O1.C c1(C(N2CCC(CN(C(C(CCC)=CCC)=O)C)C2)=O)noc2c1COCC2 C#CCCCCCC(=O)NCC(CC(=O)NC(c1ccncc1)C)OC C1(NC(Cn2c(C)ncc2)=O)CN(C(=O)CCCCC(N)=O)CC2(CCC2)C1 CC1CC(NC(=O)CCCCCN(C)C)CN(C(C2CC(n3ccnn3)C2)=O)C1 N(C(=NCC1CCCCO1)NC(c1ccccc1)CF)CCOC C(C(C)(C)C#CC(=O)N1CC2(CCC2O)C1)NC(CC1N(C)CCC1)=O c1(SC)ncc(C(=O)N)c(O)n1.C1CN(C(c2cccn2C(C)C)=O)CC12CC2 C1(OC)CC(NC(C2CC(CF)C2)=O)CN(C(=O)C(c2ccncc2C)C)C1 CCC(C)C(O)C(C)C(=O)NC1COCC1C(=O)NC1C=CCC1 c1(C(N2CCC(N(C(c3nc(COC)sc3)=O)C)C2)=O)cc2n(c1)CCCC2 O=C1CCC(CC(=O)NCCNC(C2(C(F)(F)F)CC2)=O)C1 c1(C(=O)NC)ccnc(-c2nnc(C3CC(=O)N(C)C3)n2C)c1 N1(c2cc(N(C)CC3CC3(C)C)nc(C(C)C)n2)CCC=C(c2ccncc2)C1 N1(C(C(CC(C)C)n2ccnc2)=O)CC(C)(CNC(=O)CC2CCC2)CC1(C)C c1(C(N(c2cccc(Cl)c2)C2CC(C)C2)=O)cccc2c1nnn2C C1CCC2(CN(C(c3cc(C(C)(F)F)on3)=O)C2)O1.CC(C)C(C)CC(=O)N.C C1(NC(c2cc(CCCCC)[nH]n2)=O)CCN(C(=O)CC(F)(F)F)CC1CO c1(N(CCN(C(C(=O)N(C2C(SC)COC2)C)=O)C)C)ccc(Br)cc1 N#Cc1ccc(Br)cc1C(N1CC2(CC(C(=O)NC)C2)C1)=O.c1ccnc(F)c1 N1(C(c2n(C)nc(O)c2)=O)CCN(C(c2cnc(C3CC3)o2)=O)CC(C)(F)C1 c1(NC)cccc(C(=O)N(C(C)CCNC(C2CCC2(C)C)=O)C)n1 C(CN=C(NCC1CCC1)NCC(c1ccc(Cl)cc1)(C)C)c1c(C)ccs1 N1(C(C(CCCOC)NC(c2cccnc2O)=O)=O)CCC2(CC=CCO2)C1 CC1(C)CN(C(c2csc(C3CC3)n2)=O)CC1CNC(C1CCCN1C=O)=O C1(C(N2CC(CNC(c3cn(CCCF)nn3)=O)C2)=O)CCOC1=O c1(CCCOCCN(C=O)CC)cnc2c(Br)cccn12 N1(C(C(CSC)OC)=O)CCC(C(=O)Nc2cscc2C)C12CCC2 N1(C(c2cncn2CC(F)(F)F)C(=O)N)CCCC(C)(O)C1.Cn1nnc(C)n1 C1(NC(c2c(OC)c[nH]n2)=O)CCC(C)(NC(c2scc(C)c2C)=O)CC1 C1(NC(CC(CC=C)(C)C)=O)CC2CCCC(C1)C2.C12(C(=O)N)CC(C)(C1)C2 N1(C(CCOC)=O)CCC2(NC(C3CCCCCC3)=O)CCCCCC12 c1(OC)ncc(-c2cccc(N(C)C)c2)cc1C(=O)Nc1[nH]cnc1C c1(CCC)cc(C(=O)NC2(C(F)F)CCC2)no1.C(=O)(CCC1CCC1)N c1(CCC(=O)NC(COCCCNC(c2ccc(C)o2)=O)(C)C)ccccc1Cl CC(CCCNC(=O)CCc1cncn1C)NC(C1CCCC1C(F)(F)F)=O c1(CN(C2CCC(C)CC2)C(COC)=O)cnc(Cl)c(C)c1 C1(CNC(c2cn(C)nn2)=O)CC2(CCC2)CN1C(C1CCC2(CC1)CC2)=O N1(C(C2CN(C(C)C)C(=O)C2)=O)CC(NC(C2(CF)CC2)=O)CC(C)(C)C1 S(=O)(=O)(c1ccc2c(c1)NC(=O)CC(C)S2)N1CCOc2c(ccc(C)c2)C1 C(=O)(C1c2ccccc2OCC1(C)C)Nc1ccc(OCC)cc1C(F)(F)F O=C1CCC(C(=O)NC2CCCC2CNC(=O)C(c2ccccn2)O)=NN1 C(=O)(CCCCC(C)(C)C)N1CCCC(CC)C1C(=O)NCC12CC(CCO1)C2 C1(CNC(C(C=C=C)C)=O)CC(F)(F)CN1C(c1cc(O)nc(Cl)c1)=O C1(C(N2CC3C(NC(c4cccc(Cl)c4)=O)C(C3)C2)=O)CCc2nnnn2C1 C1(CNC(Cc2cccc(OCCC)c2)=O)CCC(C)(C)CN1C(=O)C(C)O N1(C(C2CC(=C)C2)=O)CC(NC(=O)CC2(N(C)C)CCC2)C(O)C1 N1(C(c2ccc(COC(C)C)cc2)=O)CC(C2CN(C(C34CCC3C4)=O)C2)C1 C1(C(=O)NCc2c(OC(C)C)ccnc2)CSC(c2ccccc2O)=N1 n1(CC)c(C(=O)NCCN(C(=O)CC)Cc2ccccc2OC)cnc1O C1(C(=O)NC2CC(C)SCC2)CC12CCN(C(=O)CCCCCF)CC2 c1(CC)cc(CNC(=O)C(O)C2CN(C(=O)Cc3ccnn3C)C2)no1 C1(CC(=O)NCCCOCCCC)CN(C(c2cc(C)[nH]n2)=O)CC1C CC(CC(C)(C)C)NC(C1CCCCC1NC(c1ccc(C(N)=O)o1)=O)=O N1(C(CCOC)C)CCC(NC(=O)C=Cc2cccs2)C(CN)C1 CCC(CC(=O)N1CCC(CNC(C2CCn3cncc3C2)=O)CC1)C(C)(C)C c1(NCC2(OC)CCSC2)cc(N2CCOC(c3cccnc3)C2)ncn1 N1(C(C2CCCC(OC)C2)=O)CCN(C(=O)Cc2ccon2)C2CCCC2(C)C1 c1(CN2CCC(C(=O)Nc3ccc(-c4ccno4)cc3)C2)cnc(Cl)nc1Cl N1(CC(=O)NC(CC)CNC(=O)C(C)(C)n2cnc(C)c2)Cc2ccccc2C1 c1(COC(C)C)ccc(C(=O)N)cc1.c1(C=O)[nH]ncc1C#N.C1(CC)CC1 Cc1cc(C(=O)NC2(C)CCCCC2)cc(O)c1.C1(C)(CC=O)CC1(Cl)Cl.N C1(CNC(CC(C)N(C)C)=O)CC(O)CN1C(=O)CC1CCCCO1 Cc1ncc(Cl)cc1CC(N1CCOC(C)(CNC(=O)CCn2cccn2)C1)=O C(=O)(C(S(N)(=O)=O)c1ccccc1)N1CC(C(=O)NCCCC)OCC1 N1(C(c2[nH]nc(CC)n2)C(=O)NCC)CCN(c2ccc(C(=O)OC)nn2)CC1 Cc1cnc(NCC(O)C(N)=O)c(S(=O)(=O)NCC(N2CCOCC2)(C)C)c1 C(=O)(C1CCc2nccn21)NC1CN(C(Cc2ccc(CC)c(F)c2)=O)CC1O c1(C(=O)NCC(C)CC2CCC2)cncc(CNC(=O)C(CO)N(C)C)c1 C(=O)(C1=NN2CC(C)CN=C2N1)N1CC(CCC)N(C(=O)C2=COCCC2)CC1 c1(CN2CC(CC)N(C(=O)C(C)(C)CC)CC2)ccc2cc[nH]c2n1 N1(C(C)=O)CCN(C(c2cnn3c2OCC3)=O)CC1c1ccncc1 N1(C(C(CC)(C)O)=O)CCOC2(CCN(C(=O)NCc3ccco3)CC2)C1 [N-]=[N+]=NC1CC(C(=O)NCC2CC(F)CN2C(=O)Cn2nnc(=N)[nH]2)C1 C12(CNC(C3CCN(CCC)CC3)=O)CCN(C(=O)NC3CC3)CC1C2 CC1C(C)N(C(=O)CCOC2CN(C(C3C(C)(C)C3(C)C)=O)C2)CCN1C CC1(CCC(=O)NCC=CC)CCC(=O)N1.c1(C=O)cnn(C2CC2)c1Cl.N c1(C(=O)NC23CC(CNC(CC4C(C)CCC4)=O)(C2)C3)ncc(Br)cc1O C1(NC(CN(CCCC#C)C)=O)CCC(C(=O)N(C)C)CC1 C1(NC(c2ccc(NC(C)=O)c(C)c2)=O)CN(c2ncns2)C2CCCCC12 NS(=O)(=O)c1ccsc1C(N1CCN(CC2NC(=O)CC2C(F)(F)F)CC1)=O c1(COCC)ccc(F)c(F)c1NC1CC1C=O.c1ccc(C=O)cc1 c1(C(N2CCC(F)(CNC(C(CCCC#C)C)=O)C2)=O)ccc2nc(=N)[nH]n2c1 N1(C(C2C(C=C)C2)=O)CCCC(N(C(=O)Cc2cccc(Cl)c2)C)C1.C1CC1 Cc1cc(C(=O)NC2(CF)CCN(C(c3cc(Cl)no3)=O)C2)c2c(C)n[nH]c2n1 c1(CC)ccccc1CC(=O)NC1CC(CNC(c2cc(C)c(C)o2)=O)C1 c1(C(C(=O)N(CCC)CCNC(=O)C(O)CN(C)C)C)ccccc1F c1(C(N2CCN(C(C3C(C)C3C)=O)CC2CCO)=O)cccc(S(C)(=O)=O)c1 c1(OC)cc(C(N2CCN(c3ncccn3)C(C(C)C)C2)=O)ccc1Cl N1(CC2CCCC(C)(C)O2)CC2CS(=O)(=O)C2C1 N1(C(c2ccc(NC(C)=O)o2)=O)CCC2CN(C(C3CCSC3)=O)CC12 c1(C(N(CCCCNC(c2cc(Cl)ns2)=O)C)=O)cccc2c1OCCN2 C(=O)(C1=CCC(NC(c2ccccc2Cl)=O)C1)NCC(CC)C(C)C n1(CNCC)ccc(=NC(=O)c2c[nH]nc2C2CC(NC)C2(C)C)[nH]1 C(=O)(CC(C)(O)C(F)(F)F)N1CCCC(CNC(C(C(C)(C)C)OC)=O)C1 N1(C(c2scc(C)c2C)=O)CCC2CN(C(c3cncn(C)c3=O)=O)CC2C1 C1(C(N2CCN(CC(C)NC(C(CCC)N(C)C)=O)CC2)=O)CC(F)(F)C1(C)C c1(C(N2CC(O)(C(C)NC(CNC(=O)NC)=O)C2)=O)ccnc2[nH]cnc12 c1cc(F)c(F)cc1O.c1(OC)ccc(Cl)cc1NC(C1CC(F)(F)CN1C)=O c1(C=O)c(F)cc(N)cc1F.C1(NC(c2nc(OCC)oc2)=O)CCOCC1.N c1(CC(N2CCCCC(NC(CSCC)=O)C2)=O)cccc([N+](=O)[O-])c1 N1(C(CC(C)(C)OC)=O)CC2CCOCC2(NC(=O)CN2C(=O)CCC2=O)C1 c1(OC)cncc(C(c2nnnn2C(C)C)NCc2nn(C)nc2Br)c1 CCCCCCC(=O)NC1C2CC1N(C(c1cc(OC)cs1)=O)C2C c1(OC(COC)C)nc(=NC2CCN(C(=O)OC(C)(C)C)C2)[nH]c2c1COCC2 [SH](=O)(=O)c1cccc(Cl)c1.C1CC(S(C)(=O)=O)C1.CCCC.[SH](C)(=O)=O.N C12(NC(C(C=C)O)=O)CC(CO)(C1)OC21CCN(C(=O)CC2(C)OCCO2)CC1 C12(C(N3CCC(C(=O)NC)C3C)=O)CCN(C(=O)C3=CCCCC3)CCC1C2 c1(C(N(CC(C)NC(=O)C(c2cccc(F)c2)O)C)=O)cccc2cnsc12 C(=O)(C1CCCc2scnc21)N1CCC(CCNC(c2cc(C)ncc2)=O)CC1 C1(N(C(CCCC)=O)C)CCCN(C(=O)C(C)(C)C(C)C)CC1.c1ccccc1Cl C(c1cccc(F)c1)=CCC(=O)N(CCCN(C(CC(C)C)=O)C)C.CC=O.N N1(C(c2cc(OCC)no2)=O)CCN2CCN(C(=O)Cn3cncn3)CC2C1 C1(C(=O)NC2CCN(C(=O)CCCn3cccc3)C2)CC2(CCCCO2)C1 c1(C(N(CC(CC)NC(c2nnc(S)n2C)=O)CC)=O)cccc(F)c1Cl c1(CN2CCC(NC(CCc3c(C)cccn3)=O)C(O)C2)c[nH]c2cnccc12 C1(CC(=O)NCC2CCN(Cc3ccnc(Cl)c3)CC2)NC(=O)NC1=O C1(C(=O)NC2C(Nc3ccc(C(N)=O)cn3)CCCC2)CCCC(F)(F)CC1 C1(C(N(C)CCNC(=O)CSc2ccccn2)=O)CCc2cncn2C1 CC(C)CC(CNC(=O)C(C1CC1)C1CC1)C(=O)N1CC(C)OCCC1C C1(C(N2C(C(=O)NOCCC(F)(F)F)C(O)CC2)=O)CC12C(=O)Nc1ccccc12 C1(NC(C(CC=C)NC(C)=O)=O)CCC2(CCN(C(c3cc[nH]n3)=O)C2)C1 C(=O)(CCCCC(C)(C)C)N(CC(O)CN(C(=O)COc1ccccc1)C)C C1(NC(C(C)OCCC=C)=O)CCC(NC(c2ccncc2C(F)F)=O)CC1 C1(OCC)CN(C(=O)CCCC2CCCO2)CC1C.C1(CC=O)CCC(O)C1 N1(C(C(=O)N(C(c2ccc(C3C(C)C3)o2)=O)C2CC2)=O)CC(C)CC1C N1(C(CCN(C)C)=O)CCCC(Cn2cc(CC3(O)CCCCC3)nn2)C1 c1(C(=O)NC(CC(C)C)CNC(=O)C(C)(O)C2CC2)cnc2[nH]c(O)nc2c1 c1(C(=O)NCCN(C)C(C2CC23CC3)=O)ccnn1CC1CCCO1 c1(C(N2C(c3c(OC)ccc(F)c3)CCC2)=O)ccc2c(N(C)C)nccc2c1 CC1CN(C(C2CC2c2ccc(Br)s2)=O)CCCN1C(C1(F)CC1)=O C1(C(=O)Nc2cn(COC)nc2)COCCN1C(c1cc(F)cn1C)=O C1(NC(c2c(C)onc2)=O)CC2CC(NC(=O)Cc3sccc3Br)CC12 CCCC(O)CC(=O)N1CCCCC(N(C)C(c2cc(C)nc(O)n2)=O)C1 c1(N(C(=O)CCC2CCCN2Cc2ccc(C#N)nc2)C)nc2ccccc2[nH]1 C12(NC(CC(=C=C)C)=O)CCOCC1CN(C(c1cnc(N)c(N)c1)=O)C2 N1(C(C(=O)NC(C)CN(C(=O)CC2(C3CC3)CC2)C)C)CCCCCC1 C1(Cc2cn(C3(C(N4CCCC(C(=O)OC)C4)=O)CC3)nn2)CCCCC12CC2 c1(-c2nccc(C(N3CC4C(C(=O)OC)C4C3)=O)c2)cccc(F)c1F CC(C)C(C(=O)N1CCC(O)C(N(C(=O)CC2COCCO2)C)C1)C(C)C O=C(C1=CCN(C(C2(O)CCCC2)=O)CC1)N1CC2CSCC(C2)C1 c1(OC)cc(C(=O)NCCCOCCCNC(C2CC(F)C2)=O)nn1C c1(C(CC=O)C)ccc(F)cc1.CC(O)CC.C1(C(=O)OCC)(C=O)CC1.N c1(C(N2CCC(O)(CNC(CSCCOC)=O)C2)=O)ccc2cccnc2c1N C1(N(C(=O)C(O)C2CN(C(=O)CC(C)(F)F)C2)C)CCCC1(C)O Cc1cc(Cl)ccc1NC(=O)CN1CCC(C)(C)C1C C=CCN=c1[nH]cc(C(=O)NCCCC(C)NC(=O)C(C)OCCOC)s1 c1(OC)ccccc1-c1cn(CCN(C(=O)CC2CCC3CC3C2)C)nn1 c1(N(C(CNC(c2nc(C)oc2)=O)Cc2ccccc2)C)ncnn2cccc12 Cc1ccc(Cl)cc1C(N1CC(NC(c2cc(Cl)ccc2C)=O)C(C)C1)=O C1C=CCN1C(=O)CCCc1ccncc1.CCS(=O)(=O)NC(C)C(=O)NC C(=O)(CCCc1ccc(Br)s1)NC1(CCNC(C=CC(CC)C)=O)CC1 N1(C(c2ncc(C)cn2)=O)CC2CCCC(CNC(C3(CO)COC3)=O)(C2)C1 C1(CCC)CN(C(=O)C=CC(C)CC)CCN1C(=O)Cc1ccon1 N1(C(C)=O)CC(NC(C2CCCC23CC3)=O)CC(C)(C)C1 c1(OCC#C)cc(F)ccc1.C1(c2nnnn2C2CC(F)(F)C2)(N)CC2CC2C1 C(=O)(C(C)(F)C(C)(C)F)NCC1OCCCN(C(CNS(NC)(=O)=O)=O)C1 CC1CN(C(=O)CC2C=NN(C)C2=O)CCC1.C12(C(=O)N)C(=O)C3CC1C2C3 c1(C(=O)NC2CC(C)N(C(c3cc(F)ccc3F)=O)C2)cc(F)c(N)cc1F CC1CCC(C)(C(N2CCN(C(=O)CCc3nncs3)C(CC(F)F)C2)=O)CC1 C1(CN(C)C)CCCN(C(=O)C(CN(C)C)NC(=O)CC2(O)CCCCC2)C1 C1(C(N2CC(CC3CC3)C2)=O)CCCN1C(C1COCCO1)=O C1(C(=O)NCC(CNC(C2(C#C)CC2)=O)(C)O)CC12CCC(F)(F)CC2 c1(C(N(CCC)CCNC(c2[nH]nc(OC)c2Cl)=O)=O)c(F)cccc1Cl N1(C(c2ccnc(C)n2)=O)CCCC(C)(C(=O)NC2CC3CCC2(CO)C3)C1 N1(C(C2C(COC)C2)=O)CC2CCN(C(c3n[nH]c(C)c3C)=O)CC2C1 Cc1cccc2oc(=NCC3CN(C(C4(CO)CCCCO4)=O)CC3C)[nH]c12 C#CCC(CC(F)F)NC(=O)C(CC(=C)Cl)NC(c1cc(C)c(CC)o1)=O n1(CC=C)cc(C(=O)NCC2(F)CCC2)cn1.C1(O)(CC=O)CCC1.N CC1CCC(C(=O)NCC(c2ccccc2)NC(c2c[nH]nc2Br)=O)O1 N1(C(c2cc(C)cc(F)c2)=O)CC(C)CN(C(=O)C2=C(Cl)CC2)C(C)C1 Cc1noc(C(C)C)c1NC(c1cc(CNC(=O)C(C)C#N)cs1)=O N1(C(COCC#C)=O)CC2CCN(C(=O)Cc3cc4ccccc4o3)CC(C2)C1 c1(C(=O)OCC)cc(C(N2CC(O)C2)=O)n(C)n1.C(=O)C(C)C1CCOC1 N1(C(C2CC(OC)CN2C(=O)Cn2ccc(C)c2)=O)CC2CC1CS2=O CCC(C)(C)CC(=O)N1CCCC(NC(c2cn(-c3ccccc3)nn2)=O)CC1 C1(NC(C=CC(C)C)=O)COCCN(C(=O)C(C)Oc2ccc(Cl)cc2Cl)C1 C#Cc1c[nH]nc1C(N1CC=CC(NC(=O)CS(=O)(=O)NC)C1)=O c1(C(N(CCN(C)C(c2c(N)cccc2F)=O)C)=O)cnc2c(cnn2C)c1O C(=O)(C1=C2CCN=C2NC=C1)N1CCC(CCNC(c2c[nH]nc2[N+](=O)[O-])=O)C1 C(=O)(C1CCc2ccccc21)N1C(C)(C(N2CCNC3(CCC3)C2)=O)CC1 N1(C(c2cc(C)ncc2)=O)CC2(C)CCC1C2.C1(=CC=O)CCC(C)(C)CC1.N c1(NC(=O)Nc2ccc(SC(CC)C)cc2C)cc(Br)c(C)cc1Cl N1(C(CSC(C)C)=O)CC(=O)CC1C(=O)Nc1cn(C)nc1Cl n1(CC)nc(C)cc1C(N1CC2CC1C2NC(C1CCC(C)(CC)O1)=O)=O n1(CC(=C)C)nc(-c2ccc(OC(C)C)cn2)nc1-c1ccc(CN(C)C)cc1 N1(C(C2N(C(CC)=O)CSC2)=O)CCC(CF)(NC(=O)C(C)CC)C1 C1(CNC(C(C)N(C(C)=O)C)=O)C(O)C(O)CN1C(c1cccnc1S)=O C1(C(=O)NCCNC(CCCCCC=C)=O)COc2ccc(F)cc2C1 c1(-c2c(C)cns2)nc(Cc2ccncc2)nn1C(C1CCC1)C C(=O)(CCCC(C)NC(C1CC12CCCC2)=O)NCc1cc(C)ncn1 N1(C(=O)OC(C)(C)C)CCC(C(=O)O)(C(=O)NCC2CCC(=O)O2)C1 C(CC(F)F)(C(=O)NCC1(CCO)CC1)NC(C(C1CCC1)OC)=O C1(CC(=O)NCC(CNC(c2cc(C(N)=O)co2)=O)OC)CCCCC1 c1(CC)cn2c(n1)CC(C(=O)NCCC1(O)CCN(C(=O)CCCS)C1)CC2 C1(C(N2CCC(C)(CNC(C(Br)=C(C)C)=O)CC2)=O)CCN2CCCC2C1 C1(CNC(C2(C)CCCS2)=O)CC2(CCC2)CN1C(C1CC(F)(F)C1)=O C1(NC(Cc2c(C)cc(C)s2)=O)CCN(C(C2(C(F)F)CCCO2)=O)CC1(C)C C1(NC(c2ccccc2)=O)CCN(C(=O)CCN2CCOCC2)C(C2CC2)C1 N1(C(c2cccc(C)c2Cl)=O)CCC2C(CCN2C(=O)CC2CCCO2)C1 C(C(COC)C(=O)NC(C1CCCN1C(C1CCC1(C)C)=O)C)OC C1(NC(=O)CN2C(=O)CNC2=O)CCCCN(C(c2c[nH]c(Br)c2)=O)C1 C(CS(=O)(=O)c1ccc(Cl)cc1)OC.C12(CC=CCC1)C(=O)OC2 C1(CC)(CC)SCCNC1C(=O)NCC(c1ccncc1)C c1(CC)cccc(C(N2CC(CCC)C2)=O)c1O.C1(CC(=O)N)NC(=O)NC1=O C1(C(=O)NC2(CC=C)CCN(C(=O)CC3OCCO3)C2)CC(C)OC(C)C1 c1(CC)ccc2cc(C(N3CC=CC3CC)=O)ccc2n1 c1(C(=O)NC2CCC(N(C(CCOCCOC)=O)C)C2)cnc(N)c(N)c1 c1(C(=O)NC)onc(NC=O)c1C.C1CC2(C1)CC2C=O.C(C)(C)C.N CC(C#N)CCC(=O)N1CCCC(CCNC(=O)CCCOC(C)C)C1 c1(OCC)cncc(C=O)c1.C1(C=O)(C(F)F)CC(F)(F)C1.C1CCC1.N Cc1cncc(C(=O)NCC(C)(CO)NC(c2cn(C3COC3)nn2)=O)n1 N1C(=NCCc2ccco2)NC2CC2C1.OC1CCCCC1OCc1ccccc1 CN1CCOc2ccc(NC(C34COCC3CN(C(C3CC=CC3)=O)C4)=O)cc21 N1(CC(=O)NC(C)C)CCCS1(=O)=O.N1(CC=O)CCCC(N(C)C)C1 N(C1CCc2ccccc21)(C(=O)CN1CCc2ccccc2CC1)CCO N1(C(CC=CC=C)=O)CCC2(CC1)CCN(C(c1ccc(CC)cc1)=O)C2 Cn1nccc1C(C(N1CC=C(F)C1)=O)NC(c1cnnn1C)=O Cc1oc2ncnc(O)c2c1C(=O)NC1CC2CC1CN2C(c1cnsc1)=O Cc1nc2cccc(C(N3CCCN(C(=O)CC(C)CF)CC3)=O)n2n1 N1(CCC#C)CCC(C(N2CCC(C)C2)=O)CC1.n1(CC=CC=O)cncn1.N C1(NC(c2cc(C)sc2)=O)CCCC12CCN(C(c1ncc(C#N)cc1C)=O)C2 C12(NC(CCC(C)SC)=O)CCC(NC(=O)CC3CN4CCC3CC4)(CC1)C2 C1(NC(CC2OCCN(C(C=Cc3n(C)ncc3)=O)C2)=O)CCC=CCCC1 C1(C(=O)NCC(C)NC(c2c(N)cccc2Cl)=O)CC2CC1C1CC21 N1(C(c2nc(C)sc2C)=O)Cc2[nH]nc(C(=O)NCC3(N(C)C)CC3)c2C1 CC(CC(=O)N1CCC(O)(CNC(c2coc(C#N)c2)=O)C1)C(C)(C)C C1(CC)(CC)CCN(C(=NCC(C)N2CCCC2)NCc2ccsc2Cl)CC1 c1cc(-c2nnc(COCc3cccnc3)o2)ccn1 Cc1c(NC(c2ccc(N3CCOC3=O)cc2)C)ncnc1N1CC=CCC1 C1(CC(=O)N)COC(=O)C1.C1(CC(N2CCC2)=O)OCCC1c1ccccc1.C N1(C(C(C)n2cncn2)=O)CCN(C(=O)COC2CC=CC2)C(C)C1 c1(C=O)cccc2nc(O)[nH]c12.c1(C(=O)NC2COCC2C)cc(=O)cc[nH]1.N Cc1noc(C)c1C(C)CC(=O)NCCNC(c1nocc1Br)=O c1(C(N2CC(F)CC(NC(=O)Cc3sccc3Cl)C2)=O)cccn2ccnc12 CCC(C(=O)NCC(C)(C)NC(=O)C(n1ccc(C)n1)C)C(C)C N1(C(N2CC3CCC2C3)=O)CCOC(c2cccc(OC(F)F)c2)C1 C(CNC(=O)Cn1cnccc1=O)(CC(F)(F)F)NC(=O)CO C1(C(=O)NCCOC2CN(C(C(C(C)C)=O)=O)C2)Cc2ccccc2C1C N1(C(CN(S(C)(=O)=O)C)=O)CCCC(O)C1.c1(C=O)coc(N(C)C)n1.C C1(C(=O)N(C2CC3CC3C2)C)(NC(c2scc(COC)c2)=O)CCCCC1 O=C1CCC(CC(N2CCC(=CCNC(C3CC34CCOC4)=O)CC2)=O)C(=O)N1 c1(CNC(c2nnnn2CCCC)CCOCC=C)c(C2CC2)cnn1C N1(C(C(C#C)(C)C)=O)CC(NC(=O)CN(CC(=O)N)C)CC(F)C1.C(C)C c1(CC)nocc1NC(=O)C(=O)NC1COCC1F C(C(CC(C)C)C(=O)NC1(C(=O)NCc2[nH]nnc2C)CCOCC1)OC N1(CCNC(C2(NC(C3C(C(C)C)OCC3)=O)CSC2)=O)CCCCC1=O C1(C(=O)NC(C(OC)OC)C)CCC(n2cc(-c3ccnc(C)c3)nn2)CC1 C(C1=NOC2CN(C(=O)CCNC(=O)CO)CC12)NC(C1(C=C)CC1)=O C1(CNC(=O)CSCC(F)F)C(O)C(O)CN1C(C1CC1(F)F)=O c1(C(N(CCCC)C)=O)cnc2c(c1)c(C)nn2C.C1(C(=O)N)CC(C(C)C)C1 C(=O)(C1=CC2CCCC12)NC(C1CCN(C(C2(n3cccn3)CCC2)=O)CC1)C N1(C(=O)CC(F)(F)Cl)CC2OCCN(C(c3occc3Cl)=O)C2C1 c1(OCC)ccccc1S(=O)(=O)N(CCC1CNC1)CCOCC C1(C(=O)NCC(CC)NC(=O)C(C)(C)C2CCOCC2)COC2(CCC2)C1 Cc1cc(Br)cc(F)c1C(N1CC2CC1CN2C(=O)COC1CCOCC1)=O C1(N(c2ncccn2)C)CCCC2CN(C(=O)CNC3Cc4ccncc4C3)CC12 CC(C)(CNC(=O)C=CCF)CC(=O)NOCCN1C(=O)CCC1=O C12(CN(CCN(C)C)CCN(C)C)CCC(F)(CC1)C2 C1(C(=O)NC(C(C)NC(c2cc(-c3ccccc3)c[nH]2)=O)(C)C)CC2CCC1C2 C(=O)CC(CN(C)C)C(F)(F)F.c1(C(C)=O)ncc(C(=O)N)s1.C1CC1.C C(=O)(C1=CC2CCCC12)NCCCN(C)C(c1ccsc1C#N)=O N1(C(Cc2nc(C)sc2)=O)CCC2(C(=O)NCC(N3CCOCC3)=O)CCCC12 Cc1ccc(Cl)c(N)c1C(N1CCC(CNC(=O)C(O)C2CCCC2)C(C)C1)=O CN1CCn2ncc(C(=O)NC3CCCC3CNC(=O)CS)c21.c1cn[nH]c1 Cn1cccc1-c1cc(C(=O)N(CCC#N)Cc2cnn[nH]2)n[nH]1 N1(C(C2C(C#C)C2(C)C)=O)CCOC2(C1)CN(C(C1CC13CCCCC3)=O)C2 C1(NC(C2(C)C(C)(C)C2)=O)CC2(C1)CN(C(=O)C=Cc1ccccc1)C2 CS(=O)(=O)c1nccc(N2CCC(F)(C(=O)Nc3cc(Br)nn3CCO)C2)n1 C1(CNC(CCNC(=O)OC)=O)CCN(C(=O)Cc2cnc(C)[nH]2)C1.C N1(C(c2c(CC)onc2)=O)CCC2CCC(C1)N2C(c1c[nH]nc1C)=O C1(C(C)(C)C)CCN(C(C2CC(C)(F)C2)=O)CC1.c1(C(C)O)ncc(C(=O)N)s1 N1(C(C2CC(=C)C2)=O)CC(C2CCN(C(c3cc(C(N)=O)co3)=O)CC2)C1 c1(C(N(CC(O)C(F)(F)F)CC)=O)cc2n(n1)CCCO2 c1(C(=O)NC2C(NC(=O)COCCCF)CC2)cnc(O)s1 CCCCCCCC(=O)NC(C)(CC)CCNC(=O)CC1(N(C)C)CCC1 C#Cc1ccc(C(N2CC(C)N(C(c3nc(C)nn3C)=O)CC2C)=O)c(F)c1 CN1CC(F)CC1CNC(=O)NCc1ccc(CC#N)cc1 C1(CNC(c2ccc(F)c(Br)c2)=O)CN(C(=O)CC2CCC2)CCCO1 C1(C(=O)NC2C(NC(c3c(CC)nco3)=O)CC2)(CF)CCOCC1 N1(C(C(Br)=C(C)C)=O)CC(NC(c2cccc(C(=O)C(F)F)c2)=O)CCC1C c1(C=O)c(C)[nH]c2ncccc12.c1(OCC)ccc(C(=O)NC2CCC2)nn1.N C1(N(C2CCN(C)CC2)C(=O)Cc2ccc(F)c(F)c2)CCC2(CC1)CNC2 N1(Cc2nc(C)c(C)s2)CCC2(CCN(C(c3cccc4c3OCC4)=O)C2)C1 C(=O)(CN=c1ccc(C#N)c[nH]1)NCC1CC(NC(C(C(C)SC)O)=O)C1 c1(C(=O)NCC2CC(NC(C3(C#C)CC3)=O)C2)nccc2occc12 N1(C(CCC(=O)OCC)=O)CCC(NC(c2csnc2Cl)=O)C(C(C)C)C1 NS(=O)(=O)c1ccc(C(N2CC3CC2CN(C(C2CCCC(=O)O2)=O)C3)=O)cc1 C1(C(N(CC(C(C)C)OC)C)=O)CCN(C(c2cccc[n+]2[O-])=O)C1C n1(CC)ncc(C(N2CC(NC(C)=O)C(c3ccccc3)C2)=O)c1C CC1CN(C(C2(CCF)CC2)=O)CC(CCNC(=O)C=CSc2ccccc2)O1 c1(C(=O)NC(C(=O)NC(CC=C)(C)C)COC)cncn(C)c1=O c1(OC)cc(C)c2cc(C(=O)Nc3ccc4c(c3)nnn4C)oc2c1 CC1(C)CC(CSCC(=O)NC(C)(C)C)CN(C(=O)NC2CC2F)C1 C1(C(=O)NC2CCN(C(=O)C=C3CCOCC3)CC2O)C2CCC3C(C2)CC13 C12(C(=O)Nc3cccc(CNC(C(C)OC)=O)c3)CCCC1CCC2 C1(CC(=O)NC2CN(C(C(C)(C)CC#N)=O)CC2O)CCCCCC1(F)F N1(C(CN(CC)CC)=O)C2CCCC1CC(NC(c1coc(C)c1)=O)C2 c1(C(N(CCCNC(=O)COC2CC(F)(F)C2)C)=O)nn(C)cc1N C(=O)(CC(C)(C)C#N)N(C(CCNC(c1cc(CCC)nn1C)=O)C)C N1(C(C2(OC(C)=O)CC2)=O)CCN(C(=O)CCC2CCCC(=O)N2)C(CF)C1 Cc1ccc(CC(=O)NC2CCOCC2NC(C2CC23CCC3)=O)cc1 C1(CNC(c2c(CC)non2)=O)CCN(C(c2cnccc2Cl)=O)CC1C c1(CC(=O)N(CC(C)NC(c2cc(C)[nH]n2)=O)CC)cc(Cl)ccc1O.O c1(C(N2CCCC(NC(CN(C)C3CC3)=O)CC2)=O)cnn2c1OCC(F)C2 CC1CCN(C(=O)CCCn2cc(-c3ccncc3F)nn2)C1c1cn(C2CC2)nn1 C1(C(=O)NCc2c(C(N(C)CC3C(C)C3)=O)cccn2)CN2CCC1CC2 c1(C2(C(=O)NC3C(CN(C(c4n(C)cnn4)=O)C)CCC3)CC2)cccnc1Cl C(=O)C1=CCOCC1.c1(C2CN(C(C=CC(=O)OCC)=O)C2)ocnc1.C c1(C=O)cc(=O)c2ccncc2o1.C1(CC(=O)NC2(C)CC2)CC(=O)NC1=O c1(NC2(CO)CCCN(C(CC3(OCC)CC3)=O)C2)ccc([N+](=O)[O-])cc1Br c1(CCC)nc(C)c(C(=O)Nc2cncc(C(=O)O)c2)o1.C12CCN1C2 N1(C(c2cncc(OC)n2)=O)CCC2CC2(C(=O)NCc2ncsc2C)CC1 CC(C(=O)NCC1(F)CCC(NC(c2cccc(C3CC3)c2)=O)C1)C(F)F c1(C(=O)NCC2(CNC(=O)CC3CC3)CCCC2)cc(C)ccc1F.S c1(NC(C(N2CC(OC)CC2COC)C2CC(CC)C2)=O)cccc(I)c1 N1(C(=O)CCCCF)CCC2(CCCN(C(C3CCCC34CCOCC4)=O)C2)C1 c1(CNCC(c2ccc(Cl)nc2)O)ccc(C(=O)O)cc1 c1(C(=O)N(c2nccc(-c3ccccc3)n2)CC2CCCN2)cccc(O)c1F c1(C(=O)OCC)ncnc(NC2CCN(C(C3CC34CC(OC)C4)=O)CC2)c1F c1(OC)nc(C)ccc1NC(C1CC(N=[N+]=[N-])CN1)=O Cc1ccc(NC(=O)C(C)CN(C)C(c2ccc(O)cc2F)=O)cc1C#N c1(C(=O)NC(CNC(c2cc(C)cc(F)c2)=O)(C)CO)ccc(C#N)c(O)c1 C1(CN=C(NCCc2ncc(C)s2)NC2CCCCC2C)CCC2(CC1)CC2 Cc1cnc2nccc(C(=O)N(CCNC(c3csc(Cl)n3)=O)C3CC3)c2c1 C1(C(=O)NC2CC(NC(C(c3cn(CC)nc3)=O)=O)C2)CC2(CCOC2)C1 c1(C(=O)NC23CC(NC(C=CSC)=O)(C2)C3)ccc(C2CCCC(=O)N2)cc1 Cc1cncc(CC(N2CC(N(C)C(C3CCCC3C)=O)C2)=O)c1 CC(C)C(C(=O)N(C1CN(C(=O)C(c2ccn(C)c2)C)CC1O)C)n1cnnc1 C1(c2cn(C(C)CNC(C3(C(=O)O)CCCCO3)=O)nn2)CCCC(F)(F)C1 N1(C(C(CC)(C)F)=O)CC(CO)C2(CCN(C(=O)CC(=O)OC)CC2)C1 C1(C(=O)NCC2N(C(CC(=O)N(C)C)=O)CC=C2)CC12CCC(C)(C)CC2 N1(C(Cc2cccc(C#C)c2)=O)CC2CC(NC(C3CCCC3F)=O)CC(C2)C1 N1(C(c2ccc(SC)s2)=O)CCC2(CC1)CC2.C1(C=O)(C(C)C)CNC(=O)C1 c1(SCCN2CCOCC2)cc(O)c2ccoc2c1.c12scc(c1Cl)C(=O)OC2=O N1(C(c2n(CCC)ncc2)=O)CCCCC(NC(c2ccc(C)nn2)=O)C1 CC1(C#N)CCCN(C(C2CCN(C(=O)C34CCCN(CC3)C4)O2)=O)C1 N1(C(CN(CCOC)C)=O)C(C(=O)NCC2(CCO)CCC2)CC1C Cc1ccc2sc(=NCC3(C)CCN(C(c4ccc(C)o4)=O)C3)[nH]c2c1 c1(C(C)=O)ccc(C(=O)NC(CCN(C(=O)CCc2nncs2)C)C(C)C)nc1 C1(C(N2C(C3CC3)CCC2)=O)CC2(C1)CC1(CCC1)C2.Cc1nnc(C=O)s1.N Cc1cc(C(=O)N(C)CCN2CCOC(C)(C)C2)cc2c1CCC2 c12ccc(Br)cc1CS2.c1(-c2ccc(C(=O)O)s2)ccc(C(F)(F)F)nc1 n1(CC(N2CC(NC(c3csc(O)n3)=O)C(O)C2)=O)ccc(Br)cc1=O N1(C(c2c(C(C)C)n(C)nc2)=O)CCC(CO)(NC(c2c[nH]c(Br)c2)=O)CC1 N1(CCCNC(NC2CC(N3CCC3)C2)=NCc2cc(C)on2)CC(C)CC(C)C1 C(C(C)CC(=O)NC1CC(CNC(c2cn(C3COC3)nn2)=O)C1)OC c1(CC)oncc1C(N1CCC(CNC(C2CCC(=O)O2)=O)C1)=O O=C(CCCCn1ccnn1)NC1CC(F)(CNC(c2ccc[n+]([O-])c2)=O)C1 CC#CCC(C(=O)NCCc1ccncc1)NC(c1sccc1CO)=O N1(C(C(=O)NCc2cn(CCN3CCC(C)CC3)nn2)=O)CCN(CC)C(=O)C1 c1(CCC(=O)NCC2C=CCN2C(C2(F)CCOC2)=O)ccc2ccccc2n1 C1(NC(c2ccc(CC)o2)=O)C2CC1CN(C(c1cc(F)ncc1OC)=O)C2 c1(C(=O)NC2C(CNC(C(N3CCSCC3)C)=O)CC2)c(Cl)nc2ccccn12 N1(C(CCc2onc(C)n2)=O)C2CCC1C(C(=O)NCC1CCOC1C)C2 c1(C(N2CCC(N(CC#C)C(c3cnn(C)n3)=O)C2)=O)ccc2occ(C)c2c1 c1(C(=O)NCC2C(NC(CCN(CC)CC)=O)C2)ccon1.N(C)C C(=O)(C(CC)C(F)(F)F)N(CC(CN(C(CCc1ccc(C#C)cc1)=O)C)O)C N1(C(c2c(C)n[nH]c2)=O)CC2=C(C1)CN(C(=O)CCc1ccnc(Br)c1)C2 c1(CC(=O)NC2C(NC(c3ccc(C)cc3)=O)CCOC2)nsc2ccccc12 c1(N2CCC(C)(CC)C2)nc(=NCC2CCCCO2)[nH]c2c1CCC2 N1(Cc2n(C)c(-c3ccc(F)cc3)cn2)CCCCCC1C1CC1 C1(CNC(C(CSC)O)=O)CC(C(=O)N2CC(N3CC(F)C3)C2)=NO1 c1(C(=O)NC2CC(NC(CS(N)(=O)=O)=O)C2)cc([N+](=O)[O-])c(N)cc1F C(CNC(=O)C(CO)NC(=O)C1CC1)(C(C)C)NC(C(F)=CC)=O c1(OCC#C)ccccc1OC(C)C.N12CCN(CC1)CC(=O)N(C)CCC2 C(=O)(C1=CCN(C(=O)C(C(C)(C)C)N(C)C)C1)N1C(C)C(N(C)C)CC1 N1(C(CC(C=C)(C)C)=O)Cc2ccccc2C(NC(=O)CSS(C)(=O)=O)C1 O=C(CC(C(F)(F)F)NC(=O)Cn1c(O)nnc1O)NCC(O)C1CC1 Cc1ccc(C(=O)NCC(C)NC(=O)Cc2c(C)cnn2C)cc1[N+](=O)[O-] CC(F)CC(=O)NCCNC(C1CN(C(c2coc(C(N)=O)c2)=O)C1)=O C12(NC(C3CCCC3c3nc(S)n[nH]3)=O)CC1CN(C(c1ccccc1Cl)=O)C2 C1(C(N2CC(C(=O)NCCO)C2)=O)(NC)CCOCC1.C1(C=O)SCCC1C CC(C)C(N=[N+]=[N-])C(=O)N1CCC2(CC2)CC1C(=O)NCC(C)C(C)O c1(NCCC(C=C)(C)C)ncc(S(=O)(=O)NCc2cc(C)ccn2)cc1Cl C1(C)(CNC(c2c(OCC)cccn2)=O)CCCCC1.C(=O)C(C)(Cl)Cl.N c1(N2CC(C(C)NC(C(CC)C)=O)OCC2)nnc2c(c1C(=O)OC)CCC2 C1(NC2c3ccccc32)CCc2nc(CC)cn2C1.c1(CC)cccc(Cl)c1F C1(NC(C(C)OCC)=O)CN(C(c2cnc(C(C)C)n2C)=O)CCC1C c1(C(N(C(C)CNC(=O)C=Cc2ncco2)C)=O)ccc(SC(F)(F)F)nc1 CCC1c2ccccc2CCN1C(=O)NC1Cc2ccccc2CC1O Cc1[nH][nH]c(=N)c1C(=O)NCCC(O)CNC(C1CCN(C)C1=O)=O Cc1cccc(CN2CC3CC2(c2cn(CC(O)Cc4ccccc4)nn2)C3)c1 C1(OC)C2CCN(C(=O)COC(C)(C)C)CC12.C12(C3CC3)CN(C1)C2=O C(N=c1ccn2ccnc2[nH]1)C1(CNC(Cc2nc(C)[nH]n2)=O)CC1 CC1CC(NC(=O)CCc2ccsc2)CN1C(=O)CCSc1ccccc1Cl C(=O)(CS(=O)(=O)N)N1CC(C)(NC(C2CCC(C(N)=O)C2)=O)C1.C1CC1 N1(C(c2ccn(C(C)C)c2)C(=O)NCCC)CC2(COC(C)C2)C1 C=C(C)CCCC(=O)NCC=CCNC(c1cccc(OC)c1)=O CN1CCCC1CCC(=O)NC(CC1CC1)C(=O)NCCC1CC=CCC1 c1(C(=O)NCC(O)CNC(=O)C(O)CC2CC2)cc(Cl)c(Cl)c(Cl)c1 CC(CC(=O)NCCC1CCCCN1C(=O)COc1ccc(O)cc1)C(C)(C)C C1(C(C)C)CN(C(=O)CCc2ccc(O)c(F)c2)CCN1C(=O)C(C)N(C)C c1(OC)ccccc1C=CC(=O)NCC.C(=O)(CS(=O)(=O)CC1CCC1)N c1(CNc2c(C#N)nccc2)cccc2c1C(=O)OC2 Cc1cc(C(N2CC(O)(C(C)NC(C3OC4CCC3CC4)=O)C2)=O)nnc1O Cc1cnc(C)c(NC(C2CCC(=O)N(c3cnn(C)c3)C2)=O)n1 C(C(C)CC(=O)NCC(C)C1CC1)OC.C(=O)(CN(C)C(=O)C1CC1)N CC1CCC(O)CN1C(=O)C(C)Oc1ccccc1F c1(C(=O)NCCC)ccccc1C1CC1(F)F.c1(C=O)cn(C)nc1C1CC1 C(=O)(CC1COCc2ccccc21)N1CC(NC(=O)COCCF)C(F)C1 c1(OC)cc2c(cc1C)CN(C(c1c(Cl)sc(Cl)c1C)=O)CC2 C1(OCCOc2ccc(OC)cc2)CCC2CNCC12 C1(C)(C(=O)OC)CCCN1C(c1coc(C2CC2)n1)=O.C(C)(C)(C)O c1(-n2c(C3CCCC3CF)nc(CCCCN(C)C)n2)cc(Cl)nc(Cl)c1 C1(C(N(CCN(C(C(CC)SC)=O)C)C)=O)CC(=O)C12CCCC2 c1(C(=O)NC2C3(CN(C(C(CCSC)O)=O)C3)CC2)cc(F)cc2ccoc12 C(C(C(=O)N(C1CN(C(c2cc(C)sc2C)=O)C1)C)C(C)(C)C)OCC=C c1(-c2cn(C)nc2)cncc(C(=O)NC2(C)CN(C(=O)CS)C2)n1.c1cccs1 c1(C(=O)NCC2C(NC(CCCn3c(C)ncc3)=O)C2)cccc(C2CC2)c1Cl C1(C(N2CC(C#C)(O)C2)=O)CN(C(c2cn3c(n2)CCC3)=O)C2(CCC2)C1 c1(C(N2CCCC2C2CCCOC2)C(=O)NCCCCCC)cc(Br)cnc1OC C1(C(=O)NCCN2CCCCC2)CC(F)CN(Cc2cccc(O)c2Br)C1 c1(CC)c[nH]c(=O)c(C(N2CCCCC(NC(C3CCCNS3(=O)=O)=O)C2)=O)c1 C1(C(=O)Nc2n(C(C)(C)C)ncc2C#N)CN(Cc2cncc(C)c2)CCC1O Cn1nc2c(c1C(=O)NCC1CN(C(C3(Br)CC3)=O)CC13CC3)COCC2 c1(OC)ccc(CN2CCSC(C(=O)NCc3ncc(C)s3)C2)cc1Br N1(C(CCCC(C)C)=O)CC2CCC(C1)N(C(=O)Cc1ncccn1)C2 Cc1cc(C)c(C(=O)CN(C)CC2(C#N)CCC2)c(C)c1O C1(CNC(C(C)OC2COC2)=O)CN(C(=O)CC2COC(C)(C)C2)CCO1 c1(C(=O)N)ccc2cccnn12.c1(NC(C)=O)ccc(C(=O)NC(C)CCC)s1 c1(C(N(CCCNC(C=CC(C)C)=O)C(C)C)=O)ccc(C#N)cc1F C1(CC)CN(C(c2ccccc2F)=O)CCC1NC(c1scnc1C(F)F)=O CC1CC(CO)CN1C(=O)C(=O)NCC(c1ccc(C(C)(C)C)cc1)(C)C CC(C)(CO)C(C1CC1)NC(=O)CC(O)CNC(c1ccoc1)=O C1(CC#C)(C(=O)NCCC(C)NC(=O)Cc2csc(SCC)n2)CCCO1 N1(C(=O)NC)CCC(C(=O)NC2CCC2)CC1.C1(C=O)CC(C)(C)CO1.C C(N=c1ccnc(NCc2cnn(CC3CCC3)c2)[nH]1)c1n(C)nnn1 C12(CNC(C(C(CC)O)C)=O)CC(C1)C1(CCC1)O2.C(=O)C(F)C1CCOC1 c1(NC(C2C(CCC(N3CC(c4nc(C)[nH]n4)C3)=O)C2)=O)cc2occc2[nH]1 N1(C(C(C)n2cncn2)=O)CCN(C(c2ccccc2)=O)C(C2CCCC2)C1 Cc1c(C(=O)NCCC(C)(C)NC(=O)Cc2cc(Cl)sc2Cl)cccc1N n1(CC)cc2ccc(C(=O)NCC3CN(C(c4cnc(Cl)s4)=O)CC3C)cc2n1 n1(CC(=O)N)cc(C)c(O)nc1=O.N1(C(c2cc(C)sn2)=O)CCC(C)(CC)C1 C=CCCCCCC(=O)NC(CNC(C1CC(F)CN1C)=O)CCCC C(c1ccnn1C)=CC(N1CC(CC=C)(NC(CCOCC#C)=O)C1)=O CCCC(C)C(=O)NC(CO)C(=O)NC(C)(C)CCF N1(C(C(C)OC)=O)CCC12CCN(C(C1CCc3ccccc3C1)=O)CC2 CC1(C)CCC(c2noc(-c3cn[nH]c3)n2)C1 C#CC1(C(N2CCSCC(C)C2)=O)CCN(C(c2cnc(C)cc2C)=O)C1 c1(C(N(CCC(C)NC(C(CC)N(C)C)=O)C)=O)nc(Cl)sc1C(C)C C1(CCC)C(=O)NCCN1C(c1n[nH]c(C)n1)C(=O)NCc1ccccc1Cl O=C(CC1=NNC(=O)C1)NCC1CN(C(=O)CC2SC3=NCCN3C2=O)C1 N1(C(c2ccc(CN(C)C)nc2)=O)CCC2(CCN(c3nccnc3C#N)C2)C1 c1(CC(=O)NC2CC2)ccc(F)cc1.C1CCCN1C(=O)CC1CCC1.C c1(C(C)=O)ccccc1OCC(=O)NC1CN(C(=O)C(F)C2CCOC2)CC1C c1(NC(C2CSCCN2Cc2ncc(C(F)(F)F)[nH]2)=O)ccc(F)cc1Cl Cc1cc(C(N2CC(NC(c3c(C)cccc3F)=O)C(F)C2)=O)cnc1F CC(C)CCCC(=O)N(C(=O)C(N)C(C)N(C)C)c1ccccc1 c1(CCC(=O)NCC2CC(NC(=O)COCCCF)C2)cnc(O)[nH]1 c1(NC(=O)NC2(c3c(CC)cccc3)CC2)cccc(S(N)(=O)=O)c1Cl C(=O)(CCCc1cncs1)N(C1CC(C(=O)NC2(C3CCCO3)CC2)C1)C c1(C(=O)N)noc2c1COCC2.C(C)(CO)NC(=O)C=CC(=O)NC1CC1 C1(NC(c2c(CNC(C3(C#N)CCCC3)=O)ocn2)=O)COCC1C1CC1 C(CN=c1ccnc(NCCc2ccc(F)nc2)[nH]1)(C1CCOC1)OC Cc1nc(=NCC2C(C)CCC2C)[nH]cc1Br CC1(C)CCC(NC(=O)CC2CC3(CC3)CN2C(=O)CCCF)CC1 c1(C(C)C)ncc2c(n1)CCN(C(c1cnc(C(F)(F)F)cc1Cl)=O)C2 C1(NC(=NCC)NCc2nc(OC)c(C)s2)CCCN(c2ccc(F)c(F)c2)C1=O N1(C(CC(C=C)(C)O)=O)CCOCC(C)(CNC(=O)CCC(C)C)C1 n1(CC(N2C(C)CC(NC(c3ccc(Cl)c(F)c3)=O)C2)=O)ncc2cccnc12 C1(CC(=O)NC2(CNC(=O)C=CC3CCOC3)CCOC2)CCOCC1.C N1(C(c2ccn(C)n2)=O)CC(NC(c2ccc(F)c(C(F)F)n2)=O)CC(F)C1 Cc1c(C(N2CCCC(CN(C)Cc3ncc(Br)s3)C2)=O)cccc1O C1(CNC(C2(C=C)CC2)=O)CN(C(c2cocc2Br)=O)CCC1(F)F CCC(C(=O)OC)C(=O)NCCNC(=O)Cc1cnco1 N1(C(C)=O)CCCC(C(N2CC(CNC(=O)CC)C2)=O)C1.C1(C=O)CCC1 c1(C(=O)NC2CN(CCOC)C2)cccc(C(C)C)c1 c1(C(=O)NC2C(NC(CC3(C)CC3)=O)C2)cc2ccc(C(F)(F)F)cc2[nH]1 C1(CC=O)CS(=O)(=O)CCN1C.N1(C(C=CCC)=O)CCC(C(F)(F)F)CC1 CCS(=O)(=O)CC(=O)NCC(C)NC(C1CCC1CF)=O N1(C(C#CC(C)(C)C)=O)CCCN(C(=O)CSCc2cccs2)CC1CO N1(C(CC2(C=C)CC2)=O)CCC(C(C)NC(=O)C(C)OC)CC1 C(=O)(CCCN(C)N=O)N1CCN(C(CC(C)OC)=O)C(C2CC2)C1 c1(C(N2CCC(NC(C3CC(=C)C3)=O)C(F)C2)=O)sccc1S(=O)(=O)NC c1(C(=O)NC2CN(C(c3cn(C)nc3Cl)=O)CC2F)ncnc2c1CCC2 C#Cc1ccc(C(=O)NC(C)(CNC(=O)CC23CCCC2C3)C(C)C)cc1 C(=O)(C(CC1CCC1)NC(C1CCCN1C(C)C)=O)NC(CC)CN(C)C C1(CCC)CCCN(C(=O)C=C(C)C(C)(C)C)C1.C(=O)C(C)(C)C1CCNC1 c1(C(N2C(CNC(C3CCCCC3O)=O)CC(F)C2)=O)cnn2c1CCCC2 N1(C(c2cc(C)sn2)=O)CCC(NC(c2nc(Cl)sc2Cl)=O)C(C)C1 C1(C(=O)NOCCCC=C)(CC#C)CCN(C(C2C3CC(=O)CC23)=O)C1 C1(CNC(C=CC(CC)=CC)=O)CC(C)CO1.C(=O)(C(C)(F)F)N C1(=O)CCC(C)N1.C(CCC(C)C)OCC(=O)N(C(CC#C)C)CCO N1(C(C)=O)CCC(N(C)C(C2CC(C)(NC(=O)COC3CCC3)C2)=O)C1 N1(C(C2(C)CC(=C)C2)=O)CC2CCCC2(NC(=O)C(CC(C)C)n2ccnc2)C1 N1(C(CNC(COC)=O)=O)CCC2(CC1)CC2NC.c1ccccc1.C(C)C CCCCC(=O)C(=O)N1CCN(C(c2c(OC)noc2C)=O)CC1C1CCC1 S(=O)(=O)(c1ccc(F)cc1)N1C(C(=O)Nc2cnccn2)CC(F)C1 C1(C(=O)NCCCCC)CCCCC1(C)NC(=O)CCNC(N)=O N1(C(CCC=C(C)C)=O)CC2(C1)CN(C(=O)COC1(O)CCOC1(C)C)C2 c1(N(C(C(n2c(C(CSC)(C)NCCOC)nnn2)C)=O)C)cccc(C)c1C C12(C(=O)NC(C)CCCCNC(c3ccncc3O)=O)CC3CC(C(=O)N1)C2C3 CC1(Cc2ccc(F)cc2)CCCN1Cc1c(Cl)cnn1C(C)(C)C C1(C)(NC(CCN(S(C)(=O)=O)C)=O)CN(C(=O)CO)C1.C1CCCOC1 C1(C)(C(=O)Nc2c(C)ocn2)CCCN1c1nccc(Oc2ccccc2)n1 C1(C(N2CCC(C(=O)NCC3C(CC)C3)CC2)=O)CCC(C2CC2)C1 C1(CC=C)CN(C(=O)C)C1.n1(CC=O)cnc(C(F)(F)F)n1.C1COC1.N C1(C(N(CC(F)F)C)=O)CC12CCN(C(C1(C)CCCCCC1)=O)C2 C1(C(N(C2CN(C(C3(CC)CC3)=O)CC2F)C)=O)CC2(CCCC2)C1 N1(C(COC)=O)CCN(C(=O)C=CCF)CC(C)C1 C(C(=O)Nn1nnc2c1CCCC2)C1CCN(C(CC)=O)C1 C1(COCC)(CNC(=O)CC2CNCCC2C)CCCCC1 c1(NCCCC(=O)NC2(CF)CCN(C(C(C)SC)=O)C2)ccccc1[N+](=O)[O-] N1(C(c2ccc(C(C)=O)cc2F)=O)C2CCC1CN(C(C1CC1(F)F)=O)CC2 C(CCCCCC(=O)N1CCOC(CF)C1)NC(C1C(C)(C)C1(F)F)=O Cc1nn2c(C(=O)NC)c(C)nc2s1.C1(C=O)CCCC(O)C1.C12CC(C1)C2 Cc1nc2c([nH]1)C(C(=O)NC1CCCN(C(=O)C(Cl)=CCl)CC1)CCC2 Cn1cnc(C(=O)NCCCCc2cn(CC3CCCCC3)nn2)c1 S(=O)(=O)(c1ccc(OC)cc1)NC1CN(CCOC)CC1C c1(CNC(C2(NC(CC(=O)OC)=O)CCC2)=O)cc(=O)cc(C)[nH]1 C=C=C(C)CC(=O)N1CC2C(CN(C(=O)CN3CCC(OC)C3)C)C2C1 C1(NC(C2(CC)CCN(C(c3cc[nH]n3)=O)C2)=O)CC2CCCC2C1 c1(C=O)nc(C(F)(F)F)ccc1N.C(C)(C(=O)NC)OCCCC.C1CCC1 c1(OC)ncccc1NC(C1C=CCN(C(=O)C(C)(O)C2CC2)C1)=O N1(C(C2CC(OCC)C2)=O)CCCC2CCN(C(c3ccnn3C)=O)CC12 CCC(C)C(C)CN=c1nc(N2CCC(N(C)C)CC2)c2cc(Cl)ccc2[nH]1 C1(NC(C(COC)(C)C)=O)CC(OC)CN(C(c2cnn(CC(C)C)c2C)=O)C1 C1(CCNC(c2c(C)nn[nH]2)=O)CN(C(=O)C=Cc2cncn2C)CC1C C1(CCC(=O)NC2(CSC)CCC2)CCN(C(C2CCC(CN)C2)=O)C1 C1(CNC(C2N(C(C)C)CCC2)=O)CCCN(C(=O)CC2(O)CC2)C1 N#Cc1ccncc1C(=O)NC1(CC(N2CCC3(CCO3)C2)=O)CCCCC1 N1(C(=O)CC2CCC(O)C2)CCOCC1c1ccc(F)cc1 c1(OC)nccc(=NC(=O)C2CC3CN(C(c4cc(C)c(Br)cc4C)=O)CC3O2)[nH]1 C(C(C)(O)C(=O)N1CC(CC(C)NC(=O)CC2CCCS2(=O)=O)C1)OC N1(C(CNC(C(CC)C)=O)=O)CC2(C1)CN(C(c1cc(F)ccc1N)=O)C2 C(=O)(C(C(C)C)NC=O)NCCN(C1CC1)CC.c1(CCC)c[nH]cn1 N1(C(C=CC)=O)CCC2(CC1)CN(C(c1ccc(SC)c(SC)c1)=O)CC(C)O2 CCC(C)(C(=O)NCC1CC1NC(=O)Cc1ccccc1)C(N)=O.CC c1(C(c2nnnn2C2CCCC2)NCC(C)(C2CC2)OC)cccc(C)c1Br C(CN=c1ccc(Cl)n[nH]1)NC1C(C)CCOC1 N1(C(CC(C)F)=O)CCCCC12CC(NC(C1CCc3nn[nH]c3C1)=O)C2 C1(CNC(c2n(CC)ccc2)=O)CC2(CCN(c3nc(OC)ncn3)C2)CO1.O C1(C(N2CCCC(C(F)(F)F)CC2)C(=O)NC2(C)CC2)CC2(C1)OCCO2 c1(OCC)ccc(CCC(=O)NCCC(O)CNC(c2ccnn2C)=O)cc1 n1(CC(=O)NCC2C=CCN2C(=O)CCC2CCCCCC2)cnccc1=O n1(CCC)cc(C(=O)NCC2(NC(C3CCOCC3)=O)CCC2)c(C)n1.C C(=O)(CC(C)P(C)(C)=O)N1CC(CNC(CCCc2c(C)ccs2)=O)OCCC1 C1(CC)(NC(=O)COC2CCCOC2)CCCN(C(C2(CCO)CC2)=O)C1 N1(C(C(C=C)(C)O)=O)CC2CCCC(NC(c3ccc(C(F)F)c(F)c3)=O)C2C1 C(C)(C)(CCCCC(=O)NCC(CC(C)C)NC(=O)CCN1CCCC1=O)OC C1(C(=O)NCCS(C)(=N)=O)CC(NC(=O)CNc2ncccn2)C1(C)C c1(C(C(=O)NCC2CN(C(C3(O)CC3)=O)CC2O)O)ccc(Cl)cc1Br N1(C(=O)NC(CC2(CC(=O)OC)CC2)(C)C)CCC(C)C(C(F)(F)F)C1 c1(-c2c(C(N3CCC(C)(O)C3)=O)cccn2)cccc2c1OCC2 C1(NC(C2C=CCCC2)=O)(CF)CCN(C(c2cc(=O)cc[nH]2)=O)C1 c1(CC(N2C(CNC(CCC=C(C)C)=O)CCC2)=O)cncc(O)c1 c1(C(NCCC)=O)c(C(C)C)nn(C)c1Cl.C(=O)(C=O)NCC.C1CC1 C1(NC(=O)Cc2ccc(Cl)cc2)CC2COCC(C1)C2NC(=O)CCN1CCC1 c1(N(C)C)cccc(C(=O)NC2CC(F)(CNC(C3C=CCC3)=O)C2)n1 C#CC1CCCCCN1C(=O)C(Cc1ccc[nH]1)NC(=O)OC(C)(C)C N1(C(C(n2cc(Cl)cn2)C)=O)CC2CCN(C(c3ccn(C)c3)=O)C(C2)C1 c1(CO)ccsc1NC(c1nnnn1CC1CC1)(C1CCOCC1)C Cc1c(C(N2CCC(F)(C(=O)NCCC(N)=O)C2)=O)cccc1Br CCCCC(C(=O)N1CC(CC(C)NC(=O)Cc2nccs2)C1)ON=C(C)C CC(C(C)(O)C(=O)NCCC1(C)CC1)c1ccccc1.C1(C=O)CSCN1C.N c1(NCC2(C)CCCC(=O)N2)[nH]c(=NCc2cn[nH]c2)nc2sccc12 C1(C(=O)NCC=C2CCN(C(C(C)S(C)(=O)=O)=O)CC2)CCCCC(F)(F)C1 C1(CNC(C(CNC(Cn2c(C)nnn2)=O)(C)C)=O)C(=O)NCCC1C c1(C(=O)N)cnc2cc(Br)ccc2c1.c1(CNC(C2CC2)=O)cc(F)ccc1Br C(=O)(C(F)C(C)(C)O)N(C)CC1CN(c2nnc(C(F)(F)F)s2)CCO1 CCCCCC(C)CC(=O)N1CC2(C1)CN(C(=O)C(C)(O)C(F)(F)F)CCO2 N1(C(C2C(C)(C)C2)=O)CC(NC(C2(C(F)F)CC(O)C2)=O)C(O)C1 N1(C(CSCC#C)=O)CCC(C(C)NC(c2cnc(N(C)C)nc2)=O)CC1 C1(C(=O)NCC2C(CNC(c3c(CC)n[nH]c3)=O)C2)CC2CCC1CC2 C1(C(=O)NCC(CCC)NC(CC=C)=O)CCCC(CF)C1 CC(C)C(CN1CCCCC1)NC(=O)Nc1nnc(O)s1 C1(NC(c2nsnc2O)=O)CN(C(c2ncsc2C(F)(F)F)=O)CCC1F N(C(=NCCN1CCOCC1)NC1CCS(=O)(=O)C1)C(C1CCOCC1)C#C Cc1ccccc1-c1ncc(CNCc2n[nH]cc2Br)cn1 C1(NC(c2n(CC)nc(C)c2)=O)CN(C(c2cnn(C)c2Cl)=O)C2CCCC12 n1(CC)nc(C)c(C(=O)N(CCCC(C)(C)C)C)c1C.C(=O)(CS(N)(=O)=O)N C(=O)(N=c1nc[nH]n2cccc12)C1CCC2(CN(C(c3cc(Br)cs3)=O)C2)O1 N1(C(C(C)=C(CC)C)=O)CC(OC)C(C(=O)NCCC(O)CC)C1 C(C1CN(C(=O)CP(C)(C)=O)Cc2ccccc21)NC(C1COC(C)(C)O1)=O c1(C(N2CC(C(C)NC(=O)C(C)Cc3ccncc3)C2)=O)cccnc1O CC1(C)CN(C(=O)C2CC2)CCC1NC(C1CCN(c2cccc(Cl)c2)C1=O)=O c1(C(c2n(C(CC)(C)C)nnn2)NCCC(C)(C)F)cnn(C)c1C(C)C N1(C(C=COCC)=O)CCCC(C)(NC(C2CC2c2ccccn2)=O)C1 C1(C(=O)NC2CCC2c2ccccc2)(OCC)CCOCC1 c1(CNC(=O)NC(c2nc(Cc3ccccc3)no2)C)csc(Br)n1 C1(NC(CS(N)(=O)=O)=O)CCC12CCN(C(C1CCCC(F)(F)C1)=O)CC2 c1(C(N2C(CN(C(C=CC=CC)=O)C)CCC2)=O)cc(Br)c(C)cc1C C1(C(=O)NCCCCCN(C(=O)C)C)COCCC1(F)F.c1(C(=O)N)ccoc1 N1(C(Cc2ccc(C)c(Cl)c2)=O)CCC2CCN(C(c3occc3C)=O)CC2C1 C1CC2(CCC2)CN1C(C1(CCO)CC1)=O.CN1CCC(OCC(=O)N)CC1.C c1(C(N2CCCC(NCc3n(C)cnc3)C2)=O)cc2cccnc2cc1F C1(CC(=O)N(CCN(C(=O)COC2CCC2)C(C)C)C)CCC(=O)NC1 c1(C(N2CCN(C(C(CC=C)C)=O)C(C)C2)=O)cc2cccc(O)c2[nH]1 c12cccc(c1)NC2=O.C1(NC(=O)COC2CC2)CCN(CC2CC2)C1 C1(C)(C(=O)NCCSCC(=O)NCC(C(C)(C)O)F)CC2CCC1O2 N1(C(CC=C)=O)CC2CC(Nc3nccc(C(F)(F)F)n3)C2C1 C1(NC(C2CCC(C)O2)=O)CN(C(c2csc(C(F)F)n2)=O)CCC12CCC2 c1(-c2n(CCC(=O)NC)c(N3CCS(=O)CC3)nn2)ccc([N+](=O)[O-])cc1C c1(C(N(CCN(C(C2C(C)(CC)C2)=O)C)C)=O)cc(Br)cc(F)c1F C1(NC(c2nn(C)c(O)c2)=O)CN(C(=O)C(F)(F)Cl)CC12COC2 [nH]1cccnc1=O.C(=O)(C(O)C(F)F)NC1(C)CN(C(=O)Cc2cn(C)nn2)C1 C(C(C)(C)C(C)(C)C)NC(C1C(NC(C2(C=C)CCCC2)=O)CCOC1)=O C1(C(N2CCC(N(C(=O)C(C)=CC)CC#C)C2)=O)COCCOC1 C1(F)(CNC(c2coc(Cl)n2)=O)CCCCC1.C12(C=O)CC3CC1C2C3.C C(=O)(C(C)CC(C)(C)C)N(C(CC)C(=O)NCC1CN(C(C)C)C1)C c1(N(C)C)cccc(CCC(=O)NCc2ccc(C)cn2)c1.C(=O)C(C)(C)O.N C#CCCCC(=O)NCC1CC(OC)CN1C(=O)CCCCN(C)C C1(C)(C(=O)NCCN(c2nnc(C3CC3)s2)CCC)CCC(F)(F)C1 Cc1ccc(C(C)NC(c2cc(F)cc(Cl)c2)(C)C)c(Cl)n1 C1(C(=O)NCCOCC(C)O)CCC(NC(C2CC(N=[N+]=[N-])C2)=O)CC1 C(N=c1ncnc2[nH][nH]c(C)c1-2)C1(C)CCN(C(CCCSC)=O)CC1 N1(CC(=O)N(CCC)C)C(=O)CC(C)(C)C1=O.CC=O.C(=O)OCC.N c1(C(=O)NCCCO)cn2c(n1)CCN(Cc1cnoc1)CC2 c1(C(=O)NC(C)CNC(C2(CO)CCCO2)=O)cccc([N+](=O)[O-])c1N c1(C(=O)NC(C)CCCNC(=O)CC2CCC2)ccc(O)nc1 c1(C(N2CC(C)N(C(c3cc(Cl)c(Cl)n3C)=O)CC2)=O)cnc2n(c1=O)CCS2 N1(C(c2cc(CC)oc2C)=O)CC(NC(c2c(Cl)n[nH]c2C)=O)C2CCCCC12 Cc1cc(-c2ccc(CNC(c3cncc(F)c3)=O)cn2)cnc1O Cc1nc(CNC(=O)CN2CCCC(C(C)(F)F)C2)sc1Br Cn1cncc1C1CC1C(=O)OCC(c1ccccc1)F N1(C(c2cc(C(=O)OC)sc2)=O)CCN(C(C2C=CCC2)=O)CC(C)(F)C1 c1(C(=O)NC2CN(C(=O)Cc3cn[nH]c3)CC2C(F)F)cnn2c1NCCC2 c1(C(=O)OCC)cccnc1C=O.n1(CC=O)ccnn1.C1(CC)CC1.N c1(C(=O)OC)cc(C(=O)NC(C)Cn2cc(C3CCC(=O)CC3)nn2)ccc1Cl C(=O)(C1=CC2(CCN(C(=O)COCCS)C2)C1)Nc1cc(CC)c(C)nc1 O=C1NC2CN(Cc3cnc4cnccn34)CC2NC1=O c1(OC)nc(C(=O)NCC(C2CCC2)NC(=O)C(C)SC)sc1C N1(C(c2cnc(SC)nc2O)=O)CC(N=c2[nH]nc(-c3cccnc3)s2)CC1C C(=O)(C1=NN(C)C(=O)CC1)NC1C(C(=O)NCc2c(C)nn(C)c2)C1 CC(C)S(=O)(=O)CC(=O)NCCN(C(=O)CC(C)n1ccnc1)CC(C)O C[S+](C)CCC(O)C(=O)N1CCCC1C1(NC(=O)CC2COCCOC2)CC1 C1(C(C)C)CC(NC(C2CCC(NC(=O)C(C3CCCCC3)=O)C2)=O)CO1 C1(CC(N2C(C(=O)OC)CC2)=O)C2CCCC2N1C(=O)C(O)CN1CCCC1 c1(CN2CCCC(F)(C(=O)Nc3cccc(CC)c3)C2)c[nH]c2cccc(F)c12 C(=O)(C1=COCCC1)NCC(C(=O)NCCc1onc(CC)n1)N(C)C c1(C(N2CCN(C(CC(C)NC(N)=O)=O)CC2)=O)ccc2cnnn2c1 CCCC(C)C(=O)NC(Cn1cncn1)C(=O)NCc1cscn1 c1(C(N2CC(C(=O)N(C3COC(C)(C)C3)C)CC(C)C2)=O)ccn2nccc2c1 Cc1cccc(C(N2CC(CNC(C3(C)CCCS3)=O)C3(CC3)C2)=O)c1C N1(C(c2c(C)c[nH]c2)=O)C(C(=O)Nc2cncc(Cl)c2)CCC1C1CC1 c1(C(=O)NC2CCC(NC(Cc3cc(C)ns3)=O)CC2)cccc2c1OCO2 C(=O)(C1=NOC(C)C1C)N(CC(=O)NC1CCC(=O)NC1(C)C)CCOC C(C(=O)NCC(C)(O)CC(C)C)(C(C)(C)C)NC(C(CC)N(C)C)=O C(=O)(CC(CC)C(C)C)N1C(CCCC)CN(C(C2C(C)C2C)=O)CC1 CCCC(CNC(=O)CC1(OC)CN(C(C2(C)CC(=O)N(C)C2)=O)C1)CCO CCCC(CNC(=O)C(C)(C)C(N)=O)C(=O)NCCOC(CC)CC C1(NC(c2cc(CSC)c(C)s2)=O)CC2CN(C(=O)C3=CCSC3)CCN2C1=O C(=O)(CCCC(F)(F)F)NCC1(C)CCN(C(c2cccc3[nH]ncc23)=O)CC1 C1(C)(C(=O)NC(CC)CN(C(=O)C(Cl)=CCl)C)CCC(=O)N1 C12(NC(c3nccc(OC)c3)=O)CCC(F)(CC1)C2 CC(CC(=O)NCC1(C2(O)CN(C(=O)C(N)=O)C2)CC1)P(C)(C)=O C(=O)(C(CNC(=O)C(O)C1CCC1)CCC)NCC(CCC=C)O N1(C(c2ccc(C(=O)OCC)cc2)=O)CCC(C)CC1.C(=O)(C1=CCC1)N c1ccc(Cl)nc1.c1(C(=O)NCCNC(C2C(C)(C)C2)=O)csc(Cl)n1.C C1(C#N)(C(=O)NC(C)CC2CN(C(=O)C(C)CC(N)=O)C2)CC2C=CC1C2 C1(NC(C(Cn2cccn2)NC(c2nc(CC)oc2)=O)=O)CC12CCCCCC2 N1(C(C(C)(C)c2cccnc2)=O)C2CC1CN(C(C1CCCC(CF)C1)=O)C2 c1(C(C)C)c[nH]nc1C(=O)NCC(C)NC(=O)CN1CCOC1=O Cc1ccc(C(=O)N(CCCCNC(c2cn(C)cn2)=O)C)c(F)c1F C=CCC(C(=O)NCC=CC)NC(C)=O.c1(C(CC(=O)N)C)ccccc1C c1(OC)cnc(C(=O)NC2CCC(CC(=O)NCCN3CC=CCC3)CC2)cn1 CC1CCC(NC(=O)CC2CCN(C)CC2)CN1C(=O)CSc1ccccc1 C1(C(=O)NCC(COCC)C)CCN(C(c2cc(Cl)c[nH]2)=O)C(C)(C)C1 c1(C(N2CC(NC(c3nc(C(C)OCC)sc3)=O)C(O)C2)=O)cccc(O)c1Cl O=C1CC(C(N2CCOCCC2C(=O)NC2CN(CC(F)F)C2)=O)NC(=O)N1 N1(C(c2c(C)con2)=O)CC(NC(=O)C(C)(Cl)Cl)C(C)(C)C1 c1(C(N2CCC(c3ccco3)C2)C(=O)NCCOC)cccn(C)c1=O C1(CNC(=O)CCC2CCCCCC2)CC2(CCC2)CN1C(C1SCCCS1)=O c1(CC)c(C(N2CCCC(N(C)C(C3C4CC5C(C4)C35)=O)C2)=O)cccc1C C(C(C)(O)C(=O)NC1CCCCC1CNC(=O)C(C)=C1CCC1)OC CCCC(O)C(=O)N1CC(C)(OCC(=O)N(C)Cc2cc(C)ccn2)C1 CCC(C)(C(=O)N1CC2CC1CN(C(c1cnc3cc[nH]c3c1)=O)C2)C(F)F C=Cc1ccc(C(N2CC(NC(=O)C(F)(F)C(O)C3CC3)C(C)C2)=O)cc1 C1(C)(CNC(C2C(C)C2)=O)CN(C(c2cc(Cl)n(C)n2)=O)CC1C c1(CC)ccc(C(N2CCC(C)(C)C2)=O)c(N)c1.C(=O)C(C)S(C)(=O)=O.C C1(C2CCN(C(c3ccncc3F)=O)C2)(NC(c2c[nH]c3cccnc23)=O)CC1 C(=O)(C(C)N1C(=O)C(C)Oc2ccccc21)Nc1ccc(NC(CC)=O)cc1 CC1(C)COc2c(C(=O)NC3CN(C(=O)CC4=CCCCC4)CC3O)cnn2C1 c1(N(C2CCC(C)C2)C)ccc(-n2cc(-c3cnn(C)c3C(F)(F)F)nn2)cc1 c1(CC)ccc(C)c(C(=O)N(CC(C)(C)NC(C2C3CCC(=O)C23)=O)C)c1 N1(C(C(Cc2c(OC)cccc2)=O)=O)CCOCC(CNC(=O)C(O)C2CC2)C1 CCC(C)C(=O)N(C1CCN(C(=O)CC2(O)CCCC2)C1)CC N1(C(CCNC(=O)OCC)=O)CC2(CC(NC(=O)CC(CO)C)C2)C1 N1(C(Cc2nc(COC)sc2)=O)CC2(CCC2)C1.C1(CC=O)CCC2CC12.C C(C)(C(=O)NOCCN(C)C)(N(C)C(C1CC(C2CC2)C1)=O)C1CC1 C(=O)(CCCCCCCSC)NC1C2CN(C(C3CCN(CC)C3)=O)CC1C2 c1(CC=C)ccccc1C(=O)NCCCNC(c1c(C)cnn1C)=O.C1CC1 C1(NC(c2cccc(CSC)c2)=O)CCN(C(=O)CCO)CC1(C)C.C1CC1 C1(C(=O)NCC2CC(NC(Cc3n(C)cnn3)=O)C2)COc2cc(F)ccc2C1 C(=O)(CC(O)CNC(C1CCO1)=O)NC(C)Cn1cnnc1 N1(C(C2(C)CCC(=O)NC2)=O)CCC2(CCCC2NC(C2(F)CCCC2)=O)CC1 C1(NC(C(CC)Oc2ccccc2C)=O)COC(C)(C)CO1 c1(C(N2C(C)CN(C(c3coc(Cl)n3)=O)CCC2)=O)ccc2ccccc2c1F CC1Cc2cc(F)ccc2CN1C(=O)Nc1ccc2c(=O)[nH]ccc2c1 c1(C=O)cc2n(n1)CCCO2.C(C)C(=O)N(C(C)C1CC1)C.C(C)OCC N1(C(=O)Nc2c(CCN)cccc2)CCC2CC(NCCN3CCOCC3)C2C1 C(=O)(C#CC1(C)CCCO1)NC12CCCN(C(c3n(C)cc(Cl)c3)=O)CC1C2 c1(C2C(C=O)C2)cc(F)cc(C#N)c1.n1(CC)cnc(C(=O)NCCC)n1.N C(c1cccnc1)=CNC(=O)C=CCNC(=O)C=Cc1cn[nH]c1 N1(S(=O)(=O)Cc2ccc(F)c(F)c2)CCCC2(CCC2O)C1 c1(SC)ccc(C(=O)NCC2CC(F)(C)C2)cc1.c1(C=O)cnccc1C.N C(C(=O)NCC(=O)OCCCC)(C(C)(C)O)NC(COCCC=C)=O c1(C(=O)NC2C(OC)CN(C(=O)C(C)O)C2)csc(S(C)(=O)=O)c1 Cc1cccc2c1CN(C(C1CCCC1NC(c1nccn1C)=O)=O)C2 c1(CN2C3(C#C)CC(C2)C3)ccc2ccc3ccccc3c2n1 c1(CC2CC(OCC)C2Nc2ccccc2)ccc(C(F)(F)F)nc1 CC(C)CC(CNC(=O)Cn1cnnn1)C(=O)NCC1CC(CN=[N+]=[N-])C1 C1(c2cn(C3C(NC(COCCCC)=O)COC3)nn2)(CO)CCCOC1 C1(C(=O)NC(C)CNC(C2(CF)CC2(F)F)=O)CCCC(CF)C1 N1(CC)CCOCC1CNC(=O)N(CC(F)(F)F)C C1(CNC(=O)CCc2cnc[nH]2)CCCCN(C(C2(C(F)F)CCCO2)=O)C1 C1(NC(C2N(Cc3n(CC)ncc3)CCC2)=O)CC(=O)N(CC)C1.C(C)C CC1CN(C(c2cc(O)ccc2O)=O)CC(C)N(C(=O)Cc2ccco2)C1 C=CC1(CNC(=O)CC2CCN(C(C3CCOC3)=O)C2)CCC1 C(=O)(C1=CC2C=CC1C2)NC(C1CC(NC(c2cccc3c[nH]nc23)=O)C1)C N1(C(CSCC)=O)CC2CN(C(C34CCCN(CC3)C4)=O)C(CO)C2C1 S(=O)(=O)(c1ccc(Cl)cc1)NCC1(C(=O)O)CC2CCC1CC2 c1(N2CC(CN(C)C(C34CCCC(C)(C3)OC4)=O)C2)nc(Cl)nc2[nH]ccc12 CCC(C(C)(F)F)NC(=O)CCN(CCCO)C(=O)Cc1ccns1 Cc1cccc(C)c1C(N1CC(NC(c2cc(Br)nn2C)=O)CC(O)C1)=O C1(CCNC(c2cnn(CCN3CCCCC3)c2)=O)CC2(CCO1)CC2 C=C(F)C1(CC(=O)NC23CC2CN(C(=O)Cc2ccnc(O)c2)C3)CCC1.C C(=O)(C(CC=CCl)c1ccccc1)N1CCC(NC(C2(C=C)CC2)=O)C1 Cc1cc(=NC2CCN(C(C3CC(C(C)(C)C)=NO3)=O)C2)[nH]cc1C#N CC(C)(C)C(CC(=O)N1CCC2(CC1)CC(NC(=O)C1=CCCC1)CO2)C(F)F C1(C(N2C(C)CC(NC(=O)CCc3cccnc3)CC2)=O)CN2CCN1CC2C N1(C(c2c(N)ccc(N(C)C)c2)=O)CCC2(COC(CNC34CC(C3)C4)C2)C1 c1(C(=O)NCC2C3CN(C(C(COC)OC)=O)CC32)cn2c(n1)CCCC2 CC1CN(C(=O)CCC2(C)CC2)CCC1NC(C1(C)CCCS1)=O C1(NC(c2n(CCCC)ncc2)=O)CCCC(NC(=O)C(C2CCC2)OC)C1 c1(C(N(C2CCN(C(=O)CCCF)C2)CC)=O)cc2c(o1)CCCC2 c1(C(C)(C)C)ocnc1C(=O)NCC1CCN1CC(=O)NC.c1ccco1 C1(C(N2C(C(C)NC(Cc3c(C)cccn3)=O)CCC2)=O)CC(C(C)(C)C)=NO1 c1(C(=O)OCC(C)C2CC2)ccn(CCOC(=O)NC(C)(C)C)n1 N1(C(CN(CC)CC)=O)CC(C)N(C(=O)CCc2c(C)n[nH]c2C)CC1C C1(C(=O)NCCN(C(=O)C(CO)NC(=O)C(F)(F)F)CC)CCCSC1 N1(C(C=C(C)c2cccs2)=O)CCC2CC(C1)CN(C(=O)C(C)C1CCCC1)C2 c1(CC)nc(C(c2nnnn2C2CCOCC2)NCCCNS(N)(=O)=O)cs1 Cc1cc(C(N)=O)cc(CCC2CC2)c1.c1ccc(N2CCN(C(C)C)CC2)cc1 C(C)(N=c1cc(C)nc(N2CCC(F)C2)[nH]1)c1ccc(NC(CCC)=O)cc1 Cc1cc(C(=O)N(CC(O)CNC(c2cn(C)ccc2=O)=O)C)c2occc2c1 CC1CN(C(=O)CS(C)(=O)=O)CCC1CNC(=O)COc1cn[nH]c1 N(C)(C1CCCc2ccccc21)C(CNc1cc(CC)c([N+](=O)[O-])cc1)=O C1(NC(C(CC#C)O)=O)CC2(NC(c3n[nH]cc3OC)=O)COC1C2 C1(OCCCNC(CCC2CCC(C)O2)=O)CCN(C(=O)CC2(O)CC2)CC1 c1(CNC(C2C(C)CC2)=O)cc(C(=O)NCCC2(C)CCOC2)no1 S(=O)(=O)(c1ccc(NCC2CC(C)(C)CCC2O)c(Cl)c1)N(CCC)CC C12(CNC(c3c(C)c(N)ccc3)=O)CCCC1CCN2C(=O)CSC(F)F C1(C(N2CC(C)(NC(C3CC(C4CC4)=NO3)=O)C2)=O)CC12CCC1(CC1)CC2 Cc1ccc(NC(c2cnc(OCCN3CCC3C)s2)=O)cc1 C1(C(N2CCC(C)(NC(c3cnc(N(C)C)o3)=O)C2)=O)CN2CCN1CC2 C(=O)CC1CCc2cc(Br)ccc21.CC(C(=O)NC1(C)CC1)OC(C)(C)C.N C1(C(=O)NCc2c(CC)nn[nH]2)CCN(C(=O)CN)C12CC2.c1ncccn1 CC1CSCCCN1C(=O)C(CC(F)F)N(C)C(c1csc(F)c1)=O C1(CC)CN(C(=O)CN2CCCS2(=O)=O)CCN1C(c1cc(CO)ccn1)=O C(=O)(C1=CC2CCCCCC12)N1CCC(NC(C2(O)CC(C)(C)C2)=O)C(O)C1 C(=O)CC(C)CC(C)(C)C.N1(C(c2n(CC)ncn2)=O)CC(COC)CC1C c1(CC)cccc(F)c1.c1(CC)cccc(Cl)c1.C12(C=O)CC(C=O)(C1)C2.N N1(C(c2cc(C(C)C)[nH]n2)=O)CCC(C)C1C.c1(C(=O)N)cncs1.C1CC1 c1(NCc2ccc(C=CC(=O)OCC)cc2)cc(C)nc2c(C)cnn12 N1(CC2CC(C)CC(C)C2)C2CCCC1CSC2 C(C(O)CC(=O)NC(CO)(CO)CO)NC(C(CC)OC)=O c1(CNC(=O)Nc2cc(C(CC)CC)no2)cc(OC)ccn1 c1(OCC(N2CCC(NC(C34COC(CO)(C3)C4)=O)C2)=O)c(Cl)cccc1Cl n1(CCC(=O)NC23CC(NC(c4nc(C)sc4)=O)(C2)C3)cnc(C)cc1=O N1(C(c2cc(NC)nn2C)=O)CC(O)CC1(C)C(N1CC(C)(CSC)C1)=O N1(C(CCC2(C)CC2)=O)CC(C(N2CCC(C(F)(F)F)C2)=O)CCC1(C)C C1(OC)COCCC1CC(N1CC(NC(C2CCN(C(N)=O)CC2)=O)C1)=O C12(CCC(C)(C)C1)C(=O)N2.C1(CCNC(c2c(C)ccs2)=O)CCCC12CC2 N1(C(CC(CC)CC)=O)CC(C)(C(=O)NCC(O)Cn2cccn2)CC1(C)C C#CC1CN(C(=O)C(CNC(=O)C(C)(O)C2CC2)N(C)C)CCN1C c1(CN2CC3C(C(=O)NCCn4cccn4)C3C2)ccc(Cl)cc1F N1(C(C(c2c(C)ccc(C)c2)C(C)C)=O)CC(C)CN(C(=O)C2CC2)C(C)C1 C1(NC(C(C)OCOC)=O)C2CCC(C2)C1C(=O)NCCCc1nc[nH]n1 c1(CCC(N2C(CC)C(NC(C3CC3(Cl)Cl)=O)CC2)=O)cc(OC)ccc1.O C1(NC(C=Cc2ccc(C)o2)=O)CN(C(=O)C(O)C(C)(C)C)C2(CCCC2)C1 CCCC(C)(O)CC(=O)NC1CCC(CNC(C2CCC(C)(C)O2)=O)C1 C1(CCNC(CCCOCC)=O)CCCN(C(C2(O)COC2)=O)C1 Cc1ccc(CC(=O)NC2CCN(C(c3cnn(C)n3)=O)CC2F)cc1C C1(OC)CC(C)N(C(c2ccc(C(F)F)nc2)=O)C1.C1(C=O)CCC(O)CC1.N N1(C(CCN(CC)CC)=O)CCN(C(c2cc(C3CCC3)on2)=O)CC(C)(F)C1 c1(C(N2C(CCNC(C3(C)ON=C(C)C3)=O)COCC2)=O)cc2occc2s1 N1(C(c2ccc(NC)c(F)c2)=O)CCC2(CC1)CN(C(C)=O)CC2CO N1(C(C2C(CC)C2)=O)CC2(CNC(=O)C(=Cc3c[nH]cn3)F)CC1CO2 c1(C(C(=O)NCC(CNC(CSC)=O)C(F)(F)F)C)cccc2ccccc12 C1(CC)CN(C(=O)CCNC(c2sncc2C)=O)C(CC)CO1 C(C(=O)NCC(F)C)(C(F)(F)F)OC(C)=O.c1cccc(F)c1.C(=O)C.N Cc1ncc(Cl)cc1CC(=O)N(C)CCN(C(=O)COC1CCCC(C)C1)C Cc1ncc(CC(=O)NCCC(C)N(C(=O)CC2CC2C)C)[nH]1 C=C1CCC(C(=O)NCC2CC2CNC(c2csc(Br)n2)=O)CC1 N1(C(C(COCC)(C)C)=O)CCC(C)(C)CC1.c1(C=O)n[nH]c(C2CC2)n1.C C1(CC)CN(C(C2C3CC(=O)CC23)=O)CCO1.c1(C(=O)N)cn[nH]c1.C1CC1 c1(C(N2CCC(CCC=O)CC2)=O)cnn2c1OCC2.C(=O)CC1CC1.CC.O CC1CN(C(=O)CNC(=O)CCCC(=O)C2CC2)CC(C)(C)C1 N1(c2ccnc(N(C)Cc3ccco3)n2)CCN2C(=O)N(C)C(=O)C2C1 c1(NC(C(C2CN(C(C3CC4(CCC4O)C3)=O)C2)OC)=O)ccc(Cl)cc1C N1(C(C(C)SC)=O)CC(NC(c2csc(C)n2)=O)C(C)C1 N(C(=NCCCCl)NC1CC(c2ccncc2F)C1)C(C)CC1CCOC1 c1(C(=O)NC(CNC(c2n[nH]c(C)c2C)=O)C2CCC2)ccc2ccncc2n1 C1(CCNC(CC(=C=C)C)=O)CC2CCC(C1)N2C(=O)Cc1cccc(F)c1F N1(CCCCC)CCC2(CC1)CC2(C)CNCCCOCc1ccc(F)cc1 N1(CCCCNC(C(C(C)C)F)=O)CCCN(C(c2cnsc2)=O)CC1 c1(CNC(=NCCC#C)NCCCc2nnc(C)s2)ncccc1S(C)(=O)=O N1(C(CC2CCC(=O)N2)=O)CC2(CC(NC(=O)C(CO)c3ccccc3)CO2)C1 N1(C(CCCCC=CCCC)=O)CC(O)CC2(CCCC2)C1 c1(CC)cc(CNC(=O)C(C(C)C)NC(=O)C(O)CN2CCCC2)ccn1 c1(-n2ccc(C)n2)ccc(C(=O)NCCCn2cc(C3CCN(C)C3)nn2)cc1 c1(C(=O)NC(CC2CCN(C(C(C=C)O)=O)CC2)C)cccc2cnn(C)c12 C1(C(C)C)Cn2nccc2CN1C(=O)C(n1cc(C(C)(C)C)nn1)C c1cccc(C2(C(=O)N)CC2)c1.c1(NS(CC)(=O)=O)cc(C(=O)O)on1.C c1(OC)cc(C(C)CC(=O)N2CCCC2CNC(=O)C=CC2CC2)ccc1C N(C1CCCc2ccccc21)(C(c1cnc(COC2CC2)s1)=O)CC N1(C(C(CCSC)N(C)C)=O)CCN(C(c2c(Cl)cnn2C)=O)CCC1C n1(CC(=O)NC(c2cccc(C)c2)CNC(=O)CCS(C)=O)ncc(O)nc1=O C1(C=O)C2CN(C(C3CC(O)CN3C(=O)CC3CCC(C)(C)C3)=O)CC12.C c1(CCC)ccc(C(=O)NCCC2CCCCN2C(=O)CN=S(C)(C)=O)cc1N N1(C(c2c(OC)n(C)nc2)=O)CC2CCCC(C1)N2C(=O)C(C)CCCC(C)=O C1(C(N(CC(=O)N(C2CN(C(C)C)C2)C)CC2CC2)=O)COC(=O)N1 N1(C(CNC(=O)OCC)=O)CC2CN(C(c3ccc([N+](=O)[O-])s3)=O)CC12 C1(NC(CCNC(=O)OC)=O)CC2(C(=O)NCc3cccs3)COC1C2 C1(NC(c2cnc(Cl)s2)=O)CC12CCN(C(=O)C=Cc1cnccn1)CC2 N1(C(C=CC=CCC)=O)CCC(NC(=O)C(F)=C2CCCC2)C(CO)CC1 c1(C(CC)NC(C(=O)N(C(CSCC)C)C)=O)ccc(Cl)c(Cl)c1 N1(C(C2(Cc3n(C)ccn3)CC2)=O)CCCCC(NC(=O)C)C1.C(N)(=O)N N1(C(C(CCOC)NC(c2c[nH]c(=N)o2)=O)=O)CCCC(C)(C)C1C c1(C(=O)NC(C)Cc2nn[nH]n2)cc2ccc(Cl)cn2c1 c1(C(N2CC(CNC(c3c(C)ccnc3)=O)CC2(C)C)=O)ccn2nnnc2c1 CCC(C)(C(=O)NC1CN(C(c2cccc(CC(C)C)c2)=O)CC1O)C(N)=O c1ccc(F)cc1.C(=O)(CCC(=O)N1CCCC1CNC=O)NC.C(C)C.N C(=O)(CC(C)C(F)F)NC1(CC(=O)NCCC(C)N(CCC)C)CC1 C(=O)(C1Cc2ccc(F)cc21)N1CCCC(NC(=O)CCSC(F)(F)F)(CO)C1 C=CC(C)(O)CC(=O)NC(C1CCCC1)CC1CCN(C(=O)Cn2ncnn2)CC1 C1(NC(c2c(C)[nH]nc2CO)=O)CC(NC(c2cnncc2O)=O)C12CCC2 N1(C(c2cnc(OC)nc2)=O)CCC(NC(c2cnc(O)n2C)=O)CC1C C1(NC(Cc2c(C)non2)=O)CC(N=c2nc(C3CC3)[nH]s2)C12CCC2 c1(OC)cc(C(=O)N)nc(C)n1.C1CCN(C(=O)C(C)P(C)(C)=O)C(C)C1.C c1(C(CNC(=O)NC(c2ccccc2)Cc2ccon2)O)ccc(F)c(F)c1 C(c1ncc(C)[nH]1)=CC(=O)N(C1CCN(C(c2ccn(CCCC)n2)=O)C1)C C1CCN(C(=O)CC2CCC2)CC1C.c1(CC)noc(COCC(=O)N)n1.C Cc1ccc(C(N2CCC(C(C)(C)NC(c3nncn3C(C)C)=O)C2)=O)cc1C C(C(CC(C)C)Nc1cccnc1)(c1nnnn1CC)NP(C)(C)=O.CCCCCC Cc1ccn(CC(N2CCCC(N(C(=O)CCc3cnco3)C)C2)=O)c(=O)c1 N1(C(CN(C)CC)=O)CC2CC3CC2C1C3NC(c1ccc(C)s1)=O C1(C(=O)NC2C(C(N(CC(COC)(C)C)C)=O)C2(C)C)CCCN1C=O n1(CC)cnc2c(N3CC4CCC3C4)[nH]c(=NCC(CCOC)OC)nc12 c1(CNc2ccc(C(=O)Nc3c(OCC)cccn3)nc2)ccc(Br)cc1Br N1(C(C=CCCC)=O)CCN(C(c2noc(C3CC3)c2C)=O)C2CCC12 N1(C(CN(CC)CC)=O)CCCC(N(C(=O)C(C2CCOCC2)O)CCO)C1 CCCCC(C(=O)N1CC2CC(C)C2C1)NC(C1CC2(C1)CC21CC1)=O C=CC1(C(=O)NCC2CN(C(c3onc(CC)c3C)=O)CCC2C)CCCCC1 C(CC(=O)N)(C(F)(F)F)NC(c1cc(C(C)C)no1)=O.C12CCC(CC1)O2.C c1(CC)ccc(C(=O)N(CCCNC(C23CCCN(CC2)C3)=O)C)cc1Br N1(C(CSC)=O)CCC(C)C(CNC(c2n[nH]c(CC)c2C)=O)C1 N1(C(CCC#CC)=O)CCOCC(C(=O)NC(CO)CCC)C1 Cc1[nH]nc(C(=O)NCC(CC2CCCC2)C(=O)NCC2CCN(C)CC2)c1O c1(C=O)ccc([N+](=O)[O-])o1.CCCCCC.C12(C=O)CC(C(C)(F)F)(C1)C2.N C(CCCC(C)NC(C1(C)CC1Br)=O)NC(CN(C(=O)OC)C)=O C(=O)(CS(=O)c1ccc([N+](=O)[O-])cc1)NCCCN(C(c1ccnn1C)=O)CC N1(C(C2(NC(C)=O)CC2)=O)CC2(CO)CC1(C(N1CC3(CCOC3)C1)=O)C2 C1(C2CCC2)(CNC(CC(CC)(C)C)=O)CCN(C(c2ccncc2)=O)CC1 c1(NC2(CNC(c3cnoc3C)=O)CCCC2)ncnc2c1ncn2C1CC1 C1(CNC(C(CC)(C)C)=O)CC(NC(=O)CCc2ccc(F)nc2)C12CCC2 C1(NC(CCc2n(C)ccn2)=O)CC(NC(c2cccn(C)c2=O)=O)C12CCC2 Cc1cc(=NCCC(C)(C)CO)[nH]c(NC2CCc3c(C)cccc32)n1 C1(CNC(c2c(C)nc(C)s2)=O)CN(C(C2CC3CC2CO3)=O)C(C)(C)C1 CCC(CC(=O)NC1CC(C)(NC(=O)CC2CCOCC2OCC)C1)C(F)F N1(C(c2nc(C3CC3)cs2)C(=O)NCCOC)CC(CO)C(CO)C1 c1(C(=O)NC2(CCNC(C(C(C)C)SC)=O)CC2)ccc2c(c1)SCCN2 N1(C(C2C(C=O)C2)=O)CCC(C)(CC)CC1.c1(C=O)c(Cl)cnn1C.CC.O c1(CC(=O)NC2CCC3(C2)CN(C(=O)CC2CCC2)C3)cnc2ccccn12 C1(C(N(C2CCOC2)CCNC(C)=O)=O)=CC=CN(C(c2cc(Br)cs2)=O)C1 Cc1ccc(Cl)c(C(N2CCOCCC2C(=O)O)=O)c1 C1(CCOC)(NC(=O)CCc2cn(C)nc2C)CCN(C(C2CCCN2C)=O)C1 C1(NC(c2c(OC)csc2)=O)COCCN(C(c2cc(F)ccc2I)=O)C1 C1(C(C)C)CN(C(=O)C(N)=O)CCCN1C(=O)Cc1ccc(Br)cc1 c1(CC(=O)NC(C2CCCN(C(C(C(C)C)N(C)C)=O)C2)C)ccc(O)c(F)c1 c1(C(=O)NCCN(C(CCC=C=C)=O)C2CC2)cnn2ccncc12 c1(C(=O)NC(C(C(C)C)C)CNC(=O)CC2=CCCC2)ncsc1S(N)(=O)=O N1(C(C(N2CCCC(NC(C)C)C2)=O)=O)CCCC2(CCC(=O)N2)C1 c1(C(=O)NC(CN(C(=O)CC(C)OC)CC)C)ccc(S(=O)(=O)NC)o1 c1(SC)ccccc1C(=O)NC1CC1CNC(=O)CCC1CC1(Cl)Cl C1(C(N2CC(C(C)NC(c3cc(C(F)(F)F)cs3)=O)C2)=O)CC2CCC1C2 c1(C(N2C3CC(CNC(C4C(C)(C)CC4)=O)(OC3)C2)=O)cnc2[nH]cnc2c1 C1(c2ncc(C)s2)CCCN(C(c2snnc2C)C(=O)NCCCF)C1 N1(C(c2ncn(CC)n2)=O)CC2CCC2(C)C1.C1(C=O)CC2C(C1)C2(F)F.N C(CN=C(NCc1c(C)nn(C)c1C)NC1CC1C)N(C1CC1)CC Cc1cc(C)n(CCC(=O)NC2(CO)CCN(C(=O)Cc3ncoc3C)C2)n1 N1(C(c2ncc(CC)s2)C(=O)NCCCCCC)CCC(O)(COC)C1 C1(C(=O)NCC(CNC(CNS(CC)(=O)=O)=O)CO)CC=C(C)CC1 C(C(C)CC(=O)N1CC(NC(c2cnc(S)[nH]2)=O)C(n2ccnn2)C1)OC C(=O)(CCCS(C)(=O)=O)N(C1CCC(NC(=O)COC(=O)CO)CC1)C Cc1cnc(=NCCNC(c2ccc3c(C(C)(C)C)csc3c2)=O)[nH]c1 c1(CCc2cn(Cc3scc(C(=O)OC)n3)nn2)cc(Cl)ccc1Br C1(C(=O)NC2(C(=O)NCCOCC(N)=O)CC2)OC2CCC1C2 C1(Cn2cc(CC(=O)O)nn2)Cc2ccccc2CN1C(=O)C(F)n1ccnc1 c1(N(C)C(N2CCC2)=O)cnn(CC2CCC2)n1.[nH]1cc(C2(C)CC2)nn1.C c1(C(=O)NCC2(C)CC(NC(c3c[nH]c(=NCC)s3)=O)C2)ccc2nc[nH]c2n1 c1(C(=O)NC(c2ccccn2)C)ccc(Br)cc1[N+](=O)[O-] N1(C(c2ccc(C(C)C)s2)=O)CCN(CC(C)NC(c2ccncc2Cl)=O)CC1 C1(NC(C(CC)SC)=O)CCN(C(c2cccc(F)c2)=O)C1CC C1(NC(C=CSC)=O)CCCC(C)C1.c1(CC(=O)N)cc(C(F)(F)F)n(C)n1 C(CCCCCC(=O)N1CC(NC(=O)C(F)=CCCF)CCC(O)C1)SC C(=O)(C(C)CC(C)C(C)=O)N1C(CC(=O)N(C(CC)C)C)C2CCCC21 C(C(F)(C(=O)NCC(C)CCCO)C(C)C)NC(c1ccnc(OC)n1)=O C(CCCCC(=O)NCCC(=O)NC1CC1)NC(CC(C)F)=O c1(CCC)cc(C(=O)NC(Cn2cncn2)C(=O)NC(c2cscn2)CO)n[nH]1 C1(NC(C2C(C)C2)=O)(CF)CCN(C(C2(c3ccccc3Cl)CCCCC2)=O)C1 c1(C(N2CCCC(CC(=O)N(CC#C)CC)C2)=O)ccc2cc[nH]c2c1 CC1CCCCC1CC(=O)N(C)CC1CN(C(C23CCC(C2)OC3)=O)CCO1 C(=O)(C(F)(F)C(F)(F)F)OC(c1nnnn1-c1ccccc1)C c1(C(N2C(CNC(c3ccnc(O)c3)=O)CC(OC)C2)=O)nn(C)c(Cl)c1Cl C(=O)(C#CC1CCCOC1)NC1CC2(CCN(C(CN3CC(C)(C)C3)=O)C2)C1 c1(OCC)ccc(C(c2nnnn2C2(C)CC2)NC(C)C(C)(C)C)cn1 N1(C(c2c(OC)cncn2)=O)CCC2CCN(C(=O)C(C)CC(F)(F)F)CC12 C1(C(C)C)CN(C(c2nccn2C)=O)CCN1C(=O)CCCOc1cccnc1 Cc1ccc(CC(N2CCCCC2CCNC(c2ccnn2CC#N)=O)=O)cc1 C(=O)(CCC(=O)N(C1CN(C(=O)C(C2CCCCCC2)O)C1)C)NCC C(=O)(N=c1cnn(C2CCC2)[nH]1)N1CCCC(CN2C(=O)CCC2)C1 c1(C(N(CCNC(CCCN(C(=O)OC)C)=O)C)=O)c(Cl)ccc(F)c1F C1(C(N(CC(C)NC(c2ccccn2)=O)C)=O)COCC(C)(C)O1 c1(-n2c(C(c3ccc(C)cc3)C)nc(CCCOC)n2)cc(F)ccc1C N1(C(c2c(OC)scc2)=O)CCCN(C(C2CC2(F)F)=O)C(C)C1 C#CCC(CC(F)F)NC(=O)C(O)C1CN(C(=O)C(COCC)N=[N+]=[N-])C1 CCCCCCCC(=O)N1CCCC(C(=O)N(CCCCO)C(C)C)CC1 c1(C(=O)NC(CCN(C(c2cc(C)c(CO)cn2)=O)C)C)cccc2sccc12 C(=O)(C#CC1CCCCO1)N1CCN(C(c2c(NC)snc2C)=O)CC1C(C)C n1(CCNC(CNC(CNC(C)=O)=O)=O)cc(CC(O)CO)nn1 C(C)(CCC(=O)NCC1(C(=O)NCC2(C)CCC2)CC1)OCC C(=O)(CC(C)C(=O)NC1CC(c2n[nH]c(C)n2)CC1O)c1ccc(OCC)cc1 c1(OC)cc2oc(C(=O)NN3CCCCC3C(=O)N(C)C)cc2cc1C C(C(CC(=O)Nc1cncc(CO)c1)NC(=O)Cn1c(O)nnc1O)OC C#CCCCCCCC(=O)NCC(O)CC(=O)NCC1CCCSC1 C1(C=O)CCN(C(=O)N(C)C)CC1.c1(CC)c[nH]nc1C=O.C(C)C(C)C.N C1(N(C)C(c2cc[nH]c(=NCCCC3CC3)n2)=O)CCc2ccccc2NC1=O CCN=C(NCCC(F)(F)F)NC1CCOC(C)C1 c1(C(=O)NC(CC)(CNC(c2sncc2C)=O)CC)c[nH]c2ccccc2c1=N c1(C(=O)OC)cc(=NCC2CC2NC(=O)C(c2ccccc2Cl)C)[nH]c(C)n1 c1(CCC)cc(C(=O)NC2C=CCN(C(=O)C=C3CCCCC3)C2)ccn1 c1(C=O)nsc2ccc(C)cc12.C(CC)(C(=O)NCc1nccs1)OCC.C C1(C(=O)NC2C(C(C)C)N(C(=O)COC(C)(C)C)CC2)CC2CCC1CC2 C1(NC(C(COC)OC)=O)CCN(C(c2ccc(F)cc2OC)=O)C1(C)C CN1CC(C(=O)NC2CCC(NC(=O)CC3COC(C)(C)C3)CC2)CC1=O CCC(CCc1ccccc1)C(=O)N1CC(CNC(=O)CC2CN(C)C2)CC1C c1(OCc2ncc(-c3c(OC)cccc3)o2)cc(F)cc(F)c1OC c1(OCC(=O)NC2CCCC(CN(C(CCOC)=O)C)C2)ccc(F)cc1O c1(C=O)cc(C)c(O)c([N+](=O)[O-])c1.C(C(C)(C(=O)N1CCC(C)C1)OC)OC Cn1c(C(=O)NC2CCCC2CC(=O)NC2CC=CCC2)cnc1Cl C1(N(C)C)CCCN(S(=O)(=O)CC2CC(=O)C23CCC3)CC1 C12(CNC(C(C)(C)SC)=O)CCC1CCN2C(=O)CC1(O)CCCC1 C1(CNC(C(C(C)C)NC(N)=O)=O)CCCC2CN(C(=O)C(C)(C)Br)CC12 c1(CC)cc(C(N2CCCC(C)(NC(c3ccnnc3)=O)C2)=O)cc(O)n1 c1(SC)cc(C(N2CCC3C(NC(=O)CN4CC5CC5C4)C23)=O)c(C)o1 c1cc2oc(C)cc2[nH]1.N1(C2CN(C(C)=O)C2)CC(NC(=O)CC(C)(C)C)CC1=O C1(C(=O)NCC(CCOC)NC(=O)Cc2cc(C)ns2)CCCC(O)C1 N1(C(C(C2CN(C(CC3CC(=C)C3)=O)C2)O)=O)CC2(CNC(=O)OC2)C1 N1(C(C(C)NC(C2COCCN2C)=O)=O)CCC2C(O)CC12 CC1(NC2COC(CCC(=O)O)C2)CCN(Cc2ccccc2)C1 C(CC(C)C)(C(=O)NCC(CO)C1CCC1)NC(C(CSC)OC)=O C=CCC(F)(F)C(=O)NC1CCC1NC(=O)C(C)(F)CC c1(C(=O)NC2(C3N(C(CC=C)=O)CCCC3)CC2)nc2nc(C(F)F)ccn2n1 Cc1ccc(C(=O)NCCOC(C)(C)CNC(=O)CC(F)(F)Br)cc1 c1(C(=O)NC2(CO)CCN(C(C3(C)CC4CC4C3)=O)C2)cc2nc[nH]c2cn1 C(=O)(CCCCC(C)C)NCc1oc(C)c(C(=O)Nc2cncc(Cl)c2)n1 N1(C(C(CC)=CC)=O)CCC2(CC1)CN(C(c1ccnn1CCOC)=O)C2 C(=O)(CCCCC(=O)NCC(F)CNC(=O)C)NC.c1(C=O)ccc(F)cc1 O=C(C1=CCCN(C(c2cncc(F)c2)=O)C1)Nc1c(O)cccc1Cl C=C(C)C(CC(=O)NCCC(=O)NCC(C)(O)CC)OCC C1(CC)CN(C(=O)C(C)N2CCCC2)CCC1NC(=O)CN1CCCNC1=O N1(C2CN(C(CNS(NC)(=O)=O)=O)C2)CCN(C(=O)C=CC=C(Cl)Cl)CC1 N1(C(CCC#N)=O)CCC(CNC(=O)C(F)(F)C2(O)CCC2)C(O)C1 C1(C(=O)NCCCN(C(=O)CS)CCC)C2CC(=O)CC12.C1CCCCC1 c1(C(=O)NCC2C(NC(C3(SC)CCC3)=O)C2)c(OC)nn(C)c1Br c1(N(CC(=O)OC)C)nnc(NC(CN2CCCS2(=O)=O)CO)n1C C1(NC(c2ccc(SC)cc2)=O)CN(C(=O)Cn2nnc(=O)[nH]2)CCC12CCC2 C(CCN(C)C)(C(=O)NCC1CC(O)CCO1)NC(C(COCC)C)=O CCC(C)C(C(=O)NC1(C)CN(C(c2ccc(Cl)nc2C)=O)C1)OC C1(C(N2CCC(CNC(=O)CCc3cncnc3)C2)=O)CCC(F)(F)CO1 C1(NC(Cc2nc(C)sc2C)=O)COCCN(Cc2nccn2C(C)C)C1 N1(C(CCSC)=O)CCC(C2CC2)C1C(=O)NCC1CCC1 c1(OC)cc(NC(C2CC2C(=O)Nc2cccc(OC)c2O)=O)cc(C)c1 C12(NC(C(CC)COC)=O)CC(CNC(c3coc(Br)n3)=O)(C1)OC2C N1(C(CC(C)OC)=O)CCOC2CN(C(c3ccc4c(c3)CCCO4)=O)CC12 CCCC(O)C(=O)N1CCC(NC(=O)C(c2cnn(C)c2)C)CC1 c1(C=O)cc(C)c(N)cn1.C1(C(=O)OC)(NC(C2CC2C)=O)CCOC1 CCN=c1[nH]c(C)c(C(=O)NC(C2CCOC2)CNC(=O)C2=C(C)CCCC2)s1 N1(C(C(CC=C)N(C)C)=O)CCC2(CCCN(CCNS(C)(=O)=O)C2)C1 N1(C(C(C)OCC#C)=O)CC2CC(NC(C3(O)CCCC(C)(C)C3)=O)CC1C2 CCC(CC)C(C(=O)NCC(C)=CC(=O)N(C1CC2(CCC2)C1)C)OC c1(CC(N2CCC(NC(=O)CN3CC(=O)NC3=O)C2)=O)cc(Cl)cnc1C.C c1(C(N2C(CNC(C(CCC)CC)=O)CCC2)=O)ccc2c(c1)CCC(C)(C)O2 N1(C(c2cc(-n3ccnc3)cs2)C(=O)NCC)Cc2ccc(C(=O)OC)cc2C1 Cc1cc(C(=O)N(CCC(N2CCCC2CCN(C)C)=O)C)c[nH]1 c1(NC(COC2CN(C(C(c3cccs3)SC)=O)C2)=O)ccncc1Br Cc1nn(C)c(Cl)c1C=CC(=O)NC1CC1.c1(C=O)cc(O)cc(=O)o1.C CN1CCN(C(C2CC(C)(C)CN2C)=O)C(C)C1.c1(C(=O)N)nc(O)[nH]c(=O)n1 Cn1nc2c(c1C(=O)NC1COC3(C1)CN(C(=O)CCS(C)(=O)=O)C3)CCCC2 Cc1nc(C(=O)NCC(C2CCOC2)NC(=O)C(C)(C)c2ccns2)nn1C N1(C(=O)CC2CC=CC2)CCCC1C1CCCN1C(c1ccccc1O)=O N1(c2c(Br)cnc(C)n2)CCC2CN(C(C3C4COCC34)=O)CC12 C(=O)(C(C)(F)C(=O)NCC(c1ccccc1)NC(=O)Cn1cncn1)OC c1(C=O)sc(C(C)C)nc1C.c1(CC)nocc1C(=O)NC1CCCC1C.N C(C)(C)(CCC)NC(c1[nH]cc(C(=O)OC)c1)=O.C1(C(=O)N)CCC(C)C1 CCC1=C(C(=O)NCC(CC(C)C)NC(c2csnc2OC)=O)CCCO1 N1(C(C=COCC)=O)CCC(CO)(CNC(=O)C(C)C(C)(F)F)CC1 c1(C(N2CCN(C3CCN(C(CCCC=C)=O)C3)CC2)=O)c(F)cc(Cl)cc1F c1(C(C)=O)cc(Cl)n(Cc2ncc(-c3ccc(Cc4ccccc4)cc3)cn2)n1 C1(C(=O)N)CN(C(=O)Cc2ncn(C)c2C)CC1C1CC1.C1(O)(CC)CCCCC1 c1(C(N(C2CCN(C(C3C(OCC)C3)=O)C2)CC)=O)n[nH]c2c1CCSC2 c1(OC)nc(Cl)ccc1C(N1CC=CC(NC(=O)CC(C)c2ccncc2)C1)=O C=Cc1ccc(C(=O)NC(CCCC)C(=O)NCC(CO)C(C)(C)C)cc1 N1(C(C(C2CC2)OC)=O)CC(C2CN(C(=O)C=Cc3ccc(F)c(Cl)c3)C2)C1 N1(C(c2ccc(C)nc2C(C)C)=O)CCC(C)N(C(C2CC2)=O)CC1.N(C)(C)C S(=O)(=O)(c1ccc(NC(c2ccc(C(F)(F)C(F)(F)F)cc2C)=O)cc1)NC c1(OC)ccc(Br)c(C(=O)NC)c1C.C12CC(C1)C2.c1(CC=O)ccoc1 C(C(C)S(C)(=O)=O)NC(C1C(C)C1)=O.C(=O)C(C(C)(C)C)C1CCCC1.N C(=O)(C1CCCc2nc[nH]c21)N(CC(C)NC(=O)CSc1nc[nH]n1)C N1(C(CNC(CC2CCC(=O)N2)=O)=O)CCCCCCCCC1 c1(C(=O)NC(c2noc(C)n2)CC)ccccc1N(C)C(c1ccc(S)cc1)=O c1(C(=O)NCC2C(NC(CCCc3c(C)ccs3)=O)C2)n[nH]c(C)c1O N1(C(c2cc(C)sc2)=O)CCC2(NC(=O)C(F)C(C)C)CCCCCC12 N1(c2snc(C(C)(C)OC)n2)CCN(C(C)C(N)=O)CC1 C(CC(C)C)(C(=O)NCCc1ccsc1)NC(c1cc(C)sc1N)=O C(=O)(C1CCc2ccccc21)NC(CNC(CSC)=O)(C)Cn1cccn1 c1(C(N2CC3(OCC(NC(CCC(C)C)=O)C3)C2)=O)ncn2cc(Cl)ccc12 C(=O)(N=c1ccn(C2CC2)[nH]1)NCC(C)(O)c1cccs1 C(=O)C(C)C(C)(C)C.Cc1nc(C2CC2)sc1C(=O)NC(C)C(C)(C)C.N C(=O)(CC(CC1CC1)CC)NCCC(C)N(C(COCCC=C)=O)C Cc1cc(F)ccc1C(F)(F)C(=O)NC(C)C(CO)NC(=O)C(C)(O)C(C)C C1(CC(=O)NC2(C(=O)NCC3(OC)CC3)CSC2)OCCC1(C)C c1(OCC)cccc(CC(=O)NC2CC2)n1.c1(CC=O)cnn(C2CC2)c1 c1(C(C)C(=O)NCC2CCN(C(C3CC3C(C)(F)F)=O)C2)ccccc1Cl C#CCCN=C(NCc1ccnc(F)c1)N1CCOC(CF)C1 N1(C(CC(CC)C2CC2)=O)CC=C(C)CC1.C1(C=O)C(c2nc(C)no2)C1(C)C.N C1(C(=O)NC(CC)CN(C(=O)CCC2CC2CC2CC2)C)CCN(C)C1 N1(C(C(CC)OCC)=O)CCC(CNC(=O)C=Cc2cnccc2C)C(O)C1 C1(NC(=O)Cn2cnnc2O)CCC2CCN(C(C3CC(Cl)(Cl)C3)=O)C1C2 c1(C(N2CC(C)(C)C2c2ccccc2)C(=O)NCC)ccc2ccc(O)nc2n1 C(C(C(C)C(C)C)NC(c1nnc(S)n1C)=O)NC(CC1(OC)CCCCC1)=O N1(C(C)=O)CCC(C(=O)NCC(C)C(C)(C)C)C(C(F)(F)F)C1 C=CCC(C)(CC)C(=O)NC1C2CC(NC(=O)CCn3cncn3)CC12 c1(C(N2CCC(N(C(C3N(CC)C(=O)CC3)=O)C)CC2)=O)ccc2oncc2c1 c1(C(=O)N)n[nH]c2c1CCC2.Cc1c(C(=O)NCC2CCC2)cnn1C(C)C c1(OC)c(Cl)ccc(C(=O)NCCC(C)CCNC(=O)Cc2cncn2C)c1F N1(Cc2snc(OC)c2Cl)CC2CC1CN2c1ncncc1Cl c1(C=O)cc2sc(N(C)C)nc2s1.Cc1nocc1C(=O)NC1CC(O)(C)C1 Cc1cc(C=CC(N2CC(N(C(=O)CC(C)n3cccn3)C)C2)=O)ccc1Br n1(CC)cnc(C(=O)NCC2COCC2)n1.c1(C=O)c[nH]nc1C(C)(C)C C1(NC(N2CCOCC2)=O)CCN(CC2CCCC2(C)Nc2ccco2)CC1 C1(CC)CCCCN1C(C1C(C)(C)C1(C)C)=O.C12CCN(CC1)C2=O.C(N)=O N1(C(C(c2n(C)ccc2)=O)=O)CC2CC(C(=O)NCCS(C)(=N)=O)C(C2)C1 C1(CC(=O)NC(CCF)C(=O)NCCC23CC(CCO2)C3)CCCC2CC12 CC1CC(C(=O)NCCCC2CCCN2C(c2ccon2)=O)CC(=O)N1 N1(C(C2(CC(C)C)COC2)=O)CCN(C(c2ccccc2)=O)C(C)C1.N(C)(C)C Cc1cc2sc(C(N3CC4CC(C3)N(C(=O)C=Cc3cnn(C)c3)C4)=O)cc2s1 C=Cc1cncc(C(=O)NC2(CCC)CCCN(C(C3CC(=O)N(O)C3)=O)C2)c1 C1(CCN(C)C(c2n[nH]cc2F)=O)CCCCN1C(C1CC1(C)C)=O CC1(CS(=O)(=O)NCC2(C(F)(F)F)CC2)CC2CCC1C2 C1(C(C)NCCF)CCCN(C(c2ccccc2OC(F)(F)F)=O)C1 CC1CN(C(=O)C(C)(C)n2cnnn2)CCC1N(C(=O)CCC1CCCCC1)C c1(N(C(C(C)NC=O)=O)CC(c2ccns2)=O)cccc(Cl)c1.C(C)(C)C.O CC1CC=CCC1CNCc1csc(C(=O)O)c1.c1ccccc1 c1(NC(C2=CCC(NC(C(CSC)C)=O)C2)=O)cncc([N+](=O)[O-])c1 CC1C2CN(C(C3(N(C)C(C4CC4[N+](=O)[O-])=O)CC3)=O)CC12 C(C(CNC(=O)CCCn1cccc1)CO)NC(C=C(CCC)C)=O C12(CC(N3CC(NC(c4cn(C)nn4)=O)C(F)C3)=O)CCC(CC1)C2(C)C Cc1ccc(C(=O)N(C2CCC23CCNCC3)Cc2cnn(C)c2)c(I)c1C c1(C(=O)N)ccc(C#N)cc1F.c1(C(N(C)CC2(C)CC2)=O)nc(Br)c[nH]1 S(=O)(=O)(c1cc(F)c(Br)cc1F)N1CCC2(CC(NC(=O)C(=O)C3CC3)C2)CC1 N1(C(C(C)(F)F)=O)CCCCC2(CCN(C(c3cn4ccncc4n3)=O)C2)C1 c1(C(N(C)CC2CCCN(C(C(CCC)N(C)C)=O)C2)=O)nccc(N)c1Cl Cc1nn(C)c(C)c1-c1cn(CCOCC)nn1.c1(C(=O)N)cc[nH]c(=N)c1Cl C1(CN(C(CCOC)=O)C)CCCN1C(=O)CC(=O)NCC(F)(F)F C1(NC(C(C)=CC=C)=O)CC2CC1CC2C(=O)N.C1(O)CCC(C)(C)C1 C(=O)(C1=CCCC(C)(C)C1)NC1CCC(c2cn(Cc3n(C)ccc3)nn2)CC1 C(c1ccc2c(c1)OCO2)=CC(=O)NC1CCCCN(C(C2C(C)C2)=O)C1 CCC(C)CC(C(=O)NC1CCCCCC1)NC(c1ccncc1Cl)=O C#CCCCCC(=O)N(CC(C)O)CCNC(=O)C(C(C)C)SC c1(C(=O)NCCNC(c2cnc(O)s2)=O)cnnn1C1CC1 CCCCC(C)C(=O)N1CCN(C(c2cnc[nH]2)=O)CC1c1cc(F)ccc1F N1(C(CC2(CC=C)CCCC2)=O)CC2CC1CCN2C(=O)C(C)OCCOC CC1CN(C(=O)CCC2CC(NC(C3COCOC3)=O)C2)CCC1N(C)C C(=O)(CCCCCCCCCO)N1CCC(N(C(COCC#C)=O)CC)CC1 C1(C(=O)NC(COC)C)CC2(CCC2)CN1C(C1CCCC(=O)C1)=O Cc1cccc(C=O)c1-n1cccc1.N(S(=O)(=O)N(C)C)CC(N1CCC1)=O.N C1(CC(=O)NC)C=CS(=O)(=O)C1.C1CCCCC1.c1(CC=O)cccc(O)c1 C(=O)(CCCCNC(N)=O)N(C1CCCN(C(=O)C(=O)N)C1)C.CCC(N)=O c1(-c2cn(C(C(=O)N(CC(=O)NC(C)C)C)C)nn2)cc(F)cc(Cl)c1 c1(OCC)cccc(C(=O)NCCC(C)(C)NC(C2CC23CCOC3)=O)c1 CCC(F)(F)C(C)(C)C(=O)NCC1CC2(CCC2)CN1C(=O)CCCCCC#N C1(C(=O)NCC(CC)NC(c2ccsc2)=O)CCC(=C(F)F)CC1 C(CCC(=O)NN1CCCC1C(=O)N(C(C)CC1CC1)C)OC Cc1nn(C2CCC2)cc1C(=O)N(C1CCN(C(C2CCN(C)C2=O)=O)CC1)C N1(C(C)C)CCC(N(c2nnnn2C)C)CC1.C1(C=O)C2COCC12 c1(C(C)O)nc(-c2cc(C(C)(C)C)ccn2)n(-c2cncc(Br)c2)n1 c1(CC)cc(NC(=O)C(C)(C2CC2)N(C(=O)Cn2cnnn2)C)cnc1C N#CCCCCCC(=O)N1CC(O)CCC1C(=O)NOCCO Cn1ccc(CNC(=O)NC(C)(C)C(=O)Nc2ccc(Cl)c(F)c2)cc1=O C1(N(c2ccncn2)C)CN(C(C2CCCCCCC2)=O)CC12CC2 N1(c2nnc(C)c(C)n2)CCC2(CN(C(c3ccc(F)cc3Cl)=O)CC(C)O2)C1 N1(C(C)CN2CCOCC2)CCCC(NS(=O)(=O)CC2CCOC2)C1 Cc1ccc2nc(C)c(C(N3CCCN(C(=O)C(C)(C)CO)CCC3)=O)cc2c1 Cc1nc2cncc(NC(N3CCC(N)CC3C)=O)c2nc1C c1(C(=O)NC(C(=O)NCC2N(CC)CC2)Cc2ccoc2)cnc(S)nc1 C1(O)(C(CNC(COCC=C)=O)C)CCN(C(c2ocnc2C)=O)C1 c1(OC)ccccc1-c1ncc(CN(C)CC2CCCCN2)cn1 CCC(c1ccccc1)=CC(=O)NCC(CNC(=O)C1=CCC(C)CC1)CO c1(C(=O)NC(CN(C(c2c(CC)occ2C)=O)C)C)c(OC)ccn2ccnc12 c1(-c2cn(CC(c3cc(C)nn3C)=O)nn2)sc(=O)n(C)c1Cl N1(C(CC2(C=C)CC2)=O)CCC2(CC(NC(c3ccc(C)n(C)c3=O)=O)C2)C1 C1(C2CCOCC2)(C(N2CC(N(C(CCN(CC)CC)=O)C)C2)=O)CC1(F)F N1(C(=O)NC(c2ccccc2)C)CCCC(C)(NC(c2ccc(Cl)cc2F)=O)C1 N1(C(c2cccc(CO)c2)=O)CC2CC(C1)N(C(c1cn3cccnc3n1)=O)C2 N1(C(CN(C)C)=O)CCCC2CN(C(c3ccccc3OC3CCC3)=O)CCC12 CCCCC(CNC(c1ccsn1)=O)NC(=O)C(C)CO C1(C(N2CCC(C)C2CNC(C2(F)CCOCC2)=O)=O)CCC([N+](=O)[O-])CC1 N1(C(CCC2N(C(C(C)OCCC=C)=O)CCC2)=O)CC2COC(=O)C2C1 C1(C(=O)NCC2CCCN2C(=O)C=Cc2cncs2)OCCOC12CCC2 c1(OC)cccc(C(=O)NC2CN(C(=O)C(C3CC3)S)CC2C(F)F)c1 C(=O)(CC(C)(C)F)N(CC(C)NC(c1n(C(CC)CC)ncc1)=O)C c1(NC(C(C(C)OC)NC(=O)CC2CCCCN2C)=O)cn(C)c(=O)cc1C Nc1ccc(Cl)cc1C(=O)NC(C1CCOC1)C.c1(C(=O)N)ccc2c(c1)CC2 C(C)(N=c1ccnc(NC(c2cnccc2C)C)[nH]1)c1cc(OC)ns1 c1(CNC(C2(C)CC2F)=O)ccc2c(c1)CCN(C(c1cc(CO)ccn1)=O)C2 Cc1c(C(=O)NCC(CO)NC(=O)CC2(C)CCC2)oc2c(Br)cccc12 c1(COC)c(C(N2C3CCC2C(NC(=O)CCS)C3)=O)sc2cccc(F)c12 N1(C(C(N(C(c2nnn(CC)c2C)=O)C)C2CC2)=O)CC(CO)C2(CC2)C1 C1(C(=O)OC)CCCN(c2cc(NC3C4CCC(F)C34)ncn2)C1 N1(C(C(C(C)C)C#N)=O)CCC2(CCCN(C(c3ns[nH]c3=O)=O)C2)CC1 C1(CC)(CN2CCC23CC(C(=O)OC)C3)CCCCCC1 N1(C(C(C2CCOCC2)OC)=O)CCC(n2cc(COC3CCOC3)nn2)C1 c1(CC)nc(C(=O)NCC(O)C)c(C)o1.C1(C=O)COCCN1C1CCCC1.N c1(C(=O)NC(C(CC)C)C)cccc(S(=O)(=O)NCC2CCCO2)c1 CN1CCc2cc(C(N3CCC(C)(NC(=O)CC4=NNC(=O)C4)C3)=O)ccc21 c1(C(=O)NC(C2CCCO2)CC)ccoc1C.C(=O)C=CC(=O)N(C)C C1(C(N(CC(C)C#N)C)=O)(NC(=O)C(C)CN(C)C)CCCC1 N1(C(CCC2C(=O)NC(=O)N2)=O)CCOC2(CCN(C(c3ccc[nH]3)=O)C2)C1 C(=O)(CCC(C)O)NCC(CC)NC(c1csc(C)c1)=O Cc1ccncc1C(=O)NC1CC(C)N(C(=O)C(F)=C2CCCC2)C1 c1(C(=O)NCC2N(C(c3cnc(COC)s3)=O)CCC2)cccc(OC)c1 C1(O)(Cc2cn(C(C)CNC(=O)CCc3cccnc3)nn2)CCCCC1 C1(C(=O)NCC(O)CN(C)C(c2ccccc2C)=O)(OC)Cc2ccccc2C1 C1(NC(Cc2nc(C)[nH]n2)=O)CN(C(c2ccc(F)cc2Cl)=O)CC(C)(C)C1 c1(CC)[nH]nc(C(N2CC(C)(CC(N3CCOC(=O)C3)=O)C2)=O)c1F CN1CCC(=CC(=O)N(CC(O)CNC(=O)CC2CCNC2=O)C)CC1 N1(C(CCC)=O)CC(CNC(=O)C(C)Sc2nncn2C)OC2COCC12 Cc1cc(O)c(F)cc1NC(C1(CO)CCN(C(=O)C(C)CC2CCCC2)C1)=O C1(C=O)CC12CCS(=O)(=O)CC2.C(C(C)(C)CC(=O)N)OC.C1(CC)CCC1 c1(CN2C(CNC(c3ccnn3C3CC3)=O)CC2)ccccc1.C1CC1.C C12(C(=O)N)CC3CC(C1)CC(C)(C3)C2.CC1CCCCN1C(=O)CCC1CCC1 CC1C(NC(=O)C(F)(F)F)C(C)CCN1C(=O)C(C)(C)C1CCCNC1 C1CC2(CCC2)CN1C(=O)C.Cc1nc(C(C)C)sc1C(=O)NC.C1CC1 C1(C(N(CCCNC(c2cn(CCCF)nn2)=O)C)=O)Cc2cccnc2C1 CCC(C)C(O)CC(=O)N1CCC(C(NC[Si](C)(C)C)=O)C(C)C1 c1(NCCSC23N(CC4CC(F)(F)C4)C(CC2)CC3)ccc2ccncc2c1 O=C(C#CC1CCOC1)N1CCN(C(=O)Cc2ccsc2Br)CC1 c1(NC(N2CC(OCc3nccc4n[nH]cc34)C2)=O)cccc([N+](=O)[O-])c1 n1(CC(N2CCN(C(c3c(C)cccc3)=O)C3C2C3)=O)sc(=O)c2ccccc12 Cc1cc(C(=O)NC2(C(=O)NCC3CCCCS3)CCOCC2)c(C)o1 N1(C(c2cc(CC)no2)=O)CC(F)(F)CC1CNC(c1cscc1CC)=O C1(CNC(c2nn(C)c(O)c2)=O)COCCN(C(=O)C=CC(=O)N(C)C)C1 N1(C(C(C)(C2(C)CC2)OC)=O)CCC2(CC1)CC2C.c1(C(=O)N)cnns1 N1(C(C)C(F)F)CCN(C(=O)C(O)c2ccco2)CC1.CC=O.CC(=O)N.C(C)=O N1(S(=O)(=O)Cc2ccc(Cl)cc2Cl)CC2(CCCCC2)C1 C1(N(C)C(C2CC(N)CN2C)=O)CC2CC1N(C(=O)Nc1ccccn1)C2 C1(NC(C2CCCN(CC)C2)=O)CCC2(CCCN(C(c3ncsc3C)=O)C2)C1 C1(NC(CC(C)C)=O)CC12CCN(C(=O)CCn1cncn1)C2 N1(C(C(CCC)NC(c2n[nH]c3c2COC3)=O)=O)CCN(C)C(C(=O)NC)C1 C1(CNC(c2nc(C(C)(C)C)oc2)=O)CN(C(=O)CC(F)(F)F)CCC12CCC2 C1(NC(=O)C2CC2)CCC2(CCN(C(=O)C3CC3)C2)C1 C1(C(N2CCCC(CNC(C3(C4CCCO4)CCC3)=O)C2)=O)(OC)CCSCC1 N1(C(c2c(OCC)scn2)=O)CCN(C(C2CCC2OC)=O)CC1C1CC1 C(CCCCNC(C1C(NC(c2cnn(C)c2)=O)C1(C)C)=O)N(C)C CCCCCCCCC(C(=O)Nc1ccc2c(c1)OCCO2)N1CCC1COC C(=O)(C1=CN2CCS(=O)(=O)N=C2C=C1)N1CC(CNC(C(CCCC)C)=O)C1 c1(NCC#CCC)cc(=NC(C)CCc2ccccc2)[nH]c(COC)n1 Cc1cc(C)c(C(N2CCC(O)(CNC(=O)C=O)C2)=O)cn1.c1ccccc1.N N1(C(c2n(COC)ncc2)=O)CC(CNC(=O)CC2(C)CC2)CC12CCC2 C1(N(C(=O)CCC#N)C)CCCN(C(C2CC3C=CC2CC3)=O)CC1 C(=O)(CC(=O)OC)NCC(CC)NC(C1CCSC1)=O c1(C(N2CCC(C(N(C)CCC3CC3)=O)(CF)C2)=O)ccc(=O)n(C)c1 c1(C(=O)NC2(CCCNC(C3CCC(N(C)C)C3)=O)CC2)cccc(C)c1Cl Cc1nc(NC2CCCCN(C(=O)Cn3nnc(C(C)(C)C)n3)C2)ncc1Br Cc1c(C(=O)NCCOC2CN(C(=O)C(C)C3CC3)C2)sc2ccc(F)cc12 Cc1cc(C)n(C(C)C(N2CCCC2CNC(=O)C=CCO)=O)n1 c1(C2(C(=O)NCC(CNC(=O)CC(O)C3CCCC3)O)CC2)cccc(F)c1 c1(C(N2CCC(NC(c3cc(C)on3)=O)C(O)C2)=O)cnc2ccc(C#N)cn12 N1(C(c2nc(CNC(CCOC(C)C)=O)oc2)=O)CCc2nn[nH]c2C1 C=CCC(C)(C)CC(=O)NC1CCC1NC(=O)C(C)c1cc[nH]n1 N1(C(C2OCC(C)C2)=O)CCC(CO)(NC(c2csc(Br)c2)=O)CC1 c1(CC)occ(C)c1C(=O)NC1CCC1.c1(C=O)ccc(-c2ccon2)cc1.N C1(NC(c2c[nH]c(=NC)o2)=O)CN(C(c2ccoc2Br)=O)CC1C1CC1 N1(C(c2c(C)n(C)cn2)=O)CC2CC1CCN2C(c1cn(CC(N)=O)nn1)=O N1(C(C(CC)c2cccnc2)=O)CC(NC(c2ccc(F)cc2O)=O)C2(CC2)C1 N1(c2cc(C(=O)NC)ncc2)CCN(N2CCOC3(CC2)CCS(=O)(=O)C3)CC1 CC1CCN(C(=O)C(C)CC(C)(C)C)C(C)C1NC(c1snc(Cl)c1Cl)=O c1(C(N2C(CNC(Cn3c(C)ncc3)=O)CC2)=O)cnn(-c2ccccc2)c1Cl O=C(CCCC(F)F)NC1CC(NC(=O)Cc2ccnc(Br)c2)C1 C1(NC(C2C(COC)C2)=O)CCN(C(C2CCC3(C2)N=N3)=O)CC1F C(=O)(C(C)(O)CCN(C)C)N1CCCC(NC(C(CCOC)C)=O)C1 C(C)(C(=O)Nn1ccnn1)C1N(C(C2C=C(C)CS2)=O)CCC1 C1(C(N2C(CC=C)(C(=O)NCC3(C)CCCC3)CCC2)=O)CCOCC1(C)C C(CCCCC(=O)NC(C)CCCNC(=O)CCOc1ccc(C)cc1)OCC O=S1(=O)CCC(N2CCC(NC(=NCc3cccs3)NCC3=CCCC3)CC2)C1 Cn1nc(C(=O)NC(C2CCCC2)CNC(=O)CCCS(N)(=O)=O)c2c1CCC2 C1(NC(c2cc(-c3cn(C)nn3)on2)=O)CCCCN(C(=O)CO)C1.C(C)(C)C C1(C(=O)N)CN(C(=O)C(c2cccc(F)c2)C)CC1C.C(=O)(CC1CC1)OC N1(C(C2(SC)CCCC2)=O)CCC(C)N(C(C2CN(CC(C)C)C2)=O)CC1 N1(C(c2cc(C)on2)=O)CCCOC(CNC(c2cc(F)cc(Br)c2)=O)C1 C1(CC)CCCN(C(c2cccc(CNC(C3CCCN(CC)C3)=O)n2)=O)C1 C12(C(=O)NCC(CC(=O)NC(c3c[nH]ccc3=O)C)O)C(=O)C3CC1C2C3 C12(C(=O)NC3CC(C(=O)NC4CN(CC)CC4C)OCC3)CCCN1CCC2 N1(C(C23OCC(C(=O)OC)(C2)C3)=O)CC2CCC1CC2.c1(C(=O)N)ccc[nH]1 Cc1cccc(C(=O)O)c1S(=O)(=O)N1CCCC(c2cnn(C)c2)C1 Cc1cnc(Br)cc1NC(N1CCOC(CC2CC2)C1)=O Cc1ccc(C(N2CC(C(=O)NCCCS(C)=O)C(C(C)C)C2)=O)nc1C Cc1ccc(CC(C)C(=O)NC2CCCC(NC(=O)CC(F)(F)F)C2)cc1 C1(N(C(c2cc(C(C)C)no2)=O)CC)CCN(C(=O)C(C)N2CC(C)C2)C1 CCCCC(CNC(c1cn(CCNC(=O)C(C(C)C)NC=O)cn1)=O)CC C1(CCNC(CSC)=O)CCCN(C(=O)C(c2cccc(Br)n2)(F)F)C1 C(Cc1cccs1)(CC(=O)Nc1cccnc1I)NCc1c(C)n[nH]c1 N1(C(C(CC)NC(C)=O)=O)CCCCC(NC(=O)C(=C2CCCCC2)F)C1 C(=O)(CC1=CCOCC1)NC(C1(O)CCN(C(CS(=O)(=O)NC)=O)C1)C C1(CC(=O)N)CCCNC1=O.C1(C(=O)NC(C)C)(SC)CN(C(=O)C)C1 c1(C(=O)NCCCSC)cc(C(F)(F)F)ccc1I S(=O)(=O)(c1cccnc1NCC(C)O)N1C(c2cc(C)[nH]n2)CCCC1 N1(C(C)=O)CCN(C(c2c(CN)nn3c2CCC3)=O)CC2(CC2)C1 C(C(CO)(CO)NC(=O)CNC=O)N(C)C(c1cnn(CCF)n1)=O C#CC#CC(C)(C)NC(=O)CNC(=O)CNC(C1(C)CCNC1=O)=O C=CCCCCCC(=O)N1CCC(NC(c2cnn(C(C)(C)C)c2Br)=O)C1 C(=O)(C(=O)C(C)CC)N1CC(CCC=C)(C(N2CCC3(CC3)C2)=O)C1 c1(C(N2CCCC(C)(NC(C(C)CC(F)(F)F)=O)C2)=O)c(N)cccc1[N+](=O)[O-] c1(C(=O)N)cn(C)c2ncccc12.CN1CC(O)CC1C(=O)NCCOCC CC(c1cnn(C)c1)=CC(=O)NC1CCCCC1NC(=O)C(C1CCCCC1)O C1(C(=O)NC(CC#C)C(=O)OC)CCN(C(C2(CC)CCNC2=O)=O)CC1C C1(NC(c2c(SC)snn2)=O)COCCC1NC(C1CCNC(=O)C1)=O C12(C(=O)NC3(C(=O)NC4C(N(C)C)CCC4)CCN(C)C3)CCCC1C2(F)F CC1(C#CC(=O)N2CCC(c3c[nH]c(=N)[nH]3)CC2)CCCO1 C=CC(C)(C)CC(=O)NCC1CC(NC(c2ncccc2Cl)=O)CCO1 N1(C(C(C(C)C)n2cnnc2)=O)CC2CCC(NC(=O)CCC3CC3)CC2C1 N#Cc1ccc2c(C(=O)NCC)c[nH]c2c1.C1(CO)CCCC(C=O)O1 N1(C(CCc2cccc(C(=O)O)c2)=O)CCN(C2=NCC(C)S(=O)(=O)N2)CC1.CC C1(NC(CC2CC(CC)OCC2)=O)COC2(C1)CN(C(=O)CCCS(N)(=O)=O)C2 N1(C(C(CC#C)C)=O)CCN(C(C2CC(CF)C2)=O)CC1c1nccn1C c1(CC(=O)NC2CN(C(C(CC=C)C)=O)CC2O)ccc(F)c(C)c1 C(=O)(C(CC(C)(C)C)NC(=O)COCC1CCCC1)NC(C=C)C N1(C(C2CN(C(N(C)C)=O)C2)=O)CCC2CN(C(c3ccc(Cl)s3)=O)CC12 C(=O)(CCCCCC#N)NCc1c(C(=O)NCC2(C)ON=C(C)C2)cco1 c1(C(=O)NCC(C)CN(C)C(c2cccc3c2CCC3)=O)ncnc2c1CCC2 c1(-c2cn(C(C)CSc3cccs3)nn2)cc(F)ccc1OC(F)F C1(NC(C2(C#C)CCCC2)=O)CC2(C1)CCC2.c1(C(=O)N)coc(C(F)F)c1 Cn1cnc(C(N2CCC(N(CCO)C(C3CCS(=O)(=O)C3)=O)CC2)=O)cc1=O Cc1nnc2n1CC(C(=O)NC(C)CN(C(=O)CCSC(F)(F)F)C)C2 C(N=c1nc(-c2ccccc2)[nH]c(=NCC2CCC2)[nH]1)C1Cc2c(nc[nH]2)CC1 N1(C(c2c(C)c(Cl)ccc2)=O)CC(C2CN(C(C3CCS(=O)(=O)N3)=O)C2)C1 C1(NC(C2C(OC)CN(C(c3ccccn3)=O)C2)=O)CCCCC12OCCO2 C1(C(=O)OC)N(C(c2c[nH]nc2)=O)CC1(C)C.C(=O)C(O)CN1CCCC1.C C(C)(C=O)(C(=O)N)OC.C1(C)CCN(C(c2cc(Cl)c[nH]2)=O)C1.C(C)(C)C c1(C(C)=O)cc(C(=O)NC2CCCC(C(=O)NCc3nc[nH]n3)C2)ccn1 c1(C(=O)NC2C3CC(NC(c4c(C)nncc4)=O)CC32)cc2ccncc2o1 C(=O)(C1CCc2cccnc21)N(C1C(O)CCN(C(C(CC=C)C)=O)C1)C C(C1(C)COC1)=C(C)C.C(=O)Cc1cscn1.C1CN(C=O)C1.C(C)(C)C C1(C(=O)NCC2CCCCS2)CN(C(=O)CCc2cncs2)CCO1 c1(C(=O)NC2CCCCC2NC(C2CC3CCC3C2)=O)ccn2nnnc2c1 C(=O)(C(O)C1=CCCCC1)NCC1(C)CCN(C(=O)CC=C(Cl)Cl)C1 C#CC1CN(C(C2CCCC2CNC(C2(SC)CC(C)(C)C2)=O)=O)CCN1C C(=O)(C#CC(C)(C)C)NCCN(CCC)CC.c1(C(=O)N)ccc(O)cc1 N1(C(C2C(CC)CN(C(c3cc(C)cc(C#N)c3)=O)C2)=O)CCCC2(C)CCCC12 c1(C(N2C(C(N(CCCN3CCCC3)C)=O)CC(=O)C2)=O)cncn(C)c1=O C1(NC(c2cnc(C(C)C)n2C)=O)CC1C1CCCN(C(C2CNC(=O)N2)=O)C1 c1(CC(=O)NCC2C=CCN2C(c2cc(O)nc(O)n2)=O)ccnc(Cl)c1F c1(OC)ccc2ncnc(N3CC(NC(c4cnc(O)cc4O)=O)C(F)C3)c2c1 C=CCCCCC(=O)NC1CC(NC(c2sccc2I)=O)C1 c1(-c2cn(CC(=O)OC)nn2)ccc(C)cc1C.c1(CC(=O)N)c(C)noc1C C1(SC)CN(C(C2CC2[N+](=O)[O-])=O)CC1NC(c1cnn(-c2cccnc2)c1)=O c1(SCC)cc(C(=O)N(CC(CC)NC(c2cc(O)n(C)n2)=O)C)ccn1 C1(CCNC(Cn2nnc(C)n2)=O)CCN(C(=O)C(C)CC(C)C)CC1(F)F N1(C(CC2CCC(C)(C)O2)=O)CCC2(CC2NC(=O)Cc2cccnc2)C1 CC(CN1CCOCC1)C(=O)NCCCN(C(=O)CC1CCCC1)CCO CCC(CC)CC(F)C(=O)NCC1(C)CCN(C(C2(OC)CCCOC2)=O)C1 c1(OCCN)cc(Cl)ccc1C.CCCCCCN(C(=O)CCC)C c1(C(=O)NC2CN(C(CS(=O)(=O)N(C)C)=O)CC23CC3)ccc2cc[nH]c2c1F c1(C(=O)NCC(CO)NC(=O)CCCC2CCOCC2)ncncc1F N1(C(C(CN(C)C)NC(CC(CC)C2CC2)=O)=O)CC2(CCN2C)C1 Cc1ccc(C)c(SCC(=O)NCCC(O)CNC(c2cc(C)n(C)c2)=O)c1 c1(SCC)ccc(CC(N2CC(N(C)C(c3cnc(C(C)C)nc3)=O)C2)=O)cc1 CC(C)C(C)C(=O)NCC(CO)NC(=O)CCc1ccccc1C N1(C(C(c2cnn(C)c2)NC(C(C(C)C)C)=O)=O)CCS(=O)C(C)C1 c1(C(CC)=O)ccc(NC2CCCCC2C)c([N+](=O)[O-])c1.C(=O)(C(C)(C)CF)N C(C)(CCC(=O)NC1CCC1NC(c1cccnc1OCCO)=O)OCC C1(NC(C(Cc2ccco2)NC(CNC(CC)=O)=O)=O)CC2(C1)CN(C)C2 N1(CC(N)=O)CCC2CC(NC(=O)COCCC[SH]=Cc3ccccc3)C2C1 c1(CN(CCNC(C2CC2C2CC2)=O)C2CC2)csc(C(F)(F)F)n1 Cc1cn(CC(=O)Nc2cccc(COC(F)F)c2)c(=O)nc1O C1(OCC)CN(C(=O)Cc2cccc(OC)c2)CC1C.c1(C=O)cnco1.N C1(CCNC(=O)NCC(CNC)C)CCOCC1 N1(C(C2C(NC(C3CC(=O)N3)=O)C2)=O)CCOC(O)C1 C1(CCNC(c2[nH]c(=N)sc2)=O)CN(C(c2ccc(OC(F)F)cn2)=O)CCO1 c1(NC(CCNC(CC(CCC)OC)=O)=O)ccc2c(c1)OCO2 C1(SC)CN(C(c2nc(Cl)oc2C)=O)CC1NC(C1CCCC(CF)C1)=O Cc1cc(CC(=O)NC2CCCC2NC(=O)C(C)Cc2cnc[nH]2)sn1 O=C(CCC(F)(F)F)NCC1CCN1C(C1(C2CCC2)CCC1)=O N1(C(C(C)=CC)=O)CCN(C(=O)CN=S(C)(C)=O)CC1C1CCC1 N1(C(CN(C2CC2)CC)=O)CCC(NC(C2CC2C2CCOCC2)=O)C12CCC2 C=CC(C)CC(=O)NCc1cc(C2CCN(C(=O)C(CC)SC)CC2)no1 C1(CNC(C2(F)C(C)C2)=O)COCCN(C(c2cnc(N(C)C)c(Cl)c2)=O)C1 C(=O)(CCC)NCC(C)CN(C)C(C1CC12CC2)=O.C(=O)(C(C)(C)C)N c1(OCCC(N2CC(C)OCC2)=O)cc2n(c1)CCCC2 C(C(=O)NOCCN(C)C)(C1(O)CCC1)NC(c1ccc(OC)o1)=O C1(C(=O)NC2(C(=O)NCCCc3cn(C)nc3)CC2(C)C)CCCC(O)C1 C1(NC(=O)C2=CCN(C(C3CC(F)C(=O)N3)=O)C2)CCOC2(CCC2)C1 Cc1c(Cl)ccc(F)c1C(=O)NCc1ncc(Br)cc1Cl Cc1ccncc1C(=O)NCc1nnn(C)c1C(=O)NCC(N1CCCC1)C Cc1c(C(=O)NCCCN(C)C(C2CCCS(=O)(=O)N2)=O)cncc1Br C(c1ccc(Cl)cc1Cl)=CCOC(=O)NCCSCCCOCC(F)F c1(-c2c(CCNC(C(N)Cc3cn[nH]c3)=O)cno2)ccc(F)cc1Cl C=CCCCCCN(C(=O)C(C)(CO)NC(=O)Cc1ccccc1O)C Cc1nc(-c2cccc(Nc3nccc(N4CCCC(F)C4)n3)c2)c(C)s1 C12(NC(=O)C(O)C3CC3)CCCN(C(=O)CCCCCF)CC1C2 Cc1cc(C(=O)NC2CC(O)CN(C(=O)CC(Cl)Cl)C2)c(F)cc1F C1(NC(c2ccc(CCC)[nH]2)=O)(C)CC2CCC1C2.C1(C)(CC=O)CCCC1 c1(C(c2nnnn2CC2CCOCC2)NC2(C)COC2)ccc(Br)cc1F C1(C(N2CCC(=C)C2)=O)CN(C(=O)C(O)CC)CCO1 CC1(C)CCCOC1C(=O)NCC1(NC(C2CC3(CCO2)CC3)=O)CCOC1 c1(C(=O)NC(CCCNC(CCC#C)=O)C)cncc(OC)c1C N1(C(CN(CCOC)C(C2CNC(=O)N2)=O)=O)CCC12CCCC2 N1(C(C2(C)CCCC2)=O)CCOC(CNC(c2cc(N)ccn2)=O)C1 CC(C)(CNC(=O)C1=CCCCC1)CC(=O)NCCC(=O)OC(C)(C)C N1(C(c2ccn(CC)n2)=O)CC(C)C(C(F)(F)F)C1.c1(C=O)cc(Cl)cn1C c1(C(N2CC(NC(=O)C(C)CC3CCC3)CC(OC)C2)=O)ccc(C)c(C)c1N c1(C(=O)NC2C(CNC(Cc3nc(C)oc3)=O)CCC2)ccc2c(c1)COCO2 C1(C(=O)NCC(C(C)C)NC(=O)C2=C(Cl)CC2)CS(=O)(=O)CC(=O)N1 N1(C(C(n2ccc(C)n2)C)=O)CCC(F)(C(=O)N(C(C)(C)CO)C2CC2)C1 N1(C(C2OCC(C)(C)C2)=O)CC(N=[N+]=[N-])CC1C(N1CCCC(O)CC1)=O CC1CCCCN1c1cc(C(=O)OCCc2cnccc2Br)cs1 Cc1cn2c(n1)C(C)CC(C(=O)NC)C2.C1(O)CN(C(c2cnc(C)o2)=O)C1 C1(NC(=O)CCn2cccn2)CCC2(CC1)CN(C(c1cc3cscc3s1)=O)C2 C(=O)C1=C(C)CCC1.c1(CC)ocnc1C(N1CC(C(C)(C)O)(C)C1)=O.N C=CC1CCCN(C(CC2C=CCC2)C(=O)NC2(C)CC2)C1 C1(Cn2ncc(C)c2)CCCCN1C(=O)Nc1ccccc1C1(C)CC1 Cn1ccc(C(=O)NCC(F)CNC(=O)C(C)(O)C2CCC2)n1 C1(CC(=O)N(CCCN(C(=O)COc2ccccc2)C)C)CCC(F)(F)C1 c1(C(N(CCNC(Cn2c(C)cc(C(F)F)n2)=O)C)=O)cnc2c(n1)CCCC2 CC1(C(=O)NCC2CCC(=O)O2)CC(O)CN1C(=O)CCCn1ccnn1 Cc1nc2c([nH]1)CN(C(CCC1OCCO1)C(=O)NCC(C)C)CC2 N1(Cc2cc(OC)c(OC)cc2)CCc2[nH]nc(C(N3CCC(OC)C3)=O)c2C1 c1(CC(N2CCC(O)(C(C)NC(C=CCC)=O)C2)=O)c(F)cccc1Cl CCC(CC(=O)NC1(CCCNC(=O)CCc2cccc(C)c2)CC1)OC C1(C(N2CC(OCC(=O)NCC(C)CC3CCC3)C2)=O)COCCN1CC CCCCCCCC(C(=O)NCCO)N1CCN(C)CC1C(C)C.C1CC1 C=CCCCCN(C(=O)CCNC(c1cccn1C(C)C)=O)C c1(CNC2C(C(=O)Nc3ccc(CCC)cc3)C2)ccc(C)nc1OC Cc1ncncc1C(N1CC(O)CC1C(=O)NCC1(F)CCN(C)C1)=O C(CCNC(C1CCC1C(C)(C)C)=O)(C(=O)N(c1cccc(C)c1)C)OC CC1COCCC1NC(=O)NCC1CCCCN1Cc1ccc(C(=O)O)cc1 c1(C(N2C(CC(=O)NC(CC(C)(C)OC)C)CCC2)=O)cc2cccn2cn1 N1(C(c2c(C)nn(CCO)c2)=O)CCC(CO)C(NC(=O)CN2CC(C)C2)C1 C(CC1=CCN(C(=O)CC2CCCC(F)(F)C2)CC1)NC(C=C(CC)CC)=O Cc1ncc(NC(C2C3CC3CN2C(C2CC(=O)N(C)C2)=O)=O)cn1 CCC(C(=O)N(CC(C)CNC(=O)C(c1ccncc1)C)C)n1ccnc1 CCCC(CCC)CCCOc1ccc(C=CC(=O)OC)cc1 c1(SC(CC(CC)C)C)nc2sc(CO)c(C)c2c(=O)n1CCCN c1(OC)cc(CNC(c2cnn(C3CNCCOC3)c2)=O)c(Br)cc1C C1(C(C)(C)C)CCC(CNC(C2(O)CCOC2)=O)CC1 c1(CN2CCC(CNC(c3n[nH]c4c3CCCC4)=O)C2)cc(F)ccc1[N+](=O)[O-] C1(NC(CCCC#C)=O)CCN(C(c2c(C)nn3c2CCCC3)=O)CCC1(F)F c1(C(=O)NC(C(=O)NC2C(C)(CC)C2)CC2CCCC2)cc(C)nnc1C N1(C(CCC2CC(OC)C2)=O)CC(CNC(c2c(C)cnn2C)=O)CC(C)C1 C1(N(C(c2c[nH]c(=NC)s2)=O)C)CN(C(c2cnn(C3CC3)c2C)=O)CC1(C)C N1(C(=O)NC2CCC(C)CC2)CCC2C1CCN2C(c1ccoc1)=O Cc1ccc(C(F)F)c(C(N2CCCCC(CNC(C3CC3C)=O)C2)=O)c1 C#Cc1ccc(C(N2CCCC2CCC(=O)NC2CCCC(CO)C2)=O)o1 c1(C(C=O)=O)ccc(F)cc1F.CC(C)(C)C.C1(CCOC)(C(=O)N)CCC1 c1(C(=O)NCCCC)ccc(Nc2ccncc2)cc1.C(=O)(C=CC1CC1)N C1(C(=O)NC2CN(C(CC3CCN(C(C)=O)C3)=O)C2)CC(C)C1.C1CCC1.C N1(C(C(C(C)C)NS(C)(=O)=O)=O)CC2CCN(C(c3ccccc3F)=O)C2C1 C(CC(N)=O)(C(=O)NCC(C1CCCO1)O)NC(C(c1cncnc1)C)=O N1(C(CCC=C)=O)CCC2C(C1)NC(=O)CCN2C(c1ccc2ccsc2c1)=O C1(NC(CCC=CC(C)C)=O)COC2C(NC(C3(CCO)CC3)=O)COC12 N1(C(C2(CNC(c3cnn(C)n3)=O)CC(=C)C2)=O)CC2CC2C2CC12 N1(C(c2cnn(C)n2)=O)CC2(CCN2C(c2cc(=O)n(C)cn2)=O)C1 C1CC(F)CN1C(C1CCCCN1S(C)(=O)=O)=O.C1(C=O)CC1.CC=O.O C1(NC(CCC=CC)=O)CC2(C1)CC2C(=O)NCc1ccc(C)cn1 C=CC1CN(C(=O)Cc2ncoc2C)CC1NC(=O)CC1CCCS(=O)(=O)C1 c1(C(=O)NCC2C(NC(=O)C=Cc3cccs3)CCC2)ccncc1O C1(C=O)C2CCC(C2)C1C(=O)O.N1(CC2(CCC=C)CC2)CCC(C)C1.N N1(C(CCP(C)(C)=O)=O)Cc2ccccc2C(CNC(C2CC3C=CC2O3)=O)C1 c1(C=O)ccc2occc2n1.CC1(C)OCC2CC12C(=O)NC(C)C(C)(C)C.N c1(C(=O)NCC2(C)CCCN(C(C(CC)C)=O)C2)cc2nc(C)cc(C)n2n1 C1(C(N2CCC(C)(F)C2)=O)CCN(C(=O)CCc2cnn[nH]2)CC1(C)C C1C(C2CC2)CCN1c1ncc([N+](=O)[O-])cn1.N1(CC)CC(C(=O)NC)CC1=O C1(NC(c2cnn(CCOC)c2C)=O)CCCCN(C(=O)CC2CCCOC2)C1 c1(C(=O)NC2CC3CC2CN3C(c2ccsc2)=O)cc2ccccc2oc1=O Cc1c(C(=O)NC2CCCC2NC(C2C=CCC2)=O)sc2cncn12 C(=O)(C(O)CC(F)(F)F)N1CC(n2cc(CNC(C3CC(=O)NC3)=O)nc2)C1 c1(N2CCCC(CC=C)C2)ncnc(C(=O)OC)c1OC C=C=CCCC(=O)NCCC1CCCN1C(=O)CC(=O)OCCC(C)C CCC(C)CC(C(=O)N(C1CC2CCC1O2)C)NC(c1cnn(CCO)c1)=O N1(CC(N2CCC(NC(CC(C)NC(N)=O)=O)(CF)C2)=O)CCCCCC1=O C1(C)(C(=O)N)CN(C(C2CC3CC3C2)=O)C(C)(C)C1.Cc1cc(C)cc(F)c1 C1(CC=C)CCCN(CC2CC2C(C)(F)F)C1.c1(C=O)ccc(C(N)=O)o1 C(C(CNC(=O)Cn1ncc(Cl)c1C)C(F)(F)F)OC.c1(N)cc(O)ncn1 c1(C(=O)NC2(CNC(C(n3cc(Cl)cn3)C)=O)CC2)cccn2nncc12 Cc1cccc(OC(C)C)c1NC(C1(C2CCCCO2)CCOCC1)=O c1(C(=O)OC)c(C)cc[nH]c1=NCCCNC(=O)CC(n1nc(C)cc1C)C C1(CC)CN(C(c2sccc2Cl)=O)CCC1NC(=O)C=Cc1cc(C)no1 Cc1cnn(C)c1C(=O)NC(C)CC1CN(C(=O)CC2COCCN2C)C1 C1(C(=O)NC2CCN(CCc3cn(CCO)nn3)CC2)CC1C1CCCC1 c1(NC(C2CC(NC(C3CCCSC3)=O)C2)=O)c(Cl)cccc1[N+](=O)[O-] c1(NC(CC(CNC(c2ccc(C(C)=O)[nH]2)=O)OC)=O)c(C)[nH]c(C)cc1=O C1(C(N(CCN(c2snc(C=O)n2)C)C(C)C)=O)CCS(=O)(=O)C1.CO N1(C(C2(NC(C(CC(C)C)N(C)C)=O)CC(F)(F)C2)=O)CCC2(C1)CC2(F)F C1(C(N(C2CCN(C(C3C(C=O)C3)=O)C2)C)=O)CCC(NC)CC1.C#CC c1(C(N2CC(NC(C(C)NS(CC)(=O)=O)=O)(C)C2)=O)noc2c1COCC2 C(=O)(C(CC1CC1)NC(=O)COC1CCCC1)NC(COCC)C C=CCC(C)(C)C(=O)NC1CN(C(=O)Cc2[nH]cnc2C)CCC1C c1(C(=O)OC(C)(C)C)ccccc1OCCSc1ncccn1 c1(C(N(C2CCN(C(=O)C(C)NC(C)=O)C2)CC)=O)ccoc1C.C(C)C c1(CNC(=O)NCc2ccc(F)cc2F)cnn2cc(Br)ccc12 N1(C(=O)CC2CCCCO2)CCC(C(N2CCN(c3ccnc(Cl)n3)CC2)=O)CC1 CC(C)C#CC(=O)N(C1CCN(C(=O)C(C)(O)C2CCCCC2)CC1)C c1(C=O)cc(C(F)F)ccc1F.C1(C(F)(F)F)(C(=O)NCCC)CCCCO1.N n1(CC(=O)NCC2(F)CCC(NC(c3cn[nH]c3)=O)C2)nc(O)ccc1=O c1(C(N2CCC(C(C)C(N3CC4CC=CC3C4)=O)CC2)=O)ccn2ccccc12 N1(C(c2ccn(CC)n2)=O)CCCC1C(C)(C)C(=O)NCC(C)OCC c1(C(N(CC(=O)NCC23CCCCC2C3)C2CCC2)=O)cc(F)cc(F)c1 Cc1cc(C(N2CCN(C(=O)CC34CCCC3C4)CC2C)=O)cc(F)c1 C(C)(CC(=O)NC1CC(C)(CNC(=O)C(F)(F)C2CCOCC2)C1)OC C12(N(C(C)(C)C)C(=O)OCC(=O)NC(C)(C)C)CSCC1C2 CCC(Cc1ccccc1)C(=O)NC1CC(NC(=O)C(O)C(C)c2ccccc2)C1 c1(C(=O)NC2CCCN(C(N)=O)C2)cccc(OCc2nccs2)c1F N1(C(CN(CC)CC)=O)CC2CCC2(CC)C1.C(C)(c1ccncc1)=CC=O c1(C=O)cc(C2CC2)cs1.C1(CC)CCOC1.C(C(=O)N)=CCN(C)CC c1(C=O)ccc(I)c(F)c1.C1(CC(=O)NCc2n(CC)cnc2)CCCCC1 CCCCCC(C)(CC)C(=O)NCC1C=CCN1C(c1cn(C2CC2)nn1)=O c1(CC)ccc(C(N2CCCCC2c2ncccn2)=O)c(C)c1 c1(NC(C2C3CN(Cc4ccc(Cl)nn4)CC23)=O)ccc(Cl)c(CO)c1 c1(CC(=O)NC2CCCC23CC3)csc2nc(-c3ccccc3)cn12 Cc1c(C(N2CCCC(C)(NC(=O)CC3(C)CCCO3)C2)=O)cccc1CO Cc1sc(Br)nc1C(N1CC(N(C(=O)C(O)CC2CCCCC2)C)C1)=O C(=O)C1CNC(=O)c2ccccc21.c1(CC)ccsc1C(=O)NC1CCC1C.N N1(C(=O)OC(C)(C)C)CC=C(CC(=O)Nc2ccccc2SC2CCC2)CC1 N1(CC)CC2CCCC2C1.c1(C2CC2)cc(COCCOC)on1.C(=O)N C1(C(=O)NCC(C)NC(C=CC)=O)CCC(O)(Cc2ccccc2)CC1 Cc1ccc(C(=O)NCC(CC(C)C)NC(=O)CCc2cccnc2C)cc1O C(=O)(C(F)CC(C)(C)NC(C1CC(N(C)C)C1)=O)NCC(CC)O C#CCCC(C(=O)NCC1CCC(=O)N1)NC(=O)COCC1CCC1 c1(C(=O)NCCC(CC)(C)NC(c2cccc(C(N)=O)c2)=O)cc(F)ccc1F Cc1coc(C(=O)NCC(O)CNC(=O)CC2COC(C)(C)C2)c1C N1(C(C(c2ccccc2)C)=O)CC2CCCC(C1)N2C(C1C(C)(C)C1(F)F)=O c1(NC(C2CN(Cc3ccn(C)n3)CC(F)(F)C2)=O)cc(Cl)cc2ncoc12 CC(C)CCC(=O)N1CCC(CC(C)NC(=O)CC2CCC(C)C2)CC1 C1(O)(CCNC(c2c(F)cccc2Cl)=O)CCCN(C(C2CCCOC2)=O)C1 N1(C(CCC2CCN(C(C3CCC(O)CC3)=O)CC2)=O)CCc2cccc(F)c21 N1(C(CCc2cccc(C)c2)=O)CCCC(NC(=O)C(C)(C)c2ccno2)C1C N1(C(c2n(C=C)ncc2)=O)CC(C)(C)CC1C.c1(C=O)cccc(C2CC2)n1.N N1(C(C2CS(=O)(=O)C2)=O)CCN(C(=O)CCCC2CC2)C2CC12 n1(CC=C)cc(C(=O)NC(Cn2cncn2)C(=O)NC(C)C(F)F)cn1 C1(C(N2CC(NC(c3c(CC)nco3)=O)(CO)C2)=O)CC2(COCCO2)C1 N1(C(C2(C(C)=O)CC2)=O)CCCCC1.c1(C(N(C(=O)CC)C)=O)ocnc1C C1(C(=O)Nc2cccc(-c3nnco3)c2)CC2(CCC2=O)C1 S(=O)(=O)(C1CC1C)NCCC(=O)NCCC(=O)OC C(=O)(C1CCc2cccnc21)NCC(C)(C)c1ccsc1 Cc1c(CCNC(=O)C(C2CCN(C(C3CN(C)C3)=O)C2)F)cnn1C Cc1c(C(=O)NCC2(C)CCC2)[nH]c2c(C)cccc12.c1(C=O)sccc1Cl.N C1(CC(=O)NC2C(CNC(Cc3ccn(C)c3)=O)CC2)CC(C)(C)CO1 c1(C(N2CC(C(N3CC4C(CC)(C4)C3)=O)(CC)C2)=O)cc(C)ccc1O CON1CCC(C(N2CCN(C(C3CC3C(=O)OC(C)C)=O)C(C)C2)=O)CC1 c1(C(N2CCC(CCOC)(NC(C3CCC3)=O)C2)=O)c(O)ccc(Br)c1C CS(=O)(=O)CCCCCCCC(=O)N1CCC(c2cnccn2)C1 C(C(CC(=O)N1CCC(NC(C23CCC(CC2)CC3)=O)C(O)C1)C(F)F)N(C)C c1(C=O)cc(F)cc(F)c1F.CC(C)C(CN(C)C)C(=O)N(CC(C)(C)C)C.N CCC(C)(O)C(=O)NC1CCOCC1NC(=O)Cc1ccn(-c2ccccc2)n1 N1(C(c2c(C)snc2)=O)CCC(NC(=O)CC2CCOC2(C)C)C(C)(C)C1 c1(C(=O)NCC2N(C(c3c[nH]c(=NC)o3)=O)CC2)ccc(Br)c(F)c1F N1(C(c2c(C)[nH]cc2)=O)CC2C(CC(N3CCCCC3CC(C)C)=O)C2C1 C=CC1(C(=O)NCC2C3CCCOC23)CCN(C(=O)CCCn2cccn2)C1 C1(C(N(C(CCNC(C2(COC)CC2)=O)C)C)=O)CNc2ccccc2O1 C(C(C)(C)C1=CCCC1)CCCN(C1(C(=O)N)CCOCC1)C.C(=O)C(Cl)Cl N1(C(c2cc[nH]c2C2CC2)=O)CCC2C(CCCN2C(=O)CCOCC(F)F)C1 CCCCC(C)(F)C(=O)NC1CN(C(=O)C(C)(C)C(C)O)CC2(CC2)C1 N1(C(=O)C2CC2)CC2CC1CN2Cc1ccncn1 N1(C(C2(C(=O)NC)CCC2)=O)CC(NC(C2(Br)CC2(C)C)=O)C(O)C1 N1(C(C(C)CO)=O)CCCN(C(C2(c3ccno3)CCC2)=O)CC1C C1(O)(C(N(C(C)CN2CCCCC2)C)=O)CCOC1(C)C C1(CCOC)CN(C(=O)CC(=O)OC)CCN1C(=O)COCCCF C(=O)(C(O)CCC(C)C)NCC1CN(C(CCCOCC=C)=O)CC1(F)F C1(C(=O)NC2(C)CC(NC(c3ccsn3)=O)C2)COc2cc(F)ccc2C1 CC1COCC(C(=O)NCC(C)(C)NC(=O)CCCc2ccccc2)O1 c1(C(N2CCC(C)(CNC(C(CC#C)(C)CC)=O)C2)=O)cc(C#N)c(F)cc1F C(=O)(CCCCCCCCC1CC1)N1CCC(NC(CC(C(C)C)OCC)=O)C1 CC1C(NC(=O)C(C)CCCc2ccccc2)CCCN1C(=O)CN1CCCC1 C1(NC(c2cc(N)c(N)nc2)=O)CC12CCC(NC(=O)C(Cl)=CCl)CC2 C1(NC(=O)C(c2cccc([N+](=O)[O-])c2)O)CCc2nccn2C1 Cc1ncc(C(=O)NCC2CN(C(c3cc(C)sc3C)=O)C2)c(C2CC2)n1 C(C)(N=c1[nH]c(=NCCCN(C)C2CC2)[nH]c2ccsc12)c1c(C)nns1 C1(C(=O)NCCC2CCCC3CC23)C2CCN(C(C3CC4CC3CC4=O)=O)CC12 c1(C(=O)NCC(CNC(C(c2cccc(C)c2)C)=O)O)c(C)cnnc1O C1(C(N2C(C)C(NC(c3sccc3C#N)=O)CC2)=O)CCS(=O)(=O)CC1 C12(CCN(C)C(C3CCOCC3)=O)CC3CC(CC(C3)C1)C2 C1(C(=O)NC2(CF)CCN(C(CC(=O)OC)=O)C2)CCC(N=[N+]=[N-])CC1 Cc1ccnc(C(F)(F)C(=O)NCCN(C(=O)CCCF)CC(C)O)c1 c1(C(=O)N)ccc2nc[nH]c2n1.C(C)(CNC(=O)CC1(C)CCC1)(C)OC Cc1sc(C(=O)NCCCc2cnn[nH]2)cc1Br Cc1ncsc1C(=O)NCC1CC1.c1(C(NC)=O)sccc1-n1ccnn1.C c1(CC)ncc(C(=O)NC(C)(C)CNC(c2ccc(C)cc2N)=O)c(O)n1 c1(C(N2CC(OC)(CNC(=O)CC)C2)=O)c(C)cnnc1O.c1ccccn1.S C1(NC(CCC#C)=O)CN(C(c2cccc(OCC3CC3)c2)=O)CCC1CO CC1=NOC(C(=O)N(C2CCN(C(=O)COC3CCCOC3)CC2)CCO)C1C N1(C(c2c(CC)con2)=O)C2CC=C(C(=O)NCc3cccnc3C)C1CC2 C1(C=O)CCOCCN1C(=O)CCc1cc(C)no1.C(=O)(CCC1CC1)NC.N N1(C(CCSCCCC)=O)CCN(C(=O)CCF)C(c2cccc(Cl)c2)C1 C(=O)(C1=COCCO1)NCCN(C(C1CCCN(C(=O)C2CC2)C1)=O)CC C(=O)(C(C)(C)CC(C)(C)C)N1CC2C(CCNC(C=CCOC)=O)(CC2)C1 C(C(CC(C)C)C(=O)NC1C=C(C)CCC1)NC(c1scc(C)c1)=O C1(CNC(C2C(C)C2)=O)(NC(=O)C(C)(F)c2ccon2)CCOCC1 C(=O)(N(CCC(=O)NC1CCCCCCC1)OC)c1n(CC)ccc1 N(C=CC(=O)C(F)(F)F)Cc1cc(C)nn1C.N1(CC)CCC(F)(C=O)CC1 c1(CC(=O)NC2(CNC(Cn3c(C)nnn3)=O)CC2)cccc(O)c1 Cc1cc(C(N2CCOC(CNC(c3cncc(CO)c3)=O)C2)=O)ccc1F Cc1cccc(F)c1CC(=O)NCC(C)CNC(C1(C2CC2)CC1)=O c1(C(=O)NC2CC(CC)(CC)N(C(C3CCC3OC)=O)C2)cc2cnccc2[nH]1 CC(C)CC(C)CNC(C1CCC(C#N)CC1)=O.C1(N(CC=O)C)CCCC1.N N1(C(CC2(CSC)CC2)=O)CCCC2CCCC12.C1(C(=O)N)CC1.C1CCC1 O=S(=O)(c1sccc1F)NCC1C2Cc3ccccc3C12 C(=O)(CCCCC1CC1)N(CCCCNC(=O)C)C.C12(C=O)CCCC1C2.N Cc1nc(O)ccc1C(=O)NC1(C(=O)NOCC(=O)N(C)C)CCC(C)(C)C1 N1(C(c2cc(CC)on2)=O)CC2CCC1C(CNC(C1(C)CCCO1)=O)C2 c1(C(=O)N)ncc(C)cc1C.c1(C(N2C(C)CC(OC)C2)=O)nn(C)c(Cl)c1Cl Cc1sc(Br)c(CNCC2OC(=O)CC2(C)C)c1C c1(OC)ccc(Br)nc1NC(C1CC(F)(F)CN1C(c1cccc(O)n1)=O)=O Cn1ccc2c(NC(C3CC(O)CN3Cc3cccc(C(N)=O)c3)=O)ncnc12 C(=O)(CCC(F)(F)F)N(C1CCCN(C(=O)CC2COCCOC2)CC1)C n1(CC(=O)NC(C)CC2CN(C(C3OCCO3)=O)C2)cnc2c(cnn2C)c1=O c1(NC(c2ccnc(Cl)c2)C)nc(N2CC=C(C(C)(C)C)CC2)nc2sccc12 c1(C(=O)NCC2(O)CCN(C(CCC=C)=O)C2)cnn2cc(S(C)(=O)=O)cnc12 N1(C(c2cnc(Cl)s2)=O)CCN(C(C2(c3ncco3)CC2)=O)CC1 CCCCC(O)CC(=O)N(CCC(=O)Nc1ccc(CC)cc1)CCCO c1(CC2(C(N3CC4CC3C4)=O)CC2)ccccc1Br n1(CCC)cc(NC(=O)N(CC)CC2CCCO2)cn1 n1(CC)ccc(C(=O)NCCC2CN(C(C3CC3c3ccncc3F)=O)C2)c1C N1(C(=O)NCCC2CCOC2)CCC(C(=O)Nc2ncc[nH]2)CC1 c1(Cn2cc(-c3c(C(=O)OC)cccc3)nn2)ccc(-c2ccncc2)cc1F c1(-c2ccn(C(C)C)n2)cnc2n[nH]c(C(N3CCNC(C)(C)C3)=O)c2c1 C12(CNC(C(CC(C)C)n3ccnc3)=O)CCCCC1N(C(=O)CN(C)C)CC2 N1(C(CCNC(=O)NC)=O)CC2CCC1C(CNC(c1ccc(S)o1)=O)C2 c1(CCC(=O)NCCC(C)(C)NC(C=CSC)=O)ccc(Cl)nc1 N1(C(C(CC=C)C)=O)CC(C(=O)NCC2(CCOC)CC2)C2(CC2)C1 N#Cc1cncc(C(=O)NCCC2(O)CCCN(C(=O)Cc3cnc[nH]3)C2)c1 Cc1nc(C(N2CCC(C3CCCCN3C(C3CC34CCC4)=O)CC2)=O)c(C)o1 C1(NC(c2ccncc2Br)=O)CN(C(c2ccc(O)nc2)=O)CC2CC12 C(CCF)(C(=O)N1CCC(C)(N(C)C)C1)NC(COCC(=O)OC)=O C1(NC(C2CC23CC3)=O)CCCC12CN(C(c1sccc1-n1ccnn1)=O)C2 c1(CC)occc1C(=O)NCC1CC1(F)F.C1(C=O)CC1(C)C(F)F.C n1(C2CC(C(=O)NC3C(=C)C3)C2)cc(C(C)(C)CC)nn1 N#CC1(C(N2CCC(CCNC(C3CCS(=O)CC3)=O)C2)=O)CC2(CCC2)C1 N1(C(c2onc(OC)c2Br)=O)CCCC(NC(=O)CC(C)C(F)F)CC1 C12(NC(c3cccc(CC)c3)=O)CCCC1N(C(c1cccc(N)c1)=O)CCC2 c1(N2CC(c3n(CC)cnn3)OCC2)nc2ccc(C)cc2s1 CN1CCC(C(=O)NCc2nncn2C)(NC(=O)CC#N)C1 C1(C(=O)NCC(c2cnc[nH]2)C)(NC(CC(C)SC)=O)CCC(C)(C)C1 O=S(=O)(c1ccc(NCC(Cl)Cl)c(Cl)c1)NCCCc1c(F)cccc1F N1(C(c2c(C)n(C)cc2)=O)CCC(NC(=O)C(C)Cc2cnco2)C(CO)CC1 C1(NC(C(CC)(C)F)=O)CCN(C(C2CC=CC2)=O)CC1CO C1(COC)CCCN(C(=O)CC2CC(F)(F)C2)C1.C(=O)CCC.C(N)=O.N C12(NC(c3cn[nH]c3)=O)CCC1CN(C(=O)C=Cc1sccc1Br)C2 C=CCC(C)(CC)C(=O)N1CCC(C)(NC(=O)CN2CCCS2(=O)=O)CC1 C1(NC(c2c(C)nn[nH]2)=O)CC2CCC1CN2C(c1ocnc1C)=O C(C(=O)NCCC1CCCO1)(C(C)(C)C)NC(CCCOC(C)(C)C)=O c1(C(=O)NCC(CN(C(CCNC(=O)NC)=O)C)C)ccnc2[nH]nnc12 C1(C(N2CCC(O)(CC)C2)=O)CC(CC)CCN1C(=O)CCc1cnoc1 CC1(C)C(NC(=O)CCC2CCOCC2)CC1C(=O)NCC1CSCCO1 C(CC(COC(=O)CCN1CCOC1=O)OC)OC C1(C)(CC)CC(NC(C2(C(C)C)CC2)=O)CN1C(c1cncc(F)c1)=O c1(CC)ccc(C(N2CCC(O)C(C(=O)NC3CCCOC3)C2)=O)cc1[N+](=O)[O-] c1(OC)ccc(C(=O)NCC(O)CNC(=O)Cn2nc(O)ccc2=O)cc1C C1(C(=O)NCC(C)NC(C2(CC)COC2)=O)CCS(=O)(=O)N1 O(N=C1CCCCCC1)CC(N1CCC(NC(C(CC)N(C)C)=O)C(CC)C1)=O c1(OC)cccc(CC(=O)NC2CC2C)c1Cl.c1(C(=O)N)cc(C)nc(O)c1 N1(C(C(C)NC=O)=O)CC(C(=O)NCc2nocc2C(N)=O)C(F)(F)C1 C1(NC(CCNC(NC)=S)=O)CN(C(=O)CC2CCCC2)Cc2nccn2C1 c1(C(=O)NCC(C)N(C(C2CCCCO2)=O)CC)cc2sc(C)nc2[nH]1 N1(C(COCCC)=O)CCC(CNC(=O)C(C)CC)C1(C)C N1(C(C2CCC(=O)C2)=O)CCC2C(NC(=O)COCC3CCCCO3)C12 C(=O)(C(CC)C(C)C)NCC(C)(C)OCCNC(C1ON=C(CC)C1)=O CC(C)CC(CNC(C1CCCN1C=O)=O)NC(=O)C(c1ccccc1)C1CC1 c1(C(=O)NCC(CCCC)NC(c2n[nH]cc2SCC)=O)ccc(C)c(O)c1 CC1CN(C(c2ncn3c2CCC3)=O)CCN(C(C2CCOC2)=O)C1 c1(C(N2CC(OCCNC(CCC)=O)C2)=O)cc(=O)oc2ccc(O)cc12 C12(C(=O)OC)COC(C(=O)N(CC(O)C)C)(C1)C2.C1(C=O)CCN(C)CC1 C1(NC(c2n(CCC)ncc2)=O)CCOCC1NC(=O)C(C)=CCOC N1(C(c2ncc(OCC)cn2)=O)CCC(C=CC=O)CC1.N1(C)CCC(O)CC1 c1(C(N2CC3N(C(CCOCC)=O)CC(C3)C2)=O)c(N)cc(F)c(Br)c1F N1(C(C(n2ccc(C)n2)(C)C)=O)CC2CCC1C1CN(C(C3(C)CSC3)=O)CC21 N1(C(C2(C(C)NC(C3CC34CCC4)=O)CC2)=O)CCC2(CNC(=O)O2)C1 C1(NC(c2c(OC)csc2)=O)CC(F)CN(C(C2(C)CC=C(C)CC2)=O)C1 C(=O)(C1c2ccc(O)cc2CCN1C(c1ccc(-c2cscn2)cc1)=O)OC Cc1ccn(C)c1C(=O)NCC(CNC(=O)CCc1ccccc1)CO n1(CC)cc(C(=O)NCCS)c(C)n1.C1(N(C(C)=O)CCO)C2CCCC12 CC1C(NC(=O)Cc2ccc(F)cn2)CC2CCC1N2C(=O)C#CC1CC1 n1(C(C)C)ccc(=NC(=O)C23CC(CO2)N(C(=O)C(c2ccn(C)n2)C)C3)[nH]1 N1(C(c2c(C)n[nH]c2C)=O)CCC(C)C(NC(C23CC2C3)=O)C1C C1(O)(CN(C(c2cc(C)n(C)c2)=O)C)CCN(C(=O)CC2C=CCC2)CC1 N1(C(c2ccc(CCC#N)cc2)=O)CC2CCC2(CNC(c2ccoc2)=O)C1 N1(C(CNC(CNC(C)=O)=O)=O)CC2CN(c3nc(Cl)ncc3Cl)CC2C1 c1(C(=O)NC2(C)CC(NC(CCOC(C)C)=O)C2)ccc2nccnc2n1 N1(C(c2c(CN(C)C)nccc2)=O)CC2CCC2(NC(C2CNC(=O)C2)=O)C1 C(=O)(CCCCCCNC(=O)CC12CCC(CC1)C2)N(C)CC1CN(C)C1 C1(Oc2cc(C(=O)OC(C)(C)C)nc(C(=O)O)c2)CCCCN(CC)C1.C C#CCCCCCC(=O)N1CCC(NC(=O)CN(CC)CC)C1C C1(NC(C(CC=C)OC)=O)CN(C(c2cnn(CCOC)c2)=O)CC(F)(F)C1 C1(C(=O)NCC2C(NC(c3ccc(C)nc3)=O)CC2)CCOCC12CCC2 N1(C(CCCC)=O)CCOC(C(=O)NCC2CC2(F)F)C1 C1(C(=O)NCc2cocn2)CCC2(CN(C(=O)CCN3CCOCC3)C2)O1 c1(C(=O)NC2C=CCN(C(Cc3cc(C)no3)=O)C2)cc(Br)cc(Cl)c1C C(=O)(C1=NOC2(CCC2)C1)N1C(CNC(=O)C(c2ccccc2F)O)C=CC1 C1(CNC(C2(C)CCN(C)C2)=O)CN(C(C2(C)CCC2)=O)CCN1C.C1CC1 C1(CNC(C2CNC(=O)N2)=O)CCC(C(=O)NCCCCc2cnc[nH]2)CC1 c1(C(=O)NC(C(C)NC(CCOC(C)=O)=O)C)cc(-c2ccoc2)on1 N1(C(CCCC(CC)NC(C2CC3(CCO2)CC3)=O)=O)CCn2c(O)nnc2C1 C1(NC(C2(CC#C)CC2)=O)CN(C(c2snc(Cl)c2Cl)=O)CC1C(F)F Cc1nc(N(C)Cc2cccc(OCC(=O)O)c2)c2c[nH]nc2n1 C1(C=O)CC(C)CC(C)C1.Cc1onc(C2CC2)c1C(=O)NC.C1C=CCC1 N1(C(Cc2cncc(C)c2)=O)Cc2n[nH]cc2C1C(=O)NC(C)Cc1ccco1 c1(C(N2CCCC(NC(CSSC)=O)C2)=O)ccc(F)c(C)c1 Cc1cccc(CN2CCC(CCS(C)(=O)=O)CC2)c1N C1(NC(C(C)C(C)(F)F)=O)CC12CCN(C(c1cccc[n+]1[O-])=O)CC2 c1(NS(CCOCCOC)(=O)=O)c(C)noc1C(C)C N1(C(C2CC(C)(CC)C2)=O)CC2(C)CCC1CC2.c1(C=O)ccc(C#C)cn1.N C(=O)(C1CSc2ccccc21)N1C(CNC(c2nc(C)oc2)=O)CCC1.C1CC1 C1(C(=O)NCC2(O)CCOCC2)OCCCC1c1ccccc1.n12cc(nn1)C2 N1(C(C(=O)NC(C)C)=O)CC2(C1)SCCC2.C1(CC=O)CC(C)(C)CCO1.N c1(C(C(=O)NCCCN(C(C=CCCC)=O)CCO)C)cccc(Br)n1 N(C(=NCC1CC1)NC1CCCC1)CCNCc1n(C)ncc1.C(C)(C)C.O C(=O)(CC(C)P(C)(C)=O)NCCC1CCN(C(c2n[nH]c(C)c2O)=O)C1 N1(C(C(CCCC)NC(c2ccc(F)cc2F)=O)=O)CCC2(CNC(=O)O2)C1 Nc1cc(Cl)cc(F)c1C(N1CCOC(C)C1)=O.c1(C(=O)N)cn(C2CC2)cn1 C1(NC(c2cnc(C)[nH]2)=O)CCCN(C(=O)Cn2cc(C3CCC3)nn2)CC1 c1(C(=O)NCCN(C(C2(COC)CCCO2)=O)C)ccc(C2CC2)cc1 N1(C(c2c(C(C)C)occ2)=O)CCCCC(NC(C23CC(C)(CCO2)C3)=O)C1 C#CCC(C)C(=O)NCC1CN(C(c2ccc(SCCC)cc2)=O)CCO1 C1(NC(c2n(C(C(=O)OC)C)nnn2)C2(CO)COC2)CCCCCCC1 c1(C(=O)NC(C(C)NC(=O)C(CO)N(C)C)CO)cc2ccncc2s1 CCC(C(C)(C)C)NC(=O)CONC(=O)CC1NC(=O)NC1=O C(=O)(C(F)C(C)(C)O)N(C1CCN(C(C2(C)CCN(C)C2)=O)CC1)CC(F)F C1(NC(C2CC(=C)C2)=O)CC2CC1CN(C(c1ccc(F)cc1C1CC1)=O)C2 c1(CC(=O)NC2(CN(C)C(C3C4CCC3CC4)=O)CC2)ccc2nc[nH]c2c1 C1(C(N2CCCC2C=C)=O)(CNC(CCCOCC=C)=O)CC12CCC2 C(=O)(CCCCCC#N)N1CCC(O)(CN(C(C2OCCC(C)C2)=O)C)C1 c1(C(N2CCC(CCOC)(NC(c3cnoc3)=O)C2)=O)cc(F)c(N)cc1.O c1(NC(C(C(C)(C)C)CNC(=O)Cc2cn[nH]c2)=O)cccc2cnc(Cl)cc12 N1(C(CCC=CC)=O)CC(NC(=O)Cc2c(F)cncc2Cl)CC(O)C1 C12(C(N(CC(CCC)O)C)=O)CC(CO)(CN1C(=O)CC1CC1C1CC1)C2 N1(C(c2[nH]cc(C)c2)=O)CC2(CCN2C(=O)C(C)C2CCCC2)C1 C1(C(C)NCC(=O)Nc2ccncc2)CN(C(c2ncccc2F)=O)CCC1C C1(CNC(=NC)NCC2CCCN(C)C2c2ccnn2C)CCCC(C)(C)C1 Cc1nccc(C(=O)NC2COCCN(C(=O)C(C)c3cc[nH]n3)C2)c1N N1(C(C=CC(C)C)=O)CC2CCCC1C2CNC(=O)CCC(F)F c1(OC)ccc2c(c1)CN(C(C1C=CCN1C(=O)CC(C)O)=O)CC2 c1(C(N2CCC(C(C)(C)C)(CNC(CCCCC)=O)C2)=O)cc(Cl)ccc1C C1(NC(CCOCCC)=O)COC2(CCN(C(c3ccc(CO)cn3)=O)C2)C1 N1(C(c2c(SCC)nccn2)=O)CC(N(C)C(c2ccccc2C)=O)C2(CC2)C1 N1(C(C(c2cccnc2)NC(c2cc(C)sc2C)=O)=O)CCN(C)C(C(=O)O)C1 N1(C(CCCCC=CC)=O)CC(CNC(C2CC(C)N(C)C2)=O)CC(C)(C)C1 N1(C(c2sc(C)c(O)n2)=O)CCCC2(CCCCC2NC(=O)C(Cl)=CCl)C1 CN1CCN(C)CC(NC(C2CCCN(C(c3ccccc3)=O)C2)=O)C1 N1(C(c2ccnc(C)n2)=O)CC2(CCC2NC(=O)CCC2CC2(C)C)C1 c1(COC(CCSCCCC)=O)cc(C)c(F)c(Cl)c1 C1CCC(C=O)CC1.CCC(C)C(=O)N.C12(CC=O)CC(C1)C2.C(C)(C)C C(=O)(CCCCC(C)(C)OC)NCC(CNC(C1(CC#C)CCC1)=O)O C1(NC(c2c(C#C)c[nH]n2)=O)CCCCCN(C(=O)Cc2cc(F)ccc2F)C1 c1(N2CC(C)CCC(C)C2)nc2ccsc2c(=NCc2ccncc2)[nH]1 c1(C(=O)NCCC2CCCN(C(=O)C3=NOCC3)C2)c[nH]cc(Br)c1=O C1(CC(N2CC(CCn3cc(CC(=O)OC)nn3)C2)=O)CCCC1(F)F C1(NC(C2(N(C)C)CCCC2)=O)CCCN(C(c2cccc(N(C)C)c2)=O)C1 N1CCCC(CC(F)F)C1.c1(C(=O)O)ccc(C(F)(F)F)[nH]1.c12c[nH]nc1CN2 c1(C=O)c(F)cc(C(F)(F)F)c(F)c1F.C1(CCNC(CSC)=O)CCOC1 C1(CC)CN(C(c2cn(C)cn2)=O)CC1NC(=O)C=Cc1cccnc1 c1(NC(C2CC3CC3N2C(c2ccnc(F)c2)=O)=O)c(F)cc(F)cc1Br c1(C(C(=O)NCCN(C(C(CC)NC(C)=O)=O)C)C)ccc(OC)c(O)c1 c1(C(=O)NCCCC(C)NC(Cc2c(C)n[nH]c2C)=O)c(N)cccc1Cl C(c1ccn(C)c1)=CC(=O)N(CCCC)C.C(=O)(C(C)C)N(CC=O)C.N c1(C(=O)NCC(CNC(C2(C#N)CCC2)=O)OC)ccc(NC=O)cc1 c1(C(N2CCN(C(c3cc(C(=O)OCC)n(C)n3)=O)CC2)=O)ccc(N)cc1C N1(C(C=Cc2cnc(C)s2)=O)CC2CCN(C(=O)C(C)(C)N(C)C)CCC2C1 CC(CC(=O)N1CC(CO)(NC(=O)CC(F)F)C1)CC(F)(F)F S(=O)(=O)(c1cc(C(=O)O)cc(C(=O)O)c1)N(C(c1c(C)nc(C)s1)C)C c1(C=O)ccoc1C1CC1.c1(C2C(C(N(CCO)CC)=O)C2)ccco1.CC CC#CCCCC(=O)NCC1CCCC1NC(c1nc(C)n(-c2nc[nH]n2)n1)=O c1cccc(C(=O)N(N)C)c1Cl C1(C(=O)NC2CCC(NC(CCNC(=O)CO)=O)CC2)Cc2cccnc2C1 C(C)(C)(C(=O)N(CCC(=O)NCCc1ccncn1)CCCO)N(C)C CC1=CCN(C(c2ccc(C(C)O)cc2)=O)CC1.C1(C(=O)OC)CC(C=O)C1.N N1(C(=O)NC(CNS(CC)(=O)=O)C)CCC(C(=O)OC)C(C)C1 Cc1cc(N2CC(OCCNC(C3CC4CCCC34)=O)C2)n2nc(C)nc2n1 N(S(=O)(=O)N1CCCCCC1)Cc1nc(-c2cccc(C(=O)O)c2)sc1 Cc1ncc(C(N2CC(NC(=O)CC(F)(F)Cl)C(C)C2)=O)n1C N1(C(C(C)(C)F)=O)CCC(C#N)(NC(c2c(Cl)cncc2Cl)=O)C1 C1(O)(CNC(C2C(CC)CCC2)=O)CCN(C(c2ncc(OC)cn2)=O)C1 CS(=O)(=O)C1(C(=O)NC2CCC2)CCCC1.c1(C(=O)N)ccc(F)c(Cl)c1F Cc1ccccc1C(N1CCC(CO)(NC(C23CSC(C2)C3)=O)C1)=O N1(C(CC2(OCC)CC2)=O)CCC(C(C)C(=O)NCCc2cccnc2F)CC1 C1(NC(c2cn(C(C)C)nn2)=O)CN(C(=O)C(O)P(C)(C)=O)C2(CCOCC2)C1 C(=O)(C(C(C)(C)O)NC(C1OC2CCC1C2)=O)NCC(C)C Cc1nc(C(=O)OCc2nnc(C(C)C)s2)c2c(ncn2C)n1 C1(CC(=O)N(C)C)CCN(N2CCCC3=CCCCC23)CC1 c1(C(=O)NCC(C)NC(c2cc(O)n(C)n2)=O)cc(Cl)cc(Cl)c1N C12(C(=O)NC(C)CN(C)C)CCC(C=O)(CC1)CC2.c1ccnc(C2CC2)c1 Cc1cc(Cl)c(C(=O)NCC)s1.C1(C(C=O)(C)C)CCC(O)CC1.C1CC1.N C1(O)(C(N(C2CC2c2ccccc2)C)=O)CCCN(C(N)=O)C1.Cc1ccsc1 N1(CCNC(=O)CSc2cn[nH]c2)CCCC1=O.C1(c2ccco2)C(=O)N1 C1(C(N(CCCNC(c2cccc(OC)c2)=O)C2CC2)=O)CC12CCSCC2 CCCCCCCCC(CO)NC(=O)CSCC(N1CCOCC1)=O c1(OC)nc(Cl)c(C(N2CCC(OCCCNC(=O)C3=CCCO3)CC2)=O)s1 c1(C(=O)NC2CCCN(C(=O)C(F)=C3CCC3)C2)nccc2c(Cl)cccc12 c1(C(=O)OC)cc(Cl)cnc1NC(C1CCCN1C(=O)N)=O.c1cccnc1Cl c1(C(=O)NC(CNC(C2C(C)C2)=O)(C)C2CC2)cn(C)c(=O)n1C C1(NC(CN(C(C)C)C)=O)(CNC(C2CCC2F)=O)CCCCCC1 C(=O)(C#Cc1ccc(F)cc1F)N1CC(C(F)(F)F)CC(C)C1 C(=O)(C(C(C)(C)C)OC)N1C(CCCNC(C=CC)=O)CCCC1 C1(C(N2CCN(C(c3n(C)ccn3)=O)CC2CCO)=O)CCCCC(C)(C)C1 c1(OC)ccc(C=Cc2nc(CSC3(CO)CC4CC4C3)no2)cc1 C1CC2CCCC2C1.N1(C(C2C(COC)CCO2)=O)CCCC1(C)CCC(=O)NC c1(OC)nccc(C(=O)NC2CC(NC(=O)CC3CCN(C)CC3)C2)c1Cl Cc1nc(C)c(CNC(c2c[nH]nc2-c2ccc(F)c(Cl)c2)=O)nc1C Cc1cc(C(=O)NCC2CCC2NC(C2CC2C#N)=O)cn1C CN1CC2(CCN(C(=O)C(c3cccnc3)NC(=O)CN3CC4CC4C3)C2)C1 C1(C(=O)NCCC(C)F)CCCC(NC(c2ccon2)=O)CC1 c1(COC)ccsc1C(=O)N(C)CC1CCN(C(=O)C(C)N2CCC2)C1 N1(C(c2nc(C)sc2C)=O)CCCC(F)(C)C1.C1(C(=O)N)CCN1C1CCCC1 C1(C(C)C(=O)NCC2(N(C)C)CCC2)CCN(C(C2CC=CC2)=O)C1 N1(C(c2c(OC)nccc2)=O)CC2(CCCC2NC(c2c(Cl)cnn2C)=O)C1 C1(C)CCCN1C(C1C2CCC1(c1cccnc1)C2)=O.C(C(=O)N)=CCOC c1(C(=O)NCC(CNC(c2cnc(OCC)s2)=O)O)ccc(Cl)c(F)c1 Cc1ccc(I)c(C)c1NC(C1CC12CCN(C(c1cc(F)cn1C)=O)C2)=O N1(C(c2ncc(OC)cn2)=O)CCCC(F)(C)C1.C(=O)C(C)(C)CC1CC1.N C(=O)(C(O)P(C)(C)=O)NC(CNC(c1nc(CCCC)sc1)=O)(C)CO N1(Cc2cc(C)cc(Cl)c2)CCC(=O)N(Cc2cc(C(C)C)on2)C1=O c1(CCC(=O)NC2CN(C(C(COCC)C)=O)CC2C)ccc2ncccc2c1 CCC(CC)C(C(=O)N1CCN(C(=O)C=Cc2nc(C)co2)C(C)C1)OC Cc1cc(N)ccc1C(=O)NCCN(C1CCCC1)C(c1ccc(=O)oc1)=O Cc1c(CC(CNC(C2CNC3CC23)=O)CO)cccc1Br c1(C=O)c(F)ccc(Cl)c1N.Cc1cc(C(=O)NCC2COC(C)C2)n(C)n1 Cc1c(C(N2CC(CNC(c3cncc(Cl)c3)=O)C(F)(F)C2)=O)ccc(F)c1F c1(OC)cccnc1-c1nc(-c2ncc(Br)cn2)n(C2CCCSC2)n1 N(C(=NCCCC(=O)NCCN1CCOCC1)NCCC(=O)C1CC1)CCC(C)C N1(C(C(N)=O)=O)CCC(CC2CCN(C(=O)C=CC(N3CCOCC3)=O)C2)CC1 c1(CNC2C(CNC(CC(C)c3ccccc3)=O)CCCC2)ccc(Cl)nc1O N1(C(C(CC#C)(C)NC(C2COCC(C)O2)=O)=O)CCc2n[nH]cc2C1 c1(N(c2n(CCCOCC)c(-c3cnc(O)nc3)nn2)C)cccc(C)c1Br c1(CNC(=NCC)NCC(c2ccccc2)O)ccc2cnn(C)c2c1 C(C)(c1ccccc1)=CC(=O)NCC(CCCC)NC(=O)CCC1(C)CC1 c1(CNC(C(C)NC(C2CCO2)=O)=O)ccccn1 CC1=CCCN(C(c2sccc2OC(F)F)=O)C1.C1(C(=O)N)CC2(C1)CC(O)C2 C(CC(C(=O)NC1CC(CCC(N)=O)C1)NC(=O)CCC1CCCO1)SC Cn1nc2c(c1C(=O)NCC(O)CNC(=O)CC1CCCCCO1)CCCC2 C1(F)(CNC(CSCCCC)=O)CN(C(=O)C(C)OCC2CCCO2)C1 c1(C(=O)OC)ccc(N2CCCCC2CNC(C2CC(CC(F)F)C2)=O)nc1 C12(NC(c3ccc(NC=O)cc3)=O)CCCC1N(C(C1(C3CC3)CC1)=O)CC2 C1(CC(=O)N)CCN(C(C2CC(C(=O)N)C2)=O)C1.N1(C2CC2)CCOC1=O c1(CC(=O)NC2CC23CC(NC(=O)C2=COCCO2)C3)cc(F)cc(Cl)c1 C12(NC(C3CC4(CCC4)CO3)=O)CCCCC1CN(C(c1cc(F)cs1)=O)C2 N1(C(CC2(OCC)CC2)=O)CC2CCC2(C(=O)N(C2CCOC(C)C2)C)C1 CC(C)C(C#N)C(=O)N1CCN(C(C2CCCN(C(C3CCC3)=O)C2)=O)CC1 C1(C(N2CC(OCCNC(C(CC)OCC)=O)C2)=O)CCn2ccnc2C1 c1(N2C(CCNC(C(C)(C)S(C)(=O)=O)=O)CSCC2)nc2cc(Br)ccc2o1 c1(C(=O)NC2CCC(NC(c3ncc(CC)nc3)=O)C2)c(F)cc(Cl)cc1Cl C1(C(=O)NCC(CNC(CCc2onc(CC)n2)=O)F)CCCC(OC)C1 c1(C(=O)NCCC2(C)CC2)ccccc1-n1cccn1.C1(C=O)CCC1.N N1(C(=O)OC(C)(C)C)CC(C(F)(F)F)OCC1CC(=O)N.C1OCCCC1(C)C C(=O)(C(CC(C)C)OC)NCc1oc(C(=O)NCC(=C)Br)c(C)n1 N1(C(c2cc(OC)n[nH]2)=O)CCC(C)C(CC(=O)NCCCC(N)=O)C1 C(=O)(CC(CNC(=O)Cc1scnc1C)C1CCC1)NCCC(=C)C c1(CC(=O)Nc2ccccc2Cl)[nH]nc(NC(C2CC=CC2)=O)c1Br Cn1nc(C(F)F)c(C(=O)NC2CC3(C2)CCC3)c1C#N.C(=O)COC(F)F C(c1ccc([N+](=O)[O-])cc1)=CC(=O)NC1CC(NC(=O)CC)C1.C1CCCC1 N1(CCOC)CCCC1C(=O)N(C)CC1(O)CCCC1 c1(OC)nc(C(=O)NC2(CC)CCCC2)cc(O)n1.c1(C=O)ccc(C)nn1.N CN1CC(C(=O)NC2CC(NC(=O)C(F)(F)c3cnccn3)C2)NC1=O N1(C(c2cc(OC)nc(F)c2)=O)CCC(C2CCN(C(c3csc(C)n3)=O)C2)C1 C1(O)(c2cn(CC(=O)NCC3CCCC(C)C3)nn2)COC(C)(C)OC1 C12(NC(C(CC)F)=O)CC3CC(C1)CC(C)(C3)C2.c1(C(=O)N)ccn(C)n1 C12(CNC(CCC#CC)=O)CN(C(c3cccc(=O)o3)=O)CC1CCO2 N1(C(=O)COC2CCN(C(C3C4CC5C(C4)C35)=O)C2)CCC2(CCCC2)C1 C12(NC(C3CN(C(C)C)C3)=O)CC1CN(C(c1ccccc1)=O)C2 C1(C(=O)NC(CC)CN2CCCC2)CC12CC(NC(c1cc[n+]([O-])cc1)=O)C2 O=C(CS(=O)(=O)CCO)NCCC1CCN(C(C2CCCCC23CCC3)=O)C1 C1(CCNC(C2CCC(NC(C3(Cl)C(C(C)=O)C3)=O)C2)=O)CC2CCC1O2 C1COCC(=O)N1C.C1(CC=C)(C(=O)NC)CCN(C(=O)C(C)=C2CC2)C1 c1(C(N2C(C)CC(NC(=O)C=C3CCOCC3)CC2)=O)cnc2ccsc2c1 N1(C(c2[nH]n(C)c(=O)n2)=O)CC(NC(C2CCCNC2=O)=O)C(N=[N+]=[N-])C1 Cc1cc(OCC(O)CN2CC(O)C(F)(F)C2)cc(C)c1 C1(N(C(C=CCC)=O)C)CCC(CNC(C2CCOC2=O)=O)CC1 C(=O)(C1CCCc2n[nH]cc21)NCC(C)(O)CNC(=O)C1=CCOC1 CC1(C)OCCC1(O)C(=O)NCC(C)(C)Cn1cc(C2C(C)(C)C2(F)F)nn1 C1(CC)CN(C(=O)C(F)(F)c2nccs2)CCN1C(c1cccc(CO)c1C)=O CC1CCN(C(c2cnc(OCC(F)F)cn2)=O)CCN1C(C1CCC(C)O1)=O N1(C(CCCC#C)=O)CCCN(C(=O)CN(c2ccccc2)C)C(C(C)C)C1 C(C)(CCCNC(C1CCCCC1)=O)NC(C1(CC)CCC1)=O N1(C(CCC=C=C)=O)CCOCC(NC(=O)COc2ccccc2Cl)C1 N1(C(c2cc(CC)nc(O)c2)=O)CC2(C1)SCCC2NC(C1COCCN1C)=O C1(NC(CN(C)C2CC2)=O)COCCC1NC(c1cscc1C(F)(F)F)=O C1(C(=O)NC(C=CC(=O)NC(CCOC)COC)(C)C)CCC(C)CC1 c1(C(=O)NCC2CN(C(CC3(C#N)CC3)=O)C2)coc2c(Br)cccc12 Cc1cc(C)c(C)c(C(N2CCC(CNC(c3occc3F)=O)C(C)C2)=O)c1C c1(C(=O)NCC(C)(C)NC(C(N2CCOCC2)C)=O)ccc(S(N)(=O)=O)s1 C1(CNC(C=COCC)=O)CCN(C(C2CN3CCC2CC3)=O)CC1(F)F N1(C(C)=O)CCCCC1CC(=O)NCC(O)CNC(c1cc(C)c(Br)o1)=O c1(OC)ccc(C(=O)NC2CCCN(C(=O)Cc3ccc(C)s3)C2C)cc1F CC1(C(=O)NCC2CC2C(N2CCC2CC2CCCC2)=O)CC(=O)C1 CC(CC(F)F)C(=O)NNC(=O)C(C)(C)CCCCNC(C1(C)CC(F)(F)C1)=O c1(N(C)C)ccncc1C(=O)NCCCNC(c1ccnn1CC(F)F)=O CCCCCC(CCCCC)C(=O)N1CCC(NC(=O)CO)C(C)C1 C1(NC(C2C(CC)N(C(=O)CNC=O)CC2)=O)CCCC2(CC1)CC2 c1(NC(C)=O)ccc(Cl)c(C(N2CCCC(NC(C3CCOC3C)=O)C2)=O)c1 C1(CNC(CC2(OC)CN(C(C3CCCCC3O)=O)C2)=O)CC12CC2(F)F C1(NC(c2coc(C(=O)NCC(CO)SC)n2)=O)(CO)CCSC1 c1(NCC(C(C)C)OCC)nccc(=NCCOCCNC(C)C)[nH]1 C1(CNC(COC2CC(NC(c3c(C)ncnc3)=O)C2)=O)CCOCC12CCC2 C1(NC(c2c(OC)cccn2)=O)CC2CN(c3ncc(I)cn3)CC2C1 C1(C(=O)NCC(=C)CCNC(=O)Cn2cnc(Br)n2)COCCOC1 c1(C(=O)NCC2=CCN(C(C(F)=CCC)=O)CC2)cc(C)c(C)c(Br)c1 C(CCN(C)C(c1cnc(SC)s1)=O)(C(C)(C)C)NC(C(CC)=CC)=O C1(C(=O)NC(CCOC)C)(NC(c2nccc(C)c2N)=O)CCC(C)(C)C1 C=CC(CCC)CC(=O)NC1CCC(NC(c2ncc(F)cc2C)=O)CC1 CC(CNC(=O)CC1CCC(NC(c2nnsc2N)=O)C1)C(C)(F)F C(c1ccc(C)cn1)=CC(N1CC(OC)C(NC(=O)C2=C(Cl)CC2)C1)=O N1(C(CCCCc2ccc(C)cc2)=O)CCCC(NC(c2ccnnc2)=O)C1C c1(C(=O)NCCNC(c2c(C)coc2)=O)ccc(OCC(F)F)nc1 Cc1nn2cc(C(N3CCCN(C(C4CN(C)CCO4)=O)CC3CO)=O)nc2s1 N1(C(Cn2nnc(C)n2)=O)CC(C2CCCN(C(=O)Cc3nc(C)c(C)o3)C2)C1 c1(C(=O)NCCCN2C(=O)CNC2=O)cc2c(=O)[nH]ccn2n1 c1(OC(C)C(N2CCN(C(C3NC(=O)CC3C)=O)CC2)=O)ccc(C(N)=O)cc1 c1cc(O)c(F)c(F)c1.c1(OC)cc(NC(C2CC(F)(F)CN2C)=O)ccc1C N1(C(C(COC)Cl)=O)CC=CC(NC(c2cc(C)[nH]n2)=O)C1 CC1CC(NC(C2(c3ccno3)CCC2)=O)CN(C(=O)CCCC(F)F)C1 N1(C(C=C=C(C)C)=O)CCC(C)(CNC(c2ccns2)=O)CC1 c1(C(=O)NC(CCCC)CNC(=O)Cc2cc(C)on2)cnn2c(C)cccc12 N1(C(C2(CC=C)CCC2)=O)CC2(C)CC1(C(=O)Nc1ccc(CC)nc1C)C2 C1(C(N2C(CC(C)C)CCCC2)=O)CC2CN(C(=O)C#CC3(C)COC3)CC2C1 OCC(CN=c1cc[nH]cc1S(=O)(=O)NCC1=CCCOC1)c1ccccc1 Cn1cc(C(=O)NC2CCC2)c(C(F)F)n1.C1(C2CCCO2)(C=O)CCC1.C c1(OC)ccc(Br)cc1CC(N1CC(O)(CCNC(C2(C)CC2)=O)C1)=O c1(C(C(=O)N(C2CN(C(CC(C)OC)=O)C2)C)O)ccc(F)cc1 Cn1c([N+](=O)[O-])cnc1C(N1CC(CNC(=O)COC2CCC2)C1)=O C1(C(N2CCCC2CF)=O)(NC(c2cc[nH]c2)=O)CC(O)C1 CC1(CCCNc2ncc(Br)cc2C(F)(F)C(F)(F)F)NC(=O)NC1=O C(C1=NOC2CCCC12)NC(C1C(NC(C2CC3CCCC3C2)=O)CC1)=O C=C=CC(C)C(=O)NC(C)(C)CCNC(C1CCCCC1C(N)=O)=O CCCCCC(O)CC(=O)NC1(CO)CCCN(C(C2CC3(CCCO3)C2)=O)C1 CN=c1[nH]c(=NCCc2ccc(N3CC(OC)C3)cc2)[nH]c(=NCCCC#N)[nH]1 C(C(C(C)C)NC(=O)CC1CC(OC)C1)(c1ccccc1)NC(CCCC)=O CC1CC(C(=O)NCCC(C)(C)CNC(C23COCC2C3)=O)CN1C C(=O)(C(CCC)CC(C)C)N1CCC(C(N2CCOCC(CC)C2)=O)CC1 c1(CNC(C2C(CNC(CCCOC)=O)OCC2)=O)cc(C)ccc1F c1(C(N2CCN(C(=O)CN3CCCCS3(=O)=O)C3CC23)=O)cncc([N+](=O)[O-])c1 c1(NCC2CC(C)C2)[nH]c(=NCC2CCC(C)(C)CO2)nc2c1ncn2C(C)C N1(C(C(Cc2c(Cl)ccc(SC)c2)N)=O)CC(C)(C)OC2(CCOC2)C1 C1(CC)CC(CC(N2CC(NC(=O)CCn3cncn3)C(C)C2)=O)CCO1 CCCS(=O)(=O)C(C)C(=O)N(C)CCNC(=O)C1=CCCC1 CC1CCC(NC(c2ccc[n+]([O-])c2)=O)CN1C(=O)Cc1csc(Br)c1 c1(C(CNC(c2nnsc2C(F)F)=O)NC(C(C)O)=O)ccccc1F c1(C=O)cccc(S(=O)(=O)CF)c1.C1(F)CCC1.CC1CCN1CC(=O)NC S(=O)(=O)(c1ccc(C(N2CCC(C)(NC(c3ncccc3C)=O)CC2)=O)o1)NC CN1CC(NC(=O)C(CCF)NC=O)CC1C(=O)O.C(C)(C)(C)O Cc1ccc(Cl)c(C(=O)NCC2(F)CCC(C)CC2)c1.C(=O)(C1=CCCC1)N C(=O)C(C)CCC(C)(C)C.Cc1n[nH]c(C)c1C=CC(=O)NC1CC(O)(C)C1 N(C1CC2(CN(C(=O)C(C)=C(C)C)C2)n2ccnc21)C(C1(CC)CCNC1=O)=O N1(C(C2N(C(c3c(Br)c(C)n(C)n3)=O)CCCC2)=O)Cc2cccc(O)c2C1 c1(CNCCC(C)S(C)(=O)=O)ccc2ccccc2n1 N1(CCNC(CC2N(C(CCn3ccc(C)n3)=O)CCC2)=O)CCCCC1=O c1(C(=O)NCCCN(C(=O)C=CBr)C2CC2)cc2c(F)cc(F)cc2o1 c1(CNC(c2cn(C3CCOC3)cn2)=O)cc(Cl)ccn1 Cc1cccc(C(=O)NC2C3CC4C2C4C3C(=O)NC(C2CSC2)C)c1C#N Cc1cc(OCC(=O)NC(CN(C)C(=O)C2CC2)Cc2ccccc2)ccc1F C1(CNC(c2c(CC)nccn2)=O)CCCCCN1C(=O)C=Cc1ccncc1 C1(Nc2nccc(-n3ccc(C)n3)n2)C2CCN(CC2)C1C C=CCC(C)(C(F)F)NC(C12CC(CN(C(=O)CN3CCNC(=O)C3)C1)C2)=O C(=O)(CC(CNC(C1(COC)COC1)=O)C1CCC1)NC(CCC)C CCC(CC(=O)N1C2CCC1CN(C(=O)C(C)(C)CO)C2)C(C)C c1(C(N2CCCC(C)(O)CC2)C(=O)NCCC)ccc2c(c1)OCC2(C)C CS(=O)(=O)C1CN(C(=O)CC2C3CCCC3N2C(=O)C(O)CN2CCCC2)C1 C(=O)(C1Cc2ccccc21)N1CCN(C(c2c(C)nn[nH]2)=O)CC(C)C1 c1(CC)cc(C(=O)NCC(C)N(C)C(C2C3CC(F)(F)CC23)=O)cc(N)c1 Cc1nn(C)c(Cl)c1CC(N1CCC(CNC(C2CC3C=CC2O3)=O)C1)=O C1(CNC(C2CC(OC)C2)=O)(NC(=O)CCCCF)CCC(C)(C)CC1 N1(C(C2CC(C)(O)C2)=O)CC2CC1C2NC(=O)CC.c1(CC=O)ccccc1 c1(C(=O)NCC(C(C)(C)C)NC(=O)C(O)c2ccsc2)cnc2ccnn2c1N Cc1ccc(F)c(C(=O)NC2CC(=O)N(Cc3ccccc3)C2)n1 C(C(=O)N1CCCN(Cc2ccc(F)cc2)CC1)(C(C)(C)C)N(C)C C1(C(=O)OCC)CCCN(CC(N2CCC(OCC)C2)=O)C1 c1(C(=O)OCC2OCCN(C(C(C)SCC)=O)C2)cccc(C2CC2)c1.O n1(CCCC)nc(C)c(C(=O)NCC2CCCN(C(c3cc(F)c[nH]3)=O)C2)c1Cl c1(C(=O)NC2C(C)(C)CN(C(C3CC4(CCC4)C3)=O)C2)nc2ccccn2n1 C1(C)(C(=O)NC2CC3CN(C(CC(CC)CC)=O)C2C3)COC(C)(C)CO1 CC(C)CC(C)C(=O)NC1C2CCC1N(C(=O)CCCc1cccc(Br)c1)C2 CCC(CC(=O)N1CCC(OC2(CC(=O)N(C3CCCC3)C)CC2)CC1)C1CC1 CCCCS(=O)(=O)NCC(=O)NC1(CNC(=O)CC2C=CCC2)CC1 C(=O)(C(C)CCN(C)C)NCC(CN(C(C(c1ccccc1)OC)=O)C)C C1(C)(C(N(C)Cc2cccc(C)c2)=O)CN(C(=O)CC(C)(C)C#N)CC1C c12ccc(cc1)c(=O)n2CC.c1(CN(CC(CC)O)C)ncc(C)o1 c1(C(=O)NC2(CCNC(c3ccncc3)=O)CC2)cccc(C2CCOC2)c1 C=CCC(C)(O)C(=O)N(CCCCCC(=O)NC1CC(CC(=O)OC)C1)C c1(OC)ccc(C)c(C(=O)NC2CCC(CC)C2)n1.C(=O)C(C)=C1CCCC1 c1(CC)cc(C(N2CCCC2)=O)nn1C.c1(C(NC)=O)n[nH]cc1C(F)(F)F.C C1(C)(C(C)C)CCN1C(=O)COC1CCN(C(=O)CCN(C)C)C1 C1(NC(CC(=C)C)=O)CC2CC(C1)N(C(c1cccc3cnsc13)=O)C2 N1(C(CCOCCC)=O)CC2CCC1CN2C(c1cccc(CO)n1)=O CC(CC(=O)NCCCNC(C1(C)CC1C)=O)N(C)C N1(C(=O)C#CC2CC2)CC2(CCN(C(c3cnn4ccc(O)nc34)=O)CC2)C1 c1(OC)ccc(Cl)cc1C(=O)NCC1CN(C(C2(F)CCCN(C)C2)=O)C1 c1(C(N(C2CCC(NC(c3ccsn3)=O)C2)C)=O)n[nH]cc1F C1(OC)CCCN(C(=O)CCN(C)C(c2cc(C)n(C)c2C)=O)C1C C1(C(=O)OC)CC(C(=O)O)CN(C(=O)CCCC(=O)c2ccc(OC)c(F)c2)C1 Cc1cc(C(=O)NC2CC3C(NC(=O)CN4CCOCC4)C3C2)cc2c1CCC2 CC1CC=C(C(=O)N2CCC(F)(C(=O)NC3CCCOC3)CC2)CC1 c1(C2C(C=O)C2)ccc(F)cc1.O=C1CCC(C(=O)NCCC2CCC2)N1.N CCC(CNC(C1(OC)CCC1)=O)CC.C12(C(=O)N)CC(C(C)C)(C1)C2 C(=O)(C1=CS(=O)CCC1)NC1(CNC(CC2CN(C)CC2O)=O)CC1 C1(NC(Cc2c(C)cccc2)=O)(CO)CCN(C(=O)CN(C)CCO)CC1 C1(C2CCCO2)(C(=O)NC(CNC(CSc2nc(C)[nH]n2)=O)C)CCOCC1 c1(C(N)=O)cnc(COc2ccccc2OCCSC2CCCC2)cn1 c12ccc-1cc2.Cc1cc(-c2nnc(-n3nnc(-c4ccccc4)n3)o2)on1 c1(OC)ccc(C(N2CCCC(C#N)C2)=O)c(OC(C)CC)c1 N1(C(CN2CCN(C(C3=CC(C)(CC)C3)=O)CC2)=O)CC(OC)CC12CCC2 c1(NCCCCOCCOCC)cc(=NCc2ncoc2C2CCC2)[nH]cn1 c1(OCCOC2CCN(c3ncc(C)c(C)n3)C2)ccc2nccn2c1 N1(c2nnc(-c3c(C)nccn3)n2CCC(=O)N(C)C)C(CO)CC2COCC12 N1(C(C(CC)C)=O)CC(C2CCCN(C(c3cc(Br)nn3C)=O)C2)C1 Cc1cc(C)c(C(=O)NCC2(CN(C)C(C3CC3(F)Cl)=O)CC2)s1 N1(C(C(C)(C)NC(=O)OC)=O)CCCC(F)C1.c1(CC(=O)N)cccnc1Cl C1(CC)CCN(C(=O)Cc2ncn(C)c2C)C1C(=O)N(CCC(C)(C)C)C Cc1ncnc(O)c1CCC(=O)NC1CCCN(C(c2cnn(C)n2)=O)C1C CC1CC(C(=O)NCC2(C)CCN(C(=O)C(O)Cc3cnc[nH]3)C2)CCN1C C12(C(=O)NCCn3ncc(C)c3)CCC(CN(C(C3CC4(CCC4)C3)=O)C1)C2 C1(O)(CC)CCN(N2CC(c3ccc(OC)cc3)C2)CC1 c1(C(N2CCN(C(C(CCSC)O)=O)C(C)CC2)=O)c(C)[nH]c2ccc(Cl)cc12 N1(CC(=O)NC(COC)CO)CCN(C(=O)C=Cc2ccc(C)o2)CC1 C1(NC(C=CC(C)(C)C)=O)CCN(C(c2ccc3ocnc3c2)=O)CCC1CO CCCC(C)CC(=O)N1CCN(C(=O)C2=NNC(=O)C2)C(C(F)F)C1 C1(C(F)(F)F)(COC(=O)Cn2ccnn2)CC2CCC1CC2 Cc1nc2cc(C(=O)NC3CC(C)CC3O)ccc2s1.C(=O)(C(C)CN(C)C)N n1(CC)ccc2nc(N(C3CNCC3(F)F)Cc3cc(F)cc(Cl)c3O)ncc12 C1(NC(c2c(OCC)nccc2)=O)CCCCN(C(=O)C(F)CC(C)C)C1 CCC(C)C(C)N=c1[nH]c(=NCCc2ccccc2OC(C)C)c2sccc2[nH]1 c1(OCCOC)cncc(C(=O)N(CC(C)(C)NC(C2SCCC2C)=O)C)c1 C1(CNC(=O)CCn2cncn2)CCCCC1NC(=O)CC1CC1 C1(C)(NC(c2ccnc(N3CCCCC3)c2)c2n(C)nnn2)CC2(CCC2)C1 O=C(C#CC1CCCC1)NCCCNC(c1cc(Br)cnc1S)=O Cc1ccc2c(c1)CN(N(C)C(C(C)C)c1ccccc1)CC2 Cc1cc(C(N2CCOC(C)(CNC(=O)C=CC3CCCN3C)C2)=O)nc(O)c1 N1(C(C)=O)CC(O)CC1C(=O)NCC1CC(F)C1.c1(C=O)[nH]c(C)cc1C c1(C(C)C)cc(NC(c2c(C(F)(F)F)nn(C)c2Cl)=O)ccc1O C(C(CNC(C1CN(C(N)=O)C1)=O)C(F)(F)F)NC(CC1C(C)C1)=O N1(C(Cc2cc(C)ncc2)=O)CC(C)(C)CCC1CNC(=O)CS.CC(N)=O N1(C(c2c(C)ccs2)=O)CCCCC(NC(=O)C(C)(C)C2CCCC2)C1 N1(C(c2c(CC)cns2)=O)CCC(O)(C)CC1.C(=O)(C(C)CC1CCCCC1)N N1(C(c2ccc(C)o2)=O)CCC(C=CC(=O)NCC(F)Cl)CC1 C1CC2(C1)CN(C(=O)CC)C2.[SH](=O)(=O)C(F)(F)F.C1CC12CC(O)C2.O=C CC1CN2CCN1CC2C(N1CCCC1CN(C)C(C1CCCCNC1=O)=O)=O Cc1cc(S(N)(=O)=O)oc1C(=O)NC1CCCN(C(=O)C#CC(C)C)C1C N1(C(C)=O)c2ccccc2CC1C(N1CCCC(NC(c2cn(C)cn2)=O)C1)=O C1CN(C(=O)CN2CC=CC2)C2CC12.c1(C(=O)OC)sccc1C(=O)N.C c1(C(N2CCN(C(CNC(CC(C)C)=O)=O)CC2)=O)cc(F)c(F)c(N)c1Cl N1(C(C(C)C2CCC2)=O)CC2(CC(NC(c3cccc(N4CCCC4)n3)=O)C2)C1 CC1CC(=O)NCC1C(N1CC(C)(NC(c2nc(Cl)c(Cl)s2)=O)C1)=O CC(C)(C)C(O)C(=O)N1CCC(O)CC1C(=O)NC1(C#N)CCOCC1 C1(NS(CC)(=O)=O)(C)CN(C(=O)C(c2cccnc2)(C)C)C1.C(=O)(C)N N1(C(c2cnc(C)n2C)=O)CCCC(C2(NC(=O)Cn3ccccc3=O)CC2)C1 Cc1nn(CC(F)F)cc1Cc1nc(-c2ccco2)nn1-c1cccc(F)c1 Cc1cc(C2CCC2)ncc1C(=O)NC(C)(C)C(C)C.C1(C(=O)N)CCCCS1 n1(CC)nc(Oc2ccc(Cl)cc2)nc1-c1cnc(-c2ccccc2)o1 N1(CC(=O)N(C2CC2)Cc2c(C)nsc2)CCN(c2ccccn2)CC1 c1(CC(=O)NCC(CCCC)NC(=O)C#CC(C)C)ccc(C#N)cc1 C1(C(N(CC)C2CC2)=O)CC(S(C)(=O)=O)C1.C(C=O)C(C)C.CCO c1(C(N2C3CN(C(C45C(C)(C)OCC4C5)=O)CC2C3)=O)ccc2c(c1)CCC=C2 Cn1ncc(CNC(C2CCC(F)CC2)=O)c1C(=O)N.O(C(F)(F)F)CCC C=CCC(C)(C)C(=O)N1CC2CC1CC2NC(=O)Cc1c(C)nn(C)c1C Cc1oc(CO)cc1C(N1CC2(NC(c3ccccc3CC#N)=O)CC1C2)=O CCC(C)C(O)C(=O)N(CCNC(=O)C(c1cccs1)SC)CC Cn1cc(C(=O)NCC2CC2)ncc1=O.N1(CCC2(C=O)CC2)CCCCC1 N1(C(c2cc(Cl)ncc2O)=O)CC2CN(C(c3ccc(O)nc3Cl)=O)CC2C1 C(=O)(CCC(=O)NC(C)(C)CC(=O)NC(C)(C)CCCOC)NCC CCCCC(CC)C(=O)N1CC(CC(N2CC(C)(F)C2)=O)CC1(C)C N1(C(c2c(CC)n(C)nn2)=O)CCC(C)(NC(C2CN(c3nncs3)C2)=O)CC1 C=C(C)C(CC(=O)NCC(C(=O)NC(CCO)C(C)(C)C)N(C)C)OCC N1(C(CNC(=O)OC)=O)CC(NC(=O)C(C)C(F)F)CC12CCC2 C1(NC(COC(CC)C)=O)CN(C(C2(CCOC)CCC2)=O)CC1OC N1(CC)CCC=C(c2nc3c(s2)COC(C(N2CC4C(C2)C4(F)F)=O)C3)C1 Cc1nn(C)cc1CC(=O)NC1CCN(C(c2ccc(Br)cc2)=O)CC1 n1(CCOC)ccc(=NC(=O)C2(C)CN(C(c3ccnnc3C)=O)C(C)(C)C2)[nH]1 c1(C(=O)NC2CC(NC(CC(CC)OC)=O)C2)c(C)nn(C)c1Br C(CC(C(C)(C)C)NC(c1ccncn1)=O)N(C(C1CC(C)(CC)C1)=O)C Cc1ncc(Br)cc1NC(=O)C(=O)NCC1(C)CC1Br c1(C(=O)NC2CC(CCNC(C3(C)CCCCO3)=O)C2)ccccc1C#N C(=O)(C1=CCC(NC(c2cc(C(C)=O)c[nH]2)=O)C1)N(CC#CC)C c1(C(C)=O)ccnc(COC(C)(C)C)c1.c12cc(c[nH]1)COC2=O C(C(=O)NOCC1CCOC1)(C1(C)CC1)NC(=O)CC(Cl)Cl c1(OC)ccc(C(C)NC(c2cccc(CCN)c2)=O)cn1 N1(C(c2n(CCC)ccc2)=O)CCC2(CC1)CC(NC(c1cnnn1C)=O)CO2 c1(C(=O)NC(CC)CNC(c2cnc(SC)s2)=O)ncn2c1COCC2 C1(C(=O)NC2(CC=C)CN(C(=O)C(C)(C)F)C2)CCCCC12CC2 C1(C(N2CCC2c2ccccc2)=O)CN(CC=Cc2ncc[nH]2)CC(F)(F)C1 C=CC1(O)CCN(C(=O)C(CNC(c2ccnn2C(C)C)=O)C(C)C)C1 c1(C(=O)CN2CCN(C(=O)COCC3CCC3)CC2)cccc2c1OCCO2 CN1CC(NC(=O)C(F)CC2CN(C(=O)CC3OCCO3)C2)C(F)(F)C1 Cc1cc(C(N2CCC(C)(NC(=O)C3=CCOC3)C2)=O)nn1C(F)F C(=O)(CC1=NN(C)C(=O)C1)N1C(C)CN(C(c2ccc3c(c2)COC3)=O)CC1 n12c(nnc1C(=O)NC(c1ccc(F)cc1)CF)N(C)CC2.C(C)(C)S.CO C12(CC(=O)N)CC3CC(CC(C3)C1)C2.CCCN(C(=O)C=CC1CC1)C c1(C(N2CC(SC)C(NC(C3CC34CC(F)(F)C4)=O)C2)=O)c[nH]c2ncccc12 C(CN=c1cc(-c2ccccn2)nc(Cl)[nH]1)NC(c1c(CC)scn1)=O C1(CCNC(C2C(C=C)C2)=O)CN(C(c2ncc[nH]c2=O)=O)CCCO1 CC1=NN(C)C(=O)C1CC=O.C1CCN(C(=O)CN2CC(C)(C)C2)C12CC2.N C1(c2cn(CCOC)nn2)N(C(=O)CN2CC=CC2)CC12CCOCC2 N1(C(=O)Cn2cc(Cl)cn2)CCCC1C1CCCN1C(c1ncccc1O)=O n1(C(CO)C2CCC2)cnc2c(N3CC4CCC3C4)ncnc12 C1(Nc2ncc(C(N3C(c4onc(C)n4)CCCC3)=O)s2)CC1C1CCCC1 c1(NC(C2(F)CCN(C(C(C)n3cccn3)=O)C2)=O)cnc2ccnn2c1 C1(NC(C(C=C)O)=O)C2CC3C1C3C2C(=O)NCc1ccc(CC)cc1 CN1CCOCC1CC(N1CCCC1C)=O.c1(C=O)[nH]c(=N)sc1C(F)(F)F.N c1(C(N2C(CNC(C3CN(c4ccncc4)C3)=O)CC2)=O)ccc[n+]([O-])c1 Cc1ncc(C(N2CCC(O)(C(C)CNC(=O)C(C)(C)F)C2)=O)c(C)n1 C1(C(N(CCCCN(C(c2c(C)ocn2)=O)C)C)=O)C2CCC1(c1cscn1)C2 C1(C(N(CCNC(c2cccc(C(C)C)c2)=O)C)=O)CC2CC1CC2(F)F N1(C(c2c(C)snc2)=O)CCC(C)N(c2ncc(C#N)cc2Cl)CC1 c1(C(N2CC(C)(CNC(c3cccnn3)=O)OCC2)=O)cnc(P(C)(C)=O)cn1 N1(C(c2ccn(C)n2)=O)CC(NC(=O)Cc2nc(C3CC3)cs2)CC2(CCC2)C1 N1(C(c2c(OC(C)C)cccc2)=O)CCC2CCC(C1)N2Cc1cccc(Br)c1 N1(C(C2=NNC(=O)C2)=O)C2CCCC1CC(NC(=O)CSC1CCOC1=O)C2 n1(CC)cc(C(N2CC3(NC(c4cc(Cl)no4)=O)CC2C3)=O)c(C(C)C)n1 Cn1c(C(=O)NC2CCC(CCNC(C3(CF)CCOCC3)=O)C2)nnc1S Cc1ccc(CC(=O)NCC2CC2C)c(C)c1.c1(C(=O)N)ccc(O)nc1C n1(CC)nncc1CN(C(=O)C(=O)N(C1CCSC1)C)C c1(CC(=O)NC2CCCCCC2NC(C2(CO)CC2)=O)ccc(F)c(F)c1 N1(C(CC2(C)CCOCC2)=O)CCC(C2CN(C(C3C=CCCC3)=O)C2)CC1 N1(C(C2CC(=C)C2)=O)CCCC(C2CN(C(c3cn(C)c(C)n3)=O)C2)C1 C=C(C)CCC(=O)NCC(CNC(c1cccc(-c2csc(C)n2)c1)=O)CO c1(NC(c2nc(CC)[nH]n2)C)ncnc(NC)c1C.c12cccc(n1)SC1CC21 Cc1ccc(C(N)=O)cc1C(=O)NCC(CNC(c1c(C)ncn1C)=O)CO c1(C(N2CCN(C(=O)C3CC3)C3(CC3)C2)=O)cnc(O)c2ncccc12 C1(CC(=O)OC)(C(=O)N(CC(F)(F)CO)C)CCCCC1 CC1CCC(CNC(c2nnnn2C2(C)CC2)C2CCC2)CC1.OC N1(C(c2ccccc2Cl)C)CC=C(CCNC(=O)C(F)CC2CCCCC2)CC1 C1(NC(CCCC#C)=O)CCN(C(C2CC2c2ccoc2C)=O)C12CC2 C(=O)(C1=CCCSC1)N(C1CCN(C(c2ccnn2CCC)=O)CC1)CC#C N1(C(C(C)OCC(C)C)=O)CC2CCCC(N(C(=O)CC3CCCC3C)C)C2C1 N1(C(C(c2c(C)n[nH]c2C)C)=O)CC2(CCC2)C1.N(C)(S(N)(=O)=O)CC=O C(=O)(C(C)(F)C(=O)OC)N1C2C(NC(c3c(CC)occ3)=O)C(C2)C1 CC(C)C(C(=O)N(CCCNC(=O)COCCO)C(C)C)N1CCCC1 C1(NC(c2ccncc2)=O)CCCC(NC(C2CC3(C2)CC3F)=O)C1.C1CC1 C1CCc2nncn2C1.C(C1CCCC1)=CC(=O)NCC(=O)NCC=O.CC=C.N C1(CN(c2ccc(C(C)(C)C)s2)CC)CCN(C2CCCc3ccccc32)CC1 C=C(C)CCCC(=O)NC1CCOCC1NC(C1CC(=O)N(O)C1)=O c1(C2CCN(C(c3cc(Cl)cs3)C(=O)NC3CC3)C2)ccc(F)cc1 N1(C(CN(C)C)=O)CCC(C(=O)NCc2cc[nH]n2)C2OCCC12 Cc1cc(C(N2CCC(NC(=O)C(c3ccccc3)F)C2(C)C)=O)cnc1O CC(O)CC(=O)N1CCCC1CCC(=O)NCC(C)(C)C#N C1(CNC(Cn2ccc(C)n2)=O)(NC(=O)C(C)(C)c2nccs2)CCCCC1C c1(-c2ccc(OC)c(OC)c2)csc(=Nc2cccc(O)c2)n1C1CCSC1C c1(CC(N2CCC(O)(CC)C2)=O)c(F)cccc1Cl.c1(CC)ccc(C(=O)N)s1 C1(C(N(CC(C)(C)CO)C)=O)CN(C(=O)C2=CCOCC2)CC1(C)C CC(C)C(CNC(=O)CC1(O)CCC1)C(=O)N=c1ccn(CCCO)[nH]1 C1(C#N)(OCC)CN(C(C2CCCC2NC(C2CC(=O)C2(C)C)=O)=O)C1 C1(C(N2CCC(F)C2)=O)CCCC12CCC2.C1(C(=O)NC)(NC(N)=O)CC1 Cc1ccccc1C=CC(N1CCCC(CCNC(=O)CC2CC3(CC3)C2)C1)=O CC1(C)C2CCC(C2)C1C(=O)NCC1C2CCCCC12 Cc1ccsc1CC(N1CCCC1C1(O)CN(C(C2CCSC2)=O)C1)=O C(C(CC(=O)NCC(F)Cl)OC)NC(C1(CC)COC1)=O c1(NC(C(COC)NC(=O)C(C2CC2)C2CC2)=O)cnc(Cl)nc1C c1(C(=O)Nc2cn(C)c(S(=O)(=O)N3CCOCC3)c2)cccc2ccc(Br)nc12 C1(C(N(C(CC)CO)CC)=O)CCN(C(=O)CCC2CCCC2)C1 C=CC(CC)CC(=O)N1CC(N(C)C(c2cc(Cl)cn2C)=O)C2(CC2)C1 C1(NC(c2ccc(C#N)[nH]2)=O)CCCN(C(=O)CC2CC(CF)C2)CC1 C1(C(N2CC(CNC(CCCOC)=O)C2)=O)OCC2CCCC12 C1(C(=O)NCCSCC(C)C)CNC(=O)CN1C(=O)CCc1ncccn1 C1(CNC(CCN(C(C(C)NC(CC)=O)=O)CCO)=O)CCC(O)CC1 C(=O)(C(C)CC(N)=O)NCCC1(NC(CCC2CC(C)C2)=O)CCC1 c1(CNCC23C(CN(C(c4cc(Cl)cnc4O)=O)C2)C3)ccc2occc2c1 c1(C(N2C(C)CC(NC(=O)C(=O)N=S(C)(C)=O)C2)=O)cc2cnc(Cl)cc2s1 Cc1ccc(SCCO)c(O)n1.c1(-c2nnn(C3CCCCC3)n2)cc(O)ncc1F N1(C(C(=O)NCC(C)C)C2CCOC2)CCOC(CC(C)C)C1 C(CC(N)=O)(C(=O)NCC12CCN(CC1)CC2)NC(c1ccc(C)[nH]1)=O c1(C(=O)OC(CC)COC)cc(C)cc(Cl)c1Br C1(N(C(=O)Cc2ccnn2C)CC)CCCN(C(c2ccc(CO)nc2)=O)CC1 c1(C(=O)NC(C)CCCCNC(c2nn(C)cc2Cl)=O)ccc2nccnc2n1 c1(NC(C=COCCOCCOC)=O)ccc(OC)cc1C c1(CCC(N2C(CNC(C3C(C)CC3)=O)CCC2)=O)ccc(O)nn1 N1(CC(=O)NC2CCCN(C(CCC=CC)=O)C2)CCCCS1(=O)=O CC1CC(C)CN1C(=O)C=Cc1ccncc1.c1(C2(C(=O)N)CC2)ccccn1 Cc1nn(C)c2cc(NC(C3CC(NC(c4cn5cccnc5n4)=O)C3)=O)ccc12 N1(C(C(C)N(C)C)=O)CCc2nc[nH]c2C12CCN(C(C1CCOC(C)C1)=O)C2 C(=O)(CCC(C)C)NCC1(COC)CN(C(=O)CN2CCOCC2)C1 c1(CC(=O)NC(C)CC(C)NC(c2ccc(N)c(F)c2)=O)c[nH]c2ccccc12 CC1(C)OCCC1C(=O)NCCCN1CCN(C(C2CC(N(C)C)C2)=O)CC1 N1(C(c2cccc(SC)n2)=O)CC2CC1CCC2NC(c1n[nH]c(O)n1)=O C1(C(=O)NCc2ccccc2)CCCN(C(c2[nH]cnc2-c2ccccc2)=O)C1 C(=O)(CC1C(=O)Nc2ccc(C)cc21)N(C(CCNC(CC1(C=C)CC1)=O)C)C N1(C(CC=C(C)C)=O)CCN(C(C2CCCN2c2cnccn2)=O)CC(C)(F)C1 C#CCCCC(=O)NC1(CCNC(=O)C(C)(C)Cc2ccccc2)CCCC1 C(=O)(CC(F)(F)Cl)NC(CN(C(C1CCC(CC)O1)=O)C)C Cc1cccc(C(N2CC(NC(c3ccnc(C4CC4)n3)=O)C(O)C2)=O)n1 C1(CNC(CN(C)CCO)=O)CN(C(=O)C(C2CC(F)(F)C2)O)CCCO1 CC(C)CCCC(=O)N1CCCC1C1CCN(C(=O)CC(O)CN(C)C)CC1 C1(C(C)C)C(NC(c2cccn2C)=O)CCN1C(c1cccc(C(F)F)n1)=O c1(NC(c2c(NC(c3c(OC)ccs3)=O)ccs2)=O)cc(O)c(Cl)cc1F C1(CC(=O)N(C2CCC2)CCC2CCC2)CCC1O.n1(CC=O)cccn1 N1(C(C2CCN(C(CCCCOC)=O)C23CC3)=O)CC(=O)N(C)CC1C N1(c2ccc(-n3c(C)cc(C)n3)nn2)CCOc2c(C(C)(C)C)cccc21 CC1(C)Cc2cc(S(=O)(=O)NC3COC4(CCNCC4)C3)ccc2O1 c1(C(C)C(=O)NCC2(CCNC(c3ccn(C)n3)=O)CC2)cccc(Cl)c1 Cc1ccc2c(c1)CC(C(N1CCC(C(C)(C)NC(C3CCC(C)C3)=O)C1)=O)S2 N1(C(C(Cc2ccco2)NC(C(n2c(C)ncc2)C)=O)=O)CCC2(CSC2)C1 C1(CN(C(CN(C2CCC2)C)=O)C)CCn2cncc2C1.C12C3CN(CC13)C2=O C1(CC)CCN(C(=O)CC)C1.C1CN(C(N)=O)C1.C(=O)(C)N.C(C)(C)C C(=O)(CCC(F)(F)CN=[N+]=[N-])N1C(C)C(NC(c2cc(Cl)cn2C)=O)CCC1 N1(C(C2C(C)(NC(c3cc(C)sc3)=O)CCCC2)=O)CCc2nn(C)cc2C1 CCC(COC)C(=O)NCC(CCOC)NC(c1cccc(C)c1)=O C1(OC)CC(C)N(C(=O)Cn2nnnc2-c2ccsc2)C1.c1(C=O)cncs1.N Cc1ccc(COCC(N2CCOC(CNC(=O)C(C)C3CC3)C2)=O)cc1 N1(C(CN(C(C(C=C)C)=O)CCOC)=O)CCC(O)C(F)(F)C1 c1(CC)ccnc(C(=O)NCCCNC(c2cncc(C(C)=O)c2)=O)c1 C1(NC(C(c2ccoc2)N(C(C)CC2CC2)C)=O)CCC(F)(F)CC1 C1(C(NOCCC#C)=O)C2CC2CN1C(=O)CCn1cnnn1 C=C1CC(C=O)(CNC(=O)C=CC(=O)N)C1.C1CCCC1N(C)C Cc1occc1CNC(C1CCCC1C)=O.C1(C(C)CCO)(C=O)CCC1.N c1(C(N2C(C=O)CC(F)C2)=O)ccc(Br)c([N+](=O)[O-])c1.c1ccc(Cl)c(F)c1.N N1(c2nc(N3CCCOC(C)C3)cc(C)n2)Cc2ccncc2C1 c1(C(N2CC(C(C)NC(CCN(CCC)C)=O)C2)=O)coc(SC)n1 CCCCC(O)C(C)C(=O)NCCCCCCN(C)C(c1cscc1OC)=O N1(C(C(CCC)OC)C(=O)NCCCSC)CC2CC(C1)C2(C)C N#Cc1ccc(S(=O)(=O)NCC2CCSC2)cc1NC1CCC(CO)CC1 c1(NC(C2CCCCN2C(c2ccc(Cl)s2)=O)=O)c(-n2cccn2)ncnc1Cl C1(N(C(COCCCC)=O)C)CCC(NC(=O)Cc2csc(C)n2)CC1 c1(CC)nc(Cl)nc(NC(C)(C)C)c1Cl.c1(C(=O)N)nccnc1C(F)(F)F CC1(C)CCC(C(=O)NC2(C(N3CC4CCC3C4)=O)CC(O)C2)O1 Cc1cc(CCC(=O)NC2CN(C(=O)CC3CCCCCO3)C2)nn1C N1(C(C2CCN(CC)C2)=O)CCCC2(C1)CN(C(=O)CC1CNC(=O)C1)C2 C1(NC(c2ccc(COC)cc2)=O)CCC(C)N(C(c2c(C)n[nH]c2C)C)C1 c1(C(C)C)ccc(C(C(=O)OC)NC(CO)CCSc2ccc(Cl)s2)cn1 N1(C(CCCOC)=O)CCC2(NC(c3cc(C(N)=O)cc(F)c3)=O)CC2C1 c1(C(=O)OC)ccc(CCNC(C2CC2)=O)cc1F.c1(C(=O)N)cc[nH]c1 Cc1ccc2snc(C(=O)NC3CCCCC3CNC(=O)CC(O)C3CC3)c2c1 c1(NC(COC)CNC(=O)C(=O)NC2CC2)ccc(COC)s1 c1(CN2CCC(CC(=O)NC(CC)CO)C2)cc[n+]([O-])cc1 c1(C(=O)N)ccc2nnn(C(C)(C)C)c2c1.c1(C(=O)NCCCC)cn(C)cn1 N1(C(C(C(CC)C)NC(C)=O)=O)C2CCCC1CN(C(=O)C(C)(C)c1cnsc1)C2 C(=O)(CCC(C)(C)N(C)C)N.C(=O)(CCC(=O)NCC1COCC1)OCC c1(C(=O)NC(C)(C)CNC(=O)COC(F)(F)F)ccc2occc2n1 c1(C(N2C(C(C)NC(COC)=O)CCCC2)=O)cccc2c1COC2 C1(NC(c2n(CCCSC)nnn2)c2conc2C)COC2CCCCC12 C(=O)CC(C)C(F)(F)C(F)(F)F.c1(COC)nc(C(N2CCC2C)=O)co1 CC12CN(C(=O)COC3CCC3)C(C(=O)NC)(C1)C2.C1CCC(=O)NC1 N1(C(CCCOCC=C)=O)CCC2(CO)CN(C(=O)C3=COCC3)CC2C1 C(=O)(C1CCc2ccccc21)NC1CC(CNC(=O)CCc2cccc(Cl)c2)C1 C1(CN(C)C)CCCN1CC(=O)NC(C1CCOCC1)C1CC1 C(CC(C)C(C)C)NC(c1cccc(OCC)c1)=O.c1(CC=O)nonc1C.N C1(CC(N2CC(OCCNC(CC(CC)SC)=O)C2)=O)CCCC2CCCCC12 C1(N(C)C(C2CC(F)(F)C2)=O)CCCN(Cc2nccn2C)C1 N1(C(C(CNC(CSCC=C)=O)O)=O)CCC2(CC(CO)C2)C1 c1(CCC(N2CC3(C(NC(CC(C=C)C)=O)CC3)C2)=O)ccccc1[N+](=O)[O-] C1CCCCN(C(=O)CN(c2ccccc2)C)C1.C(=O)(CCC(=O)NC)NCC O=C(NNC(=O)C1OCCCO1)NCC1(c2ccc(Cl)cc2)CCCCC1 C(=O)(C(C)C(C)CO)N1CC(CNC(C2(C#C)CCCC2)=O)(OCC)C1 N1(C(c2nccc(N)c2)=O)CC2(C1)SCCC2NC(C1CC2(CC2)CO1)=O C(=O)(C#CC1CCOC1)N1CC(CC(C)NC(c2ocnc2C2CC2)=O)C1 C(C(=O)NCc1occc1C(=O)N(CC(C)(C)N(C)C)C)(C(C)C)OC c1(CN2C(CCC(=O)Nc3c(C#N)ccs3)CCC2)cccc(Cl)c1C(F)(F)F N1(C(C(C)=C(C)C)=O)CC(CNC(=O)C(F)(F)c2cncs2)C2(CC2)C1 C1(N(CC(C)C)C(C2(COCC)CC2)=O)CCN(C(c2cnn[nH]2)=O)C1 C1(NC(C2C(=C)C2)=O)CCN(CCNC(c2cn(C(C)C)cn2)=O)CC1 CC1(C)CCOC(C(=O)NC(Cc2ccoc2)C(=O)NCC#CCCO)C1 C1(CC(=O)NC)CCC2(CCC2)O1.C12CC1CN(C(=O)C=Cc1ncc[nH]1)C2 c1(N(C)C)cccc(CN2CCN(CC(=O)NC3CCC3)CC2)c1O C(C)(C)(CC(C)C)NC(C(C)NS(CC)(=O)=O)=O.c1ncnn1C.C(=O)C c1(C(=O)NCC2N(C(C3N(C=O)CCC3)=O)CCC2)cc(Cl)cc(F)c1F c1(C(=O)OC)c[nH]c(=NCc2ccc(C(C)C)nc2Cl)s1 C(N=c1[nH]c(N2CC3CCC(O)C3C2)nc2c1CSC2)C1CN(C2CC(C)C2)C1 CCCCCC(CC)C(=O)N1CCC(CNC(=O)C(CC(C)C)N(C)C)CC1 CN=c1[nH]c(=NCCC2CCCCCC2)[nH]c(=NC2CCCCC2C(N)=O)[nH]1 C(CN=c1[nH]c(=NCCC(N)=O)c2c(F)cccc2[nH]1)(CC(C)C)OCC N1(C(c2c(OC)ccc(F)c2)=O)CCOC2(C1)CN(Cc1ncc(Br)cc1C)C2 N1(C(C2CCC(CC)CC2)=O)CCCN(C(c2cnc(C(F)F)s2)=O)C(C)C1 N1(C(Cc2nc(C)oc2)=O)CCC2C1CCCN2C(=O)Cc1cc[nH]n1 N1(C(COc2cn(C)nc2)=O)CCC2CC2(C(=O)NCCc2cocn2)CC1 C(C(C)(C)C)N(C(c1cc(C(C)(C)C)n[nH]1)=O)CC.C(=O)CCC1CC1 c1(CC)cncc(C(=O)NC(C2CN(C(=O)CCc3cccc(C)c3)C2)C)c1 c1(OC)cc(C(=O)N)nn1C.C1(C2CC2)CCCN1C(=O)C(O)CN1CCCC1 N1(C(C(=O)NCC(CC)(C)c2ccncc2)=O)CCc2c(C(=O)OC)cccc21 C1(OCC)CN(C(=O)C(c2nc(C)cs2)C)CC1CNC(=O)C(C)C.O C1(NC(C2(OCC)CCOC2)=O)CC(NC(C2SCCS2)=O)C12CCC2 CCCCCCCCCCSCn1c(O)nc2ccccc12 N1(C(c2cc(C)c(C#N)cc2)=O)CCc2cc(O)ccc2C1C CC(=O)C(C)(C)CC(=O)N1CC(C)(C(=O)NCC2(O)CC3CCC2O3)C1 N1(C(CC=O)=O)CCCC(C)(C)C1.CC(C)CC.CC(C)C.C(=O)CC1CC1.O C1(C=O)CCCN(S(N)(=O)=O)C1.N1(C(c2ccc(CC)[nH]2)=O)CCC(C)(C)C1 c1(C(=O)NC(CNC(C(C(CC)C)O)=O)C)ccc([N+](=O)[O-])cc1O c1(CN2CC(C(=O)Nc3c(C#N)cccc3Cl)OCC2)c(Cl)[nH]c2ccccc12 C(CCCC(=O)N1CCC(C(F)CNC(=O)CCN2CCN(C)CC2)CC1)SC N1(C(c2cn(C(C)C)nc2)=O)CCC(C)C1C.n1(C2(CC=O)CC2)cccn1 C1(CNC(C2(CC)CCC2)=O)CN2CCCCC2CN1C(c1cnsc1)=O CC1CN(C(c2cc(F)cnc2O)=O)CCC1CNC(c1ccco1)=O c1(NC(C2CCN(C(c3c(OC)cccc3)=O)CC2O)=O)c(I)cccc1C#N N1(C(C2(C)CCCC2)=O)C2CCCC1CN(C(C1CC1c1ccc(Cl)cc1)=O)C2 c1(C=O)ccc(S(N)(=O)=O)o1.C1(CC)CCN(C(=O)C)CC1.[SH](C)(=O)=O C(c1ccc(C(F)(F)F)cc1)=CC=O.n1(CC)cc(C(N2CCC2)=O)cn1.C N1(C(CCCCCSC)=O)CCN(C(C2C(C)(C)C2(C)C)=O)CC(C)(F)C1 C(=O)(CC1=CCCCC1)NCC1CCCCN(C(c2c(OC)cccn2)=O)C1 N1(c2cn(C)nc2)CCC(O)(C(N2CCN(c3cnsn3)CC2)=O)CC1 C(=O)(C(C)(C)S(C)(=O)=O)N1CCCCC1.C1(C(=O)N)(CN(C)C)CC1.C C(CCN=C(NC1COC2CC1C2)N1CCC(COC(F)F)C1)OCC N1(C(=O)C=CBr)CCC2C(CCCN2C(=O)C(c2ccc(F)cc2)O)C1 c1(COCC)nc(C)c(C(=O)NCCC)s1.c1(CCC=O)nc(C)cs1 CC1CN(C(=O)NCc2cc[nH]c(=N)c2)c2cccc(F)c2O1 N1(C(C2CN(S(CC)(=O)=O)C2)=O)CC2(C1)CN(C(=O)C(C1CC1)O)CC2 N1(C(COc2c(C)cccc2Cl)=O)CCC(C)N(C(=O)Cc2ccccc2)CC1 Cc1cc(N)c(C(=O)N(C)CCN(C)C(C2CN(C)CC(C)O2)=O)nc1C c1(-c2ccc(C(=O)NCCCC=C)s2)ccc(C)c(C)c1.C1(C(=O)N)CC1C=C C1(C(=O)NC(c2nncn2C)C)COCC1NC(=O)CCCn1cccc1 C1(C(C(=O)NC(C)(C)C)N(CCCN(C(C)=O)C)C)CCC2CC1C2(C)C c1(C(=O)NCC(CCOC)NC(c2cnn(C)c2N)=O)ccc([N+](=O)[O-])o1 CC(C)(C)C(C(=O)N1CC=CC1CNC(c1ccc(F)s1)=O)N1CCNC1=O CCCN(OC)C(=O)C1CCCN(C(c2ccc(CC)c(F)c2)=O)C1 N1(C(CC)=O)CCC2(CC2C(=O)NCC(C)C(=O)OC)C1 C(=O)(CCC(C)(C)C)NCC(C(C)C)NC(c1nc(C(C)OC)sc1)=O Cc1ncc(C=CC(=O)Nc2ccc(OC(C)C)nc2C)c(O)n1 C1(N(C(CC2CCN(OC)CC2)=O)C)CC2CCC(C1)N2C(C1CC1(F)F)=O c1(N(C(C)C)C)ccccc1C(=O)NC1CCCN(C(=O)CC2CCOC2)C1 C1(C(=O)NCC2CN(C(C(=O)NCCOC)=O)C2)ON=C(C)C1C.C n1(CC(=O)NCCC(C)NC(=O)CCC(C)C(C)(C)C)cnc2c(N)ncnc12 C1(N(C(=O)CSC2CC2)C)CCC(C)CC1.C(=O)CCCN1CCOC1=O.N C#CC1(NC(=O)C(CC(C)(C)C)NC(=O)CCC(CC)OC)CCC(C)(C)C1 N1(C(CCCN(C)C)=O)C2CCC1C(CNC(=O)CC)C2.C1(C(=O)N)CCCO1 C(=O)(C1=C(Cl)CCOC1)NC1(CC(=O)NCC2(OC)CCOC2)CC1 c1(CC)ccc(C(=O)NC2CCN(C(=O)C(C)(O)CC)CC2F)cc1Br c1(NC(C2(C)N(C(C(CC)COC)=O)CC=C2)=O)ccc2ccccc2c1 Cc1cc(CC(N2CCCC2(C)CNC(C2CCCC2)=O)=O)cc(C)c1 N1(CCN(S(C)(=O)=O)C)CCS(=O)(=O)C(CC)C1.C1(CC=O)CCOC1 c1(OC)cc(C(c2nnnn2CCCF)NCC2(CC(N)=O)CC2)cc(F)c1 C1(C(=O)NC2(CNC(CC(c3cn(C)nc3)O)=O)CCC2)OCC2CCCC1C2 C#CCC(O)C(=O)N1CCCC1C=CC(=O)NC(C)(C)CCCOC C=CCCC(C)(C)C(=O)NC1CCCCN(C(c2cc(CC)on2)=O)C1 C=CCCN=C(NCC1C=CCCCC1)NC1CC1C(F)F c1(CC(=O)NCCN(C(c2cc(C#N)n(C)n2)=O)CC)cc(C)ccc1 C1(C=O)CCOC(C)(C)C1.c1(C(N(CC(C)(C)C)CC)=O)ncoc1C.N C(C(=O)N1CCCC(N(C)C(c2ccoc2Br)=O)CC1)(C(C)(C)C)NC(C)=O N1(C(C(C)N(c2cccc(S(C)=O)c2)c2ccccc2)=O)CCn2cnnc2C1 c1(C(=O)NCC)c(Cl)ccc(F)c1F.C1CCN(C(=O)C)C1.C1CC1(F)F.O c1(C(C(=O)NC(C2(O)CCC2)C)NC(C=CCC)=O)cn(C)nn1 C1(OC)CC(CNC(C2CC(C)(C)C2)=O)N(C(C2CCC(C)O2)=O)C1 C(=O)(C(C(=O)N(CCCCN(C)C(c1c[nH]nc1F)=O)C)OC)OCC Cc1sc(C(=O)N(CCC(C(C)C)NC(C2CC2(F)F)=O)C)cc1Br n1(CC(N2CC3C(CNC(c4cc(C)n(C)n4)=O)(C3)C2)=O)cc(F)ccc1=O c1(C(N(C)CC2COCCN2C(c2cnn3c2CCC3)=O)=O)cnc(N)c(Cl)c1 C1(N(C(C(CC)NC(C)=O)=O)C)CN(C(c2cncc(Cl)c2)=O)CC1(C)C Cc1cc(C)c(N2CCN(c3ncc(Cl)cc3C#N)CC2)c(Br)c1 C(=O)C1CNC(=O)c2ccnn21.CC(C)(C)C1=NOC(C)(C(N2CCC2C)=O)C1 Cc1cccc2nc(C(N3CC4(C3)CN(C(=O)CC3(CO)CCCC3)C4)=O)cn12 C1(O)(C(=O)NC2CN(C(C(c3ccc(F)cc3)OC)=O)C2)CCSCC1 c1(CC(=O)NC2CN(Cc3c(C)scn3)CC2O)ccc(Cl)c(Cl)c1 Cc1c(C(=O)NC(Cn2cncn2)C(N2Cc3ncsc3C2)=O)cccc1F CN1CCN(C(C2COCOC2)=O)CC1C(N1CCCCCC1CO)=O c1(C(=O)NCCC(CNC(C(C)OCCC=C)=O)O)nnn2ccccc12 Cc1ccc(C(=O)N(C2CCC(NC(C3NC(=O)CC3C)=O)CC2)C)cc1C#N N1(C(CNC(CC(C)C)=O)=O)CCC(C(=O)NCCCCCCSC)C12CCC2 C1(C)(C(N2CC(OCCC(=O)NC3C(C)CCC3)C2)=O)CCSCC1 O=S(=O)(c1ccc(N2CCC3(CC2)CC(O)CCO3)cc1Br)N1CCC(CF)C1 Cc1cc(C(=O)NCc2ncoc2CCNC(=O)CN(C)C)ncc1F C=CC(CC)CC(=O)NC(C)C(C)(C)NC(c1ccc(OC)c(OC)n1)=O c1(C(N2CCN(c3c(C(C)=O)ccc(CN)n3)CC2)=O)ccc([N+](=O)[O-])cc1F c1(CCC(=O)NC2CC(NC(=O)Cc3ccsc3Cl)C2)nnc(O)nc1O C1(NC(c2onc(C)c2C)=O)CC2CCC1(NC(c1ccnc(Br)c1N)=O)C2 c1(C(N(C)Cc2cncnc2)=O)n[nH]c2c1CN(C(C1CN(C3COC3)C1)=O)C2 n1(CC=O)cnc([N+](=O)[O-])c1.Cc1ncccc1C(=O)NC1(C)CCCCC1.N c1(C(N2CC(O)(CCNC(=O)Cc3ccnc(F)c3)C2)=O)noc2c1CCCC2 C(CC(=O)NC(C)CC(C)NC(=O)C(F)C1CCC1)(C(F)(F)F)OC C1(C(=O)NCC2(CC)CC2)CC2(CCC2)CN1C(c1cnn(C)c1)=O.O C(=O)(CC1OCc2ncccc21)NCC(CC=C)NC(c1nc(C)oc1OC)=O CC1(C)CN(C(c2cn(C(C)(C)C)cn2)=O)CC1.c1(CC=O)ccc(Cl)s1.C C1([SH](=O)=O)(C)CC1.n1(CN(Cc2cn(CC(CC)C)nn2)O)c(C)nnc1S.N Cc1cc2c(cc1NC(C1CCC1c1nc[nH]n1)=O)sc(=O)n2C C1(C=O)(CC)CCN(C(=O)C=CC(=O)N(C)C)C1.c1(C(C)O)ccncc1.N c1(C=O)ccc(C(F)(F)F)c(O)c1.C#CC(C)(C)C(=O)NCC(C)(C)C.C CC(CCO)N=c1[nH]c(=NC(CC2CC2)CC2CC2)[nH]c2c1CCCC2 S(=O)(=O)(c1ccc(N)nc1)N(C(C)CS(C)(=O)=O)C.C12CC(C)(CCO1)C2.C c1(C(=O)NC2CN(C(CSC)=O)C3C2C3)cc(=O)n(C)cc1Br N1(C(CC2CN(C(C)=O)C2)=O)CCCC(CO)(NC(=O)CN2CCCCC2)C1 CCC(CC)C(C(=O)NC(C(=O)NCCC(C)(C)F)c1cccs1)OC C1(C(N(CCC(N2C(CC)CC2)=O)C2CC2)=O)CN2CCC1C2 N1(C(=O)NC(c2ccc(C)cc2)c2ccco2)CCS(=O)(=O)CC1CO c1(C(C(=O)NCCOC)N(C(C)(C)C2CC2)C)ncc(C(F)(F)F)[nH]1 n1(CC)nccc1C(=O)NCC(C)N(C)C(c1sccc1CO)=O c1(C(=O)N)cc2occc2n1C.N1(C(CNS(CC)(=O)=O)=O)CCC(C)C(C)C1 N1(CC(=O)Nc2c(C)sc(I)c2)CCN(C(=O)OC(C)(C)C)CC(C)C1 C1(NC(CC(=C=C)C)=O)C2CC3C1C3C2C(=O)NCc1nc(CO)n[nH]1 N1(C(C(=O)NCC)=O)CCC(C(C)(O)C)CC1.CCC(F)(F)F.C(=O)C.N C1(C(=O)NC2CCC(NC(=O)CC(C)COC)CC2)(COC)CCCCO1 n1(CC)nnc(C(=O)NCC(C)(F)CNC(c2cc(C(C)C)sn2)=O)c1C c1(OC)ccc(NC(C2CCC(O)CN2C(=O)C(C)COC)=O)cc1O c1(C(CC)N(C(=O)C(n2cc(C3(C)CC3)nn2)C)C)ccccn1 CCCC(COC(c1ccc(OCC)c(F)c1)=O)C(=O)OC CC(CS(=O)(=O)N(C)C)N=c1[nH]c(=NC2CC3C(C2)C3(F)F)c2ncccc2[nH]1 CC1CN(C(=O)CC2CCC(F)(F)CC2)CCN1Cc1cccc(Cl)n1 N1(C(C2N(CC)CCC2)=O)CC(F)CC1C(N1CCC(F)(CF)C1)=O N1(C2CCC(NC(C(=O)N(C)C)=O)C2)CCN(C(c2ccc(Cl)cc2)=O)CC1 CCC(CC(=O)NCC(C1CC1)NC(=O)C=Cc1cnc(C)s1)OC N1(C(CN(C(C(C)C)=O)C)=O)CSCC1C(=O)NCCc1cc[nH]n1 c1(Cn2ncc(NC(N3CC4(CC(O)C4)C3)=O)c2)cc2ccccc2s1 C#Cc1cccc(C(=O)NCC(C)N(C(c2cc[nH]c2C)=O)CC)c1Cl N#Cc1cc(S(=O)(=O)NC2CCN(C(C3CCCS3)=O)CC2)ccc1Br Cc1ncc(NC(=O)CC2(NCc3cccc(O)c3O)CCC2)c(C)n1 Cc1cc(C(=O)NC2CCC2NC(c2cc(C3CC3)cs2)=O)nc(C)n1 CC(C)CCC(F)C(=O)NCC(C)(CC(C)C)NC(=O)C(C)OC1CCOC1 N1(C(C2CCCCN(C(CCc3c(C)noc3)=O)C2)=O)CCN2CC(C)CC2C1 C1(NC(C=C(C)Cl)=O)CC(O)(CNC(=O)CC2CC2C2CC2)C1 Cc1ncoc1C(=O)NCc1cc(C(=O)NCC2CCCS2)no1 c1(C(=O)NC2CCN(C(C3CCCOCC3)=O)C2)c[nH]c2ccc(F)cc12 C(CC(C)N=c1[nH]c(=NCc2ncccc2N)c2cccc(F)c2[nH]1)SC c1(C(=O)NCC2CN(C(CC(C)OC)=O)C(C)C2)csc2c1CCC(C)C2 C(=O)(CCCc1csc(=N)[nH]1)N(C1CCN(C(=O)CS)C1)C.c1ccccc1.C C(=O)(CCCCCC(c1nnnn1C)NC1(c2ccn3ccnc3c2)CC1)OC CCCCC(CCC)N(CCN1CCOCC1)C(=O)Nc1c(OC)ccc(Cl)c1F c1(C=O)cccc(F)c1.C1(CNC(C2(COCC)CC2)=O)CCC1.N C(=O)(C1=C2CCN=C2NC=C1)NCCCNC(=O)C=Cc1ncco1 C(=O)(C1CSc2ccccc21)N1C(CN(C(=O)CNCC(C)(C)C)C)CCCC1 N1(CCN(C(C(N2CCN(C(C(CC)CC)=O)CC2)=O)=O)C)CCOC(C)(C)C1 N1(C(c2cc(C(F)(F)F)no2)=O)CCN(C(c2nn[nH]c2Cl)=O)C2CCC12 C#CCC(C(=O)NCC(c1cnn(C)c1)O)NC(c1csc(C)n1)=O C1(C(=O)OC)(NCc2nc(N(C)C)no2)CCOC1(C)C c1(C(N2CC(C(C(=O)NCC(C)(C3CC3)OC)OC)C2)=O)nnsc1C CCCC(CCC)CC(=O)NCC1CC2CC2N1C(c1cc(SC)ccc1C)=O c1(C(N2CCCC(NC(c3cnc(CC)[nH]3)=O)(CO)C2)=O)occ2c1CCCC2 C1(NC(=O)C2=CSCCO2)COC2(CCN(C(c3cc(O)cc(=O)o3)=O)CC2)C1 C(C)(C)(C(C)CC(=O)N(C1CCOCC1C)C)NC(CS(CC)(=O)=O)=O c1(CC)cccnc1C(=O)NC(C1CCN(C(=O)CNc2nccs2)CC1)C C1(C(N(C2CCN(C(c3scnc3C(C)C)=O)CC2)CC)=O)CCC2CC2C1 n1(CC)c(C)cnc1C.C1(O)(C(C=O)F)CN(C(=O)CC23CCCC2C3)C1.N C#Cc1cccc(CC(=O)NC2CCCC(NC(c3cncc(NC)c3)=O)C2)c1 c1(CC(=O)N)ccc(F)cc1C(F)(F)F.CC(C(C)C)NC(=O)C(Cl)=CCl N1(C(CCN2C(C)CCCC2)=O)CC2CC(C1)N(C(C1SCCS1)=O)C2 C(N=c1cc[nH]cc1S(=O)(=O)NCc1cnn(CC2CC2)c1)C1(C=C)CCOCC1 N1(C(C(C)CO)=O)CC=C(CC(=O)NC2CCCCC23CC3)CC1 N1(C(c2c(CC)occ2)=O)CCCC(CC)C1C(N1CC(CO)C(O)C1)=O N1(C(C(CCCC=C)NC(=O)C(C)OC(C)=O)=O)CC(C)(C)OC(C)(C)C1 CC1CCC(NC(c2ccc(NC=O)cc2)=O)CN1C(=O)CCC1CCCCO1 c1(CC)cn2c(n1)CCCC2.c12cc(O)ccc1CN=C(NC1CC1)N2 C1(F)(NC(C2C3CN(C(c4ccccc4-n4ccnc4)=O)CC23)=O)CCOCC1 C1(NC(c2cc(OCC)n[nH]2)=O)CCN(C(=O)CN)CC1C.c1cnn(C)c1 c1(C(=O)NC(C=CC(N2CC(COCC)C2)=O)C)cnccc1OC N1(C(CN2CCC(OC)C2)=O)CC(O)CC1C(N1CCC(N(C)C)C1)=O N1(C(CCc2cnc(C)s2)=O)CCOC(C(C)NC(C2CN(CC(C)C)C2)=O)C1 C1(C(N2CC(C(=O)NC(CC)(C)C(=O)OC)C(OC)C2)=O)CC12CCCCC2 C(=O)(CC(C(C)C)C(C)C)N1CCN(C(c2cc(C)n(C)c2)=O)C(C)C1C c1(CNC2CCN(C(C(CC)N(CC)CC)=O)CC2F)c[nH]c2cccc(O)c12 N1(CC)CCOC(C(=O)NCCC2CC(C(=O)Nc3cncc(Cl)c3)C2)C1 Cc1ccc(C=CC(=O)NCC2CC2NC(=O)CC2CC2)c(C)c1 CCCC(C(O)C(=O)NC(C1(O)CCCCC1)C)NC(c1ccn(C)n1)=O n1(CC)nnc(C)c1C(N1CC2C(C(=O)NOC3CC4CCC3C4)C2C1)=O N1(C(C=CC(=O)Nc2c(N)nccn2)=O)CCC(CN2CCCC2=O)C12CCC2 C1(NC(CC2N(C)CCOC2)=O)CCCN(C(c2ccsn2)=O)CC1 C(CC#CC(C)(C)O)OC(C1CN(C)CC1c1ccccc1)=O C1(OC)CN(C(=O)CNC(c2cccnc2)=O)C(C)(C)C1.C(=O)C(N)=O C1(N)(C(=O)NCc2cn(CCOC)nc2)CCC(O)CC1 N1(C(c2c(C)cc(SC)s2)=O)CCN(C(=O)CN2CCCOC2=O)CC(O)C1 C1(C(=O)NCCC2CCCCC2)(CNC(=O)CC(O)C2CCCC2)CCCCC1 C(=O)(CC(C)c1cccnc1)NCCC(C)N(C(CC=CCC)=O)C C1(NC(C(N2CCNC2=O)C)=O)CCCN(C(C2CCC(=O)N2)=O)CC1 CC1(C)C(CNC(=O)CC2CS(=O)(=O)C2)CCN1C(c1nccnc1N)=O C1(C)(CNC(C2(COC)CCCCO2)=O)COCCN(C(C2CCOCC2)=O)C1 N1(C(c2c(CC)n[nH]c2)=O)CCOC(C(C)NC(=O)C(C2CCC2)OC)C1 C1(CC(=O)NC2C(CNC(c3ccc(C)cc3)=O)COC2)CCC(C)(O)CC1 C=CCCCCCNC(CC1CCCCC1)C(=O)NCC=C c1(C(=O)NC(CC)CNC(c2cc(C)c(C)s2)=O)c(C)cc(C)cc1C c1(CCC(=O)N)ccc(C)c(C)c1.c1(CCNC(C(C=C)O)=O)ccc(F)cc1 CC(=O)CCCC(C)C(=O)N1CCN(C(=O)Cc2cncc(C)c2)C(C)C1C c1(C(N2CCCC(CC)C2)C(=O)NCCC)cnc(N2CCCC2)nc1 C(=O)(C1COc2ccc(F)cc21)OCC(c1cc(C)n(C)n1)=O c1(C(=O)NCC2(F)CCCC2)ccccc1.C(=O)C(O)C1CC1.C1CC1.N c1(C(=O)NC2CCC(NC(=O)C=Cc3cccs3)C2)ccc(F)cc1 C1(C(=O)NC(c2ccncc2)CO)CN(C(c2cnccc2Cl)=O)CCO1 c1(N(c2cc(C)nc(N3CCCC(N=[N+]=[N-])C3)n2)C)ccc2n[nH]cc2c1 c1(C(N(C(C)CNC(=O)C(C)c2ccco2)CC)=O)ccc(Cl)c(C)c1O c1(N2CCC(C(C)O)C2)ccc(Br)c(S(=O)(=O)N2CCN(CC(C)O)CC2)n1 c1(OCC)oc(C)nc1C=O.C1C2CN(C(C3CCN(C4CC4)CC3)=O)CC12 c1(CC)cccc(C)c1NC(=O)C(N1CCC(CO)(SC)CC1)CCC c1(C(=O)NCCC2(C(N(C3CCN(C(C)=O)C3)C)=O)CC2)ccc(=N)[nH]c1 c1(COCC)ccccc1.C1(C)(C=O)CCN(C)C1.C(=O)CCC1CC1.N N1(C(C(CC)(C)C)=O)CCC(NC(=O)CC2CCCCC2(C)C)C(O)C1 C1(C(=O)NC(CN(c2nccc(SC)n2)C)C)CCC2C(C1)C2(F)F C(=O)(CC1=NN(C)C(=O)C1)NC(C(C)C)CCN(C)C(C1C(C)C1C)=O C1(NC(C2C(C(N)=O)C2)=O)(C)CCC(F)(F)CC1.c1(C(=O)N)c[nH]cc1Br C(c1cn(C)nn1)=CC(=O)N.C(C(=O)N(CC)C1CC1)(C1CCC1)OC c1(CN(C(C)C)Cc2nc(C3CCOCC3)no2)ccccc1Cl N1(C(CC)=O)CC(C)C1C(=O)N(CC(c1cnn(C)c1)O)CC.C(C)(C)C c1(OC)cc(C)cc(C(=O)NC2CC(CCNC(C3CCCCS3)=O)C2)c1C c1(C(N2CC(NC(=O)C3=CCCOC3)C3(C2)CC3)=O)ccnc2cc(F)cnc12 c1(C(N2C(CNC(c3nccc(C)c3)=O)CC2)=O)ccc2ccccc2c1C N1(C(CC2C(CC)C2)=O)CCC2(CC1)CC(NC(=O)C(CO)C(F)(F)F)C2 c1(NC(N(CC=C)Cc2ccncc2)=O)cc(C)nc(C)c1 O=S(=O)(c1cnc(Cl)cc1Cl)NCC1(O)CC2CCC(C2)C1 c1(NC(CSCC(C)OCC)=O)ccc(OC(F)F)cc1 C(=O)(CC(C)(C)O)NCCn1ccc(C(N(C)CC2(OC)CCC2)=O)c1 c1(C(=O)NC2CN(C(c3cc(C)no3)=O)CC2C)cnc2cnc(Cl)cc2c1 CC1CCCN(C(=O)C(=O)NCC(F)CNC(=O)CCC(=O)c2ccc[nH]2)C1 C1(C)(CC)C=C(C(=O)NC2CCN(C(c3cnoc3-c3ccco3)=O)C2)C1.C C1(C(N2CC(C3(C)CC3)OCC2)=O)CN(C(=O)C(c2ccccc2)O)CCN1C c1(C(C)=O)ccc2nc(N3CCC4C(CCN4C(=O)N(C)C)C3)sc2c1 C(CCCOC)(C(=O)N(C)Cc1cnc(C)s1)NC(C1N(CC)CCOC1)=O C(P(C)(C)=O)(c1cccs1)NC(N(C1CCCC1)CC=C)=O C1(C(=O)NCc2ccccn2)CCC2(C1)CN(S(=O)(=O)CC1CCC1)C2 C1(NC(C2(C3CCCO3)CC2)=O)CC2(CCCCCC2)C1 N1(C(C2N(C(=O)OC)CCC2)=O)CC2CCC(N(C(=O)Cn3cccn3)C)C2C1 N1(C(c2c(OC)ccs2)=O)CCC(NC(=O)Cc2nc(C)sc2C)C12CCC2 CCC(CC(=O)NC1CC12CCN(C(C1CCC(N(C)C)CC1)=O)C2)CC(C)C N1(C(c2cc(C)no2)=O)CCC2(NC(=O)CCc3ccccc3C)CCCCC12 c1(OC)ccc(C(F)(F)C(=O)NC2CCN(CCF)CC2)nc1 C1(C(=O)NC2CCN(C(=O)NC)CC2)CCCS(=O)(=O)C1 c1(CC(N2CC(=C(CNC(C(N3CCSCC3)C)=O)F)C2)=O)cnc(F)c(Cl)c1 C12(NC(c3occc3Br)=O)CCCC1N(c1nccn3nnnc13)CC2 C(=O)(C1=NOC(C)(C)C1)N1C(C(C)(C)NC(C(CSC)C)=O)CCC1 N1(C(c2scc(C)c2)=O)CC(NC(C2CCN(CC3CC3)CC2)=O)CC(C)C1 c1(C2(C(N3CCN(C(=O)NCc4ccncc4Cl)CC3)=O)CC2)cccc(F)c1 N1(C(C)=O)CCCCC1CCCNC(=O)C(n1ccc(C)n1)C N1(C(C2(C(=O)NC)CC2)=O)CC(C(C)NC(=O)Cc2nncs2)C1 n1(CC)nccc1C(N1CCC(CN(C)C)C1)C(=O)NC1COC1.C1CCOC1 Cc1cc(C(=O)NC2(C)CCCN(C(C3CC(C(C)C)C3)=O)C2)cc(C)c1F C(=O)(C1=C(C)S(=O)(=O)CC1)N(C1CN(C(CCCCCC#C)=O)CC1O)C N1(CC)CCN(CCC(=O)N(C)CC2CCCCN2C(C2CC3CC3C2)=O)CC1 C(c1cccs1)=CC(N1CCCC1C(O)C(=O)O)=O C(=O)(C(C#N)C(C)C)N(CCC(=O)NCCCC#C)C(C)C C=CCCC(CC(C)C)C(=O)N1CC(NC(c2ccnc3[nH]ncc23)=O)CC1C c1(SC)ccc(Cl)c(NC(=O)C(=O)NCCn2nc(C)cc2O)c1 c1(C(=O)NC(CN(C)C(c2c[nH]nc2S(N)(=O)=O)=O)(C)C)ccc2nncn2c1 Cc1cc(C(N2CC(NC(c3ccc(O)cc3O)=O)C(C)(C)C2)=O)cc(Cl)n1 C(C(O)C(=O)NCC1(C(=O)NCCN2CCOCC2)CCCO1)N(C)C N1(C(C2(N(C(=O)CCc3nccs3)C3CC3)CCC2)=O)CCCC(CCO)CC1 C=C1CCN(C(=O)C(C)N(CC)CC)C(C(=O)NCc2csc(C)c2)C1 C1(COC)C(=O)NCCN1C(C1CCCN(CCN2CCCC2)C1)=O N1(C(C2CCC(=C)CC2)=O)CC=C(C(=O)NCC2(CC3CCC3)CC2)CC1 c1ccc(Cl)s1.C1(F)(C(N(C)C)=O)CN(C(c2ccco2)=O)C1.C(C)(C)C N1(C(CCOC)=O)CCC2(NC(c3cnc(OCC(F)F)cn3)=O)CC2C1 C(=O)(C1=CCC(C)(C)CC1)N1CCCC(O)C1.c1(C(N(C)C)=O)cccc(=O)o1 c1(C(NC)=O)ccc(=O)n(C)n1.C1(O)CN(C(=O)C=CC(F)(F)F)C1.C N1(C(C=C(CC)CC)=O)CCN(C(c2cnoc2C(C)C)=O)CC(C)(F)C1 N1(C(C2CCN(C(C(C)C)=O)CC2)=O)CC2CCC1CN2C(C1CCCC1O)=O CC1CN(C(=O)CN2CCCCC2)CCN1C(=O)Cc1cc(Br)cs1 C(=O)(C1=COCC1)NC1CC(C(C(=O)NC(C)C2CC2)F)C1 c1(C(=O)NC2C(C)N(C(c3coc4c3CCCC4)=O)CC2)cccc2nsnc12 C1(C(=O)O)CN(C(=O)CC)CCC12CN(C(c1cc(F)c(C)c(Br)c1)=O)C2.CC C1(C(N(C)Cc2cccnc2)=O)C(C2CC2)CCN1C(=O)CCS(C)(=O)=O C(C)(C(C)(C)C(=O)NCCCCCCCO)NC(C1CC(C#N)(OC)C1)=O c1(OCC)ccccc1NC(C1COCCC1NC(C1(CO)CCOC1)=O)=O N1(Cc2cccc(OCCC)c2)CCC(C)C(NC(c2n[nH]cc2C)=O)C1 C1(COC)CCN(C(=O)C(F)n2ccnc2)CC1.c1(CC(=O)N)ccc(F)cc1 C1C2CC(O)C1N(C(=O)C)C2.c1(C(=O)N)ccncc1C(F)(F)F.C1CCC1 n1(CC)nncc1C(N1CCCC1C)=O.C(=O)(C(C)(C)C1(C)CC1(F)F)N c1(NC(=O)NCC2(C)COCCO2)nc2cc3c(cc2s1)OCO3 C(=O)(C(O)CC(C)(C)C)NCc1cc(C(=O)NC(C)C(=O)N(C)C)on1 N1(C(c2cnn[nH]2)=O)C2CCC1CN(C(C1(CCF)CCOCC1)=O)C2 c1(C(=O)NCCN(CC(C)O)C(=O)CC2CCNC2=O)cc(Cl)ccc1O N1(CC(=O)Nc2cccc(Cl)n2)CCN(C(=O)CCc2cccc(Br)c2)CC1=O c1(CCC)nc(C(=O)NCCN(C(c2occc2Br)=O)C2CC2)cs1 C(N=c1[nH]c(=NCCC2CCOCC2)[nH]c2ccsc12)C1(SC)CC1 N1(C(C2(CNC(=O)OC(C)(C)C)COC2)=O)CCC(O)C2CCC12 C(c1cccnc1)=C(C)C(=O)NCC(C1CCCC1)NC(C1(N=[N+]=[N-])CC1)=O c1(C(=O)NCC)cc2[nH]ccc2cc1-c1cc(C(F)(F)F)ccc1C CC(C(=O)NC(c1cccc(Cl)c1)CNC(C1CC(F)(F)C1)=O)C(C)O C1(C(N(CCC(=O)O)CC)=O)CCC(CS(=O)(=O)Cc2ccccc2)O1 C1(C)(CNC(=O)NC(Cc2c(C)noc2C)C)COC(C)(C)CO1 c1(C(=O)NCC2CN(C(C3CC4CC4C3)=O)C2)cnn2c1CCCC2 N(C(=NCCCCl)NCC(c1ccccn1)(C)C)Cc1c(C)n[nH]c1 c1(C(N(CCCCCNC(=O)CCc2cnoc2)C)=O)cc2ccnc(Cl)c2[nH]1 C1(CNC(c2cccc(C)c2C)=O)C2CCCC1N(C(C1CCS(=O)(=O)N1)=O)C2 c1(C(N2C(COC)CC2)=O)cc2cnccc2nc1C c1(OC)ccnc(CNC(=O)CC2(C)CCN2C(C2CC(C)(F)C2)=O)c1 c1(C=O)scnc1C.c1(CC(=O)NCC(C)OC)cccc(O)c1.C(C)=O C=CCC(C(=O)N1CC(O)(CNC(C2(CCCC)CC2)=O)C1)C(C)(C)C CN=S(C)(=O)c1cccc(C(=O)NC2CCC2NC(c2cnc(O)nc2)=O)c1 C1CN(C(=O)C(N2CCCC(O)C2)C)C(C)(C)C1.c1(C=O)ccc(C=O)o1.CO c1(C(=O)NC(CNC(C2(O)CCC(CC)C2)=O)(C)C)cnc2ccncc2c1 n1(CCCc2cc(-c3ncon3)ccc2C)cnc2c1c(=O)[nH]c(=O)n2CCC(C)C C1(NC(C(CCCCC)O)=O)CN(C(=O)CCCSC(C)(C)C)C2CCCCC12 c1(CCC)c(C)noc1C.C1(C(=O)OCC)(S)CCC1.C(C)(C)C.C=O C1(C(N2CC(C(N(CC(CC)(O)CC)C)=O)C(OC)C2)=O)CC2(C1)CC(C)C2 c1(C(N2CC3CN(C(=O)CCCCCCCBr)C3C2)=O)cn2cccc(Br)c2n1 N1(C(CC(=O)OC)=O)CC(C(=O)N(C)CC2COCCO2)C(C)(C)C1 C1(C(=O)OC)CCCN1NC(=O)C(C)c1cccc(Br)c1 C12(CC(=O)NC3CC(F)CN(C(c4occ5c4CCC5)=O)C3)CCC(CC1)OC2 C(=O)(C1(C)CCn2ccnc21)NC1CC2(CCC(C(=O)OC)OC2)C1 Cc1cc(C)c(S(=O)(=O)NCCN(S(=O)(=O)c2cccnc2C)C)c(C)c1 Cc1c(C(N2CC(CCNC(=O)CC3CNC(=O)C3)C2)=O)sc2nnc(S)n12 C1(C(=O)NC(C(=O)N2C(CC)CCC2)C(C)O)CN2CCC1CC2 c1(CC)cc(Br)ccc1CN1CCC2(CC2C(=O)Nc2ccc(Br)cc2)C1.O N1(C(c2c(C)nn(C3CC3)c2)C(=O)NC2CCCCC2)CCOC(C(F)F)CC1 N1(C(C(CC)O)=O)C2CCCC1CC(NC(=O)CCc1ccc(OC)c(O)c1)C2 c1(C(=O)NCC2C(C)CCN(C(CC)=O)C2)ccc2nnc(O)n2c1 c1(C(=O)NC(C2CC2)C)cnccc1OC.CC(C)=CC(=O)N.C1CCC1 c1(C(C(=O)NC2C(NC(c3ccccn3)=O)CCC2)=O)cc(F)ccc1F N1(C(C(=O)NC(C2(O)CN(C(CC=CC=C)=O)C2)C)C)CCP(C)(=O)CC1 C1(C=O)CCC2C(CC1)C2(F)F.C(c1ccc([N+](=O)[O-])s1)=CC(=O)N.CCC N1(C(C2C(=C)C2)=O)CC(CNC(c2ccc(F)cn2)=O)OC2COCC12 c1(C(=O)NCCC(=O)NCC(CCCC(C)C)C)[nH]c2cccnc2c1Br CC1CN=C2NC(C(=O)NC3CCCN(C(=O)CCC(N)=O)C3)=NN2C1 N1(C(c2cnc(C(N)=O)s2)C(=O)NCCCOCCOC)CC2CC2C1 C(=O)(C(C)S(=O)(=O)C(C)C)NC1C(NC(c2c(C)cnn2C)=O)CCC1 c1(CC(CC(C)SC2CCC2)c2nnnn2-c2ccc(F)cc2)cnc(C)nc1 N1(C(c2n(C=C)ncc2)=O)CCCCCCC1C(=O)NCCC1CCCCC1O c1(C(N(CCCNC(c2c(CC)nn[nH]2)=O)CC2CC2)=O)cnccc1 C1(CC(N2CC(CN(C(c3nc(CC)oc3)=O)C)C2)=O)CCCC2CCCCC12 C1(CCC(N2CC(C3N(C(c4c(C)nn[nH]4)=O)CCC3)(O)C2)=O)CCC(=O)NC1 Cc1c(C(=O)N(CCCNC(c2cncs2)=O)C2CC2)ccn1C(C)C N1(C(C=Cc2n(C)cnc2)=O)CC(C)C2(CCC2)C1.C1(=CC=O)CCSCC1.N C1(CCNC(c2ccon2)=O)CC(F)(F)CN1C(C1CC(F)(CO)C1)=O CCC(C)CC(=O)N1CCCC(C(=O)NCCNC(=O)CC2(C#N)CC2)C1 c1(CCC)cc(C(=O)NC2CCCCC2CNC(c2csc(C)n2)=O)nn1C C1(C(=O)NCCC#C)COCCN(C(=O)Cc2ccc(C)cc2C)C1 Cc1ncn(O)c1C(=O)NC1(C)CCCC1.c1(C(=O)N)cnc(N(C)C)nc1 Cc1c(C(N2CCC(CNC(C3CN(C(N)=O)C3)=O)C23CC3)=O)[nH]ccc1=O CCCC(O)C(CO)NC(C1CCCN1C(c1c(C)coc1CC)=O)=O c1(C(=O)NC(CC(C)C)CNC(=O)C(C)C2CCCC2)n[nH]c2c1CCCCC2 CCC(C(=O)OC)C(=O)NCC(CC)NC(c1ccc(Cl)cc1C(F)(F)F)=O c1(C(=O)NC2CC3C2CCN3C(=O)CN2C(=O)CCC2=O)n[nH]c2c1CCCC2 N1(C(c2c(C)nsc2)=O)CCC(C)(C)C1C(=O)N(CC(O)C(F)(F)F)C [SH](=O)(=O)c1cccc(F)c1.C(=O)(C#CC1CC1)N(C(C)CCNC(=O)C)C.N CC1(C)C2CC1CN(Cc1ccc(-n3cccn3)nc1)C2 C1(NC(Cc2c(Br)cn(CC)n2)=O)CCC12CN(C(=O)Cn1cnnn1)C2 C1(C(N2CCC(C(C(=O)OCC)(C)C)C2)=O)COCC2(CCNCC2)O1 CCC(F)(F)CC(=O)N1CC(=O)NCC1C(N1CC2CC1CC2CF)=O Nc1c(C(N2CCC(CNC(C3C(F)(F)C34CC4)=O)C2)=O)ccc(Cl)c1Cl c1(C(=O)NC(CC2CN(C(CSCC=C)=O)C2)C)ccc(CO)cc1 c1(OC)cncc(C(=O)N(CC(C)CNC(c2cnc(-c3cccs3)o2)=O)C)c1 N1(C(C23C(C(N)=O)(CCC2)C3)=O)CCC2(CC1)CC2NC(C1CCCO1)=O.C C1(C#CC(=O)NCC(CO)NC(C2CC(O)C2)=O)(CC)COC1 CCCC(C(C)CC)Nc1cncc(C(C)(C)F)c1 N1(C(C(CC#C)(C)C)=O)CCCN(C(c2ccc(C)nc2O)=O)C(C(C)C)C1 C12(C(=O)NC(c3ncc[nH]3)C)CCC(CC1)N(C(=O)COc1ccsn1)C2 c1(C(=O)NC(C(C)NC(CC(CCC)C)=O)(C)C)coc2c1C(=O)NCCC2 Cc1ccccc1C=CC(=O)NCCOCCOCC.C1(C=O)CC1Cl.N CCCC(C)(CC)C(=O)NCC(C)N(C(=O)CSCc1cccnc1)CC C=C(C)C(CC(=O)NC1CC2CC1N(C(c1nc(C)n(C)n1)=O)C2)OCC C1(OC)CCN(C(C2CC(C)CN(C(=O)C)C2)=O)C12CCC2.C(=O)(C1CC1)N N1(C(CCNC(CC(C)C)=O)=O)CCC2CCCCC2C1 C1(CNC(C(CCC)(C)C)=O)CC2(CCC2)CN1C(=O)C#CC1CCOC1 c1(C(=O)NCC(CSCC)SC)cccc(NC(C2(C)CCC2)=O)n1 Cc1nc2[nH]c(C(=O)NC3CCC(CNC(C4CCCN(C)C4)=O)CC3)cc2s1 C1CC2CCCC2N1C(c1cc2n(n1)CCO2)=O.C1(C(N)=O)CC1C(=O)NC Cc1cccc(C)c1C(=O)N(C)CC1CCN(C(=O)C(O)Cc2ccccn2)C1 N1(C(C2CC(CCC)OCC2)=O)CC(F)(F)CC1C.C(=O)(C(C)n1cncn1)N C1(c2nc(COC)nn2C)NC(=S)N(C2CC2C)C(CCl)=C1C(=O)OC C1(C(N2CC3CCN(C(C4(C(C)C)CC4)=O)CC32)=O)Cc2cc(F)cc(F)c2O1 C1(CCC=C)CCCN(C(C2CC(NC(c3ccnn3C3CC3)=O)C2)=O)C1 c1(C=O)ccnnc1O.Cc1oncc1C(=O)NCC(=O)NC1CCCC1C.N Cc1ccc(CCNC(C2CCC(C)N2C(c2cnc(O)[nH]2)=O)=O)cc1C c1(CCCC)ccc(C(C)C(=O)NCC(Cc2ccc(Br)cc2)CO)cc1 C(=O)C(C)S(N)(=O)=O.Cc1ccc(C(C)(C)C(=O)NC(C2CCCC2)C)cc1 c1(CNC2C(C)CC2)nc(-c2ccc[nH]2)cs1 N1(C(C(C)SC)=O)CC2(CCC(NC(C3CS(=O)(=O)C3)=O)CC2)C1 Cc1nc[nH]c1CC(O)C(=O)N(CC(C)CNC(=O)CN1CCCCC1)C Cc1noc(C(=O)N(C2CCN(C(=O)CCCC3CCOCC3)C2)C)c1C CCC(O)CC(=O)NCC1CCCN1C(c1cccnc1N)=O CC1CCN(C(=O)C2=NOCC2)C1CNC(C1(C(=O)N)CC1)=O.C1CC1 N1(C(=O)CC2CC2CNC(C2(F)CC2)=O)CCC(n2cncn2)C1 N1(C(c2c(C)nc(O)s2)=O)CC(N=[N+]=[N-])CC1C(N1CCOC(CN=[N+]=[N-])C1)=O Cc1c[nH]c(C(=O)NCCNC(c2coc(C3CCCCC3)n2)=O)c1 CC(CC(=O)NCc1cn(CCNC(c2cc(Cl)cs2)=O)nn1)C(C)(C)C C(C1CCCn2cc(C)nc21)NC(c1n(CC)ccn1)c1nnnn1C1(C)CC1 N1(C(=O)CCF)CCN(C(=O)COc2ccc(F)cn2)C2(CCC2)C1 c1(C(N2CCC(CNC(C3C(=C)C3C(=O)OC)=O)C2)=O)nc(C)nn1C c1(CC)[nH]nc(C(=O)NC2CCN(c3cc(O)nc(O)n3)C2)c1[N+](=O)[O-] N1(C(c2cccc(N(C)C)n2)=O)CCC2CCC(NC(C3CCC=CO3)=O)C1C2 C=CCC(C)(O)C(=O)N1CC2C(CC(=O)NC(c3ccc(F)cn3)C)C2C1 c1nc(C)c(C)o1.C(C(C(=O)NC)n1cc(C2(C(C)C)CC2)nn1)OCC C1(N(C(C2(C(C)NC(=O)CCc3nc(O)n[nH]3)CC2)=O)C)CCCC(C)C1C N1(C(C2(COC)CCCC2)=O)CCC(F)(CC(=O)N(CC(C)CO)C)CC1 CC1=C(C(=O)NC2(C)CN(C(c3ncsc3C3CC3)=O)C2)CCCC1 N1(C(N(C)C)=O)CC(NCC2(F)CC2)C1.C1CC(=O)NCCO1 C1(CC(=O)NC)CCCCN1C(=O)CCOCCCO.C1(=O)C(CC)N1C N1(C(C2CC(=C)C2)=O)CC(CNC(c2csc(Cl)c2)=O)CC12CCOCC2 c1(CCCC(=O)OC)cc2c(nc1C)N(C(=O)C(n1ccccc1=O)C)CCC2 C1(C(C)C)OCCC1CNCc1csc(C2CCOC2)n1 C1(NC(c2n(CCOCC)nnn2)C2CC2)CC(=O)N(c2cn[nH]c2)C1 C#Cc1cc(C(=O)NCC2CCN(C(C3CCC3)=O)C23CC3)ccc1Cl S(=O)(=O)(c1ccc(F)c(C(=O)NCCCCC)c1F)NC.c1(C(=O)N)ccsc1 c1(C(=O)NC2C3CC2N(Cc2ccc(C(=O)O)s2)C3)cnn2c1CCC2 C1(CN(C(C2CC(SC)C2)=O)C)CN(C(C2(O)COC2)=O)CCO1 N1(CC)CCCC(C(=O)NCCC2(O)CCN(C(c3ccnnc3)=O)C2)C1 C1(C(N(CCCOCC)C)=O)CN(C(=O)C)CC1C(C)C.C1CC=CC1.O c1(C(=O)NC2CC(NC(C(C)c3cc[nH]n3)=O)C2)ccc(C(F)(F)F)cc1 N1(C(C(CC)COC)=O)CC(OC)CC1(C)CNC(c1cn(C(C)C)nn1)=O c1(C(=O)NC2CC(NC(c3c(C)cno3)=O)C2)cc(C(C)(C)C)n(C)n1 c1(CC)cnc(CC(=O)NC(C)Cc2ccccc2)[nH]1.C(=O)(CC1CC1)N c1(CN(C(=O)CCc2cccnc2)C)cc(C)[nH]c(=NCC2CCCC2)n1 c1(C(=O)OCCCCC(C)C)cnc2c(c1)c(C1CC1)nn2-c1ccccc1 CC(C)C(CCO)NC(c1ccc(NC(c2ccc(Br)cc2)C)cc1)=O CC12COC(CO)(CN1C(C1CN3CCCN1CC3)=O)C2 Cc1ncc(C#N)c(NC2CCC(NC(c3cccc(C(C)(C)C)c3)=O)C2)n1 C=CCC(CC(=O)N(C)CCc1noc(C)n1)NC(=O)C(c1cnn(C)c1)O c1cc(O)nc(Cl)c1.C1(CC(=O)N)CCCCN1C=O.CCCCOC(=O)C c1(C(=O)NCC2CN(C(C(CC)(C)CC)=O)CC23CC3)ccc(Cl)cc1[N+](=O)[O-] c1(C(=O)NCCN(C(c2ccc(C)cc2)=O)CC)cc(OC)cc2c1CCC2 N1(C(c2c(SC)ccc(N)c2)=O)CC2CCCN(C(=O)C(F)OC(F)(F)F)C2C1 c1(CC)ccc(C(N2CC(O)(CNC(=O)CCC3CCCCO3)C2)=O)c(F)c1 N1(C(C2C(=C)C2)=O)CCC(NC(c2cc(C(C)C)c(O)cc2C)=O)CC(O)C1 N1(C(C(CCC)OC)=O)CC(C)(C)OCC1CNC(=O)Cc1ccon1 n1(CCC#C)c(C2CNC(=O)C2)n[nH]c1=Nc1cnn(CCC#N)c1 Cc1ncc(C(=O)NC2(c3ccccc3)CCN(C(=O)C3=CCC3)C2)n1C c1(C(C(=O)NCC2CCC23CCC3)OC)cc2ccccc2o1 N1(C(C(C2CCC2)NC(c2c(C)coc2)=O)=O)CCN(C2CCC2)CC1 c1(NC2C(C)CCCC2)ncccc1S(=O)(=O)NCc1cc(F)cnc1Cl c1(OC)cnc(C(=O)NCC=CC)c(F)c1.C(=O)(C(C)CC1CCC1)N N1(C(CCc2n(C)ncn2)=O)CCCCC1C1(NC(c2ccc(Br)cc2)=O)CC1 c1(C(=O)NC(C2CN(C(c3cccnc3)=O)C2)C)coc(C2CCC2)n1 N#Cc1ccc(CNC(=O)CNc2ccc(N3CCOCC3)cc2Cl)cc1 c1(OC)cc(C(N2CC(C)(C(=O)NC3COC(C(C)C)C3)C2)=O)sn1 c1(C(N(CC(=O)O)CC)=O)ccc(-n2c(C)cnc2O)cc1 CCCCCCC(C)C(=O)NC1CCCN(C(=O)Cc2cccs2)C1CC N1(S(=O)(=O)c2ccns2)CC=CCC2(CCCC2)C1 Cc1cccn2c(CC(N3CC4CC4(CNC(c4cc(Cl)no4)=O)C3)=O)cnc12 C1(CC(=O)N(CC(C)(C)OC)C)C2CCC(C2)N1C(=O)CS.C1CC1 c1(C(=O)NC(C)(C)CCNC(C2COC(=O)O2)=O)cc(Cl)cnn1 c1(C(=O)N)cccnc1.c1(CNC(C2CC(CC)C2)=O)cocc1.N(C)C N1(C(CC2CC3(CN(C(C)=O)C3)C2)=O)CC2COC(=O)C2C1.C=CCOC=O C1(NC(Cc2nc(C)[nH]n2)=O)CC(N=c2[nH]c(C3CCCCC3)nc(=N)[nH]2)C1 C1(C(=O)NC2CCN(C(c3ccc(OC)s3)=O)C(C)C2)CC2(C1)CC1(CC1)C2 CC(CC1CC1)C(=O)N1CCC(N(CCO)C(c2csnc2Br)=O)C1 Cc1ccc(OCCC(=O)NC2COCC2)c(Cl)c1.C1(CC(=O)N)CCN(C)C1 C1(C2CC2)CCN(C(=O)C(C)CC2CCC2)C1.n1(CC)nnc(C)c1C(=O)N N1(c2nc(N3CCC(COC)CC3)nc(C)c2)CC(C)OC2(CCCOC2)C1 C(=O)(C1=NOC(C)(C)C1)NC(C1(C(N2CC3CC2CS3=O)=O)CC1)C C(CC(C(C)(C)C)NC(=O)Cc1ccno1)N(C(C(CC=C)OC)=O)C C=CCC(C)(C)CC(=O)N1CCCN(C(c2cc(O)nc(Cl)c2)=O)CC1CO C(=O)(C1=CCCC1)NC1C(NC(CC(c2cccc(Br)c2)C)=O)CCC1 C(=O)(C=C1SCC(=O)N1C)NC1(C2CCN(C(C(CSC)OC)=O)C2)CC1 O=C(N=c1[nH]onc1C1CC1)C1CN(C(=O)Cc2ccc(Br)cn2)CCS1 N(C(=NCCC(=O)N1CCCC(C)C1)NCC1CC1)C1C(OC)CCC1 N(C(=NCCCOC)NCc1cc(-c2ccccc2Cl)on1)C(COC)C N1(C(CC(COC)(C)C)=O)CC2(CC(NC(c3ccn4nccc4n3)=O)CO2)C1 N1(C(CSCCC)=O)CCC(C2CCCCN2C(=O)Cc2cnc[nH]2)CC1 c1(C(=O)NC(C2CCOC2)CC)ccc(CNC(C2CCCC(=O)C2)=O)cn1 C1(NC(c2cnc(O)[nH]2)=O)COC2(CCN(C(C3CC(F)(CO)C3)=O)C2)C1 CC(C)(C)CC(F)C(=O)N1CCC(NC(C2CC3CCC2CC3)=O)C(O)C1 C#Cc1ccc(NC(C2(NC(=O)C(n3cc(C)cn3)C)CCN(C)C2)=O)cn1 Cc1nnc2n1CC(C(=O)NCC1C3CN(C(=O)Cc4nn(C)cc4Cl)CC13)C2 CN1CCOC2CN(C(=O)CSCC(=O)N(C3CC(C(=O)O)CCO3)C)CC12 C1(CC)C(NC(C2(O)CC2(C)C)=O)CCN1C(C1CCN(C(N)=O)CC1)=O C1(O)(CC(=O)NCC=CCC(=O)NC(C(C)C)C2CCC2)CCCC1 C1(NC(=O)C2CC2)CCC(C(F)(F)F)(NC2CC=CC2)C1 c1(C(N2CC(C)C(NC(c3cccc(O)n3)=O)C2)=O)ccc2nccn2c1 C1(C(CO)NC(CSCCOC)=O)CCN(C(=O)C(C(C)O)N(C)C)CC1 c1(-c2scc(O)c2)ccc(F)c(-c2ccc(Nc3ccnc(SC)n3)nn2)c1 C1(OC)CCCC1C(=O)N(C(C)C(=O)Nc1ccccc1)C(C)C C#Cc1ccc(C(=O)NC(C)C(C)NC(c2ccc(COC)o2)=O)o1 C1(NC(Cn2c(C)ncc2)=O)CC(C(N2CC(c3ccncc3)C2)=O)C1(C)C N1(C(c2cnc(C)nc2)C(=O)NC2CC2)CCCC2C1CCCN2C(C)C c1(N2CCC(CC)CC2)nc(N2CC3CC(C)(C)C3C2)nc2c1ncn2C(C)C N1(C(CC(COC)C)=O)CCCN(C(=O)CCSC2CCCC2)CC1 Cc1cc(CC(=O)NCCCCN(C)C(c2sccc2C#N)=O)n(C)n1 CC1CC2CN(C(C3(Cl)CC3(C)C)=O)CC2N1C(=O)CSc1ccncc1 C1(C(=O)NCC2CN(C(C3C(C(=O)OC)CCC3)=O)C2)C2CCCOC12 Cn1c(C(N2CCC(NC(=O)CCOC3CCOC3)C2)=O)ccc1[N+](=O)[O-] C1(C=O)CCCC(=O)N1C.c1(COC)nocc1C(=O)NC1CCC1C.N C1(N(C(=O)Cc2ccn(C(F)F)n2)CC)CCN(C(C2CCOC2C)=O)CC1 c1(C(=O)NCC2N(C(C(CC#C)O)=O)CCOC2)ncc(C)cc1OC N1(C(C(C(CC)C)O)=O)CCCC2(CCCCC2NC(c2[nH]c(C)nc2C)=O)C1 C1(C(N(C)CC2N(C(c3cnc(C(C)=O)s3)=O)CCC2)=O)CC(OC)CC1.O CCCCC(C)C(=O)N1CCN(C(c2cc(CC)oc2C)=O)C(c2cn[nH]c2)C1 c1(C(=O)NCC2N(CC(=O)NC(CC)C)CC2)cnc(Cl)c(Cl)c1 CC1C(NC(C2COCCOC2)=O)CCN1C(=O)CCCc1cccs1 C1(N(C(CC2(NC(C)=O)CC2)=O)C)CC2CCC(C1)N2C(C1(C)COC1)=O C1(C(N(CCN(C)C)CCO)=O)CN(C(=O)C#CC(C)(C)C)CC1C1CC1 N1(C(CCC2CCCN(C(C(COC)(F)F)=O)C2)=O)CC2(C1)CC2(F)F n1(CC(=O)N)ncc2ccccc12.Cc1ncc(C=CC(N2CC=CC2C)=O)s1 Cc1c[nH]nc1C(N1CCC(CCC(=O)N(C)CC2CCCOC2)C1)=O Cc1cnc2n1CC(NC(c1ccc(N3CCOCC3)c(F)c1)=O)CC2 C1(CNC(=O)CO)C=CCC1.C(C)(C)(C)OC.C(=O)C.CC(C)C c1(C(N(CCCNC(c2cnc(C)s2)=O)C)=O)cccc(OC2CC2)c1 N1(C(CCC(=C)Cl)=O)CCN(C(=O)C(C)NC(c2cccc(C)c2)=O)C(CO)C1 N1(C(CCC2OCC(C)(C)C2)=O)CCOCC1(C)C(=O)O C1CN(C(C2(O)CCOCC2)=O)CC1(F)F.c1(CC(=O)N)cccc(C(F)(F)F)n1 Cc1cccc(C(C)C)c1C(=O)NC1CCCC1.C12(C(=O)N)CC1COC2(C)C C(=O)(N=c1[nH][nH]c2c1CN(c1ncc(Br)cn1)C2)c1c2c([nH]n1)CC(C)CC2 C(C(C(C)C)NC(=O)C(C1CCCCC1)NC(=O)CC(C)O)OC CCCC(C(=O)NC1CC12CCN(C(=O)CS(=O)(=O)NC)CC2)S(N)(=O)=O c1(CC(=O)N(C)CCNC(=O)CC2(O)CC2)csc(-c2ccoc2)n1 c1(CCC(=O)N)cccc(F)c1Cl.C1(CCC(=O)N(CC)CC)CCN(C)CC1 c1(CC)c(OC)cccc1C(=O)NCC(C)NC(=O)C(C)(C)c1nncn1C Cc1cc(C)cc(C=CC(N2CCOCC2C)=O)c1.c1(CC=O)coc(C)n1.N C1(n2cc(CCN(C(c3cn(CCC)nn3)=O)C)nn2)C2CC3C(C2)C13 N1(C(c2cc(C)sn2)=O)CC2(CCCN(C(C3(N4CCOCC4)CC3)=O)C2)C1 CC(C)(C)CS(C)(=O)=O.c1(CCC(=O)NC(=O)C(F)(F)F)ccc(F)cc1Cl Cc1nscc1N(C(=O)C(C1(O)CN(C(C2CC23CC3)=O)C1)F)C N1(C(c2ccnc(C)n2)=O)CCC(C2CCN(C(=O)CC3CCCCC3)CC2)C1 C1(C(N2CC(OCCNC(CCCC#CC)=O)C2)=O)CC(c2ccccc2)=NO1 c1(C(N(CC(C)O)CCNC(=O)Cn2cnnn2)=O)cocc1Br O=C(CCCCCNC(=O)C(C1CCOCC1)F)NCc1cscn1 C1(NC(CC(C)(C)C)=O)CC2CC1N(C(c1ccc(Br)nc1N)=O)C2 N1(C(c2n(CC)ccc2)=O)CCCN(C(=O)CCc2cccnc2Cl)CC1CO N1(C(c2ccn(CCOC)n2)=O)CCCC(NC(c2ccc(F)cc2)=O)C1 N1(C(c2ccc(N(CCC)CC)nc2)=O)CC2CCC2(NC(=O)C(C)C)C1.S c1(CCC(=O)NCC2CC(F)CN2C(=O)C2=CCSC2)cnc2ccccc2c1 N1(C(C=C(CC)C)=O)CCCC(N(C(=O)C(N2CCSCC2)C)CCO)C1 C1(NC(=O)CC2CCCOC2)CN(C(C2C3(CC3)C23CC3)=O)C2(CCCCC2)C1 c1(C(N2C(CNC(CCC(C)OCC)=O)CC2)=O)cc(S(C)(=O)=O)cs1 CC1CC(NC(=O)C=C2CCCC2)CN(C(=O)CCc2ccsc2Cl)C1 C(=O)(CC(O)(CC)c1ccccc1)NCCN(C(=O)CCC1CCCCO1)CC C12(NC(c3nnn(CC)c3C)=O)CCN(C(c3cc4occc4[nH]3)=O)CC1C2 c1(N2CCC(CNC(=O)C(c3ccccc3)n3cccn3)C2)ncc(I)cn1 C1(C2CCC2)CCN(C(c2n[nH]c(C)n2)=O)CC1.C1(CCC)CC(C(=O)NC)C1 Cc1c(C(=O)N(C2CCC(NC(=O)C=CCO)C2)C)cnn1C(C)C c1(N2CC(C(C)NC(C(C)=CC)=O)C2)cccc(F)c1C#N C(C)(CCC(=O)N1CCCC1C(C)(C)NC(C1CC1(C)C(C)C)=O)SC c1(OCC)nc(NC(C)CNC(=O)C(CC)C2CCOCC2)ncc1Br N1(C(c2cnn(CC)n2)=O)CCOCC1CNC(=O)C(C1(O)CCCC1)F c1(C=O)cncc(C=O)c1.c1cccc(F)c1.C(=O)(CO)N(C(C)C)CC.N C1(CNC(Cn2c(=N)scc2)=O)CC2COCC2N1C(c1cc(O)cc(O)c1)=O CC1OCC2(CCNCC2)C1N(C(=O)C(C)NC=O)Cc1cc[nH]c1 N1(C(c2cccc(C#C)c2)=O)CCN(C(=O)CN(S(=O)(=O)CC)C)CC(C)(C)C1 N1(C(=O)Nc2ccc(CC(C)O)cc2)CCC2(CC1)OCc1ccccc12 c1(OCCOC)ccc(CC(C)NC(=O)C(c2cccnc2)OC)cc1 C1(NC(C=CC)=O)CCCOC12CCN(C(c1cc(F)c(CO)c(F)c1)=O)CC2 n1(CC)cnnc1C(N1CCCC1C1CCN(C(=O)C=CC(C)C)C1)=O N1(C(C(CCC)OC)=O)CCC=C(C(=O)NCCCC2CCOC2)C1 C(=O)(CS(=O)(=O)c1ccccc1Cl)NCCC(C)NC(C1CCSC1)=O N1(C(c2nc(C)n(C)c2)=O)CC(C)C(C)(C)C1.C1(C(=O)N)CCN1C1CCCC1 C1(CNC(C(CC)(C)C)=O)CCC2(CC1)CCC2.C1(C(=O)N)CC(C2CC2)C1 C(=O)(CCCC(C)(C)C)NC(CCCCNC(c1c(Cl)cc(C)nc1)=O)CO C(=O)(C(C(=O)NC12CC1CN(C(c1ccccc1)=O)C2)OC)OC.C1CC1.S N1(C(CCOCC(C)C)=O)CCCC2(NC(=O)CCc3nncs3)CCCC12 C1(C2(O)CCOCC2)(C=O)CC1.C1(COC)CCN(C(=O)CC(F)(F)F)C1.C c1cc(C(=O)N(C(C)CN(C(=O)CCc2cccc(Cl)c2)C)C)cc(Cl)n1.CO C1(COC)(NC(C2CCC(C)O2)=O)CCN(C(=O)CCc2ncnn2C)C1 Cc1cn2cc(C(=O)NCC3CCN(C(=O)CS)C3)nc2s1.c1cccnc1.C C1(N(C(c2c(C)scn2)=O)C)CCCCN(C(=O)C(F)(F)C(F)F)C1 Cc1c(C(=O)N(C)CC2CCCN(C(C3CC(O)C3)=O)C2)ccc2c1CCC2 C1(C(N(C2CCCN(C(=O)CCSc3ccc(Cl)cc3)C2)C)=O)CCC(F)CC1 N=c1nc[nH]c(=NCC(=O)N2CCOC(CNC(=O)Cc3ccccn3)C2)[nH]1 Cc1cc(C(=O)C(C#N)C(=O)NCCc2noc(=O)n2C)c(C)n1-c1ccon1 c1(NCCC2CCN(C(C(CC)C)=O)C(C)C2)ccc([N+](=O)[O-])cc1 C1(C(=O)NCC(C)NC(=O)C(C)c2cc[nH]n2)CCCN1c1nccs1 c1(CN2C3C(C(N4CCCCC4CO)=O)C(C3)C2)ccc2ccccc2n1 C1(CNC(=O)CN2CCCC2)CN(C(C2CCCS(=O)(=O)C2)=O)CC12CC2 C(=O)(CCC(=O)NCC(CC(C)C)NC(=O)CCN(CCCCOC)C)NC N1(C(C(Br)=C(C)C)=O)CC(C)CN(C(c2csc(C)c2N)=O)CC1C CC(C)C(C(=O)NCC1(CCNC(CC(C)(C)C)=O)CC1)c1ccncc1 N1(C(C2(CCOC)CC2)=O)CCC2(CC1)CCN(C(C1CCC3CCC13)=O)C2 N1(C(CC=CCNC(c2n[nH]c3c2CCC3)=O)=O)CCC2CCC(O)C1C2 C1(C(=O)NCCOCCOCC)CCC(C)CC1.C(=O)C(C)(C)C.N c1(OCC)nccc(C)c1C(=O)NC1CCCC1O.c1(C=O)cccc(O)n1.N c1(CC)nn(C)c(C(=O)NCC(C)(C(C)C)NC(=O)CCc2cnn[nH]2)c1Cl CC(C)(CC=CC(=O)N(CC(O)CO)CCO)NC(=O)CCC1CC1 CCCC(C(=O)N(CCNC(c1cccc2c1OCO2)=O)C(C)C)S(N)(=O)=O c1(C(=O)NC2(C)CC(NC(=O)C3=CC4CCCC34)C2)csc2c1CCC(C)(C)C2 C(=O)(C1CCc2nccn21)N1CC(NC(=O)C(=O)NC2CC2)CC(OC)C1 c1(C(=O)NC2CCN(C(C(C)OCCCC)=O)C2)ccn2c(Br)cnc2c1 C1(N(C(=O)Cc2cc[nH]c2)C)CCC(NC(c2csc(-c3ccoc3)n2)=O)CC1 Cc1nscc1CC(=O)NC(C(=O)NCC1(CO)CCC1)c1ccoc1 N1(C(CCC(=C)C)=O)CCCCC2(CCN(C(=O)C(C)(C)C3=CCSCC3)C2)C1 Cc1cc(Cl)cc(C(N2CCN(C(=O)COCC(C)(C)C)C3CCC23)=O)c1C C1(CC)CCCCN1C(=O)C(O)C(C)C.c1(CC)noc(COCC(=O)N)n1 c1(CC)ccnc(C(N2CCC(C)(NC(=O)CCC3C(=O)NN=C3C)C2)=O)c1 Cc1cc(C(=O)NOC(CC(C)C)C(=O)NC2CC3CCC2O3)c(C)cn1 C(=O)(C1CCCc2ccnn21)N1CC2(C(NC(Cc3nnc(C)s3)=O)CCC2)C1 C1(OC(C)(C)C)CCCN(Cc2sc(Cl)cc2Cl)C1 Cc1cc(C(=O)NC2CCCCC2NC(=O)CC(C)C(C)(C)C)c(N)c(F)c1 C1(C)(C(N2CC(COC)(C)C2)=O)CCCN1C.c1(CC(=O)N)ccccn1 c1(C(N2CCC(N(C(COC(CC)(C)C)=O)CCO)C2)=O)cn(C(C)C)cc1C S(=O)(=O)(c1cc(C(=O)O)ccc1Cl)NC1CCN(C(N2CCCC(C)C2)=O)C1 Cc1c(C=CC(=O)NC2CN(C(c3cn(C)nn3)=O)CC2O)cnn1C.C1CC1 N1(Cc2cc(C)no2)CCN(C(c2cccc(C(=O)O)c2)=O)CC1 O=C(CCCCCI)N1CCN(Cc2cn(Cc3oncc3C(=O)O)nn2)CC1 C(=O)(C1CN(CC)c2ccccc21)N1CC(O)(CNC(CC(C=C)(C)C)=O)C1 C1(C)(C(N(CCCN(C(CC(C)c2cnn(C)c2)=O)C)C)=O)CC=CCO1 C1(CC)CC(C(=O)NCCCCC(C)NC(=O)CC2(CO)CCOCC2)CCO1 c1(C(N(C2CCCN(C(=O)CC34COC(CF)(C3)C4)C2)C)=O)nccnc1O C(C)(C(=O)NCCC(=O)NCC(=O)NCC(C)C)OCCC=C.[SH2]=O c1(C(=O)NC(CCC)C(=O)N(C)CC2CCN(C)C2)ccc(C)c(F)c1 N1(C(c2c(C)nn(CCO)c2)=O)CCN(C)CC1CNC(c1cccnc1C)=O C1(C(C(=O)NC(C(=O)OC)(C)C)C)CCCN(C(c2cnc(Cl)n2C)=O)C1 C1(CC)CN(C(c2cnc(Cl)[nH]2)=O)CCC1NC(c1cc(C)n(CC)n1)=O C1(SC)COC2(CCC2)CN1C(=O)CCCOC(=O)C(C)(C)C c1(OC)cccc(SCC(=O)NCCC2CCCN(C(c3cnc(C)o3)=O)C2)c1 CCC(CCC(=O)NC(C(=O)NC(C)C(C)(C)C)c1ccco1)OC CCC(C)CC(=O)NC1CC(O)C1CC(=O)NC1CC(N2CCC2)C1 C(=O)(C1=CCCOCC1)N(CC)C(C)C.c1(OC)ccc(C(N)=O)cc1C=O c1(OC)ccc(C(=O)NCC(CO)NC(C2CCC(=O)N2)=O)cc1 CCCC(C)(O)C(=O)N(C1CCN(C(=O)CC(C)c2ccco2)C1)CC CN1CC(NC(C2C=CCN2C(=O)Cn2ccnc2)=O)CC1CO C(CCCC)(C(=O)NCC(n1cccn1)C)NC(CC(=C=C)C)=O C1(O)(C(C)NC(C(F)OC)=O)CCN(C(C2CCN2C2CCCC2)=O)C1 CC(C)S(=O)(=O)C(C)C(=O)NCC1CCN1C(=O)CSc1nncn1C CC1=CC(NC(C2C=CCN(C(=O)CCOC3CCCC3)C2)=O)CCC1 C12(NC(COCC#C)=O)CC1CN(C(c1ncnn1CC)=O)C2 C12(OCC)CCCC1(NCCn1cc(C)c(C(C)C)n1)CCO2 c1(C(=O)NC2C3CN(C(C(COC)OC)=O)C2CC3)cc2cc(Cl)cc(C)c2[nH]1 Cc1cn2c(n1)CC(C(=O)NC1CCC(C)CC1)CC2.c1(C(=O)N)cnc(S)[nH]1 S(=O)(=O)(C1CCN(c2ccncc2S(=O)(=O)NCC(C)(C)F)C1)NCC c1(N2CCCCC2)ccc(N)c(NCC(N2CC(OC)C(C)C2)=O)c1 C1(C(=O)NCc2c(CC)con2)CCC2(CC2)N1C(c1cc(O)ccc1C)=O C(=O)(C1=CSCCO1)NCC1N(C(CCc2n(C)cnn2)=O)CCC1 C(CCCC(=O)NC1CCCCCC1C(=O)NCCCOC1CCC1)(OC)OC CN1CCc2ccc(CNC(N3CC4CC(C3)C(O)C4O)=O)cc2C1 C=Cc1cnn(C)c1C(=O)N(C)CCN(C)C(C1CC(OC)C(OC)C1)=O c1(O)ccccc1.c1(OC)ccc(C(=O)NC2CCC2NC(=O)CSC)o1 C1(CC)CN(C(=O)CCOC)CC1C(=O)NCCc1cnn(C)c1 C(C(CNC(c1ccc(C(N)=O)cc1)=O)C(F)(F)F)OCCOC CC1CC(NC(c2cnn(C)c2)=O)CN(C(c2ccc([N+](=O)[O-])[nH]2)=O)C1 C(=O)(C#CC(C)(C)O)NC(C(=O)NC(COC)CCO)COC(C)C CC1(O)CCC(NC(C2(C)CCN(C(=O)CC3CNC(=O)O3)C2)=O)CC1 C1(C(=O)NCC(CNC(=O)CC(C)C(C)C)CO)(CC)CCC(O)CC1 Cc1cc(C)n2nc(C(N3CC4CC(NC(C5CC=CCO5)=O)C4C3)=O)nc2n1 C1(=CC(=O)NCCOCCCN(C(CSCC)=O)C)CCCCC1 N1(C(c2nc(C)oc2)=O)CC2CCCN(C(=O)CSc3ccc(F)cc3)C2C1 C#CCCC(O)C(=O)N.C1CN(C(c2c(Cl)n[nH]c2C2CC2)=O)CC1C(F)(F)F Cc1cc(C(=O)NCC(C(=O)N2CCCC2CC(C)O)N(C)C)nnc1O C1(C(=O)NC2CCN(C(C34CC(C)(OCC3)C4)=O)CC2O)CCCCC12CCC2 C1(NC(c2c(C(C)C)n[nH]c2)=O)CCCN(C(c2coc(CO)c2)=O)CC1 Cc1cccc(CN(C)C)c1F.N12CCCC(C1)CN1CCC1(C)C2=O C12(CNC(c3ccn(C)n3)=O)CC(NC(=O)CCc3cncn3C)(CO1)C2 Cc1ccc(NC(=O)C(N)Cc2cccc(Br)n2)c(OC(C)C)c1 Cc1cc(C)n(C)c(=O)c1CNC(=O)Cn1cc(CC(C)O)nn1 n1(CC(C(=O)Nc2cccc(C(C)F)c2)C)ccc2ccccc12 C(=O)(CC(F)(F)C(F)F)N1C(C)(CCC(N2CCC(CCN(C)C)C2)=O)CCC1 C1C(C)C(=O)N=CCC(=O)N1C.C(C(=O)NC(C)C)N(C1CC1)CC c1(C(=O)NC2(C)CCN(C(C3CC(C)(F)C3)=O)C2)cc(Cl)cc2ccncc12 N1(C(C(CC)(C)OC)=O)CC2CC(C1)N(C(c1cn(CCC3CC3)nn1)=O)C2 c1(CCC)cc(C(=O)NCC(C)NC(c2cc(CC(C)C)[nH]n2)=O)ccn1 C1(NC(c2c(C(C)C)noc2)=O)CCCC2CN(C(C3CC4(CC4)C3)=O)CC12 C1(NC(C2C3CCCC23)=O)CC2CCC(C1F)N2C(c1ccccc1F)=O N1(C(CCN2C(=O)C(CC)CCC2)=O)CCOC2CC12.C(N)(=O)NC C(=O)C(C(C)(C)C)N(C)C.c1(OC)nc(C(=O)NCC2CCC2)sc1C.N C1(c2n(CCC)nnn2)(NCCNC(=O)OC)CCCC(SC)C1 c1(C(=O)NCC2=CCN(CCCCC3CCOCC3)CC2)ccc2cccnn12 C(c1ccsc1Br)=CC(=O)NC1CC(NC(=O)CC2CC(=O)NC2=O)C1 c1(C(N(C2CN(C(c3cncnc3)=O)CC2F)C)=O)c[nH]c(=O)c2ccncc12 c1(C=O)cn2c(n1)CC(C)CC2.c1(OC)c[nH]nc1C(=O)N.C1(O)CCC1.C N1(CC)CC(C(=O)NC(C2(O)CN(C(c3ccnnc3)=O)C2)C)CC1=O C1(CNC(CCSCCC)=O)CCC2CN(C(=O)CC3OCCCO3)CC12 N1(C(c2c(CC)non2)=O)CCC2CN(C(c3cncc(OC)c3)=O)CCC2C1 Cc1cc(C(=O)N(C2CCCCN(C(c3cscc3C)=O)C2)C)cc(C)n1 Cc1cc(NC(c2ccc(SCc3ccc(C)n3C)o2)=O)c(Br)cc1F N1(C(C(=Cc2ccccc2)C)=O)CCC(C(N2CC3(CSC3)C2)=O)C(O)C1 c1(OC)nc(Br)ccc1CNC1CCCN(C(c2ccc(C)cc2C)=O)C1 c1(C(=O)NC2(CO)CCN(C(C(C(=C)C)(C)C)=O)C2)n[nH]c2c1CC(C)CC2 CC(C)C(C(=O)N(C)CC1CCCN1C(=O)CC1(CO)CC1)c1cnn(C)c1 C#CC1(C)CCN(C(c2cnc(C)nc2)=O)CC1.N1(CC(=O)N)C(=O)CNC1=O CCCC(C)(C)C(=O)NC1(CO)CN(Cc2ccc(Cl)c(F)c2)C1 C(=O)(C1=CCC(NC(C2CCCOC2)=O)C1)NC(C(=O)OCC=C)(C)C c1(C(N2CC(OCCNC(C3C(C)(C)CC3)=O)C2)=O)cc2cccc(F)c2s1 N1(C(c2c(CNC(c3cccc(O)c3)=O)cco2)=O)CC2C3CCC(O3)C2C1 Cc1ccc(C(=O)NC2C3CC2N(C(C2OCCC2C)=O)C3)c(Cl)c1C c1(C(=O)NCC2(C)CCN(C(=O)CC3CC4CC4C3)C2)cc2nn[nH]c2cc1F n1(CCCC(=O)NC(C)CCNC(c2cocc2Br)=O)ccccc1=O C(C(C=O)NC(=O)OC(C)(C)C)OC.c1(C=O)ccco1.CC(C)C.N c1(C(C(N2CC(CNC(c3c(C)ncnc3)=O)C2)=O)C)ccc(F)cc1F Cc1cc(C(=O)NC23CCCCC2N(C(=O)CCF)CC3)cc(S(C)(=O)=O)c1F c1(C(=O)NCC2CN(C(=O)CC3=CCCC3)C3CC23)cccc2c1CNC2=O CCC(C)(C)C(O)C(=O)N1CCC(C(=O)NC(c2ccc(O)nc2)C)C(C)C1 c1(OC)ncc(C(=O)Nc2ccsc2C=O)cc1C.c1cnn(C(C)(C)C)c1.N C=CCC(CC)C(=O)N1CC(CC(C)NC(c2cc(F)c[nH]2)=O)C1 C(=O)(C(C)C1=CCCC1)NC(C(C)C)CCN(C)C(c1csnn1)=O N1(C(C(C2CN(C(c3n(CC)nc(C)c3)=O)C2)O)=O)CC(C2(C)CC2)C1 Nc1c(C(N2CCN(C(C3CC3c3ccco3)=O)CC2C2CC2)=O)cccc1Cl c1(OC)cnc(Cl)c(NC(=O)Cc2ccc(N3CCCC3)cc2)c1 C1(NC(C(CC)(F)F)=O)CN(C(c2cccc(OC3CCC3)c2)=O)CC2CC12 CCC(C)(C)C(C)NC(C12CC1CCN2C(=O)COc1ccn(C)n1)=O C1(C(N(CC=C)Cc2ccc(Cl)s2)=O)CCn2c(cnc2-c2ccccc2)C1 c1(C(N2C(C(=O)Nc3c(OCC)nccn3)CCC2C)=O)c[nH]c2ncccc12 N1(C(c2cccc(C)c2)=O)CCC2C(NC(=O)Cc3csc(S)n3)CC12 c1(OC)ccc(C(C)C(N2CCN(C(=O)COc3cccnc3)CC2)=O)cc1F CC1SCCCC1C(=O)NC(C1CCCCC1)C(=O)NCCCC(F)F CCCCCC(O)CC(=O)NC1CN(C(c2ccc(N)c(C)c2)=O)CCC1C N1(C(=O)Nc2n(CC)nnc2)CCC(C)(C)C2OCCC2C1 N1(C2CCC2)CCOCC1.C1(NC(=O)CC2CC2CO)CCOC1 c1(C(=O)NC(CCNC(CC(c2cccc(OC)c2)C)=O)C)cccc(=O)n1C CC1(NC(=O)CN(C(=O)CSCC#N)CC2CC2)CC(O)C1 C1(CNC(c2cnc(OC)c(C)c2)=O)CN(C(c2cnsc2)=O)CC12CCC2 C(C)(C)(CCC)NC(C1CC(C(F)F)(OC)C1)=O.c1(CCC=O)nccn1C C(=O)(C1CCCc2c[nH]nc21)NCC1CCN(C(C(C=C)(C)O)=O)CC1 N1(C(C(C2CCCCC2)C)=O)CC(C)(NC(=O)Cn2cc(N(C)CCO)nn2)C1 c1(C(N2CCN(C(CN(CCC)C)=O)C(COC)C2)=O)cc(=O)n2nccc2[nH]1 C1(NC(CC(CC)SC)=O)C2CC(O)C1N(C(=O)CC1OCCO1)C2 N1(C(C(C)(C)n2cncn2)=O)CC2CCCC2(C(=O)NC2CC(C3CCC3)C2)C1 N1(C(C(N2CCCCC2)C)=O)CCOCC1CN(C)C(c1cnnn1C)=O N1(C(CCOC(C)=O)=O)CCCC(NC(C2(N(C)C)CCC2)=O)C(F)C1 c1(C(=O)NCCCN(C(C2C(C)(COC)C2)=O)C)ccc2ncccc2n1 c1(CC)cc(C(=O)NC(c2ccccc2)C(=O)NCC(C)CC)nn1C N1(C(CC2(C#N)CC2)=O)CC2CC(NC(c3coc4c3COC4)=O)C(C2)C1 CCCCCC(O)CNC(c1oc(CNC(=O)CCCCCOC)nc1C)=O CCCCC(F)C(=O)N1CCC(C(=O)NCC2(O)CC(C)(C)C2)(CO)C1 c1(CCNC(C(N2C(COC)CCCC2)=O)=O)cn(C)c2cc(C)ccc12 C1(CCCNC(C2CSC2)=O)CCCN1C(C1CCCCC1)=O C12(C(=O)NCCNC(CCOC)=O)CC1CN(C(c1ccc(O)nn1)=O)C2 N1(C(C2(C)CCN(C)CC2)=O)CC2CCC(C(=O)N=c3ccn(C(F)F)[nH]3)(C2)C1 CCC(CC)C(O)CNC(=O)CCN(C(=O)C(C(C)C)C1CCC1)C(C)C c1(OC)nc(Cl)c(C)cc1NC(=O)C(=O)NC1CCC2(CC1)CNC2 c1(NC(CCN(C)C)=O)ccccc1NC1CC2(C1)CC2C(=O)O c1(C(=O)NC(CNC(CC(C)O)=O)(C)CO)snc(Cl)c1Cl C(COCCO)(CC(C)(C)C)NC(c1ccc(C(C)C)cc1)C C(CN=c1nc(N2CCc3ncn(C)c3C2)cc[nH]1)c1scc(CC)n1 C(CC(C)(C)CC(=O)N1CC(NC(C2(C3CC3)CCCO2)=O)CC1C)OC N1(C(CCc2scc(C)n2)=O)CCC(CNC(C2CC2[N+](=O)[O-])=O)C1(C)C C(CC(C)C)(c1ccccn1)N(C(c1ccccn1)C(=O)NC)CC c1(CC)n[nH]cc1C(=O)NCC(CC)NC(c1ccc(C2CCCCC2)s1)=O C1(NC(CC(=C=C)C)=O)CN(C(c2ccc(-c3ccccn3)nc2)=O)CCC1C C(=O)(C(C)(O)C(C)(C)C)NCC1CC(NC(c2cc(C)[nH]n2)=O)C1 C#CCCCCC(=O)NC(CC1CC1)CC(=O)NCc1ccncc1Cl c1(OC)cc(C(=O)N(CCNC(C2CCCN(C)C2)=O)C2CC2)ncn1 C12(CNC(C(CC)C(C)C)=O)CCCC(CN(C(=O)C=Cc3cnc[nH]3)C1)C2 CC1CN(C(=O)Cc2csc3nccn23)C(C)CN1C(=O)CCc1ncco1 C1(O)(CC(=O)OCC)CCCN(Cc2cccc(Oc3cccc(Cl)c3)c2)C1 C(=O)(N=c1[nH][nH]cc1I)C1CCN(C(=O)Nc2ccc(C)c(O)c2)C1 CC1CN(C(c2cc(C3CC3)no2)=O)CC1CNC(C1CC2CC2C1)=O C1(C(N(CC(C)O)CC)=O)CCN(C2CCCCC2)C1.C(C=O)N(CC)CC C1(OCC)CC(c2nnnn2C(C)(C)C)(NC2(c3cccc(Cl)c3)CC2)C1 CCC(CC(C)C)C(=O)N1CC(NC(c2cc(C)ccc2Br)=O)CC(F)C1 C1(NC(C2CCC(C)(C)CC2)=O)CC2CCC(C1)N2C(C1NC(=O)OC1(C)C)=O c1(C(=O)NCC2(C)COCCO2)cc(S(=O)(=O)N(C)C)on1 c1(-c2ccc(CONCc3nc(Cl)nc(C4CC4)c3Cl)cc2)nnc2n1CCCCC2 n1(C(CC)C)nc(C(=O)NCC2(F)CC(NC(=O)C(C)(C)O)C2)cc1C c1(CC(N2CCC(N(C(C(C=C)(F)F)=O)C)CC2)=O)cccc2c1OCCO2 N1(c2cc(CC(C)C)ncn2)CCCC2(NC(=O)C(C)SC(F)(F)F)CCCC12 C12(NC(C(=Cc3ccccc3)OC)=O)CCCN(C(C3CC3(C)CC)=O)CC1C2 c1(C(N2CC(NC(C=C(C)C)=O)C(C(F)(F)F)CC2)=O)csc2ccc(C)cc12 C(=O)(C(C)(C)C(C)(C)O)NCC(CC(C)C)NC(c1c(CCC)occ1)=O N1(C(c2c(N)cn(C)n2)=O)CCCC(NC(=O)CC2C=CCCC2)CC1 C(C(C)(C)C(C)(F)F)NC(COC1CCN(C(c2c(C)nccn2)=O)C1)=O c1(CC(=O)N(C)CCNC(C2CCC2F)=O)ccc(Cl)c2cccnc12 CCC(C)CCCC(=O)NCC12CC(C)(CO1)C2.c1cccc[n+]1[O-].C(=O)(C)N C(=O)(C(C(C)C)NC(=O)CCn1cccc1)N(C)Cc1ncc(C)o1 c1(NC(C2(F)CN(Cc3ccncc3)C2)=O)ccc2[nH]ccc2n1 C1(C)(C(=O)NCC2CCC(C(N3CCC(CCOC)C3)=O)C2)CCCCO1 CC1(C2CCN(C(=O)C(Cn3cccn3)NC(=O)CC3CCC3)CC2)CC1 CC1(C#CC(=O)N2CC3CCCC(NC(C4CNC(=O)N4)=O)C3C2)CCCO1 c1(C(N2CCC(CCC(=O)N(C3(CC)CC3)C)C2)=O)ccc(C)nc1 N1(C(c2n(C(C)C)nnc2)=O)CCCC(C2(NC(C3CCCC(O)C3)=O)CC2)C1 c1(C(N2CC(NC(CC3N(CC)CCC3)=O)C(F)C2)=O)cnc2ncnn2c1O C1(NC(c2cc[nH]c3nccc2-3)=O)CCC2CN(C(=O)CN3CCCC3)CC2C1 N1(C(c2ccc(C(F)F)o2)=O)CC2(C1)CN(C(C1CC3OC1C1CC31)=O)C2 c1(-c2scc(C(=O)Nc3c(C(=O)OC)nc[nH]3)n2)ncnc(C)c1C C12(CNC(c3cnc(SC)n3C)=O)CCCC1CN(C(=O)C=CCF)C2 S(=O)(=O)(c1ccc(-c2ccccc2)s1)N1CC2C(C(=O)O)(C2)C1 c1(C(N(CCC)C(C)C)=O)cnc2c(c1)CCC(=O)N2.c1(C=O)cnc(Cl)s1.N C1(NC(CC2C(C)CCO2)=O)CC2(C1)CN(C(=O)CCc1ccc(F)nc1)C2 S(=O)(=O)(c1ccc(=NCCCCC2CC2)[nH]c1)NC(C1CCOCC1)CC C1(CNC(CC2(C)CC2)=O)CC2(CO1)CN(C(c1ncc(Cl)cc1Cl)=O)C2 n1(CC)nc(C)c(CC(=O)NC2CC2NC(=O)CO[Si](C)(C)C)c1C CCCCC(C(=O)NOC(C)(C)C(=O)OC)NC(=O)CN(C)C(=O)C1CC1 C1(C(=O)NCCCc2ccncc2)CCC2(CC2)N1C(=O)C(C1CCCCC1)O C(CC(C(=O)NCC1CC1C(=O)O)NC(C)=O)OC.c1ccc(C)nn1 C#CCC(C)(CC)C(=O)NC(CN(C(=O)COCCC1CCCC1)C)CC C1(CNC(=O)NC2CN(C(C)=O)C2)CC2CC1C1CC21 Nc1ccnc(C(=O)NC2CCCCC2NC(=O)CCC(F)(F)F)c1Cl c1(C(NOCC(=O)NC2C(OC)COC2)=O)cc(O)nn1C C1(NC(CN(CC)CC)=O)CC(F)CN(C(c2ccc(F)cc2OC)=O)C1 Cc1ccnc2c(C(=O)NCC3CCN(C(=O)COCCO)CC3C)cnn12 C1(C(=O)Nc2c(C)noc2)CCC2(CN(C(C3CCC(=O)NC3)=O)C2)O1 c1(C2(C(=O)NCC(CO)NC(C3C=CCC3)=O)CCCC2)cc(F)ccc1F c1(C(=O)N)cnn2c1NCCC2.C12CC(CO1)N(C(=O)CC1(O)CCOC1)C2.C c1(CC)oc(C(=O)N(C2CCCN(C(c3cnc(S)[nH]3)=O)C2)CC)cc1C C1(NC(C(CC)O)=O)CC2(CCC(CNC(C3CC(OC)C3)=O)OC2)C1 C1(CCC(=O)N(C2OCCC2CC)CC)CCCN(C(C2CCN(C)CC2)=O)C1 Cc1ncsc1CCNC(=O)CCNC(C1CCCO1)=O C1(NC(c2c(C)csc2)=O)CC(O)CN(C(=O)Cc2ccccc2)C1.C(N)=O.N C=CC(C(=O)N1CCC(n2cc(C3CC(=O)C3)nn2)C1)c1ccccc1 Cc1nc(Br)oc1C(=O)NC1(C)CC(NC(=O)CC(C)N(C)C)C1 c1(SC)nc(N2CCCC2CNC(=O)CC2CCC=CCC2)cc(C)n1 c1(C(=O)NCC(CNC(C(CCC)=CCC)=O)F)ccc([SH](=O)=O)nc1.N CC(C)C(CNC(=O)CCOCC(F)F)C(=O)NCc1ncc(F)cc1F C1(C(C)(C)C)(NC(C(CO)NC(C)=O)=O)CCN(C(C2CC2CF)=O)C1 C1(NC(COCC=C)=O)CN(C(=O)C(C)CCc2cccc(F)c2)CCC1CO C(=O)(C1=COCCO1)N(CC)CC.C1(C(=O)N)(CC)CC(C)(C)C1.CCO C1(CC)C(C(=O)NC2(CN(C)C)CCCC2)CCN1C(c1cnncc1O)=O c1(C(=O)OC)ccc(Cl)cc1NC(=O)NC.c1cccc(C2(C#N)CC2)c1 N1(c2nc(C)cc(OC)n2)CCC2(CC1)OCCCC2c1nc(C)no1 C1(CCNC(=O)CCC2CCCOC2)CCN(C(=O)CNC2CCCC2)CC1 CCC1C(=O)Nc2ccc(C(N3CCC(C(=O)OC(C)(C)C)C3)=O)cc21 C(=O)(C1SCc2cccnc21)N(CC(C)NC(c1ccnc(C(F)F)c1)=O)CC C1(C(N)=O)CN(C(c2cc(C(=O)O)nn2-c2ccccc2)=O)CCO1 c1(N(CC)C)nn(C)c(C)c1Br.C12CCN(C1)C2=O.C(OCC)OCC N1(C(CC(=O)OCC)=O)CCC2(CC1)CN(C(C1CCC1c1nc[nH]n1)=O)C2 N1(C(C(CCOC)C)=O)CCOCC(NC(=O)CC2CCC(F)(F)CC2)C1 C=CC(F)(F)C(=O)NCc1ccc(C(=O)NCC(c2nncn2C)C)o1 N1(C(c2cc(CC)nc(O)c2)=O)CCOC2CN(C(=O)CCC3CC3(F)F)CC12 N1(CC(=O)N(CCCN(C(C(C)SC(F)(F)F)=O)C)C)CCCCCC1 c1(NCCCc2cn(CC)nn2)ccc(S(=O)(=O)N2CCOCC2CO)cc1Br C(CCCCC(=O)N1CCCC(C(=O)NCCNC(=O)CC(C)F)C1)=CCCC C1(NC(CC2N(C)C(=O)CC2)=O)CCC2CCN(C(=O)CCC(C)(C)C#N)C1C2 N1(C(c2c(SC)cn(C)n2)=O)CCN(C(=O)COC(F)F)C2CCCCC2C1 N1(C(=O)CCN2CCCC2)CC2CCN(C(c3cccn4cncc34)=O)C2C1 N1(C(C(=O)NC(CC)C)CC2C(OC)C2C)CCCN(Cc2occc2C)CC1 C=C(C)C(CC(=O)NC(C)(C(N1CCCC(C)(CO)C1)=O)C1CCC1)OCC C1(C(N(C2CCN(C(c3conc3C3CCC3)=O)C2)CC)=O)CNC(=O)C1 C1(c2cccc(COC)c2)CN(C(C)=O)CCN1C(c1nn(C)c(C)c1Cl)=O S(=O)(=O)(c1ccc(=NCC(C)(C)C)[nH]c1)N1CCC(C(CC)CC)CC1 c1ccc(C(F)(F)F)c(Br)c1.CC1=CCC=CC1C(N1CC2CC2(CN)C1)=O C1(C(C)(F)F)(C(N2CC(C)(NC(c3ccncc3)=O)C2)=O)CCOCC1 N1(C(C=C(C)C2CC2)=O)CCC(Nc2nccc(CC#N)n2)C(CO)C1 C1(CNC(c2ccc(CC)o2)=O)CC(F)CN1C(=O)C(C)NC=O CCCCC(O)C(C)C(=O)N1CC2(C)CC1(C(=O)NCCC(O)CO)C2 C1(C(N2CC(CCCCNC(C(C)(C)SC)=O)C2)=O)CC2(C)CC1CO2 N1(CC)C(=O)CCC1C(=O)NC1CCC(F)C1.N1(CC=O)CCCCC1=O.C C1(NC(C(CCCOC)C)=O)CN(C(=O)CCc2nccn2C)CC1S(C)(=O)=O c1(OC)ccc2[nH]c(-c3ccc(NCc4cccc5nn(C)cc45)nn3)cc2c1 c1(C=O)ccn(C(F)(F)F)n1.c1(C(C)C(=O)NC)cncnc1.C1(CC)CC1 C1(NC(C(C2CCCC2)NC(Cc2scc(C)c2)=O)=O)CNC(=O)OC1 c1(C(=O)NCCCCC2CN(C(C(CCCC)O)=O)C2)cc2ccccc2cn1 c1(C(N2CC(O)CC(NC(c3c(C)cc(C)s3)=O)C2)=O)cnc2sccc2c1 c1(C(=O)NC(COC)C(=O)N(C)CC)nn(C)cc1SC.C(=O)(C=CBr)N N1(C(C2(CC)COC2)=O)CCC(N(C)C(C2(C3CCCO3)CCC2)=O)C1 c1(C(=O)NC2CN(C(C(C)n3ccnc3)=O)CC2C)ncc(Br)cc1N c1(NC(C2CCN(C(c3cc(O)ccc3I)=O)C2)=O)cc(Cl)ncc1[N+](=O)[O-] C1(NC(C(C2CC2)OC)=O)CCCC1(C)CN(C(=O)CSC1CC1)C C=CC(CCC)CC(=O)N1CCCCC(NC(c2ccc(O)nn2)=O)CC1 C1(CC(=O)N)COCC(C)(C)O1.Cc1nc(C(=O)N(C2CCCC2)CC)sc1C C1COC2(CCN(C(=O)C3=C(Cl)CCOC3)C2)C1.Cn1ncc(C2CC2)c1C(=O)N Cc1cc(C(N2CCC(C)(CNC(c3cc(Br)n(C)n3)=O)C2)=O)c(C)n1C C(=O)C(CO)C(C)(C)C.N1(C(c2cc(OCC)no2)=O)CCCC(O)(C)C1.N c1(C(N2CCC(CCNC(C(CC)n3cncn3)=O)C2)=O)cc([N+](=O)[O-])cn1C C1(F)(C(=O)NC(C#C)C(C)OC)CCN(C(C2CCCN2C(C)=O)=O)CC1 C1(CN)CCC(CNC(C2CC23CC(O)C3)=O)CC1 C(c1cccnc1)=C(C)C(=O)NC(C1CCCCC1)CNC(C1CCNC1=O)=O c1(CC(=O)NC(C(=O)NCC(CC)OC)Cn2ccnn2)ncccc1F c1(C(=O)NC(CCCNC(Cn2ncc(C)c2)=O)C)cc2c(F)c(Cl)ccc2[nH]1 N1(C(CC2(C#N)CCOCC2)=O)CCCC(O)(CNC(C2CCC(=O)N2)=O)CC1 c1(OC(C)C)ccc(CC(=O)NCCOCCN(C)C(C2CC2)=O)cc1 C12(C(N3C(C(C)C)CCC3)=O)COCC1CN(C(=O)CC1CC(C3CC3)C1)C2 Cc1cnc2n1CCC(NC(=O)C(=O)NC1CCN(c3ccc(F)cc3)C1=O)C2 C1(NC(c2cc(-c3ccc(F)c(F)c3F)on2)=O)CCC2CCCCC2C1 N1(C(C(C(C)C)F)=O)CC2(CCN(C(=O)CS(=O)(=O)N3CCCCC3)C2)C1 CCC(C)(CC)C(=O)NCC12CC(CO1)N(C(c1cc(C#N)c[nH]1)=O)C2 CN1CCN(C)CC(C(=O)NCC2CCN(C(=O)CN3CCCC3)C2)C1 C(C(C)(C(=O)NCC(O)C1CCC1)NC(=O)CC1CCOC1(C)C)SC CCS(=O)(=O)c1ccc(NC(=O)C(N2CCCC(c3cccc(Cl)n3)C2)=O)cc1 c1(C(=O)N)cccc(C2CC2)c1.CC1(CC(=O)NC2CCCC2C)CC1(Cl)Cl N1(c2snc(CCC)n2)CCCC12CC2.C(=O)CC(F)(F)F.C(=O)(C=CC)N c1(CNC(=O)CCN2CCCC2C(N2CCCCC2)=O)cccnc1 C(C(=O)N=c1cc(C)o[nH]1)c1[nH]c(=NC(CC(C)NC(=O)OC)C)[nH]c(=N)n1 CC(C)C(O)CC(=O)NC1(CCNC(=O)CC2(O)CCOCC2)CCCC1 C1(n2cc(C(C)O)nn2)CCCN(C(=O)NC2CCSCC2)C1 C1(C(N2CCC2)=O)CCC(=O)C1.C1(OC)CC(C=O)C1.C(=O)CC.CC.N N1(C(c2c(C)nn(CC)c2C(F)F)=O)CCC2(CCN(c3ncc(F)cn3)C2)C1 C(C)(C)(CCC(=O)NCC1COC(C)(C)C1)NC(c1c(CC)n(C)cc1)=O Cc1cc(C(N2CC(F)CC2CC(=O)NC(C)CCCO)=O)cc(O)c1 N1(C(CCCC(=C)C)=O)C2CCC(C(=O)Nc3cnccc3C)C1CC2 CCCC(C(=O)NC1CN(C(c2cccc([N+](=O)[O-])c2)=O)CC1(C)C)C(C)C N1(C(C(CC(C)C)ONC(C2CC23CCOCC3)=O)=O)CCCC2C1CCN2C Cc1ccc(CC(N2CCC(C(C)NC(=O)C(C(C)O)N(C)C)CC2)=O)c(F)c1 C(=O)(CC(C(F)F)n1ccnc1)NCC(C)NC(C(C)OCCC(C)C)=O CC1(NC(=O)C(O)Cc2cnc[nH]2)CCN(C(C2(CF)CC2)=O)C1 CC1CC(=O)c2c(N3CCN(C4CCCCC4(C)O)CC3)ccc(F)c21 C=C(C)CCCC(=O)NCC(CC(F)(F)F)NC(=O)CCCNC(=O)COC N1(C(c2cnc(-c3cccs3)s2)C(=O)NC2CCOC2)CC2NC(=O)OC2C1 C(=O)(C(=O)C(C)(C)C)N.c1(OCC=C)ccc(C(N2CCCC2C)=O)cc1 C(=O)(C(CCSC)OC)N1CC(CC(C)NC(c2cc(CC)on2)=O)C1 Cc1cc(C(=O)NCC(C)=CC(=O)NC2CC(C)(CO)C2)ncc1N c1(C(C)=O)cc(NC(C2(C)CC(NC(=O)C(C)n3cncn3)C2)=O)ccc1C CCC(C)CCC(=O)NCc1nnn(C)c1C(=O)NCC1CC1Cl Cc1ccc(C(N2CCC(C)C(NC(=O)CN(C)C3CC3)C2)=O)cc1C#N C1(CCNC(CN(C)C(=O)C2CC2)=O)CC(C(=O)NC2CC2(C)C)C1 CCC(C(=O)NCCCC(=O)NCCc1ncn(C)n1)OC c1(C(=O)NCC2OCCN(C(c3scc(C)c3C)=O)C2)cc(=O)ccn1C C1(NC(CC(C)C2CC2)=O)CC2(CCCN(C(=O)CC3=CCCCC3)C2)C1 C(=O)(C(O)CCNC(=O)CCC1CC1C)N(CCCN(C)C)CCC C1(C(N(CC=C)CCO)=O)(NC(C2CCC(CC)O2)=O)CC1(C)C c1(C(=O)NCC(CCC)NC(c2ccsc2OC)=O)nccnc1OC N1(C(C(N2C(C=C)CCCC2)=O)CCC)C(=O)C2C3CCC(O3)C2C1=O CCCCCC(CC)C(=O)N(C(C)CC(=O)NC(C1CC1C(=O)OC)C)C C(CC(C)C(=O)NC(CCN(C(=O)C=NOC)C)c1cccs1)=CC C1(C)CCCN(C(=O)C(=O)NCC)C1.N1(CCOC)CC(C(=O)O)CC1=O CCC(CC(F)F)C(=O)N1CCN(C(=O)COCC(F)(F)F)C(CCO)C1 c1(OC)cc(C(N2CCC(C(C)C(N3CCCC3CC3CCC3)=O)C2)=O)ccn1 C1(C(N2C3C(NC(c4cc(C)c(O)nc4)=O)C(C3)C2)=O)CCCC2CCCCC12 c1(C(C)NC(C(CC=C)CC=C)=O)ccc2c(c1)CN(C(=O)CC(C)N(C)C)C2 C(C(C)C(F)C(=O)NCc1cnn(C)c1C)NC(CN1CC(C)(OC)C1)=O C1(N(C(Cc2cc(C)on2)=O)C)CCCCN(C(=O)C(F)(F)C(C)O)C1 N1(C(CCSCCCC)=O)CCCC(NC(C2CCNC2=O)=O)C1CC c1ccc(F)c(Br)c1.Cc1cc[nH]c1C(=O)NCC1(O)CN(C(=O)CO)C1 Cc1ncc(C(N2CCC(C)C2)=O)c(C(C)C)n1.c1(C=O)ccc(C2CC2)o1.N N1(C(=O)CC2C=CS(=O)(=O)C2)CC2CCCC(C1)N2C(C1CC12CC2)=O N1(C(CCCCSC)=O)CC2(CC(C(=O)Nc3cnccc3C)CO2)C1 c1(CC=O)ccccc1.C1(CC=O)CN(C(=O)C(=O)C2CC2)CCO1.CC.O C1(C)(NC(COCC=C)=O)CC(NC(c2coc(C(C)(C)C)n2)=O)C1 c1(C(=O)NCc2cccc(OC)c2SC)ccccc1N=c1ccn(C)[nH]1 C1(NC(COCC=C)=O)CC2CN(C(=O)Cc3c[nH]nc3C)CCN2C1=O c1(-c2cc(C(=O)O)cc(Cl)c2)ccc(S(=O)(=O)N2CC=CC2)c(Cl)c1 C(CCCC(=O)N1CCC(CC(C)NC(C2CCCCN2C)=O)CC1)OCC Cc1oc(C(C)C)cc1C(=O)NC(C)CC(C)C.C1(C=O)(C(F)F)CCCO1 c1(CN(CCCN(C(C(=O)NCc2ccco2)C2CCSC2)C)C)ccccc1 N1(C(c2c(OC)csc2)=O)CC2CCN(C(C3CC(C)(C)CCO3)=O)CCC2C1 N1(C(C2(C)COC2)=O)CC2CN(Cc3ccc([N+](=O)[O-])cn3)CC2C1 O=C(CC=C(Cl)Cl)Nc1cccc(NC(c2nncs2)=O)c1 N1(c2ccnc(C)c2N)CCc2ccc(Oc3ccccc3)cc2C1 c1(C(=O)NCC2CN(C(COCCCOC)=O)C2)cc(OC)no1 C1(C(=O)NC(CNC(Cc2c(F)ccc(C)c2)=O)C)CCn2nnnc2C1 C1(CCCC)CCC(c2nnnn2CCSC)(NC2CC(CO)C3CC23)C1 c1(C(N2CCC(C)C(NC(C3(CCF)CC3)=O)C2)=O)cc2ncccc2[nH]1 Cc1nccnc1-c1cn(CCCNC(=O)C(c2ccccc2Br)(F)F)nn1 CCC(C)CCCCC(=O)NC1CC2CCC1N2C(=O)C=Cc1cccs1 N1(C(C(C2CCC2)NC(c2c(OC)cccc2)=O)=O)CC=C(C(C)(C)C)CC1 c1(N2CCC(=C)C2)nc(N2CCOCC2)nc(N2CCC(OC)CC2)n1 c1(N(C)C)cncc(NC(C2OCCC2C)=O)c1.C(=O)(C(C)(O)C1CCC1)N c1(C=O)cc(-c2ccncc2)[nH]n1.C1(C(N(C)CCOCC)=O)COC(=O)C1 C(=O)(CC(C)(C)C)NC1(C(=O)NCC=C2CCSCC2)C(C)C1 Cc1nc(C2CC2)sc1C(=O)N(C(C)CN(C(=O)C(O)C1CC1)C)C N1(C(C2N(C)CCCC2)=O)CCC2CCC(C1)N2C(C1(CO)CCC1)=O C(CC(C)(C)C)(C(=O)N(C(CO)CO)C)NC(C(C)C(F)(F)F)=O c1(C(=O)NCCCCNC(c2cccnc2-n2ccnn2)=O)cc(O)cc(F)c1 CC1CCC(NC(c2cnn(C3CC3)c2)=O)CN1C(=O)CCCN1CCOC1=O N1(C(c2ccncc2)=O)CCC(C2(Nc3nc(Cl)ncc3Br)CC2)CC1 C1(CC)CCc2o[nH]c(=NC(=O)Nc3ccc4ccccc4c3C)c2C1 CC(C)C(CS(=O)(=O)N1CCN(C(C2CCCN2)=O)CC1)C(C)C c1(C(N2CC(OCCNC(C(c3ccccc3)C)=O)C2)=O)cnn2c1OCCC2 N1(C(C(F)OC)=O)CCCC1(C)CNC(c1cccc(C(C)C)n1)=O c1(CC(C(=O)N)O)c(F)cccc1Cl.C(CCCC)NC(CN(C(=O)OC)C)=O C=C(C)CCC(=O)NCC(C1CCCCN1C(c1cncc(Cl)c1)=O)(C)C C1(CNC(CCSCC)=O)CN(C(c2cc(CC)nn2C)=O)C(C)(C)C1 CC1(C)C(CC(=O)NCC2CC2Cl)CCN1C(c1ncc(F)cc1N)=O c1(CC)c(C(=O)NCC2CC(OC)CN2C(c2c[nH]cc2C)=O)nnn1C CC(C)CCC(O)C(=O)N(C1(CC(N2CC(O)C(C3CC3)C2)=O)CC1)C c1(C(N(CC(O)CN(C)C(C2CC2(C)Br)=O)C)=O)cc2nn[nH]c2cc1F C1(C(=O)NC(c2ccc(C)cc2)C)(CC)CCCN1C(=O)C1=CCSC1 C1(O)(CCNC(COCP(C)(C)=O)=O)CCCN(C(c2ccccn2)=O)C1 N1(C(C(CN)c2ccccc2)=O)CC2CC1CC2N(C(=O)C(=O)O)CC=O.C C1(CC(N2Cc3c[nH]nc3C2)C(=O)NC2CCOC2)CCCCC12CC2 CN1CCN(C(c2cncc(Cl)c2)=O)CC1C(=O)NC(c1cncn1C)CO c1(C(=O)NCC(C)NC(c2ccc(C(N)=O)o2)=O)n[nH]c(C(C)(C)C)n1 C1(C(=O)NC23C(CN(C(C4CCCN(C)C4)=O)C2)C3)C2CC(F)(F)CC12 CCCC(C)(C)CC(=O)NCC1CC(F)CN1C(C1(C2CCCO2)CCC1)=O c1(C(N2CC(NC(C3(CC=C)CCCC3)=O)C(O)C2)=O)cnc2c[nH]nc2c1 C=CCCC(F)(F)C(=O)N1CC2CC(C(=O)NCC)C(C2)C1.c1cc(C)nn1C.C n1(CCC(=O)NC23C(CN(C(C(C(C)(C)C)=O)=O)C2)C3)c(=O)oc2ccccc12 C1(N(C(C(C2CN(C(C(CCSC)O)=O)C2)O)=O)C)CCCC(C)C1C C1(CC(=O)NCc2n(C)nnn2)N(C(c2nonc2N)=O)CCC1(C)C c1(CNC(c2c(CC)cncc2)=O)n[nH]c2c1CN(C(c1ccsc1C)=O)CC2 Cc1cc(C)c(C(=O)NCCn2cc(C(=O)NC(C(C)C)C3CC3)cn2)o1 c1(C(N2CCC(CCC(=O)NC(C)CCCO)C2)=O)cc(Cl)n(C)n1 C1(c2n(CC(=C)C)nnn2)(NC2CC(CCO)C2)CCCN(C)C1 N1(C(CCCCSC)=O)CCN2CCN(C(C3CCOC(=O)CC3)=O)CC2C1 c1(C(=O)NC2CC(NC(C3C(CC)C3)=O)C2)cccc2cc(O)ccc12 c1(C(=O)NC2(C3CN(C(CCC=C)=O)C3)CC2)cc(C)nc2ccccc12 C1(NC(C2C(NC(COC(C)=O)=O)CC2)=O)CCCC1.CCN(C)C.C CC1CCCC(NC(C2CCN2Cc2ccn(C3CCCC3)n2)=O)C1 N(C1CCc2c(Br)cccc21)C(=O)COc1ncccc1OCC(F)F c1(C(=O)NCC2N(C(CCNC(COC)=O)=O)CC2)cc(Br)nn1C Cn1ncc(Cl)c1C(=O)NC1CC1CNC(=O)C(c1ccc(F)cc1)O CCC(C)C(=O)C(=O)N(C(CC)CC(=O)N(c1ccc(O)cc1C)C)C C1(C(N2CCC(NC(C3(C)CC3)=O)C2)=O)(OC)CCCCCCC1 N1(C(c2ncn(CC)n2)=O)CCC(NC(C2OCCO2)=O)C(C(C)C)C1 c1(C(N2CCC(CF)C2)C(=O)NCC2CC2)cccc(-n2cncn2)c1 N1(C(C(CNC(=O)C(F)C(F)(F)F)OC)=O)CC2(CCOC2=O)C1 c1(C(=O)NC(c2ccc(Br)cn2)C)sc(-c2ccccc2)nc1C(F)(F)F C(=O)(C(C)C(O)CC(C)C)NC1(COC)CN(C(CCSCCCC)=O)C1 C1(CNC(C(C)CC2CCC2)=O)CCCCN(C(=O)CC#N)C1 Cc1cccc(Cl)c1NC(C1CCN1C(c1cccc(Br)c1Br)=O)=O N1(Cc2cc(OC)c(C#N)cc2)CCC2CN(C(=O)C(O)C(C)C)CCC12 C1(CC(=O)NCC=Cc2ccccc2)CCCC(NC(=O)C(O)C2CC2)C1 CCCCCC(O)C(=O)N1CCC(C2CCCN2C(=O)C=Cc2cc[nH]n2)C1 C1(O)(CC(=O)NC(CN(C(C2(C#C)CCC2)=O)C)CC)CCCOC1 C1(C(=O)NC2C3CC2N(C(C2CC(OC)C2)=O)C3)(OC)CCCC(C)(C)C1 C1(NC(C2N(CCC)CCCC2)=O)CC(F)(F)CC1NC(c1ccc[nH]1)=O.C c1(NC(C(Cn2cccn2)NC(c2cc(C)on2)=O)=O)ccc(O)cc1 c1(C(=O)NC2CC3CN(C(c4ccc(CC)s4)=O)C2C3)ccc2c(c1)ncn2C C(=O)(C1CCCc2cccnc21)N1CC(CNC(c2cc(C3CC3)ccn2)=O)C1 N1(C(c2n[nH]c(CC)c2Cl)=O)CC2CC(NC(=O)CC3(C)CC3)C1C2 Cc1cncc(C(=O)N(CC(C)CNC(c2cnn(C)c2F)=O)C)n1 C1(NC(CCCC=C)=O)CC2CC1N(C(c1csc(-c3cccc(Cl)c3)n1)=O)C2 N1(C(c2ncc(-c3cccnc3)s2)C(=O)NCC(C)C)CCS(=O)(=O)CC1 CCCCCCC(F)C(=O)N1CCCN(C(=O)C(c2c(C)n[nH]c2C)C)CCC1 C1(C(C)(C)O)(Cc2ncc(Cl)cn2)CCN(C(=O)Nc2cc(C3CCC3)no2)C1 Cc1ccc(C(=O)NC2CC2NC(C2CC2c2cccc(Br)c2)=O)cc1C#N C1(CNC(c2cc(C)n(C)c2)=O)(CNC(=O)C)CC2CCCC2C1.CCC#N c1(OC)cc(OC(c2cn(C)c3cnccc23)=O)ccc1[N+](=O)[O-] C1(NC(C(C2CCOCC2)OCC)=O)CN(C(c2scc(C)c2C)=O)CC1F N1(CC)CCOC(C(=O)NCC(O)CCNC(=O)C(c2cnccc2C)(C)C)C1 C1(NC(c2c(C)ocn2)=O)CC2CN(C(=O)C(C)Oc3ccc(F)cc3)CC2C1 C(=O)(C(CNC(C1CCCC(=O)C1)=O)C(C)C)N(C)Cc1n(CC)cnn1 S(=O)(=O)(c1sccc1I)NCCC(=O)NC(C1CCCO1)C N1(C(CCSC)=O)CCN(C(=O)C(C)C)C(CC(C)(C)C)C1 Cc1ccc(OC(C)C(=O)NC2CCCN(C(c3nnn(C)c3C)=O)C2)cc1 C=CC1(C(=O)NCc2cncc(Cl)c2)CCN(C(c2cc(CO)[nH]n2)=O)C1 C=C1CC(C(=O)NCC2CCNC2=O)(NC(=O)OC(C)(C)C)C1 C(=O)(C(C)CCCC(C)=O)NC(CC(=C)Cl)C(=O)NCC1(O)CCCC1(C)C N1(C(c2cnc(C)s2)=O)CCC(C2(O)CN(C(=O)CC3CCC(C)C3)C2)CC1 c1(CC(=O)NCc2nc(C)cs2)cc2ccccc2o1.C1(CC=O)CC12CC2 c1(C(=O)NCC(CN(C)C(c2scnc2Cl)=O)O)cccc(C(F)(F)F)c1N C1(CNC(CC=C=C)=O)CCN(C(=O)C(C)CCOC)CCC1(F)F C1(NC(=O)C(F)C2CCCC2)CCCN(C(c2cc(O)ccc2F)=O)CC1 N1(C(CSCC#C)=O)Cc2[nH]nc(C(=O)NCC(C)(C)C(C)O)c2C1 C(=O)(N=c1[nH]oc2cnccc12)C1N(C(c2c(C)n[nH]c2)=O)CCSC1 c1(CC(=O)N(C)CC)nnc(O)c2ccccc12.C1(C=O)CCCC1C(=O)O.N N(C1CSc2ccccc21)C(c1cccc(OCc2ccccc2)c1)C N1(C(CCSCC)=O)C2CCC1CC(Cn1cc(-c3cnn(C)c3OC)nn1)C2 C1CN(C(=O)Cc2cnccc2C(F)(F)F)C2CC12.c1(C=O)ccc(F)cn1.N c1(C(N2C(C)CCC(C(N(CCCC)CCCC)=O)C2)=O)cccc2c1C(=O)NC2 N1(c2n(N3CCC(Cc4ccc(O)c(C)c4)C3)nnn2)CCCC2(CCCC2)C1 CCC(C)(C)C(O)C(=O)N1CCC(C(=O)Nc2ccccc2)C1 C1(CC(N2CC(O)(C(C)C)C2)=O)CCCN(C(C2CC(C)(C)CO2)=O)C1 C=C(C)CC(C(=O)NC1CC12CCOCC2)NC(c1cc(C)no1)=O c1(CCC(=O)NCC2CCN(CCF)C2)cccnc1 c1(SCCCC(N2CC(NC(C=CC)=O)C(CO)CC2)=O)nc2ccccc2s1 N1(C(C=C(CCC)CCC)=O)CCC(c2cccc(Br)c2)(C(C)(C)C)CC1 N1(C(c2c(CNC(CC=CC(C)(C)C)=O)noc2)=O)CCCCC(CO)C1 C1(CC=C)(C(=O)NC(c2nc[nH]n2)CC)CCCN1C(c1nn(C)cc1Cl)=O N1(C(CC(=O)NCC)=O)CC2CCC1CC2NC(=O)C(C(C)(C)C)OC c1(N2CCCC(C(=O)NC)C2)nc(C)cc(=NCC2CC(O)C23CCC3)[nH]1 Cc1cc(OCC(N2CCC(C3CC(N)CCO3)CC2)=O)ccc1-n1ccnc1 c1(CC(N2CC(NC(Cc3n(C)ncc3)=O)(CO)C2)=O)nc2ccccc2s1 c1(NC(C2CC(O)CN2Cc2cnc(Cl)cc2Cl)=O)ncc(F)cc1Cl N1(C(c2c(Cl)nsc2Cl)=O)CCC2C(CCCN2C(=O)CCc2cnccn2)C1 N1(C(C(CCC)C)=O)CCC(NC(C2(O)CCC2)=O)C(CO)CC1 C(=O)(CC(C)(C)C(F)F)NCCOCCNC(c1cnn(C)c1F)=O CCC(C(=O)NCC1(C)CN(C(c2cccc(F)c2NC)=O)CCO1)C(F)(F)F N1(C(C(CCCOC)NC(C2CC(C#N)(OC)C2)=O)=O)CC2(C1)CC(C)(C)C2 C(=O)(C(C(C)C)c1ccncc1)N1CCCC1.C1(C)(C=O)CC(C(=O)OC)C1.N C1(NC(C2C(C(C)(F)F)C2)=O)CCC12CCN(C(c1cocc1Br)=O)CC2 C1C2CN(C(=O)Cc3ccc(Cl)cn3)CC12.C1(C(=O)N)CCOC1C1CC1.C c1(CC(=O)NC2CN(C(=O)CN3CCCCC3=O)CC2F)cc2cc(Cl)ccc2[nH]1 Cc1cc(C(N2CC3CCC3(C(=O)NOCC(O)C(C)C)C2)=O)cc(O)c1 c1(SC)ncc(Br)c(=NCC2CCN(c3nc(O)cs3)CC2)[nH]1 C1(NC(CN(S(C)(=O)=O)C)=O)CCCC1C.c1(C(=O)N)csc(=N)[nH]1 N1(C(C(CCC)C)=O)CCC(C2=NOC(C(=O)OCC)C2)CC1 c1(C(=O)NC2C(CNC(C(C)OCC)=O)C2)cc2cc(Br)ccc2o1 c1(OC(C)=O)ccc2c(OCC#CC3CCCCO3)cc(=O)oc2c1 C(=O)(CCN(CCC)CC)N.CCC=O.C(C)C.C(C)=O.CCN(C)C Cc1ccnnc1C(N1CCC(CC(C)NC(=O)C(C)C#N)CC1)=O N1(C(C2(C(C)C)CCCN2C(C2CCCN(C)C2)=O)=O)CC2(CCCO2)C1 C1CN(C(=O)Cc2ccn(C)n2)C2CC12.C1(C(=O)N)(NC(C)=O)CCC1 N1(Cc2c(CC)noc2)CC(NC(c2cnc(OC)c(C)c2)=O)C(C)(C)C1 N1(C(=O)C=Cc2ccsc2)CC2CN(C(C3CC(C(F)F)C3)=O)CC2C1 N1(C(=O)NC(C#C)CC2CCC2)CC2CCC2(C(=O)O)C1 N1(C(c2cc(OC)ns2)C(=O)NCCC2(C)CC2)CCc2cccc(C)c21 c1(CC(=O)NC2CN(C(C(C(CC)O)(F)F)=O)CC2C)ccc2oc(O)nc2c1 c1(NC(C2CCCCC2)C#C)cc(C)c(OCCCC)cc1C N1(C(C(n2cnc([N+](=O)[O-])n2)C)=O)CC2CN(C(=O)CC(=O)N(C)C)CC2(C)C1 Cc1cc(Br)c(CN2CC(NC(=O)C=Cc3cnccn3)C(F)C2)cc1[N+](=O)[O-] C(=O)(CC1=NNC(=O)C1)NCCCCCNC(c1cc(C)c(N)cn1)=O C1(NC(C2CN(C)C(=O)N2)=O)CCC(O)CN(C(=O)Cc2ccc(C#N)cc2)C1 C=CCCCCC(=O)NCC(C1CCN(C(=O)C=Cc2ccc(C)cc2)CC1)F N1(C(CNC(C)=O)=O)C(CNC(C2CC3CCC2C32CC2)=O)CC2COCC12 c1(NC(c2c(CC)c[nH]n2)=O)cccc(NC(C23CCCC2C3Br)=O)c1 C1(NC(c2cccc(NC(CC)=O)c2)=O)CCCCCN(C(=O)C(C)OCC)C1 c1(C(=O)NCC(C(C)C)NC(C2CCC(=O)CC2C)=O)c[nH]c2ccccc12 c1(C(N2C3CCC2CC3)=O)cc2c(s1)CCS(=O)(=O)C2.c1(C(=O)N)cn[nH]c1 N1(C(C2(CCCC)CC2)=O)CC(C)(OCC(N2CCC(C)C2)=O)C1.C1CCC1 S(=O)(=O)(c1cnccc1N1CCC=C(Br)C1)NC(COCC)C CC1(C)C(C(N2CCC2CF)=O)CCN1C(=O)CCC1CCCOC1 C=Cn1ccnc1C(c1nnnn1CCC1CC1)NCC(CC(C)C)OC C(=O)(C1=CC2(CCOCC2)C1)NC1CC(C)(C)CN(C(=O)C(C)(O)C2CCC2)C1 Nc1ccc(C(=O)NCC2CCCCN2C(C2CCSC2)=O)nc1Cl N1(C(Cc2cccc(OC)c2)=O)CCC(NC(=O)CCN2CCC2)C(F)C1 CCCCCC(C)CC(=O)Oc1nnc(CSC(C)C(=O)Nc2ccccc2)s1 C(=O)(C(C)(C)C)NCCOC.C1CCN(C(=O)CCC2(C)CC2(F)F)C1 Cc1cccc(C(=O)NCCC(O)CNC(C2CSCCS2)=O)n1 n1(CCC)ccc(=NC(=O)C2CC(NC(=O)C(CC)CC(C)C)C(O)C2)[nH]1 N1C(CC(C(=C)Cl)(C)C)=CC=CC=C1[N+](=O)[O-] C(=O)(C1CC(=O)c2ccccc21)NC1CC(C)(C)CN(c2nc(Cl)ncc2Cl)C1 c1ccc2c[nH]nc2c1.c1(OCC)ccc(CNC(C23CC2CN(C)C3)=O)cc1 N1(C(CC2(CSC)CC2)=O)CCC2CN(C(=O)C(C)(C)c3nncn3C)CCC12 C(C)(CO)(CS(C)(=O)=O)NC(C1C(c2cn(CC(C)C)nc2)C1)=O C1(C(c2n(CC)nnn2)NCC2(CC)CC2)CC12CCOCC2 C1(CNC(Cc2c(C)con2)=O)CN(C(C2C(C#N)C2(C)C)=O)CC1O N1(C(=O)Cn2cccn2)CC2(CCCCN2C(=O)C(F)(F)c2cscn2)C1 C1(NC(C2CC(C)OC2)=O)COC2(C1)CN(C(c1ccc3ocnc3c1)=O)C2 CON(CCC(=O)NCCc1ccccc1O)C(=O)CC(C)n1cccc1 N1(C(CC2CC(C)(C)C2)=O)CCC2(CCC(CNC(=O)C(F)(F)CO)O2)CC1 C1CN(C(c2ccc(C(F)(F)F)cn2)=O)CC1C.c1(OCC)cc(C=O)[nH]n1.N O=C(C(O)CC(F)(F)F)NC1CCC12CCN(C(=O)Cc1sc(O)nc1O)C2 c1(C(C(=O)NCCC)O)ccc(O)cc1.CC C1(C)(COC)CC(NC(c2csc(C)c2)=O)CN1C(c1cn(C)cc1C)=O C(=O)(CC(O)C(C)C)N1C(CN(c2ccnc(C(CC)C)n2)C)CCC1 c1(C(=O)NC(CC(C)NC(c2c(CC)non2)=O)C)c[nH]nc1C(C)C.C c1(C(=O)OC)ccc(NC(C2CCCCC2)=O)cc1I.C12CC(C1)NC2=O.S CN=c1[nH]c(C(N2CCCC2CCCNC(c2cccc(=O)[nH]2)=O)=O)cs1 c1(C(CNC(Cn2cc(CN(C(C)=O)C)nn2)=O)=O)ccc(F)cn1 c1(C(=O)O)ccc2c(c1)S(=O)(=O)NC2.C(C(F)(F)F)N(C(=O)C)C(C)C C1(O)(CC(N2C(CN(C(=O)C(C)c3ccsc3)CC)CCC2)=O)CCCCC1 C=Cn1nccc1C(N1CC=CC1CNC(=O)C(c1cccnc1)O)=O c1(CC)ccccc1C(=O)NCC(C)(CNC(C1CCCC1(C)C)=O)OC c1(NCC2C(CC)C2)ccc(C)o1.N1(C(C(N2CCC2)=O)C)CCOC1=O CC1CN(N2CCN(c3c(-c4nn[nH]n4)cccc3F)CC2)CCC1N(C)C N1(C(c2c(C(C)=O)coc2)=O)CCC(C)C12CC2.C(=O)CCC(C)CN(C)C.N C(CC(CNC(=O)CC1(OC)CC1)NC(=O)CCC1(C)CC1)OC c1(C(N(C2CN(C(=O)CCc3cncs3)C2)C)=O)cccc(N2CCOC2=O)c1 C1(NC(C2CCN(C)C2)=O)CCSC12CN(C(c1ocnc1C(F)F)=O)C2 C1(CCNC(C2(OC)CCOC2)=O)CN(C(=O)C(C(C)C)N(C)C)CCO1 c1(-c2ccc(C)o2)nc(=NCc2ccccc2CNC(=O)CO)s[nH]1 C1(C(=O)NC(c2cnc[nH]2)C)CCC2(CCN(C(c3sccc3F)=O)CC2)C1 N1(C(c2cc(OC)no2)=O)CC23CCCC2(C1)CN(C(C1C=CCS1)=O)C3 N1(C(C2CCC(OC)CC2)=O)CC2CCCC2(C(=O)N(C2CCCOC2)C)C1 C1(C(=O)OC)CC2(CCN2S(=O)(=O)Cc2cccc(C)c2C)C1 C1(OC)CC(C(=O)O)N(C(=O)C(N2CCCC(c3nc[nH]n3)C2)=O)C1 O=Cc1cccc(-c2cc(C(=O)OCC(C3CC4CCC3C4)=O)on2)c1 C1(N(C(C23CCC(OC)C2C3)=O)C)CCCC2CN(C(C3CCCC3F)=O)CC12 c1(C(N(CC(CN(C(C(CC)CO)=O)C)O)C)=O)cc(F)cc(Cl)c1N C(C(N=c1cc[nH]c(=NCCCc2ccccn2)[nH]1)C1CC1)c1cccc(C)n1 CN1C(=O)CC(NC(=O)C(=O)NCC2(c3ccc(C#N)cc3)CC2)C1=O C1(NC(=O)NCCc2ccc(CN3CCCCC3)cc2)CCC2CSCC12 C(=O)(C1=CCN(C(=O)C(C)SC)CC1)NCCC1CC(SC)C1 c1(OC)ccccc1C(C)=CC(=O)NC(C)C(CO)Nc1ncc(C(F)F)cn1 C1(C#N)(CC(=O)N(CC(C)NC(C(C)C#N)=O)C)CCCCC1 C(=O)(C(CC1CCCCC1)N(CCCO)C)NCCCSC C=CCCCCCCCCC(=O)N1CC(O)(C(C)NC(=O)C(C)(F)F)C1 Cc1ccc(NC(C2(C)CCN2C(=O)Cc2cccc(Cl)n2)=O)cc1Cl c1(C(N2CCCCC(NC(C3CC3C3CCC3)=O)C2)=O)cnc2[nH]ccnc1-2 C1(C(N2CCN(C(CCCC)=O)CC(O)C2)=O)Cc2nn(C)cc2C(=O)N1 n1(CC)nnnc1C(c1ccc(SC)o1)NCC1(CCO)CCOC1 C1(C(N(CC(O)CC(C)(C)C)C(C)C)=O)Cn2ccnc2NC1=O Cc1ccc(CN2CCC(O)(C(=O)NCC3CCOC3)C2)c(F)c1F N1(C(c2cc(-c3ccccn3)no2)=O)CC2CC(CO)(CO2)C1 C(CC(C)C)(C(=O)N1CCCC(NC(=O)C(C)(C)Cc2ccccc2)C1)OC CCC(C)C(CC(=O)NCC(N1CCCC1)C)NC(c1cc(C)on1)=O C1(NC(C2CC(=C)C2)=O)COCCC1NC(=O)C(F)(F)c1cscn1 C(=O)(C(F)(CNC(=O)Cc1ccsc1)C(C)C)NC(C#C)C1CC1 C(=O)(C(C)(C)C(=O)NCCCCC)N(C)C.C(=O)(C(Cc1ccsc1)NC=O)N N1(C(C2(C(C)C)COC2)=O)CC(C)C(O)C1.c1(CCC=O)nc(C2CC2)no1 C1(=O)CC(C(F)(F)F)O1.C1(NC(=O)OC(C)(C)C)CCCCC12CCC2 C1(O)(CNC(c2c(C)ocn2)=O)CCN(C(c2cc(C(F)F)ncn2)=O)C1 N1(C(c2c[nH]nc2Cl)=O)CC=C(C(=O)N2CCCC(O)(CO)C2)C1 C=CCCCCCC(C)C1CCN(CC(F)(F)F)CC1.c1ccncc1F N1(C(CCCC)=O)CC(CNC(c2[nH]nc3cnccc23)=O)C2(CCOCC2)C1 c1(OC)ccc(C)cc1C(=O)NC1C2CN(C(=O)C=Cc3sccc3C)CC12 c1(C(N2CCC(NC(CCC)=O)C(C)C2)=O)cc2c(F)ccc(F)c2[nH]1 N1(C(C2C(OCC)C2)=O)CC2(CCN(C(c3cc[nH]c4nccc3-4)=O)CC2)C1 Cc1nc(C)n(CC(=O)NC(C)CNC(C2CC2c2cccc(Br)c2)=O)n1 CCCC(C(=O)NCC1CCCN1C(c1cccn1C1CCCC1)=O)OC CCC(CC(=O)N1CC(CO)(NC(c2cc(-c3cccs3)on2)=O)C1)C1CCC1 N1(C(c2c(O)cc(C)nn2)=O)CCC(C)N(c2ncncc2Cl)CC1 C(=O)(CC(C)(C)C)N.Cc1cc(C(=O)NC(C)(C)CCNC(=O)C)ns1 CCCC(CC)CC(=O)N1CCN(C(=O)CCCC(=O)OCC)C(CF)C1 c1(C(=O)NC2C(CNC(c3cc(C)[nH]n3)=O)C2)ccncc1F C1(C(=O)NC(CC(C)NC(CCC=CC(C)C)=O)C)CCCCN1N=O C1(NC(CCCOC)=O)CCCCCC1NC(N1CCOCC1)=O C1(C(N2CC(CNC(Cn3c(C)ccn3)=O)C(O)C2)=O)OC(C)(C)OC1(C)C CC(CC(=O)NC1CCOCC1NC(C1C2CCC1CC2)=O)C(F)F c1(C(=O)NC2CC(CNC(C3CCC(F)C3)=O)C2)ccccc1CO C1(C(=O)N)CCN(CCO)C(=O)C1.C1(C(C)C)(C(=O)NCCC)CNC(=O)C1 Cc1cc(C(=O)NCCC2CCCN2C(=O)CO)cc(Cl)n1 C1(CNC(c2n(CC)ncc2)=O)CN(C(C2CC2Br)=O)C2(CCC2)C1 N1(C(c2cc(C)cc(C)n2)=O)CC(NC(C2C3(CC3)C23CC3)=O)CC12CCOC2 C1(C(=O)N)C2C3CC4C1C1C2CC3C41.C1(CC)CCC1.n1(CC=O)cnnn1 N1(C(c2ncc(C)cn2)=O)CCN(C)CC1CNC(=O)CC1CCOCC1 Cc1nn(C)c(=O)c(C(=O)NC2CN(C(=O)Cn3ncnn3)C3CC23)c1C c1(C(=O)NC2C(C)N(C(c3cn4ccccc4n3)=O)CC2)n[nH]c2c1CSCC2 c1(CNC(C(=O)N(C)C)=O)cccc(-n2cc(C3CCC(C(=O)O)CC3)nn2)c1 c1(C(=O)NC(C(=O)OC)C2(C)CC2)cc(F)ccc1NC(=O)NC C1(C(=O)NC2CC2c2ccco2)CC2CC2N1C(=O)COC.C1CCC1 CC(CC(=O)NCC1CCC1NC(c1cncc2n[nH]cc12)=O)C(C)(C)C C1(C(=O)NCCCC2CCN(C(C3=CC(C)(C)C3)=O)CC2)OCCOC12CCC2 CC(C)CCC(=O)NC(C1CCCCC1)C.C1(C(=O)N)CCCN(S(C)(=O)=O)C1 N1(C(C=COCC)=O)CCOc2ncc(-c3cc(C)ccc3OCC)c(C)c21 c1(C(=O)NCC(CO)NC(=O)C(O)CC(F)(F)F)cc(O)c2sccc2c1 N1(C(CN(CCOC)C)=O)CCCCC1CNC(=O)CSc1ccccn1 C1(C(=O)O)(CNC(C(CO)NC(C)=O)=O)CC2(CC2)C1 C1(C(=O)NCCN2CCC(OC)C2)CC(C)CN(C(c2ccsc2C#N)=O)C1 N1(C(C2N(C(C3CC(N(C)C)C3)=O)CCC2(C)C)=O)CC2(C1)CC(C)(C)C2 C(=O)(C1=CCCCCC1)NCCn1cc(-c2c(F)ccc(OC)c2)nn1 N1(C(C(C(C)C)O)=O)CC(N(C)C(c2n[nH]cc2C(F)(F)F)=O)C(C)(C)C1 c1(C(=O)NC(CC=C)CNC(c2ccn(CC)n2)=O)cc(=O)c2ccccc2o1 C(C(C(=O)NC1C=CCC1)C(C)C)NC(C(C)(C)NC(=O)OC)=O N1(C(C)=O)CC(O)CC1Cn1cc(CNC(=O)CCn2cncn2)nn1 C#Cc1ccc(C(=O)NCc2nnn(C)c2C(=O)NCC2CCCS2)cc1 C=CCC(C(=O)N1CCC(NC(c2[nH]ccc2C2CC2)=O)C1C)C(C)C C12(C(=O)NC)COCC1CN(C(C1CN(C(=O)OC(C)(C)C)CCCO1)=O)C2 N1(c2ccnc(NC(c3c(C)nc(C)s3)C)n2)CCOC(C(F)F)CC1 C1(CNC(COC)=O)CN(C(=O)CO)CCC1(F)F c1(C(N(C)CC2CN(C(C3CN(CC)C(=O)C3)=O)C2)=O)cc(C)cc(O)c1 c1(C(C)NC(=O)C(=O)NC(C)C)ccc(Cl)cc1Cl.C(C)(C)C.C=O.N C1(C(=O)NC2(CC=C)CC2)(OC)CCN(C(c2ccnc(C)n2)=O)CC1 C(C1CCCO1)=CC(=O)NCC1CC(NC(c2ccc(C(F)F)s2)=O)C1 C1(C(N2CC(N(C(C3CN(CC(C)C)C(=O)C3)=O)C)C2)=O)Cc2cccnc2C1 C1(C(=O)Nc2ncccc2C(F)(F)F)CCN(Cc2ccccc2)CC1 [N-]=[N+]=NC1CC(C(=O)NC2CC2C(F)(F)F)N(C(c2scnc2Cl)=O)C1 C1(C(N(CC(NOC(C=C)C)=O)C)=O)CCC(C)(O)CC1 c1(C(C(N2C(C3CC3)CCC2)=O)=O)ccc(O)cc1.C(C)(C=O)(C1CC1)OC N1(CCNC(C2CC3C=CC2C3)=O)CCN(C(c2ccc(CO)cc2)=O)CC1 C1(NC(C(C(C)C)N(C)C)=O)CCCCCC1NC(=O)CC1CN2CCN1CC2 C1(C)(CC)C=C(C(=O)N(C)CCN(C(=O)C(O)CSC)C)C1 N1(C(CCOCC(C)C)=O)CCC(C)(C)C1CC(=O)NC1CSC1 Cn1cnc2[nH]c(C(=O)NCC(CNC(C3(CO)CCCCO3)=O)CO)cc12 N1(C(C(CC#C)CC#C)=O)CCN(C(=O)CC(C(N)=O)NC(C)=O)CC(C)(C)C1 c1(NC(c2c(CNC(C(CCC)F)=O)n[nH]c2)=O)ccccc1N=[N+]=[N-] C(=O)(CCCCC1CCSS1)N1CCC(OCCNC(C2C(CC)OCC2)=O)C1 N1(C(CCCC#C)=O)CCCC(C2CCN(C(=O)CCCc3nncn3C)C2)C1 c1(C=O)cc(F)cc(F)c1O.CC1CCCC1(C)C(=O)NCC1(C)CCCC1.N S(=O)(=O)(c1cccc(F)c1)N1CC2C(C2)C1.c1(C(=O)NC)ccc(Cl)c(O)c1 c1(NCC2(NC(=O)CC34CNC(=O)C(C3)C4)COC2)ncnc2cnccc12 C(=O)(C1=C(Cl)CCOC1)N1CC(C)C(NC(c2cnc(O)n2C)=O)CC1 Cc1ccccc1C=CC(=O)N(CCCCCC(=O)N(c1cnn(C)c1)C)C C1(CNC(c2c(OC)n[nH]c2)=O)COCCN(C(=O)C(c2cnn(C)c2)C)C1 C1(CNC(C(CC)=CC)=O)CN(C(C2(C)CC3(CCC3)C2)=O)CC12CC2 c1(CCC)cc(C(N2CCCC2CNC(=O)Cc2cnn(C)c2C)=O)n(C)n1 c1(C(=O)N)cc2ccc(F)cc2cn1.CC(C)(CF)C(=O)NCC12CC(C1)C2 c1(SC)ccc(CCNC(=O)Nc2c[nH]nc2-c2ccccn2)cc1 N1(C(C2N(CC)CC2)=O)CC(NC(c2cncn2C)=O)C(c2cccc(F)c2)C1 c1(NC(N(C)C(c2ccc(Cl)cc2)C2CCOC2)=O)nc2c(s1)COCC2 CCC(C(=O)N1CCCC1CCCNC(c1cnn2ccccc12)=O)C(F)(F)F CC(C)CCCC(=O)NC1CC(O)(CNC(=O)CN2CCN(C)C(=O)C2)C1 N1(C(C2CCC(CC)CC2)=O)C2CCC(C2)C1C(=O)N(C1CC(OC)C1)C C1(C)(C(=O)NCc2n(C)cnc2)CC12CCN(c1ccc(F)cn1)CC2 N1(C(C(C)OCCC=C)=O)CCN(C(c2cccc(C3CC3)c2)=O)C2(CCC2)C1 Cc1c(NC(C2CCCC2NC(=O)CC(=O)NC2CC2)=O)cnn1C C#CC1CN(C(C2CSCC(=O)N2)=O)CCN1C(c1ccc(C)nc1OC)=O C(=O)(C1=C(C)S(=O)(=O)CC1)N(CC(C)N(C(c1cc(OC)n[nH]1)=O)C)C c1(C(=O)NC2CC(F)(CNC(c3cc(C)c(Cl)s3)=O)C2)cc(C)c(C)cc1C c1(C(N2C(CCNC(c3sc(C)c(O)n3)=O)COCC2)=O)cc2n(n1)CC(F)C2 N1(C(c2sc(CC)c(C)c2)=O)CCN(C(=O)Cc2cnoc2)CC1C(F)F CCC(C)CC(=O)C(=O)NCC(C)(C)OCCNC(C1(C)CCCO1)=O C1(CNC(C2(COCC)CCC2)=O)CCCN1C(C1C2CCCC12)=O Cc1cc(C)n(C(C)CC(=O)NC(C)Cc2ccc(Cl)cc2)n1 C1(C(=O)NCC(COC)(F)F)CC=CC(NC(=O)C(N2CCCCC2)C)C1 N1(C(c2coc3ccccc23)C(=O)NC(C)C)CC2(CCCC2)OCC1C c1(C(=O)OCC(C2CCC(N)CC2)=O)cccc2nc(Cl)cn12 C1(C(N2CCCC(OC)C2)=O)CCN(C(=O)C2=C(C)OCC2)CC1(C)C CC1CCC=C1C(=O)NC1CC12CC(NC(c1cnc(C3CC3)nc1)=O)C2 c1(C(N(C2CC3CN(C(CCSCC(C)C)=O)C2C3)C)=O)ccc2cnnn2c1 C1(CNC(c2n(CCC)ccc2)=O)CC2CCC1N2C(c1cccn1CCC)=O c1(C2(C(N3CC(SC(CC(=O)OCC)C)C3)=O)CCC2)cccc(Br)c1 c1(C(N(C2CCN(C(C3CCSCC3)=O)C2)C)=O)ccnn(C)c1=O N1(C(C(CC=C)C)=O)C2CCC1CC(NC(=O)C(c1ccc(F)cc1F)(F)F)C2 C(=O)(C(CC(F)F)C1CCC1)NCCN(C(c1nncc(CCC)c1)=O)CCC C1(NC(C2C(C)C2)=O)COC2(C1)CN(C(C1(C)CCC(F)(F)CC1)=O)C2 Cc1cccc(C(=O)NCCCOCCC(=O)NCC(F)(F)C(C)C)c1 N1(C(CCCCNC(C(CC)(C)CC)=O)=O)CCC2OCCCC2C1 CCC(CC)(CO)C(=O)N(CC(C)NC(c1cc(C#N)c[nH]1)=O)C c1(CC)nn(C)c(Cl)c1C(=O)N(C)C.C1CCN(C(c2c(C)n[nH]c2C)=O)CC1 C(c1ccc(Cl)cc1F)=CC(=O)NCCCC.C1(C(=O)N)CC2C(C1)C2(F)F c1(C(=O)NC(C)C(C)NC(=O)C(F)(F)C(F)(F)F)cc2ccncc2[nH]1 C1CS(=O)(=O)C12CCNCC2.c1(-c2scc(NC=O)n2)cccc(C(F)(F)F)c1 N1(Cc2c(OC)cco2)CCC(C)(C(=O)NCCC2CCCC(C)C2)C1 C1(CCCCCNC(C2CCCC23CC3)=O)CCN(c2nncs2)CC1 n1(CCN(C)C)cc(C2CN(C(C3CCCN3C3CCCC3)=O)C2)nn1 N1(C(C(=O)NCC)=O)CCN(C(c2ccc(-c3ccsc3)cc2)=O)CC(C)(C)C1 N1(C(C(C)(Cl)Cl)=O)CCC(C2CCCN(C(C3CCCC4CCCN34)=O)C2)CC1 C1(O)(NC(COC2C(CC)CCCC2)=O)CCc2ccccc2C1 C(=O)(C(C)S(N)(=O)=O)N1CCC(CC)C1C(=O)NCC(O)CC1CCC1 N1(C(c2c(C)cc[nH]2)=O)CCC2(C(N3CC(c4ccon4)C3)=O)CCCC12 C1(NC(COCCC)=O)C2CC3CN(C(=O)CCc4cc(OC)no4)C1C3C2 C1(OC2CCN(C(C)(C)CC#N)C2)CCCN(C(=O)C(F)Br)C1=O C1(CN(C(=O)CCSc2ccccn2)C)COCCN1C(c1cc(Cl)ccn1)=O c1(C(=O)NCC(CNC(=O)CC(O)c2cnc(Cl)s2)O)nnc(O)cc1O n1(CC)nnc2c(NC(C)CN(C(=O)CCS(=O)(=O)N(C)C)C)ncnc12 CN=c1[nH]ccc(C(=O)NCC2COCC2NC(=O)C2=CCCOC2)c1[N+](=O)[O-] N1(C(c2c(C)con2)=O)CCN(C(=O)CCOCC2CCC2)CC1C(C)C C=C(Br)CC(C)(C)C(=O)NCC(C)CNC(c1cnccc1C(=O)OC)=O N1(C(C(=O)NC2C(CCCC)CCC2)=O)CCC(C#N)(C#N)CC1 c1(C2CC(NC(C3(N4CCOCC4)CC3)=O)C2)cn(CC)nn1.c1ccncc1.O c1(CN2CC(C(=O)NC(c3cccnc3)CC)C2)c(OC)cc(Br)cc1F c1(CCC(=O)NC2CCC3CC23)cnc2c(Br)cccn12 C(C)(C(O)C(=O)NCCC1(NC(=O)Cc2ccccc2F)CC1)OCC N1(CC)OCC(NC(=O)C(C)(C2CC2)N(C(=O)Cc2cccnc2)C)C1=O C(=O)(C(=O)C(C)(C)C)N.N1(C(C)C)CC(C(N2CCC(C)(CC)C2)=O)CC1=O C(=O)(CC(C)NC(c1occc1C1CC1)c1nnnn1C(C)C)NC C1(NC(C2C(C)CC(=O)NC2)=O)CCSC12CN(C(=O)CN(C1CCC1)C)C2 C1(NC(CC(C)C)=O)CCN(C(c2cocn2)=O)CC1(C)C.C(=O)(C(C)(C)C)N c1(N2CC3C(CNCc4c(Cl)nsc4)C3C2)ncc(C(F)(F)F)cc1Cl C#CCCCCC(=O)NC1(C)CN(C(C2(C)CCC(C)C2)=O)C1 C1(CNC(c2nc(C)sc2)=O)CCCC(NC(=O)CP(C)(C)=O)C1 C(CC(F)F)(C(=O)N1CCC(N=[N+]=[N-])C1)N(C(=O)CCc1ncccn1)C S(=O)(=O)(c1cc(Cl)c(Br)cc1F)N1CCC(CCOC)C1 C=C(Cl)C(C)(C)C(=O)NC1CC1CNC(c1scc(Cl)c1Cl)=O CC1(C(N2CCC(NC(C34CC(F)(C3)C4)=O)C2)=O)CCOC1 Cn1cc(-n2cnc(C(=O)NCCCNC(C3CC3(C)C(F)F)=O)c2)cn1 CC1(C)OCCC1C(N1CCOC(c2cnn[nH]2)C1)C(=O)NC1CC1 C1(C(=O)Nc2cccn(C3CCSC3)c2=O)CCn2cnnc2C1 C1(CNC(N2C(C)(c3ccccc3)CC2)=O)CC2CCCCN2C1=O Cc1c(C(=O)NC2CC(NC(C3CC34CC4(F)F)=O)C2)c2ccccc2n1C Cc1cc(C(N2CC(CN(C)C(c3ccc(O)c(Br)c3)=O)C2)=O)c(C)cc1Br N1(C(c2c(C)c[nH]n2)=O)CCC2(CCOC2)C(CNC(=O)CCCC(F)F)C1 CC1CC(C(=O)OCC2CCCO2)CCN1C(=O)OC(C)(C)C.C1CO1 C1(C(=O)NC(c2cccc(C)c2)C)CC(F)CN(Cc2cccc(C#N)c2)C1 C1(OC)CC(NC(=O)CCC2CCCN(C)C2)CN(C(C2C=CC=CC=C2)=O)C1 C(C(CCNC(C12CC(NC(=O)Cc3coc(C)n3)(C1)C2)=O)O)OC C(=O)(CCC1=CCCCC1)NC1C(C(=O)Nc2cccc(OC)c2C)COCC1 N1(C(C(=O)NCC)CC2CCOC2)CCOCC(CO)C1 N1(C(C(CC#C)C2CC2)=O)CCCC(F)C1.n1(CC(=O)N)cnc(C(F)(F)F)n1 C(C(C)(C)C(=O)NC1CN(C(=O)CC2CC2(C)C)CC1C(F)F)OC C1(C=O)(CNC(c2cc(C)oc2)=O)CC12CCC2.C12(CC)CC(CO1)C2.N c1(CC)ncc(C(=O)NC)[nH]1.c1ocnc1C=O.C(C)(C)C=O.C(C)=O C1(C(=O)NC2CCN(C(C3CCCCC3O)=O)CC2)CC2CSCC(C1)C2(F)F c1(OC)ncc(Cl)c(=NCC2CCCC2NC(c2ncoc2C(F)(F)F)=O)[nH]1 Cc1cc(O)ncc1C(=O)NOCC(=O)NCCC1CC(C)C1 CCCC(C(=O)NCCCC(=O)OCCOCC)NC(=O)C=C(C)C CCCCC(CNC(=O)CSCC)NC(=O)Cc1sc(S)nc1C C(=O)(C(C)C(O)C(C)CC)N1CCC(C=C)(C(=O)NOCC(F)F)C1 c1(-c2c(C)nc(CC)s2)ccc2c(C(=O)Nc3cccc4c3CCC4)noc2c1 Cc1nc(N2CCCC2)cc(N(CCSc2n[nH]c(C)n2)C2CC2)n1 c1(CC)ccc(NC(=O)C=CC(C)NC(C2(C)CCCC2O)=O)c(F)c1 c1(C=O)cnn(C)c(=O)c1.C(=O)(Cc1ccco1)N(CC#C)CC1CC1 C1(CC)C(NC(=O)Cc2cscn2)CCN1C(=O)C(C)CC1CC1 N1(C(C2(NC(C)=O)CCOC2)=O)CCC(C)(C)C1.C(=O)C(C)=C1CCC1.N C(CC(C(=O)Nc1ccsc1C(C)C)NC(=O)Cc1ccoc1C)OC N1(C(CC(CC)C2CC2)=O)CCOCC(C(=O)NCc2ccn(C)n2)C1 c1(N(CC#CC)C)ccncc1S(=O)(=O)NCCCOc1ccccc1 N1(CC)CCN(C(=O)C(C)(C2CC2)N(C)C(C2COC(=O)N2)=O)CC1C Cc1cc(C(N2CCC(NC(=O)CCc3nncn3C)C2C(C)C)=O)nc(C)n1 N1(C(C(CC)CC)=O)CC2CC(NC(=O)CCOC3CCOCC3)CC1C2 c1(N2C3CN(C(c4cccc(Cl)c4Cl)=O)C(C3)C2)ccn2ncc(Br)c2n1 C1(CC(=O)NCC(=O)OCC#C)CCN(C(=O)CCCN2CCCC2)C1 C(C(=O)NCC1CC(O)C(O)C1)(C(C)(C)C)NC(CC1C(C)(C)CCO1)=O C#CC1(C(=O)NC2CC=CCC2)CN(C(C2CN(C3COC3)C2)=O)C1 c1(CS(Cc2cc(C)nn2C)=O)nc(Cl)c(Br)cc1[N+](=O)[O-] N1(C(C(CCCCC)CC)=O)CC2(C1)CN(C(c1cccs1)=O)CC(C)(C)O2 Nc1c(C(=O)NC2CS(=O)(=O)CC2NC(=O)C2=COCCC2)cccc1F C1(CC(N2CC(C(CC)C)C2)=O)C2CCC(C2)N1C(=O)CN(c1cnccn1)C C1CCN(C(C2CCC(=O)NC2)=O)C12CCC2.n1(CC=C)cc(C(=O)NC)nn1 c1(C(=O)NCC2CCN(C(c3cc(C(C)C)no3)=O)C2)cncn(C)c1=O C1(NC(C(CCN(C)C)O)=O)CC2CC(NC(=O)CCc3ccc(O)nc3)C2C1 C(=O)(CC1=NN(C)C(=O)C1)NCC(CCNC(Cn1c(C)nnn1)=O)O c1(C(=O)NC2CN(C(C3(C)ON=C(C)C3)=O)CC2C)coc2c1CCCC2 O=C1CCC(=O)N(Cc2cn(C3CC(NC(=O)CO)C3)nn2)C1.C1CCOC1 CC1(C)COC(C(=O)NCC2CCC(NC(C34CCC(C3)C4)=O)C2)CO1 C1(C(=O)NC2C(NC(CCCCOC)=O)COC2)CC2C=CC1CC2 CCN=c1ccc(C(N2CC(NC(=O)CCC(C)CC)C3(CC3)C2)=O)c[nH]1 C1(C(=O)NC(c2nc(C)[nH]n2)C)CCOCCN1C(c1cnc(=N)[nH]c1)=O N1(C(CCC)C)CC(C(=O)NCC2CN(CC3CCC(C)O3)CCO2)CC1=O n1(CC)cc(C(=O)NC2CN(C(=O)CCOc3ccccc3F)CC2O)c(C)n1 N1(CC)CCOCC1C(=O)NC1CC(C)C1.c1(C2(C(=O)N)CC2)ccno1 C(CCCC(=O)NC1CCCCC1NC(=O)C=CC(C)(C)SC)OCC N1(C(c2cnn(CC)n2)=O)CC23CCCC2(C1)CN(C(=O)Cn1cccn1)C3 N(C(=NCCF)NCC1(O)CCN(C(=O)OC(C)(C)C)C1)Cc1c(C)coc1 N1(C(c2ccc(CCCC)cc2)C(=O)NCC)CCC2CN(C)CCC12 C12(NC(CC=C=C)=O)CCN(C(c3cncc(-c4cccc(F)c4)c3)=O)CC1C2 C1(n2cc(C3C(C(=O)OC)C3)nn2)CCC(NC(C2CCCOCC2)=O)CC1 C(=O)(C1CCCc2sc(=N)[nH]c21)N(CCN(C(c1c(OCC)cccc1)=O)C)C Cc1ccc(C)c(C(N2CC(O)CC2CNC(c2cc(Br)oc2C)=O)=O)n1 O=C(C#CC1CCCOC1)N1CCN(C(c2ccoc2Br)=O)CC1 C1(C(N2CCC(CNC(C3N(C(C)=O)CC(O)C3)=O)C2)=O)CCn2nncc2C1 c1(C(C)=O)cccnc1NCCCNC(=O)Cn1cccc1 C1(C#N)(C(N2CCCCC2)=O)CC2CC2C1.C(=O)(C)N(CC=C)C.C1CC1 N1(C(C)=O)CCCC(C)(NC(C(F)(F)F)c2nccn2C)C1 N1(C(C(C)O)=O)CC2CC(NC(c3cccc(C(N)=O)n3)=O)C1C2 C=CCC(CNC(=O)COC(C)(C)CC)C(=O)N1CCS(=O)C(C)C1 O=C1NC2(CO1)CC(C(=O)NC1CC3C(C1)C3(F)F)C2 CCC(C)(C)C(O)C(=O)NC1CCC1NC(c1ccc(Cl)c(N)c1)=O CC1Oc2ccccc2N(CC(=O)N(C(=O)CN2CCC2)CCNC(N)=O)C1=O CCC(CC)C(=O)NCC1CCN1C(c1ccsc1Br)=O c1(C(=O)NCC(C)CN(C)C(c2cnoc2)=O)ncoc1C1CC1 C1(CC)COC(C)(C)CN1C(=O)CC(C(F)F)NC(c1cc(COC)[nH]n1)=O N1(C(CC2(OC)CN(C(C3C4CC(=O)CC34)=O)C2)=O)CCCC(O)(CO)C1 CCC(C)(CNC(c1cnc(C2CC2)o1)=O)C(=O)NC1CCC(O)C1 C1(C(N2CCOC(C)CC2)=O)(NC(C2CC(N(C)CC)C2)=O)CCC(C)(C)C1 Cc1cc(=O)c(C(N2CCC2)=O)cn1C1CC1.N1(C(C=O)=O)CCCC(C)C1.C C(=O)(CC(C(F)F)n1cccn1)N(C(C)C)CCNC(C12CCC(CC1)O2)=O CC(=NOCCCN1CCCCCC1)c1nc(N)sc1C C(=O)(C(C)CCC)N1CC(OCC)(CNC(c2n[nH]cc2C2CCC2)=O)C1 c1(N(CCCC)C)nc2cc[nH]c2c(=NCC2CC3(CCC3O)C2)[nH]1 Cc1cccc(C)c1C(c1nnnn1C)NCc1cnc(O)s1 CCC(C)(C)CC(=O)N1CCOCCC1C(=O)NCCC1CC(F)C1 c1(CCNC(C2(F)CCN(C(CC(=O)OC)=O)C2)=O)c[nH]c2ccc(Cl)cc12 N1(C(c2nc(CCC)sc2)=O)CCC(C)C(NC(=O)C=C(C)c2ccsc2)C1C c1(COC)nnc(N2CC(C(C)NC(=O)C(C)OCC(C)C)C2)s1 c1(SC)nn(C)cc1C(=O)NC1CC(CNC(c2c[nH]nc2C)=O)C(O)C1 C(CC(C(C)(C)C)NC(C1(C#N)CCSCC1)=O)N(C)C(C1CNC(=O)N1)=O C1(C(N2CCCC(NC(c3cnc(Cl)cn3)=O)C2)=O)CCCCC1(F)F C1(C)(C(=O)NCC(C)C#N)CCCN(c2ccc(C(=O)O)nn2)C1 C(CCC(=O)NC1CCC1NC(c1csc(Br)c1)=O)N(C(C)=O)C c1(OCOC)cccc(S(=O)(=O)N(C)Cc2ccc(SC)cc2)c1 c1(C(N(CC(C)NC(C2CCC2CF)=O)C)=O)ccc(Br)c(F)c1F C1(NC(C(CC)OC)=O)COC2C(NC(c3nc(OC)cc(OC)n3)=O)COC12 N1(C(CN(C)S(N)(=O)=O)=O)CC(NC(c2ccc(CO)c(F)c2)=O)CC(O)C1 N1(C(CCC=C(C)C)=O)CCC2CC(NC(C3CCC(=O)NC3)=O)CCC2C1 CS(=O)(=O)C=CC(=O)NC.C1CN(C(C2CC3CC3C2)=O)CC1C(F)(F)F C(=O)(C(C)(F)C(=O)N1CCCC(N(C(=O)C(C)(C)C)CC2CC2)C1)OC c1(C(=O)N)cc(F)cc(C)c1O.C1(OCCC)CCCCC1C(N1CC(C)C1)=O N1CC(C)OCC1C(=O)O.Cc1noc(C)c1Cn1cc(C2CCN2)nn1 C1CC2(C1)CC2(F)F.[SH](=O)(=O)CC(=O)N1CC(O)CC1C1CCCCC1.CC.S N1(CCC(=O)NC(C2CC(NC(CCOC)=O)C2)C)CCOCC1 c1(C(N2CCC2)=O)cccc2c[nH]nc12.CC(CCc1cn(CO)nn1)CCO C1(CC)CCCC(CNC(c2cc(CNC(=O)C=CSC)no2)=O)C1 C1(OC)CN(C(=O)CCn2cncn2)CC1NC(C1C=CC=CC=C1)=O C1(NC(=O)C=Cc2cn[nH]c2)CCN(C(c2ccccc2-c2cn[nH]c2)=O)CC1 c1(C(=O)NC2C(CNC(Cc3c(C)ccs3)=O)C2)ccccc1SC(F)F C1(CCNC(C(c2cccc(Cl)c2)SC)=O)CCCN(C(C2CCC(=O)N2)=O)C1 C=CC(C)(O)CC(=O)N1CCN(C(CNC(c2nnc(C)s2)=O)C(F)(F)F)CC1 CC(C(=O)NCC1CN(c2cc(C3CC3)nc(Cl)n2)CCCO1)S(C)(=O)=O c1(C(N2CC(C)(NC(C(C(C)OC)O)=O)C2)=O)cc(F)c(O)c(Br)c1 CC1CCN(C(=O)CC2C=CS(=O)(=O)C2)C(C)C1.c1(CCC=O)ccncc1.N CCC(CC)(CO)C(=O)NCC(C1(O)CCN(C(=O)COC(C)=O)C1)C N1(C(CC23CC(NC(=O)OC(C)(C)C)C(C2)CO3)=O)CCC(C)C12CCC2.N c1(C(N2CC(NC(c3c(C)[nH]nc3Br)=O)C(O)C2)=O)cc2ccccc2s1 C(C(C)(C)CC(=O)NC1CN(C(c2cnn(CC3CC3)c2)=O)CC1C)OC N1(C(c2c(CC)nns2)=O)CCC(CCNC(=O)Cc2ccsn2)CC1 C1(CC=O)CC2(C1)CN(C(=O)Cc1ccc3c(c1)CC3)C2.CCC(C)(C)O.N C1(NC(CCSCC)=O)CC(NC(c2ccncc2)=O)C12CCC2.C(C)C.O C(=O)(C(CC)CCCCC)NCC(CC=C)NC(c1cccc(OC)n1)=O Cc1ccc(C(=O)NCC2CCCC2)cc1.n1(CC=O)nnc(C(C)(C)C)n1 c1(Cc2nnc(N3CCC(c4ccc(C)cc4)CC3)n2C)cccc(C#N)c1 N1(CC(=O)NCc2cn(C3CCN(C(COCC)=O)C3)nn2)CCCNC1=O CC1(CNC(=O)CCCc2ccsc2)CCCN1C(=O)CCC1CCOCC1 N1(C(Cc2c(C)n[nH]c2)=O)CCC2CC12C(=O)NCC(O)C(C)(C)C C#Cc1ccc(C(N2CCC(C(C)NC(=O)CCN3CCC3)C2)=O)cc1 C(=O)(C(C(C)(C)C)O)N(CC(=O)O)C(c1cn(-c2ccc(OC)cc2)nn1)C Cc1cc(F)cnc1C(=O)N(CC(=O)NCC1(C)C=CCCC1)C1CC1 N1(C(C(CCC)C)=O)Cc2ccnn2CC(NC(C2(CC)CC2)=O)C1 N1(C(CCc2onc(C)n2)=O)CC(N=c2ccn3nccc3[nH]2)CC(C)(C)C1 N1(C(C=C(C)C)=O)CCC2CC(C1)CN(C(c1nnn(C)n1)=O)C2 C12(CNC(CCCC)=O)CCCN(C(=O)COc3cccc(Br)c3)C1C2 CC(C(=O)N(C)CC)NC(=O)CC1CCCC1.c1(C=O)cscn1.C(=O)C C12(C=O)CC1COC2(C)C.C(C)(CO)(C(=O)N1CCC(C(C)(C)C)CC1)OC.N N1(C(=O)NC)CCC(C(=O)NCC2CC2)C1.C(=O)C(O)c1ccco1.C C1(CNC(C(N2CCN(C)CC2)CC)=O)CCCN(C(c2csc(C)c2C)=O)C1 C(=O)(CCS(C)(=O)=O)NC1(CCOC)CCN(C(c2cccn2C)=O)C1 C1(CC=O)SC2=NCCN2C1=O.c1(C(=O)OCC)nc(C=O)cs1.CCC.N C12(C(=O)NC3CCCN(C(c4c(CC)nccn4)=O)C3)CCCC1C2(F)F C1(NC(CC(CC=C)(C)C)=O)CC2COCC(C1)C2NC(c1cc(OC)cs1)=O N1(C(c2c[nH]c3cccc(C)c32)=O)CCc2ccc(NC(=O)C(C)O)cc2C1 N1(C(CCCNC(C)=O)=O)CCOCC(C)(CNC(=O)C(O)C2CC2)C1 N1(C(CC)=O)CCn2ncc(CN(C)C(C3CC(C(F)(F)F)C3)=O)c2C1 C1(CNC(C2(CC)CC2)=O)CCC(C(=O)NOCCCF)C1 c1(C=O)cc(C)cc(N)c1.N1(C(C2CC2)=O)CCC(C(C)(C)C)CC1.CC.O C(=O)(C(C)CC(F)(F)F)N.c1(C(N2CCC(OC)(C)C2)=O)cnc(N)c(Cl)c1 n1(CCC)nc(-c2cc(SC)ccn2)nc1C1CCCN1Cc1ccccc1 C1(C)CN(C(C2(C(N)=O)CC2)=O)CC1C.c1(C(C)F)ccc(C(=O)N)cc1.C N1(C(C2C(=C)C2)=O)CC2CC(NC(c3ncc(C(F)F)s3)=O)CC1C2 CC1CCCC(CCNC(=O)Cn2cc(C)nn2)C1.c1(C=O)ccc(Cl)cn1.N c1(C(c2ccc(Cl)cc2)NC(=O)NCC(C)(C)C)c[nH]c2ccccc12 C(=O)(C(C)(C)C(F)(F)F)N1CC2C(CCNC(c3cc(C)c(O)nc3)=O)(CC2)C1 C1(C(=O)NCC2(F)CN(C(c3nnn(CC)c3C)=O)C2)CCc2n[nH]cc2C1C c1(N2CCN(C)C(CNC(C3CN(C)C(=O)N3)=O)C2)nc2cccnc2s1 Cc1cc(C(=O)NCC2CN(C(c3cc(Cl)cc(F)c3F)=O)C2)cc2nn[nH]c12 [SH](=O)(=O)c1c(C)noc1C.C(=O)(C(C)(F)F)N(CC)CC.C(=O)CC.C Cc1cccc(S(=O)(=O)N2CCC3CN(c4ncnc5cc[nH]c45)CC3C2)c1 c1(CN2CCCC(NC(=O)CC3CCCC(=O)N3)C2)ccc2cccc(F)c2n1 C(=O)(C(=O)CC(C)C)NCC(CC=C)NC(c1ccc(CO)c(F)c1)=O C=C=CCC(=O)N(CC(C)O)CCNC(c1ccnn1C(C)C)=O Cc1cc(C(N2CCC(NC(C3CN(C4CCOC4)C3)=O)C2)=O)ccc1O CCCC(C)(C(=O)OC)NC(=O)CCc1ccccn1 c1(NC(C2N(CC)CC2)=O)ncccc1CSc1ccsc1C(=O)OC CCN=C(NCCC(=O)N(C)C)NCC1CCC1(F)F c1(C(N2CC3C(N(C(C(C)NC(CC)(C)C)=O)C)C3C2)=O)cccn2ccnc12 Cc1cccnc1CC(=O)NCC1CCC1NC(=O)CN(C)S(N)(=O)=O C1(C(N2CC(CN(C)C(c3cnc4[nH]ccc4n3)=O)C2)=O)CCn2ncnc2C1 N1(CCOCC=C)CC2CCC1CN2C(=O)Cn1cc(C(F)(F)F)cn1 c1(C(=O)NC2CC(C)(NC(=O)C3CC3)C2)cc2c(Cl)cccn2n1 Cc1nn(C)c(C(=O)NCCCCC(C)NC(C2C3CCCCC23)=O)c1Cl C(CC(C(C)C)NC(=O)CC1CC1C)NC(C1(OCC)CCOC1)=O CC1(CO)CCCN1C(=O)CC1(C)CCN(C(c2cc(Cl)cs2)=O)C1 C1(c2nc(CNC(C3CCCC3)=O)[nH]n2)CCCN(C(=O)C(O)C2CCC2)C1 C(C)(C)(CC(F)C(=O)Nc1cn(C)nc1OC)NC(CC(CC)SC)=O C(=O)(CC(C)CC(=O)N1CC(F)CC1CNC(=O)C)OC.c1cncc(Cl)n1 C(=O)(C1(C)CCn2ccnc21)N1CC(C(C)NC(C=Cc2n(CC)ncc2)=O)C1 N1(C(C2N(C(COCCCC#C)=O)CC(OC)C2)=O)CC(C)OCC(C)(C)C1 C=CC(O)C(=O)N(C)CC1CCN(C(=O)CCc2cn[nH]c2)C1 c1(C(N2C(CNC(c3cc(Br)c[nH]3)=O)CCCC2)=O)cccc(=O)n1O Cc1c(F)ccc(C(=O)NC2CCCCC2NC(c2cncs2)=O)c1N C(C1c2ccccc2CN1C)NC(=O)NCc1c(OC)cccc1Cl C1CCCCC1.c1(N(CC=O)C(C)=O)ccnc(Cl)n1.CCCC=CC(=O)N N1(C(c2ccc(C#C)cc2)=O)CCC2(NC(c3cc[nH]n3)=O)CCCCC12 N1(C(C2(C)CC(O)CN2C(=O)C2=CCCC2)=O)CCC12CCOCC2 C(C(C)(C(=O)N1CCN(C=O)CC1)NC(=O)CC1(N(C)C)CCC1)SC.O N1(C(C(C)(C)C)=O)CC(NC(c2cnn(C3CCC3)c2)=O)CC(O)C1 c1(-c2n(C)cnc2)cccc2ncc(C(=O)NCCc3nccs3)n12 c1(CC(=O)N(C)CC2CC(F)CN2C(=O)CC(F)F)cccc(O)c1F c1(OC)ncnc(C)c1NC(=O)CC1CCN(CC(F)(F)F)CC1 c1(CC)c(C(N2CCCC2)=O)cnn1C.c1(C(NC2CC2)=O)cn(C)cc1C.C c1(C(N2CC(CN(C(CCN(C)CC)=O)C)OCC2)=O)ccc(OC)nc1Cl N(C)(C(=NCCC(C)C)NCC1CC1c1ccsc1)Cc1c(COC)noc1 Cc1nn(C)c(C(N2CC3CC(C2)C3NC(C2CCCC2)=O)=O)c1[N+](=O)[O-] C(=O)(CS(=O)CCC(F)(F)F)N(CCC)C.c1(CCC(=O)N)cnc(C2CC2)o1 N1(C(C=CC)=O)CCC(C2CCCN2C(=O)CSCC(=O)OC)C1 C1(c2nnc(C3N(C)CCOC3)o2)CC2CCC(C1)N2C(=O)OC(C)(C)C N1(C(C2CC(C)NC(=O)C2)=O)CCC(NC(c2ncn(C)n2)=O)C(F)(F)CC1 C12(CNC(C3CCCCC34CC4)=O)CCC(CN(C(=O)Cc3ccsc3)C1)C2 C1(OC)CCC(C)(C(=O)NCCC2CCC2)CC1.C1(C=O)NC(=O)OC1C.N N1(C(C2CCn3cncc3C2)=O)CCCC2(C1)CN(C(C1CCCC1)=O)C2 C1(NC(c2nc(CC)oc2)=O)CCCN(C(=O)CCn2ccnn2)C1 CC(C)CCCC(=O)NC1COCCN(C(c2cc(-c3cccnc3)no2)=O)C1 c1(SC)nc(N2CC=CC(NC(=O)CC(O)C(C)C)C2)c(C)c(Cl)n1 c1(CNC2CC(CC(=O)Nc3ccnc(F)c3Br)C2)c(F)cc([N+](=O)[O-])cc1F N1(Cc2cnc(CCCC)[nH]2)CC2CC(C1)N(c1nccc(C(C)C)n1)C2 C1(C(N(CC(C)(C)C)C)=O)CC(NC(C2(C)CNC(=O)N2)=O)C(O)C1 C12(NC(Cc3c(C)ncs3)=O)CCCC1N(C(c1ccc(=N)[nH]c1Cl)=O)CCC2 N1(C(CC(C(C)C)C)=O)CCC2(CC(NC(=O)CC3(n4cccn4)CC3)C2)C1 CCC(CCC(=O)N(CC(O)C1CCC1)C)NC(c1ccc(CO)o1)=O N1(C(CC(C)(C)NC(=O)NC(C)Cc2ccco2)=O)CCCCC1 c1(C(=O)NC2C(NC(CCCOC(C)C)=O)CCOC2)cc(C(C)C)nc(O)c1 C1(C(=O)NC2CC(CNC(=O)C(C)n3ccnn3)C2)(OC)CCCCCCC1 c1(C(=O)NC2CC(CCNC(CC3CC(OC)C3)=O)C2)cnnc(O)c1 c1(C(=O)NCC(CCOC)NC(C2COCCC2(F)F)=O)ccc(OC)c(F)c1 N1(Cc2c3n[nH]c(C)c3ccc2)CCc2cc(OCc3ccccc3)ccc2C1 N1(C(c2ncc(C)[n+]([O-])c2)=O)CC2(CCCC2)C1C(N1CC(C)(C)CCC1C)=O c1(C2(NC(=O)CN3CCC(NC(=O)C4CC4)C3)CC2C)cccc(Cl)c1 C1(F)(C(=O)NCC(C)CN(C)C(c2[nH]ccc2C2CC2)=O)CCCC1 CCC(CC)C(C)C(=O)NCCOCCCNC(C1C(C)C1C)=O N1(C(C(COC(C)=O)C)=O)CCC(C)(NC(C2CCCSC2)=O)CC1 Cc1cn2c(C(=O)NCC(C)NC(=O)CCc3ccc(N)cn3)cnc2s1 CCCC(CCC)C(=O)N1CCC(CO)C(NC(=O)CCc2nccn2CC)C1 CCCC(CC)CCC(=O)N1CCC1CC(=O)NC(C)(C)COC N1(C(=O)CCN(CCCO)C(C23CCCCC2C3)=O)CC2(CCC2O)C1 C=CCCCCCC(=O)NCC12CCC1CN(C(c1cnc3[nH]ncc3c1)=O)C2 N1(C(C(C(C)(C)C)O)=O)CCCC12CCN(C(=O)C1=CC3C=CC1C3)C2 N1(C(c2cccc(COC)c2)=O)C(C)CN(C(c2cccc(C#N)c2)=O)CC1C N1(C(C(c2ccc(C)nc2)N)=O)Cc2cc(Cl)ccc2CC1CO c1c(F)c(F)c(F)c(F)c1F.c1(C(C)CC)ccnc(C(F)(F)F)c1 O=C(N=c1[nH]oc2ccc(Br)cc12)NC(CO)CC(F)F O=C(C1=C(Cl)CCC1)NCc1ccc(C(N2CCOC3CC23)=O)nc1 C1(CN(CC(=O)O)CC2(CC)CCC2)CCCN(Cc2coc(C)n2)C1 C(=O)(C1CCCCc2ccccc21)NC1CCN(C(C(CC)COC)=O)CC1 c1(C(=O)NC(C)CCCNC(=O)C(C)CC(C)(C)C)cc(F)cc2ccoc12 c1(C(=O)N)ncc(Br)cc1C.C(CC)(C(C)C)NC(c1nc(OCC)oc1)=O N1(C(C(C)Cn2ccnc2)=O)CC(NC(C2(c3ccc(Cl)nc3)CC2)=O)C(F)C1 N1(c2cn(CCOC)nc2)C(=O)C2CCC3(CCOCC3)CN2C1=O c1(C(N(C2CCN(C(=O)COC)C2)CC)=O)cnc2ncc(Cl)cn12 C1(C#C)(C(N2CCC(CC#C)C2)=O)CN(C(C2CC(CC)(CC)C2)=O)C1 CC(CC(C)NC(C1(CCF)CC1)=O)Nc1ccncn1 C1(C(=O)NCCC(C)CO)(CNC(C2CC(=C3CCC3)C2)=O)CCCCC1 C1(NC(c2n(C)nc(C3CC3)c2)=O)CCN(C(=O)CCc2nc(O)n[nH]2)CC1F N1(CCC#C)CCC(C(=O)NC2CCCN(C(C3CC(C)=NO3)=O)C2)CC1 Cc1cccc(-c2cn(C3CCCC(NC(C4CC(=O)N(C)C4)=O)C3)nn2)c1 N1(C(C(c2c(F)cccc2F)C)=O)CC(NC(=O)Cn2cccc2)C(C2CC2)C1 C(CCC(=O)NCCC(C)(C)NC(=O)C(=O)NCC(F)F)SC(C)(C)C c1(C(c2n(CCSC)nnn2)NCc2nc(C(C)C)ns2)c(C)noc1C c1(OCC(=O)NCC(C)C)cccc([N+](=O)[O-])c1.C12(C=O)CC(C)C1C2 C1(NC(C2C=CCC2)=O)CC2CC(C1)N(C(=O)CC(O)c1ccccc1)C2 Cc1ccc(C(=O)NCC2(C)CCC(NC(c3ncn(C)c3C)=O)C2)cc1Cl C#CCC(C)C(=O)NC(C1CCN(Cc2ccc(NS(C)(=O)=O)cc2)CC1)C N1(C(C(C)(C)OCC)=O)CCCCCC1.c1(C=O)ccc(CS(C)(=O)=O)o1.N C1(NC(C(C)=CC)=O)CC(O)CN(C(=O)C=C2CN3CCC2CC3)C1 C1(C=O)C2CC(O)C(C2)N1C(=O)CC.C1(COC)CCCC1.CCC(C)C.N C(=O)(C1=CC2CCCCCC12)NCC(CNC(c1c(C)nn(C)c1Cl)=O)C N1(C(C=CCC)=O)CC2CCC1CN2C(c1coc(COCC(F)(F)F)c1)=O C1(CNC(c2[nH]cc(C)c2)=O)CN(C(C2CCC3(CCC3)C2)=O)CCN1C C12CC1CN(C(=O)C(C)C)C2.C(C)(C(=O)NC)N(CC)CC.C(C)=O N1(C(C2C(CC)C2)=O)CCN(C(=O)CC(C)c2ccco2)C(CO)C1 C(=O)(C1=CCCCC1C)N(CC(=O)NC(C(=O)OCC)C)CC N1(C(C(n2c(C)ncc2)C)=O)CCSCC1CCNC(=O)Cc1ccco1 C(=O)(C1=CCCOCC1)N1CC(CNC(C=CC=CCC)=O)OCC1 C(=O)(CCN=c1ccc(C)c[nH]1)N1CCCC(NC(C(C(CC)O)C)=O)(CO)C1 C(CCCC(=O)NCCCC(C)NC(=O)C(C1CCC1)OC)OCC c1(C(N2CC(CCNC(=O)COCC3CCCOC3)C2)=O)ccc2nc[nH]c2n1 c1(C(=O)NC(CNC(C(C)CO)=O)C2CCC2)ccc2c(c1)OCCNC2=O CN=c1ccc(C(N2CCCC(C(=O)NCCC3(C)CCOCC3)C2C)=O)c[nH]1 c1(N(CCC)CC)ccc(CNC(N2CC(O)(c3cncnc3)C2)=O)cc1 C1(C(=O)NCCCCNC(c2ccc(CO)s2)=O)CCS(=O)CC1 S(=O)(=O)(c1c[nH]ccc1=NCc1cc2c(cn1)OCCO2)NC(COCC)C N1(C(c2cc(C(N)=O)ncc2)=O)CC2(CNC(C3CCCO3)=O)CC1CCO2 C(C)(C(=O)NC1CC(NC(C2CC2c2ccco2)=O)C1)OCCCC c1(N(C)C)ncc(C(=O)NCC2CN(C(=O)C)CCO2)cn1.C1CC(F)(F)C1 C1(NC(C(Cn2ccc(C)n2)C)=O)CCN(C(c2cc(Br)no2)=O)CC1F N1(C(C(F)=C(C)C)=O)CC(NC(c2cnccc2)=O)C(C2CC2)C1.N(C)C.C C=CCCC(C(=O)NCCC(CO)C(C)C)NC(=O)CCc1cccs1 C12(NC(CS(CC)(=O)=O)=O)CCCN(C(C3(C(N)=O)CCC3)=O)CC1C2 C1(NC(=O)CN2CCCCCC2)CCN(C(c2c[nH]cc2Br)=O)CC1F C1(N(C(C=C(COC)C)=O)C2CC2)CCN(C(=O)CCc2cn(C)cn2)CC1 C(=O)(CCC(C)NC(c1scnc1Cl)=O)N(CC(C)C)CCN(C)C Cc1ncc2n1CCN(C(=O)CC1(N(C)C(C3CC34CC4)=O)CC1)C2 CCCC(C#N)C(=O)NCC1CC1NC(=O)Cc1cc(F)ccc1OC C#CC1(C(=O)NCC(C2CCC2)NC(c2c(C)ncnc2C)=O)CCOCC1 c1(C(=O)NC2(C)CN(C(C3CC(C4CC4)=NO3)=O)C2)c[nH]c2cccc(C#N)c12 c1(C(=O)NCC2CCN(C(c3c(C)n(C)cn3)=O)C2)cncc2nc[nH]c12 C1C2CC1CN(C(C13CC=CC(C1)OC3)=O)C2.c1(OCC)ncccc1C=O.N N1(C(c2ccc(OC)c(F)c2)=O)CC2CN(C(C3(C(N)=O)CC3)=O)CC2(C)C1 C(=O)(C(C)CNC(=O)CCn1cc(C)cn1)NC(C#C)C1CCC1 c1(-c2nc(CC(C)(C)CO)nn2-c2cc3ccccc3s2)cc(S(=O)(=O)F)c[nH]1 C(CN=C(NCCCCCCF)NC1C(F)(F)C12CC2)c1n(C)ccc1 S(=O)(=O)(c1ccc(C(F)(F)F)cc1)N1CCC1.Cc1c[nH]c(C(=O)N(C)C)c1C c1(C(=O)NCCC2CSCCN2C(c2cnn[nH]2)=O)ccc2cccnc2n1 C12(C(N(C3CCCN(C(c4c(CC)n(CC)nc4)=O)C3)C)=O)CCCC1C2(F)F CC(C)C(CC(=O)N(C1CC(C)OC(C)C1)C)NC(C1OCCC1C)=O C1(NC(Cc2cc(C)sc2)=O)CC(C(=O)NC(C)CCF)CC1O c1(C(N2CC(COCC)OCC2)C(=O)NCCC2CC2)ccc(F)cc1F C1CN(C(C2CC(O)C2)=O)CC2(CCC2)O1.c1(SC)cccc(CC(=O)NC)c1 C1CCCCN1C(=O)Cc1ccc(C2CC2)cc1.c1(CC)cc(C(=O)N)ns1.C CCCC(CNC(=O)C=C1CCC(C)CC1)C(=O)NC(CO)CCC(C)C N1(C(C(C)C(F)F)=O)CCC2(CCCN(C(c3cc(P(C)(C)=O)ccn3)=O)C2)C1 N1(CC2C(OC)C2)CCCC2(CC2C(=O)OC(=O)N(C)C)C1 C1(CC)CCCN(CC(=O)NCC(C)Cn2cccn2)C1.C(=O)(C)N.C1CC1 N1(C(C2(SC)CCC2)=O)CCCC(C2CC2NC(C2(OC)CCSC2)=O)C1 N1(C(C2(NC(C(CO)OC)=O)CCCC2)=O)CC2(C)CCC2(C)C1 n1(CC)ncc(C)c1C(=O)N(CC(N1CCC1(C)COC)=O)CC N1(C(C(CCC)CC)=O)CCCN(C(c2ccc(F)c(C)c2)=O)C(C(C)C)C1 c1(OC)ccc(C(N2CCC(c3n[nH]cc3C(N3CCC(=O)C3)=O)CC2)=O)cc1 c1(C(=O)NCC(CNC(C2CN(C)CC(C)O2)=O)C)csc(=NC2CC2)[nH]1 c1(CCC)cc(C(=O)N(CC)Cc2ccccn2)cc(OC)c1OC Cc1cc(Cl)cc(C)c1OCCN1CCOC(C)CC1 c1(OC)cc(C2SCCS2)ccc1OC(=O)C=Cc1cncc(F)c1 C#CC1(C(=O)NCc2cc(CC)no2)CCN(C(C2CC(=C)C2)=O)C1 c1(N2CCC(N3CC(C)(C)C3)C2)nc2c(c(=NCCC3CCOCC3)[nH]1)SCC2 C1(N(C(C(CC)SC)=O)CC2CC2)CCN(C(=O)CC2CN(C)C2)CC1 c1(C(=O)NCCN(C(=O)CC2COCC2(C)C)C)ccc(Br)c(N)c1 C1(C(=O)NCCN(C(=O)CN2CCC2C)CCC)CC(C)(C)C1 c1ccc(F)cc1C(N1CCC2(CC2C=O)C1)=O.c1nccnc1C(N)=O.CO Cc1c(C(=O)NC2CC(CCC(N3CC(C)C(O)C3)=O)C2)cnn1C c1(CC)ccc(CC(N2CCC(C(N3CCC(COC)C3)=O)CC2)=O)cc1.N(C)C S(=O)(=O)(c1cccc(N2CCC(CCO)C2)n1)NCC1C(C(C)C)OCCC1 c1(OC)ccc(F)c(C(=O)NC2CC(C)C2)c1.c1(CC=O)c[nH]c(=N)nc1O N1(C(C(CC#C)C)=O)CC2(CCN(C(c3cc(O)c(F)cc3N)=O)CC2)CC1C C1(NC(C2CCCN(C(C3CC3)=O)C2)=O)Cc2ccc(-c3nn[nH]n3)cc2C1 N1(C(C2C(C)(C)C2)=O)CC2CCC(NC(=O)CSc3n[nH]c(O)n3)(C2)C1 C1(CC(=O)NCC(C)NC(=O)C=C2CC2)(NC(C)=O)CC1 N1(C(Cc2ccc(C)cc2C)=O)CCCC(C2CN(C(c3nnsc3N)=O)C2)C1 N1(C(c2c(CC)scc2)=O)CCN(C(=O)C(C)(O)C2CCC2)CC(O)C1 C1(NC(c2cnnc(Cl)c2)=O)CN(C(C2CC=CCC2)=O)CC12COC2 CC1CN(C(=O)C=CBr)CCC1N(C(=O)CCN1C(=O)CCC1=O)C c1(C(=O)NCCC(=O)NCC(CC)NC(=O)CC(C)CF)cc2ccccc2[nH]1 C1(C(N(CCCNC(C(CCC)N(C)C)=O)C)=O)CC(C)CCC1C(C)C N1(C(c2ncn(C)n2)=O)CCC2(NC(=O)CSc3nnnn3C)CC2C1 c1(CC(=O)OCC)ccc(=O)n(CC)n1.c1(C2C(C=O)C2)cncn1C N1(C(CCCc2nc(C)sc2)=O)CC(CNC(C2CC3(C2)CC3F)=O)CC1C c1(C(C(=O)N(CC)C(C)C)C)c(C)noc1C.c1(COC)ccc(C=O)[nH]1 Cc1cc2cc(C(N3CCCC3CN)=O)ccc2[nH]1.C1(=O)C(C)N1C N1(C(C(Br)=C(C)C)=O)CCN(C(C2CCNC2=O)=O)CC1c1cccnc1 CCC(C(C)(F)F)NC(=O)C(C1CCCC1)NC(C1CCC(OC)CC1)=O c1(C(N2CCN(C(CC3CC(CC)OCC3)=O)CC2)=O)oc2ccccc2c1Cl C1(CCCNC(c2c(CC)occ2)=O)CN(C(c2cc(Cl)cs2)=O)CCO1 Cc1cc(N2C3CC2CN(C(=O)COc2ccc(Cl)c(C)c2)C3)nc(C)n1 c1(C(=O)NCCN(CCOC)C(c2ccnc(O)c2)=O)nc(OC)ccc1Cl CCCCCCC(C)(c1nnnn1C)NCC(S(C)(=O)=O)c1ccccc1 Cc1cc(C)c(NC(=O)CC2CC3(C2)CN(C(=O)CCCC(C)C)C3)c(Br)n1 CCC(C)(O)C(=O)NCC.C1(C(=O)N)CCCN(C(=O)Cc2cc(C)cs2)C1 CC(C1CCCCC1)=CC(=O)NC1CCCC1NC(c1cc(O)ccc1C)=O CCC(C(=O)N1CCC(C(C)NC(=O)Cc2ccnn2C)C1)n1cccn1 C1(NC(CC=C)=O)CC2CC1N(C(c1ccc(CSCC)cc1)=O)C2 CC1OCCC1(C)C(=O)NCC1CCC1.c1(C=O)ccnn1CCN(C)C.C CCCCS(=O)(=O)NC1CC1NCc1nc(CO)n[nH]1 C1(N(C(CCOCC(C)C)=O)C)CCCN(C(C2CCC(C(N)=O)C2)=O)C1 Cc1cnc2cc(C(N3CCC(CO)(NC(C4CC4CF)=O)C3)=O)ccn12 C1(C(N(C(C(=O)OCC)C)C)=O)COC2(CN)CC1C2 c1(C(=O)OC)nc(Br)cnc1NC1CC1C(C)C CN1CCC2C(CCN2C(C2(CNC(C3CNC(=O)C3)=O)CC2)=O)C1 C#CC12CCCC1(F)CN(Cc1ccc(C3(C(F)(F)F)N=N3)cc1)C2 c1(C(=O)NC(CCCNC(C(CCC#C)O)=O)C)cc(Br)c2ncccc2c1 Cc1cc(N2CCC(CS(N)(=O)=O)CC2)c2cnn(C)c2n1 C(C1CCCN1C(=O)C=Cc1cnccn1)=CC(=O)N.C(=O)(C(O)C)OC Cc1ncc2n1CCC(C(=O)NC1CCCN(C(c3cc(N)ccn3)=O)CC1)C2 c1(SCC)c(NC(N2CCCC(n3cc(C4CC4)nn3)C2)=O)cccc1F CC1CC(NC(=O)C(F)(Cl)c2ccccc2)CN(C(c2ccccc2)=O)C1 CCC(CC)C(C(=O)N(CCCCN(C)C(C1CC1CF)=O)C)OC C1(NC(C(CC)OC)=O)CC2CCC1C2.c1(C(=O)N)ccc(F)cc1.C(C)=O C1(C2CCCOC2)(NC(=O)C2=CCN(C(c3cn(C4CC4)nn3)=O)C2)CC1 C(=O)(CC(C(F)(F)F)NC(=O)CCC1CCCN1C)NCc1nnn(CC)n1 c1(CC)n[nH]c(CC)c1CC(N1CCC(C)C1)=O.c1(CC=O)ccc(Cl)cn1.N C1(CNC(CCSCC)=O)(OC)CCN(C(c2cc(C)oc2C)=O)C1 c1(C(N2CC(NC(c3ccccn3)=O)C(F)CC2)=O)cnc2ccsc2c1 N1(C(CNC(=O)NC)=O)CCC(O)(C)CC1.C1(C=O)CCN(CC(F)F)CC1 N1(CC(=O)NC(C2CCN(C(CCC3C(C)C3)=O)C2)(C)C)C(=O)CCCC1=O C1(C(=O)NC(C2N(C(CSCC)=O)CCC2)C)(OC)CCCOC1 N1(C(C2CCC(C)CC2)=O)CCN(C)CC1CNC(=O)Cn1cccnc1=O N1(C(C(CC)(C)OC)=O)CC2CN(C(=O)CN3CCC(C)(C)C3)CC2C1 c1(-c2cccc(C(N3C4CC(C(=O)OCC)C3CC4)=O)c2)coc2ccccc12 C1(c2cn(C)nn2)CCCC(F)(F)C1.c1(C(=O)NCCCOCC)ccccc1 N1(C(C23N(C(CC=C)=O)CC(CO)(C2)C3)=O)CCNC(=O)CC1C N1(C(C(C)S(C)(=O)=O)=O)C(C)CC2CCCC12.c1cccc(F)c1.C1(C=O)CC1 C(=O)(N=c1cc[nH]cc1F)C1(C)CN(C(c2csc(Cl)n2)=O)C1 N1(C(C2(C)CC2(Cl)Cl)=O)CCC2C(NC(=O)Cc3cccnc3)C2C1 c1(CC(N2CCC(N(C(=O)CCc3ccsc3)CC)C2)=O)c(C)nc(O)nc1O N1(C(CC2C(C)C2)=O)CCC(C)(NC(=O)CCN2CCP(C)(=O)CC2)CC1 c1(C(C(=O)NCC2CCCN2C(=O)CCC2CC2)N(C)C)ccccc1Cl C(=O)(C1CCCn2ccnc21)NC1C(C)CN(C(=O)C(c2ccc(Cl)s2)=O)C1 CCC(F)(F)C(C)(C)C(=O)NCCCC1CCCCN1C(=O)C=CCCC(C)C CCS(=O)CC(=O)OCC1CCN(c2nccc(OC3CCOCC3)n2)CC1 Cc1[nH]nc(Cl)c1C(=O)NCC1CCCC1.c1(C=O)cccc(C(F)(F)F)c1 c1(OC)ccc2c(c1)CCC(C(=O)NCC(O)CNC(c1cc[nH]n1)=O)C2 C1(NC(c2cc(OC(C)C)ncc2)=O)CCC12CN(C(=O)C(O)c1cnc[nH]1)C2 N1(C(c2c(C)cnc(C)n2)=O)CC2CCCN(C(=O)CCc3cnn(C)n3)C2C1 N1(C(CCc2cccc(OC)c2F)=O)CCC2(CC1)CC2NC(C1(O)CC1)=O C(=O)(CCC(C)NC(C1(C(N)=O)CCC1)=O)N(CCn1ncc(C)c1)C CCCCCCCCC(=O)NCCOCCCNC(=O)C(CCCC)N(C)C N1(CC(=O)NC2CN(C(C3CCC(C)S3)=O)C2)CCCOC1=O C(CCCCC(=O)NC(C)(C)CN1CCN(C(=O)CNC(N)=O)CC1)OC c1(C(=O)OC)cc(N2CCC(NC(=O)C=CS(C)(=O)=O)C(O)C2)nc(Cl)n1 N1(C(c2ccc(-c3cscn3)nc2)=O)CCN(C(C2CCCS2)=O)C(CF)C1 C1(N(C(C2CCN(C(c3c(CC)ncs3)=O)C2)=O)C)CCC2(CC1)CC2 N1(C(C(C2CN(C(=O)CCc3ncccn3)C2)OC)=O)CCC(CSC)C1 c1(C(=O)NCC=CCNC(C2C(CC)OCC2)=O)cn(C)nc1OC c1(OCC)sccc1C=O.c1(C(N(CC)C(C)C)=O)ccon1.NC.N Cc1cc(O)cc(=O)n1CC(N1CCCC1CCNC(=O)CCc1nccs1)=O Cc1cc(C(=O)N(CC(O)CN(C)C(c2cnoc2C(C)C)=O)C)c(Cl)cc1N CC(C)CCC(F)C(=O)N(CCNC(c1cc2c(s1)CCC2)=O)C(C)C N1(C(COC(C)C)=O)CCSC(C(N2CCOC(O)C2)=O)C1 C(=O)(CCCF)N(CC(C)C)CC(=O)N(C1CCOC1)C c1ccc(F)c(Cl)c1F.Cc1cccc(C(N)=O)c1NC(C1CCC(NC)C1)=O c1(OC)ccc(C(CF)Nc2nccc(-c3ccnn3C)n2)cc1 CCCCC(CN(C(=O)C1=CCC(NC(c2cnc(NC)cn2)=O)C1)C)CC C(=O)(C(CC(C)(C)C)O)NCC1(CNC(C2CCN(C)C2)=O)CCCCC1 C1(NC(CC2CC(N(C)C)C2)=O)CN(C(=O)C(CCO)N(C)C)C2(CCCC2)C1 C1(C(=O)N)CCCCC1.Cc1cc(C(F)(F)C(=O)NCC(O)C)cs1.C(N)=O c1(CC)nnc2n1CCCC2C(=O)N(CCN(C)C(C1(Cl)CC1)=O)C(C)C c1(C(=O)OC)ccc(C(c2nnnn2CCSC)NC2CCCN2C)s1.C c1(CNC(C(C)N(C(C2(C)CC=CCC2)=O)C2CC2)=O)ccc(C#N)cc1 c1(C(=O)NC2CC(NC(C(C)OCCC=C)=O)C2)ccc(C=C)cc1 C(CNC(=O)CC1CCC(C)CO1)(CC)(CC)NC(CN(CC)CC)=O C1(NC(C2CCOC(=O)CC2)=O)CCCC12CCN(C(C1CC(O)C1)=O)CC2 N1(C(C(C)N(C(C2(OC)CC(C)C2)=O)C2CC2)=O)CC(O)C(N=[N+]=[N-])C1 C1(S(N)(=O)=O)(C(=O)NC2C3CN(C(c4n(C)nnc4)=O)CC32)CCC1 C(C(C)(CC(C)C)NC(=O)CN1CCC1C)NC(C=CCC)=O C1(CCCC)CCC(NC(c2ccoc2Cl)=O)CC1.C12(CCOC1)C(=O)NC2 CC(CCCc1ccccc1)C(=O)NC1CCN(C(C2CN3CCN2CC3)=O)C1 c1(N2CCC(C=C)(COC)CC2)ncnc2c1cnn2Cc1ccc(Cl)cc1Cl Cc1nsc(Br)c1C(=O)NCC1C=CCN1C(c1ccc[nH]1)=O C1(NC(CCc2onc(CC)n2)=O)C=CCN(C(c2cnc(C(C)(C)C)o2)=O)C1 C1(C(N(C)CC2CN(C(C(C)NC(N)=O)=O)C2)=O)CCCOC1 c1(C(=O)NC(C(C)C)CNC(=O)C(C(C)O)N(C)C)cc([N+](=O)[O-])cnc1N N1(c2n(CCOC)c(Cc3ccc(Br)c(F)c3)nn2)CC2(CCCCCO2)C1 c1(C(N2C3CCC(CNC(=O)Cn4nccn4)(C3)C2)=O)cncc2ccccc12 c1(C(C(=O)NC(CNC(c2cc(CC)on2)=O)C)(F)F)ncccc1C C1(NC(Cc2ccn(CC)n2)=O)C=CCN(C(C2CC2F)=O)C1 Cc1cc(Cl)c(Cl)cc1NC(=O)CC1COCCN1Cc1ccc(Br)c(C#N)c1 C(=O)(CCC(=O)NC1(C)CCN(C(c2cnn(CC(F)F)c2)=O)C1)NCC C1(CNC(C2C(C)CC2)=O)(NC(C2CC(O)C2)=O)CCCCC1 C1(CC(N)=O)(NC(C2CC(O)C2)=O)CCN(C(=O)C(=O)NC2CC2)CC1 O=C1COC(CNC(C2CCN2C(=O)CCN2CCOCC2)=O)CN1 Cc1ccc(C)c(C(=O)NC2CCCCC2CNC(c2occc2C)=O)c1 C1(NC(CC=CC=C)=O)CCC2CCN(C(=O)C(F)=C3CCC3)C1C2 CC1(C(N2CCCC(O)(CNC(C3CCCCC3O)=O)C2)=O)CC2(CCC2)C1 N1(C(C=CCOCCOC)=O)CCCC(CC(=O)NC2CCC2C=O)C1 CC(C)CC(CC(=O)NCC1(NC(c2cocn2)=O)CCCC1)CC(N)=O C(=O)(C(F)C(C)(C)O)NC(C)CCNC(=O)CCc1nnc(C2CCCC2)o1 c1(NC(C(=O)NC(CC)(C)C)=O)cc([N+](=O)[O-])c(C)cc1Cl CC1(C)CC(C(=O)NCC2(F)CCOC2)CCN1C(=O)CCc1ncccn1 C1(NC(C(Cn2ccc(C)n2)C)=O)CC12CCC(NC(=O)C(F)(F)CO)CC2 N1(C(CC2CN(C(C(C)C)=O)C2)=O)Cc2cc(Br)cnc2C1 CC1(C)C2CCC(CCNC(C3(P(C)(C)=O)CC3)=O)C1C2 c1(OC)cncc(C(=O)NC2CCN(C(c3cnnc(C4CC4)c3)=O)C2)c1 CC(C)C(C)CNC(=O)OC(C)(C)C.c1(C=O)nccnc1C(C)(C)O N1(C(c2cnc(CC)nc2)=O)CCCCCCC1C(=O)NCC(O)C(N)=O C(=O)(C(C(C)NC(=O)CN(C)C(=O)OC)C(C)C)N1CC(=CCC)C1 C(=O)(C(F)CC(C)C)NC1(CCCNC(c2c(CCC)occ2)=O)CC1 Cc1ccc(O)cc1C(=O)N1CCC(C(=O)NCC(O)C(F)F)O1 c1(C(=O)NC2(CNC(C(C=C)O)=O)CCOC2)cccnc1N1CCCCC1 c1(C(N2CCC(C)C(NC(c3nnc(O)nc3O)=O)C2)=O)ccc2c(c1)OCO2 C(C(=O)N1CCC(CO)(NC(=O)CC2(C)CC(F)(F)C2)C1)(C(C)C)OC C1(CNC(C(COC)(F)F)=O)CC2(CO1)CN(C(c1ccccc1CO)=O)C2 N1(CC)CCOCC1C(N1CCCC(NC(C2CN(c3nncs3)C2)=O)C1)=O c1(-c2n(CC)c(N(C3CC3)CC3CCCO3)nn2)ccc2nn[nH]c2n1 N1(C(C(OC)OC)=O)CCN(C(C)=O)C(CCO)C1 c1(C(=O)NC2CC(C(=O)NC3C(C(=O)OC)CCC3)C2)ccc(C)cn1 CC1CN(C(=O)C=CCO)CCCN1C(c1occ2c1CCCC2)=O c1(C(=O)NCC2CN(C(c3c(NC)scn3)=O)CC2O)ncc2ccccn12 C=CCCCCCCC(=O)NCC1(NC(c2cc(O)n(C)n2)=O)CCC1 c1(CC)nccnc1C(=O)NCCC(C)N(C)C(c1cnoc1C1CCC1)=O C1(C(N2CC(C(=O)NC)C2)=O)CC2CC1CC2NC(C1CCOCC1)=O CC(N=[N+]=[N-])C(=O)NCCn1cnc(C(=O)NC(CO)C2(C)CC2)c1 c1(NC(C2(c3ccc(C)n(C)c3=O)CC2)=O)ccc(O)c([N+](=O)[O-])c1 N1(C(c2c(C)n(C)cc2)=O)CCC(NC(c2cc(C(C)(C)C)nn2C)=O)CC1C C=CCC(CC=C)C(=O)NCC1CC1.C1(CC(=O)NC)COC(C)(C)CO1.C N12C(C3CCCC13)CC(=O)O2.c1(OC(C)(C)C)nc(Cl)ccc1C(N)=O c1(CC)cc(C(N2CCC(CNC(c3ccncc3Br)=O)C2)=O)ccn1 c1(C(=O)NC(C2CCCCC2)CO)nnc2n1CCOC2 CCCCC(F)C(=O)NC(C)(C(=O)NCc1ccc(Cl)nc1)C1CCC1 CCC(C)(C)C(O)C(=O)N1CC(C(N)=O)(C)C1.c1(C(=O)N)ccc2sncc2c1 CC(CCC(=O)NCc1ncn(C)n1)NC(=O)CCn1cnnn1 C1(C(=O)NC2C(OC)C2)C2CCC(C2)N1C(=O)Nc1nc(C)ccc1Br N(C(=NCCc1cccc(OC)c1)NC1CC1C)CC1(CC)CCOCC1 Cc1ccccc1C(F)(F)C(=O)NC1CC(CC)C1.C1(C)(C(=O)N)CC=CC1 CC(c1cccc(Cl)c1)=CC(=O)NCC1CC(C)N(C(c2ccnc(Cl)c2)=O)C1 C1(C(=O)OC)CCCC(COc2nccs2)O1.N12CC(O)(C1)SCCC2=O Cc1cnc(NC(CNC(=O)CC2COC(C)(C)C2)C(C)C(C)C)nc1O c1(OC)c(C=O)csc1NC(C1CN(CC)CCO1)=O.c1(C=O)conc1C.O C(N=c1[nH]c(=NCC(C)c2ccccc2)c2[nH]ccc2[nH]1)C1N(CC)CCCC1 N1(C(CSC)=O)CCN(C2CN(C(c3ccnc(-c4ncc[nH]4)c3)=O)C2)CC1 c1(CNC(C(CNC(C(C)C#N)=O)C)=O)ccc(O)cc1F C(=O)(C#CC1(C)CCCO1)NC(CCCC)C(=O)NCC1COCC(C)O1 C(=O)(CC1CCc2ccccc21)N1C(CNC(CCCCCSC)=O)C=CC1 c1(N(C(C(CC#N)N)=O)C2CC3CNC2C3)ccc2nc(CO)[nH]c2c1 C1(NC(C2CCC(CC)C2)=O)CCN(C(c2cccc(N)c2C(F)F)=O)CC1O c1(C(N2CC(NC(=O)C=CCCC(C)C)CC(OC)C2)=O)cc(C#N)ccc1Cl N1(C(CN(CCOC)C(c2csc(C#N)c2)=O)=O)CCOC(COC)C1 n1(NCC(n2cc(C3(C4CC4)CC3)nn2)C)cccc(CC2COC(=O)O2)c1=O c1(C(=O)NCCNC(c2cc(C3CCC3)on2)=O)cccc2c1CCS2(=O)=O n1(CC(=O)N)nnc2ccccc12.c1(OC)nc(C)ccc1C(=O)NCC(O)C Cc1cccc(C)c1C(=O)NCCC(C)CC.c1(C(=O)N)c[nH]cc1C(C)(C)C c1(C(=O)NC(C(=O)NC(c2cccs2)C)Cc2cc[nH]n2)ncc(F)cc1N CC(C)(Cl)C(=O)NOCC(=O)NCC1CC1Cl N1(C(Cc2cccc(OC)c2)=O)CC2(CCCN2C(=O)C(C)S)C1 N1(C(CN(C)C)=O)CCN(CCCC2CCCN(C(C34CCC3CC4)=O)C2)CC1 C1(NC(C(N2CCOCC2)C)=O)C2CN(C(c3ccc(CC(C)(C)O)s3)=O)CC12 C1(C(=O)N)CCN(c2ccncc2)C1.C(C(C)C)N(C(=O)CCC1CC1(F)F)C CCC(C)CC(C(=O)NOCc1nc[nH]n1)NC(=O)CCc1ccncn1 CC(C)(C(=O)NOCC(=O)NC1CCCCC1=O)c1ccc(C(F)(F)F)cc1 c1(CNC(COCCC=C)=O)conc1C(=O)NCC(C)(CC)SC c1(C(N2CCC(C)C(O)C2)C(=O)N)cc(C(F)(F)F)ncc1F.CC1(CC)CC1 C=CCCCCC(=O)NC(C)(CNC(c1c(C)nsc1C)=O)C1CC1 c1(C(N(C2CC(C(=O)NCCC(C=C)(C)C)C2)C)=O)cc(C)c(C)nn1 C12(C(=O)NC(C)CC3(O)CCC3)CCC(C1)C(F)(F)C2 N1(C(CCCCC)=O)CCC(CC(=O)NC(CCO)C2CC2)C1(C)C Cc1cccc2c(C(N3CC4CC(O)C3C4NC(=O)CC(C)(C)C)=O)coc12 c1(C=O)[nH]nc(C2CC2)c1Cl.C(C)(C(=O)NC(C)C1CCC1)OCC=C.N C12(CNC(CCCOCCC)=O)CC(CN1C(C1(c3cc[nH]n3)CC1)=O)C2 C12(C(=O)NCc3ccc(C#N)cc3)CCCC1CCN2C(C1CC12CCC2)=O C=CCCN=C(NCCc1cccc(OC)c1OCC)NCC1CNC(=O)C1 C1(NC(CCC2N(C)CCC2)=O)CN(C(C2CCCC(O)C2)=O)C2(CCC2)C1 C(=O)(C(O)CC(C)(C)C)NCC1N(C(CC(=C=C)C)=O)CCC1CC N1(C(CS(CC)(=O)=O)=O)CC(NC(c2cc(F)ccc2F)=O)C2CCCCC12 c1(C(N2CC3C(CNC(C(COC)(C)O)=O)C3C2)=O)cnn2c1C(=O)NCC2 c1(C(=O)NCC2CCCC(NC(c3sccc3Cl)=O)C2)cc2cscc2s1 C1(O)(C(N2CCC(NC(CC(C)C(F)(F)F)=O)C2)=O)CC2(CCOCC2)C1 c1(NC(C)C)ccc(C(=O)OC(C2(C)CN(C(C(CC)C)=O)C2)=O)n1C N1(C(C(=O)NCC=C)C)CCC2C(CCCN2C(=O)C(Br)=CC)C1 c1(C(=O)NC(C2CCN(C(=O)CCc3cncn3C)C2)C)cccc2nsnc12 C(C(COC)CC(=O)NCC(=O)N(C(C)C(C)(C)O)C)OC C=CCCCCCCCCC(=O)NC(C)C(C)(C)NC(c1cncc(F)c1)=O N1(C(c2ncccc2Cl)=O)CCC(O)(NC(c2ccccn2)C2CC2)CC1 CC(C)(F)CCC(=O)NC1CCCC1CC(=O)NCCC1(O)CCCC1 c1(C(=O)NC(C(C)NC(C(C)NC(C)=O)=O)C)c(C)ccc2nsnc12 CC(C)C(C(=O)NCC(CC(F)(F)F)NC(C1CC2(CCC2O)C1)=O)C(C)C CC1(C)CC(=O)N(CC(=O)NC2(C)CC(NC(C3CC3(F)Cl)=O)C2)O1 C(C(F)(F)CCC(=O)NC1CCCSC1)n1cc(C(C)(O)CCO)nn1 C1(NC(C2CC(C)C2)=O)COCCC1NC(c1ccccc1-c1cc[nH]n1)=O c1(OCC(N2CCCC2C(=O)NCc2cc(Br)cs2)=O)ccccc1 C(C)(C)(CCNC(=O)C1=CCC1)NC(C(c1ccccc1)OC(C)C)=O c1(C(N2CCC(F)(C(=O)NC(C)CCO)C2)=O)cc(F)c(F)cc1O CS(=O)(=O)c1cncc(C(=O)NC2CCOCC2NC(C2CC2(Cl)Cl)=O)c1 Cc1nnc2n1CC(C(=O)NC1C3CN(C(=O)C#CC(C)(C)O)CC13)CC2 c1(OCC)cc2ccccc2cc1C(=O)N.C(C1CCOC1)=CC(N1CCC1)=O C1(NC(C2(C(C)C)CCC2)=O)C=CCN(C(=O)C=C2CCN(C)CC2)C1 c1(C(N(CC(C)C)C)=O)cc2c(C)c(C)ccc2[nH]1.C#Cc1ccc(C(=O)N)o1 C1(NC(c2cn(C)nc2C2CCCO2)=O)CN(C(C2CC=CC2)=O)CC1N=[N+]=[N-] c1(OC(CC)C(=O)NCC2CN(C(=O)CN3CC(C)C3)CC2O)ccccc1C C#Cc1cc(F)c(C(=O)NC(C2CCCN2C(c2ccccc2Cl)=O)C)c(F)c1 N1(C(c2c(C)nsc2)=O)CC(C(=O)NC2(CCF)CC(O)C2)CC(C)(C)C1 O=S(=O)(c1ccc(N(CCCSc2ccc(Cl)cc2)CCO)cc1)N1CCCC1 C1(C(N(CCC)C)=O)COc2cc(Cl)ccc2C1.c1(COC)ncc(C=O)s1.N C12(C(=O)NC3(CC=C)CN(C(c4ccccc4Cl)=O)C3)CC(C)(C1)OC2C.S c1(N(C(=O)C(C2CC2)NC(=O)CC2CCSC2)CCN(C)C)ccccc1 C1(CNC(c2ncn(C)c2)=O)CCCCC1NC(c1csc(O)n1)=O C=CCC(CCCCC)C(=O)N1CC(CO)(NC(=O)CCCNC(N)=O)C1 C=CC1(C(=O)NCc2c[nH]nc2)CCN(C(=O)C(CN(C)C)N(C)C)C1.C C1(NC(C2CC(C(F)(F)F)(OC)C2)=O)CCSC12CN(C(C1CCC1)=O)C2 N1(C(CN(C)CC2CCCCC2)=O)CCC(c2cnco2)C1 N1(C(C2(NC(=O)CN3C(=O)CNC3=O)C(C)C2)=O)CCn2cnnc2C1 C1(CC(=O)N(CCCn2cc(CNS(C)(=O)=O)nn2)C)CCC(C)CC1 N1(C(C2(F)CCN(C(C(n3c(C)ccn3)C)=O)C2)=O)CCC2(CCOC2=O)C1 S(=O)(=O)(c1ccc(C(=O)NCCCNC(=O)CC2OCCC2C)o1)NC N1(C(CCCNC(N)=O)=O)CC(F)(F)CC1C.C1(C=O)CCS(=O)(=O)N1.N c1(C(N2CCN(C(C(F)OC)=O)C(C)CC2)=O)ccc2c(c1)COC2=O C1(CCC(N2CCC(CCNC(C3ON=C(C)C3)=O)C2)=O)NC(=O)NC1=O c1(CNC(C(CC=C)C)=O)c(C)nc(N2CCN(C(=O)C=CCO)CC2)nc1C N1(C(CSCC(C)C)=O)CCC(OCC(=O)NC2(C3CCCO3)CC2)C1 C1(NC(C2C(C)OCC2)=O)CC1C1CCCN(C(=O)CSc2nncn2CCF)C1 C1(CN)CCCC2(CC(C(=O)NC(c3cccc4ccccc34)CO)C2)O1 C1(CC)C(C(=O)NC(c2nn(C)cc2O)C)CCN1C(c1cnn(C)c1Cl)=O N1(C(CCNC(=O)OC)=O)CCN(C(=O)C=Cc2ccccc2Br)C2CC12 N1(C(C2(CC)CC2)=O)CCCC(F)(F)CC1.c1(C=O)ccn(C)n1.C1CC1.N C=CC(C)(C)CC(=O)NC1CCN(C(c2cc(OC)ncn2)=O)C(C2CC2)C1 N1(C(CC(C)SC)=O)CC(NC(c2cnc(C(C)C)nc2)=O)C(N=[N+]=[N-])C1 N1(C(Cc2ccn(C)n2)=O)CCN(C(C2CC(C)(O)C2)=O)CC1 c1(OC)cc(C)nc(N2CC3CC(Nc4cc(F)ccc4OC)C3C2)n1 C1(C(NC)=O)CCS(=O)(=O)CC1.c1(CCC)[nH]ccc1C(=O)NC1CC1.C c1(C(=O)NCC2N(C(Cc3c(C)ccs3)=O)CCC2C)cnn2c(=O)cc[nH]c12 Cc1ccc(C(=O)NCC(C)CNC(C2(C)COCCO2)=O)n1C c1(C(N(CC)C)=O)cc2n(n1)CC(O)CO2.CN1CCC(=CC(=O)NCC)C1 C1(N(C)C(C2CCCN2C=O)=O)CN(C(c2ccc(CO)nc2O)=O)CC12CC2 c1(C(=O)NC2CC(NC(c3nn(C)c(F)c3)=O)CC2O)c(F)cncc1Br Cn1nncc1C(N1CCCC1C(=O)NCC1(C#N)CC1)=O c1(OC)cc(CN(CCCNC(C2CCCCC2C)=O)C(C)C)ncn1 C1(CCC(N2C(CC)CCC2)=O)CCCCC1.C12(C=O)CC(F)C1C2.C(N)=O c1nccc2ccccc12.c1(C(C)(C)C)nocc1C(=O)NC1CC1.C(=O)(C)N CC1CCN(C(C23CCC(F)(CC2)CC3)=O)CCN1C(=O)CCCN.[SH](C)(=O)=O C1(NC(C(C)OCC)=O)CCN(C(c2cc(=O)n(C)o2)=O)CC1F C1(NC(C(c2cscn2)N(C)C)=O)CCN(C(=O)C=CC2CC2)C1 N1(C(c2ccc(C)[nH]2)=O)CCC(C)(C)CC1C(=O)NC(C)CN1CCCC1=O C(=O)(C(C)CCC(C)(C)C)N1CCCN(C(C2C(CC)C2)=O)CC1CO C1(NC(CONC(C=Cc2cc(C)no2)=O)=O)CN(C)C2(CCC2)C1 CC1CCN(C(c2ccc(C3(C)CC3)cc2)=O)C1CNC(c1cocn1)=O C1(C)(CNC(CC(C)n2ccnc2)=O)CCCN(C(=O)CCOCC(F)F)C1 Cn1ncc2c1CC(CCC(=O)NCCCNC(c1cnc(N)cn1)=O)CC2 C(C(C)(C)C(F)(F)F)NC(=O)NCc1cccc(C(OC)OC)c1 C1(C)(C(=O)OC)C=CCN1C(=O)CCCN(C)C(c1nnsc1C)=O N1(C(C2(CC)CCOC2)=O)CC(NC(=O)CCC(=O)NC)CC(C)C1 N1(C(c2c(COC)nn(C)c2)=O)CCC2(CCCN2C(=O)C(F)CC(C)C)C1 N1(C(CCCOCC=C)=O)CCN(C(C2(CCOC)CCCC2)=O)CC(C)(C)C1 c1(C(C(=O)N(CCn2cc(-c3csc(C)c3)nn2)CC)(C)C)ccccc1C N1(c2cc(N3CCCCC(COC)C3)ncn2)CCC2(CCC(O)C2)C1 c1(C(N(C2CC(NC(=O)C(O)Cn3cncn3)C2)C)=O)ccc(F)o1 C1(C)(C(=O)NC(C#C)C2CC2)CCCN(C(=O)CC2CC(OCC)C2)C1 c1(C(=O)NC2CC(CNC(C(CN(C)C)(F)F)=O)C(O)C2)cnc2n1CCCC2 C1(C(N(C)CCNC(C2CCC3CC2CO3)=O)=O)CC(c2ccccc2F)=NO1 N#CC(C(=O)NCC(F)CNC(c1cc[nH]n1)=O)C1CC1 c1(CCC(N2CC=CC(NC(C(C)N3CCC3)=O)C2)=O)ccc2ccccc2n1 CC1CC(c2cn(CC3CC4CC4C3)nn2)CCN1C(C1CC2CCCC2C1)=O Cc1ccc2c(c1)ncn2CC(=O)N(C)CCN(C)C(C1(CCO)CC1)=O c1(C(C(=O)N(CCCCN(C(C(C=CC)O)=O)C)C)CO)ccc(Cl)cc1 c1(C(=O)NCCC(CNC(C(C)OCCC=C)=O)O)cc(Cl)cc(C)c1N c1(C(=O)NCCC)ccc2cc(NC(C3CCCCC3O)=O)ccc2c1 n1(CC(=O)NC(CCCC)CNC(c2oc(C)cc2C)=O)nc(C)c(Cl)c1C Cc1cc(C)c(C(=O)NCCC(C)NC(C2CC2c2ccn(C)n2)=O)c(S)n1 C1(CNC(C2(C=C)CCC2)=O)C(C)CCN1C(=O)C=Cc1cncn1C c1(C(=O)NCC(CCC)NC(c2ccc(N)cc2C)=O)ccc(F)c(OC)c1F C1(C(=O)NCCCCC2CN(C(c3c(C#N)scc3)=O)C2)COC2COCC12 N1(C(CCC(=C)C)=O)CCN(C(c2cc(C(C)(C)C)[nH]c2C)=O)CC1C1CC1 N1(C(c2nc(CNC(c3c(CC)nco3)=O)oc2)=O)CCCC(C#N)C1 C#Cc1c[nH]nc1C(=O)NC1COCC1C(=O)NC1(C(=O)OC)CC1 CN(C)NC(=O)CCC(=O)N1CCC2CN(C(=O)C3=CCCCC3)C2C1 C12(CC)CCC(C(=O)NC3CC34CCC4)(CC1)CO2.C1(CC=O)CC12CC2 C1(C(=O)NC2C3CN(CC4CC45CCOC5)CC23)CC12CCc1ccccc12 c1(CC)cc(C(=O)NC2CCCC(NC(=O)CC34CCCC3C4)C2)cc(N)c1 c1(CC)nc(C(=O)NC2CCC(NC(=O)CCn3cc(C=O)cn3)C2)cs1 C(C)(CCC(c1nnnn1CC(F)F)Nc1ccc(-n2cncn2)cc1)OC c1(C(=O)NC(CNC(C2C(C=C)CC2)=O)CC)ccc(Sc2ccccc2)cc1 N1(C(CSCC(=O)OC(C)(C)C)=O)CCOCC1.C1(C)(C=O)SCCCS1.C c1cccc(Cl)c1.C(CSC)(C(=O)NCC)OC.C1(C(=O)N)CC1[N+](=O)[O-] c1(N(C2CN(Cc3nc(Br)cs3)C2)C)ccc(C(F)(F)F)cn1 CN1CCC(C(N2CC(F)C2)=O)(NC(C2CCOC2(C)C)=O)C1 C=C1CC(C)(C(=O)NCCOC2CCN(C(c3ccn(CCC)n3)=O)C2)C1 c1(C(=O)NCC(CC(C)C)NC(=O)CCCC#N)c(O)ncc2c1CCC2 C1(F)(CNC(C2(CC)CCC2)=O)CN(C(=O)CC2CC(F)C2)C1 N1(C(c2c(CC)onc2)=O)CCCC2CCN(C(=O)C=CSC)CC12 Cc1nc(C)c(CC(N2CCCC(CNC(=O)CN3CCC(C)C3)C2)=O)s1 C(=O)(CCC(CF)CF)NCc1cc(C(=O)NC(C#C)(C)CC)ncc1 C(=O)(C(C)(C)CS(C)(=O)=O)N(CCCCNC(CC(C(CC)C)O)=O)C C1(NC(C2CCC(NC(C3C(CC(C)C)C3)=O)C2)=O)CC(C)(C)OC1=O N1(CC)CCCC(N=c2[nH]c(=NCC3CC3CO)[nH]c3c2CSC3)C1 N1(C(C=CC2(C)CCOCC2)=O)CCC2(COCC(C)O2)C1.C1(C)(C=O)CC1.N c1(C(N2CCC(CN(CCN3CCCCCC3)CC)CC2)=O)cc(Cl)ncc1Cl N1(C(C2N(C)C(=O)CC2)=O)CCC2(CCCN2C(=O)C2CCc3nccn32)CC1 CC1(C(=O)NC(CC(=O)NCC(O)CF)C2CC2)CCC2CC2C1 N1(C(CCOc2cccc(OC)c2)=O)CC2CN(C(=O)C(C)C(C)C)CC2(C)C1 CC1OCCC1CC(=O)NCCOCCNC(=O)C(c1cccnc1)O c1(C(N2CCC(C(C(=O)NCC(C3CC3)SC)F)C2)=O)ccc(C)nc1 Cc1n[nH]c(C)c1C(=O)NCC1(F)CN(C(c2cccc[n+]2[O-])=O)C1 CC(C(=O)N1CCN(CCN(C(=O)CCOCC2CC2)C)CC1)P(C)(C)=O C=C(Cl)CCC(=O)NC1CC(O)(CNC(=O)COC2(C)CCCC2)C1 N1(S(c2c(CC(=O)OC)ccc(Br)c2)(=O)=O)CCC2(CCCC(C)(C)C2)C1 C#CCCCC(=O)N(C)CC1(O)CCN(C(C2(C#C)CC(=O)C2)=O)C1 N1(C(c2n(C)ccn2)=O)CCC2(NC(=O)CCc3cc(F)ccc3Br)CCCC12 Cc1ccc(F)c(N)c1C(=O)N(CCCC)C.c1(C(=O)N)nc[nH]c1C(C)(C)C N1(C(CC2C(=O)OCC2)=O)CC2C=CC1C(C(N1CCC(F)(F)CC1)=O)C2 c1(C(N(C)C)=O)cc(C)c(O)c(C)c1.CC1=CC(C(=O)NC2CCCC2)SC1 C(=O)(CCCCCC(C)O)N1CC=C(CNC(CCC(C)OC)=O)CC1 C1(C(=O)Nc2cc(OC)cc(F)c2)N(C(=O)CCc2nncs2)CC12CCCC2 Cc1nn(C)c(C)c1OCC(=O)N.C1(C=O)CCC(=O)N(C2CC2)C1.CCC CC1(C)CC(CC(N2CCC(CNC(=O)CCc3ccc(=N)[nH]c3)C2)=O)CO1 c1(CN(C(=O)Nc2cnc(CC)s2)C)cnc2ccc(Cl)cn12 N1(C(c2c(C)sc(O)n2)=O)CCC(NC(=O)C(C)N2CCCC2)C(CO)CC1 c1(C(=O)NCCN(CCCCCC)C(=O)C(C)O)cc(C(=O)O)ncc1F.C c1(C(C(=O)NCCC)N(CC)Cc2ccc(Cl)cc2Cl)c(C)nn(CC)c1C C1(CC(=O)OCC2N(C(=O)OC)CCC2)CCN(S(C)(=O)=O)CC1 c1(CC)nc(C(=O)N(C2CCCN(C(=O)C(c3ccnn3C)O)C2)C)c(C)o1 N1(C(CC=C)=O)CC(NC(c2ccsc2C(=O)OC)=O)CCC1C C12(CNC(C(Br)=C(C)C)=O)CC(NC(=O)CCc3ccncc3)(CO1)C2 C(CCC(O)C(=O)NCP(C)(C)=O)NC(C(CSC)OC)=O C(=O)(C#CC1CCCCC1)NC(CCC)C(=O)N(C)CC1COC(=O)N1 c1(CC(CC(=O)NCCSC(F)F)NC(CN(C)C)=O)ccc([N+](=O)[O-])cc1 N1(C(CC(C)n2cccn2)=O)C2CCC1C1CC1(NC(=O)Cc1cscn1)C2 c1(CC)cccc(C(=O)NC2CC(C)(NC(C3CC(C)CO3)=O)C2)c1 CC1CCN(C(C2CCCC2)=O)CC1NC(=O)Cc1cncc(F)c1 c1(OC)ccc(C(=O)C(=O)NC(C)C(C)C)cc1.C1(C=O)CC=C(C)CC1.N Cc1noc(C)c1C(=O)NC1CCOCC1NC(=O)C(c1ccccc1F)C Cc1ccc(Br)cc1C(N1CCOCC(NC(=O)CC(C)n2ccnc2)C1)=O C1(C(=O)NC2(CNC(=O)CCc3ccncc3F)CCCC2)CCC2(C1)N=N2 C1(NC(C(C(C)C)OCC(C)C)=O)C2CC1CN(C(c1cccc(N)c1F)=O)C2 C1(NC(CSc2n(C)cnn2)=O)CCN(C(c2cc(N)nc(Cl)c2)=O)CC1F N1(C(c2c(C)cc(OC)nc2)=O)CCN(C(=O)CCOCCS)CC(C)(C)C1 C1(NC(=O)NC(C)C)CCCN(C(c2ncccc2Br)C(=O)N)C1.CCC1CC1 c1(NC(C(=O)NCc2scc(C)c2)=O)cccc2c1OCCC2=O C1(C(=O)NC2C(OCC)COC2)CC(F)(F)CN1C(c1cccc(Cl)c1)=O C(=O)(C1CN(CC)c2ccccc21)NCCCN(C(c1ccccn1)=O)CC C1(C(=O)NC(c2nc(C3CC3)no2)CC)COC2CN(C(=O)C(C)O)CC12.C C1(n2cc(C(=O)OC)nn2)CON(C(=O)CC2COCCO2)C1 c1(C(=O)NC(C(C)NC(C2(CC#C)CCCO2)=O)CO)c(C)ccc(F)c1O C(C(=O)N1CC(NC(=O)Cn2nc(C)nc2C)C(F)C1)(C(C)C)OC C1(O)(SCC(CO)SCCOC(c2ccn[nH]2)=O)CCOCC1.c1ccco1 c1(OC)ccc(C(C)C)cc1CN(C)C.C1CCCN(C(C2CC(O)CN2)=O)C1 Cc1cc(C(N2CC(F)(CNC(=O)CC(C)(C)O)C2)=O)cc(C)c1 N1(C(c2nc(C#C)sc2)=O)CC=C(CCNC(=O)C(=Cc2cccs2)C)CC1 N1(C(C(=O)NCCC)C)CCC(C2CCN(C(=O)Cn3ccc(C)n3)CC2)C1 C1(NC(=O)CN2CC3CCC2C3)COC2(C1)CN(C(=O)CS(=O)(=O)C1CC1)C2 c1(N2CCN(c3scc(C)n3)CC2)cc(C)[nH]c(=NCCC2COCC(C)O2)n1 CC1(C)CCC(CNC(=N)NCc2nccn2C2CC2)O1 c1ccccc1.c1(CCCOCC(C)(C)NC(=O)NC2CC2)cccc(F)c1 C1(C(N2CC(C(=O)NC(C#CC#C)(C)C)C(CC)C2)=O)CN2CCN1CC2 CCCCCC(C)CC(=O)NC1CC2(C1)CC(NC(C1CC1C(C)(F)F)=O)C2 C1(NC(CC2(OC)CN(C(C3(C)C=CCC3)=O)C2)=O)CCc2c[nH]nc2C1 c1(CC)cncc(C(N2CC3C(NC(=O)C=CCN(C)CC)C3C2)=O)c1 C1(C(=O)NC(C)Cc2ccno2)CCCC1NC(=O)C(C)Sc1ccccn1 C1(NC(C(C)CF)=O)CN(C(c2ccc(CSC(F)F)o2)=O)CC12CC2 C1(C(=O)O)C2CC2CN1C(=O)C(c1cccc(C(F)(F)F)n1)(F)F C1(NC(CC(CC)SC)=O)CN(C(c2ccnc(Cl)c2OC)=O)C(C)(C)C1 N1(C(C(N2CCC(C)C2)=O)=O)CC2(CC(NC(=O)Cn3cc(Br)cn3)CO2)C1 Cc1ccc2[nH]nc(C(=O)N(C)CCNC(=O)CCC(=O)c3cnn(C)c3)c2c1 Cc1c(C(=O)NC2CC(C)N(C(=O)CSCc3cccs3)C2)nn(C)c1N c1(C(C)C)nocc1CNC(=O)Cn1cc(-c2cncnc2)nn1 N1(C(C(C(=O)OC)C)=O)C(C(N2CC=CCC2)=O)CCC12CC2 c1(C(=O)N)c(O)cccc1Cl.N1(Cc2cc(C(=O)OCC)[nH]c2)CCC(F)C1 N1(C(c2ccc(C)cc2O)=O)CCCC1C1CCCCN1C(=O)CCC1CCC1 N1(C(c2ccc(C)nn2)=O)CC(C(N2CCSCCC2C)=O)C(F)(F)C1 c1(COC)nc(C(=O)NCCO)cs1.C1(C(N(CC)C)=O)CCC2CC12 C(CCCN=c1nc(N(C)CC2CCCO2)c2ccccc2[nH]1)N(CC)CC C12(C(C)(C)C)CCN(C1)C2.C1(C(=O)O)(NC(=O)NN)CC1 N1(C(c2sc(CC)c(C)c2)=O)CCC(NC(C23CCC2C3)=O)C(F)C1 C1(OC)(CNC(c2cnc(C)[nH]2)=O)CCN(C(c2cc(Br)oc2C)=O)C1 Cc1c(CC(N2CCC(N(C(=O)CSC(F)F)CCO)C2)=O)cnn1C N1(C(c2c(C)scc2)=O)CCC(NC(=O)Cc2ccc(C(F)F)cc2)CC1C Cc1c[nH]c(=NCCC2CCN(C(C3CC(O)C3)=O)CC2)nc1C c1(CC(=O)OCc2cnn(C(F)(F)F)c2)c(F)ccc(Cl)c1Br c1(OCC)ccc2cccc(CNC3CCC(N)CC3)c2c1 c1(COC(c2c(F)ccc(OC(C)C)c2)=O)ccc2c(c1)C(C)C(C)O2 C(C(O)C(=O)N(CC(=O)NCc1n[nH]c(CC)n1)CC)=CC C(C)(N=c1cc(C)nc(N(C)Cc2ccccc2Cl)[nH]1)c1c(C)ncs1 C1(C)(C(=O)NCc2n(CC)cnn2)CCN(c2ccc(C)nn2)CC1 c1(C(=O)NC2CC(CC(=O)NCCc3cccnc3O)C2)cnc2n1CCC2 CC(C)(CCCNC(C1(O)CC1)=O)NC(=O)CN1CCNC(=O)C1 c1(-c2c(C)nc(F)cc2)ccc2c(CC(=O)NCCc3ccncc3)n[nH]c2c1 C1(N(C(CNC(C(CC)C)=O)=O)C)CCN(C(=O)C(C)C(F)F)CC1 N1(C(CC2N(C(C)C)CCC2)=O)CCOCC(NC(C2CCC2C#N)=O)C1 N1(C(c2ccc(CC)[nH]2)=O)CCCCC(C(=O)NC2CC(C)CCC2O)C1 C(C)(C(=O)N(CCO)OC)N(C(c1cc(CCC)on1)=O)C(=O)C1CC1 C(C#Cc1ccc(I)cc1)Nc1cn(C)nc1-c1ccc2cccnc2c1 N1(C(c2cnc(CC)nc2)=O)CCN(C(c2cnc(OC)s2)=O)C(CO)C1 C12(C(N(C)CCc3cccs3)=O)CCC1CN(C(=O)CN1CC=CC1)C2 CC12CNC(C(=O)NCC3CCN(C(=O)C(F)(F)F)C3)(C1)C2 C12(NC(c3nc(CC)oc3C)=O)CCC1CN(C(=O)CN1CCOCC1)C2 C12CCC(c3cn(C(C)C(=O)O)nn3)(CC1)CC2.C(=O)(CC(C)(C)C)NCC c1(C(=O)N)cnc2cccnn12.C12(COC)CC(CN1C(C1CCCC1C)=O)C2 Cc1ccc(C(N2CCCCC(N(C)C(C3CC(F)(F)CS3)=O)C2)=O)cc1O CC(C)(C)C(=O)N(CC)C(C)C.C(=O)C(F)(F)CC1CCCO1.CCC.C CCCC(C(=O)N1CCC(CNC(=O)C#CC2CC2)(COC)C1)OCC C#Cc1cncc(C(=O)NC2CCCN(C(C3CCC(=O)NC3)=O)C2)c1 C(CCCCC(=O)NC1CCC(CNC(=O)CC)CC1)NC(N)=O.C1COC1.O C1(CCC(=O)NC(c2ccccn2)C)CCN(C(C2(N(C)C)CC2)=O)C1 c1(C(=O)NC2COCCN(C(C3(C)CCC(C)C3)=O)C2)cccc2ncccc12 n1(CC(N2C(CNC(C)=O)CC2)=O)nnnc1Cn1nccc1C(=O)O N1(C(c2cnc(CC)[nH]2)=O)CCC2(CC(NC(=O)CO)CO2)C1.c1nc[nH]n1 c1(C(=O)NCC#CCNC(C(COC)C)=O)cccc(OCC(=O)OC)c1 Cn1cc(C(=O)NC2CCCCC2)cc1S(N)(=O)=O.C1(C=O)CC2(CC2)C1.C C(=O)(C(C)(C)C(F)(F)F)NC1CCCN(C(c2c(N)cc(CC)c(F)c2)=O)CC1 c1(CC(=O)NC(CC)CN(C(=O)CCC=CC(C)C)C)coc2cc(F)ccc12 c1(NC)cnc(C(=O)NC2CCN(C(C3CC3c3ccn(C)n3)=O)C2C)cn1 CC1(C)CCC=C(C(=O)NCCC2CC(NC(c3csc(Cl)n3)=O)C2)C1 Cc1cc(C(N2CC(NC(C3CC(C)C3)=O)C(C)(C)C2)=O)ccc1Br CC1(CCO)CCN(C(C2(C)CCN(C(C3CC3(F)Cl)=O)C2)=O)C1 N1(C(C(C)OCC)=O)CCC2(CC1)OC1(C)CC2C1.C(=O)C1=CCC(C)CC1.N N1(c2nnc(C(C)C)o2)CCCC(CCNC(c2ccnc(O)c2)=O)C1 Cc1ccc(C(C)OC(C2(C(F)F)CCCO2)=O)c(Br)c1 CCC(C(=O)NC1(C)CN(C(=O)COc2ccsc2Cl)C1)SC C1(N(C(C(C)C#N)=O)C)CCN(C(=O)CN(c2ncccn2)C)CC12CC2 C1(NS(CCC)(=O)=O)CCN(N2CCC(c3n[nH]c(C)n3)CC2)CC1 c1(C(=O)NC2C(C(=O)NCc3c(F)cncc3Cl)CCC2)ccc2c[nH]nc2c1 C(C(=O)N1CCCC1C)(C(C)C)N(CC)CC.c1(C(C=O)=O)csc(=N)[nH]1.N C(=O)(C#CC1CCOC1)N(CC(C)O)CCNC(=O)CN1C(=O)CCCC1=O C1(NC(C(CC)COC)=O)CCC(C)(CNC(c2cnoc2C)=O)CC1 c1(OC)ccc(CCC(C)NCC2CC3CCC2C3)cc1OC CC1CN(C(c2cn(C3CC3)nn2)=O)CC1CCNC(=O)CC.C(=O)C=CCl C(=O)(CN=c1cc[nH]cc1)NC1C(CNC(c2cn(C)c(Br)c2)=O)COC1 CC(C)CCCNC(=O)Cn1cnnn1.c1(C(=O)N)ccnn1CCN(C)C N1(C(c2ccc(OC)cc2)=O)CCC(C)(NC(=O)COC)CC1.C1CCOC1 C1(NC(c2cccc(Br)c2)c2n(C(C)(C)C)nnn2)CCN(C(N)=O)CC1CO N1(C(C2CC(C)(O)C2)=O)CC2(C1)CN(C(=O)C1=CC3CCCC13)CCO2 CC1CN(C(=O)C2=C(Cl)CCC2)CC(C(=O)NC2CC(C(F)F)C2)O1 CCC(C)(COC)C(=O)N1CCC(CC(=O)NCc2cc(C)no2)CC1 N1(C(C(C)n2ccnn2)=O)CCC2(CC1)CCN(C(=O)CN1CCNC(=O)C1)C2 C1(NC(C2(C)COC2)=O)COC2(C1)CN(C(=O)COCc1ccccc1)C2 c1(OC)cnc(Cl)cc1C(N1CC(NC(c2n[nH]cc2C)=O)CCC1C)=O C1(CNC(C2C(=C)C2)=O)CCCCN(C(c2ccc(Br)cc2OC)=O)C1 Cc1nc(C(N2CCC(OCC)C2)=O)c(C)n1C.c1(CC(=O)N)ccc(Cl)cc1 CCC(CN(C(c1ccc(C(C)C)s1)C(=O)NCCCF)C)CCC1CCCC1 C1(C(=O)NCC2CCCN(C(C(CSC)C)=O)C2)CC2CCC(C1)S2(=O)=O C(CCCCC(=O)NC(CCO)C(C)(C)C)N(C(=O)CCc1cscn1)C C1(CC)(NC(c2nc(Br)nn2C)c2nnnn2C2CC(F)(F)C2)CCCOC1 N1(C(C2C(CC)N(C(c3scc(C)c3C)=O)CCC2)=O)CC(O)C(N=[N+]=[N-])C1 C(=O)(C(F)(CNC(C1CC1)=O)C(C)C)OCC.n1(CC=O)cnnc1 C(CC(=O)N1CC(CO)C1(C)C)(C(F)F)NC(CC1N(C)CC=CC1)=O C1(C(N(C2CCN(C(=O)C(C)OCC)CC2)CCC)=O)CCCS(=O)(=O)N1 N1(C(c2cccc(C)c2N)=O)CC2CC(C1)N(C(c1ccc3snnc3c1)=O)C2 C(=O)(CC(C)(C)C)NC(C1CCN(C(C2(C=C)CCC2)=O)C1)C C1(C(N2CCC(C3(C)CC3)C2)=O)CC(O)C(O)CC1.CC(C)(C#N)CC(=O)N.C Cc1nc(CC(=O)NCC(F)CNC(=O)C(O)Cc2[nH]cnc2C)n[nH]1 c12cc(Cl)cnc1N2.C1(C(=O)OC)(CBr)CC(c2nnnn2C)(OC)C1 c1(C(N(C2CN(C(=O)CCc3cnoc3)CC2F)C)=O)ccc2nnn(C)c2c1 S(=O)(=O)(c1ccc(C(=O)NC2CN(C(C3CCS3(=O)=O)=O)CC2C)o1)NC C1(NC(C2(COC)CC2(F)F)=O)CN(C(c2nc(C)sc2C)=O)CCC1C N1(C(C2CC(C)CN2Cc2cc(Cl)c(Cl)c(Cl)c2)=O)Cc2ccc(F)cc2C1 C1(C(=O)NC(CCNC(C(C)SCCCC)=O)C(C)C)CCCCC(=O)N1 C1(C)(C(=O)NC(C(=O)N(CC)CC)C)CC(c2cc(Cl)cc(Cl)c2)=NO1 C=CCCC(F)(F)C(=O)N(C(C)CNC(=O)CC1CCN(C)C1)CC c1(C(=O)NCC2N(C(c3cc(C)sn3)=O)CCC2)cnncc1O N1(C(=O)CC2OCCCO2)CCC2C1CCCN2C(c1cc2c[nH]cnc-2n1)=O C#Cc1ccc(F)cc1C(N1CCN(C(c2cc(C)c[nH]2)=O)CC1CC)=O c1(OC)c(Cl)cc(C(N2CCCC(NC(=O)C(C)CC(C)C)CC2)=O)cc1Cl S(=O)(=O)(CC(=O)NC(CC1CCCC1)C(=O)N)NC.c1(C(C)C)nc[nH]n1 C1(NC(c2ccn(CC)n2)=O)C2CC1CN(C(=O)Cc1ccc(Cl)cn1)C2 c1(-c2n(C(c3cnn(C)c3)C)nc(CC3(C)CC3)n2)cc2cnccc2[nH]1 c1(C(C)NCC2CC2)ccc(-c2cscn2)cc1.C1(C(C(=O)N)O)CCCCC1 C1(C(=O)NC2CCN(C(C=C(C)C)=O)C2C2CC2)C2(CCC2)C12CCC2 c1(C(C(=O)N(CCCNC(C(CSC)C)=O)C2CC2)O)ccc(Cl)cc1F Cc1nc(CN2CCCC(CNC(c3cc(Cl)no3)C)CC2)cc(O)n1 N1(C(c2c(CC)occ2C)=O)Cc2cccc(CNC(C3CCCSC3)=O)c2C1 CCC(CC)C(C)C(=O)NC1CC(O)(CNC(=O)CCc2cn[nH]c2)C1 C1(C#N)(NC(C2C(C(=O)OC)C2)=O)CCOCC1.N12CC=CC1C2=O N1(C(c2cc(CS(C)(=O)=O)on2)=O)CCN(C(=O)C(O)C2CC2)C(CO)C1 C1(C(=O)NC2CC(CNC(COCCC)=O)C2)CCCC2(CCOCC2)O1 N1(C(C(F)OC)=O)CCOC2(CCCN(C(C3CCCCCC3)=O)C2)C1 c1(CC)cc(F)ccc1C(N1CCCCC1CN(C(c1conc1C)=O)CC)=O N1(C(C)C)CCCC(N(C2CCN(C(=O)CSC(F)F)CC2)C)C1 N1(C(c2c(CC)ccs2)=O)CC(NC(=O)C(C)(C)C(=O)N(C)C)CC12CCC2 C(=O)(C(O)CCCNC(=O)CC1CCCC(=O)N1)N1CCC(C(CC)C)CC1 CC1C(C(=O)NCC2CC2NC(=O)Cn2nnc(C3CC3)n2)CCN1C C1(C(=O)NCC(CCC)OC)CN2CCCN1CC2 C(=O)(C(C)(C)S(=O)(=O)C1CC1)NC1CN(C(c2c(C)scc2)=O)C2C1CCCC2 C12CCC(CC1)N(C(c1cc(S(C)(=O)=O)co1)=O)C2.CCS(=O)(=O)CC(=O)N CCCC(C(=O)NC(=O)NC)NC(=O)CN(C)CCc1ccco1 c1(OCC)ncc(C(N2CC(CNC(C3(O)CCC3)=O)(O)C2)=O)cc1Cl c1(NC(C(C)N(CCC)C(C2CC(O)C(O)CC2)=O)=O)cc(C#N)ccc1C CC1(C)CC(NC(c2nc[nH]c2C(F)(F)F)=O)CN1C(=O)CCC#N c1(NCC(CCCC)NC(=O)CCc2ccc(C)nc2)ncc(C#N)cc1Br n1(CC)cc(C(=O)N(C(C)CN(C(=O)CCCCc2ccccc2)C)C)c(C)n1 c1(C(N2CC(CCC)C2)=O)cn2ccccc2n1.C1(C(=O)N)(CSC)CCC1 C1(C(N2CC(F)(CNC(C(C=C)CC)=O)C2)=O)CCCCC1(C)C CCC(C(=O)NCC1(F)CCCC1)C(C)C.c1(C=O)ccc(C(F)(F)F)[nH]1.C C1(CC=C)(NC(c2n[nH]cc2Cl)=O)CCN(C(c2n[nH]c(CC)n2)=O)C1 N1(C(CCN(C(C(CC)NC(N)=O)=O)CC)=O)CCC(CN(C)C)CC1 Cc1cc([N+](=O)[O-])cc(C(=O)NC)n1.C1CN(C(=O)CC2CCOC2)CC12CC2 CCC(C)(C)C(=O)N1CC2CC1C2NC(c1cncn1-c1ccccc1)=O CCCC(C)C(=O)NC1(CO)CN(C(c2nccnc2SC)=O)C1 Cc1ccc2cnc(C(=O)NCC3CCCCN3C(C3CC3CF)=O)cc2c1 N1(C(C2N(CCC)CCC2)=O)CCN(C(c2ccnc(S)c2)=O)CC(C)C1 C(=O)(CCCCC(N)=O)NCC1C(C)CCCN1C(=O)CCC1CC1 C(=O)(CS(=O)(=O)C1CC1)NC.c1(CC)ncncc1C(=O)NC1CCCC1.C c1(C(=O)NC2(C)CC(NC(c3cncnc3)=O)C2)cccc(OC2CCC2)c1 c1(C(N(CCC(C)NC(c2cc(C)nc(C)c2)=O)C)=O)cc(C)c(C#N)cn1 C(=O)(C1=COCCC1)NC(CCNC(C(n1nnc(-c2ccccc2)n1)C)=O)(C)C N1(C(C2(COC)CC(=C)C2)=O)CCC(C(=O)NCC)CC1.C1CCCC(O)C1 N1(C(CN(C(C)C)C)=O)CCCC2CN(C(c3cc(O)nn3C)=O)CCC12 CC(C)CC(C(=O)N1CCC2(C1)CN(C(=O)CC1OCCO1)C2)C(N)=O c1(C(N2CCCN(C(CC3(C)CCCO3)=O)CC2)=O)n[nH]c2c1CS(=O)(=O)CC2 C(CNC(=O)CC(C(F)F)n1cccn1)(CC(F)(F)F)NC(CCCC#N)=O c1(OC)c(C)cc(C(=O)NC2(C)CN(C(=O)CCC(C)C)C2)cc1C N1(C(C(OC)OC)=O)CCCC(C(=O)Nc2ccc(O)cc2C)CC1 N1(C(CN(C(=O)CC2CCCCC2O)CCC)=O)CCC(=O)N(C)CC1 N1(C(CNS(NC)(=O)=O)=O)CCOC(CCNC(=O)C(C)Cc2cnc[nH]2)C1 N1(C(C2(C)CCN2C(c2cncc(Cl)c2)=O)=O)CCn2nccc2C1 c1(C(=O)N)sc([N+](=O)[O-])cc1Cl.C1C2CN(C(c3ccn(CC(F)F)n3)=O)CC12 N1(C(c2nc(C)n(C)n2)=O)CCC2(NC(c3cc(F)c(F)cc3F)=O)CCCC12 N1(C(C2(C(C)C)CCC2)=O)C2CCC1CN(C(=O)C(C)(C)c1cncnc1)C2 Cc1cncc(C=CC(=O)NC(C)C(C)(C)C)c1.C1(CC=O)CC2CCC1O2 N1(C(CCC(=C)C)=O)CC2(C1)C(NC(c1conc1C)=O)CCS2(=O)=O C(=O)(C(CNC(=O)CC1CC2CC2C1)OC)N(CCCCC)C C#Cc1ccc(NC(C2CC(C)N2C(=O)CC2C(C)(C)C2(C)C)=O)cc1 c1(C(N(C(CC)CC)Cc2ccsc2)=O)ccc(SC)cc1 C1(N(C)C(c2cnn(C(F)F)c2)=O)CCCN(C(=O)Cc2ncc(Cl)s2)C1 N1(C(Cn2nc(C)c(Cl)c2)=O)CCC(F)C(NC(=O)Cc2nc[nH]n2)C1 N1(C(CCC=C=C)=O)CC(CNC(C2CCCCC2OC)=O)CC(C)C1 CC(C)(CNC(=O)C(C1CCN(C(=O)C(C)(C)N=[N+]=[N-])C1)F)CN=[N+]=[N-] N1(C(CC(C=C)C)=O)CC2(C1)CN(C(c1cccc(Br)c1C)=O)CCO2 C(=O)(C(C)(O)C(F)(F)F)N1CCN(C(C(C)n2cncn2)=O)C(CCO)C1 c1(C(=O)NCCC(C)NC(=O)CCC)ccc(C(=O)NC)o1.c1ccccc1 C1(C(N2CCC(C)(COC)C2)=O)(NC(C2C(CC)C2)=O)CCCCCC1 c1(C(=O)NC2C3CN(C(C=CCC)=O)C2CC3)c(C)[nH]c2ccc(OC)cc12 c1(OC)cc(C(N2CC(F)(C(=O)Nc3sncc3C#N)C2)=O)cc(Cl)c1O CN1CC(C(=O)N(CCCN(C)C(c2cccn2C)=O)C)C(C(F)(F)F)C1 C(=O)(CC(C(F)F)C(C)(C)C)N1CC(C)C(CNC(=O)CN=S(C)(C)=O)C1 c1(OC)ccc(C(=O)NCC(O)CNC(=O)C(CC(F)F)C2CCC2)cc1Cl N1(C(C(=O)NC)CCc2cccc(F)c2)CCC2(CCC(O)C2)CC1 CN1CCCC(C(N2CCCCC2CNC(=O)C)=O)C1.C1(C(=O)N)CCCCC1 CC1CN(C(=O)CCOCC(F)(F)F)CC(C)N(C(=O)Cn2ccccc2=O)C1 c1(C(N2CC(CO)(CF)C2)=O)cc(CNC(C2(CF)CC2)=O)cs1 C1(C(N(C(C)C(F)F)C)=O)CCN(C(C2CCN(C)C2)=O)C1C c1(N(CC(=O)NCCC)C)nc2c(c(=NC3CS(=O)(=O)CC3C)[nH]1)CCC2 C1(NC(=O)NC2CCCN(C(Cn3c(C)ncc3)=O)C2)CCCN(CP(C)(C)=O)C1 N1(C(C2N(C(C)(C)C)CC2)=O)CC(F)(F)CC1(C)C.C1(C=O)CCC1(C)C.N C1(C(=O)NCCCCCNC(C(C)c2cc[nH]n2)=O)CCOCC12CCCCC2 Cc1nn(C(F)F)c(C)c1CC(N1CC(CC(C)NC(C2(O)CC2)=O)C1)=O C1(NC(C2N(C(C)C)CCC2)=O)CC(C)CN(C(=O)Cc2cccc(C#N)c2)C1 C1(CC)(C)CCN(C(=O)CC)CC1.C(=O)CN(S(C)(=O)=O)C.C=O.N c1(C(C(=O)NCCC(C)NC(C2(C)CCOC2)=O)(C)C)ccc(F)c(Cl)c1 c1(CC)c(C(=O)NCC(Cn2cc(C(C)OC)nn2)OC)cccc1F C1(C(=O)NCC2(OC)CCN(C(c3ccn(C)c3)=O)C2)CCCCS1(=O)=O Cc1cnc(C)c(C(N2CCC(C)(CCNC(c3cc(=O)cc[nH]3)=O)C2)=O)c1 Cc1nccc(C(N2CCC3(CC3NC(C3CCC4CC34)=O)C2)=O)c1C C1(NC(C(C)=CC)=O)CCN(C(=O)COC(C)=O)CC1c1ccccc1 N1(C(c2c(CC)n(C)nc2)=O)CC2CCC1C(CNC(=O)CC(O)C(C)CC)C2 C1(CCC(=O)N(CCC(=O)OC)C)CCN(C(=O)CC23CCCC2C3)C1 C(C#Cc1cn(Cc2ccc(Br)cc2)nn1)NC(C1CC12CCOC2)=O CC(C)C(C)C(CNC(=O)C(C)(C)c1ccccc1)NC(=O)CO.C1CC1 N1(C(C2(CC=C)COC2)=O)CCC(C(C)NC(c2sc(C)cc2C)=O)CC1 c1(C(=O)OC)cccc2c1CCCC2NC(C1(CO)CC(O)C1(C)C)=O CCC(CC)C(=O)NCC(C)(C)OCCNC(c1cnc(S)n1C)=O n1(CC)cc(C(=O)NCC2CCCCC2)c(C)n1.C(=O)C(C)(C)N1CCCC1 N1(C(CN(C)C=O)=O)CC(O)CCC1C(N1CC(C(N)=O)C2(CC2)C1)=O.C C(=O)(C(CC(C)C)C(C)C)N.Cc1oc(C)c(C(=O)NC(C)CC(F)(F)F)c1C N1(C(c2c(OC)cc(F)cc2)=O)CC2CCC(NC(C3(CO)COC3)=O)CC2C1 n1(CC=O)cnc([N+](=O)[O-])c1.CC1=C(C(=O)NC2(C)CC(F)(F)C2)CC1 c1(CN2C(C(=O)Nc3cnccc3CO)CC(C)C2)cc(Br)cnc1Cl C(=O)(C1CCCc2c[nH]nc21)NCCCCCNC(C(C)C1CCC1)=O N1(Cc2nc(CCCC)sc2)CCCC(CCNC(C2CCCN2CC)=O)C1 CCCCCCCCNC(=O)NCC1CN(C(=O)CCC(C)N(C)C)CC1(C)C N1(C(C2(CNC(c3occ(C)c3)=O)CC=CC2)=O)C2CCC1CC1(C2)N=N1 Cn1cc(C(N2CC3CC3C2)=O)c(C(C)(C)C)n1.C(c1cscn1)=CC=O.C C1(C(=O)NC(c2ccc(C)s2)C)CC=CCC1NC(c1ccc(Cl)o1)=O CC1(C(N2CC(CN)CC23CCC3)=O)CC2CCC(C1)S2 Cc1cc(Cl)c(C(N2CCN(C)C3CC23)=O)cc1F N1(C(c2cc(C(C)=O)sc2)=O)CCCN(C(=O)C(O)CC2CC2)CC1 N1(C(C2C(C=O)C2)=O)CCN(C(=O)CCN(CCC(C)(C)C)C)C(C)C1.CO CC1(C)CC2(CO1)CN(C(=O)NC(CO)CS(C)(=O)=O)CCO2 C1(C(NCCNC(C2CCC(C)(C)OC2)=O)=O)Cc2c(C)cccc2O1.CC N1(C(C(C2CCCO2)NC(c2cnn(C)c(=O)c2)=O)=O)CCn2c(O)nnc2C1 N1(C(CC2C(C)(C)C2)=O)CCC(C2CCOCC2)CC1 c1ccc(C(C2CCCC2)N(S(=O)(=O)CC2CC2(F)F)CCO)c(F)c1.C c1(C(N(C)CCN(C)C(C2C=CCCC2)=O)=O)cc(C2CC2)nc2c1cnn2C C1(NC(c2nn(C)c(C(F)F)c2)=O)CCN(C(c2cocc2C(N)=O)=O)CC1F C1(CC)CN(C(=O)CC2CNCC2O)CCC1c1ccccc1 C#Cc1ccc(C2CC2NC(=O)NC2CCCN(CC(=O)OCC)C2=O)cc1 C1(C=O)CC12CCCOC2.C1(CCC)(CNC(CN(C(C)=O)C)=O)CCCC1.N C(=O)(CCCC(=O)NOC(C)(C)C)NC1C(C)CN(C(=O)Cc2cocn2)CC1 c1(C(C(=O)N(CC(CC)NC(=O)C(C)(C)C2CCCC2)CC)O)ccccc1Cl C1(C(=O)NCC(CC(F)(F)F)NC(C(CSC)(C)C)=O)CCCCCC1(F)F C1(C(=O)NC2CC(C(F)(F)F)SCC2)CCCC(c2ccccc2)CC1 CC1(C)CCN(C(c2ccc(Br)cc2N)=O)C1CNC(=O)C(O)C1CCC1 C1(C(=O)NC2(COCC)CCC2)C2CC1N(C(C1CC3(CC3)C1)=O)C2 CC1NC(=O)C2=C1N(c1cccc(F)c1)C(=S)NC2c1cccc2cc[nH]c12 Cc1ccc(C(N2CCN(CCn3cc(-c4ccnn4C)nn3)CC2)=O)cc1Cl N1(C(C2(C)CCCN(C(=O)CC3CC3)C2)=O)CCCC(C)(C#N)C1 C=C1CON(C(=O)C(C)(C)C2(NC(=O)CN(C3CCC3)C)CCC2)C1 C(=O)(C1CCCn2ccnc21)N1C2CN(C(=O)CCC3CCOC3)CC1CC2 N1(C(C2C(C)CC=CC2)=O)CC2OCCN(C(c3nnc(S)n3C)=O)C2C1 c1(C(=O)NCC(CNC(=O)C(CCSC)NC=O)OC)cc(F)n(C)n1 c1(NC(=O)NC(C2CCCOC2)CC)ccc(CNC)cc1F C(=O)(C(O)CC(F)(F)F)N1CC=CC(C(=O)NC(C(=O)NCC(C)C)C)C1 N1(C(CC(COC)NC(c2cn(C)nc2C)=O)=O)CCC2(CCCOC2)C1 C1CC(C)(C)CN1C(c1cccc(Br)c1)=O.C(C(=O)N)=CCC.C(C)=O.C O=S(=O)(c1c[nH]ccc1=NCCNCCC(C(F)F)NCCN1CCCC1)CCC c1(C(=O)NCC(=C)CCNC(C2CNC(=O)N2)=O)cccc(F)c1CC c1(C(N2CCN(C(C(CC=C)C)=O)CC2COC)=O)cc2c(F)cc(Cl)cc2[nH]1 CC(C)(C)C(=O)N1CC(O)(CCNC(=O)C(=O)NC2CC2)C1 c1(C(=O)NCCNC(C)=O)noc2c1CC(NC(n1cccc1)=O)CC2 C1(OC)CN(S(=O)(=O)C=Cc2ccccc2)CCC1(c1ccccc1)OC c1(CC)ccc(OC)cc1C(=O)N.c1(C=O)ccc(O)c(C)c1.C1(CC)CC1 CC(CC(=O)N1CCC(N(C(=O)CC2(CO)CCC2)CCO)C1)CC(F)(F)F N1(C(C(CC)(F)F)=O)CCCC2(C1)CN(C(c1cccc3oc(C)cc13)=O)C2 C1(CNC(c2sc(C)c(O)n2)=O)CC2(CO1)CN(c1cc(=O)n(C)cn1)C2 C1(=CC(=O)NC2CCN(C(c3cnc(C#N)s3)=O)C2)C2CC3CC(C2)CC1C3 N1(C(C(CCC)(C)CC)=O)CCn2ncc(CN(C)C(C3CC3(C)C)=O)c2C1 c1(CC)ccc2c(C)cc(=O)oc2c1.N1(CC(=O)O)CC(C(F)(F)F)CCC1=O N1(C(C)=O)CC(C(=O)O)C2(C1)CN(C(c1cc(CC(C)C)c[nH]1)=O)C2.CCC.S C1(O)(CNC(C(=O)N(C)C)=O)CCN(C(=O)CN2CCOC2=O)C1 N1(C(CNC(C2C(C)C2)=O)=O)CCN(C(=O)CCC2CCCCC2)CC1CO N1(C(c2conc2CO)C(=O)NC(CC)C)CCN(CC(N)=O)C(=O)C1 CC(CC(F)F)C(=O)N1CCCCC1C(C)(C)CNC(=O)CCn1cnnn1 C1(C(N(C)CC2(O)CN(C(=O)CC(O)c3ccccc3)C2)=O)CN2CCN1CC2 CC(C)C(C(=O)N(CCCNC(C1(Cl)CC1)=O)C)c1ccc(Cl)cc1 CCC(C)CC(C(=O)N(C)Cc1ncc(C)o1)NC(c1ncccc1F)=O C(=O)(CC(C)CNC(=O)C(C1CC1)N(C)C(C1CCCCC1)=O)OC C1(NC(=O)NC2CCC(C(C)C)CC2)CC2COC(C)CN2C1 C=C1CCC(C(=O)NC2CCC2C(=O)NCC2COC(=O)N2)CC1 C(C1=CCN(C(c2cc(C3CC3)cnc2Cl)=O)CC1)NC(CCC1C(C)(C)C1)=O C12CC1CN(C(c1cnn(C3CCCC3)c1)=O)C2.C(C(=O)NC)N(C)C1CC1 N1(C(c2ccc(CC3CC3)s2)C(=O)NCC)CCC(OC)C(C(=O)O)C1 C1(C=O)CC2(C1)CC(F)(F)C2.CCCCCCNC(=O)C(O)Cc1cnc[nH]1.N N1(C(C(CC2CCC2)NC(c2cc(C)on2)=O)=O)CCC(C(=O)N(C)C)CC1 N1(C(C(CC(C)C)N(C)C)=O)C2CCC1CN(C(C1C(C)C1C)=O)CC2 C(=O)(C1SCCc2sccc21)NCC1C(NC(=O)CCc2cnoc2)COC1 C(=O)(CCCC(F)(F)CO)N1CC(CC(C)NC(Cc2ccc(OC)nc2)=O)C1 Cc1ccccc1C(=O)NC(C(=O)N(C(C)CC(F)(F)F)C)C1CCOC1 N1(C(C(C)Cc2ccnn2C)=O)CC(CNC(c2nccn2C)=O)CC(C)(C)C1 c1(CNC(C(C(C)C)C)=O)n[nH]c2c1CN(C(C1CCCCS1(=O)=O)=O)CC2 c1(C(=O)NCC2N(C(C(CO)NC(N)=O)=O)C3C(C2)C3)ccc2n[nH]cc2c1Cl N1(C(C2CC(C)N(c3nnc(-c4ccc(F)cc4)o3)C2)=O)CCc2ccccc21 C(CN=c1cc(Cl)nc(C2CC2)[nH]1)(C1CCCC1)NC(=O)C#CC1CCCOC1 C(=O)(C(O)CC(N)=O)N(C(CC)C(=O)NC(C)C(F)(F)F)C c1(C(=O)NCC2CCC(C)CN2C(=O)CS(=O)(=O)CCO)[nH]nc([N+](=O)[O-])c1Cl C(=O)(C(C)(C)C(C)O)NCc1ccc(CCNC(CCC)=O)cc1 C1(C(=O)NCC(CNC(=O)Cn2cccn2)OC)CCC=CCC1 CC1=C(C(=O)N2CCN(C(C3CCC3)=O)CC2CO)CCC(C)(C)C1 C1(O)(CC#C)CC(C(=O)NCCC(CNC(=O)C=Cc2ccco2)O)C1 Cc1cc(NC(C23CC(C)(CN2C(C2Cc4nccn4C2)=O)C3)=O)c(O)cc1F C1(CNC(C(F)=CCC)=O)COCCN(C(=O)C)C1.c1ccc(C)c(C)c1.S C1(NC(C(CC)OC)=O)CC2(CCC(NC(=O)CCCn3ccnc3)CC2)C1 CC(C)(C(=O)N1CCCC(N2CCN(C(c3cc(Cl)c[nH]3)=O)CC2=O)C1)C(F)F C1(C(=O)NCCN2C(C=C)CCC2)CN(C)CCN1C(=O)C(C)C(F)(F)F C1(C(N2CCCC(C3(C(=O)OC)CC3)C2)=O)CCC2(CCCCC2)NC1 CCCCCC(O)CC(=O)NC1COCC1NC(=O)C=Cc1cncnc1O N1(C(CSC(C)(C)C)=O)CC2(C(=O)NCC(O)C(C)(C)C)CC1CO2 N1(C(CC(=O)NCC)=O)CCN(C2CCN(C(C3(CC)CCOCC3)=O)C2)CC1 CC(C)(CC(=O)N1CC2CC1(CNC(=O)CCN1CCCC1)C2)C(F)(F)F CN1CC(O)CC1(C)C(N1CC2CC1C2C)=O.c1(C(=O)N)cncc(C2CC2)c1 C=CC(C)(C)C(=O)NCCC(C)CCNC(c1n[nH]c(C)c1F)=O n1(CC(=O)NC2CN(C(CCC=C)=O)C(C)C2)c(C(F)(F)F)nc2ccccc12 CC1=CC(C(=O)NCC=CC(=O)N(C(C)CC(N)=O)C)SC1 C1(C(N2C(C(C)(C)NC(c3cnc(O)s3)=O)CCC2)=O)CCc2nncn2C1 n1(CC)nc(C)c([N+](=O)[O-])c1N1CCC(CCC)CC1.C(=O)(CCS(C)(=O)=O)N C12(C(N(CC(Cl)Cl)C)=O)COC(C1)C(NC(=O)CC1CCC(=O)C1)C2 C(=O)(C1=CCCOCC1)NC1CC(CNC(c2sc(CC)c(C)c2)=O)CC1O C(CCC(C)(C)C(=O)Nc1cccn2ccnc12)NC(C1CC(OC)(OC)C1)=O N1(C(CCCC(=O)NCCC)=O)CCOC2(C1)CN(C(C1CS(=O)(=O)C1)=O)C2 N1(C(CSc2n(C(C)C)cnn2)=O)C2CCC1C(NC(c1cc(CO)on1)=O)C2 C(=O)(CC(O)c1ccccc1)NCCC(C)NC(C(C1CC(F)(F)C1)OC)=O C1(N(C(CC)=O)C)CCCCN(C(=O)Cn2ncc(C#N)c2N)C1.C(=O)(NC)N CCC(CC)C(C)C(=O)N(CCCNC(c1cnc(C2CC2)o1)=O)CC c1(C(=O)NC2CCCC(NC(c3cc(C)sc3C)=O)C2)ccc([N+](=O)[O-])[nH]1 CC1CC(NC(C2CCCO2)=O)CN1C(c1c[nH]nc1C1CCCO1)=O c1(OC)cc(O)c(C(N2CC(F)(CNC(C3CCCCC3F)=O)C2)=O)cc1.O N1(C(CC)=O)CCC2CCN(C(c3cc4c(Cl)ccc(Cl)c4[nH]3)=O)CC2C1 Cc1scnc1C(=O)N.n1(C2CCC2)cc(C(O)(CO)CO)nn1.CC.C=O.C N1(C(C)C)CC(C(=O)NC2CN(C(c3ccc(C(N)=O)o3)=O)CC2C)CCC1=O CC(C)C(O)CC(=O)NC1COCCC1C(N1CC2CC1CC2CF)=O C12(CNC(c3c(C)c[nH]n3)=O)CC(CNC(=O)CC)(CO1)C2.C1CC1 C1(N(C(CCSC)=O)C)CCCN(C(C2CC(=O)N(c3cn[nH]c3)C2)=O)CC1 Cc1nn(C)c2c(N(CCC(C)(C)C)C)nc(NCCS(C)=O)nc12 S(=O)(=O)(c1ccc(C(N2CCC2)=O)cc1)N(C)C.c1(C=O)ccc2c(c1)CC2.N C1(CNC(C(C=CC)O)=O)CC(C)CN(C(c2cc(Cl)n(C)n2)=O)C1 C1(NC(c2c(C)cns2)=O)CCN(C(C23CC4CC2C3C4)=O)CC1C Cc1cnn(C(C)C(=O)N)c1.c1(C(N(CCC)C(C)C)=O)coc(N(C)C)n1 N1(C(C=Cc2ccc(=N)[nH]c2)=O)CCC2(NC(=O)C3=CCCC3)CCCC12 c1(C(=O)NCCCC(C)NC(C=NOC)=O)ccc(C(OC)OC)nc1O C12(C(=O)NCCC(C(=O)OC)C)CCN(C(=O)CCCC3CC3C)CCC1C2 C1(C(=O)NC23CC2CN(C(c2cc(C4CC4)cs2)=O)C3)CCn2c(O)nnc2C1 c1(N2C3CCC(NC(C)(C)C)(CC3)C2)ncc2c(Br)cccc2n1 C(C(C)CC(=O)N(C)CCC1CCCCN1C(c1ccnnc1C)=O)OC C(=O)(C1OCCc2ccccc21)NCC1N(C(CSCC)=O)CCOC1 n1(CCCC(=O)NC2C(NC(C(C)=CC3CC3)=O)CCC2)cnc2ccccc12 C1(S(C)(=O)=O)(C(N2CCC(NC(c3cncc(C)n3)=O)C2)=O)CCCC1 Cc1ncc(C(=O)NCCC2CCCN(C(c3csnc3C3CC3)=O)C2)n1C CCC(CC(=O)NC(C1CN(C(=O)Cc2cnccc2O)C1)C)SC C12(C(=O)NCC(CSC)C)CC1CCN2C(=O)CC1CSC1 N1(C(C(n2cc(C(C)(C)C)nn2)C)=O)CC2(CCCO2)C1C1CC1 c1(OCc2nc(C(C)C)on2)ccc(C(=O)N(C2CCCCC2C(=O)O)C)cn1 c1(C(N(CC(CC)NC(=O)C(C)NC=O)C)=O)ccnn1C(C)(C)C.N C=CC(CCC)CC(=O)NCC(CNC(C1(OC)CCC(C)(C)C1)=O)CO C1(CN(C(=O)CC2CC2)C)CCN(C(C2CCCN2c2cnccn2)=O)C1 N1(C(c2nccc(OC)c2)=O)CC2(CCC(NCc3ccc(C)nc3Cl)C2)C1 C1(C(=O)NCC#CCC)CCC2(CC2)N1C(=O)C(CC)NC(N)=O N1(C(c2ccc(C)nc2)=O)CC(NC(=O)Cc2ccon2)C2(CCOCC2)C1 Cc1nsc(C(N2CCOC(CC(=O)NC(c3ccncc3)C)C2)=O)c1N C1(NC(c2cncs2)=O)COC2(C1)CN(C(=O)CC1CSCCS1)C2 n1(CC)ncc2c1CCCC2NC(=O)CCn1cc(-c2cn(C)nc2C)nn1 CCC(C(=O)NC1CCCC(NC(c2cc(F)cc(Cl)c2O)=O)C1)C(C)(F)F O=C(C#CC1CCCO1)N1CCC(N2CCN(C(=O)COCCCF)CC2)C1 C1(C(N2CCC(O)(C(C)NC(c3cc(Cl)ccn3)=O)C2)=O)(CC)CCCCC1 N#CC1CCCC(C(=O)NC2CCN(C(=O)CCc3cscn3)CC2CO)C1 c1(CCCC(=O)NC2CCN(C(Cn3ccc(C)n3)=O)CC2)c(F)cccc1F C(CCCCC(=O)NC(C1(O)CN(C(c2c(C)cncc2C)=O)C1)C)OCC CC(O)C(C(=O)NC1CC(CCNC(=O)C(c2ccnn2C)C)C1)N(C)C C1(CC#C)(C(=O)NCC(C)OC(C)C)CCN(C(=O)COCCC)C1 C1(CNC(CC(C2CC2)NC(=O)CCc2ccoc2)=O)CC2C=CC1O2 C1(N)CC2CC1CC2(C)O.c1(CN(OC)CC2CC2)oc2ccccc2c1C N1(C(C(c2ccccc2)C)=O)CCC(F)(CNC(=O)Cc2ccc(Cl)cn2)CC1 N1(C(=O)C2=CS(=O)(=O)CCC2)CCC2(CC1)CCN(C(c1cccc(Cl)c1)=O)C2 Nc1cc(C(=O)NCCC2(C(=O)N)CCCC2)cc(F)c1.C12CC(CCO1)C2 c1(C(N(CCNc2ncc(C)c(C)n2)CC)=O)cn(C)c(=O)cn1 c1(C(N2CCN(C(=O)C3=CCCC3)CC2CC2CC2)=O)ccc2ncsc2c1 c1(N2CC(C)C(F)(F)C2)nc(N2CCC(CCC#N)CC2)c2ncn(C)c2n1 C(=O)(CCC[N+](=O)[O-])NC(C(C)C)CCN(C)C(c1ncoc1C(F)(F)F)=O N1(CC(=O)NC(CN(C(C2C(C)OCCC2)=O)C)C)CC(=O)N(C)C1=O N1(C(c2cnc3sccn23)=O)CC2(CCC(NC(C34CCC(C3)OC4)=O)CC2)C1 C(=O)(CN1C(=O)CCc2ccccc21)NCCCCCN(C(C=C(CC)C)=O)C N1(C(C)C)C(=O)CCC1C(N1CC(CNC(=O)C=CCO)CC1C)=O C(C)(C(C)(C)C(=O)N1CCOC(C#N)C1)NC(CCn1ccc(C)n1)=O C(=O)(C(C)(C)S(C)(=O)=O)NC(C1N(C(C=NOC)=O)CCC1)C Cc1cc(CNC(=O)CC2CC(C)N(C(=O)CN3CCCC3)C2)ccn1 C1(CNC(CN(C(=O)OCC)C)=O)CC2CCc3ccccc3C12 CS(=O)(=O)C1CCCN(C(C23CC2CN(Cc2cc(Cl)cnc2Cl)C3)=O)C1 C1(NC(=O)OC)COc2c(OC)ccc(Br)c2C1.n12cc(nn1)C2 C=C(C)CCC(=O)NC1CCC(NC(c2ccccc2NC)=O)CC1 N1(C(COC)=O)CCN(C(=O)C(CO)NC(c2ccc(F)cc2)=O)CC1CCO C#Cc1cc(F)c(C(=O)NC2(C)CCN(C(c3nc(=N)cc[nH]3)=O)C2)cc1F Cc1nc(C(=O)NC2CCN(C(=O)C=CC3CCCO3)C(C)C2)cc(O)n1 CCC(C)CC(=O)NCCC1CCCCN1C(=O)CCc1cnn(C)c1 C1(C(=O)NC(C2CCCN2C(C2(O)CC2(C)C)=O)C)C2CCC3C(C2)CC13 Cc1ncc(N)cc1C(N1CC(CNC(=O)Cc2cnn(C)c2)CC1(C)C)=O N1(C(Cc2c(C)ccs2)=O)CCC2C(CCCN2C(=O)C(C)OCCN(C)C)C1 N1(C(c2ccc(C)c(O)c2)=O)CC(C)(C)OCC1C.C(=O)(CS(=O)(=O)C(C)C)N N1(C(C(C)(C)F)=O)CCC2CCC(NC(c3cc(CC4CC4)on3)=O)C1C2 C1(C2(OC)CCC2)(NC(C(CC)NC(c2ccnc(OC)c2)=O)=O)CC1 CCC(C)CC(=O)NCCN(CCNc1nccc(OC)n1)CC CN1CCN(C(c2sccc2C#N)=O)C(CNC(C2CCC(C3CC3)O2)=O)C1 N1(C(C(C)=CC=C)=O)CCOCC1CC(=O)NCc1cc(=O)cc[nH]1 C(C)(C)(CCCNC(=O)CCC1CCCOC1)NC(c1ccc(CC)s1)=O c1(-c2nc(CNc3c(C(=O)OCC)n(C)cn3)on2)cc(Cl)c(OC)c(Cl)c1 N1(C(c2cc(C)c(C#N)[nH]2)=O)CCCC2(C1)CN(C(C1CCCN1C1CC1)=O)C2 CC1CCCC(C(=O)N(C2CCCCC2)CC2CCOC2=O)N1C=O.C(C)(C)C C1(NC(CC2(OC)CCC2)=O)CCCCN(C(=O)C(C)S(N)(=O)=O)CC1 Cc1noc(C(F)(F)F)c1C(N1CCCC(NCC(=O)N)C1)=O.CC(C)C(C)C C(N1CCC2(Cc3ccccc3C2)C1)c1cc2nc(C)n(C(C)C)c2cc1 N1(C(C(C)(C)C2CCCO2)=O)CC2CC(NC(C3(F)CC3)=O)CC1C2 C1CN(C(=O)CC2CC(=O)C2)CC12CCC2.CCC(C(=O)NC)NC(C)=O C(=O)(C1CCCc2c1ncn2C)N1CCCC(NC(c2cc(C)n(C)c2)=O)CC1 CC1CN(C(c2csnc2Cl)=O)CCC1C(=O)NCCc1nc[nH]n1 c1(C(=O)NCCNC(c2cc(OCC)no2)=O)ccc(N(C)C)cn1 c1(OC)ccc(CCC(N2CCCC(C(N3CCCC(O)C3)=O)C2)C)cc1 N1CCCC(C(=O)N(CCN(C(=O)C)C)C(C)C)C1.c1ccc(C)cc1.CC N1(C(=O)OC)CC2CCC1CN2C(C1CCN1C(C)(C)C)=O.C1CC(=O)N1 c1(CN(CCCN(C)C(=O)N)CC)c[nH]nc1C(F)(F)F.CC(C)(C)O c1(OC)ncc(-c2cn(CC(N3CC4C=CC3C4)=O)nn2)n1C N1(CC)C(=O)CCC1CC(=O)NCCCC1CC1.C1(C(=O)N)CCN(C)C1 N1(C(C(CCSC)(C)C)=O)CCC=C(C(=O)NC2CCCCC2(C)C)C1 c1(C(=O)NC(C)C(C)(C)NC(=O)Cc2cnsc2)cccc(N(C)C)n1 c1(NCc2csc(C)c2C)[nH]c(=NCC2(CO)CC2)nc2sccc12 O=C(CCC(=O)c1cc(Cl)sc1Cl)NC1CCN(C(=O)CC2CC=CCC2)C1 N1(CC(=O)N)CCN(C)CC1.C1(C)(CC(=O)N(CCCC)CC)CC1(F)Cl C12(Cn3cc(C(C)NC)nn3)CC3CC(C1)CC(O)(C3)C2 C1(NC(CN(C)S(N)(=O)=O)=O)CC12CC(NC(=O)C(F)(F)C1CC1)C2 CCC(CNC(C1COC(=O)N1)=O)(CC)NC(=O)CC.c1(C=O)ccncc1 C(C(=O)N(c1ncc(C)s1)C)(C(C)(C)C)n1cc(COC)nn1.C1CCOC1 Cc1cc(C=CC(=O)NCC2CCCN2C(c2cnc(O)cc2O)=O)c[nH]c1=N C1(CC(=O)NC)SC(=Nc2cc(-n3nc(C)cc3C)ccc2Cl)NC1=O N1(C(C2CCCN(C(C)=O)C2)=O)CCN(C(c2cccc(C)n2)=O)CC1C(C)C CCCCCCC(C)C(=O)NC(CNC(=O)CCc1nc(C)no1)C1CCC1 c1(C(N2CC3C(CNC(C(CC=CC)CC)=O)(C3)C2)=O)cccc2nn(C)cc12 C(=O)(CCCCCSC)NC1C(C(N(C(C)C2CC2)CC)=O)CCC1 Cc1cc(O)cc(=O)n1CC(=O)N(C(C)CCC)C.C1(C=O)CC1.C(N)=O CCCCC(O)C(C)C(=O)NC(c1cccnc1)C(=O)NC(C)CSC C(C)(CCCCNC(c1cnnn1C)=O)NC(C=CC(C)C)=O N1(C(c2ncon2)=O)CCCC2(CCN(S(=O)(=O)c3ccccc3F)CC2)C1 N1(C(CCc2ccc(C)s2)=O)CCn2c(nc(C(N3CC4CC(C3)O4)=O)c2Cl)C1 C(C)(CCC(C)(C)C)(c1nnnn1CCC1(C)CC1)NC(CCCC)C(=O)OC C#CCC(CC(=O)N1CC(O)C1)NC(=O)C=CCCC CC1(C)CCCN1C(=O)CC1NC(=O)NC1=O.C1(O)(CC(=O)N)CCCOC1 CC(C(=O)NC(C)C(=O)NCC1CN2CCC1C2)C(C)N(C)C N1(c2c(S(=O)(=O)NC(CO)C3CCC3)cncc2)CCC2(CC(C(F)F)=NO2)C1 C(=O)(C(C)C(C)C(C)(C)C)N1CC(C(C)C)N(C(=O)C(C)(C)S(C)(=O)=O)CC1 N1(CC)CCCCC1C(=O)NCC(O)C(=O)NCCC1CC1C1CC1 N1(C(CCC(C)OCC)=O)CCC2CCN(C(=O)C(CCSC)OC)CC12 C1(C(=O)NC2C(CC)C2)C2CC1N(C(=O)Nc1ccccc1C1CC1)C2 O(S(=O)(=O)c1c(OC(F)F)cccc1F)c1c(C)cc(Br)cc1 Cc1c(Cl)ccc(C(=O)NC2(CO)CN(C(C3Cc4nccn4C3)=O)C2)c1Cl n1(CCOCC)nc(C2CCCO2)nc1-c1csc(CC2CCCC2)n1 N1(C(C2CC(CN(C)C)C2)=O)CCC(F)(C(N2CCC(C(C)(C)O)C2)=O)CC1 C(=O)(CCCc1ncc(C)o1)NCCCN(C(C(C1CCOC1)OC)=O)CCO C(=O)(CCCCCCNC(C1CC2C=CC1C2)=O)N1CC(C#N)OCC1 c1(OC)ccc(OCCC(=O)NC)cc1.C1CCOC1.C(=O)C(F)CC1CC1 c1(C(N2CC(N(C(C3CN(C(C)=O)C3)=O)C)C3(C2)CC3)=O)cc(C#N)cc(C)n1 C(=O)(C1CCCn2nncc21)NC1(COC)C(C)C1C N1(C(CC2CCC(C)CO2)=O)CCC2(NC(=O)CCCNS(C)(=O)=O)CC2C1 S(=O)(=O)(c1ccc(NCc2cncc(C)c2)cc1Cl)NCC(C1CC1)OC c1(C=O)ccc(C)c(C)c1.C=CCC(CNC(=O)C=CCO)NC(=O)C N1(C(C(CC=C)CC)=O)CCC(C2(O)CC(NC(=O)C#CC3CCCO3)C2)CC1 c1(C(N(C(c2ccc(CO)cc2)C(=O)NCCOCC)C)=O)ccccc1 C(=O)CS(=O)c1ccc([N+](=O)[O-])cc1.C1CCCOC1.C(=O)(C)N(CC)CC.N C(C(=O)NCc1ccc(C)cc1)(C(C)CC)N(C(c1ccc(CC)[nH]1)=O)C C1(NC(CC(C)CNC(C2CCCC2O)=O)=O)CCOC(C)(C)C1 Cc1cc(N2CCCC(Cn3cc(CC(C)(C)C)nn3)C2)nc2cc(F)ccc12 CC1CC(C(=O)N2CCCC(CO)(NC(c3cc(C4CC4)ccn3)=O)C2)=NO1 Cc1noc(N)c1C(N1CCCC1CCC(N1CCCCC1CCCO)=O)=O C1(NC(c2nn(CC)c(C3CC3)c2)=O)CNCC1S(C)(=O)=O C1(CCC)CCCN(C(=O)CC2CCC(NC(=O)C(C3CCOCC3)O)C2)CC1 Cc1cnc2n1CCCC2C(=O)NC(C)CN(C(=O)Cc1cccc(F)c1O)C c1(OC)ccc2c(c1)C(C(=O)NC1CCCCN(C(=O)C3=CCCS3)C1)CC2 CCC(CCCC(=O)N1CC2CCCC2C1)NC(=O)CC1CNC(=O)O1 C(=O)(C(C(C)C)NC(c1ccccc1)=O)N(c1ccc(Br)cn1)CC Cc1cc(O)ncc1C(=O)NC(CC1CCOCC1)C(=O)NCc1ccoc1 N1(C(c2cn(C(C)(C)C)nn2)=O)CCN(C2CN(C(c3c[nH][nH]c3=N)=O)C2)CC1 N1(C(c2cn(C(C)C)nc2)=O)CCC(NC(=O)CN(C)S(N)(=O)=O)CC1C C(F)(F)C(F)(F)F.Cn1ccnc1C(N1CCCC1CCNC(=O)CO)=O c1(OCC)cc(C(=O)N)oc(=O)c1Br.C1CC1.C(=O)(C=C1CC1)NC Cc1cc(C(N2CCN(C(=O)CC(C)(C)CN(C)C)CC2CF)=O)c(C)cc1Cl c1(SC)cc(C(N2CCC(O)(CCNC(c3csc(Cl)n3)=O)C2)=O)n(C)n1 C(C(CC1CC1)C(=O)Nc1ccc(F)cc1)NC(CC1N(C)CCC1)=O N1(C(CC(n2c(CC)ncc2)C)=O)CC(NC(=O)CCC2CCOC2)C(C)C1 N1(C(CN(CC#C)C(C2CC3C=CC2O3)=O)=O)C2CCC1COC2 c1(SC)cn(C)nc1C(=O)NCCN(C(=O)CC1CCC(C)CO1)C N1(C(C(C)NC(=O)NC)=O)C2CCC1CN(C(=O)CCc1ccccn1)C2 c1(C=O)c(F)cc(F)c(O)c1F.Cc1nc(CC(=O)NC2(C)CC2)c(C)s1.N C12(NC(C=Cc3ccc(C)nc3)=O)CCCC1N(C(C1CC3C=CC1C3)=O)CC2 C(=O)(C1=CCCC1P(C)(C)=O)NC(CNC(CSC)=O)C(C)(C)C C1(NC(C(CCC)(C)CC)=O)CN(C(c2cccc(C)c2F)=O)CC2(CCC2)C1 CCCC(CC)C(=O)NC1CN(C(C2(c3ccno3)CCC2)=O)CC1C C(=O)(C(CC(C)CC)NC(=O)C=Cc1cc[nH]n1)NC(C#C)C(C)(C)C c1(CC(=O)Nc2ccsc2C(=O)Nc2cccc(F)c2O)cc(Br)ccc1Br C1(N(C(=O)C=CC2CCC2)CCF)CCCN(C(=O)CCc2ccc[nH]2)C1 CC(CCC(=O)NCC(C(C)(C)C)NC(C1(CCF)CCC1)=O)c1ccccc1 c1(C(N2CC(N(C(CC3(CC=C)CCCC3)=O)C)C(F)C2)=O)ccc(N)c(Cl)n1 c1(C=O)cc(C)cnc1C(F)(F)F.N1(C(C(COC)OC)=O)CC2CC2(C)C1 c1(C(N2CCC(NC(C=C(C)C)=O)C2)=O)cc(C(C)C)ccc1F c1(N2CCC(C(C)NC(=O)C=CBr)C2)nc(Cl)nc2ccccc12 N1(C(c2c(C)cc(C)[nH]2)=O)CC(CNC(c2sncc2C)=O)N2CCC1C2 N1(C(=O)N)CC2CCC2C1.C1(CC=O)CC(C(C)(C)C)C1.C(C)OCC C1(C(=O)NC2(C)CN(C(C(C)n3ccnc3)=O)C2)COC(C)(C)C1 N1(C(CC2(C)CCCO2)=O)CC2(C1)C(NC(=O)CC1(C)CC1)CCS2(=O)=O c1(NC(C23CN(C(COCC(=C)C)=O)C(C2)CO3)=O)cncc([N+](=O)[O-])c1 C1(NC(CC=CCCCCC)=O)CC12CC(NC(C1CC3(CC3)CO1)=O)C2 c1(C(=O)NCC)ccc(C(=O)NC2CCC(CCOC)CC2)c(O)n1 [SH](=O)(=O)c1c[nH]c(C(N)=O)c1.CC1CN(C(=O)C)C1.c1(C(=O)N)csnn1 C1(CNC(c2nc(CCC)oc2)=O)CCC2CN(C(C3CC(C)C3)=O)CC12.O CCC(F)(F)C(C)(C)C(=O)N(C)CCN1CCN(c2ncns2)CC1 N1(C(=O)CN2CCCS2(=O)=O)CCOC2(CCCN(C(c3ccon3)=O)C2)C1 C(C(CC(F)(F)CNC(=O)NCC1(O)CCCSC1)OC)OC N1(C(c2ccc(CC)[nH]2)=O)CCC(C2CCN(C(C34CC(OC)(C3)C4)=O)C2)C1 Cc1ccc(C(N2CC3CC3C2C(=O)NCCCN(C)C)=O)nc1 C1(OC)CN(C(C2CC(n3ccnc3)C2)=O)CC1NC(=O)C.c1nnnn1C.S C(=O)(CCC1=CCc2ccccc21)N1CCC2(C(NC(CCC)=O)CC2)CC1 Cc1ccsc1C(=O)NC(C)(CNC(c1cccn1C(C)C)=O)C1CC1 O=[N+]([O-])c1cc(Cl)c(Cl)cc1CN1CCCc2ccc(C(F)(F)F)cc21 C1(CC#C)(C(=O)NCC2C3CN(C(=O)CC(F)(F)Cl)CC23)CCCCO1 N1(C(C(=O)Nc2cn(CC(C)C)nc2)=O)CCOC(CCC(F)(F)F)C1 C(CC1=CCCCC1)N(C(=O)C(F)C1CC(NC(C2CC(F)(F)C2)=O)C1)C C1(NC(C2C(CCC)C2)=O)COC2C(NC(c3c(C)nn(C)c3)=O)COC12 C#Cc1ccc(C(=O)N(CCC(=O)NC(CCF)C(=O)OC)CCO)o1 c1(C=O)cc(Cl)cc([N+](=O)[O-])c1.Cc1ccc(C(=O)NCC(=O)NCC)cc1 C(=O)(C(C)(C#N)CC)NCC(C)(C1CC1)NC(C1CC(CC)C1)=O c1(C(N(CC(C)O)Cc2c(OC)cccc2)=O)ccc(=O)n(C(C)C)c1 N1(C(CCOC2CN(C(c3cc(F)cc(F)c3)=O)C2)=O)CCC(F)(F)C(O)C1 CN=S(C)(=O)c1ccc(C(=O)N(C)CC2CCCCN2C(C2CC(F)C2)=O)cc1 N1(C(CC(C)O)=O)CCC2(CC1)CN(C(=O)CC1C(=O)ON=C1C)C2.CC=O.N C1(C(=O)NC2C(NC(C(CC)n3cccn3)=O)COC2)CCS(=O)(=O)CC1 C=CCCCCCCN=c1cc(C)[nH]c(=NCC2(OC)CCCSC2)[nH]1 C#CCCCCC(C(=O)NC(c1ccccc1)C)N1CCCC(C(O)C(F)F)C1 c1(C(=O)NC2CN(C(C(C)CC3CCCC3)=O)C(CO)C2)cc(O)ncc1F C(=O)(CC(C)CCC=C(C)C)N1C2CN(C(c3c(OC)ccs3)=O)CC1C2 C(=O)(C1=CC(C)(C)C1)N1C(C(N2CC(N(C)C3CC3)C2)=O)CC=CC1 C(=O)(C#CC1CCOCC1)N1C(CCNC(=O)C(O)C2CCC2)CCCC1 c1(C(=O)OC)sc(N2CCC(CNC(=O)C(C)(F)F)C2)nc1Cl C(CC(C)C(=O)NC1CCC1NC(c1cc(C2(C)CC2)on1)=O)=CC N1(C(c2ccc(=NC)[nH]c2)=O)CC(C(=O)Nn2cncn2)CCC1(C)C C=C1CCN(C(c2cnn(CC(F)F)c2)C(=O)N(c2ccccc2)C2CC2)CC1 Cc1c(-c2cc[nH]c(=N)c2)cnc2c1N(C(c1sccc1OC(F)F)=O)CCO2 N1(C(C2(C)C(C(=O)OC)C2)=O)CC(NC(c2ccccc2SC)=O)CC(C)C1 c1(C(N2CCN(C(c3ccc(C)c(N)c3)=O)C3C2C3)=O)ccc(S(C)(=O)=O)[nH]1 C(=O)(CC(C)(C)CC(C)=O)N1C(C)CC(NC(c2nnc(CC)s2)=O)C1 O=C(C1=CCCCO1)NCC1CN(C(=O)C2=C(Cl)CC2)CC1O N1(C(CC2C(=O)NCC2)=O)CCCC(C(N2CCN(c3ccccc3)CC2)=O)C1 C(=O)(CCCS(C)(=O)=O)N1CCCC1.Cc1cccc(-n2ccnn2)n1 c1(C(=O)NCC2C(CNC(c3[nH]c(=N)sc3)=O)C2)snc(O)c1Cl N1(C(c2ccc(OC)nn2)=O)CC(NC(=O)CCN)C(C)(C)C1.c1ccccn1 Cc1nc(N2CC3CC2CN3C(=O)C=Cc2ccccc2)cc(SC(C)C)n1 N1(C(C(CC)Oc2cccc(C)c2)=O)C2CCC1CC(NC(C1(O)CC1)=O)C2 C(=O)(CCCC1CCCCC1)NC(CC)CNC(=O)C(C)=CC(C)(C)C N#Cc1ccc(Br)cc1C(N1CC2(CCC(Nc3ccn4nccc4n3)C2)C1)=O C1(NC(C2C(CCC)C2)=O)CC2CC(C1)CN(C(=O)C(O)C(C(C)C)OC)C2 N1(C(C23C(=O)C4CC2C3C4)=O)CCC2CN(C(C34CCC(CC3)C4)=O)CC12 C1(NC(CC(CCSC)O)=O)CC2CN(C(c3cnc(CC(C)C)s3)=O)CC2C1 c1(C(C)C)ccc(C(=O)NCC2C=CC(NC(=O)CC3CCOC3=O)C2)o1 n1(CC(N2C(Cn3cc(CCCC)nn3)C=CC2)=O)nc2ccccn2c1=O c1(C(C)CNC(C)(CCc2ccncc2)c2nnnn2C)ccc(F)c(Cl)c1 CC1(C)C2CCC(C2)C1(C)c1nc(-c2ccc(OC(F)F)c(Cl)c2)no1 Cc1cc(C(N2CCC(C)(C(=O)NCC(c3nccs3)C)C2)=O)ccn1 c1(CC(=O)NCC(C(C)C)NC(CS(CC)=O)=O)ccc(F)c(Cl)c1F N1(C(CCCOC)=O)CC(CNC(c2cc(C)no2)=O)C(C)C1 N1(C(c2cc(C)ncc2)=O)CCC2(CC1)CC2NC(=O)Cc1csc2nccn12 C(c1cnc[nH]1)=CC(=O)NCC(C)NC(=O)CC(C)C1CCCO1 Cc1nc(C(N2CC(NC(c3cnns3)=O)CC23CCOC3)=O)c2n1CCCC2 c1(CC(N2CC(NC(c3cnccc3Cl)=O)C3C2C3)=O)c[nH]c2ccc(Cl)cc12 N1(C(C(C)NC(C2CCC2)=O)=O)CCC2C(C1)CN2C(=O)C1=CCCC1 c1(C(=O)NCC(CC=C)NC(c2c[nH]nc2OC)=O)cc2c(nn1)OCCS2 C1(N(C)C)CN(C(=O)C(=O)NC(c2ccc(C(F)(F)F)cc2)C2CC2)CC1F C#CCN(OC)C(=O)C(F)(CNC(c1nccnc1N)=O)C(C)C C1(C(N2C(CNC(C3(C(C)C)COC3)=O)CCC2)=O)CCc2nccn2C1 N1(C(C(C=C)OC)=O)CCCC2C(NC(=O)CCCOC)C(C)(C)C12 Cc1cc(C(=O)NC2CC(Nc3nccn(C)c3=O)C2)cc(C)c1 Cc1cccc2c(CCC(=O)NCC34CCC(CC3)O4)c[nH]c12 Cc1ccc2oc(C(=O)NC3CCN(Cc4ccc(I)c(O)c4)CC3O)cc2n1 c1(C(=O)NC2CC(C)C2)cc2c(Cl)nccc2s1.C1(C=O)CCS(=O)(=O)N1 C12CCC(CC1)CN2C(=O)C=C(C)C(F)F.c1(OC)cccnc1C(=O)N C1(n2c(CC3CCC(F)(F)CC3)nc(C3C(C)(C)C3)n2)CC2CS(=O)(=O)CC2C1 c1(OC)cc(C(=O)NCCC(C)NC(=O)C(C)C(C)(C)C)c([N+](=O)[O-])cc1F C(N=c1cccc(S(=O)(=O)N(CC(O)C2CC2)C)[nH]1)C1CC2(CC(OC)C2)C1 C1(CN=c2[nH]nc(C(F)F)o2)CCCC2(CNC2)O1 Cc1cc(=NC2CCC(F)(F)C2)nc(NC2C3CCCC23)[nH]1 C1(C(N2CCC(CC(C)NC(=O)C(F)(F)CC3CC3)CC2)=O)CC12CCOCC2 C(C(O)CC(=O)NC(C)CC1CCC1)NC(CNC(C)=O)=O c1(C(=O)NCC(C)(CO)NC(=O)Cn2cnc([N+](=O)[O-])n2)ccc(Cl)cc1F c1(C(CC)C(=O)NCCC(C)N(C(=O)CSCC(F)(F)F)C)cccc(Cl)c1 C(=O)(N=c1ccn(CC(C)C)[nH]1)C1CC(CC)N(C(=O)C2=C(Cl)CC2)CC1 c1(C(=O)NC(CC=C)CNC(=O)CC2C=CCC2)ccc2c(C)cc(O)nc2c1 N1(C(C(C)S(N)(=O)=O)=O)CCN(C(C2C3C4CCC(C4)C23)=O)CC12CC2 c1(OC)c(F)c(F)cc(NC(C2CSCCN2C(c2cnc(C)cn2)=O)=O)c1F C(CCCCC(=O)N1CCN(CCO)CC1)N(C)C(c1ccc(CO)o1)=O C12(C(N(CCC)C)=O)CCC(CC1)N(C(C1CC(C)(C)CO1)=O)C2.C1CC1 C(CC#CC(C)(C)C)NC(C1OCCN(C(C2(OC)CCCOC2)=O)C1)=O Cc1ncc(Cl)cc1C(=O)NC1CN(C(=O)CC#N)CC1F.C(CCCO)C1CC1 c1(C(=O)NCC(CNC(c2cn(CCC)nn2)=O)(C)O)cccc(F)c1O C1(NC(CCOC)=O)C2CC1N(C(c1ccccc1-n1cccn1)=O)C2C C(=O)CCCC.C(=O)(C(C)CN(C(=O)CC1CCCCC1)C)OC.C(C)=O.N C(=O)(C1CCCc2c[nH]nc21)N1C(CCNC(C2C=CC=CC=C2)=O)CSCC1 N1(C(c2noc(CC)c2C)=O)CCC(C=CC(=O)NCCCN2CC=CC2)CC1 c1(CC)cc(C(=O)NC2CC(C(N3CC(O)(CC4CC4)C3)=O)C2)nn1C N1(C(=O)Nc2cccc(CNC(CC)=O)c2)CCCCCC1C(C)C c1(NC(C(C)N(CC(C)NC(C2(F)CC2)=O)C)=O)ccc(F)cc1 C1(C(=O)NC2CCC(NC(C=CSC)=O)CC2)COc2c(F)cc(F)cc2C1 c1(OC)ccc2c(c1C(=O)NC(CNC(C1CSC1)=O)C1CC1)CCC2 C#Cc1cc(C(=O)NC2CCN(C(=O)CC3CCCC3(F)F)CC2O)cc(F)c1 N1(C(c2c(Cl)cn(CC)n2)=O)CC2CCCC1C2CNC(=O)C(O)C(C)C C(=O)(C(=O)N=S(C)(C)=O)N1C(C)CC(CNC(=O)Cc2cnoc2)CC1 CS(=O)c1ccc(CC(N2C3CCC2(CNC(C2CCCSC2)=O)CC3)=O)cc1 c1(C(=O)NCCNC(Cc2c(C)ocn2)=O)ccn2nncc2c1 c1(N(C)Cc2cc(Br)ccc2F)nc(=NCC2CC(F)(F)C2)[nH]c2c1COCC2 N1(C(Cn2c(C)cc(C)n2)=O)CCC(C)CC1CNC(=O)C(F)CC(C)C CCCCCC(O)CC(=O)NC1COC2(C1)CN(C(=O)CSSC)C2 Cc1ncc2n1CCC(C(=O)NCCC(C)NC(=O)CN(C)CCO)C2 CCC(F)(F)C(=O)NCCC(O)C(=O)Nc1cc(C)sc1C Cc1cc(C(N2CCC3C(NC(=O)C=CC4CCOC4)C23)=O)cnc1C C1(C(N2CCC(O)(C(C)NC(CCC=C(C)C)=O)CC2)=O)CCCC12OCCO2 C1(CC(N2C(C3CCN(C(=O)COC(F)F)CC3)CCC2)=O)CC2(CCC2)CO1 Cc1c(CC(N2CCOC(CN(C(=O)CCC(F)F)C)C2)=O)oc2ccccc12 C1(CNC(c2c(CC)onc2)=O)C(C)CCN1C(=O)CCCCF c1(CSCC)cc(C(=O)NCCC(O)C)no1.C(=O)CC(O)C1CCCC1.N C=CCC(C(=O)N1CC(C(=O)NOCCO)CC(C)C1)C(C)C CC1COC2(C1)CN(C(=O)C(c1ccco1)NC(=O)Cn1cnc(C#N)n1)C2 c1(C(=O)NC2(CNC(C=CC)=O)CCC2)ccc(OC)c(Br)c1 C1(CNC(c2cn(CCOC)nn2)=O)CCCCC1.c1(C=O)cc(Br)n[nH]1.N C(=O)(C(C)CCC(C)(C)C)NCC1C(CC(=O)NC(C)CC2CC2)C1 c1(-c2nc(C(F)F)nn2C2CCOC2)cnc2c(Br)n[nH]c2c1 C1(C(N2C(C(C)NC(C(C3CCC3)OCC)=O)CCC2)=O)CCC=CCC1 Cc1ccc(-c2nc(CN(C=O)C(CC3(N4CCCC4)COC3)C3CC3)co2)cc1 C(CC(=O)NCC(O)(C1CC1)C1CC1)OCCCNC(COCC=C)=O C(=O)(C(CNC(=O)CO)C(C)C)N(CC=CC)C1CC1 c1(OC)ccc2[nH]c(=NCCSC(C)(C)C)[nH]c(=NC(C)C3CC3)c2c1 N1(C(=O)Nc2nccc3cc(C(F)(F)F)ccc23)CCc2ccc(O)cc2CC1 Cc1ccncc1CC(=O)NCC1CCC(NC(C2(C(F)(F)F)CC2)=O)C1 S(=O)(=O)(c1ccc(F)cc1)N1CCN(C(Cc2nc3scc(C)n3c2)=O)CC1 C12CC(C1)CCO2.c1(CC)nc(C(=O)NC)c(N)s1.C1(C=O)CC12CCC2 N1(C(C2(C)CCC2)=O)CCC(C2CCN(C(c3ccc(S(N)(=O)=O)o3)=O)CC2)C1 C(C)(CC(=O)NCC(CO)NC(=O)CCc1cnco1)SC c1(C(=O)NC(CCCC)CNC(=O)Cn2ccnn2)cncc2c1CCC2 C(CC(=O)N(OC)C1CCCC1)N(C(C1CCCCC(=O)N1)=O)CC C1(OC)CC2(C1)CC(C(N1CCN(CC)CC1)=O)C2.c1(C(=O)N)cc(C)sc1C C1(CC)(NC(C2CC2CF)=O)CCN(C(c2c(C)ncnc2C)=O)CC1 c1(C2(C(=O)NC3C(NC(C4CSC4)=O)CC3)CC2)cc(F)ccc1F C1(CC)(NC(=O)CC(C)c2ccccc2)CCN(C(c2ccncc2)=O)CC1 c1(NC(c2cccnc2N2CCCCC2)=O)cc2n(c1)CCNC2 C#CC(CC(C)(C)C)NC(C1C=CC(NC(=O)CC2CC(C)(C)CO2)C1)=O N1(C(c2n(CC)nc(C)c2)=O)Cc2ccnn2CC(NC(=O)C(C)(F)F)C1 C1(OC)CCC2(C(N3CC(C(=O)NC(c4cccnc4O)C)(CO)C3)=O)CC12 C1(CC)CN(C(c2c[nH]nc2OC)=O)CCN1C(c1coc(C(C)(C)C)n1)=O N1(C(C(CC)CO)=O)CCN(C(c2ccon2)=O)CC1CCO C1(CNC(C2CCCC3(CCC3)C2)=O)CC(N=c2[nH]nc(CO)s2)C1 N1(C(CCCC#CC)=O)CCC(NC(=O)CC(C)CF)C12CCC2 C(C(=O)NCC(C)NC(=O)C(C1CCCO1)C1CC1)(C(C)C)OC C1(C(=O)NCCCC=CC)CN(C)CCN1C(=O)C(N1CCOCC1)C C1(C(=O)NCCCCCOC)CCCN(C(=O)C(=O)Nc2c(C)n[nH]c2C)CC1 c1(-c2scc(C)c2)cnc2c(c1)N(C(=O)Cc1cc[nH]n1)CC2(C)C C1(CNC(=O)CCCC2CCC2)C2CN(C(c3cscc3Cl)=O)CC12 Cc1ccc(C(N2CCC3C(NC(c4ccc(F)cc4C)=O)CC23)=O)c(O)c1 C1(NC(=O)Cc2ccno2)CC(F)CN(C(c2cc(Br)co2)=O)C1 N(C1CCOc2c1ccc(Cl)c2Cl)C(=O)Nc1cc(C(F)(F)F)ccc1Br CCC(C(=O)N(CC)CC)Nc1ccccc1.C1CCC(=O)N1 c1(OC)ccc(CNC2CCCC2C(=O)OCC2CCO2)c(O)c1OC c1(C(C)SCC)nnc(N(C)CCOc2ccccc2Cl)n1CC1CCCO1 c1(C(C)NC(C(C)Oc2c(C)cc(Cl)cc2)=O)cc(F)c(Cl)cc1Cl c1(-c2cn(C(COCC)C(=O)N3CCC(COCC)C3)nn2)ccc(C)nc1Cl Cc1cccc(C)c1C(N1CCCCC(N(C)C(c2cccc(Cl)c2Cl)=O)C1)=O c1(CC)cc(C(=O)NCCC2(c3ccccc3)CCCC2)ccn1 CC(C)C(C)CNC(c1n[nH]cc1C1CC1)=O.C(=O)(CCCc1ccccn1)N O=C(NNc1cnnc2ccccc12)C1CCN(C2=NCCS2)C1 N1(C(C(C2CCN(C(C3C(C#N)C3(C)C)=O)C2)C)=O)CCC2(CC1)N=N2 c1(C(=O)NC(CNC(c2c(CC)cncc2)=O)CC)ccc2c(c1)CCCC2 c1(CC(=O)NC2CC(NC(C3CCC(OC)C3)=O)C2)cc(C)nn1C C(C)(C)(C(=O)NCC(C)NC(C1(c2ccccc2)CCCC1)=O)OC(C)C C(C(=O)N(CCCO)CCCO)(C(C)O)NC(C(C1CCCC1)OC)=O N1(C(CC=CC)=O)CCC(C)C(F)(F)C1.c1(C(=O)N)cncs1.C(C)(C)C C1(N(C)C(C2CC(NC(c3ncoc3C3CC3)=O)C2)=O)CCCOC1 N1(C(C2CC(OC)C2)=O)CCC2(NC(c3cnc(S)nc3)=O)CCCCCC12 CCCC(C)(O)C(=O)N1CC(CC(C)NC(c2ccc(C(N)=O)c(Cl)c2)=O)C1 c1(C(N2C(C)C(NC(=O)COC3CCCOC3)CC2)=O)n[nH]c2c1CCSC2 c1(C(=O)NCC(C)CN(C(=O)C(F)(F)C2CCCC2)C)cnccc1Cl N1(C(=O)CCc2cccs2)CC(=O)NC2CN(C(=O)C(F)(F)C3CC3)CCC12 N1(C(CC2(CC=C)CCCC2)=O)CC2(CCN(C(=O)CC(C(F)(F)F)OC)C2)C1 C=CCCCC(C(=O)NCC12CCCC1OCC2)NC(=O)Cc1cnn(C)c1 C=C(Cl)CC(C(=O)NCCC(O)C(C)C)NC(c1cc(C)nn1C)=O c1(C(=O)NC(CCCNC(C2CCCC(OC)C2)=O)C)ccc(Cl)cc1Cl C(CC1=CCN(C(=O)C=Cc2ccc(C)o2)CC1)NC(c1cnc(C)nc1)=O c1(C(N2C(C(=O)Nc3ncc(O)cc3Cl)C(O)CC2)=O)cc(Br)ccc1[N+](=O)[O-] c1(C(=O)NCC(CNC(COC(C)C)=O)CO)ccc(N=[N+]=[N-])cc1 C1(C(=O)NCC=CCNC(CCSCCCC)=O)CCC(N(C)C)CC1 N1(C(=O)Nc2cncc(OCC(F)F)c2)CCCC(C2CC2)CC1 N1(C(C(F)=CC)=O)CC2CC2(CNC(=O)CC(F)(F)F)C1 c1(CC(C)C(=O)NC2CCC2CNC(c2cccc(O)n2)=O)ccccc1F C1(N(C)C(c2cscc2F)=O)CN(C(c2cn(C)cn2)=O)CCC1O N1(C(C2C(=C)C2)=O)CC2C(C(N3CCC=C(C)C3)=O)C2C1 N1(C(C(CNC(CN(C)C2CC2)=O)N(C)C)=O)CC2COC(=O)C2C1 CC1CC(NC(C2C3CCCOC23)=O)CCN1C(=O)Cc1ccc(O)cn1 CC(C)C(C)C(CNC(=O)COC(F)(F)F)NC(=O)C=CCO c1(OC)ccccc1-c1cc(C(N2CCCC(c3ccccc3)C2)=O)n[nH]1 C=CC1(O)CN(C(C2CCCC(NC(c3sccc3OC)=O)C2)=O)C1 c1(OC)ncccc1C(=O)NC(CNC(=O)C(c1ccc(O)cc1)=O)CO C(=O)(C(=O)N=S(C)(C)=O)NCC(CNC(c1ncnc(C)c1C)=O)O N1(C(c2cc(C(C)C)[nH]n2)=O)CC(C(F)(F)F)CC1C.C(=O)CC.C(N)=O CC(C)(C)S(=O)(=O)CC(=O)NCC1(O)CCC1.C(C1CCOC1)=CC=O N(C1CCCn2ncnc21)C(CC(C(F)F)NC(=O)C(O)C1CCC1)=O c1(C(C)C)ncc(C(=O)NCC(C2CCC2)NC(=O)CCN(C)CCO)s1 c1(C(=O)NCC2(O)CCN(C(=O)CO)C2)ccc(Cc2cnn[nH]2)c(F)c1 C1(C(=O)NCCC)CCC(C)N(C(=O)CC2CSCCO2)C1 C1(C(=O)NCCC(C)NC(COCCCCC)=O)CCOC1C c1(OCCOC)ncccc1C(=O)N.C12CC1CN(C(=O)CC)C2.C(C)=O c1(CC)ccc(C)c(C(=O)N(CC(C)O)CCNC(=O)CC2CCC2)c1 C1(NC(Cc2nnc(C)s2)=O)CCN(C(=O)C(C)Oc2ccc(F)nc2)CC1F C(c1cc(Cl)ccc1Cl)=CC(=O)NCCCN(C(C1N(CC)CCOC1)=O)C C1(CNC(C)=O)CCCN(c2nnc(-c3nc(C)cs3)n2CC2CCCCO2)C1 c1(CCC=O)ccc(Cl)c(F)c1.C1(C#N)(C(NCC)=O)CC2(CC2)C1.CC C1(COC)CCN(C(c2cn(C3CC3)nn2)=O)C1.c1(C(=O)N)sc(C)cc1 C1(C(=O)N)CCS(=O)CC1.C(C(C)(C)C)N(C(=O)C(c1ccccc1)O)CC c1(C(N2CC(C)(CNC(C3(C=C)CC3)=O)OCC2)=O)coc2c(F)cccc12 c1(C(c2cn[nH]c2)NC(C2(CC)CCCCC2)=O)cccc(F)c1F c1(C(=O)NC(C)CC(C)NC(c2ccn(C)c(=O)c2)=O)cc(F)c(N)cc1F N1(C(C=CC(=O)OCC)=O)CCC(C)C(CC(=O)N)C1.C(C)(C)C(C)O CON(CCC(=O)NC(c1ccsc1)(C)C)C(=O)c1cncc(Cl)c1 c1(C(=O)NC(C2OCCN(C(CCCCC#C)=O)C2)C)ncnc2c1ccn2C c1(CC)onc(C(N2CC(NC(c3cn(CCO)nc3C)=O)C(O)C2)=O)c1C C1(C)(NC(COCCCC#C)=O)CCCN(C(c2ccc(F)c(CC)c2)=O)C1 C1(NC(CC(CC)C2CC2)=O)CN(C(C2(C)CC2)=O)CC1C1CC1 N1(C(=O)Cn2cc([N+](=O)[O-])cn2)CCCC1C1CCCCN1C(=O)C1CC1 C1(NC(C2CSCCN2C(c2coc(C(F)F)c2)=O)=O)CCC2CC1CO2 Cc1cccc(C(O)C(=O)NC(CNC(C2CCCN2C=O)=O)C(C)C)c1 N1(C(C(C)SCCCC)=O)CCCC(F)(CNC(=O)C(CC(C)C)OC)CC1 C(c1cnc(O)nc1O)=CC(=O)NCC1(C)CCN(C(=O)CCC2CCCC2)C1 C1(C(N(CC(CC)NC(=O)COCC(F)F)C)=O)Cc2cccc(F)c2O1 C1(CC)CN(C(=O)CN(C)C(C)C)CCC1.C(CCC=C(C)C)=CC=O C#Cc1cccc(CC(N2CCOCC2CC(=O)N(CC(O)C2CC2)C)=O)c1 c1(COc2c(N(C)Cc3c[nH]c(=N)s3)cccc2)ccc(-c2nn[nH]n2)cc1F C1CN(C(=O)C(O)CC(N)=O)CC(C)(C)O1.C1(C(=O)N)(OCC)CCOCC1 C1(NC(=O)CC2CSC2)CC2CN(C(C3(C(F)(F)F)CCOCC3)=O)CC2C1 N1(C(c2cc(C)sn2)=O)CC(C(N2CCC(C(C)C)C2)=O)C(F)(F)C1 c1(OCC(CN(CC(=O)NCc2ccccc2)CCC)O)ccccc1C N1(C(c2c(CC)cc[nH]2)=O)CC(NC(c2nccnc2N)=O)C(n2ccnn2)C1 C1(CCN(C(=O)CCCC2CCC2)C)CCN(C(=O)CCCC2CCC2)CC1 S(=O)(=O)(c1c[nH]ccc1=NCCCC1CCCC1)N(CC)CC1CCCO1 C=CC(C)(O)C(=O)N1CCN(C2CN(C(c3ccc(NC)cn3)=O)C2)CC1 CC1(C)CCCC1C1CCN(C(c2n[nH]c3ccc(F)cc23)=O)C1 c1(C(=O)N)cc(C)nc(O)n1.C1(NC(c2nc(OCC)sn2)=O)CCOCC1 C(C1CCN(C(=O)C(C)n2cccc2)CC1)=CC(NOCCCOC)=O C(CC(F)F)(C(=O)NC1(CO)CC(F)(F)C1)N(C(C=C(C)C(F)F)=O)C CC(C)C(C)C(CNC(c1nccn1C)=O)NC(c1csc(Br)c1)=O N1(C(CSCCC)=O)CCCC(O)(CCNC(=O)CCOC)C1 C1(C(=O)NC(C)(C)C(C)C)(OC)CCN(c2cc(-n3cccn3)ncn2)CC1 C1(N(C(=O)CC2OCCO2)C)CCCC(N(C(=O)CC2CC=CC2)C)C1 [N-]=[N+]=NC1CCC(C(N2CC3(CC3)CC2CC(=O)NC2CCOCC2)=O)C1 C1(CNC(c2cc(C)oc2C(F)(F)F)=O)CCN(C(=O)C2=NOCC2)CC1C c1(C(=O)NCC(C)(C)NC(=O)CCCC(=O)c2cccs2)ccc([N+](=O)[O-])o1 n1(CCC)ncc(C(N2CCCC2CN(C)C(c2nnn(C)n2)=O)=O)c1C n1(CCCC)cc(C(=O)NC2CN(C(C3CC(=O)N(C)C3)=O)CC2O)c(C)n1 Cc1nonc1CC(=O)NCC(C)(C1CC1)NC(=O)CCC.[SH](C)(=O)=O.N C#CCC(C)(CNC(c1csc(C)c1)=O)CO.C(=O)(C(C)(C)n1ccnn1)N N1(C(C2CCC(CNC(c3cncc(CC)c3)=O)O2)=O)CCN2CCC1C2 CCC(CC(F)F)C(=O)N1CC2CCC1C(CNC(c1c(C)nn(C)c1Cl)=O)C2 N1(C(C2(F)C(C)C2)=O)CCCCC(CNC(=O)CN2C(=O)CN(C)C2=O)C1 c1(C(N(C)CC2N(C(c3nc(C)oc3)=O)CCCC2)=O)cnc2scc(C)n12 CC1CN(Cc2cccnc2)CC(C)O1.c1(C2CNC(=O)N2)cc(Cl)cc(Cl)c1 N1(Cc2cn(-c3c(CC)cccc3)nn2)CC(=O)Nc2ccccc2C1 C1(CC)CN(C(C23CC(F)(C2)C3)=O)CC1C(N1CC2CC2C1)=O C1(C(N(CC(CNC(c2nc(C)oc2)=O)(C)C)C)=O)SC2C=CC1C2 c1(-c2cncc(C(=O)NC(COC)C(C)C)c2)ccc(OC)c(OC)c1 C=CCC(C(=O)NCc1cc(C)c(C(=O)NCCC2CCCO2)o1)OC c1(OC)cncc(C(=O)NCC2CC2NC(=O)CC=CC(C)(C)C)c1 C1CC2(CCN(C(=O)C(O)CC(C)(C)C)C2)CO1.n1(CC)ncc(C(=O)N)n1.C C1(C(N(CCC)CC)=O)CC(NC(c2cnsc2)=O)C(O)C1 c1(C(=O)NCC(C)N(C(C(C)Cc2ccc(F)cc2)=O)C)cc2ccsc2n1C N1(C(CCCN(C(C)=O)C)=O)CCC(CF)(NC(=O)CC2CC(F)(F)C2)C1 C(=O)(C1=NN2CCCN=C2N1)NC(CCNC(c1ccn(C)c1)=O)(C)C c1(N2CCC(NC(=O)NC3CC(F)(CF)C3)C2)ccc(F)cc1 C(CN=c1ccnc(N2CCOCC2)[nH]1)=CCCNC1C(C)CCC1 N1(C(CCCC)=O)CCC(NC(=O)Cc2csc(Cl)n2)CC1 CC1CCc2[nH]c(=NCCCC3CC3)[nH]c(=NCC3CCCS3(=O)=O)c2C1 c1(CC(N2C3CC(OC)C(C3)C2)=O)n[nH]c2c1CCCC2 CC1CCCC1(C(N1CCCC(CF)C1)=O)NC(c1cc(O)n(C)n1)=O N1(C(c2cc(CC)c(Cl)cc2)=O)CC2(CCCCN(C(=O)Cn3cccn3)C2)C1 c1(OC)ccccc1C(C(N1CCC(F)(CNC(=O)C2=NOCC2)C1)=O)OC c1(C(C(N2C3CC(NC(C(CCSC)O)=O)C(C3)C2)=O)=O)cc(F)c(F)cc1F CC(O)C(C)C(=O)NC(C)(C)CCCNC(c1conc1C(F)(F)F)=O O=C1COc2ccc(S(=O)(=O)N3CC(CNC(c4ccc(O)cn4)=O)C3)cc2N1 C1(CCNC(CCCCC=C)=O)CCN(C(=O)Cc2ccc(F)cn2)CC1(F)F Cc1n[nH]c(C)c1C(=O)NCC1CCC1NC(C1CC(OC(F)F)C1)=O C=CCCC(C(=O)NC1CC2C=CC1C2)NC(c1cc(C)nn1C)=O C12(C(=O)NC(CC)CO)C(NC(c3cnc(C)s3)=O)C3CC1C2C3 Cc1nc(N2CCCC2CN(C(=O)CC2CCC=CCC2)C)c(Cl)cc1C#N c1(OC)ccc2oc(CN3CC4CCN(C(=O)C(N)=O)C4C3)cc2c1 C1(C(=O)NC2C(NC(c3ccc(OC(F)F)cc3)=O)C2)(CO)CCCCC1 c1(-c2onc(C(C)[SH]=CCCNC(=O)OC(C)(C)C)n2)ccc(Cl)cc1 c1(CN2C(C(=O)NCCc3ccccc3F)CC(C)C2)cc(O)ccc1Cl N1(C(C(c2cccnc2)NC(CCCCOC)=O)=O)C2C=CCC1CC2 c1(C2C(C(N(CCCC)CC)=O)C2)ccnn1CC(C)C.C1(C=O)CC1F.N N1(C(C=C(CCC)C)=O)CC(NC(=O)Cn2nc(O)ccc2=O)C2CCCC2C1 C(CC)C(C)C.c1(COC)nocc1C(=O)N.c1(C=O)ccn(CC(F)F)n1 c1(OC)ncc(CNC2CCCC2C(=O)Nc2cc(I)ncn2)cc1Br C(=O)(CCCCCC(C)C)NC1CCN(C(CSc2ccc(C)cc2)=O)C(C)C1 c1(C(N(CCC(C)NC(CCN(C)CC)=O)C)=O)cc(Cl)c(C)cc1Br c1(C(N2C(CC)CN3CCCC3C2)=O)cc(Br)cc2cccnc12 S(=O)(=O)(c1ccc(C#N)c(N(C)CC2(F)CCC2)c1)NC1CC(C)SC1 CON1CCC(C(N2CC(NC(=O)CN(C)C(N)=O)CC(O)C2)=O)CC1 c1(CC)cc(C(N2CCC(CN(C(=O)CSc3ccccn3)C)C2)=O)ccc1C Cc1ccc(=O)n(CC(=O)N(C(C)CCNC(=O)CC2CC(C)(C)CO2)C)c1 C1(CNC(c2n[nH]c3c2CCC3)=O)CCN(C(c2ccc(F)c(F)c2)=O)C12CC2 c1(C(N2CC(C)(CC=C)C2)=O)cc(S(=O)(=O)NCC(N)=O)ccc1F C1(CCOC)CC(N=c2[nH]c(N3CCN(C4CC4)CC3)nc3cc(C)ccc23)C1 C1(NC(C(C)=C(C)C)=O)CCCCC1NC(=O)CCS(C)=O C1(C(=O)NCC(CC=C)NC(=O)Cn2ccc([N+](=O)[O-])n2)CCn2nccc2C1 C(c1csc2ccccc12)=CC(=O)NCCC(C)NC(CC(=O)NCC)=O c1(CC(=O)NC2CCCC(NC(C(CCC)OC)=O)C2)cn2cc(C)sc2n1 C1(NC(=O)CCN2CCCCCC2)CCCOC12CCN(C(=O)CCCF)CC2 n1(CC)nc(C)cc1C(N1CCC(C(C)(C)NC(c2ccns2)=O)C1)=O c1c[nH]c2cccnc12.C1(N(CC(C)C)C)CCN(C(=O)C)C1.C1(C)(C)CN1.O C1(C(=O)NCCC(C)F)CN(C(=O)OC(C)(C)C)CC1OC1CCSCC1 C1(NC(C(COC)OC)=O)CC2CCC(C1C)N2C(c1cnc(N)c(O)c1)=O CC1CC(C(=O)NCCOc2ccc(Cl)cc2)CN(C(=O)C)C1.C1CCCC1.S N1(C(C2(CC)CCC2)=O)CCc2c(-c3ccc(S(C)=O)cc3)cccc2C1 C#Cc1cccc(OCC(=O)NCCC(C)NC(=O)CC(C)C(=O)OC)c1 C(=O)(C1COc2ccc(F)cc21)N1CCC(NC(C(C)S(N)(=O)=O)=O)(CO)CC1 N1(C(C(c2ccco2)NC(C(COC)COC)=O)=O)CCC2(CCC2)C1 C(C(=O)OC1(F)CC1)(c1cscn1)NC(=O)OCCOC(C)(C)C C1(F)(C(N(C(C#C)C2CCC2)C)=O)CCN(C(=O)C(=O)C(C)C)CC1 CC(C)(CCCO)C(=O)NC1(CO)CCCN(C(C2CCOC(=O)CC2)=O)C1 n1(CC)nc(C)cc1C(=O)NCC1(C(N2CC3CCC3C2)=O)CCCCC1 CC(C)CC(C)(O)C(=O)NC1CC(C(=O)NC(C)(C)CF)CC1O CCCCC(CNC(C1(SC)CCC1)=O)NC(C1CCC(CN(C)C)O1)=O C1(C(C)NC(CCN(CCCCC)CC)=O)CCCCN1C(=O)Cc1ccoc1 c1(CC)cncc(C(=O)NC(C)(CNC(=O)C(n2nc(C)cc2C)C)CC)c1 c1(C(=O)NCCCCCN(C(C(C)CO)=O)C)cc(C(F)(F)F)ncc1F N1(C(C(C2CCOC2)NC(C2CC3C=CC2C3)=O)=O)Cc2ccc(O)cc2C1 Cc1ccn(C(C)CC(=O)NCCCCCN(C)C(c2n[nH]cc2Br)=O)n1 C(C)(C)(C(=O)N1CCC1C(=O)NC(c1nncs1)C)OCC C(C(C)(C)C#CC(=O)N(C1CCC1O)C)NC(CCC=C)=O C1(NC(CS(C)(=O)=O)=O)CCCC(CNC(=O)Cc2ccc(C#N)nc2)CC1 C12(C(=O)NCc3cn(CC(CC)O)nn3)CCC(CC1)OC2 C1(NC(CN(CCC#C)C)=O)COC2CN(C(c3cnn(C)c3N)=O)CC12 C(C(C(=O)NC1(C)CC(F)C1)NC(c1cc[nH]c1CC)=O)OCC c1(C(N2C(C(=O)NCC(CC)OC)C=CC2)=O)cc(O)ccc1C C(=O)(CS(=O)(=O)Cc1csc(C(C)(C)C)n1)NC(CC)COC N1(C(c2n(C)ccn2)=O)CCN(c2ccc(NC(=O)CC3CCC3)cc2)CC1 c1(C(NCCCC)=O)ccc2c(c1)CC(C)O2.C(CC(=O)N)OCCOC c1(N2CCC(C(CC)CC)CC2)nccc(=NCc2ccc(N)c(C)c2)[nH]1 c1(C(=O)N)cc(O)cc(F)c1.CC(C)C(C)C.c1(CC=O)cncn1C1CC1 C(CC(C)C(=O)N1CCCC(N(C(=O)CCSC)CC2CC2)C1)OC N1(C(c2[nH]cc(C)c2)=O)CCC2CCCC12C(=O)NC(CN(C)C)C(C)C c1(C(C(=O)N(C)CC2C3CN(C(=O)CCC(N)=O)CC23)O)ccc(Cl)c(F)c1 C(=O)(C(CNC(C1CC(C)CC(C)C1)=O)CC(C)C)N(CC(C)C)CCC CC1(C2CCN(C(=O)CCCCCCNC(C3CCC(=O)CC3)=O)C2)CC1 c1(NC(C2CC3CC3N2C(=O)CCN2CCOCC2)=O)ccc2c(c1)OCO2 c1(NC(CN(C2CC2(Br)Br)C)=O)ccc(Cl)cc1 C1(NC(C(N2CCSCC2)C)=O)CC(=O)N(C2CN(C(=O)C(C)N3CCC3)C2)C1 C#Cc1ccc(C(=O)NCC(C)(C)CSC)cn1 C1(NC(C=CCOC)=O)CCCC(C(=O)N(C(C)C(N)=O)C)C1 NC12CCC(C(N3CCCC(c4ccc(F)c(O)c4)C3)=O)C1CC2 CCCC(CNC(=O)C=CCO)C(=O)NCc1cc(C2CC2)no1 c1(C(=O)NC2C(CNC(C(C)Sc3ccccn3)=O)CCC2)cc2scnc2[nH]1 c1(C(N(C(C)CNC(c2cccnc2)=O)CC)=O)sccc1C#N N1(C(CCc2cncc(C)c2)=O)CC2CC(NC(C3(N4CCCC4)CC3)=O)C2C1 C(=O)C(F)(F)c1ccsc1C(F)(F)F.C(C(F)C)NC(C1C=CCC1)=O.N CCC(C(=O)NCC1(C)CCCN1C(c1cnc(C(F)(F)F)nc1)=O)C(C)C C=C(C)C(CC(=O)NC(C)(C)CC(=O)N(C)Cc1cncnc1)OCC N=c1ccc2c(CNC3CC4CC3CN4CCc3ccccc3)cc(O)nc2[nH]1 C(=O)(C(O)CC(F)(F)F)N(CC)CC.c1(C=O)ccc(Cl)cc1.C(C)=O.N N1(C(CC=C=C)=O)CCC(O)C(NC(c2ncoc2-c2ccco2)=O)C1 C1(NC(C(OC)OC)=O)CCC(C(=O)NC(c2ccc(Br)cn2)C)CC1 N1(C(c2n[nH]c(C3CC3)c2)=O)C2CCC1CC2.C1(C=O)CN(C(N)=O)C1.CC N1(C(=O)CC2CC2)CCC(C2CCCN2C(C2CCSCC2)=O)C1 Cc1ncc(Br)c(N2CC3CN(C(C4CCC(CO)CC4)=O)CC23)n1 C(=O)(C(CC(F)F)N(C)C(c1ccsc1Cl)=O)NC(CC#C)CC c1(COCC(N2CC(NC(c3c(C)nn(C)c3)=O)C2)=O)ccc(C#N)cc1 c1(OC)cc(C)cnc1C(N1CCCC1CCCNC(c1n[nH]cc1C)=O)=O c1(C(=O)NCC2C3CC2N(C(c2cncc(F)c2)=O)C3)cc2ccccc2s1 CC1(C)CC(O)CCN(C(=O)CC2CN(C(c3ccoc3C3CC3)=O)CCO2)C1 CN(C)NC(=O)CCC(=O)N1CC(CNC(C2CCC(=O)NC2)=O)CC1(C)C N1(C(c2nnn(C(C)(C)C)n2)=O)CCC2(CC2C(N2C3CSCC2C3)=O)C1 C1(COC)CCN(C(C2CCCC23CC3)=O)CC1.C12(C(=O)N)CCCC1C2(F)F C1(OCC)CC(C)N(c2ccnc(C(C)(F)F)n2)C(C)C1 N1(C(C(CC)(C)C)=O)CC(OC)CC(NC(=O)COc2cc(F)cc(F)c2)C1 N1(C(C2N(C)C(=O)CCC2)=O)CC2CCC(C1)N2C(c1ccc(F)s1)=O C12(C(N3CCCC3)=O)C3CC(CC13)C2(F)F.n1(CC(N)=O)cc(C=O)nn1.N c1(C(N2C(CCC(N3CCOC(C4CCC4)C3)=O)CCC2)=O)ccc(F)cc1F C1(C=O)CCCCC1n1ccnc1.c1(CCC(=O)NCC2CC2)cc(Cl)no1.N C1(NC(C(C=C)(C)C)=O)CCC2(CCCN(C(=O)CC3(C)CC(F)(F)C3)C2)C1 C1(C2CCCN(C(=O)C(F)OC)C2)(NC(c2cn(CC=C)nc2)=O)CC1 N1(C(C2C=CCC2)=O)CCC2(CCCN2C(c2cn3ccccc3n2)=O)C1 C(=O)(CCN=c1[nH]ccs1)N1C(CNC(=O)CC2(C3CC3)CC2)CC1 C1(c2ccn(C)c2)CCCN(C2COCC2O)C1 C=CCCCCCCC(=O)NC(CCSC)C(=O)NC12CC(C1)C2 C1(NC(C2CCCC2)=O)CN(C(C2CCCC2(F)F)=O)CC2(CC2)C1 C(=O)(CCC(F)(F)C(F)(F)F)N1C(CNC(CC(C=C)CCC)=O)CC(O)C1 C#CC1(NC(=O)CNC(C2CCCOC2C)=O)CC2CCCC12 Cc1ccc(O)c(C(=O)NCCn2ccc(C(N3CCS(=O)CC3C)=O)c2)c1 N(C(=NCCC1CCCS1(=O)=O)N(C)Cc1ccc(OC)cc1)CC(=C)C Cc1cn2c(C(=O)N(CC(C)N(C)C(C3CCC4(CCC4)C3)=O)C)c(Cl)nc2s1 N1(C(C2(CC=C)CCN(C(=O)CC)C2)=O)CCC(F)(F)C(F)C1.C(=O)(CO)N N1(C(C)=O)CC(CC(=O)NOCCCO)C2(CC2)C1.Cc1noc(N)c1 c1(CN(C(C2CC(CC(=O)O)C2)=O)CC2CCCSC2)ccncc1 [N-]=[N+]=Nc1ccc(C(=O)NCCOCCNC(C2CCC(F)C2)=O)cc1 c1(CC)nc(C(=O)NC(C)CN(C(=O)C(C)OC2COC2)C)cs1 N1(C(C(CCC)OC)=O)CCN(C(c2ccccc2)=O)CC1c1cn[nH]c1 N1(C(COCC=C)=O)CCN(C(c2cn(C3CC3)nn2)=O)CC12CC2 c1(CC)cc(C(=O)NCCN(C(=O)CC2CC(F)(F)C2)C)ccn1 N1(C(c2cnc(CC)s2)=O)CC2CC(C(=O)NC3C=CC(C)(C)CC3)C(C2)C1 C1(C(C)NC(C(C)=C(C)C)=O)CN(C(c2noc(C)c2Br)=O)CCO1 C1(NC(CCCOC)=O)C2CC1CN(C(=O)C(C)=CC1CC1)C2 c1(C(N2CC=CC(NC(C(C)C3CCC3)=O)C2)=O)cccc2c1CCCCC2 C1(CNC(C=CC2N(C(COCC)=O)CCC2)=O)CCC(C)(C)CO1 c1(C(N(C(CN(C(C2C=C(C)CS2)=O)C)C)C)=O)ccc(-c2ccccn2)nc1 N1(C(C(=Cc2cccs2)C)=O)CCC2CN(C(=O)COCP(C)(C)=O)CCC2C1 CCC(CCC(=O)NCC1CCC1(F)F)NC(C1(COC)CCCC1)=O c1(C(N2CCN(C(CC3(C)CCCCC3)=O)CC2)=O)cc2nc[nH]c2cc1N C(C(C)(C)CN(C)C)N(C(C)C(=O)NC(C1CC1C)=O)C.c1ccccn1 CC1CCCC(N(C(=O)C(CC2CC2)NC(=O)C=CC2CC2)C)C1C C1(CC=C)(NC(C2CCOC2C=C)=O)CCN(C(=O)Cc2ccc(C)o2)C1 N12CCC3CCC(C1)N3C(=O)CC2.N1(CC(CC)OC)CCCCCC1 Cc1c(C)c(C)c(-c2csc(-c3ncccc3C(F)F)n2)c(C)c1C c1(CC(=O)NCC(O)C)sc(C)cc1C.c1(C=O)cn(CC(N)=O)nn1.CC N1(C(=O)Nc2c(C)cnc(Br)c2)CCC2(CC1)CC2(F)Br c1(OC)cccc(C(=O)NC2CCC(CNc3cccc(OC)c3)C2)n1 N1(C(C2(CC)CCOC2)=O)CCC(C(=O)NCc2conc2C)C(C)C1 N1(C(C(C)NC(C)=O)=O)CCC(CN(C(=O)C(C)(C)N(C)C(C)C)C)C1 C1(CCNC(c2cn(CC=C)nn2)=O)CN(C(c2cncc(C)c2)=O)CCCO1 C(=O)(C1CCCc2cccnc21)N1C(CNC(CC=C)=O)COC(C(F)(F)F)C1 C1(C(N2CC3C(c4cn(C(c5ccccn5)C)nn4)C3C2)=O)CC2(C1)CC21CC1 c1(C(=O)NC2CCN(C(CCN3CCN(CC)CC3)=O)C2)ccc2[nH]ccc2n1 C(=O)(C(C)C(O)CCCCC)NC1CN(C(CCC=C=C)=O)CC(F)C1 C12(C(=O)NC(C(=O)N(C3CC3)C)C3CCC3)CC(C1)C2.c1ccoc1 N1(C(C(C)(C)C2CC2)=O)CC2CCCC2(NC(C2CCCCS2)=O)C1 c1(C(=O)NCC(C)CN(C)C(C2CCCS2)=O)cccc2nccn12 N1(CC(=O)NCC(CC)NC(=O)C=Cc2cocn2)CCCC1CO C12COCCN1C(=O)CN(C(=O)Cc1cnns1)C2.C(CSC)(C(=O)N)OC.C C1(C=O)CC12CC(F)(F)C2.c1(SCC(=O)NC(C2CC2)C)ccccn1 c1(CNC(C(Cn2ccnn2)NC(C2C(C)OCC2)=O)=O)cccc(C#N)n1 c1(C(N2CC(CC)OC(CC)C2)C(=O)NCCC)cc(OC)c(Cl)cc1F Cc1nc(C)n(CCC(=O)NCC2(F)CCN(C(c3ccc(CO)cc3)=O)C2)n1 C(CC(C)(C)C(=O)N1CC2CC(CNC(c3cc(Cl)ccn3)=O)C2C1)OC C(=O)(C1=CC2C=CC(C1)C2)NC1CC(C)CN(C(C2CN(C(N)=O)C2)=O)C1 C1(CC(=O)NC2CCCSC2)(OC)CN(C(=O)CC2CCC(=O)C2)C1 N1(C(Cc2c(C)nc[nH]2)=O)CCN(C(c2cscc2C(F)F)=O)C2CCC12 C1(NC(CCc2ncc(C)[nH]2)=O)CN(C(c2cnn(CC(F)F)c2)=O)CC12CC2 C=CCC(C)C(=O)N(C(C)CNC(c1ccc(NC(C)=O)cn1)=O)C N1(CC(=O)N(C2CCCCC2N(C)C(C2CC2(Cl)Cl)=O)C)C(=O)CCCC1=O c1(CC(=O)NC(C)CN(C(=O)Cc2nc[nH]n2)C)ccc(F)cc1[N+](=O)[O-] c1(C(N2C(CCNC(C3C(OC)CC3)=O)COCC2)=O)ccc(Cl)cc1N C12(NC(CCC(=O)NC)=O)CCN(C(c3cccc4cncn34)=O)CCC1C2 c1(CC)nc(N2CCCC2C2CCN(C(c3c(C)cnn3CC)=O)C2)cc(C)n1 c1(C(=O)NC2CCC(CNC(CC(C)C3CCCO3)=O)C2)cccnc1F C(CC(C(C)(C)C)NC(c1cc(C)co1)=O)N(C(CN1CC(CC)C1)=O)C N1(C(CCCn2ncc(C)c2)=O)CC(CC(=O)NCc2c[nH]ccc2=O)CC1C c1(SCC(=O)NCCC(O)C)ccc([N+](=O)[O-])cc1.C(=O)C(F)n1cccn1.N C1(NC(C(F)OC)=O)CCN(C(c2n[nH]c(C)n2)=O)CC1C C1(C(N(CCCN(C(COCc2ncc(C)o2)=O)C)C)=O)CCN2CCOCC12 N1(C(C2C(CC)C2)=O)C2CCC1(CNC(C1C(F)(F)C13CCC3)=O)CC2 N1(C(CC2CCN(C)C2)=O)CCCC(O)(C)C1.c1(C2C(C=O)C2)ccc(F)nc1.N Cc1ccc(SCC(=O)NCc2cnn(C(C)(C)C(=O)O)c2)cc1 C1(CNC(CCc2ncc(C)[nH]2)=O)COCCN1C(c1ccc(Cl)cc1)=O C(=O)(C(C(C)(C)O)NC(=O)CC1CCSC1)N(C12CC(C1)C2)C CCN=C(NCCCNC(C)=O)NC1CC(C)N(C2CC2)C1 C1(C(C(=O)NC2C(C)C2(C)C)(C)C)CCCN(C(=O)CCN2CCCC2)C1 N1(C(Cn2cc(SCC(N)=O)nn2)=O)CCC(C2(CC3CC3)CC2)C1 C1CC2CN(C(=O)C#CC(=O)N(C)C)CC2C1.Cc1ncsc1COCC(=O)N N1(C(C(C)N=[N+]=[N-])=O)CCC2CC(C1)CN(C(=O)CCCC(F)(F)F)C2 c1(SC(C(=O)NC(CNC(c2c(C)coc2)=O)C(C)C)C)nc2ccccc2[nH]1 CN1CCC(N2CCC(NC(C3CC3C(F)(F)F)=O)C2)CC1 O=C(N=S1(=O)CCC2(CC1)OCCO2)c1cnn(Cc2ccccc2)c1Cl C1(C)(NC(C=CCCC)=O)CC(NC(=O)Cc2ccc(Cl)s2)C1 N1(C(C2C(C#C)C2(C)C)=O)CC(NC(c2c[nH]nc2Br)=O)CCC1C N1(C(c2c(CC)nns2)=O)CCCC(C)(C(=O)NC(c2nc(C)cs2)C)C1 C(=O)(C(C)(F)C(C)(C)F)NCCCC.c1(C(=O)N)cnc(CCC(F)(F)F)s1 C12(C(=O)NC3(CC=C)CN(C(c4c[nH]cc(C)c4=O)=O)C3)CSCC1C2(F)F Nc1ncc(O)cc1C(=O)NCC1CCCCC1.c1(C=O)ccc([N+](=O)[O-])s1.N CC1(C)CCCC2(CCN(C(C3(N)CC(O)(C(F)(F)F)C3)=O)C2)C1 c1(CNC(c2ncc(C)c(C)c2)=O)ccc2c(c1)CN(C(C1CC1C)=O)C2 C(=O)CCC(=O)NN(C)C.C(=O)CCC.C(=O)(CC1CC1)N.C(=O)(C)OC C#CCCCC(C)C(=O)N(CCCC(N1CC(CO)OC(C)C1)=O)C C1(CNC(=O)NC)CCCCN1C(c1ccccc1OCC(F)(F)F)=O c1(CNC(C(c2ncc(Cl)s2)N(CCC#N)CC)=O)cccc(Br)c1 CN(C)C1CCc2cc(NC(=O)NC(c3cccnc3)C3CCCCC3)ccc21 c1(C=O)cc(C)nc2c(C)cccc12.C12(CNC(C(C)SC)=O)CC(C1)C2 C(=O)(C#CC1(C)COC1)NC(CC=C)C(=O)N(CCCCCC)C N1(C(c2cc(C)no2)=O)CCC2(CCCN(C(C3CCn4cncc4C3)=O)C2)C1 C(=O)(C(F)(F)C1=CCOCC1)NCC1CCCN(C(=O)CC2CCCC23CC3)C1 N1(C(C2(CC)CCOCC2)=O)CC2CCC(C1)C2NC(=O)CCc1cc(C)cs1 N1(C(C(CCC)F)=O)CC(C)(C(=O)NCC(O)CCOC)CC1(C)C C1(NC(CC=C)=O)CN(C(c2cccc(F)c2C(C)C)=O)CC1C1CC1 C(=O)(C1=C(Cl)CCCC1)N.n1(CC(N2C(C(C)C)CCC2)=O)cc([N+](=O)[O-])cn1 N1(C(C2CCCO2)=O)CC2C3CCC(C2C1)N(C(=O)C1CCc2c[nH]nc21)C3 c1(CCC=O)ccc(C=O)nc1.C(=O)(CC1(CC(=O)NCC)CC1)OC C(=O)(CCCS(N)(=O)=O)NC1CCN(C(C(CCOC)(C)C)=O)CC1C C(=O)(C1Cc2ccccc21)N1CCC2(CN(C(c3n(C)nc(O)c3)=O)C2)C1 c1(CC(=O)NC2CN(C(C(C)Oc3cccnc3)=O)CC2C)cccc(F)c1O C1(C(N2CC(CC(C)(C)C)C2)=O)(OC)CC(CF)C1 C(=O)(C(CC(C)C)O)NCC1(C(C)NC(c2cncc(NC)c2)=O)CC1 c1(OC)ncc(C(N2CC=C(CO)CC2)C(=O)Nc2ccccc2)cc1Br C1(C(N(CCNC(C)=O)C)=O)CC(F)(F)CN1C(=O)C1=CCCCC1 C1(NC(CCCN(C)C)=O)CC(F)CN(C(C23CCCC2(C(N)=O)C3)=O)C1 C(=O)(C1=CC2CCCC12)N1CCC(CCC)CC1.n1(CC)nc(C)cc1C(=O)N Cc1cccc(CN2CCCC2CNC(=O)CN2CCCC2=O)c1 Cn1cnc(C(=O)NC(C)(C)CC)cc1=O.N1(CCCC(=O)N)C(=O)CCC1=O N(C(=NCC12CC(CN1C)C2)NC(CC)CC)CC(COCC)(C)C N1(C(C2CCN(OC)CC2)=O)CCC(NC(c2cocn2)=O)C12CCCC2 N1(C(CCOCCOC)=O)CC2COCC(C1)C2.C1(C(=O)N)CCCC(F)(F)C1 Cc1cc(C)c(C(=O)NCCCCC(C)NC(=O)CC2(C)CCCC2)c(O)n1 N1(C(Cn2ncc(C#C)c2)=O)CCN(C(=O)C(C)Cc2ccco2)CC12CCC2 N1(C(CNC)=O)CC2CC(C1)N2C(c1ccc(C(N)=O)o1)=O.c1ncccn1.C C1(NC(c2cnn(-c3ccccc3)n2)C)CC(C)(C)SC(C)(C)C1 CCCC(C)(C)C(=O)NC1CN(C(c2ccnc(Br)c2F)=O)CC1(F)F c1(C(=O)NC2CN(C(C(CCOC)OC)=O)CC2CO)cc2n(n1)CC(O)CO2 C1(C(=O)OC)CC2CC1(CNC(c1ccc(N(CC(C)C)C)nc1)=O)C2 C1(NC(CC2CN(C)CC2O)=O)CC2CC(NC(c3cc(N)cc(O)c3)=O)C1C2 C1(c2nnnn2CCC)(NCCCC(=C)C)CC2(C)CCOC12 CC1CC=C(C(=O)NCc2cc(O)nc(CNC(=O)CC(F)F)n2)CC1 C1(OC)CCC12CC(C(=O)N(C1CCC(NC(c3ccccc3Cl)=O)CC1)C)C2 c1(C(N2C3CN(CC=Cc4cccc(OC)c4)CC32)=O)noc2c(Cl)cccc12 C1(CCNC(c2c(OC)ccs2)=O)CN(C(=O)CSC2CC2)CC(C)O1 N1(C(c2nc(C)sc2)=O)CC2CCN(C(c3occ4c3CCC4)=O)CC12 Cc1nc2c(s1)CN(C(C1CN(C(C3(CC4CCC4)CC3)=O)CC1C)=O)C2 C1(CNC(=O)CO)CC2CN(C(c3cc(Cc4ccccc4)on3)=O)CC12 C#Cc1ccc(CCNC(c2nnnn2C2(C)CC2)C(C)C2CCCC2)cc1 C(=O)(C(C)C(C)(C)C)NCCCNC(C)=O.C1(CC=O)CC(=O)NC1=O c1(C(=O)NCC2(NC(c3c(C)nc(C)[nH]3)=O)CCC2)ccc2c(c1)CC2 C1(NC(C2CCC2)=O)CC2CN(C(=O)C(F)(F)c3ccccc3)CCN2C1=O C#CCC(C)C(=O)NCCC1(NC(=O)CC)CCC1.c1(C=O)ncccc1O.N c1(OC)cc(CC(=O)NCC2CCCC2)ccn1.C(=O)(CC(C)(C)C1CC1)N Cc1cc(OCCC(=O)NCCCNC(c2cocc2C)=O)c(C)c(C)c1 N1(C(c2cnc(OC)nc2)=O)CCC(CO)C(NC(=O)CC2CC2(C)C)C1 c1(C(=O)NC2CCN(C(c3cccc(C4CC4)c3)=O)C2)ccc2nccn2c1 N1(Cc2c(C(C)C)cccc2)C(=O)CCN(CCOC2CCCCC2)C1=O CCCCCCC(C)C(=O)N1CC2CC(C1)N(C(=O)CCN1CCC1)C2 c1(C(=O)NCCNC(CC(=C)Br)=O)cc(C)n(-c2ccc(C(C)C)cc2)n1 N1(C(c2c(NCC)scn2)=O)CC(C)N(C(C2CCCC2CC)=O)CC1C C1(NC(CCN(C(CCn2c(C)ncc2)=O)CCCO)=O)CNC(=O)OC1 N1(C(CC(C)c2cnn(C)c2)=O)CCC(NC(C2CC(=O)NC(C)C2)=O)C(F)C1 C1(C(=O)NCCCNC(=O)C)(COC)CCC1.C1(CS)CCOC1 c1(C(N2CC3(C(C(=O)OCC)C3)C2)=O)ccc(B(O)O)cc1 C1(NC(C2C(=C)C2)=O)C=CCC(C(=O)N(C(C)CC2CC2)C)C1 c1(C(=O)NCC2CC3CCC2N3C(=O)CCCC=CBr)cnn2c1NCCC2 c1(C(N(C(=O)CCN(C2CCCCC2)C)CCOC)=O)nccc2c(Cl)cccc12 C(=O)(CC1=CCN(C(=O)C(F)CC2CCOC2)CC1)N1C(CC)C(C)CC1 N1(C(c2c(CC)cno2)=O)CCC2(C1)CN(C(=O)C1=NOC(C)(C)C1)CC(C)O2 C#CCC(C(=O)NCC(C)(O)C(F)F)NC(=O)C(C)SC(C)C C=C(C)CC(C(=O)NCC(C)(CC(C)C)NC(=O)Cc1scnc1C)OC c1(C(N2CCC(CO)(COC)C2)C(=O)NCCC)cncc(C(C)C)c1 N1(C(C(C)Cc2cnc[nH]2)=O)CC(F)CC1CN(C)C(C1CC(O)C1)=O C1(N(C(CC2CN(C)C2)=O)C)CCCC2CN(C(=O)COCCCF)CC12 C1(CC(=O)NCC2(O)CN(C(C3CC(OC)C3)=O)C2)C(=O)NN=C1C c1(C(=O)NCCC(C)(C)NC(C=Cc2c(C)cccn2)=O)cnc2c(c1)CCC2 c1(SCC2CC(NCC(C3CCOC3)OC)C2)cccc(C(F)(F)F)c1 N(C(=NCc1ccc(F)cc1)NCC(Cl)C(F)(F)F)C(CC)C C1(CNC(=O)Nc2ccc(C(=O)NC(CC)C)cc2)C2CCOC2C12CCC2 N1(C(C2CCC(OC)C2)=O)CCN(C(c2cnc(SC)nc2O)=O)C2CCC12 c1(C(N2CCC(CNC(CC(C=C)(C)O)=O)C(C)C2)=O)cccc2ncoc12 c1(C(=O)NCCCN(C(=O)CCS(C)=O)CC)cn2nc(C)sc2n1 c1(C(=O)NC2CCCCCN(C(c3n(C)ncc3)=O)C2)nnc2ccccc2n1 CC1CC(NC(=O)C(C)CC2CCCC2)C(=O)O1.c1(CCC(=O)N)cccnc1 N1(C(Cc2cccc(OCC)c2)=O)CCCOC(CNC(=O)C2=CCCC2C)C1 N1(C(c2nc(C)nc(O)c2)=O)CC2(C1)SCCC2NC(=O)CCN1CCOCC1 C(=O)(C#CC1CCCC1)N1CCC(C(C)NC(c2c(C)cc(Br)o2)=O)C1 N1(C(c2ccc(OCC)nc2)C(=O)NCCOC)CCC(O)(C(N)=O)CC1 C1(C(=O)OC)(OC)CCN(N2CCN(c3nc(F)c(F)cc3F)CC2)C1 c1(C(=O)N)cc(C)c(C)cc1Cl.Cc1cc(C2(C(=O)NC(C)CCC)CC2)on1 N1(Cc2cnn3c2CC(C)CC3)CCC2(CC1)CC(NC(=O)C(F)(F)F)CO2 C(CCC(C)CC(=O)NC(C)C(C)(C)NC(=O)C(=O)N)=C(C)C.c1ncc[nH]1 CC1(CNC(C2CCCC3(CC3)C2)=O)CCCN(C(C2(N=[N+]=[N-])CC2)=O)C1 c1(OCCOC)cc(NC(=O)C(F)C2CN(C=O)C2)ccc1F.C(C)(C)C C1(C(=O)OC)CCCCN1C(=O)C(F)CC1CN(C(=O)C#CC(C)C)C1 c1(NC(C2(O)CCN(C(=O)CO)C2)=O)cc(Cl)nc2ccccc12 N1(C(COc2cccc(C#C)c2)=O)CC2COCCC2(NC(c2ccco2)=O)C1 N1(C(CN2CCC(C)C2)=O)CC2CCN(C(C3(C4CC4)CC3)=O)CC12 C(=O)(C=C(Cl)Cl)N(CC(CC)NC(=O)CCc1nc(C(C)C)no1)C N1(C(c2ccc(C#C)o2)=O)CC(NC(=O)C(=O)NCCC(N)=O)CCC1C N1(C(CCN(C)CC)=O)CC(CNC(=O)C(c2ccccc2OC)O)CC1C c1ccc(F)c(C)c1.C1(C(N2CC(C(C(=O)N)OC)C2)=O)CC2(C1)CC(O)C2 Cc1[nH]nc(C(=O)NC(C2CC(NC(C3CC(=C4CCC4)C3)=O)C2)C)c1Cl Cc1cc(CN=C(NC2CCCCC2)NC2CCC3CCOC23)cnc1C c1(C(=O)NCCOC2CCN(C(C(C)c3cc[nH]n3)=O)C2)cccc(O)n1 c1(CCC(=O)N)cncc(C)c1.C1CCN(C(=O)CC2CC(C)(C)C2)C1.CCC N1(C(C(C(C)C)C)=O)CCC2(CCCN(C(c3ccc(S(N)(=O)=O)cc3)=O)C2)C1 CC1CN(C(C23CSCC2C3)=O)CCN1C(=O)COCc1nc[nH]n1 C12(NC(c3ncncc3Cl)=O)CC1CN(C(=O)C=CC(F)(F)F)C2 N1(C(C2(C)CC(=C)C2)=O)CCC2(CC1)CCN(C(=O)C(CO)N(C)C)CC2C N1(CC2(NC(CC3CC(=C)C3)=O)CC2)CCN(C(=O)CC2CCC2)CC1.O C12(CC)CC(C(N3CC(O)(C)C3)=O)(CO1)C2.c1(C=O)cnc(C2CC2)s1 C1(NC(C2C(c3n(C)ccn3)OCC2)=O)C=CCN(C(C2(C)CCOC2)=O)C1 C(=O)(C(C1CC1)C1CC1)NCC1C(NC(COC)=O)C1 Cc1nc(NC2CN(C(=O)C(O)CC(C)(C)C)CC2(C)C)ncc1[N+](=O)[O-] CC(O)C(C(=O)N1CCCC1C(C)(C)C(=O)NC(c1ccc(F)cn1)C)N(C)C N1(C(CC(C)(C)N(C)C(c2cnn3c2OCC3)=O)=O)CC(=O)NC(C)(C)C1 c1(NC(C(N2C(COC)CC(O)C2)c2sncc2C)=O)ccc2c(c1)OCO2 N1(C(c2nn(CC)c(C)c2)=O)CCN(c2nc(C(C)C)cc(C)n2)C(C)C1 N1(C(=O)NC2(C)C(OC(C)(C)C)CCC2)CCCC12CCC(F)(F)CC2 c1(CC(=O)N(CC)CC)ccncc1.C1CCCO1.CC(C)NC(=O)CO Cc1nccc(C(=O)NCC2CN(C(=O)C(C)(C)c3cc[nH]n3)CCN2C)c1C C(C(C)C(F)C(=O)NCC1(CC)CCCO1)NC(C(C=C)C)=O C(C(=O)C1CCOc2ccccc21)N1CC(=O)N(CCC23COC(C2)C3)C(=O)C1 CCCC(CCCNC(c1cncc(C)c1)=O)NC(=O)C(c1cccc(Cl)c1)O C12(NC(c3c(CC)onc3)=O)CC(C)(C1)OC21CN(C(C2CCCCO2)=O)C1 C1(NC)CCN(C(c2cccc(NCC(=O)O)c2)=O)CC1 Cc1cn2nc(C(=O)NC(c3cccnc3)CCN(C)C)cc(C)c2n1 c1(OC)ccc2c(c1)N(C(C(=O)Nc1ccccc1Cl)c1nc[nH]n1)CCO2 c1(C(N2CCC(N)C2)=O)ccc2cc(C(=O)O)oc2c1 C1(NC(c2nn(C)c(Cl)c2)=O)CC2CCC(C1)N2C(C1CC2CCC1CC2)=O CC1(NC(=O)NCC2(C3CCCCC3)CC2)COC(C)(C)OC1 CS(=O)CCC(=O)NCC1(NC(c2nccnc2N)=O)CCOC1 c1(C(=O)NCCCNC(C2(CC#C)CCCOC2)=O)ccnc(Cl)c1OC N1(C(C2C(C)(C)C2(F)F)=O)CC=C(CC)CC1.C1(c2cc[nH]n2)(C(=O)N)CCC1 C1(NC(c2[nH]cc(C)c2C)=O)CCN(c2ncc(I)cn2)CC1F C#CCCCC(C)C(=O)NC1C(C(N2CC(C)(N(C)C)C2)=O)C1(C)C C1(c2ccccc2)(C(=O)N(c2ccccc2)CC2CCCO2)CCCCO1 c1(NC(C)CC2CC2)ccc(S(=O)(=O)N2CCc3cnccc3C2)cn1 C12(C(=O)NC3CCN(C)CC3)COC(C1)C(NC(C13CCN(CC1)C3)=O)C2 C1(NC(CSCc2cccc(C)c2)=O)CC(C)CN(C(=O)CCC2CC2)C1 Cc1noc(C)c1CC(=O)NCC(C)COC1CCC(=O)NC1 N1(C(CC(COC)C)=O)CCC(O)(CNC(C2CC23CCOC3)=O)CC1 C(CC(C(=O)NOCC(F)F)NC(=O)C=C1CCOCC1)=CC n1(CC)nnc2c(NC3(C4CCN(C(=O)C(C)(O)C5CC5)CC4)CC3)ncnc12 C(CCCC(C)(F)F)NC(C1OCCN(C(C(C)n2cccn2)=O)C1)=O C1(CCNC(C(C2(O)CN(C(CCc3n(C)cnn3)=O)C2)F)=O)CCC(C)(C)C1 C(=O)(C1=CCS(=O)(=O)C1)NCCC.c1(C=O)cccc(F)c1C(F)(F)F c1(CNC(CC2(CSC)CC2)=O)cnn2c1CN(C(C1CC1C)=O)CC2 [N-]=[N+]=NCCCCC(=O)NC(C(=O)NCCCC1CC1)C1CCOC1 S(=O)(=O)(c1nc(N2CCC(c3ccno3)CC2)ccc1Br)NC(C)CF C1(NC(c2ccsn2)=O)CCC2(CC1)CCN(C(c1cc3ncccc3s1)=O)C2 c1(C(=O)NC2C(OC)CN(C(C3CSCN3C(C)=O)=O)C2)cn(C)ccc1=O S(=O)(=O)(c1ccc(F)c(Cl)c1)N1CC2CN(C(c3ccncn3)=O)CC21 CC1CCC(=CC(N2CCCC(C(C)(C)C(=O)NC(C)CCCCO)C2)=O)CC1 C1(NC(c2ccc3ncnn3c2)=O)CCCC12CCN(C(C1CC(Cl)(Cl)C1)=O)C2 N1(C(C2N(C(CC=C)=O)CSC2)=O)CC(C2CC2(F)F)C1 CC(CNC(=O)C(C)C1CCOC1)CC1CCC1.C12(CC1)C(=O)N2 CC(C)C(C(=O)N(C)C)NC(=O)CC1CCCO1.C12(N)CC(C=O)(C1)C2 c1(OC)ccc(F)cc1CN1CCCC(NC(C2CCN(C(C)C)CC2)=O)C1 N12CCN(CC1)C1CN(C1)C(=O)C1C(=C)C1C2=O.C1(C(=O)O)CCN(C)CC1 CCC(C)(CC(=O)OC)NC(=O)COCc1ccc(F)cc1 N1(CC(=O)N(CC)C)C(C)CCC1C.C1(C(=O)OCC)CC1CC(=O)N Cc1ccccc1OC(C)C(N1CCN(Cc2sc(Br)cc2C(=O)O)CC1)=O C1(CNC(CN(C(COC)=O)C)=O)CC12CCN(C(C1CCCN1N=O)=O)CC2 Cc1cccc(CC(=O)NCC#CCNC(c2n[nH]cc2-c2cnn(C)c2)=O)c1 C(N=c1[nH]c2cc(C(=O)O)ccc2o1)c1c(NC(C)=O)ccc(OC)n1 c1(CC(=O)NC)ccccc1Cl.c1(CCC)nc(C(=O)NCC2CC2)cs1.C c1(CC(=O)NC2C=CCN(C(c3nc(CCC)oc3)=O)C2)ccc(F)c(C)c1 c1(Nc2cc(OCC)c(C)cc2)ncnc2c1ncn2C1C(=O)OCC1CO c1(C(=O)NCC(C(=O)OC)OC)n[nH]c2c(C)cccc12 C=CCCCC(=O)NCC(C)CNC(=O)CCc1ccc(F)cc1 CN1CCC(C(=O)NC2CC2NC(C2CCCCS2)=O)CC1 c1(OC)cc(C(=O)NC2CCC(N(C)C(c3cncn3C)=O)CC2)c(N)c(C)c1 N1(C(=O)Cn2ncnn2)CCCC(C2CCN(C(=O)C(F)(F)C(F)(F)F)CC2)C1 c1(C(=O)NC2CCCCN(C(c3c(CC)nn[nH]3)=O)C2)cccc2c1CCN2 Cc1nn(C)c2c(NCC(Cl)(Cl)Cl)nc(=NC(CC(N)=O)C3CCCCC3)[nH]c12 C(CC(=O)N1CCC1CNC(C1CC(C)(C)C1)=O)(C(F)(F)F)OC C1(CNC(=O)Cc2csc(-c3ccccc3)n2)CCCCCN1C(=O)CO CC1CN(C(C23CCC(CC2)CO3)=O)CCN1C(c1cc(Cl)c(Cl)s1)=O N1(C(c2c(NC)cccc2)=O)CCC(O)C(NC(=O)CC(C)c2ccccc2)C1 C1(CCNC(CC2CC(OCC)C2)=O)CCN(C(c2cc(Br)co2)=O)C1 C1(F)(CNC(C2CCSCC2)=O)COCCN(C(C2CC2C2CCC2)=O)C1 c1(CCC)nnc(S)n1CC(N1CCC(N(C(=O)C(C)N(C)C)C)C1)=O C(=O)(C(C)(C)C1=CCN(C(=O)C2=C(Cl)CCOC2)C1)N(C)CC1CCCOC1 N1(C(C(C)Sc2ncccn2)=O)CCC(NC(=O)CCC[N+](=O)[O-])C(F)C1 c1(OC)nc(C(=O)NCC(N2CCN(C(=O)C(C)C(C)C)CC2)C(F)F)sc1C C12(NC(c3ccc(CC)o3)=O)CCCC1N(C(=O)CC1CCC(C)(C)O1)CCC2 c1(N2C(C)C(C)N(C(=O)OC(C)(C)C)CC2)cc2ccc(Br)nc2[nH]1 Cc1cc(F)cnc1C(=O)NCCC(C)N(C)C(c1cc(N)ccc1F)=O Cc1ccc(S(=O)(=O)n2cccc2CN2CCC(O)C2)cc1.C1(O)(C=O)CC1.N C1(C(N(C2CCN(C(=O)CCn3ccnc3C)C2)CCC)=O)CC2(CCCO2)C1 c1(C(=O)NCC(C)(C2CC2)NC(c2cnc3n2CCS3)=O)nc2cccnc2s1 N1(C(c2c(SC)n(C)nc2)=O)CCc2sc(C)nc2C1.C(=O)(C(=O)C(C)(C)C)N CCS(=O)(=O)CC(=O)NC(Cc1cn(C2CCN(C)C2=O)nn1)C(=O)OC C1(NC(c2cc(OC)ns2)=O)CC(C(F)(F)F)C1.C(=O)C=C1CCC1 CN1CCC2C1CCCN2C(=O)N(c1cccc(C#N)c1)Cc1ccccc1 C(=O)(C(C(C)(C)C)NC(=O)Cn1ccnn1)N(CC(C)OC)C CCCCC(C)(F)C(=O)NC1CCCCCN(C(C2CCN(C(C)=O)CC2)=O)C1 c1(CC)onc(C(=O)NC2CC(NC(c3ccncc3Cl)=O)C2)c1C c1(C(N(CCCNC(=O)C(C)OCCC(C)C)CC)=O)cc2ccoc2cc1F C1(C2CN(C(c3cn(CC(F)(F)F)nc3C)=O)C2)CC1.CC(C(F)F)=CC=O.N C=CCCCCCC(C)(c1nnnn1C(C)(C)CC)NCC1(CO)CC(C)C1 C=CCCC(C)(c1nnnn1-c1ccccc1C)NC(CCC)C(=O)N(C)C C#Cc1ccc(C(=O)NCc2nocc2C(N2CC(S(C)(=O)=O)C2)=O)cc1 C1(CC=C)(C(=O)NC(C2CCCN2C(=O)CC=C(C)C)C)CCOCC1 c1(C(N2CCC(NC(C(CCCC#C)C)=O)C2)=O)cc(F)cc2nc[nH]c12 CS(=O)(=O)C1(CNC(=O)N)CCC1.N1(c2ccccn2)CCS(=O)(=O)CC1 C(=O)(C1CCCc2ccccc21)NC1C(NC(c2cccc(N)n2)=O)C1 c1(C(=O)N)cc2ccc(Cl)nc2s1.C1(CNC(CCOC(C)=O)=O)CCCCC1 Cc1ccc(C(F)(F)C(=O)N2CCCC2CNC(=O)C(F)(F)C2CCCC2)cc1 CC12CN(C(=O)C(F)n3ccnc3)C(C(=O)NCc3ncsn3)(C1)C2 C1(CNC(c2nccc(SC)n2)=O)CN(C(C2CC(N(C)C)C2)=O)CCC1C N1(C(c2ncc(OC)nc2)=O)CCC2(CCOCC2)C(NC(=O)C(O)C(F)F)C1 C1=C(CCNCc2cscc2Br)c2ccccc2OC1 c1(C(=O)NCC(C2CCOCC2)N(C2CCCCC2)C)cccc2c1OCO2 Cc1cc(C(=O)NC(C)CCCNC(=O)Cc2sccc2C)n(C2CCC2)n1 C(=O)(CCCCC(C)(C)C)N1CCC(N(C(=O)C2=C(C)OCCS2)CC#C)C1 CC1(c2ccccc2)CCCCN1CCCc1ccccc1.c1(C=O)ccccc1Cl C(=O)(C1=NOC(CNC(c2ccncc2)=O)C1)NCCc1cc(C)ncc1 c1(OC)ccc(C(N2CCCCC(NC(=O)CCc3ccon3)C2)=O)c(F)c1F C(=O)C1=CC2(CCOC2)C1.N1(C(C)=O)CCC(CNC(c2conc2)=O)C1.C C1(CC=C)(NC(=O)CCC2CC2)CCCN(C(=O)CC(C)N(C)C)C1 c1(CC(=O)NC2(CN(C(C(=O)NCC)=O)C)CC2)cnc(C)o1 C1(C)(OC)CCN(C(=O)CCCN(C(=O)C=Cc2ccco2)C)CC1 c1(C(N2CCCC(NC(C3(F)CCC3)=O)C2)=O)cc2c([nH]1)CCOC2 S(=O)(=O)(c1ccsc1C(=O)NCCC(C)NC(=O)CSC(F)F)NC C1(CNC(C2C(=C)C2)=O)CC2(CCC2)CN1C(=O)Cc1csnn1 C1(CC(=O)NC(CC#C)C)CCN(C(c2nn(CC)nc2C)=O)C1(C)C c1(CNC(C2CCN2C2CC2)=O)cc2n(n1)CCCO2 C(=O)(CCS(C)(=O)=O)NCC1(COC)CCN(C(=O)CC(C)C)C1 C1(CNC(COCC#C)=O)(C)CC(F)(F)C1.C1(C=O)(CCC)CCC1 N1(C(Cc2c(C)cccn2)=O)CCC(O)C1.C1(C)(C(NC)=O)C(C)(C)C1(C)C.C c1(C(N2CC(NC(Cn3c(C)nnn3)=O)C(CO)CC2)=O)cc(Cl)c(N)c(Cl)c1 C(C(C)(O)C(F)(F)F)NC(CCOCCCNC(c1c(C)cncn1)=O)=O N#Cc1ccnc(N2CC(C(N3CCC(O)C3)=O)(Cc3ccc(F)cc3)C2)n1 N1(C(C(CCC)C)=O)CCOCC12COCCN(C(c1cnoc1)=O)C2 c1ccccc1.CC(C=O)n1cncn1.C(=O)(C(C)NCC(F)(F)F)NC1CC1 C(C)(CCC(=O)NC(C(=O)NCC1(O)CC1)C1CCCC1)OC C1(NC(C(CCNC(=O)Cc2ccsc2C)OC)=O)CC2(C1)CC21CCC1 Cc1sccc1C(=O)N(C1CCN(C(c2ccnn2CCF)=O)C1)C C1(NC(c2c(Cl)cn(CC)n2)=O)CCC2CC1CN2C(=O)CN1C(C)CCC1C CC1(C)CC(NC(c2cocn2)=O)CCN(Cc2cc(F)cc(Br)c2)C1 C(CC(C(=O)NC1CN(C(=O)CCC(=O)N(C)C(C)C)CC1C)NC=O)SC N1(C(c2ccc(C(C)(C)C)[nH]2)=O)CCN(CCS(N)(=O)=O)CC1 N1(C(c2c(OC)ccs2)=O)CCN(C(=O)C=C=C(C)C)CC12CCC2 C1(C(=O)NCC=CCNC(=O)CCC2CC2)COCCC1c1ccccc1 C1(CC(=O)NC2COC(C3CC3)C2)(OC)CN(C(=O)C=C2CCC2)C1 C1(C(N(CCN(C)C)CCO)=O)N(C(c2cccc(CO)c2)=O)CC12CCCC2 c1(NC(CCCC)CCC)cc(C)c(S(=O)(=O)NC2CN(CC)C2)cn1 NC1(CNC(=O)COc2cncc(Br)c2)CCOCC1 N1(C(=O)C(O)Cc2cnc[nH]2)CC2(CCN(C(C3CCC4CC3CO4)=O)CC2)C1 Cc1cccc(C(=O)NC2CCN(C(c3scnc3C(C)C)=O)C2)c1F C1(NCC2CC(S(C)(=O)=O)C2)CCCC2(C1)OCCO2 N1(C(c2ncc(Cl)cc2Br)C(=O)NCCCSC)C2CCC1CC(O)C2 CC1(C(N2CCN(C3CCN(C(C4(C)CC4F)=O)CC3)CC2)=O)CCSCC1 C1(CNC(c2c(SC)csc2)=O)CN(C(C2OCC3CCCC23)=O)CC1(F)F c1(CCC(=O)NCC(CNC(C(=O)N(C)C)=O)O)c(Br)cncc1Br c1(COCC(C2CC2)(OCC)OC)ccnc2cc(OC)ccc12 c1(C(N2CCCC(NS(=O)(=O)C3CC3)C2)=O)cc(C(F)(F)F)cc(Br)c1 C(C)(C)(C(=O)NOC(CC(C)C)C(=O)NC1(c2cc[nH]n2)CC1)OCCC c1(CC)onc(C)c1C(=O)N(C(C)C(=O)NCC)C1CC1.C1CC1.C C1(CC)CN(C(=O)CN2CCN(C(c3nccnc3C)=O)CC2)CC(=O)N1 C1(C(N2CCN(CC)CC2C)=O)CC2CC1CN(C(=O)C(CSC)OC)C2 c1(C(=O)NC2C3CN(C(c4ncc(CC)cn4)=O)CC32)ccc2c(c1)ncn2C C1(C=O)CCC2CCC(=O)N12.n1(CCNC(c2cnc[nH]2)=O)cc(C)nn1.N N1(C(c2nc(COC)oc2)=O)CCCC12CCCC2.C(=O)C(F)(F)C(C)(C)O.N N1(C(c2c(C)oc(C(C)C)c2)=O)CC(NC(=O)NCCCl)C2(CC2)C1 C1(CC)CCC(CN(C(=O)C(C)N(C(C2CCCC(O)C2)=O)CC)C)CC1 N1(C(c2ccccc2)=O)CCC(C2CCN(c3nc(O)c4nc[nH]c4n3)C2)CC1 CCCC(C)CC(=O)NC(C1(O)CN(C(=O)CSc2cccc(F)c2)C1)C C(c1cn(C)cn1)=CC(=O)N(CC(C)NC(=O)C(O)C1CC1)CC CC1(C)CC(NC(c2cc(Br)ccn2)=O)CN(C(C2CC3CC3C2)=O)C1 C1(CNC(=O)C#CC2CC2)CN(C(c2occc2Cl)=O)CC12CC2 CCCC(CC(=O)NCCC12CC(CO1)C2)NC(=O)CC1COCCO1 C(C(F)(C(=O)N1CC=CC1CF)C(C)C)NC(c1cn(CC)nn1)=O c1(C(N(CC(C)O)CCNC(CCCC#CC)=O)=O)cc2sccc2cn1 N1(C(C2C(OC)CCC2)=O)CCN(C)C(CNC(=O)C2=CCN(C)C2)C1 C1(NC(C2N(C)CCCC2)=O)CC(F)CN(C(c2coc(CC3CC3)n2)=O)C1 C(c1cccc(Cl)c1Cl)=CC(=O)N(C(CCNC(C(C1CC1)SC)=O)C)C N1(C(c2cnn(C(C)C)c2C2CC2)=O)CCCC(CNC(c2ccon2)=O)CC1 C1(CCNC(Cc2c(C)nc(S)s2)=O)CCN(C(c2nnn(C)c2N)=O)C(C)C1 c1(C(N(CCNC(C2CCCC2O)=O)C)=O)cc2n(n1)CCCC2O.C1CC1 c1(OCC)cncc(CNC(c2cn(C)nn2)c2nnnn2CCOC)c1 N1(C(C(C)(C)CC(F)(F)F)=O)CCC2(C1)CN(C(=O)CCC1CC1(C)C)CCO2 c1(C(C)=O)ccc(Br)c(NC(C2CN(Cc3ccc(I)o3)C2)=O)c1 CCCCC(O)C(=O)NC1CC(O)CN(C(=O)CN(C)C2CC2)C1 c1(C(N2CC(NC(C3(COC)CCCC3)=O)C(C)C2)=O)ccc(=N)[nH]c1Cl C(=O)(C(CCCC)C(C)C)NC(C(=O)N1C(C#C)CC1)CCC1CC1 c1(C(N2CC(C)C(CNC(=O)C(C)S(C)(=O)=O)C2)=O)cnn2ccnc(N)c12 c1(C(N(CCNC(C(CCC)O)=O)C)=O)cnc(O)cc1O c1(C2C(C=O)C2)ccccc1Cl.C1(C(=O)OCC)(C(=O)NCC)CCC1 C(=O)(C1=CS(=O)(=O)CCC1)N1CC2C(NC(c3ncc(C)cc3F)=O)(CCC2)C1 CC1C(C(=O)NC)C(O)C(=O)N1C.c1(C(N2CCC2)=O)cc([N+](=O)[O-])cn1C N1(C(c2c(OCC)nccc2)=O)CCCC(C)C1.C1(C(=O)N)(C(C)C)CCC1 C12(C(N(CCC)C)=O)CCN(CC1)S(=O)(=O)C2.Cc1n[nH]c(C)c1CC(=O)N N1(C(CSC)=O)CCOC(C(=O)NC(CO)(CO)CO)C1 C(C(O)C(=O)NC(Cn1cccn1)C(=O)NC(c1cn[nH]c1)C)SC C1(CCC=C)CCCN1C(c1nc(Cl)cs1)C(=O)NC(C)(C)C C1(C(N2CCCC(CN(C(c3c(C)n(C)cc3)=O)C)C2)=O)CCC(C)(C)OC1 N1(C(C)=O)CCCCC1CCN(C)C(c1cn(-c2cccc(Br)c2)nc1C)=O CN1CCN(C(=O)CC2COCCO2)CC1CNC(c1cc(Cl)ccc1Cl)=O Cc1cccc(CO)c1NC(c1ccc(Cl)c(Cl)c1)=O.c1(OCC)ccc(F)cc1 C(=O)(C(CC)(CO)OC)NC(CC)CC(=O)NCc1[nH]nnc1C c1(C(=O)NC(CC)C)cn(CCNC(=O)C(C)NC(=O)C(C)C)nn1.O C(=O)(C(F)(F)C(F)(F)F)Nc1cc(OC(C)C2CC2)ncc1 C12(CCNC(C3CC(=C)C3)=O)CCC1CN(C(c1cccc(=S)n1O)=O)C2 C1(C(N(C2CC(C(=O)NC3CC4(CC4)C3)C2)C)=O)C2CCCCCC12 c1(NC(C(C)NC(CC=C)C#N)=O)cc(C)cc(C)c1 C1(NC(C(C)c2ccco2)=O)CCOCC1NC(c1c(Cl)cnn1C)=O C1(OC)CN(C(=O)CCC2CC2(C)C)CCC1NC(=O)CN(C1CCCC1)C C1(CNC(Cc2n(C)cnc2)=O)CN(C(=O)CNC(C2CCC2)=O)CCCO1 C(COC)(CC(=O)NCCC1(CO)CC1)NC(C(C)OCC=C)=O C1(C(=O)Nc2cccc(-c3n(C)c(O)nn3)c2)CC(=O)c2ccccc2C1 c1(C(=O)NC(C(C)NC(=O)CCSC(F)(F)F)CO)cc(N(C)C)ccc1N c1(C(N2CCC(C(C)NC(C3C(=C)CC3)=O)CC2)=O)c(F)ccc(F)c1Cl c1(C(N2C(C)CC(NC(=O)C(C)(C)N(C)C)C2)=O)cc(O)ccc1OC(F)F N1(C(C(C)C#N)=O)CC2CCC1C(NC(=O)Cc1ccc(F)c(Br)c1)C2 C(=O)(C(C)C(C)(C)C)N(C(C)C(N)=O)C1CC1.c1(C=O)ncc(F)cc1N.N CC1(C)CCN(CC(=O)NCC(C2CCCC2)NC(C2CCCSC2)=O)C1 N1(C(Cc2c(C)nn(C)c2Cl)=O)CC2CC(NC(C3CC34CC4)=O)CC(C2)C1 C1(CCC(=O)NCCCS(C)=O)CCCN(C(=O)CN2CCC(=O)CC2)C1 C(=O)(CC(C=C)CCC)N(C1CCN(C(CCCC#C)=O)CC1)C c1(C(N(CC(C)(C)C)CC)=O)ccc(F)cc1.CCC=O.C(=O)(C1CC1)N c1(C(N2C3C(N(C(CC(=O)NCC)=O)C)CC(C3)C2)=O)cc(C)c(C)cc1C c1(C(N(CC(C)NC(c2ccccc2)=O)CC)=O)ccc2c(n1)OCC(=O)N2 C(=O)(C(C)(C)COC(C)C)N(CCCC)C c1(COC(c2ccc(-n3ccnc3)cn2)=O)n[nH]c2cc(Br)ccc12 Cc1ccc2cc(C(=O)NC)[nH]c2c1.C1C2CN(C(=O)CC3CNC(=O)C3)CC12 N1(S(=O)(=O)CCCCl)CCC2CN(Cc3csc4ccccc34)CC12 O=C1CC2CCCC2(C(=O)NC2CC(CNC(=O)COCC(F)F)C2)C1 C1(CC#C)(C(=O)NCC=CCS)CCN(C(=O)Cc2c(C)noc2C)C1 C1(NC(C(C=C)OC)=O)CN(C(=O)Cn2cc([N+](=O)[O-])cn2)CC1N=[N+]=[N-] N1(C(C(CC)(CC)CO)=O)CC2(C1)CN(C(=O)C(O)C(C)C)CC2CO C(=O)C(C=O)C(C)C.C1(CC(N2CCC2)=O)(C(F)(F)F)CC(=O)N(O)C1 N#Cc1cc(Cl)ccc1NC(C1C2CC1N(C(c1csc(Br)c1)=O)C2)=O C1(C)(C(N2CCC2)=O)CC2(CCC2)C1.C1(CCOC)(C(=O)NC)CCC1 C(=O)(C(CC(F)F)N(C)C(c1nccn1CC)=O)N1CC(CC#C)OCC1 Cc1ccc(C(N2CCC(NC(c3cccnc3C3CC3)=O)C(O)C2)=O)c(C)n1 N1(C(C(CC)C)=O)CCCC(C)(CNC(c2sc(N(C)C)nc2C)=O)C1 C(CO)(CCCCNC(=O)CN1CCSCC1)NC(Cn1c(C)ncc1)=O N1(C(=O)Nc2cnc(C)c(C3CC3)c2)CCCS(=O)(=O)CC1C1CC1 c1(CN2CCC(C#N)(NS(=O)(=O)c3cccnc3)C2)cc(F)ccc1[N+](=O)[O-] O(NC(=O)N=c1[nH]n(C)cc1CC)CC#C c1(CC(=O)OCC)ccccc1-n1cc(C2(C)CCCN2C)nn1 C(N=c1ccc(S(=O)(=O)N(C)C)c[nH]1)C1CN(C(C2(OC)CCSC2)=O)CC1C C12(NC(CCN(C)CC)=O)CCC(C1)N(C(c1cn(C(C)(C)C)nn1)=O)C2 C(c1ccc(OC)c(Cl)c1)=CC(=O)NC(CCCC)CNC(=O)CCC(C)C Cc1cc(N)cc(C(=O)NCCN(C)C(c2cc(Cl)c(F)c(Cl)c2)=O)c1F C1(NC(Cc2cnc(CC)s2)=O)CCCN(C(=O)CCN2CCOC2=O)C1 c1(C(N2CC3C(CNC(C(CC=C)(C)C)=O)(C3)C2)=O)ncc2n1CCCC2 c1(C(C)NC(CCC(C)C)c2n(-c3c(C)cccc3)nnn2)ccc(F)c(C)c1 C1(C(=O)NCC(O)CC(=O)NCC(c2ncc[nH]2)C)(OC)CCOCC1 C(=O)(C1CCc2ccccc21)NCC(CCCC)NC(c1cnc(N(C)C)s1)=O c1(C(N2CC3(CN(C(C4(CC)CC4)=O)C3)C2)=O)cccc2c1OC(C)C2 C1(C(=O)NCC(CCOC)NC(=O)Cn2ccc(C)c2)CCC(=O)N(C)C1 C(=O)(CC(=O)N(CC(C)N(C(=O)Cc1cnn(C(F)F)c1)C)C)OC C1(C(N2CC(CCn3cc(C(C)(C)C4CC4)nn3)C2)=O)(OC)CCCCCCC1 C#CC1(CNC(C2CC(C)CN(C(c3csc(=N)[nH]3)=O)C2)=O)CCOCC1 n1(CCSC)nnnc1C(C1(C)CCCS1)NCCCCF c1(CC(=O)N(CCN(C(=O)C(C)C2CCCC2)C(C)C)C)csnn1 CC(CC(=O)NCCN(C(=O)C(=O)N(C)C)C1CC1)C1CC1.C1CN1 c1(N2CCC(CCOC)C2)nc2c(c(=NCCc3ccc(Cl)c(Cl)c3)[nH]1)CCC2 C1(N(C(c2c(C)nc(COC)s2)=O)C)CCN(C(=O)C2=CCOCC2)CC12CC2 N1(C(C=COCC)=O)CC2(CCCN(C(c3c(C)ccc(C)c3C)=O)C2)C1 C#CC1(C(=O)NCC2(C)CCCN(C(=O)C(C#N)C(C)C)C2)CCOCC1 N1(C(CC2C(C(=O)OC)CC2)=O)CC(NC(c2ccoc2Cl)=O)C(N=[N+]=[N-])C1 N1(C(CC(C=C)(C)C)=O)CCN(C(C2CCC3C(C2)C3(F)F)=O)C2COCC12 Cc1cc(C(N2CC(NC(=O)Cc3ccc(Br)cn3)C2)=O)c([N+](=O)[O-])cc1F c1(C(C(=O)NCCCN(CC(C2CCC2)OC)C)C)cnn(C)c1 N(C(=NCCc1ccccc1F)NCc1ccc(Cl)o1)CC1N(CC)CCC1 C1(CNC(C(F)=CCC)=O)CC(C)CN(C(C23CCC(C2)C3)=O)C1 C1(CNC(C(CC=C)C)=O)CC2(CCN(C(c3cc(C)c(C)[nH]3)=O)C2)CO1 C1(N(C)C(c2cocn2)=O)CC2CC1N(C(c1conc1-c1ccccc1)=O)C2 c1(C(=O)NCC2N(C(C3OCC(C)C3)=O)CCCC2)cc2c(O)ncnc2cn1 C1(C)(CNC(=O)NC(C2CC2(C)C)CC)CCCC(F)(F)C1 c1(OCC)ccc2nc(N3CCCC4(NC(=O)C5=NNC(=O)C5)CC4C3)sc2c1 N1(C(c2c(C)cc(F)cn2)=O)CC2CCCC(C1)N2C(C1CC1C#N)=O N1(C(CCN(CCC)C)=O)CCCN(C(=O)COc2cc(C)ccc2F)CCC1 N1(C(c2cc(C)cc(C)c2)=O)CCC2CCCC12C(=O)N(C1CCC=CCC1)CC CC1C(=O)N(C)CCN1C(c1ccc(CNC(C2CC2(F)F)=O)cc1)=O C1(C(N2CCC(C)(NC(=O)C3=CCC3)CC2)=O)CC2CCCC(C1)C2 C1(c2n(C(C(=O)OCC)C)nnn2)(NCCCCC(C)(C)C)CCOC(CC)C1 c1(NC(C2(O)CC2)=O)cnn(CCO)c1C1CC1 c1(OC)ccc(C(C2CC2)SCC(=O)Nc2ccc(Br)cn2)cc1 N1(C(C2(C#C)CCCC2)=O)CCC(CO)C(NC(c2cncc(OC)c2C)=O)C1 C1(CN(C)C(C2COCCN2C)=O)CN(C(c2ccoc2C(F)(F)F)=O)CCO1 C1(NC(C2CCN2C(=O)C(F)CC2CCOC2)=O)CCN(c2ccccc2)CC1 C1(CCNC(CC(=C)C)=O)CCCN(C(=O)CC2C(=O)ON=C2C)C1 C1(C(N2CC(=CCC)C2)=O)CN(C(=O)CC2=CCCC2)CCN1C Cc1cc(C(=O)NCc2csc(C(N3CCCC3CCO)=O)c2)nc(C)c1 Cc1cccc(C(CNC(c2csnc2Cl)=O)NC(=O)C(F)=C2CCC2)c1 CC1CN(C(=O)CC(C)(C)O)CC1CNC(=O)CC(=O)Nc1nccs1 C1(NC(c2ccc(CC)cc2)=O)CC12CCN(C(=O)C(C(C)C)SC)CC2 CC(C(=O)N(C)CC1(CNC(C2CCCS2)=O)CC1)C1CCC1 c1(C(c2nnnn2CCCF)NC(CC)C2CC2)cn(C)nc1C S(=O)(=O)(c1ccc(-c2ccc(C#N)s2)s1)N(C1CS(=O)(=O)CC1O)CC(C)C c1(CC)c(C(=O)NCC2(CNC(c3ncsc3C)=O)CCCC2)cccc1C C1(NC(COC)=O)CN(C(=O)CCCc2ccc(CC(C)C)cc2)CC1OC Cc1cn2c(C(N3CCCCCC(NC(C4C5CCCOC45)=O)C3)=O)cnc2s1 N1(C(CC2CC(CNC(c3c(N)c(F)ccc3)=O)C2)=O)CC2CCC(CO)(C2)C1 CCC(CC)(CC)C(=O)N1CC(O)(C(C)NC(c2cnc(S)[nH]2)=O)C1 C(=O)(CCCCCC(C)O)NC(CC)(CC)CCNC(=O)C(n1cc(C)cn1)C c1(C(N2CCOCCC2)=O)c(F)ccc(C)c1N.C(C(=O)N)(C1CC1)OCC.C c1(C(=O)NCC(C)OC)ccc([N+](=O)[O-])s1.c1(C(C(=O)N)C)ccccc1C c1(C(N2CCC(CN(C(C(C(CC)(C)C)O)=O)C)C2)=O)cccc2oc(O)nc12 C(=O)(C(O)C(C)CC)N1CCC(N(CCCC)C(c2nc(Cl)sc2C)=O)CC1 CC1C(N(C)CCO)CCN1C(=O)CCC1(C)CN(C(=O)CCCC2CC2)C1 N1(C(Cn2ccc(C)n2)=O)CC2CN(C(=O)Cc3[nH]cnc3C)CC2(C)C1 N1(C(C(CCC)C)=O)CC2CCCC1C2CNC(=O)CC=CC(C)(C)C C12CCC(CO1)C2.c1(C(=O)NC)nc(C(F)(F)F)ccc1F.C(=O)C1CC1 C1(CN(C(=O)CCC2CCC2)C)CN(C(=O)CS(=O)(=O)N2CCCCC2)CCO1 N1(C(c2ccn(CC)n2)=O)CCCC(NC(c2cnc(S)nc2)=O)C(F)C1 C1(NC(=O)CCn2ccnn2)CN(C(C2CC3CCC3C2)=O)CCC1O Cc1ccc(CC(N2CCCC2C(N2CCC(C(C)(C)O)C2)=O)=O)cc1[N+](=O)[O-] c1(NC(c2ccc(CC)cc2C(F)(F)F)=O)cc(F)cc(F)c1O N1(C(C2N(C(C3C=C(C)CS3)=O)CCSC2)=O)CCCOC(C)C1 c1(C(c2nnnn2-c2ccc(F)cc2)NCC(=C)F)c(F)cccc1Br N1(C(c2nnn(CC)c2C)=O)CC2(CCCN(C(=O)CC3CCCCCC3)C2)C1 N1(C(C#CC)=O)CC2C(C1C(=O)NCc1ccccc1C(C)(C)C)C2(C)C CC1CN(C(c2coc(C(F)F)n2)=O)CC1NC(c1scnc1C(F)F)=O c1(CCC(=O)NCC(CO)NC(=O)Cc2cnccc2Cl)cc(F)ccc1F C1C2CCC(C2)N1C(c1cc(O)n(C)n1)=O.C1(CC=C)(C(=O)N)CCC1.C c1(C(N2CCC2C(F)F)=O)ccc(O)c([N+](=O)[O-])c1 C1(NC(c2cc(C)n(CC(F)(F)F)n2)=O)CC2CC1N(C(=O)C=O)C2.C(C)C C(=O)CC1=NN(c2ccccc2)C(=O)C1.C(F)(C(=O)NC1CC1C)=C(C)C C1(C)(C(N(CCC)CC)=O)COC(C)(C)CO1.C1(C=O)CC(n2cnnc2)C1 CCC(C)(CO)C(=O)NCC(C)(C)CCNC(C1(c2cccs2)CC1)=O C(=O)(C1=C(Cl)CCCC1)N1C2CC(NC(C3C(C)CCOC3)=O)(C2)C1 c1(C(=O)NCC2CNCC(C)C2)ccc(Cl)c(Br)c1 C1(C(N2CCN(CCN(C(=O)CSc3cccs3)C)CC2)=O)CCCC(=O)N1C FC1(C2CC2)CCN(CC(c2ccncc2)c2cccs2)CC1 c1(NC2CC(CCNC(C3C(=C)CC3)=O)C2)cc(OC)c([N+](=O)[O-])cc1Cl C1(C(N2CC(N3CCN(C(C=CC=O)=O)CC3)C2)=O)CCc2nn(C)cc2C1.C c1(C=O)cccc(S(C)=O)c1.N1(C(COc2cc(C)on2)=O)CC2CC2(C)C1.N CC1NC(=O)CCC1N=c1[nH]c(=NCC23CC(CN2C)C3)c2[nH]ccc2[nH]1 CC1(C)CC(O)CN1C(C1C2CC3C(C2NC(=O)C2=NNC(=O)C2)C13)=O C1(NC(c2ccc(COC)o2)=O)COCCC1.n1(CCC=O)nc(C)cc1C.N CN1CCOC(CN(C(c2cnn(CCCl)c2)C(=O)Nc2ccccc2)C)C1 N1(C(=O)CC2CCC(NC(C34CSCC3C4)=O)C2)CC2COCC(C2)C1 c1(CC(=O)Nc2sc(C)c(C3CC3)n2)c[nH]c2c(Cl)cccc12 c1(OC)cc(Cl)c(Cl)cc1CC(=O)NCC(C)C1CC1.C1(C=O)CCCN1C.N c1(C(N(C)CC2CCN(C(=O)C(C)(C)CC#N)C2)=O)cc2sc(=O)n(C)c2s1 C(c1ccccc1)=CC(=O)NCC(=O)N(CC(C)NC(COC)=O)C CC1CN(C(c2nccn2C)=O)CC(C)N(C(c2ccc(C3CC3)s2)=O)C1 Cc1cnc(C(N2CCC(NC(C3CC(C)(C)CO3)=O)C(O)C2)=O)cc1C N1(C(c2c(C)onc2)=O)CCOC(CNC(=O)CCC(=O)OC(C)(C)C)C1 N(C1CCCc2n[nH]cc21)C(C1(CC=C)CCN(C(=O)C(CO)NC(N)=O)C1)=O c1(OC)ccc(C(=O)NCC2CCN2C(=O)COc2ccccc2)c(F)c1 C(=O)(CC(C)(C)C(F)(F)F)NCC(C)NC(C(CC)N(C)C)=O C1(CNC(CCCSC)=O)(NC(c2ccc(C(F)F)nc2O)=O)CCCCCC1 c1(C(=O)NC2CCC(=C3CCC3)CC2)ccc(=O)n(Cc2cccc(Cl)c2)c1 c1(C(N(C)CC2CN(C(C(C)n3cccn3)=O)C2)=O)cc(-c2cccnc2)on1 C(=O)(CC(CCC)NC(=O)CC1CCCC(=O)C1)NC(C#C)(CO)CO N1(C(C(C)C2CC2)=O)CCCCC1C1CCN(C(c2c[nH]c(=O)cn2)=O)C1 c1(C(=O)NCC(C)(CO)NC(C2COC(C)(C)O2)=O)cc(O)nc2cnccc12 Cc1ncccc1CCC(N1CCCC1C(C)(C)NC(C1CCCCN1C)=O)=O CC(C)C(O)(C(=O)N1CCC(F)(CNC(=O)CCCC(F)(F)F)CC1)C(F)(F)F N1(C(c2ccn(CCOC)n2)=O)CCC2C(C1)CN2C(=O)CCc1ccccc1 N1(C(CCCC=C)=O)CCC(NC(=O)C=Cc2ccn(C)c2)C(CO)C1 C(C)(CC(F)(F)F)NC(C1C(=C)C1)=O.c1(C(=O)N)cnn(C(C)(C)C)c1 c1(CCNC(C2(SC)CN(C(C3CC3)=O)C2)=O)ccc(O)cn1.C1CCC1 Cc1ccc(CCCC(C(=O)NC2CCC2)N2CCCCCC2CCO)cc1C C1(NC(C(C)OCC=C)=O)CN(C(=O)C)CC12CC2.c1cccc(C#N)c1.S N1(C(C(CC=C)(F)F)=O)CCOCC(C)(CNC(C2CCCC(=O)N2C)=O)C1 S(=O)(=O)(c1cn(C)c(=O)n(C)c1=O)NC(c1c(F)cccc1Br)C c1(C(=O)NC2C(C(N(CCCC)CCO)=O)C2)nn(CC)cc1Cl C1(NC(C2(N(C(CCC(C)N(C)C)=O)C)CC2)=O)CCCCCCC1 N1(C(c2ccc(C=C)cc2)=O)CCCN(C(c2cccnc2C2CC2)=O)CC1C Cc1[nH]c(C(=O)NC(C)C(C)C(C)C)c(C)c1[N+](=O)[O-].C(=O)C.C1CCC1.N Cn1cc(C=CC(N2CCN(C(=O)C=Cc3csc(C(F)F)c3)CC2)=O)cn1 C(=O)(CCC(F)(F)C(F)F)N(C)CC1N(C(Cn2c(C)nnn2)=O)CC(F)C1 c1(C(N2C(CC)CCC2)=O)ccc2c(c1)COCC2.C1(C=O)CCS(=O)(=O)C1.N c1(C(C)=O)ccc(C(=O)OCC23CC(NC=O)(C2)C3)cc1.C(C)C.N C1(CCC(=O)N(C2(C(=O)OC)CC2)C)CCN(C(c2ccns2)=O)CC1 C(=O)(C(CCOCCO)NC(=O)CC1COCCOC1)NC1(C)CC(=C)C1 c1(CN2CCCC(NC(=O)C=CC3CCCC3)C2)cc(B(O)O)co1 N1(C(c2cc(Br)c(Cl)s2)C(=O)NCC=C)CCn2c(C(=O)OC)cnc2C1 C12CCCC(CN1C(C1(C3CCCO3)CCC1)=O)C2.Cc1coc(C(=O)NC)c1 C1(C(N(CCCNC(c2cnn(CC(F)(F)F)n2)=O)C)=O)CCOC(=O)CC1 c1(C(=O)NCc2cnc(C(=O)O)cn2)c(F)c(Br)cc(Br)c1F c1(C(=O)NCC(C)(CC)NC(C2CC(=C)C2)=O)cnn2c(=O)cc[nH]c12 C1(CC(=O)NC(C(C)NC(=O)CCc2nncs2)CO)CCC(=O)NC1 CC1CN(C(C2(C(F)(F)F)CCCCC2)=O)CCCN1C(C1CC=CCO1)=O CC1(CNC(=O)Cc2cnc[nH]2)CCC(NC(c2cocn2)=O)C1.C1CC1 C(CO)(C(=O)N1CC(=C(F)CNC(c2cc(Cl)cs2)=O)C1)NC(N)=O C#CCCC(=O)NC(C)CNC(c1csnc1Br)=O C1(C#N)(C=O)CC2CCC1C2.C1(C)(C(N2CCC(CC)C2)=O)CCC(=O)CC1.N C(=O)(CCCCCC#N)N1C2CC(NC(c3n(CC(C)C)ncc3)=O)C(C2)C1 C1(CNC(C2(C)CC(=C)C2)=O)CCN(C(=O)Cc2ccc(O)cc2)CC1(F)F N1(C(C2CC(NC(C3CCCOCC3)=O)C2)=O)CCC(O)(C(F)F)C1 C(=O)(C1CCc2nccn21)NC1(CO)CN(C(C23OCCC(C)(C2)C3)=O)C1 c1(CNCC(O)Cc2ccc(F)cc2)cc(F)cc(F)c1 C1(COC)(NC(=O)C(C)OC)CCCN(C(c2ccc3c(c2)CC3)=O)C1 C(CC)(CCCC(=O)Nc1ccc(C)c(F)c1)NC(CC1CC(CC)C1)=O n1(CC)nc(C(=O)NC2CC3(C2)CC3C(=O)NC2CCCCCC2)c(C)n1 C(=O)(C#CC1CCCCC1)NC1(C(=O)NC(C=C)C)CCCC1 CCC1=NOC(C(=O)NC(C)C(CO)NC(=O)CCn2ccnc2)C1 c1(C(N2CC(O)(C(C)NC(=O)CCCCC3CC3)C2)=O)c(F)cc(F)cc1Cl CCCCC(F)C(=O)N(O)Cc1cn(-c2ccn3ccnc3c2)nn1 C1(CCNC(c2c(COC)ccs2)=O)CSCCN1C(=O)CN1CCCCC1C c1(CC(=O)NC(C2CCCCC2)CNC(C(CC)(C)O)=O)c[nH]c2cnccc12 C1(C(=O)NC2CCN(C(c3c(COC)cc[nH]3)=O)C2C)C2CCC(F)(F)C12 C1(CC)C(C(=O)NCCSC)CCN1C(=O)C=CC.N1CCCNC1=O.C CCCCCCCCCCCCCC(=O)NCC(CO)NC(=O)CCCC(C)=O C(C)(C)(C(O)C(F)F)NC(C(CC)N(C(=O)CC1CCOCC1)C)=O C1(SC(C)C(=O)NC(=O)CNc2ccccc2)CCC(CO)CC1.c1ccccc1 C1(C(N2CC(C#N)(COC)C2)=O)CN(C(C2(C)CCCOC2)=O)CC1(C)C N1(C(c2c(C)cno2)=O)CC(CNC(=O)C(C(C)C)N2CCCCC2)C(O)C1 CC(C)(C)CC(O)C(=O)NC(CCCNCc1ccc(O)cc1)c1ccccc1 c1(CC(=O)N)ccccc1.Cc1ncc(C(=O)NCC2CCCC2)s1.C1CC1 c1(C(=O)NC2(CC)CCOC2)cc(N2CCOC2=O)ccc1F c1(C(N2CCCCC(C(NOCCC=C)=O)C2)=O)ccc2n[nH]cc2c1 N1(C(C)=O)CCN(C(C2(C)CCCO2)=O)C(C)C1.N1(CC(=O)N)CCCNC1=O C1(NC(c2cnn(C(C)C)c2N)=O)CCN(C(C2(C)CCCS2)=O)CCC1CO c1(CC(N2C(CC(=O)N(C)Cc3ccccc3)CCC2)=O)ccc(C#N)cc1 c12ccc(cc1Cl)NC(=O)OCC(O)CNC2.C(C)(C)(C)OCC C1(CNC(c2ccnc(C)n2)=O)CCN(C(C2COCCO2)=O)CC1(F)F N1(C(c2cn(-c3nc(C4CC4)ns3)cn2)=O)CCCC(O)C1 C1(C)(C(=O)NCCC(=O)NC(c2nc[nH]n2)CC)CC2(CCC2)C1 C1CCN(C(C2CC(C)C2(C)C)=O)CC1.c1(OCC)cc(C(=O)NC)on1 Cc1nc(C(C)C)[nH]c(=NCC2C(C)CCCN2C(c2cc(Cl)cs2)=O)c1Br n1(CC)ccc(C(N2CCC(C)(NC(=O)C(CCOC)OC)C2)=O)cc1=O c1(C(N(CCC(C)NC(Cc2cnc(C)s2)=O)C)=O)noc2ncccc12 N1(C(C(C2CCC2)NC(C(C)SC(C)C)=O)=O)CC2CCCC(C1)N2C C#CC1(CNC(C2CCCCC2(C)NC(=O)CCC)=O)CCOCC1.C(C)=O.O c1(N(CC(CNC(C2(COC)CCCC2)=O)C)C)nc(C(=O)N)c(C)s1 C1(c2nnnn2C2(C)CC2)(NCc2cnc(C)o2)CCOC1C C1(CNC(C=C(COC)C)=O)CCCCN(C(c2ccc(F)cc2F)=O)C1 C1(C=O)CCC(C(F)(F)F)CC1.C1(C(N(CCC)C)=O)CC(N2CC(O)C2)C1 c1(OC)cc(C)nc(N2CCC(NC(c3ccc(CO)nc3)=O)C2C)n1 N1(C(c2c(=O)cc(C)[nH]c2)=O)CCN(c2ccnc(C(F)(F)F)n2)CC(C)(F)C1 C1(C(=O)NC(C)CCF)C2CC3C(C2NC(=O)CC2CC2)C13 N1(C(c2ccn(CC)n2)=O)CC23CCCCC2(C1)CN(C(=O)CC(O)C1CC1)C3 N1(C(C(C)(C(C)C)OC)=O)CCC2(CC1)CN(C(C13CC1C3)=O)C2C(C)C C1(NC(Cc2c(F)ccc(C)c2)=O)CCCCN(C(=O)C(F)(F)CO)CC1 N1(CC)CCN(CCC(=O)NC(CNC(C2CC2OC)=O)C2CC2)CC1 N1(C(C(CCCNC(C(C)n2ccnc2)=O)O)=O)CC2CSCC(C2)C1 C(=O)(C#CC1CCOC1)NC1C(c2n(C)ncc2)CN(C(=O)Cc2ccoc2)C1 Cc1c(C(=O)NC(C2CCN(CCSc3cccc(F)c3)CC2)=O)cccc1Cl C1(C(=O)NC(CCC=C)(C)C)CC1C1CN(C(c2n[nH]c3c2CCC3)=O)C1 c1(-n2c(C)cnn2)ccc(NC(=O)C(=O)Nc2nc(C3CC3)cs2)cc1 N1(C(=O)CC2CCN(C(C3CC34CCCC4)=O)CC2)CCN2C(=O)CCC2C1 Cc1cccn2nc(C(=O)N(CCC(C(C)C)NC(=O)CN3CCC3)C)cc12 C1(OC)CC(CNC(c2n[nH]c(C)c2Cl)=O)N(C(=O)C=Cc2ccncn2)C1 Cc1cc([N+](=O)[O-])c(Oc2cc(F)ccc2[N+](=O)[O-])cc1F CC1CN(C(=O)CCCN2CCOCC2)CCN(C(=O)C=CC2CCCCC2)C1 N1(C(C=CCC)=O)CC(CNC(=O)CC(c2ccccc2)N(C)C)CC1(C)C c1(N2CCC(N(C)C)CC2)nc2ccccc2c(=NC2C3COCC23)[nH]1 Cc1ncc(C(=O)NCC2(C(N)=O)CN(C(=O)C(C(C)C)N(C)C)C2)cn1 C1(C(=O)NC(CC)(CC)CCO)CN(C(=O)CCC2CCC(C)O2)CC1C1CC1 C(=O)(C1CNC(=O)c2ccnn21)NCCCCNC(=O)C1=CCCCC1 C(CCC(=O)NC1CCCC(C=C)C1)(C(C)C)NC(C(CC=C)NC(C)=O)=O c1(SCC(=O)N(C(c2cccnc2)CO)C)cc2ccc(C(=O)O)cc2o1 C(C)(CC)(CCNC(=O)Cn1ccccc1=O)NC(C=CC=CCC)=O c1(CC(=O)NCC(CNC(c2cc(C)ns2)=O)CO)csc2cc(C)sc12 C(CCCCC(=O)N(c1ccc(Cl)cc1)CC(c1cc(Cl)ccc1F)=O)OCC c1(C(C(N2CCCC(NC(Cc3nc(C)sc3)=O)C2)=O)(F)F)cc(F)cc(F)c1 c1(C(=O)N)ccnc2ncnn12.C1(COC)CN(C(=O)C(c2ccc(C)o2)C)C1 CCC(CC)(CC)C(=O)NCCN(C(c1[nH]nc(C(F)(F)F)c1C)=O)C(C)C c1(C(N2CCC(COC)C2)=O)sccc1S(C)(=O)=O.C1(C=O)CCCN1N=O.N C1(NC(CCC(=O)Nc2nnc(CC)s2)=O)CCOCC1.C(=O)CC1CC1.C S(=O)(=O)(c1cccnc1)N1C(C2(COC)CC2)COCC1.C(CS(N)(=O)=O)N C12(CCCC1)C(=O)N2.C(CC(=O)N1CC(Cn2ccnn2)C1)C1(C)CC1 c1(-c2nccc(C(N3C4CCC3CC(O)C4)=O)c2)c(F)cc(F)c(O)c1F N1(C(C2CC(C)OCC2)C(=O)NC(C)(C)C)CCN2C(=O)NC(=O)C2C1 N1(C(C(CC(=C)Cl)NC(=O)C(CC)CCOC)=O)CC2C3CCC(O3)C2C1 N1(C(c2cc(C)ns2)=O)CCN(C(C2CCCC(C)(C)O2)=O)CC1c1cn[nH]c1 C1(OC)CN(C(=O)C=C(C)C(C)C)C(C)(CNC(C2(Cl)CC2)=O)C1 C(C1CCc2c(Br)cccc21)NC(c1sc(C#N)c(Br)c1)=O C1(C2CCCC2)(C(=O)NC2C(CNC(c3c(C)nccc3)=O)CC2)CCNC1=O N1(C(C2C(C)CN(C(C3(C#N)CC34CCC4)=O)C2)=O)CC=CC12CCCCC2 CC1CC(C)N(C(=O)C2=CCCOC2)CCN1C(=O)NCc1ncc(Cl)cc1F C1(C(=O)NCc2ccc(C(=O)NC3CC=CCC3)o2)OCC2CCCC12 C1(C(N(CCNC(c2cc(C)[nH]n2)=O)CC)=O)CC2(CCC2)CO1.CCO.O c1(C(=O)NCC2(COC)CCN(C(C3CC3Cl)=O)CC2)cccn2nccc12 n1(CC)cnc(C(=O)NC(Cn2cccn2)C(=O)NCC(C)C(C)C)c1 Cc1nc(C)c(CNC(C2CCC(COC(C)C)C2)=O)[nH]1 n1(CC=C)nnnc1C(c1ncoc1C)NCc1cc(CC)no1 c1(CC)cc(CNC(C2CCCO2)=O)cc(C)c1.c1(CC=O)cncnc1.C C1(N(C(=O)CC2(CC(=O)O)CC2)C(C)=O)CCCCC1.C1(N)CCCO1 C1(C(N2CCC(Cn3cc(CNC)nn3)CC2)=O)CC(C)CCC1C(=O)O C(N=c1[nH]c(=NCC2CCCS(=O)(=O)C2)[nH]c2c1CCCC2)C1OCC(C)(C)C1 N1(C(CN2CCN(C)CC2)=O)CCC2(CC1)CN(Cc1c(Cl)cccc1Br)C2 C(CCOC)(C(=O)NCC1(CCO)CCC1)NC(C(C)OCC#C)=O c1(C(=O)NC2C(C)N(C(=O)CC(F)(F)F)CCC2)cc(Cl)c2ccccc2c1O c1(C=O)n[nH]cc1[N+](=O)[O-].c1(SCC(=O)N(C(C)C2CC2)C)nccn1C.N C1(CC)CCCC(C(=O)NC2(C)CCSCC2)N1C(=O)OC(C)(C)C C12(Nc3ccnc(N4CC5(OCC(N)C5)C4)n3)CC3CC(C1)CC(Br)(C3)C2 N1(C(C(CC=C)OC)=O)CC(C)CCC1C(=O)N(C)CCc1noc(C)n1 C1(NC(C=C(CCC)C)=O)CC2CCC1N(C(c1cccc3c1CCC3)=O)C2 c1(C(=O)NCC(CC)NC(=O)C(C)NC(N)=O)csc2ccccc12 c1(C(=O)NC(C(C)(C)C)C(=O)NCC2CC23CC3(F)F)cccc2ccoc12 c1(C(C)C)nn(C)c2sc(C(=O)NC)cc12.C1(C=O)CC(F)(F)C1.C1CC1 c1(C(=O)OC)cccc(C(CN2CCSCC2)N)c1.c1sc(CS(C)(=O)=O)nc1C C=CC(C)(CCOC)C(=O)N1CCC(CO)C(NC(c2cnc(F)c(F)c2)=O)C1 C(=O)(C(F)C(C)C)N1C(CNC(CCn2c(C)ncc2)=O)CC1 C1(SC(C(N2CCCC(CC)C2)C)=O)CC=C(C)CC1 c1(C(=O)NC(C)CNC(C2(C#N)CC3(CC3)C2)=O)cncc2cscc12 C(N=c1[nH]c(=NCCNC(=O)OC(C)C)[nH]c2c1COCC2)c1cc(C)ncc1 C1(NC(C(C)NC(CC)=O)=O)CCN(C(=O)CCP(C)(C)=O)CC1F C1(C(=O)Nc2ccc(C3CC3)cc2)CC1C1CCCC1 N1(C(COCC=C)=O)CCC(C(=O)NCC23CC(CCO2)C3)(CC)C1 C(=O)(CCC(F)(F)F)NCCC(C)NC(=O)C(C)(C)C#N C1(CC=C)(NC(c2cnn(CC)c2Cl)=O)CCCN(C(c2cc(C)c(C)o2)=O)C1 c1(CC(=O)N(CCC(OC)OC)C2CC2)ccc(-c2nn[nH]n2)cc1 c1(C2(C)CC2)ccccc1.C1(NC(C2(COC)CC2)=O)CN(C=O)C1.C N1(C(C2CN(C(C)C)C2)=O)CC(C2CC2C(=O)NC2(CO)CCC(C)C2)C1 C#CC1CCCCN1C(c1ccnn1CC(F)F)C(=O)NC1COC1 C1(C2c3nnnn32)CC12CCCCCC2.CCCOCCSC N1(C(C(C)OC)=O)CC(C)(NC(=O)CC2(n3cncn3)CC2)C1 C(C)(C(=O)NC1CCC1NC(=O)Cc1cnoc1)OCC#C CC1(NC(C2CCC(=O)N2)=O)CC(NC(C2CCCCS2)=O)C1 C(c1cncc(C)c1)=CC(=O)N(CCNC(C1CCS1(=O)=O)=O)CC N1(C(c2cnc(CC)s2)=O)CCCCC1C(=O)NCC1CN(C)CCO1 Cc1ncc2ccc(C(=O)NC3CC4CC3CN4C(c3sccc3F)=O)cn12 C(=O)(CN=c1[nH]c2c(c(=NCc3ccncc3)[nH]1)CSC2)N(C1CCCCC1)C C1(COC)CC(C)N(C(=O)CC)C1.C1(C(=O)N)CCCC1F.CCN(C)C C1CN(C(C)=O)C1.C(c1cccs1)=CC(=O)OCC.C12(C=O)CCC1C2 c1(N2C3(CNC(c4c(C)coc4)=O)CC(C2)C3)cc(C(N)=O)ccc1[N+](=O)[O-] N1(C(c2c(N(C)C)cncc2)=O)C2CCC1CC(CCNC(=O)C(C)(C)C)C2 C1(NC(CN(C=O)C)=O)CCN(C(=O)CCC2CC2(F)F)C1.C1CC1.CO c1(CNC(=O)Cn2cc(C3(O)COC3)nn2)nc(Cl)ccc1F c1(CCC(=O)NCC2(C)COC(C)(C)O2)nc(O)c2ccccc2n1 C1(NC(c2sc(C)c([N+](=O)[O-])c2)=O)CCC12CCN(C(C1(CF)COC1)=O)CC2 CC(C(=O)N1CC=CC(NC(C2CCC(C)(F)CC2)=O)C1)C(C)(C)C C(CC(CC)C(=O)NCC1COCC1NC(C1NC(=O)OC1C)=O)=CC N1(C(C(CN(CC)CC)F)=O)CCCCC1c1cn(Cc2cncc(C)c2)nn1 N1CCC(CC=O)CC1.N1(C(CCCOC2(C)CCCC2)=O)C2COCC1C2 c1(N(C)CC)nc(=NCc2ccncc2C(F)(F)F)[nH]c2c1CCC2 C1(NC(c2c(OC)cccn2)=O)CN(C(C2COC(=O)N2C)=O)CC2(CCC2)C1 N1(C(C2CCN(C(C)=O)C2)=O)CCCOC(CNC(c2c(C)n[nH]c2C)=O)C1 C(=O)(C(C)CCCCCC)NCC(=C)CCNC(c1cc(SC)oc1C)=O Cc1cc(C(N2CC(OCC(=O)N(C(C)CC(C)C)CC)C2)=O)nc(O)n1.O c1(SCC)ncc(C(=O)N(C2CCC2)C)cc1C.C1(C=O)CN(C)CC(C)O1.N c1(N2CCC(CC=C)(NC(C3CCCC3OC)=O)C2)cccc(F)c1[N+](=O)[O-] C(=O)(CCCC(F)(F)F)N1C(CNC(c2[nH]cc(C)c2C)=O)CC(OC)C1 c1(C(=O)NC2CCCN(C(C(C(C)C)(C)O)=O)CC2)cccn2nnnc12 C1(CC)CCC(C)N1C(=O)COCCNC(=O)CC1(C)CCOC1 c1(CN(C)C)nc(-c2ncccc2C(F)(F)F)nn1CCC(=O)NC(C)(C)C c1(CC(=O)N(C(C(=O)NCC2CCCC(=O)N2)C2CC2)C)cncc(F)c1 C(C)(C(C)S(C)(=O)=O)NC(=O)NC(COC)COC C1(N(C(C)=O)C2CC2)C(C)CN(C(c2c(C)nc(C3CC3)nc2S)=O)CC1C C12(C(N3CC(COC)(NC(C4CCC4)=O)C3)=O)CCC(F)C1CC2 C1(NC(=O)C=CI)CCN(C(c2ccc(C(F)(F)F)cc2)c2ccccc2)CC1 C1(NC(C(C)SC)=O)CCC(CNC(c2cc(C(C)C)[nH]n2)=O)C1 N1(C(C(C(C)(C)C)O)=O)CCCC(F)(F)CC1.c1(C(=O)N)cc(C(F)(F)F)on1 c1(C(=O)NCCCCCN(C(C(C)n2cncn2)=O)C)cccc(OCCF)c1 C1(C(C(N)=O)NC(=O)NCC2(CF)CCC2)CCOCC1 C12(C(N3CC(NC(c4nn(C)nc4Br)=O)C3)=O)COC(CCO1)C2 C(=O)(C(C)(O)CO)N(CC)C.CC(C)NCCOCC c1(C(=O)NCCN2CCN(C(=O)C3=CCCS3)CC2)csc([N+](=O)[O-])c1 CC1CCCN(C(C2CCSCC2)=O)C1CNC(c1cn2c(n1)CCC2)=O c1(OC)cc(C)sc1C(=O)NC(CNC(C1CCC(C)O1)=O)CC(C)C C(=O)(C1=NNC(=O)CC1)NCC(CNC(C(c1cc(C)sc1)(C)C)=O)(C)O c1ccc(C(C)C)cc1.C(C(O)C(=O)N(CCCNC(=O)C)C)=CCC#C.S c1(-c2cn(Cc3occ(C(=O)NC4CCC4)c3)nn2)ccc2sccc2c1.C1CC1 N1(C(c2sc(C)c(O)n2)=O)CCC2CCCN(C(c3cc(CO)ccn3)=O)C2C1 c1(CNC(C2N(C(c3c(C)cccn3)=O)CCOC2)=O)ccc(Cl)c(C)c1 C1(C(N2CCCC(N(C)C)C2)=O)CC2CN(C(C3CCC4(CC4)C3)=O)CC2C1 C1(NC(C=CSC)=O)CCN(C(c2c(N)sc3c2CCC3)=O)CC12CCC2 Cc1ccc(C(=O)NC23CC2CN(C(=O)C=Cc2nccs2)C3)c(=O)n1C C(=O)(C(=O)C(C)CC)N1C(C(N(CCCC)CCCC)=O)CCC1C(C)C Cc1nc(C(=O)NC2CCN(C(c3n[nH]c4c3CCC4)=O)C2)cc(O)n1 C1(C=O)Cc2nnc(C)n2C1.N1(C(COCCOCC)=O)CCC(C)CC1.C C1(C(=O)NCCN(C(=O)C(C)(c2cccs2)N(C)C)C)CCCC(=O)O1 N1(C(C2C(C)C2)=O)CCC(O)(CN(C(=O)CN(C2CCCCC2)C)C)C1 N1(C(c2cnc(C)s2)=O)CCOC2CN(Cc3cc(Br)ncc3Br)CC12 c1(C(=O)NCC2N(C(CCCOCC)=O)CCOC2)cc(CC)cc(F)c1 C(CC(C)C(=O)N1CCC(C)(NC(=O)CC(C)(C)OC)C1)OC.c1ccccc1 C(=O)(C#CC1(C)COC1)N1CC(CC)C(NC(C2(CC(C)C)CC2)=O)C1 Cc1coc(CN2CCN(c3cc(OCc4ccccc4)ccn3)CC2)c1C n1(CC)ncc2c1CC(C(=O)NC1CC(NC(c3ccoc3)=O)C1)CC2 CC1CN(C(c2cc(C#N)c[nH]2)=O)CC(C)C1NC(=O)CN(c1ncccn1)C C1(CC(=O)NC)CN(C(c2ccn(C3CCC3)n2)=O)CCN1C(=O)C1=NOCC1 CCC(=O)CCC(=O)NC1CCCC(C(=O)N(C)CC2(C)CCC2)CC1 C1(C(N(CC(C)(C)NC(c2cnn(C)c2)=O)C)=O)COC2COCC12 Cc1cc(C(C)C)ccc1C(=O)NCCC1CCCN(C(C2(CCF)CC2)=O)C1 C(=O)(C(F)CC1CN(C(=O)C(C)c2cc[nH]n2)C1)N(CC(C)O)C C1(NC(CCC)=O)CC2CC1CN(C(c1c(C3CCCC3)noc1C)=O)C2 CC1CC(NC(=O)Cn2ncnn2)CCN1Cc1ccc(-n2cccn2)cc1 Cc1cc(OC(F)F)c(C(=O)NCCCNC(=O)C(C)C(C)O)s1 c1(CNC(C(C2CCCN2C(C2CN(C)CCN2C)=O)C)=O)ccc(O)c(F)c1 Cc1nc2ccc(C(=O)NCC3CCN(C(C4CC=CCC4)=O)C3)cn2n1 Cc1cc(-c2csc(Oc3cccc4c3OCC4)n2)cc(C)c1C#N C1CCN(C(=O)CC)C1(C)C.c1(C=O)ccoc1.CC(C)(C)OC(=O)NC N(C(=NCCCCl)N1CC=C(c2ccc(Cl)cc2)CC1)CC(CN(OC)C)O C1(CN(C(c2cnc(S)n2C)=O)CC)CCCN(C(=O)C(c2ccnn2C)O)C1 c1(C(N2CC(N(C(c3csc(C)c3C)=O)C)C(C)CC2)=O)cccc2oncc12 CCC(CCOC)C(=O)NCC1CC(NC(c2ccn(CC(F)F)n2)=O)CC1O C1(NC(CCc2cn(C)nc2)=O)CC(NC(c2c[nH]nc2Br)=O)C12CCC2 c1(C(c2ccc(C(Cn3ccnn3)OC)cc2)NC)cc(F)ccc1S.CC(C)C c1(OCC)ccc(C(c2ccccc2)NC(=O)CC2CCOC(CC)C2)cc1Cl c1(C(=O)NC(c2ccc(OC)cc2)C(F)(F)F)c(Cl)cccc1[N+](=O)[O-] CCC(C)(C(=O)NCC1CC(F)(CNC(=O)CCC2CCCCO2)C1)OC C(=O)(CC(C)O)NCCC1(NC(C(C)OCC(C)C)=O)CC1.C(C)C C1(CC)CN(C(c2ccoc2CNC(=O)C(C(C)(C)C)OC)=O)C(C)CO1 N1(C(c2c(C)ccc(F)c2)=O)CC(C2CCCCN(C(c3cn[nH]c3)=O)C2)C1 CC1(CC(=O)NCc2nc[nH]n2)CCN(C(=O)COCC2CCCO2)C1 N1(C(C2CC(=C)C2)=O)CCC2CN(C(C3CCn4cnnc4C3)=O)C2C1 c1(C(C)O)ccc(-c2csc(Oc3ccccn3)n2)cc1F C1(C(=O)NCC2N(C(c3c(SC)nn(C)c3)=O)CC2)CCC(C)(C)CC1 C(=O)(CCC(N)CN)C1C(c2ccc(C3(C)OCCO3)cc2)C1 CC1CC(CNC(=O)Cc2cnn(C)c2)CN(C(=O)CSc2nc[nH]n2)C1 C(=O)(C(F)(F)C(F)(F)C(F)(F)F)N1CCC(N(CCC)C(c2cnns2)=O)C1 c1(OC)ccc(C(N2CCC(NC(=O)CCc3cccc(Br)c3F)C2)=O)c(Br)n1 c1(C(=O)NCC(CCNC(c2cc(C)c(Cl)cn2)=O)O)nc[nH]c2nccc1-2 C=CC(C)(C)C(=O)NC1CCCC(NC(=O)Cn2nc(C)cc2C)C1 c1(NCC(C)Cc2ccccn2)cc(N2CCC=C(Cl)C2)nc(C(F)(F)F)n1 N1(C(c2c(C)onc2Br)=O)CC2CC(NC(c3cnc[nH]3)=O)C(C2)C1 c1(NC(c2n(C)ccn2)C2CCOCC2)ncnc2c1c(Br)nn2C C1(NC(CCSC)=O)CCCC2CN(C(c3cnc(-c4cccnc4)s3)=O)CC12 C=CC(C)(C)CC(=O)NCCC1(NC(c2cc[n+]([O-])cc2)=O)CCC1 C1(NC(CC(C)CF)=O)CC2CCC(C1)N2C(c1cc2ccsc2s1)=O C1(CNC(C(N2CCSCC2)C)=O)CC2CCC(C1)N2C(=O)C(C)C1CCOC1 O=S(=O)(c1cnc(O)c(Br)c1)NC1CCOCC1F CCCC(CC(C)C)C(=O)N1CCC(C)(C)C(C(N2CC3(CCCCC3)C2)=O)C1 O=C(N(O)CCc1cccc(F)c1)C1CCCCC1.C1CCC2CC12 CC1CCN(C(=O)CC2CC(O)CN2C(=O)Cc2nncn2C)CC1 C1(OCC)(C)CN(C(=O)C(C)Cc2ccnn2C)C1.C1(C=O)CNC(=O)C1 c1(C(=O)OCC(=O)N(c2ccc(Cl)cc2)CCOC)cc(C)n(C)c1C N1(C(C=NOC)=O)CC2=C(C1)CN(C(=O)C(C1(OC)CCOCC1)(F)F)C2 Cc1cc(C)n2ncc(CNC(=O)NCCCN3CCNC(=O)C3)c2n1 c1(CNC(CCOC(C)=O)=O)cc(C(=O)NCCC2CC2C)no1 C(CCCCCNC(C1CCOC1C(C)C)=O)NC(C1(SC)CC1)=O Cc1nn(C)c(C)c1CC(=O)NCC1(C)CN(C(C2(C)CCCC2)=O)CCO1 C(=O)(C1OCCc2ccccc21)NCCN(C(C(CC(=C)C)C)=O)C(C)C c1(C(CNC(C2(SC)CC(F)C2)=O)(C)C)cncc(O)c1 c1(C(=O)NC(CC)CN(C(=O)C(C)(O)CC)C)cnc([N+](=O)[O-])n1C c1(C(N2CCN(C)C(CNC(=O)CC3CC3)C2)=O)cc(Br)c2nccn2c1 C1(CNC(c2c(C)occ2)=O)C(C)CCN1C(c1nc(C2CC2)cs1)=O CC1(C(=O)NC2CCCC(C(N3CC(Cc4ccoc4)C3)=O)C2)C=CCCC1 N1(C(=O)CCSC(F)(F)F)CCC2CN(C(=O)CCn3cc([N+](=O)[O-])cn3)C2C1 C1(O)(C(=O)NCC2N(C(CC3C(CC)C3)=O)CCC2)CCCC(C)(C)C1 C1(NC(c2ccccc2I)=O)CCC12CN(C(=O)COC(F)F)C2 c1(C(N(C(CN(C(c2cc(C)[nH]c2C)=O)C)C)C)=O)cn(C)c(=O)n1C CC1(CNC(=O)C(O)C2CCCC2)CCN(C(c2csc(-c3cn[nH]c3)n2)=O)C1 Cc1cccc(C)c1CC(=O)NCC(C)(O)CNC(C1CCS(=O)(=O)N1)=O c1(C2N(C(CC(CCC)NC(=O)C=CCO)=O)CCC2)cccc2ccccc12 N1(C(c2c(C)c(O)ccc2)C(=O)NC2CCOC2)Cc2nccn2CC(CO)C1 CCC(CC)(C(=O)NCC(C(C)C(C)C)NC(=O)CC(=O)OC)c1ccccc1 Cc1ccc(-n2cc(CCC3CCCN3C(=O)Cn3cnnc3O)nn2)cc1Cl C=CC(CCC)CC(=O)N1CC(NC(c2cnccc2C(F)F)=O)C(C)C1 C1(CNC(=O)CCn2ccnn2)CCN(C(=O)Cc2cc(Cl)cs2)CC1O C(=O)(CCCCC(=O)NCC#CCNC(C1CCC2(CCOC2)O1)=O)OC C1(NC(C2C(CNC(C3OCC(C)(C)C3)=O)OCC2)=O)CC12CCCCC2 CC(O)C(F)(F)C(=O)NCC1(C(C)(C)O)CN(C(c2ccccn2)=O)C1.C C(C(CC(C)C)C(=O)NCCCC1(O)CCC1)NC(c1c(CC)cco1)=O C1(NC(Cc2c(C)n[nH]c2)=O)CCCCC1N(C(=O)CCNC(=O)N(C)C)C CC(C)C(C)(C)c1cn(CCCCCNC(=O)CSc2nnc(S)s2)nn1 N1(C(CC2(NC(C)=O)CCC2)=O)CC=CC(NC(=O)C(C)n2cnnn2)C1 Cc1c(C(=O)NC2CN(C(C3CC4CCC(C3)S4)=O)CC2C)ccc2c1CCC2 Cc1ccc(O)c(C(N2CC(NC(=O)C3=CCOC3)C(F)C2)=O)n1 C(C(=O)N1OC2CCC1C2)N(CCOC)C(c1cscc1C)=O c1(C(=O)NC2C(CNC(COCCC)=O)C2)cc(CC)ccc1C N1(C(C(CC#C)O)=O)CC(C2CCCN(C(c3cc(Br)oc3C)=O)C2)C1 C1(NC(CC(=O)NCC#C)=O)CCCCC1.c1(C=O)cnn(C(C)C)c1C.C c1(CC(N2CC(F)(CNC(Cc3cccc(C)c3)=O)C2)=O)ccc2c(c1)CCC2 C1(c2cn(-c3n(C)nnc3)nn2)CCN(C(=O)COCC2CCCOC2)CC1 c1(C(N(C)C)=O)ccc(-n2cccn2)cc1Cl.C(C(=O)NCC1CC1)=CC c1(C(=O)NCCCOCCN(C(C2(CC)CCOC2)=O)C)ccc(C)cc1 C(=O)(C1(C)OCCc2ccccc21)N(CCC(C)NC(C(C(=O)NC)(C)C)=O)C c1(CC(N2CC(N(C)C(C3(c4ccno4)CCC3)=O)C2)=O)cnn(C)c1 C(=O)(C(C)(F)C(=O)NC)OC.C1CC(F)CN1C(C1CC(n2cnnc2)C1)=O C1CC2(CCO1)CC2.C1(CC(C=O)NC(C2(C)CCCS2)=O)CCC2(CC2)C1.N c1(CN(CCCOC(F)F)C)cn(C2CCOC2)nn1 N1(C(CCc2c(C)ncs2)=O)CCC2(CCCCC2NC(C2CCC(C)C2)=O)C1 C1(C(=O)NCCCN(C(C(CCC)CC)=O)C)CCC(=C(F)F)CC1 C1(N(C)C(C2(N(C)C)COC2)=O)CCN(C(=O)CN2CCC(F)CC2)CC1 C12(C=O)CC(C)(C1)OC21CCC1.C(C)(C=O)OCCC=C.C1(CC)CC1.N C#CC1(O)CN(C(=O)CC2(C)CCN2C(=O)CCCOCCOC)C1 n1(CC)c(C)cc(C(N2CCC(O)(CC)C2)=O)c1C.N1(CC(=O)N)CCSCC1 C1(NC(C2CCCN(C(=O)CN3CCCC3=O)CC2)=O)(CO)CC2CCCC12 CC(C)S(=O)(=O)C(C)C(=O)N1CC(NC(=O)CCCCn2ccnn2)C2(CC2)C1 c1(C2(C(=O)NC(CC)CNC(c3ccncc3)=O)CC2)ccnc(Cl)c1 C(=O)(CC(C)(C)C=O)N(CC(C)NC(c1ccc(OCC)c(Cl)c1)=O)C.O c1(C(=O)NC2CN(C(COCCCC)=O)CC2O)ccc2nc(S)oc2c1 N1(C(CC(c2cc(OC)c(C)cc2)C)=O)CCC2CCCCCC2C1 N1(C(C(C)CSC(F)(F)F)=O)CCN(C(=O)CNC23CCCC2C3)CC1 c1(CC(=O)NCCCCN(C(c2ccnc(C)n2)=O)C)ccc2c(c1)CCOC2 C(C)(CO)(C(=O)N)NC(CCNC(=O)OCC)=O.c1(CC)ncc(C)s1 c1(NC(C2(F)CCN(Cc3cnc(Br)s3)C2)=O)ccc([N+](=O)[O-])cc1 Cc1ccc2scc(C(=O)NC(C3CCN(C(c4cnc(S)[nH]4)=O)C3)(C)C)c2c1 c1(C(N2CC(C(=O)Nc3c(C)cc(OC)c(Br)c3)C2)=O)cnc2cc(C)nn2c1 C(C(C)CC(=O)NC(c1ccccc1)CNC(=O)C(c1cnn(C)c1)C)OC c1(C(N2C(Cn3cc(C(N4CCCC4)(C)C)nn3)CC2)=O)sc(F)cc1Br c1(CC(N2CCC(NC(=O)C(=Cc3cscn3)F)C2)=O)nnc2n1CCCC2 c1(C(=O)NC2CCC(N(C(C3CN(C)C3)=O)C)C2)c(F)c(F)c(F)c(F)c1F C1(NC(c2c(CC)ncs2)=O)CCCC(N(C(=O)CNC(=O)NC)C)C1 N1(CC(=CC2CCCC2)C)CCCC(C(C)NC(C2(C)COC2)=O)C1 c1(C(N2CCN(C(c3n(CC)nc(C)c3)=O)C(C)C2)=O)ccc(S(C)(=O)=O)cn1 c1(C(=O)NC(C2CCCN2C(c2ccsc2)=O)C)cc(C(C)(C)C)n(C)n1 N1(C(C(CCCOC)C)=O)CCN(C(=O)C2=C(C)OCC2)C2CCC12 N1(C(Cc2ccc(C)nc2)=O)CCN(C(=O)CSc2c(C)n[nH]c2C)C2CCC12 C(CCC(=O)NC1(C(C)O)CC1)(C(C)C)NC(C(CC)NC(N)=O)=O Cc1cc(CC(=O)N(CC(O)CN(C)C(c2cc3scnc3[nH]2)=O)C)ccc1Cl N1(C(c2cnc(CCC)s2)=O)CCC(C)C1.c1(C(=O)N)cnn(C2CC2(F)F)c1 c1(SC)ncc(C#N)c(N(CC(C)C(=O)NC)C)n1.C(C)=O C12(NC(=O)NCc3cn4ccc(C)nc4n3)CC3CC(C(=O)N1)C2C3 c1(C(CC)NC(=O)C=CCn2cc(Br)cn2)ccc(OC(C)C)cc1 N1(C(C(CC)C2CCOCC2)=O)CCN(C(C2CCCC2O)=O)CC12CCC2 C(=O)(CC1=CCCCC1)NCCC1N(C(C2C(C)(C)OCCO2)=O)CCC1 n1(CC(=O)NC(C)CCCNC(C2CC(=O)CO2)=O)cc2ncccc2n1 C(=O)(C1=COc2ccccc2O1)N(C1CCC(NC(CC(=C)Br)=O)C1)C C(=O)(C(CC(C)C)C1CCC1)NC(CNC(C(C)OCC#C)=O)CC(C)C CC1C(C)N(C(c2cc(C(F)(F)F)nn2C)=O)CCN1C(C1(F)CCCC1)=O NC1(C2(C(=O)Nc3cncc(OC(F)F)c3)CCC2)CCC1 c1(C(C)NC(C(C)NC(=O)OC)=O)ccccc1-c1nn[nH]n1 Cc1cc(NC(=O)CC(C(C)OF)NC(C2(C)CNC(=O)N2)=O)cnc1F CC1C(c2noc(C3CCCSCC3)n2)CCCN1C(=O)CCC=CBr Cc1ccc(CNC(=O)C(CO)NC(=O)Cc2csc(C)n2)c(F)c1 c1(CC)nc(N(C2CCN(C(c3cccc(Cl)c3F)=O)C2)C)c(CC)c(Cl)n1 C1(C)(C(=O)NCCC(COC)(C)C)CC(O)CN1C(c1nnc(S)n1C)=O c1(CC(=O)NC2CC(NC(C3N(CC)CC3)=O)C2)cc(Br)ccc1OC N1(C(CCC2CCN(C(c3cc(OC)n[nH]3)=O)C2)=O)CC2C(C1)C2(F)F CCCC(C(O)C(=O)N1CCSCCC1C)NC(c1nccn1CC)=O c1(C(=O)NCC23C(CN(C(CC4(C)CC4)=O)C2)CCO3)[nH]nc2c1CCC2(C)C C(N=c1[nH]c2c(c(=NC(C)C(C)CC)[nH]1)CCCCCC2)c1nc(CC)sc1 N1(C(C2N(CCC)C(=O)CC2)=O)CC2CC1CCN2C(=O)CN(C)CCOC CC1(C(N2CCC(N3CC(O)C3)C2)=O)CCCN1C(=O)CCc1cccs1 c1(C(=O)NCC(CNC(C2C(C=C)C2)=O)OC)cc(OC)cnc1F O(NC(=O)CCC1CCC(NC(c2occc2CC)=O)C1)C(C=C)C c1(C(C)C)nnc2n1CC(CNC(=O)C(C1CS(=O)(=O)C1)N)CC2 Cc1cccc(C(N2CCC2CNC(c2ccc(OC3CC3)cc2)=O)C)c1 Cc1nccc(CCC(=O)NCCCN(C(=O)CC(=O)N)CCO)n1.C1CC1.C N1(C(CC)=O)C2CCC1CN(C(C1(Cl)CC13CCC3)=O)C2 C1(NC(CC2C(C)(C)C(O)C2)=O)C2CC1CN(C(c1ccn(C(F)F)n1)=O)C2 n1(CCN(C(c2ccc(Cl)s2)=O)CC)cc(C(C)(O)CC)nn1 c1(C(=O)N)oc(S(N)(=O)=O)cc1C.C(CC(C)(C)C(=O)NC1CCCC1)OC C(=O)(CCCN=[N+]=[N-])N1CC(OC)(CNC(=O)C(N2CCC(O)CC2)C)C1 c1(NC(C2CCN(c3ccnc(OC)n3)C2)=O)cnc(Cl)c(Br)c1 C1(NC(=O)COc2ccccc2)CN(C(=O)CCC(F)(F)F)C2(CCCCC2)C1 N1(C(C)=O)CCCC1(C)C(N1CC(F)(CNC(=O)C(C)(F)F)C1)=O c1(C(=O)N)cnc(C)c(C#N)c1.C1(C(NOCC(=O)OCC)=O)CC(C)C1 C(C(=O)NC1(C(=O)N(C(CO)C2CC2)C)CCN(C)C1)(C(C)C)OC c1(C(=O)NC2CCCN(CC)C2=O)cc2cncc(Br)c2s1 C#CC1CN(C(C2(F)CCN(C(c3c(CO)n[nH]c3C)=O)CC2)=O)CC1O C1(O)(CC(=O)NC2C(C)(C)C2)CN(C=O)C1.c1cc(-c2cccnc2)[nH]n1.N C1(C)(CC)CC(NC(c2cccc(=O)o2)=O)CN1C(=O)COCCSC C1(C(=O)NC(C(C)NC(=O)CCCc2cnn[nH]2)C)CC2CCC2C1 CC(F)(F)CCC(=O)NC1CCN(C(C2(c3cccc(Cl)n3)CC2)=O)CC1O C1(NC(c2ccnc(C(C)C)n2)=O)CCSC12CN(C(=O)C(C#N)C1CC1)C2 c1(C(=O)NCCC(CNC(=O)C2=CCCSC2)O)c[nH]c2ccc(F)cc12 c1(CNc2ccc(CNC(c3ccccc3)C#N)cn2)ccc(F)c(Br)c1F N1(C(=O)NCc2c(C#C)cccc2)CC2CCCN2CC1CO N1(C(c2c(C)cno2)=O)CC(C)CCC1CNC(C1CCS(=O)CC1)=O N1(C(CC)=O)CC(CNC(=O)C(C2CCCCCC2)OC)C(C)(C)C1 C1(CNC(c2c(C)snn2)=O)CN(C(=O)CCOC(C)CC(C)C)CCN1C c1(OC)ccc(C)cc1C(=O)NC(C1CCN(C(=O)CCC(C)(C)F)C1)C N1(C(=O)CC2CC(F)(F)C2)CC2(CCN(CCn3cccn3)CC2)C1 [N-]=[N+]=Nc1cnccc1C(N1CCC(CCNC(=O)CSC2CC2)C1)=O Cc1nc2nccc(N3C4CCC3CN(C(c3cnn(C5CCC5)c3)=O)C4)n2n1 C1(C(=O)NCCSCC)CCN(C(C)=O)C1.c1(C(=O)N)cncc(C)c1 Cc1ccc(C(F)(F)C(=O)NC2CCCC2NC(c2ccco2)=O)nc1 c1(CC=O)cccc2c1CCC2.c1(CC)nccnc1C(=O)NC1CCC1C.N c1(OC)cc(CC(N2CCCC(N(C)C(c3coc(O)n3)=O)CC2)=O)cc(Cl)c1 Cn1cc2c(n1)CCN(C(C1CCCC1CNC(c1ccc(C#N)n1C)=O)=O)C2 C1(C)(C(N2CC(CC(C(=O)N)F)C2)=O)CC(=O)N(C)C1.Cc1ccsc1C N1(C(c2c(C)nc(CC)o2)=O)CCN(C(=O)CCC(C)(C)[N+](=O)[O-])CC(C)(F)C1 c1(OCC(=O)NC2CCC2NC(=O)Cc2csc(S)n2)ccsc1Cl c1(OCC)ccc(C(=O)NCC(CNC(C2CC2C)=O)OC)cn1 C(CC(CNC(C1CC(CCO)C1)=O)NC(c1coc(C)c1)=O)OC C(C)(C)(CCNC(=O)CC=CC(C)(C)C)NC(C(C1CCCC1)OC)=O Cc1nc(C(N2CCCCC2CCC(=O)NCC(C)N(C)C)=O)sc1C C1(CNC(c2ccc(C)c(Cl)c2)=O)CC2COCC2N1C(c1ccncc1)=O c1(C(=O)NC(C2N(C(CCC=CCC=C)=O)CCC2)C)ccc(OC)nc1OC C(=O)(C(C(C)C)NC(C1CCCC1)=O)N1CCC(C(C)NC(C)=O)C1 CN1CCC(C(=O)NCC2CCC(C(=O)NCC#CC(F)(F)F)CC2)C1=O c1(CC)nocc1C(=O)NCCSCC(N1CC(CCO)(CC)C1)=O C(=O)(C(C)(F)C(F)(F)F)N.c1(C(N(CCC)CC)=O)ccncc1.C(C)C C1(O)(C(N2CCN(C(C)=O)C(C)C2)=O)CCC(C)(C)CC1.C(C(=O)N)NC(C)=O C(=O)(C(F)(CNC(=O)Cc1ccsc1)C(C)C)NC(C=C)C1CC1 C1(OC(CCNC(=O)NC)C)CC(F)(C(=O)OC)C1 c1(C=O)cn(CC(C)C)c2ccccc12.C(C(=O)NC(C)C1CC1)SCC=C CC(=NO)C1CC(C(=O)NC(C)(C)CN(C)C(C2CCC2)=O)C1(C)C Cc1cccc(C)c1C(N1CC2(CC2)CC1C(=O)N(C)CCc1scnc1C)=O C1(NC(CN(C(c2cccnc2N)=O)CC)=O)CCCC(OC)CC1.C1CC1 c12cc(N)c(cc1F)NC(=O)C2.C1(C(=O)OC)CC(CF)C1 c1(C(C)C)ncc(C(=O)N(C2CCN(C(c3coc(CC4CC4)n3)=O)C2)C)cn1 C(C)(C(C(=O)NC1CCOC1)NC(=O)CCC1CC(C)C1)OC CCC(CC)(C(=O)NCCCC(=O)N(C1CCC2(CC1)CC2)C)OC c1(CN(C(CC2(C#N)CC2)=O)C2CC2)cn(CCc2ccccc2)nn1 c1(-c2cn(C(C)=O)nc2)ccc2nnc(C(=O)Nc3nc(Cl)ccc3O)n2c1 C1(C(=O)NCC(C)(C)NC(C2(Cl)CC23CCOCC3)=O)CCc2ccnn2C1 N1(C(c2c(C)[nH]nc2Br)=O)CCCCC2(CCN(C(c3cc[nH]c3)=O)C2)C1 N1(C(c2c(C)occ2C(F)(F)F)=O)CC(NC(C2CC=CC2)=O)C(C)(C)C1 c1(CC)ncnc(N(C2CN(C(c3ncc(F)cc3F)=O)C2)C)c1F N1(C(=O)C=Cc2cccnc2)CCC2CCN(c3ncc(F)cn3)CC2C1 Cc1cc(C(=O)NC2CC(C)(NC(=O)CCS(N)(=O)=O)C2)cc(C)c1 c1(C(C(=O)NC(C2CN(C(c3cncs3)=O)C2)C)C)cn(C)c2ccccc12 N1(C(=O)CC2(O)CCOC2)CCCC2(CCN(C(c3ncccc3O)=O)C2)C1 N1(C(c2nnc(C)s2)=O)CCOC(C(C)NC(c2ccccc2Br)=O)C1 C1(CC)CCN(C(c2cccc(-c3ccccc3C(C)(C)C)c2)=O)CCO1 S(=O)(=O)(c1csc(C2CC2)n1)N1C(C)CC(N(C)C)CC1 N1(C(c2cn(C(C)(C)C)nn2)=O)CCC2(CC1)CC(C(=O)NC)C2.c1ccc[nH]1 C1(C(N(CCCCN(C(=O)CCC2CCCO2)C)C)=O)COC(=O)N1C C=CCCCCC(=O)NCC(CNC(C1CCC(C(C)(C)C)O1)=O)S(C)(=O)=O c1(NC)snc(C)c1C=O.c1(CCC(N2CC(CC)C2)=O)nc(C(C)C)no1 C1(C(C)C)CCC(C(=O)NC2CCC(O)C2)N1C(C1CCCC1)=O C1(CC(=O)N(C(C)CN(C)C(c2cn(C)ccc2=O)=O)C)SC2=NCCN2C1=O C1(C(=O)NC(C2(C(=O)N(CC(Cl)Cl)C)CC2)C)CC(O)(CO)C1 CON(CCC(=O)N1CCCC(O)(C2CC2)C1)C(=O)C1CC(=O)C1 C#CCCCCC(=O)NCC1CC(C(=O)N(C2(c3cc[nH]n3)CC2)C)=NO1 C1(NC(CCCCCNC(N)=O)=O)CC2CCC1CC2NC(C1CCCCS1)=O c1(C(=O)NC2C(NC(C(C)(C)c3cccnc3)=O)C2)ccc(O)cc1 c1(C(=O)NC2CC3(CN(C(C(C)C(C)(C)C)=O)C3)OC2)cnc2nccnc2c1 CC12CCC(C(N3CC4CCN(C(=O)C(C)(C)O)CC(C4)C3)=O)(CC1)C(C)(C)O2 N1(C(c2cc(CC)oc2C)=O)CC2(CCN(C(=O)CC3CCCC3C)C2)C1 S(=O)(=O)(c1ccccc1C(=O)N(C)C)NC1(c2cccc(C)c2)CC1 N1(C(C(C)(C)OC)=O)CC2CCC1CN2C(=O)C(=Cc1ccccc1)OC CC(CC(=O)NCCC1(O)CCN(C(=O)C(C)(C)c2cnsc2)C1)C(C)(C)C Cc1cccc(C(N2CC(NC(=O)CN(CC(C)(C)C)C)C(C)C2)=O)c1C S(=O)(=O)(C1CCN(C(=O)C(=O)NC(C2CCCC(F)C2)=O)C1)N(C)C N1(C(C2N(CC)CCOC2)=O)CCCC2(CCCN2C(=O)C(F)C(C)(F)F)C1 CCC(C)CC(C)NC(=O)CN1CCN(C(=O)C(CC)OC)CC1 C(CNC(=O)C=CCN(C(=O)CC1CCCO1)C)(C(C)C)OC c1(C(N2CCN(C(C(C=CCCC)O)=O)CC2)=O)cc(C)nnc1CC C(C)(C(=O)OCC(=O)N(C1CCCC1)C(C)C)OCC C1(C2(O)CN(C(C3CS(=O)(=O)C3)=O)C2)CC1.CC1CCCC1C(=O)NC N1(C(CCC2N(C)CCC2)=O)CC=C(C(=O)NCCC2(C)CCOCC2)C1 c1(C2C(C(N(CCN(C(=O)CCCc3nccs3)C)C)=O)C2)ccc(O)cc1 N1(C(=O)C=CC2CCOC2)CCN(C(=O)Cc2csc(NC=O)n2)C(CO)C1 c1(N2CC(C(N)=O)(CNC(C(C)OCC)=O)C2)cc(N(C)C)ncn1 CCC(C(F)(F)F)NC(C1(OC)CCN(C(c2cc(OC)ccn2)=O)C1)=O Cc1ccnn1CC(=O)NC(CNC(=O)C)C(C)C.c1ccccn1.C=O.N Cc1coc(C)c1C=CC(N1CCCC1CCCNC(C1(C)CCCCO1)=O)=O c1(OC)c(C(N2CCC(CCCNC(c3cnnn3C)=O)CC2)=O)cccc1F N1(C(C(C2(O)CN(C(C3CC(C)C3)=O)C2)F)=O)CC(C)OC(C)(C)C1C C1(CC(=O)O)CNCCN1C(c1cccc(SCC#N)c1)=O c1(CCC(=O)NC2CN(C(=O)C=C(Cl)Cl)CC2O)cc2ccccc2o1 CCCCC(O)C(=O)N1CCCC(CNC(=O)CNC(=O)CCC)CC1 c1(NC(CC2C(C=O)C2)=O)ccc(C(=O)NC2CC(C)(CC)C2)cn1.O N1(C(Cc2c(C)ccs2)=O)CC(NC(=O)CCNC(=O)C=CCl)CC(C)C1 c1(C(=O)NC(C(C)NC(C(CCSC)O)=O)C)cccc2nn[nH]c12 Cc1nc(NC2CCC(NC(c3ccc(N(C)C)cc3)=O)C2)ncc1Br C1(C(=O)NCC2CC(O)C(O)C2)(CC)CCN(C(=O)CCC)C1.C(C)C.O C1(CNC(C(CNC(CCNC(C)=O)=O)O)=O)NC(=O)NC1=O N1(CC)CC2CCC(NC(C3SCCCS3)=O)CC2C1 C(=O)C1=CS(=O)CCC1.N1(C(CN2CC(C)(C)C2)=O)CCC(C(C)(C)C)(C)C1 C12(C(N3C(CN(C(c4ccc(C)s4)=O)CC)CCC3)=O)CCCC1C2(F)F CC1CC(C)(C(=O)N(CCCC(=O)NCC2(F)CC(O)C2)C)C1 Cc1cccc(CN(C)C(N2CC(Cc3cccc(-c4nc(C)cs4)c3)C2)=O)c1 c1(NC(CN(CCC)C(c2cc3ncccc3[nH]2)=O)=O)ccc2c[nH]nc2c1 c1(CC)ncccc1C(=O)NCC1(O)CCC1.c1(CCC(=O)N)cncn1C C(=O)(C(F)(F)CCn1ccnn1)N.c1(C(=O)NCC(C)OC)ccc(Cl)o1 C1(C(C)(C)C)CC(C(=O)N2CCCCC(CNC(c3nocc3Cl)=O)C2)=NO1 n1(C(C)C)cc(C(=O)NC2CCC(NC(=O)CSC3CCCCO3)C2)cn1 CC1(C)CCOC(C(=O)NC2CCC2CNC(c2cnn(CCO)c2)=O)C1 C1(CNC(c2c(C)nsc2C)=O)CC(C)(C)CN1C(c1coc2c1CSC2)=O N1(C(c2c(CC)nccn2)=O)CC(C)CCC1CNC(c1ccc(Cl)cc1F)=O C=C1CCN(C(=O)C(O)C(C)(C)C)C(C(=O)NCc2cc(F)ccc2O)C1 CCCCC(CNC(=O)C(Cc1ccoc1)NC(=O)CCCC(=O)NC)CCC c1(CC(=O)NC(C)CCN(C)C(C2(C)CC=CC2)=O)c[nH]c2nccc(Cl)c12 c1(C(=O)Nc2cncc(F)c2I)ccc2c(-c3cccc(C4CC4)c3)c[nH]c2c1 Cc1cc(C(C(=O)NCCC2(C)CC2)N(C)CCc2nccs2)sc1Cl Cc1c(C(=O)N(CC(O)CN(C)C(c2ncccc2N)=O)C)noc1C1CC1 C1(C(=O)NC2(COC)CN(C(C3CC3F)=O)C2)Cc2cc(Cl)ccc2O1 C1CN(C(=O)C=C(C2CC2)C2CC2)CC12CC2.C1(C=O)CCCC1C=O.C C(=O)(CCCC(OC)OC)N1CCCC(C(=O)NC2(CC=C)CCCC2)C1 N1(C(C(C(C)C)=O)=O)CCCC(C(=O)NC(C)CC2(O)CCC2)CC1 c1(NC(C(=O)OCC2ON=C(C(=O)OC)C2)=O)ccc2c(c1)CCC2 Cc1cc(C)c(NC(C2CCC(NC(c3cc(N)cc(F)c3)=O)C2)=O)c(C)n1 C1(C(N2CC(NC(Cc3n(C)ncc3)=O)C2)=O)C2C3CC4C1C1C2CC3C41 N1(C(c2cc(OC)n[nH]2)=O)CC(=O)NCC1C(=O)Nc1cncc(Cl)c1 N1(C(C2(CC#C)CCCC2)=O)CCN(C(=O)CC2C(C)(C)C2(C)C)C(CC)C1 c1(C(=O)OC)ccccc1CS(=O)(=O)NC(c1cncn1C)CO c1(C(N2CC(NC(C(C)N(C(C)=O)C)=O)C(F)C2)=O)ncc(N)cc1C C1(NC(Cc2c(C)noc2C)=O)CC(C2CCN(C(=O)CC#N)C2)C1 C1(O)(C(C)NC(C2CC(F)(CO)C2)=O)CCN(c2nccc(-n3ccnc3)n2)C1 C(=O)(CCC1=NNC(=O)CC1)N1CC2C(NC(C(=Cc3cccnc3)C)=O)(C2)C1 N1(C(C(=O)NCCOC)C(C)C2CCCC2)CCN2C(=O)OCC2C1 c1(-c2ccc(NC(C=C(C)C)=O)cn2)cc2cc[nH]c2cc1F C1(CN(CC(C)OC(N)=O)C)CC(=O)N(Cc2ccccc2)C1 Cc1ncnc2c1CC(C(N1CC(C3(NC(C4CC(C)(C)O4)=O)CC3)C1)=O)CC2 c1(CCC)cc(C(=O)NCC2COCCN2C(c2ccnc(C)c2)=O)ccn1 N1(C(C(CSC)C)=O)CCN(C(c2cc(F)ccc2C)=O)C2CC12 c1(C(=O)NCC(CC)NC(C2(CC=C)CCCC2)=O)sc(Cl)c(Cl)c1O O=C1CSCC(C(=O)NCC2CCCN2C(=O)CC2CC3CCC2C3)N1 N1(C(CNC(CC)=O)=O)CCC(CC)(NC(c2csc(C(F)(F)F)n2)=O)CC1 Cc1cn(C)nc1C(=O)NCCC(C)NC(=O)CCc1nnc(-c2ccsc2)o1 c1(N(CCSC)C)nnc(Cc2cc(C)no2)n1CC(C)(C)O C1CC2(C1)CN(C(=O)C(C(C)C)C1CCC1)C2.C(C)(C)C=O.C(=O)N.CC C1(NC(C(C(COC)C)C)=O)CN(C(=O)CCc2ccccc2)CCC1(C)C CCC(C)CCC(=O)NC1COCC1NC(=O)CCCOc1ccc(F)cc1 C1(NC(c2cn3c(n2)CCC3)=O)CC2(CCCN(C(C3(O)CCCCC3)=O)C2)C1 N1(C(c2n(CC)ccn2)=O)CCCC(C)(NC(=O)Cc2ccoc2)C1 S(=O)(=O)(c1cccc2scnc12)NC1CCN(Cc2c(C)ccs2)CC1F c1(NC(c2cc[nH]c2C2CCC2)=O)cnc(CO)nc1 Cc1ccc(C2CC2)c(C(=O)NC2CCN(C(=O)C=C3CCC(C)C3)C2C)c1 Cc1nccc(C(N2CCC(C(F)C(=O)N(C)CC3CC3)C2)=O)n1 C1(OC2C(C(=O)NC3CCCCC3)C2C)CCC2CN(CC(=O)NCC)CC2C1 C(C1=COCCC1)(c1n(CCOC)nnn1)NCCC(C)C(F)F C1(C(=O)NC(C)(CNC(=O)Cc2nnc(O)s2)C2CC2)CN2CCN1CC2 C=C(C)c1cncc(C(C(=O)NC2CCOC2)N(CC)Cc2ccc(C)o2)c1 N1(c2ncc(CC)cn2)CCCN(Cc2ccn(C)n2)CC1C CCCC(C)CNC(=O)C(Cc1ccoc1)NC(=O)C(=O)NCC(F)F C(C(C)(C1CCC1)NC(=O)COC(F)F)NC(COC(C)(C)C)=O Cc1c(C(N2CCN(C(C3CC34CCCOC4)=O)CC2)=O)[nH]c2c(C)cccc12 C1(N(C(C2CC3CC2C3)=O)CC)CCN(C(C2CCCCC2F)=O)CC1 N1(C(C(C)(C)SC)=O)CC(CNC(c2cc(C3CCCC3)no2)=O)CCC1C c1(C(c2nnnn2C)NCC2(CCC=C)CC2)cncc(Br)c1C c1(C(=O)NCC2N(C(c3nc(OCC)oc3)=O)CCOC2)ccc(O)nc1F c1(C(=O)NC2(CC=C)CCN(C(=O)C(C)=O)C2)ccn(C(C)C)c(=O)c1 c1(NCC(n2cc(C(N3CCn4nccc43)=O)nn2)C)ccn2ncnc2c1 c1(C(=O)NCC(C)N(C(=O)C(F)=CCCF)C)ccc(F)c(Cl)c1 c1(C(C)=O)ccccc1C(=O)NC(C)(CNC(C1CC1C(F)F)=O)CO c1(COCC)ccc([N+](=O)[O-])cc1-c1noc(C2CCCC3(CCC3)O2)n1 CC(CC(C)(F)F)C(=O)NCCCC1CCCN1C(=O)CCc1ccccc1O c1(CN2CCCC(CNC(c3occc3Br)=O)C2)ccnc(Cl)c1Br c1(C(=O)NC(CN(C(C(CC#C)C)=O)C)CC)c(C)cc(F)cc1Br c1(OC)cccc(Oc2sccc2C(=O)NCC2CN(C(=O)CC)C2)c1.O N1(C(c2ccc(OC)cc2)=O)CC2(CCCN(C(=O)CC3CC34CC4)C2)C1 CC(C)C(O)C(C)C(=O)N1CCN(C(=O)C2=CCN(C)C2)CC1C1CC1 Cc1nc(=N)[nH]cc1C(=O)NC(C1CN(C(=O)C=Cc2ccnn2C)CCO1)C C(C(=O)NCCCC(C)C)(C(F)(F)F)OC(C)=O.c1(C(=O)N)snc(O)c1Cl c1(C(=O)NCCN(C(C(CC)=CCCC)=O)CCO)ncncc1Cl.CCC=C c1(C(N2C(CNC(c3ccc(CC)s3)=O)CC2)=O)cc(-n2cccc2)ccc1Cl C(=O)(C(COC)OC)N1C(C(=O)NCCC(=O)NC(CC)C)CC1 C1(NC(CC(C)SC)=O)CCCC12CCN(C(c1cncn1C)=O)CC2 Cc1ccc(C=CC(=O)NC2CCC2CNC(=O)C(c2ccccc2)O)s1 N1(CC(=O)NCC(CCNC(C2CCN(C(C)=O)C2)=O)O)CCCOC1=O N1(C(c2cncc(C)c2Cl)=O)C2CCC1CC(N(C)C(c1cnc(S)n1C)=O)C2 N1(CCC)CC(C(=O)NC2CC2CNC(c2cc(C)co2)=O)CC1=O.C N1(C(c2c(C)cc(C)[nH]2)=O)CCC(CNC(=O)C(F)(F)C(F)F)C(F)(F)C1 c1(C(N(CCCCN(C(C2C(C)OCC2)=O)C)C)=O)cc2n(c1)CCCNC2=O N1(C(C2C(C)CC3CC3C2)=O)CC2CC(C1)N(C(c1nc(O)[nH]c(=O)n1)=O)C2 N1(C(CC2C(OC)CC2)=O)CCN(C(c2ncc(F)cn2)=O)C2COCC12.C(C)=O c1(C(N(CC)Cc2cc3ccccc3o2)=O)c(C)nc(-c2cccnc2)nc1O C1(NC(COc2c(OC)cccc2)=O)CCCN(C(=O)C(F)n2cccn2)CC1 CC(C)(CCCNC(c1cnc(S)[nH]1)=O)NC(=O)COc1ccccc1 CC(=Cn1ccnn1)C(=O)NCc1cn(C2CN(CC3CC34CC4(F)F)C2)nn1 c1cccc(Cl)c1.C=CCC(CNC(=O)C=CC)NC=O.C(C)(C)C.O C(=O)(C1CCCc2ncnn21)NCC1N(C(COCC(C)(C)C)=O)CC=C1 C(=O)(CCC(C)(C)C#N)N1C2C(C(N(C3CCCCC3(F)F)C)=O)C(C2)C1 N1(CC(=O)Nc2nnc(C(C)C)s2)CCC(NC(C2(C)CCN(C)C2)=O)CC1 N1(C(CNC(N)=O)=O)CC2CC(NC(c3cc(C4CCC4)on3)=O)C1C2 C1(C(=O)NC(c2cccc(F)c2)C)C2C(CN1Cc1ccc(Cl)cc1)C2(C)C c1(OC)ccc(C(=O)NC2CN(C(=O)CC3C=CCCC3)CC2C)nc1 c1(NCCC2CCC(NC(c3c(C(C)C)onc3)=O)C2)ncnn2c(Br)ccc12 C(CCCOC)(C(=O)NCC1CC1Cl)NC(CC(CC)C)=O C1(C(=O)NC(c2cc(C)on2)C)CCN(C(=O)C(C)C(F)F)CC1(C)C N1(C(c2cc(CCC)[nH]n2)=O)CC2(CO)CC1(C(=O)NCCCCCCO)C2 Cc1ncccc1C(=O)NC(C)C(=O)NC1CCCC(CO)C1 N1(C(CCC2CCN(C(C3(C)C(C)(C)C3)=O)C2)=O)CC2CC1CS2 N1(C(c2c(C)cno2)=O)CC(CO)C2(CCN(c3snc(C)c3C#N)CC2)C1 CC1=NNC(=O)C1CC(=O)N.C1CCCCC1.C(O)(C(F)(F)F)C1(C=O)CC1 C#Cc1ccc(OC)c(-c2nc(-c3ccc(Cl)s3)no2)c1 CCC(O)(CC(=O)NCCC(C)N(C(=O)C(O)C(C)C)C)c1ccccc1 N1(C(C2CC(C)(O)C2)=O)CC(NC(=O)CNC(c2ccsc2)=O)C(F)C1 c1(CC)ncc(C(=O)NC(c2cnn(C)c2)C(=O)N2CCC2C(=O)NC)cn1 C1(C=O)CCCC(C)(C)C1.N1(C(C(c2n(C)ncc2)(C)C)=O)CC(C)C(O)C1.N c1(C(N2C(CCNC(C(C(C)C)SCC)=O)CCCC2)=O)cc(N)ccc1.S CC1CN(C(C2(n3nccn3)CC2)=O)CCN1C(=O)C(CO)N(C)C N1(C(c2ccccc2)=O)CCN(C(C2(c3cccnc3Cl)CC2)=O)CC1 C(c1nc2ccccc2[nH]1)=CC(=O)NC1C2CN(C(CCC(=C)C)=O)C1C2 CCCCC(CNC1CN(CCF)C1)CC C1(C2N(C(CC(C)F)=O)CCC2)CCCN(C(c2cc(C(F)(F)F)no2)=O)C1 C1(NC(c2cc(C)sn2)=O)CN(C(=O)CC2C(C)(C)C2(C)C)CC1C N1(C(C=C(CC)CC)=O)CCC(CNC(C23CCCC2C3)=O)(OC)CC1 CC1(C)CCC(NCC2NCCC23CC3)CC1C#N c1(CC)ccc(C(=O)NC(C)CCCNC(=O)CCOC(C)C)nc1 C(=O)(C(C(C)(C)C)NC(N)=O)NCC(CCCC)NC(C1(CO)CC1)=O S(=O)(=O)(c1cccnc1NCCC(C)CC(C)(C)C)NCCC(C)O C1(C(=O)NC2CCCCC2NC(C2CCCS2(=O)=O)=O)CN2CCC1CC2 Cc1ccc2ncccc2c1C(=O)NCCC1(O)CCOC1 c1(C(N2CC(NC(CCC3CCN(C)CC3)=O)C(F)C2)=O)nc[nH]c2ncnc1-2 c1(NC2CCCN(C(=O)Cn3ccccc3=O)CC2)ncnn2cccc12 C(=O)(C1=CCCC1P(C)(C)=O)N1CC2CCN(C(C=C(CCN(C)C)Cl)=O)C2C1 C1(C(=O)NC)CCCN(c2ccncn2)C1.CC(F)(F)F.CC.CC.CCO.O CCC(C)C(C(=O)NCCCNC(C)=O)N(C)C(c1ccc(O)nc1C)=O C1(O)(CC)CCCN(C(=O)C=CC2CCCO2)C1.CC(C)(CC1CCC1)C=O.N C(=O)(CC(C)(C)NC(C1C=C(C)CS1)=O)NCCCOCC=C C1(C)(NC(C(CC(=C)C)NC(=O)CC2CCC(=O)N2)=O)CC(C)(C)OC1=O CC(C)CC(O)C(=O)NCC(c1ccccc1)NC(=O)C(O)C(F)(F)F c1(C(=O)NC(CNC(=O)CCOC2CCOC2)CO)ccc2cccnc2n1 C1(NC(C(C)(C)OCC(F)(F)F)=O)CC2CCC2C1.C1(C=O)CSCC(=O)N1 N1(C(C(COC)C)=O)CCC(C2(NC(=O)Cc3cc(Cl)ccc3Cl)CC2)CC1 N1(c2nccc(=NCC3N(S(C)(=O)=O)CCCC3)[nH]2)CC2(CCCCC2)C1 CCC(C(=O)NCCC(=O)NCCc1ccccc1)N(C)C c1(C(N2CC(CC)N(C(C3CN4CCC3CC4)=O)CC2)=O)c(N)cc(Cl)cc1F C(=O)(CC(O)CC(C)(C)C)NCC#CCNC(c1c(C(C)C)occ1)=O CCC(C)CC(C)NC(=O)CN(C(=O)CC1CCC(C)(C)C1)C N1(C(C(CC)(F)F)=O)CCC2(CCC(NC(=O)CC=C(Cl)Cl)C2)CC1 c1(C=O)ccnn1C1CCCC1.C1(CC)CCN(C(=O)Cc2nc(=N)[nH][nH]2)C1.N CC1CNc2c(CNC(=O)C(=O)N3CC(N4CCCC4=O)C3)cnn2C1 C(=O)(CCC(C)OC)N1CC(OCC)(CNC(c2snnc2CC)=O)C1 Cc1ccc2cc(C(=O)NCC(C)NC(=O)C3=NOC4(CCC4)C3)[nH]c2c1 c1(CNCC2OCCN(C(C(C)(C)NC(C)=O)=O)C2)cc(F)c(O)cc1F N1(C(CCc2cccc(C)c2)=O)CCC(O)C(NC(c2cn[nH]c2)=O)C1 C1(CC(N2C(CNC(CCC(=O)NC)=O)CCC2)=O)CCn2cncc2C1 c1(C(N2C(CCN(C(=O)Cc3nc[nH]n3)C)CCCC2)=O)ccc([N+](=O)[O-])cc1 C1(CNC(c2c(CC)c[nH]n2)=O)CC(C)N(C(=O)Cc2nncn2C)C1 C1(NC(=O)NCC2CCCCC2)CC12CCc1ccccc12 C1(C(N2CC(C)(C)C2)=O)CC2CC2N1C(c1ccc(-c2ccccc2)nc1)=O C(=O)(CCCCCN(C)C(c1ccn(C)n1)=O)N1CCCC(C(C)C)C1 C12(C(=O)NC(CCCC)COC)CC(C)(CN1C(C1(N(C)C)CC1)=O)C2 C1(C(=O)NC2C(NC(CC(CC)C3CC3)=O)COC2)CC2(C1)CC(C)(C)C2 N1(C(C(CSC)C)=O)CCCC(C)(C(N2CCCC(CF)C2)=O)C1 c1(C(=O)NC(C)CN(C(=O)CC2CC2)C)cccn1Cc1ccccn1 N1(CC(=O)NC)CCC(C(N2CCCC(C(C)=O)C2)=O)(OC)CC1 N1(C(c2cn(CC)nc2)C(=O)NC)CCN(C)C(c2cc(F)cc(F)c2)C1 C1(NC(Cc2ccc(C)o2)=O)CCCCCC1NC(=O)Cn1nc(Cl)ccc1=O C1(CNC(C2CCN(C(c3cc(C)c(C)[nH]3)=O)CC2)=O)CCC(=O)NC1C CC(C)CCCC(=O)NCC(C(=O)NC1CCC(C(C)O)CC1)N(C)C N1(C(C(C)=C(CC)C)=O)CCN(CC2(NC(C3CCOC3C)=O)CC2)CC1 C1(C(C(C)C)O)CCN(C(c2cccc(CCF)c2)C(=O)O)CC1 C1(OC)CCC(C(N2CCC(CC(=O)N(C(C)C(F)F)C)CC2)=O)CC1 C(CCNC(=O)CCc1ccsc1)(C(=O)Nc1cccc(C(C)=O)c1)OC CCCCC(C(=O)N1CCCCCO1)NC(=O)C1=CC2C=CC(C1)C2 c1(NC(C(N2C(C=C)CC2)=O)=O)ccc2c(C)nn(C)c2c1 N1(C(C(n2cc(C)nc2)(C)C)=O)CC2CC(NC(=O)C(O)C(C)C)CC1C2 N1(C(C(C2CCOCC2)C)=O)CCOC(CNC(=O)C=Cc2ccccn2)C1 c1(CC)cccc(CC)c1C(=O)NC1(CNC(C2(C)CC2Br)=O)CCC1 C1(CC)CC(C)CCC1O.c1(C(C(=O)N)NC(CN(CC)CC)=O)cccnc1 c1(C(N(C)CC2N(C(C(C(C)C)SC)=O)CCC2)=O)cc(O)c2ccccc2c1 C=CC1CCCN1C(=O)CC(C)CNC(c1cnn(CC)c1)=O N1(C(C2(C)N(C(CCNC(COC)=O)=O)CCC2)=O)CC2CN(C)CC2C1 C1(NC(C(CC)CC2CCCC2)=O)CC2C1CCN2C(c1[nH]c(=N)ccc1C)=O C1(C#N)(C(=O)NCC2CC(NC(CCN(C(C)=O)C)=O)C2)CC12CCCC2 N1(C(C2N(C(C)(C)C)CC2)=O)CCC(C(=O)N)C12CC2.C1(CCO)CCCC1.C C1(C2N(C(=O)NC3C(COC)CC3)CC2)CCCCC1 n1(CC)cc(CC(=O)NC2CC(NC(C3CCCO3)=O)C2)c(C)n1 C1(NC(C=CC)=O)CC12CC(NC(c1ccc(OCC)cc1)=O)C2 C1(C(=O)NC(CCCC)CNC(=O)C(F)(F)COC)CCc2nc(C)cn2C1 C(=O)(CC1=CCOCC1)NC1C(NC(=O)C=CC2CCOC2)CC1 CC1CCN(C(=O)CCNC(N)=O)C(C(=O)NCc2nn(C)c(=O)o2)C1 CCCCC(CC)CC(=O)N(CC(O)CN(C(=O)C(=O)CCC(C)C)C)C CC(C)CC(CNC(c1ccc(C(C)F)cc1)=O)NC(C1CC(C)(O)C1)=O C1(C(=O)NC(C)C(CO)NC(=O)CCc2ccccc2F)CCC(=O)N(C)C1 Cc1cnc2n1CCCC2C(=O)NC1CCCCC1NC(C1CC(F)(F)C1)=O c1(-c2cc(C(=O)OC)no2)ccc(COC(c2cnc(=N)[nH]c2)=O)cc1 c1(C(=O)NCC2CCCC(NC(c3ccc(C)o3)=O)C2)cnc(Cl)cc1N Cc1cc(CC(=O)NCC(CNC(c2n[nH]c(C)c2Cl)=O)CO)c(C)s1 C(CCCCCNC(=O)CCC1CC(F)(F)C1)N(C(CC(C)C1CCCO1)=O)C N1(C(=O)CN2CCC2)CC2(C(=O)NCCn3cncn3)CC1CO2 C1(Nc2nc(C(C)C)nc(N3CCCC(C)(O)CC3)c2)CCCCC1S(C)(=O)=O Cc1[nH]c2ccccc2c1C1CCN(C(=N)NCc2ncc(C#N)cc2Br)C1 n1(CC(N2CC(C)OCC(C)(C)C2)=O)cnc2ccccc2c1=O Cc1nn(C)c(Cl)c1CC(N1CC(n2cc(CC3CCC3)nn2)(C(=O)O)C1)=O N1(C(C2(NC(C)C)CC2)=O)CCCC2(C1)CN(C(=O)C=C(Cl)Cl)CCO2 C1(NC(C2(C)CC(NC(Cc3n(C)nnc3)=O)C2)=O)CC2CCCC2C1 C(C(=O)N=c1cc(C)n(C2CC2)[nH]1)(C1CCOC1)NC(CSC)=O N1(C(CCNC(C(CC)N(C)C)=O)=O)CCC=C(F)C1 C1(NC(C2C(=C)C2)=O)CCOC2(CCN(C(c3cc(C4CC4)ccn3)=O)CC2)C1 CC1CN(C(=O)C(c2ccc(Cl)s2)=O)CCC1NC(=O)C(C1CCC(=O)N1)C n1(CC(=O)NCCCCN(C)C(C2CC23CC3(F)F)=O)cnc2ccccc12 c1(C(=O)NCCCC2N(C(C3CC(C#N)C3)=O)CCC2)cccc(Cl)c1F Cc1cc(C(C)C(=O)NCCNC(C2(C)CS(=O)(=O)C2)=O)c(C)o1 c1(C(=O)NC2CC(CNC(CCC#C)=O)C2(C)C)cc2ccncc2[nH]1 N1(CC(=O)N(CC(C)C)CC(=O)NCC(O)CO)CCSCC1 CC1CCCC(CC(N2CCC(Cn3nccn3)CC2)=O)C1 c1(CNC(C2N(C(c3c(OC)cnc(Br)c3)=O)CC2)=O)ccccc1[N+](=O)[O-] CC(C)(C)C(CNC(C1(F)CC=CC1)=O)C(=O)N1CCCC(C)(N(C)C)C1 c1(OC)ccnc(C(=O)NC2C3CC(NC(=O)C(C)C(C)(C)C)CC23)c1C C1(COC)CN(C(=O)C(C)=O)CCN1C(C1CC2CC1CN2)=O N1(C(C(OCC)OC)=O)CC2CC(NC(C3CN(CC(C)C)C3)=O)C1C2 c1(CN(C)C)ccnn1CC(=O)NCC(C1CCCCC1)(C)N n1(CC)nc(C(N2CCC(C)C2)=O)cc1O.C1(CC=O)(C(F)(F)F)CCC1.N C1(C=O)C2CC3C(C2)C13.c1(C=O)ncoc1C.C=C1CC(C)C1.C1CC1.N CCC(CC(=O)N1CCC(C)C(N(C(=O)CN2CC3CC3C2)C)C1)C(F)F N1(C(c2cnc(C)nc2)=O)C2CCC1C(C(=O)N(C)CCN(C)CCO)C2 n1(CC)ccnn1.C(C)C=O.C1(C(NC2CC2)=O)CCOC1.C(CO)OC Cc1cc(N2CCCC(CO)C2)ncc1S(=O)(=O)NC1CC(Cl)(Cl)C1 Cc1nc(C2CC2)[nH]c1C(N1CCN(C(C2(C)CC2F)=O)CC1)=O N1(C(C2C(=C)CC2)=O)CC23CCCC2(C1)CN(C(=O)C=CC(C)=O)C3 c1(CNC(C(=O)NCC2(C)CCC(=O)N2)=O)c[nH]c2ccc(C#N)cc12 c1(CNC(N(C2C(OC)COC2)C)=O)ccc(F)nc1Br C1(C(=O)NCCc2nccs2)COCCN(C(=O)CCc2ccc(O)cc2)C1 C(CC(F)F)(C(=O)N(CC)Cc1cccnc1)N(C(CCC=CCC=C)=O)C C(CC(C)C)NC(CCNC(=O)OCC)=O.S(S(C)(=O)=O)CC=O.N c1(C(N2CC(OCC)C(C)C2)=O)nn2c(c1C)CCCC2.C1(C=O)CCC1C.N C1(NC(CC(c2ccccc2F)C)=O)CCCN(c2ncnc(=N)[nH]2)C1 c1(C(C(=O)NCCCN(C(=O)Cc2occc2C)CC)O)cccc(C)c1 C1(c2ccccc2)(C(=O)OC)CNN(Cc2ccccc2)CC1.c12cc(on1)C2 C1(CC(=O)NC(CNC(COCC)=O)(C)C(C)C)CCC(F)(F)CO1 c1(C(=O)OCC)[nH]c(C)c(CN2CCOCCC2)c1C.C(CC(=O)O)C(=O)O.C C1(CNC(C(C)(C)F)=O)(C)CC(F)(F)C1.C(=O)CCCCN1CCOCC1.N C(=O)(C(C)(C)CS(C)(=O)=O)N.c1(OC)cc(C(=O)NC2(C)CC2)sn1 Cc1nccc(CCNC(=O)CC2CCCO2)n1.C12(C(=O)N)CC(F)(C1)C2 C1(C)(SCC)CN2CCC1CC2.N12CC(CC(=O)N)(C1)N(C)CC=CC2=O C1(CO)CCC(N=c2[nH]c(-c3cccnc3OC(F)F)cs2)CC1 Cc1cc(N)cnc1C(=O)NCC(c1ccccc1)CNC(=O)C.CC(F)F.O C1(CC(=O)NCCC2CN(C(C3(C)CCCOC3)=O)C2)CCc2sccc2C1=O N1(C(C(CCC)NC(C)=O)=O)CC(CC(=O)N(C)CC)C2(CC2)C1 c1(C(=O)NCC=CCNC(C2CCOC2)=O)csc2nnsc12 C1(C(=O)NC2CCOCC2OC)(CC)CCCN1C(C1CC(=O)C1)=O c1(C(CN2CCN(C(C)=O)CC2C)O)ccc2ccccc2c1 c1(C(N2C(C)(CC(=O)N(C)Cc3snc(C)n3)CC2)=O)ncccc1O C1(NC(C(C)OCC#C)=O)CCCCC1.c1(C=O)ccccc1C(C)(F)F.N Cc1nn(C)c2sc(C(=O)N(C3CCCCN(C(C45CC(O)C4C5)=O)C3)C)cc12 [SH](=O)(=O)c1ccsc1C(N1CCC(O)C1)=O.C1(C=O)CN(C(C)=O)C1.CN C1(C(=O)NCC2N(C(C(c3ccn(C)n3)C)=O)CCC2)CCCCC1CF C(=O)(C1Cc2ccc(F)cc21)NC(CCN(C(CCOC)=O)C)C N1(C(CC(C(F)(F)F)OC)=O)CCC2(CCN(C(c3cnn(C(C)C)n3)=O)C2)C1 C=C(C)C(C)(C)C(=O)NC1CC(CNC(c2cc(O)nc(Br)c2)=O)C1 N1(C2CN(C(CCc3n(C)ccc3)=O)C2)CCN(C(=O)CC2CCCCC2)CC1 C(=O)(CCC=O)N(C(C)C)C.C1(O)(CC)CN(C(c2ccc(C(N)=O)s2)=O)C1 C(CC1CCCCC1)(C(=O)NC1COCC1NC(=O)Cc1nonc1C)OC N1(C(CCN2CCN(C)CC2)=O)CC(N(C)C(C2CCC(C)(C)O2)=O)C2(CC2)C1 N1(C(C=CCCC=C(C)C)=O)CCC(CNC(c2cc(Cl)no2)=O)C12CCC2 c1(OC)cc(C(N2CCC(O)(C(C)NC(=O)CC(C)SC)C2)=O)cc(Cl)c1 C1(NC(CC2C(C)(C)C2)=O)CCOC12CCN(c1cc(O)ncn1)CC2 c1(C(=O)NC(CC)(C)CNC(C2(F)CCC2)=O)ccc(C)c(N)c1 c1(C(=O)NC2CC(NC(C(CC)c3cccnc3)=O)C2)cc(C)ccc1N C(=O)(C1CCc2ccccc21)O.N1(C(c2cn(C)nc2)=O)CCC2(CC1)CC2 c1(C(=O)NCC2C(OCC)CN(C(=O)C(C)C)C2)nc(C2CC2)ncc1Br C(=O)(C1CCCCn2ccnc21)NC1CC(C(C)C)OCC1 c1(SCC)ccc(NC(=O)C(=O)N(CC(C)C)C)cc1.C(=O)C.C1CC1 Cc1cccc(C)c1.N1(CC(=O)N(CCN(C(C)=O)C)C)CCP(C)(=O)CC1.O c1(OC)nccc(CCCNC(N2CC(C)CC2c2ccc(OC)cc2)=O)n1 C1(NC(c2cc(O)ccc2F)=O)CCC2(CC1)CN(C(c1cc(Cl)ccn1)=O)C2 N1(C(c2occ(C)c2C)=O)CCC2CCCC12CNC(=O)CCN1CCCC1=O c1(C(N2C(CCCNC(C3(C)CC=CC3)=O)CCC2)=O)cc2n(n1)CCOC2 CC1C(NC(c2cnc(C(C)(C)C)s2)=O)CCCN1C(C1CC(C)(C)CN1C)=O C1(NC(C2CC(OCC)C2)=O)(C)CC2CCC1CC2.C(=O)CCC1CCC1 N1(C(C(c2cccnc2)=O)=O)CCN(C(c2csc(O)n2)=O)CC2CCCCC12 Cc1cc(C(N2CC3CC(NC(c4nc(=O)n(C)[nH]4)=O)C3C2)=O)cc(C)c1 n1(CC)ccnc1C(N1CCC(C(=O)NC(CO)CCSC)C1)=O C1(C)(NC(CNC(CCNC(C)=O)=O)=O)CCCC1.C(C)(C)C.C=O.N c1(C=O)coc(S(N)(=O)=O)c1.CCC(=O)N(CCC)C(C)C.C(C=O)OC n1(CC(=O)NCC(C)(C2CC2)NC(CN(C)CC)=O)[nH]cnc1=N C1(OC)CN(C(=O)CCC=CC(C)C)CC1C(=O)NCCCN1CCCC1 c1(CN2CCN(C(c3cc(F)ccc3C(F)F)=O)CC2)cn2cc(Br)ccc2n1 C1(NC(C(CCN(C)C)NC(C2CCS2(=O)=O)=O)=O)CC(F)(F)C1(C)C CC(C)CC(CNC(c1cnn(C)c1Cl)=O)C(=O)NC1(C)CCOC1 c1(N(CCCNC(c2cncc(Cl)c2)=O)CC)ccc2c(n1)CC(C)(C)CC2=O C(C)(CC1=CCCCC1)NC(CC1C(NC(CCCCC#C)=O)CCC1)=O C1(OC)CC2(CCN(C(=O)C(C)CNC(=O)C(F)F)C2)C1 c1(C=O)cc2n(n1)CCCNC2=O.O=C(CCCC1CC1)NCC1(C)CC1.N C1(C(=O)NCC(C)NC(C2CCC2C)=O)(CC)Cc2ccccc2C1 N1(C(C=CC(CC)C)=O)CC2CC1CN2C(=O)CC1CC2(CCO1)CC2 c1(OC)cc2c(C(=O)N)c[nH]c2cc1Cl.C1CN(C(=O)C(=O)N(C)C)C2CC12.C c1(CNC(C2C(CC)CN(C(C3CCCSC3C)=O)C2)=O)c(F)cncc1F C(=O)(C1CCCc2c1ccn2C)N1CC(O)(CCOC)C1 N1(C(CC(=C)Br)=O)CC(CNC(c2cnn(CCC)c2)=O)CC1C C12(C(N3CC=CC(NC(CCC(=C)Br)=O)C3)=O)CCC(C1)S(=O)(=O)CC2 c1(NC)nc(C)ccc1C(=O)NC1CN(C(=O)C(O)COC)CC1(C)C c1(C(=O)OC)cc(Br)c(OC)cc1NC(C1(OC)CCSCC1)=O N1(C(c2c(OC)n[nH]c2)=O)CCC(C2CC2)(NC(=O)CCc2cncc(C)c2)C1 CC1CN(C(=O)C(N)=O)CCN1C(C1C2CCC1(c1cccs1)C2)=O c1(SC)ncc(Br)c(=NCC(CC(C)C)NC(C2C3CC4CC(C3)CC2C4)=O)[nH]1 c1(CC)cnn(CC(=O)NCCCC(=O)NC(c2ccncn2)C)c1 c1cc2cc(N)ccc2[nH]1.C1(N(C)C)CCCCCC1NC(=O)OC.C(C)(C)C c1(OC(C)C(N2CCN(C(c3ccon3)=O)C(CCO)C2)=O)ccc(C#N)cc1 C(CCCC(=O)N1C2CCC1(CNC(=O)CC(C)CF)CC2)(OC)OC Cc1[nH]c2ccc(F)cc2c1C(=O)NC1CCN(C(=O)Cc2cnnn2C)CC1 N1(C(C2(C=O)C=CCC2)=O)C2CCC1CC2.C(C)(C(C)(C)C)=CC=O.C c1(C(=O)NCC23C(CN(C(CCC(=O)N(C)C)=O)C2)C3)ccc(F)c(F)c1F C(=O)(C1Cc2c(Cl)cccc21)N(C1CCCN(Cc2cccc(C#N)n2)CC1)C Cc1cc(C(=O)N(CCNC(C2CCOC2C)=O)Cc2ccccc2)cnc1F CC(N=c1[nH]c(N(CC(F)F)C)nc2ncn(C)c12)c1cccc(F)c1F C#CC1(C(N2CC3CC2CN3C(=O)CCCn2cncn2)=O)CCCCC1 C(=O)(CCC(CC)CC)NCC1N(C(C=CC=CCCCCC)=O)CCOC1 N1(C(C2(COC)COC2)=O)CC2CCCC2C1.c1(C2(C(=O)N)CC2)cc[nH]n1 C1(NC(c2cc(C)cc(C)n2)=O)CC2CC(C1)N(C(C1CCCN1C=O)=O)C2 C1(CCCNC(COCCC=C)=O)CCCCN1C(=O)CSC.c1cscn1 C12(NC(c3c(=N)cc[nH]c3)=O)CCOCC1CN(C(=O)CC1CC=CC1)C2 c1(C(C(N2CC(NC(c3ncc(C)s3)=O)C3C2C3)=O)=O)ccc(Cl)cc1O CC(CC(N)=O)N(C(=O)CC1(N(C(=O)CN(C)CCO)C)CC1)C C1(CC)CC(CC(=O)NCC2CCCN2C(=O)C=C2CCC(C)CC2)CCO1 Cc1ncc(Br)c(=NC(=O)c2nc(NS(=O)(=O)C(C)C)cn2C)[nH]1 c1(CCC)cc(=NC(C)CN(C)C(C)=O)[nH]c(Cc2cccc(Cl)c2)n1 C1(OC)CN(C(=O)CCOc2cccnc2)CC1N.C1CN(C(=O)COC)C1 c1(C(N2C3CN(C(CSCC)=O)C(CC3)C2)=O)ccc2cc(Br)ccc2n1 C(C1=CCN(C)CC1)NC(CCC1CCCN(C(c2ccc(SC)o2)=O)C1)=O Cc1cc(=NCCC2CCSC2)[nH]c(=NCCOCC2CC2)[nH]1 C(=O)(C(C)C(C)(C)C)N(CC(C)C(=O)NCc1cccc(C#N)c1)C C1(C2CCN(C(C(c3cccnc3)C)=O)C2)CCCCN1C(=O)CN(C)CCO Cc1nc(C)n(O)c1C(N1CCC(O)(CNC(C2CC2CF)=O)C1)=O C1(C(N2C3(CNC(c4cc(C)n(C)n4)=O)CCC2CC3)=O)CCc2ncnn2C1 C1(C(N(C)Cc2n(CC)ccn2)=O)CC2CCC1N2C(=O)CN(C)C(C)C C1(C)(NC(=O)NCC(n2cccn2)C)CN(C(C2CNC(=O)C2)=O)C1 c1(C(N(C2CC(C(=O)NC(C3(CO)CC3)C)C2)C)=O)cccc[n+]1[O-] C1(C(=O)NC(C)CC#N)CC=CCN1C(c1ccncc1Cl)=O C1(C(C)NC(Cc2scc(C)c2)=O)CCCN(C(=O)Cn2cnc(C#N)n2)C1 C1(NC(C2(CCNC(CC(CC)C)=O)CCC2)=O)CC2(CCC2)C1O Cc1cn2c(C)c(COC(C3(c4cc(F)cc(Br)c4)CC3)=O)nc2s1 C1(NC(=O)NCCn2cc(Br)ccc2=O)C2Cc3ccccc3C12 C(=O)(C(C)(C)CCc1ccccc1)NCC1=CCCN(C)C1.C12CCCC1NC2 C=C(C)CN=C(NCC1(N(C)C)CCOCC1)N(C)CC1(OCC)CCOC1 Cc1nc(=N)[nH]cc1C(C)NCC1CCCC(c2ccccc2)O1 C(=O)(CCCCCCNCc1nn(C)c(C)c1I)OCC C1(CNC(C(C=C)(C)C)=O)CCC(C)N(C(c2coc(CCO)n2)=O)C1.C N1(C(CCOCC)=O)CCC(NC(C2CN(C(C)=O)C2)=O)C12CCC2 C(=O)(C1CCCc2nc[nH]c21)N1CCC(C)C1CNC(=O)CC1CC(C)(C)CO1 C=CCCCC(C(=O)NC1CN(C(=O)C2CC2)C1)NC(C1CN(C)CCO1)=O c1(C(=O)NC(C2CCCN(C(CSCCC)=O)C2)C)ccc(F)c2c1OCC2 c1(N2CCC(C3N(C(CS(CC)=O)=O)CCCC3)C2)ccc([N+](=O)[O-])cc1 C(CN=C(NCc1ccoc1)NC1CC(O)C12CCC2)c1ccc(OC)cc1 c1(COC)cc(C(N2CC(CNC(C3CC3C)=O)(OC)C2)=O)n(C)c1 N1(C(c2c(COC)onc2)=O)CCN(C(c2nn[nH]c2Cl)=O)CC12CCC2 C1(NC(C2(CC)CC2)=O)CC2CN(C(C3CCCCCCC3)=O)CC2C1 CC(=O)CCN=C(NCc1cccc(C(C)(C)C)n1)NCC1CCCN1C(C)C C(CC1=CCN(C(=O)C(C)SC)CC1)NC(Cc1ccc(OC)cc1)=O N#Cc1nnc2ccccc2c1N1CCN(C(=O)CNC(c2cccs2)=O)CC1 C(=O)(CS(=O)CCC(F)(F)F)N1CCC2CN(C(c3cnc4sccn34)=O)CC21 N1(C(Cc2c(C)nc(S)s2)=O)CC2(CCN(C(C3CCC4CC4CC3)=O)CC2)C1 C1(NC(c2cnc(C)nc2O)=O)C2CCCN(C(c3cnccn3)=O)C2C1(C)C C#CC1CCCN(C(c2cc(OC(F)F)ccc2F)C(=O)NC)C1 Cc1sc(C(=O)NC(C)(CNC(=O)CCc2ccn(C)n2)C2CC2)nc1O c1(C(N2CCCC(NC(c3ccns3)=O)CC2)=O)c(Br)nc2n1CCOC2 CC(C)CCCCC(=O)N1CCC=CC1C(N1CC(N(C)CCO)C1)=O c1(C(=O)NC(C)CCNC(=O)CCCn2cncn2)ccc(Cl)cc1F C(=O)(CCC(C(=O)O)NC(=O)C(c1sncc1Br)N(C)Cc1cscn1)OC c1(N2CCC(NC(c3cccc4nonc34)=O)(CF)C2)nc(Cl)nc2c1CCC2 CCCCCCC(C)C(=O)N1CCN(C(C2(CCC)CC2)=O)CC1CC N1(C(C(=O)NCCCOCC)C)CCC(C)C1.N1(C(C(=O)N)C)CCOCC1 S(=O)(=O)(c1ccc(C#N)cc1)NC(C(=O)Nc1ccc(OC)cc1)C(C)O.O C1(NC(Cn2c(C)nnn2)=O)C2CC3C(C2)C13C(=O)N(C(C)C(C)SC)C N1(C(C2(CC)COC2)=O)CCC2(NC(=O)Cn3ccccc3=O)CC2C1 N1(C(C2CCN(C(C3(C)CCCCCC3)=O)C2)=O)CC(C2=NOCC2)C1 c1(C=O)nccc2cc[nH]c12.c1(OCC(=O)NC2CC2C)cc(F)ccc1F.N c1(C(N2C(C(C)(C)NC(=O)CSS(C)(=O)=O)CCC2)=O)cn2ccncc2n1 Cc1ccc(CN(C(C)C(C)N(C)C)C(=O)Cn2cc(CCCCO)nn2)o1 c1(CC)nc(C(N2CSCC2C(=O)NC2CCCOC2)=O)c(C)o1 Cc1nn(CC(F)F)cc1C=O.C(CCN(C(=O)C)C)C(C)C.C(C)(C)C.N CC(CC(F)(F)F)C(=O)NCC(C)Nc1ncnc2ccsc12 CC(CC(F)(F)F)C(=O)NCC1N(C(c2nocc2Cl)=O)CCCC1(C)C CC1(NC(=O)COCC2CCC2)CN(C(C23CC2C3)=O)C1 C(=O)(C1CCCc2ccccc21)NC12CCC(CN(C(c3c(C)c[nH]n3)=O)C1)C2 Cc1ccc(F)c(C(=O)N(CCC(C(C)C)NC(c2cn(C)ccc2=O)=O)C)c1 C1(C(N(CC(C)N(C(CCOc2c(C)cccc2)=O)C)C)=O)CCCC(C)(C)O1 c1cscc1Cl.N1(CCCN(CC(=O)OCC(=O)N(CC)C)CC)CCCC1 C1(N)CC2(CCC2)C1.O=C(CNC(c1ccccc1)=O)CCC1CCCCO1 C1(CCCNC(C2C(C)(C)C2)=O)CCN(C(C2(O)CCOC2)=O)CC1 N1(C(C2CC2c2ccccc2)=O)CCC(C2CCCN2)CC1 Cc1cc(O)ccc1N(C)C(C1CCCC(NC(=O)C(O)CN(C)C)CC1)=O C(CN=C(NCC(C(C)C)OC)NC1CCOCC1)(c1ccc(Cl)cc1)OC Cc1cc(F)ncc1C(=O)NC.C1(CC=O)CCCCC1.C1CN(C(=O)C)C1 C1C(C)CCCN1C(C1CN(C(N)=O)C1)=O.Cc1noc(Cl)c1CC(=O)NC C(=O)(C#CC1CCCO1)N1CCC(N(C(Cc2ccc(OC)cn2)=O)CCO)CC1 N1(C(C(c2cccc(F)c2)(C)C)=O)CCN(C(=O)Cc2ccsc2)CC(CO)C1 C(C1CCN(C(=O)Cn2ncnn2)CC1)=CC(=O)NC(c1nn[nH]n1)CC N1(C(CC(C)N(C)C)=O)CC2CC(C(=O)NCC3CCC=CCC3)C(C2)C1 CC1CC(CNC(C2CC2C)=O)CCN1C(C12CCC(F)(CC1)C2)=O CCC(C)N(OC)C(=O)CC1CC(NC(c2sccc2C)=O)C1 C1(N(C(C(N2CSCSC2)C)=O)c2ncc[nH]2)CC2(CNC2)C1 c1(C(=O)OC)ccc(Br)c2c1CN(C(C)C)CC2.c12ccc(cc1)S(=O)(=O)N2 N1(C(Cc2c(C)occ2)=O)CC2CCN(C(c3cnoc3C3CC3)=O)CC(C2)C1 N1(C(CCN(C)C)=O)CC2CCCC(C1)C2C(=O)NCc1ccncc1O c1(NC(=O)NCCCn2ccnc2O)cccc(S(=O)(=O)N2CCCCC2)c1 C(=O)(CC(C)CC(F)(F)F)N1CCCCCC(NC(COCCC)=O)C1 c1(C(C)=O)cncc(C(=O)NCC2CCN(C(=O)CCc3c(C)noc3Cl)C2)c1 C1(NC(Cc2cn(C)nc2Cl)=O)CC2CC(C1)N(C(c1cc[nH]c(=N)c1)=O)C2 CN=c1[nH]ccc(C(N2CCC(NC(C34CC(C)(C3)OC4C)=O)C(F)C2)=O)c1N c1(C(=O)NC(C2CCN(C(C(COC)(C)C)=O)CC2)C)cncc(F)c1C c1(-c2c(OC)cccc2F)cn2cnc(C(N3CCOC(O)C3)=O)c2s1 CC(CCCCNC(=O)CCc1nc[nH]n1)NC(=O)CC1CCCCC1C c1(C(c2n(C(CC)C)nnn2)NCCCC(=O)NC)nc(Br)c(C)cc1Cl N1(CC(C(=O)NC(C)=O)C)CCCC(CCc2ccc(CCS)cc2)C1 C(C(C)(C)C(C)(F)F)NC(C(CCOC)NC(CCSCCC)=O)=O C=C(C)CN=C(NCC1CCN1C(C)(C)C)NN1CC(C)OCC1 N1(C(CCSC)=O)CC(O)CCC1C(=O)NC1CC(CCF)C1 C=C=CCCC(=O)N1CC(C)(OCC(N2CCCC(C(C)O)C2)=O)C1 N1(C(C(CC)(C)O)=O)CCC(C(=O)NCCN(C(C)C)C2CC2)C(O)C1 c12nnc(n1C)C(C)OCCN2CC#C.S(C)(=O)(=O)NCC(=C)C C(c1ncc[nH]1)=CC(=O)NC1CC1NC(c1ccc(SC(F)(F)F)o1)=O c1(OCC)c(C)cc(NCC2(C)C=CCN2C(=O)O)cc1C.C(C)(C)C C(=O)(CC(C)C(=O)N1CCCCC1C(N1CCOCCC1C)=O)OC Cc1nnn(CC(=O)NCC2CCC(NC(C3(C(F)F)CCCO3)=O)C2)n1 N1(C(CCOCC)=O)CC2(CCC(N3CCC4(CC3)CC(F)C4)CC2)C1 Cn1ncc(Cl)c1CC(=O)NC1CC(NC(=O)CCC2(C)CC2(F)F)CC1O Cc1cc(C)nc(N2CCCC(C(=O)NCC)C2)n1.c1(C(=O)N)nc(O)c(C)s1 CC(CS(C)(=O)=O)C(=O)N.C1(CC(N)=O)CCN(C(C2(O)CC2(C)C)=O)CC1 Cc1cc(C)c(C(N2CCC(C)C2)=O)c(C)c1.c1(CC(=O)N)cc(O)nc(O)n1 c1c[nH]c2nc(Cl)ccc12.c1(NC(C)=O)ccc(NC(=O)CC2CN(C)C2)cn1 N1(C2CN(C(C(C)=C3CCC3)=O)C2)CC(NC(C2CCS2(=O)=O)=O)CC1=O C1(C)(CNC(CC)=O)CN(C(=O)CNc2cnn(C)c2)C(C)(C)C1 N1(C(C(S(CCC)(=O)=O)C)=O)CCCC12CCCN(C(c1sccc1C#N)=O)C2 N1(C(c2c(CC)nns2)=O)CC2CC(NC(c3nc(O)[nH]c(=O)n3)=O)CC2C1 N1(C(CN(C)C)=O)CCC2(CC1)CCN(C(c1ccc(-c3cccs3)cc1)=O)C2 CC1=C(C(=O)NC(C)CN(C)C(c2nc(C)ccc2O)=O)CCCC1 C#CC1(C(=O)NC2CCC(C#N)CC2)CCN(C(c2ccncc2)=O)C1 CCCCC(F)C(=O)N1CC(C2CC2C(=O)Nc2cnc(OCC)nc2)C1 Cc1nnc(CN2CC(CC)C2)s1.C(=O)(CN(S(C)(=O)=O)C(C)C)N CC(C)CC(C)CC(=O)N1CCC1CNC(C1C2CC(=O)CC12)=O c1(C(=O)NC(C2CN(C(C(CCC)N(C)C)=O)C2)C)ccc(Cl)c(C(=O)O)c1 N1(C(C(C)n2ccnn2)=O)CCC2C1CCN2C(c1cc2ccoc2cn1)=O Cc1nn(C(C)C)cc1C(N1CCCC1)=O.c1(C(=O)N)cnn(C2CC2(F)F)c1 Cc1c(C(=O)NC2CC2C)oc2c(C)cccc12.c1(CC=O)csc(Br)c1.N CC(Cn1cccn1)N=c1nc(-c2ccccc2)[nH]c(=NC2CCCN(C)CC2)[nH]1 C1CCCN(C(c2[nH]nc(C(F)(F)F)c2C(C)C)=O)C1.CC(CC(=O)N)C1CC1 C1(NC(Cc2nc(C)c(C)s2)=O)COC2(C1)CN(C(=O)Cc1cccnc1Cl)C2 C1(C#N)(C(N2CC(CC(C)NC(C(C)=C3CC3)=O)C2)=O)CC1C CC(C)CC(CNC(C1CCCC1NC(c1cscc1Cl)=O)=O)CO C(=O)(C#CC1CCOC1)NCC1N(C(=O)CC2CCOCC2)CCN(C)C1 C(O)(C(F)(F)F)C1(C(N(CCCNC(COCCC)=O)C)=O)CCC1 Cc1cc(C(N2CC(O)CC2C)=O)nn1C(C)C.C(=O)(CC(C)c1ccco1)N Cc1cc(NC(C2CN(Cc3cccn4ccnc34)CCS2)=O)cc(C)c1C n1(CC=O)cc(S(N)(=O)=O)cn1.C1(CC=O)CCC2(CC1)CC2.CCC.CN c1(C(C)C)ccccc1C(=O)NCC(C)N(C(=O)Cn1ncccc1=O)C N1(C(C(=O)NC(CC)C)C2CCCC2)CCN(C)C(c2ccccc2)C1 CCCCC(C(=O)NC1CCN(C(=O)C(c2nc(C)cs2)C)CC1O)NC(N)=O c1(C(=O)N)ccnn1C.c1(CCNC(C=C(C)C)=O)cc(C)no1.C(N)=O CCCCCCCCC(=O)NCCC1(Nc2cc(Cl)c(O)nn2)CCC1 c1(C=O)ccc(C(F)(F)F)c(C)c1.C1(C(=O)NC(C)CCC)(OC)CCCC1 c1(C(=O)NCC2(O)CN(C(COC(C)=O)=O)C2)cn(C)c(=O)cc1C C(=O)(C(O)CC(F)F)NCC1C(NC(c2sc(CC)c(C)c2)=O)CCCC1 c1(C(N2CC(CC(=O)NC3CC=C(C)CC3)OCC2)=O)cnc(C)cc1C C1(C(=O)NCC2(C)CC(C)C2)CN(C(=O)C(c2ccn(C)n2)C)CC12CCC2 N1(C(C(N2CC(C)CC(C(=O)OC)C2)=O)=O)CCC=Cc2ccccc21 N1(Cc2cc(OC)ncc2Br)CCC2CN(C(=O)C=Cc3ccc(Br)cc3)CC12 CC1COCCN1C(=O)CC1(C)CCN1C(=O)CSc1ccccn1 C(CCCCC(=O)NC1CC2(C1)CC(NC(=O)CCSCC(C)C)C2)=CC N1(C(c2ccc(C(C)=O)[nH]2)=O)CC(C(=O)N(C)CCC2CCCCC2)C(C)(C)C1 n1(CC#C)cnnc1C(N1CCC1(C)CC(=O)N(C)C(c1cnn(C)c1)C)=O O=C(C1=NN(c2ccc(Cl)cc2)C(=O)CC1)N1CC2(CCC(O)CC2)C1 C1(NC(CC2OCC(C)(C)C2)=O)CCSC12CN(C(=O)Cn1nccn1)C2 c1(C(CO)NC(CC(C)SC)=O)ccc(Br)c(F)c1 N1(C(CCCOC)=O)CCCC12CCN(C(c1cc3scc(Cl)c3[nH]1)=O)CC2 CC1(C#CC(=O)NCC2CN(C(=O)CSCc3cccs3)CCO2)CCCO1 N1(C(CC(=O)OC)=O)CCC(C(=O)Nc2ccccc2N(C)C)(CF)C1 N1(C(C2CC(CC=O)C2)=O)CC(N(C)C(c2cnc(O)n2C)=O)C(O)C1.CO S(=O)(=O)(c1ccc(NC2CCN3CCCC3C2)c(Br)c1)NCCCN(C(C)C)C C=CC1(C(N2CC(C)C(C(F)(F)F)C2)=O)CCOCC1.S(C(F)(F)F)CC=O C(=O)(CC(C(C)CC)NC(C1CC1C(C)C)=O)N(CC#C)C(C)C C1(OC)Cc2ccc(S(=O)(=O)NCC3CCN(C4CCCCC4)CC3)cc2C1 N1(C(CNC(c2ccc(C)s2)=O)=O)CC2CCC2(NC(C2CC(CF)C2)=O)C1 CCCCC(CC)CCC(CNC1CCCC(CC)C1)CC Cc1noc(C)c1C(=O)NC12CC1CN(C(c1coc(-c3ccccn3)n1)=O)C2 c1(OCC(=O)NC2CN(C(C)=O)CC2C)ccc(Br)c(C)c1 N1(C(C2CC(CC)C2)=O)CC(C)CCC1CNC(=O)CCc1ccsc1 c1(C(=O)NC(C)C(CO)NC(c2ccc(Cl)nc2N)=O)cncc2nc[nH]c12 c1(OC)cccc(NC(C2CC2NC(c2ccc(Cl)s2)=O)=O)c1C#N C=CCC(CNC(c1cc(O)n(C)n1)=O)C(=O)N1CCC(c2ncc[nH]2)C1 C1(C(N2CCC(OC)C2)=O)N(C(=O)Cc2ccc[nH]2)CC12CCCC2 N1(C(C(C(C)O)N(C)C)=O)CC2(CCN(C(c3cc(N)ccc3Cl)=O)CC2)C1 N1(C(c2nnc(C)o2)C)CC=C(CNC(c2ccc(F)cn2)=O)CC1 c1(CNC(CCOC)=O)ccc(CC)cc1.C(=O)(C=CC(=O)N(C)C)N CC(C)C(C(=O)NCC(C)NC(C1CCC(=O)NC1)=O)NS(C)(=O)=O c1(C(N2CC(N(C(C3(CCOC)CCCC3)=O)C)C2)=O)cc(F)c(Cl)cc1F Cc1cn(C)nc1NCC(C)NC(=O)C(F)CNC(=O)OC(C)(C)C C1(S(=O)(=O)N(C)C)(C=O)CCC1.c12cnn(c1)CCNC2=O.C(C)(C)C C(=O)(n1cccc1CS(C)(=O)=O)N1CCC(C(N(CC(F)(F)F)C)=O)CC1 Cc1c(-c2c[nH]c(=NCC3CCCC3)s2)cccc1C#N.c1cc(C)nn1C(C)C C(=O)(C(CC(C)(C)C)OC)NCC(CC=C)C(=O)NCc1c(C)nn(C)c1C C(CC(C)(C)C(=O)NC1CCN(C(=O)CC(F)(F)F)C1Cc1ccccc1)SC C=CC(CCC)CC(=O)NC(CC1CCC1)C(=O)N1CCC(c2nc[nH]n2)C1 c1(NC(CN(C2CCCCC2)C(C2C(C)C2C)=O)=O)cnn(CCO)c1 c1(C(=O)NC2CC(NC(C3(n4cncn4)CC3)=O)C2)[nH]nc([N+](=O)[O-])c1Cl N1(CCNC(c2ccnc(CC(C)C)n2)=O)CCCN(C(C2(F)CCC2)=O)CC1 C(C(=O)NC1CCN(C(=O)COc2ccccc2F)CC1O)(C(C)(C)C)SC C1(O)(CC)CCN(C(c2ccc(Cl)cc2F)=O)CC1.C1(CC(=O)N)COC(=O)C1 C1(NC(C(C(C)C)O)=O)CCCC12CCN(C(C1C3C=CSC13)=O)CC2 C1(NC(C(C)(F)F)=O)CCC(F)(CNC(c2coc(C3CCC3)n2)=O)C1 c1(C(=O)OC)cccc(NC(c2[nH]nnc2C)c2nnnn2C2CCOC2)c1C C1(NC(c2cc(Br)c[nH]2)=O)CN(C(C2CCC(F)(F)C2)=O)CC2(CCC2)C1 Cc1nc(C)c(CNC(=O)CC2(C)CCN2C(c2cn(C)c(C)n2)=O)o1 C12(C(=O)NC3CN(C(=O)CCn4cnnn4)CC3C)COCC(C1)OC2.C1CC1 Cc1nc2c([nH]1)CC(C(=O)NC1CCC(NC(c3nc(=N)cc[nH]3)=O)CC1)CC2 C#Cc1cn(C)nc1C(=O)NC(C(=O)N(C(C)C(C)C)C1CC1)C(C)C c1(SC(COC(c2cc(C(CC)=O)c(F)cc2)=O)C)ccc2c(c1)OCCO2 C1(NC(c2occ(C)c2)=O)CC(NC(C2CCC3(CCC3)O2)=O)C12CCC2 C(=O)CCC(=O)N1CCOCC1.CC(C)C1CC1.C1(C(=O)N)CC1C(F)(F)F N1(C(c2cc(C)sc2C)=O)CC(C)CN(C(c2cc3cccn3cn2)=O)CC1C C1(C)(NC(CC2C3CN(C(C(c4cncnc4)C)=O)CC32)=O)CCCC1(C)C C1(NC(c2cc(Cl)ccc2F)=O)CC2(C1)CC(NC(=O)C1CC1)C2 C1(CNCc2cccc(OC#N)c2)CCCc2ccccc2C1 C(=O)(CC(CC(C)C)NC(=O)CC1CCCN(C)C1)N(CC)CC1CCCO1 c1(-c2n(Cc3onc(CC)n3)ccn2)ccc(-c2ccc(=N)[nH]c2)cc1 C1(C)(NC(C(c2ccc(Br)s2)C)=O)CC(NC(c2ccccc2)=O)C1 CC1CN(C(c2nccc3cc[nH]c23)=O)CCCN1C(C1C(C)(C)C1(F)F)=O C(CC)(C(C)C)NC(COCCCCC)=O.c1(C(C(=O)N)(F)F)ccc(F)cn1 c1(C(=O)NC2CCN(C(c3cnc(CCC)s3)=O)CC2F)cc2n(n1)CCCC2 Cc1ccc(Cl)c(F)c1C(=O)NCC1CC2CC2N1C(=O)C(c1ccccc1)C N1(C(CSCC)=O)CCCCC1C(=O)NCCNC(C(CSC)C)=O Cc1ccc(C(N2CCCC(CCNC(=O)CO)C2)=O)c(Cl)c1C.CC(C)(C)C CCS(=O)(=O)CCn1nc(-c2cnn(CCO)c2)nc1-c1cc(F)n[nH]1 c1(CCC)c(C(N2CCCN(C(=O)CCF)CC2)=O)[nH]c(C)c1C(C)=O C12(C(N3CC(O)(CNC(C(CC)n4ccnc4)=O)C3)=O)CCCCC1NC(=O)C2 N1(C(CCCOCC)=O)CC(C(=O)NC(c2ccc(C)cn2)C)C(F)C1 C=C(C)C(CC(=O)NC(C)CNC(=O)C(C1CCOCC1)O)OCC c1(C(N2CCCC(O)C2)=O)n[nH]cc1N=c1ccn2ncc(Br)c2[nH]1 C12(C(=O)O)CCC(F)(F)CC1CN(C(c1ncc[nH]1)=O)C2 C(=O)(CCCCC(=O)N1CC=CC1CNC(c1cc(-c2ccoc2)[nH]n1)=O)NC C1(CCNC(CC=C)=O)CCN(C(=O)C(F)(F)CN(C)C)CC1(F)F c1(CCC(=O)NCC=CCNC(C2C(C)(Br)C2)=O)cnc2ccccc2c1 c1(OC)ccc(Br)nc1C(N1CCOC(C#N)C1)C(=O)NCCC1CC1 c1(N(C)C)cnnc(C(=O)NC2CCCC2CNC(=O)CN2CCCCCC2)c1 C1(CC)CN(C(=O)C(c2ccc(CC(C)C)cc2)C)CCN1C(=O)C(C)C1CC1 c1(C(C)C)nccc(C(=O)NCCN(C)C(C2(CCO)CC2)=O)n1 C1(O)(CN(C)C(C2CC(F)C2)=O)CCN(C(C2(Cl)CC2(C)C)=O)CC1 n1(CC)cc(C(=O)NC2(C)CC(C(N3CC=CC3COC)=O)C2)c(C)n1 C1(C(C)NC(C(C)C)=O)COCCN1C(=O)CC1CN(C(c2ccccc2)=O)C1 C1(C)(C=O)CC(C)OC(C)C1.C(C(C)(C)CCNC(c1cccs1)=O)OC.C C1(C(=O)NC(CN(C(c2ccnn2CC)=O)CC)C)CCOC(=O)N1 C(=O)(C(CSC)c1ccccc1)N(CC(C)NC(CC=CC)=O)C n1(CC)nc(C)c(CNC(=NCCF)NC2CC(c3ccc(F)c(F)c3)C2)c1C CCCN(C(=O)CNC(C)(C)C)C.C(=O)(CN(C)C(C1CC1)=O)N N1(C(C)C)CCCC(CC(=O)NCCCN(C)C(C2(C)CC(C#N)C2)=O)C1 C=CCC(C)(C)CNC(C1CC=CCC1NC(=O)CCC1CCCCO1)=O C1(C2CCCO2)(C=O)CCOCC1.c1(COC)cc(C=O)no1.CC=CC.N C1(NC(c2coc(Br)c2)=O)CCC(O)CN(C(C2CCC2(F)F)=O)C1 C(=O)(C(CC(F)F)N(C(=O)Cc1ncoc1C)C)NCc1snc(CC)n1 Cc1c(C(=O)C(=O)C(C)OC(=O)C(F)(F)F)sc2ccccc12 c1(C(=O)NC(COCC)C(=O)N(C2CCOC(C)C2)C)cc(C)c(C)cn1 CC(C)C(C(=O)N(C(CNC(=O)C(O)C(C)C)C1CC1)C)n1cc(Br)cn1 c1(OC)nc(NCC(O)CNC(=O)CCOc2cc(C)ccc2C)nc(C)c1F n1(CC)ncc([N+](=O)[O-])c1C(N1CC(NC(=O)CCCCCn2cnnn2)C1)=O CC1(CNC(C2CCCOC2)=O)CCCN(C(C2(C(F)F)CCCO2)=O)C1 c1(OC)n[nH]c(C(=O)N(C2CCC(NC(=O)C(OC)OC)CC2)C)c1Cl Cc1ccc(C#N)cc1NCc1cc(=NC(=O)C2C3CCC(C3)N2)[nH][nH]1 N1(CC(=O)NC(CC)CNC(=O)CCN2CCCC2=O)CCN(CC)CC1 CC1(CNC(c2ccc(Cl)c(F)c2)=O)COCCN(C(=O)C(O)P(C)(C)=O)C1 C(=O)(C(CC(C)C)NC1CCCCC1)NC.C1(C)C(C)(C)S1 C=CCC(CC=C)C(=O)N1CCN(C(C2CCC23CCC3)=O)CC1C1CCC1 N1(C(CC)=O)CCCC(CN(C(=O)Cc2cscc2Br)C)C1 C=CC(C)(C)CC(=O)NCC1CC(C)CO1.c1(C(=O)N)ccccc1.CC=C Cc1cc2ccccc2nc1C(N1CC(CNC(=O)CC(C)C(C)C)C1)=O N1(C(C2CC2NCc2c(O)cccc2O)=O)CCOCC(O)C1 N1(CC)CCN(C(=O)CCCCCN(C)C(C2C(C(C)=O)C2(C)C)=O)CC1=O c1(C(N2CCC(CCOC)C2)=O)snc(C)c1I N1(C(CC(C)F)=O)CCC2(CCC2NC(=O)C2=NNC(=O)CC2)CC1 C(=O)(CN1C(=O)Cc2ccccc21)NC1C2CN(C(C(C(CC)O)C)=O)CC21 C1(C(NOCCC=C)=O)CCCN(C(=O)CCc2nccn2C)CC1 C1(c2ccc(C)cc2)CN(C(=O)Cn2cc(COCCCO)nn2)CC(C)O1 Cc1cc(Cl)cc(N)c1C(=O)NCCN(C)C(c1cccc(C2OCCO2)c1)=O N1(C(=O)C(F)=CCCF)CCCC2C1CCCN2C(c1cc2c[nH]cnc-2n1)=O c1(C=O)cc(C2(O)COC2)on1.C(C)(C(=O)NCC(O)C)OCC(C)C.N N(C(=NCC(C)c1ccsc1)NCc1c(C)cccc1Cl)C(C=C)C N1(C(C2N(CC)CC2)=O)CCCCC2(C1)CN(C(C1(SC)CC1)=O)C2 C12CCC(CC1)C2.c1(C2(C(N(CC(C)C)CC(=O)N)=O)CC2)ccno1.C N1(C(C2CCC(CC)CC2)=O)CCCC(F)C1.c1(CC(=O)N)cc(C2CC2)no1 c1(CN(C(CC)C)C)cc(F)ccc1NC(=O)NC(c1ccc(F)cc1F)C c1(C(=O)NC2CCC(NC(Cc3cc(C)n(C)n3)=O)C2)cccc2ncsc12 N1(C(CN2CCC(OC)C2)=O)CC2CCN(C(=O)CCC)CC2C1.C(=O)(C1CC1)N c1(CC)ccccc1CC(=O)N(C)CC1CCCCN1C(=O)Cc1c[nH]nc1C c12ccc(cc1)CNC(=O)C2.C1(O)(C(N(C)CC)=O)CCSC1 C(=O)(C1CC=Cc2ccccc21)N(CCCCCCNC(=O)C1=CCCSC1)C C1(C(=O)NCCOC2CN(C(c3c(CC)cno3)=O)C2)CCCC(C)C1.O N1(C(C2(C)C(C)C2)=O)CCC2(CCN(C(c3cccc(-n4cncn4)n3)=O)C2)C1 Cc1cc(=NCCC(C)N(C)C)[nH]cc1S(=O)(=O)NCC(S(C)(=O)=O)C1CC1 c1(CC)oc(C(=O)NCCC2CC2)cc1C.c1(C(=O)N)c[nH]cc1C1CC1 C1(CNC(=O)CC2CCCN2C2CC2)CC2CCC1N2C(=O)C1=COCCC1 C(=O)(C1=CCCCC1C)NC1C(SC)CN(C(=O)CCc2c(C)n[nH]c2C)C1 Cc1ccc(C(N2CCC(C)(NC(=O)C3=CSCCO3)C2)=O)c(C2CC2)c1 c1(C(=O)NC23C(CN(C(C4(C)ON=C(C)C4)=O)C2)C3)cc(C)c(C)nc1O C1CCCCN1C(c1cn[nH]c1)=O.c1(C(=O)NC2CC2)cnn(C(F)(F)F)c1 C(C)(C)(CC=CC=O)NC(CN(C(C(C)C)=O)C)=O.C1(CC)CC1C1CC1 CC1CN(C(=O)C#CC2CC2)CCCN1C(=O)Cc1noc2ccccc12 CON(C)S(=O)(=O)c1ccc(NC(C2CCOC3(CCSCC3)C2)=O)cc1 c1(C(N2C(CNC(CCC=C)=O)COCC2)=O)cnc2cc(C)[nH]c2c1 C1(OC)CN(C(=O)Cc2nnc(C)o2)CC1NC1CCCCC1C C(C(=O)NCCn1ncnn1)(C1CCOC1)NC(C1CC(O)C1)=O.C1CC1 C1(CC(=O)NCC2OCCN(C(CCc3ccc(C)s3)=O)C2)CC(=O)NC(=O)C1 CC1C(C(=O)N)C(O)C(=O)N1C.C1CCN(C(c2nc(=O)n(C)[nH]2)=O)C12CCC2 C1(NC(c2cc(O)ccc2Cl)=O)C2CCC1CN(C(=O)CCC1CCCCC1)C2 CC(C)(C(=O)NCC(C)(F)F)c1csc(-c2ccsc2)n1 C=CCC(C(=O)NC1CC(NC(=O)CCCC2(C)NC(=O)NC2=O)C1)C(C)C N1(C(c2cc(C(N)=O)[nH]c2)=O)CCN(C(=O)CC2(C3CCCC3)CC2)CC1CO N1(C(c2c(OC)noc2C)=O)CCC(C)(C)C(C(=O)Nc2cnn(C)c2)C1 C1(NC(=O)OC(C)(C)C)CC2(C1)CCC2.C1(C=O)CCCN(c2nccs2)C1 N1(C(CCC(=O)OC)=O)CCCC2(CCCN2C(C2(C)COC2)=O)CC1 n1(CC(CCCC)CC)c(-c2cccnc2C)csc1=Nc1cnn(C)c1 c1(NC(=O)NC(c2ccc(CC)cc2)C=C)cc(COC)ccc1C O(NC(=O)C(O)C(C(C)C)OC)CC.C12CCCCN1C(=O)c1c[nH]nc12 c1(-c2nc(C3C(C)C3)nn2C(c2cnn(C)c2)C)snc2ccccc12 N1(C(c2n(CC)ccn2)=O)CCC2CCN(C(C3CCN(C(N)=O)CC3)=O)C2C1 N1(C(C2(OC)CC2)=O)CCC(NC(c2ncoc2C2CC2)=O)C(O)C1 C1(NC(c2c(OC)nsc2)=O)CCOCC1C(=O)NC1(CC(N)=O)CCC1 N1(C(CC2CCCC(NC(C(CCC)C#N)=O)C2)=O)CCCC(O)(C2CC2)C1 Cc1nc(C#N)ccc1C(N1CCC(C)C(NC(c2coc(CO)c2)=O)C1C)=O N1(C(c2c(C)cc(F)s2)=O)CCCN(C(c2cnn(C)c2C)=O)CC1CO O=C(CC1CCc2ccc(O)cc21)N1CCC(C(=O)NC23CC4CC2C3C4)C12CC2 N1(C(c2nccc(C)c2)=O)CC2(CC2)CC1CNC(C1CC1(Cl)Cl)=O C1(CC)CC(C(=O)O)CN(C(c2nnc(-c3occc3C)o2)=O)C1 c1(C(=O)NC2C(C)CN(C(C3CC(C)(C)CO3)=O)C2)c2c(nn1C)CCC2 C1(NC(C(CCC)N(C)C)=O)CN(C(c2ccncc2Br)=O)CC2(CC2)C1 N1(C(CC2CC(CC)OCC2)=O)CC2CCN(C(c3cc(C)cc(F)c3)=O)CC12 CCCC(F)C(=O)NCC(C)CNC(c1cccnc1C1CC1)=O c1(CNC(Cc2ccc(Nc3nc(C(C)C)ncn3)cc2)=O)ccc(Br)c(F)c1 c1(C(C(=O)N)(C)C)cccc(Cl)c1F.C=C(C)CCNC(=O)CCOCCC C1(CC)CCCN(C(=O)CN(CC(C)C)C(c2cc(C(C)=O)c[nH]2)=O)CC1 c1(C(=O)NCC(CC)N(C(=O)Cc2cc(C)nn2C)C)cccc2ncnn12 C#Cc1ccc(OCC(=O)NCC#CCNC(C2CCCC(O)C2)=O)cc1 c1(CC(N2CCC(NC(C(C)C3CC3)=O)(CF)C2)=O)ccc(Br)c(Cl)c1 N1(C(CN(C)C)=O)CCC2(CCCN(C(=O)CCC3CCCO3)C2)C1 c1(NC(c2ccc(Cl)cc2)CSC)cc(NC(C)C)ncn1 C=CCCCCCC(=O)NCCOC1CN(C(=O)CC2CCCCCC2)C1 C1(OC2CC(NC(=O)NC3C(C=C)OCC3)C2)CC2(C1)CC(C#N)C2 C1(C(=O)NCC(C(C)(C)F)(C)F)CCN(C(c2ccncn2)=O)C12CCC2 CCCC(C)C(=O)NC(C1CCCN1C(=O)CCc1ccc(Br)nc1)C C(CC(C)(C)CC(=O)N1CC(NC(=O)Cn2nccc2N)C(C)C1)OC N1(C(c2cccc(Cl)n2)C(=O)NCCCSCC)CC(C)c2ccccc21 CS(=O)(=O)c1ccsc1C(=O)NCCC1CCC1.C1(C(=O)N)CC1C1CC1 N1(C(c2oc(CC)c(C)c2)=O)CCN(C)CC1CNC(C1CCCN(CC)C1)=O C1(NC(CC2C(CC)C2)=O)CCC(NC(c2scc(C)c2C)=O)CC1 N1(C(CCOCC#C)=O)CCCN(C(=O)C(C2CCCCC2)O)CC1 C(CNC(=O)C(C1CCC1)C1CCC1)(CC(F)(F)F)NC(=O)CC(Cl)Cl N1(C(CC2(OC)CN(C(C3CC(OC)C3)=O)C2)=O)CC(C)=CC(C)C1 c1(C(N(C(C)C)CC2CCCCO2)=O)ccc(NCc2nccn2C)cc1 N1(C(C(=O)NCC)=O)CCC(C)(C)C1C(=O)N.c1(CCC)cc(C)[nH]n1 C(=O)(C(C)(C)C(C)C)N(CC(CC)NC(c1csc(-c2cn[nH]c2)c1)=O)C C1(C)(NC(CC=C)=O)CCCN(C(c2cnns2)=O)C1 CC(C)C(O)C(C)C(=O)NC1C=CC(C(=O)NCc2cc(Cl)ccn2)C1 C(C(CO)C1CC1)N(C1CC1)CC1CC1.C1(CC)(COC)CC1 N1(C(C(CC#C)C)=O)CCN(C(c2cncc(F)c2)=O)C(COC)C1 CC1CCN(C(=O)C(F)=C2CCC2)C1CNC(c1cnc(-c2cccs2)s1)=O N1(C(CCCc2cc(C)no2)=O)CC2CCCC1C2CNC(c1cnc(O)s1)=O C(C)(C)(C=O)NC(=O)OC.c1(C(C=O)C)nc(C)cs1.CCC1CC1.N C1(C=O)CC2CCC1CC2.C(=O)(C(F)C(=O)NCC1CCCC1)OCC.C C=C(F)C1(CC(=O)NC(COC)C(=O)N(C)Cc2cc(C)nn2C)CCC1 N1(CC(=O)NCc2ccc(-c3nnn(C)n3)cc2)CC2CC(F)(C2)C1 C1(N(C)C(C2CC=CCC2C(F)(F)F)=O)CCN2CCOC1C2 C1(NC(c2cc(C(C)=O)oc2)=O)CCCN(C(=O)CSCC2CCCO2)C1 Cc1cc(O)c(Cl)cc1C(=O)NCCNC(C1(c2cccs2)CC1C)=O C(=O)(CCCC(C)C)N1C(C(=O)NCCc2cnc(C)[nH]2)(CC)CCC1 C=Cc1ccc(C(=O)N(CCC(=O)NC2COC(C(F)F)C2)CCCO)cc1 C(c1sc(Cl)nc1Cl)=CC(=O)NC(C)(C)CNC(C1CC(C#N)C1)=O N1(CCC)CCC(NC(C2(CC)CN(C(C3CCCCC3F)=O)C2)=O)CC1 c1(CCNC(=O)Nc2c(OC)ncnc2C)cccc2c1OCCO2 c1(C(=O)NC(CNC(C2C(C=C)C2)=O)C2CCC2)cc(Cl)c(N)cc1F CCCC(CC)CC(=O)N1CCN(C(=O)C(C2CCCCCCC2)O)CC1 C1(C(C)NC(C(CC)OC)=O)CCN(C(=O)C(C)Cc2ccco2)CC1 C1(C#N)(C(N2CC(C(C)NC(CCCOC)=O)C2)=O)CC2CCC1CC2 n1(-c2cc(C)on2)c(C)cc(C(=O)N(CC(C)CNC(c2ccoc2)=O)C)c1C c1(C(C(=O)NCCC)N(c2ccc(OC)cc2)CC)snc(OC)c1Br C1(NC(c2cncc(C3CC3)c2)=O)CCN(C(c2ccnnc2)=O)CC1O C1(C#N)(CC)CCN(C(=O)C(C)CNC(c2nnc(O)nc2O)=O)CC1 C1(NC(c2n(CCCC)nnn2)c2cnco2)CCSC(C)(C)C1 c1(C(=O)NCC#CC(N2C(C)COCCC2)=O)ccc2occc2c1 c1(C(=O)NCCCN(C(C2OCC2(C)C)=O)CC)ccc(O)nc1C c1(C=O)ccc(S(N)(=O)=O)c(F)c1.N1(C(CC(C)F)=O)CC(C)C(C)(C)C1.N c1(CC)nc(C)c(C(=O)NCC2CCCCC2)s1.C1(C(=O)N)CC2CCC1O2 C1(CNC(=O)NC2CCC23CCOCC3)CCC2(CC1)OCCO2 C1(O)(CNC(C(C)SCCCC)=O)CC(N=c2[nH]c3c(cc2C#N)COCC3)C1 C(C)(CCC(=O)NC(c1cn(C)nn1)C(=O)NCCOCC1CC1)OC N1(C(C2C(CCC)CCC2)=O)CCC(N(CCC)C(C2CCS(=O)CC2)=O)CC1 c1(C(C(N2CC3C(COC)C3C2)=O)(F)F)cccc2ccccc12 N1(Cc2c(C)cc(Cl)cc2)CCC(F)(F)C(NC(c2cccnc2C)=O)C1 c1(CC)cc(C(=O)N(C2CN(C(c3ccc(C(F)(F)F)[nH]3)=O)C2)C)on1 Cc1sc(C(=O)NC2CN(C(=O)C(O)C3CCCC3)CC2C)nc1Br N1(C(CC2N(C(c3scc(C)c3)=O)CC(F)C2)=O)CC(=O)NCC1C CCC(CCC(=O)NCc1ncc(C)s1)NC(=O)C(C)(C)C(=O)N(C)C c1(-c2nc(CSC)n(CC3CCCC3(F)F)n2)nccn2nccc12 n1(CC)nc(C(N2CCC(O)C2C(=O)N(C)CC2(O)CN(C)C2)=O)cc1C Cc1nc(CO)ncc1C(=O)N(C1CCCN(C(=O)CSc2cccs2)C1)C C1(NC(c2c(C)c[nH]n2)=O)CN(C(=O)CCc2nc[nH]n2)CC1N=[N+]=[N-] C1CCC2(CN(C(=O)C=C3CCN(C)C3)C2)O1.c1(COC)ccoc1C=O c1(C(=O)NCCCNC(C(C)SC)=O)ncncc1C#N CC(C(=O)N=c1ccc(C(c2ccccc2)=O)n[nH]1)N1CC(=O)NC1=O CCCC(CC)C(=O)N1CCC(CF)(NC(=O)C(c2ccccc2)OCC)C1 C(c1ccccc1C#N)=CC=O.C1CCC1.C1(CC(=O)NC)(OCC)CC1 c1(C(N2CCC(C)(NC(c3ccc(=N)[nH]n3)=O)CC2)=O)cn2cc[nH]c(=O)c2n1 N1(C(C2CCN(C)CC2)=O)CC2COCCC2(NC(=O)Cc2ccon2)C1 N1(C(C)=O)CCn2ncc(-c3ccc(NCc4cscn4)cc3F)c2C1 c1(C(=O)NCC(CC=C)NC(=O)C(C)Oc2cccnc2)cc(F)cc(Cl)c1N N1(C(CCC(=O)C2CC2)=O)C(C(N2CC(CO)C3(CC3)C2)=O)C2CC(O)C1C2 c1(N(CCOC)CCNC(c2cccc(CS(C)=O)c2)=O)nc(O)ncc1Cl C(=O)(C(C)(C)S(C)(=O)=O)N(C1CCCCN(C(C2COC(=O)N2)=O)C1)C N1(C(c2n(C)c(Cl)c(Cl)c2)=O)CCN(C(C2CCCN2C=O)=O)CC(CO)C1 C=CC(C)(O)C(=O)N1CC(C)(CCC(=O)NC2CCOCC2F)C1 CC1=C(C(=O)NCC2CN(C(c3ccc(Cl)cc3)=O)CCC2C)C(C)(C)CCC1 c1(C(N2CCC3C(NC(C4CC(C)(C)C4)=O)C32)=O)ncnc(O)c1Br N1(C(C2(NC(c3cc(C)c(C)o3)=O)CCCC2C)=O)CCSC(C)(C)C1 Cc1ccc(NCCCCN(CCCN(C(=O)Cc2cn(C)nc2Cl)C)C)nc1 CC1(CNC(=O)CCC2(O)CCC2)CCN(C(C2CCCC(F)C2)=O)CC1 c1(C(=O)NCC(c2ccc(Cl)cc2)C(C)C)cc2c(oc1=O)CCCC2=O C1(NC(C2(COC)CC(=C)C2)=O)CN(C(=O)CC(C)CC)C2(CCCC2)C1.O CCCCCC(O)CC(=O)N1CCN(C(c2ccn3nncc3c2)=O)CC1CO C12(C(=O)NC(CC)(CNC(C3CCC(=O)N3)=O)CC)CC1COC2(C)C C(C1(CO)CCc2ccccc21)NC(=NCCOCC=C)NC1CC(OCC)C1 C1(NC(C(=O)NCCCOC)=O)C2CCCC1CC(C(=O)O)C2 CCC(CC)CC(=O)N1CC2(CC(CNC(=O)COc3cnn(C)c3)C2)C1 C12(C(=O)NCCC(C)OC)CC1CN(C(c1ccon1)=O)C2 CC(C)CCCCCC(=O)N1CC(O)CCC1C(NC[Si](C)(C)C)=O C1(CCNC(C2(C)CCCOC2)=O)CCCN(C(c2c(O)cccc2O)=O)CC1 n1(CCN(C(=O)CC2(C)CC2)C)cc(C(C)CC2CCC2)nn1 C1(C)(C(N(CC(C)N(C(=O)CCCc2ccncc2)C)C)=O)CS(=O)(=O)C1 N1(C(C2C(NC(C(COCC)C)=O)CC2)=O)CCOC(CCO)C1 C(CCCCC(=O)N1CCC(O)(CNC(C2(n3cccc3)CCCC2)=O)C1)SC N1(C(C(CC(C)C)C)=O)CCC2CCC(NC(=O)C(C)Cc3cnco3)C1C2 C1(CC(=O)Nc2c(OC)nsc2)CC(F)CN1C(c1ccc(CC#N)cc1)=O N1=C=C(CC(=O)NC2CC(CCNC(c3[nH]ccc3C3CC3)=O)C2)C=N1 n1(CC(=O)NC)ccc2ccccc12.C(=O)(C=O)N.c1(CC2CC2)nn[nH]n1 N1(C(c2cnc(N(C)C)s2)=O)CCC(NC(c2csc(Cl)c2)=O)C2(CCC2)C1 C#CCCCCC(=O)NC1CC(NC(=O)Cc2ccc(Br)c(Cl)c2)C1 C1(NC(C2CC(C)(CC)C2)=O)CCN(C(=O)CCC=CBr)C1C Cc1nc(C)c(C(=O)NC(C2CCCN2C(=O)CCNC(=O)CO)C)[nH]1 Cc1nn(C)c(C)c1C(c1nnnn1C(C)C)NCc1cc(Br)c(Cl)s1 CC1(C)CC2(CC(C(=O)NC3CN(C(C4COCCC4(F)F)=O)CC3CO)C2)C1 C=CCC(C)C(=O)NCC1CCC(N(C(=O)C(CC)Oc2ccccc2)C)CC1 c1(CCC)c(C(N2CCCCC2CN(C(=O)CCC)C)=O)nnn1C.C(C)(=O)N C(=O)(CCCC(F)F)NCC1CN(C(c2ncn(CC)c2)=O)CC1C(F)(F)F c1(C(N(CC(C)NC(c2c(OC)ccs2)=O)C)=O)cc(Cl)cc2c1OCC2 S(=O)(=O)(c1cnc(N)c(Cl)c1)NC(c1ccc(C)cc1)CC.C1(C)CCCO1.C C1(C=O)C2C3CCC(C3)C12.C1(C)(C(N2CC(COC)C2)=O)CC(C#N)C1 N1(C(Cc2cn(CC)nc2)=O)CC2CCCC2(NC(=O)CC2CNC(=O)C2)C1 N1(C(C2CC(O)C2)=O)CCCCC1c1nn(-c2ccccc2)cc1Cl C1(NC(c2cc(C)on2)=O)CC(F)CN(C(=O)CC2CCC(C)(O)CC2)C1 c1(CC)nc(C(=O)NC(c2n[nH]cc2)C)cs1.C1(C)CC1C(=O)N.C c1(C(=O)NC2C(NC(CCCCOC)=O)CC2)c[nH]c2nccc(Cl)c12 C1(NC(C2(NC(C)=O)CCCCC2)=O)CN(C(c2cscc2SC)=O)CCC1C c1(NC(C2CC3CC3N2Cc2cncc(Cl)c2Cl)=O)ccc2sncc2c1 n1(CC)nc(C)cc1C(=O)NCC=CCNC(=O)C=Cc1ccoc1 N1(C(CC(=O)OC(C)(C)C)=O)CC(NC(=O)Cn2ncnn2)CC(O)C1 C1(NC(c2cnn(CCC)c2C)=O)C(C)CN(C(=O)C(=O)NOC)CC1C Cc1ncc(Cl)c(C(=O)NC(C)C(C)(C)NC(c2ncncc2Cl)=O)n1 Cc1ccn2nc(C(N3CCOCC3CNC(=O)C(F)n3cccn3)=O)nc2n1 CN1CCN(C(=O)C=Cc2cccs2)CC1CNC(=O)C1=CCOCC1 CC1C(NC(=O)C=C(Br)Br)CCCN1C(=O)CN(C)CCO C12CCCC1NC(=O)CONC2=O.C1(CCOC)(OC)CCOC1 c1(C(=O)NC(CC)CN(C(=O)C(F)(F)CC)C)ncc(Br)cc1O c1ccc(C)c(F)c1.C(C)(CCC(=O)NC(COC(C)C)C=O)OCC.N C1(NC(C(CSC)OC)=O)CN(C(c2cc(C)[nH]n2)=O)CC2(CCC2)C1 C(=O)(C1=CCCCC1P(C)(C)=O)N(CCNC(C(C(C)SC)O)=O)C C1(CN(CC(C)C)Cc2n(CC)ccc2)CCN(C=O)CC1.C(C)(C)C.O c1(OC)ccc(C)cc1CNC(=NCCOCCO)NC(c1ccccc1)C c1(OC)ccc(O)cc1C(=O)N(C)CCNC(C1CC1(c1ccccc1Cl)C)=O C12(NC(COC(CC)(C)C)=O)CCCC(CN(C(=O)CC(O)C(C)C)C1)C2 c1(C(N2CCC(CC(=O)OC)C2)=O)cccc(C)c1N Cc1cnc2nc(NC(N3CCN(C)C(C(C)C)C3)=O)sc2c1 c1(C(=O)OC)cc(NC(c2cc(NC34CC(CO)(C3)C4)n[nH]2)=O)ccc1C Cc1[nH]c(C#N)cc1C(=O)NC1CCOCC1NC(c1ccnn1C1CC1)=O c1(CCC=O)ccc(OC(F)(F)F)cc1.C(C#CC)NC(C1(CC)CC1)=O.N c1(C(=O)NCC(CNC(C(CC(C)C)F)=O)C)ccc2cncn2c1 C(CC(=O)N=c1cc(C(N)=O)n(C)[nH]1)C1CCN(C(COCCCC)=O)C1 c1(CNC(C=CCN(C)CC)=O)ncc(C(=O)NOCCO)cn1 c1(COC)nc(N)cc(N(CC(F)(F)F)C)n1.C1CCCN(C(=O)N(C)C)C1 C1(NC(=O)CC2COCCO2)CCOCC1NC(c1cc(Br)n[nH]1)=O c1(CC(=O)Nc2c(C)ccc(C(N)=O)c2)cccc(S(=O)(=O)N(C)C)c1 C1(CNC(c2n(CCOC)ncc2)=O)CN(C(=O)CCCCCF)CCC1(C)C Cc1cccc(C(=O)C(=O)NC)c1.C1CC(C)N(C(=O)Cc2ccc(F)cc2)C1 C=C1Cn2c(C(=O)NCCC3CSCCN3C(=O)CC3CC=CCC3)nnc2S1 CCC(C)CCCCC(=O)NC(C)(CNC(=O)CCCCCOC)C(C)C C12(CNc3nnc(C)c(C)n3)CCC(CC1)CO2.C(=O)(CCS(=O)(=O)N(C)C)N C12(C(=O)NCC(C)C(C)(F)F)COCC1CN(C(=O)C1=CCCC1C)C2 c1(CC)nc(C)c(C(=O)NC(C2CCCN(C(C3SCCS3)=O)C2)C)o1 Cc1cc2ccc(C(=O)NCCN(C)C(c3cccn(C)c3=O)=O)cn2c1 N#CC1CC2(CC(NC(C3CC=CC(NC(C4C=CCS4)=O)C3)=O)C2)C1 c1(CC)nc(C(=O)NC(C)CNC(=O)CCc2ccn(C)n2)c(C)o1 Cc1nsc(C)c1C(=O)NC(C)CCC(=O)NC(c1cn(C)nn1)C N1(C(CNC(=O)NC)=O)C(C(=O)N(CC(C)(C)C#N)C)CC1C Cc1cc(C(=O)NC2CC2NC(C2CCOC2C)=O)c(O)nn1 Cc1ccc(CN2CC3(C2)CN(c2ncc(F)cn2)CCO3)c2ccccc12 c1(C(=O)NC(C)CC(C)NC(C2(C)CCNC2=O)=O)n[nH]c2ccc(F)cc12 C1(CC)(NC(c2cc(C)n(CCO)n2)=O)CCCN(C(c2cc(Cl)no2)=O)C1 c1(C(=O)NC2(C3CN(C(C=C4CCN(C)C4)=O)C3)CC2)noc2ccc(Cl)cc12 S(=O)(=O)(CCCNC(=O)Nc1n[nH]cc1-c1ccccc1)NC c1(CNC2CC(C(=O)Nc3cc(C)nc(F)c3)C2)c(F)ccc(F)c1O c1(CC)cc(C(=O)NC(C)CNC(=O)Cn2nnc(C)n2)ccn1 c1(OCC)ccc(CCNC(=O)C(n2cc(CCC(C)=O)nn2)C)cc1 c1(N2CCc3c([nH]n(C)c3=O)C2)nc(C#N)nc2ccccc12 C(=O)(CS(=O)(=O)c1ccc(Cl)cc1)N(CCC)CC.C1(CC=O)CCCCO1.N N1(C(C(CCC#C)O)=O)CC2CC(NC(=O)C(C)=CC)CC(C2)C1 Cc1ncn2ccc(C(=O)NC3C=CCN(C(=O)C(C)CSC(F)(F)F)C3)cc12 C=CCC(C)C(=O)NC1CCCC1CC(=O)NCCc1cn(C)cn1 N1(C(CCNC(N)=O)=O)CC2(CCCN(C(C3(O)CCSC3)=O)C2)C1 C(C(O)CC(=O)N1CC(O)(c2nn[nH]n2)C1)N(C(C)=O)C1CC1.CC.CCO N1(C(CNC(N)=O)=O)CCC(CO)C(NC(=O)Cc2ccccc2F)C1 C(=O)(N=c1[nH]n(CC(=O)O)cc1C)c1ccc(N(C2CCCO2)CCC)cc1 C12(CCNC(CC(C)(C)c3ccc(F)cc3)=O)CC3CC(CC(C3)C1)C2 c1(CCC(=O)NC(CN(C(Cc2cn(CC)nn2)=O)C)C)ccccc1Cl C1(NCc2scc(C(=O)OC)c2)CN(C(=O)C(C)CN2CCOCC2)CCO1 C1(C(N(C(C#C)C)C)=O)CCN(C(=O)C(C)(F)c2ccon2)C(C)(C)C1 Cc1n[nH]c(C)c1CC(C)C(=O)NC1CC(C)C1.C(c1ccsc1)=CC=O.N c1(-c2cn(CCNC(C(C)(C)NC(C)=O)=O)nn2)ccc(F)cc1 C1(N(C)C(c2ncn(C(C)(C)C)n2)=O)CCCCC1NC(C1CC12CCC2)=O CON(C)CCCNC(C1C=CCN1C(c1ccsc1Cl)=O)=O N1(C(c2ccc(C(=O)OC)o2)=O)CCC2CS(=O)(=O)CC2C1 c1(OC)cc(C(=O)NCCC2COCCN2C(=O)Cc2occc2C)ccc1C c1(C(=O)NCC2CN(C(CCC)=O)CC2O)c[nH]c2cc(C)ccc12 N1(C(C(C)F)=O)CCOC(c2ccccc2C(F)(F)F)C1.CC(C)(C)OC(=O)N N1(C(CC2C(OCC)COCC2)=O)CCN(C)C(CNC(=O)CC(CC)OC)C1 c1(OC)ccc(C(=O)NCCC2(O)CN(C3CCCN(C)C3=O)C2)c(OC)c1 c1(CC(=O)NC2CCN(C(c3csc(Cl)n3)=O)CC2F)cn2ccccc2n1 c1(-c2n(CCCOCC)c(N3CCC(C(C)C)CC3)nn2)cccc2ncnn12 C1(C2(O)CCN(C(C3Cc4ccncc4C3)=O)CC2)(NC(C(C)CCO)=O)CC1 c1(C(=O)NCC(N2CCC(NC(=O)O)C2)C)nnc2ccccn12.C(C)(C)C N1(C(C)=O)CCCC1CC(=O)NC1(C)CC1.c1(C=O)n[nH]cc1C1CC1.N N1(C(CC(CC)NC(=O)C(C)Cn2cccn2)=O)CCC(F)(CF)CC1 Cc1cc(C(N2CC(CCCCNC(C3CCCC(=O)N3)=O)C2)=O)cc(N)c1Cl CC(CCC(C)(C)C)C(=O)N1CC(N(C)C(c2ccnc(O)c2F)=O)C(O)C1 C1(NC(C(C2CCC2)NC(C2CCCC(O)C2)=O)=O)CCCCCC1CO C(C(=O)NCC(C)(C)CNC(C1(NC(C)=O)CC1)=O)(C(C)C)OC C=CC1OCCC1C(=O)NCc1cc(C(N2CC(OCC(C)C)C2)=O)ccn1 CCC(C)(CO)C(=O)NC(c1cccc(C)c1)CNC(=O)CCC1CC1 c1(CC)cc(C)nc(N(C2CCC(N)C2)Cc2cc(OC)cc(OC)c2)n1 c1(N2CCN(CCNC(CC=C)=O)CC2)ncnc2c(Cl)cc([N+](=O)[O-])cc12 c1(C(N2CCC2CN)=O)cc(Cl)cc([N+](=O)[O-])c1Cl.[SH](=O)(=O)c1ccccc1Cl CC1=CCC(C)(C(=O)NCCOCCC)CC1.c1(C=O)cn(CCCF)nn1.N n1(CC)nncc1C(=O)NC(c1cn(C2CCCC2O)nn1)C C(=O)(CC1C(=O)Nc2ccccc21)N(C1CC(NC(=O)CS(N)(=O)=O)C1)C n1(CCC(=O)N2CCC2Cn2cc(-c3cncc(Br)c3)nn2)cnccc1=O N1(CC)CC(NC(C2CC(O)C2O)=O)CC1=O c1(C(=O)NCCNC(CC(CC)OC)=O)c(C)nn(-c2ccc(F)cc2)c1Cl C1(C(=O)NC(C2CCN(C(C3(F)CC3C)=O)CC2)C(C)C)CCc2cncn2C1 S(=O)(=O)(c1cccnc1NCCSC(C)(C)C)NCC(C)CC(N)=O C(=O)(C1=NNC(=O)CC1)NC1CC(C)CN(Cc2cc(F)ccc2Br)C1 CC(C)CC(CNC(C1CCC(C)C1)=O)C(=O)NCC1(F)CCOCC1 C=CC1OCCC1C(=O)NCC1C2CN(C(c3cncn3C)=O)CC12 c1(C(C(=O)N(CC(C)C)C)=O)ccc(F)cc1.c1(C(=O)N)ccnn1C1CC1 N1(C(c2ncc(C)c(C)c2)=O)CC(NC(C2CC3CCC2C3)=O)C2CCCCC12 C=Cc1ccc(C(=O)NC2CCN(C(c3ccc(F)c(Cl)n3)=O)CC2F)cc1 Cc1ccc(C(N2C(C(=O)NCC3(F)CCN(C)C3)CCC2C2CC2)=O)nc1 N1(C(c2c(CC)occ2)=O)CC2C(CN(C(=O)C(c3cccs3)S)C)C2C1 c1(CC)nc(C)sc1C(=O)NC(C)(CNC(=O)CCCC1CC1C)CO CCCS(=O)(=O)CC(=O)N(CC(C)N(C(=O)CCc1ccc(Cl)c(OC)c1)C)C C1(N(C(=O)C(F)=CC2CC2)C)CCCN(C(C2(CF)COC2)=O)CC1 N1(C(C(C)OC(C)(C)C)=O)CC2CC(C1)CN(C(C1CC3(C1)CC3F)=O)C2 c1(C(=O)NC2CC(C(=O)NC(c3cnn(C)c3)CC)C2)cc(O)ncn1 CN=c1nc(C(=O)NC2CCCN(C(=O)CCCNS(C)(=O)=O)C2)cc(C)[nH]1 C1(C(=O)Nc2c(OC)cnc(Cl)c2)CC2CC1CC2(C)OC N#Cc1c(NC(C2CCCN(Cc3cccnc3F)C2)=O)sc2c1CCCCC2 N1(C(C(C)OCCC#C)=O)CCN(C(c2c(O)cccc2Cl)=O)CC1C1CC1 CC1ON=C(C(=O)N2CC3CC3(NC(=O)C)C2)C1C.C1(CC=O)CCCCC1.N Cc1nn(-c2ccccn2)c(C)c1CC(=O)NC(C)CNC(C1(F)CC1)=O c1(C(=O)NCCCN(C(=O)COC2CCC2)C)cc(C#N)cs1 N1(C(CN(C(COC)=O)C)=O)C2CCCC1CN(C(=O)CN1CCC(C)C1)C2 N1(C(c2cc(OC)n[nH]2)=O)CCC(C)C(NC(c2cnccn2)=O)C1.C(C)C.O N1(C(CC2(OC)CC2)=O)CCCC2(CCN(C(C3(C)CC3(F)Cl)=O)C2)C1 C(CC(C)C)C(=O)O.c1(CN(CCC)C=O)ccc(NC)cc1.c1ccccc1.N CCC(C)C(C(=O)N1C2COCC1C2)N(C)C(c1cocc1C)=O N1(C(C(C=C)OC)=O)C2CCC(C(N3CCCC(CCCO)C3)=O)C1CC2 C(=O)(CC(C)C(=O)N1CC(OCC(=O)NCC(C2CC2)C2CC2)C1)OC c1(C(N2CCC(O)(C(C)NC(Cc3nnc(C)o3)=O)C2)=O)nc(C)n(C)c1C CCCC(C)(CC)C(=O)NC(C)(C)CN1CCN(C(C2CCNC(=O)C2)=O)CC1 C1(CNC(C(C=C)O)=O)CCN(C(=O)CC2(O)CCCCC2)CCO1 n1(CC(N2CCC(NC(C(C=C)(F)F)=O)C(CC)C2)=O)sc(=O)c2ccccc12 C1(NC(c2ccc(CC)s2)=O)(CC)CCN(C(=O)CO)CC1.c1cnn(C)c1 C1(NC(CNC(CCC)=O)=O)CCN(C(=O)CCSc2ccccn2)C1CC c1(C(N2CC(CNC(CCC(=O)NCCC)=O)OCC2)=O)ccnc2ccsc12 C1(CNC(CCC(=C)C)=O)COC(C(F)(F)F)CN1C(c1ccc(O)nc1)=O c1(C(NC2CCCN(C(=O)C=CC(F)(F)F)C2)=O)ccnc(C2CC2)n1.C CC1COc2c(C(N3CC(CNC(C4(C)CCCCC4(F)F)=O)C3)=O)cnn2C1 CCCCCC(CCCCC)C(=O)N1CC2CC1C2NC(C1CCC(=O)NC1)=O CC(C(C)(O)c1ccccc1)NC(=O)CCN1CCCCC1 N1(C(C(C2CC2)OC)=O)CC(C)CN(C(C2CC(OC(F)(F)F)C2)=O)CC1C c1(CC(=O)OC)occ(C)c1C(=O)N.C(C)CCC.C(=O)CC=C(C)C c1(C(C(=O)NCC(C)NC(=O)C(c2cccc(F)c2)(C)C)C)c(F)cccc1F CC1CC(NC(=O)C(C)(C)C)CN1C(C1(c2cccc(Cl)c2)CC(F)(F)C1)=O c1(C(N(CC(CNC(CNC(CC)=O)=O)(C)C)C)=O)ccccc1.CC#N.O c1(OC)cc(C(=O)NC2CCC(C(=O)Nc3cc(SC)n[nH]3)C2)ccc1F C12(CNC(c3c(C)nn[nH]3)=O)CCC1CCN2C(=O)CCC1CCOCC1 CC1(C(=O)NC2CC(C)C2)CCC(F)(F)C1.c1cccc(F)c1.C(=O)(C)N c1(CN(C)Cc2ccc(-c3cc(C(=O)O)ncn3)cc2)cccc(OC)c1 c1(CN(CCCN(C(c2cc(OC)ncc2)=O)C)C)nc2ccccc2o1 Cc1nccn1C(C)C(=O)NCC1(C(N2CCC(N(C)C)C2)=O)CCC1 C(CC1C(=O)NCC2(CCCC2)N1)SC.C1CCCC1.C(C)(C)C.C(=O)N N1(C(Cc2cn(C)nc2)=O)CC2CC(C1)CN(C(c1cc(Br)nn1C)=O)C2 C(=O)(CC(O)CC(C)C)N1CC(NC(c2ccc(C)n2C)=O)C2(C1)CC2 N1(C(C2CCCN(C(C(C)C)=O)C2)=O)CCN(C(=O)CCF)CC(O)C1 N1(C(=O)Nc2c(C(=O)OC)nccn2)CC23CCC2(COC3)C1 N1(C(C2(CCC)CCC2)=O)CCC2(CCC2)C1.c1(C=O)cc(S(N)(=O)=O)co1 C(C)(C(C)(C)CN(C)C)NC(CNC(CCc1cc(C)on1)=O)=O CCCCN=C(NCc1csc(CC)n1)N1CCC(C2CCCC2)C1 c1(C(=O)N)c(C)c(C)c(Br)c(C)c1C.C=C(C)CC(=O)NCC1(O)CCC1 c1(C(CC(=O)NCC2(OC)CN(C(C3(S)CCC3)=O)C2)O)ccc(Cl)cc1 N1(C(C2N(S(C)(=O)=O)CC2)=O)CCC(F)(C)CC1.C(=O)C=CC1CC1.N CC#CCC(C(=O)NCCSCC)NC(=O)CCc1nccs1 C1(C(=O)NC(CNC(CNS(CCCC)(=O)=O)=O)C)CCC(C2CCC2)CC1 C(C)(C)(CC(=O)N1CCSCC1CCNC(C1CN(C2CCC2)C1)=O)SC c1(C=O)cc(S(N)(=O)=O)n(C)c1.C1CN(C(C2(N(C)C)CC2)=O)CC1.C CCC(C)(CC)C(=O)N1CCC(OCCNC(=O)C#CC2(CC)CC2)CC1 C=CC(CC)CC(=O)NCCCN(C)C(C1CC12CCC2)=O C(=O)(C(C(=O)OC)NC(=O)CC(Cl)Cl)N1C(C=C)CC1 C(=O)(C(C)C(C)C(C)(C)C)OCC(=C)C=O.O(CC)CC C12(C(=O)OC)CCCOC1CN(C(=O)NCC(C)CS(N)(=O)=O)C2 C1(C(=O)NCCC(O)C)(OC)CCS(=O)(=O)C1.c1(C=O)ccc(F)c(C)c1 C1(C(=O)NCCCC=CC)(CC)CCN(C(=O)C(C)c2ccsc2)CC1 C1(CNC(CSCC)=O)C(C2CC2)CCN1C(c1ccn2ncnc2c1)=O c1(C(=O)NC2CS(=O)(=O)CC2NCCN2CCCC2=O)cnc2ncnn2c1O C1(c2n(C(CC)(C)C)nnn2)(NC(C2CC2)C2CC2)CCOC(C(C)C)C1 N1(c2cc(OC)ncn2)CCC2C(CCN2C(=O)Cc2c(C)cc(C)cc2C)C1 CC(C)CCC(C)N(C)C(C12CC(NC(=O)CCC3CCC(=O)C3)(C1)C2)=O N1(C(=O)OC(C)(C)C)CCCCC(COc2ccc(F)cc2C(=O)CF)C1 C1(CNC(C=C(CC)CC)=O)CC(OCC)CN1C(=O)C.C1CCCOC1.S c1(C(N2CCC(NC(c3c(C)onc3CO)=O)CC2C)=O)ccc2c(c1)CCC2 c1(C(N2CCC(O)(CNC(CCCCNC(C)=O)=O)C2)=O)cncc(F)c1C Cc1ccc(C)c(C(=O)N(CCN(C(=O)CO)C)C(C)C)n1.C1CCOC1 N#CC1CN(C(C2(Br)CC2)=O)CC1NC(c1ccc[n+]([O-])c1)=O c1(SC)nccnc1C(=O)NC1CN(C(=O)Cc2occc2C)CC1C Cc1cnc2c(C(=O)NC(CNC(C3(C)CCCO3)=O)C3CC3)cccn12 C(=O)(CCC#Cc1ccccc1)N(CCCNC(C1C(CC)OCC1)=O)CC C(=O)C1=CC2C=CC(C1)C2.CC(C)CCCC(=O)NC(CC1CC1)CC1CC1 C1(C(=O)NCCCOCCN(C(CSCCC(C)C)=O)C)CCCC1(F)F c1(C(=O)NC2CN(C(C(F)=C(C)C)=O)CC2C)ccccc1F.C(=O)C(C)C C12CC3CC3N1C2=O.C=CCCC.C(=O)(CCNC(=O)N)CNC.CC C1(C(N2CCC(C)(CNC(C3(Br)CC3)=O)C2)=O)COC2(CCC2)CO1 C1(NC(C=CC)=O)COC2(CCN(C(=O)CCC3CCC3)C2)C1 c1(CN2CCCC(C)(C(N3CC(O)C(O)C3)=O)C2)c(O)ccc2ccccc12 C1(C(=O)NC(C(=O)OC)(C)C)CCOCC1NC(=O)CC1CCCSC1 C(C)(C)(CC(C)C)NC(C1(CCCC)CC1)=O.c1(CC=O)c(C)n[nH]c1C.N c1(C(=O)NCc2ncc(CC)o2)ccncc1N=[N+]=[N-] C=C(C(=O)N(C(C)Cc1ccc(Cl)cc1)C)C1CC1 c1(OC(c2ccc(C#N)cc2)C(=O)NC)cc(C)cc(C)c1 c1(CC(=O)NC2(C)CN(C(C3N(C(CC)=O)CCCC3)=O)C2)ccc(Cl)cc1F CC(C(=O)NCC=CCNC(c1cc(C2CCCCC2)on1)=O)C(F)F C1COCCN(C(C2(F)CCOCC2)=O)C1.CC(C(=O)NC)NC(C1CCC1)=O N1(C(Cc2scc(C)c2)=O)C2CCC1CC(C(N1CC3CC(C)C3C1)=O)C2 c1(C(N2CCOc3ccccc3C2)=O)ccc2c(c1)S(=O)(=O)NC2 [N-]=[N+]=NCCCC(=O)N1CCC(CNC(c2ccc(F)cn2)=O)CC1 Cc1ccncc1CN(C(=O)Cc1cn(C)nn1)C.C(=O)(C(C)c1ccsc1)N C12(C(=O)NC(CCCC)CC)CNCC1S(=O)(=O)CCO2 N1(C(C2C(c3cn(C(C)C)nc3)OCC2)=O)CCC(CCC(=O)OC(C)(C)C)CC1 C(=O)(C(CC#CC)NC(=O)CCC(F)(F)F)N(CC#C)CCF CS(C)(=O)=NC(=O)C(=O)NC1CCN(C(c2cnn(C)c2)=O)CC1F.C1CCC1 O=C(N=c1[nH]nc(Cl)cc1O)NCC1CC12CCC2 C(CC(C)(C)C)NC(c1nc(CC)oc1)=O.c1(CC(C(=O)N)C)ccccc1Cl CN1CCC(OCC(=O)NC)CC1.C1C2CN(C(=O)CC)CC12.[SH](C)(=O)=O Cc1cccc(NC(C2CC2NC(=O)CCc2ccc(Cl)cc2Cl)=O)c1C#N C1(CNC(c2n(C)ccc2)=O)CCCCC1NC(=O)Cc1ccc(Cl)s1 C=CC(C)(C)CC(=O)NCC(CCC)C(=O)N1CCC12CN(C)C2 Cc1cccc2c1C(C)CC2CC(=O)NC1(CNC(c2cc[nH]c(=N)c2)=O)CC1 c1(C(CC)NC(N2CC3CC2C3NCC(=O)N(C)C)=O)cc(C)ccc1C N1(C(c2ccnn2C2CC2)=O)CCC2(C1)CN(C(C1Cc3nccnc3C1)=O)C2 CCCC(C)C(=O)NC(C1CCCCC1)C(=O)NCC(C1CC1)C1CC1 C1(C)(CC)CC(Nc2ncc(C(=O)OC)s2)CN1C(=O)C1=CCC1 N1(C(CNC(c2n[nH]c(=N)[nH]2)=O)=O)CCN(C(C2CSC2)=O)CC1 CCS(=O)(=O)CC(=O)N1CC(c2cn(C(c3cccnc3)C)nn2)C1 c1(C(N(CC(CNC(c2cn(CCC)nn2)=O)(C)C)C)=O)nc(OC)ccc1F c1ccccc1C1CCC(=O)N1.N1(C(C2(NC(=O)OC)CC2)=O)CCCCC1.N c1(C(=O)NCC(COC)NC(c2sc(F)cc2C)=O)cn(C)c(=O)cn1 N1(C(C(=O)NCC)=O)CCC(C2CCCN(C(C3(F)CC3C)=O)CC2)CC1 CCC(CCOC)C(=O)NC(C)CCCC(=O)NC(C)CC(C)(C)O C(=O)(C1CCc2ccccc21)NCCN(C(c1nc2ncc(Br)cn2n1)=O)CC C1(OC)CN(C(=O)CCc2n[nH]c(=N)s2)CC1NC(=O)CCc1cncnc1 C1C2CN(C(=O)CC)CC12.C1(N(C)C(=O)N)CC1(C)C.C(=O)C1CC1.C c1(C(=O)NC2CCN(C(c3nc(CC)sc3N)=O)C(C)C2)c(C)cc(C)nc1O C1(CC=C)(C(=O)NC2CC2CNC(=O)CCCF)CCCC1 C#CC1CCCC(NC(c2cc3sccc3[nH]2)C(=O)NCCCSC)C1 Cc1ccc2oc(C(=O)NCC3CN(C)CCN3C(=O)C#CC3CCC3)cc2n1 CC(CC(=O)NC1CC(F)(CNC(c2ccns2)=O)C1)c1cnn(C)c1 C1(C(C)C)CN(C(=O)CO)CCN1C(c1cc(CS(C)(=O)=O)on1)=O Cc1cccc(C)c1NC(c1ccc(OCC2CCCC(C)(C)O2)s1)=O C12(C(=O)O)COCC1CN(Cc1cnc(-c3ccccc3)nc1)C2 N1(C(C(C)(C)c2cncs2)=O)CCCC(C)(CNC(C2COCCO2)=O)C1 c1(CC(N2CC=CCC2)=O)cc(Cl)c2c(c1)OCO2.NS(=O)(=O)C1(C=O)CC1 Cc1ccc(CC(N2CCCC(N(C(=O)CN(C)C)CCF)C2)=O)c(F)c1F c1(C=O)cc(C(F)F)cc(F)c1.C1(C(C)(C)O)(C)CN(C(C2CCSC2)=O)C1 c1(CC(=O)NC2CCN(C(C(F)OC)=O)C2(C)C)cc(Cl)cc2c1OCC2 C(CCC(CCC)NC(=O)CC(C)OC)NCc1c(NC(CCC)=O)cccn1 N1(C(C2N(C(C(C(C)C)OC)=O)CC(O)C2)=O)CCC12CCOCC2 C1(CC)CCC(O)(C(=O)NCC(C)(C)CNC(c2cnc(OC)cn2)=O)C1 c1(SCC)ocnc1C(=O)N(C(C)C(=O)NC1(C)CN(C(=O)O)C1)C c1(CN2C(C(=O)O)CC(=C)C2)cc2c(C)cc(OC)cc2[nH]1 N1(C(CC(C)SC)=O)CCN(C(c2ccccc2C2CCC2)=O)CC1C C(COC(C)(C)C)(CF)(c1nnnn1C1COC1)N(CC(=O)OC)CCC C(=O)(CC1CN(C(=O)C2=NOCC2)c2ccc(Br)cc21)OC Cn1ncc(C(c2nnnn2CC2CCCO2)NCCS(C)(=O)=O)c1Br C1(C(=O)NCC(CC(C)C)NC(c2cnccc2Cl)=O)C2Cc3ccccc3C12 C1(C(=O)NC23C(C)OC(CC2)C3)COC2(C1)CN(C(=O)CCCc1ncco1)C2 N1(C(C(C)N2CCC2)=O)CCOCC(NC(=O)Cn2ccnn2)C1 c1(N2C(C(=O)Nc3n(C)ncc3)C3CCC2C3)ncnc2c1CCC2 N1(C(CC=C=C)=O)CCC2CCN(C(c3ccc(O)c([N+](=O)[O-])c3)=O)CC2C1 n1(-c2c(C)n[nH]c2)nc(C2(N3CCOCC3)CCCCC2)nc1C N1(C(C)C(=O)NCc2csc(CNC(=O)C)n2)CCCCC1=O.C1CC1.S O=S1(=O)C2CCC1CN(c1nc(NCC(F)CO)c3ccsc3n1)CC2 N1(C(CCCOCC)=O)CC2CC2(CNC(=O)C(c2ccccc2)(F)F)C1.N CC1(CO)C=CCN1C(=O)NCc1ccnc(Cn2nnc(=N)[nH]2)c1 Cc1cc(CCC(=O)NC(C)Cn2cc(C3CC34CC4)nn2)no1 N#Cc1c[nH]ccc1=NC1CCCC(NC(c2nnc(O)c3ccccc23)=O)C1 c1(C=O)ccc2c(c1)CCC2(C)C.C(CCCNC(=O)OC(C)(C)C)C1CC1 c1(C(C(OC)OC)C)cn(CCNC(c2ocnc2C2CC2)=O)nn1 c1(NC2C(C(F)(F)F)CCN(C(c3cnsc3)=O)C2)c(F)cc([N+](=O)[O-])cc1F CC1OCCN(C(c2ccc(NC)nc2)=O)C1C(N1CCC(n2ccnc2)C1)=O Cc1nc(NC2CCC(CNC(C3CCCCO3)=O)CC2)c(Cl)cc1C#N N1(C(C(F)OC)=O)CC2(CCOCC2)CC1CNC(=O)C(C)(O)C1CC1 N1(C(Cc2c(C)nc[nH]2)=O)CCN(C(C2CC(=O)NC2(C)C)=O)CC2(CC2)C1 c1(-n2cc(CC(C(N3C(C(=O)O)CCC3)=O)O)nn2)ccc2c[nH]nc2c1 N1(C(CCCC)=O)CCC(NC(C2CCN(c3ccccc3Cl)C2)=O)CC1CC CCCC(CCC)C(=O)N1CCC(N(CCO)C(c2ncsc2C)=O)C1 CC1CCN(C(C2(n3cccn3)CC2)=O)C(C(=O)NCC2(C3CC3)CC2)C1 Cc1nc2[nH][nH]cc-2c(=NCC(C)N(C)C(c2cnc(C(C)(C)C)o2)=O)n1 c1(C(=O)N)n[nH]nc1C.C1(C(=O)OCC)CCCN1C(C1COC(C)C1)=O C(=O)(CCCCC(F)(F)F)N1CC(CNC(C2C(C(C)(F)F)C2)=O)C2(C1)CC2 c1(C(=O)NC(C)CN(C)C(C2(F)CC=CCC2)=O)cc(S(N)(=O)=O)cs1 C1(C(=O)NCCNC(c2cnn(C)n2)=O)CC(=O)c2cc(Cl)ccc2O1 c1(OCCCC(=O)NCC(CNC(CCCSC)=O)OC)ccccc1Cl CC(CC(F)F)C(=O)N1CCCCC1CCC(=O)NCC(F)C1CCC1 C1(CC=C)CCN(C(=O)C(C)NC(=O)OCC)CC1.c1(N)ccc(C#N)cc1 Cc1ccccc1NC(=O)CCNC(=O)C=O.C1(c2ccccc2)CC1(F)F.N CC1CCC(CC(=O)NCC(C2CC2)N(C(=O)CSc2ccccc2)C)O1 C1(O)(C(N(C)Cc2nnc(CC)s2)=O)CCN(CCSC)CC1 CN1C(=O)CCCC1C(=O)NCC1CC1C(=O)NC1CC(O)C1O N1(C(c2c(OC)c(Cl)sc2)=O)CCC(C)(C)C(C)C1.C(=O)(CC1(O)CC1)N C1(CNC(C)=O)CCCCN1C(C1CN(C(=O)CCC(C)NC(C)=O)C1)=O S(=O)(=O)(c1ccc(C(=O)NC2CC2)cn1)N(C)C.c1(C=O)nc(Cl)cs1.C C1(NC(C(F)=C(C)C)=O)CC12CC(NC(=O)CCCc1cccs1)C2 C1(C(=O)NCCC(CNC(Cc2c(SCC)cccc2)=O)O)CCCCC1(F)F Cc1nc(C(N2CC(CNC(c3c[nH]c(C#N)c3)=O)CC2C)=O)[nH]c1C c1(C(=O)NC(CNC(c2nc(COC)oc2)=O)(C)CO)nc(OC)ccc1C C12(CC)CCC1CN(C(c1nc(C)c(C)s1)=O)C2.C(C)(C)(C=CC=O)SC CC#CCC(N)C(=O)N1CCCC(N2CCC2)C1 N1(C(=O)C2=COCC2)CCC(C(=O)NCC2CC(F)C2)C(O)C1 Cc1nc(C)c(F)c(=NCC(C2CC2)NC(=O)CCCc2ccccc2Cl)[nH]1 N1(C(c2cc(C)sn2)=O)CCC2(NC(=O)CCc3cnc[nH]3)CCCC12 Cc1nc(NC2CCC(NC(C3CCS3(=O)=O)=O)CC2)c2ccsc2n1 N1(C(CCC(=O)NCCC)=O)CCC(C(=O)NCC2CC2Cl)C12CCC2 c1(C(=O)NC2(CN=c3nc(COC)[nH]s3)CCCCC2C)cccc2nccn12 C(=O)(CC(O)C(C)C)N.C1CC(c2cn(CC)nn2)(N(C)C)C1.[SH](C)(=O)=O CC1(C)C(NC(=O)CCC2CC2)CCN1C(c1ccc(-n2ccnc2)nn1)=O C(=O)(C(C(CC)CC)OC)NCC1COCCN(C(c2nc(CC)sc2)=O)C1 c1(C(N2CCC(CCNC(C3CCSC3)=O)C2)=O)ccccc1SC(F)(F)F C1(NC(c2c(F)cc(C)c(O)n2)=O)CN(C(=O)OC(C)(C)C)CC12CCOCC2 n1(CC=C)nc(-c2ccccc2)nc1CN(C1CCOCC1)CC1CCOC1=O c1(C(N(CC(N2CCC(CC3CC3)C2)=O)C(C)C)=O)cc2cccn2cn1 CC1CC(C)CN(C(C2(C)CC(C)(C)C2)=O)C1.c1ccc(Cl)nc1.C(=O)(C)N N1(C(C(CCOCC)NC(=O)CC=CC(C)(C)C)=O)CC(C)C(N=[N+]=[N-])C1 N1(C(c2c(C)n[nH]c2)=O)CCC(C)C(NC(c2ncnn2C)=O)C1C c1(N2CCN(c3nnc(C)o3)CC2)ccc(S(=O)(=O)NC(C)C(C)(C)C)c(Cl)c1 CCC(C)(C)CC(=O)N(C)CCN(C(=O)C(C)(F)CC)C N1(C(c2c(N(C(C)=O)C)cccc2)=O)CCCCC(NC(c2cc(C)no2)=O)C1 c1(CC)cc(CN2CC(=O)N(CCc3ccncc3)C2=O)cc(C)c1.[nH]1cccn1 C1CC2(CO1)CN(C(=O)C)C2.c1(CC)ccsc1C(=O)N.c1cc(C)on1.C C(=O)(C1=CC2C=CC1C2)N1C(C)(CNC(C(C2CCC2)OC)=O)CCC1 N1(c2c(C#N)nccn2)CCC2(CCN(C(=O)C(O)Cc3ccccc3)C2)C1 C1(CC=O)CN(C(C23CC(CC(F)F)(C2)C3)=O)CCN1CC1CC1(C)C C(=O)(C(=O)N=S(C)(C)=O)N(C1CCCN(C(=O)CNS(C)(=O)=O)C1)C C(=O)(CCC(CF)CF)NC1CC(O)(CNC(COc2cc(C)on2)=O)C1 C1(CN(C)C(C2CCN2C(=O)C(F)n2ccnc2)=O)CCCC1 c1(C(N2CCC(N(C(COCC(=O)OC)=O)C)C2)=O)cn2ccc(O)cc2n1 C1(CC(=O)N(C)CCN(C(=O)C(C2CCCCC2)=O)C)CCCOCC1 C1(OC)COCCC1NC(=O)C(=O)N(CCF)C(C)C Cc1nc2ccc(C(N3CC4CC3CN(C(C3CCN(C)CC3)=O)C4)=O)cc2[nH]1 c1(NC(C23CC(NC(c4cnc(Cl)cc4I)=O)(C2)C3)=O)nccc2occc12 C1(C(=O)NC2C=CCN(C(=O)C(C3CCCCC3)O)C2)CCCC2(CC2)C1 N1(C(C2(OC)CCOC2)=O)CCC2CC2(C(=O)NCC(C)(C)SC)CC1 CC(C)CC(C)(CNC(c1cccc(C2CC2)n1)=O)NC(=O)C1=CCCOC1 C#CCCCC(C(=O)NC(C)CC)N1CCN(CCOC)CC1C N1(C(C2C(CC)N(C(c3cccc(C)c3)=O)CC2)=O)Cc2ccsc2C1 C(CCCCCNC(=O)Cc1sccc1Cl)N(C(=O)CC1CCC(=O)N1)C C1(CNC(c2c(CC)onc2)=O)CN(C(c2cc(C)ns2)=O)CC1C O=C1NCC2(C(N3CCOCC3C(F)F)=O)CCC1C2 C(=O)(CCCCC1CC1)NCC(COC)NC(=O)Cc1nocc1C(C)C C1(C)(NC(c2ccn(CCC)n2)=O)CCCN(c2nn[nH]n2)C1 c1(NC(CC2(N(C)C(C3CC3[N+](=O)[O-])=O)CC2)=O)cn(C)c(=O)nc1O C1(C2CN(C(C3CC=CCC3)=O)C2)(NC(c2cn(-c3cccnc3)nn2)=O)CC1 C1OCCOC1(C)C.n1(CCNC(C2C(OC(C)C)C2)=O)cc(CO)nn1 c1(CC(=O)NC2C(c3cn(C(C)CO)nn3)C2)ccc(CN2CCNC2=O)cc1 CC1CN(C(=O)C=Cc2ccn(C)c2)CC(C(=O)NCC(C)(C)CO)O1 C1(C(=O)NCC2CCCN(C(c3cn(C)nc3O)=O)C2)CC2(C1)CC21CCC1 c1(CCNC(N(C2CCS(=O)(=O)C2)CCOC)=O)c[nH]c2ccc(Cl)cc12 c1(C(N2CC3CN(C(c4c(C)n[nH]c4)=O)C3C2)=O)ccc(Cl)c2cc[nH]c12 O=[N+]([O-])c1cc(CNCc2nnc3ccccn23)cc(C(F)(F)F)c1 C=CC(C)(O)CC(=O)N1CCN(C(=O)C(SC)SC)C(CF)C1 N1(C(CC)=O)CCS(=O)(=O)C(CC)C1.C(=O)C(F)=C(C)C1CC1.CC(=O)N C(=O)(C(O)P(C)(C)=O)N(C)CC1(C)CC1.c1(C=O)nccs1.C1CC1 C1(NC(c2ccc(C)o2)=O)CCN(C(=O)Cc2ccc(C)c(F)c2)CCC1CO c1(OCC)cccc(C(=O)NCC2CN(C(=O)C)C2)c1.c1ccc(C)cc1 n1(C(C)C)c(O)nc(N2CC(C)(NC(=O)CC3CCCCC3O)C2)cc1=O Cc1ccc(C(=O)NCCCO)cc1S(C)(=O)=O.c1(C(=O)N)ocnc1C1CC1 c1(C(N2C3CN(C(c4cnc[nH]4)=O)CC2CC3)=O)cc2cc(Cl)ccc2[nH]1 N1(C(c2cc(C)no2)=O)CC2C(CNC(=O)Cn3cnccc3=O)C2C1 c1(CC(=O)N(C(C(=O)N(C2CCCOC2)C)C2CC2)C)cccc2c1CCC2 C(=O)(CCC(C)CN(C)C)N1CC2C(C(N3CCN(C(COC)=O)CC3)=O)C2C1 C1(C(C)NCc2ccccc2-n2cc(C(C)(C)O)nn2)CCc2ccccc2O1 C1(C)(NC(C(N2CCCCCC2)C)=O)CCCN(c2nnc(C(N)=O)s2)C1 C1(C(N(C2CN(C(C3CCOC3c3cccnc3)=O)C2)C)=O)CC2C=CC1CC2 CC1CC(NC(=O)CN2CCCCC2=O)CN(C(c2ccc(CO)nc2)=O)C1 c1(N2CCC(C3N(C(c4n(CC)ncc4)=O)CCCC3)C2)nc(C)nc(Cl)c1C c1(C(=O)NCC(CNC(CC2CN(C)C2)=O)C(F)(F)F)[nH]c2ccccc2c1Cl C1(C(N(C2(CC(=O)NCCc3nncs3)CC2)C)=O)CCSC1 C1(CC(N2CC(C)(O)C2)=O)(NC(c2coc(CO)c2)=O)CCCCC1 N1(C(CNC(C=CCC)=O)C)CCN(C(=O)Cc2ccc(F)cc2)CC1 c1(C(=O)NC2C(F)CCN(C(c3cc(N)c(Cl)cn3)=O)C2)c(F)ccc(F)c1Cl c1(OC)cncnc1NC(=O)C(=O)NCC(c1ccccc1)N1CCCC1=O N1(CCOC(C)C)CCC(C(=O)NCC=C(Cl)Cl)C1C c1(C(N(C(C)C(=O)C(COC)=O)CC)=O)ccnc2c(Cl)c(C)ccc12 N(C(=NCCc1ccc(F)cc1)NCc1cccs1)CC1(C)CCC1 C1(CNC(c2c(CCC)nco2)=O)CC2CCC1C2.c1(C=O)cc(C)ccn1.N CC12CCCC(C(N3CCC3CNC(c3cncc(N)n3)=O)=O)(CO1)C2 N1(C(CNC(CC)=O)=O)CCCCC(C(=O)NCC(CO)C(C)C)C1 C1(NC(CC2(C#N)CC2)=O)CCC12CCN(C(c1cc(C3CC3)[nH]n1)=O)CC2 C1(OC)(O)CC(C=O)C1.C1(C(C(=O)NCC)O)CC(F)(F)C1.C1CC1 N1(C(COCC#C)=O)CCC(CNC(=O)Cc2sccc2-c2ccccc2)C1 CS(=O)(=O)c1cccc(C(O)CNC(=NCCCCl)NCC2=CCCOC2)c1 n1(CCC=O)cc([N+](=O)[O-])cn1.n1(C(C)C)ncnc1C(=O)N.C1(CC)CC1 c1(C(=O)NC2C(NC(C(=C)F)=O)CCC2)cnc(C)c(C)c1 C(=O)(CC(C)C(F)(F)F)NCCCNC(c1cnc(NC(C)=O)o1)=O C(CCC(C(=O)N(C)C)NC(c1ccc(Cn2nc(C)cc2C)cc1)=O)OC C1(CC=C)(NC(=O)C=CCF)CN(C(C2C(CN=[N+]=[N-])C2(C)C)=O)C1 C1(F)(CNC(c2c(COC)cccc2)=O)CCCN(C(=O)C(F)C(C)C)CC1 CC1CCC(C)(NC(=O)C(O)C2CN(C(=O)CC3CC4(CCC4)C3)C2)C1 C1(N(C(COCC=C)=O)C)CN(C(=O)CC2C=CS(=O)(=O)C2)CC1O CC1CN(C(=O)CC2CC2)CCC1NC(=O)COc1ccc(F)c(F)c1 C(=O)(CCC(C)CN(C)C)NC1(CC)CN(C(c2occ3c2CCC3)=O)C1 c1(C(N(C)CCNC(C2CCC23CCCO3)=O)=O)cc2c(F)cccc2[nH]1 N(C(=NCCc1cccs1)NC(C)CC#C)C(C#C)CC1CCOCC1 CC(C)CC(CC(=O)N1CC2(CCN2C(C2CC3(C2)CC(O)C3)=O)C1)CC(N)=O c1(C(=O)NC(CNC(C(CCC)C#N)=O)C2CC2)cc(F)c(F)c(F)c1F c1(OCC(=O)NCC2CC3(CC3)CN2)ccc(C(F)(F)F)cn1.C1CCC1 c1(N(CCCOC(C)C)C)nc(=NCCc2cc(Cl)cc(Cl)c2)[nH]c2c1SCC2 C(=O)(C1(C)CCCc2ccccc21)N1C(CNC(COC)=O)c2ccsc2CC1 CCC(C)C(C(=O)NC1CCN(C)CC1)N(C(=O)COC1CCOC1)C N1(C(C)=O)CC=C(c2ccnc(NCc3cc(OC(C)C)ccc3O)c2)CC1 N1(c2nc(C#N)c(Cl)s2)CC(CNC(c2cc[n+]([O-])cc2)=O)OC2(CCC2)C1 C1(N(C(c2c(C)cccc2)=O)C)CN(C(=O)Cc2ccccc2Cl)CC12CC2 C1CC2CN(C(C34CC5CC3C4C5O)=O)CC12.C(C)(C(=O)N)NC(COC)=O C(=O)(C1=NOC2(CCOC2)C1)N(CC(C)NC(c1cnc2[nH]cnc2c1)=O)C C1(NC(C(CC=C)N(C)C)=O)(CO)CCCN(C(c2cnn(CC)c2CC)=O)C1 C1(NC(COCC)=O)CCN(C(=O)CCc2ccc(O)nn2)CC1C c1(C(N(C2CCN(C(=O)C(Cl)=CCl)C2)CCC)=O)ccn(-c2ccccc2)n1 CC(CC(N)=O)C(=O)NCc1ccc(C(=O)NCC2CCCSC2)cn1 C(=O)(CC1=CCN(C(=O)CC2CSC2)CC1)NC(C)(C)CC1CCOC1 CCC(O)C(=O)NCC(=O)NC(C)CN(CCCF)C C1(C2CN(C(C3CC34CC(O)C4)=O)C2)(NC(C(N2CCCCC2=O)C)=O)CC1 C1(C=O)CCc2nn[nH]c2C1.N(C)(S(=O)(=O)N(C)C)CC(=O)NCCCCC.N C(=O)(CC(C)(C)c1cccc(Br)c1)NC(CC)CSC CC1(C(=O)NCCO)CCCC1(F)F.c1(C(N2CCCC2)=O)cc2c(s1)CCC2 N1(C(c2ccc(C)c(Br)c2C)=O)CCC2CN(C(=O)C(N)=O)CCC2C1 CC1CC(NC(=O)Cc2ccon2)CN1C(=O)CCC(=O)c1ccc(Cl)s1 c1(NC(=O)NCC(C#C)OC)cc(C(=O)OC)c(C)s1 N1(C(c2c(CC)n(C)nn2)=O)CC(NC(=O)C=O)C(F)C1.CC.C(C)=O.N C1(C(=O)NCC(=O)NCC2CC2)CC1.CC(=O)NCC c1(N2CCC(=CCNC(Cn3c(C)cnc3)=O)CC2)ncc([N+](=O)[O-])cc1C#N N1(C(C(CC)Cl)=O)CC2CC(NC(c3ncn(C)c3C(F)(F)F)=O)C1C2 C1(C(C)(C)NC(CCN(C(C(C2CCCC2)OC)=O)CCO)=O)CCCCO1 C1(C(=O)NCC(C)NC(c2cc(Br)no2)=O)CNC(=O)CC12CCC2 O=C1CCCCN1CCC(N1CC2C(C(N3CCC(C(F)(F)F)CC3)=O)C2C1)=O Cc1cccc2c1CCCC2NC(=O)NCCCOC1CCCCCC1 c1(CNC2C(C(=O)Nc3c(C)ccc(Br)n3)C2)cc(C)c(F)c(F)c1 C(=O)(C(COC)CC(C)C)N1CCN(CCNC(CC(CC)CN(C)C)=O)CC1 C1(C(=O)NC(C)CCNC(C2(C)CC2)=O)Cc2ccc(Cl)cc2C(=O)O1 C1(NC(c2ccc(CC)cc2)=O)CN(C(C2CCCCO2)=O)C2(CCOCC2)C1 N1(C(C(NOC)=O)=O)CCN(C(=O)C=CC2CCOCC2)C(C2CC2)C1 C1(C(N2CCCC2)=O)CCC2(CCC2)OC1.C(CC(=O)NC)NC(=O)OCC c1(OC)cc(-c2ccc(CN3CCOCC3(C)CO)cc2)cnc1Br N1(C(C(C)N(C(CCC=C(C)C)=O)C)=O)CCCOC(C)C1 c1(C(=O)OCC(C)C)cc(N(C)C)c2ccccc2n1.C1(CN(C)C)CCC1 N1(C(C(CC)C#N)=O)CC(CNC(c2cn3cccnc3n2)=O)CC12CCC2 C(=O)(C(F)(F)C(O)C(C)C)NC(C1CCCC1)CNC(CCCCCC)=O CCCCCCCN(C)N1CCCC1Cc1cccc(S(C)(=O)=O)c1 CC(C)C(C)C(=O)NC(Cn1cncn1)C(=O)N(C)CCN(C)C(C)=O C(C(=O)NCC)(C(C)C)OCC.c1(CC=O)cccc(CC(F)(F)F)c1.N c1(CC(N2CC3C(N(C(c4c(C)nco4)=O)C)C3C2)=O)cc2cc(Cl)ccc2[nH]1 C(=O)(CCCCCN(C)C(c1cnc(N)cn1)=O)NC(C(CC)C)CO Cc1c(C(N2CCCC(CN(C(=O)CC(C)(C)F)C)C2)=O)cccc1Cl c1(OC)ccc(NC(=O)C(C)C(C)NC(C2(F)CCCCC2)=O)cn1 C1(NC(C(CNC(=O)C(C2CCC2)OC)OC)=O)CCCC2(CC1)CC2 c1(CC)nc(Cl)c(CC)c(=NCC2CCCN2C(=O)C(C)C)[nH]1 Cc1cc(C(=O)NCC(C)NC(=O)Cc2sc(SC(F)F)nc2C)sc1C C1(NC(C)=O)CC2(C1)CN(C(=O)C=Cc1ccco1)C2 C1(C(N2CC3(CCN3C(c3sccc3Cl)=O)C2)=O)CS(=O)(=O)CC12CCC2 Cc1oc(Br)cc1C(=O)NC1(C2CCCN2C(c2cc(C(C)C)[nH]n2)=O)CC1 c1(C(=O)N)nc2ccccc2s1.C(C)(C(C)C)NC(c1cnc(OCC)s1)=O C1(C(=O)NC)COCCN1C(C1CC(NC(=O)C(=O)C2CCCC2)C1)=O c1(NC(c2ccc(COc3c(C)cccc3)cc2)=O)ncc(Cl)cc1Cl C1(CC(NOCC=O)=O)C=CS(=O)(=O)C1.c1(CC)ccccc1Cl C1(C)CN(C(=O)CC2(C)CCS(=O)(=O)N2)CCO1.C(C(=O)N)OCC.C C(=O)(C=CS(C)=O)NCC(c1ccccc1F)NC(c1nc(C(C)C)oc1)=O C1CC(F)(F)CN1C(=O)C=CC(C)(C)C.c1(SC)ccc(C(=O)N)s1.C N1(CC2(NC(CCC3C(C)C3)=O)CC2)CCN(C(c2cn(C)[nH]c2=N)=O)CC1 C1(C(N2C(CN(C(CCCC=C)=O)C3CC3)CCC2)=O)CC2OC1C1CC21 CC(CCC(=O)NCC1(C)CCN(C(c2cc(O)n(C)n2)=O)C1)c1ccccc1 CCC(F)(F)CC(=O)NC(C)(CO)C(=O)N1CCC(N2CCC2)C1 c1(NC)ccccc1C(=O)NC(C)(CSC)C(=O)NCC1(F)CCOCC1 C1(NC(c2csnn2)=O)CC(O)CN(C(=O)C(F)(F)c2nccs2)C1 c1(OCC(=O)N(CCOCC)C)ccc(F)c(Br)c1.N12CCC(C1)C2=O [nH]1c(C)nn(CC(=O)N(C)CCN(C(C23CCC2C3)=O)C(C)C)c1=O.CC N1(C(CCCC(C)C)=O)CCCC(NC(=O)COc2ccsn2)CCC1 C12(CCNC(C3CCCS3)=O)CCC(C1)N(C(=O)CSCC(F)(F)F)C2 c1(C(=O)NCC(CNC(CCn2c(C)ncc2)=O)C)cn(C)nc1C1CC1 C#Cc1nccc(C)c1NC(C1C=CCCN1C(=O)CCOCC(C)C)=O CCC(C)C(=O)N1CSCC1C(=O)NC1CC1C.c1(CC(=O)N)ccsc1 Cc1cc(Br)cc(F)c1CNC(=O)Nc1cncn1-c1cccnc1 C1(CC(=O)Nc2c(CC)noc2)C2CN(C(=O)CC(C)CC)CC12 C(C1CCN(C(=O)CS)CC1)=CC(=O)NC(c1ccc(O)nc1)C.C1CC1 N1(C(c2ccn(CCC)n2)=O)CCC2(CC1)CC(NC(=O)CC(C)(C)O)CCO2 N(C1COc2ccc(Cl)cc21)C(=O)Nc1cc(CC=C)no1 CON(CCC(=O)N1CC(CC2CCCC2)C2(CC2)C1)C(=O)OC(C)(C)C n1(CCC)cc(C(=O)NCCC(=O)NCC(C)C)nn1 C=CCC(CNC(c1[nH]nnc1C1CC1)=O)C(=O)NCC(C)C(C)(C)C N1(CC)CC2CCC(C1)N2Cc1ccc(C=CC(=O)Nc2cn(C)nn2)cc1 Cc1ccc(C(=O)NC(CC2CC2)C(=O)NC2(CO)CC3CCCC23)cc1C c1(N(c2nc(C)cc(C(=O)OC)n2)CC2CCNC2)nc(SC)nc(C)c1Br CC1(C2CCN(c3nc(N4CCN(C5CCC5)CC4)nc(C4CC4)n3)C2)CC1 c1(C(=O)NC2C(NC(C3(OC)CCCC3)=O)CCCC2)cc2c(cn1)OCCO2 c1(OC)ccc(Cl)cc1CC(N1CCCCC1C(=O)NCC1(O)CC1)=O C#CC1(C(N2CCCC3COCC23)=O)CCN(C(=O)CC2CCCN2C)CC1 c1(C(=O)NCCC(C(C)C)C)c([N+](=O)[O-])cc(S(C)(=O)=O)cc1[N+](=O)[O-] C1(NC(c2cnn(CCF)c2)=O)CCCCC1NC(C1(C2CCCO2)CCC1)=O N1(C(C(CC)n2ccnc2)=O)CCC2(CCN(C(c3ccn(C)n3)=O)CC2)C1 C(c1cccs1)=CC(=O)NC1CC(F)(CNC(c2cc(F)n[nH]2)=O)C1 Cc1ccc(-c2ccccc2C(=O)NCC(C)CNC(=O)CC)cc1.C(C)C.S C1(NC(=O)C(C2CCCC2)NC(C2CC23CCCC3)=O)CCCCCC1O C1(C(=O)NCCSCC)OCCC1NC(=O)CCC1CCCCO1 c1(C(=O)NCC(CCC)NC(=O)C=CSC)ccc2nn[nH]c2c1 Cc1nn(CCNC(c2ccc(-c3ccccn3)o2)=O)c2ncc(S(N)(=O)=O)cc12 c1(CC(=O)N(C2CCN(C(C3(O)CC3)=O)C2)CCC)ccccc1OC C1(NC(c2cnn(CC)c2C)=O)CN(Cc2ccn(C3CCCC3)n2)CCC1C N1(C(C(C)NC(=O)NC)=O)CCCC1C(C)(C)C.C(=O)CCC.C=O.N C(=O)(CC(O)C1CCCC1)N(C1CCC1C(N1CC(NCCO)C1)=O)C N1(S(CCC(C)OC)(=O)=O)CCC2(CCCCO2)CC1 C(=O)(C(CC)CCCCC)NC(CC=C)CNC(c1ccc(CO)c(Cl)c1)=O C(=O)(CCCCC(F)(F)F)N(CCC(C)NC(=O)COCc1cnn(C)c1)C C1(NC(=O)CCc2nc[nH]n2)CN(C(=O)CC2CCC(O)C2)CC1CC1CC1 N1(C(C(c2cnccn2)C)=O)CCC(C2(NC(C3CC34CC(O)C4)=O)CC2)C1 N1(C(C2N(C(C3(C=C)CCC3)=O)CCC2)=O)CCn2c(O)nnc2C1 c1(C(N2CCn3ncnc3C2)=O)cscc1C1=Cc2ccccc2C1 CCCCC(C(=O)N1CCC(CC)(CC)C1)NC(=O)CN(C)C(C)=O C12(COC(c3c[nH]c(=NC)s3)=O)CC(C(=O)OC)(C1)C1(COC1)O2 C(=O)(C(F)CC(C)C)NCC1N(C(CCC(=O)NCCC)=O)CC=C1 CC(C)C1=CCC(NC(C2CCCCCCN2C(c2nccs2)=O)=O)CC1 C(=O)(CC(O)C(C)C)N1CCN(c2nc(C)c(CNCCN(C)C)s2)CC1 C1(CC=C)(NC(=O)C2CC2)CN(C(=O)C(C)N(C2CCCCC2)CC)C1 Cc1cc(C)c(C(=O)NC2(C(=O)NCCN3CCCC(O)C3)CCCC2)cn1 N1(C(C2C(COC)(COC)C2)=O)CC2CC(C1)CN(C(=O)C(C)C)C2.S CC(C)(C)C(CO)C(=O)N1CC2CC(NC(=O)Cc3cccc(Cl)c3Cl)CC1C2 N(C1CN(C)Cc2ccccc21)C(C1CC(N)(OC)C1)=O Nc1ncccc1CC(=O)NCC1CCCCN1C(c1cnnc(C2CC2)c1)=O c1(C(=O)NC2C(CNC(c3c(OC)cncn3)=O)C2)ccc2cc[nH]c2n1 C1(NC(C2CCC3CC3CC2)=O)CC1C1CCCN(C(c2cc(Cl)no2)=O)C1 C1(C(N2CCCC(C)C2)=O)(COC)CCN(C(=O)CS(C)(=O)=O)CC1 C1(C=O)CC1C1(C)COC1.C1(N(C)C(c2cc(C(N)=O)co2)=O)CCCCC1.N N1(C(CCCOCC=C)=O)CC2CC(C1)N2C(c1cc(CC)c[nH]1)=O N1(C(c2cc(CNC(C3(O)CCOC3)=O)on2)=O)Cc2cc(O)nnc2C1 N1(C(c2c(CC)ncnc2)=O)CCC2C(C1)CN2C(C1CCC2CC12)=O Cc1cc(C)c(C)c(S(=O)(=O)N2CCC(C(=O)OCCCCCBr)CC2)c1C CC1CCC(CNC(c2cc3ccsc3s2)=O)CN1C(=O)Cc1ccno1 c1(-c2cc(F)c(SC)c(F)c2)cnn2c1CN(C(c1cncc(F)c1)=O)CC2 N1(C(C(COC)N(C)C)=O)CCN(C(c2cnn(C)c2C)=O)C2CCC12 S(=O)(=O)(CC(=O)NC12CC(C1)N(C(c1ccc(COC)s1)=O)C2)NC C(=O)(C1OCCn2ccnc21)NCC1(C)COCCN(C(CC(C)(C)O)=O)C1 C#CC1(C)CCCN(C(=O)CCC2CCN(C(C3(CC)CC3)=O)CC2)C1 CC(CC(=O)NC(C)(CNC(=O)C(C)(C)c1ccccn1)C1CCC1)C1CC1 c1(C(N(C(C(C)C)C)C)=O)ncoc1CNC(=O)CC1CSCCO1 c1(C(N)CNC(c2nn[nH]c2-c2ccccc2)=O)ccc(Cl)c(Cl)c1 Cc1cccc(C(=O)C(=O)N(C)CCN(C(=O)CSC2CC2)C)c1 CCCCC(CNC(c1cnn(CCF)c1)=O)NC(=O)C(C)CF C(=O)(CCCC(C)CC)NC(COCC)C(=O)NC1CNC(=O)C1 C(CCO)(C(=O)N1CC2C(CNC(C3(c4cccnc4)CCC3)=O)C2C1)N(C)C c1(NCC(COc2ccc(SC)cc2)O)ncc(Cl)cc1O CCC(C)CCCC(=O)N1CCC1CC(=O)NCCC(F)(F)F N1(C(c2cccs2)CC)CCN(C(=O)Nc2conc2-c2ccccc2)C(C)C1 C1CC(=O)N(C)C1=O.N1(CC)CCOCC1C(=O)N(C(C)(C)CC(=O)N)C.C C12(C(=O)NC3CCN(CCCC)CC3)CC(C)(CN1C(=O)O)C2.C(C)(C)C Cc1cc(C(c2nnnn2CC2CCCO2)Nc2ccccc2)ccc1C1CC1 CC1(C)CC(CC(=O)NCC(C)(O)CNC(c2cn(CCCF)nn2)=O)CCO1 N1(C(c2ccc(CSCC)cc2)=O)CCCC(C)C1.c1(C(=O)N)cnn(C)c1 C1(NC(CCN(CCC(C)(C)C)C)=O)CC2C1CCN2C(=O)Cn1cccc1 Cc1cc(C(C)(C)C(=O)NCC2CCC2)ccc1F.C(=O)C(=O)C(C)(C)C.C C1(F)(CNC(CCc2scc(C)n2)=O)CCN(C(=O)CC2CC(O)C2(C)C)CC1 C(c1c[nH]c(=N)c(C)c1)=CC(=O)N(CCC=O)CCO.C(=O)NC.CC N1(C(C2CC(SC)C2)=O)CCC(C(C)(O)C)CC1.C1(C)(C=O)CC(C)(C)C1 C1(C2CN(C(=O)OC(C)(C)C)C2)(N(C)C(C2(F)CCC2)=O)CC1 C1(CCOC)CCN(C(=O)C(O)CCNC(=O)CN(C)C2CC2)CC1 c1(C(=O)NC(C)CNC(c2cnc(O)cc2O)=O)cccc2nc[nH]c12 C1(CNC(C2N(C)C(=O)CC2)=O)CCCC2(CCN(C(C3OCCO3)=O)CC2)O1 CC1=C(C)CC(C(=O)NC23CCC2CN(C(=O)CCn2cccnc2=O)C3)CC1 CC1CN(C(C2CCC(NC(C3(C)COC3)=O)C2)=O)CC(C)N1C c1(N(C2CCC(NC(C(CCCOC)C)=O)CC2)C)ccc(S(C)(=O)=O)cn1 C(=O)(CC(O)CC(C)C)N1CCN(C(CCCCC#C)=O)CC1C1CC1 C1(NCC2(P(C)(C)=O)CC2)CCCN2CCCC12 C(=O)(C=C1SCC(=O)N1C)NC1CC(C)N(C(c2cc(F)ccc2N)=O)CC1 C1(CC)CCCN(C(c2nc(C)c(Br)s2)C(=O)NCC(F)F)CC1 C1(C(F)(F)F)(C=O)CC(F)(F)C1.c1(C(N(CC=O)C)=O)ccoc1.CCC c1(C(N2CCC(NC(C(C)OCC#C)=O)C(O)C2)=O)nc2ccccc2cc1Cl c1(-c2cn(CCC(=O)N3CC(CC4CC4)C3)nn2)ccc(SC(F)(F)F)cc1 C1(F)(CNC(C(CC)COC)=O)CCN(C(=O)C(c2cc(C)cc(F)c2)C)CC1 N1(C(C2C(CC)OCC2)=O)CC2(CCN(C(c3ccc(=NC)[nH]c3)=O)CC2)C1 C1N(C(C2CC2C(F)(F)F)=O)CCCC1(C)C.CC(C)(C)OC(=O)NC C1(CC(N)=O)(NC(c2c(C)nc(CO)s2)=O)CCN(C(c2cccnn2)=O)CC1 n1(C(CC)CC)nc(Cc2cccnc2)nc1-c1ccnc(CO)c1 N1(C(CSC)=O)CCCC12CCN(C(=O)C(C1CCCO1)N(C)C)CC2 C1(NC(CCC(CC)C)=O)CCS(=O)(=O)C12CN(C(=O)CCC(C)(C)OC)C2 Fc1cc2c(cc1F)C(Nc1nc3c(c(=NCCC4CC4(Cl)Cl)[nH]1)COC3)CC2 C1(CC(=O)NCC2N(C(CCCOC)=O)CC3(CC3)C2)CCCC2(CCC2)O1 Cc1ccc(C(=O)NC(C)CC(C)NC(c2c[nH]c(C)cc2=O)=O)c(O)n1 S(=O)(=O)(c1cccnc1NC(C)C1CC1)N(C)CC1CCN(CCC)CC1.O c1(C(N2CCCC(CCNC(C(CCC)C)=O)C2)=O)cc(C)nc2c1cnn2C c1(C(N2CCC(N(CC(=O)NC(C)C)C)C2)=O)ccc2nnn(C)c2c1 C(=O)(C(CCC)C(C)C)NC(C(=O)NC(C#C)C(C)C)COCC C(C)(C(=O)N1CCC(C(=O)N(C)C)C1)(N(C(C(C)c1ccsc1)=O)C)C1CC1 N1(C(CCCC#CC)=O)CC2CCC1C1CN(C(=O)C(C)CC(N)=O)CC21 C(c1ccncc1)=CC(=O)NCC(CCC)NC(C1NC(=O)CC1C)=O C#Cc1ccc(C(N2CCC(C(=O)O)C(C(C)C)C2)=O)cc1F N(C1CCCc2c[nH]nc21)C(C1N(C(c2c(C)cc(C)nc2)=O)C2C(C1)C2)=O C=CCCCC(=O)N1CCC(N(C)C(c2cc(Cc3ccccc3)[nH]n2)=O)C1 CC#CCCCC(=O)NC1CCC(NC(c2csnc2-c2ccccc2)=O)CC1 Cc1cccc(SCC(=O)NC(C2(O)CN(C(c3cccnc3N)=O)C2)C)c1 C1(C(=O)NC(C)(C)CNC(C2CCC3(CC3)C2)=O)CNC(=O)CC12CCC2 C1(F)(C(=O)NCC(n2cc(C3(CO)CC3)nn2)C)CCCC1 C#CCC(C)(C(=O)NCc1cncs1)NC(c1cncc(Cl)c1)=O C1CCCN(C(=O)CC(C)CN(C)C)C1.C1(O)(CC(=O)N(CC)C)CCC1 N1(C(c2cc(C)c(Cl)c(C)c2)=O)C(C)CC2CN(C(=O)Cc3nnc(O)s3)CC12 C1(C(=O)OC)COC2(CCC2)CN1C(=O)Cc1cc(C)cc(F)c1 N1(C(c2c(C)nsc2)=O)CCC2C(CCCN2C(=O)C=Cc2cnc[nH]2)C1 O=C(N=c1[nH]n(Cc2ccccc2Cl)cc1I)c1nccc2ccncc12 N1(C(c2ccn(CC)n2)=O)CCCC2(C1)CN(C(C13CCC(C1)C3)=O)CCO2 c1(NC(c2ncc(C)cn2)C)ccc(S(=O)(=O)NC(CCO)CC(C)C)cc1Br C1(NC(Cc2c(C)nn(CC)c2C)=O)CC2CC1CN(C(C1CC1(F)F)=O)C2 C(CCCCC(=O)N(C1CCOCC1)C)N(C)C(C1(C)CC1(C)C)=O c1(C=O)cc(Br)cc2cccnc12.C12(NC(c3cnco3)=O)CC(C)(C1)C2.N C1(C)(CC)CCCN1C(=O)Cc1cc(F)ccc1C(C)C.C(=O)(CCCC#N)N C=CC(CC)CC(=O)NCCSCC(=O)NCc1snnc1CC c1(-c2nc(C(C)N(CC(F)(F)F)C)[nH]n2)ccc(N2CCOCC2)cc1 C(C(F)(F)C(=O)N1CC(F)(c2cn(Cc3ccccc3COC)nn2)C1)OC c1(C(C)NC(CCCCNS(CC)(=O)=O)=O)ccc(C#N)cc1F C=C(C)C(CC(=O)NCC1CC1C(=O)NCC1CCCCCCC1)OCC Cc1ccnc(C(N2CCC(CO)(CNC(=O)Cc3cccnc3Cl)C2)=O)c1 C1(N=[N+]=[N-])(C(N2CCN(CC#CC)CC2)=O)CCN(C(=O)C=CC(C)C)C1 C(C)(CCCC(C)C)NC(C1CCN(C(c2c(OC)nccc2)=O)CC1)=O N1(C(=O)CN2CCCC2)CCC(C2CN(C(C3(F)CCC3)=O)C2)CC1 N1(C(C=CC(CC)C)=O)CCCCC1CC(=O)NC1CCOC1C N1(C(c2cccc(C)c2F)=O)C(C(=O)N(CCCC(C)C)C)CC2CCCC12 N1(C(CC(C)(C)N(C(C2=CCCC2C)=O)C)=O)CC2(CCC2)C12CCC2 CCCC(CC(=O)N(C1CCC1C)C)NC(C12CCC(C1)C2)=O C(=O)(C#CC(C)(C)C)NCCCN1CCN(C(CCCOC(C)C)=O)CC1 C=C=CC(C)C(=O)NCCC1CN(C(c2ccn(C)c2)=O)CCO1 N1(C(c2cccc(CC)c2F)C(=O)NC)Cc2ccc(O)cc2C1 CCCC(CC)C(=O)NCCC1(O)CCCN(C(=O)COc2ccccc2C)C1 c1(C(c2n(C)nnn2)NCc2ccoc2)cc(Cl)cc(Cl)c1F Cc1ncc(N)cc1C(N1CCC1CNC(C1CN2CCC1CC2)=O)=O c1(C(=O)NC2CC(NC(Cc3cc(OCC)ncc3)=O)C2)cnn2c1NCCC2 Cc1ccc(C(=O)NCC2CN(C(c3nccs3)=O)CCC2C)c(Cl)c1 N1(C(c2cnccn2)=O)CC(C2CC2)(C(=O)NC23CCCCC2C3)C1 C(=O)(C(C(C)(C)C)N1CCC1)NCC1CCC(C(NC[Si](C)(C)C)=O)CC1 C1(C2CC2)(NC(Cn2cc(C(C)O)nn2)=O)CCN(C(=O)C)C1.CCN(C)C N1(C(C2CCNC2=O)=O)CCC(O)(CC)CC1.C(=O)C(C1CC1)N(C)C.CC N1(Cc2cnc(SC)nc2)CCCC(O)C1C(=O)O Cc1ncc2c(n1)CCC(C(=O)N(C)CC1CCN(C(=O)C3=CCSC3)CC1)C2 C1(O)(CCNC(C(c2ccccc2)N(C)C)=O)CN(C(=O)COCCF)C1 c1(CN2C(C(=O)NCc3cn(C)nc3)CC(O)C2)cccc2nc[nH]c12 N1(C(CCCOCCC)=O)CC(NC(C2CC3CCC3C2)=O)CC1(C)C C1(CNC(C(n2cc(C(C)(O)C(=O)O)nn2)C)=O)CC12CCOC2 CCC(CCC(=O)NC1CC(C)(C)OC1=O)NC(=O)C(C)(C)O CC1CN(C(C2CC3(CCO2)CC3)=O)CC(C)C1NC(C1CCCC(O)C1)=O N1(C(Cc2ncc(C)s2)=O)CC2(COC(CNC(=O)C(CC(C)C)N(C)C)C2)C1 c1(CN(C(c2ccnn2CC(F)F)C(=O)NC)C)cccc(O)c1.C1CCCO1 CC(N=c1[nH]c(N(C)CCF)nc2c1CSC2)c1cncc(F)c1 C(=O)(C(C)(C)C1=CCSCC1)N.Cc1cc(CC(=O)NCC2CCC2)cc(C)c1 CC1(C)COC(CC(N2CCC(C)(NC(=O)Cn3nccn3)C2)=O)C1 C1(NC(c2cnc(C(C)C)[nH]2)=O)CN(C(c2snnc2C(C)C)=O)CC1C Cc1ccc(C(=O)NC2(CNC(c3cn(C4CCCC4)nn3)=O)CC2)n1C C(c1c(Cl)cccc1Cl)=CC(=O)N(CC(C)NC(=O)C(C)C(C)(F)F)C C1(NC(c2c(CC)scc2)=O)COCCN(C(=O)Cn2cccc(N)c2=O)C1 C1(NC(CC2C(C)OC(C)C2)=O)CN(C(C2CCC2)=O)CC1(C)C [SH](=O)(=O)c1cccc(Cl)c1.CC(C)(C)CS(N)(=O)=O.CC(C)COCCC.N C1(CNC(C2(C)CC=C(C)CC2)=O)CC2(CCN(C(=O)C3=CCCCO3)CC2)C1 CCCCCCCCC(=O)NC1CCCC1NC(c1ncnc2sccc12)=O C=CC1CN(C(=O)CN(C)CC2CCCC2)CC1NC(=O)CCO.C1CC1 CCCCCC(O)C(=O)NCC1CC(C(=O)Nc2cc(O)cc(F)c2)C1 N1(C(=O)CCCc2ccccc2)CCC2CCCC(C1)N2C(=O)C(F)=C1CCC1 c1(N2CCCC(N(C(c3c(C)ocn3)=O)C)CC2)nc(Cl)nc2cnn(C)c12 C1(C(=O)NC(C=C)(C)CC)(OC)CCN(C(c2ncccc2O)=O)C1 c1(CCNC(N2CCC(N3CCN(CC)CC3)C2)=O)cccc2ccn(C)c12 n1(CC)c(=O)n(CC(=O)NCC(C)CC)c2ccccc12.C(=O)C(C)=C1CC1 c1(C(=O)NCC(CC)NC(=O)Cn2nnc(=O)[nH]2)cnc(OC)cc1OC C12(NC(Cc3cc(C)[nH]n3)=O)CCCC1N(C(c1cccnc1S)=O)CCC2 N1(C(CC(C=C)(C)C)=O)CC2CCC(NC(=O)COC(F)(F)F)(C2)C1 N1(C(C(CCCC)C)=O)CCN(C(=O)C(F)(F)C2CC2)CC(O)C1 n1(CC(=O)N(CC(=O)OC)Cc2ccccc2)cc(C(F)(F)F)nn1 c1(C(C)=O)cc(C(N2CCOC(CN(C(=O)CC3CC34CC4)C)C2)=O)cnc1C C1(NC(c2cc(C)oc2C)=O)CN(C(=O)CC(=O)NCC2CC2)CCC1.C c1(C(C)OCC)nc(CSCc2cncn2C)n(-c2nc(Br)nn2C)n1 N1(c2ccnc(SC)n2)CCC2(CCOC2)C(CNC(=O)C(C)C2CC2)C1 C1(NC(CCC)=O)CN(C(=O)C=Cc2ccccc2OC(F)F)C(C)(C(C)C)C1 C1(C(N(CCN(CC(C)OC)C)C)=O)COC(C)(C)OC1 Cc1ccccc1CC(N1CC(NC(=O)Cc2conc2C)C2CC12)=O C1(NC(CN(CCC#C)C)=O)CCC2CC1CN2C(c1ccco1)=O.N(C)(C)C N1(C(C)C2CC2)CC(C(=O)NC2COCC2)CC1=O.C(=O)CCC1CCC1.N CC1CN(C(c2ccccc2)=O)CCN1C(C12CC(CO)(C1)OC2C)=O C(C(C(F)(F)F)c1ccon1)NC(C1CCCCCN1)=O C1(C(=O)NCCc2ccccn2)C2CCN(C(c3cnc(O)o3)=O)CC12 C#CCC(CC#C)NC(c1ccc(CNC(c2ccc(O)cc2)=O)cn1)=O c1(C(=O)NCCN(C(=O)CCc2nc(-c3ccsc3)no2)CC)nccnc1N N1(C(C2N(C(CCCC(=O)OC)=O)C(C)C2)=O)CCCCCCCCC1 CC1CN(C(=O)CC2(C)CCCCC2)CCC1NC(=O)C(F)(F)c1nccs1 c1(C(=O)NCC2C=CC(NC(=O)CCCc3ccccn3)C2)cccnc1Cl c1(CC)c(C(=O)NCC2CCN(C(=O)CC(O)c3ccccc3)C2)cccc1C C1(C(N(CCCCCC)CCO)=O)CCC(C2CC2)CC1 c1(OC)cc(OC)c(C(=O)OCC2CCC(C(=O)O)C2)cc1N.O N(C(=NCc1cccs1)NCC(CC)CC)CC(=O)N(CC)CC.C(C)=O.N O=C(C1CCCn2nccc21)NCC1CC2CCC(C1)N2c1ccc(C#N)nc1 CCCC(CC)C(=O)N1CCCN(CCNC(c2nn(CC)cc2[N+](=O)[O-])=O)CC1 C1(c2n(C)ncc2)CCCN(C(C(=O)N(Cc2ccccc2)CF)c2cnn[nH]2)C1 c1(CCC)cc(C(=O)NC(C)(C)C)nn1C.C1(C=O)CCCCC1.C(C)=O.N c1(NC=O)cnc(O)c(C(F)(F)F)c1.c1ncc(F)cc1Br.C1CC1C=O.N N1(C(CN2CCC(C)CC2)=O)CCN(C(C2CCC=CO2)=O)CC1CCO Cc1nn[nH]c1C1CN(C(=O)N(CC(=O)OC(C)(C)C)C)C1 c1(C(=O)NCC(C)N(C(CC(CC)(F)F)=O)C)cnn2c(C)cc(C)nc12 C1(C)(NC(c2cc(CC)on2)=O)CCCCC1C(=O)NCCC(C)C c1(C(=O)NCc2ncoc2C2CN(C(=O)C=CBr)C2)ncc(Br)cc1O c1(C(=O)NCC2CC(C)N(C(=O)CO)C2)cccc2c1NCC2.C1CCCC1.C C1(NC(=O)CC(F)F)CC2CC1N(C(c1conc1-c1ccc(Cl)cc1)=O)C2 C1(C)(CNC(COC2(C)CCC2)=O)CCCC1NC(=O)CC1CCOC1 N1(C(C(CC(C)(C)C)O)=O)C(C)CC2CCCCC12.C1(CC(=O)N)CC(F)(F)C1 C1CC2(CCN(C(C3(F)CCCC3)=O)C2)CO1.c1(C(=O)N)ccc(Cl)c(Cl)c1.C C1(NC(C#CC)=O)CN(C(c2cccnn2)=O)CC1(F)F c1(C(=O)NCC2N(C(CCc3ccnc(C)n3)=O)CC(O)C2)cc2n(n1)CCC2 c1(CNC(CC2N(C(C(C)=C3CCCC3)=O)CCC2)=O)cccnc1O Cc1nn(C)c(Cl)c1CC(=O)NC1CCCC(CNc2cnc(C#N)cn2)C1 Cc1cccc(C(=O)NC2CC(CC(=O)NCC(C)CO)C2)n1 O=C(C1=CCS(=O)(=O)C1)NC1CCC2CN(C(c3cnccn3)=O)CC12 C(=O)(C1CCCc2nncn21)NC1CN(C(C(C(C)C)N(C)C)=O)CC2(C1)CC2 CCCCCC(O)CNC(=O)C(O)CNC(C1CCCC1O)=O c1(C(=O)NCC(C)NC(=O)C(C)O)ccc(C(F)(F)F)cc1.c1ccccc1 c1(C(=O)NCC(C)CNC(=O)COc2cn[nH]c2)cc2ccccc2[nH]1 C(=O)(CCP(C)(C)=O)N1CCC(NC(c2cncc(OCCOC)c2)=O)C1 c1(N(CCNC(C)=O)C)nc(=NCC(C)(C)C(C)(F)F)[nH]c2cc[nH]c12 CN1C(=O)CSC1=CC(=O)NCC1(F)CCC(NC(=O)C(CO)N(C)C)C1 Cc1ccc(SCC(=O)NC2CC(CNC(c3ncccc3C)=O)C2(C)C)cc1 c1(OC)ccc(CC(C)NC2(c3ccccc3)CC2(C)C)cn1 C1(OC)CCOCC1NC(=O)CC1(NC(c2ccccc2Cl)=O)CCCCC1 CC1(NC(=O)Cc2cncs2)CCC(NC(=O)CCCc2cnccn2)CC1 C(CCN(C)C)(C(=O)NOC1CC2CCC1C2)NC(CC(C)C(F)F)=O CC1OC(=O)NC1C(=O)NC1C=CCN(C(c2csnc2Cl)=O)C1 C(C)(CNC(c1ccc[n+]([O-])c1)=O)(CC(C)C)NC(C(CCC)OC)=O C#CCCC(C(=O)NCC1CCOC1C)NC(=O)CCOCC(C)C CC(C)C(C(=O)NC(C1CC(NC(C2COC(=O)N2C)=O)C1)C)N(C)C CCC(C(=O)NCC(C)N(C(=O)CCc1ccc(C)o1)C)N(CC)CC C(=O)(C1=COCCC1)N(c1ccccc1C#N)C.c12ccc(nc1)n2CC(F)F c1(C(N2CCC(OCCNC(C(C(CC)O)C)=O)C2)=O)cc2c([nH]1)CCCC2=O c1(C(=O)NC(C)CC(C)NC(=O)C(F)=CCCF)cc(=O)c2ccccc2[nH]1 c1(OC)ccc(Br)c(CN2CC3(CC3C(N3CCC(C)C3)=O)C2)c1 c1(C=O)ccc(P(C)(C)=O)nc1.C(C)(CCC)NC(CNC(=O)OC)=O.N N1(C(c2ccc(SC)cc2)=O)CC2(C)CC1CO2.C1(C=O)CC2(CC(=O)N2)C1 CCCC(C(=O)N1CCC(C(N2CC[Si](C)(C)C2)=O)(N(C)CC)C1)NC(C)=O C1(CN(CCC(=C)C)C)CCN(C(C2CCCN(C)C2)=O)CC1 C(c1ccc(C(C)C)cc1)=CC=O.c1(C(N(C(C)C)CC)=O)ccc(F)nc1 Cc1ncc(F)c(N2CCC(CCNC(c3cccc(OC(F)F)c3)=O)C2)n1 C1(NC(c2n(CCC)ccc2)=O)CC2CCC(C1)N2C(=O)C(C)C CC(C)CS(=O)(=O)CC(=O)NC1CN(C(=O)CCc2cccc(O)n2)CCC1O C1(C(=O)NC(C(C)C)CNC(c2csc(C3CC3)n2)=O)CCC(F)(F)CO1 N1(C(C2CCC(SCC)CC2)=O)CCN(C(c2cncc(C)n2)=O)CC1C1CC1 CC(=O)CCCC(C)C(=O)N1CCOCCC1C(=O)NC(C)CO CN=C(NCC1CC(=O)N(c2ccc(Cl)cc2)C1)N1CCCC(C)C1 Cc1cc(Cl)cc(C(N2CCN(C)CC2CNC(c2ncccc2Cl)=O)=O)c1N c1(C=O)cccc(CC(F)(F)F)c1.C(C(=O)N1CCC1)(C1CCOC1)OCC.N c1(C(c2nnnn2C(C)C)C)cccc(F)c1I.c1(CC)cnc(C(C)(C)C)o1 CCC(CC)(C(=O)NCC(C(C)C(C)C)NC(C1CC2(CSC2)C1)=O)OC C1(NC(CC2CC(N(C)C)C2)=O)C2CC1N(C(=O)CN1CCCC1=O)C2 CC(F)CC(=O)NC(CNC(c1coc(C(C)(C)C)n1)=O)C1CCC1 C1(C(=O)NCC2CCN(C(C(CCSC)O)=O)CC2)COc2cc(O)ccc2C1 C#CC1CC2(CC(C(N3CC4(C3)SCCC4NC(=O)CC)=O)C2)C1.C1CC1.O C1(C(=O)NCc2ccc(C3(C)CC3)cc2)CN(C(N2CCCC2)=O)CCC1O N1(C(c2c(OC)cncc2)=O)CC2CCC(C2)C1.C1(C=O)CC2(C1)CC2(F)F.N N1(C(c2cccc(OCCC)c2)=O)CCC(NC(c2n[nH]cc2CC)=O)C(F)C1 Cc1nn(C)cc1C(C)C(=O)NC1CC(CCNC(c2ccnnc2O)=O)C1 C=C(C)C(C)(O)C(=O)N(CC(C)NC(C1(c2ccc(Br)cc2)CC1)=O)C C(C(CC(C)C)C(=O)NC1CC2CC1N(C(c1ccc3[nH]ccc3n1)=O)C2)OC Cc1c(C(N2CC(NC(c3cccn4nncc34)=O)C2)=O)[nH]c2c1CCCC2 N1(C(C(CC)F)=O)CC2CC(N(C)CCO)C1C2 N1(C(C(C)SC)=O)CCn2nc(C)c(CNC(=O)C(C)Cc3ccnn3C)c2C1 N1(C(CC=C)=O)CCCC(C2(NC(c3ccc(C)c(F)c3)=O)CC2)C1 C(=O)(CCCC(C)C)NCC(CC=C)NC(C1(COC)CCCC1)=O c1(NC(=O)Nc2cncn2-c2ccc(F)cc2)ccc(F)c(F)c1 c1(C(N(CCOC)CCNC(C2CCNC2=O)=O)=O)cc(Cl)c(Cl)[nH]c1=N CC1(C)C(=O)CC1C(N1CCC=CC1C(=O)NCCC1C=CCC1)=O C12(NC(c3cccc(C)n3)=O)CC(C)(C1)OC21CCN(C(=O)C(C)O)CC1 C1(CNC(C(C)=C(CC)C)=O)CC(C(=O)NC(CC(C)C)C(N)=O)=NO1 N1(C(c2ccnc(C)c2C)=O)CCC(C2CCC2)(CNC(C2(C)CC2F)=O)CC1 c1(C(=O)NC(CNC(C23CC(OC)C2C3)=O)(C)C)ccc([N+](=O)[O-])cc1 N1(C(C2(OC)CCOC2)=O)CCN(C(=O)C)C(c2cccc(F)c2)C1.C(N)=O.N C1(C(N2CCCC2CO)=O)CN(CCCc2cc(O)n[nH]2)CC(F)(F)C1 N1(C(CSSC)=O)CC(NC(=O)CCOc2cc(C)cc(C)c2)CC(C)(C)C1 N(C(=NCCc1cccs1)NC(c1snnc1C)C)CC(C(F)(F)F)OC c1(C(N2CCC(N(C(C3CCCC(C)(C)C3)=O)CC)C2)=O)cccc2oncc12 C(=O)(C1Cc2ccc(Cl)cc21)NC(C)C(CO)NC(=O)COc1ccon1 C(Cc1ccccc1)(CN=c1cc[nH]cc1S(=O)(=O)N1CCCC1C1CC1)OCC c1(C(=O)NCC(CC)NC(C2CC(OC)(OC)C2)=O)cc2c(cn1)COCC2 C1(NC(C=CC(CC)C)=O)COCCN(C(=O)Cn2nc(C(F)(F)F)cc2C)C1 n1(CCC=O)cc[nH]c(=O)c1=O.c1(CNC(C(C)=C2CC2)=O)ccccc1.N c1(NCCN(C(C(c2ccc(Cl)s2)C)=O)C)cc(=O)n(C)c(=O)n1C C1(CC)(CO)CN(C(C2CCN2C(=O)CCC2CCCCO2)=O)C1 c1(CN2CC(C)(C(N3CCCOCC3)=O)C2)ccc2cc[nH]c2n1 C(C(=O)N1CCC1CNC(C1CCCN1C)=O)(C(C)C)NC(C(C)C)=O C1(NC(CSCC#C)=O)CCC2CN(C(=O)C(F)(F)c3ccccc3)CC12 N1(C(c2ccc(C(C)=O)nn2)=O)CC2CCC(C1)C2NC(=O)CSC(C)=O C1(C(C)(C)C)CCCCN1C(C1CC=CC(n2cc(CC3CCCO3)nn2)C1)=O C1(C=O)CC(C)(C)CCN1C(=O)C(C)S(N)(=O)=O.Cc1ccc(F)cc1C.N C(=O)(C(CN=[N+]=[N-])NC(c1cnn(C(C)C)n1)=O)NC(CC#CC)C c1(NC2C(C)C2)nc(N2CCOCC(C3CC3)C2)c2cccc(F)c2n1 c1(CCNC(N(CCOC)C(c2ccc(Br)s2)C)=O)cc(F)ccc1F C=CCC(CC=C)C(=O)NC1CN(C(=O)C(C)=CCC)C(C)(C)C1 C1(C(C(=O)NCCO)N(CC(C)C)CC)CC12CCOCC2.c1cccnc1.C N1(C(C(CC)C)=O)CCN(C(c2ccc(Oc3ccccc3)cc2)=O)CCC1C N1(C(C2CC(C)N2C(c2ccc(C#N)n2C)=O)=O)CCC12CC(O)C2 N1(c2[nH]c(N3CC(=O)N(C)C(C)C3)nc(=NCC)n2)CCCC2(CCCCO2)C1 Cc1cnccc1C=CC(N1CCCCC(NC(c2cscc2C(N)=O)=O)C1)=O c1(OC)ccc(OC)c(CNC(c2cccnc2)C(C)C)c1 C12(C(N(C(C)C(F)F)C)=O)COC(C1)C(NC(c1ccsc1C#N)=O)C2 N1(C(=O)NCC(N2CCCC2C(=O)NCC2CC=CCC2)C)CCCCC1 C1(NC(C(Br)=C(C)C)=O)CCCCC12CCCN(C(=O)CCn1ccnn1)C2 N1(C(CN(C(COC)=O)C)=O)CCOCC(F)(CNC(=O)C(C)(C)C)C1 C(=O)(NNc1ccc(C(F)(F)F)cc1F)c1cc(C)c(Br)cc1F c1(C(CC)(C)C)n[nH]c(=NCC2CC(NC(=O)C3=NNC(C(F)(F)F)C3)C2)o1 c1(CC(=O)NCC(CO)NC(c2cnc(C)s2)=O)nn(C)cc1Cl C#CC1(O)CC(C(=O)NCCC2CCCCN2C(=O)C(O)Cc2cnc[nH]2)C1 CCC(CC(=O)NCc1nocc1C(=O)Nn1cccn1)C(C)C c1(C(=O)NC(CC)CNC(C23CC(CN2C2CC2)C3)=O)c(C)cccc1O N1(C(C2C=CC(N)C2)=O)CCC(O)C(O)C1.c1cccc(F)c1OC(F)(F)F.C c1(C(N2CC(CNC(C(C)(F)F)=O)C(F)(F)CC2)=O)ccc2cnnc(O)c2c1 C1(S(C)(=O)=O)(C(=O)NC(C2(O)CCN(C(c3cnsn3)=O)C2)C)CC1 C=C(Cl)CC(C(=O)N(C)CCN1CCCC1=O)NC(c1ccc(C)cc1C)=O N1(C(C(C)(C)C2CC2)=O)CC2CCC1C1CN(c3ncc(F)cn3)CC21 C1(NC(=O)CC2CCOC2)CN(C(C2(CCO)CC2)=O)CC12CCOCC2 c1(C(=O)NC(C2CCN(C(c3cn(C)nc3Cl)=O)CC2)C)ccc(CCF)cc1 C1(NC(C2=CC(C)(CC)C2)=O)COC2CN(C(c3cc(C)ncn3)=O)CC12 CN1CCC(O)C(NC(=O)C(C2(O)CCC2)NC(c2ccc(C#N)o2)=O)C1 C1(C(N2C(CNC(C(c3ccccc3Cl)C)=O)CC2)=O)Cc2ccc(F)cc2O1 c1(N2CCN(C(C3(C)CCNC3=O)=O)CC2)nc(C(F)(F)F)ccc1C#N N1(C(c2c(F)cc(F)cc2Br)=O)CCc2ccc(-c3ccc(F)c(O)c3)cc2C1 N1(C(C(C)(C)C2CCCO2)=O)CCCC(C)(NC(=O)Cn2ccnn2)C1 C1(C(=O)NCCCCN(CCCNC(CC=CC)=O)C)CCS(=O)(=O)N1 C1(C(N2C(C)(C(=O)OC)CC2)=O)CC2CCC1N2C(=O)CSCC(N)=O C(c1ccc(Cl)s1)=CC(=O)NCC(C1CC1)NC(COCCCCC)=O CCCCC(CO)NC(=O)C(CO)NC(c1cc(C)nn1CC)=O c1(N2CCCC(CNC(C)=O)C2)ccncc1S(=O)(=O)NC1CCCO1 O=C(C#Cc1ccc(Cl)cc1)NC1CCC(CNC(c2ncccc2F)=O)CC1 C(=O)(C1CCc2cc(F)ccc21)NC1CCN(C(CCC(C)(F)F)=O)CC1CO Cc1cc(F)cnc1C(=O)NC(C(=O)NC1CCC(O)CC1)c1cccs1 C1(C(N2CC(NC(c3nc(C)oc3)=O)C(n3ccnn3)C2)=O)CCCC(F)(F)C1 N1(C(c2n(CC)ncn2)=O)CCN(C(=O)CCc2nnc(C)n2C)CC1C(F)F N1(C(C2(C)CC2)=O)CCC(C(=O)NCC2SCCS2)=C(F)C1 c1(C(=O)NCC2(F)CC(NC(CC(CCC)O)=O)C2)cnc2cnn(C)c2c1 C1(C(N(CC(C)C)CCOC)=O)CN(C(=O)C2=CCSC2)CC1C(C)C Cc1ccnnc1C(N1CCC(N(C(=O)Cc2cncn2C2CC2)C)C1)=O C(=O)(CCCCC(=O)N1CCC(C(=O)NC2CC=CCC2C)C1)OC c1(OC)cc(C(=O)N)ccc1[N+](=O)[O-].C1CCCN1C(=O)C=Cc1cnc[nH]1.C N1(C(c2c(C)cc(C)[nH]2)=O)CC(C)(C)CC1CNC(C1CCCN1C=O)=O C(=O)(C(C)C(CC)CC)NCC1(C(N2CCCC(C#C)C2)=O)CCCCC1 C1(NC(c2csc(C)c2C)=O)CC(C2CCN(C(=O)CCOCC(F)(F)F)C2)C1 C1(N(C(=O)C#CC2CC2)CC)CCCN(C(=O)CSc2ccccc2C)CC1 c1(C(N2CCCCC23CC3)C(=O)NCC(=C)C)cn2cccc(F)c2n1 N1(C(CCNC(=O)CO)=O)CC(NC(c2cncc(CO)c2)=O)CC12CCOC2 CCC1=C(C(=O)N2CCC(NC(=O)C3=C(Cl)CCOC3)C(F)C2)CCCO1 CS(=O)(=O)C(C(=O)NCCCCNC(C1CNC(=O)N1)=O)C1CC1 C1(C(N2CC(C)(CCC(=O)NC34CC(C)(C3)C4)C2)=O)CCCC1C1CC1 CCCC(O)CC(=O)NCC(C)CNC(c1nnn(-c2cccc(Cl)c2)c1C)=O C(=O)(C(C)(C)C(C)NC(C1CCCC(=O)CC1)=O)N(CCSC)C C(=O)(CS(=O)(=O)CC(=O)OC)NCC1N(C(COCC=C)=O)CC(O)C1 N1(C(c2ccc(C)cn2)=O)CCN(C(=O)Cc2ccoc2)C(CO)C1 c1(CC)nn(C)c(C(=O)NCC2C3CN(C(c4c(Cl)csc4Cl)=O)CC23)c1Cl C(CSC)(C(=O)NC1CCC(NC(=O)CCN(CC(F)(F)F)C)C1)OC c1(C(=O)OC)csc2c1CCN(Cc1cccc(OC(C)C)c1Cl)C2 Cc1ccc(C)c(CC(=O)NC2CCCCN(C(=O)C3=CCC3)C2)c1 N1(C(c2cc(CC)ncc2)=O)CCCCC(NC(=O)C(C)(C)CO)C1 C1(C(=O)NCCC2CCN(C(=O)CCCC3CCC3)C2)CCS(=O)(=O)N1 c1(C(N2CC3C(CNC(C4(C(C)C)CC4)=O)(C3)C2)=O)cc2ccc(F)cc2o1 N1(CC(N2CCCC2)=O)CCC(C)(O)C1.Cc1csc(C(F)(F)C(=O)NC)n1.C Cc1cc(CCC(=O)NCC(C)(C)OCCNC(C2CCCCN2C)=O)c(C)s1 c1(NC(C(N2CCC23CCC3)C)=O)cccc(Br)n1 c1(C(=O)NC2C(CNC(CC(C)C3CCCCC3)=O)C2)nn2cccnc2c1Cl C1CC2(CC2)CN1C(=O)CC1CC2CCC1O2.C(c1ccccc1)=CC(=O)N.C N1(C(C(C)C)=O)CCC(O)(CCNC(=O)COC2CCCCCC2)C1 N1(C(C2(C)CC(=C)C2)=O)CCC2CCN(C(c3cn(CC4CC4)nn3)=O)C2C1 C(CN=c1ccnc(NCc2onc(C)c2Br)[nH]1)N(C)CC C(=O)(C1=CCCC(C)(C)C1)NC(CN(C(C1CC(F)C1)=O)CC)C C(=O)(CCS(=O)(=O)c1cc(Cl)ccc1Cl)NCc1c(F)ncc(C)c1 c1(C(=O)NC(C(C)NC(C(C)=C2CCCC2)=O)C(C)C)cnn2cc(C)cnc12 Cc1nn(C)cc1CCC(=O)NC(C1CCCN(C(=O)CCc2cncs2)C1)C NC(=O)CC(O)C(=O)NCC1CN(C(=O)CSc2nc[nH]n2)CCO1 Cc1nc(O)nc(O)c1NC(C1CC2CC2N1C(=O)Cc1ccc(Cl)cc1)=O Cc1cc(C(F)(F)C(=O)N2CCC(NC(c3occc3C)=O)C2)cs1 Cc1cc(O)cc(C)c1NC(=O)C(=O)NCC1COC(=O)N1 C1(C)(NC(C(C)NS(C)(=O)=O)=O)CCCN(C(=O)CCC2(O)CCC2)C1 C1(F)(CNC(CN(C)CC)=O)CCC1.C(=O)C(F)(F)c1csc(C)c1.C N1(C(c2cccc(F)c2F)=O)CC2COCC2(C(N2CC3CCCC3C2)=O)C1 Cc1ncc2cc(C(=O)NC3(C)CCN(C(=O)CS(=O)(=O)N(C)C)C3)ccn12 c1(C(=O)OCC2CCCO2)ccc(S(=O)(=O)NC2CCc3ncnn3C2)cc1 c1(C(N2CC(NC(C(C)CC(F)F)=O)C(C(F)F)C2)=O)ccn2nccc2c1 C1(O)(CCNC(C2CCC3CC3C2)=O)CCN(C(c2cnn(CCO)c2)=O)CC1 CC(C)CC(CNC(c1ccc(C(F)F)cc1)=O)NC(C1(C)CC1Br)=O C12(C(N3CCN(CCCNC(=O)Cc4cnoc4)CC3)=O)CCC(F)(CC1)C2 N1(C(=O)NC2CCN(c3cccc(Cl)c3)C2=O)CCCC2CCC12 Cc1ccc(CN(C(=O)C(=O)NC2CCC2CF)C)o1 C1(C(=O)NCCC=CCCC)(NC(=O)C(C(C)(C)C)S)CCC(C)(C)C1 c1(C(=O)NC2CCN(C(=O)CC3CC(C(F)F)C3)CC2O)nc2c(s1)CCCC2 S(=O)(=O)(c1cccc(=NCCCN(C)C)[nH]1)NCC(CC)OC c1(C(=O)NCCCNC(CC2(C)CC2(F)F)=O)ncc2cc(Cl)ccn12 C1(N(C(c2ccc(C)nc2)=O)C)CCCN(C(c2ncc(Cl)cc2Cl)=O)CC1 C1(C(=O)NCC(C)NC(Cn2ccc(C)n2)=O)CCN(Cc2ccncc2)CC1 C1(CC)(CC)CC(C(=O)N(CCCNC(=O)CC(C)C2CCCO2)C)C1 N1(C(c2nccc(-n3c(C)ncc3)c2)=O)CC=C(CCNC(=O)C=CS(C)=O)CC1 N1(C(c2ccc(C)nc2O)=O)CC2(CCC2)CC1C(=O)NC(C)C(O)C(F)F CCC(Cc1ccccc1)CC(=O)N1CC(NCC=Cc2ccoc2)CC(C)C1 C1(C(N(CC(=O)NCc2ccc(Cl)o2)CCOC)=O)CCCC(C)CC1 C1(O)(CN2CC(CC(C#C)C)C2)CCC(c2ccccc2)CC1 N1(C(C2C(C(=O)OC)C=C2)=O)CCC(O)(C)C1.c1(C(=O)N)cn(C)nn1 c1(OC)cnnc(C(=O)NC(C)C(C)NC(=O)C(C)(C)Cc2ccccc2)c1 c1(C(=O)NC(CCCNC(C2CCN(CC)C2)=O)CO)cc2ncccc2o1 CC(C)(CCCNC(C1CC1F)=O)NC(=O)Cc1cncs1 N1(C(C2C(C)(C)C2)=O)C2CCC1C(NC(c1csc(C(N)=O)n1)=O)C2 N1(C(C(C)SCC)=O)CC(NC(=O)C)CC2(CCC2)C1.c1cccc(F)n1.O c1(C(N(C2CCCC2O)C)=O)c(F)cccc1Cl N(C(=NCCC(=O)OC(C)(C)C)NCCCCn1ccccc1=O)C(CC)C N1(C(C(CC)SC)=O)C(C(N2CC(OCC(F)F)C2)=O)CC2CC12 c1(CC(=O)NC(CN(C)C(C2OC3CCC2C3)=O)(C)C)noc2ccccc12 C1(CC=C)(C(=O)N(CC(O)C2CC2)C)CN(C(=O)C(=O)N(C)C)C1 C1C(C)CCCN1C(c1cc(C(N)=O)no1)=O.C(CCC(=O)N)N(C(C)=O)C.C CCC(=O)CCC(=O)Nc1ccc(OCOC)cc1 C1(NC(c2c(C)ccs2)=O)CC2CC(NC(c3cc([N+](=O)[O-])n[nH]3)=O)C2C1 C1(C)(C=O)CCC(F)(F)C1.c1(C(N(CCC)CC)=O)coc(-c2ccsc2)c1 C1(NC(Cn2c(C)ccn2)=O)CC(C(=O)NCCO)C1(C)C.CCN(C)C c1(C(C(=O)NCCC2(O)CN(C(CCCOC)=O)C2)O)cc(Cl)cc(Cl)c1 C1(C(=O)NC(CC#C)C(=O)NC)CN(C(=O)CC(C)C(C)C)CC(C)(C)C1 Cc1nccnc1NC(C1COCCN1C(c1cccnc1C(F)(F)F)=O)=O C(=O)(C(O)P(C)(C)=O)NC1CCC(N(C)C(c2nc(C3CC3)cs2)=O)CC1 c1(CC)cc(N)ccc1C(=O)NCC1CCCC12CC2 N1(C(C=CC=CCC)=O)CCC(F)(CNC(=O)CCc2ccccc2Cl)C1 CCCCS(=O)(=O)NCC(=O)NCC(CO)NC(C1(CSC)CCOCC1)=O C(=O)(C1=C(C)S(=O)(=O)CC1)NCC(CC=C)NC(c1cnsc1)=O c1(NC(C2C3(CN(C(Cc4cnc(C)s4)=O)C3)C2)=O)ccc(F)cc1Cl N1(C(c2c(C)ccc(C(=O)OC)c2)=O)CCC(C2CC2)CC1.C(=O)(C1CC1)N C1(C(=O)NCCc2ccc(CN(C)C)cc2)CCC(N=[N+]=[N-])C1 c1(C(=O)NC(CN(CC)CC)C)c[nH]c2cc(C(=O)OC)ccc12 c1(C(=O)NC(CSCC)C(=O)NC(C2CCOC2)CO)cc(OC)nn1C n1(CC(N2CC(CCNC(CC(n3ccc(C)n3)C)=O)C2)=O)cccc(C)c1=O N1(C(C2CCC(C(F)(F)F)C2)C(=O)NC(CC)C)CC2C3C=CC(O3)C2C1 C#Cc1ccc(C(=O)N(C2CCCN(C(c3ccccc3CC)=O)CC2)C)nc1 N1(C(C(CNC(=O)CCC2CCCCC2)N(C)C)=O)CCOC(CCO)C1 N1(C(CCC=CC)=O)CC(O)(C2(CNC(C3CC4CCC3O4)=O)CC2)C1 C(=O)(CCC(C)(F)F)NC(C(C)NC(c1cc(Br)c(Cl)s1)=O)C C#Cc1ccc(C(=O)NCC2CC(C)N(C(c3[nH]ncc3C#N)=O)C2)c(F)c1 c1(C(=O)NC2C(CNC(CSC)=O)CC2)ncn(C(C)C)n1 C1(NC(=O)C(F)C2CCCC2)CCN(C2CN(C(C3CCS(=O)(=O)N3)=O)C2)CC1 C1(C(N2C3CC(CN(C(C(C)(C)C4CC4)=O)C3)C2)=O)CC2CC1C1C2C1(F)F CCC(C(=O)NCCN(C)C(C1(C)CCCO1)=O)N(C)Cc1ccccc1 C(=O)(C1=C(C)OCC1)N(C1CCN(C(=O)Cc2ccc(Br)cc2)CC1)CC C1(CNC(C2CCCN(CC)C2)=O)CCC12CN(C(c1cnc(C)s1)=O)C2 c1(C(=O)NCCCCC)cc2cccc(-c3ccc(OCCC)cc3)c2[nH]1 c1(C(=O)NC2CC(NC(c3c(CC)scn3)=O)C2)cc(F)cc(Cl)c1O C1(c2n(C)nnn2)CC2(CCC2)C1.N1(C(CNCCSC)=O)CCCC1 C1(OC)CCN(C(=O)C(C2CCCCC2)NC(C2CCCCC2)=O)CC1F Cc1nc2ncnn2c(C)c1C(=O)NCC1CC(C(=O)Nc2conc2C)CO1 CCC(C)C(O)C(=O)NCC(C)(C(C)C)NC(c1nocc1Cl)=O c1(C2(C(N3CCN(C4(CC)CCC4)CC3)=O)CC2)c(Cl)ccnc1OC CCC(CNC(=O)NC1CC(C(=O)O)CC1O)C(C)(F)F Cc1nc2c(N(Cc3cc(C(C)C)cc(Cl)c3)CC3CCNC3)ncnc2[nH]1 c1(OC)ncccc1C(C(=O)NC1CC1)N(C1CC(C)C1)C.c1ccccc1.O N1(C(CCC2CC(C)C2)=O)CC(CCNC(=O)CC2(CO)CC2)C(O)C1 N1(C(=O)Nc2cccc(N(S(C)(=O)=O)C)c2)CCN(C)c2ncnc(Cl)c2C1 C12(C(=O)NC(CC)CNC(c3cccc(Cl)c3)=O)CCC(C1)C(C)(C)O2 C1(C(=O)NOCC(=O)NCCC2CCCN2C)(CC)CC(=O)C1 C1(COC)(NC(c2scnc2C)=O)CCN(C(C2CCCC(N(C)C)C2)=O)CC1 C1(c2nc(C(C)NC(N3CC(n4cc(Cl)cn4)C3)=O)on2)CCC2CC1CO2 Cn1nnc2c(NCC(C3CC3)NC(c3cc(Cl)c(Cl)s3)=O)ncnc12 N1(C(CC2(OC)CCCC2)=O)CC(NC(c2nccnc2C)=O)CC(F)C1 Cc1ccccc1CN(Cc1ccccc1)CC1CC(=O)N(c2ccccc2)C1 C1(C)(C(=O)NC2CC(CCNC(C=C(C)C(F)F)=O)C2)CCN(C)C1=O Cc1cc(C(=O)NC(C(=O)NCCCC(O)CO)c2cccs2)n(C)n1 N1(C(c2c(CC)nns2)=O)CCC2(CC1)CCS(=O)(=O)N2C.C(=O)(CC(C)F)N N#Cc1c(NC2CCN(C(N3CCCC3)=O)CC2)ccc([N+](=O)[O-])c1N C(c1ccc(Br)cc1)=CC(N1CCN(C(=O)C2=CCCOC2)C(CF)C1)=O c1(C(N(C(=O)CCc2cccc(Cl)c2I)C)=O)nc(C(F)(F)F)n2ccccc12 CC(C(C)(C)C(=O)NCC12COC(C1)C(O)C2)NC(=O)C(F)C1CCCC1 c1(C(=O)NC(CN(C(c2scc(C)c2)=O)C)C)ccc(NC(N)=O)cc1 C1(C(N2CCCC(n3cc(CC(O)C4CC4)nn3)C2)=O)CC2(CCOCC2)CO1 c1(C(=O)NC(C(=O)NC2C(SC)CCC2)C2(C)CC2)ccc(=N)[nH]n1 C=Cc1cc(C(N2CC(NC(=O)CCOC(C)C)CC23CCC3)=O)cc(F)c1 O=C1CC2(CCN(C(c3ccc4cc(O)ccc4c3)=O)CC2)Oc2ccccc21 C1(C(N(C)Cc2ncc(C)o2)=O)CC(C)(C)CN1C(=O)Cc1cccn1C CCC(CC(=O)N1CCC(CCC(=O)N(C)Cc2nc(C3CC3)no2)C1)C1CC1 C(CCCC1C(=O)NN1CCOC(F)F)OC.C1(C(=O)OC)CCOC1 C(CCCCCCC)NC(CCC1N(C(C(=C)Cc2ccccc2)=O)CCC1)=O Cc1cccc(S(=O)(=O)NC2CC2(c2ccccc2Br)F)c1Br CCCCC(C)C(=O)NCC(c1ccc(C)cc1)NC(=O)Cc1ccoc1 N1(C(c2ccc(NC(c3ccc(C)cc3Cl)=O)nc2)=O)CCCCC(C)(F)C1 N1(C(c2c(C)nns2)=O)CCC(O)(C)CC1.C(=O)CS(=O)(=O)CC1CCCO1.N C(=O)(CC(O)CCCCC)N1CC(C)(CCC(=O)N(CCCCCC=C)C)C1 C1(N(C(C(C)SCC)=O)C)CC2CC1N(C(C1CN3CCC1CC3)=O)C2 c1(C(=O)NCCC(C)NC(=O)C(C)(C)Cc2cnn[nH]2)ccc2c(c1)OCO2 C1C(C)(C)C1(F)F.C1(O)(C(C=O)NC(C2(OC)CCSC2)=O)CCCCC1.N C(=O)(C1=C(C)CCOC1)N1CCC(c2nc(-c3c(C)cccc3F)no2)(OC)C1 C1(OCCC)CCC(CC(=O)N(CCCCCCNC(=O)CC2CC2C)C)CC1 C1(NC(c2cccc(C)n2)=O)CN(C(c2ncoc2C)=O)CC1S(C)(=O)=O C1(NC(C(C)N=[N+]=[N-])=O)CCC(C)N(C(c2cnn(C(F)F)c2)=O)C1 c1(NC(N(CCCOC)Cc2ccccc2I)=O)ccc(C)cc1C C1(NC(c2cnc(-c3cccnc3)s2)=O)C2CC1N(C(=O)CC1CSCCS1)C2 c1(CC)ccc(F)cc1C(N1CCC(NC(=O)C(C)C(C)O)C1)=O C=CCC(CNC(=O)C=Cc1cnccn1)C(=O)N1C(CO)CC1C C1(NC(=O)CC2CC=CCC2)CN(C(c2n[nH]cc2Br)=O)C2(CCCC2)C1 n1(CC(=O)Nc2ccc(C(N3CCCC(C)C3)=O)c(Cl)c2)ccc2cccnc12 C1(NC(C(CCCOC)C)=O)CC2CCC(C1C)N2c1nnc(C)c(C)n1 Cc1ccc(C(=O)NOC(CC(C)C)C(=O)NC(c2nnnn2C)C)cc1C C1(C(=O)NC(C2CCCN2C(c2cc(Cl)ns2)=O)(C)C)CC2(C1)CC2(F)F CC1(O)CCC(CC(=O)NC23CCC2CN(C(c2nncn2C2CC2)=O)C3)CC1 N1(C(=O)CSCc2ccc(Cl)s2)CC2CCC1CN2C(C1CCCO1)=O N1(C(CCC=C=C)=O)CCC(C)(NC(c2ccc(CN(C)C)cc2)=O)CC1 N1(C(CCn2cc(C(CC)(C)O)nn2)=O)CC2CCCCCCC2C1 C1(CC(=O)NCc2c(C)scc2)CN(C(=O)COCCCF)CC12CC2 C1(C=O)CCCC(O)C1.O=C(C=CC(=O)NC1CC1)NCCO.CCC C(=O)(C(CC(C)C)NC(=O)CCCn1cccc1)NCCOC(C)=O c1(C(=O)NCC=CCC(=O)NC(CCC)C2CCC2)oc(C)cc1C c1(OC)cc(S(=O)(=O)N2CC(CN(c3cccc4nccn34)C)C2)ccc1Br C1(NC(c2cccc(C)c2C)=O)CCN(C(c2ncc(F)cn2)=O)CC(C)(C)C1 Cc1nc2c(n1C)CCCC2C(=O)Nc1ccc(Cl)c(Cl)c1C#N C(=O)C1=NN(C)C(=O)CC1.CCC(C)(CNC(c1ccc(C)cn1)=O)C(C)O c1(C(=O)NCC2CN(C(CNC(CC)=O)=O)CC2C)ccc(=NC)[nH]c1 C(CCC(C)(C)C(=O)N1CCC(F)(C(=O)NCCC2CCCC23CC3)C1)OC C1(CC)CCN(C(=O)CC(C)n2cccn2)C(C(=O)NC)C1.C1CC(C=O)C1 C1(N(C(C(C)NC(C)=O)=O)C)CN(C(=O)CN2CCNC(=O)C2)CCC1C c1(OC)cccc(C(=O)NC2CCCCN(C(=O)Cc3csnn3)C2)c1C N1(C(CC(C)NC(N)=O)=O)CCN(C(c2ccsc2)=O)CC1c1cccc(Cl)c1 CC1C(NC(c2cc(=O)cc(Cl)[nH]2)=O)CC2CCC1N2C(C1CC(=O)CO1)=O S(=O)(=O)(CC(=O)N1CCCC1C(C)C)NC.C(=O)CC(O)Cc1ccccc1.N c1(C(C(CC)CNC(=O)C(C)(C)OC)=O)cncc(N2CCCC2)n1 C(=O)(C1=C(C#N)CCC1)N(C)CC1CCN(C(C2C(OCC)C2)=O)C1 N1(C(c2cc(C(=O)OC)n[nH]2)=O)CCOC(CN)C1 c1(C(=O)NCC(C(N2CCCC2(C)C(C)(C)C)=O)OC)nc(C)sc1C C(=O)(CCC(C)SC)NC(COC)CNC(=O)Cc1ncoc1C Cn1ccc(C(N2CC=CC2CNC(c2cnn(C3CCCC3)c2)=O)=O)n1 c1(-c2ccsc2)cn(Cc2ncoc2CN2CCCC2)nn1 Cc1c(C(N2CCC(NC(=O)C(C)O)C2C(C)C)=O)cnn1-c1ccc(F)cc1 Cc1cnc(C(=O)NCC(C)(C2CC2)NC(=O)C=C2CCC2)c(C)c1 Cn1c(NCC2CCCC(F)C2)cc(O)nc1=O.C12(CC1)CCNC2=O C(CN=C(NCc1ccn(C)n1)NCc1nnc(C)s1)OCC C1(C(=O)NCc2c(C(=O)NCc3n[nH]c(C)c3C)occ2)CCCCC(=O)C1 C1(CCn2cc(-c3c(C)c[nH]n3)nn2)CCCN(C(c2ccccc2)=O)CC1 c1(C(=O)NCC(CCC)NC(c2ccc(C=C)cc2)=O)nccc2cc[nH]c12 C(=O)(C1CCCc2nn[nH]c21)NC(CNC(C1C(C(C)(C)C)C1)=O)CO C(=O)(C(CO)C(F)(F)F)N1CCC(CCNC(C=C2CCC(C)C2)=O)C1 c1(C(=O)NCCC2C(C)CN(C(c3csc(C(F)F)n3)=O)C2)cc(N)ccc1F c1(NC(C(N2CCCC(C(c3csc(C#N)c3)=O)C2)C)=O)ccc(F)cc1 Cc1ccc(O)cc1C(=O)NC1CC(NC(C2(C(C)(F)F)CC2)=O)C1 c1(C(=O)NC(c2cccc(OC)c2)(C)CC(=O)O)ccn2c(N)cnc2c1 c1(C(=O)NC2CN(C(C(C)OCC)=O)CC3C2C3)c(Cl)ccc([N+](=O)[O-])c1Cl c1(OC)ccc(Br)cc1C(N1CCC(NC(=O)CC2CC=CC2)C(O)C1)=O n1(C2(CNC(=O)COCCNC(C3CCC3)=O)CC2)cnnn1 CC1CCCN(N2CC(C(=O)N(C)C)CCC2(C)C)C1C N1(C(C(CC)CC(C)C)=O)CCN(C(C2CCc3n[nH]cc3C2)=O)CC2(CC2)C1 C1(C(C)C)N(C(c2ncc(Cl)n2C)=O)CC12CCN(C(C1OCC1(C)C)=O)CC2 c1(C(=O)NCC2N(C)CCN(C(=O)C(F)F)C2)onc2ccccc12 c1(CC)cccc(C)c1NC(=O)C(CC1CC1)NC(=O)CC(CC)SC c1(OC)ncc(C(=O)NC2C3CN(C(C4CC5CC4C5)=O)CC23)cn1 n1(CC)ccc(C(=O)N(C2CC(NC(C3SCCCS3)=O)C2)C)n1 CCN=c1cc(C(N2CC(O)(CNC(=O)C(F)(F)C3CC3)C2)=O)cc[nH]1 C1CN2CCC1C2.n1(CC(=O)NCCNC(C2(C=O)CC2)=O)nccn1.N C(CCCCCNC(C1C2CN(C)CC12)=O)NC(C(C)CC1CCC1)=O O=C(CC1CCCc2ccccc21)NC1CCCC1NC(=O)CC1CC=CC1 c1(CC(=O)N(CC(C)(C)CNC(=O)CC2CC2)CC)cncc(F)c1 c1(CC)cccc(CNC(=O)C(C)NC(C2CC2CC)=O)c1 C(=O)(C1=CCN(C(=O)CC(O)CC)C1)N(CCC#C)CCO N1(C(C2C(N(C)C)CCC2)=O)C(C)CC2CC12.C(=O)CCN(CC(F)(F)F)C Cn1cc(NC(c2ccnc(C3CC3)n2)=O)cc1C(=O)Nc1ncc(F)s1 C(C)(C(=O)NCC1(C(=O)N(C(CC)CC)C)CC1)OCCC C12(C(N3CC(CCNC(C(C)(C)OCC)=O)OCC3)=O)CC1CCC2(F)F c1(N2CCC(C(N(C)C)=O)CC2)cc(NCc2nncs2)nc(C(F)(F)F)n1 [N-]=[N+]=NC1(C(=O)NC2CC3CCC2O3)CCN(C(=O)CC2CCCSC2)C1 N1(C(C(C)N2CCC2)=O)CC2(CC2)CC1CNC(c1coc(CO)c1)=O CC1CN(C)CC(C(=O)NCCC2(O)CN(C(=O)C(F)CC3CCOC3)C2)O1 C#CCC(CC#C)C(=O)N1CCC(CO)(CNC(=O)CCCC(=O)N(C)C)CC1 Cc1cc(C(=O)NCCSCC(N2CCC(N(C)C)CC2)=O)ccc1O C#Cc1nc(C(=O)NCC(c2ccccc2)N(C)C(C2COCCN2C)=O)cs1 CCCC(C(=O)NCC1CN(C2CC2)C1)NC(=O)C(C1(O)CCCC1)F CCC(CO)C(=O)N1CCN(C2CCN(C(=O)COC3CCCC3)C2)CC1 N1(C(C(C)(C)C(F)c2ccccc2)=O)CC2(CC(NC(c3cccs3)=O)CO2)C1 N1(C(c2ccc(C)cc2)=O)CCC(NC(C2(C)CCCN2C)=O)C(CO)C1 C1(C(N2CC(C)(OCC(=O)NCc3ccncn3)C2)=O)CCCCC1O C(C(C(=O)NC(C)CC1CC1)C(C)C)NC(c1c(CC)onc1C)=O C(=O)(N1OC2CCC1C2)c1c(CNC(c2n(C)nc(O)c2)=O)ocn1 C1(C(=O)NC2C(C)CCN(C(C3(C=C)CCC3)=O)C2)CCc2nnc(C)n2C1 C(CCN=c1cccc(S(=O)(=O)NCC2(c3ccccc3)CC2C)[nH]1)OC(C)C c1(NC(c2c(Cl)ccc(OCC)c2)=O)cc2n(C3CC3)cnc2cc1F c1(C(C(=O)NC2CC(F)(F)C2)NCC(=O)OC)n[nH]c(C)c1Cl C1(C(=O)NCc2c(C)nsc2)CCN(C(=O)C(C)C(C)C)C1(C)C C=C(C)CC(C(=O)NC(CNC(=O)C(O)CC1CCCC1)C1CC1)OC CN1C(=O)c2ccccc2C1CNC(=O)NCc1noc(C2CCCO2)n1 CC1CN(c2cc(C(N3CC(N4CCOCC4)C(F)C3)=O)ccn2)CCO1 C1(C(=O)NCc2cn(CCC)nn2)CC(F)(F)CN1C(C1CC1CC)=O Cc1ccc(CSCC2CCCCC2C)c(O)c1 N(C(=NCCCN(c1ccccc1)C)NC(CO)CCF)C(C=C)C c1(C=O)[nH]c(C)c([N+](=O)[O-])c1C.Cc1cc(C(F)F)oc1C(=O)NCCCC.N N1(C(C2(CC)CC2)=O)CCC(CN(C)C(c2cccc(-c3ncon3)c2)=O)CC1 c1(OC)ncc(Br)c(=NCC(C)(C)NC(=O)COc2ccccn2)[nH]1 C1(C)COCCN(C(=O)C(=O)C(C)(C)C)C1.C1(CC(C)C)(C(=O)N)COC1.C CC1(C)CC(C(=O)O)N(C(c2cc3n(n2)CCO3)=O)C1 C(=O)(C1(C)CCc2ccccc21)NC(C1(O)CCN(c2ncc(C)c(O)n2)C1)C c1(CC)cccc(C(N2CCC2CNC(c2ccccc2I)=O)=O)n1 c1(C(N(C)C[Si](C)(C)C)=O)ccnn1C.C(CC1CCCC1)(C(=O)N)SC C=CC1CCCC(NC(=O)CC(C)C2CCNCC2)C1 N1(C(C2(OC)CCCC2)=O)CCC(C2CCN(C(=O)CCC3CCCCC3)C2)C1 c1(C(N2CC=CC(NC(c3cc(OC)ncn3)=O)C2)=O)oc2ccccc2c1Cl C(CCCCC(=O)NCC1(F)CC(NC(=O)C(C)C)C1)OCC.C(C)=O CCC(C(=O)NCC1CCCN1C(=O)CCc1ccn(C)c1)OC C1COC2(C1)CN(C(c1cc(C3(Cl)CC3)n(C)n1)=O)C2.C(CCC=O)=C(C)C.N C1CCCC(F)(F)C1.N1(C(CC2C(OC)C2)=O)CC(OC)CC1C(=O)N.CC N#Cc1ccc(C(=O)NC2(F)CCN(C(=O)COc3ccccc3)C2)c(Cl)c1 C(=O)(CCC(C)SC)NC(c1cn(C)nn1)C(=O)NCc1occ(CC)n1 N1(C(CCc2cc(C)[nH]n2)=O)CC(NC(C2(C)CCN(C)C2)=O)C(C)C1.C1CC1 N1(C(C(C)OC)=O)CC(CNC(=O)CCOCC(F)F)CC12CCC2 C(=O)(C(O)C(F)(F)F)NC(CCCNC(=O)CN1CC2CC2C1)c1ccccc1 N1(C(C2(C(=O)OCC)CCO2)=O)CC(F)C1.C(=O)C(F)(F)c1cnnn1C Cn1cc2ccc(C(N3CC4CN(C(=O)Cc5ccsc5)C4C3)=O)cc2n1 C12(C(=O)NCCOCCC#C)CC(CO)(CN1C(C1CC3CC3C1)=O)C2 CC(C)C(C)C(CNC(c1cncc(Br)c1)=O)NC(c1cncnc1)=O Cc1nc(C2CCC2)oc1C(=O)NC1CCC1.c1(C(=O)N)cccn1C1CC1 N1(C(C=CC)=O)CCN(C(=O)C(c2ccc(Cl)cc2)C)CC1COC c1(C(=O)NCC2CC(NC(CC3(OC)CC3)=O)C2)cn(C)nn1 C1(C(=O)Nc2cc(C)cc(F)c2)CN(C(=O)CCC2CC2(C)C)CC1C1CC1 Cc1csc(Cl)c1C(=O)NCC(O)C.c1(C(=O)N)cnn(CCO)c1C(C)C C1(CC)NCCCC1C(=O)NNC(=O)c1cc(-c2ccccc2)on1 N1(C(C(C)=C2CCCC2)=O)CCCC2CN(CCOCC3CC3)CCC12 c1(C(N2CC3C(CCNC(CC#N)=O)(CC3)C2)=O)ccc2oc(S)nc2c1 C1(CC=O)NC(=O)NC1=O.C1(C(N(CCCOCC)C)=O)CCNC(=O)C1 c1(C(=O)NC2CNCC(=O)OC2)nc(C)cs1.c1(CC)ccccc1 c1(CC)nn(C)c(C(=O)N(c2ncc(SC)cn2)CC2CCNCC2(F)F)c1Cl C1(C(=O)Nc2ccc(OC)cc2)(COC)C=CCN1C(C1CCCN1C)=O N1(C(CC2(CSC)CC2)=O)CCC2CN(C(c3ccc(F)s3)=O)CCC12 C1(C(=O)NCCCC(O)CO)(CNC(C2CCCOCC2)=O)CC2(CC2)C1 N1(c2ncc(C(=O)OC)s2)CC2CCN(C(=O)CCC(C)C)C2C1 N=c1[nH]c2ccc(C(N3CCCC(CCNC(C4CCOC4)=O)CC3)=O)cc2s1 c1(C(=O)OC)ccc(C(=O)N(C2CCN(C(c3n[nH]c(C)n3)C)CC2)C)c(Cl)c1 C1(N2CC(OC)C(F)C2)CCC2(CC1)CCN(C(=O)CCc1ccc[nH]1)C2 N1(C(=O)OC)CCCC(OCc2ccc(N3CCOC3=O)cc2)C1 C1(CNC(C=COCC)=O)CCN(C(c2cc(OC)ns2)=O)C(C)C1 N1(C(CC(C)OC)=O)CCCCC2(CCN(CC(O)Cc3ccc(F)cc3)C2)C1 c1(C(=O)NCC2C(COC)C2)cnn(C2CCOC2)n1 CC1(O)CCCN(C(C2CC23CCN(C(=O)Cc2ccc(Br)cc2I)C3)=O)C1 C1(NC(c2c(C)cns2)=O)CCC2(CCN(C(=O)CCCCC#N)C2)C1 C1(C(N2CC(C)C(CNC(c3cnco3)=O)C2)=O)Cc2ccccc2N1 N1(C(c2c(C)sc(Cl)n2)=O)CC=C(CCNC(C2C3CC(F)(F)CC23)=O)CC1 N1(C(C2C(=C)C2)=O)CC2(CCN(C(=O)C(CCC)S(N)(=O)=O)CC2)C1 N1(CC(N2CCCC(C(N(C)Cc3cccnc3)=O)C2)=O)Cc2ccccc2C1 C(=O)(C(O)CC(C)(C)C)N1CC(NC(c2occ(C)c2)=O)C(n2ccnn2)C1 Cc1cn(CC(=O)NCC2CCCC2O)nc1C(F)(F)F.c1(C=O)cnco1.N n1(CCOC)c(C(=O)NC2CN(C(C3CC3C)=O)CCC2F)cc2ccccc12 c1(C(C=O)=O)cccc(C)c1.C(c1ccco1)=CC(=O)N(CC)C.C(N)=O c1(N(C(=O)C(F)C2CCC2)C2(C=O)CC2)cccs1.C(=O)C1CC1.CO N1(C(c2cc(C)cc(O)c2)=O)CCC2(CO)CN(C(C3(C)CCC3)=O)CC2C1 CC1COCCN1C1CCN(CCNC(c2cccc(CC(=O)O)c2)=O)C1 c1(CC)ccc(C(=O)NC(C)(CNC(C2CC2F)=O)C2CCC2)o1 N1(C(CCC)=O)CCC(C(C)(C)C)CC1.C1(CC(=O)N)CCC(=O)C1.C(N)=O C1(C(NOC(COC)COC)=O)CCCN(C(c2ccn(CCF)n2)=O)C1C C(C(=O)NCC(=O)OCC1CC1)(C(C)(C)C)NC(CC(C)F)=O C1(NC(c2cc(-c3ccccc3)[nH]n2)=O)CCN(C(C2CCCC2O)=O)CC1 N1(C(c2c(OC)c(Cl)ccc2)=O)CCC(C)C(NC(c2csc(C)c2)=O)C1C C1(C(=O)N)CCC(F)(F)CO1.C(C)(CC)N(C(CC1(C(=O)OC)CC1)=O)C S(=O)(=O)(CCCC(F)(F)C(F)(F)F)NC(c1ccc(O)c([N+](=O)[O-])c1)=O c1(C(=O)NCC(O)CNC(C2COCCO2)=O)ncccc1F C1(C(F)F)(CNC(C(CC)SC)=O)CCN(C(c2ncn(C)c2C)=O)C1 CC1CC2(CO1)CN(C(c1csc(-c3cccnc3)n1)=O)C2 c1(C(N2CCC(CCC)(Nc3cncc(Cl)n3)CC2)=O)ccnc2[nH]nnc12 c1(CN2CCCC(C(=O)Nc3cnc(Br)nc3)C2)c[nH]c2ncc(Br)nc12 c1(C(N2CC(NC(=O)C(O)C(C)(C)C)CC(C)C2)=O)c(F)cccc1[N+](=O)[O-] C1(CNC(C(C)OCC)=O)CCC(C(=O)NCCCCO)CC1.C(C)C N1(C(c2nc(CC)sc2)=O)CCCC2(CCCN2C(=O)CC2CCCCO2)CC1 C=CCCCCCC(=O)N1CC(F)(F)CC1CNC(c1nocc1C(C)(C)C)=O C1(NC(C2N(C(CC)=O)CCCC2)=O)CCCN(C(c2oc(C)cc2C)=O)CC1 C1(C)(CCC(=O)NC(c2noc(C)n2)CC)CN(C(C2CCCCC2)=O)C1 C1(NC(c2cc(C)no2)=O)CCCN(C(c2coc(C(C)C)n2)=O)CC1F C1(NC(C(C)C2CC2)=O)CC(F)(CNC(c2cccnn2)=O)C1 C1(NC(C(CNC(CC(=O)NCC)=O)O)=O)CCC(O)CC1 Cc1c(C(=O)NCC2CCN(C(=O)CC3CC(F)C3)C23CC3)cnc2ncnn12 C1(C(N(C)CC2CCCS2)=O)CN(C(C2(C(N)=O)CC2)=O)CC1F N1(CC)CCCC(C(=O)NCC(CC(=O)NCC(Cl)=CCl)C2CCC2)C1 C1(NC(=O)C=CC(C)(C)C)CCN(C(c2cc(SC(F)(F)F)c[nH]2)=O)C1 c1(OCC)cnc(C(=O)NCCCN(C)C(C2CCC(C)(C)C2)=O)cn1 N1(C(c2c(NC)nccc2)=O)CCCCCCC1C(N1CCC2CC12)=O C(=O)(C#CC1CCCC1)NC(CC(=C)C)C(=O)NCC1(CCO)CN(C)C1 C1(CNC(C(=O)N(C)C)=O)CN(C(c2cncc(C(F)(F)F)n2)=O)C2CC12 N1(C(C(CCF)NC(c2c(C)oc(C#N)c2)=O)=O)CCn2nccc2C1 c1(C(N(CCN(C(C)C)C(C)C)C)=O)nnc(N2CCCC2)o1 Cc1cnccc1C(=O)NCCC1CCCN(C(c2nscc2N)=O)C1 c1(CSC)ccc(C(=O)N(CC(C)CNC(c2ccnn2CCF)=O)C)o1 Cc1ncc(C(=O)NC(CCN(C)C(C2CCN(C)C2)=O)C(C)(C)C)c(=N)[nH]1 C(=O)(CCO)NCC1N(CC)CC1.C1(C(=O)NCC)CCCC1 CCCCCC(=O)NCC(C1CCC1)NC(=O)C(CCC)OCC c1(N2CC=CC(OC)C2)ccn2c(Br)cnc2n1 C1(C(=O)NC(CC2CCC2)CO)C2CC2CN1C(=O)CCC(=O)N1CCC1 N1(C(c2c(CC)scn2)=O)CCC2(CCC2)C(NC(C2CCCC3(CC3)C2)=O)C1 c1(C(N2CCCC(NC(C(c3cn(CC)nc3)=O)=O)C2)=O)ccc(F)c(C)c1 C1(OCC)CC2CN(C(=O)CC=CCNC(C3COC(C)C3)=O)CC12 c1(C(N2C(C)CC(NC(C=NOC)=O)C2)=O)cc(O)ccc1Br C(=O)C(C)(C)c1cscn1.c1(CC(=O)NCCC)cc(C(F)(F)F)cs1.C CCCCCCC(=O)NC(C1CN(C(c2cnoc2C)=O)C1)C C1(NC(=O)CCc2cnn[nH]2)COCCN(C(=O)Cc2sccc2Cl)C1 C(C(F)(F)C(=O)N1CC(C)C1)OC.C(=O)CCC(=O)N1CCOCC1.C(=O)C.N Cc1ccn(CC(=O)NC2CCCC2CNC(c2cc(C3CC3)cs2)=O)c1 c1(COCC)ccccc1NC(=O)Cc1nccc(C)n1.CCCCCC N1(C(c2ccc(C3CC3)cc2)=O)CCC2CN(C(=O)C(O)C3CCCC3)CCC12 Cc1cc(C(N2CC(CCNC(=O)COc3ccccc3)C2)=O)c2n[nH]cc2c1 C=Cc1cnn(C)c1C(=O)NCC(C1CC1)N(C)C(C1CCC(=C)CC1)=O C(CCCCC(=O)NC(CCSC)C(=O)NCCC(C)(O)CC)=CC CCCS(=O)(=O)C(C)C(=O)N1CCC(C)N(C(=O)Cc2nocc2C)CC1 C(=O)(C(C)(C)CN(C)C)N1CC(OC)(C)C1.C(=O)C(C)(C)C1CCOCC1 C(CC(C(=O)NCC12CC1CN(C(c1sccc1F)=O)C2)N(C)C)SC N(C1CCOc2c(NC)cc(C)cc21)C(=O)NCCSCC#C C1(c2cccnc2)(CNC(N(C(C)C)CC2CC2)=O)CCCCC1 CC(=O)CCCCC(=O)N1CCOC(CCCNC(=O)C(c2cnccn2)C)C1 C(N=c1ccc2nnnn2[nH]1)C1(C)CCN(C(C(c2ccccn2)C)=O)C1 CC(C)N=c1nc2c(cnn2C(C)C)c(NCCC2CCCO2)[nH]1 C1(NC(C=C(C)C(C)(C)C)=O)CN(C(=O)Cc2ncc(C(C)C)[nH]2)CC1C c1(C(N2CCN(C(CC3(OC)CC3)=O)CC2)=O)ccn2c1CSCC2 Cc1noc2cc(C(=O)NCCCC(C)NC(=O)CC(C)C(F)(F)F)ccc12 N(C(=NCC(O)Cc1ccccc1)NCc1csnn1)C(C1CCCO1)C N1(C(C2CC2C(F)(F)F)=O)CC2CCCC(C1)N2C(C1CCS1(=O)=O)=O N1(C(CN(CCC)C)=O)CC(CCNC(=O)CCN2C(=O)CCC2=O)C(C)C1 Cc1nc2ncnn2cc1C(=O)NC1CN(C(c2scnc2C(F)F)=O)CC1C C(=O)(CC1=NN(C)C(=O)C1)NC(CCC(C)C)C(=O)NCc1ccc(C#N)o1 C(=O)(CCC1=CCCCC1)NC1CN(C(C=Cc2nc(C)c(C)[nH]2)=O)CC12CC2 CC(C(=O)NC)S(C)(=O)=O.c1(CCC=O)cc(C(F)F)ccc1F.C1CCC1 C1(OC)(C)CCN(C(C2CCC2)=O)C1.C1(C=O)CCN(S(C)(=O)=O)CC1.N C(=O)(C1=NOC(CNC(c2cc(F)ccc2F)=O)C1)NCCCNC(N)=O c1(C(=O)NCC2CCN(C(Cc3c(C)nccc3)=O)CC2)cnn2ccncc12 C1(C(=O)N)C2C3CC4C1C2C34C=O.c1n[nH]c(C(F)(F)F)n1.C1CC=CC1 N1(C(C2CCCN(C(C)C)C2)=O)CCC(NC(C2CSCC(=O)N2)=O)C(C)(C)C1 N1(C(c2cnc(C)s2)=O)CCN(C(c2ccc(CCC(N)=O)cc2)=O)C2CCC12 c1(N(C(C(=O)N(CCC)C(c2nccs2)C)=O)CC)cc(F)cc(F)c1F c1(C=O)ncccc1OC(F)F.C1(CC(=O)N(CCC)CC)CC(C)=NO1.N c1(C(N2CC3CC2CN(C(C2(Cl)CC2(F)F)=O)C3)=O)ccnc2c1CCC2 c1(C(=O)NCC(C(C)C)NC(c2cccs2)=O)ccnc2ccnn12 N1(CC(=O)NCCc2c(CNC(C(CC)F)=O)nco2)CCCCC(O)C1=O N#CCCCCCC(=O)NCC(O)CNC(c1ccnc(Cl)c1)=O c1(OC)c(C)ccc(C(=O)Nc2cccc(C)c2)c1F.C1(CC(=O)N)CCOC1 CC#CCC(CO)NC(=O)C(CNC(C1CCC(N(C)C)C1)=O)CC1CCCC1 Cc1nc2c(C(=O)NCC3(C)CCN(C(=O)CC4CCC(C)C4)C3)cccc2o1 c1(CC)nc(C(=O)NC(C)CN(C(=O)C(C)N(C)C)CC)cs1 c1(OC)ccc(F)c(C(N2CCC(NC(c3nnc(C)s3)=O)C(CO)C2)=O)c1F Cc1ccc(CCC(=O)N(CC(C)(C)NC(=O)C(C)n2cccn2)C)c(C)c1 N1(C(=O)C=CBr)CC2(C1)CN(C(C1CC13CCSCC3)=O)C2 c1(C(N(CCC)CCNC(=O)CCC(C)C#N)=O)ccc2occ(C)c2c1 Cc1nc(C(=O)NC(C2CCN(C(=O)Cc3ccn(C(F)F)n3)CC2)C)nn1C C1(C(C)(C)O)CN(C(=O)Cc2cn(C3CC3)cn2)C1.C1(C=O)(CC)CC1 N1(C(C2(C#N)C(C)(C)C2)=O)CCC2C(C(=O)NCCCC3CCCCO3)C2C1 CCCC(C)C(=O)NCCOC1CCN(C(c2ccn(CC(F)(F)F)n2)=O)C1 C1(CC(=O)N(CC=C)CC2CC2)C(NC(=O)CSC)CC1O C1(C)(CC)CC(NC(=O)C2CC2)CN1C(=O)C=C(C)C(C)C N1(C(c2cc(COC)[nH]n2)=O)CCC(NC(c2ccoc2Br)=O)C1C(C)C Cc1cc(C)c2c(c1)N(C(c1cnn(C3CCC3)c1C)=O)CCC2 C1CCCN(C(C2CC(F)C2)=O)C1.CC(F)(F)F.C(=O)(C=CC)N(C)C C1(CCCC)CN(C(=O)CC2CCC(=O)NC2)CCN1C(C1CC(C#N)C1)=O CC(C)C(C(=O)NC(CNC(C1CSCCS1)=O)CO)NS(N)(=O)=O c1(C(N2CCC(CC)OCC2)C(=O)NCCOC)cn2c(F)cccc2n1 c1(C(N2CCCC3CC23)C(=O)NC2CC(F)(F)C2)ccc(-n2ccnc2)nc1 N1(C(CC2CC(OC)C2)=O)CC(NC(=O)C2CC2)CC12CCOCC2 c1(C(=O)NC(=O)CC2CCCC2C(=O)O)c(Br)ccc2ccccc12 N1(C(CC(COC)C)=O)CCC2(CCCCC2NC(c2ncc(F)cn2)=O)CC1 C1(C(N(CCNC(=O)C=C(C)C2CC2)CC)=O)Cc2ccccc2S1 C(C(C)(C)C(C)(F)F)(c1n(C)nnn1)NCCc1ncc(C(=O)OC)s1 C1(NC(C(CC)CN(C)C)=O)C2CCN(C(=O)Cn3ccnc3C(C)C)CC12 N1(C(=O)CN2C(=O)C=CC2=O)CC2(CNc3nc(CO)cc(O)n3)CC1CO2 C1(CC(=O)NC(CCC)C)C2CCC1CN(Cc1cc(Cl)cnc1Cl)C2 c1(C(=O)NCC2CN(C(C3C(OC)CCC3)=O)C2)cccc(O)c1Br CC1C(CC(=O)NCCCN(C(=O)CCc2ccc[nH]2)C2CC2)C1(F)F CON(CCC(=O)NC(C)CCC=C(C)C)C(=O)C(SC)SC.C(C)(C)=C N1(C(C(CC#C)O)=O)CC2CC(C1)C(CO)C2NC(c1ccc(CC#N)cc1)=O c1(C=O)ccnc(C(C)(C)O)c1.c1(CCC)ccc(C(=O)N)s1.CCC1CC1 C(=O)(C1CCCn2cnnc21)NCC1OCC2(CN(C(CCCCC#C)=O)C2)C1 C1(C(=O)NCCC(C)(C)NC(=O)CCCC2CCC2)C2CC(=O)CC12 CCCC(CCC)CC(=O)N1CC(NC(=O)CS(=O)C(F)(F)F)CC1CO c12cccc(c1)OC2=O.Cc1csc(C(C)NC(=O)CN(C)C)n1 C(=O)(C(O)C(C)(C)C)NC(CC=C)CNC(=O)C(C)Cc1ccc(OC)cc1 C1(Nc2c3nc(C)sc3ncn2)CN(C(=O)C=CC2CCC2)C2(CCCCC2)C1 N1(C(C(C(C)C)C2CCC2)=O)CCC(C)C(NC(c2ccc(CO)c(F)c2)=O)C1 c1(CSC)cn(CC(=O)N)nn1.c1cnn(C)c1.C(C)C.C(=O)C.C=O C1(C)(CNCCC)CCNCC1.c1(C(c2ccon2)CC)cnoc1-c1ccco1 C1(NC(C(C)CCO)=O)CCS(=O)(=O)C12CN(C(=O)Cn1cnc(=N)[nH]1)C2 C(=O)(C1=CCC(F)(F)CC1)NCC(CC)(CC)NC(CCCCCC=C)=O c1(C(=O)NCC(N2CCC2CNC(CC)=O)=O)ccc(Cl)cc1F c1(C(=O)NC(CCNC(c2c(CC)nns2)=O)(C)C)cccc2scnc12 c1(C(N(C2CCCC2)CCCNC(=O)Cc2ccon2)=O)ccn2ncccc12 CCCC(O)C(=O)NC(C1CN(C(=O)CNC(c2ccc(Br)o2)=O)C1)C C1(O)(CN(C(C2(COC)COC2)=O)C)CN(C(=O)C(F)C2CCOC2)C1 C(=O)(CCS(=O)(=O)C1CCCC1)NCCCC1OCCN(C(C2(C)C(C)C2)=O)C1 C1(NC(CN(c2ccccc2)C)=O)CCCC(NC(=O)C2=CCSC2)C1 c1(CN2CCC(NC(c3cnc(OC)c(F)c3)=O)C2)c(F)cc(C(=O)O)cc1F C1(C(=O)O)CCC2(CC1)CCN(C(=O)NCC1(CO)CCC1CO)CC2 C1(O)CCCN(C(C2C(C)(C)C2(C)C)=O)C1.C(C)(C(=O)N(C)C)SC(C)C N1(CC(N2C(CNC(C(C)(C)C)=O)COCC2)=O)C(=O)NC(C)(C)C1=O c1(NC(=O)CCC2CCN(C(=O)CCCC3CC3)C2)ccc(CCO)cc1 C1(C(N2CCCC(C(=O)NC(CF)C(F)(F)F)C2)=O)CC2(CCO1)CC2 c1(C(=O)NCC2CCN(C(C3N(C)CCC3)=O)CC2O)cnc2n1CCOC2 Cn1c(O)nc(NC2CCC3CN(C(=O)CS(N)(=O)=O)CC23)c([N+](=O)[O-])c1=O C(=O)(CCCC1CCCO1)N1CC(C(C)NC(C(C)c2ccsc2)=O)C1 c1(CC)nc(NC(=O)CC(Cc2ccccc2)Cc2ccccc2)cc(O)n1 C1(C(N(c2ncccn2)C)=O)CC2OCCC2N(C(c2ccc(Cl)c(Cl)c2)=O)C1 Cc1cccc(Cl)c1C(=O)NCC1CCC(C)CN1C(=O)CC1CCN(C)CC1 C1(C(=O)NC2CC(N(C(C(F)=C(C)C)=O)C)C2)CC12CCC2.C(C)(C)C Cc1ccc(C(N2CCOC(C)(CNC(=O)CS)C2)=O)c(N)c1.c1ccccn1 C1(CC(=O)N(CCCCO)CC)CC(O)CN1C(C1CC1)=O.C(C)(C)C.O C1(NC(C2(C)CCN(C)C2)=O)COC2(C1)CN(C(c1cc3c[nH]cnc-3n1)=O)C2 c1(C(=O)NCC(O)CNC(c2ccnn2CCF)=O)ccc(C2CC2)nc1 c1(CNCc2ccc(-c3cncc(N(C)C)c3)nc2)nc2ncccc2o1 C1(CN(C(CC2CC(CC)C2)=O)C)CCCN(C(=O)CC(F)F)C1 C1(NC(CCN(C(c2c(C)ncnc2)=O)C2CC2)=O)CCCC(C)CC1 c1(C(N(CCN(C(C2CC3CCC2O3)=O)CC)CC)=O)csc2ccccc12 N1(C(C(COC)(C)C)=O)CCN(C(c2cn(CCCF)nn2)=O)CC(CO)C1 c1(CC(C(=O)N)=O)ccc(F)cc1.CC1(C(=O)NC(C2CCCC2)C)CSC1 c1(OC)ccnc(C(=O)NC(C2(O)CCN(C(c3cc(C)sn3)=O)C2)C)c1F C1(OCC)CC2CCC1N2C(=O)Cc1cc(OCC(F)(F)F)cc(OC)c1 C1(NC(c2c(C(C)C)cco2)=O)CN(C(=O)C2=CCSC2)C2(CCCC2)C1 Cc1ccc(CNC(=O)CC(c2ccc(F)cc2)N)c(C)c1.c1cc(Br)c[nH]1.C C1(CC(=O)NC2CCC(NC(C3(SC)CCC3)=O)CC2)CCCCC12CC2 C1(C(=O)Nc2cnc(C(C)(C)C)[nH]2)CCC(n2ccnn2)CC1.NS(N)(=O)=O.C C(C(C)CN=c1nc(OC)cc(C)[nH]1)NC(C1(CC#C)CC=CCC1)=O c1(C(=O)NCC2OCCN(C(C3CCC(CC)CC3)=O)C2)coc2c1COC2 CC(C)S(=O)(=O)CCN=C(NCCC1(O)CCOC1)NC1CCS(=O)(=O)C1 c1(OC)cccc(C)c1C(=O)NCC(CO)NC(C1CC1C=O)=O.CCO C=C1CCC(C(=O)NCC2C=CCN2C(=O)COCCOC)CC1 CN1C(=O)CN(C(C23CC(CN2C(C2CC(C4CC4)=NO2)=O)C3)=O)CC1=O CC1(C)CN(C(c2cc(C(F)(F)F)no2)=O)CC1CNC(c1ccoc1)=O C1(CC(=O)Nc2c(C)nccc2)CC(C)(C)CN1C(=O)C#CC(C)(C)C c1(C(=O)NCC2CCN(C(c3ccno3)=O)C2)ccnc(C2CC2)n1 c1(CC(=O)NC(CC)CN(C)C(c2[nH]c(C)nc2C)=O)cc(C)ccc1C c1(C(N2C(CC(=O)OC)CC(F)C2)=O)cc2c(cc1[N+](=O)[O-])n(C)c(=O)n2C C1(CN(C(C2CCC(C)C2)=O)CC)CCN(C(=O)CSc2ccoc2)CC1 C(C(C(=O)N(O)Cc1cn(-c2nccnc2OC)nn1)OC)OC C=CC1CCN(C(CC(C)c2ccccc2)C(=O)NCCCC)CC1 C=CC1CN(C(c2c(C(C)C)cccc2C)=O)CC1NC(c1cncnc1C)=O C(CCCC(=O)NC1COC(C(F)F)C1)N(C(C(C1CCCCC1)C)=O)C C1(NC(CC(=C=C)C)=O)CC2CCC1C(NC(=O)C(O)C(C)CC)C2 c1(Cn2c(C3(NC(C)(C)CCF)C(C)CCC3)nnn2)ccc2c(c1)OCCO2 C(=O)(C(CCC(N)=O)n1cc(C2CCNC(=O)C2)nn1)NC1CC(C)(C)OC1 C(=O)(C(CC)C(C)(C)CC)N1C(C(N2CCC(C)(CC)C2)=O)CC(F)CC1 Cc1ccnc(S(=O)(=O)N2CCC(CC(=O)O)S(=O)(=O)CC2)n1 C1(C(=O)NCCCS)CCCC2(CCC2)C1.c1ccccc1.C12CC1C(=O)N2 Cc1ccc(C(=O)NC23CCN(C(c4ccc(F)s4)=O)CC2C3)c(N)c1Cl c1(C2(C(N(CCCCNC(C(C=C)O)=O)C)=O)CC2)cncc(Br)c1 c1(C(C(N2CC(O)C2)=O)NC(CC(CC)SC)=O)c(C)cccc1Br CCCCC(CNC(c1[nH][nH]c(=N)c1Br)=O)NC(=O)CC(C)CN(C)C C1(NC(C(CC)SC)=O)CCCC(C(=O)NC)C1.c1(C2CC2)nn[nH]n1 C=CCCN=C(NCCCN(C)C(=O)OC)NCC1(O)CCC(C)(C)CC1 C1(CNC(C(CNC(=O)CC(=O)NC2CC2)OC)=O)Cc2nccn2C1 C1(F)(C(=O)NCC2N(C(C(C)SC)=O)CCCC2)CCC(F)(F)CC1 N1(Cc2ccc(C#N)s2)CCN(C(=O)C=Cc2cccc(Cl)c2)C2CC12 N1(C(C(C)NC=O)=O)CCC(C(=O)N(C(CN2CCCC2)CO)C2CC2)CC1 C1(C(=O)NC2CCCC2)(CC)CCCCC1.C1(C=O)CCCN1C(=O)C1CC1 S(=O)(=O)(c1ccc(C#N)c(N2CC(C3CC3)OC(C)C2)c1)N(CCCS)CC c1(CCC(=O)NC2CCCC(NC(C(C)(C)SC)=O)C2)nnc(O)nc1O C=CC1OCCC1C(=O)NC1C2CC(NC(=O)Cc3cc(C)on3)CC12 c1(C2C(C=O)C2)ccc(Cl)c(C)c1.N1(C(CNC(=O)OC)=O)CCCCC1.N CC1CC(=O)NCC1C(N1CCC(C)CC1)=O.C1(C(C(=O)N)O)COC(C)(C)O1 C=CCC(C)(C)CC(=O)NCCCN(C(=O)CC(C)O)C.C(C)(C)C.C=O.N c1(CN(C2CN(C(c3ccc(Br)cc3O)=O)C2)C)csc2ccc(Cl)cc12 C1(C(=O)NC2CC(CC)OCC2)CC(C)(C)CCN1C(c1ccncc1O)=O C(=O)(CCCC(C)(C)CC)N1CCCC2(NC(C3N(CC)C(=O)CC3)=O)C(C1)C2 c1(C(=O)NC2C(NC(=O)CCC=CBr)CCOC2)ccc(O)cc1F CC(=Cn1ccnn1)C(=O)NCC(C)(F)CNC(c1ncn(C)n1)=O C(=O)(CC(CN(C)C)C(F)F)N1CC(CNC(c2cccc(C)n2)=O)C(O)C1 c1(C(=O)NC2CN(C(C3CC(C(C)C)C3)=O)C(C)CC2)ccc2c(n1)OCCO2 c1(CC)ccc(C(N2CC(NC(c3ccc(F)s3)=O)C(C)(C)C2)=O)c(C)n1 CC(C)P(=O)(CC(=O)N1CCCC1C(C)NC(C1CNC(=O)N1)=O)C(C)C C1(NC(=O)CC2CC3CC3C2)CCN(C(c2cnc(Cl)cc2Cl)=O)C12CCC2 CCCC(CC(C)C)C(=O)NC1CN(C(=O)C(C)NC(N)=O)CC2(CC2)C1 c1(OC)cc(C(=O)N(C)CCN(C(=O)C(O)C2CC2)C)ccc1C(N)=O c1(OC)ccnc(C(=O)NCC(C)NC(c2cccnc2OC(F)F)=O)c1F c1(C(=O)NC2(CC=C)CCCN(C(=O)CN3CC(C)C3)C2)nc2cnccc2s1 C(CC(C)C)(C(=O)NCc1ncnn1C)ONC(c1cc(CC)sn1)=O c1(C(=O)NC2CN(C(CCCOC)=O)CC2(C)C)ccn2cc(C3CC3)nc2c1 Cc1onc(C(F)(F)F)c1C(=O)NC1CCC(NC(C2CCC(C)S2)=O)CC1 C(C)(CSC)(C(=O)NCC=CC(O)(CC)CC)NC(C(C=C)O)=O c1(C=O)cc(O)n(C)n1.N1(N(C(=O)C(F)(Cl)c2ccccc2)C)CC2CC2C1 Cc1ccc(O)c(C(=O)NCC2(F)CCC(NC(=O)CCC)C2)c1.C(N)=O c1(CC(N2CCCC(n3cc(COCC)nn3)C2)=O)c(C)cc(Br)cc1C N1(C(CNC(c2cc(C)on2)=O)=O)CCC2(CC1)COC(CNC1NCCC1O)C2 C1(CC(=O)NCc2c(C)scn2)CN(C(C2(C)CCCOC2)=O)CC12CC2 C1(NC(C2C3CN(C(CN4CCC(C)C4)=O)CC32)=O)CCCN(C)CC1 N1(C(c2cc(CC)[nH]n2)=O)CCOC(CNC(C2(Cl)CC2(C)C)=O)C1 N1(C(C2C(C=C)C2)=O)CC2CCN(C(c3cc(OC)c(O)c(Cl)c3)=O)C2C1 C(=O)(CCCCCCNC(c1cc(C)n(C)c1C)=O)N(CC(C)(C)O)CC N1(C(c2cc(CC)oc2)=O)CCC(N(C)C)CC1.c12c[nH]cc1C(=O)NC2 N1(C(c2c(OCC)ccs2)=O)CCC(O)C(NC(=O)C(C)C2CC2)C1 CCCS(=O)(=O)C1CCN(C(C(=O)NC2CCOCC2)C(C)C(C)(C)C)CC1 c1(C(N2CCCC(NC(C(=O)NCC)=O)(CC)C2)=O)ccc2c(c1)CCO2 CC(C(C)(C)C(=O)N1CCC(C(C)CO)CC1)NC(=O)C=Cc1cnn(C)c1 C(C)C(O)C(F)F.C1CC(=O)N1.C(=O)(C(C)N1CC(C)C1)N(CC)CC.O CCC(CC(=O)N1CCN(C(=O)CC(C)C(F)F)C2(CCC2)C1)C(C)(C)C C1(C(F)(F)F)CC(F)(F)C1.C1(N(C(C(C)n2cncn2)=O)CCO)CCNC1.C C1(CNC(Cc2c(C)nsc2)=O)CN(C(=O)CNc2ccccn2)CCO1 O=C(N=c1ccn(CCO)[nH]1)C(=O)N1CC2(CCC2)OCC1CO c1(C(N2CC(CN3CCN(C(C=CCCC)=O)CC3)C2)=O)nc2cccnc2s1 C(=O)(C1=COCCO1)N(C1CN(C(c2cc(C)nn2CC(F)F)=O)CC1O)C CC(CCC(C)(C)C)C(=O)NC1CC2CCC1N2C(=O)C=Cc1ccco1 c1(C(=O)NCCOCCCN(C(C(CC#C)C)=O)C)cccc(Br)c1Cl c1(CC(=O)NCC(CNC(c2c(CCC)nco2)=O)F)cccc(F)c1Cl C1(C(N(CCCCCC=C)C)=O)C(C2CC2)CCN1C(=O)Cc1cnns1 C(=O)(C(C(C)NC(c1ccoc1)=O)C(C)C)Nc1cnc(SC)nc1 CCC(CC(=O)NC1CC(CCC(=O)N(C)CCc2cc[nH]n2)C1)C1CC1 Cc1ccc(NC(=O)C(=O)NCCC2(O)CCCNC2)nc1.C1(N)CC1 C(O)(C(C)C)C1(NC(CC2(OCC)CC2)=O)CC1 c1(CNC(C2CC(C=O)C2)=O)cccc(OC)c1.c1cccnc1.C1CC1 c1(C=O)cscc1C=O.C1(C(=O)NCCCN(CCC)C)(CC)CCC1.N C(C)(C)(CC(F)C(=O)N(C)OCC(=O)OC)NCc1c(CC)cns1 C1(C(=O)NCC2CCCC(NC(C(CC)(C)C)=O)C2)CCS(=O)(=O)CC1 c1(C(=O)NC(C(C)NC(C(CC)(C)C(N)=O)=O)CO)ccc2c(c1)COCC2 c1(CN(C(C(C)C#N)=O)C)cccc(CNC(C2CCS(=O)(=O)C2)=O)c1 N1(C(C)=O)CCCC1(C)C(=O)NCC1(O)CN(C(=O)CCC(C)N(C)C)C1 c1(C(=O)NC(C(C)NC(=O)CC2(CO)CC2)C)snc(O)c1Cl Cc1ncnc(C)c1OCC(=O)NCC1CC1C.C(=O)CCS(C)(=O)=O N1(C(c2cn(CCCOC)nc2)=O)CC(NC(c2cccc[n+]2[O-])=O)C2CC12 Cc1ccsc1C1CC1C(=O)N(CC(C)(C)NC(C1CCS1(=O)=O)=O)C N1(C(c2cn(CC(CC)O)nn2)=O)CC(C2CN(C(c3n[nH]cc3Br)=O)C2)C1 C12(C(=O)O)COCC(CN(C=O)C1)C2(F)F.N#Cc1ccccc1SC(C)(C)C c1(C(=O)NC)c(F)cc(F)c(F)c1F.C1(C=O)C2CC3C(C2)C13.C1CC1 c1(NC(c2c(C(C)C)c3c(o2)cccc3)=O)ncc2c(n1)CCOC2 c1(NCCC2OCCN(C)C2)nc(N2CCC(N(C)C)C2)nc2c1ncn2C c1(COC)nc(CC(=O)NC(C2CCCN2C(C2CCCCC2)=O)(C)C)cs1 c1(SC)cc(N2CC3C(NC(=O)CCCSC)C3C2)nc(SC)n1 C(C)(C(=O)N1OC2CCC1CC2)NC(C1C(C)CCOC1)=O N1(C(C(CC(C)C)=O)=O)Cc2occ(C(=O)N(CC(C)C)CCO)c2C1 C(=O)(C(=O)C(C)(C)CC)N1CCC(C(=O)NC(C2CCCC2)C#C)C1 CC1(C)CN(C(=O)Cc2ccno2)CC1CNC(C1(C)CNC(=O)C1)=O C=CCC(C)(C)C(=O)NCc1ccc(C(N2CCNC(=O)C2)=O)cn1 N1(C(c2c(CC)ocn2)=O)CCC(CC)C1COC.C1(CC(=O)N)CCOCC1 N1(C(C(C)(C)c2ccccn2)=O)CCC(CCNC(=O)C)C(F)(F)CC1.C1CC1 C1(O)(CN(C(=O)CC2OCCO2)C)CCN(C(C2(C)CC(F)(F)C2)=O)C1 c1(C(C)NC(N2CC(C(F)F)(OC)C2)=O)c(-n2cccn2)cccc1F C1(CC#N)(CC)CCCN(C(=O)Nc2ccc(C)c(F)n2)C1 N1(C(C2CC3CC3C2)=O)CCOC2(CCC(Nc3ncc(C(F)F)cn3)CC2)C1 C(CCN=c1cccc(S(=O)(=O)NC2CC(CC#N)C2)[nH]1)c1ncn(C)n1 C(=O)(C1CCCc2ncc(C)n21)N1C(CNC(CC2CC(=C)C2)=O)CCCCC1 c1(OC)cccc(OC)c1C=O.c1(C(N(CCC)C2CC2)=O)cc(Br)no1.N S(=O)(=O)(c1ccc(NC(C)COC2CCOC2)cc1Br)NCCOC(C)C C(CN=c1[nH]c2c(c(=NC3CCCC(O)C3)[nH]1)COC2)c1n(C)ncn1 CCC(CN(C)C)CC(=O)NCC(F)CNC(=O)C(=O)NCC(F)F c1(N(C)Cc2cccc(F)c2)nc2cc[nH]c2c(=NCc2cccc(Br)n2)[nH]1 CCC(C(=O)N1CCCC(O)(CNC(C23CC(C)(CCO2)C3)=O)C1)C(C)C N1(c2nnc(-c3c(=N)[nH]c(C4CC4)nc3)n2CC2CC2)CCN2C(=O)OCC2C1 C(=O)(C1CCCn2c(Br)cnc21)N1CC(NC(C2CN(c3ncc(F)cn3)C2)=O)C1 N1(C(=O)Nc2ccc(CC)c(C)c2)CC2(CCC2)CC1COC C1CN(C(=O)CCc2nccs2)CC1n1ccnn1.O=C(CC1(C(F)F)CC1)N N1(C(C(COCC)(C)C)=O)CC2CCC(C1)N2C(C1CC(O)C(F)C1)=O C(CCC(C)(F)F)N(CCC(C)(C)C)C(=O)C(=O)N1CCCC1 C(=O)(C(COCC)NC(=O)CC(C)n1ccnc1)N(CCCC=C)C C(=O)(C(C(=O)O)C(C)C)N1CC(C(C)NC(C=CC(CC)=CC)=O)C1 c1(NC(=O)CC2CN(Cc3ccoc3)C2)cc(Br)c(O)cc1Br C(=O)(C1=CC2(CCN(C(=O)C(=O)NC3CC3)C2)C1)NCC(C(C)C)C C1(C(=O)NCC23N(c4c(C)cnc(C)n4)CC(C2)C3)CCc2c[nH]nc2C1 C(=O)(CS(=O)(=O)C(C)C)NC1C(CC)N(C(c2cnc[nH]2)=O)CC1 C1(NC(CN(C(C)=O)C)=O)CN(C(=O)Cc2coc(-c3ccsc3)n2)CCC1C Cc1cc(C(=O)NC(C2CN(C(=O)C=C3CCCCC3)C2)C)cc2nn[nH]c12 N1(C(c2nc(C)sc2C)=O)CC2=C(C1)CN(C(=O)CCC1COC(C)(C)O1)C2 c1(N(S(C)(=O)=O)CCC#N)nc2c(s1)CCc1sccc1-2.C1C(=O)N1 N1(C(c2ccc(SC)o2)C(=O)NCC(=C)C)CCOC2CCCCC12 c1(C(=O)NC(C)CCCNC(C2CCC(O)CC2)=O)ccc(C2CC2)cc1F c1(OC)ccc(Cl)c(NC(C2CCC(NCc3cnc(Cl)cc3C)CC2)=O)c1Cl C12(C=O)CC(CN(C(=O)CC3COCCO3)C1)C2.C(=O)(NCC)NCC C1(NC(C2(SC)CCC2)=O)CCC(CNC(=O)C=C2CCSCC2)CC1 c1(C=O)ccc(Cl)c(F)c1.c1(CC)ccccc1.C1(CCOC)CC1C(=O)N C(=O)(CC1CCCc2ccccc21)N1C(COC)(CNC(=O)CC(C)C)CCC1 CC(CC(F)(F)F)C(=O)N1CC2C(N(C)C(C3CC(=C4CC4)C3)=O)C2C1 N1(C(Cn2c(C)c(Cl)cn2)=O)CC2(C1)CN(C(=O)C(C)CC(C)(C)C)CC2CO c1(C(N2CC(NC(c3n(C)ncc3)=O)C(F)CC2)=O)cnc2ccc(Br)cn12 N1(C(c2cc(C(F)(F)F)n[nH]2)=O)CCN(C(C2(CO)CCCO2)=O)CC(O)C1 c1(C(=O)NC2CCN(C(=O)C(O)CC3CC3)C2)cnc(O)c(Br)c1 c1(CN(C(CC)C(=O)NC2CCS(=O)(=O)C2)C)ccc(C)cc1Cl C12(NC(c3cc(C)nc(C)n3)=O)CCCC1N(C(=O)CSc1cnn(C)c1)CC2 C#CCC(CC#C)NC(=O)CC1CC(NC(c2nc(C)c(C)s2)=O)C1 c1(C(=O)NCCC(C)NC(C2CCC=CO2)=O)cnc(O)o1 C(=O)(CCC(C)CC)N(CCCNC(c1ncn(CC)n1)=O)C(C)C c1(-c2ncn(C)c2C(=O)N2CC3=NNCC23)ccc(C#N)c(F)c1 N1(C(Cc2c(C(=O)OC)cccc2)=O)CC(NC(c2ccoc2)=O)CC(F)C1 N1(C(C2ON=C(CC)C2)=O)CCC(C(=O)NCCc2ccc(O)nc2)C(O)C1 CC1(C)CCCCC1C(=O)NC1CCCC1NC(=O)CCc1ccc(F)cc1 CC1CCC(CNC(=O)C)CN1C(=O)CCn1cnc([N+](=O)[O-])c1.C1CCC1 N1(C(C)C)N=C(C(=O)NCC(C(C)C)NC(C2CC(F)C2)=O)CCC1=O c1(NC(c2c(-c3c(OC(C)C)nccc3)c[nH]n2)=O)cnc(Br)c(I)c1 CN1CCN(C(c2ccc([N+](=O)[O-])o2)=O)C(C(=O)NCC2(O)CC2)C1 c1(C(C)C)nc2n(n1)CC(NC(=O)NCCCN1CCCC1)CC2 CC1CCC(Cc2ccc(F)cc2)CC1.c1(C(=O)OC=O)cc(CO)c(Cl)s1 C1(C(=O)NC2C(NC(=O)CC(O)c3ccccc3)C2)CC2CCCC(C1)C2 Cc1cnc(CN(C(=O)C(CNC(=O)CC2CC3CCC2O3)N(C)C)C)cn1 Cc1cccn(CC(N2CC(NC(c3c[nH]c(Br)c3)=O)C(C)(C)C2)=O)c1=O C(=O)(C1=CCCC(C)(C)C1)NCC1CCN(C(Cc2cc(C)n(C)n2)=O)C12CC2 C(C(O)C(=O)NCC(O)C(=O)NCc1cn(C2CC2)cn1)N(C)C c1(CNC(C2C3CN(Cc4nc(C)[nH]n4)CC32)=O)cc2n(n1)CCCC2 C1(CC(=O)NC(c2c(C)ncs2)C)CCCCN1C(C1CC1C(C)(F)F)=O c1(CCC(=O)NCC(C)C)nc(-c2ccsc2)no1.C1(CC=O)CCNC1=O.N C(=O)(C1=NN(CC)C(=O)CC1)NCC(CCOC)NC(C(CC)F)=O c1(-c2cnc(OC)c(C)c2)n[nH]c2c1CN(C(c1cncn1C)=O)CC2 c1(C(N(CCCN(C)C)CC)=O)cc(O)cc(=O)o1.CC1CN(C(=O)O)C1 C1(C(=O)N)CC(C)CN(C(C2COCC2C(N)=O)=O)C1.C(C(C)(C)CO)OC C(CCCCCNC(C1CN(C2CCOC2)C1)=O)N(C)C(C1CCC2(CC2)C1)=O C#CCC(C(=O)NCC(F)CO)NC(C1CCC(F)(F)C1)=O C(=O)(CCCC(N)=O)N(C(CNC(=O)CNC(=O)C1CC1)C1CC1)C N1(C(C(=O)N(C)Cc2ccc(C3C(C)C3)o2)=O)CC2(C1)OC(=O)NCO2 c1(C(CNC(c2ccc(F)cn2)c2n(C(C)C)nnn2)(C)C)ccncc1Cl C12(NC(CCC=CCC=C)=O)CC1CN(C(C1CCCN1C=O)=O)C2 C1(C(=O)NCC(C(=O)NC(C)C(C)(C)CO)(C)C)CCCC(C)(C)C1 N1(C(c2ccn(CC)n2)=O)CC2=C(C1)CN(C(=O)Cc1csc(CO)n1)C2 C1(CCNC(C(C)OC2CCOCC2)=O)CSCCN1C(=O)C1=CCCS1 CCC(C)(CCNC(c1ccc(C2CC2)cc1)=O)NC(=O)C.c1ccccc1.O c1(COCCOC)nnc(C)c(C)c1C(=O)NNC(C)=O C1(CC)(NC(=O)CC(C)CNC(=O)Cc2cnsc2)CCOCC1 C1(C(=O)NCC2(CNC(C3CCCC3)=O)CCC2)CCCCC12OCCO2 CCC(C)CCCC(=O)N1CCN(C(C2Cc3ccccc3C2)=O)CC(CO)C1 C1(NC(C(C)C=Cc2ccccc2)=O)CC2(CCN(C(=O)CC3CC3)C2)C1.C Cc1cc(C)c(C(=O)N)c(Cl)n1.c1(CC(N2CC(=C(C)F)C2)=O)nnc(C)s1 c1(C(N(C(C)(C)CC(=O)NCc2c(O)cccc2F)C)=O)cccc(F)c1N C(C1=CCCN(C(C2CCN2C)=O)C1)NC(CC1ON=C(C)C1)=O C1(OC)(CNC(C2CCC(=O)N2C)=O)CCN(C(C2CC(=O)C2C)=O)C1 n1(CC(=O)NCC(CC)NC(=O)CC(C)COC)nc2n(c1=O)CCCCC2 c1(C(N2C(CNC(CCCCCC(C)C)=O)CC2)=O)cccc2c1CC(C)(C)C2 CCCCCC(F)C(=O)NCC(C)CN(C)C(c1cccn1CCC)=O n1(C(CC)C)nnnc1C(C1CCCO1)(C)NC(C)(C)CF CS(=O)(=O)CCCCCCCC(=O)N1CC2=C(C1)CN(C(C1C3CCCC13)=O)C2 N1(C(C2CCC(=O)O2)=O)CCCC(N(CCF)C(c2cnsc2)=O)C1 Cc1csc(C(N2CCCC(CC(N3CC(SC(F)F)C3)=O)C2)=O)c1C CN1CCC(CN(CC(O)C(C)(C)C)CC2CC2)CC1 c1(NC(N2C(CO)CC(OC)C2)=O)ccc(N2CCOCC2)c(C)c1 c1(CN(C(c2ccc(C)nc2)C(=O)NCCC)C)c(C)nn(C)c1Cl c1(C(C)=O)cc2ccccc2o1.c12ccc(cc1)C(c1ccccc1)N2 c1(N(C)Cc2cn(C)cn2)nc(=NCC(C)(C)C(N)=O)[nH]c2c1CCCCCC2 N1(C(c2ncc(CC)cn2)=O)CCC(NC(c2ccco2)=O)C(C)(C)C1 N1(C(c2cnn(C)c2Br)C(=O)NCC2CCCO2)CCOCCC1C(F)F c1(CN2CCN(C(=O)CSc3nc[nH]n3)C3C2C3)cc(F)cc(F)c1Br C1(C(N(CCC)Cc2ccccc2OCC)=O)Cc2cc(Cl)ccc2C(=O)O1 C(=O)(CC(F)(F)C(F)F)N1CC(C)CC1.Cc1nn(C)c(C)c1CCC(=O)NC c1(NC(=O)Nc2cccc(I)c2)ccc(OCC(F)(F)F)nc1 N#Cc1cc(F)ccc1CNC1CC(NC(c2n[nH]c3ccccc23)=O)C1 c1(C(=O)NCC(CN(C(C(C)N(C(C)=O)C)=O)C)C)cc(C)c(Cl)cc1C N1(C(C(=O)NC(C)C)=O)CCC(CO)(NC(=O)CN2CCCCC2)C1 C1(CNC(C2C(CC)C2)=O)CN(C(c2cc(C)cc(F)c2)=O)C(C)(C)C1 C1(NC(c2cc(C3(C)CC3)n[nH]2)=O)CCCCC1.C1(CC=O)CCC(=O)N1C.N C1(C(=O)NCC2(NC(CC(CC)SC)=O)CCCC2)Cc2cc(F)ccc2O1 c1(CC(N2CCC(CC(=O)NC(CC)C)C2)=O)cc(C)nn1C Cc1cccc(CNC(=O)CC)c1.C1(C(C)C)CCCN1C(=O)CNC=O.N c1(CC)ccc(C)c(NC(=O)C=CC2CCCN2C(=O)CC2COCC2O)c1 c1(CN2CC(CC(N3CC4CCC3CO4)=O)OCC2)ccc(F)cc1Br N1(C(C#C)=O)CCCC2(CCN2C(c2csc(C)c2C)=O)C1 c1(C=O)cc2n(n1)CCCC2.c1(C(C)C)oncc1C(=O)NC1CCC(C)C1.N c1(C(=O)NCCCCCNC(C(C)C2CCCO2)=O)ccc(O)c2ncccc12 NC(=O)CCCCC(=O)NC1CC2CC1N(C(=O)C(F)(F)C(O)C1CC1)C2 C12(NC(COC(C)=O)=O)CCC(NC(=O)CCCCCN(C)C)(CC1)CC2 C(CC(C)CC)NC(C1CCC(OC)C1)=O.n1(CC(=O)N)cc(C2CC2)cn1 CS(=O)(=O)C1CCCC1C(N1CCC(CNC(C23CCCN2CCC3)=O)C1)=O Cc1ccc(F)c(C(=O)NCC(O)CNC(=O)CC2CCC3(CCC3)CO2)c1N C#CC1CCN(C(C23CC(CO2)N(C(c2cnn(C)c2OC)=O)C3)=O)CC1 NS(=O)(=O)CCCC(=O)NCCC1CN(C(c2ncn3c2CCC3)=O)CCO1 N1(C(CC=CC)=O)CCN(C(=O)CCOC2CCOC2)CC1c1ccncc1 N1(C(C2(F)CN(C(C(C)SC(C)C)=O)C2)=O)CC(CO)CCC1C Cc1ncncc1C(=O)N(C)CCN1CCN(C(=O)C=Cc2ncco2)CC1 C#CCC(CC#C)C(=O)N(C1CCC(NC(C2CN3CCCN2CC3)=O)CC1)C C1(NC(CSC)=O)CCCCC1CNC(=O)CC1CC2(CC2)CO1 n1(CC(=O)NCCNC(c2c(C)nncc2)=O)ccc([N+](=O)[O-])n1.C1CC1 C1(C(C(N2C(C(=O)NCC3CCCS3)CC2)=O)O)CCOCC1 C(CC1CCC1)(C(=O)N=c1ccn(CCO)[nH]1)NC(c1c(C)snc1)=O C1(C(N2CC(CN(C(CC3C(C)CCO3)=O)C)C2)=O)CCc2nc(O)[nH]c2C1 c1(C(N2CCC(C(C)(C)NC(=O)C=CC=C(Cl)Cl)C2)=O)cccc2cncn12 N1(C(C2C(C)(C)CC2)=O)CC(F)(F)CC1(C)CNC(c1ccc(O)nn1)=O c1(CCC(=O)N(C(C)CNC(c2ccc(Cl)nc2O)=O)C)ccc2c(c1)OCO2 CCCCC(C(=O)NC(CN(C)C)C(C)(C)C)NC(=O)CCc1cnc(C)o1 C1(CC=C)(NC(=O)C(C2CCOCC2)=O)CCCN(C(=O)CC2CCCC2C)C1 C1(C(=O)NC(C2CCN(C(c3c(C)ccn3C)=O)CC2)CO)CCCCC1(C)C c1(OCC)ccc(CC(=O)NC2(C)CCN(C(c3cc(CF)on3)=O)C2)cc1 C(=O)(CCCN=[N+]=[N-])NC1C=CCN(C(C2(C)N(C)CCC2)=O)C1 c1(C(N(C2CCN(C(C(COC)OC)=O)C2)CCO)=O)nn(C(F)F)cc1Cl CC1CN(C(c2ccc(Cl)cc2Cl)=O)CCCN1C(=O)C1=C(C#N)CCC1 C1(C(=O)NCC=CCNC(c2n(C)c(S)nn2)=O)CCS(=O)(=O)C1(C)C c1(CC(=O)NCCC2CCN(C(C(CO)N(C)C)=O)CC2)ccc2c(c1)COC2 C(=O)(C1CCCc2sccc21)NCC1(F)CC(NC(=O)CCn2cccc2)C1 C(=O)(CCCC(C)(C)C)N1C(C(C)NC(c2c[nH]c(=N)s2)=O)COCC1 Cc1cc(O)cc(O)c1C(N1CCC(F)(C(=O)NC(C)(CO)CO)CC1)=O C1(C(=O)NC(C)CC2CC2)C2CCC(C2)N1C(c1cc(C(F)F)[nH]n1)=O C(=O)(C1CCCn2cnnc21)N1CCC(CN(C(=O)C(F)CC(C)(C)C)C)C1 N1(C(c2cnc(CC(C)C)s2)=O)CC(NC(c2cncc(Cl)c2)=O)CC(F)C1 N1(C(C)=O)CCN(C(c2ncc(C)cc2O)=O)CC(O)C1 n1(CCC)nnnc1C(C)(CCc1ccncc1)NC(CC)CC N1(C(c2cc(C)c(F)cc2)=O)CCC2CN(C(=O)Cc3cc(C4CC4)on3)CC12 Cc1cc(CN2CCC(C(=O)Nc3nccc(C)c3Br)C2)c(O)c(C)c1 C1(NC(C(c2scc(C)n2)C)=O)CCCCC1NC(c1cnsc1C)=O C1(C(=O)NC(CCCOC)C)CCCN(C(=O)NCCC(C)(C)O)C1 c1(C2(F)C(C(N3CCN(C(=O)CC4CCCO4)CC3)=O)C2)ccccc1Br c1(C(N2CC3(N(C(C(C)(O)C4CC4)=O)CC3)C2)=O)cc2nc(F)ccc2o1 Cc1ccc(C)c(CC(C(=O)NC2CC2NC(=O)C2=NNC(=O)C2)C(C)C)c1 C(N=c1cc(Cl)[nH]c(C(F)(F)F)n1)C1C(NC(c2ccc(CO)o2)=O)CCCC1 CCC(C)C(C(=O)NC1CCOCC1)NC(=O)OC.C(C(C)CC)=CC=O.C N1(C(c2c(C)ccc(OC)n2)=O)CCCC12CCCN(C(=O)C(C)SC)C2 c12cccc(c1)O2.c1(C(N(CCN(CC)CC)CC)=O)cc(C#N)no1 n1(C(C)(C)C)nnnc1C(c1ccn[nH]1)NCCOCC(N)=O.C1CC1.C c1(C(=O)NC2CCN(C(C3CC(=C)C3)=O)C2C)nc2cc(F)ccc2s1 c1(NC(C2N(C(c3cnc(C)nc3)=O)CC(F)C2)=O)ccc2nc(C)sc2c1 C1CC(F)(F)CN1C(=O)CN1CCC(=O)NC1=O.Cc1cnn(C)c1C(=O)N N1(C(c2c(Br)c(C)nn2C)C(=O)NCCCSCC)CC2CCC2(OC)C1 N1(C(c2ccn(C)c2)=O)CCCCC1CNC(=O)Cc1cccnc1Cl N1(C(c2c(C)onc2)=O)CCC(F)(F)C(NC)C1.c1ccc(F)c(C(F)(F)F)c1 c1(C(N2C3(C(=O)NC4CCC(N(C)C)C4)CC(C2)C3)=O)cc2n(c1)CCCC2 C12(C(=O)NC3CN(C)C(=O)C3)CC(CCO1)N(C(=O)C=Cc1ccnn1C)C2 C1(NC(CC(C)(C)OC)=O)CN(C(c2nc(C)ccc2F)=O)C(C)(C=O)C1.N c1(C(=O)N)c(F)ccc(F)c1O.c1(C(C)C(=O)NC2CC2C)nc(F)ccc1Cl c1(CC(=O)N)ccc(C)c(O)c1.c1(OC)nn(C)cc1C(N1CC2CC2C1)=O S(=O)(=O)(c1ccc(C(N2CCN(C(C)CO)CC2)C(=O)N)cc1)NC.C1CC1.C C1(C2CCN(C(c3csc(Cl)n3)=O)CC2)(NC(c2ccc([N+](=O)[O-])[nH]2)=O)CCC1 C(CN=C(NC1CC1)NC1CC(=C2CCC2)C1)c1ccc(C#N)s1 C1(C(=O)NCCc2cc(C)no2)CC2CCC(C1)N2C(=O)C(N)c1ccco1 C1(NC(c2n(C)cnc2)=O)CN(c2ncc3c(n2)CCCC3)CC2(CCC2)C1 Cc1cc(CC(=O)NCC2CC3CC2CN3C(=O)C=CCO)cc(C)c1 C#Cc1ccc(F)c(C(N2CCC(N(CCC)C(c3ccnc(C)c3)=O)C2)=O)c1 N1(C(CN2CCC(C)C2)=O)C(CC(=O)NOCC2CCC2)C2CCCC12 C1(C(=O)OCC(=O)Nc2ccncc2)CC2CCC1O2 c1(C(N2CC(O)(CNC(C3(C(=O)OC)CC3)=O)C2)=O)c(C)nsc1C C1(C2CC2)CCCCC1.c1ccc(C=O)cn1.C1(OCC)CCC1C(=O)NC CC1CN=C2NC(C(=O)NCCCNC(c3cccc(OC(F)F)c3)=O)=NN2C1 C1(C(N2C(CNC(c3cncc(Cl)c3)=O)CC2)=O)CC2CS(=O)(=O)CC2C1 C(C(=O)NCC(C)(C)O)(C(C)(C)C)N(C)C.C12(C=O)CCC(CO1)C2.CC C(C(O)CN=c1cc(NC(=O)CCn2c(C)cc(O)cc2=O)nc[nH]1)OCC c1(C2C(C(N(CC(=O)N(CCNCC)CC)C)=O)CC2)nncn1C Cc1ncccc1CC(=O)NC1COCC1N1CCN(C(=O)C(=O)N(C)C)CC1 c1(CCC(=O)N(CC(CC)NC(=O)C#CC2CCOC2)C)nc2cccnc2[nH]1 N1(C(Cc2ccc(C)cc2Br)=O)CCC2CN(C(=O)CCc3cnc[nH]3)CC12 C1(O)(CCNC(c2c(C)coc2C)=O)CCN(C(C2CN(C)CCO2)=O)CC1 C(=O)(C(CC)C(=O)N1CCC2CC12C(=O)N(C)Cc1cnnn1C)OCC C(=O)(C#CC1(C)CC1)NC(C)Cc1cccc(Cl)c1 N1(C(Cc2ncc(C)o2)=O)CC2C(CNC(=O)COc3cccnc3)C2C1 C1(C)(NC(C(C)NC(C2CCCS2)=O)=O)CCC(=O)N(C)C1 N1(Cc2ccc(-c3cc4ccn(C)c4cc3)cn2)CCC2(CCCCC2)CC1 C(=O)(CCC(C)S(C)(=O)=O)NC(CC)CNC(=O)C=C1CCCCC1(C)C C=CCC(C(=O)NCc1nnnn1CC)NC(c1cn(C)c(C)n1)=O c1(C(=O)NCC(C)(C)C)ccc(O)cn1.C1(C(=O)N)CCCN1c1ncccn1 C1(CC)CN(C(=O)C(c2cccnc2)C)CCC1NC(c1sccc1C(F)F)=O Cc1ccc2[nH]cc(C(=O)NC3(C)CC3)c(=O)c2c1.C(=O)C(C)c1ccsc1.N c1(C(=O)NC(CC)C(C)(C)c2ccc(O)cc2)cnc(OCC(F)(F)F)c(F)c1 N1(C(CCN(C(CC)CC)C)=O)CCOCC(NC(=O)C(C)n2cncn2)C1 c1(COC)c(C(N2CC(C)(NC(=O)CC3CCCC3O)C2)=O)cnn1C N1(c2c(F)cnc(C)n2)CCCC12CCN(C(=O)COc1c(C)cccc1C)C2 N1CCC(C)C1.c1(NC(C(=O)NCCOC)=O)ccccc1OCC(C)O N1(C(C=CCN(C)CC)=O)CCCN(C(=O)C(C)(C)n2cccn2)CC1CO CC(C)C(F)(CNC(=O)CC1CSCCO1)C(=O)N(C)CC1CCCS1 c1(OC)c[nH]c2ccccc2c1=NC(C)c1cc(F)ccc1SC c1(C(=O)NC23CC(C2)C3)cncc([N+](=O)[O-])c1.C1(C(=O)N)CC12CCCC2 Cc1nc(C(=O)NC2CN(C(C3CCN(Cc4cccnc4)C3)=O)C2)cs1 N1(C(CC(c2ccc(OC)cc2)C)=O)CC(NC(c2sccc2Cl)=O)C(C)(C)C1 C(=O)C1=CC(C)(C)C1.N1(CCC)CC(C(=O)NCC2CCCCC2)CC1=O.N C12(CNC(CN(CCC)C)=O)COC(C)(C1)C2.C1CCOCC1.C(=O)CC C1(C)(CC(=O)NC(CNC(C(C)=C2CCC2)=O)(C)C)CC1(F)Cl C1(CCC(=O)N(CCCNC(=O)Cc2ncc(C)[nH]2)CC)CCOCC1 C1(CC(=O)NC(C)C=O)CCCCC1.C1(C(=O)N)CC(O)CN1C.C(C)(C)C c1(OC)ncc(Br)cc1C(c1nnnn1-c1ccccc1)NC(C)C(C)C c1(C(=O)NCC(C)NC(=O)C(C)O)csc(-c2cccs2)n1 C1(OC(C)(C)C)CC(=O)N(CC2CCCC(C(F)(F)F)O2)C1 C(=O)(NNc1ccc(F)c(Cl)c1)NC(C1CC(=O)OC1)=O.C1CC(=C2CCC2)C1 CC1=C(C(=O)NCC2CC(NC(=O)C(O)C(C)C)C(O)C2)SCCO1 c1(-c2nc(Cc3cn(C)nc3)nn2-c2cncc(Br)c2)cc2cccnn2n1 C(C)(C)(C(F)(F)F)N(C(CSCC)=O)C.c12cnc(o1)C(C)N2 C1(N(C(C2(C(C)NC(=O)CCC3CCCN3C)CC2)=O)C)CCCC(C)C1C Cc1ccc2oc(NC(C3CN(Cc4ccccc4)CC(C)O3)=O)cc2c1 c1(C(C)NC(=O)NCC(O)C(C)(C)O)ccc([N+](=O)[O-])cc1 C(=O)(NNC(=O)CSCCC1CCCC2CC12)Oc1cccc(C)c1 c1(NC(C2CC23CCN(C(=O)CC2CCSC2)C3)=O)cnc2cc[nH]c2c1 CC1CCCC(O)(C(N2CCN(C(c3cccnc3O)=O)CC(O)C2)=O)CC1 C1(C#N)(OC)CC(C(=O)NCCc2cc(C(N3CCCC3CO)=O)no2)C1 S(=O)(=O)(CCC(=O)N=S(C)(=O)c1ccc(F)c(F)c1)NCC(=O)OC C1(NC(c2cnc(CNC(C(C)C3CC3)=O)nc2)=O)C(=O)NCC1(C)C N1(C(CC(C)O)=O)CCC(NC(C2(C(F)(F)F)CC3(CCC3)C2)=O)C(CO)C1 c1(C(=O)NCC(C(C)C)NC(c2cocn2)=O)ccc(OC2CCOC2)cc1 C1(C)(CNC(C2(C#C)CCC2)=O)CCCN(C(=O)C(C(C)C)n2cnnn2)C1 c1(OCC)ccc(C(=O)NC2CC2CNC(c2ncn(C)n2)=O)cc1C C1CN(C(=O)Cn2ccc([N+](=O)[O-])n2)CCN1C(=O)C(C)CN(C)C.CO.C C(=O)(C(C)(C)C(F)(F)F)N1CC(CC=C)(NC(=O)Cn2ccnn2)C1 C1(C(N2C(CC)CCC2)=O)CC2(C1)CC1(CC1)C2.Cc1ccc(C(C)C=O)s1.N C12(c3nnc(COC)o3)CCN(C(c3c(C)nn(C)c3C(F)F)=O)CCC1C2 C1(NC(c2cc(C)n(CCO)n2)=O)C2CCCCCC12 CC1CC2(CC2)CN1C(C12CCC(NC(=O)C(O)CCN(C)C)(CC1)C2)=O N1(C(c2n(CC)ccc2)=O)CCC2(CCN(C(c3ccoc3CC(N)=O)=O)C2)C1 C(=O)(C(F)(F)C(O)C1CC1)NCC(CNC(CC(C)C1CC1)=O)(C)C N1(C(c2n(COC)ncc2)=O)CC(NC(=O)C(O)C2CCCC2)CC2(CCC2)C1 C12(CNC(CCCOC)=O)CN(C(=O)Cc3ccoc3C)C(COC)(C1)C2 c1(OC)c(C(N2CCN(C(=O)C(F)(F)Cl)C(C(C)C)C2)=O)ccc(F)c1F N1(C(CCSC(=N)N)=O)CCCC2(CC(C(=O)NC(n3ccccc3=O)C)=NO2)C1 c1(N(CC)CC)ccc([N+](=O)[O-])c(C(=O)NCC2CCCC3CC23)c1 N1(C(C2=C(C)CCC2)=O)CCN(C(=O)COCCCF)C2CCCCC2C1 N1(C(C(C)(C)OCC)=O)CCC2(CCCCC2NC(=O)CCS(C)=O)C1 CC1=C(C(=O)N2CCN(C(C3CCC3c3nc[nH]n3)=O)C(CCO)C2)CCC1 c1(C(N2CC(N(C(C(CC)C#N)=O)C)C(C)(C)C2)=O)cc2ccncc2cc1F C1(N(C(C)(C)C)C(c2cn(CC3CCC3)nn2)=O)CC2CC(O)CC(C1)C2 c1(C(=O)NC2C(NC(Cc3nc(C)[nH]n3)=O)COC2)cccc2c1CC(=O)N2C C1(NC(c2cnc(OCC)s2)=O)CC(C)N(C(=O)C(OC)OC)C1 Cc1cc(CC(=O)NC(C2CCN(C(=O)C(F)CC3CCC3)CC2)C)c(C)s1 c1(C(=O)NCC2CCCN(C(c3n(CC)cc(Cl)c3)=O)C2)cnc(O)cc1.O N1(S(C)(=O)=O)CCCCC1C(=O)NC1CC1.c1(C=O)ccccc1OCF.C c1(C(=O)NC2(C)CCN(C(=O)C3=CCCS3)CC2)ccn2ncnc2c1 C1(NC(c2onc(C)c2C)=O)CCN(C(C2CCC(C)(C)CC2)=O)CC1(C)C c1(OC)cc(C)c(C(=O)NC2CC(N(C(=O)Cc3cscn3)C)C2)cc1Cl c1(C(=O)NC(CN(C)C(c2cc(C(F)F)cs2)=O)(C)C)ccc2ccccc2n1 N1(C(C(c2c(C)cncc2)C)=O)CC2CCCC2(NC(c2n[nH]cc2F)=O)C1 CC(C)C(C)CNC(c1c[nH]ccc1=O)=O.C1(C=O)CCCN(S(C)(=O)=O)C1 N1(C(C(C)OCC=C)=O)CC(C(=O)Nc2cnc3ncnn3c2)CCC1(C)C C(=O)(C(F)(F)C1=CCOCC1)NCCN(C(=O)C(F)C1CCOC1)CC c1(OC)ccc(OC)c(CNC(=O)CC2CCCN(C(=O)CCCC(C)C)C2)c1 CN1CC2CN(C(=O)CCNC(C3(c4ccno4)CC3)=O)CC2C1 C(=O)(CCC(C)(C)C)NC(C1CCN(C(CCc2ncn(C)c2)=O)CC1)(C)C N(C1CCc2ccc(Cl)cc21)C(=O)NC(c1ccc(C)cc1C)C c1(C(=O)NC2C(NC(C3N(C)CC(F)C3)=O)COC2)ccc([N+](=O)[O-])cn1 c1(SCCOCC(c2cccc(C)n2)=O)ccc2c(c1)CCC2 N1(C(C2C(OC(C)=O)C2)=O)CC(NC(c2nn(C)c(C)c2Cl)=O)CC(F)C1 Cc1c(CC(=O)Nc2ccccc2-c2ncc[nH]2)ncn1C c1(C(=O)NC2CC(NC(C3C4CCCC34)=O)C2)cc(Cl)ccc1-n1cnnn1 Cc1cnccc1C(=O)N(CCC(C(C)C)NC(c1ccc(F)cc1)=O)C C1(NC(CC(C)n2cccc2)=O)CN(C(c2cn(C)cn2)=O)C(C)(C)C1 C12(NC(=O)C#CC3CC3)CCCN(C(=O)Cn3cc(Br)cn3)CC1C2 C(=O)(CCCC(C)(C)C)NC1(C(=O)NC(CCC)C(=O)N(C)C)CC(F)C1 C1(C(N2CCCC(CNC(c3c(C)cccn3)=O)C2)=O)CSc2ccccc2O1 c1(N2CCC(CSC)C2)nc(=NC2CC(CC(N)=O)C2)[nH]c2c1CCCCCC2 C(C(CO)C(F)(F)F)NC(C1(NC(c2ccc(CO)s2)=O)CCC1)=O C#CCCCC(=O)N1CCC(C(C)C(N2CCC(OC(C)=O)C2)=O)CC1 O=C(C1=C(Cl)CCOC1)NC1CCC1NC(C1(c2ccncc2)CC1)=O C1(C(=O)NC(CC)CNC(c2cc(Cl)c[nH]2)=O)CCc2c(n[nH]c2C)C1 c1(C(=O)NCC(=C)CCNC(=O)CC(C)F)c(CC)nn(C)c1CC c1(C(=O)NC(CCNC(C2CCC(C)C2)=O)C)ncc(C#N)cc1Cl c1(C(=O)NCC(CNC(C2C(OC)C2)=O)O)c(Cl)ccnc1C c1(C(N2CC3N(C(C(C)OCC=C)=O)C3C2)=O)cc(F)c([N+](=O)[O-])c(F)c1 CC(C)C(C)(CNC(=O)CN(C)CCO)NC(=O)CC1(C(F)F)CC1 C(=O)(CC(O)CCSC)NC1(CC=C)CCN(C(c2cnn(C(F)F)c2)=O)C1 C(=O)(C1=NOC2COCC12)N1CCC(C)(CC(=O)N)C1.c1(OCC)ccccc1 C1(NC(C(C=C)OC)=O)C=CCN(C(=O)CSc2ccc(O)cc2)C1 c1cnc2ccccn12.N1(C(c2ccc(C(F)(F)F)[nH]2)=O)CC2CC2(CN)C1.C CC1(NC(C2CC2(F)F)=O)CCN(C(C2(C)CCOC(C)C2)=O)CC1 N1(C(CCOC)=O)CCC2(COC(CNC(C3CC(F)(F)C3)=O)C2)C1 C1(NC(c2c(Cl)ccc(C)c2)=O)CN(C(=O)CCC2CC2)CC12CCC2 N1(C(C(N2CC(CCNC(C(CC)CC)=O)OCC2)=O)C)CCP(C)(=O)CC1 C1(C(N(CCCCCNC(COC(CC)C)=O)C)=O)CC2CCC1O2 C1(NC(C2(CCC)CC2)=O)CCCC(N(C)C(c2ns[nH]c2=O)=O)C1 Cc1ccc2c(CC(N3CCC(CF)(NC(=O)Cc4ccon4)C3)=O)c[nH]c2c1 C1(NC(=O)C(=Cc2cccnc2)F)CN(C(c2cncnc2)=O)CCC1F c1(CC)nc(C)ncc1C(=O)N(C)CC1CN(C(c2nncs2)=O)C1 N#Cc1cccc(CNC(C2CC(NC(c3csnn3)=O)C2)=O)c1 C(CCN(C)C)(C(=O)NCCC1CCCO1)NC(c1cnc(OC)s1)=O C1(C(C)C)CN(C(=O)CC2CC(CF)C2)CCN1C(c1ccc([N+](=O)[O-])o1)=O C(CC(C)C(=O)NCCCC(c1ccccc1)NC(=O)CO)=CC.CC(F)F c1(OC)c(Cl)cc(Br)cc1S(=O)(=O)N1CC2(CCOC2)C1 Cc1ccnn1C(C)C(=O)N(CC(C)O)CCNC(=O)COc1ccon1 C1(NC(C2N(C(CC(C)C)=O)CCCC2)=O)CN(C(=O)CC(F)(F)F)CC1(C)C Cc1ccc(C(F)(F)F)cc1CCNCC1CC1C(F)F C1(CC=C)CN(C(=O)CC2CC2C2CC2)C1.c1(C(=O)N)ccco1.C(C)=O C1(NC(N2CCCCCCCC2)=O)CCn2nnnc2C1 O([Si](C)(C)C(C)(C)C)C(C)CNC(c1cccc(OC(F)F)c1)C(F)(F)F N1(C(CCC2(NC(Cc3ccc(C)o3)=O)CCCC2)=O)CCNC(=O)C1C C(=O)(C1=CCCC(C)(C)C1)N1CCC(CNC(C2(CC)COC2)=O)C1 N1(Cc2c(CCN)ocn2)CCC2(CCOCC2)C1 Cc1c(C(N2CC3CC3(NC(c3c[nH]ccc3=N)=O)C2)=O)oc2c(Cl)cccc12 c1(COC(C)C)nc(CC2OCCCO2)n(-c2ccnc(Br)c2)n1 N1(c2nc(OC)c(C)cn2)CC2(CCC(C(=O)Nc3ccc(OC)c(Cl)n3)O2)C1 S(=O)(=O)(c1ccc(N2CCC3(CCCC3)C2)c(F)c1)NC(CCSCC)C C12(C(N3C4CC(NC(c5cccc(OC)n5)=O)C(C4)C3)=O)CC3CC1C2C3(F)F CC1OCCC1(C)C(=O)N(C1CC(CNC(=O)C=CC=C(Cl)Cl)C1)C C1(CNC(c2noc(CC)c2C)=O)CCN(C(=O)Cc2cccs2)CC1(F)F Cc1cc(C(=O)NC(C)CCC(=O)NCC2CCC=CCC2)cnc1O c1(CC)c(C(=O)NCC2(C(N3CC(CCO)C3)=O)CC(C)(C)C2)ccn1C C1(C(=O)NCC2(C)CC3(CC3)C2)CCCCN(C(C2CCCOCC2)=O)C1 N1(c2ncc(C(=O)OC)cn2)CCC(NC(C2CC2(F)F)=O)C(CO)CC1 C#Cc1cccc(C(=O)NC)c1.c1(CCC=O)ccc(N)c(F)c1.C1(O)CCC1 O=S(=O)(c1ccc(C(F)F)o1)N(C(c1ncc[nH]1)CO)Cc1ccco1 n1(CC(=O)NCC(CNC(C2CCCCCC2)=O)OC)cc(F)ccc1=O N1(C(c2n(C)cnc2)=O)CCCC1C1CCCCN1C(=O)Cc1csc(Cl)n1 C=CC1(C(=O)NC2CC3CC2N(C(C2CC(O)C2)=O)C3)CCCCC1 Cn1ccc(C(N2CC(C)(F)CC2C(=O)NCC2CC23CC3(F)F)=O)cc1=O C1(C(N(C2CC3CCC2CC3)C)=O)CC12CCN(CCC1CC1)CC2 C(CNC(=O)CCC1CC1(F)F)(CCNC(C1(C)CSC1)=O)OC N1(C(CCC=C)=O)CC(C2CCN(C(=O)CN3CCCC3)CC2)C1 c1(OC)cc(OC(=O)Cc2cccc(N(C)C)c2)ccc1[N+](=O)[O-] C1(NC(CCNc2cccc(OC)c2)=O)COC2(C1)CN(C(=O)C(C)O)C2 c1(C(=O)NC(CN(C(=O)CC2CCCO2)CC)C)ccc2c(c1)COCC2 N1(C(C(C=C)(C)C)=O)CC2(C)CN(C(=O)C(O)C=CCCC)CC2(C)C1 C1(C(N(C2CCCC2)CC(=O)OC)=O)(NC(=O)CCN(C)C)CCC1 N1(C(C2C=C(C)CS2)=O)C2COCC1CC(NC(=O)Cn1cccnc1=O)C2 C1(C=O)CCC2(CCC2)C1.c1(C(=O)NC)ccc(C(F)F)c(Cl)c1.C1CC1 CCCCC(CC)N=c1[nH]c2c(c(=NCCOCCOC)[nH]1)COC2 C1(CC(=O)NCCC(C)NC(C23CCC(CC2)CC3)=O)CCC(C)(O)CC1 CN1CC(NC(C2CCCCCN2C(c2nocc2Cl)=O)=O)C2(CC2)C1 c1(OC)ccc(CC(=O)NC2(C3CCCCN3C(=O)C=C(C)Cl)CC2)cc1F C1(NC(C(C)OCC(F)(F)F)=O)CCN(C(=O)C(F)(F)c2cccnc2)C12CC2 c1(CNC(C2C(C)CC2)=O)ccccc1CNC(c1cnc[nH]1)=O N1(C(C2CCN(C)CC2)=O)CCC2(CCCC2C(=O)Nc2nc3c(s2)CCC3)C1 Cc1nc2nccc(N3CCN(C)C(CNC(=O)CS(N)(=O)=O)C3)n2n1 c1(C(CN2CCC(C(C)C(=O)NC(=O)CC(C)(C)C)CC2)=O)csc2nccnc12 C1(C)(C(N(C2CN(CC3CC(=O)N(C)C(=O)N3)C2)C)=O)CCCCC1(F)F c1(C(N(CCCNC(C2CN(C3CCOC3)C2)=O)C)=O)ccc2ncncc2c1 C1(CC)CCN(C(c2c[nH]c(=NC)o2)=O)C1C(=O)NCC(Cl)C(C)(F)F C(c1cncnc1O)=CC(N1C(C)CC(NC(c2cc(Br)n[nH]2)=O)C1)=O c1(CC(N2C(CC=O)COCC2)=O)ccc(O)cc1Cl.C1(C(=O)O)CC1.CC c1(C(C2CCCCC2)N(CC(c2nn[nH]n2)C)C)cc(Br)cnc1F Cc1nc(C(C)C)ccc1C(=O)NCCNC(C1(Cl)CC12CCC2)=O N1(C(C2CCCN(CCC)C2)=O)CCC2C(CCN2C(c2n[nH]c(C)n2)=O)C1 C1(NC(C(c2ccc(CC)cc2)(C)C)=O)CCCN(C(=O)C=C(C)C)CC1 CC1CCS(=O)(=O)CCN1C(C(=O)NCC1CCOC1)C1CC1 C12CCC1CN(C(C1CCC(C(N)=O)C1)=O)C2.c1(CC)nc(C)c(C(=O)N)s1 N1(Cc2cc(C)c(F)nc2)CCC=C(C(=O)Nc2nc(Cl)ccc2F)C1 Cc1ccn(CC(=O)NCC2(C(=O)NC(c3ccsc3)C)CC=CC2)c1 c1(C(=O)NCCN(C(CC2CC(=C)C2)=O)CCOCCO)ccc(Cl)o1 c1(N(C(C)=O)C(c2nn[nH]n2)C2CCOC2)ccc2c(c1)nc(O)n2CC(C)C Cc1cc(Cl)cc(Cl)c1OCC(=O)NC1CN(C(=O)Cc2ccoc2C)CC1C N1(C(c2c(C)ccs2)=O)CCN(C(=O)CCc2ccncn2)CC2CCCCC12 C1(C(=O)OCC)(C(=O)NC(C)C(c2ccc(C)cc2)OC)CCC(O)C1 C1(CC)CN(C(=O)C(C)O)CCC1NC(=O)Cn1cnnc1O C1(CNC(c2c(C)cncc2C)=O)CN(C(=O)C2=CCCOC2)CC(C)(C)C1 c1(C(c2n(C(CC)C)nnn2)NCCOCCF)ccc(Br)cc1OC Cc1cn(C(c2ccccc2)C)[nH]c1=NC(=O)Nc1ncc(Cl)c(I)c1F C1(C(=O)Nc2ccnc(F)c2)CC12CCN(Cc1cc(Br)co1)C2 c1(OC)ccnc(F)c1C(N1CCCC1c1cn(CC(F)(F)F)nc1C)=O c1(CCC(N2CC(N3CCOCC3)(CC)C2)=O)ccc2cccnc2c1 N1(C(C=NOC)=O)CC2CN(C(C34C5CC(CC35)C4(F)F)=O)C(CO)C2C1 C(=O)(C(C(C)(C)C)NC(=O)CCOC1COC1)N1C(C#C)CC1 N1(C(c2n(C(C)C)ncc2)=O)CCCC(F)(CNC(C2CCCC2C2CC2)=O)C1 C1(CC(=O)NC(C)CCCNC(C2CCCOC2)=O)CCC(=O)N1C C(C(C)(C(=O)N1CCC(NC(=O)CC(C)(C)OC)C1)OC)OC CC(C)C(C(=O)NC1(C)CC(O)C1)NC(C1COCC1C(N)=O)=O C(=O)(CCCCCC=C)NC1CC(NC(c2ccc(CCC=C)cc2)=O)CC1O CC(C)(C)CCC(=O)NCCCN(C(=O)CC1CCC(F)(F)CO1)C1CC1 C12(C(=O)NCCC=C)CCC(NC(c3cc(Br)cc(Cl)c3F)=O)(CC1)CC2 C(=O)(CC1=NN(C)C(=O)C1)N(C1CN(C(c2c(C)n(C3CC3)nc2)=O)C1)C C(N=c1nc(N2CC3C(C(=O)NC)C3C2)c2c([nH]1)CSC2)c1ncc(OC)nc1 CC(C)C(C(C)NC(c1ccc(C(N)=O)nc1)=O)NC(=O)CCN1CCCC1 C(C(C)(C(=O)N)OC)OC.C1CN(C(C2(C)COC2)=O)CC1c1ccccc1.C N1(C(C)=O)CCCC12CCCN(C(=O)C(c1ccc(Cl)cc1F)F)C2 C1(C)(NC(C2(C(C)C)N(C(CCCSC)=O)CCC2)=O)CCCCC1(C)C c1(C(=O)NC(C2CCOC2)C)cnc(CNC(=O)Cn2cccn2)nc1 CC(C)C(CC(=O)N(C)Cc1ccns1)NC(=O)CC1CC2CCC1O2 C1(CN(C(CSC)=O)C)CN(C(c2ccc(C(F)F)s2)=O)CCO1 c1(OC2CCN(CC#N)C2)ccc(F)cc1F.c1(C(C)C)cccc(C(C)(CO)N)c1 N1(C(CN(C2CC2)CC)=O)C2CCC1CCC2.C1(O)(C(=O)N)CC(C)(C)C1 Cc1cc(C(=O)NC2CCN(C(c3cnn(CCN(C)C)c3C)=O)C2)oc1C c1(-c2cccc(C)c2)nc(=NC2CC(NC(c3ccnn3C)=O)C2(C)C)s[nH]1 N1(C(=O)NCc2n(CC)nc(Br)c2)CC(C)(C(=O)O)C(F)(F)C1 N1(CC(=O)N(C(CCNC(CSCCC(C)C)=O)C)C)CCC(=O)NC1=O Cc1ncncc1C(N1CC(F)CC1CC(=O)NCCn1cnnc1)=O C(CS(=O)c1ccccc1)NCc1ccc(SCC)nc1 C(CCCC)NC(C=CCOC)=O.C1(C=O)CC1(F)F.C(C)(C)C.C=O C1(NC(C2CCCN(C(=O)CCn3cccc3)C2)=O)CC2C(C1)C2(F)F c1(OC)ccnc(CC(=O)N(CCC(C(C)C)NC(C2CC(C)CO2)=O)C)n1 N1(C(c2cc(C)nc(O)c2)=O)CCCC(C2(NC(=O)CC(C)P(C)(C)=O)CC2)C1 N1(C(C=CC(=O)OCC)=O)CCCC12CCOCC2.c1(CC(=O)N)cnoc1 C(=O)(C(C)(C)CCCNC(C1OCCC1(C)C)=O)N(C)C[Si](C)(C)C C(=O)(C#CC1CCCO1)N1CCN(C(C(C)(C)N2CCCC2)=O)CC1C(F)F CN1CCN(C(=O)OCc2nc(CO)n[nH]2)C(C(=O)NC(C)(C)C)C1 C(=O)(C(C)(C)C(=O)NCc1cc(C(=O)NC2CC2)cs1)OCC.C Cc1c(C(N2CCC(CC(=O)NCc3ccccc3)C2)=O)ncn1C c1(C(N(CCNC(=O)Cc2nonc2C)CC)=O)ccc2snnc2c1 C1(NC(=O)C=Cc2ccc(F)nc2)CCC2CCN(c3cc(Cl)ncn3)C1C2 c1(N2CCC(SC)CC2)ncc(C)cc1S(=O)(=O)NCCC(C(C)(C)C)C1CC1 c1(CN2CCCC(C(=O)Nc3occ(C)n3)C2)ccc(F)c(C)c1Cl N1(C(CC(C)OC)=O)CCCC2C1CCN2C(c1ncnc2c1ccn2C)=O C(CC(C)C(=O)NCC12CC1CN(C(=O)C(C1CCOCC1)OC)C2)OC C1(C(=O)Nc2ccc(C(CN3CCN(C)CC3)=O)cc2)OCCNCC1(C)C c1(-c2ccc(CCC)cc2)cnc(O)c(CNC(C2(c3ccsc3)CC2)=O)c1 c1(-n2ncc(-c3c(N4CCC(O)C4)ccc(OC)c3)c2)ccc2c(c1)CC(C)O2 C1(CCNC(C(CC)OC)=O)CCCCN1C(C1CSC1)=O c1(C(=O)NC(C2CN(C(=O)CN(C)CCO)C2)C)ncc2n1CCCC2 C1(C(N2CCCCC2)=O)CC2(CCCO2)C1.Cn1nc(C2CC2)cc1C(=O)NC O=S(=O)(c1cnccc1NC1CC1c1c(F)cccc1F)NC1CCCC(F)(F)C1 c1(C(=O)Nc2ncc(N(C)C)nc2)cccc2nc(Cc3nccn3C)cn12 c1(C(N(C2CCN(C(c3cscc3C#N)=O)C2)CCC)=O)cc(C)ccn1 c1(C(N2C(CCNC(C=C(C)C)=O)CSCC2)=O)ccc2c(c1)CC(C)O2 N1(C(CC(C)(C)O)=O)CCN(Cc2ncco2)CC1CC#N C1(NC(c2cc(F)c[nH]2)=O)CCCC2CN(c3nncs3)CC12 c1(C(=O)NC(C2CCN(C(C(C)N(C)C)=O)CC2)C)cc(F)c(Br)cc1N C=CC(CC)CC(=O)N1CCC12CN(C(=O)CCC(=O)N(C)C(C)C)C2 Cc1ccc(I)c(NC(C2C=CCN2C(=O)C(C)O)=O)c1 c1(C(=O)NC2C(NC(c3cnc(OC)s3)=O)CCCC2)c(C)cccc1C CCCCC(O)CC(=O)N1CCCCC(NC(c2cc(C)cc(Cl)c2)=O)C1 Cc1sc(Cl)c(C(=O)NCC2(O)CCN(C(=O)CC#N)C2)c1C Nc1nc2c(cc1C(N1CC3C(NC(=O)CO)C3C1)=O)CCCC2.C1CC=CC1 C1(C)(CC)CCC(C(=O)NCC2CN(C(=O)C(C)CO)CCO2)O1 c1(C(=O)NC2CCCC(NC(CCCCC#C)=O)CC2)cc2c(s1)CN(C)CC2 CC1CN(C(=O)CCc2cc(Cl)no2)CCN1C(c1cnc(C(C)(C)C)[nH]1)=O Cc1ccc(CC(=O)NC2CC2NC(=O)C(C)C#N)c(F)c1F CC(C)(O)CC(=O)NC(C1CCCCC1)CNC(=O)C=Cc1nc[nH]n1 Cc1cc(O)ncc1C(=O)NC(C1CN(C(C2(N(C)C)CCCCC2)=O)C1)C N1(C(CC2CCN(C(=O)OC(C)(C)C)C2)=O)CC=C(CO)CC1 N#Cc1ncc(F)cc1NC(C12CC1CN(Cc1ccc(Cl)c(F)c1)C2)=O Cc1ncc(Cl)c(C(=O)NCC(CC(F)(F)F)NC(C2(C)CNC(=O)C2)=O)n1 N1(C(CS(CCOC)(=O)=O)=O)CCC(C2CCCN(C(C3(F)CCC3)=O)C2)CC1 C1(NC(CC2(C)CN(Cc3ncc(OC)s3)C2)=O)CCc2ccccc2O1 N1(C(C2(OC)CCCC2)=O)CC(CO)C2(C1)CN(C(C13CCCC(CO1)C3)=O)C2 n1(C(C)C)cnc2c(N3CCC(CCO)CC3)[nH]c(=NCC(C)CN(C)C)nc12 Cn1c(NC2CCCC23CCN(C(=O)C=CC2CC2)C3)cc(=O)n(C)c1=O Cc1c(C#N)c(CCNC(=O)CNC(=O)C2=CCOC2)n(-c2ccccc2)c1C C(=O)(CCCCCCC(=O)OC)N1C2CC(NC(C(CC=C)C)=O)(C2)C1 C(=O)(C(CCN(C)C)NC(c1ccc(C#N)o1)=O)NCc1c(C)nsc1 C1(C)(C(=O)NC2CCN(C(CC(CC)SC)=O)C2)CCC(C(=O)N(C)C)C1(C)C CC(CC1CCCO1)C(=O)NCC1CN(C(=O)CCc2cccn2C)C1 Cc1ccc(=N)[nH]c1C(N1CC(O)(CC)C1)=O.n1(CC=O)c(C)c(C)sc1=O C(=O)(C1=CC2CCCCCC12)N1C(C)CCC(NC(c2n(CC)ccc2)=O)C1 N1(C(c2c(C)ccc(OC)n2)=O)CCN(C(=O)C(C)C(C)(F)F)CCC1C N1(C(=O)OC(C)(C)C)CCC2(CCCCN2C(=O)C(O)C(F)F)C1 C(=O)(CC(C)(C)CC(F)F)N(CC(C)N(C)C(C12CC(C)(C1)OC2(C)C)=O)C Cc1cc(C)c(C(=O)NCC2CC3CC(C2)N(C(c2nocc2C)=O)C3)cc1C C1(CC(=O)N(CC(C(C)C)O)CC(C)C)CCCC(C)(C)CC1 C1(NC(C(C(CC)C)N(C)C)=O)CCN(C(c2coc(C(C)C)n2)=O)CC(O)C1 c1(CNC(C(CC)n2cncn2)=O)nc2c(s1)CCN(C(C1(SC)CCC1)=O)C2 N1(C(c2cc(C3CC3)ccn2)C(=O)NC(C)C)CCCC2CC(C)CCC12 C1(NC(C2C(C)(C)C2)=O)CCCCCC1C(N1CC(F)(C#N)C1)=O c1(C(=O)NCC2(O)CN(C(C(C)OC3CCCCC3)=O)C2)cccc(O)c1F N1(C(c2c(C)cccn2)=O)CC(NC(c2ncccc2OC(F)F)=O)C2(CC2)C1 C1(NC(C(c2ccccc2)NC(CC)=O)=O)CC12CC(O)C2 CC(CO)(C(=O)NCCCn1cccn1)NC(c1ccc[nH]1)=O N1(C(c2n(CC)ncn2)=O)CCOCC12COCCN(C(=O)C(C)N1CCC1)C2 c1(C(N2CC3C(CNC(CC4(C#N)CC4)=O)(C3)C2)=O)nnn2c1CCCC2 CCC(CCC(=O)NCCS(C)(=N)=O)NC(=O)CNC(=O)OC c1(C(=O)NC2CN(C(=O)COCC3CCOC3)C2)cnccc1Cl N1(C(c2c(CC)nco2)=O)CC=C(CC(=O)NC[Si](C)(C)C)CC1 c1(NC(=O)NCC)cccc(CNC(=O)C=O)c1.C(=O)C(C)NC=O N1(CC(=O)N(C)CC2CCCN(C(c3c(C)[nH]nc3)=O)C2)Cc2ccccc2C1 c1(NC(=O)Nc2c(OCCC)cccc2)nc2cccc(Br)c2o1 C1(C(N(CCC)CCO)=O)CCN(C(C2CC(C)(C)CO2)=O)CCO1 C(C#Cc1cnn(C)c1)NC(=NCC)NCc1cnn2c1CCC2.C1CCCCC1 N1CCN(C(=O)C(O)c2ccsc2)CC1.c1(OC)csc(C(=O)NC2CC2)c1.C CC(C)(CNC(=O)C=CC1(C)COC1)CC(=O)NCC1CC1 C1(CN(C(=O)C(C)(C)n2cccn2)C)CCCN(C(c2ccn(CCF)n2)=O)C1 O=C(C#CC1CCCO1)NCC12CC(C1)C2.C1(CC=O)CC(=O)NC(=O)C1 C1(C)(C(=O)NC(c2cccnc2O)C)CCN(C(=O)CC(C)O)CC1 C1(NC(c2[nH]cc(CC)n2)=O)CCN(C(C2(F)CCOC2)=O)CC12CCC2 N1(C(CNC(c2ccccc2)=O)=O)CCC2C(CCN2Cc2cncc(F)c2)C1 c1(CC)cc(C(N2CC(NC(=O)Cc3csc(Cl)c3)CCC2C)=O)cc(O)n1 C(=O)(C(CN=[N+]=[N-])NC(=O)CCC1CCC(=O)C1)NCC(C)(C)N(C)C c1(C(C(N2CCC(CNC(C(C)OC3COC3)=O)C2)=O)(C)F)ccc(F)cc1 c1(C(=O)NC(C)CNC(=O)CCc2cc[nH]n2)nc(Br)n2ccccc12 N1(C(C2C(OC)(OC)CC2)=O)CCC(CO)C1C.c1(C(=O)N)cnc(C)[nH]1 c1(C(C)=O)ccc(C(=O)NCCCc2ccccc2)[nH]1.C(=O)(CC(C)N(C)C)N C12CCN(CC1)C1CCN2C1.C1(CO)C=CCN(c2nnnn2C2CCOC2)C1 N1(C(C(COC)OC)=O)CC2CC(C(=O)NOCC(=O)OC)(C2)C1 c1(N(CCCNC(C(C=C)O)=O)C2CC2)ncnc(Cl)c1CO N1(C(C(=O)NCC)=O)CC2(CCCC2NC(c2cnc(SC)s2)=O)C1 C1(NC(c2ccc3occc3c2)=O)CCC2CC1CN2C(=O)CN1CC2CC2C1 CCC(C)CCC(=O)NC1(C(=O)N(CCC(O)CO)C)CC1(C)C C1(NC(COCCOC)=O)C2CC1N(C(=O)CN1CCC(C)(O)C1)C2C CC(=O)CCCC(C)C(=O)NC1CN(C(c2cocn2)=O)CC1C1CC1 N1(C(c2nccs2)=O)CCN(C(=O)C(=O)NC(C)Cc2ccccn2)CC1 C(=O)(CC(C)C(C)(C)CC)N(CCCNC(=O)C(O)CCC(C)C)CC C1(NC(N(CC(C)C)CCC#N)=O)CCN(C2CCCCC2)C1 C1(S(N)(=O)=O)(C=O)CCCC1.c1(COC)cccc(C(=O)N)c1.C1CCC1 C1NC(=O)CC1(C)C.C(=O)(C(C(=O)NCC1OCCC1C=O)OC)OC.N Cc1nnc2n1CC(C(=O)NCC1COCCN(c3cc(Cl)c(O)nn3)C1)CC2 c1(CNC2CCC(C(=O)Nc3cc(C)nn3C3CC3)C2)cccc2ncccc12 C=CC(C)(CC)C(=O)OCC1(c2c(F)cccc2F)CCC1 CCCCCC(C(=O)N1CCC(NC(c2c(C)nsc2N)=O)C(C)(C)C1)C(C)C c1(C(C)(C)SC)nc(CC(N2CCOCC2)=O)nn1-c1ccc(Cl)cc1 Cc1cnc(C(=O)NC2CCOC(C(N3CCCC34CC4)=O)C2)cc1C CC1CC(NC(C2CCC(O)CC2)=O)CN1C(c1cc(CF)on1)=O C(=O)(CCC(C)(C)C)NC(C1(O)CCN(C(c2ccncc2F)=O)C1)C c1(C(N2CCC(CCC(=O)N(C3C(OC)COC3)C)C2)=O)ncc2ccccn12 C(CCC(C(=O)NCc1cn(C)nc1C)NC(=O)CCc1ccc[nH]1)OC N1(C(C2(C)CC2(Cl)Cl)=O)CCC2(CC1)CN(C(=O)Cc1cnco1)CCO2 C(=O)(N=c1cc[nH]c(C)c1C)c1n(C)cc(NC(c2c(OC)cc(Cl)cc2)=O)n1 Cc1nccc(C(=O)NCC2CN(C(=O)C(=O)NCC(F)F)CCO2)c1O c1(OC)nc(Cl)ccc1CN1CC(O)CC1C(=O)NCc1nn[nH]n1 C1(N(C)C)CCCN(C(C2CC(C)(C)CN2C(c2csc(=N)[nH]2)=O)=O)CC1 CC1CCC(C(=O)N(C(c2ccccc2)CNC(=O)CN2CCOCC2)C)O1 N1(C(c2nc(CC)[nH]n2)=O)C(CNC(c2ncsc2C)=O)CC2COCC12 c1(CC)cccc(C(=O)NC2CCCC(NC(c3cc(CCO)on3)=O)C2)c1O c1(CNC(N2CCCCC(NC)C2)=O)ccc2c(c1)CCCN2C C1(NC(CNC(=O)NC)=O)C2CC3CN(C(=O)C#CC(C)(C)C)C1C3C2 O=C1CC2OCCC2(C(=O)NC2COCC2CNC(C2(F)CC2)=O)CN1 C(c1ccccc1F)=CC(=O)NC12CN(C(C(C=C)O)=O)C(C1)C2 c1(CNC(C)=O)cn(CC(=O)NCCCNC(c2ccccc2)=O)nn1 C1(C(=O)NOCC(=C)C)(CC=C)CCCN1C(=O)C(C)CC=CCC N1(C(C2N(CC)CCOC2)=O)CC2CC(NC(c3c[nH]cc(C)c3=O)=O)CC1C2 N1(C(C2(CC)CCOC2)=O)C2CCC1(CNC(=O)C(C(C)C)SC)CC2 CC1=NNC(=O)C1CC(N1CCC1(C)CC(=O)NCc1ccc(F)cn1)=O C1(CNC(C(C(CC)O)C)=O)CCN(C(=O)C=CC(C)=O)CCC1(F)F c1(C(=O)NC(C(=O)NCCCC(=C)Br)CC)ccccc1C CC(C)CC(=O)NCC=CC.C1(O)(CC=O)CCC1.C(C)(C)C.C=O C1(C(=O)NC(c2ccc(C)s2)C)CSCCN1C(=O)C=CC1CCCN1C N1(C(CCCC#C)=O)CCC2(CNC(C3C4CNC(=O)C34)=O)CCCC12 Cc1cc(NC(=O)CS)ccc1.c1nncn1C.C(=O)C(F)(F)C12CC(C1)C2 C1(C(N(CCN(C(c2c[nH]nc2O)=O)CC)CC)=O)CCC2(CCC2)C1 C(=O)(C#CC(C)(C)C)NCC1(C)N(C(C2CCC(C(=O)OC)CC2)=O)CCC1 N1(C(C=CC)=O)CC2C=CC1C(C(=O)N(CC(F)(F)Cl)C)C2 N=c1nc2c(c[nH]1)CC(C(=O)NC(C)CC(F)(F)F)CC2.c1(C(=O)N)cscn1 N1(C(C(C)OCC(C)C)=O)CCCC(C)C1.c1(C=O)nocc1C(C)(C)C.N CC(C)CC(CNC(=O)CNS(C)(=O)=O)NC(=O)CO.C1CCC1 N1(C(c2n(C)ncc2Cl)=O)CC2(C)CC1CO2.C1(C(=O)N)CC(F)(F)C1(C)C C1(C(N2CCC2CC)=O)(NC(c2c(CC)c[nH]n2)=O)CCC(C)(C)C1 C(CSC)(C(=O)NCC#CCCO)NC(C(C)SC(C)C)=O c1(OCC)ccc2oc(N(c3nc(SC)ncc3C#N)C34CC(N)(C3)C4)cc2c1 C(=O)(C#CC1CCCC1)NC1CC(N(C)C(c2csc(C3CCCCC3)n2)=O)C1 Cc1cnn(C)c1CC(=O)NC1(CF)CN(C(C2CC23CCOC3)=O)C1 c1(C(N(C2CCN(C(CCOCC)=O)C2)C)=O)ccc(C#N)c(C(F)(F)F)c1 Cc1oc(S(N)(=O)=O)cc1C=O.c1(C(N(C2CCCC2)C)=O)cnc(O)n1C.N C1(C2CCOCC2)(C(N2CCC(NC(CCSC)=O)(CF)C2)=O)CC1 C(C)(CCCC(=O)NCC(O)C(=O)OC)NC(C1(CC=C)CCOC1)=O c1(C(=O)NCCN(C(=O)C(C)(C)C2CCOCC2)C)cc2ccccc2oc1=O c1(C=O)cc(=O)c2ccncc2o1.N1(C(COC(C)(C)C)=O)CC2CC2(C)C1.N c12cc3c(s1)CN(CC3)C2.c1(SC)cccc(C(=O)N(C2CCCC(C)C2)C)c1 N1(C(C=CC(C)(C)NC(C=CC)=O)=O)CCC(C)(C)CC1.COC=O c1(C(N2CCC(CNC(C(CC)OC)=O)(OC)C2)=O)c(C)ccc(Cl)c1O N1(C(C(CNC(C2(C(C)C)CC2)=O)CC2CC2)=O)CCOC(C2(C)N=N2)C1 CCC(O)C(F)(F)C(=O)NCC(C)NC(c1cc(Cl)cc(C(F)(F)F)n1)=O C1(C(N2CC3(COC(CNC(C4(CF)CC4)=O)C3)C2)=O)CCCC2CCCN12 c1(C(N2CC(CC(C)NC(CC3ON=C(C)C3)=O)C2)=O)cncc(OC)n1 S(=O)(=O)(c1cccnc1NC1CCCCC1O)NC(C)C(C)(C)C N1(C(CN2CC(C)C2)=O)CC2CCN(C(=O)CCc3ccc(OC(F)F)cc3)C2C1 c1(N(C)Cc2nnc(O)o2)nc(N2CCC(N3CC=CC3)CC2)nc2scnc12 C1(CC=O)CCCS(=O)(=O)C1.Cc1cccc(COCC(=O)N)c1.C1CC1 c1(C=O)c(C)c(C)nn(C)c1=O.N1(C(C2C(CC)C2)=O)CCCC(O)(C)CC1 N1(CCN(C)C(C2CCCC2)=O)CCC2CCC(C1)N2C(=O)C.C(C)(C)C.O CC1(C)CCC=C1C(=O)NC(CNC(C1(C)CC=CCC1)=O)CC(F)(F)F c1(C(N2CC(NC(Cc3ccn(CC)n3)=O)C(C)C2)=O)cncc(S(N)(=O)=O)c1 c1(C(N2CCC(C)(CNC(=O)CNC=O)CC2)=O)ccc(F)c(F)c1N CC(C)CC(CN=c1ncc(O)c[nH]1)NC(=O)CC(C(F)F)n1ccnc1 CN1CC(C(=O)NC2CCN(C(C3COC(=O)N3)=O)CC2)CCC1=O C(=O)(CCCCCCCCCO)N1CC(CNC(C(C(C)(C)O)F)=O)C(O)C1 c1(CCC)c(C(=O)NCC(C(C)C)NC(=O)C(C)CO)cnn1C C1(C)(NC(c2c(C)ncnc2)=O)CCN(C(=O)C(C(C)C)n2ncc(N)n2)CC1 N1(Cc2c(C)nc[nH]2)CCN(CC(=O)Nc2cc(F)c(Cl)cn2)C(=O)C1 C(C)(CNC(c1cnn(C(F)(F)F)c1)=O)(C(C)C)NC(C1C(C)=C1)=O N1(C(Cc2c(C)nn(C)c2C)=O)CCCC12CCN(C(c1cc(C)n(C)n1)=O)C2 C1(C(=O)NC2(CC)CCOC2)COCCN1C(=O)CCC1CCC1 c1(C(N2CCOCC2C(N2CCCC2c2nn[nH]n2)=O)=O)cc(O)c(O)c(O)c1 N1(C(=O)Cc2csc3ccc(O)cc23)CCOc2c(Cl)cccc2C1 N1(C(CC2CCN(C(C)C(=O)NC3CCCC3)C2)=O)CC2CC(=O)NC2C1 C1(C)(CC(=O)NCC(NOCC)=O)CCN(C(=O)C(C)N(C)C)C1 Cc1cc(Cl)cnc1CNCCOC1(C)CCOCC1 C=Cc1cnn(C)c1C(=O)NC(C)CNC(c1ccc(C(C)CC)cc1)=O C1(CC=C)(NC(=O)CCC2CC2)CCN(C(=O)C=C)C1.n1(CS)cncn1 C(C)(CNC(C1(C)CC1C)=O)(C(C)C)NC(c1nc(C)oc1)=O c1nocc1C(=O)N(CC(C1CCCC1)O)C.C(C(=O)N)(OCC)OCC c1(C(=O)NCC2CC(NC(C(COC)(C)O)=O)C2)cc2ccnc(Cl)c2[nH]1 c1(C(=O)NCC2N(C)CCN(C(CS(CC)=O)=O)C2)nc2c(cc1Cl)OCCO2 C1(NC(CC(C)SC)=O)CC(NC(c2nnn(C)n2)=O)CC1O N1(C(c2cnc3ccccc3c2)=O)CCC2C(CCCN2c2cnc(F)cn2)C1 CC(CS(C)(=O)=O)C(=O)N1CCN(C(=O)Nc2ccc(S(C)(=O)=O)[nH]2)CC1C C#CCCCCCCCC(=O)NC1CCC(CNC(=O)C#CC2CCOCC2)C1 N1(C(c2cc(CC)nn2C)=O)CCC2C(NC(c3ncc(F)cc3F)=O)C2CC1 c1(C(=O)NCCCCNC(C2(CSC)CC2)=O)cnc(C#N)s1 C(=O)(CC(C)P(C)(C)=O)NCC(CCNC(CCCC(=C)C)=O)OC C1(NC(c2[nH]cc(C(C)=O)c2)=O)CCCC2CN(C(=O)Cc3nccs3)CC12 c1(C(=O)NC2CC(n3cc(CCCC(C)O)nn3)C2)cccc(C(=O)O)c1 Cc1cc(C)c(C(=O)NCCC(O)CNC(=O)C(C)S(N)(=O)=O)cc1N N1(C(C2(CC)CCCC2O)=O)CCC2(CC2C(=O)NC(C2CCC2)C)C1 N1(C(=O)Cc2cncnc2)CCC2(CCCC2Nc2ccccc2[N+](=O)[O-])CC1 N1(C(CCC(C)=O)=O)CCCC(C(=O)NCCN2CCC3CC23)(C(C)C)C1 C(=O)(C1=CC2C=CC(C1)C2)NCC(N1CCN(C(C(CN(C)C)O)=O)CC1)=O N1(C(CSCC(N)=O)=O)CC2CC(NC(=O)C)C2C1.N1(C(C)C)CCCC1.O c1(C(=O)NC2C3CN(C(c4c(C(C)C)nns4)=O)CC32)cncc2c1CCCC2 N1(C(CCCCOCCC=C)=O)CC2CC(NC(=O)CN3CCC(C)C3)C1C2 c1(C(N2CCCC(CN(C(C3C(C)C3)=O)C)C2)=O)nc(C2CC2)ncc1Cl C12(CNC(c3c(C)c[nH]n3)=O)CCCC1N(C(c1ccnc(F)c1Cl)=O)CCC2 C1(C(N(C2(C#C)CC2)C)=O)CCN(C(c2csc(C)n2)=O)C1C(C)C Cc1cc(C)c(C(N2CC(N(C(=O)COC3(C)CCCC3)C)C(O)C2)=O)[nH]1 C1(NC(c2c(CC)csc2)=O)CC2(CCCN(C(=O)Cc3cn(C)nn3)C2)C1 C1(C(=O)NC(C2(CNC(=O)C(C)(C)F)CC2)C)CCC(C(N)=O)O1 N1(CCNC(c2n(C)cc(Cl)c2)=O)CCCN(C(C23CCC2C3)=O)CC1 N1(C(CC)=O)CCC(CNC(c2coc(C)n2)=O)C1.C1(C=O)CCCSC1 N#Cc1ccc(N2CCN(CC(=O)NCCC3CCCNC3)CC2)cn1 N1(C(C(C(CCC)NC(=O)C2=C(Cl)CCCC2)O)=O)CC2CCCC(C1)N2C C(CCC(O)C(=O)N1CCC12CC(O)C2)NC(c1cncc(C)n1)=O N1(C(CCCC(C)C)=O)CC(C)N(C(=O)CCOc2ccc(Cl)c(F)c2)CC1C c1(SC)nc(N2CCC(=CCNC(c3[nH]nnc3C)=O)CC2)cc(C)n1 C12(NC(C3C(=O)NCCC3)=O)CCCC1CN(C(c1c(F)cc(F)cc1Cl)=O)C2 C1(CN(C(C=CC)=O)C)CCCC(NC(=O)CC2CC3(CC3)C2)C1 C(CC(=O)N(C1(C)CC1)C)(C(C)(C)C)NC(C(CC)CCOC)=O C=C1CC2(C1)CC(C(=O)N)C2.c1(C=O)cc(C(N)=O)c[nH]1.CC(C)C1CC1 c1(C(=O)NC2CCCN(C(c3n(C)nc(C4CC4)c3)=O)C2)c(F)cccc1Br C1(C)(c2n(CCCSC)ncc2C)CCCN(C(=O)OC(C)(C)C)CC1 N1(C(CSCCN(C)C)=O)CCN(C2CCCN(C(=O)Cc3ccco3)C2)CC1 C1(C(=O)NC2(CCCC)CC2)CC12CCN(C(=O)C(C)S(N)(=O)=O)CC2 C12(CC(N3CCC3)=O)CCC1CN(C(C1CN(C(C)C)C1)=O)C2.CC(C)C.O C12(c3cn(C(C)CNC(=O)Cn4cnnc4)nn3)CC3CC(CC(C3)C1)C2 N1(C(=O)Cn2cccn2)CCOC2CN(Cc3cc(F)cc([N+](=O)[O-])c3)CC12 C1(C(=O)NCC(C)SC)CC(C)(C)CCN1C(c1cccc(C)c1C)=O S(=O)(=O)(c1ncc(Cl)cc1C)NC1(C(=O)OC)CC(OC)(OC)C1 C(=O)(CN=c1cc[nH]cc1)NC1(C(=O)NCCC2CCC(=O)N2)CC1 N1(C(Cc2c(C)cccc2)=O)CC2CCN(C(=O)C(C)n3ccnn3)CC(C2)C1 C(=O)(CC(C)(C)CCC)NC1CCC(C#C)CC1 C1(NC(=O)Cc2cnc[nH]2)CCN(C(=O)Cc2ccc(Cl)cn2)C12CCC2 N1(C(C=CSC)=O)CC2(CCNC(=O)Cc3[nH]cnc3C)CCC1C2 N1(C(C2CCN(C)S2(=O)=O)=O)CCCC12CCN(C(=O)C(F)=C1CCC1)C2 Cc1cc(C(N2CCCC(NC(c3n[nH]c(C4CC4)c3Cl)=O)C2)=O)c(N)cc1F C1(CC(N2CC(O)(CC)C2)=O)CCOC(C)(C)C1.C(=O)(CCc1cc[nH]n1)N N1(C(=O)Nc2ccc(C(CC)C)cc2)CCCc2c1ccc(F)c2Cl c1(CC)cc(C(=O)N(C(C)C(C)C)C2CC2)no1.C(CC=O)OCCCC.N C1(C)(C(=O)NCC2(C)CCCN(C(C(C)(C)CF)=O)C2)COc2ccccc2O1 CC(C)CCCC(=O)N1CCN(C(=O)CCC2CCCC2)C(C2CC2)C1 N1(C(c2ccc(C(C)C)cc2)C(=O)N)CC(C)OC2(CCOC2)C1.C1(C)CCC1 n12nc(nc1-c1cnn[nH]1)OCC2.c1cc(C2CC2)ccn1 C1(C(=O)NC(CNC(c2c(N)cc(OC)c(F)c2)=O)C)CCC(C2CCC2)CC1 Cc1cnn(CCC(=O)N(C(C)CN(C)C(C2CC(c3ccccc3)C2)=O)C)c1 C=C(C)C1OCCCC1C(N1CCCCC(CNC(c2cccnn2)=O)C1)=O CCC(CC)CC(F)C(=O)NC(C)CNC(=O)CC(C)c1cnn(C)c1 C1(CC(=O)NC)CCN1C(=O)CC1(N(C)C(=O)OC)CC1 c1(C(=O)NCC2CCN(C(c3nc(C)oc3)=O)CC2C)cc(F)c(N)cc1F c1(NC)cc(Cl)ccc1C(=O)NC1CC(NC(c2ccncc2)=O)C(O)C1.O CCC(CC(=O)NCCN(C(=O)C(c1ccnn1C)O)C1CC1)C1CCC1 CCC(CC)(CCNC(=O)CC=C(Cl)Cl)NC(=O)CC1CCN(C)C1=O C1(NC(c2cc(CC)on2)=O)COC2(CCN(C(C3CC(O)C3)=O)CC2)C1 c1(C(=O)NC(C(=O)NCC2CC(C(C)C)C2)(C)CO)ncn2ccccc12 c1(N(C)Cc2c(C)ccs2)nc(N2CCC(c3nncs3)C2)nc2c1cnn2C N1(C(c2cccc(C)c2C)=O)CCC2C(CCN2C(c2ncccc2F)=O)C1 Cc1oc(C(F)(F)F)c(C(=O)NCCC(C)NC(C2CCOC2(C)C)=O)c1C c1(OC)noc(C)c1C(=O)NCCCCC.c1(C=O)ccccc1C(F)(F)F.N C12(NC(c3c(C)n[nH]c3)=O)CCCC(CN(C(=O)CCN3CCCC3)C1)C2 N1(C(C(CC)OC)=O)CC(C)(C)CCC1CNC(c1cc(Cl)cn1CC)=O C(C)(C)(CC(=O)N1CCOC(C)C1)n1cc(CSCCNC(=O)OC)nn1 c1cccc(C2CC2)c1.n1(CC(=O)NCC2(C(=O)N)CCC2)nnc(=O)[nH]1 CCN=c1ccc(C(N2CCCC(N(C(=O)CCCCCN(C)C)C)C2)=O)c[nH]1 CN1C(=O)c2ccccc2C1C(=O)NC1CC(NC(=O)C(O)P(C)(C)=O)C1 C(C(CNC(=O)C=NOC)C(F)(F)F)NC(c1c(C(=O)OC)cccc1)=O C1(C(=O)OC)CCOC1C(=O)NCC(C)C.C1(C=O)CCCN1C1CC1.N CN1C(=O)CC(CNc2nnc(-c3ccccc3)n2-c2ccccc2Cl)C1=O C1(C(F)(F)F)(C=O)CC2(CCC2)C1.C1(CC(=O)NC(C)C)CCCC(C)O1 N1(C(c2c(CC)n(C)nn2)=O)CC=C(CC(=O)N(C)CC2CCCC2(C)C)CC1 C1(CNC(c2nccc(C)n2)=O)C2CCCC1N(C(=O)C(C)n1cccc1)C2 C12(C=O)COC(C1)C2.C1(CNC(C=CC=CCC)=O)CC(C)CO1 N1(C(=O)CCOC2CCC2)CCCC2C(CCCN2C(c2ccc(Cl)o2)=O)C1 C1(C=O)Cc2c(F)cccc2O1.c1(C(=O)OCC)ccc(C(=O)NCC)cc1 N1(C(C(C)n2ccnc2)=O)CC2CCN(C(C3CCC=CO3)=O)CC2C1 c1(N2CC(c3ccccc3)(CC)OCC2)ncnc2[nH]c(C(F)F)nc12 C(C(COC)CC(=O)NCC1(C(N)=O)CN(C(=O)C(C)(F)F)C1)OC O=C1CC(CC(=O)N2CCN(C(=O)CCCc3ccc(Cl)cc3)CC2C2CC2)=NN1 C(=O)(C1=C(C2CCC2)N(CC2CCCS2)C(=S)NC1c1c(C)cccc1F)OC N(C1CCCn2nccc21)C(C(CC(=C)Cl)NC(=O)COC1CCCC1)=O N1(C(c2c(C)ocn2)=O)CC2C(C(=O)NCC3CCCC3)C2C1 N1(C(C2CC(CCC)C2)=O)CC2CCC(C1)N2C(C1Cc2nccn2C1)=O C1(C(=O)NC2(C3N(C(CSCCOC)=O)CCC3)CC2)CCc2nnnn2C1 C(CN=C(NCc1cccnc1O)NC1CCCC1)C1OCC(C)(C)C1 C1(N(C(CC)=O)C)CCN(C(=O)COC(C2CCN(C)C2)=O)CC1.C1CC1 C1(C(=O)N(C)CCNC(=O)CC2CCCCC2)(OC)CC(C)CC(C)C1 CC1CN(C(C23CC2CN(Cc2ccc(C(C)(C)C)nc2)C3)=O)CCC1=O c1(C(C(=O)NCCOCCOC)N)ccccc1CSC C1(F)(C(=O)NC2CCN(CCCNC(C(C3CC3)OC)=O)C2)CCCCC1 N1(C(C(CCC)(C)C)=O)CCC2(C1)CN(C(=O)C(C)(C)NS(C)(=O)=O)C2 C=CC(C)(CC)C(=O)N(CCNC(c1cnn(CC)c1N)=O)C.c1ccccc1 N1(C(c2ccc(OCC#C)cc2)=O)CCCC(C)C1.C(c1ncco1)=CC=O.N C1(CC=C)(NC(C23COCC2C3)=O)CCN(C(=O)C=C(C)CCC)CC1 N1(C(C2(C(C)C)CCN(C(c3cc[nH]n3)=O)C2)=O)CC2(CCOCC2)C1.COC C#CC1CN(C(=O)CN(C(=O)COC2CCCOC2)CC)CCN1C C1(C)(C=O)CC(O)CN1C(=O)C=Cc1cc[nH]n1.n1(CC)cnc(CC)c1.N CC(C)(C)C(C)(O)CNC(=O)C(Cc1ccc(Cl)cc1Cl)NC(=O)C(F)F CCC(F)(C(=O)OC)C(=O)N1CCC(NC(c2sncc2C)=O)C(O)C1 CN=c1[nH]cc(C(=O)NC(c2ccccc2)CNC(=O)CC(C)F)s1 C1(NC(c2scc(COC)c2)=O)CCCN(C(c2cnc(OC)nc2C)=O)C1C C1(OC)CC2=CCON(C2=O)OC2CN(C(=O)OC(C)(C)C)CC12 C1(C(=O)NCC(CNC(=O)CCc2scnc2C)OC)(COC)CCOCC1 N1(C(C(C)C(C)O)=O)CCCN(C(C2CC(O)(C(F)(F)F)C2)=O)C(CO)C1 C1(NC(CC2(NC(Cc3c(C)ncs3)=O)CC2)=O)CC(C)CCC1O c1(C(C)=O)cn(CC(=O)NC(CNC(c2cncn2C)=O)C2CC2)nn1 C(CCN(C)C(C1CCOC1)=O)(C(C)(C)C)NC(C1CN(C)C1)=O CC12CC(C(=O)NCC(CO)NC(=O)CC3(C)CCCO3)(CCO1)C2 CC1(C(=O)NCC2CC2)CCS(=O)(=O)CC1.c1(CCC(=O)N)ccncc1 C(=O)(C(=O)NOC)N1C(CCNC(C2CC(OCC)C2)=O)CCC1 CC(C)C(O)C(C)(C)C(=O)N1CCC(C(=O)Nc2cnn(CCF)c2)C1 c1(CC)ccc(C(=O)N(C2CCN(C(=O)Cc3ncn(C)c3C)C2)C)c(C)n1 C=CC(C)(CC)C(=O)NC1CN(C(=O)Cc2sc(O)nc2O)CC1CC C1(NC(c2nc(COC)oc2)=O)CC=C(C(=O)NC(C)C(C)F)C1 c1(N(C(c2ccncc2)C(=O)NC(C(=O)OC)C)C)cc(C)cc(Br)c1F c1(OC)ncc(C(=O)NC2(C#N)CCN(Cc3ccsc3)C2)cc1C c1(C(=O)NCC(CN(C)C(c2cscc2Cl)=O)O)cccc2c1C1CCC2O1 C1(NC(CCCC)=O)CN(C(=O)CC2OCCC2C)C2(CCOCC2)C1 CC1(CNC(c2cccc(CO)n2)=O)CCN(C(C2CC2C2CC2)=O)C1 c1(C(=O)NC2CC(NC(CC3C(C)OCC3)=O)C2)cnc2ccc(Cl)cn2c1=O C(=O)(C(F)OC(F)(F)F)NCCCN(C(=O)CCC1CCC1)CC n1(CCC)cc(Cl)c(C(N2CC(NC(=O)C=CCO)CC2C)=O)n1 N1(C(C2CCCCN2C(=O)CC2CCCO2)=O)CCCC2(CC2)C1 c1(C(=O)NC(CCOC)CNC(c2cc(C)no2)=O)ccc(C=O)c(F)c1 C(=O)(C(C)C(C)C(C)(C)C)NCC1CN(C(c2cc(OC)ns2)=O)C1 CCC(CC(=O)NC1(CC(=O)N(C2CCCNC2=O)C)CCCCC1)OC N1(C(c2cn(CC(CC)O)nn2)=O)CCCC(O)C1.C1(CC=O)CS(=O)(=O)C1 C(CC(C)(C)C(=O)N(CC(C)C(=O)Nc1cnc(Cl)nc1)C)OC C1(C(=O)NC2CC3CCC2N3C(=O)Cc2cnc[nH]2)CCCC2(CCC2)C1 Cn1nnc2cccc(C(=O)NC3CCC(NC(=O)C)C3)c12.c1n[nH]c(=N)s1.S Nc1ccnc(C(N2CCN(C3CCCN(C(C4CCCO4)=O)C3)CC2)=O)c1Cl CCCC(CC)C(=O)N(C1CN(C(=O)CCc2ccnn2C)CC1O)C CC(=O)CCCC(=O)NC1(C2CCCCN2C(c2ccns2)=O)CC1 C1(CC(N2CCC(NC(c3ccco3)=O)C23CC3)=O)CCCC2(CCC2)O1 c1(C=O)ccccc1C1(C)CC1.C1(NC(CNC(=O)OC)=O)CCC1.C N1(C(c2cc(C#N)no2)=O)CC(NC(=O)Cn2cc(Cl)cn2)C2CCCCC12 c1(C(=O)NC2CCC(NC(C3(C)C=CCCC3)=O)CC2)cc(F)c(F)c(F)c1N n12c(nnc1SC1CC1)N(CC)CCOCC(C)OCCC2.C(C)=O Cc1nc(C(F)(F)F)sc1C(=O)N(CC[Si](C)(C)C)CCc1ccc(Cl)cc1 n1(CC(=O)NCCCN(C(c2ccccc2)CCOC)C)nc(O)ccc1=O CCCS(=O)(=O)CC(=O)N1CCN(C(=O)CCCC2CCCCC2)CC1CF C1(C)(CNC(C(C)N(C)C)=O)CCN(C(=O)C=C(C2CC2)C2CC2)CC1 N1(C(C=CCC)=O)CC(C)(C)OC2(C1)CN(C(=O)C=C(CCC)CCC)C2 C(=O)(CC(C)(C1CCC1)NC(N)=O)NC(C(C)C)CN(C)C C1(NC(c2cccc(COC)c2)=O)CN(C(=O)C2=CCSC2)C(C)(C)C1.O C(=O)(C(=O)N=c1cc(C)o[nH]1)N1CCCC(C(N)=O)C1.c1(CC)cc(C=O)no1 C1(OC)C(NC(C2CCCCC2NC(=O)Cc2ccn(C)c2)=O)CC12CCC2 C1(OCC)CC(N(C)C(=O)Nc2ccncn2)C12CCC2 c1(C(N(C2CC(=O)N(C(=O)CCl)C2)CC2OCCN(C)C2)=O)ccn2nccc2n1 Fc1ccc(Cn2cc(C3CCCNC3)nn2)cc1 C1(NC(c2ccc(C(C)C)cc2)=O)CN(C(C2Cc3cscc3C2)=O)CCC1C c1(OC)ccc(CN(C(C(=O)NCCCF)C(C)CC2CCOCC2)C)cc1F CCCCC(F)C(=O)NCC1(C)CCC(NC(=O)Cc2cccnc2O)CC1 CC(C)(CC(F)C(=O)NC1CC(=O)N(O)C1)NC(=O)Cc1ccc(O)cn1 CN1CC2CCC(C1)N2C(=O)CC1CCCN1C(C1(CCN=[N+]=[N-])CC1)=O c1(C(=O)Nc2cncnc2Br)cc(-c2cccc3c2CCC3)cc2cc[nH]c12 C(CC(C(=O)NCCC(=O)N1CCCC1)NC(C1CCCCC1O)=O)N(C)C N1(C(C(CC)N(C)C)=O)CCN(C(c2cc(C3CC3)ns2)=O)CC1CCO C(c1csc(Br)c1)=CC(=O)NCCN(C(C)C)C(C1CC2CC2C1)=O CN1CCn2ncc(C(=O)NCC3CCN(C(c4sccc4F)=O)CC3)c2C1 c1(OCC)c(CCNC(=O)CNC(=O)Nc2cccnc2)cccc1O c1(NC(CCC)(c2nnnn2C2CCC2)C2CCC2)ccc(F)c(O)c1 C1(C(N2CCC(NC(C=C(C)c3ccco3)=O)CC2)=O)CCC2C1C2(F)F C(=O)(C1CCCc2cc(O)ccc21)NCC(CNC(c1c(C)nc[nH]1)=O)(C)C C1(CNC(C(C)CF)=O)CN(C(=O)CCS(C)(=O)=O)CC12CC2 N1(C(CC(=C)Br)=O)CCC2(CC(NC(c3[nH]cnc3CC)=O)CO2)C1 c1(C(N2CC(NC(Cc3c(C)ocn3)=O)C2)=O)ccc(-c2cn[nH]c2)cn1 C1(O)(CNC(C(N2CCC(C)CC2)=O)=O)CCN(C(C2(C)CCOCC2)=O)CC1 C=CCCCCCC(=O)NCC(c1ccccc1)CNC(=O)C#CC1(C)COC1 C(=O)(CCCC(N)=O)N1CCC(C)(CCNC(c2ccnc(O)c2)=O)C1 N1(C(CCN(CC#C)C(C2CN(C(C)=O)C2)=O)=O)CC(CO)CC1C c1(C(=O)OC)ccc2[nH]nc(CC3(C)CCC3)c2c1 C12CCC(C1)N(C(c1cc(C=O)no1)=O)C2.C(C(C(=O)N)N(C)C)OC.C c1(C(=O)NCCC2CN(C(CNC(=O)NC)=O)C2)cncc(Cl)c1Cl Cc1cc(C(=O)NC(C)(CNC(C2CCOCC2)=O)C2CCC2)cnc1O CC1CN(C(c2nnc(Cl)cc2N)=O)CCC1CNC(c1cc[nH]n1)=O C(=O)(C(C(C)C)NC(c1cnncc1O)=O)NC(C1CCCC1)CC c1(CC)cc(CC(N2CCCC2Cn2cc(C3(N(C)C)CCCC3)nn2)=O)on1 CC(CC(N)=O)C(=O)NCC(C)CN(C(=O)C=C1CC1)C C(c1cccc(F)c1)=CC(=O)NC(C(C)NC(=O)CCCF)CO c1(CCCCC)nc(C(=O)NC2CCC2NC(=O)CCC2CC2(C)C)cs1 c1(C(=O)NCC2C(CC)CCC2)ccc2nc(C)n(C)c2c1 C(=O)(CCC(F)(F)C(F)(F)F)NCC1(C)CCCN1C(=O)CC1CC=CCC1 C1(OCC)CC2(C1)CC2C(N1CCCC(n2ccnn2)C1)=O.[nH]1cc(Cl)cn1.C c1(OC)ccc(-c2cn(C3CN(C(c4cn[nH]c4)=O)CC3SC)nn2)cc1 CC(C)C(CN(C)C)NC(C1CCC(CNC(=O)CC2COCC2O)O1)=O CC1(C)CC2OCCC2CN(C(C2CC(=O)N(c3ccc(Cl)c(Cl)c3)C2)=O)C1 O=C(CCN=C(NC1CC1)NC1CCc2nnnn2CC1)NC1CCCC1 CC1(CCO)CCN1C(=O)C(C1CCOC1)NC(c1cnn[nH]1)=O Cc1nc(C=CC(N2CCC(CNC(c3cnnn3C)=O)C2(C)C)=O)[nH]c1C C1(C(N2CCC(O)C2)=O)CC2CCCCC12.c1(SCC)ccccc1C(=O)N.C C(CC(=O)NCC(O)CN(C(=O)C(C)n1cccn1)C)=C(C)C C(=O)(CN=c1cc[nH]cc1)NC1CC(N(C(C(C2CCC2)OC)=O)C)C1 C(C#Cc1cn(CCCC(F)(F)F)nn1)NC(c1ccc2c(c1)OCC2)=O C(=O)(C(Cc1cnc[nH]1)NC(C1CC(CF)C1)=O)OC.CC(C)C#N CN1CCC(C(=O)NC2(C(N3CCC(c4cnco4)C3)=O)CC2(C)C)CC1 c1(N2CC(C)(C)C(O)C2)c(Br)cccc1C#N C1(OC)CN(C(=O)CN2CC(C)(C)C2)CC1C(=O)NC1(CF)CCC1 Cc1cc(C(=O)NCC(C)NC(C2(N3CCCCC3=O)CC2)=O)n(C2CC2)n1 c1(C=O)ccccc1.C(C)(CC)NC(CC1C(CC)C1)=O.C=O.C(C)C.N C(C(=O)N1CC(F)(C(=O)NCC2CCC(F)(F)C2)C1)(C(C)C)OC CCCC(C(=O)N(C)CC1CCC(CNC(=O)C(O)C(F)F)CC1)C(C)C N1(C(CN2C(C)CC2)=O)CC(NC(=O)C=CC2CCC2)CC(F)C1 c1(C(=O)NC(CC)(CNC(=O)Cn2nnc(=N)[nH]2)CC)csc2cncn12 C(CC(=O)N(CCCO)CCO)N(C(C1(NC(CC)=O)CC1)=O)CC C(=O)(C(C)(CC)CC)NC(C1CCN(C(c2c(OCCC)cccn2)=O)C1)C C1(NC(c2c(C)snc2)=O)CCCCC1NC(c1ccc(Cl)[nH]1)=O CC1(C)NC(=O)N(CCC(N2CC3(NC(c4cocn4)=O)CC2C3)=O)C1=O N1(C(CC(CC)C)=O)CC2CC(NC(=O)CC3C=CCC3)CC2C1 C1(NC(=O)C2=CCCC2)CC2CC(NC(c3cncc(Br)c3)=O)CC12 c1(C(N2C(CN(C(c3c(C)nc(C)[nH]3)=O)C)CCC2)=O)c(C)nc2ccccn12 C(C(C)(C)CC(=O)NC1CCCCC1NC(c1ccn(CCO)c(=O)c1)=O)OC C1(C(N2CC(O)(C(=O)OC)C2)=O)(NC(c2sccc2O)=O)CCN(C)C1 C1(NC(CC(C)(C)F)=O)CC2(C1)CC(NC(=O)CC(=O)OC(C)(C)C)C2 N1(C(c2nc(C(=O)OC)oc2)=O)CC(CNC(=O)C2=C(C)CC2)CC1C Cc1c(C(=O)NCC2CC(NC(C3CCCCC3(F)F)=O)C2)[nH]c2ccccc12 N#Cc1ccc(C(=O)NC(CNC(c2c(Cl)nsc2Cl)=O)CO)[nH]1 C1(NC(c2c(CCCC)ocn2)=O)CCCCCC1NC(c1n[nH]cc1OC)=O c1(CC)cccc(C(CO)NC(=O)CC)c1.C(=O)NCCN(C)CCN(C)C C1(CNC(COCCC#C)=O)(C)CC(F)(F)C1.C1(C=O)CCC(=O)N1 Cn1nc(C(=O)NC2CC(C(=O)NC(CO)C(C)(C)C)C2)cc1CO c1(CC)ccc([N+](=O)[O-])cc1C=O.C(C)C(C)C.c1(CC=O)ccc(Cl)s1.N C1(NC(=O)Cc2ccon2)CN(C(=O)CC2CCCC2(F)F)C2CCCCC12 CN=c1[nH]c(=NCC23CCN(CC2)CC3)[nH]c(=NCC2(C)CC(C)(C)C2)[nH]1 CN1CCC(CC(=O)NCC2CCCC2NC(=O)CSC(F)F)C1 N1(C(C(CCCC)C)=O)CC(NC(c2cnoc2CC)=O)Cc2ccccc21 c1(C(N2C3(CN(C(c4cc(C)cc(O)n4)=O)C3)CC2)=O)ccccc1S(C)=O N1(C(C2(NC(=O)CC3CCSC3)C(C)(C)C2)=O)CC(O)C(F)C1 C(=O)(C(O)CC1CC1)N(CC(C)N(C(=O)CC1CSCCO1)C)C C1(CNC(c2c(C)snn2)=O)CCCC(CNC(c2cnccc2Cl)=O)C1 N1(C(CC(C)C2CCCCC2)=O)CCN(C(C23CCC(F)(CC2)C3)=O)CC1C1CC1 C1(C(=O)OC)Cc2ccccc2N(C(c2nc(Br)sc2C)C(=O)NCCC2CC2)C1 c1(CCNC(=NC)NCCc2ccc(F)cc2)ccc(Br)c(OCC)c1 C1(NC(CSC(C)(C)C)=O)CCOC(C(=O)NCCCc2cn[nH]c2)C1 C(C(C)NS(=O)(=O)CC1CC1)=CCC C1(CC(C)C)(C(N2CCC(NC(=O)CCc3ncc[nH]3)CC2)=O)CCNC1=O C1(SC)CN(C(c2ccc(Cl)cn2)=O)CC1NC(=O)CC1CCC(F)(F)C1 c1(C(=O)NC(C(C)NC(=O)COc2ccccc2O)C)cccc2nc[nH]c12 O=C(O)C#CC(=O)N1CC2C(C(N3CCCCC3CCO)=O)C2C1 N1(C(C=Cc2c(C)ccnc2)=O)CC(C)CN(C(=O)C(C)(C)CC#N)CC1C N1(C(C(=O)NC2CCCN(S(CCC)(=O)=O)C2)=O)CCOC2CCCC12 c1(OC)cc(C)cc(C(=O)NC)c1C.C1CCC1.c1(C2(C=O)CC2)cccs1 C1(CCC(=O)N(C)CCc2cc[nH]n2)CCCCN1C(=O)CC1OCCC1(C)C C1(C(=O)NC(C)C(CO)NC(=O)CSC(C)(C)C)CN2CCCN1CC2 c1(N2CCC(C)C(NC(c3n[nH]c(O)n3)=O)C2C)ccc2nccnc2n1 c1(CCNC(c2ccoc2CNC(C2CC23CCC3)=O)=O)ccccc1O C1(CCNC(CCC)=O)(NC(=O)CSCCC#N)CCCC1 CC(C)CCC(=O)N1CCC(C2CCCN2C(c2ccc(C3CC3)cc2)=O)CC1 C1(C#N)(C(=O)NCC(C(=O)NCCc2nnc(C)s2)O)CCOC1 N1(C(CCC2(C)CC2)=O)CC(NC(=O)Cc2ccc(Br)cn2)CC(F)C1 Cc1nc(=NCC2CCN(C(c3ccnn3CCN(C)C)=O)CC2C)[nH]cc1Br C(=O)(C1CCCCc2ccccc21)N1CC2(N(C(c3scc(C#N)c3)=O)CC2)C1 N1(C(CN(C)C(C2CC2C(N)=O)=O)=O)CCN(C(c2occc2F)=O)CC1 c1(C(N2C3CN(C(c4ccc(I)c(I)c4)=O)C(C3)C2)=O)c[nH]c2ccncc12 c1(C(C)OC)nc(C)c(C(=O)N(CCc2csc(C)n2)C)s1.C(=O)CCF C1(C(N2CCN(C)CC2CNC(=O)CC2CCCN2C)=O)CC2CCCC(C1)C2 c1(C(=O)NC(C2CCOC2)CNC(C=CCC)=O)c[nH]cc1CC C12(CNC(C(CC)SC)=O)CC1CN(C(=O)C(C)n1cnnn1)C2 N1(C(c2c[nH]c(=NCC)s2)=O)CCC2(CCCN2C(=O)C(C2CC2)SC)CC1 c1(C(C(=O)NCC)N(C)Cc2nc(C(=O)OCC)n[nH]2)nn(C)cc1Cl c1(-c2ccc(-c3n(CCC=C)ccn3)cc2)n[nH]c2c1CCC2 c1(NC(CCCCC)C)ccc(-c2ccccc2)c(F)c1 c1(C2(C(=O)NC3CC(c4nn[nH]n4)C3)CC2Br)ccccc1 c1(OC)cc(C)nc(N(C2(C#N)CCNC2)Cc2c(Cl)cncc2Cl)n1 C(=O)(C1=NOCC1)N(C)CCOCCNC(C1CCC1c1nncn1C)=O C1(NC(c2c(OC)ccnc2)=O)CC2CN(c3nc(Cl)ncc3C)CC12 CC1(NC(C2CC2c2ccccc2)=O)CC(NC(=O)CC2CCCCC2)C1 C1(CNC)CCC(CNC(C2(N)CCSCC2)=O)CC1 n1(C2CN(C(CCOCCC)=O)C2)cc(CNC(C2COCCO2)=O)nn1 c1(N2CCCC(C=C)C2)nc(NCC2(C)NC(=O)NC2=O)c2ncsc2n1 C1(C#N)(C(=O)NC(CN(C(c2cnc(C)nc2C)=O)CC)C)CC2CCC1CC2 C1(C(=O)NCc2nc(C)on2)CN(Cc2ccn(C(C)(C)C)c2)CCC1O n1(CC(=O)Nc2cncc(C#N)n2)ccc(=NCc2occc2Br)nc1O C1(NC(C#CC(=O)O)=O)C2CCCC1CN(C(=O)CSc1nc[nH]n1)C2 N1(C(CSCC(N)=O)=O)CCCC1CC.c1(C=O)scnc1.C=O.CCF.N c1(COC(C2CC(CF)C2)=O)ccc(Br)cc1Br c1(C(=O)Nc2ccccc2C(F)F)cc(Cl)cc2cc[nH]c12.c12cc(ncn1)N2 C(C)(N=c1cc(C)nc(COC)[nH]1)C1CCN(C(C(C(CC)C)OC)=O)C1 c1(C(=O)NCC(C)NC(c2cc(C)c(O)nn2)=O)c(Cl)ccc(Br)c1F c1(C(N2CC(O)(CN(C(c3c(C)ccnn3)=O)C)C2)=O)cc2ncccc2o1 c1(OC)ccc(Cl)cc1C(=O)NC1(C#N)CCN(Cc2cnc(O)c(Br)c2)C1 c1(C2C(CNC(=O)NCC(C)(C)C3CNC3)C2)ccc(F)cc1Br C12(C(=O)N)CCC(CC1)C2.C1(C=O)C2CCCCC12.CCS(=O)(=O)NCC Cc1ccc(C=c2sc(=C(C#N)C(=O)c3cc(I)sn3)n(C)c2=O)c(Cl)c1 N1(C(c2cnc3sccn23)=O)CCN(C(C2CCOCC2)=O)C2CCCCC2C1 Cc1nc(NCC(S(C)(=O)=O)C2CC2)cc(=NCC(C)(C)c2nncn2C)[nH]1 c1(C(=O)NC(C(C)C)C(C)NC(=O)CCSc2ccccn2)cnn2c1CCC2 c1(C(N(CCOCCOCCOC)C)=O)cncnc1C1CC1 C(C(C)(C)C#CC(=O)NC1CCCCCC1CO)NC(CSCC)=O CC(CCNC(=O)Cc1ccnn1C)CCNC(C1(C)COC(=O)C1)=O C=C(C)CC(C)C(=O)N1CCN(C(c2csnn2)=O)C(CCC)C1 C(=O)(C1=CCC(C)CC1)NCC(CC(F)(F)F)NC(CC(C)=C(C)C)=O CCC(C#N)C(=O)N1CCOC(CNC(C23CCCC2(C(N)=O)C3)=O)C1 c1(-c2nc(C)nn2CCCO)ccc(S(=O)(=O)N(C2CCCCC2)C)o1 c1(C(N2CCC(O)C2)=O)ccc2nccn2n1.C1(C(=O)N)(COCC)CC1 C1(COC)(CNC(=O)C(C)N2CC(C)C2)CCCN1C(c1cncn1C)=O C1(CNCC=CCC)(NCc2ncn(C(C)(C)C)n2)CCCCC1C c1(C(N2CC3CCN(C(=O)CN4CCCC4)C3C2)=O)cc(Br)cc([N+](=O)[O-])c1Cl c1(C(C)C)ccc(C(N2CCCC(NC(c3ccncc3Cl)=O)CC2)=O)c(O)n1 C(C(COC)CC(=O)NC1(CCOC)CCN(c2ccnc(C#N)n2)C1)OC CCC(C)C(O)C(C)C(=O)N1CC2(C)CC1(C(=O)NCC1(O)CC1)C2 C(=O)(CS(=O)(=O)C1CCCC1)N1CC(C)(NC(=O)CCc2cncnc2)C1 C1(C)(C)CC(=O)N2CCCC2Cc2cn1nn2.C1(C(C)(C)NC)CCCCC1 CN1CCN(C(C2CCOC2)=O)C(CNC(=O)CSc2cccs2)C1 C1(C(=O)NCCNC(=O)Cc2c[nH]ccc2=O)CCS(=O)(=O)CC1 N1(C(c2ccc(N3CCC(C)CC3)cc2)=O)CC(=O)NCC1C C(CC(C)(C)C(=O)N(C)CC1CCCN1C(c1snc(O)c1Cl)=O)SC N1(C(CSCCC)=O)C2CCC1CN(C(c1ccc(Br)cc1F)=O)C2 C12(C(N3CCCC(NC(CSC(C)C)=O)C3)=O)CC3CC(C1)CC(O)(C3)C2 C1CN(C(C2C(F)(F)C23CC3)=O)CCC1C(F)(F)F.C(c1nccs1)=CC=O N1(Cc2ccc(S(=O)(=O)N(C)C)cc2Br)CCC2(CC1)C(=O)NCCN2C C(C)(C)(CCC)NC(C(CC)OCCOC)=O.C(=O)C(F)OC(F)(F)F.N C1(CSC)CC2CCC1N(C(C1(CC)CCCN1C(=O)C(COC)OC)=O)C2 c1(C(=O)NC2(CC(=O)NCC(C)(C)F)CC2)ccc(N)c(F)n1 c1(CC)nnc(O)c(C(=O)NCCCN(C(=O)CCc2cncnc2)C)c1CC N1(C(c2ncc(CC)s2)=O)CCCC(C)C1C.C12(C=O)CC(C)(C1)OC2C.N c1(C=O)nsc2c(Cl)cccc12.c1(C(=O)NCCOCC)cccc(O)c1F.N N1(C(CN(CCC)C)=O)CCC(N(C)C(c2cncc(N(C)C)c2)=O)C2(CC2)C1 c1(N2CCC(CNC(c3c(C)nn(C)c3C)=O)CC2)cc2nnc(C)n2cn1 N1(C(c2c(N)cc(Cl)nc2)=O)CCN(C(C23CCCN(CC2)C3)=O)C2CCC12 C(=O)(CCCCCc1cccs1)NCC(C1CCOC1)NC(C1CC(OC)C1)=O C1(CCC(=O)NCCCc2ncc[nH]2)CCCCN1C(C1CCSC1)=O CC1CC(C(N2CC(F)(CNC(=O)C(F)(F)c3nccs3)C2)=O)CCO1 C1(CCC(=O)N(C2CN(C)C2)C)CCN(C(c2cncnc2)=O)CC1 c1(C(N2CCC(O)(C(C)NC(CC(C)OC)=O)CC2)=O)cc(C)c(C)c(F)c1 C1(CNC(=O)C(=O)NCC2CCNC2)NCCC1C1CC1 C(=O)(C1=CC2CCCCCCC12)NCCCN(C)C(c1cc(N)cc(F)c1)=O N1(C(c2c(F)ccc(C)n2)=O)CC2CCCCN2CC1CNC(=O)CS.C(C)C Nc1c(F)ccc(C(=O)NCC2CCCN2C(=O)CCC2CCCO2)c1F C1(C(=O)N(CCCC(=O)O)C)(COC)CC(F)(F)C1 N1(C(Cn2c(C)csc2=O)=O)CCCC(O)(C)CC1.C(=O)(CC(C)(C)C1CC1)N C1(NC(CN(C(=O)OCC)C)=O)CC(C)C1.C(=O)CCCc1ccsc1.N c1(CNC(=O)NCC2CCOC2)nc(C2CCCO2)n[nH]1 C(c1cnn(C)c1C)=CC(N1CCCC1C1CC1)=O.C(CCC=O)OCC=C.N c1(C=O)[nH]c(C)cc1-n1cc(C2(O)CN(C(=O)C(C)CC3CC3)C2)nn1.CO Cc1c(CNCCN2CCN(CCO)CC2)sc2nnccc12 N1(C(CS(CC)(=O)=O)=O)CCC2(CC(NC(=O)Cc3ccc(C)nc3)C2)C1 Cc1cccc(OCC(=O)NCCCCC(C)NC(C2CCCC(C)C2)=O)c1 CC(C)C(C#N)C(=O)NCC(N1CCN(C(C2CC=CCC2)=O)CC1)=O CC1=C(C(=O)NC2CCCC2C(=O)N(CC(C)C(C)(C)C)C)CCO1 CCCC(C(=O)N1CC2(CCC2)CC1C(=O)NCCCCNC(N)=O)C(C)C c1(OC)ncc(F)cc1C(N1CCC(NC(c2cc(Br)ccc2I)=O)C1)=O Cc1ccc(CN(C)C(C2CN(C(=O)C(C)CN(C)C)CC2C)=O)cc1 n1(CC(N2CC(CC)C(NC(c3cnccn3)=O)CC2)=O)cc(C)c(O)nc1=O CC(C)CS(=O)(=O)CC(=O)N1CCC2(CCCC2NC(c2cc(F)n[nH]2)=O)C1 C1(NC(c2ccc(-c3ccco3)o2)=O)CCCC12CN(C(C1CSCCS1)=O)C2 N1(C(C2(OC(C)=O)CC2)=O)CC(NC(C2(C)CSC2)=O)C1 C1(C(=O)NC(CCNC(c2c(CC(C)C)onc2)=O)C)CN(C)C(=O)N1 c1(C=O)ccc(C(F)(F)F)c(O)n1.C(C)C(C)(C)C.Cn1nccc1C(=O)N c1(C(=O)NC2CC(C(=O)NCC3CCC3)C2)ccc2nc(O)[nH]c2c1 c1(C(=O)OC)cccc(C(N2C3CCC2C(NC(=O)Cc2ccoc2)C3)=O)c1C N1(C(C(CC=C)NC(=O)CN(C)CCOC)=O)CCCC2C(O)CC12 C(=O)(CCC(=O)OC)NC(CC)CN(C)C(c1cn(CC2CCOCC2)nn1)=O N1(C(CCCn2cc(Cn3c(C)nnc3Br)nn2)=O)CCNC(=O)CC1(C)C C1(NC(C(C)OCCOC)=O)CC2CC(NC(c3cc(Cl)no3)=O)C1C2 N1(C(CCc2ccn(C)n2)=O)CC2(CC(C(N3CC(C#N)C3)=O)CO2)C1 C1(C(=O)NCCCC(F)F)OCCC1NC(C1CC=CC1)=O C1(CN(C)C(C2CC2C)=O)CCC(CNC(=O)C(O)c2ccsc2)CC1 Cc1ccc(C(=O)NC(C)(C)CCCNC(C2(C)CCC(C)C2)=O)nc1 N1(C(C2(CC)CCCO2)=O)C(CC(=O)Nc2cnn(C(F)F)c2)C2CCCC12 C(=O)(C1=CCC2CCC1N2C(C1CCCS1)=O)NCC(=O)N(CC)CC C(CN=C(NCc1cnnn1CC1CCC1)NC(c1cccs1)C)OCC Cc1sc(Cl)c(C(N2CCC(CN(C(=O)CC3CN(C)C3)C)C2)=O)c1C CC(C)CC(C)(CNC(=O)C=CBr)NC(=O)Cn1cnc([N+](=O)[O-])c1 C12(C(N(C(CCNC(c3cc(C)nn3C)=O)C)C)=O)CC1COC2(C)C N1(C(C2N(Cc3ccc(OC)nn3)CC(O)C2)=O)CCOCC(O)C1 C(=O)(C(C)(O)C(C)C)NCCCCNC(c1ccn(CCOC)n1)=O N1(C(C(CC=C)(C)C)=O)CC(NC(c2cc3c(s2)CCC3)=O)C2(CCOCC2)C1 C(=O)(CC(C)(C)C#N)NC1CCC(C(=O)NC2CN(CC)CC2C)CC1 C1(C(=O)NCC#CCOC)CC2(CCC2)CN1C(=O)CC(C)C.C(C)(=O)N C1(C(N(CC(O)CC2CC2)C)=O)CC12CCN(C(=O)CN)CC2.c1cccnc1 C(=O)(C(CC)C(=O)N(C)C)OCC.C1(O)CN(C(=O)C(C2CCCCC2)C)C1 O=C(CC1CCc2cc(Br)ccc21)NC1CN(C(C2CCC(F)(F)C2)=O)C1 C#CCCC(O)C(=O)N1CC2CCC2(CNC(c2cccc(F)c2OC)=O)C1 c1(-n2c(CCc3csc(C4CC4)n3)nc(CC(C)C)n2)cc(F)cc(F)c1 Cc1ccccc1CC(=O)N(CC(=O)NCCSC(C)(C)C)C N1(C(c2sc(C)cc2C)C(=O)NCCSC)CCC(c2ccco2)CC1C Cc1cc(C(N2CCC(N(C)C(c3cn(C)c(C)n3)=O)C2)=O)c2c(c1)CCO2 N1(C(C(=O)NC2CC2)=O)CC(C2CC2)(C(=O)NCC2CCOC2)C1 C(=O)(CC(F)(F)F)N.C1(O)(CC)CN(C(=O)CC2(O)CCOC2)C1.O=CC N1(C(C=NOC)=O)CCC(O)(CNC(=O)C2=C(C)CC2)C1 [N-]=[N+]=NCC(C(=O)NOC1CC2CCC1C2)NC(c1cncnc1)=O c1(C(=O)NCC2CCCCC2)ccc2nonc2c1.C1(C(=O)N)CCC(F)(F)C1 C(=O)(C(C)CC(C)(F)F)NC1(CO)CCCN(C(c2cc(C)nnc2)=O)C1 C(=O)(C1=C2CCN=C2NC=C1)N1C(CNC(C(C)N(C)C)=O)C(C)(C)CC1 C1C=CC(C=O)N(C=O)C1.C1(C(=O)OCC)CCC1N.C(C)(C)C.C n1(CC(N2C(C)CC(CNC(C(CC)F)=O)C2)=O)nc(C)c(Cl)c1C N1(C(CC(=O)NCC)=O)CCCCC12CN(C(=O)C(CN(C)C)CC)C2 C1(C(=O)NC2CC(CNC(C(CC)(C)O)=O)C2)CCc2ccccc2C1 N1(C(C(CO)NC(N)=O)=O)C2CCC1CN(C(c1ncccn1)=O)C2 C1(CNC(C2CC3(CCO2)CC3)=O)CC12CCN(C(c1cn[nH]c1)=O)CC2 C(=O)(C(c1cccs1)NC(c1cccs1)=O)N(CCCC)C N1(C(C2CC(=C)C2)=O)CCC2(CCC(C)O2)CC1.C12(C(=O)N)CCCC1C2(F)F c1(N2CC(C)C(NC(c3cnc(O)nc3O)=O)CC2)nc2cccnc2s1 c1(OCC#C)ccc(CNC2CCCC(CO)C2)cc1 c1(C(=O)NC2CN(Cc3ccc(C#C)s3)C2)ncnc2c1ccn2C1CC1 C1(NC(C(C#C)(C)C)=O)CCCCCN(C(=O)COc2ccc([N+](=O)[O-])cc2)C1 N1(C(CCn2c(C)ncc2)=O)CCN(C(C2CC(C)CCC2C(C)C)=O)CC1C C1CCN(C(=O)CCc2cncnc2)C1C(C)C.c1(OCC)cc(C=O)sn1.N N1(C(Cn2cc[n+](C)c2)=O)CCCC(O)(CNC(C2CCC(=O)O2)=O)C1 C(=O)(C(C)N(C)C)NC1CCN(C(c2coc(C)n2)=O)C1.C(C)(C)C.CC C1(CCC)CCN(C(=O)C=CC2CCCC2)CC1.C1(O)(CC#C)CC(C=O)C1.N N1(C(C(F)=C(C)C)=O)CCCC(C(=O)NCCNC(=O)CC(F)(F)Cl)C1 C(=O)(N=C1CCN(c2cccc(C3CC3)c2)N1)N1CCc2c(c(C)cc(C)c2)C1C CC1CC(C(N2CCOC(CN(C)C(c3cnn(C)c3)=O)C2)=O)CC(C)C1 c1(C(=O)NC(C(C)(C)NC(c2c(C)nns2)=O)C)cc2scc(Cl)c2[nH]1 N1(C(C=CC(C)(C)C)=O)CC(CNC(=O)CC)C2CC12.CC(F)(F)F.O S(=O)(=O)(c1ccc(NC(C)(C)CF)cc1Cl)NCCC1CCN(C)C1 c1(C(N2CCCC(C)C2CNC(C23CCCCC2C3)=O)=O)nn(C)cc1[N+](=O)[O-] c1(C(=O)NCC(C(=O)O)CC2CCCC2)cccc2[nH]ccc12 N(S(=O)(=O)N=S(C)(=O)C1CCCCC1)Cc1occ(C(C)(C)C)n1 CC1CCN(C(=O)Cc2ccno2)C1C.c1(CC=O)nnn(C(C)(C)C)n1.N N1(C(C2OCCC(C)(C)C2)=O)CCCC(C)(C)C1C(N1CC(CN=[N+]=[N-])C1)=O CC1(NC(=O)CCc2ccccn2)CCCN(C(c2ccc(C(F)F)cn2)=O)C1 c1(C(N2CCC(=CCNC(C3CC(O)C3)=O)CC2)=O)cccc(Cl)c1F c1(C2C(=O)NN(c3cn(CC)nc3)CCO2)ccncc1.C(C)(C)(C)C N1(C(C(CC)O)=O)CC2CCN(C(=O)COc3ccc(C(=O)OC)nc3)CC2C1 C1(NC(C(=O)Nc2c(Sc3cc(C)no3)cccc2)=O)C2CCOC2C1(C)C C1(CCC(=O)NCC(C(C)C)(F)F)CCCCN(C(C2CCC(=O)C2)=O)C1 N1(C(C2C(NC(c3nc(CC)oc3)=O)CCO2)=O)CCC(CC)(CO)C1 N1(C(CC=CCNC(C(CC)(F)F)=O)=O)CCOCC(F)(F)C1 N1(C(C(CC=C)C)=O)CCOC2(CCCN(C(C3(COC)CCC3)=O)C2)C1 n1(CCCN(C)C(c2cn(C)nc2-c2ccccc2)=O)cc([N+](=O)[O-])ccc1=O C(C)(C(=O)NC1CC(NC(=O)C(C)c2ccco2)C1)OCCC=C C(CCC(=O)N1CC(O)(CN(C)C(c2csc(CS(C)(=O)=O)n2)=O)C1)OC CC(C(=O)NC1(C(N2CC(F)CC(F)C2)=O)CC1C)C(F)(F)F N1(C(CC2N(C)CCC2)=O)CCN(C2CN(C(=O)CN3CCOCC3)C2)CC1 C#CCC(C)(C(=O)NC(CC1CC1)CO)NC(=O)C(n1nccc1C)C C(=O)(CC(C(F)F)NC(c1cc(C(N)=O)c[nH]1)=O)N(C1CCN(C)C1)CC N#CC1CCN(S(=O)(=O)NCc2ccc(N3CCCC3=O)cc2)CC1 C(C(=O)N1CC(C(C)NC(=O)CC(O)C(C)C)C1)(C(C)(C)C)NC(C)=O CC(C)(O)CCCC(=O)N1CCCC(C)(F)C1 c1(C(=O)NC2CC(NC(c3ncnc(C)c3C)=O)C2)cc2cccc(Cl)c2s1 C12(C(=O)NCCC(C(C)C)Nc3ncncc3Cl)COC(CCO1)C2 C1(NC(C2C(C=C)C2)=O)CCC(C)(NC(c2nnc(Cl)cc2N)=O)CC1 O=C(NNS(=O)(=O)c1ccc(C(F)(F)F)c(Cl)c1)NCC(c1ccc(Cl)cc1)F c1(C(=O)NC2CC3CC(NC(C(NOC)=O)=O)C3C2)ccc2occc2c1 c1(OC)cncc(C=CC(=O)NC2CCCN(C(C34CCCC3CCC4)=O)C2)c1 C1(NC(c2nc(CC)oc2)=O)CN(C(=O)CCc2ncco2)CC1O C1CCN(C(=O)CN(S(C)(=O)=O)C)C12CCC2.CCC1=NOC(CC(=O)N)C1 N1(C(CN(C(=O)OC)C)=O)CCCC(C(C)C)C1.C1(C=O)CC1.C(C)C.N C1(CNC(c2c[nH]c(=NC)o2)=O)CC2CCC1N2C(=O)C.C(=O)C1CC1.N Cc1cc(O)nc(C)c1C(=O)NC1CCN(C(c2ccccc2O)=O)C1C(C)C N1(C(C(CSC)C)=O)CCN(C(=O)CCCc2ncc(C)o2)C2(CC2)C1 c1(C(=O)NC(CNC(CC(COC)C)=O)(C)C2CC2)cccc2cncn12 c1(C(N2CCN(C(CCOC)=O)C(c3ccccc3)C2)=O)snc2ccccc12 C(N=c1nc2c(Br)csc2c[nH]1)C1(O)CN(C(=O)Cc2ccc(Cl)c(F)c2)C1 S(=O)(=O)(c1ccncc1)Nc1ncc(-c2ccc(C(=O)OC(C)(C)C)nc2)cn1 n1(C(C)C)nc(C2CC2)cc1NC(=O)CCC1CCC(C)O1 C12(NC(=O)Cc3csc(S)n3)CCCC1CN(C(C1CN3CCC1CC3)=O)C2 N1(C(Cc2cccc(OC(=N)O)c2)=O)CC2CCC1C2.C1(C=O)C=CCCC1.C(C)=C C(N=c1[nH]c(=NCC2(F)CCC2)[nH]c2ccccc12)c1n(CC)ccc1 C(=O)C(C)(C)S(C)(=O)=O.C1CCCC1.C1(C(=O)OCC)(C=O)CC1.N N1(C(C(C)CC2CCC2)=O)CC2(CCN(C(C3(C)CCCOC3)=O)C2)C1 Cc1scc(C(=O)N(CCCC(=O)NC2(C)CCC(C)C2)C)c1C c1(C(=O)N)cc2c(C#N)c(F)ccc2[nH]1.C1(CC(=O)N(CC)CC)CCC1 C(C)(C(=O)NOCC1CCCO1)N(C(C(CC1CCC1)OC)=O)C C1(CNC2CN(C(C3CCC(C(=O)OC)C3)=O)C2)CCC(C(N)=O)CC1 N1(C(C(C)SC)=O)CC2(CNC(=O)C(C)(C)N(C)C)CC2(C(F)F)C1 CC1CN(C(C2CS(=O)(=O)C2)=O)CCN(C(=O)Cc2ccn(C)c2)C1 c1(C(NC)=O)cc(S(N)(=O)=O)ccc1F.N1(C(C(C)C#N)=O)CCC2(CC2)C1.C Cc1cc(CC(=O)NC2(CNC(C3CC4CCC3C4)=O)CCCCC2)ccc1Cl C1(NC(=O)CC2CCCCCC2)CC(O)CN(C(C2(F)CC=CC2)=O)C1 C(=O)(C1=C(C)CCC1)N1CCC(C(C)NC(c2cnc(CC)[nH]2)=O)CC1 c1(C(C)C(=O)N2CC(CC(C)NC(C3(C4CCCO4)CCC3)=O)C2)cccnc1 Cc1ncc2c(n1)CCC(C(N1CCC(C)N(C(=O)Cc3cccs3)CC1)=O)C2 N1(C(c2c(C)[nH]cc2)=O)CC2(CCCC2CC(N2CCC(CO)C(O)C2)=O)C1 c1(CN2CC3(CC(CC(=O)NCc4cc(Br)cs4)C3)C2)cc(F)cc(F)c1O C1(C(=O)NC2C3(CC(OC)C3)C2)CN2CC3CC2(CO1)C3 CC1Cn2nc(C(=O)N)cc2C(=O)N1.C12CC1CN(C(=O)CC1CC=CC1)C2.C C1(C)(C(N(CCCNC(=O)COCCCF)CC)=O)CCNC1=O c1(C(=O)NCCNC(Cn2nc(C)c(Cl)c2C)=O)[nH]cc2c1CCCC2 C1(NC(C(C)=C2CCCC2)=O)(CO)CN(C(C2CCCC2n2cccc2)=O)C1 c1(C=O)ccc(C2SCCS2)cc1.CC(CNC(=O)CCC1CC1)C1CCC1.N C(=O)(C(C)CC(=O)N1CCC(F)(CNC(c2nc(C)nn2C)=O)C1)OC C(=O)(CC(O)CCCCC)NC1C(NC(CC2(C=C)CCCCC2)=O)CCOC1 N1(c2cccc(S(=O)(=O)N3CCC=C(C)C3)n2)CCC2(CCC(O)C2)CC1 c1(C(=O)OC)cc(CC)ccc1Br.C(=O)(C(=O)N)NC(c1cnsc1)C CN1CCC(C2(C(=O)NCCCCCNC(=O)C(C)(C)c3ccno3)CC2)CC1 C1(C(N2CCC(OC)C2)=O)C2CN(C(=O)CCCC3CCCO3)CC12 N1(C(C(C)(C)N(C(C)=O)C)=O)CCC(c2ccccc2Cl)(C(F)(F)F)C1 C1(C)(CC)CCC(Cn2cc(Cn3cc(C(O)C(C)C)nn3)nn2)O1 C(=O)(CCCCNC1CC1c1c[nH]c(C)c1C(=O)OC)OCC N1(C(CCC2(C)CC2)=O)CCC(NC(=O)C(O)c2ccsc2)C2(CC2)C1 N1(C(CNC(N)=O)=O)C2CCC1CN(C(C13CC(CF)(CO1)C3)=O)C2 C1(c2n(C)ccn2)CN(C(C2CCOC2)=O)CCN1C(c1cc(F)n[nH]1)=O N1(C(CCc2cncc(OC)c2)=O)CC(NCc2cncs2)CC(C(F)(F)F)C1 CC1(F)COCCN(C(C2(F)CCN(C(c3ncc4ccccn34)=O)C2)=O)C1 C1(CN2C(C(C)O)CC(C)CC2)CCC(C)(C)N(C(=O)OC(C)(C)C)C1 C1(C(N)CNC(=O)NCc2cn(C3CCCC3)nn2)CCOCC1 C1(NC(C(C)C2CCOC2)=O)(CNC(=O)C#CC2CC2)CCOCC1 c1(C(N(C(CNC(C2(OC)CCSC2)=O)C)C)=O)cccc(C#C)c1Cl Cc1c(C(=O)NCCC(C(C)C)NC(C2(C)CCC(=O)N2)=O)ccc2n[nH]cc12 c1(C(=O)NCC2N(C)CCN(C(=O)CCC(C)(F)F)C2)ccc2ccncc2c1 C(=O)(CCC(C)(C)[N+](=O)[O-])NC1C(C(N(C2(CO)CC2)C)=O)OCC1 c1(CCC)[nH]ccc1C(=O)N(CC(=O)N(C)Cc1cccnc1)C(C)C C1(C(=O)NC2(CC=C)CC2)(CC=C)CCCN1C(=O)C(C)Cn1cccn1 c1(C(N(C2CCN(C(c3cc(C)c(F)cn3)=O)C2)C)=O)[nH]c2ccccc2c1Cl C1(C(N(C)CC2N(C(C(C)SC(F)(F)F)=O)CCC2)=O)CC(=O)N(O)C1 c1(C(=O)NC2CC3CC(NC(COCCCC)=O)C2C3)[nH]nc2c1CC(C)CC2 C1(CC(=O)OCC)CCN(N2CCC(c3cccc(OC)c3)CC2)C1 N1(C(CC2(C=C)CCC2)=O)CCCC(C(C)(O)CNC(c2ccsc2C)=O)C1 C(=O)(C(C)CC(=O)N1CC(C)(Cc2ccc(Oc3ccccn3)cc2)C1)OC N1(C(C2(CCC)CC2)=O)CCC2(CCN(C(C3(O)CC(F)(F)C3)=O)C2)C1 S(=O)(=O)(c1ccc2c(c1)CCC2)NC1CN(C(CC#N)=O)CC1O c1(C(=O)NCC2OCCN(C(CCOCCC)=O)C2)cccc2nccnc12 C(CCSC)(C(=O)N(CCCNC(C1(CCF)CCC1)=O)C)OC C1(C(=O)O)C2CC3CC1CC(C1CCN(C(c4n(C(C)C)ncn4)=O)CC1)(C3)C2 C1(NC(C2(CC)CCC(O)CC2)=O)CC2CN(c3nccc(OC)n3)CC2C1 C1(C(N(C)Cc2ccncn2)=O)CCN(C(C2CCCSC2)=O)CC1 C1(N(C(=O)CCC2CC(NC(c3c[nH]c(=N)o3)=O)C2)C)CCCC1(C)O c1(C=O)ccnc(O)c1F.N1(C(C)=O)CCCC1CNC(C1CCC(C)O1)=O C1(O)(CC=O)CCCCC1.C1(CN(C)C(C2COC(C)C2)=O)OCCC1(C)C C1(C(=O)NCC2(NC(=O)CCCC(F)F)CCC2)CC2CCCC(C1)C2(F)F Cc1nc(Cl)ncc1NC(c1ccc(NC(c2cc(Cl)ccc2F)=O)nc1)=O N1(Cc2cc(-c3cc(OC)cc(OC)c3)n[nH]2)CCOc2cccc(C)c21 c1(C=O)cc2c(C)cccc2[nH]1.C1(NC(C(C)OCCOC)=O)CCCCC1.N C1(NC(C2CC(C)(CC)C2)=O)C2CC1CN(C(C1CCCN1C=O)=O)C2.N N1(C(C(C2CC2)OCC)=O)CCCC1C1CCN(C(=O)C(C)O)C1.CC(C)C CCC(F)(F)C(C)(C)C(=O)N1CCC1CNC(c1[nH]nc2ncccc12)=O C12(CNC(CCCOCC)=O)CCC(CC1)CO2.C(=O)(CCC)N.C(C)=O Cc1cccc(-c2noc(-c3cnc[nH]3)n2)c1O C(C(O)C(=O)NCc1nnnn1C)NC(C(C)NC(=O)OC)=O N1(C(c2cnc(CCOC)s2)C(=O)NCCC2CC2)CCCC(CO)CC1 N1(C(C=CC=CCC)=O)CCC2(CCC(NC(=O)C3Cc4ccccc43)C2)C1 N1(C(Cn2ncc(C)c2)=O)CCC(C(=O)NCC(F)(F)C(C)(C)O)C12CCC2 c1(CC(C)C(C)NC(C2CCOC2)CO)ccccc1[N+](=O)[O-] CCC(C)(CC)C(=O)N1CCN(C)C(C(=O)NC(C)Cc2nn[nH]n2)C1 c1(-c2cc(C(N3CCN(C(C)=O)CC3)=O)c(Cl)nc2)ccn2cnnc2c1 c1(CC(N2CCN(C(Cc3scc(C)c3)=O)CC2C)=O)cccc2sccc12 C1(C(N(CC(=O)NCCCN(CC)CC)C)=O)CCCC1C(C)C CC(C)(F)C(C)C.c1(C(=O)NC(C2(C=O)CC2)C)cocc1C(N)=O.N N1(C(C(CC)OC2CCCC2)=O)CC(C)(C)CC1CNC(=O)C.C(C)C.S n1(CC)cnc2nc(=NC3CCCc4ccoc43)[nH]c(NCC3CC(O)C3)c12 c1(SCC(CNC(C2(S(C)(=O)=O)CC2)C)F)cccc(Cl)c1 N1(C(=O)NCc2ccc3ncsc3c2)CCC2CCCc3cccc1c32 C1(C=O)CC(O)C1.C1(CCCC)COC(C(C)(C)C)C1.CC(C)C.C=O.O c1(C(N2CCC(O)(CN(C(C(NOC)=O)=O)C)C2)=O)[nH]nc2ncccc12 CC1=C(C(=O)NCC2(NC(c3cc(C4CCC4)no3)=O)CCOC2)CCCO1 N1(C(c2c(CNC(=O)CC3CCOC3=O)ccs2)=O)CCc2ncncc2C1 c1(CC)nc(C)c(CC(=O)NC2(C)CC(NC(=O)C3=CCCC3)C2)c(C)n1 C1(CN(C(=O)COC2CCCC2)C)CCCCN1C(=O)CC1(CO)CC1 Cc1cccc(OCCC(=O)NC(C)(C)CO)c1.c1(CC(=O)N)c(C)noc1Cl c1(OC)cccc(CCC(=O)NC2CC(NC(=O)CCC(C)SC)C2)n1 N1(C(c2ncc(NC)nc2)=O)CC(NC(C2CCCC2)=O)CC12CCC2 C1(CC(N2C(C)CC(NC(C3CS(=O)(=O)C3)=O)CC2)=O)CCc2ccccc2C1 C12(C(=O)NC3C(CNC(CCc4c(C)ncs4)=O)C3)CCC(C)(CC1)OC2 C(=O)(C(F)(F)C1=CCOCC1)NC1C(C)CN(C(c2nccc(Cl)c2F)=O)C1 C#Cc1cccc(CSC2CCC(CC)C2)c1 N1(C(C(C)SCC)=O)CC2(CCCN(C(c3ccnc(C4CC4)n3)=O)C2)C1 N#Cc1cncc(C(N2CCC(CNC(C3CCCS3(=O)=O)=O)C2)=O)c1 C1(C(N2C(CN(C(C3(COC)CC3)=O)C)CCCC2)=O)CC(C)(C)CN1C n1(CC(N2C(C)CC(NC(c3[nH]cc(C(C)=O)c3)=O)C2)=O)nc(O)ccc1=O C1(C)(CC)CCN(C(=O)CC2N(C(=O)Cc3cnnn3C)CCC2(C)C)CC1 c1(C(=O)NC2CC2NC(c2nnc(O)nc2O)=O)cc(F)c(Br)cc1F C(C)(C)(CCC(=O)NCC1COCC1O)NC(c1c(C#C)c[nH]n1)=O c1(C(=O)NC2CC(CNC(C3CC(C)OCC3)=O)C2)cc2n(n1)CCCO2 C1(C#N)(C(=O)NCC2N(C(CCCC#C)=O)CC2)CC12CCCC2 C1(NC(c2c(O)cccc2F)=O)CCCC(NC(c2nncn2C2CC2)=O)CC1 CC1(C(N2CCC2CNC(=O)C(=O)NCC(F)(F)F)=O)C=CCCC1 C1(C(N2CCC(CN(C(Cc3c(C)n(C)cn3)=O)C)C2)=O)CC(C)CC(=O)N1 C=C(C)CC(C=O)NC(C)=O.n1(CC=O)cnc(C(N)=O)c1.C(C)CO.N c1(SC)cc(C(N2CCOC(CS(C)(=O)=O)C2)C(=O)NCCC#N)n(C)n1 N=c1[nH]nc(C(=O)NC(CNC(C2CC2CF)=O)CO)s1 Cc1ncc(N)cc1C(=O)NC1(C)CC(NC(=O)CCSc2ccccn2)C1 c1(C2(NC(c3nc(C(=O)NC4COCC4O)sc3)=O)COC2)cccc(Cl)c1 c1(C(c2nn[nH]n2)NC(C(c2ccc(Br)cc2)C)=O)cccc(Br)c1 CC(CC(=O)N1CC2(C1)CN(C(c1cnc(-c3ccoc3)s1)=O)C2)C(C)(C)C c1(C(N(CCN(C(C=C(CCC)CCC)=O)C)C)=O)cc(Cl)c(OC)cc1Cl Cc1nc(C)c(C(=O)NC(CNC(=O)CC23CC(C2)C3)C(C)C)nc1C C1(C(=O)N)CCC2CC1CO2.c1(C(N(CCN(C)CCO)C)=O)cc(C)ccn1 c1(OC)cccc(O)c1C(=O)NC1CN(C(c2cscc2C)=O)CC2CC12 C1(CNC(C2CC(F)CN2Cc2ccoc2C(F)(F)F)=O)CCC(O)CC1 N1(C(Cc2cc(C)[nH]n2)=O)CCCC(NC(=O)CC2CCC(C(F)(F)F)O2)C1 C1(C(=O)NCC(CCC)NC(c2c[nH]nc2Cl)=O)CC2CCC2C1 NS(=O)(=O)C1(NC(=O)NCCS(=O)(=O)CCO)CCCC1 N1(C(C(C)SC)=O)CCC2(CC1)CCN(C(C1C3CCN1CC3)=O)CC2 C1(NC(C(C)=C2CC2)=O)CC(NC(C2C(C)C2C)=O)CC1O Cc1ccc(NC(C2(NC(c3ccc(C(C)(C)C)cc3)=O)CC2)=O)c(C)n1 c1(C(=O)NCC(C)N(C(=O)CCc2ccncc2Br)C)cnn2ccccc12 c1(OC)cccc(C(=O)NCC2CN(C(=O)CC(C)n3cccn3)CCO2)c1F C1(CC(C)O)CCCN(C(=O)CN(C(=O)COCc2ccccc2Cl)C)C1 C1(NC(C(C2CCCOC2)N(CCOC(CC)CC)C)=O)CCC(C(=O)OC)C1 C12CN(CCS1)C2=O.c1(CC)conc1CNC(=O)CC1CC(C)=NO1 C(=O)(CCC(=O)NCCC1(C)CCN(C(=O)CCC(C)OC)C1)NCC N1(C(c2c(CC)nnc(C)c2)=O)CCCC2(CCC2)C1.C(=O)(C(F)=C(C)C)N c1(OC)ccc2[nH]nc(N3CC4C(C(=O)NCCN(C(C)CC)C)C4C3)c2c1 CCC(F)(F)C(=O)NCCN(CCOCCO)C(c1[nH]c(C)nc1C)=O Cc1ncoc1C(=O)C(c1c[nH]nn1)O.c1ccoc1.C1CC1.C(=O)O.NC CCC(C)(CO)C(=O)NC(CNC(C1CCN(C)CC1)=O)CO C1(NC(C2CC(OC)C2)=O)CC(N=c2nc(C3CCCC3)[nH]s2)C12CCOCC2 Cc1[nH]cc(C(=O)NC2CN(C(=O)CSc3ccccc3)CCC2C)c(=O)c1Cl N1(C(c2nc(=O)cc(N)[nH]2)=O)C2CCC1CC(NC(c1ccncc1Cl)=O)C2 c1(C(N(CCCN(C(c2cnc(C)s2)=O)C)C)=O)cc2c([nH]1)CCC(C)(C)C2 C1(C2CCCN(C(C3(O)CCCCC3)=O)C2)(NC(C2Cc3nccn3C2)=O)CC1 C1(CCC(=O)OC)CC(C(=O)O)N(C(C2CCC(c3ccccc3)C2)=O)C1 N1(C(C2(F)CN(C(C)=O)C2)=O)CCC(n2cccn2)C1.C(=O)CN(C)CCC C#CCCCCCC(=O)NC(CNC(=O)COCC1CCOCC1)C1CC1 C1(CC(N2CC(C)(C(N)=O)C2)=O)CCN(C(c2n[nH]c3c2COC3)=O)C1(C)C c1(C(N(C)CC2CCN(C(C=C(COC)C)=O)C2)=O)cnn2cccc(OC)c12 Cc1ccc(C(=O)NCC2CCCCN(C(=O)CCN3CCCC3=O)C2)cc1N CCCCCCCCNC(=O)C(=O)NC1CC(C)(NC(=O)CCF)C1 CC(CC(=O)N(CCNC(C1CCOC1c1ccncc1)=O)C1CC1)C1CC1 N1(C(C2(NC(c3ccc(C#C)o3)=O)CCCCC2)=O)CCOC2C(O)CC12 Cc1cc(C(N2CC3CC3(C(=O)NCC3(C4CC4)CCCO3)C2)=O)c(C)o1 C=CC1(C(=O)NC(C)CC2CCC2)CCN(C(=O)COC2CCCC2)CC1 N1(C(C2(OC)CCN(C(=O)C=CC(C)(C)C)C2)=O)C2CCC1CN(C)CC2 C1(C2(O)CN(C(=O)CC(c3ccc(F)cc3)C)C2)CC1.O(C=CC(=O)NC)CC C=CC(O)C(=O)NC1(CNC(c2nccn2C)=O)CCOC1 N1(C(CCc2onc(C)n2)=O)CC=CC(NC(=O)CNS(=O)(=O)C2CC2)C1 C=CCC(C(=O)NC(C)CCC1CC1)NC(=O)CCc1cnccn1 c1(C(N2CCCC(N(C(C(CC(=C)C)C)=O)C)CC2)=O)c(N)sc2c1CCC2 C1(C(=O)NC2CCN(C(C(C)OC)=O)C2C)CC(C2CCCC2)C1 c1(OC)ccc(C(N2CCC(CNC(C3C4(CC4)C34CC4)=O)CC2)=O)cn1 c1(CC(=O)NCC2C(CNC(C3(C)CC=CC3)=O)C2)cc(Br)ccc1F c1(C(=O)NCC2C3N(C(C=CS(C)=O)=O)CC(CC3)C2)cc2c(nc1N)CCC2 C1(N2C(=O)CSC2)CCCN(C(c2ccc(-c3ncco3)cc2)=O)C1 n1(CCCNC(C2CC(N3CCCC3)C2)=O)cc(C2CCC2)nn1 Cc1ncccc1CC(N1CCC(C)(CCNC(C2(C(N)=O)CCC2)=O)C1)=O C(C(=O)NC1CN(C(=O)CCC=CBr)CC1c1cnn(C)c1)(C(C)C)SC CC1=C(C(=O)NCC2CN(C(=O)C(C)(C)C(=O)N(C)C)CCO2)SCCO1 N1(C(CCCC)=O)C(CNC(=O)CC2CC2CC)CC2CCCCC12 CC1CCCCN1CCNC(C12CC1CCN2C(C1CCCN1C)=O)=O CCCC(C#N)C(=O)NCC(C)CNC(=O)CCCOC(C)=O N1(CC)OCC(NC(C2CCCCC2CNC(=O)Cc2cc[nH]c2)=O)C1=O C1(O)(C(N2CC(NC(c3cncc(SCC)n3)=O)C2)=O)CC2CCC1C2.C S(=O)(=O)(c1ccc2sc(C(=O)O)cc2c1)N1C(CC)CCC1 C(=O)(C#CC(C)(C)C)NCC1(CC)CCCCO1.c1(C=O)ccc(N)c(F)n1 CC(CCNC(C1COC1)=O)NC(=O)CCOCC(F)(F)F c1(CC(=O)N)ccc(F)cc1Br.CC(F)(F)C1CC1C(=O)NC1CC1C n1(CCC)ccc(CN(CCNC(=O)C2=C(C)OCC2)CC)cc1=O.CCO CCCC(CC)C(=O)N1CC(O)CC1CNC(=O)C(O)c1ccsc1 C(=O)(C1CCCc2sccc21)N1CCCC(C)C1CNC(c1cnc(C#N)s1)=O c1(-c2onc(C3CCCN(C)C3)n2)cn(C2CCc3cc(Cl)ccc32)nn1 c1(CC(=O)NC2CCCC2CNC(c2ccco2)=O)ccccc1F c1(C(N(CCCNC(C2COCC(C)O2)=O)C2CC2)=O)cn(C)c2ccccc12 C1(C)(NC(C2N(CC)CC2)=O)CN(C(C2CCC(OC)C2)=O)C1 C=C(C)CCCC(=O)NCCC1CCC(NC(=O)C)C1.c1(C=O)ccoc1C.N Cc1ccc2sc(=NC3CCCC(NC(=O)C4=CCCS4)C3)[nH]c2c1 n1(CC(N2CCC(NC(c3c(C)cns3)=O)C2C)=O)cc2ccccc2n1 N1(C(C2(C=C)CC2)=O)CC(NC(C2(C(F)F)CCOCC2)=O)C(n2ccnn2)C1 n1(CC(N2C(CNC(c3ccco3)=O)CCC2)=O)cc(-c2ccco2)cn1.C S(=O)(=O)(c1ccc(Cn2c(C(=O)OC)nnc2)cc1)N(CC)CC c1(C(=O)NC2C(NC(c3c(C)noc3N)=O)CCC2)ccnc2c1CCC2 C1(C(=O)NC(C#C)C(C)C)CCCCC1CNC(=O)C=C1CCC1 C#CCC(CC#C)C(=O)NC1CN(C(=O)CSc2ccc3c(c2)CCC3)CC1C Cc1cc(N)cnc1C(N1CC(C)(C(=O)N(C2CC(C)OC(C)C2)C)C1)=O N(C(=NCCNS(=O)(=O)CC)NC(C)C1CC1)C1CCC(C(=O)NC)CC1 C1(C(=O)OCC)CCCN(CC(=O)N(CC(C)C)Cc2ccc(O)cc2)CC1 N1(C(COCCN(C)C)=O)CCCOC(CNC(=O)COC2CCC2)C1 C(C(CC(=O)N(C1CC(F)(F)C1)C)C1CCC1)NC(c1c(NC)n[nH]c1)=O N1(C(CCCCC(N)=O)=O)CCC(NC(c2coc3c2COC3)=O)C(F)(F)CC1 Cc1cc(-c2nc(C)c(NC(c3cncs3)=O)s2)ccc1[N+](=O)[O-] c1(OC)nc(C(N2CC(OC)CC2C)=O)cc2ccccc12.C(=O)CC1CC1.N c1(CC=O)ccc2nc(O)[nH]c2c1.N1(C(C2C(C(C)C)C2)=O)CCC(C)(C)C1.N c1(N2CCC(CCNC(c3n(C)ncc3)=O)CC2)ncnn2cccc12 C(C(C(C)(C)C)C(N1CCC1)=O)NC(C(C)(C)C)=O.c1(C(=O)N)ccoc1 c1(C(N2CCC(C)C(NC(c3cc(Cl)c[nH]3)=O)C2)=O)ccc2nonc2c1 CCC(CN1CC=CC1)NC(=O)CCSC(=N)N N1(C(c2c(C)snn2)=O)CCCC(O)(CNC(=O)C(c2cnn(C)c2)=O)C1 Cc1ccccc1CC(N1CCC(C)C1CNC(c1ccon1)=O)=O C(CC(C)(C)C(=O)N(CCCCCC(=O)NCCCc1nccs1)C)SC C1(C2(NC(CC=C=C)=O)CC2)CCCCCN1C(=O)C(c1ccccc1)=O c1(C(=O)O)cc2ccc(S(=O)(=O)NCC3(C)C=CCCC3)cc2s1.c1ccccc1 C1(NC(=O)CCc2cccnc2F)CCN(C(C2CCC(O)C2)=O)CC1O c1(C(N2CCN(CC(C)NC(C(C)CC3CC3)=O)CC2)=O)nnc(O)cc1O C1(N(C(=O)CCc2nc(-c3nc[nH]n3)no2)C)CCCN(C(=O)C(O)C2CC2)C1 Cc1cc(F)ccc1C(N1CCC=C(CNC(c2cccc(F)c2)=O)C1)=O C=CCC(C(=C)C)C(=O)N1CC2CC2(C(=O)Nc2ccccc2OC)C1 C1(C(=O)NC(C2(O)CCC2)C)CC(O)CN1C(=O)CCOCC(F)F Cc1cc(F)c(-c2nn[nH]n2)cc1NC(=O)CCc1nc(C2CCOCC2)no1 C1(NC(C(=O)N(C2C3CCCC23)CC=C)=O)CCC(O)C(C)C1 N1(C(C(C)=C(C)C)=O)CCC(C(F)(F)F)CC1.c1(C=O)n[nH]cc1C1CC1.C N1(C(C2(COC)CC=CC2)=O)CCCCC(C)CC1.C(=O)C(O)CC(F)(F)F.N N1(C(COC(CC)C)=O)CCC2CCCC(C1)N2C(c1cc2cscc2s1)=O C12(C(N(C(CC)C(N3CCN(CCO)C(C)C3)=O)C)=O)CC(C)(CCO1)C2 N#CC1(C(=O)NC(C2CCOC2)CNC(C23CCC2CC3)=O)CCCC1 C(=O)(C#CC1CCCCO1)N1CCC(CCNC(C(C(CC)(C)C)=O)=O)CC1 C(N=C(NC(C)C)N1CCC(F)(C#N)C1)c1cncc(OC)n1 N1(C(=O)OC)CC(C(c2nc(C)no2)c2ccccc2)C(C)(C)C1 C1CCCCN1C(=O)C(C)n1ccnc1.N1(CC(=O)NCC)CC(C)(C)C1.C c1(C(CCC)=O)ccccc1C(=O)OC(C)C(=O)OC(C)(C)C CCCCC(O)C(=O)NCC(C)(C)CN(C)C(c1c(Cl)c(CC)nn1C)=O O=C(C1=CCCN(C(=O)CC2CSC2)C1)NC1(C2CC2)CCC1 C1(NC(c2cnc(O)o2)=O)CCC12CCN(C(c1cc3n(n1)CCCC3)=O)CC2 Cn1cc(C(N2CCC2)=O)ccc1=O.c1(CCC(=O)NC2CC2)nc(O)n[nH]1.C C(=O)(CCCCCn1cc(CCC(=O)O)nn1)N(C)Cc1cn(C)nc1C(F)F Cc1sc(C)c(S(=O)(=O)N2CCOC(c3nc(C(C)(C)C)n[nH]3)C2)c1C c1(NC(C2(SC)CN(C(C(CC)SC)=O)C2)=O)ccc2ncnn2c1 C(CS(=O)(=O)Oc1cc(F)ccc1Br)(OCC)OC N1(C(c2c(OC)csc2)=O)CCC(F)(CNC(=O)CC(F)F)C1 C1(NCc2c(C(F)(F)F)nc(C)s2)CCC(O)(C2CC2)CC1 c1(C(N2CC3C(NC(C(C)C4CCC4)=O)C3C2)=O)c(N)sc2ccccc12 c1(CC)ccc(C=CC(=O)NCC2CC(NC(=O)CCS)C2(C)C)o1 C(=O)(C1=CCC(NC(C2CCCC(=O)N2)=O)C1)N(C(C1CCCCC1)C)C N1(C(C2CCN(C(C(CCC)NC(C)=O)=O)C2)=O)CCc2nc(C)nc(O)c2C1 N1(C(CCOCC)=O)CCC(NC(=O)CCOc2cccnc2)C12CC2 N1(C(C(C)C)=O)CCCN(C(=O)CNC=O)C(C(C)(C)C)C1.c1cccc(Cl)c1.O C(=O)(C1Cc2c(Cl)cccc21)NC1CC(C)(C)CN(C(C2(O)CCOC2)=O)C1 Cc1cnnc(O)c1C(N1CCC(C)(NC(c2ncc(F)cc2F)=O)C1)=O N1(c2cc(NCCN(C)C3CC3)ncn2)CCC2(CC(C(F)F)=NO2)C1 C12(C(=O)Nc3cncc(C#C)c3)CCCC1CCN2C(=O)C(=O)NCC(F)F C1(CC(C)C)CCCN(C(C2(NC(c3c[nH]c(=S)cn3)=O)CCC2)=O)C1 CC(C)C(F)(CNC(=O)CCc1ccnn1C)C(=O)N(C)C[Si](C)(C)C CCCCC(CNC(c1cn(-c2cnn(C)c2)cn1)=O)NC(=O)C(C)CO N1(C(C=Cc2nc(C)sc2)=O)C2CCCC1CN(C(=O)CC1(CO)CC1)C2 c1(C(C)C)nnc(C(=O)NCCCC(C)NC(=O)CCc2nc[nH]n2)s1 Cc1nn(CC(=O)NCC2CCN(c3ncnc(=N)[nH]3)C23CC3)c2ncccc12 C1(C2(NC(C(C)OCCC=C)=O)CC2)CCCCN1C(C1(O)CCCC1)=O C1(NC(Cc2nc(C(C)C)sc2)=O)CCN(C(=O)C=CC2CCOCC2)CC1O c1(CN2CC3CN(C(c4cc(OC)cc(C)c4)=O)CC32)ccc(F)c(F)c1F c1(C(=O)NCC(C)OC)cc(C)c2ncccc2c1.c1(C(=O)N)nnc(S)n1C CN(C)S(C)(=O)=Nc1nc(-c2nc(Cc3cccc(F)c3)nn2C2CSC2)cs1 N1(C(=O)COC(F)F)CCC(CC2COCCN2C(c2ncc(F)cn2)=O)CC1 N1(C(CCCCOC)=O)CC2CC(N=c3ccc(C(F)(F)F)n[nH]3)C2C1 C1(CC(N2CC(OCCC(=O)NC(C3(O)CCC3)C)C2)=O)CCCN1C c1(OC)cccc(C(=O)NCc2ocnc2C(=O)NC)c1.c1cnn(C)c1.C C1(C2CCN(C(=O)CNC=O)CC2)(NC(Cc2c(C)cccn2)=O)CC1 c1(C(=O)NCCCN(C(C2(C)CC=CCC2)=O)CCO)ccc(CO)c(F)c1 C1(C(c2nnnn2CCCOC)NCc2nnc(CC)o2)(OC)CCCOC1 C1(OC)CCN(c2cc(NCCN3CCCN(C)CC3)nc(C)n2)CC1C N1(C(c2sncc2Br)=O)CCC(n2cc(C3CCC3C(F)(F)F)nn2)C(O)C1 N1(C(c2cn(CCC=C)nn2)=O)CCC(C)C1CNC(c1sc(C)nc1C)=O c1(CC(CC(=O)O)Nc2cc(C)cc(C)c2)cn(C)c2ccccc12 c1(C(=O)NC2C=CCC(C(=O)NCc3ccccc3)C2)cc2n(n1)CCO2 C1(NC(c2ncoc2C2CCC2)=O)CC2(NC(=O)C(O)C3CC3)COC1C2 C1(C(=O)NC2CC(NC(=O)CSCC(F)F)C2)CCc2nn[nH]c2C1 n1(CCOC)nc(-c2ccsc2)nc1C1CC(F)(F)C1 c1(C(=O)NCCC(C)NC(=O)Cc2ccccc2)cc(C(F)(F)F)ncn1 C=CCC(CNC(=O)CCN(CC)CC)NC(=O)CCC1CC1(F)F C1(C)(C(N(C(C)COC)CCOC)=O)CC2(CCC2)C1 c1(C(c2n(CCSCC)nnn2)N)ncc(Cl)cc1F.c1cccnc1OC N#CC1(C(=O)NC2C3CC(NC(=O)CCc4cscn4)CC23)CCCC1 c1(C(=O)NCC(S(C)(=O)=O)CNC(=O)COC(F)F)occ2c1CCCC2 N1(C(c2cccc(C)c2F)=O)CC2CC1CN(C(=O)CC1CC13CC3)C2 C1(C(=O)OC)CCCC(NC(=O)NC23CCOC(C)(C2)C3)CC1 N1(C(C2C(OC)CN(C(=O)CC(O)CC(C)C)C2)=O)CCc2cc(F)ccc21 CC(CC(C)(C)C)C(=O)N1CCC(C(=O)Nc2cnc(O)c(F)c2)(CO)C1 Cc1c(C(=O)NC(c2ccc(F)c(F)c2)(C)C)nn2c1CCCC2 CC(C)CCCC(=O)NC1CC2CCC1N2C(=O)C(C)(O)Cn1ccccc1=O c1(C(N2C(CN(C(CC3CN(C)C3)=O)C)CCCC2)=O)cncn(C)c1=O c1(C(=O)NCCC)cccc(CNC(N2CCCCC2CCN(C)C)=O)c1 c1(C(N2C3(CNC(C4C(C)OCC4)=O)CCC2CC3)=O)cnc(O)n(C)c1=O C1(CC#N)CN(C(c2ccc(O)cc2)=O)CCN1C(=O)CSc1ccc(F)cc1 C1(CNC(C(C)=CC)=O)CN(C(=O)CCC(=O)NCC)CCO1 N1(C(C(C)(C)OC(C)C)=O)CCC(C2(NC(=O)C#CC3CCOC3)CC2)C1 N1(C(C2CC2(Cl)Cl)=O)CCCC(C(N2CCN(CC=Cc3ccco3)CC2)=O)C1 C1(C(=O)N)Cc2nccnc2C1.C1(COC)(C)CN(C(C2(F)CCCC2)=O)C1 C1(CNC(C(CC)OC)=O)CC2(CC2)CN1C(=O)C(C)(C)CC1CC1 C#CC1(C(=O)Nc2cncn(C)c2=O)CCN(C(C2CC(OC)C2)=O)CC1 C1(OC)CC(CNC(=O)CCCC2OCCO2)N(C(=O)C(=O)N)C1.C1CC1 c1(C(=O)NCC2C(NC(CC#N)=O)CC2)cc(C(N)=O)cc(F)c1 Cc1ncc(C=CC(N2CC(C)C3CC23)=O)s1.C1(C=O)C(C)(C)C1(C)C.N N1(C(C)=O)CCC(C)(CNC(C2CCCN(CC3CCCOC3)C2)=O)C1 c1(C(=O)OC)cnc(=NCCOCC)[nH]c1.C1(C=O)CCN(S(C)(=O)=O)C1 c1(C(N2CCCC2)=O)cc2ccccc2[nH]1.C1(C(=O)NCC(=O)N)CC(CF)C1 N1(C(C(C)CC2CCCC2)=O)CCCC(CC(=O)N(CCCC(O)CO)C)C1 C1(N(C)C(c2cnc(S)nc2)=O)CCCCN(C(=O)CCCC2CCC2)C1 N1(C(c2cc(CC)n(C)n2)=O)CCC(C)(C(=O)NC(CO)CCOC)CC1 Cc1nc2c(s1)CN(C(C1CC3(CC(NC(c4nccs4)=O)C3)C1)=O)C2 Cc1nn(CC(F)F)cc1C(=O)NC(C1(O)CN(C(=O)CC2CCCC2)C1)C CCCCC(C)C(=O)N1CCOC(C(N2CCN(C)C(CC)C2)=O)C1 c1(C(=O)N)ccnc(S)c1.N1(C(C(C)NC(=O)OC)=O)CCC(C(C)C)C1 C(=O)(CC1OCCc2ccccc21)NC1(CC)CCN(C(=O)C(F)F)CC1 C(=O)(CCC)N(C1CC1)C.n1(CC=O)cnc(C#N)n1.n1(CC)nccc1 C1(C=O)CC1C1CCC1.c1(CCCC)cn(Cc2ncoc2C)nn1 C1(C2CC2)(CC)NC(=O)N(CC(=O)NCC(C2CCCCO2)C)C1=O Cc1cc(=NCC2(C)CCCN(C(=O)CCNC(=O)C=CCl)C2)[nH]cc1[N+](=O)[O-] C1(C(=O)OC)CC(C(=O)NCCC(C)N(C(=O)COCC(C)C)C)C1 N1(C(=O)NC(C(=O)OC)C)CCN(C(=O)Cn2ccnn2)CC1.C1CN1 Cc1cn(C)cc1C(=O)NCC1CCOC1C(=O)N.C(C(C)C)c1nc[nH]n1 C#Cc1ccc(C(N2CCC(C(=O)N(C)Cc3cnccn3)(OC)C2)=O)cc1 C=CCCCC(C(=O)NCCSCC=C)NC(C1CCN(C)C1C)=O c1(C(=O)NCC(C2CCC2)NC(C2CC=CCO2)=O)ccnc2c1CCC2 c1(C=O)cnn(CCO)c1C.CCC(C(=O)N(CC)CC)Sc1nc(=N)[nH][nH]1.N c1(OC)ncc(C)cc1.C1(C)(C(=O)N)CCCN1C(C1CC1C(C)(C)C)=O C1CN(C(C2(CC(C)C)CCCC2)=O)CCN1C.C(C)(C(=O)N)OCC(C)C.C Cc1c(C(=O)NC2CN(C(c3ccccc3O)=O)CC2F)cncc1Br c1(C(C)C)cc(C(=O)NC2CCCC2NC(=O)CCCCn2ccnn2)nn1C C1(N(C(C2C(NC(c3cc(C)[nH]c3)=O)CCO2)=O)C)CNC(=O)C12CC2 C1(C=O)CC(C2CC2)=NO1.Cc1cnc(C=CC(=O)N)[nH]1.C1(C)CCCC1.C N1(C(CCOCCOC)=O)CCC2CCCN(C(=O)CC(=O)NC3CC3)C2C1 c1(CNc2c(OC)nccc2)cc2c(s1)CCN(Cc1c(F)cc(O)cc1F)C2 C(C)(CCC(C)C)NC(C1(CC)CCCN1C(=O)Cc1cccc(F)c1)=O CC1CCN(C(C2CC(=O)C2)=O)CC1NC(c1c[nH]nc1-c1ccncc1)=O C1(F)(C(N2CCC(CNC(CCCNC(N)=O)=O)C2)=O)CCCOC1 C1(C(=O)NC2(C3OCCN(C(C=CCC)=O)C3)CC2)CCc2c[nH]nc2C1 C1(NC(C=CCC)=O)CN(C(C2(c3cc[nH]n3)CCOCC2)=O)CC(F)(F)C1 c1(C(=O)N)c[nH]ccc1=O.C=CCCCNC(=O)CCc1ncc(C(C)(C)C)o1 N1(CC2CC(n3c(Cl)cnn3)C2)CCC(Cc2ccccn2)CC1 C12(NC(CC(C)(C)SC)=O)CCCCC1N(C(=O)Cc1cccnc1)CC2 C(N=c1[nH]c(=NCCN2CCCCC2)[nH]c2c(F)cc(F)cc12)C1NC(=O)OC1 Cc1ccc(C(N2CC3CC(C2)C3(C)C)C(=O)NC2CC2)c2c1CCC2 C(CC(C)O)N(C(CN(C(C=CCC)=O)CCOC)=O)C C(CC(F)=C(F)F)NC(=O)CC1C=CC(NC(c2occc2C2CC2)=O)C1 C(CC(C(C)C)(c1nnnn1-c1ccccc1Cl)Nc1ccc(Cl)cc1)OC C=C1CC2(C1)CN(C(=O)CC1(C)CCN1C(C1(C)CCCCO1)=O)C2 c1(SC)ccc(Cl)c(C(=O)N(C2CCN(C(c3ccccc3S)=O)C2)C)c1 c1(C(=O)NCC23C(CN(C(C(C#C)(C)C)=O)C2)C3)coc2c1C(O)CCC2 c1(CC)nn(C)c(C(N2CCC(C#N)(NC(=O)C)C2)=O)c1Cl.c1ncccn1.N C(=O)(C(F)C(C)CC(C)(C)C)N1CCC(CC)(NC(=O)Cn2nccn2)CC1 C=CCCCC(=O)NC(C)(C)CCC1CCN(C(=O)C(C2CC2)SC)CC1 C(=O)(CC(CC(C)C)NC(=O)CC1CCCC1O)NCc1c(C)nccn1 Cc1sc(C(=O)NC2CN(C(=O)CP(C)(C)=O)CC2F)cc1[N+](=O)[O-] c1(OCCCC)ccc(C=O)cn1.N1(CC(=O)N(CC(C)C)C)CCC(C)C1 c1(NC(CC2CC3(CN(C(C4CCC4)=O)C3)C2)=O)ccc2ccc(O)cc2c1 N1(CCCCC)C(=S)NC(c2c(Br)cc([N+](=O)[O-])cc2Br)C2=C1CC(C)NC2=O N1(C(c2cnc(CCC)s2)=O)CCN(C(C23CCC(CC2O)C3)=O)CC(C)(C)C1 CC1CCCC(C(=O)NC(C)CCNC(c2ccc(-n3ccnc3)nc2)=O)O1 N1(C(CCOCC#C)=O)CC2CS(=O)(=O)CC2(NC(c2sccc2F)=O)C1 N1(C(C(F)=CCNC(C2(CC#C)CCC2)=O)=O)CC2(CO)CCC1CC2 C1(C)(CC(N2C(CC(=O)NC)CC2)=O)CN(C(c2cc[nH]c2)=O)C1 CCCCCCC(C)C(=O)N1CCCC(CN(C(=O)CS(=O)(=O)CCO)C)C1 C1(NC(CC2N(C(C)=O)CCC2)=O)CC12CC(NC(c1cc(C)nn1C)=O)C2 Cc1csc(C=CC(=O)NCCCC(C)NC(c2coc(C3CCC3)n2)=O)n1 c1(C(=O)NC2(CC=C)CCN(C(c3cccc(F)c3F)=O)C2)csc2nccn12 C1(NC(c2c(C)n(C)cn2)=O)CCC(C)N(CC(=O)NC=O)C1.C(C)(C)C.N C12(NC(C3CC(CC)OCC3)=O)CCCC1N(C(c1ncsc1C)=O)CC2 S1(=O)(=O)c2ccc(cc2)N1.N1(C(C)C(N2CCOCC2)=O)CC(C)N(C)C(C)C1 N1(C(c2cnco2)=O)CCC(C2(O)CCN(C(c3sccc3F)=O)C2)CC1 c1(C(N(CCCN(C(=O)CSC2CCCCO2)C)C)=O)cnn(C)c1N C1(CNC(c2cc(C)c(F)cn2)=O)C2CCCC1N(C(c1ncccc1Cl)=O)C2 c1(C(=O)NC2C(NC(CCCCOCC)=O)CC2)cnc2ncnc(O)c2c1 CCCCCC(=O)N1CCCC(CNC(C2(C(F)(F)F)CCCCC2)=O)C1 c1(C(=O)N)ccc(C2CC2)nc1.C(=O)(C(F)(F)c1nccn1C)N1CC(CC)C1 c1(CC)nc(C)oc1C(N1CCC(C)(C(=O)NC2(CC)CCOC2)C1)=O CC(C)C(C(=O)N1CC2CC2C1)NC(=O)C(F)(F)F.C1(CC=O)CC(F)C1 CC(C(C)C(=O)N(C)CCN(C)CCO)NC(=O)C(O)Cn1cncn1 C12(C(N3CC4C(CC(=O)N(C(CC)CC)CC)C4C3)=O)CC(C)(CCO1)C2 CC(C)C(Cc1ccccc1)C(=O)NCC(O)C.c1(C(=O)N)cnoc1C1CC1 N1(C(CCNS(CC)(=O)=O)=O)CCCN(C(c2sc3ccsc3c2C)=O)CCC1 Cc1ccc(CC(=O)NCCOCCN(C)C(C2CC3(CCC3)C2)=O)cc1C C(=O)(CC(O)CN(C)C)NC1(CCC(=O)NC2C(OCC)C2)CCC1 C1(CNCC(CC)NC(=O)OC(C)(C)C)CCC(S(C)(=O)=O)CC1 C1(N(C)C)CCc2ccccc2C1NC(N1CCC(Cc2cccnc2)CC1)=O NC(=O)C(F)(F)CNC(C1CN(C(=O)CN2CC3CC3C2)CCO1)=O CC1(CNC(=O)C(N2CCCC(COC(F)F)C2)=O)CS(=O)(=O)CCO1 N1(C(c2ccc(COC)[nH]2)=O)CCCCC1C.C1(CC(=O)N)CCC(C)(C)CC1 Cc1ccc(F)cc1NC(=O)C(=O)NC1CN(Cc2cnc(Cl)s2)CC1O Cc1n[nH]c(C)c1C(c1nnnn1C)Nc1ccc(-c2nc(=O)o[nH]2)cc1 C1(C(N2CCC(COC)(C)C2)=O)CCC(C)=C(C)C1.C(=O)CC(C)(F)F.N Cc1nn(C)cc1CCC(=O)N1CC(NC(C2CCN(CCF)CC2)=O)C1 c1(NCC2CC(OC)C2)cc(=NCC2(C)CCC(=O)N2C)[nH]c(C(C)C)n1 N1(c2cc(CC)ncn2)CC(NC(=O)CCc2nc(O)n[nH]2)C2CCCCC12 N1(C(C(C2CCN(C(C3N(C)C(=O)CCC3)=O)C2)(C)C)=O)CC2COCC2(C)C1 c1(C(N(CC(O)CNC(C2CC2CF)=O)C)=O)cncc(-c2ccccc2F)c1 C1(CC(=O)N(CC(C)CNC(=O)COCC(F)F)C)CSCCS1 O(NC(=O)C(F)C1CCN(C(c2occc2C)=O)C1)CC=C c1(OC)cc(C(N2CC3CC2C3NC(c2cocc2C)=O)=O)cc(Br)c1O C1(NC(C(C2CCC2)NC(C)=O)=O)CCN(C(c2snnc2C)=O)CC(O)C1 C(=O)(C(C(C)CC)NC(c1nccnc1C)=O)NCc1c(CC)nn[nH]1 c1(OC)ccc(C(C)C(=O)NC(C)C(C(C)C)Nc2ncc(Cl)cn2)cc1F C(=O)(C(CC(C)CC)NC(c1nccnc1C)=O)NCCN(CCCC)C CC1CCCC1(C)C(=O)NCCCCCNC(c1cc(C2CC2)on1)=O C1(C)(N(C)C)CCN(C(=O)C(C2CCOC2)NC(C2(O)CCCCCC2)=O)CC1 N1(C(C(N2C(c3nnc(C)o3)CCC2)=O)=O)CCCc2c1cccc2S(C)(=O)=O N1(C(c2ccc(C3CC3)cc2)C(=O)NC)CC2(CCCC2)CC1C(=O)OC c1(OC)cc(C)cc(CN2CCCC(C)(C(=O)Nc3cc(O)ccn3)C2)c1O c1(NC(C)=O)ccc(C(=O)N)cc1.c1ccc(C(N2CCC(=O)CC2)=O)cn1.C CC1COC2(CCC2)CN1C(=O)CC1(C)CCN1C(c1cc(C#N)ccc1N)=O Cc1cc(C(N2CCOCC2CC(=O)Nc2nc(Cl)ccc2O)=O)ccc1Br C1(C(N(C)CCn2cccn2)=O)CCC=CC1NC(c1csc(Cl)n1)=O c1(C(=O)NC(C(C)(C)NC(CC2(NC(C)=O)CC2)=O)C)cn(C)nc1C N1(C(c2cnc(C)nc2)=O)CC(NC(C23CCCCC2C3(F)F)=O)CC(C)(C)C1 C(=O)(C(CC)CC(F)F)NC1CC(CNC(C(C2CCCC2)OCC)=O)C1 C1(C(=O)Nc2cnoc2)C=CCN1C(c1cnc(O)[nH]1)=O C1(CC(=O)NCC2C(NC(CCc3ccn(C)n3)=O)CCC2)CN2CCC1CC2 Cc1ccc2c(c1)C(C(=O)NC1CCC1NC(c1ccc(SC(F)F)cc1)=O)C2 C1(NC(CCN(CC=C)C(C2CCCN2C)=O)=O)CCCCC1C c1(CCCN(C(C)C(N2CCOCC2)=O)C)nc(Cc2ccccc2)cc(O)n1 N1(C(C(n2cc(-c3cccc(C(=O)OCC)c3)nn2)C)=O)CCC2CCCC12 CCC(C(=O)NCCC1CN(C(c2cc(C)ccc2OC)=O)C1)C(C)(F)F N1(C(CC2CC(=O)C2)=O)CCN(C(c2cc(C3CC3)ccc2Cl)=O)C2(CCC2)C1 c1cc(O)ncc1C=O.C1(C2CC2)(CC(N2CCC2)=O)CC1.C(C)(C)C.N Cc1cccc(C(O)C(N2CCC(O)(CNC(=O)CC3CSC3)C2)=O)c1F CCC(C)(F)C(=O)NCCCNC(=O)CCC(=O)OC(C)(C)C Cc1ccc(Cl)cc1C(N1CC(=C(F)CNC(C23CCCCC2C3)=O)C1)=O C(CCCCC(=O)NCCCNC(C1CC(O)(C(F)F)C1)=O)NC(C)=O C1(CC)(NC(=O)Cc2ccn(C)c2)CCN(C(C2CC(C)(F)C2)=O)CC1 CC(C)C(C(=O)N)NC(=O)C(F)(F)F.C1(C(N2CCCC2)=O)CCC(=O)NC1 C(CC(C)C(=O)NC1CC(C(F)F)C1)=CC.c1(CC(=O)N)ccc(F)nc1 C1(C(=O)NCC2CCN(C(=O)COC3CCOCC3)C2)COC2CCCCC12 N1(C(CCC2(O)CCN(C(CCCC#C)=O)CC2)=O)CCC(C)(C)C(CO)C1 C(CC(O)C(=O)N1CCC(C)(C(=O)N(CCC(C)(C)O)C)C1)N(C)C CCC(CC)C(F)C(=O)NCC(CC(N1CC2CCC(OC)C2C1)=O)OC CC1(C)CC(NC(C2CCSCC2)=O)CN(C(=O)Cn2cccc(N)c2=O)C1 c1(C(N2CC(C(=O)NCC)C2)=O)n[nH]c2cc(Cl)ccc12.C(CC=O)OCC C1(CC(c2cncnc2)=O)COCCN1C(=O)Nc1cccc(N2CCCC2)n1 C1(N(C(N2CCN(C3CCC3)CC2)=O)CC2CC2Br)CCC=CCCC1 c1(C(=O)NCCC2CCC(NC(C3CCOCC3)=O)C2)cnc2c(Cl)cccn12 Cn1cncc(C(N2CCCC(F)(CNC(C3(C4CCCO4)CC3)=O)C2)=O)c1=O C1(C(NOCC(=C)C)=O)CC(F)CN1C(c1ccsc1C#N)=O c1(N(CC#C)C)ccc(C(=O)N(C)C(C2CCCC(OC)C2)=O)cc1 C1(C)(C=O)CCC2(CC1)CC2.c1(C=O)ccc(C(F)F)nc1.C(C)(C)OC.N c1(C(=O)NCCC2CCN(C(C3N(CC)CCC3)=O)CC2)ccc(F)c(Cl)c1N c1(C(N2CCC(NC(c3c(C)cco3)=O)C2C)=O)ccc(CO)c(Cl)c1 C=C(Cl)CCC(=O)N1CC(CNC(=O)Cc2cncn2C)C(C)C1 C1(CNC(C(C)C)=O)CCN(C(=O)CC2CNC(=O)C2)CC1CO CC1(C)OCC(n2cc(C(c3ccc(Br)cc3Br)O)nn2)C(c2ccccc2)O1 CC1(C)OCCOC1CC(=O)NCC(CO)NC(c1cscc1C(F)F)=O C(=O)(C1COc2ccc(F)cc21)NC1CC(NC(c2cnn(CC)c2C)=O)C1 C(C(O)C(=O)N1CC(OCCC(=O)NCCSC(C)C)C1)=CC C1(C2CN(C(=O)CC3(C)CC3)C2)(NC(C(C)Oc2cccc(F)c2)=O)CC1 c1(SC)ccc(O)c(C(=O)N)c1.C1C(C)CCCN1C(C1CC(C(C)C)C1)=O CC1CN(C(C2C(F)(F)C23CC3)=O)CCN1C(=O)Cc1c(F)cccc1F C1(CNC(c2nc(Cl)c(Cl)s2)=O)CC(F)(F)CN1C(c1cncc(Cl)c1)=O N1(C(C(C)O)=O)CCC(C)(NC(c2cnc(-c3ccccc3)o2)=O)CC1 N1(C(CN(C2CCSC2)C)=O)CCCCCC(NC(c2cccc(=O)n2C)=O)C1 N1(C(Cc2c(CC)cccc2)=O)CC(CNC(=O)CC(C)OC)C2(CCC2)C1 c1(CC(N2C(C)CC2C(=O)NC2(CO)CC(F)C2)=O)ccc(C#N)cc1 N1(C(c2c(CC)noc2)=O)CC2CN(C(=O)C(F)(F)C(O)CC)CC(C1)O2 Cc1c(NC(c2scnc2C2CCCC2)c2nnnn2C)cccc1N(C)C N1(C(CC2CCC(C)CO2)=O)CCN(C(=O)CN(c2cnccn2)C)C(CO)C1 C#CCCCCCC(=O)NC(C)(CNC(C1(C)CC=CCO1)=O)CC(C)C N1(C(C(C=C)(F)F)=O)CCN(C(C2CC2c2c(Cl)cccc2Cl)=O)C(CC)C1 C(=O)(C1CCc2nccn21)NCC1CCCN(C(c2cc(C)on2)=O)CC1 C1(CN(C(=O)NC2COC(C)C2C)C2CC2)CC2CC1CC2N.c1ccccc1 N1(Cc2nc(C)oc2)CC2(CC2)CC1C(=O)NC(CO)C(C)C c1(C(=O)NC2CCC23CN(C(c2cnns2)=O)C3)ccc2nn(C(F)F)cc2c1 C1(CC(=O)NCCc2c(C)ncs2)CCCN(C(c2ncoc2C(C)C)=O)C1 CC1(C)COC(CNC(=O)C(=O)NCC(c2ccc(Cl)cc2)(C)C)CO1 C(C(CO)NC(=O)CCNC(=O)Nc1ccsc1)NC(C=CCCC)=O C1(C(N2C(CC(=O)NCC(CC)OCC)CC2)=O)C2CC3C(C2)C13 C=CCC(C)(C)C(=O)NCCOCCCNC(c1ccc(NC)cn1)=O N1(C(c2cc(Br)c[nH]2)=O)CCN(Cc2cccc(O)c2F)CC1C(F)(F)F N1(C(=O)Cn2ccc3ccc(Br)cc23)CCCc2ccc(F)c(F)c21 c1(OCC(=O)NCCCC(C)NC(Cc2c(C)nc[nH]2)=O)ccc(F)cc1 c1(C(N2CCC(COC)(NC(=O)CCC(C)OC)CC2)=O)cc2n(n1)CCCN2 C1(NC(c2c(C)n(C)nc2)=O)CCC2(CCN(C(C3CCCCCN3C)=O)C2)C1 C(=O)(CCCCCCS(N)(=O)=O)NCCCNC(C(C(CC)CC)C)=O c1(C(N2CC(O)(C(C(=O)NC(CC)CO)F)C2)=O)c(C)nsc1N CC(CC(=O)N1CCC(C)(CNC(=O)C(c2ccccc2)=O)C1)C(F)F C(CN=c1nc(C)c([N+](=O)[O-])c[nH]1)C1CCN(C(CCc2cc(C)[nH]n2)=O)C1 c1(C(=O)NC23C(CN(C(Cc4scc(C)c4)=O)C2)C3)c[nH]c2cccc(C#N)c12 C1(CNC(=O)C(F)n2ccnc2)(NC(C2(c3ccno3)CC2)=O)CCCC1 c1(C(=O)NCC(C)(CO)NC(C(C)OCC=C)=O)cc2cnn(C)c2s1 n1(CC=C)ncc2c(O)nc(=NCC(C3CC3)NC(c3cnc(C)n3C)=O)[nH]c12 N1(C(C=COCC)=O)CCCC(C(C)NC(C2(O)CCCCC2)=O)C1 CC(CC(=O)NCCNC(=O)CCN1CCN(C)CC1)C(F)(F)F.C1CC1.C C=C(C)C(O)CC(=O)NC1(CNC(C2(O)CCCCCC2)=O)CCOC1 c1(OC)c(C(N2CCC(NC(=O)C(C)SC)C(C)(C)C2)=O)cccc1[N+](=O)[O-] N1(C(CC(C)n2cccn2)=O)CCCC(O)(CNC(=O)C=Cc2ccco2)CC1 N1(C(C23CC(C)C2C3)=O)CCC(O)C1.c1(C=O)cn(C)nc1-c1cnn(C)c1.N C1(C#N)(C(N(CCNC(C23COC(C2)C3)=O)CC)=O)CC2CC2C1.C C1(C2CC2)(C(=O)NCC2(CCC)CC2)CN(C(c2cscc2OC)=O)C1 c1(CN2CCC(c3cccc(CC)c3)(F)C2)cccc2nc(O)oc12 c1(CC(=O)N(C)CCNC(C2CC23CCCC3)=O)ccc(O)cc1Cl c1(OC)ccc([N+](=O)[O-])c(C=O)c1.C12(CC=O)CCC(C)(C1)OC2.C1CC1 c1(C(N2CC3CC3(C(F)(F)F)C2)C(=O)NCC=C)nc(Cl)ccc1Br c1(COC)nc(C)ncc1C(=O)NCC(C)CO.c1(C=O)cc2occc2[nH]1.N C1(CC(C)C)(C(N(CCNC(Cc2nc(C)oc2)=O)C2CC2)=O)CCNC1=O N1(c2nc(=N)nc(N(CCCOCC)C)[nH]2)CCOC2(CCSC2)C1 CC1(C)CCC(=CC(=O)NC2CC3CC(NC(c4ccncc4Cl)=O)CC23)CC1 C1(CC)COCCN(C(=O)C(CC2CC2)NC(=O)Cn2cccc2)C1 C(=O)(CC1CN(C(=O)C=C(C)C2CC2)C1)NCC1C(CCC)C1.O CCC(CC(=O)NCC1CCN1C(c1ccc(Br)c(F)c1N)=O)C(C)C c1(CC(N2CCCCC(N(C(C=COCC)=O)C)C2)=O)c[nH]c2ccc(O)cc12 Cc1cn(C)cc1C(=O)NCC1(CC(=O)NCC2CC2Cl)CC1 c1(C(=O)NCC(CC)NC(C2(c3ccccc3Cl)CCC2)=O)cc(C)nc(O)c1 N1(C(C(C)O)=O)CC2(CC(NC(=O)Cc3cnn(C)c3)c3nccn32)C1 CC1=C(C)CC(C(N2CCCC(NC(c3cn(C)cn3)=O)C2)=O)CC1.C1CC1.C c1(-n2c(C)cc(C=O)n2)ccc(C)c(F)c1.C(C)(C(=O)N)OCC=C.CCC CC1CCCN1C(=O)CCC1CCN(C(c2cccn2C)=O)C1 Cn1ncc(C(N2CCC(NC(C3CCCCC3C(N)=O)=O)CC2)=O)c1C(F)F C1(NC(c2[nH]nnc2C2CC2)=O)CCCC12CN(C(=O)C=Cc1nccs1)C2 C1(=CCNC(c2coc(Cl)n2)=O)CCN(C(=O)Cc2ccncc2)CC1 N1(C(C2C(CNC(C(C)(C)C3CCCC3)=O)OCC2)=O)CC2OCCOC2C1 C1(CS(C)(=O)=O)CCN(CC(=O)Nc2cn(C3CCCCC3)nn2)CC1 C#CCC(C)(C(=O)NC1CC1C1CCCC1)NC(c1cnnc(C)c1)=O N1(C(C(C)C2(O)CCC2)=O)CC2CCCC(C1)N2C(c1cc2occc2n1C)=O Cc1nc(NCc2ccncc2)cc(NC2CCC(C3CC3)C2)n1 CC1CCCC(CC(=O)NCC(O)C(=O)NC2CC(=C3CC3)C2)O1 C(=O)(CC1=CCN(C(=O)C=C(C)C)CC1)NCC=C C1(CCC(N2CC(NC(C(CC)=CCCC)=O)C2)=O)CC2CCC1C2 N1(C(CCC)=O)CC(CNC(C2(c3cccnc3)CCC2)=O)C2(CCOCC2)C1 N1(CC(N2CC(N(C(=O)C(C)(C)CF)C)C(F)C2)=O)CCCCS1(=O)=O c1(C(CC(=O)NCC2C(NC(CC3(OC)CCC3)=O)C2)C)ccccc1F c1(NC(C2CC(NC(Cc3ccc(OC)cc3)=O)C2)=O)c[nH]c2ncccc12 C1(CC2(NC(C3C(CNC(=O)C)OCC3)=O)CC2)CCSCC1 S(=O)(=O)(c1ccc(=NCc2ccsc2Cl)[nH]c1)N1CC(CC)OC(C)C1 CCC(CC(=O)NC1CC2(C1)CC2)C1CCC1.c1(CCC=O)nc(C)c(C)o1.N C12(C(N3CCN(C(=O)COCCCF)C(CO)C3)=O)CCCCC1NC(=O)C2 C(CCC(C)(C)NC(=O)C(c1cccc(F)c1)F)NC(C1C(C)C1)=O N1(C(CC2CC(C)(C)OC2)=O)CCC2(CCN(C(=O)C=CC(N)=O)C2)C1 C1(C(=O)NC(C(=O)NCC)C)CCC(C)(C)C1.C1(C(=O)N)CCCCC1 N1(C(COCCC)=O)CC(C)OC2(CCN(C(c3ccc(C(N)=O)cc3)=O)C2)C1 CCCCC(O)CC(=O)N1CCC(C(F)C(N2CCC(CC3CC3)CC2)=O)C1 C(CCC(=O)N1CC=CC1CNC(c1cscc1Br)=O)OC(C)(C)C Cc1oc(C#N)cc1C(N1CC(NC(c2ccc(-c3ccccc3)nc2)=O)C1)=O c1(C=O)ccc2c(c1)CCC2.C(=O)(C(C)S(C)(=O)=O)N1CC(COC)C1.N CCC(=O)CCC(=O)N1CC(C(=O)NCc2ccc(F)cc2F)CC(C)C1 c1(SCCNC(NCCC(=C)C)=NC)ccc(C(=O)OC(C)(C)C)cn1 c1(C(=O)NC(CN(C(C2CCC(O)C2)=O)CC)C)cccc2c1OCC2(C)C c1(OC)cc(C(N2CCC(CF)(NC(c3nn(C)cc3Cl)=O)C2)=O)cc(OC)n1 C1(N(C(C=CCN(C)C(c2ccoc2)=O)=O)C)CCCC(O)C1 CCC(O)CC(=O)NCCC1(C(=O)NC(c2nccs2)C)CCCC1 C12(NC(N(C(CO)SC)C)=O)CC(NC(=O)OC(C)(C)C)(C1)C2 c1(NC)ccc(C(=O)N(CCNC(=O)CC2CCCC2C)C2CC2)cc1 N1(C(C2(CCC)CC2)=O)CC2CCN(C(=O)CCc3ccnn3C)C(C2)C1 C1(CNC(=O)CS(=O)(=O)C2CC2)COCC2(CCN(C(c3cocn3)=O)C2)O1 CCC(C)CCCC(=O)NCCN(C(C1CC(=O)N(C(CC)CC)C1)=O)C(C)C c1(CC(=O)N(C2CN(C(c3sccc3Cl)=O)CC2O)C)ccc2c(c1)CCCO2 N1(C(C)=O)CCOC(C(N2CC(NC(=O)CS(N)(=O)=O)C(C)C2)=O)C1 C(=O)(C1=CC2(CCOCC2)C1)NCC1CN(C(C2C(C)C2)=O)C(C)(C)C1 c1(C(=O)NC2(CC=C)CCN(C(=O)CCF)C2)ccc2c(c1)CCOC2(C)C Cc1ccc(OCc2cn(CCC(=O)NCC3(C4CCCCO4)CC3)nn2)cc1 n1(CC)ncc(C(=O)NC(C)CC2CN(C(=O)C(C3CCC3)OC)C2)n1 N1(C(C(C)=C(C)C)=O)CCC2(CC1)CC2.c1(C=O)sccc1S(=O)(=O)N(C)C N1(C(CC2(C=C)CCC2)=O)CC(NC(=O)CC2CCC(C)(C)O2)C2(CC2)C1 c1ccccc1.C(C=O)OCC.C1(CC(N)=O)(N(C)C=O)CC1.C(C)(C)C c1(C(=O)NCC(=O)NCCC(C)NC(c2nnn(C)n2)=O)cnn(C)c1 C=CCCCCCC(=O)NC(Cc1cn[nH]c1)C(=O)N(C)C(C1CCOCC1)C N1(C(C(C)(C)C2CCCN2C(C2CCCSC2)=O)=O)Cc2c[nH]nc2C1 CC1C(NC(=O)Cn2nnc(=O)[nH]2)CCCN1C(=O)Cn1cnc(Br)c1 C(=O)(N1CC2COCC2O1)C1CN(C(c2c(COC)cc[nH]2)=O)CC12CC2 C1(NC(Cc2cc(C)c(F)cc2)=O)CC2CCC(C1)N2C(C12CC(C1)C(C)O2)=O C(C)(CCF)C(=O)O.c12ccccc1-n1cc(nn1)C1CCN1C(=O)CC2.CC CN1CCC(c2nc(CC(=O)NC3CCOCC3)no2)C1=O C1(C(=O)NCC(C)NC(c2ccn(C3CCC3)n2)=O)(C(F)F)CCCC1 c1(CC)cc(C(=O)NCC2C=CCN2C(=O)CSC(F)F)ncn1 c1(C(=O)NCC(CC)NC(=O)C)cc(Cl)c(C)cn1.c1(C=O)ccncc1.N c1(CCCC(=O)Nc2nc3ccccc3s2)ccc(O)c2ccccc12 C(=O)(CC(C(F)F)c1ccccc1)N1CC(O)C1.CC1CC(C#N)(C(=O)NC)C1 O=C(CC(CC1CC1)NC(c1cnoc1C1CC1)=O)NCCN1CCC1 c1(C(N2CC=CC(NC(c3c(OCC)cncc3)=O)C2)=O)c(C)nn(C)c1N C(=O)(N=c1[nH]n(C)c2ncc(I)cc12)Nc1nc(F)cc(C)n1 C(=O)(C(CNC(C1(C)CSC1)=O)CC1CC1)N1C(C)CC1CO Cc1cc(O)c(C(C)C)cc1C(N1CCCC1C)=O.C(=O)C(F)CC1CC1.N c1(CC(=O)NC2CCCCC2CNC(C2(CCF)CC2)=O)ncn2c1COCC2 C(=O)C(F)(F)C(F)(F)F.C1(CN(C(c2ccn(CC)n2)=O)C)CCCCC1.N C1(O)(C(C)NC(c2cnc(C)[nH]2)=O)CCN(C(C2CCCS2(=O)=O)=O)CC1 N1(C(C(CC=CC)NC(C2CN(C)C2)=O)=O)CCC2C(C(N)=O)C2C1 C=C(C)CCCC(=O)N1CCN(C(C2(F)CCOC2)=O)C(C2CCCC2)C1 c1(C(=O)NC2(CNc3ncc4ccsc4n3)COC2)cccc2ccncc12 N(C1CCc2cccnc21)C(c1ccc(S(C)(=O)=O)cn1)c1n(CC=C)nnn1 C(=O)(CC(C)P(C)(C)=O)NC(CN(C(C=CC(CC)C)=O)C)(C)C Cc1ccc(CCCC(=O)NC2CCC(CNC(C3(CF)CCC3)=O)C2)cc1C C1(C(N(C2CCOC2)C)=O)C2CC3C(C2NC(=O)CC2CCOC2(C)C)C13 C1(C(=O)NCC2COCCN(C(C(CO)NC(N)=O)=O)C2)CCOC2(CCC2)C1 N1(C(C2CCC(C#C)CC2)=O)CCc2c(C(C)C)ncnc21 CC(CS(C)=O)C(=O)NCC1CC1.c1(C=O)cn(CCN2CCCC2)nn1.C c1(C(=O)NC2CN(Cc3ccc(OC(F)F)c(O)c3)C2)nc2ccccc2[nH]1 C1(COC)CCN(C(=O)C=C2CCC2)C1.c1(C=O)ccc(C(F)F)cn1.C C1(OC)CCN(C(=O)C(N2CCOCC2)C2CC2)C1.C(=O)C=C1CCC1.C Cc1ccc2cc(C(N3CCC(N(C(=O)Cc4cn(C)nn4)C)C3)=O)[nH]c2c1 c1(CN(C(=O)N(c2ccc(F)cc2)C)Cc2nccc(C)c2)cc(Br)cc(Br)c1 c1(C(N2CCNCC2C2CC2)=O)cn2cccc(Br)c2n1 S(=O)(=O)(c1cccc(N2CCC(C)C2)n1)NCc1c(OCCC)nccc1 CCCCC(C)C(=O)NC(C)(CNC(c1cc(C)nc(O)c1)=O)C1CC1 N1(C(C=C(C)C(F)F)=O)CC2C(CC(=O)NCc3nncn3C(C)C)C2C1 Cc1ncc(NC(c2nnnn2C2CCOC2)C2CC2n2cccn2)n1C(F)F C1(NC(C(CC#C)C)=O)CC2(C1)CN(C(c1cc(-c3ccccc3)co1)=O)C2 C1(CNC(c2c(CNC(=O)Cc3cncnc3)nccc2)=O)CCC(O)CC1 N1(C(C2(COC)CC=CC2)=O)CCCC(C)C1.C1(CC=O)CCCCC1(F)F.N C(=O)(CCCC(C)C)N1CCCC(CC(=O)NCc2[nH]nc(C(C)C)n2)C1 N1(C(C=CC(C)(C)C)=O)CCOCC1CC(N1CCN(CC(F)(F)F)CC1)=O N1(C(c2snc(C)c2N)=O)CCC(O)(CNC(C2CCCCC2C)=O)CC1 N1(C(c2n(C)nnc2)=O)CC(N(C)C)C(CNC(=O)Cc2ccon2)C1 C1(C(C)C(=O)NCC2CCO2)CCN(c2ncncc2F)CC1 c1(NC(COCc2nnc(C)s2)=O)cc2occc2[nH]1.C1(C=O)CC1(C)C.C C=CCCCCCCNC(=O)CC1CCN(C(c2cocn2)=O)CC1 c1(C(N2CCCCC2)=O)c(S(C)(=O)=O)cnn1C.c1(CC)nc(C)c(C=O)s1.N CC(C)C(CN(C)C)C(=O)N(C(C)C(N1CC(C)(O)C1)=O)C c1(OC(C)(C)C(N2CCCC(NC(=O)C3=CCOC3)C2)=O)ccc(C(N)=O)cc1 C1(OC)CCN(C(c2ccc(N(C)C)nn2)=O)C1.C(=O)C(C)=CC(C)(C)C.C C=CCC(C)(C)CCNC(=O)C1=CCC(NC(=O)CC2(OCC)CC2)C1 C1(COC)CN(C(C2COCC2NC(=O)CC(C)n2cccn2)=O)CCO1 C(CC)(CC(=O)NCC(F)(F)CC)NC(C(=O)NCC)=O C1(NC(=O)NCCC(C)C)CN(C(C2CC3C=CC2C3)=O)CCO1 C1(C(=O)NC2C(CC=C)CCC2)CCN(C(=O)CC2CCCO2)C(C)C1 c1(C=O)ccc(-n2cncn2)cc1.O=C(CCCC1CC1)NCC1CC1C.N C(=O)(C(F)C(C)CNC(c1sccc1F)=O)NCCCN(CC(C)C)C C1(C(N2CCC(NC(CCN(CC)CC)=O)C2C2CC2)=O)COCCC1(F)F N1(C(C=C(C)C2CC2)=O)CCN(C(=O)C=Cc2cnn(C)c2C)CC(C)(F)C1 C1(C(=O)OC)C2C=CC(C2)C1Nc1ncccc1Cl n1(CCOC)nnnc1C(C1COCC1c1ccccc1)NCC.C(N)(=O)N C(=O)(CC(C)(C)C(F)(F)F)NC1C(SC)CN(C(c2cc(F)ncc2C)=O)C1 C1(CC=C)(NC(=O)CCc2ccnc(C)n2)CCCN(CC2CCC3CC3C2)C1 C1(NC(C(CC)SC)=O)COCCN(C(=O)C(C)(C)CN(C)C)C1 C1(CNC(=O)C(C2CCCCC2)O)C2CC1N(C(C1CCCS1(=O)=O)=O)C2 C(=O)C(O)P(C)(C)=O.c1(C(=O)OC)cccc(CC(=O)N(C(C)CC)C)c1.N c1(C(N2CC(NC(Cc3cc(C)sc3C)=O)C(C)CC2)=O)cc2n(n1)CCCC2 C1(NC(C(CCC)C)=O)CCS(=O)(=O)C12CN(C(c1cccc3c1CCC3)=O)C2 C1(O)(CC(=O)N(CC(C)CNC(=O)C(C)O)C)CCCCCC1.C1CCCO1 CCC(C(=O)N1CCCC(Cn2cc(-c3ccc(F)cc3)nn2)C1)C(F)(F)F N1(C(CCCC)C(=O)NCCCSCC)CCSC2CCCCC12 c1(OC)cccc(Cl)c1CN1CCC(CNC(c2cccc(C)c2Cl)=O)C1 c1(C(N(CCCNC(c2cnn(C)c2C#N)=O)CCO)=O)sc([N+](=O)[O-])cc1Cl C12(Sc3nccc(C(=O)NCCCN4CCCC4)c3)CCCC1CS(=O)(=O)C2 N1(C(C=C(C)Cl)=O)C(C)CC2CN(C(=O)CCP(C)(C)=O)CC12 N1(C(c2sc(C)c(Br)n2)=O)CCCCC(NC(=O)CC2(C)CCCO2)C1 C12(CC)CN(C(=O)C(C)(C)CC)C(C)(C1)C2.c1(C=O)cccc(CCO)c1.N C(=O)(C(CC(C)C)ONC(c1ccc(O)c(F)c1)=O)NC1(c2ncc(C)o2)CC1 S(=O)(=O)(c1ccc2c(c1)CCC2)NC1=C(C=O)CCC1.C(=O)(C(C)C)OC.N c1(CC)ccc(C(=O)NCC2CN(C(=O)CCC3CCCC3)CCO2)c(OC)c1 C1(CC)C(NC(c2cnc(C)nc2)=O)CCN1C(=O)CNC(=O)C(C)CC C1(CS(C)(=O)=O)CN(C(C2(C)CCCC2)=O)CCN1C(=O)C=C.[nH]1cncn1.C N1(C(C(n2c(C)cc(C)n2)C)=O)CCC(C2CCN(C(c3cocn3)=O)CC2)C1 c1(OC)cccc(C#N)c1C(=O)NC1CCC(C(=O)Nc2sncc2C#N)CC1 N(C1CCCn2cnnc21)C(C(C1N(C(CC(C=C)CCC)=O)CCC1)(C)C)=O c1(C(N(CCNC(C(C(CC)CC)C)=O)C2CC2)=O)ccc2c(c1O)CCCC2 Cc1noc2nc(CO)cc(C(=O)NC3CC3)c12.C1(C2CC2)(CC=O)CC1.C C1(NC(c2ncc(SCC3CCCOC3)s2)=O)CCCCC12CCC2 N1(CC(=O)NCc2ccc(Cl)s2)CCN(c2ccccc2OCC(F)F)CC1 C=CCC(CNC(c1cc(C)sc1C)=O)C(=O)Nc1cnc(C)c(OC)c1 Cc1n[nH]c(C)c1C(C)C(N1CCCC(CN(C)C(c2ccccc2)C)C1)=O Cc1ccc(C(=O)NC2CCCN(C(C3CCCN3C3CC3)=O)C2)c(N)n1 N1(C(C2N(C(C)C)CCC2)=O)CCC2(CCN(C(c3c(C#N)cnn3C)=O)C2)C1 C(=O)(CC(C)(C(F)F)N(C)C)N1CCC(O)C1.C1(C(NC)=O)(N(C)C)CC1 c1(C(=O)NCC2C(NC(C(CC)CC)=O)CCC2)nc(C)c(C)[nH]c1=O c1(C2(C)CC2)ccc(Cl)cc1C(N1CC(NC(=O)C=CBr)C1)=O C1(NC(C2(CCOC)CC2)=O)COC2(CCCN(C(=O)CC3CC3)C2)C1 c1(C=O)ccco1.C(=O)(CC1CC1C1CCC1)N.C=CCCC1(C)CC1 C1(NC(CCOC(CC(C)C)C)=O)CN(C(=O)C(F)(F)C2CCCC2)CCC1O N1(C(C=CC(C)(C)C)=O)CCCC(F)(C(=O)NCCC2CC=CC2)C1 Cc1nn2cccnc2c1C(=O)NCC12CC1CCN2 C(=O)(C1CCCc2nccn21)N(C1CC2CCC(C1)N2C(c1cnc(S)[nH]1)=O)C N1(C(CCc2cn[nH]c2)=O)CCC12CC(C(N)=O)C2.c1(CC)nc(C=O)co1.N C12(C(=O)NCCc3n(C)nnc3)CC(CN(C(c3ccncn3)=O)C1)C2 N(C1CCc2cc(C(=O)O)ccc21)S(c1n(CC)ncc1)(=O)=O C1(C(C)(O)CNC(=O)Cn2cnnn2)CCCN(C(c2ccc(N)cn2)=O)C1 C(=O)(C(F)C(C)C)NCCCN(C(C)C)C.C12(C(=O)N)CC(C)(CCO1)C2 c1(OC)cc(C(=O)NC2CCN(C(C3(OC)CCSC3)=O)C2)c2ccccc2n1 N1(C(c2cccc(C(=O)OC)n2)=O)CCOCC(NC(c2cn(C)cn2)=O)C1 C(=O)(C(C)(C)C)NCc1nnc(CC)s1.C1(C(=O)N)C(C)(C)C1(C)C C1CCC(F)(F)C(=O)N1.C=CC1COCC1NC(=O)N(Cc1ccccc1)C c1(C2N(C(=O)Cc3cc(C(=O)Nc4ccccc4)no3)CCC2)cncc(Br)c1 CC1CCC(C(=O)N(CC)C2CC2)CC1.c1(CCC=O)cccc(C(F)F)c1.N Cc1ccc(C=CCC(=O)NC23CC2CN(C(=O)CSC(C)C)C3)cc1 c1(C(C)=O)cn(C)nc1C(=O)NCCC1CN(C(c2ccc[n+]([O-])c2)=O)CC1C C1(NC(CC=CC(C)(C)C)=O)CC(F)C1.C(=O)C(C)(C)C.C(=O)CC.C CC(C)CC(C(=O)N1CC(NC(=O)CCc2cc[nH]n2)C2(CC2)C1)C(C)C C1(CC#C)(C(N2CC(O)(C(F)C=O)C2)=O)CCCO1.CCC(C)C.C(C)=O.N C1(C(N(CC(F)F)CC)=O)CCCC12CCN(C(c1c[nH]c3ncccc13)=O)C2 CN1CCC(C(=O)NC(C)(C)CCCNC(=O)CC2(CO)CC2)C1=O CC1(C)CC(Sc2ccc(NC(N3CCC3CF)=O)cc2)CC(O)C1 Cc1c[nH]nc1C1(C(=O)NC(C)CNC(=O)CCSc2cccnc2)CC1 C#Cc1ccc(C(=O)NCc2cn(CCNC(c3cscc3)=O)nn2)cn1.S C#Cc1cncc(C(=O)NC(C)CCNC(=O)CS(=O)CC)c1 C1(O)(CC(N2C(C(N(C)Cc3nc(C)on3)=O)CC2)=O)CCCCC1 C12(CNC(CCC)=O)CCCN(C(c3cnc(C4CC4)cc3C)=O)C1C2 c1(C(=O)NC(C2OCCN(C(CN(C)CC)=O)C2)C)ccc(F)c(C)c1N C(=O)(C1=CCCC1(C)C)N1CC(NC(CC(=C=C)C)=O)C(C)CC1 N1(C(c2cnn(C)c2N)=O)CC(NC(=O)CC2CCC3CC23)Cc2ccccc21 C1(NC(C2(CC=C)CN(C(c3ccnn3C=C)=O)C2)=O)CC12CCCCC2 CCC(CC(F)F)C(=O)NCCCCC1CN(C(c2cnc(CC3CC3)s2)=O)C1 Cc1cn2c(n1)C(CN1C(=O)NC(Cc3cncc(F)c3)C1=O)CCC2 C1(C(N2CCC(F)C2)=O)CC2(C1)CC1(CC1)C2.c1(C(NC)=O)cc(Cl)cnn1 N1(C(C(=Cc2cn[nH]c2)C)=O)CC(CC(=O)NCC2(CCO)CCC2)CC1(C)C c1(C(N2CC(NC(C34CC5CC3C4C5O)=O)CC(C)C2)=O)cc2scc(Cl)c2[nH]1 C1CCCN(C(=O)C=Cc2ccc(C)s2)C1.C(CC(=O)N(C)C)OCCOC C1(NC(c2cc(C)on2)=O)CN(C(=O)CC=CCc2ccccc2)CCC1C c1(C(N2CCCC(F)(CNC(C3(O)CCC3)=O)C2)=O)ccc2ncnc(O)c2c1 N1(C(C2C(C)(CC)C2)=O)CCC(NC(c2ccnn2CC2CC2)=O)CC1C C(=O)(C(=O)C(C)CC)N(CCC1CCN(C(CCC#CC)=O)CC1)C O=C(C1=CCCCO1)NCC1CCCC(NC(c2nc(Br)c[nH]2)=O)C1 N1(C(c2c(C)occ2)=O)CCC(C)(C)C(C(=O)N(CC(O)CF)C)C1 n1(CC=C)c(N(C2CCSC2)C)nnc1-c1c[nH]nc1CC c1(CC)ccc(C=CC(=O)NC2CC(C)N(C(c3nn(C)cc3Cl)=O)C2)cc1 c1(C(=O)NC23CC(NC(C(F)OC)=O)(C2)C3)cc2c(cnn2C)nc1C c1(OC)c(C(=O)NCC(C)CNC(C2(C)CCC(C)C2)=O)c(C)nn1C C#CC(CC(C)C)NC(C1CCC(C2CC2)N1C(=O)C=CC1CC1)=O c1(C(=O)NC(C(C)(C)NC(C(CCC)OC)=O)C)ccn2ncccc12 N12CCC(C1)CNC2=O.c1ccccc1.C1(c2nccs2)(NC=O)CCC1.N N1(C(CCc2cnc(C)o2)=O)CCC(CC(=O)NCCCCCCCO)C1(C)C N1(C(=O)NCCOC(C(=C)C)=O)CC2(CC2)CC1C=O.C1CCOC1C.N C1(CCOC)CCC(C)N1C(=O)Cc1n[nH]c(C)c1Br Cc1cc(C(=O)NCC2(CNC(=O)C(F)C(C)(F)F)CCC2)nnc1C c1(C(=O)NCC(CNC(C(C)Oc2cccnc2)=O)CO)cc(Cl)ncc1O C1(C)(C(N(CC)Cc2ccncc2)=O)CCCN1C(=O)CCCc1ccccn1 C1CN(C(=O)CS(=O)(=O)N2CCN(C)CC2)CC1S(C)(=O)=O.C=C1CC1C=O N1(C(c2ccc(C)n2C)=O)CC(C)N(C(c2cc(O)nc(O)n2)=O)CC1C c1ccc(F)cc1O.C(C(C)CC(=O)N)NC(C1C(C(=O)OCC)C1)=O.C c1(C(=O)NCC2CC(NC(CNC=O)=O)C2)cc2nccc(C(F)F)n2n1 n1(CC)ncc([N+](=O)[O-])c1C(N1CCCCC(CNC(c2cnns2)=O)CC1)=O C1(NC(C(=Cc2cccs2)C)=O)CCCCCN(C(=O)C(CO)N(C)C)C1 c1(C(N2C(C3CC3)CCC2)=O)cc(F)c(F)cc1O.CCC(C=O)NC(C)=O.N CCC(CS(=O)(=O)NCc1csnc1C(F)F)OC N1(C(c2cnc(-c3ccccc3)n2C)C(=O)NCCCOC)CCCC(CF)C1 CC1(F)CC2(CN(C(=O)CC3CC(O)CN3C(=O)CNC=O)C2)C1 CCCCC(CNC(=O)C=CC(=O)N(C)C)NC(=O)C(F)CC1CCOC1 c1(C(=O)NC(C2(CNC(CCC=CC(C)C)=O)CC2)C)cccc(N)n1 C(=O)C(C1=CCCCC1)N(C1CCC2CC12)C.c1(C(=O)OCC)ccc(C)o1.N Cc1coc(C(=O)NCCCOCCCNC(C2CC2(F)F)=O)c1 N1(CCNC(C(N2CC(C(=O)OC)C(N)CC2)=O)=O)CCN2C(=O)COCC2C1 CC1COC(C)(C(=O)NCC(C)(C)OCC)CO1.C1(CC(=O)N)CCSCC1 c1(C(=O)NC2(CO)CCN(C(=O)C3=CCOCC3)CC2)cc2n(c1)CCCC2 C1(C(=O)NC(C)C(C)NC(C2(F)CC=CC2)=O)C(C)(C)OC1(C)C c1(CC(=O)NCC(CNC(Cc2c(C)ccs2)=O)CO)ccc(C(N)=O)nc1 Cc1nc(C2CCC2)sc1CC(=O)N(C1CCCN(C(=O)C(F)C2CCC2)C1)C N1(C(CN(C(CC=C(C)C)=O)C(C)C)=O)CCOC(C2CC2)C1 O=C(CN1C(=O)C(NC(C2C3COCC23)=O)CCc2ccccc21)NCC(F)F C12(CNC(=O)CN3CSCC3=O)CCC1CCN2C(c1cn2ccnc2s1)=O C1(C(=O)NC2CCS(=O)(=O)C2)CN(c2cc(OC3CCC3)ncn2)CCC1O C1(C(=O)NCC(CC)NC(c2ccn(Cc3ccccc3)n2)=O)CCCC1(F)F N1(C(C(C(C)C)NC(=O)C(C)(C)n2cnnn2)=O)CCN2C(=O)NCC2C1 O=C(CN=c1cc[nH]cc1)NC1CN(C(c2coc(O)n2)=O)C2(CCOC2)C1 c1(CC)cc(CNC(=O)C(C)N(C)C)n[nH]1.C(=O)C(O)CN1CCCC1.N c1(CC)cccc(C(=O)N(CC(=O)NCCCCCC2CC2)C)c1 c1(C(C)(F)F)ccc(C(=O)NCCN2CCN(C(C3CCC3)=O)CC2)nc1 c1(C(=O)NC2C3N(C(CCC(=C)C)=O)C(CC3)C2)ccc(S(C)(=O)=O)o1 C1(CNC(=O)CC2CCOC2)C2CN(C(C3CC3c3cccc(Br)c3)=O)CC12 Cc1cc(F)sc1C(=O)NC1CC(C)N(C(c2cccnc2N2CCCC2)=O)C1 N1(C(=O)C(F)CC2CC2)CCN(C(c2ccc(O)c(CO)c2)=O)C(C)C1.C1CC1 c1(NC(=O)NC2ON=C(CC)C2)ccc(C(=O)N(C)C)c(Cl)c1 c1(C(=O)NCCCC(C)NC(=O)Cc2cccc(Cl)c2F)cccc(N)c1F CCCCC(CC(=O)NC(CCO)C(C)C)NC(=O)CNC(N)=O C1(C(=O)N)OC2CCC1C2.c1(C(=O)OC)cc(C(=O)NC2CC(C)C2)c[nH]1 N1(C(C(C)O)=O)CCCC2(NC(=O)C=CCN3CCOCC3)CC2C1 c1(NCC2(OC)CCC2)[nH]c(=NCc2cccc(C(C)C)n2)nc2c1cnn2C N1(C(C2(CC=C)CCCCC2)=O)CC=C(CNC(=O)CCC(C)C)CC1 C1(C2CC2)(CN(C(=O)CN(C(=O)C(F)C2CCOC2)C)C)CC1 c1(C(N(CCCNC(=O)C(=O)NC2CC2)C)=O)cc2n(n1)CCNC2=O c1(C(N2CC3(CCC(C(=O)NCC(F)CO)O3)C2)=O)cc2cc[nH]c2cc1Cl C1(NC(C2=NNC(=O)CC2)=O)CCCCC12CCN(C(=O)CN1CC(F)(F)C1)C2 CON(CCC(=O)N1CC2CC3CC2C1C3O)C(=O)C1Cc2nccn2C1 C1(C2CCN(C(=O)C(C)(C)CC3CC3)CC2)CCC1.n1(CC)ccnc1C=O.N N1(C(C2CCCCC2O)=O)CC2CCCC2(C(N2CCSCC2CO)=O)C1 c1(C(N(C(CC(=O)NCC(CCC)O)CC)C)=O)cccc(F)c1C N1(C(C#CC(=O)N(C)C)=O)CCN(C(=O)Cc2cscn2)C(C2CCC2)C1 N1(C(c2c(CC)cccc2)=O)CCOC(C)(CNC(c2c(C)ncn2OC)=O)C1 N1(c2ccc(SCC)cc2)CCCN(NC(c2cc(Cl)c(Cl)nc2Cl)=O)C(C)C1 N1(C(c2cc(SC)ncc2)=O)CC2(CCN(C(=O)Cn3cnnc3)CC2)C1 C1(NC(=O)NCc2ccc(OCCC)cc2)CN(C)CC(F)(F)C1 c1(CC(N2CC(O)(CNC(C(C)(C)F)=O)C2)=O)ccc2c(c1)CCOC2 C1(C#N)(C(=O)Nc2cccc(CNC(CCC=C=C)=O)c2)CC12CCOCC2 C=CC1(C2(C(N3CCC4(NC(=O)CCCCN(C)C)CC4C3)=O)CCC2)CCC1 C=CCCCC(=O)N(CCCNC(=O)C(C1CCOCC1)O)C(C)C N1(C(CCC2CC(NC(Cn3ccc(C)n3)=O)C2)=O)CC(C)OC(C)(C)C1C C12(NC(CC=CCC)=O)CCCN(C(c3ccc(OCC)c(C)c3)=O)CC1C2 C(=O)(C1=CC2C=CC(C1)C2)NC1(C)CC(O)CN1C(=O)CSc1nc[nH]n1 C1(CC=O)(C(F)(F)F)CC(=O)N(O)C1.C1CCCC1.O=CCOCCF.N N1(C(C2C(C(C)C)CCC2)=O)CC2(COC(CNC(=O)CCCCCF)C2)C1 c1(SCC)ccc(C(=O)NC(C)CC)cc1.C(c1cn(C)nn1)=CC=O.N CCCC(C#N)C(=O)NC1CCCN(C(c2ccc(C)c(F)c2)=O)C1 C1(C=O)CCC2(CC1)CC2(F)F.c1(C(C)(C)O)cnc(NC2(C)COC2)nc1.N Cc1c(Br)ccc(O)c1C(N1CC(NC(=O)CN2CCC2C)C(O)C1)=O C1(NC(=O)C2=CCC2)CC2CCC1C1CN(C(=O)C(c3ccccc3Cl)O)CC21 N1(C(c2ncc(N(C)C)cn2)=O)CCN(C(c2ccc[n+]([O-])c2)=O)CC(O)C1 Cn1c(C(N2CC3CC2C3)=O)cc2occc12.C1(CC(=O)N)CC(=O)NC(=O)C1 c1(C(N2CC(O)(C(C)NC(CC(=C)C)=O)C2)=O)ccc(-n2nc(C)cc2C)cc1 C1(NC(c2c(Cl)cc(C)s2)=O)CCCC12CCN(C(=O)COC(C)(C)C)C2 c1(C(CNC(=O)CC(C)F)NC(C(C=C)O)=O)ccc(N(C)C)cc1 C1(C(=O)NCc2cc(C)n(C)n2)CC(C)(C)CCN1C(c1cc(O)ncc1F)=O N1(C(C(=O)NCCCn2c(C)nc(C)n2)=O)CCc2cc(O)ccc2C1 CC1C(NC(=O)C(C)(O)c2ccccc2)CCCN1C(=O)C=Cc1cnccn1 CCC(CC(=O)NC1CC2C(NC(c3cnn(C)c3OC)=O)C2C1)SC N1(C(=O)OC)CCC(NCC(=O)NC(c2ccccc2CC#N)=O)CC1 N1(C(c2cc(C)cc(Cl)c2)=O)CCCC2(CCCN2C(=O)COCCC(C)C)C1 c1(OC)nc(C)ccc1C(N1CCC(C(C)C)C1)=O.C1(C=O)CC2(CC2)C1.N N12C3CCC1CC(C3)C2=O.c1(C(C)N(C)C)ccco1.CC(C)(C)OC(=O)N C=CC(CC)CC(=O)NCC1CN(C(c2nn(CC)nc2C)=O)CC1C(F)(F)F C1(N(C(=O)CCc2ccc(Cl)s2)C)C2CN(C(=O)C=CC3CCCC3)CC12 Cc1ccc(C)c(C(=O)C(C)OC(=O)CC2CCC2(C)C)c1 n1(CC)[nH]c(=NC(c2cc(C)cnc2Cl)c2ccccc2OC(F)F)cc1CO c1(C(N2CCCC(NC(C(CC=C)(C)C)=O)C2C)=O)ccc(Cl)c(C#N)n1 c1(C(N2CCC(C(C)(C)NC(c3n[nH]c(C)c3Cl)=O)C2)=O)cnc2ncccn12 C1(C(NOCC2CC(=C)C2)=O)CCCCC1NC(c1ccn(C)n1)=O c1(C(N2CCC(N(C(=O)C3=CSCS3)C)C2)=O)cnc2onc(C3CC3)c2c1 C(=O)(CS(=O)c1ccc(Cl)cc1)N1CC2C(NC(C(C3CC3)OC)=O)C2C1 C1(C(=O)NCC=CC(C)(C)C)CC(NC(=O)CCC2CC2)C(O)C1 C(N=c1[nH]cnc2c(Cl)cc(Cl)cc12)C1CCCN(C(=O)C2=CC3CCCC23)C1 Cc1cc(F)cc(C#N)c1S(=O)(=O)NC1CC(COCc2ccccc2)C1 C(CC(C)C(=O)N1CC2C(C(N3CC(c4ncc[nH]4)C3)=O)C2C1)OC C12(C(=O)NC3CCC(NC(=O)CC4(C5CC5)CC4)C3)COCC(C1)C2 N1(C(C2CCN(OC)CC2)=O)CCC(C2CCN(C(C3CC3C)=O)CC2)C1 c1(C(=O)NCC2C(NC(COCCC#C)=O)C2)nn(C)cc1Br Cc1nnc(O)c(C(=O)NCC2CC(C)N(C(=O)C=CCCC(C)C)C2)c1C c1(N2CCC(CC(=O)NC)C2)nc(=NC)nc(N2CCC(=C(F)F)CC2)[nH]1 CC(CN=c1[nH]c(N2CCCC(CCF)C2)nc2c1CCC2)c1cccc(O)n1 N1(C(C=CSC)=O)CC2CCC1C2NC(C1CCCC2(CC2)C1)=O c1(OC)c(C)csc1C(=O)NCC.c1(C(=O)N)cnn(C)c1C(C)(F)F N1(C(CN2CCN(Cc3c(C)n[nH]c3)CC2)=O)CCc2cc(F)ccc2C1 C(=O)(C#CC1CC1)NC(C1N(C(c2nnc(C)s2)=O)CCC1)C c1(C(=O)NC2CCN(C(CCS(=O)(=O)NC)=O)CC2C)ccnc2[nH]cnc12 C1(NC(=O)CCc2nncs2)C=CC(C(=O)NCc2nc(CO)n[nH]2)C1 c1(CC)c(NC(=O)C=O)sc(C=O)c1C(C)C.C1(C)CCOC1C.C(C)C C(=O)(C(C)C(O)C(C)CC)NCC(CC)NC(c1ccnc(N2CCCC2)n1)=O C12(CC=O)CC3CC(C1)CC(O)(C3)C2.CCC(C#N)C(=O)NCCC(C)(C)C C(=O)(C(=O)C(C)(C)C)N1CC(CCNC(C(CN(C)C)(C)C)=O)OCC1 CC1(C)CC(NC(=O)NCCc2nccs2)CC(C)(C)C1 N1(C(c2c(C)[nH]cc2)=O)CCC2(NC(=O)Cc3nn(C)cc3[N+](=O)[O-])CCCC12 C(CO)(CCCNC(c1ccnc(C(F)F)c1)=O)NC(CCCN(C)C)=O C1(NC(C(CCC)OC)=O)CN(C(=O)C=C(C)c2cnn(C)c2)C2CCCCC12 c1(CN2CCCC(C)C2)cc(-c2nc(-c3cnc(N(C)C)s3)no2)oc(=O)c1Br C1(NC(=O)NC(c2ccc(OC)cc2)CC)CCC2CC(C)CN2C1 CCC(C)CCNC(=O)C(=Cc1cccn1C)F.C(=O)C(F)(F)F.C(=O)C.N C12(CNC(c3ncn(CC)n3)=O)CC1CN(C(=O)CC=O)C2.CCC(C)C.O N1(C(CCCCCOC)=O)CC(C)OC2(CCN(C(=O)CCS(C)(=O)=O)C2)C1 c1(N(C)C)ccnc(N2CCN(S(=O)(=O)CC3(C)CC(F)(F)C3)CC2)c1 c1(OCC)cccc(CN2CC(C)C2)c1F.c1(C=O)ccc(C2CCC2)cc1.N C#CC1CN(C(C2CCCN2C2CC2)=O)CCN1C(=O)COCC(F)F C(=O)(C(C)(O)C(F)(F)F)N1CCC(O)(CC)CC1.C12(C=O)CC3CC1C2C3.N N1(C(c2cc(CC)no2)=O)CC(NC(c2ccoc2C)=O)C(C2CC2)C1 C1(NC(c2ccn(CC)n2)=O)CCCC(N=c2cc(Cl)nc(C3CCCO3)[nH]2)C1 C(=O)C1=CC2(CCN(C(=O)C(C)(C)C)C2)C1.C(CC)OC.CC.C(C)=O.O N1(C(c2cnc(CC)[nH]2)=O)CC(C)CCC1CNC(=O)C(COC)COC CCCCCC(C)(CC)C(=O)N1CCCC(O)(CNC(=O)C(CC)CC)CC1 C1(N(C23CC(C=O)(C2)C3)C(CC2(C)CC2)=O)C2CCC1CNC2.CO c1c(F)c(F)cc(F)c1F.C1(C=O)CCS(=O)(=O)C1.CNCCOCC.N c1(CCC(=O)NC(C)C(C)NC(C2(Cl)CC2)=O)ccc(C(C)(C)C)cc1 C(=O)CS(=O)(=O)c1ccccc1F.C1(C)(CC)C=C(C(=O)NCC)C1.CC.O C1(NC(C2C(C)C2)=O)CN(C(c2csc3c2CCCC3)=O)CCC1(C)C N1(C(c2cnc(C)n2C)=O)CC2(C1)CN(C(=O)CC(C)CN(C)C)CC2CO C(=O)(CC(C)(O)c1ccccc1)N1CCC(C(=O)NC2(CN(C)C)CCCC2)C1 c1(C(=O)NC(CC)CNC(=O)CCOC(C)C)ccc2c(c1)CC(C)O2 C(=O)(CCCC(F)F)NC1(CC=C)CN(C(=O)CC2CCCOC2)C1 Cc1cc(CC(=O)N(CCN(C)C(c2cc(N)nc(Cl)c2)=O)C(C)C)ccc1F C(=O)CC(C)(C)CC(F)F.N1(C(COCc2cc(C)on2)=O)CC2(CCC2)C1.N C1(OC)CCCCC1OC(=O)C(C)(C)NC(C1CCOC1c1nccn1C)=O Cc1nc(Cl)ccc1S(=O)(=O)N1CCCCC1C(N1CCC(C)(C)CC1)=O C(C(C(=O)NCC1CCC1)N(C)C)NC(CCOCCC)=O CN1C(=O)OCC1C(=O)NC(CC1CCOCC1)C(=O)NCCCc1nccs1 C1(CCCC)CC2CCC(C1)N2C(=O)NC1(C(=O)OC)CC(OC)C1 CN1CCN(C(=O)CCCCC#N)C(C(N2CCCCCC2)=O)C1 C1(OC)(CNCC(C2CCOCC2)OC)CCC(C)C1 C(=O)(C1=CC2(CCN(C(=O)CC(C)(C)CC(F)F)C2)C1)NC(CC)CO C1(CC)(NC(=O)COCCSC)CCN(C(=O)CC(C)(C)CC)CC1 C1(CC)CCC(C)CN1C(c1ccc(CNC(c2nonc2N)=O)o1)=O C=CCC(C)(C)CC(=O)NC1CCC(CC(N2CCC(C(=O)OC)C2)=O)CC1 CCCS(=O)(=O)CC(=O)NCC1(NC(c2cnc(S)nc2)=O)CCOCC1 CCC(C)C(CC(=O)NCc1cnc[nH]1)NC(=O)CCNC(C)=O C1(OC)CCC12CC(C(=O)NCC1CCCN1C(=O)CC1(CO)CC1)C2 c1(NC(c2n(CCC)nnn2)c2cc(C3CC3)ns2)cnc2n1CCCCC2 C1(C(=O)N(C)Cc2ccc3cc[nH]c3c2)(OC)CCCC(C)(C)C1 c1(C(N(CCC(C)NC(c2c(C)nsc2)=O)C)=O)ccc(F)c(N)c1F CCC(C)CCC(=O)NCC(C1CCN(C(=O)CC(C)CN(C)C)CC1)(C)C C(=O)(CC=C(Cl)Cl)NC(C1CCN(C(C2CC(=C)C2)=O)C1)C C(CCCCC(=O)NCC1(C)CCCN(C(=O)C(O)CC(F)F)C1)NC(C)=O N1(C(C=COCC)=O)CCC2CC(NC(C3CCOC(C)C3)=O)CCC2C1 C(CC(C(=O)N(C1CC(F)(F)C1)C)NC(=O)Cn1ccnc1)N(C)C N1(C(C2C(C(=O)OC)C2)=O)CCC(O)C(N(C)C(c2ccc(C)s2)=O)C1 c1(C(=O)OC)cc(C(C(=O)NCC(F)F)N(C)Cc2nc(C)no2)ns1 c1(OC)cc(C)c(NC(C2CN(C(c3cc(C(C)C)on3)=O)C2)=O)cn1 C1(C(C(=O)NCC(C)C)N(C(CC)C)CC)CCN(Cc2ccccc2)CC1 N1(C(CCCSC)=O)CC(CO)C2(C1)CN(C(C1CCCCO1)=O)C2 c1(C(=O)NCC(=O)NCC=C)cccc(-n2cc(CC(O)C(C)C)nn2)c1 C12(CNC(c3ncc(C)nc3)=O)CCCCC1N(C(=O)CCN1CCCC1)CC2 c1(OCCCNC(C(C)(C)C)=O)ccc(S(C)(=O)=O)cc1 C#CCC(O)C(=O)N1CC(C(=O)NCC(C)OCCOC)(CC)C1 c1(C(=O)NC(CNC(C(C=C=C)C)=O)CC=C)cc2c(cn1)OCCC2 Cc1cc(CNC(=O)Cc2cn(C)nn2)c(C)s1.C12(CC=O)CCCC1C2 C(=O)(CCCC(F)(F)C(F)(F)F)N1C2C(NC(C(S(CCC)(=O)=O)C)=O)C(C2)C1 C1COCCN1C(c1csc(C(F)F)n1)=O.c1(COC)csc(C(=O)N)c1.C N1(C(C)=O)CCC2(C1)CN(C(=O)CCc1cccc(Br)c1)CCO2 C1(F)CCCN(C(=O)C(c2ccn(C)c2)C)C1.c1(C(C)C)ocnc1C(=O)NC N1(C(c2ccc(C)cc2Cl)=O)CC2(CCCCN(C(=O)C3=CCS(=O)(=O)C3)C2)C1 C12(C(=O)OC)CCN(C)CC1CN(C(=O)Nc1nccc(Cl)c1I)C2 CN1CC(=O)N(CCCCNC(=O)CNC2(c3cccc(F)c3)COC2)C1=O C12(C(=O)NCC3N(C(C(C)=C(CC)C)=O)CC(OC)C3)CCC(CC1O)C2 c1(CN(C)C(=O)OC(C)(C)C)ccc(-c2cccs2)s1.c1(C=O)ccco1 C(c1cccnc1)=CC(=O)NC(C1CCCCN1C(=O)C(F)CC1CCCC1)C N1(C(C(C(C)C)OC)=O)CCCC2(CCCN2C(c2cn3c(n2)CCC3)=O)C1 C1(N(C(CN2CC(C)C2)=O)CC(C)C)CCN(C(c2cnn[nH]2)=O)CC1 N1(CC)CCN(CC(=O)NC2CN(C(C3CSCC(=O)N3)=O)CC2C)CC1 c12ccc(cn1)C(=O)N1CCN(CC1)C(=O)N2.C1(C(=O)O)COCCN1 N1(C(C(CCOCC)NC(=O)COc2cccnc2)=O)CCSCCC1C C1(C(N2CCC2CO)=O)(CNC(c2n(CCC)ncc2)=O)CC(C)(C)C1 CCC(C)(CO)C(=O)N1CCN(C(c2ccc(Cl)c(Cl)c2)=O)C(CCO)C1 c1(CC(=O)NCCC(C)NC(=O)C(O)C(F)(F)F)csc2c(Cl)cccc12 C1(F)(N(CC(C2CCOC2)O)C(=O)OCC(F)(F)F)CCCC1 CC(CCCO)NC(C1CCC(CNC(C2C3COCC23)=O)O1)=O N1(C(CCC2C(C)=NOC2=O)=O)CCCC12CCN(C(c1cc(O)cs1)=O)C2 C1(OC)CC2(CCC(C(N3CCN(C)C(CNC(=O)CCC(C)C)C3)=O)CC2)C1 C(=O)(CCC(C)(F)F)NC(C1CCCCC1)CNC(Cc1c(C)nsc1)=O C=Cc1ccc(C(=O)N(CCC(=O)NCCCc2cc(C)no2)C)cc1 N1(C(c2ccnc(C)c2N)=O)CCCC2(CNC(=O)COCCF)CCCC12 C(C)(CCC(=O)N(c1ccsc1)C)NC(C(F)=CCC)=O C(c1c(Cl)cccc1Cl)=CC(=O)NC1CCN(C(C2CCC(C)O2)=O)CC1C N1(CC(=O)N(C2(C(N(CC(COC)O)C)=O)CC2)C)CCC(OC)C1 N1(C(C2C(C(C)(C)C)CC2)=O)CCCC(NC(c2cc(O)ncc2F)=O)C1CO N1(C(C2(CC#C)CCOC2)=O)CC2CCN(C(=O)CCC(=C)Br)C(C2)C1 Cc1nc(F)ccc1-c1cn(CC(N2CCCCC2)=O)nn1 CCC(CNC(=O)C(F)OC)(CC)NC(c1ccc(N(C)C)nc1)=O C1(NC(CC(CCC)C)=O)CN(C(=O)Cn2cc(C)cn2)CC(F)(F)C1 CC1(C)C(=O)NCC1NC(N1CCN(C(c2cc(Cl)cc(Cl)c2)=O)CC1)=O c1(CCCNC(=O)NCC(C2CCC2)OC)cnccn1 c1(OCC#C)ccc(CC(c2ccc(C)cc2)=O)cc1.C1C(=O)N1 CC(C)(C#N)CCC(=O)N1CCCC(C(=O)NC2CC(C3CCCC3)C2)C1 N1(C(c2cc(Cl)cc(OC)n2)=O)CC2(CCC(CN3CC4CC3CN4C)O2)C1 c1(NC(N2CC(C(=O)OC)C(O)C2)=O)ccc(I)cc1Cl Cc1nn(C)c2cc(-c3cnccc3CN3Cc4n[nH]cc4C3CO)ccc12 C(=O)(C1=CSCCO1)NC1CCC(N(C)C(c2cccc(=O)o2)=O)C1 C1(CCC(=O)NCC(C)NC(=O)CCc2ccc(Cl)cc2)NC(=O)NC1=O c1(C(N2C(CNC(c3n(C)c(O)nc3)=O)CC(F)C2)=O)cc2n(n1)CCCC2=O N1(C(c2ccnc(C)n2)=O)CCC(C(N2CC3CC(C2)O3)=O)C(O)C1 N1(C(c2[nH]n(C)c(=O)n2)=O)CCCC2(C1)CN(C(=O)CCC1CCCCCC1)C2 CON(C(=O)c1nccn1Cc1ccccc1)C1CCN(Cc2ccccc2)C1 C1(c2cccnc2)(C=O)CC2(CCC2)C1.CC(C)CCOCC(=O)NC1CC1 c1(N(C)CC)nc(NCCCOc2cccc(C)c2)c2ccsc2n1.C1CCOC1 N1(C(C2C(NC(C(C)Cn3cccn3)=O)COC2)=O)CCC2C(O)C(C)(C)C12 O=C(CCC(F)F)NCCOCCCNC(c1ccc(C(F)(F)F)[nH]1)=O c1(SCC(=O)NC(CC)CNC(=O)Cc2cc(C)on2)cccc(F)c1 CCC(CC)(CC)C(=O)NCC(C)NC(C1CN(S(N)(=O)=O)C1)=O C(=O)(C(C)(C)CCC(=O)NC1CCC(NC(=O)CC2=CCCCC2)C1)OC Cc1ccc(C(N2CC(O)(C(C)NC(=O)C(C)CC(C)(F)F)C2)=O)c(F)c1Cl C1(C(=O)Nc2snc(-c3ccccc3)c2Cl)CCC2(CCOCC2)CC1 Cn1cc(C(=O)NCc2cccc(OC3CCCCC3)c2)c2c(Br)ccnc12 C1(N(C(=O)CN2CCN(C)CC2)C)CCN(C(=O)C(=O)N)CC12CC2.C1CC1 C1(CC)CN(C(c2cc(OC)cc[n+]2[O-])=O)CCC1NC(c1cnc(C#N)s1)=O c1(-c2cnc(CC(=O)NCc3n(C)ncc3)nc2)cc(C(F)(F)F)ccc1O c1(CCC=O)cc(F)c(F)c(F)c1.CC(CNC(=O)C(F)=C1CCCC1)CO N1(C(C(C)SC)=O)C2CCC1CC(N(C)C(c1cc(-c3ccncc3)no1)=O)C2 C1(CNC(c2c(C)nccc2)=O)C(C)CCCN1C(c1ccco1)=O.N(C)C.C C1(CNC(c2c(C)nc[nH]2)=O)CC2COCC2N1C(c1nnc(C(C)C)s1)=O c1(C(=O)NC2CCN(C(=O)CNc3cccnc3)CC2)cncc2[nH]ccc12 C=CC(C)(C)C(=O)NCC1CCC(F)(C)C1.c1(C=O)cc(C2CCC2)no1 C(=O)(C(C)CC(F)F)N1CC(NC(C(CC)OC2CCCC2)=O)C(CO)C1 N1(C(c2c(CC)occ2C)=O)CC(C)C(F)(F)C1.n1(CC=O)nnnc1C.N CCC(CC(F)(F)F)C(=O)NCCNC(c1ccccc1OC1CC1)=O.C Cc1nccn1CC1CCCN1C(=O)NCc1cocn1 C1(NC(c2cc(C)ncc2)=O)(CNC(c2cnc(C)[nH]2)=O)CCCCC1C C1(C(=O)NC(C(=O)NC(C(C)C)C2CC2)C2CC2)CCCC(=O)N1C c1(SCC)ccccc1CC(=O)N(C1CC(C(=O)NCCCCCSC)C1)C N1(C(C(CCC)CC)=O)CCCC(C2(NC(=O)C3=CCSC3)CC2)C1 C1CN(C(C2(C(F)F)CCCC2)=O)CC2(CC2)C1.c1(OC)ccncc1C(=O)N C1(N(C(C(C)SCCCC)=O)CC)CCN(C(=O)CN(CC(C)(C)C)C)C1 C#Cc1ccc(CC(=O)NC(CCNC(C2(O)CCSC2)=O)C(C)C)cc1 C1(NC(C2(C)CCCO2)=O)CC2CCC(C1)N2C(=O)Cn1cccn1 c1(SC)cn(C)nc1C(=O)NC(C)(C)CN(C)C(C1CC1Cl)=O C1(NC(c2n[nH]c(C)c2F)=O)CCCCCN(C(=O)C(C(C)C)NC(N)=O)C1 C1(NC(CCCOC)=O)CC2CCC1N2C(=O)C=CSc1ccccc1 c1(CC(=O)NCCN(C(=O)COC)CCC)cc(C)no1 CC1C(O)CCCN1C(C12C(NC(=O)CC3(C)CCC3)C3CC1C2C3)=O c1(C(C(N2CC(CC=C)(NC(=O)CC(C)F)C2)=O)CC)c(C)noc1C N1(C(CCCOCCC)=O)CC(=O)CC1C(N1CCCC(C(C)(C)C)C1)=O S(=O)(=O)(c1ccc(Cl)c(Cl)c1Cl)NC1CCN(Cc2ccc(C(C)C)cc2Br)C1 N1(C(CSCC#C)=O)CCC(C(=O)NCc2cccnc2O)C1C(C)C N1(c2cc(N3CCC(COC)(CO)C3)ncn2)CCc2c(ccn(C)c2=O)C1 C(=O)(C(C)CCCC(C)=O)NC1C2C(C(=O)NC(CC)CC)C3C(C2)C13 Cc1cscc1C(=O)NC1CC(OC(C)C)C1 Cc1c(C(N2CC(NC(=O)C(C)C3=CCCC3)C2)=O)cc([N+](=O)[O-])cc1Br c1cn(C)nc1C1CC1.C(C)(C)(C(=O)N)OC.C1CCC(C=O)C1.C1CC1 C12(NC(c3cc(N)c(F)cc3)=O)CCCC1CN(C(c1cc(CCO)on1)=O)C2 c1(CNC(C=COCC)=O)nc2c(s1)CCN(C(=O)C(C)SC(F)(F)F)C2 c1(C(=O)NCC2C(C=O)C2)cccc(O)c1[N+](=O)[O-].n1(C2CC2)cccn1 N1(C(CC=C(C)C)=O)CC2CCOCC2(NC(c2n[nH]c3c2CCCCC3)=O)C1 CS(=O)(=O)c1ccc(C(=O)NC(CNC(c2cnn3cccnc23)=O)CO)s1 c1(CC)c[nH]c(C(=O)NCC2(C)CC(NC(=O)CC(C)SC)C2)c1 CC(C)(CCC#N)C(=O)N1CC2CC(NC(=O)CC3CCC(=O)NC3)C2C1 C(CCC)(C(=O)NC(c1cccnc1)C(=O)NC(C)C(C)SC)=CCC CC1(C(=O)NCC2CCC(=O)NC2)CCN(S(=O)(=O)C(F)(F)F)C1 CC(Cc1ccncc1)C(=O)NC1CC(NC(c2ccn[nH]2)=O)C1.C1CCC1.C CC1=CC(C)CN(C(C2CCCN(C(c3ccncc3N)=O)C2)=O)C1 C1(C=O)(N(C)C)CCCSC1.C1(C(=O)NC(C)C(C)C)(COC)CCCC1 c1(OC)ccc(Br)c(C)c1C(=O)NC.N1(CC=O)CCC(C)CC1.C1CC1 N1(CC2(C)CCC(C)CC2)CCCC2(CCN(C(=O)CC3CCC4CC4C3)C2)C1 c1(CN2C(C(=O)Nc3cc(OC)nc(OC)n3)C=CC2)cn2cc(F)ccc2n1 c1(NC)nc(C)ccc1C(=O)NCC(c1ccc(Cl)c(C(F)(F)F)c1)N N1(C(c2c(C)cc(C)cc2O)=O)CCC2(CCCN2C(=O)C(O)C2CC2)C1 C1(COC)CN(c2nnc(-c3ccccn3)n2CCSc2ccccc2)CCO1 c1(N(CC)CC)cccc(N(C)C(=O)NCCn2ccc(C3CC3)n2)c1 N1(C(C2C(CCC)C2)=O)CCCCC1Cc1cn(CCN2CCCCC2=O)nn1 c1(C(N2CCCCCC2c2ccco2)=O)c(C2(CO)CC2)cc(Br)cc1F C1(C=O)CC2(C1)CC21CCC1.C1(C(N2CCC(O)C2)=O)CC2(C1)CC(O)C2.N c1(C(=O)N)cnn2c(=N)[nH]cnc12.Cn1nccc1C(=O)NC(C)(C)C1CC1 C#Cc1cc(C(=O)N(CC(C)NC(c2cc(C(N)=O)c[nH]2)=O)C)ccc1Cl c1(C(N2CCCC2)=O)ccc([N+](=O)[O-])s1.c1(CCC(=O)NCC)cn(C)cn1 CN=c1[nH]cc(C(=O)NC2C=CCC(C(=O)N(C)Cc3nncn3C)C2)o1 C1(C(=O)NOCC(C)(C)C)(CCC=C)CN(C(=O)CSC(F)(F)F)C1 C(=O)CCC(F)(F)F.CC(CNC(C1(C(=O)O)CC1C)=O)C.C(C)(C)C N1(C(Cc2nc(C)[nH]n2)=O)CCC2(CCC(CNC(=O)C(C)(C)CO)CC2)CC1 C1(C2CC2)CCN(C(C2(O)CCSC2)=O)C1.O=C(CCC(=O)NC1CCC1)N.C CCC(C(O)C(F)(F)F)NC(c1cnn(C)c1Cc1ccccc1)=O C(CN=c1[nH]nc(-c2cccnc2)s1)N(C(=O)Nc1cc[nH]n1)CC C1(CCOC)(C(N2CC3CCC2C3)=O)CCN(C(=O)CC2(C)CCOC2)CC1 C1(COC)(NC(c2cnn(C)c2Cl)=O)CCN(C(=O)CC)C1.c1ccccn1.N C1(CNC(c2cccc(C3CCC3)n2)=O)COCCN(C(=O)C2=C(Cl)CC2)C1 C1(CNC(c2cn(CC)nn2)=O)COCCN1C(=O)CC1CC1C1CC1 CCCC(C)(O)CC(=O)NCCn1cnc(C(=O)NCCc2noc(C)n2)c1 N1(C(CCC=C)=O)CCN(C(c2cc([N+](=O)[O-])n[nH]2)=O)C(C(F)F)C1.C(C)(=O)N c1(N2C(C(N3Cc4ccc(Br)cc4C3)=O)CC(F)C2)ncc2c(Cl)cccc2n1 C12(NC(c3ccncc3Cl)=O)CCN(C(c3ccc(C(F)(F)F)o3)=O)CC1C2 C1(NC(c2c(C)nn[nH]2)=O)CCC(C)(C)CC1C.c1(C=O)ccn(C)c(=O)c1 c1(NC(C2N(C(C3CCC(=O)NC3)=O)CCC=C2)=O)ccc2c(c1)CCC2 C(S(=O)C1CCCCC1)c1cccc(C(=O)Nc2ncccc2C(F)F)c1 C(=O)(C1=C(C)OCC1)NCC(CC)N(C)C(c1csc(C)c1OC)=O C1(CC(=O)NCC2CC(C)N(C(=O)CCC3CC3)C2)(COC)CCOCC1 C1(NC(c2ncnc(C)c2C)=O)CC2CCC(C1)N2C(=O)CN1CCC(O)CC1 c1(CC)ccc(C(N2CCC(NC(=O)C(C)C3CC3)C(C)C2)=O)c(O)c1 C1(CC)CN(C(c2nccc(C)n2)=O)CCC1NC(=O)COCCCF N1(C(C(C)N(C(=O)CCC2CCOCC2)CC)=O)CCC(CC2CC2)C1 c1(C(N2CC(NC(c3nc(OCC)oc3)=O)C2)=O)nccc(OCC)c1F CC1CCc2c(C(N3CC(NC(=O)Cc4cnnn4C)CCC3C)=O)csc2C1 N1(C(C2CCN(C(C3CCC4(CC4)C3)=O)CC2)=O)CC2CC(C1)C2(C)C.CO.C c1(CC)cc(NC(=O)C=CC2CCCN2C(=O)CN2CCCC2C)ccc1C N1(C(c2c(C)nc(C)c(C)n2)=O)CC2CC(NC(c3n[nH]cc3F)=O)CC(C2)C1 C1(NC(c2[nH]cc(CC)n2)=O)COCCN(C(C2(F)C(C)(C)C2(C)C)=O)C1 N1(C(C(C)NC(CC)=O)=O)CC2(CC2)CC1CNC(c1ccc[nH]1)=O.C N1(C(C=CC(C)C)=O)CCC(C(=O)NCc2ncccc2Cl)(OC)C1 C1(C(=O)NC2(C(N)=O)CC2)CC2(CC2)C1.c1(C=O)coc(C(F)F)n1.C N1(C(c2ccn(C(C)(C)C)c2)=O)CCSCC1CCNC(C1CC2CCC1C2)=O C(CC(C(=O)NCc1noc(C(N)=O)n1)NC(c1ccnn1C)=O)OC N1(C(C2(COC)CC2)=O)Cc2ccc(O)cc2CC1C(N1CCC(Cl)C1)=O C(c1cn(C)c2ccccc12)=CC(=O)N(C(CN(C(CSC(C)C)=O)C)C)C C(=O)(C#CC1(C)CCCO1)NCCCN(C(=O)Cc1ccccc1O)C(C)C C1(NC(C2C(OCC)C2C)=O)CC2CN(C(=O)CCC(=O)c3cccs3)CC2C1 c1(NC(C2N(C(Cc3nc(C)on3)=O)CCOC2)=O)ccc(Br)c2cccnc12 O=C(CCC1CCN(C(C2CCC2(F)F)=O)C1)N=c1ccn(CCF)[nH]1 n1(CCCC)cc(C(=O)N(CC(C)CNC(=O)CCSCC(N)=O)C)nn1 C1(NC(CCOCCOC)=O)COCCN(C(=O)C(C)N2CC(C)C2)C1 C1(NC(=O)Cc2ccc[nH]2)CCC(CNC(c2cnc(-c3ccsc3)s2)=O)C1 c1(C(=O)NC2CC(NC(C(C)SC(C)C)=O)C(O)C2)ccc(C(F)F)cc1Cl CC1=C(C(=O)N2CCCC(C(C)NC(C34CCCC(C3)OC4)=O)C2)CCO1 N1(CC)CC(NC(C2CCN(C(=O)C(C)(C)c3ccno3)CC2)=O)C(C)C1 C(=O)(N(CCC(=O)NCCC1(CO)CCC1)OC)C1C(CC)CCC1 Cn1cc(C#N)cc1C(=O)NCC1(O)CCCN(C(=O)C)C1.c1ccccc1.O N1(C(=O)OC)CC(C)(NC(=O)C(C2CCOCC2)O)C1.C12(C)CC(C1)N2 CC(C(=O)NCC1(O)CCCN(C(c2cc(Cl)c(F)cc2O)=O)C1)C1=CCCC1 CC1CN(CCCC(c2ccccc2)O)CCC1NC(=O)CC1CC2(CC2)C1 c1(OC)cnc(F)cc1C(=O)NC1CN(C(C2CCC2)=O)C2CC12 C12(CNC(CCC=C)=O)CC1CN(C(=O)C(C)Oc1ccc(Br)cc1)C2 C1(OC)CC(C)N(C(c2n[nH]c(C)c2Cl)=O)C1.N1(CC=O)CCC(C)(C)C1.N C=CCCCCC(=O)NCC1(C)CCC(NC(c2ccccc2CO)=O)CC1 C1(NC(C=C(CCN(C)C)Cl)=O)CCN(C(C2CCCCC(=O)N2)=O)CC1O Cc1c(C(N2C(C(N3CCN4CCC3C4)=O)CC3CC23)=O)cccc1O CCC(C)N(OC)C(=O)C1CN(C(C2CCCC23CCC3)=O)CC12CC2 C=CCCC(=O)N1C(C(=O)NCCOCCO)CC1C C(=O)(CC(C)C(F)(F)F)NC(C)CCN(CC(N1C(C)CCCC1C)=O)C N1(C2CN(C(C(C)CO)=O)C2)CCN(C(=O)C=Cc2cn(C)nn2)CC1 c1(NC(Cn2cc(C3(C(=O)OCC)COC3)nn2)C)ccc(Br)nc1 c1(N(C)CC2(OCC)CCOC2)nc(=NCC(C)OC)[nH]c2c1COCC2 c1(C(N2CCC(C)(NC(c3[nH]cc(CC)n3)=O)C2)=O)cnc(O)c([N+](=O)[O-])c1 C1(C(=O)OC)(NC(=O)Cc2c(F)cccc2F)CC2(CC(C(F)(F)F)C2)C1 C1(CCC)CN(C(C2CC(CC)=NO2)=O)CC1NC(c1occc1Br)=O C1(CCC)(NC(C2C=CCC2)=O)CCCN(C(c2cn(CCC(C)C)nn2)=O)C1 O=C(CC1NCc2ccccc21)Nc1ccc(-c2ncco2)cc1 CC(CS(C)(=O)=O)C(=O)N1CCCC(c2cn(Cc3csc(Br)n3)nn2)C1 c1(C(C(=O)NC2COC2)N(CCOC(C)(C)C)CC)cccc2nc[nH]c12 Cc1conc1C(=O)NCCC1CC(NC(=O)C(c2cscc2Br)=O)C1 c1(CC(N2CC(CC)C2)=O)cccc([N+](=O)[O-])c1.CN1C(=O)CCC1CC=O.N C1(N(C(C(C)n2ccnn2)=O)C)CN(C(C2CC(Cl)(Cl)C2)=O)CCC1O c1(NC(=O)NCCC(C(=O)OC)C)ccc2nc(-n3ccnc3)sc2c1 C=Cn1nccc1C(=O)NCC(C(C)(C)C)NC(=O)CC.c1ccc(C)cc1.S C1(NC(=O)CCC2CCCOC2)CC2CCC1(NC(c1cc[nH]c1C1CC1)=O)C2 C=CCN=c1[nH]cc(C(N2CCN(C(=O)CN(C(=O)CC(C)C=C)C)CC2)=O)s1 C1(C(N(C(C#C)C)C)=O)CCN(C(=O)C(CC=C)NC(C)=O)CC1O C12(CC(=O)NCC(CNC(COCCCCCC)=O)C)CCC(CC1)C2(C)C N1(C(CCCCC#C)=O)CCCCCCC1C(=O)NC1CCCN(C)C1=O CC(C(=O)NC(c1ccccc1)CNC(=O)CCCN=[N+]=[N-])C(C)S(C)(=O)=O c1(CCC(=O)NCCCCOC)c(C)noc1C.C1(C=O)(C(N)=O)CCC1.N N1(C(C(C)OCC=C)=O)CCN(C(=O)CCc2c(C)n[nH]c2C)CC1CCO N1(C(c2cccc(Cl)n2)=O)CC2Cc3ccccc3C12.c1(C2NCC2)cn(CCO)nn1 c1(NC(C(n2ccc(C3CC3)n2)C)=O)nc2cccc(I)c2[nH]1 c1(C(=O)OC)cc(C(=O)NC(C2CCOC2)C)cc(O)c1.c1(C=O)cnco1 C#CC1CN(C(C2(O)CC2)=O)CCN1C(=O)CC1CCOC1.C(CC)O CCCCNC(=O)C.C(=O)(C(F)=CC)N.C(C)(C)C.C=O.C(N)=O N1(C(CN2C(=O)CSC2)=O)CCC(F)CC1C(=O)NCCOC1CC1 c1(C(N2C(C(N3CCCC(C)(O)C3)=O)C(O)CC2)=O)cc(F)c([N+](=O)[O-])c(F)c1 C1(NC(C2N(C(CC)=O)CSC2)=O)CCCC12CN(C(=O)C(COC)COC)C2 CC(C)(C)C(=O)O.c1(C(C)(C)NC(=O)CC2CC(C(F)(F)F)C2)c[nH]nn1 c1(CC)nnsc1C(N1CC(C(C)NC(=O)CCc2cncs2)C1)=O Cc1cc(-c2csc(NCc3noc(-c4ccccc4)c3Br)c2)cc(F)c1 n1(CC)c(O)nc2cc(C(N3CC(C)(NC(C)=O)C3)=O)ccc2c1=O c1(C(=O)NCC(C)(CO)NC(C2CCN(C)C2)=O)cncc(C(F)F)c1 c1(C=O)cccn(CC(F)(F)F)c1=O.C1(C)(C(N(C)C)=O)CCCC1.C1CC1 Cc1cccc(C(=O)NCC(=O)N)c1.C(C)(C)CO.C1(C=O)CC1C(C)C N#Cc1cc(F)c(Cl)cc1NC(N1CC(CC(N)=O)C1)=O C=CCC(CC(C)C)C(=O)NC(C)(C)CN(C(=O)CC(C)CC)C c1(NC(C2(CF)CCN(C(CN(C(C)=O)C)=O)C2)=O)cc(F)c(O)cc1C Cc1nsc(N)c1C(=O)NCC1CC1NC(c1ncn(C)n1)=O N1(C(C(C2CCOCC2)C)=O)CCOCC(C)(CO)C1.C1(=O)CCCN1.[SH](C)(=O)=O N1(C(CC=C)=O)CC(OC)CC1CCNC(=O)COC1(C(F)F)CCCC1 C#Cc1ccc(C(N2CCC(C(C)(C)C(=O)NC(CC)CC(F)(F)F)C2)=O)nc1 [N-]=[N+]=NC1CC2(C(N3CCCC(O)(CNC(c4sccc4Cl)=O)C3)=O)CC12 N1(C(C(C)CNC(C2CCC(=O)CC2)=O)=O)CC(C2CCCC2)C1 C1(C(=O)NCC(C2CCN(C(C3(CO)COC3)=O)CC2)F)CN2CCC1CC2 N1(C(CC)=O)CCOC(C(=O)NCC(C2CCCCC2)C)C1 CC(F)(F)CCCCNC(C1(N(C(c2n[nH]c(=N)[nH]2)=O)C2CC2)CCC1)=O c1(NCC2CCCCN(C(CCC)=O)C2)cc(C(C)C)nc2ncnn12 N1(C(C2N(C(c3c(CC)c[nH]n3)=O)CC(F)C2)=O)CCOCC(C)(F)C1 C1(CNC(C(CC)O)=O)(CO)CCCN(C(c2cccc(N(C)C)n2)=O)C1 N1(C(=O)CC2CC(O)C2)CC2CC(NC(C3(c4nc(O)n[nH]4)CC3)=O)C2C1 N1(C(C(CCCNC(c2c(N)snn2)=O)O)=O)CCc2ccc(F)cc21 c1(C(=O)NC2C(CNC(C3C(=C)C3)=O)CCCC2)ccc(OC)c2cn[nH]c12 c1(C(=O)NCCCCCNC(C(N2CCCCC2)C)=O)cc(O)cc([N+](=O)[O-])c1 C(C(CC)(CC)CC)NC(CCN(C(=O)CSCC(N)=O)CC=C)=O c1(C(=O)NC2CCCC(NC(C(COC)COC)=O)C2)ccc(F)c(Cl)c1F C(CC(Cc1ccccc1)N=c1[nH]nc(C#N)s1)NC(C)CC1CC=CCC1 CC(=O)C(C)CC(C)C(=O)NCC1(C(=O)NC(C2CC2)C)CC12CCC2 Cc1nnccc1C(=O)NC1C2CCN(C(=O)C(C(C)C)n3ccnc3)C12 c1(OC)ccc(C(=O)C(=O)NC2(C3CCCN3C(=O)CCC(=O)N)CC2)cc1 c1(C(=O)OC)c[nH]c2c(C(C)=O)cccc12.n12ccnc1-c1cn(nn1)CC2 CC1(C)CCC(O)(C(N2CC3CC(O)C2C3NC(C2CCC(=O)N2)=O)=O)CC1 C1(C=O)CNC(=O)CC1(C)C.c1(OC)ncc(F)cc1C(=O)NC1CCC1.C c1(C(=O)NCCCN(C(C2CC(O)C2)=O)CC)cc2c(OC)cccc2[nH]1 C(=O)CS(=O)(=O)C(C)(C)C.N1(C(C)=O)CC(F)C1.CC(C)C.C(=O)(C)O C(CCC(=O)NCCCCCNC1C2CCCC12)C1C(C)C1.C(C)N c1(C(N(CCCN(C(CC(C)c2cccnc2)=O)C)C)=O)c[nH]nc1S(N)(=O)=O c1(N(C(CNC(C2(C(=O)O)C(C)C2)=O)=O)C)ccnc(Cl)n1 N1(CC(=O)N(CCCC)C)C(=O)c2ccccc2C1=O.CC(C)C(C)(O)C(=O)N c1(C(=O)NC2CCN(C(c3ccn(CC)c3C)=O)C23CC3)ccc2nccn2c1 Cc1coc(C(=O)NCCCOCCC(N2CCC(CC(C)C)C2)=O)c1 C1(CNC(=O)Cc2ccccc2)CC2CCC(C1)N2C(=O)COC1COC1 C1(CCNC(c2c(C)oc(Cl)n2)=O)CCN(C(=O)CC(C)(C)C(F)F)CC1(F)F C1(C(=O)NC(C2CCOC2)C)(NC(c2cc(C3CC3)[nH]n2)=O)CCN(C)C1 N1(C(CCC)=O)CCC(NC(=O)Nc2ccc(C#N)cn2)C(C)C1 C(=O)(C1=NOC(C)C1)N1C2C(NC(c3cnn(C(C)C)c3Cl)=O)C(C2)C1 C(=O)(C(CC(C)C)ONC(=O)C(C)NC1CC1)Nc1c(C)n(C2CC2)nc1 CC1CN(C(c2c[nH]cc(Cl)c2=O)=O)CCC1CNC(c1cc(O)nc(O)n1)=O C1(CC(=O)NC2(C(C)C)CCC2)CCCN(C(=O)CC2CCC(=O)N2)C1 N1(C(C2C(NC(CC(C)N(C)C)=O)CCOC2)=O)C2CCCC1CC2 c1(C=O)cc2n(n1)CCCC2.c1(C(=O)NC(C(=O)OC)C2CC2)sccc1 N1(C(C(C#N)=CC(C)C)=O)CC2CC(NC(C3CC(=O)NC3(C)C)=O)CC2C1 Nc1ccc([N+](=O)[O-])cc1C(N1C2CCC1CC(NC(=O)COC(F)F)C2)=O C(C)(C(=O)N=c1ccn(CCCO)[nH]1)C1CCN(C(Cn2c(C)nc(C)n2)=O)C1 C1(C(c2n(CC)nnn2)NCC2(C)CC2)CCC(=O)NC1.C(N)=O.N CCCCC(CCCC)C(=O)N1CC2CCN(C(c3cncc(N)n3)=O)C2C1 C=C(Cl)C(C)(C)C(=O)N1CC(c2ocnc2CNC(=O)C(C)(CC)OC)C1 C(=O)(CC1COc2ccccc21)NC1CN(C(C=NOC)=O)CC12CCC2 c1(C(=O)NC(C(C)NC(=O)CN2CC=CC2)CO)csc2c(F)cc(F)cc12 n1(CCC(C)(C)C)nc(C2CCOC2)nc1-c1cccc(-c2cn[nH]c2)c1 c1(NC(N2CCC(NC(=O)OC(C)(C)C)C2)=O)ccccc1.C12CCC1C2 N1(C(C2(O)CCC(C)(C)CC2)=O)CCC2(CC(NC(c3cnc(S)[nH]3)=O)CO2)C1 CCCCCCC(C)C(=O)N1CCOCC1CN(C(=O)CCc1nncs1)C c1cccc([N+](=O)[O-])c1.N1(C(c2c(C)nsc2)C=O)CCC(C)(N(C)C(C)=O)C1.N C(=O)(C1=CC(O)C(NC(=O)CCc2nc[nH]n2)C1)NC(C#C)C1CCC1 c1(CCC(N2CC3CC3(C(=O)Nc3ccc(O)c(Cl)c3)C2)=O)cccc(Br)c1F C(=O)(C1CCN(C)c2ccccc21)N1C(C)CC(NC(c2cc(C)sn2)=O)C1 N1(C(C=CCOC)=O)CC(NC(c2ncc(C(F)F)s2)=O)CC(C)(C)C1 N1(C(C(C)OC)=O)CCC(C(=O)NCc2c[nH]nc2C(=O)O)C(C)(C)C1 C1(N(C(c2cc(C(CC)CC)no2)=O)C)CCN(C(C2(C)CCCOC2)=O)CC1 c1(CC=C(C)C)cc(C(=O)NCC2(C)CCCC2)ccc1O.C(=O)C=CBr.N n1(CC(=O)NCCC)cc([N+](=O)[O-])ccc1=O.c1(C(=O)N)ccc(F)c(F)c1 CCC(C)(C(=O)N1CC(NC(c2ncccc2CO)=O)C(SC)C1)C(N)=O CC1N(C(C2CN(C(C3CC3C3CC3)=O)CC2(C)C)=O)CCOC1(C)C c1(OC)nscc1C(=O)NC1CCCC1NC(=O)Cn1cnc(=N)[nH]1 C(=O)(C(CC1CC1)NC(=O)Cc1coc(C)n1)NCC(C)OC Cc1cnc2cc(C(=O)NCC(C)NC(C3(C)CCCN3C)=O)ccn12 N1(C(CSc2nc(C)[nH]n2)=O)CCC(C2CC2)C1CNC(=O)C(C)O c1(CC2(C(=O)O)CN(NC)C2)ccc(OC)c(OC2CC2)c1 C12(C(=O)NCCCNC(C3CCC4(CCC4)O3)=O)CCCC1CCC2 c1(C(N2CCN(C(CCN(C)C)=O)CC2CC#N)=O)cc(F)cc(Cl)c1Cl c1(C=O)cc(F)ccc1C(F)(F)F.C(C)(C(=O)NC1CC1)SCCCC.C C1(CNC(CC=C=C)=O)CC2(CCN(C(c3c(C)nc(O)nc3C)=O)CC2)CO1 c1(NC2C(=O)N(C3CCC3)CC2)cc2ccccc2c2cccnc12 c1(C(N(CCC)CCNC(c2cncc(F)c2)=O)=O)ccnc2c1CC(=O)N2 CC(CCC(=O)NCCC(O)CNC(=O)C=Cc1cncs1)N(C)C c1(C(C)C(=O)NCCN(C(=O)CC(C)(C)C)C2CC2)ccc2c(c1)OCO2 C1(CNC(C(CC=C)(F)F)=O)C(C2CC2)CCN1c1nc(Cl)ncc1F C(C)(CCCN=c1ccnc(Cl)[nH]1)NC(C1C(OC)CCCC1)=O c1(C(N2CC(C#C)(C(=O)NCCCCn3ccnc3)C2)=O)nccc(C)c1N C1(O)(CC#C)CC(C(=O)NC(C)(C(=O)NC2(C)CCC2)C2CCC2)C1 N1(C(c2cccc(OC)c2N)=O)CCC2CN(C(C3COCC3(C)C)=O)CC2C1 C(=O)(C(O)CC(C)C)N1C(CC(N2CCC(O)(COC)C2)=O)CCCC1 c1(C(c2nnnn2CCCF)NC(c2ncc(Br)s2)C)cnc2ccc(Cl)cn12 c1(C=O)c(C)cc(C#N)cc1C.C12CC(C1)C2.C1(C(C)C)CC1C=O.CC N1(C(c2c(COC)cc[nH]2)=O)CC(C)C(NC(c2cnc(Cl)[nH]2)=O)C(C)C1 CN1CCC2(CC1)CC(NC(=O)NNC(=O)c1cc(Br)cs1)c1ccccc1O2 CCC(CC(=O)NC1(CNC(C2CC(OC)C2)=O)CCOC1)C1CCC1 C1(NC(C(=O)N(C)C)=O)CC(O)CN(C(c2cc(Br)cnc2S)=O)C1 C1(NC(CSc2cccc(OC)c2)=O)CCN(C(=O)C(C)(F)F)CC1C CC1CCCCC1(C)C(=O)N(CCCNC(=O)COC1(C)CCCC1)CCO c1(C(=O)OC)nc2n(n1)CCC(C)N2CCC1C=CCCC1 C1(CNC(C2CCCN(C(C)C)C2)=O)CCC(C)(C)CN1CCC1CCOCC1 C12(NC(C(C)CCO)=O)CC(C)(C1)OC21CCN(C(=O)CCCCCO)CC1 N1(C(C(C(C)C)O)=O)CCC2(CCCN(C(c3ccc(Cl)[nH]3)=O)C2)C1 C(=O)(CCC(=O)NC1CCCC(NC(C2CCCC23CC3)=O)C1)NCCC N1(C(C2CCCC2(F)F)=O)CCN(C(c2cnn[nH]2)=O)C(c2ncc[nH]2)C1 N1(C(c2c(SC)nn(C)c2)=O)CCC(C)C(NC(c2ccc(Cl)[nH]2)=O)C1 N1(C(C(C)Cn2cccn2)=O)CCSC2(CCCCC2)C1 N1(C(c2cncc(OC)n2)=O)CC2CC(C)C2C1.c1(C(=O)N)cc(O)nc(C)n1 Cc1cncc(C(N2CCN(CCCNC(=O)C(C)CC3CC3)CC2)=O)n1 c1(C2(C(=O)NC3CCN(C(CC(C=C)C)=O)C3)CCC2)cccc(C#N)c1 C1(C(N2CC(C(=O)NCC3(N(C)C)CC3)C(F)C2)=O)CCCC2(CC2)C1 C(CC(=O)N1CC(N(C(=O)CNC2CCC2)CC)C1)OCCOCC Cn1ncc(Cl)c1C(=O)NC(C)(CNC(C1CC1C(N)=O)=O)CO C(=O)C(C)(C)C(F)(F)F.N1(C(C(C)NC(=O)Cn2cnnn2)=O)CCCC1.C C1(CNC(C2C(NC(C)=O)CCO2)=O)COCC1(C)C N1(C(C(F)=C(C)C)=O)CCC(C2CCN(C(c3cccc(N)c3F)=O)C2)C1 c1(C(N2C(C)CN(C(c3cnsn3)=O)C(C)C2)=O)ccc2[nH]ccc(=O)c2c1 C1(NC(c2c(C)cns2)=O)(CF)CCN(C(c2csc(CC(F)(F)F)n2)=O)C1 C=CC1OCCC1C(=O)NC(C1(C(=O)NCC2CC(C)(C)C2)CC1)C c1(NCCC(COC)NC)ccc(S(=O)(=O)NCCN(CCCS)C)cc1Br Cc1cc(O)ncc1C(=O)NC1(C(=O)NCC(C)CCO)CCOCC1 C1(O)(CNC(c2cnc(C)o2)=O)CCN(C(=O)C(C)O)C1.c1ccc(F)cc1 c1(C(=O)NC(C)C(C)NC(c2cc([N+](=O)[O-])cn2C)=O)cc2n(c1)CCSC2 N1(CCCCC(=O)OC)CC(=O)N(CC2CC(O)CCO2)C1=O c1(C(=O)NCCCn2cc(-c3nccs3)nn2)cc(Br)c2c(c1)OCCO2 C1(NC(=O)NC(CC(C)C)CCO)CC12CCCc1ccccc12 Cc1ccc(=O)n(CC(=O)NCC2(F)CCC(NC(C3CCCCN3C)=O)C2)n1 N1(C(c2c(C)noc2N)=O)CC2(CCCCN(C(=O)Cc3csc(S)n3)C2)C1 C(C#Cc1cnn(C)c1)NC(CN(C(=O)Cc1ccccc1)C(C)C)=O C1(C(=O)NCC(C)C)C2C(CN1C(c1n[nH]cc1[N+](=O)[O-])=O)C2(C)C C1(C(=O)NCCC2(C)CCN(C(C(CC)N(C)C)=O)C2)CC(=O)NC(=O)C1 C1(CCCC)CN(C(=O)CC(C)N(C)C)CCN1C(c1c[nH]nc1Cl)=O C1(C(=O)NC2CCN(C(=O)C)C2C)(OC)CCS(=O)(=O)C1.C1CCCCC1.O c1(N2C(C)CC(NC(C(CC)C)=O)C2)ncnc2c1ncn2C1CC1 N1(C(CC2CCC(=O)N2)=O)CC2C(CNC(c3cc(CO)on3)=O)C2C1 c1(C(=O)NCC2N(C(C(C=C)O)=O)CC(O)C2)cc2n(n1)CCNC2=O C1(NC(C(C)(C2CCC2)NC(=O)CN2CSCC2=O)=O)CCn2cnnc2C1 S(=O)(=O)(c1cccc(C(N2CCOCC2)=O)c1)NC(C(C)C)(C)CO N1(C(COCCC=C)=O)CCC2(CC1)C(NC(c1ccsc1)=O)CS2(=O)=O.O N1(C(c2c(C)[nH]cc2)=O)CCC2CC(C1)CN(C(c1csc(C(C)(C)C)n1)=O)C2 CCC(CC)CCC(=O)NCC1CCC(F)(C)C1.c1(C=O)nocc1C(C)C.N c1(C(=O)N)cn(C)c(O)n1.c1(COC)nc(C(=O)NC2CC2C)co1 c1(C(=O)NC(C2(CNC(CSC)=O)CC2)C)cc(N)c(C)cc1C c1(CNC(c2cccc(F)c2F)=O)ccc2c(c1)CCC2NC(c1cocn1)=O C(=O)(C(F)C(C)CNC(=O)CC1CSCCO1)NC1C(C)(N(C)C)CCC1 CC1C(NC(=O)Cn2nc(O)ccc2=O)CC2CCC1N2C(C1(C)CCC1)=O N1(C(c2nc(C)[nH]n2)=O)CC(NC(=O)Cc2c(Cl)cnn2C)C(C2CC2)C1 C1(N(C(C2C(CC)OCC2)=O)C)CN(C(=O)CS(N)(=O)=O)CC12CC2 CC1(C)OC(=O)CC1C(N1CC2CC2(NC(c2cnn(C(F)F)c2)=O)C1)=O C(=O)(C1=CS(=O)(=O)CCC1)N(C(c1ccccc1)C)C.C1(C=O)CCC(=O)N1 N1C(=O)CCC1C(=O)N(CCCC)C.N1(C(C2(C=O)CC2)=O)CCCC1.CC c1(C(C(=O)NCC2(NC(Cn3c(C)ccn3)=O)CC2)C)cccc(C#N)c1 c1(C(N2CC(C)(C(N3CC(C#C)OCC3)=O)C2)=O)cc(C#N)ccc1N CC(C)C(CNC(=O)C(C)(C)n1cnnn1)C(=O)NC(c1ccco1)CO C1(CNC(CSCC#C)=O)CC(C)(C)CN1C(=O)CC1OCCCO1 CCC(CC)C(=O)NCCCN(C1CCCC1)C(=O)C.c1(C(=O)N)ccccn1 C1(NC(CC(n2c(CC)ncc2)C)=O)CN(C(C2CC2F)=O)CC1(C)C C1(CNC(CCC#C)=O)CN(C(c2c(N)sc(C)c2C)=O)CC(C)(C)O1 N1(C(Cn2c(C)cc(C)n2)=O)CC2CCC1C(CNC(c1nnc(S)n1C)=O)C2 Cc1cccn2cc(C(=O)NC3CCCC3NC(=O)CCN(C)CCO)nc12 C(=O)(C1=CCCN(C(c2ccccc2)=O)C1)Nc1c(COC)ccs1 C1(N(C(C(C)OCCC#C)=O)C)CCCN(C(c2ccc(OC)cc2C)=O)CC1 c1(C(=O)NCC(CC=C)NC(C2(CC(C)C)CC2)=O)cc2c(O)ncnc2cn1 C1(CC=O)CCC(F)(F)CO1.N1(C(CCNC(=O)NC)=O)CCC(O)(C)C1 CN1CC(O)CC1(C)C(N1CCC(C)(NC(=O)CCN2CCCCCC2)C1)=O N1(C(C(CNC(C=CC(CC)C)=O)O)=O)CC2CCCCC12 N1(C(c2c(C(C)C)ocn2)=O)CC2COCC2(C(N2CCC2)=O)C1.C(=O)N(C)C C(=O)(CC(CN(C)C)C(F)F)N.C1(OC)CCCC1C(=O)NC1CC(C)C1 C1(C(=O)NCCN(CCC)C(c2cc(C#N)ccc2F)=O)CN2CCCN1CC2 N1(Cc2ccn(-c3c(C(=O)OCC)cccc3)n2)CCCC12CCNC2=O C(CCCC(=O)NC1CCN(C(c2c[nH]c(C#N)c2)=O)C1C)OCC C(=O)(C1=CCCCC1C)N(CCN(C(=O)CCOc1ccc(Cl)cc1)C(C)C)C N1(C(c2cnc(COC)s2)=O)CCCC(NC(c2cnc(O)c(Cl)c2)=O)CC1 N1(C(CN(C(C)C)C)=O)CCN(C(CNC(=O)C(C)(C)C)C(F)F)CC1 C1(O)(C(C)CNC(C2CCCO2)=O)CCN(C(c2cc[nH]c2C2CC2)=O)C1 N1(C(C2CCC(C)C2)=O)CC2CC(C(=O)NCCC3(CO)CCC3)(C2)C1 c1(C=O)ccc2cc(F)ccc2n1.CC1(C)CC2(CC2C(=O)NC(C)CO)C1.N c1cc(F)cc(F)c1.C1(C(=O)OC)C(OC)CCN1C(=O)C.C(=O)NC c1(C(=O)NCC(C)NC(C2C3CCC(F)C23)=O)ncn2cc(Br)sc12 C12(NC(c3ccco3)=O)CC(C1)N(C(c1ccccc1)=O)C2.CC(F)(F)F.O N1(C(c2cncc(SC)c2)=O)CCCN(C(=O)CC(=O)NCC(F)(F)F)CC1C Cc1nc(C2CC2)[nH]c1C(=O)NCCCCNC(C1CCCN(C)C1)=O c1(NC(COC)C(C)C)nc(SCC(C)C)cc(C)n1 c1(N(C2CC(=C)C2)CC=C)ccccc1C(N1CCSCC1C(N)=O)=O C1(Cc2n(CC(C3CCCO3)O)c(CO)nn2)(Oc2ccccc2)CCOCC1 c1(OCC2C(C)(C)C2C(=O)NC)ccc(C(F)(F)F)cc1.c1cccnc1 N1(C(C2(C)CCN(C)C2)=O)CCC(C)(C)C(C(=O)NCCCc2cccnc2)C1 C1(C(N2CCC(COC(F)(F)F)CC2)=O)CCc2[nH]nc(O)c2C1 N1(C(C(C(C)C)C)=O)CCN(C(=O)C(C)(C)c2cnn(C)c2)CC1C(C)C c1(C(=O)NC2CC(NC(C3CC(C)(C)OCC3)=O)C2)ccc(=O)n2c1CCC2 C(=O)(C1CCCn2c(C)cnc21)NCCC(=C)CNC(=O)C(C)(CC)OC c1(N(C)C)cc(N2CC3C(NCCCN4CCN(C)CC4)C3C2)ncn1 c1(C2N(C(=O)NC3CC3c3cscn3)CCC2)c(F)cccc1F c1(CC(C)C)ccccc1C(N1CCC(C(F)(F)F)C1)=O.c1(C(=O)N)cnsn1 C1(NC(c2cn[nH]c2)=O)CCN(C(=O)CSC2CC2)C12CCC2.C1CC1.C CCCCCCNC(=O)C=Cc1cccnc1.C1(CC(=O)N)C(C)(C)C1(C)C C1(NC(C2CC2(Cl)Cl)=O)CCCC12CN(C(c1ccc3ocnc3n1)=O)C2 c1(C(=O)NC(CC2(O)CCC2)C(F)F)cc(C2CCNC2=O)ccc1Cl c1(C(N2CC(CO)(CO)C2)=O)cnc2n[nH]c(-c3sccc3CO)c2c1 c1(C(C(=O)NCC2CCCCC2)N(C2CC2)CCF)cccc2nc[nH]c12 c1(CC(N2CCCC(NC(CC3C(C)(C)C3)=O)CC2)=O)cnn2ccccc12 c1(C(=O)NCCC2CCCN(C(C(C)SCC)=O)C2)c(C)nc2ncnn2c1C C1COCCN1C(c1ccn(C2CCCC2)n1)=O.C(=O)(COCC(=O)N)NC C(=O)(C(O)CCC(C)C)N1CCC(C(=O)NCCCCN=[N+]=[N-])(CC)CC1 c1(C(=O)NC2(CN(C)C(c3cnc(S)[nH]3)=O)CC2)cccc2cc[nH]c12 CC(C)(C)C(CC(=O)N1CCOCC1C1CC1)NC(C1CCCC(C#N)C1)=O N1(C(c2ccc(C(=O)OC)[nH]2)=O)CC2(CCN(C(C3CNC(=O)N3C)=O)C2)C1 C1(CC(=O)NCC(C)C(=O)NCc2cnc[nH]2)CCC(=O)N1C C1(C(=O)NC(CCSCC)CNC(=O)Cc2ccn(C)n2)CCSCC1.O C(=O)(C(C)CNC(C1CC1C1CCCO1)=O)NC1CC(C(=O)OC)C1 Cc1cc(Cl)cc2cc(C(N3CCCC(NC(C4(F)CCCC4)=O)C3C)=O)[nH]c12 c1(NC(N2CCN(CC(c3ccc(C)cc3)C)CC2)=O)cc(C#N)c(C)cc1C N1(c2c(OC)c(C)ncn2)CC(NC(C2(CC(F)F)CCC2)=O)CC(C)(C)C1 Cc1nccc(Cl)c1C(=O)NCCC1CCCN1C(c1cc2ccsc2s1)=O Cc1cc(C#N)c(O)nc1C(N1CC2CC(NC(c3cc(Br)co3)=O)CC2C1)=O c1(-c2c(C)cc(C(=O)O)cc2)ccc(F)c2occc12 S(=O)(=O)(c1ccc(C(F)(F)F)cc1)NCc1ccc(C2(N)CC2)cc1 C1(NC(=O)NCC(N2CCCCC2=O)C)CCC2CC1CN2CCO c1(C(N(C2CCN(C(C3(OC)CC3)=O)C2)CC)=O)cc(F)c(F)c(Cl)c1F C1(C(N2CCOCC2)=O)(CC)CCNC1=O.c1(C(N(C)C)=O)coc(C2CC2)n1 C(C)(N=c1ccn2c(Br)cnc2[nH]1)C1CCN(C(c2c(CC)noc2)=O)CC1 C1(NC(CCC=C=C)=O)(CNC(c2ccnc(C3CC3)c2)=O)CCCCCC1 O=C(C1=CCCCC1)NC12CCN(C(c3ccc(-c4ccncc4)s3)=O)CC1C2 C1(NC(CCc2ncc(C)[nH]2)=O)CCC(CNC(c2ncoc2C(C)C)=O)CC1 C1(CNC(C2(CC)CCCN2C(=O)CC(=O)OC)=O)CCCCN(C)C1 N1(C(c2ccc(-c3ccco3)[nH]2)=O)CCC2(CCN(C(c3cccs3)=O)C2)C1 C(=O)(C1CCCc2ccnn21)N1CCN(C)CC1CNC(c1ccoc1Br)=O c1(-c2cc(NCC(C(=O)OC)C)ncc2)ccc(=O)n(C2CCCCO2)c1 CC(C)CCC(F)C(=O)N1CC(C(=O)NC2CCCC(O)C2)C(F)C1 CC1(C(=O)NCCNC(=O)CCSc2ccc(F)cc2)CC=CCC1 c1(C(N2CCC(NS(=O)(=O)CC3CC3)C2)=O)cc(Br)c(Cl)cc1F C(=O)(C(C)C(CC)CC)N1C(CN(C(c2c(CC)c(C)sc2)=O)C)CCC1 C1(C)CN(C(C2CCC3(CCC3)C2)=O)CC1C.c1(CC)cc(C(=O)NC)ncn1 c1(COC)ccc(C(c2nnnn2C2CC2)NCCCF)o1 c1(C(=O)NC2CCN(C(C(CC)NC(N)=O)=O)C2)ccc(N(C)C(C)C)cc1 C1(O)(C(=O)NC2C(NC(c3ccc(C(N)=O)o3)=O)C2)CC(F)(F)C1 C(=O)(C1c2ccccc2OCC1(C)C)N.C(CCC)NC(CN(C)C(=O)C1CC1)=O Cn1cc2c(n1)CCC(C(N1CC(O)(CNC(c3cccnc3S)=O)C1)=O)C2 C1(CN(CCN(C)C)CCc2ccccc2)CNC(=O)C(C)(C)C1 CC(CCC(C)(C)C)C(=O)NC1CN(C(=O)CCC(C)(F)F)CCC1CO C1(CC(=O)NC2(C)CCCN(C(COC)=O)C2)CSc2ccccc2O1 CCC(CNC(=O)CCCC1(NC(=O)C(C)n2cccc2)CCC1)C(C)C C1(F)(C(=O)OCC)CS(=O)(=O)CC12CN(C(c1sc(Cl)nc1Cl)=O)C2 N1(C(C(C)n2ccnc2)=O)CCC(C#N)(NC(c2nccs2)=O)C1 c1(C(N2CCC(NC(c3c(CC)nns3)=O)C(O)C2)=O)cnc2cc(C)[nH]c2c1 C(=O)(C1NCCc2cc(OC)ccc21)NC1CCC(C)CC1Oc1ccccc1 c1(C(CCC)C)nc(-c2cccc(Cl)c2)n(C2CCCC2)n1 c1(OC)cccc(C(=O)NCCCCC(C)NC(=O)COc2ccsn2)c1F Cc1nc2cnn(C)c2cc1C(=O)NCCCNC(C12COCC1C2(F)F)=O C1(CNC(C2C(C)(C)C2)=O)CC2(CO1)CN(C(=O)CC1CC13CC3)C2 C1(CC(=O)NC(C(=O)NC23CC(C2)C3)C2CCOC2)CC2C=CC1C2 C1(N(C(c2cc(OC)no2)=O)C)CCCCN(C(=O)CC)C1.C1(C(=O)N)CCC1 NC(=O)C(O)CN=c1ccc(Br)c(S(=O)(=O)NCC2CCOCO2)[nH]1 CC1(C)C(NC(=O)CCC(F)(F)F)CCN1C(=O)COc1cnc(Cl)cn1 C1(C)(NC(CCN(C(C(c2ccc(C)o2)C)=O)CCO)=O)C(C)(C)C1(C)C Cc1onc(O)c1C(=O)NC(CNC(=O)CC1CC(F)C1)C(C)C C1(NC(C(CC(C)C)C)=O)CN(C(C2CCCC23CCC3)=O)CCC12CCC2 C(=O)(CCCC(F)(F)C(F)(F)F)N1CCC(NC(COCC#C)=O)C1(C)C C(=O)CC(C(C)C)C(C)C.n1(CCC)cccc1C(=O)NCC1CC(C)CO1 C1(C(N(C2(CC(=O)N(CCC(=O)OC)C)CC2)C)=O)CCN(C)C(=O)C1 N1(c2ccc(Cl)c(OC)c2[N+](=O)[O-])CCc2c(F)ccc(C(=O)OC)c2C1C c1(NC(C(C)NC(=O)OC)=O)cccc(NC(=O)CCC2CCC2)c1 C1C(O)C(O)CN1C(=O)CCN(CC(F)(F)F)C.CN1CCC(C(=O)N)C1.C N1(C(C2C(C)CCOC2)=O)CC2(CO)CC1(C(=O)NOCC(F)(F)F)C2 C(=O)(C1=CCCC1)N(C(CNC(C(c1ccccc1F)(C)OC)=O)C)C c1(C(=O)NCC(CN(C(=O)CCSC(F)(F)F)C)O)cncc(C(N)=O)c1 N(C1c2ccccc2CC1NC(=O)CC1CCCCC1O)C(CCC(N)=O)=O N1(C(c2c(CC)cccc2)=O)CCC(F)(F)C1.C1(Cl)(C=O)CC1C(C)=O.C CCCC(CC)C(=O)N1CC(c2cn(CCOC3CCOC3)nn2)C1 c1(C(=O)NC2CC3CC2N(C(C2(C4CCCO4)CC2)=O)C3)nc2cnccc2s1 C(=O)(C1CCc2ccccc21)N(C)CC1(O)CN(C(c2cccc(C#C)c2)=O)C1 C(=O)(C1CCCc2nccn21)NCC1CC(C)(C)N(C(c2ncncc2Cl)=O)C1 c1(OCCCOC)cccc(-c2nc(C(C)CC)nn2C2CCCC(C)C2)c1 N1(C(c2n(C)ncc2Br)C(=O)NCCC2(C)CC2)CCc2ccccc2CC1 CC(C(=O)NCC1CCCCC1)S(N)(=O)=O.C(=O)C(C)(C)CC1CC1.C N1(C(C(C(C)CNC(=O)C(c2cccn2C)=O)F)=O)CCC2(CC1)CC2C#N c1(C(N2CCC(O)(C(CNC(CC=C)=O)C)C2)=O)ccc(O)c(Cl)n1 c1(CCCC)nc(CN(C(=O)C(N)Cc2nccn2C)C)c(Cl)[nH]1 C(=O)(CCCN=[N+]=[N-])NC1(C(=O)NCc2cc(OC)ncn2)CCCC1C C1(C(=O)NCCC(C(C)C)NC(C(C=C)c2ccccc2)=O)CCC(C)C(C)C1 N1(C(C(C=C)C2CC2)=O)CC2CCCC(C1)N2C(C)C(N1CC(C)CC(C)C1)=O C(C)(CCCC)NC(CC1(NC(CCSCCCC)=O)CCCC1)=O.C(C)=O.N C1(C)(NC(C2(NC(CCCCN(C)C)=O)CC(O)C2)=O)CCCC1(F)F C(=O)(CN=c1cc[nH]cc1)N(C(CC(=O)NC(C#C)CC1CCCC1)(C)C)C Cc1nc(N2CCC(CNC(=O)C(C)C3CCCO3)CC2)c2c(C)c(C)sc2n1 CC1CN(C(=O)CCc2ccsc2)CC1NC(=O)CC1CNC(=O)C1 C1(NC(c2cnc(CC)s2)=O)CCC2(CC1)CC2.C(c1cncs1)=CC=O.N N1(C(C=C)=O)CCC(NC(c2cnc(O)n2C)=O)C(CO)CC1 C1(N(C(c2ncn(CC)n2)=O)C)CCC(NC(C23CSCC2C3)=O)CC1 N1(C(CCC=C)=O)CC2(CC(NC(=O)C(c3ccccc3F)C)C2)C1 C1(CCOC)CCN(C(=O)CN2CCCCC2)C1.C1(C=O)CC(C(N)=O)C1.N n1(C(C)C)ccc2c(N(C3CNCC3O)C(c3ncc(C4CC4)[nH]3)=O)ncnc12 N1(C(c2n(CCC)ncc2)=O)CCN(C)CC1C(=O)NC(C)CC(F)(F)F N(C(=NCCN(C(C)C)C(C)C)NC1CCCC1)C1CCN(CC)C1 C1(CC(=O)NC(CN(C(=O)C(C)(C)C2CCOCC2)C)(C)C)CCC1C1CC1 N1(C(c2cc(C)c(N)cn2)=O)CC2(C)CN(C(=O)C(C)(C)C(C)(F)F)CC2(C)C1 C1(CCC(=O)N(CC(C)C)CCCO)CCN(C(C2(CO)CCOC2)=O)C1 c1(C(N)=O)ccccc1C(=O)NCC1(C(=O)NCCCCN(C)C)CCC1 CC1CC(C(N)=O)CN(C(C2(O)CC(NC(c3ccco3)=O)C2)=O)C1 c1(C(N2CC(NC(C(CC)N(CC)CC)=O)C(O)C2)=O)c(C)ccc(C)c1C C12(NC(Cn3c(=O)ccc(C)c3)=O)CCCC1N(C(=O)CC1OCCO1)CCC2 C1(S(C)(=O)=O)(C(N2CCCC(F)(F)C2)=O)COC(=O)C1.C(CC(=O)N)=C(C)C C(c1ccccc1)=CC(C)C(N1CC(NC(=O)CCc2ccco2)C(C)C1)=O C12(C(=O)NC3CC(N(C)C(C4CC(O)C4)=O)C3)CC(C)(C1)OC2(C)C C1(CCCCNC(c2ncc(F)cn2)=O)CCCN(C(=O)C=Cc2ccc[nH]2)C1 c1(OCC(=O)NC(CCCNC(C(C)(CO)OC)=O)C)c(C)nn(C)c1C c1(C(N2C(CCNC(CC=C=C)=O)CCC2)=O)ccc(C(=O)OC)c(C)c1 Cc1csc(CCC(=O)NCC(C)NC(C2(c3ccn(C)n3)CC2)=O)n1 N1(C(C(C)SCC)=O)CCCC(NC(=O)C(C#N)CC)C1 CC(CC(=O)NCC1CCC1NC(c1csc(Cl)n1)=O)P(C)(C)=O CCC(C)CC(=O)NCC(c1cccc(Cl)c1)NC(c1ccsc1)=O C(c1ccccn1)=C(C)C(=O)N(CCCN(C)C)CC.C1(C=O)CC(C)CO1.N C(=O)(C1CCNc2c(C)cccc21)N1CCC(O)(C(C)NC(C=CCOC)=O)C1 N1(C(CCN(CC)CC)=O)CC2CC1CC2NC(=O)CCc1cncs1 N(C(=NCCC(C)(C)C1CC1)NCC1CCOC1)Cc1cc(C(C)C)no1 N1(C(c2c(OC)c(Cl)ncc2)=O)CC2CCC(C1)N2C(C1OC2CCC1CC2)=O N(C1CCCc2c(F)ccc(F)c21)CC(c1ccccc1I)O c1(C(N2C(C)CC(CNC(CSCC)=O)C2)=O)snc2ccccc12 C1(N(C(C(C(C)C)CO)=O)C)CC2CCC(C1)N2C(c1cccc(N)c1F)=O N1(CC(=O)NCCCNC(=O)Cc2cccnc2Cl)CCS(=O)(=O)CC1 c1(-c2n(CC)ncc2)cc(CN(CC(=O)O)CCO)cc2c1OCO2 C1(O)(CN(C(C(C)O)=O)C)CCN(C(=O)Cc2cncc(O)c2)CC1 n1(-c2cc(C)on2)nnc(-c2nc(C3CC3C)nn2Cc2cccc(Br)c2)c1C C1(O)(CNC(Cc2c(C)con2)=O)CCCN(C(=O)CC(=O)Nc2nccs2)C1 CCCCCC(C)(CC)C(=O)NC(C)CCCNC(=O)CC1CCCC(C)C1 c1(C(=O)NCC(C(C)(C)C)NC(Cc2ccc(C)cc2)=O)nc[nH]c2ncnc1-2 Cc1cc(C(=O)N(C2CCCN(C(C3CCC(=O)NC3)=O)CC2)C)nc(C)c1 C1(C(=O)NCCCCN(C(CCN(C)CC)=O)C)CC2(CCCCC2)CO1 c1(NC(=O)NC(C2CCN(c3nnc(C)o3)CC2)(C)C)cc(C)cc(C)n1 C(=O)(C(C)CC(F)F)NCC1C2CN(C(C3(COC)CCCC3)=O)CC21 C(=O)(CCCC(=O)NC1COCC1Cc1cnn(C)c1)c1ccc(OC)cc1 N1(c2cc(N3CCC(SC)C3)nc(C(F)(F)F)n2)CCCC2(C1)NC(=O)NC2=O N1(C(CCC(=O)NCCC)=O)CCCC(O)(CNC(c2cc(C)sn2)=O)CC1 N1(C(CCC(C)OCC)=O)CCOCC(NC(c2cc(Cl)ns2)=O)C1 N1(C(CCC(C)OCC)=O)CCC2C(C1)NC(=O)CCN2C(c1cc(C)on1)=O C(=O)(C1=NOC(C)C1)N(C1CCCCC1)C.C1(OC)(OC)CC(C(=O)N)C1.C C(=O)(C(O)C(F)(F)F)N1C(CC)C(C(=O)N)CC1.CCC(C1CC1)C1CC1 c1(C(c2n(C(CC)C)nnn2)Nc2cnsc2)scc(C)c1C C(=O)(C1=Cc2ccccc2C1)N1CC(CC)C(NC(=O)C2=C(C)CCC2)CC1 c1(C(=O)NC2C(CNC(CS(CC)(=O)=O)=O)C2)nccc2[nH]ccc12 N1(C(=O)OC)CCC(O)C1C(=O)NCC(=O)N.c1nc(C(F)(F)F)sc1C c1(C(N(C(C)CNC(C2(CF)CCC2)=O)C)=O)cc(F)cc(Br)c1O C(C(=O)N1CC2CC(C1)C2)(C(C)(C)C)SC.c1(N)cc(C(F)(F)F)nc(C)n1 C1(CNC(C2CCC(=C)CC2)=O)CC2CCC1N2C(=O)CC.CCN(C)C.O c1(CN2CCC(NC(C3CCCN(C)C3)=O)CC2)cc(I)cc(I)c1O c1(C(=O)NCCNC(CSCC(C)C)=O)cc(C2(C)COC2)no1 Nc1ccc(F)c(C(N2CC(CNC(c3ccon3)=O)C3(CC3)C2)=O)c1 c1(N(C)C)ncccc1C(=O)NCC(C)(O)CNC(=O)CC1(C)CCC1 C1(CC(=O)NCC2(O)CCN(C(=O)Cn3ccnn3)C2)CC(C2CC2)C1 c1(C(=O)NCC2CN(CC)C(=O)C2)cnc2c(Br)cccn12 c1(OC)cc(N(CC(C)CNC(=O)C(C)N2CCC2)C)nc(OC)n1 c1(CN2CC3N(C(c4cnc(Cl)nc4)=O)C3C2)cc(C(F)(F)F)ccc1O C=CC(C)(O)CC(=O)NC.C1(C)CCN(C(c2ccc(C(F)F)c(F)c2)=O)CC1 c1(C(CCSC)NCC(F)CO)nnnn1C1(C)CC1 N1(C(=O)CC2CCCO2)CCCCC(NC(C23CSC(C2)C3)=O)C1 C1(C2CN(C(C3CCCN(C(=O)Cc4cnsc4)C3)=O)C2)(NC(C)=O)CC1 C1(CC)C(NC(c2cccs2)=O)CCN1C(=O)CC(O)CN(C)C C(CC(C)(C)C(=O)N1CCOC(C2CCC2)C1)NC(CC1ON=C(CC)C1)=O c1(CC)cccc(C(N2CCCC(N(C(=O)C(CC)CO)C)CC2)=O)c1F C(CCC(C)C)NC(C1(OCC)CCOC1)=O.C1(C=O)CN(C(C)=O)C1.N N(S(=O)(=O)N1CCN(c2cc(N(C)C)nc(C(C)C)n2)CC1)(C(C)C)CC c1(OC)ccc(Cl)cc1NC(c1cnc(C)c(C)c1)c1nnnn1C1CCC1 CC1CC(NC(=O)C2=COCC2)CCN1C(c1cccc(CO)n1)=O C1(C=O)CCC2CCCCN12.n1(CC(C)C)nccc1C(=O)NCC1CCC1.N N1(C(C2(S(N)(=O)=O)CC2)=O)CCCN(C(c2cc(F)ccc2O)=O)CC1 N1(C(C2N(C(C(C(=O)OC)OC)=O)CCC(O)C2)=O)CCn2ncc(O)c2C1 C1(CCC(=O)NCCCOC(=O)NC)CCN(C(c2ccc(F)s2)=O)C1 NC(=O)CC(O)C(=O)N1CC(O)CC1CNC(=O)C(F)C(F)(F)F c1(COC)ccc(NC(=O)CCCc2ccncc2)nc1 Cc1ccc(C2CCCN2C(=O)NCCO)cc1C c1(CCOC)nnc(N2CCCC2C(C)(C)NC(=O)Cn2ccnc2C)s1 CCC(CNC(C1CC(C)(NC(C2CC(C)(C)CO2)=O)C1)=O)C(C)C Cc1nn(C)c(N)c1C(N1CC(C(N2CC3(C2)CN(C)C3)=O)C(C)(C)C1)=O N1(C(c2[nH]c(=NCC)sc2)=O)CC(NC(c2ccsc2C)=O)C2CCCCC12 N1(C(CNC(C=CCN(C)CC)=O)=O)CC(C)N(CC)CC1C N1(C(CCc2scc(C)c2)=O)CC(NC(=O)CCc2ccoc2)C(F)C1 N1(C(COCCC)=O)CCC(O)(C2(NC(c3ccc(OC)cc3C)=O)CC2)CC1 Cc1nnc2cnc(C(=O)NC3CC(NC(=O)C=Cc4ccc(Cl)cc4)C3)cn12 C(=O)(C(F)(F)C(F)(F)F)NCC12N(C(CCC(=O)N(C)C)=O)CC(C1)C2 CC1CN(C(c2coc(Cl)n2)=O)CC1NC(C1CC(N=[N+]=[N-])C1)=O CC1CCN(C(=O)C(C)(C)n2cnnn2)CC1.C1(C=O)CC(C)(C(C)(C)C)C1.N c1(OCC)cc(OC)ccc1C=O.CCC1CCC1.C(=O)C=CC=O.N C1(C(=O)NC(CC)CNC(c2ccc(OC)c(O)c2)=O)CC2C=CCC(C1)C2 N1(C(CCC(=C)Cl)=O)CC(C)(C)CC1CNC(=O)CC1COC(=O)C1 Cn1nnc2cc(C(N3CC4CC3CN4C(C3(CF)CCOCC3)=O)=O)cnc12 Cc1nn(C)c(N)c1C(N1CCN(C(c2csc(NC3CC3C)n2)=O)CC1)=O c1(SCC)ncc(C=O)cn1.N12CCOC(C1)C(=O)Nc1nc(cs1)C2=O.N c1(C=O)cc(C)n(C)c1.c1(C(C)OC)nc(CC(=O)NCC2CCC2)cs1 C=CCC(C(=O)NC1CCN(C(c2ccc(C)s2)=O)CC1)C(C)(C)C c1(NC(CNC(C2(CCC)CC2)=O)CO)ncnc2cnccc12 C1(OC)C2CC3CN(C(=O)CC(C(F)(F)F)n4cccn4)C1C3C2 N1(C(c2sccc2CC#N)C(=O)NCCC2(C)CC2)CCC(S(C)(=N)=O)C1 c1(N(C(CC)=O)C(C)C)c2c(nn1C)CCSC2.Cc1ccc(C(=O)O)c(I)c1C C1(NC(=O)NCCN(C(=O)OC)C)CCN(c2ccccc2Cl)C1=O C(=O)(C(C)CC(F)(F)F)N1CC(CC(C)NC(c2c(OC)c(F)ncc2)=O)C1 C1(C(=O)NC(C=C)(C)CC)CN(C(C2CC(N(C)C)C2)=O)CC12CC2 CC1CC(NC(=O)CC2CCCSC2)CN1C(=O)CN(C)C C1(C)(CNC(C(C(C)C)SC)=O)CN(C(c2csnc2C)=O)C(C)(C)C1 c1(C(C(=O)NCCCC)N(C)C(C)C2CC2)nc2ccc(OC)cc2s1 Cc1ncc(C(=O)NCC2(NC(=O)C(c3cccc(O)c3)C)CCCC2)n1C Cc1cc(C)c(C(N2CC3(CC(NC(=O)C(C)n4ccnc4)CO3)C2)=O)c(N)c1 CC(CC(=O)N1CCCC(F)(CNC(=O)COC2CCCC2)CC1)C(F)(F)F c1(OC(C)C)ccc(C(N2CCCCCC2)=O)c(Cl)c1.C1(C(=O)N)CC2(CC2)C1 CC1CC(NC(C2(C)CC(O)CN2C)=O)CCN1C(=O)CN1CCNC(=O)C1 c1(C(=O)NCC(CC)NC(=O)Cc2sc(C)nc2C)nnc2ccccc2n1 CCCCC(C)C(=O)NC(C(=O)NCCN1CC(CF)C1)C1(O)CCC1 C(=O)(C(CC)C(F)(F)F)N1C(C(=O)NCC(CC)N2CCCC2)CC2CC21 c1(C(N2CC(C)C(NC(C3(C)CS(=O)(=O)C3)=O)C2)=O)ccc([N+](=O)[O-])s1 N1(C(c2ccc(C)[nH]2)=O)CCC2(CCCC2NC(C2CCCS(=O)(=O)C2)=O)CC1 c1(C(N2C(C)CN(C(CCC#CC)=O)C(C)C2)=O)cncc2ncn(C)c12 Cc1cccc2cc(C(=O)N(C(C)CN(C)C(C3(C)CC(F)(F)C3)=O)C)nn12 N1(C(C(C)n2cncn2)=O)CC(CNC(=O)C=Cc2ccsc2)CC12CCC2 Cc1ncc(C(=O)NC(C)C=CC(N2CC(n3cnnc3)C2)=O)c(=N)[nH]1 c1(OC)ccc(C(=O)N(CCC(C)NC(C2(F)CCC2)=O)C)c(C)c1 c1(C(C)C)nc(Cl)cc(=NC2CC(O)(CNC(c3ccc4cc[nH]c4n3)=O)C2)[nH]1 c1(C(=O)NCC2N(C(Cc3cccc(CC)c3)=O)CC2)ccc2[nH]ccc2n1 C1(F)(C(=O)NC(C(=O)OC)(C)CO)CCCN(C(c2ccc(C#N)[nH]2)=O)C1 C1(C(N2CC(F)CCC2)=O)CNC(=O)C(C)(C)C1.Cc1csc(=O)n1CC(=O)N C1(NC(CC(COC)C)=O)(CO)CCN(C(=O)C(C)OC2CCOC2)CC1 Cc1nc(C(=O)NC2CC2NC(=O)C(c2cccnc2)NC2CC2)cn1C c1(CCC(N2CC3(CN(C(C(C(CC)C)O)=O)C3)C2)=O)ccc2ccccc2c1 N1(C(CCS(=O)(=O)NC)=O)C2CCC1CN(C(C1CCOC(C(F)(F)F)C1)=O)C2 N1(CC)CCCC(C(=O)NCC2CCCCN2C(c2nccs2)=O)C1 C1(C(N(C2CCC(O)CC2)C)=O)CC(C)(C)CCN1C(=O)C=CC(F)F N1(C(C(CC)OC)=O)CCOC2CN(C(c3cnc(-c4cnccn4)s3)=O)CC12 C(=O)(CCCC(=O)N1CCC(CNC(=O)CN2CCCCS2(=O)=O)C1)NC c1(C(=O)NC(CNC(C2(C)CC2(F)F)=O)(C)C2CCC2)nnc(O)nc1O Cc1ccnc2c(C(=O)NCC(CO)NC(c3nsnc3O)=O)cccc12 C1(NC(COCCOC)=O)COCCN(C(=O)C=C2CCSCC2)C1 C1(C(=O)NCCOCCN(C(CCCOC(C)C)=O)C)COCCC1(F)F C(CCCCC(=O)NCc1c(C)coc1C)N(C(=O)C=Cc1ccc[nH]1)C C1(C(=O)O)CCCC(NCc2ccncc2F)CC1 C1(C(N(C2CCN(C(C=CCOC)=O)C2)C2CC2)=O)CC(OC)C(O)C1 c1(C(N(CCNC(C(C)OCC=C)=O)C)=O)cccc(C(C)(F)F)n1 C1(C(=O)NCC)(OC)CCC(F)(F)CC1.c1ccccc1F.C1(C(=O)N)CC1 CC1CN(C(c2ccsc2Cl)=O)CC(C)N(C(=O)CC2CC2(C)C)C1 C1(F)(CNC(CCSCC)=O)CCCN(C(c2cc(C(C)C)oc2C)=O)CC1 CCCC(C#N)C(=O)NCCOC1CCN(C(=O)CC(C)(C)SC)C1 C1(O)(CC(=O)NC(c2ccc(C)o2)CC)CCN(C(=O)CCC(C)N(C)C)CC1 C=CCC(CC(C)C)C(=O)N1CC(O)CC1C(=O)NCC(C)(CC)C(N)=O c1(C(N2C(C(C)(C)NC(C(C)CN(C)C)=O)CCC2)=O)cc2n(n1)CCCO2 Cc1nc2sccn2c1C(=O)NCCNC(c1cnn(C2CC2)c1Cl)=O C12(NC(c3cnns3)=O)CCCC1CN(C(c1cc3ccccc3[nH]1)=O)C2 c1(-c2cn(CCNC(C(C)NC(=O)C(C)(C)C)=O)nn2)cn(C)nc1C#N C(CC(C)C(=O)N(C)CC1(CNC(c2cccc(S)c2)=O)CC1)=CC c1ccc([N+](=O)[O-])cc1.C1(NC(C(C)C)=O)CN(C(=O)C)CC1C(F)(F)F.S C1CN(C(c2cnc(C(C)C)s2)=O)CC1(C)C.CCS(=O)(=O)NC(C)C=O.N C1(NC(C(CCC)C)=O)CCC2(CCCN2C(c2cncc(C#N)c2)=O)CC1 C1(C(=O)NC2C3N(C(CCCC=C)=O)CC(CC3)C2)C2C3CC4C1C1C2CC3C41 C(C(O)C(=O)NCc1nc(C(=O)NC2C=CC(C(=O)NC)C2)co1)OC n1(CC)c(C)cc(C(N2CCCCC2CNC(c2ncnn2CC)=O)=O)c1C CC#CCC(C(=O)N(C)Cc1cccnc1)NC(=O)CCCSCCC C1(NC(CN(CCC#C)C)=O)CCCC1NC(c1cnc(Br)s1)=O CC1(CS(N2CCC(c3csc(Br)n3)C2)(=O)=O)CCCCC1 Cc1cc(Cl)c(C(=O)NCC2CCC(C)CN2C(c2cn[nH]c2)=O)cc1C c1(C(=O)NCC(C)OC)conc1CNC(c1ccsc1)=O N1(C(C(C)NC(C)=O)=O)CCCC(C)(NC(=O)C(C)OCCC(C)C)C1 C(C)(CCC(=O)NCCN1CCC(CO)C1)NC(c1nc(C(C)C)oc1)=O N1(C(COC)=O)CCC(N(C)C(c2cc(-c3ccccc3)co2)=O)C1 C12(C(=O)NC3CC4CN(C(=O)CCSC(F)(F)F)C3C4)C3CC(CC13)C2(F)F N1(C(c2cc(F)cc(F)c2)=O)CCC2CN(C(=O)Cc3cccc(Cl)c3)C2C1 N1(C(C=C(C)C)=O)CCN(C(CNC(c2ccccc2C)=O)C(F)F)CC1 C1(CC)C(C(=O)NC2(C)CC(NC(=O)CC(C)CN(C)C)C2)CCN1C c1(C(N2C(CC)(CC)CC2)=O)oc(CNC(C2C3CCC(F)C23)=O)nc1C C1(C(=O)OC)CC2CCCCC2N(C(c2[nH]c(C)c([N+](=O)[O-])c2C)=O)C1 c1(C(N2CC(CCCCNC(CCSCCC)=O)C2)=O)n[nH]c2c1CCC2 c1(C2(N(C(=O)NCc3ncc(C)o3)CCO)CC2)cccc(Br)c1 c1(C(=O)NC2C(CS(N)(=O)=O)CCCC2)c(C(F)(F)F)cncc1Cl N1(C(COC2(C)CN(C(C(CC)(CC)OC)=O)C2)=O)CC(C)OC(C)(C)C1 Cc1ccc(C(=O)C=CC(=O)NCCCCC(C)NC(C2CCC2(C)C)=O)cc1 C(=O)(C(C)CC(C)C(C)=O)NCC12CCC(C(N3CC(C=C)C3)=O)(OC1)C2 C1(CNC(c2c(CC)scn2)=O)CCCCN1C(C1COCC1(C)C)=O Cc1cc(C(N2CCCC(N(C)C(C3CC(C)(C)CO3)=O)C2)=O)ccc1[N+](=O)[O-] Cc1ccc2sc(C(=O)NC)c(C)c2c1.C1CCCN(C(=O)CN(C)C2CC2)C1 c1(C(N2CCC(O)(CN(C(C3CCCN(C)C3)=O)C)C2)=O)cc2cnn(C)c2s1 C1(NC(CCC=C)=O)CCCCC1NC(=O)COc1ccon1 C(=O)(C1=CNC2=NCCC2=C1)NC(C(C)NC(=O)CSc1ccccc1Cl)C N1(C(C(C(C)C)OC)=O)CC2CC(C)N(C(C3C4CN(C)CC34)=O)C2C1 c1(C(=O)NC2CN(C(c3cc(C)c(Br)o3)=O)CC2C)nn(C)c(N)c1C CC(C)C(C(=O)NC1(c2cccs2)CC1)C(C)NC(c1ccc(O)cc1)=O N1(C(c2n(C)ccc2)=O)CCN(C(=O)C(c2cnn(C(C)(C)C)c2)=O)C(CF)C1 C1(C(N(C2CCN(C(CCN)=O)C2)C)=O)CC2(C1)CC(F)(F)C2.CC[SH](=O)=O C1(CNC(c2csnn2)=O)CCCCN(C(c2cccc(-c3nc[nH]n3)c2)=O)C1 N1(CC(C(CC)C)O)CCCC(C)(C(=O)NC(c2ccc(Cl)cc2)C(=O)OC)C1 c1(C(N2CC(C)C(CNC(c3ccc(CCF)cc3)=O)C2)=O)cccc(Cl)c1N c1(C(C(=O)NCCCC2(O)CC2)NC(C=CC)=O)ccccc1 C1(CC)CN(C(=O)C(C)NS(C)(=O)=O)CC1.c1ccccc1C.C(=O)(C)N Cc1cnncc1C(=O)NC1CC1NC(=O)C(C(C)C)Sc1ccccc1 N1(C(Cn2ncc(C#C)c2)=O)CCC(O)C(C(=O)N(C)Cc2nnc(C)s2)C1 N1(C(C(c2ccn(C)n2)C)=O)CCN(C(=O)CC(F)(F)F)CC1C C12(C(N3CCC(NC(C4C(C)C4C)=O)C3)=O)CC(CO)(C1)OC2C C1(C(=O)NC2CCN(CC)C2)C2CC1N(C(C1(F)CCCC1)=O)C2 c1(CC(=O)NCC2(C)CN(C(=O)C(F)F)C2)ccc(OC(F)(F)F)cc1 C1(NC(c2cccc3c2OCC3)=O)CC2CN(C(C3CC3C3CC3)=O)CC2C1 S(=O)(=O)(c1cc(Cl)ccc1OCC1CCCCO1)N(CC(F)F)C C#Cc1cnn(C)c1C(=O)N(CC(=O)NCC1CCOCC1C)CCOC C(=O)(CC(O)C1CCCC1)N1CC(N(C(=O)COCC2CCCC2)C)C1 c1(C(=O)NCC(N(C(c2c(C)noc2)=O)C)C2CC2)c[nH]c2cccnc12 N1(C(c2c(OC)noc2C2CC2)=O)CCCC(C)(C)C1.C(=O)CC1CC1.N CC1(C)C2CCC(C(=O)NC)C1C2.C1(O)CCCN(C(=O)C=C2CCC2)CC1 C1(C(N(CCNC(C(CCC)OC)=O)CCOCCO)=O)Cc2ccncc2C1 C1(C)(C=O)CCC(C)CC1.C1(CNC(Cc2cnc(C)[nH]2)=O)(C)CC12CCC2 N1(C(=O)OC(C)(C)C)CC(NCc2cc(C3CC3)on2)C2CCC1C2 CC#CCCC(=O)NCCCOCCC(=O)NC1(C(O)CO)CC1 Nc1cc(F)c(C(=O)NCC23CCC2CN(C(C2CC4CC4C2)=O)C3)c(F)c1 c1(C(=O)N)c(N)ccc(F)c1F.C1(CCC)CCC(C(=O)NCC(C)(O)C)CC1 N1(C(C(CC=CC)C)=O)CCC(C)CC1CNC(c1cc(C)on1)=O S(=O)(=O)(c1cccnc1NCCc1ccccn1)N1CCCC(C)(CC)C1.OC c1(C(=O)NC2CCN(C(CCNC(C)=O)=O)C23CCC3)ncnc2c1OCCO2 c1(C(C(=O)NCC(C)OC)O)cnn(C)c1.C1(C(=O)N)CC1.C(C)=O c1(CN2CC(C(=O)NC3CC(=O)NCC3)OCC2)ccc(F)cc1O N1(C(C(COC)NC(C)=O)=O)CC(F)(F)CC1(C)C.c1(CC=O)cc[nH]n1 N1(C(C(COC)O)=O)CCN(C(c2[nH]ccc2C)=O)CC1CS(C)(=O)=O c1(C(=O)N)ccc2c(c1)N(C)CC2.N1(C(CS(=O)(=O)NC)=O)CCC2CC2CC1 Cn1c(C(=O)NC2CC23CCN(C(=O)C2=CCCCO2)CC3)cc2c1CCOC2 C1(C(=O)N)CC(c2ccccc2F)=NO1.N1(C(COCC=C)=O)CC2C(C)C2C1 N1(C(=O)C=CC(F)F)CCOC(CNC(C23CCC(C2)C3)=O)C1 c1(C(N2CCC(NC(C3C(C)(C)C3)=O)C2)=O)cccnc1OC(F)F N1(C(C(C)SC(C)C)=O)CCN(C(=O)C(c2ccccc2)=O)C2CCC12 C1(NC(C(CC)SC)=O)C=CCN(C(=O)C(C(C)C)c2ccncc2)C1 CC(C)(C)CC(O)CC(=O)N1CCC(NC(c2ncc(P(C)(C)=O)cn2)=O)C1 CCC(C(=O)NCC1CCCN1C(C)=O)N(C(=O)CCCOC)C Cc1ccc2c(c1C)N(C(=O)CCC1CCN(C)C1)CCC2 c1(CC(C)C)ncc(C(=O)NCCC)s1.c1(CCC(=O)N)nc(C(C)C)no1 N1(C(c2cccc(OC)n2)=O)CC23CCCC2(C1)CN(C(C1CCOC1)=O)C3 C1(NC(C2C(C)(C)C2)=O)CCN(CC(=O)N)CC1.C1(F)(C=O)CCC1.CC C(=O)(CC1C(=O)Nc2ccccc21)N1CCN(C(CCSCC)=O)C2C1COC2 c1(C(N2CC3CC2C3CNC(C2(O)CC2)=O)=O)c(F)ccc(F)c1Cl c1(C(=O)NCC2OCCN(C(c3cc(C)ncc3)=O)C2)cccc(C)c1C C1(C(N)=O)CCC(C(N2CCCC2CCCNC(=O)C=CCO)=O)CC1 c1(OC)cccc(Cl)c1C(=O)NCC1CCC(C)N(C(=O)Cc2cncs2)C1 n1(CC(N2C(CNC(=O)C(O)c3ccsc3)COCC2)=O)cc2ccccc2n1 c1(CC)nc(Cl)[nH]c(=NCCCNC(c2sc(C)cc2NC)=O)c1Cl n1(CC)cnc2c(NC3CCCSC3)[nH]c(=NCCCS(=O)(=O)CC)nc12 C(=O)(CC1OCCc2ccsc21)NC1(C)CCN(C(c2cccc(C)n2)=O)C1 Cc1cc(CNC(=O)NC2(C)CCCC2C)nc(Cl)c1Br CC1CCCC(C(=O)NCC#CCNC(C2CCSCC2)=O)CC1 C#CC1CC2CC1N(C(=O)C(C)Oc1ccc(CC)cc1)C2 N1(C(C(C)(C)SC)=O)CC2CC(NC(c3ccc(C#N)n3C)=O)C(C2)C1 N1(C(c2c(=O)cc(C)[nH]c2)=O)CCC(C2CC2)C1CNC(c1cncnc1)=O CC1CC(C)(CNC(C2CCN2C(=O)C(F)CC2CCOC2)=O)C1 C1(N(C(Cn2c(C)nnn2)=O)C)CC2CCC(C1)N2C(C1(C(F)F)CC1(F)F)=O c1(C(N2CC(CNC(C3C(OC)C3)=O)(O)C2)=O)ccc(C(C)C)cc1 Cc1ncc2c(n1)CCC(C(=O)NC1CN(C(c3ncc4[nH]ncc4n3)=O)C1)C2 c1(-c2ccc(CSCCCC)cc2)cc(C(=O)OC)c2nc(C(=O)OC)cn2c1 C1(NC(C2(C#C)CC2)=O)CCCCC1CNC(C1CCC(F)C1)=O CS(=O)(=O)c1ccc(NC(C2CC2NC(=O)NC2CC(O)C2)=O)nc1 CC(C)(CC(F)F)C(=O)N1CC(CNC(C2(C)CC2(Cl)Cl)=O)C(C)(C)C1 N1(C(C(C)C2CCCC2)=O)CC2(C(=O)NC(C)(C)CC3CCC3)CC1CO2 C1(C(=O)NCC(CNC(c2n[nH]cc2C2CC2)=O)OC)(C)CCCCC1 c1(C(N2C(CCNC(c3c(C(C)C)ocn3)=O)CCC2)=O)cccc2c1OCO2 n1(CC)cc(Cl)cc1C(N1CCCC1C1CCN(C(c2cc(C)sc2C)=O)C1)=O C=C(CNC(N1CCNC(C)C1)=O)c1ccc([N+](=O)[O-])cc1 C12(C(N(CCCCC)C)=O)CCN(C(c3cc(C)cc(O)n3)=O)CCC1C2 C1(NC(CNC(CCC)=O)=O)C=CCN(C(c2scnc2C(F)(F)F)=O)C1 CC1CC(NC(=O)CC(C)(F)F)CCN1C(C1C=CC=CC=C1)=O C1(N(C(C(CCC)C)=O)C)CC2CCC(C1)N2C(=O)C(c1ccccc1)F N1(C(C(C)(C)OC)=O)CC(C)CC(C)C1.C12(C=O)CC(CC(F)F)(C1)C2.N Cc1n[nH]c(C)c1CCNC(=O)N(C)CCN(C)C(C1CCN(C)C1)=O C(CCC(C)C(=O)NCCC1CCCN1Cc1ccc(Br)c(F)c1)OC c1(OC)c(N)nc[nH]c1=NCC(O)CN1Cc2cc(OC)ccc2C1=O N1(C(Cc2ccc(C)s2)=O)CCN(C(C2CCC23CCCO3)=O)CC1CO c1(C(F)(F)F)ncc(NC23CC(C2)C(c2ccccc2)N3)nc1OC CCCC(CC)C(=O)N1CCC(N(C(=O)CCOc2cc(Cl)ccc2Cl)C)C1 c1(CCC)cccc(C(C(=O)NCC2CC2)N(C2CC(C(=O)OC)C2)C)c1 c1(C(c2n(CCCC)nnn2)Nc2csnc2C)cccc(C(=O)NCCC)c1 C1(NC(CSCCOC)=O)CCC12CN(C(c1cc(OC)no1)=O)C2 c1(C(=O)NC2(CO)CCN(C(C(CC)(C)CO)=O)C2)ccc2snnc2c1 N1(CCCNC(C2C(C)CC2)=O)CCN(C(C2CC(n3cnnc3)C2)=O)CC1 Cc1c(C(=O)NC2CC2)cnn1-c1cccc(Cl)c1.C(C1CCC1)=CC=O.N C#CCC(CC(=O)OC)NC(C1CC1C1CN(C(=O)CC2CCC(C)C2)C1)=O C1(N(C(c2ncoc2C)C(=O)NCCCC)C)CC(C)(C)CC(C)(C)C1 N1(C(CC2CC(=C)C2)=O)CCC(C(=O)NCC2(O)CCCCCC2)(CC)CC1 C1(C=O)CCOC(C)(C)C1.C1(CNC(C(C)NC(C)=O)=O)CCCCC1.C N1(C(c2c(COC)cco2)=O)C2CCC1CCC2.C(=O)(C(O)Cn1cncn1)N C1(CCNC(C(CC)SC)=O)CCN(C(=O)C(=Cc2cnc[nH]2)C)CCC1(F)F C1(C(N2CCCC(CC)C2)=O)CCC2(CN(C(c3cncc(F)c3)=O)C2)O1 C(CC(C)C)(C(=O)N1CCC1C(=O)NC1CCN(CC)C1)NC(C)=O C1(C(=O)NCC2CC(NC(C3CC34CCC4)=O)C2)(CC)CCOCC1 c1(C(N2CC(c3cnco3)C2)=O)nc(Cl)ccc1F.C(C(C)=CC(=O)N)OC.C CC1(CNC(=O)C[SH](=O)=O)CCCN1C(c1ccc(CCF)cc1)=O.C1CC1 c1(CNC(c2ccc(Cl)cc2)CC(=O)Nc2c(C)coc2C)cc(F)ncc1C N1(C(=O)C=CCN2CCCC2)CCCC2(CNC(c3csnc3Cl)=O)CCCC12 C12(C(N(CC(C3CC3)NC(C3CC(N(C)C)C3)=O)C)=O)CSC(C1)C2 C1(C(=O)NC(CN(C(=O)CCc2nccs2)CC)C)COc2ccc(F)cc2C1 C1(C(=O)NCc2cccs2)(CC)CCCN1C(c1cnn(CCO)c1)=O N1(CC)CCOC(C(=O)N(CC(C)(C)C(=O)NCC(C2CCCCC2)O)C)C1 Cc1ncncc1C(=O)NCC1(CC(=O)N(C2(C)CCCC2)C)CC1 CC1CCCCN1CC(=O)NC(C12CCC(CC1)C2)C.C1(C=O)(CCF)CC1.N C1(C2CC2)CCN(C(c2cncc([N+](=O)[O-])c2)=O)C1.c1(C(=O)NC)ccnnc1 c1(C(=O)NC2(C)CCCC(F)(F)C2)cnc(P(C)(C)=O)cn1 c1(OC)c(F)ccc(C(N2CC(CNC(C3CC4CCC3O4)=O)CC2C)=O)c1F Cc1cnccc1C(C)CNC(=O)NC(C)(CN(C)C)C1CC1 C1(C(=O)NC(C)(C)C(=O)NCC2CC3(CC3)C2)CC(O)C(F)C1 C(=O)(C(C)(C)C(C)C)NCCC(=O)NC(CC(=O)OCC)C N1(C(CC2CCN(C)C2)=O)CCN(C(c2cc(Cl)c(Cl)c(Cl)c2)=O)C2(CC2)C1 CCC(CC)CCC(=O)N1CC(OC)CC1(C)CNC(C1(OC)CCCC1)=O CCCCC(O)C(C)C(=O)NCCCCC(C)NC(=O)C(C)Cc1cnn(C)c1 C#CC1(O)CCN(C(=O)C(CCC(C)C)NC(C2C=CCC2)=O)CC1 c1(CC)ccc(CNC(=O)C)cc1.C1(C)CN(C(=O)CC2C=CCCC2)C1 c1(C(=O)NCCN(C(=O)CCCN2CCCCC2)CCC)ccc(Cl)cn1 C1(NCC2ON=C(C)C2)CCN(C(=O)OC(C)(C)C)CC1(F)F C(=O)(CC1=CCCC1)NC(CCCC)CNC(=O)C(C1CCC1)OCC N1(C(COCCOC)=O)CC2CCC1C2.c1(C(=O)N)[nH]nc(C(F)(F)F)c1C c1(C(=O)NCC(C)CNC(c2cccc3nncn23)=O)cnc2n1C(C)CCC2 CC1CCN(C(c2snc(O)c2Cl)=O)C(CNC(=O)Cc2ccccc2F)C1 c1(CC)n[nH]c(CC)c1CC(=O)NCC1CCCCC1.c1(C(=O)N)nocc1C c1(N2CCCC(OCC)C2)ncnc(N2CCN(C3CCCN(C)C3)CC2)c1C CCCCCN(CCC(=O)N(CCCCN(C)C(C1CC1c1cn[nH]c1)=O)C)C Cc1ccc(S(=O)(=O)N2CC3CC2CN3C(=O)C(C)Cc2ccccc2)c(F)c1 N1(C(C(CCC)NC(C2CCC(O)CC2)=O)=O)CCn2c(O)nnc2C1 c1(C(=O)OC)cc(C(=O)NCC(O)CNC(=O)C=CCF)c[nH]1 Cc1cc(N(C)CCN(C(C2(O)CC2)=O)C(C)C)n2ncc(C)c2n1 c1(OCC)cc(CNCC2CC3CC3C2)ccc1OC(C)C C(c1cccc(F)c1)=CC(=O)N(CCCNC(C(c1cccc(C)c1)C)=O)C Cc1coc(C)c1C(N1CC(CNC(c2cn(C)nn2)=O)CC1C)=O.C1CC1 c1(C(=O)NCC2(NC(C(C(C)C)C)=O)CCOCC2)cc2c(Cl)cc(F)cc2[nH]1 Cn1ncc2c(C(=O)NC3CCCN(C(=O)CCCS(N)(=O)=O)C3)ccnc12 C(N=c1cc[nH]c(-c2ccccc2)c1)C12C(CN(C(c3ccc(F)cc3Cl)=O)C1)C2 c1(C(N2CCCC(SC)C2)=O)cc(N)ccc1Cl.C(=O)(C(F)(F)F)NC(C)C C(=O)(C1CCC(=O)c2ccccc21)NC(C1(n2cc(CC(C)O)nn2)CC1)=O C(=O)(C=C=C(C)C)NCc1ncc(C(=O)OCC)[nH]1 c1(CNC2CN(C(C3CC4C=CC3C4)=O)CC(F)(F)C2)c[nH]c2ncc(Br)nc12 C1(NC(CC(=C)C)=O)C2CC1CN(C(c1cc3cscc3s1)=O)C2 N1(C(CCCC(=O)NCC)=O)CC(C)OC2(CCN(Cc3cnn(C)n3)CC2)C1 Cc1cc(CCCC(=O)NC(C)(CNC(C2(CCO)CC2)=O)CO)on1 CC1CN(C(c2ccccc2Cl)=O)CC1NC(=O)C(O)Cc1cnc[nH]1 C(C(C)(CC(C)C)NC(c1ccc(C)c(OC)c1)=O)NC(C=CCC)=O n1(C(C)C)cccc1C(=O)NC1CN(C(C2(C)CCCO2)=O)C1 C(=O)(CCCCCC(C)O)N.c1(CNC(C2CC=C(C)CC2)=O)ccc(C)c(F)c1 c1(C(N2C3CN(C(CS(C)(=O)=O)=O)C(CC3)C2)=O)cnc2c(Br)cccc2c1 c1(NC(C2CC2C(N2CCC3(CC2)CC3)=O)=O)cc(Br)cc2cn[nH]c12 c1(CC(=O)NCCNC(=O)C2=NOCC2)ccc2c(c1)COC2 C(=O)(C1=C(Cl)CCC1)N1C(C(N(CCC2CN(C)C2)C)=O)C=CC1 c1(C(=O)NCC(CC)NC(C(C=C)c2ccccc2)=O)ccc2nc(C)oc2c1 Cc1ccc(C)c(CC(N2CCCC(NC(=O)C=Cc3cncn3C)C2)=O)c1 C=CC(F)(F)C(=O)NCC1CC1CNC(=O)C(c1cccc(C)c1)O C1(C(=O)OC)C=CC1C(=O)NCC1CC1.C(=O)(CCc1cnco1)N C1(NC(C2(N(C)C)CC2)=O)CCC(C)(C)CC1.C1(C)(C=O)CCN(C)C1=O C1(N(C(=O)Cc2cc[nH]c(=N)c2)C)CCCCN(C(=O)C(F)(F)C2CC2)C1 C(=O)(CC1=CCCC1)NC(CCOCC)C(=O)NC1CCCN(C)C1=O N1(C(CC2CCC(NC(c3c(C)ccs3)=O)C2)=O)CCC(O)C(F)(F)C1 N1(C(COCC(=O)OC)=O)CCC(O)(CNC(=O)C(F)CC(C)C)CC1 Cc1cc(C=O)n2ncnc2n1.C1(O)(CC)CN(C(=O)C=CCN(C)C)C1.N Cc1cccc(C(=O)N(C2CCC(NC(c3cccc(O)c3F)=O)CC2)C)c1F C1(NC(c2c(C)n(C(C)C)nc2)=O)CCSC12CN(C(C1CCS1(=O)=O)=O)C2 CC(C)C(C(=O)N1CC(F)(C#N)C1)NC(c1nnsc1N)=O C1(NC(c2cnc(S)nc2)=O)CCCN(C(c2n[nH]cc2C(F)(F)F)=O)C1 Cc1n[nH]c(C)c1C(C)C(N1CC(NC(=O)CCCc2cnn[nH]2)CC1C)=O C12(C(=O)NCCN(C)C(C3C4CCC3(c3cnco3)C4)=O)CCCCC1C2 c1(CC(N2CCC3C(NC(c4cc(SC)oc4)=O)C32)=O)cn2cc(C)sc2n1 Cc1coc(C(C)(C)C)c1C(=O)NC1CCCCC1N(C(=O)CC=C(Cl)Cl)C N1(C(C(C2CC2)SC)=O)CC2CCCC(CNC(=O)Cc3cn[nH]c3)C2C1 c1(C(N2C3C(NC(CCCC(=O)NCC)=O)C(C3)C2)=O)c(O)ccc(F)c1C c1(C=O)ccc(Cl)c(C(F)F)c1.n1(CC)cc(CC(=O)NC2CCC2)cn1.C C(=O)(C(=O)N=S(C)(C)=O)N1CC(N(C(=O)C(F)CC2CCOC2)C)C2(C1)CC2 c1(C(C)=O)cc(C(=O)NCc2ccc(Cn3ccnc3)o2)n(C)c1 N1(C(c2n(CCCC)ncc2)=O)CCOC(CNC(=O)C(C)CC)C1 C1(C)(C(=O)NC)CCN(C(=NCCF)NCC(Cc2ccco2)CO)C1 c1(C(N2CCCC(N(C(=O)CS(C)(=O)=O)C)C2)=O)cc(F)c2cn[nH]c2c1 c1(OC)ccc2[nH]c(=NCc3cnccn3)[nH]c(=NCC(=O)NCC(F)F)c2c1 c1(C(N(C2CCCN(C(=O)CCn3c(C)csc3=O)C2)CC)=O)[nH]c(C)cc1C CC(CC(=O)NCC1CCCN(C(=O)CC2CCCC2)C1)C(=O)c1ccccc1 C(=O)(C(C)(N)CC1CCC1)NCc1c(C(C)(C)C)noc1 N1(c2n(CCCOC)c(C(O)C3CC3)nn2)CCC2(CCC(=O)N2)C1 C12(CCNC(C3CC(N(C)C)C3)=O)CCC(C1)N(C(c1cc(Cl)ccn1)=O)C2 c1(C(=O)NCC(C)(CO)NC(Cn2ccc(C)n2)=O)snc2ccccc12 Cc1ccc(CCc2nc(CN(C)C)nn2-c2ccccc2C)cc1 c1(OC)cccc([N+](=O)[O-])c1CN1CCSCC1C(=O)NC(CO)C1CC1 N1(S(c2ccc(NC(COC)CO)nc2)(=O)=O)CCn2c(n[nH]c(=O)c2=O)C1 C(C)(CC(=O)NCCn1cc(CC2(O)CCSC2)nn1)(C(F)(F)F)N(C)C CC1=C(C(=O)NC2CCC(N(C(=O)Cc3ccc(Cl)s3)C)CC2)C(C)(C)CCC1 c1(C(N)=O)c[nH]c2ncnc(N3C4CCC3CN(C(c3c(Cl)nsc3Cl)=O)C4)c12 C1(O)(CCOC)CN(C(C2(CNC(=O)CC3CCOC3)CCCC2)=O)C1 c1(C(N2CCCC(C)(NC(=O)COC3CC3)C2)=O)cc(O)c2ccoc2c1 Cc1cc(C#N)ccc1C(N1CC2CC2(C(=O)NCCCN2CCCC2=O)C1)=O C(=O)(C(C)(C)C(=O)NCC1(CNC(c2n[nH]cc2Br)=O)CCC1)OC c1(OC(C)C(=O)N(CCCCN(C)C(C2CC2(C)C)=O)C)ccccc1Br C1(C(N2C3C(NC(c4ccc(CO)nc4)=O)CC(C3)C2)=O)Cc2ccccc2S1 c1(C(N2CCOCC2(C)C)C(=O)NCCCSCC)n[nH]c2ccccc12 c1(C(=O)NC(CCN(C(c2scc(C)c2)=O)C)C)ccnnc1C C12(NC(CC(C)CN(C)C)=O)CCOCC1CN(C(c1csc3nccn13)=O)C2 C1(C(N2CCC(C(N(C(c3nn[nH]n3)C)C)=O)CC2)=O)CC2CCC1CC2 C12(C(=O)NC(CNC(C3(OCC)CCOCC3)=O)C)CCCC1CC(=O)CC2 c1(-c2nn(CCCC)c(C3CCSC3)n2)ccc(Br)c(C)c1 c1(C(=O)NC(CCNC(C(CCCC#C)C)=O)C)[nH]c2ccccc2c1C1CC1 C1(C(N2C(C(=O)NC(COCCOC)C)C=CCC2)=O)CCCCCCC1 c1(Nc2nnc(OC)s2)ccc(-n2ccnc2)c([N+](=O)[O-])c1 N1(C(CC(CC)C)=O)CCC2C1CCCN2C(c1cnc2nccn2c1)=O Cc1nn(C)c2c(NC(C)CC(C)C(F)F)nc(N3CCC(OCF)CC3)nc12 N1(C(C(COC)C)=O)CCCCC2(C1)CN(C(=O)CSc1ccccc1Cl)C2 c1(C(=O)NCC(c2cccc(OC)c2)NC(C(CC)F)=O)c(C)nc(C)n1O C1(O)(CN(C(C(C(C)O)N(C)C)=O)C)CCCN(C(=O)CC2CCC=CCC2)C1 c1(CC(=O)NC2C(NC(C3(C)N(C)CCC3)=O)C2)cccc(S(C)(=O)=O)c1 c1(OC)c(CNC(=O)C(C)CC2CC2)cnn1C.C1(CC=O)C=CCCC1 N1(C(c2cc(C)cs2)C(=O)NCCCC)CCC(C)(N(C)C)C1 C1(C#N)(C(=O)NC2CN(C3CN(C(C(CC)CC)=O)C3)C(=O)C2)CCSCC1 C1(C(=O)NC(c2cncc(F)c2)C)CCN(C(=O)Cn2ccnc2)CC1 C12(C(=O)NCC(=C3CN(C(C=C(CC)CC)=O)C3)F)CCC(C)(C1)OC2 c1(C(CNC(=O)NC(CC=C)Cc2ccccc2)O)ccc(F)c(C)c1 C1(NC(=O)Nc2scc(C)n2)CC2CC(N)C2C1 C12(C(N3C(C)(C)CCC3)=O)CCC(N=[N+]=[N-])(CC1)C2.C(=O)(C(O)C1CCCC1)N CC(C(=O)N1CCC(OCCNC(c2cccc(CC#N)c2)=O)C1)C(C)(C)C N1(Cc2c(C)ccc(C3CC3)c2)CCC(=O)N(CC2(Cl)CC2(F)F)C1=O c1(NC2CCCCN(C(CC(CC=C)(C)C)=O)C2)nc(C)nc2sc(C)c(C)c12 c1(OC)ccc(C)c(NC(=O)C(F)CC2CN(C(c3cc[nH]c3)=O)C2)c1 C1(N(C(C(CC)OC)=O)C)CCCCN(C(=O)CC2CCC2)C1 CC(C)(F)C(C)(F)C(=O)N.CC(C)S(C)(=O)=O.N1CCCC1.C1(C=O)CC1 C=Cc1cncc(C(=O)Nc2cnc(C)nc2C(=O)OCC)c1 N1(CC)CCOCC1C(=O)NCC1C2CN(C(=O)CO)CC12.C1CCOC1 N1(CCCC(=O)NC)CC=C(c2c[nH]c3c(C(=O)OC)cccc23)CC1 c1(C(=O)NC2C(NC(CC(C)CN(C)C)=O)COCC2)cc(F)c(N)c(F)c1 C1(CNC(C(CC)n2cccn2)=O)CC2CC2N1C(C1CC2(CC2)C1)=O c1(OC(C)(C)C)ccc(CC(=O)Nc2c(C(C)C)ccc(C)c2)cc1[N+](=O)[O-] N1(C(CC(CC)CN(C)C)=O)CC2CC(C1)CN(C(C1(C)CC1(C)C)=O)C2 N1(C(CCOCC#C)=O)CC(CNC(c2ncc(F)cn2)=O)CCC1C c1(C=O)cnc2cnccc2c1.Cc1nnsc1C(=O)NCC1CC(O)(C)C1.N N(S(=O)(=O)N1CCC(O)C1)C(C1CC(n2cccn2)C1)=O N1(C(Cc2c(C)noc2)=O)CCC(C2CCN(C(C3C=CCC3)=O)CC2)C1 Cc1cccc(C(N2CC(CC(=O)NC(c3nccn3C)C)C3(CC3)C2)=O)c1N Cc1ccc(C(=O)NC2(C(N3CCCN(C)CC3)=O)CCC(C)(C)C2)cc1O C1(CC=C)(NC(c2cc(O)n(CC)n2)=O)CCN(C(c2nnc(C)s2)=O)C1 C(=O)C1CNC(=O)c2ccnn21.c1(C(=O)NCC(C)OC)sccc1C1CC1 c1(COCCC(=O)NCC2CCN(C(C3CCC3)=O)C2)ccccc1 CON(CCC(=O)N1CCCSCC1C)C(=O)C1COCCN1C C1(NC(Cc2cnc(C)s2)=O)CCC2(CC1)CN(C(C1CC(=O)CO1)=O)CCO2 c1(C(=O)NCC(C)(CNC(C2(O)CCC2)=O)OC)cc(C)ccc1C C(=O)(C1=CC2CCCCCCC12)NC1(CNC(=O)Cc2cscn2)CC1 C1(NC(=O)CC2CCC(O)C2)CC2CC(NC(c3c[nH]c(=O)cn3)=O)C1C2 C1(C(=O)NC(C)C)CCCCN(C(c2cccc(F)c2)=O)C1 N1(C(c2c(CC)c[nH]n2)=O)CCC2(CC1)CC(C(=O)O)=NO2 c1(CC)ncc(C(=O)NC2CN(C(=O)CCC(C)c3ccc(Br)cc3)C2)n1C C=C(CNC(=O)C(O)CC)CCNC(C1(CC(=O)OC)CC1)=O c1(CC)nnc2cc(N(CCNC(=O)C(C)=C(C)C)C3CC3)ncn12 C12(CNC(C3CCN(C)C3)=O)CC(CO1)C2.c1(CC(=O)N)ccc(Cl)cn1 Cc1cc(C)n(C(C)C(=O)NC2CCC(NC(=O)CCC(C)C)CC2)n1 C(C(COC)CC(=O)N1CCC(C)CC1C(=O)NCC(C)C1CCC1)OC Cc1cc(C)c(OCC(=O)NC(C2CN(C(c3nn[nH]c3Cl)=O)C2)C)c(C)c1 C(C(N=c1[nH]nc(O)s1)C(C)C(C)C)NC(C1(c2c(C)cccc2)CC1)=O Cc1ccc(F)c(C(=O)NC2CC3CC2N(C(=O)C(C)Cc2ccco2)C3)c1 c1(C=O)cc(S(C)(=O)=O)co1.CC(C)(CF)C(=O)NCC1(C)CCC1.N C1(C(=O)NC2C(CNC(C(C3CC3)OCC)=O)CCC2)CCCCCN1C C1(CC(=O)NC(C(C)C)CNC(=O)C(C)(C)c2cccnc2)CCCCC1(C)C C1(C)(CNC(CC(C)F)=O)CCCN(C(c2c[nH]nc2-c2ccsc2)=O)C1 CCCCCCC(C)(CCC)C(=O)N1CCC(CCCNC(=O)C(C)OC)CC1 Cn1nc(O)cc1C(=O)NCCc1ccccc1.c1(C2C(C=O)C2)cnc[nH]1.N C(CS(=O)(=O)CC(=O)N1CCCCC1CC(=O)NCCC(C)F)OC N1(C(c2c(CNC(C3ON=C(C)C3)=O)noc2)=O)CC23CCC2(COC3)C1 C(N=c1[nH]cc2ncnc-2[nH]1)C1CN(C(CN(C2CCSC2)C)=O)C1 C=CCCC(C)(C)C(=O)NC1CCN(C(c2ccc(C(N)=O)o2)=O)C1C N1(C(c2cc(CC)on2)=O)CCC12CCN(C(c1cc(OC)ccc1C)=O)CC2 N1(C(C2(C)CCCS2)=O)CCC(C2CC2NC(=O)C(F)(F)CC2CC2)CC1 Cc1cc(NC(=O)Cc2cnns2)ccc1NC(c1c(F)cccc1F)=O C(CN=c1[nH]c(=N)[nH]cc1I)N(C(=O)CC(F)(F)F)C C(=O)(CCCCC(F)(F)F)N1CC(N(C(=O)CCOc2ccccc2)C)C(F)C1 C1COCCN(C(=O)C(F)(F)C2CC2)C1.C1(CC)CCCCC1OCC(=O)N.C Cc1ccc(C(=O)NC2CC(C(=O)NCC3CCCO3)C2)c(Cl)c1Cl C1(NC(=O)C=Cc2ccc(F)nc2)CCCC12CN(C(=O)CCOC1CC1)C2 c1(CC)cc(C(=O)NC2CC(NC(=O)CC(=O)OC)C2)ncn1 C1(NC(C(COCC)C)=O)C2CC3CN(C(c4ccsc4OC)=O)C1C3C2 C1CN(C(C2CCC(C#N)CC2)=O)C(C)(C)C1.c1(N(C)C)nc(Cl)c(C(=O)N)s1 C(=O)(C(F)CC(C)(C)C)NCC1(CCNC(CC(COC)C)=O)CC1 c1(C(N2CC(C3CN(C(c4cc(C)oc4)=O)C3)C2)=O)cnc2nc(O)ccc2c1 C(=O)(C#CC1CCCOC1)N1CC(C(=O)OC)Cn2c(cnc2)C1 N1(C(COCCC=C)=O)CCC2(CNC(=O)CNC(=O)O)CCCCC12 C(C(=O)N1CCC(C2(C)N=N2)C1)(C(C)(C)C)NC(C1N(C)CCCC1)=O C(CCC(=O)NC(C(=O)N(C)CC1CCCS1)C1(O)CCC1)=CCC=C C1(C(=O)NC(C)CCNC(=O)C=CC2CC2)CCc2ccccc2O1 c1(OC)cncc(C(N2CC(CNC(=O)C=Cc3ccoc3)C(O)C2)=O)n1 CC(C)C(C)C(C)CC(=O)NC1(C)CCN(C(c2n[nH]c(O)n2)=O)C1 C1(NC(COc2cccc(CC)c2)=O)CCCCN(C(C2CCCCS2)=O)C1 C#Cc1cc(C(=O)NC2CCN(C(=O)CCS(C)=O)C(C)C2)ccc1C c1(C2C(C(=O)NC(C)CN(C)C(C3(C(F)F)CCOCC3)=O)C2)ccccc1F c1(OCC)ccc(C(N2CC3CC(NC(=O)C(C)CC4CC4)C2C3)=O)cc1C C12(C(N(C)CC3C(C)C3)=O)CCC(CC1NC(c1cnc(Cl)s1)=O)C2 N1(C(CCCCCOCC)=O)CCCN(C(=O)COC(C)(C)C)CCC1 C1(C(=O)NC2C3N(C(C(N)=O)=O)CC(CC3)C2)CSC(c2ccccc2O)=N1 N1(C(c2c(OC)nccc2)=O)C(C(=O)NC2CC(C)(O)C2(C)C)CCC12CC2 N1(C(C(=O)Nc2cccc(CC(=O)OC)c2)=O)CCN2CCCNC(=O)C2C1 Cc1cc(Cl)ccc1CC(=O)NCC#CCNC(c1ccnc(C(F)F)c1)=O c1(OC)ccc(Cl)c(CNCC2(NC(c3cocn3)=O)COC2)c1 c1(N(C(CCNC(CCCC)=O)C)C)nc2c(cc1Cl)C(=O)OC2 CC(C)CCCC(=O)NCCCOCCC(=O)NC1CN(C(N)=O)C1 CC(CC(F)(F)F)N(C)C(C1OCCC1NC(C1CCC(=O)NC1)=O)=O C1(C(=O)NCC2N(C(Cc3c(C)nc[nH]3)=O)CCCC2)CC2CCC(C1)N2C C1(NC(=O)OC(C)(C)C)COC2(C1)CN(C(N1CCC(O)C(O)C1)=O)C2 C1(C(N(CCCNC(=O)CC2CCSCC2)CC)=O)Cc2cccc(OC)c2O1 c1(NC)cnc(C(=O)NC2CCCC2NC(c2[nH]c(C3CC3)nc2C)=O)cn1 CC1CN(C(=O)C(F)C(F)(F)F)CCN1C(c1cncc(F)c1)=O C(=O)(CCCC(C)CCC)N(C)CC1N(C(C2CC(O)(CC#C)C2)=O)CC(F)C1 N1(CC)CC(C(=O)NC2CCC(NC(C3CC(OC)CC3)=O)CC2)CC1=O.O CCCCC(CNC(=O)C(F)=C(C)C)NC(=O)CCC(C)OCC C#Cc1ccc(C(=O)NCC(C)(CC(C)C)NC(=O)CC2CC2(Cl)Cl)cc1 C=CCCC(C(=O)NC1(CO)CC2CCCC12)NC(=O)C(C)N=[N+]=[N-] C(c1c(Cl)cccc1Cl)=C(C)C(=O)NC(C)(C)CNC(=O)Cc1nccn1C c1(C(C=O)=O)ccc(F)c(C)c1.N1(C(C2(OC)CCSC2)=O)CC2CC2(C)C1 C(=O)(C1Cc2ccc(Cl)cc21)NC1CCN(C(Cc2c(C)ocn2)=O)C1C CC1CN2CCN1CC2C(=O)NC1CCCN(C(=O)C(F)(F)C2(O)CCC2)C1 C(=O)(C(C)(F)C(C)(C)F)N1CC(NC(c2csc3nnsc23)=O)CC(C)C1 Cc1cccc(C(N2CCC(C)(C)C2C(=O)NC(c2ccccc2F)C)=O)c1N c1(C(=O)Nc2cn(C)c(C(=O)N(CCO)CCO)n2)c(O)ccc2ccccc12 N1(C(COC(CC)(C)C)=O)CC2COCC(C1)C2NC(=O)CS(=O)(=O)C1CC1 C(N=C(NCC(c1ccncc1)C)NC(C)CF)C1N(CC)CCC1 c1(C(C(C)C)N(C)CCOC)nc(CC(CO)C2CC2)no1.c1ccccc1 CC1(CNC(c2cc3c[nH]nc3s2)=O)CCN(C(C2CC23CC3)=O)CC1 N1(C(c2occ(OC)c(=O)c2)=O)CCCN(C(=O)CCc2ccn(C)n2)CCC1 Cc1c[nH]nc1C(=O)NC1CC(n2cc(C3(C(C)C)CC3)nn2)C1 c1(C(N2CCc3cnccc3C2)=O)ccc(-c2cc3sccc3s2)c2cc[nH]c12 C1(OC)(CNC(=O)C)CCN(C(=O)CC2CCCCC2O)C1.c1ccncc1.S C1(CN(C)Cc2nn(C)cc2Br)CN(C(c2n[nH]cc2I)=O)CCO1 c1(N(CC(CN(C)C(C2CCCC23CC3)=O)O)C)c([N+](=O)[O-])cnn1C CC(C)C(C)(C)C(=O)N1CC(N(C(=O)CCC(C)N(C)C)C)C(C)(C)C1 CC1CN(C(c2ccc(C3CC3)o2)=O)CC(C)O1.C(=O)(C(C)(C)n1cnnn1)N CCC(CC(=O)N(CC(N1CCC(CC)(CO)C1)=O)CC)C(C)C C(C(=O)NC1CN(C(=O)C)C1)(C(C)(C)C)NC(C)=O.C1CCN(C)CC1.O C(CN=c1ccnc(NC2CCOc3ccccc32)[nH]1)Oc1sccn1 C1(C(=O)NCC(CN(C)C)(C)C)CN(C(=O)CN2CC(C)(C)C2)CCN1C N1(C(C2(C=C)CCOCC2)=O)CCN(C(=O)CCCC(=O)NCC)CC(C)(C)C1 N1(C(c2cccc(OC)n2)=O)CCC(C2CC2)C1C.C(=O)C.C(=O)C1CC1 C1(C(N2CCC(CCCC)C2)=O)CCN(C(=O)CC2CC(=O)C2)C(C)(C)C1 c1(C(=O)NC(CC=C)CO)n[nH]c2cccc(-c3cc(C)c4n[nH]cc4c3)c12 c1(C(=O)NCC2CC2)cccc2nc(O)oc12.C1(C(=O)N)CCn2cncc2C1 c1(N(C)Cc2ncc(CC)s2)nc2ccccc2nc1NCc1cnc(O)[nH]1 C1(CNC(CNC(CCC)=O)=O)CN(C(=O)C(C)(C)CC2CC2)CCO1 C1(C(N(CC(C)(C)NC(C2CCOC2(C)C)=O)C)=O)CCC2(CCC2)C1 C1(CC(c2on(C)c(=O)c2)=O)CCC(C2CC2)C1.N12CCC(CC1)OCC2=O c1(OC(C(=O)NC(C2(C)CC2)C)C)ccccn1.c1(C(=O)N)n[nH]cc1Br Cc1ccc(Br)cc1CC(N1CCCCC1C(=O)Nc1ccc(I)c(CO)c1)=O N1(C(C(CCC)C)=O)CC(NC(=O)Cc2ccno2)CC12CCCC2 C1(NC(C(CC)F)=O)C2CC(CN(C(c3cccc4ccnn34)=O)C2)C1CO C1(CCC)CN(C(c2cocn2)=O)CC1C(=O)NC(c1ccc(C)nc1)C N1(C(C2C(C(C)C)OCC2)=O)CCC(CC(=O)N(C)Cc2cn[nH]c2)CC1 C1(O)(CNC(C2N(C)CCC2)=O)CCN(C(c2cnn(CC(F)F)n2)=O)CC1 N1(C(c2ncc(OC)nc2)=O)CCOC2CN(C(c3c[nH]nc3[N+](=O)[O-])=O)CC12 N1(C(C(N2CCn3ccnc3C2)C)=O)CCC(C)N(C(=O)C2=CCCOC2)CC1 C1(C(C(=O)NCCCOC)NC(=O)CCOC(C)=O)CC=CCC1 Cc1oc2ncnc(O)c2c1C(=O)NCC1CC(F)CN1C(c1cnc(S)[nH]1)=O CCC(C)(F)C(=O)NCCCCCCN(C)C(C1CCCN1c1cnccn1)=O CC(C)S(=O)(=O)c1ccccc1C(=O)NC1C2CCC(C2)C1c1ccccc1 N1(C(Cn2cc(-c3n(C)nc(C)c3N)nn2)=O)CC2(CCC2)CC1C N1(C(Cn2cc(C(=O)OCC)nn2)=O)CCC2CCC(C1)N2C(C1CCCS1)=O c1(C(=O)NCC(CC=C)NC(=O)CC2CCCCO2)ccc2occc2n1 CC1(c2ccc(CNC(=O)CCC(N)CC3CCCCC3)s2)NC(=O)NC1=O N1(C(C(C)N(C(c2n(CC#C)cnn2)=O)CC)=O)CCS(=O)(=O)CC1 C12(NC(CC(C)N(C)C)=O)COC(C1)C(NC(=O)C(F)(F)CN(C)C)C2 CC1(O)CCC(C(=O)NC2CCN(C(c3cscn3)=O)C(C3CC3)C2)CC1 N1(C(C(CC)SC)=O)CC(NC(C2(C)CS(=O)(=O)C2)=O)CC12CCCCC2 N1(C(C2(COC)COC2)=O)C2CCC1CC(N(C)C(c1cn3ccnc3s1)=O)C2 c1(C(=O)NC2C3CC(NC(Cn4c(C)nnn4)=O)CC32)ccc2nn[nH]c2n1 C12(NC(CCSC)=O)CCOCC1CN(C(c1ccccc1CN(C)C)=O)C2 N1(CC(=O)NC(C)(CO)CO)CCN(Cc2ccc(O)cc2O)CC1=O c1(C(=O)NCC2C(C)CCCN2C(=O)CCCC(F)F)ccc2c(c1)CCN2 c1(C(=O)NCC(CCCC)NC(=O)C(CC)OC)cccc2nn(C)cc12 C(c1cccnc1)=CC(=O)NCC1C(NC(=O)COC2CC2)C1 N1(C(c2c(C)cc(F)nc2)=O)CCC2(C1)CN(C(C1CCC(C)(C)C1)=O)CCO2 C1(C(=O)NC2CC(CCOC)C2)N(C(C2CC(N=[N+]=[N-])C2)=O)CC12CCCC2 c1(C(=O)NC(CC)(C)CNC(C2CC23CCC3)=O)ccc(-c2nc[nH]n2)nc1 N1(C(C(CC)F)=O)CCCN(C(=O)COc2ccccc2C)CC1CO N1(C(c2cccc(O)c2Cl)=O)Cc2ccnn2CC(NC(=O)C(F)(F)CO)C1 C1(CCNC(c2cn(CC)nn2)=O)CCCCN1C(=O)CNS(=O)(=O)NC O=C1CN(C2CCCN(C(=O)NCc3nc(C4CC4)no3)C2)CCN1 c1(OC)cccc(C(=O)N(CCC(C(C)C)NC(=O)CC(C)(O)C2CC2)C)c1C N1(C(=O)CO)CC2CCC(C1CO)N2C(C1CCCS(=O)(=O)C1)=O C1(C(C(=O)NC2CC2)NCc2ccc(CC)o2)CCCCCC1 C1(C(=O)NCC2C(NC(c3ccc(O)cc3)=O)CCCC2)CN2CCN1CC2 C1(C2CCC2)(C(=O)NC2C(CNC(CC(CC)C)=O)C2)CCC1 c1(N2CCC(CS(C)(=O)=O)C2)nc(N2CCC(OCCO)C2)nc2ccccc12 C1(C(=O)NCCN(C(C(c2occ(C)c2)(C)C)=O)C2CC2)Cc2nncn2C1 C1(NC(C(F)=CC)=O)CCC(NC(=O)CCCC2CC2C)CC1 C(=O)(CC1=NNC(=O)C1)NCCN(C(=O)Cn1cc(Cl)c(C)n1)CCC N1(C(c2cnc(OC)nc2)=O)CC2CN(C(C3CC3(F)F)=O)CC(C1)O2 c1(C(=O)NCC2C(C(N(C3CCOCC3F)C)=O)C2(C)C)ccc2nn[nH]c2c1 C1(C)(C(N(CCn2cc(-c3nnccc3C)nn2)CC)=O)CC(C(C)C)=NO1 Cc1nc(C=CC(=O)NCC2(C)CCC2)cs1.c1(CC=O)ccccc1.N C1(C(F)(F)F)(C(N2CCC(C(C)C#N)CC2)=O)CCN(S(=O)(=O)NCC)CC1 c1(CCC(=O)N)n[nH]c(=N)s1.C1(C(N(CCCOCC)C)=O)CCC2CC12 N1(C(c2c(NC)cccc2)=O)CCC(F)(F)C(C)C1.C1(C(=O)N)CCCN(C)C1 C12(NC(CSCC=C)=O)CCN(C(c3ccc(C(F)(F)F)nn3)=O)CC1C2 C(=O)(CC(O)CC(C)(C)C)NC(CCC)C(=O)NCC(C)CCO C12(NC(=O)Cc3ccon3)CCC(CC1NC(c1csc(Cl)c1Cl)=O)C2 c1(NC(C(=O)NC2C(C)(C)CC2)=O)ccc2c[nH]nc2c1 c1(N(C(c2c(C)cno2)C)C(=O)OC(C)(C)C)cc2n(n1)CCCC2 N1(C(c2cnn(C(CC)CC)c2C)=O)CC2CC(NC(c3cn(C)nn3)=O)C1C2 c1(NC(C2(F)CN(C(CC(=O)NCC)=O)C2)=O)cc([N+](=O)[O-])ccc1O C1(C=O)CCc2nnnn2C1.C1(CC(=O)N(CCOC)CC)CC2CCC1C2.N N1(C(c2n(C)nc(O)c2)=O)CCC(C)(C)CC1C(N1CCOC2CCCC12)=O C1(NC(COC(C)C)=O)C2CCC1N(C(c1nccnc1N)=O)C2 N1(C(c2c(C)nn(CC)c2C)C(=O)NCC=C)CC2CCCN2c2ccccc21 Cc1c(C(=O)N2CCC(=O)N2c2ccccc2)ccc2nc(-c3ccccn3)[nH]c12 c1(CC(N2CCC3(C2)CC3)=O)ccc2c[nH]nc2c1.C(=O)(C=CC(=O)N)N(C)C N1(C(C)=O)CC(NC(=O)C=CI)C(C2CC2)C1 CC1(C)CCC=C(C(=O)N2C(CNC(C3(C)CCCOC3)=O)CC3CC23)C1 c1(C(=O)NCC(CC=C)NC(=O)C(CC2CCCC2)CC)ccc(CC)cn1 N1(C(CN(C(C)C)C)=O)CCC(NC(C23CC(CO2)C3)=O)C(F)(F)CC1 c1(-c2cn(CCC(=O)N(CCCCC(C)C)CC)nn2)nccc2occc12 C1(O)(C(C)NC(c2cnsc2)=O)CCN(C(c2ccnc(C(F)(F)F)c2)=O)C1 C(C(C(C)(C)C)c1ccccc1)NC(N(CC)CC)=O C1(C(=O)NCCN(C(=O)CCc2ccccn2)C(C)C)CC1C1CCCC1 C12(C(=O)NCCCCNC(COC(CC)C)=O)CSCC1C2 c1(C(C)=O)ccc(C(=O)N(C)CC2CCN(C(c3coc(C)n3)=O)CC2)nc1 N1(C(c2ccc(C(=O)NC)c(C)c2)C(=O)NCC)C2CCC1CC(N=[N+]=[N-])C2 CN1CCOc2cc(C(N3C4CN(Cc5ncco5)CC34)=O)ccc21 S(=O)(=O)(C=Cc1ccccc1)NCC12CC(NC(C(C)S)=O)(C1)C2 c1(N(C2CCNCC2O)C(CCN(C(C)=O)C)=O)ncnc2c(Br)csc12 N1(C(CC2(OC)CCCC2)=O)CC(N(C(=O)CC2CCC(C)CO2)C)C(C)(C)C1 C12(NC(CCS(C)(=O)=O)=O)CCCC1N(C(c1ccoc1)=O)CCC2 Cc1cc(F)ccc1C.c1(C(N2CC(C(=O)N)C2)=O)ccc(OC(F)(F)F)nc1 C1(CC)CN(C(C2(C3CC3)CCC2)=O)CCN1C(c1cc(C2CCCC2)no1)=O C(C(CC(=O)NCc1cscc1C)OC)NC(COC(CC)C)=O N1(C(CC(=C)C)=O)CC2(CCCN(C(c3c(F)cc(Cl)cc3Br)=O)C2)C1 CCC(C)CC(C)N=c1[nH]c(=NC)[nH]c(=NCCC(=O)NC2CC2)[nH]1 C1(N(C(=O)C)C)CCN(C(=O)Cn2cnnc2)C1.C(=O)(CCC1CCCC1)N C(=O)(C(O)CCCCC)N1C(CNC(C2C(=C)C2)=O)CC(C(C)(C)C)CC1 CC(C)C(C#N)C(=O)N1CCCC(F)(C(=O)NC2(C(C)C)CCC2)C1 N1(C(C2N(C)CC(O)C2)=O)CCCCCC(NC(C2CCCC2)=O)C1 c1(C(N)=O)cc(C(N2CC(Cn3cc(-c4cccc(CO)c4)nn3)C2)=O)ccn1 c1(-c2ccc(C)o2)noc2nc(C)cc(NCC(C(=O)O)C3CCOCC3)c12 C1(N(C(CCOCCCOC)=O)CCF)CCCN(C(=O)Cc2ccccn2)C1 O=C(C(O)C(F)F)NC1CC2(C1)CC2NC(C1CC(n2cnnc2)C1)=O C12(C(N3CCCC(C)(NC(CNC(C)=O)=O)C3)=O)CCCCN1CCC2 N1(C(c2cnn(CCF)c2)=O)CCC(F)(C(=O)NC2(CCCF)CC2)C1 C1(NC(COCC)=O)CCC2CN(C(c3cnc4n3CCOC4)=O)CC2C1 c1(OC)cccc(NC(C23CC(C(=O)NC4CCCC=C4Br)(C2)C3)=O)c1.O C=C(C)CC(C(=O)NCCC1(O)CN(C(=O)C(CC)N(CC)CC)C1)OC C(CCCC(=O)NC(C(=O)NCC(=O)N(C)C1CC1)C1(O)CCC1)SC C(=O)(C1=C(Cl)CCCC1)N(CCCNC(c1cc(N2CCCC2)cc(Cl)c1)=O)C c1(N(C)Cc2cccc(OC)c2)nc(NC2CN(C3CCC3)C2)c2ccsc2n1 C12(CNC(C3N(C(C)=O)CCC3)=O)CC(CO1)N(C(=O)CCC(C)C)C2 N1(C(c2nc(CC)oc2)=O)CC(NC(C2(C(C)C)CCC2)=O)CC1C N1(C(c2c(C)cnnc2)=O)CCOC2CCN(C(=O)Cc3ccccc3)CC12 C(=O)(C1=CC(O)CCC1)NC(C)CCNC(c1c(C#N)cnn1C)=O C(=O)(C(C(C)(C)O)NC(C1CCN(C)C1)=O)N(CC(C)C)C N1(C(CC2CCCC(C)C2)=O)CCN(C(C2CCC3CC3C2)=O)C(C2CC2)C1 c1(C(N2CCC(C)(NC(C(CCCC#C)C)=O)C2)=O)c(C)nc2ccccn12 c1(CC(C(=O)O)NC(C2C(CC(C)(C)C)C2)=O)ccc(Cl)cc1Cl Cc1cc(C(=O)NCC2CCN(C(C3CC4CC3CC4(F)F)=O)C2)c(N)c(Cl)c1 C(=O)(C(C)C(C)S(C)(=O)=O)N1C(CC)CCC1.Cc1cccc(OCC=O)c1.N C(c1ccccc1)=CC(=O)N(CCNC(C1C(C)OCCC1)=O)C.C1(S)CC1 C1(NC(C(C(C)O)NS(=O)(=O)c2cccs2)=O)CNC(=O)CC12CCC2 c1(OC)cc([N+](=O)[O-])ccc1CN1CC(C)(CC(=O)NC2CCCOC2)C1 C(=O)(CC(C)C(C)C)N(C)CC1N(C(c2cc(C)ns2)=O)CCCC1 Cc1cc(C)c(C2CCCN2C(C2CC3(CCCCC3)N2)=O)c(C)c1 c1(CCC(N2C(CCCNC(C(=O)NCC)=O)CCC2)=O)ccc(O)nc1 C1(CC=C)(NC(=O)Cn2nnc(=O)[nH]2)CCN(C(=O)C(CO)N=[N+]=[N-])CC1 C1(CC)C(NC(=O)CCc2cnc(C)o2)CCCN1C(=O)CC(F)(F)F C1(C(N(CC(C(=O)N)C)C)=O)CC2(C1)CC(O)C2.n1(CC)ncnc1CC C(=O)(C(CC(C(C)C)SC)N1CC(C(=O)O)OC(C)(C)C1)NC1(CC)CCC1 Cc1cnc2cc(C(=O)NC3CN(C(=O)CN4CCCC4)C4(CCC4)C3)nn2c1 CN1CCC(C)(C(=O)NC2C3CC(NC(c4cn(CCO)nn4)=O)CC23)C1=O CC1(C)CC(NC(=O)C(O)C2CC2)CCN(C(=O)CCC2OCCO2)C1 N1(CC(CCC2(C(=O)OC)CCCC2)=O)CC2CCC1C2 C1CCC2(C(N3C(C(=O)N(C)CCC4CCC4)CCC3C3CC3)=O)CC12.CO N1(C(C2(C)CCN(C(c3cc(C)sc3)=O)C2)=O)CC(O)(C2CC2)C1 C1(C(N(C(CNC(=O)C(Cl)=CCl)C2CC2)C)=O)CC2C=CC1O2 c1(CC(=O)N(CC)C(C)C)cccc(F)c1F.C1(C=O)CCCCC1.COC c1(C(N2CCCCC(CNC(C3(C)C=CCC3)=O)C2)=O)c(F)cc(N)cc1F c1(C(C)C)ccc(CC(=O)NC(C)C(CO)NC(=O)COC(F)F)cc1 Cc1cncc(CC(N2CCOCC2CNC(C2(C(C)C)CCCO2)=O)=O)c1 c1(C(=O)NC(CCNC(CN2CCN(CC)CC2)=O)C)cc(P(C)(C)=O)cs1 C1(NC(C2(C(C)NC(c3ccnnc3)=O)CC2)=O)CC1C1CCOCC1 N1(C(C)CC(=O)NCCC(N2CC3(CCN3C)C2)=O)CCc2ccccc21 C(=O)(CC(C)(C)CC(F)(F)F)N1CCC(CNC(CCCOC)=O)C(C2CC2)C1 C1(C)(C(N2CC(CNC(CNC(=O)OC)=O)OCC2)=O)CCCCC1C N1(C(C(C)N2CCC2)=O)CCN(C(c2cc(Cl)n(C)n2)=O)C2(CCC2)C1 C(=O)(CC(C(F)F)c1ccccc1)N(C(C)CNC(c1cnc(Cl)s1)=O)C c1(CC(=O)N(c2ccccc2O)C)ccc2c(c1)CN(C(=O)NC1CC1)CC2 C1(C(C)NC2(CCO)CN(C(=O)CSc3ccncc3)C2)CCCCN1C n1(CC=O)nc(C)cc1C(F)F.C1CCCC1.C1(C(=O)N)(COC)CC1 C#Cc1cccc(NC(C2C=CCN(C(=O)Cn3c(C)ccc3C)C2)=O)c1 c1(C=O)ncc2[nH]ncc2n1.C1(OCC)CN(C(=O)CCC2CC2C)CC1C.N C1(NC(CCC(C)OC)=O)CC(F)CN(C(c2c(OC)nsc2OC)=O)C1 C(=O)(C=CS(C)(=O)=O)N1C(C(C)(C)NC(CCCCSC)=O)CCC1 N1(C(C2C3CN(C(c4c(CC)oc(C)c4)=O)CC32)=O)CC2(C1)OC(=O)NC2C C(C(CC(F)(F)F)NC(c1cnn(C)c1C)=O)NC(C1CN(CC)C(=O)N1)=O c1(CCC)ccc(Br)cc1.n1(CC)nnnc1CC1(C(F)F)CCC1.CCO C(=O)(CC(C)CC(=O)O)N(C(C)C)CC.c1(C=O)ccc(C(C)(C)C)nc1 Cc1cccc(C(=O)NC2CC(CNC(=O)COc3ccn(C)n3)C2)c1N C1(C(=O)NCCCCCNC(c2nccc(C)c2)=O)CC2CCCC2C1 c1(OCC)cc(Cl)ccc1C(=O)NC1CCCC1.c1(C=O)ccnc(C)c1.C N1(C(CCC#CC)=O)CCCC(C)(C)C1CNC(C1(Br)C(C)C1C)=O N1(C(C)C(=O)N)CCP(C)(=O)CC1.n1(C2(C=O)CC2)cccn1.CCC1CC1 Cc1cccc(CCNC(=O)CC2(OC(C)(C)C)CCOC2)c1.C(N)=O.N c1(C(N2C(C(=O)Nc3c(C(C)=O)cccc3)CC2)=O)ccnc2ccc(O)cc12 C1(CC=O)(C(F)(F)F)CS(=O)(=O)C1.C12CC(C1)C2.CCC=O.CN c1(-c2n(C(CC)C)nc(C3CCCO3)n2)ccc(S(=O)(=O)C2CCCC2)cc1 Cc1cc(Cl)ccc1CC(=O)N(C1CC(NC(C2Cc3nncn3C2)=O)C1)C C(C)(C)(C(=O)NCC(C)(C1CC1)NC(=O)C(c1ccn(C)c1)C)OC C1(OC)CN(C(c2ncccc2N)=O)CC1NC(c1c(Br)noc1C1CC1)=O CC1C(NC(=O)CNC2CCN(C)C2)CCN1C(c1c[nH]nc1Cl)=O C1(CC(=O)NCC2C(N)CCO2)(C(N2CCCC2)=O)CCCCC1 CCN=c1ccc(C(=O)NC2CCC(NC(=O)C3=CCC(C)CC3)C2)c[nH]1 C1(OC)(OC)CC2(COC(C)C2)C1.c1(-c2nnco2)nc(Br)sc1C.C(=O)C.O c1(NC(CCCCN(C(CCC=C(C)C)=O)C)=O)cc(C)cc(C)c1C C(=O)(C(F)CC(C)C)NC(c1ccccc1)CNC(c1cc(CCC)[nH]n1)=O C(c1cn(C)cn1)=C(C(=O)NCC(CC=C)NC(=O)CCC1CC1(C)C)F N1(C(C2CN(C)C(=O)N2)=O)CCC2(CCN(C(=O)CN3CSCC3=O)C2)C1 n1(CC(=O)NCC2N(C(c3c(C)c[nH]n3)=O)CCOC2)c(C)c(C)sc1=O N1(C(Cn2ncc(C)c2)=O)CCCC(O)(CNC(C2CC3(CCO2)CC3)=O)CC1 CS(=O)(=O)c1ccc(NC(=O)C(=O)NCCCCC(F)(F)F)cc1 N1(C(C(C)CC#N)=O)CCC2C(CCCN2C(=O)Cn2ncc3ccccc23)C1 c1(C(CC)NCc2cc(O)ncn2)ccc(Cl)cc1.C1(C)(CO)CN1 n1(CC)cnc2c(N3CC4COCC(C4)C3)nc(N(C)CC3CC3Cl)nc12 C1(CC(N2C(CC=C)C(C)(C)CCC2)=O)CCCC2(CCC2)O1 N1(C(CSCC=C)=O)CCC2(CC1)CC(C(N1CCOCC1)=O)CO2 c1(C(=O)NC2CCN(C(CC(CCC)CC)=O)C2)c(Cl)ccc2cccnc12 CCCS(=O)(=O)C(C)C(=O)N1CC2(CCN2C(=O)CCS(=O)(=O)N(C)C)C1 C1(O)(C(N(CC(C)N(C)C(c2cc(F)cs2)=O)C)=O)CC(F)(F)C1 C(=O)(C(C)CCCC(C)=O)NC(CC(=O)NC1CN(C(CC)=O)C1)CC CCC(O)C(C)C(=O)NCC1CCCC1NC(c1cc(C2CCC2)no1)=O N1(C(C(CC)C(C)O)=O)C2CCCC1CC(NC(c1cc(F)c(F)cc1F)=O)C2 C1(CNC(C2(CC)CCOC2)=O)CC(C)CN(C(=O)C#CC(C)(C)C)C1 CC1(C)CC(NC(c2ccc[n+]([O-])c2)=O)CN1C(=O)C(N)=O c1(C(=O)OC)ccc(NC(C2CN(C(C3C4COCC34)=O)CCS2)=O)c(Br)c1 C=C=CC(C)C(=O)NCC(C(=O)N(c1csnc1C)C)N(C)C CN1CCCCC1C(=O)NCC1CC1C(=O)NCC1CCC(C)(C)O1 N1(C(=O)Cn2cnnc2O)CCC(C(F)(F)F)(CNC(C2(F)CCC2)=O)C1 S(=O)(=O)(c1cnn(C)c1)NCCNC(C(c1ccccc1)OC(CC)=O)=O N1(C(C(C(=C)C)(C)O)=O)CCC2(CC1)CC(NC(=O)C(CO)OC)CO2 C1(NC(CC2(CC=C)CCCC2)=O)CCN(C(=O)CCn2ccnc2C)CC1O c1(OC)cc(N2CCC(NC(=O)C(C)(C)O)CC2C)ccc1[N+](=O)[O-] Cc1cn2cc(CC(=O)NC3CN(C(c4cnc(C5CC5)[nH]4)=O)C3)nc2s1 N1(C(c2c(C)c(=O)cc[nH]2)=O)CC(NC(=O)CC2CCC(O)C2)CC(C)(C)C1 C1(C(N2CCC3CN(C(C45CC(C)C4C5)=O)CC32)=O)C2CCC3(COC(=O)C13)O2 c1(C(N2CCC(O)C2)=O)cc2c(F)ccc(F)c2s1.C(C(C)(O)C(=O)N)OC.C C(=O)(CCCC#N)NCCC1(OC)CN(C(=O)C(=Cc2cnn(C)c2)C)C1 C1(CNC(c2ncncc2Cl)=O)CC2CCC1N2C(=O)C(O)C1CC1 CCC(C)(C)C(=O)NCC(C1CCN(C(C2COCCN2C)=O)CC1)F C=CCC(C)(C)CC(=O)NCC1(C)CCCN(C(c2cnn3c2CCC3)=O)C1 CC(O)C(C(=O)NC(C)CCCC)N(C)C.c1(CC(=O)N)ccccc1C1CC1 C(=O)(CCCNc1cccnc1)NCC(=O)NC(CNS(CC)(=O)=O)C c1(CC)c(NC(=O)CSc2ccc(C)cc2)c(=O)n(-c2ccccc2)n1C c1(NC(C2CCN(C(=O)Nc3c(Cl)cccc3Cl)C2)=O)ccc2nn[nH]c2c1 Nc1cccc(CC(F)C(=O)NCC2CN(C(=O)CCNc3cnccn3)C2)c1 N1(C(c2cnc(CCC)s2)=O)CCC(NC(c2cn(C)nc2C)=O)CC1C Cc1cc(C(=O)NCC(F)CNC(C2CCOC2C2CC2)=O)cc(C)c1O C1(NC(=O)NC2(c3ncco3)CC2)CCC(N2CCCCC2)CC1 c1(Cc2cn(CCNC(=O)CSCC3CCCO3)nn2)ccc2ccccc2c1 CC(CCCNC(=O)COc1ccccc1)NC(c1ccns1)=O S(=O)(=O)(c1ccc(N2CC3CN(C)CC3C2)cc1Br)N1CC(OC)C2(C1)CC2 C1(CNC(=O)CSCc2cccs2)C=CCN1C(=O)CC1CC2CC2C1 c1(Cc2nnnn2CCCCCC)sc(C(F)(F)F)nc1Br.C1(C)(CC)COC1 C1(C)(NC(C(CCSC)OC)=O)CCN(C(c2cnn(CCF)c2)=O)CC1 CCCC(C)CC(=O)N1CCCC(CNC(c2cccc(Cl)c2O)=O)C1 N1(C(C(CC(C)C)O)=O)CCC2CN(C(=O)CCCc3cncs3)C2C1 c1(CNC(C(COCC)NC(=O)CCC(N)=O)=O)cccc(F)c1C CC(C)CC(C)C(=O)N1CCCC1CC(=O)NCC1(F)CN(C)C1 N1(C(C(CC)C)=O)C(C(=O)Nc2nc(Cl)c(Cl)c(OC)c2Cl)CC2CCCCC12 c1(-c2n(-c3ccc(Cl)nc3)nc(CCN3CCCCC3)n2)ccc2scnc2c1 N1(C(C(CC)=CC)=O)CCc2c(CNC(C3(CCO)CC3)=O)cccc2C1 C1(NC(=O)CC2CC2C(F)(F)F)CCCC1.c1(C=O)ccoc1C1CC1.N CN1CCCC1C(=O)NCC1CN(C(C2CC(C(F)(F)F)C2)=O)C1 C(CCO)(C(F)(F)F)NC(C1(CC)CCN(C(c2cncn(C)c2=O)=O)C1)=O C(=O)(CC(C)(C)CC(F)F)NC12CC(NC(c3cn(C)nc3)=O)(C1)C2 N1(C(c2cc(OC)ns2)C(=O)NCCCC)CC2(CCC2)CC1C(=O)OC c1(-c2cncc(N(CC)CC)c2)cc(F)cc2n[nH]cc12 C12(CNC(c3cncc(Cl)c3Cl)=O)CCCC1N(C(c1coc(Cl)c1)=O)CCC2 C1(NC(=O)NCc2ccc(Cl)nc2)CCCCC1Cc1ccc(F)cc1 Cn1nc(C(N2CCN(C(=O)Cn3cc(C4CCOC4)cn3)CC2)=O)cc1Cl c1(CC(=O)OC)cc(NC(=O)C(=O)NC2C=CCC2)ccc1OC C(N=c1[nH]c(=NC2CCCN(C)C2)[nH]c2cccnc12)c1snc(CC)n1 N1(CC(=O)N(C2CN(C(=O)C(COC)OC)C2)CCC)CC(C)(C)C1 C1(C2CCOCC2)(C=O)CC1(F)F.O=C1CCC(C(=O)NCC2CCC2)=NN1.N N1(C(C(C)NC(COC)=O)=O)CCC(CF)C1.c1(C=O)coc(C2CCC2)n1 CC1(C)CC(NC(C2(n3cccn3)CCC2)=O)CN(C(=O)CC2CCOCC2)C1 C1(C)(C=O)CCS(=O)(=O)CC1.n1(C2CN(C(C3C(C)C3)=O)C2)cc(C)nn1 c1(C(=O)NCC2C(CC)CCN2C(C2CCCS2)=O)noc2c1CCCC2 N1(C(=O)OC(C)(C)C)CCC2(CC2)CC1C(N1CCC2(CSC2)C1)=O C1(C)CN(C(=O)CC2CC2C(F)(F)F)CCO1.Cc1nnnn1CC(=O)N.C C1(NC(C2CCCCC2)C(=O)N2CCC2C2CCCCC2)CC2CCC1C2 C1(C(=O)NCCOCCNC(c2cc(C)sc2C)=O)CCc2ccccc2O1 c1(C(=O)NC(C(C)NC(C(COC(C)C)(C)C)=O)C)cccc(Cl)c1F C(C)(CCN=c1[nH]c(Cl)ncc1C(N)=O)NC(Cn1c(C(C)C)nnn1)=O c1(CC(N2CC(CNC(C(COC)(C)C)=O)N(C)CC2)=O)ccc2[nH]ccc2c1 C(=O)C1=C(C)NC(=O)NC1c1ccccc1.n12cc(cn1)N(C)C(=O)C2.CC.O C1(NC(CC(C)OC)=O)CN(C(C2CCCC2O)=O)CC12CCS(=O)(=O)CC2 c1(N2CC(=C(CNC(C(C=C)O)=O)F)C2)nnc2c(c1C#N)CCCC2 Cc1ccccc1C(=O)NC(CC(C)C)c1cncs1 C1(C(N2C(CCNC(C(C)N(C)C)=O)CCCC2)=O)CCN(C)C(=O)C1 c1ccc2c(c1)CCC2.CCC(C)CC(=O)NCc1cccc(NC(=O)CS)c1 N1(C(c2ccn(COC)n2)=O)CC2CC(C)N(C(C3CNC(=O)CC3C)=O)C2C1 N1(C(C=CC)=O)CC(C)OC2(CCC2)C1.C(=O)CC(C)(C)C.[SH](C)(=O)=O c1(CC(N2CCC(NC(c3ccc(OC)nn3)=O)C2)=O)cccc2c1SCCC2 Cc1cc(C(N2CCC(C(=O)NC(C)C(C)n3cncn3)CC2)=O)c(C)[nH]1 N1(C(CN(C2CCC2)C)=O)CCCC(C2CCCCN2C(c2cn(C)nn2)=O)C1 C1(F)(CNC(=O)CN(C(=O)CCc2ccoc2)C2CC2)CC(O)C1 c1(C(=O)NCC(C2CCCC2)NC(Cc2c(C)non2)=O)c(Br)nnn1C N1(C(c2c(F)cc(OC)cc2F)=O)CCC2CCC(C1)N2Cc1nccc(C)n1 Cc1ccc(S(=O)(=O)CCC(=O)NC2CCCN(C(=O)C(C)C#N)C2C)cc1 C(=O)(C(CC(C)(C)C)NC(=O)C(=O)NC1CC1)N(C)C[Si](C)(C)C n1(CC(=O)NC(C)C(C)NC(c2ccc(O)nn2)=O)cc(C#N)c(O)nc1=O C1(C(=O)N)CCC12CCC2.c1(CN(C(=O)Cc2nccn2C)C)csc(C)n1 C1(C(=O)NC(CNC(c2c(=O)ccn(C)c2)=O)CO)Cc2c(F)cccc2O1 N1(C(c2c(CC)[nH]cc2)=O)CC2C(CNC(c3sccc3CO)=O)C2C1 C1(NC(C(CC=C)(F)F)=O)CN(C(c2ccn3c2CCCC3)=O)C2(CCCC2)C1 C1(NC(CCC=CC)=O)CCN(C(c2nnn(C3CCOC3)c2C)=O)C1CC c1(C(=O)NCC2CCC(C)N(C(=O)CC(F)(F)F)C2)ccc2c(c1)OCC2 C(=O)(C(F)CCC(C)C)N1C(CC=C)(C(=O)NCC(C)C#N)CCC1 C1(CNC(C=C(C)Cl)=O)CC(O)CN1C(c1ccc(N(C)C)cn1)=O Cc1c(N)ccc(C(=O)NC2CC2NC(c2ccc3sncc3c2)=O)c1Cl C(=O)(C1CCCc2nn[nH]c21)NC1CCC(NC(C(C)(C)c2cccs2)=O)C1 Cn1[nH]c(=NC(=O)C2CCOC2CNC(=O)Cc2ccccc2F)cc1C1CC1 N1(C(c2c(C)scc2)=O)CCC(C(C)NC(C2COC(C)C2)=O)CC1 C=CCC(C)(C)CN=c1[nH]c(N2CCC(C)C(CO)C2)nc2c1SCC2 Cc1cc(C(N2CCN(C(C3CC34CCC4)=O)C(C(F)F)C2)=O)c(C)n1C1CC1 c1(C(=O)NCC(C)NC(C2CCCSC2)=O)cn(C)nc1Cc1ccccc1 N1(C(c2cncc(NC)n2)=O)CCC(C)C12CCC2.C1(CC(=O)N)CC2CC2C1 C(=O)(CC(C)(C)N(C)C)N(CCCCCNC(C(C1CC1)SC)=O)C O=C(N=c1sccn1-c1ccccc1)C1CCC1c1ccccc1Cl C1(NC(C2C(C)(CC)C2)=O)CCCC1.n1(CC=O)ccc(C2CC2)n1.C C(C(=O)N1Cc2ccccc2CO1)(N(C)C(c1cnn(C)c1)=O)C1CC1 C=Cc1cncc(C(=O)NC2(CNC(=O)Cc3nocc3CC)CC2)c1 Nc1ccc(C(=O)NCC2CC(NC(c3ccsc3C(F)F)=O)CCO2)nc1 N1(C(C)C(=O)Nc2nc(N(C)C)ncc2Br)CC2(CC(O)CNC2=O)C1 Cc1c(C(=O)N(CCCCN(C(=O)CC2CCCN2C)C)C)cnn1CCO N1(C(C(C)(C)Cl)=O)CCC(CNC(C2C3CCCCC23)=O)C(O)C1 C1(CC(N2CC(C)N(S(C)(=O)=O)CC2)=O)Cc2ccccc2O1 CC1CN(C(=O)CCC(=O)C2CC2)CC(C(=O)NCC(C)(C)N(C)C)O1 O=C(CC(C1CC1)C1CC1)NC(=O)C(O)C1CN(C(=O)Cn2cncn2)C1 C1(C(=O)NCCC)CC2CCCN2C(=O)N1.C(=O)(CCC)N.C(=O)C(C)(C)C C(C)(C(=O)NC(C=CC(=O)NC1CCC1)C)NC(=O)OCC.C c1(CNC(C2N(c3cc(C)nc(C4CC4)n3)CCCC2)=O)cc2ccccn2c1 C1(NC(CN(C)C(N)=O)=O)COCC1NC(=O)CC(O)c1ccccc1 C1(C(=O)NCC(C(C)C)N2CCCC2)CC(O)C(N=[N+]=[N-])C1 C(=O)(C(C)(F)C=O)NCC.C(=O)(C(C)(C)N1CCCC1)N(CCC)CCC CN1CC2(CC(NC(C3(C)CCN(C(=O)CCCCCF)C3)=O)C2)C1 c1(OC)ccc(CCC(=O)NC(C)(C)C2CC2)cn1.c1(C(=O)N)cc(C)cs1 n1(CC)c(C)cc(C(N2CC(NC(=O)CCNC(N)=O)CC(F)C2)=O)c1C N1(C(=O)OC(C)(C)C)CCCC(O)(CNC(c2cc(Br)ccn2)=O)CC1 c1(C(CNC(Cn2ncc(C)c2)=O)NC(C2CC2C)=O)ccccc1F C1(C(=O)NC(Cc2cnc[nH]2)CO)CN(C(c2ccncc2Cl)=O)CC12CC2 CC1(C)CCC(C(=O)NCCCNC(c2n[nH]c(C(C)(C)C)n2)=O)CO1 C(CC(C)CCNC(=O)CN1C(=O)CCC1=O)NC(CC=CC)=O C(C(=O)Nc1ccccc1)(C(C)O)NC(=O)NC(Cc1cc(C)[nH]n1)C CC(=O)CCCC(=O)Nc1cccc(NC(=O)Cc2nncn2C(C)C)c1 C1(C(N(C(CC(CC)C)C)C)=O)CN(C(=O)CC(C)C(=O)NC)CC12CC2 C1(NC(c2c(NC(C)C)nncc2)=O)CCCC(NC(=O)C(N)=O)CC1 N1(C(CCNC(CC(C)C)=O)=O)CC2(CC)CCC1C2.C1(CC=O)CN(C)C1.N C1CCC2(CN(C(C3(C)COC3)=O)C2)O1.CC(C)(C(=O)N)NS(C)(=O)=O N1(C(C2C(C)(C)COC2)=O)CCC(C2(NC(c3ccnc(O)c3)=O)CC2)CC1 CC1(C)CC(NC(C2CC(Cl)(Cl)C2)=O)CN(C(c2cncc3nc[nH]c23)=O)C1 C1(CNC(C2(OCC)CCC2)=O)CCCC1.c1(CC=O)ccc(C)o1.C Cc1cc(C(=O)NCCc2ccccc2)cc(C)c1C.C1(CC(=O)N)CC1(C)C CCCCC(O)CC(=O)N1CC(C(O)C(N2CCOCC2C(C)(C)C)=O)C1 N1(C(C(=O)NCCCOC)CC2CCCO2)CCOC(C(N)=O)C1 N1(C(C2N(C(c3c(C)nsc3)=O)CCC(O)C2)=O)CCc2n[nH]cc2C1 c1(C(=O)NCC(O)CNC(C23CCC(CC2)O3)=O)noc2cc(F)ccc12 C1(C(=O)N)CCC(C)=C(C)C1.CNS(=O)(=O)NCC(=O)N(C)CC1CC1 c1(C(=O)NCCC(C)N(C(=O)CC(F)(F)F)C)ccnc2ccnn12 C1(C)(CC)CC(NC(=O)Cc2ccc(C)nc2)CN1C(=O)C1=CCOC1 c1(C(=O)NC(CNC(C2N(CC)CCC2)=O)C)ccccc1Cc1nc[nH]n1 N1(C(C2(N=[N+]=[N-])CCN(C(C3C(COC)CC3)=O)C2)=O)CCn2c(cnc2C)C1 C(CC(C)C)=CC(=O)NC(c1nccn1C)CC.C1(N(CC=O)C)CCCC1 C1(CC(C)C)CCCCN1C(=O)CC1CCN(C(=O)CC2COC(=O)C2)C1 N1(C(C(C(C)(C)C)NC(CC(=O)OCC)=O)=O)CCC2(CC1)CC2C#N CCCCC(O)CC(=O)NCCCOCCCNC(=O)C(C)NC(C)(C)C c1(C(C)(C)C#N)cc(C(=O)NCCCCCCO)ccc1F N1(C(C2C(c3ccc(C)o3)C2)=O)CC2CC1C2NC(C1(C2CC2)CC1)=O Cc1ccc2c(c1)CC(C(N1CCC(NC(c3[nH]c(CO)nc3C)=O)CC1)=O)O2 c1(C=O)ccoc1C(C)C.C(C)CCNCC.CC(=O)NCC.N(C)C C1(C(N(CC(CC)NC(=O)CC(F)F)C)=O)COc2c(OC)cccc2C1 c1(C(N2CC(NC(C(C)(C)OC)=O)C(F)C2)=O)cnc(O)n(C2CC2)c1=O O=S(=O)(CCCNc1ccc(OC(F)(F)F)cc1)NC1(c2ccccn2)CC1 C1(C)(C=O)CCC(=O)NC1.c1(NC(C)C)ncccc1C(=O)N(C(C)C)C.N C1(NC(C(CC2CCC2)OC)=O)CN(C(=O)C2=CCCCO2)CCC1O N1(C(C2(CC)CC2)=O)CCCOC(CNC(C2CC2F)=O)C1 N1(C(c2scnc2C(F)(F)F)=O)CCCCC1C1CCCN1Cc1cnsn1 c1(C(N(C2CCN(C(c3cc(C(F)F)[nH]n3)=O)C2)C)=O)cc2[nH]ccc2cn1 CC1(C)C(CC(=O)O)C1(C)C.c12cnc(cn1)c(=O)n2Cc1ccco1 N1(C(CS(CC)=O)=O)CCC2CCN(C(=O)C(=O)NC3CC3)CC12 C1(C(C(=O)NC(c2ncnn2C)CC)C)CCN(C(=O)C(=O)NC2CC2)C1 c1(OC)c(C(=O)NC(C2CN(C(C3(C(C)C)CC3)=O)C2)C)cccc1F CC(CCc1ccccc1)CC(=O)NC(C1CCCN1C(=O)CCC1CC1)C C1CC2(CCC2)CN1C(=O)CC1CCOC1.C1(N(C)C)(C(=O)NC)CCCCC1 C1(C(N2CC(N(CCC)CC)C2)=O)CCCN1C(C1CC1(F)Cl)=O c1(CC)cc(C)c(C(N2CCC(C(N3CC[Si](C)(C)C3)=O)C2C(C)C)=O)o1 N1(C(C2C(CCOC)C2)=O)CCC2CN(C(c3cnn(C)c3)=O)CC2CC1 N1(C(C2(COC)CCOCC2)=O)CCN(C(=O)CS(N)(=O)=O)C2CCCCC2C1 C(=O)(CCCCCC(C)O)NC1C(NC(c2cc(C)on2)=O)CCC1 N1(C(CCOCC)=O)CCC12CN(C(=O)Cc1ccc(C)cc1)C2.C(C)=O.N C1(CC)CN(C(=O)Cc2csc(C)n2)CCC1NC(=O)C(=O)C(C)C CCCCC(O)C(=O)NCc1ccc(CNC(C2CCCC(=O)O2)=O)cc1 C(=O)C(C)(C)CS(N)(=O)=O.CCC(C(=O)NC1CC(CC)C1)NC(C)=O C1(NC(c2c(C)ocn2)=O)CCCCN(C(C2CCCC(CF)C2)=O)C1 Cn1cnc2cc(NC(C3COCCN3Cc3ccc(F)c(F)c3Cl)=O)ccc12 CC1=C(C(=O)N2CCC(C)(CCNC(=O)CC3CS(=O)(=O)C3)C2)SCCO1 N1(C(=O)CC2CCN(C(=O)CCc3cnc[nH]3)CC2)CC2C(=O)NC(=O)C2C1 C1(O)(CCNC(=O)C(O)Cc2ccccc2)CCCN(C(C2CC(F)(F)C2)=O)C1 N1(C(c2ccc(CCC)s2)=O)CC2(CCN2C(C2CC(O)C2)=O)C1 CCC(CNC(=O)C(O)CC1CC1)(CC)NC(C1CCCCCC1)=O C1(CC)(CC)CC(NC(C)=O)CN1C(c1csc(CO)n1)=O c1(C(=O)NC2C(CNC(=O)C=CC3CCCCC3)CCC2)ccnc2ncnn12 CCC(CC(C)C)C(=O)N1CCN(C(c2ccc(C(C)=O)cn2)=O)C(C2CC2)C1 C12(C(=O)NCCCCCCC#C)CCC(CC1)N(C(=O)C(C)COC)C2 C1(NC(C2(CN(C)C)CC2)=O)CN(C(c2ccco2)=O)CCC12CCOCC2 CC1CCC(C(=O)NC(C23CC(CO2)C3)C)N1C(=O)C=Cc1ccoc1 C1(CNC(C=CC(C)C)=O)C2CN(C(=O)Cc3ncc(Cl)s3)CC12 N1(C(CC=CC=C)=O)CCCC2(NC(=O)CCN3CCC3)CCCC12 c1(CCNC(=O)NCCC(COC)(C)C)ccccc1S(N)(=O)=O C1(CC)OCCC1C(=O)N(CCC)C.c1(C(N(CC)C)=O)cc(C(C)C)no1 c1(N2CC3CC(=O)NC3C2)nc(N2CCc3[nH]nc(O)c3C2)nc2scnc12 N1(C(C2N(CCC)CCC2)=O)CC2CCC1C2NC(c1cc(C)ccc1F)=O C12(NC(c3cc(C)cc(O)n3)=O)CCN(C(C3(CO)CCOCC3)=O)CCC1C2 N1(CC(COCC)O)CC2CN(C(c3ccc(OC)c(OC)c3)=O)CC2C1 CC(C)CC(F)C(=O)N1CCC(NC(c2cc(C3CC3)ccc2F)=O)CC1C N1(C(c2c(CC)nn(C)c2Cl)=O)CCC(C)(C)CC1.C(=O)C.[SH](C)(=O)=O N(C(=NCC(F)F)N1CCC2C(CCCN2C2CC2)C1)C1CCN(CC)CC1 c1(C(N(C(CNC(c2n(CC=C)ccn2)=O)C)C)=O)ccc2c(c1)COCC2 Cc1cnc(Cl)c(S(=O)(=O)N2CCN(C(c3cc(Cl)ncc3F)=O)CC2CO)c1 N1(C(CN(C(C)=O)C)=O)CCN(C(=O)Cc2cc(C)n(C)n2)C(C2CCC2)C1 N1(C(C2CCN(Cc3c(OC(C)C)nccc3)CC2O)=O)CC2CCCCC2C1 c1(C(C(=O)NCCN(C(=O)Cn2nc(C)nc2C)CC)(F)F)ccccc1 C1(C(N2CCC(NC(c3nocc3Cl)=O)C(O)C2)=O)CCc2nc[nH]c2C1 CC(C)CC(O)C(C)C(=O)NNC(=O)C1CCC1 O=C(CCC(=O)N1CCCC1)NCC1CC(O)CN1C(=O)Cn1ncnn1 C1(C)(C(N(CC(C(=O)NC)C)C)=O)CCCN1C(c1cnn(C)c1Cl)=O N1(C(C(C2CCC2)NC(c2ccc(C)nc2)=O)=O)CCC(C)(C)CC1 N1(C(C2C(C)(C(F)F)C2)=O)CCC(F)(C(=O)NCCCCO)CC1 C1(C(=O)NCc2nccc(C(=O)NC)c2)CN(C)CCN1Cc1ccccc1 c1(CC(N2CC3CCN(C(C4CC4(Cl)Cl)=O)C3C2)=O)ccc2occc2c1 Cc1nc2ccc(C(=O)NCC(CO)NC(c3cc(Br)co3)=O)cc2[nH]1 c1(SCC)ccc(CC(N2CCC2CNC(=O)C(C#N)C2CC2)=O)cc1 C(=O)(CCCC(C)CC)N1C(CC)CN(C(c2cnn(CC(C)C)c2C)=O)CC1 Cc1cc(C(=O)NC2CCCC2NC(=O)CC2CCC(=O)N2)n(C2CC2)n1 N1(C(C2CCN(C)CC2)=O)CC2CCCC(NC(=O)C(=O)NCC(F)F)C2C1 C1(C(N(CC#C)C(C)C)=O)C2CN(C(c3cc(Br)c[nH]3)=O)CC12 CC(C)CCNC(=O)CSCc1cccnc1.c1(C=O)[nH]nnc1C1CC1 N1(C(C2(NC(C(C(=O)OCC)CC)=O)CSC2)=O)CC2(CC(C)CO2)C1 N1(C(c2c(C)ncc(N)c2)=O)CC(NC(c2cnn3ccsc23)=O)CC(C)(C)C1 CC(C)C(C(=O)N1CCC(O)(C(C)NC(=O)CCCCO)C1)n1ncc(N)n1 N1(C(c2ccc(C)[nH]2)=O)CCC(C2(Nc3cc(O)ncn3)CC2)CC1 C(=O)(C(CC(C)C)NC(=O)CCOC)N1CCN(C(C(COC)(C)OC)=O)CC1 Cn1ccc(C(=O)NCCOCCNC(=O)CCc2ccnn2C)n1 C1(C(=O)OC)CC2(CCC(CNC(C34CC(C)(C3)OC4C)=O)OC2)C1 CC1=C(C(=O)NCCC(C)(C)CNC(=O)C(C)C(F)F)Cn2nnnc2N1C c1(C(N(C2CCCN(C(c3cc4sccc4[nH]3)=O)C2)CC)=O)cc(F)cnc1O C(C(=O)Nc1ccc(C(=O)NOCc2cccnc2)nc1)(C(C)(C)C)N(C)C C1(OC)CN(C(c2cccc(CF)c2)=O)CC1NC(=O)CCc1ccccc1 C1(C(C)C)CN(C(C2Cc3cscc3C2)=O)CCN1C(C12COCC1C2)=O CCCCCCOC(C)C(=O)NCC(O)CNC(C1CN(C(C)C)C1)=O C(=O)(C1Cc2ccccc21)N1CC(C(N(c2c(C)cccc2)C)=O)C(C)(C)CC1 C#CC1(O)CC(C(=O)N(C(C)CNC(=O)C(C2CCCCC2)=O)C)C1 c1(NCc2nnc(O)o2)nc(N2CCC(CCC(F)(F)F)C2)nc2sccc12 c1(CO)ccc(-c2cc(-c3nccn3CC3COC4(CNC4)C3)ccn2)cc1F C1(C(N2C(C#C)CC2)=O)COCCN(C(c2ccccc2NC)=O)C1 c1(C(N2CC(OC)C(NC(C3CC3C)=O)C2)=O)ccc(Cl)c(O)c1N c1(C(N2CCC3CN(C(C(CSC)O)=O)CC3C2)=O)cccc2cccc(O)c12 C(=O)(CC(=O)NCCC(O)C(=O)N1CCC(N(C)C)C1)OCC C1(C(=O)Nc2c(Cl)cccc2Cl)CC2CC(C1)CN(CC1CC(=O)C13CCC3)C2 CC1CCN(C(C23COC(C2)C(NC(=O)CCc2ccncn2)C3)=O)CC(C)O1 C(C(C#N)(CC)CC)(c1n(CCC)nnn1)NCC1(CO)CC1(C)C Cc1c(NCC2(C)CS(=O)(=O)CCO2)nc[nH]c1=NCCSc1cccc(F)c1 N#CC1(C(=O)NCCN2CCCN(C(=O)C(F)CC3CC3)CC2)CC2(CC2)C1 N1(C(C(CC=C)NC(C)=O)=O)CCC(C2CC2NC(c2nc(O)sc2C)=O)CC1 CCCCCC(O)C(=O)N(C)CCOCCCNC(c1cc(C)nc(C)c1O)=O c1(C(N(CC(C)NC(=O)CC2CCCCC2(C)C)C)=O)cc2ccc(O)cc2[nH]1 c1(OC)cc(OC)ccc1C(N1CCCN(C(c2ncc(F)cc2C)=O)CC1)=O c1(C(=O)NC2CN(C(C3C(CC)C3)=O)CC2)c(N)sc(C)c1C.C1CC1.C c1(C(=O)NCC(CC(=O)O)C(=O)O)nccc2ccccc12 Cc1cccc(F)c1-c1noc(C2CCN(C(=O)CSS(C)(=O)=O)C2)n1 C(CCCCCC(=O)N1CCC(c2ncco2)C1)NC(CC(CC)CC)=O N1(C(c2cn(CCO)nn2)=O)CC2(CC(C(N3CCCC3C3CCC3)=O)CO2)C1 c1(NC(C2C3CN(Cc4c(OC)cc(Br)cn4)CC32)=O)cnc2ccc(F)cc2c1 C1(C(=O)NCC(c2ccc(F)cc2)NC(Cc2cnc(C)o2)=O)CCCN(C)C1 c1(CC(N2CCC(CCNC(CCSCCCC)=O)C2)=O)cccc(C)c1 C1(CN(C(C(F)=CCC)=O)C)COCCN1C(c1cn(C2CCCC2O)nn1)=O C1(CCC)CN(C(c2cccc(O)n2)=O)CCN1C(c1ccc(C(C)F)cc1)=O c1(C=O)cn(C)cc1C.C=CCCCNC(=O)COC1(C(F)(F)F)COC1 N1(C2(CN3C(c4onc(C(CCC(=C)C)C)n4)CCC3)CC2)CC(C)(C)OC1=O N1(C(COc2c(C)cccc2C)=O)CCCCC(NC(=O)C(O)C2CC2)CC1 Cc1nc(N2CCC(NC(C3CCCCO3)=O)CC2C)cc2nncn12 c1(C(C(=O)NC2C=CC(CNC(c3ccn(C)c3)=O)C2)(C)C)ccccc1Cl C1(NC(C=CC2N(C)CCC2)=O)CN(C(c2sccc2CO)=O)CCC1O c1(C(=O)NC(C2CCCCC2)C(=O)NCC(O)CCC2CC2)ccc(F)cn1 c1(CCC(=O)NCC(=O)NC(C)CC2CCCO2)ccncc1 NC1(C(=O)NCCC2CC(F)(F)CN2)C2CC3CC(C2)CC1C3 N1(C(C(C2CCC(C)CC2)N)=O)CCC2(CCCC(CO)O2)CC1 C(c1cccc(F)c1)=C.C(c1ccncc1)=C(C(=O)N(CC(C)C)C)F.C(=O)C=C.N C1(SCC(=O)NC(C)CCNC(=O)COC2CCC2)CC(F)(F)C1 Cc1nc(NCCC2CCOC(C)(C)C2)cc(N(C)Cc2ccns2)n1 N1(C(c2c(OC)nsc2OC)=O)CCC2(CCC2)CC1.C1(CC=O)CC(=O)C1 CC(CO)CCCNC(=O)C(c1cccnc1)NC(=O)CC1(C)CCCCC1 N1CCCC(O)(C=O)C1.c1(NCc2ccc(N(CC)CC)o2)cccnc1F.C C1(C(=O)NC(C)C(F)(F)F)CCCN(CCN2CCOCC2)CC1 Cc1ccc(CCC(=O)NCC2COCCN2C(c2cnn(C(F)F)c2)=O)nc1 N1(C(C2CN(C(C(C(=O)OC)C)=O)CC2F)=O)CC2CCC(C1)O2 c1(CCC)cnc(C(=O)NCc2cc(O)ccc2Br)c(C(=O)OC)c1 C1(C(=O)NC(CCC)C2CC2)CCN(C(C2(O)CCCC2)=O)CC1C C(C(=O)NC1CC12CCN(C(c1cc(C)oc1C)=O)C2)(C(C)(C)C)OC Cc1cnc(C(=O)N(C)CC2CN(C(c3csc(C)c3C)=O)C2)cc1C c1(C(=O)NC(CCNC(Cn2ncc(C)c2)=O)C(C)C)ccc2c(c1)CCC=C2 C1(NC(=O)CC2CC2)CN(C(=O)C(F)=CC2CC2)C2(CCOC2)C1 C1(O)CCN(C(C2(c3cc[nH]n3)CCC2)=O)C1.C1(CC(=O)NC)CN(C)C1.C c1(CC(=O)NC2(C)CCN(C(=O)C=CCF)C2)cccc([N+](=O)[O-])c1 C1(NC(C(C=C)O)=O)(CO)CCN(C(c2sc(CC3CC3)nc2C)=O)C1 C(=O)(C1=C(Cl)CCC(C)C1)NCC(=C)CCNC(=O)C(c1cncc(F)c1)C C(=O)(CC(CC)C(C)C)NCC1(F)CN(C(CC2CC(=C)C2)=O)C1 C1(C(=O)NCC(CO)NC(C=Cc2scc(C)n2)=O)CC2CCC1CC2 N1(C(C2CC(C(C)C)OCC2)=O)CC(C)N(C(=O)Cc2cnco2)CC1C C1(CCNC(CC2CC(SC)C2)=O)CCN(C(c2cccn2C(C)C)=O)C1 Cc1cc(C(N2CCCC(NC(=O)CC3CN4CCC3CC4)CC2)=O)nnc1C C#Cc1cc(OC)cc(C(N2CCC(CC)(CO)CC2)C(=O)NCC(C)C)c1 c1(CN2CCC(C(=O)NCc3cc(F)cc(Cl)c3)CC2)ccc2cnccc2c1 C1(C2CCCN(C(c3ccccc3CO)=O)C2)(NC(CC(CC)C2CC2)=O)CC1 Cc1onc(O)c1C(=O)NC(C)CNC(C1CCC(=O)N1C(C)C)=O c1(N2CCC(CCOC)C2)nc(N2CCN(CC(C)(C)F)CC2)nc2c1SCC2 c1(N2CCC3(OCCC(O)C3)C2)cc2nccnc2c(Cl)n1 Cc1coc(C)c1C=CC(=O)N.C1CCC12CN(C(C1(P(C)(C)=O)CC1)=O)C2 CC1OCCCC1C(=O)NCC1(CNC(c2cccnc2O)=O)CC1 C1(C(N2CCN(C(c3ccnnc3)=O)CC(O)C2)=O)CCc2ccccc2C1 N1(C(c2c(C)cco2)=O)CCC(C)(NC(=O)C(C)(C)c2ccccn2)C1 C#CC1(C(=O)NC(c2ccncc2F)C)CCN(C(c2scnc2C)=O)C1 C(CCC(CO)NC(=O)C1=NOCC1)NC(CCCOCC)=O c1(NCC=CCNC(c2ccc(C(C)=O)o2)=O)cncc(Cl)n1 N1(C(C(C)C)=O)CCN(C(C2(n3cnnn3)CC2)=O)CC(C)C1 c1(C=O)cc(C)cnc1C.C1(CNC(C2(COC)CCC2)=O)CCCCC1.N C(c1cccc(C(F)(F)F)c1)=CC(=O)N.Cc1nccn1CCC(=O)NCCC CC(CC(C)(F)F)C(=O)N1CC2CC(C1)C2NC(c1cc(F)ccc1O)=O c12cc(ncn1)N(C)CCN2.C(C(C)(C)C1CCOC1)OC C12(C(=O)NCC3(O)CCN(C(C(C)SC(C)C)=O)C3)CCC(CC1F)C2 C1(NC(=O)Nc2ccc(OCCC)c(OC)c2)CC2CC(N(C)C)CC2C1 N1(C(C2(CC)CCNC2=O)=O)CCN(C(=O)CO)C(C)C1.c1ccc(Cl)c(C)c1 N1(C(c2occ(C(C)=O)c2)=O)CCC(C)C(C)C1.c1(C=O)cc(=O)n(C)o1.N c1(C(=O)NCC(CC=C)NC(c2snc(Cl)c2Cl)=O)cc(C)cc(C)n1 CN1CCCC1CCC(=O)NC12CC(CNC(=O)C(C)(C)F)(C1)C2 c1(C(N2CCC2)=O)cc2c(C)ccc(F)c2o1.N1(CC)CCOCC1C(=O)NC C1(NC(c2ccc(C(N)=O)o2)=O)CC(NC(C2CCCCS2)=O)CC1O C=CCCC(F)(F)C(=O)N1CCN(C)C(C(=O)NCCc2cncs2)C1 Cc1ccc(C(=O)NCC(F)CNC(=O)CC2CC(F)C2)c(F)c1 C1(NC(C(C)C(F)F)=O)CCC12CCN(C(c1cn(CCF)nn1)=O)CC2 C(N=c1nc2c(ncn2C)c(NC2CC3C=CCC(C2)C3)[nH]1)c1c(C)nccn1 N1(C(c2n(C=C)ncc2)=O)CCOCC(NC(=O)CCNC(c2ccoc2)=O)C1 N1(C(CSC(=N)N)=O)CC2CCCC2(CNC(=O)CO)C1.c1cccc(Cl)c1 CC1(C)C2CCC1(C)C2C(=O)NCCC1(NC(=O)CCC(N)=O)CCCC1 C1(N(C(COCC=C)=O)C)CC2CC1N(C(=O)Cc1ccc(F)cn1)C2 O(N1C(=O)c2ccccc2C1=O)CC(=O)Nc1ccc(CCC(N)=O)cc1 c1(C(N(C2CCCCCC2)CCNC(C=CCCC)=O)=O)nccc(C)c1O c1(-c2ncc(C(N(CCC(c3ccccc3)O)C)=O)s2)cnn2cccnc12 N1(C(C2C(C)SCCC2)=O)CC(C2CCCN(C(=O)C(F)(F)CN(C)C)C2)C1 C1(C(N2CCC(C)C(NC(=O)CCC3CC3(C)C)C2)=O)CCOC2(CCC2)C1 Cc1ccc(C(=O)N(CCCN(C)Cc2ccc(-n3cccn3)cc2)C)cn1 C1(CCNC(c2csc(C(F)F)n2)=O)CCN(C(c2ccoc2Br)=O)C1 N1(C(C2CCN2C(c2cc[nH]c2)=O)=O)CC(CO)C(O)C1 CC1(C)CC(C(=O)NCC2CCCN2C(c2csc(C3CCCCC3)c2)=O)C1 c1(C(=O)NC(C2N(C(CN(C(C)=O)C)=O)CCCC2)C)nccc(C)c1N C1(CN)CCOCC1.C1(c2n(CCCCCC)nnn2)(NCP(C)(C)=O)CC=CC1 c1(OC)cc(C(=O)NC2CCCCC2NC(=O)C(F)=C2CCCC2)ncn1 c1(C(=O)NCC2(NC(C3C(C)C3)=O)CCC2)cc(F)c(F)cc1N N(C=CC(=O)C(F)(F)F)C(C1N(CC)CC1)=O.c12cccc(c1)OCCO2 C1NC(=O)CC1(C)C.Cc1nn[nH]c1C(=O)NC(Cn1cncn1)C(=O)NC c1(C(C)NC(=O)C(=O)NCC2(CS(N)(=O)=O)CC2)ccc(F)cc1 C(CCC)(CCCC)NC(CNC(C(CC=CCC)C)=O)=O c1(SC)ccccc1NC(=O)C(Cc1cn[nH]c1)NC(c1cc(C)on1)=O Fc1cccc(Cl)c1NCc1cccc(-c2cc(Cl)ncc2NC2CCOC2)c1 N1(C(c2c(C)[nH]cc2)=O)CCC(C2CC2)C1C.C1(C(=O)N)CC2C(C1)C2(F)F C(C)(C)(CC(F)C(=O)N(C(C)C(=O)OC)C)NC(C(CCC)NC(C)=O)=O c1(C(=O)NCCCNC(C2CC(C(=O)OC)C2)=O)c(Cl)cncc1Br C1(NC(C(C(COC)C)C)=O)CCCCCCC1NC(=O)Cc1ccccc1O c1(NC)scnc1C(=O)NCC1CCC1C(=O)NCCc1ccncn1 C=Cc1ccc(C(=O)NC(CCN(C)C(C2CCSC2)=O)C(C)C)cc1 N1(C(CCC)=O)CC(NC(=O)C=CC)C(N=[N+]=[N-])C1.CC(F)(F)F.C(C)C N1(C(=O)OC(C)(C)C)CCC2(CCC2C(=O)O)C1.n1(CC)ncc2ccccc12 C(=O)(C1=CC2(CCOC2)C1)N.n1(CC)c(C(=O)NC2(C)CCC2)cnc1O CCCCCC(C)NC(c1ccn(CCOC)n1)=O C(=O)(CCC(=O)CC)NC1CCC(N(C(CCC=CCC=C)=O)C)C1 C1(C)(C(=O)NC2(S(C)=O)CC2)CCN(C(=O)C2CC2)C1 C1CC(C)(C)CN1C.Cc1cc(C(N2CC(O)CC2)=O)nn1C.C(=O)C(F)(F)F.C c1(C(=O)NC2C(C)N(C(=O)C#CC3CC3)CCC2)cn2cccc(Br)c2n1 c1(CN2C(C(C)C)CN(C(=O)C(c3ccccc3)O)CC2)c(Cl)cc(Cl)nc1Cl c1(NC(=O)NCCn2ccc([N+](=O)[O-])n2)ccc2c(c1)OCCO2 c1(C(N)=O)ccc(C=CC(=O)NCC2CCOC2)o1.c1(C=O)coc(O)n1 c1(C=O)ccccc1C1CC1.c1(CC(=O)N(CC)C2CC2)cc(Cl)cs1.N CCCCCCC(=O)N1CCN(C(=O)CCC2(C)CC2)CC1CCOC N1(C(C=CCN(C(C(C#C)(C)C)=O)C)=O)CCC(N(C)C)C(C)C1 c1(C(C(=O)NCc2ccc(F)cc2)N(C(C)C)C)ccnc(Cl)c1F CC(C)CCC(=O)NCCCCC1CN(C(=O)CCC(F)F)C1 Cc1ncc(NC(C2CCN2C(=O)CN(CCO)CCO)=O)c(C)c1Br Cc1ccn(C(C)C(=O)NC2CCCC2C(=O)NCC2(C#N)CCC2)n1 c1(C(=O)NCC(O)CC(=O)NCCC(O)C(F)F)cc2occc2[nH]1 Cc1nn(C)c2ccc(C(=O)NC3COCC3NC(=O)CS)cc12.C1CCCO1 C1(CC(=O)NCC2(C)CCCS2)CCCN(C(C2(C(N)=O)CC2)=O)C1 C(C(C)C(F)C(=O)NC1CC2(C1)CC(C)C2)NC(C1(CC=C)CCOC1)=O N1(C(C(CC)OC)=O)CCOCC(NC(c2ccnc(OCCO)c2)=O)C1 N1(Cc2ccc(C)c(Cl)c2)CC2(CN(C(=O)CCC(F)F)CCO2)C1 C1(NC=O)CC2(C1)CC(F)(F)C2.CC1SCCCN1CCOC(C)(C)C.C C12(CNC(C3(COC)CCOCC3)=O)CCCCC1N(C(c1cnn[nH]1)=O)CC2 Cc1cc(C(N2CCC(NC(c3cncnc3)=O)C(C)C2)=O)c2n[nH]cc2c1 Cn1nccc1-c1cn(CCOCCCOc2nonc2C(F)(F)F)nn1 C1(CC(=O)N(C2CCN(C(C3ON=C(C)C3)=O)C2)C)CC2CCC1CC2 C(CN=c1[nH]c(=NCc2ccc(S(C)(=O)=O)cn2)[nH]c2c(F)cccc12)OC C(c1cccc(Cl)c1)=CC(=O)NC.C1CN(C(c2cc(C3CC3)no2)=O)CC1O C(=O)(C(O)CC(F)(F)F)N1C(C(=O)NC2CC(CC)OCC2)CC(F)C1 c1(OC)cc(F)ccc1CN(c1nc(C)cc(C)n1)C1(CO)CCNCC1 N1(C(=O)CC2CC3(CCC3)CO2)CC2CN(C(c3cncnc3)=O)C(CO)C2C1 c1(OC)c(C(N)=O)ccnc1Cl.c1(N)ncccc1.c12ccc(o1)C(=O)NC2 c1(C(N2C(CN(C(C(C(=C)Cl)(C)C)=O)C)CCC2)=O)cnn2c1OCCC2 C1(CNC=O)CC2CCC1N2C(=O)COc1ccccc1.c1ccc(F)cc1 C1(NC(C2CC(N(C)C)C2)=O)C(C(=O)NCC#CCCO)C1(C)C c1(OCC)ccc(SCC(=O)NCCC2CN(C(=O)C(N)=O)CC2C)cc1 C12(C(N(CCCCNC(C3C(CC)C3)=O)C)=O)CCC(C1)C(C)(C)O2 N(C1CCCc2sccc21)C(c1ccc(Cn2cc(CC(=O)OC)nn2)o1)=O C1(C(=O)Nc2ccc(I)nc2)CCC2(CN(C(C3CC(O)C3)=O)C2)O1 c1(C(=O)NCC(CC)(CC)NC(c2cc(C)c(C)o2)=O)cc(O)nc(C)n1 C1(C(N2CCC(N(C(C3(CC(C)C)COC3)=O)C)CC2)=O)C2CCCCCC12 C1(CC(=O)NC(C)Cc2ccnn2C)CCCCN(C(=O)CC2CCCOC2)C1 CCC(C)(CO)C(=O)NCC(C(C)C)NC(=O)CCC1(C(=O)OC)CCCC1 CC1(C)CC(c2ccccc2)CCN1C(=O)C(Cc1ccccn1)CCCO c1(CC)ccc(O)cc1.C(C)(C(=O)N(C)C)NC(C)=O.C1CC(CC=O)C1.N N1(C(C(n2ccc(C)n2)C)=O)CC(NC(=O)C=Cc2ccc(Cl)s2)C(O)C1 N1(c2ncc(C(C)=O)cc2C#N)CC2(CN(C(=O)CC3CC3C)CC2CO)C1 C1(C)(CC)CC(NC(c2ccsc2C#N)=O)CN1C(=O)C=CC1CC1 CC(c1ccccc1)=CC(N1CC2C(C(N3CCCCC3CO)=O)C2C1)=O C1(CC(=O)NC(CNC(C2CC2c2ccccc2)=O)C2CCC2)CSCCS1 c1(N(C)C)ncnc2c1cc(C(=O)NC1(c3ccno3)CC1)n2C C1(C(=O)NCC(CC)NC(C2CC(F)(F)CS2)=O)CC(C)(C)CCO1 N1(C(C(CC)C#N)=O)CCC2(CC1)CN(C(c1cn(CC)nn1)=O)C1COCC21 C1(NC(Cc2c(C)noc2C)=O)CCCN(C(c2cnc(S)[nH]2)=O)CC1F C1(CNC(c2c(C)noc2)=O)CN(C(c2ccc(Cl)cn2)=O)CC(C)(C)O1 N1(C(c2c(CC)onc2)=O)CC(NC(=O)C=Cc2ccc(Cl)s2)CC12CCOC2 Clc1ccc(-n2cc(CNC3CCOC3)cn2)cc1Cl N(C1COc2ccccc21)C(C1C(NC(c2c(OC)ccnc2)=O)CC=CC1)=O C(=O)(C(CN(C)C)C(C)C)NC(C(N1CC(C)(CC)C1)=O)c1cccs1 C(=O)(C(C(C)(C)O)NC(=O)CCn1cncn1)NCC(COC)(O)CO C(CO)(C(=O)N1CC(C=O)C1)NC(C=CC(C)C)=O.c1cncs1.C1CC1 c1(CNCCC2CC(OCC)C2)cc(F)c(Br)cc1[N+](=O)[O-] c1(N2CCC(C)(OCC)CC2)ccc(S(=O)(=O)N2CCCC(C)C2C)cc1Br O=S(=O)(c1nc(N2CC(F)CC(F)C2)ccc1Br)NC1CCc2ccnn2C1 c1(C(N2C(CNC(C3(OC)CCCOC3)=O)CCC2)=O)cccc2c1ccn2C c1(CNC(C2CCN(CCOC)C2)c2nnnn2C)cccc(OC)c1O C1(C(=O)OC)CCC(C(N2CCC(C(C)NC(=O)C3=CCCC3)C2)=O)CC1 C(=O)(C1=C(C#N)CCC1)N1CC(NC(=O)COC2CCCC2)CC(OC)C1 N1(C(C(C2CCC2)NC(c2nnn(C)c2N)=O)=O)CCC(C)(C#N)C1 C1N(C(c2cc(C(C)(C)C)c[nH]2)=O)CCC1(C)C.c1(CC)ncc(C(=O)N)[nH]1 C1(F)(CNC(c2cnco2)=O)CCN(C(=O)CC2OCCCO2)CC1 N1(C(CCC2C(C)C2)=O)CC(C)N(C(c2ccc(F)cc2OC(F)F)=O)CC1C C(=O)(C1OCCc2ccccc21)NC1CN(C(CC2C(C)(C)C2(C)C)=O)C1 CCC(CC)CC(=O)N(C(C)CN(C(=O)C(c1ccc(Cl)cc1)(C)O)C)C N1(Cc2n(CCOC)cnn2)CCC(O)C(C(N2CCOC(C)C2)=O)C1 CCC(CCCC(=O)OC)NC(c1ncnc2cc[nH]c12)=O N1(C(c2c(C)ocn2)=O)CC(NC(C2CCCN2CC(C)C)=O)CC2(CC2)C1 N1(C(C=C(COC)C)=O)CCC(NC(c2cc([N+](=O)[O-])c[nH]2)=O)C(C)C1 c1(C=O)nc(C(N2CCCC2)=O)cs1.C1(CC(=O)NC)CCC1(C)C.CC.O N1(C(C(F)Oc2ccc(OC)cc2)=O)CCC(F)(F)C1.C(=O)CC1CC1.C C(C)(C(C(=O)Nc1cc(Cl)cnc1C)C(C)C)NC(c1c(CC)nns1)=O c1ccccc1C#N.C(=O)(CCC(=O)NCC(O)CCNC(C1CC1)=O)NC.O C1(C)(CNC(c2n(C)nnc2)=O)CCCN1C(=O)Cc1ccc(Cl)cc1 C1(C2CCN(C(C34CCC(CC3)C4)=O)CC2)(NC(c2c(C)nsc2C)=O)CC1 C1(C(N2CCC(N(C)C(C3(C(F)(F)F)CCC3)=O)C2)=O)C(F)(F)C12CC2 c1(CCC)cc(C(=O)NC2CC2NC(=O)C(F)F)ccn1 C1CCN(C(=O)Cc2cc(C3CC3)on2)C1.c1(C(NC)=O)ccc(C2CC2)o1 C(=O)(C=CS(C)(=O)=O)N(C)CC1N(C(Cc2ccc(C)s2)=O)CCOC1 N1(C(C(CCCOC)C)=O)C2CCC1CN(C(=O)C(=O)N(C)C)CC2 c1(NC(C)=O)ccc(CC(=O)NCCCC(C)NC(C2COCCO2)=O)cc1 n1(CC)cc(C#N)c(=NC(=O)C2CC2C(=O)NCc2ccc(F)c(Br)c2)[nH]1 C(CCCC(C)C)NC(C=CC=CCC)=O.C(c1cn(C)nn1)=CC(=O)N C(=O)(CCCC(=O)N)OCC.CCCCCN(C)C(c1cncn1C(F)(F)F)=O C#CCCCCCC(=O)N1CCC(CCC(=O)NC(CN(C)C)CCO)C1 CCC(CCC(=O)N(CC(N1CCCC1)C)C)NC(=O)C(C)CC1CC1 N1(C(Cc2c(C)n[nH]c2)=O)CCC(C)(CNC(C23COC(CO)(C2)C3)=O)CC1 C#CCCCC(C)C(=O)N(C(C)C(=O)NCC(CO)C1CC1)CCC N1(C(C2CNC(=O)N2)=O)CC(NC(c2sc3sccc3c2Cl)=O)CC2(CCC2)C1 C(=O)(C1=CCN(C(=O)C2=CCCCC2)C1)N1CCC(N(C)C)C1 c1(C(=O)NCCC2N(C(c3c(CC)ncs3)=O)CCOC2)nc(OC)ccc1Cl CC1CC(O)CN1C(=O)CONC(=O)C1CS(=O)C1 c1(-n2cc(CN(C)C(C3OC4CCC3CC4)=O)nn2)ccc(Cl)cc1F C(=O)(C(C)(F)C(=O)N1CCC1C(=O)NC1CC(OC)C1)OC C(=O)(CCCC(=O)NC(C)CC(C)NC(=O)C(F)C(F)(F)F)NCCC Cc1cc(C#N)cnc1C(=O)NC(CC(C)C)C(=O)NCC1CC(CF)C1 CCCC(CCCNC(c1ccc(O)nn1)=O)NC(=O)CS(=O)(=O)NCC.C c1(C(=O)NC(C2CCOC2)CNC(c2c(C)ncn2C)=O)ccn2cccc2c1 c1(C(N2CC(CC)OC(C)C2)C(=O)NC2CC2)nc(C)c(C)nc1C N1(C(CC(CC)CN(C)C)=O)CC2(CCN(C(C3(c4cc[nH]n4)CCC3)=O)C2)C1 N1(C(C2N(C(C(C(CC)C)N(C)C)=O)C(C(C)C)CC2)=O)CC2CCCCC12C N1(C(C2N(C(CCC=C(C)C)=O)CCC(F)C2)=O)CC2(CCC2)OCC1C C1(C(N2CCC(C=C)C2)=O)CCCCCN1C(=O)C(C)CCN(C)C c1(C=O)ccc(-c2cc[nH]n2)s1.C(CC(=O)N)NC(=O)NC.CC(C)C1CC1 CN=C(NC(CS(C)(=O)=O)C(C)(C)C)N1CCCC(Oc2ncccc2F)C1 C#CCCCCCCNC(=O)C=CCN(C(=O)CC1CCC(C#N)C1)C C#CC1CC2CCC1N(C(C1CSCCN1C(=O)CC=CCC)=O)C2 Cc1cncc(-c2cnc(C3CCCN3C(c3ccccc3C)=O)[nH]2)c1 C1(C(=O)NCC2(CC)CC2)COCCC1NC(=O)CN=[N+]=[N-] C1(NC(CCc2cc(C)on2)=O)CCN(C(=O)C=Cc2cnc[nH]2)C1C1CC1 c1(C(=O)NCC2CN(C(c3cnc(C)o3)=O)C(C)C2)cccc(C2CC2)c1Cl C1(C(=O)NC2C3CCCCC23)(NC(C(SC)SC)=O)CCN(C)C1 C1(NC(C2=CC(C)(CC)C2)=O)CC2CC1CN(C(c1cc(O)ncn1)=O)C2 c1(OC)cccc(OCCCNC(N2CCCC2c2cn(CCO)nn2)=O)c1 Cc1nnc(NCC2CN(C(=O)C(C)CC(C)(C)C)CC(C)(C)C2)c(C#N)c1C C1(CNC(CC(C=C)C)=O)CC(C)(C)CN1C(=O)CCn1cc(Br)c(C)n1 C1(NC(c2cccc(Cl)c2Cl)=O)CCNCCC1CO c1(C(=O)OCc2n(CC)ncc2)ccc(-c2cc(C(F)(F)F)on2)cc1 C(=O)(C(O)CCCNC(=O)CCN1CCCCC1)N1CC2C(C(=O)NC)C2C1 C1(CNC(C2(C(C)C)COC2)=O)CCN(C(c2cc(-c3ccoc3)[nH]n2)=O)CC1 C(=O)(C1=CC2(CCOC2)C1)N(C(CC(=O)NCc1cncc(OC)n1)C)C Cc1ccc2c(C(=O)NCC(O)CNC(=O)CC3CC3(C)C)c[nH]c2c1 N1(C(C(COC)N(C)C)=O)CCOCC1CN(C)C(c1cnc(N(C)C)cn1)=O N1(C(CCCC(=O)NC(C)C)=O)CC(C)N(C(c2ccccc2)=O)CC1C C=Cn1nncc1C(=O)NCC(C(=O)NCc1cscc1C)N(C)C c1(CNC(c2c(C)ocn2)=O)cc(-c2cc[nH]c2)cnc1Cl C12(CC(=O)NOCCC(F)F)CCC1CN(C(C1C3CC4C(C3=O)C14)=O)C2 CC1(C)CC(C(=O)NCCN=[N+]=[N-])N(C(C2CCC(=O)O2)=O)C1 C=CC1(C(=O)N)CCN(C(C2CCN2C(C)=O)=O)CC1.CC(C)CC1CCCC1 N1(C(CC2C(C)(C)C2(C)C)=O)CC2(C(=O)NC3(C4CC4)CC3)CC1CCO2 C(=O)(C1CCCn2nccc21)NCC1OCCN(c2ncc(C#N)cc2Cl)C1 C(=O)(C=C1SCC(=O)N1C)NC(C)CC(C)NC(C1CC12CCOC2)=O C1(C(N2CCC(C(c3ccccc3)C)CC2)=O)COCCNC1=O C=C(Cl)CC(C)NC(=O)CN(C)C(c1csc(CO)n1)=O N1(C(CCN(CCC)C)=O)CC(CC(=O)NCC(C)(O)CCO)CC1(C)C Cc1ccnc(O)c1C(=O)NCCn1cnc(C(=O)N(C)CC2CCCCC2)c1 C1(CNC(c2ccsc2Cl)=O)CN(C(c2cscc2F)=O)CCCO1 C1(C(=O)NCCSC)CC(C)(C)CCN1C(=O)C(F)C(C)C n1(CC)cc(Cl)c(C(N2CCCC(C)C2)=O)n1.c1(CC=O)nocc1C(C)C C(=O)(C(CNC(=O)CCC(F)F)CC1CCCC1)N(C)C1CC1 CC1OC2(C)CC1(C(N1CCC(C)(C)C1)=O)C2.c1(C(=O)N)ncc(C(F)F)s1 Cc1ncc(CC(=O)NC(C)CC2CN(C(=O)CCc3csc(Br)c3)C2)[nH]1 c1(NC(C2C(C(=O)Nc3ncc(OC)nc3)C2)=O)nccc(F)c1F c1(C(=O)NCCCCN(C(c2c(C)cc[nH]2)=O)C)cccc(OCCF)c1 C#Cc1cnn(C)c1C(=O)NC1CC(NC(=O)C)C12CCC2.C1CC=CC1.O Cc1cc(C(N2CCC(C)C2C(=O)NCC2CCC(F)(F)C2)=O)cc(C)n1 CC1(C)CCN(C(=O)CCN2CCCC2)CC1C.C1(C(=O)N)CC(CC(F)F)C1 CCCCCC(C)(C)C(=O)N(CC(C)CNC(=O)C(C)(C)C(=O)NC)C S(=O)(=O)(c1ccc(NCCCOC2CCOC2)cc1Cl)NC(C)C(C)(C)C C1(NC(C2CCC(CC)C2)=O)CC2(C1)CCC2.C1(C=O)CC(N(C)C)C1.N Cc1ccc(F)c(C(=O)N(C(C)CNC(c2cc(O)cc(=O)o2)=O)C)n1 c1(CC)[nH]nc(Cl)c1C(=O)NCCCN(C(=O)C(C)O)Cc1cccnc1 N1(C(C(CC=C)(C)C)=O)CC2CCCN(C(c3cc(CC=C)ccc3O)=O)C2C1 Cc1cc(C(N2CCOC(C)C2)=O)c(C(F)(F)F)o1.C(=O)(CCn1cnnn1)N Cc1nnc(CCC(=O)NC(C)C(C)(C)NC(=O)CCC2CC(F)(F)C2)n1C N1(C(C(C)Cc2ccncc2)=O)CCN(C(C2(n3cccn3)CC2)=O)CC1 N#Cc1cccc(CC(N2CCCC2Cc2cn(Cc3ccc(Cl)s3)nn2)=O)n1 N1(C(CC2ON=C(C)C2)=O)CC(NC(=O)C(O)c2ccsc2)CC(C)C1 C1(CC(=O)NC(CC)CC)CN(C(=O)C(C)NC=O)CCC1C c1(NC(C2OCCN(C(c3cccc(C)n3)=O)C2)=O)ncc(Cl)cc1O c1(C(=O)NC2CC(C)(C)N(C(=O)C=CC3CC3)C2)sc2ccccc2c1Br N1(C(C)=O)CC(OC(C2C=CCN2C(=O)OC(C)(C)C)=O)CC12CCC2 N1(C(COCC)=O)CCCC1(C)C(=O)NCCc1cncc(C)n1 N1(C(C(C2CC2)OC)=O)CCC2CN(C(c3cnn4c(Cl)cccc34)=O)CC2C1 C1(NC(c2ncc(CC)cn2)=O)CS(=O)(=O)CC1.c1(C=O)cnc(Cl)n1C.N c1(OC)nc(C(=O)NC)cc(O)n1.C1(C(N2CCOCC2)=O)CCCC(C)(C)O1 N1(C(CCc2cccc(OC)n2)=O)CC2(CC2)CC1CNC(c1cnc[nH]1)=O C(CC)(CS(C)(=O)=O)N(c1ccccc1Oc1ccccc1)C(COC)C C#CCC(C)(C)CNC(=O)Nc1ccc(C2CCC23CCC3)cc1 C(C1=CCN(C(=O)C(CO)N(C)C)CC1)NC(C1N(C(CCC)=O)CCC1)=O C(=O)(CCCC(C)NC(=O)CNC(=O)CN(C)C)NC1CC(C)C1 C=CCC(CC(F)F)NC(c1ccncc1C)c1nnnn1CCC1(C)CC1 CC1CN(C(=O)C(c2ccccc2)O)CC1CNC(=O)CCc1ccccc1O C=C1CC2CC1CN2C(=O)C(C)NC(=O)C(C)=C(C)C C(C)(CC(=O)NCCN(C(=O)Cc1nc(C2CC2)cs1)C1CC1)OC C(CC(C)(C)CC(=O)NC1(CNC(=O)C(=O)CCC(C)C)CCOCC1)OC N1(C(CC(=C)C)=O)CCC2CCCN(C(c3ccc(C)c(OC(F)F)c3)=O)C2C1 c1(C(=O)NCC2CC(NC(CCCc3ccc(C)s3)=O)C2)c(C2CC2)noc1C N1(Cc2cnn(C)n2)CCCC1C1CCCCN1C(c1ccc2cccnc2n1)=O N1(C(c2n(CC)nc(C)c2)=O)CC2CN(C(c3ccsn3)=O)C2C1 C1(NC(C(C(=O)OC)OC)=O)CCCC12CN(C(=O)C(=Cc1ccco1)C)C2 C1(C(=O)OC)CC(F)CN1C(C1COCCN1C(C1CCC=CO1)=O)=O CC1CCN(C(=O)COCCNC(C2(n3cncn3)CC2)=O)C1 C=CCCCC(C(=O)NCC(O)CC(=O)OC)NC(=O)COCc1nc[nH]n1 c1(C(=O)NC(C#C)C2CC2)coc(CNC(C2(O)CC2)=O)c1 C1(N(C(C(c2cccnc2)C)=O)C)CCC(NC(c2ccno2)=O)CC1 Cc1cnc(C(C)CNC(=O)Cc2ccn(Cc3ccccc3)n2)s1 C=CCC(C(=O)NCC(C(C)C)NC(c1ccccc1)=O)C(C)C.[SH](C)(=O)=O c1(SCCOC)cccc(NC(=O)C(N2CCC2)=O)c1.C1CCN(C)CC1.C c1(C(=O)NCCCC(CCC)NC(=O)C(C)CC2CC2)nccn2ccnc12 S(=O)(=O)(c1ccccc1)N1CCN(C(C=C(C)c2ccccc2)=O)CC1 C1(OC)CC2(C1)CC2C(N1CC(NC(=O)C(C)OC2COC2)C1)=O C(=O)(C1=NN(CCO)C(=O)CC1)N1CC(CNC(C(CCC)(C)O)=O)C2(C1)CC2 C1(C(N(CCCNC(=O)C=Cc2cc(O)ns2)CC)=O)Cc2nnsc2S1 C(=O)(CCC(=O)N(C(C(=O)NCc1ccnc(O)c1)C1CC1)C)NCC C1(NC(C(CCNC(COC(CC)CC)=O)O)=O)CC2(C1)CC(C)(C)C2 C12CC(CN1C(C1CC1c1ccn(C)n1)=O)C2.Cc1n[nH]cc1CC(=O)N.C Cc1nsc(N)c1C(=O)NCC(F)CNC(=O)C(c1ccc(Cl)cc1)CO C(CCC(=O)N(CCCCO)C)(C(C)C)NC(C(C(CC)C)N(C)C)=O C1(CC)CCCN1C(C1CCC(F)(F)C1)=O.C1(S(C)(=O)=O)(C(=O)N)CC1 C#CC1(C(=O)N(C)Cc2cn(C)cn2)CCN(C(C23COCC2C3)=O)C1 C1(NC(CC2CCN(C(c3c(COC)cc[nH]3)=O)CC2)=O)CCN(C)CC1C#N N1(C(CC=C)=O)CCN(C(CNC(c2cn[nH]c2)=O)C(F)(F)F)CC1.C1CC1.C c1(NC(CC)(CNC(c2cccc3cc[nH]c23)=O)CC)nnc(C)c(C)c1C#N Cc1cc(Cl)ncc1NC(=O)CC1(C)CCN(C(=O)CCc2csnn2)C1 C1(CNC(CC(C)CF)=O)CN(C(c2cc(Cl)nnc2O)=O)CC1(C)C CN1C(=O)CCCC1C(N1CC(C=O)C(F)(F)C1)=O.n1(CC)ccc(=O)cc1.N c1(C(=O)NC(CC=C)C(=O)NCCC2(C)CC2(F)F)cc(C#N)[nH]c1C n1(CC)ncc(Cl)c1C(=O)NC1CC(F)(C)C1.C1(CC=O)CCCCO1.N N1(C(C(CC)(C)C)=O)CCC(NC(=O)CSc2ccccc2)C1(C)C CC1CN(C(c2cncn2-c2ccc(F)cc2)=O)CC2(CCCC2)O1 Cc1ccc2c(c1)N(C(=O)NC1CC1(c1ccc(F)cc1)C)CC(C)O2 C1(CCNC(C(C)C2CC2)=O)CCCCN1C(c1cn(CCN(C)C)nn1)=O C(C(=O)NC1CCCN(C(=O)C(C)(C)c2ccc(Cl)s2)CC1)(C(C)(C)C)OC C1(CC(=O)NCC2CCN2C(=O)CCCC2CCCO2)CCCCCCC1 CN1C(=O)CCCC1C(=O)NC(c1ccccc1)COc1ccccc1F N1(C(c2ccc(CO)s2)=O)CC2=C(C1)CN(C(c1occ3c1CCCC3)=O)C2 n1(CC)c(C(=O)NC(C)CCNC(=O)C(C)CC2CCC2)nc2ccccc12 N1(C(CC2C(=O)NCC2)=O)CCCCC12CN(C(c1ccsn1)=O)C2 C1(C(=O)NCc2ncc(CC)s2)CCN(C(=O)C(C)(C(C)C)OC)O1 C1(CCNC(Cn2c(C)ncc2)=O)CCN(C(=O)C(C(C)C)C2CCC2)C(C)C1 C1(OC)CC(NC(=O)CC2CC=CC2)CN(C(=O)C(C)(C)F)C1 Cc1ccccc1CC(=O)NC(C)CNC(C1(c2cc(C)no2)CCOCC1)=O C1CCC(c2nc[nH]n2)CC1.C(=O)(C(O)Cc1cn(C)cn1)N(CC(C)O)C C(=O)(CCC1=CCCCC1)NC(COCC)C(=O)NCC1CC2(CCO1)CC2 c1(N2CC=C(CNC(c3c(C(C)C)cccc3)=O)CC2)ncc(C#N)cc1F N1(C(C2=NNC(=O)C2)=O)CCCC2CN(C(C3CC4(CCCCC4)CO3)=O)CC12 Cc1ncc(N)cc1C(N1CCC(C)C(NC(=O)C(C)N(C)C)C1)=O CCC(C)(C(=O)NC(C1CCN(C(=O)CC2(O)CCCOC2)CC1)C)OC c1(C(N(CC(=C)C)C)=O)coc2c1CN(C(=O)CC1CC1)C2 C(CC(C)C)(C(=O)NCc1nnn(CC)n1)ONC(CC#C)=O c1(N2CC(N(C(=O)CC(c3ccc(Cl)cc3)O)C)C2)ncc2ccnc-2[nH]1 c1(C(=O)NCCCC)ccc(-n2cccn2)nc1.C1(C=O)CN(S(C)(=O)=O)C1 Cc1ccc(C(=O)NCCC(C)(C)NC(=O)CC2(N(C)C)COC2)c(O)n1 C(=O)(CC1=NNC(=O)C1)NC(CNC(C(COC)(C)C)=O)C C1(C(=O)NC2(CO)CC(OC)C2)CN(C(C2C3COCC23)=O)CCC1(C)C C1(C(=O)NC(C(=O)OC)C)CC(O)(CNC(=O)CC2CC2(C)C)C1 N1(C(CCCOCCC)=O)CC2CC1CN(C(=O)CNC(c1ccsc1)=O)C2 C(=O)(CCCC(F)(F)CO)N1CCC(C)(NC(CC2(O)CC(C)(C)OC2)=O)C1 N1(C(Cc2cccc(SC)c2)=O)CC2(CNC(=O)C(C#N)C3CC3)CCC1C2 C1(C(=O)NC2CCC2C(=O)NC(c2nc[nH]n2)C)(CC)CC(C)(C)C1 C=CCCCC(C(=O)NC(C)C(F)F)NC(=O)CN(C)CC N1(C(C(C)NC(N)=O)=O)CCC2CCC(C1)N2C(C1(S(N)(=O)=O)CC1)=O C1(NC(CC(n2ccc(C)n2)C)=O)CCN(C(c2ccc(=O)n(O)c2)=O)C(C)C1 c1(C(N(CC(C)O)CCNC(C2CC(=O)N(C)C2)=O)=O)n[nH]c2c1CCC2 C1(OC)CC(CNC(c2c(C)cnn2C)=O)N(C(c2ccoc2Cl)=O)C1 c1(C(N(CC(CC)O)CC)=O)ccnc(CNC(=O)CCCc2ncco2)c1 C1(C(=O)N(CC(C)(C)OC)C)(CC)CCCN(C(c2sc(F)cc2C)=O)C1 Cc1nnc(N2CCN(C3CCCCC3)CC2)n1CC(=O)NCCO N1(C(CCCCNC(N)=O)=O)C2CCCC1CN(C(C1(F)CCCOC1)=O)C2 N1(c2nc(NC3CN(CC)CC3C)nc(C)c2)CCC(S(C)(=O)=O)CC1 N=c1nc(O)c(C(=O)NCC2CC(NC(C3CCCC4CC34)=O)C2)c[nH]1 CN1CCN(C(=O)C(C)(C)C(=O)N(C)C)CC1CNC(c1cnnn1C)=O C1(C(=O)NC2CC(CNC(C3CCCC(O)C3)=O)C2)CCc2cnnn2C1 c1(C(=O)NCC(CCCC)NC(c2cc(Cl)nnc2O)=O)ccc(N)c(F)c1 c1(C(N2CCC3(CC3C(N3CCOCC(O)C3)=O)C2)=O)ccc(Cl)cc1O n1(CC(N2CCCC2)=O)ncccc1=O.c1(OC(C)C)cc(CC(=O)NC)on1 c1(NC(C2CCC3(CC3)C2)c2n(CC)nnn2)cccc(C2CCOC2)c1 Cc1cc(Br)cc(F)c1C(N1CC=CC(NC(C2CCCCC(=O)N2)=O)C1)=O C#CCCCCC(=O)NC1C2CC1N(C(=O)Cc1c(C)cccc1F)C2 C#CCC(C)(CNC(=O)N(CCc1cccnc1)Cc1ncc[nH]1)CO c1(CNC(=O)Nc2sc(C)c(C(=O)O)n2)cc2cc(Br)cnc2o1 C(=O)(C1CCc2c(F)cccc21)N(C1CC(n2cc(C3CCCOC3)nn2)C1)C CCC(CC(=O)N1CCCC(N(C(=O)C=Cc2cc[nH]c2)CC)C1)C(C)C CC1CCOC1CC(=O)NCC12CC(C1)C2.C1(CC=O)CC(C(F)F)C1 N1(C(c2cccc(C#C)c2)=O)CC(NC(c2cc(OC)nn2C)=O)CCC(O)C1 c1(C(=O)NC(C(=O)N(CC(CC)(C)OC)C)(C)C2CCC2)n[nH]c2c1COC2 N1(C(COCCOCC#C)=O)CCC(O)CC1C(=O)N(C(C)C#C)C C1(OC)(OC)CC(C(N2CCCC2CC(=O)NCCOC2CCC2)=O)C1 c1(OC)cc(C)ccc1OCC(N1CCCN(C(C2CCCCS2)=O)CC1)=O C(=O)(C1CNC(=O)c2ccnn21)N1CC2(C(NC(c3c(C)noc3)=O)CCS2)C1 c1(C(C)NC(CN(C(=O)CCc2ccoc2)CCOC)=O)n[nH]c(C)n1 c1(OC)cccc(C(N2CC(CNC(C34CCCC3C4(F)F)=O)CC2C)=O)c1O C1(NC(=O)Cc2c[nH]nc2O)CCC2CCN(C(=O)C=Cc3cccs3)C12 N1(C(C2(C)CCC(C)(C)CC2)=O)CCn2[nH]c(=N)nc2C1 S(=O)(=O)(C1(C(F)(F)F)CC1)NC(c1ccc(C(F)(F)F)o1)=O c1(OCC)ccc(C)nc1C(=O)NCCCC1CCCN1C(c1ccoc1Br)=O C#CC1(O)CCCC(Nc2ccccc2OCCN(C)C)C1 Cc1ccc2n1CCN(C1C3CCCN(C(=O)OCC(C)(C)C)C3C1(C)C)C2C C1(C(=O)NC(CCN(C)C)C(=O)N2CC(CO)CC2CO)CCCC2(CC2)C1 C1(COCC)CCC2COCCC2C1.N12CCCC(CC1)NC(=O)C1(CC1)C2=O n1(C(C)C)ncc(C(=O)NC(C)CNC(c2ccsc2Br)=O)c1F c1(C=O)cccc(O)c1[N+](=O)[O-].CC(C)CCCNC(=O)CCOCC(F)F.N C1(C(=O)NC(CNC(Cc2nc(C)sc2)=O)(C)CO)CCC2(CC1)CC2(F)F CN1CCN(C(C2(C#N)CCCCC2)=O)CC1CNC(=O)CCc1cnccn1 Cc1n[nH]c(C)c1CC(=O)NC1CC1NC(=O)C=Cc1ccc(Br)s1 C12(CCNC(=O)CC3CC3)CCC1CN(C(c1ccccc1)=O)C2.C1(S)CC1 C1(NC(c2cc(CC)c(CC)o2)=O)CCC2CC1CN2C(=O)CCC(C)(F)F C1(CC)CN(C(=O)C(Cc2cc[nH]n2)NC(=O)C(C)C(=O)OC)CCCO1 C1(CNC(C2C(C)C2)=O)COC(C)(C)CN1C(c1cnc(N(C)C)nc1)=O CC1CN(C(C2(S(C)(=O)=O)CC2)=O)CC2(CCN(c3ncccc3C#N)C2)O1 c1(CC(=O)NCC(c2ccc(Cl)cc2)CC)cc(C)cc(Br)c1 c1(-c2n(-c3c(C#N)c(O)nc(C)n3)nc(CC3CC3)n2)cnc2ncnn2c1C C12(C(N(C3CCCN(C(=O)C=CC=C(Cl)Cl)C3)C)=O)CCN(CC1)CC2 C1CCN(C(=O)C=CC(F)(F)F)CC1.C(C(C)C)OC.C(=O)CC.CC(F)F C1(c2n(C(C)(C)C)nnn2)(NC2(CC3CC3(F)F)CCC2)CCC2(CC1)CSC2 c1(C(=O)NCCC(C)N(C)C(c2cc[n+]([O-])cc2)=O)ccc(C#N)o1 C1(CNC(c2ccc(CCC)s2)=O)CN(C(c2cncc(O)c2)=O)C2CC12 C1(C(=O)NCCC2CCN(C(c3ccc(OC)s3)=O)CC2)CN2CCCN1CC2 C12(CNC(C3(C)CC3(Cl)Cl)=O)CCCC(CN1C(C1SCCS1)=O)C2 c1(OCCC(C)NC(c2ccc(OC)cc2)=O)ccc(C(N)=O)c(OC)c1 C1(C)(CC)C=C(C(=O)NC(CCN(C)C(c2cc(C)cnn2)=O)C(C)C)C1 N1(C(C(C(C)C)NC(N)=O)=O)CCC2(CCC2NC(c2cc[nH]n2)=O)CC1 C1(C(N2CC(CC(C#C)C)C2)=O)CN(C(C2(CCCC)CC2)=O)CCC1O c1(CN(CC(=O)NCC(C)C)CC)ccc(N)c(Cl)n1 C1(CC(=O)N(CC(C)NC(C(C(C)C)CO)=O)C)CC2CCC(C1)N2C c1(C(N(C2CCN(C(=O)CSC(F)F)CC2)CC#C)=O)cc(Cl)c(O)cc1C c1(OC(C(=O)NCCN(C(C2ON=C(C)C2)=O)C)C)ccc(F)nc1 CC(C)P(=O)(CC(=O)NC1CC(C)N(C(c2cn3cccnc3n2)=O)C1)C(C)C C#CCC(C)C(=O)N1CCC(NC(=O)C(COC)COC)C1C(C)C C1(C(C)C)CN(C(C2COC(=O)N2)=O)CCCN1C(=O)CSc1nnnn1C c1(C(=O)NC2CCCC2NC(c2c[nH]ccc2=O)=O)n[nH]c2c1CCCCCC2 CC1(CNC(=O)CCc2ccncc2)COCCN(C(C2CCNC(=O)C2)=O)C1 N(C(=NCCSC)NCC1(Cc2ccc(F)cc2)CC1)C(COC)C(C)C N1(C(C2CC(OC)CC2)=O)CCC(C)(C)C1C.C(=O)(C(C)(C)N(C)C)N C(C(CC(F)(F)F)NC(c1occ(C)c1C)=O)NC(C(CC)F)=O N1(C(CC2N(C)CCCC2)=O)CC(N=c2[nH]c(C3CC3)nc(=N)[nH]2)C1 c1(CN)cc(F)cc(F)c1F.N1(C(CN(C2CC2)C)=O)CCCCC1 Cc1c(C(=O)NCC2CCN(C(=O)C(C)CC(C)(C)C)C2)sc2ncnc(N)c12 CC1(C)CC(NC(=O)C(CO)NC(N)=O)CN1C(=O)C(F)c1ccsc1 c1(CC2(C(N3CCC(OCC4CCCC4)C3)=O)CCC2)cc(Br)cs1 c1(C(=O)O)ccc2[nH]ccc(=NC3CCCc4cccnc43)c2c1 c1(C(=O)NC(C)CNC(C2CSCCS2)=O)cc(C(N)=O)cc(F)c1 C12(COC)COC(C(N3CCC3C3CCOC3)=O)(C1)C2 C(=O)(C1CCCc2nncn21)NCC1CCN(C(CCc2ncn(C)c2)=O)CC1 C(=O)(CCCCCF)NCC(C1CCN(C(=O)Cc2cccc(Cl)c2F)CC1)C Cc1nc2c(N3CCC(O)C(C(=O)NC4CCCC(O)C4O)C3)ncnc2o1 N1(C(C(C)CO)=O)CCC2(CC1)CN(C(c1cnc(O)nc1O)=O)CCO2 c1(C(=O)OC)c(CCC(=O)N(C(C)C)C)c[nH]c1C.C(=O)(CCCCC1CC1)N CN=c1[nH]c(=NCCCCn2ccnc2)[nH]c(=NC(C)C(CO)OC)[nH]1 CC1C(O)CCN1C(=O)C(CC1CCC1)NC(=O)C(C)C1CCC1 c1(OC)cnc(C(=O)NC2CCCC2NC(=O)Cn2ncnn2)cn1 c1(C(=O)NC2CN(C(C3C(CC)OCC3)=O)C2)ccc(N)c(C)c1 CCCC(C)(O)CC(=O)NC1(C)CCN(C(=O)CCC2CCC(C)O2)C1 CC1(C(=O)NCC2(CNC(c3c[nH]c(=O)cn3)=O)CCC2)CC2CC2C1 c1(C(=O)NCC2C3CC2N(C(C2CC2(Cl)Cl)=O)C3)cccc2nn[nH]c12 N1(C(c2cn(CCNC(C3(C)CCC3)=O)nc2)=O)Cc2cncnc2C1 C(=O)CCC(N)=O.C1(C=O)CCN1C(C)(C)C.C(C)(C)(C1CC1)OC.C Cc1nccc(C(N2CC(=O)CC2C(=O)NC2CC2(C)C(F)F)=O)c1C c1(C(=O)NC2CC(N(C(C(CN(C)C)O)=O)C)C2)c[nH]c2c(Cl)cccc12 c1(CN2CCN(C(c3c(OC)cccc3SC)=O)CC2)coc(S(C)(=O)=O)c1 CC1(C(=O)NCC2CC(n3cncn3)C2)COCCO1 C(=O)(N=c1cco[nH]1)c1ccc(NC(NC2C(C)(C(F)(F)F)C2)=S)cc1 c1(OC)ncc(C(=O)N(C(C)C(=O)NCC(O)Cn2cccn2)C)s1 C12(C=O)C3CC(CC13)C2(F)F.C1(CC)CCCC1.C(C)(C=O)OCC#C.N c1(C(N2CCC(CN(C(CCc3scc(C)n3)=O)C)C2)=O)cc2ncccc2o1 Cc1cccc(C2CCCN2C(COC(C)(C)C)CF)c1.C(C)(C)C c1(C(=O)N)ccc(N)c(Cl)c1.n1(C(C)C)ccc(C(N2CCC(C(C)C)C2)=O)n1 C(=O)(C(F)C(F)(F)F)NC1CCC(N(C(C2CC(O)(CC#C)C2)=O)C)CC1 C1(NC(C2CCC(N)(C(F)(F)F)CC2)=O)CCC12CCOCC2 C1(C(=O)N(CC(O)CCC)C)(NC(CSCCC)=O)CCOCC1 CC(C)C(C)CC(=O)NCC(C)(Cn1cccn1)NC(=O)C(C)C(F)(F)F c1(NC(C(N2CCC(CSC)CC2)c2n[nH]c(C)n2)=O)cccc(Cl)c1C Cc1ccc(C(=O)NC2CC(Nc3ncnc(O)c3Br)C23CCC3)c(N=[N+]=[N-])c1 N1(C(C2(CC)CCCC2)=O)CC2CCC2(CCNC(=O)Cc2ccc(Cl)s2)C1 C1(C(N(c2cccnc2Cl)CC)=O)CCCC(NCc2cncs2)C1 N1(C(c2scc(COC)c2)=O)CC(NC(c2cncc(C)c2)=O)CC1(C)C.O C1(C(N(C)CC2COCCN2C(=O)CC2CSCCO2)=O)CC(C2CCCC2)C1 C1(N(C)C)CC(N(C(=O)CCc2nc(-c3nc[nH]n3)no2)C2CC2)C1(C)C c1(C=O)cnc(O)n(C2CC2)c1=O.C1CC(C(=O)NC)C1.C1CC1.CCO Cc1cccc(N2CC(C(=O)NCC3CC4C=CC3CC4)CC2=O)c1C Cn1c(=O)[nH]c(NCC2CN(C(C3CC(=O)N3)=O)CCO2)c(C#N)c1=O CC1CN(Cc2ccc(OC(F)F)cc2)CCC1NC(=NCCF)NC1CCC1 c1(NC(C2COCCN(C(c3ccoc3)=O)C2)=O)ccc(F)c(O)c1 CC1(C(N2CCCN(C3CC3)CC2)=O)CCN(C(=O)CCC(F)(F)F)CC1 Cc1ccc(Cl)c(C(N2CC3CCC2(CO)C3)=O)c1 N1(C(CS(CC)(=O)=O)=O)CC2CC1CCC2NC(=O)CN1C(=O)CCC1=O c1(CCCC)nc(C(=O)NC(CNC(=O)CCCc2cnn[nH]2)CC)cs1 CCC1=NOC(C(=O)NC2CCC2C)C1.c1(CCC=O)ccccc1C(N)=O c1(C(N(CCN(C(C(CCCCC)F)=O)C)C)=O)cncc2ccccc12 CCC(C)(CNC(=O)COC(C)=O)C(=O)N1CC2CCCC1C2 Cc1scc(C(N2CCC2CNC(c2nnn(C(C)(C)C)n2)=O)=O)c1N C1(C)(C(N2CCCC(CC=CC)C2)=O)CN(C(=O)CC(C)SC)C(C)(C)C1 Cc1ccc(CNC(=O)NNC(=O)c2ccc(N(C)C)cn2)cn1 c1(CNC(c2cnc(-c3cnccn3)s2)=O)ccc(S(=O)(=O)CCO)cc1 C(=O)(C(C1=NOCC1)N(CCN(C)C)CC)NCCCSCC c1(C(=O)NCC(C(C)C)NC(CC2ON=C(C)C2)=O)n[nH]c2cc(Cl)ccc12 Cc1ccc2c(C(=O)NCC3(F)CCN(C(=O)CC(C)C)CC3)c[nH]c2c1 C1(C=O)CC12CCC(F)(F)CC2.C1(NC(C2(COC)CCC2)=O)CCOCC1 c1(C(C)=O)cccc(CNc2c[nH]c(C(=O)N(CCO)Cc3ccsc3)c2)c1 N1(C(=O)CO)CCC2(CC1)CN(C(C1CCC3C(C1)C3(F)F)=O)C2.CC(F)(F)F N1(C(C(C=CCCC)O)=O)CC(NC(c2ccc(C(F)(F)F)cn2)=O)C(C)C1 N1(C(CNS(CC)(=O)=O)=O)C2CCC1C(C)C(NC(=O)CC1CC1)C2 CCC(C)(CCNC(=O)CC1CNC(=O)O1)NC(C)=O C12(C)CCC(NC=O)(CO1)C2.c1(OC(Cc2cnc(C)s2)=O)ccccc1Cl.N C1(NC(C(C)SC)=O)CC2CCC1(C(N1CCC(OC3CCC3)C1)=O)C2 CC(C)C(CNC(C1(NC(C2CC3(CCC3)C2)=O)CCC1)=O)CO N1(C(C=CCCC)=O)CCC(CF)(NC(=O)Cc2ccnn2C2CCCC2)C1 c1ccc(F)nc1C.N1(C(CCc2ccc(N(CCOC)C)[nH]2)=O)CCC2(CC2)C1 c1(CC(=O)NCCCN(C(Cn2cc(C(=O)NC)nn2)=O)C)cc(C)sc1C c1(CC)cc(NCCC2CCN(C(=O)C(F)CC)CC2)ncn1 CCC(CCC(=O)NCC(C)CNC(=O)CN1CCC(C(N)=O)CC1)OC n1(CC)ncc(C)c1C=O.c1(CC)nc(C(=O)N(C(C)CC2CC2)C)co1 C1(C(N2CCSCC2)C(=O)NC(C(=O)OC)C)COC(C)(C)OC1 C1(NC(C(CCCC)N(C)C)=O)CC12CCN(C(c1cnoc1CC)=O)CC2 C1(C(N(C2CC(=C)C2)C)=O)(CNC(C2COCOC2)=O)CC12CCC2 Cc1cc(=O)n(C)cc1C(=O)NCC1CC1.C1(C)(CC=O)CCCC1.C S(=O)(=O)(c1ccc(C#N)c(NCCn2cnnc2)c1)NCc1cc(C)on1 C(CNC(C1CC1F)=O)(CC)(CC)NC(C=NOC)=O Cc1cc(CC(=O)NCC2CC(O)CN2C(c2cccnc2O)=O)cc(C)c1 c1(C(N2C(C)CCC2)=O)ccnc2c1ncn2C.C(C)(C)(C(=O)N)OC(C)=O.C C1(C(N(CC(COC)C)C)=O)(NC(c2cc(C(C)C)no2)=O)CC(O)C1 Cc1nc(CC2CC2)sc1C(=O)NC1CCC1.n1(C(C=O)C)nccc1C.C Cc1cc(C(=O)NCC2CCCCN2C(=O)COC2CCCCC2)oc1Br C(=O)(CC1=CCOCC1)NC1C(C)CN(C(=O)C=CC(C)(C)N(C)C)CC1 C1(NC(C2CCCC(F)(F)C2)=O)CN(C(C2CCCCC2O)=O)CC12CCCC2 C(CN=c1ccc(S(=O)(=O)N(CCO)CCC2CC2)c[nH]1)OC S(=O)(=O)(c1cc(F)cc(F)c1)N1CC2(CCCC2)C1.c1(CC)ccc(CN)cc1 C1(NC(c2c(C)onc2)=O)CC2(CCCCN2C(c2ccc3sccc3c2)=O)C1 n1(C(C)C)nccc1C(=O)NCC(O)CNC(=O)Cn1ccnc1C(C)C C(=O)(CC1=NN(C)C(=O)C1)N1CC(C2N(c3ncc(CC)cn3)CCC2)(O)C1 c1(C(NOCc2cn(CC)nn2)=O)ccc(=O)n(C)c1.c1c(C)noc1C.C1CC1 Cc1nn(C)c2cc(OS(=O)(=O)Cc3nnnn3C3CCOCC3)ccc12 C1(NC(c2c(N(C)C)nccc2)=O)CCC2CN(c3ncc(I)cn3)CCC2C1 C1(CNC(c2c(C)noc2C2CC2)=O)CCCN(C(C2(N=[N+]=[N-])CC2)=O)CC1 C1(CC(N2CC(O)(COC)C2)=O)Cc2ccc(Br)cc2C1=O.C1C(C)C(=O)N1 N1(C(CC(CC)NC(C2CN3CCN2CC3)=O)=O)CCc2cccc(O)c21 C1(CC)CC(NC(=O)C2CC2)CCN1C(=O)CC=O.C1(CF)(CC)CCCC1 c1(OC)cc(C(=O)NCCC2CN(C(c3nnn(C)n3)=O)CC2C)cnc1Br Cc1ccccc1N(C(c1cn(C2CC2)nc1C)C(=O)NC1CCC1)C C(=O)(C(C)(C)C(C)(C)O)NC(CC(=O)NCCC=CC=C)CC1CC1 Fc1cncc(Cl)c1CNC1(Cc2cccc(C(F)(F)F)c2)CC1 C(=O)(C(C)(C)C(C)(F)F)NCc1ccc(C(=O)NC(C)C(O)C(F)F)nc1 c1(C(=O)NCCCN(C)C(C2CCCC(=O)N2)=O)ccc(Br)c(F)c1N C1(OC(c2ccc(C3CCCCC3)cc2)=O)CCCC(C(F)(F)F)C1 C12(NC(=O)C(F)=CC3CC3)CCOCC1CN(C(C1(O)CCCC1)=O)C2 Cc1cnc(C(=O)NC2CC3CCC2N3C(C2CCOC2)=O)c(C)c1 C1(CNC(C(CC)OC)=O)CN(C(c2c[nH]c(=NC)o2)=O)CCC1(C)C c1(C(N2CC(CCOC)N(C(C)=O)CC2)=O)cc(Cl)cc(N)c1OC CC1(NC(=O)Cn2cnnn2)CCCN(C(C2(CN3CCCC3)CCCC2)=O)C1 Cc1nc2cccc(C(=O)NCC3CC(NC(=O)Cc4cccs4)C3)c2s1 N1(C(CCCOCC)=O)CC(CNC(c2cnc(C)[nH]2)=O)C2CC12 c1(CN2CC(N3CCN(C(CN4C(=O)CCCC4)=O)CC3)C2)ncc(F)cc1F CC(CNC(=O)C(c1ccco1)NC(c1n[nH]c(=N)[nH]1)=O)S(C)(=O)=O C(C1CCCN1C)=CC(=O)NCC(CNC(CCn1ccc(C)n1)=O)(C)O N1(C(=O)CCc2nnc(C3CC3)o2)CCCCC(CNC(C23CC2C3)=O)C1 C(=O)(C#CC1CCCCC1)N1CCCC(O)(CNC(c2ccc(SC)s2)=O)CC1 N1(C(C#CC(C)(C)C)=O)CCCC2(CCCN2C(=O)CCN2CCC(O)CC2)C1 CCCC(C(O)C(=O)NC1CCC2CC1C2(C)C)NC(C1CC(=O)OC1(C)C)=O N1(C(c2c(C)nn[nH]2)=O)CC2CC1CC2NC(c1cn(C)ccc1=O)=O C1(NC(=O)C2=CCCOC2)CCCCCN(C(C2CC(Cl)(Cl)C2)=O)C1 CC1CCC(C)C(NC(=O)C(F)(F)CCn2cc(CCC(=O)CCO)nn2)C1 N1(C(C2C(C)C(=O)C2)=O)CCCC(NC(c2ccc(C(C)(C)C)[nH]2)=O)CC1 C1(NC(CCc2c(C)ncs2)=O)CN(C(=O)Cc2nncn2C)CC1C1CC1 C1(CC(=O)NCCc2ncn(C)c2)CCCN(C(=O)C=Cc2cncs2)C1 c1(C(N(C(CCNC(c2sc(CCC)c(CC)c2)=O)C)C)=O)cnc(O)nc1O N1(C(=O)CC2C=CCC2)CCC(C2CN(C(C3CC4(CCO3)CC4)=O)C2)CC1 C(=O)(C(C)(O)C(C)C)N1CC(CCNC(C(CSC)(C)C)=O)OCC1 C(=O)CCC(C)C.C(=O)(C=CC(=O)N(C)C)N(C(C)C)CCN(C)C.N O=C(CN1C(=O)Cc2ccccc21)NCC(C1CC1)NC(C1(O)CC1)=O CCC(C)C(O)C(=O)NCCC(C(=O)N1CCC1(C)CCO)OC CCC(CC(=O)N1CCCC1CN(C)Cc1nnnn1C1CC1)c1ccccc1 CC#CCCCC(=O)N1CCC1CNC(C1SCCCS1)=O c1(C(=O)NC(C(=O)OC)C(C)O)n[nH]c2c1CCN(C(c1sc(Cl)nc1C)=O)C2 N1(C(C(c2cnn(C)c2)C)=O)CCN(CCCCCNC(C2CCCS2)=O)CC1 c1(NC(CNC(c2nccc(C)n2)=O)C)cc2c(cc1[N+](=O)[O-])n(C)c(=O)n2C C1(C(N(CCOCC=C)C)=O)CC2C=CC1N(C(=O)C(C)(C)C(=O)NC)C2 Cc1nc(C(F)(F)F)oc1C(N1CCCC1CC)=O.C1(C=O)C=CC=CC=C1.N Cc1cc([N+](=O)[O-])cc(C(=O)NCC(CO)NC(=O)Cc2ccc(Cl)cn2)n1 c1(CC(=O)OC)ccc(CN(C)C(N2CCC(c3ccccc3)C2)=O)cc1 C1(NC(c2n(CC)nnc2)=O)CN(C(=O)CCc2cnc(C)s2)C2CC12 c1(-n2cc(CCC(C(N3CC(C(=O)O)OCC3)=O)O)nn2)cc[nH]c(=N)c1 C(=O)(CCC(=O)N1CCN(C(C2CC2(F)Cl)=O)CC1)NCC c1(C(N2CC(OCCNC(=O)CCCc3cccnc3)C2)=O)cnc(CCC)nc1 c1(N(C)C)ccc(-n2cc(C3COCCN3C(C3CC3(F)F)=O)nn2)cc1 C(=O)(C1=CCC(C)(C)CC1)N1C(COC)CN(C(C2CCCC(=O)N2C)=O)CC1 C1(NC(CCC(=O)NCCC)=O)(CC)CCCN(C(C2CC(OC)C2)=O)C1 C(=O)(C1CCCc2sccc21)N1C(C(C)NC(=O)COC(F)F)CCCC1 c1(C(=O)NC2C(CNC(C(C)CO)=O)CC2)sc(Br)cc1[N+](=O)[O-] CCC(CC)(CCC(=O)N1CC2CCCC2(NC(=O)Cc2cscn2)C1)[N+](=O)[O-] CC(C)(C)N(CC(O)COC1CC1)N1CC(O)CC1c1ccccc1 C1(CNC(c2ccncc2Br)=O)CC2(C1)CN(C(=O)CC1CCCOC1)C2 c1(C(=O)NC2CCC(N(C(=O)C(CO)N(C)C)C)C2)ccn2c(O)nnc2c1 C12(C=O)CCCC1CS(=O)(=O)C2.Cc1[nH]nc(C(=O)N)c1O.C1(CC)CC1.C N1(C(C2N(C(c3cc(C)c(F)cc3)=O)CC3(CC3)C2)=O)CCn2ncc(O)c2C1 C(=O)(C1=NN(C)C(=O)CC1)NC1CCCN(c2c(C#N)ccc(C(CC)C)n2)C1 c1(C(N2CC3C(NC(C(CSC)C)=O)C3C2)=O)cc(Cl)c(F)c([N+](=O)[O-])c1N CCCC(C)(C)CC(=O)NCc1cn(CC(N2CC(CO)CC(C)(C)C2)=O)nn1 c1(C(N2C(C)CCC(NC(C34CCC(CC3)O4)=O)C2)=O)ccc([N+](=O)[O-])cc1Cl C12(C(=O)NCCc3cnc(C)o3)CCC(CC1NC(=O)CCC(C)(F)F)C2 c1(C(=O)NCCCCCN(C(C2(OC)CC(CF)C2)=O)C)ccc(F)cn1 N1(C(C=Cc2c(C)n(C)nc2)=O)CC(=O)N2CCOCC2(C)C1.C(=O)(C1CC1)N C1(OC)(CNC(C2CC2C)=O)CN(C(c2ccc(C(C)C)[nH]2)=O)C1 N1(C(=O)CC2CCCCC2F)CC2CCC(C1)N2C(C12CCCN1CCC2)=O Cc1c(NC(C)C)cccc1C(=O)NCC1N(C(=O)CO)CCC1(C)C N1(C(=O)CSc2cccs2)CCC(C2CC2)C1CNC(C1(O)CC1)=O N1(C(CSCCOC)=O)CCCC2(CCC2)C1.c1(C=O)cc(C)nn1CCO.N C(=O)(CC1=Cc2ccccc2C1)NC1CN(C(c2c(C)cc(C)[nH]2)=O)CC(C)C1 N1(C(C2(N(C(c3c(C)nc(O)cc3)=O)C)CC2)=O)CCc2sccc2C1 C(=O)(C1=COCCC1)NCC1CC(C(N2CCCC2C2(N(C)C)CC2)=O)C1 C1(O)(CC(=O)NC2(C(N(C(c3nn[nH]n3)C)C)=O)CC2)CCOC1 c1(CC(C)C)ncc(C(N2CCC2CNC(=O)C(C)(F)F)=O)s1 N1(C(c2cn(CCC)nc2C)C(=O)NCC2CCCO2)CCOC2CCCCC12 C1(CC(=O)NCCC2CCN(C(c3csnc3C3CC3)=O)C2)(CC)CCOCC1 N1(C(C2CCC(OC)CC2)=O)CC2CCN(C(=O)CCCF)CC12 C(=O)(CCCCN(C)C)N1CCC(C(C(=O)NCC(C#C)(C)C)(C)C)C1 C12(C(N3CCCC(O)(CC)C3)=O)CCCC1CCN2C(=O)CCn1ccc(C)n1 C(=O)(C1(C)CCc2ccccc21)NCCCCNC(C(C(C)(C)C)C1CCC1)=O [N-]=[N+]=NC1CCC(C(N2CCC(CNc3nccc(-n4ccnc4)n3)C2)=O)CC1 C1(O)(CNC(C(N)=O)=O)CC2CCC(C1)N2C(c1ccc2c(n1)CCCN2)=O c1(N2CCC(CN(C(=O)C(N3CCC(c4ncco4)C3)=O)C)C2)ccc(Cl)cc1 C1(C(N2CCN(C3CN(C(C4C(C)C4C)=O)C3)CC2)=O)(OC)CCCC(C)(C)C1 C1(C#N)(CC)CCN(C(=O)C(O)CCCNC(c2ccccn2)=O)CC1 c1(C(C)C)cc(C(=O)N(C)CCOCCC)no1.C1(C(C(=O)N)F)CCOCC1 N1(C(c2ccc(C)[nH]2)=O)CC2CCCC(NC(=O)C=CC3CCOCC3)C2C1 Cc1c(C(N2CC(F)CC2CNC(=O)CC2C=CCCC2)=O)cncc1Br C1(C(=O)N)C2CC(=O)CC12.C(=O)(CCC1CCC1)NCCNC(CC)=O c1(OC)ccc([N+](=O)[O-])cc1C(=O)NC1CCC1.C(=O)CC(C)C.C(C)=O N1(C(CSC)=O)CC2CCC1C2NC(=O)CC1C(=O)NN=C1C c1(C(=O)NC(CCNC(C(C)OCC)=O)(C)CC)ccc(C)c(C)n1 CC1=C(C)CC(C(=O)NC(C)CNC(C2CCCN2C(C)C)=O)CC1 c1(C(=O)NC(C)CCN(C)C(c2[nH]nnc2C2CC2)=O)n[nH]c(C2CC2)c1Cl c1(C(N(CCC)CC)=O)cccc(C)c1Cl.C1(C=O)CC(O)CN1C(C)=O.N N1(C(C(C)C2CCC2)=O)CC(O)C(O)C1CNC(=O)C(c1ccccc1Cl)(C)C c1(C(=O)NC(C2CCN(C(CCc3onc(C)n3)=O)C2)C)csc2cccnc12 C1CN(C(c2cccc(CC#N)c2)=O)CC1O.CCS(=O)(=O)NCCC(=O)NC c1(C(N2CCC(N(C(C3(C(F)F)CC3)=O)CC)CC2)=O)cc(Br)cnc1N n1(CC)ccc(C(N2CC(NC(=O)C)C(C)C2)=O)c1C.c1(C=O)cccs1.N C(CCCC(=O)NC(C1CCN(C(=O)C(c2cnn(C)c2)O)C1)(C)C)OC c1(C(=O)NCC(CNC(C2C(COC)C2)=O)OC)cc(Cl)c(Cl)n1C CCC(CC(C)C)C(=O)N1CC(NC(=O)CCCCCSC)CC1(C)C Cc1ccc(-n2cc(C(C(=O)NC3CCC3)N(C)C3CC3)cn2)c(C)c1 C1(CS(C)(=O)=O)(C(=O)NC)CCOCC1.C1CC1.C(=O)C=C1CCC1 N1(C(C2C(OC)C2)=O)CCOC2(CCN(C(=O)CN3CCC(C)(O)C3)CC2)C1 Cc1cncnc1C(=O)NC1CCCCC1CC(N1CCC(F)(CO)C1)=O N1(C(C=C(C)C(=O)O)=O)CCCN(C(=O)COC2CCCC2)CC1C CCCC(F)C(=O)NCCCNC(C1CCN(CC)CC1)=O C1(NC(C(CC)=CC)=O)CCN(C(c2n[nH]c(C3CC3)c2Cl)=O)CCC1CO C1(NC(c2cc(C)c(CO)cn2)=O)CN(C(=O)C2=NNC(=O)CC2)CC1C1CC1 c1(OCC)ccc(C)cc1C(N1CCCC1)=O.C(=O)CN(C)C(N)=O.C n1(CC)cc(C(=O)NC2CN(C(=O)CN3CCOC3=O)CC2O)c(C2CC2)n1 c1(COC)cncc(C(N2CCSCC2CCNC(C2CCC(O)CC2)=O)=O)c1 C1(NC(CCSC)=O)CN(C(C2CC(C(C)C)=NO2)=O)CCC12CCC2 C(=O)(C(CC(C)C)ONC(=O)C=CC1CCCC1)NC(c1nc(C)[nH]n1)C c1(CC(N2CCC(C(F)(F)F)CC2CN)C(=O)NC)c[nH]c2cc(Cl)ccc12 c1(CN2CCCC(CNC(CSCC)=O)C2)cc(F)c(F)cc1F c1(C(N(C2CC(NC(C3CC3c3cccs3)=O)C2)C)=O)cnc2sccc2c1 C(=O)(CCCCCCCCCO)NC1C2CN(C(CCOC(C)=O)=O)C(C2)C1 C1(CNC(c2c(C(N)=O)csc2)=O)C(C2CC2)CCN1C(c1cccnc1)=O C(=O)(CC(C)(C)CCOC)N1CCN(C(C2C(C=C)CC2)=O)CC1CC(C)(C)C n1(CCC)nccc1C(N1CCCC1CN(C)C(c1cc(C=O)cs1)=O)=O.O N1(C(CCC(C)N(C)C)=O)C2CCC1C(CNC(C1(n3cccn3)CC1)=O)C2 Cc1cc(Cl)cc(C)c1C(=O)N.C1CN(C(=O)CCC2(C)CC2)CC(C)(C)C1 N1(C(CCOc2c(C)cccc2)=O)CC(CNC(=O)CCCN(C)C)CC1(C)C C(=O)(C1c2ccccc2CN1C(c1ncc[nH]1)=O)N(CC)CC1CCC(=O)NC1 C(=O)(C(C)CCCCCC)N1CCCC(CN(C(CCCOCC)=O)CC)C1 c1(NC(N2CC(C)OC(C)(C(F)F)C2)=O)nc2c(F)cc(F)cc2s1 C(c1ccccc1C#N)=CC(=O)NCC(CC)NC(c1cncc2sccc12)=O C=CC1COCC1NC(C1(F)CN(C(=O)CCN2CCCCC2)C1)=O N1(C(C(CC)NC(N)=O)=O)CC2CCCC(C1)N2C(=O)C(C)OCC(C)C c1(NCCCN(C(=O)OC)C)nc(N2CCC3OCCCC3C2)nc2sccc12 N1(C(N2CCCC2Cc2cn(CCCCF)nn2)=O)CCN2C(=O)CCC2C1 N1(C(C2CN(C(C)C)C(=O)C2)=O)CCC(O)(C2CC2)CC1.C1(C(=O)N)CC1(Cl)Cl N1(C(CCOCC)=O)CCC2(CC1)CC(NC(c1nnn(CC)c1C)=O)CCO2 c1(C(=O)NC2C(NC(=O)C=Cc3cn[nH]c3)COCC2)cc2ccccc2cn1 c1(NC2(c3n(CCCOC)nnn3)CC(C[Si](C)(C)C)C2)ccc(F)c(Cl)c1F Cc1nc[nH]c1CC(=O)NCC1(CNC(=O)CC2CCCN2C)CC1 N1(C(COCC)=O)CCC2CCN(C(c3cnc4c(cnn4C)c3N)=O)CC2C1 C(=O)(C#CC1CCCOC1)N1CCC2(CN(C(c3c(C)cc(=O)oc3C)=O)C2)C1 C1(O)(CC(=O)N)CCOC1.C(=O)(CCc1ccoc1)N(CCCN(C)C)CC C(=O)(C1=CS(=O)CCC1)N1CC(CNC(c2cc(SC)c(C)o2)=O)C(O)C1 N1(Cc2cc(C)on2)CCN(C(=NCCCS(C)(=O)=O)NC(c2cccs2)=O)CC1 N1(C(CC(CC)NC(C2CCN(C)C2=O)=O)=O)CCOCC12CC2 N1(C2CCN(C(CC(C(C)C)C)=O)CC2)CCC(N=[N+]=[N-])C1=O c1(NC(C)(CC(C)CCC)c2n(CCCOC)nnn2)cnc2ncnn2c1O N1(C(c2nc(CCOCC)oc2)=O)CCC(NC(c2coc(SC)c2)=O)C1 c1(C(N2CCC(CC(=O)NCC=CC)C2)=O)ccc(C(F)F)cc1 C=CC1OCCC1C(N1C(C(=O)NCc2cc(C)on2)CCC1C(C)C)=O C1(CNC(C2SC3C=CC2CC3)=O)CC2CCC(C1)N2C(=O)CCC1CC1 c1(C(=O)NC2C(C)N(C(c3ccc(F)cc3Cl)=O)CCC2)cnc2nccn2c1 c1(C(=O)OC)ccc(N(C)CCN(C(=O)Cc2ccoc2)C)c([N+](=O)[O-])c1 C1(C(N2C3CC(CNC(c4ccc(C)cn4)=O)C2CC3)=O)CC2(COCCO2)C1 c1(CC(=O)NC2CC(C)(NC(C(CC)n3cccn3)=O)C2)c(C)nn(C)c1Cl c1(OC)ccc(C(C)C(=O)N)c(C)c1.c1(C(N(CCC)C2CC2)=O)nncs1 C1(C(=O)O)CCC2(CCOC2)O1.c12ncc(s1)CNC(=O)C(=O)N2CC CCCC(CCCS(C)(=O)=O)C(=O)NC1CCN(C(=O)C=C(C2CC2)C2CC2)C1 C(CC1=CCN(C(c2ccnc3ccnn23)=O)CC1)NC(CCC=C)=O c1(C(N2CCN(C(CN=S(C)(C)=O)=O)CC2C2CCC2)=O)ccc2ccsc2c1 CCCCN=C(NCc1ccnn1C)NCc1cccc(C(=O)NC)c1 C1(CNC(=O)C(O)C2CCCC2)C2CCCC1N(C(=O)CCF)C2 C1(NC(C2CCC(C(C)C)CC2)=O)CN(C(=O)C(=O)Cc2cccs2)CC1(C)C N1(C(CCC2CCCN(C(c3cc(C)nnc3)=O)C2)=O)Cc2n[nH]cc2C1CO N(C1CCCc2occc21)C(C1(CC=C)CN(C(C2CC(=O)CS2)=O)C1)=O C1(NC(CCCC=C)=O)CCN(C(c2ccnc(F)c2OC)=O)C(C)C1 C1(NC(C2C(C)(C)C2(C)C)=O)CCC2CCN(C(=O)CC(F)(F)F)C12 C1(C)(NC(C2N(C(c3ncn(C(C)C)n3)=O)CCC2)=O)CCCC1(C)C c1(C(N(CC(CNC(C=Cc2c(C)nccc2)=O)C)C)=O)ccc(F)c(C)c1F c1(C(N2CCCCC2)=O)ccc(Cl)c(F)c1.C1(C(NCC)=O)CCCC(=O)O1.C C1(CNC(c2n(C)nnc2)=O)CC2(CCN(C(c3cc(Br)no3)=O)C2)CO1 S(=O)(=O)(c1ccc(-c2nn[nH]n2)cc1)N1CC2CCN(Cc3ccc(C)o3)C2C1 N1(CC)CCC(CC(N2CCOCC2c2cn(CC(=O)OC)nn2)=O)CC1 C1(C#C)(NC(C(C2CCN(C(C3CC(O)(CC#C)C3)=O)CC2)C)=O)CCCOC1 c1(NC(=O)NC(CCC)CC)cnn(C2CCNCC2)c1C c1(C(N2CC(NC(C(C(C)C)OC)=O)C3C(C2)C3)=O)cc(C)ccc1[N+](=O)[O-] C1(NC(c2ncncc2Br)=O)CN(C(C2C=CCC2)=O)CC1O c1(C(=O)N)ccc2cnnn2c1.c1(CCNC(CNS(N)(=O)=O)=O)ccccc1 C1(CCC=O)CCCN(C(=O)C=Cc2ccncn2)C1.C1(C(=O)OC)CC1.C C1(CNC(CC2C(CC)C2)=O)C2CCCC1N(C(=O)CCCC(F)(F)F)C2 N1(CC2(C)CCCCC2(F)F)CCC(=O)NC(CCC#N)C1=O c1(C(=O)NCCC(C)N(C(CC(C)n2cccn2)=O)C)n[nH]cc1[N+](=O)[O-] c1(C(N(CC)C2CC2)=O)cncc2[nH]ccc12.Cc1coc(C)c1C=CC(=O)N CC1(C)COC(CS(=O)(=O)Oc2ccc(-c3ccccc3)cc2)CO1 C1(C(=O)NC(CN(C)C)CO)(CO)CCN(C(=O)CCCF)C1 C1(C(=O)N)CCn2c(C)cnc2C1.C(CCOCC(=O)N(CCC)CCO)OC Cc1ccc(NC(C2(F)CN(C(=O)CC3CCCCO3)C2)=O)c(CO)n1 C1(CNC(=O)C=CC2CCC2)CCN(C(C2(CO)COC2)=O)C1 c1(C(N(C2CN(C(C3CCC(C)(C)O3)=O)C2)C)=O)ccc2ncncc2c1 N1(C(C(C)(C)N(C)C)=O)CCCC(C2CN(C(=O)C3COc4ccccc43)C2)C1 N1(C(CSCCCC)=O)CC2CCN(C(c3cnc(N)c(Cl)c3)=O)CC(C2)C1 C(CCN=c1[nH]ccc(=N)[nH]1)(C(F)(F)F)N(C)Cc1c(C)cncc1 Cc1cc(C(N)=O)cc(C(N2CC(C)C(O)C2)=O)c1.c1(C=O)n[nH]c(C)c1C.N C1(C)(C=O)C(C)(C)C1(C)C.CC1CCN(CCNC(C2CCCC2)=O)CC1.N N1(CCCCN(CCCC)CCC)CC(=O)N(CC23CCCC2C3(F)F)C1=O c1(C(=O)NCCCN(C(C(n2ncc(C)c2)C)=O)C)ccc2cccnn12 C#CC1(C(NC[Si](C)(C)C)=O)CN(C(C2CC=CCO2)=O)C1 c1(C(=O)NCCC(C)NC(=O)Cn2nnc(=O)[nH]2)ccc([N+](=O)[O-])cc1Br c1(C(=O)NCCCN(C(c2cc(C3CC3)ns2)=O)CC)cnn2ccsc12 C1(C(N2CC3C(NC(=O)C=Cc4cncs4)C3C2)=O)CC2CCCN2C(=O)N1 c1(OC)ccc(F)c(C(=O)N(CCCCNC(=O)C(C)P(C)(C)=O)C)c1F C1(c2cn(C)nc2)C(n2cc(C3CC4(CCO3)CC4)nn2)CC(=O)N1C1CC1 N1(C(CCN2CCC(C)CC2)=O)CCCC2(C1)CN(C(C1CCC(=O)N1)=O)C2 c1(OC)cc(Br)c(CN2CC3CN(C(c4ccccc4C#N)=O)CC23)cc1OC C1(CNC(C2N(CC)CC2)=O)CCC2CN(C(=O)CCCc3ncco3)CC12 N1(C(C2(C)CNC(=O)C2)=O)CCOC2(CCN(C(C3CC4(CCC4)CO3)=O)C2)C1 C1(C(=O)NCC#CCC)CC2CC2N1C(C1CCCN1CC)=O c1(N2CCCC2)ncnc(Cl)c1C(C)C.CCC(C(=O)NC)OCC1CCCC1 C1(CNC(c2n(CCC)ccc2)=O)C(C)CCCN1C(=O)COCC N1(C(C(C)SCC)=O)CC(C2CN(C(C3C4(CCC4)C34CCC4)=O)C2)C1 N1(C(c2cncc(C(F)F)c2)=O)CCN(C(=O)CC(O)C2CCCC2)C(CF)C1 CCCCCCCCC(C(=O)NC1CC1)N(C(C)C(=O)OC)CCCF c1(C(=O)NC2CCC(C)CC2)ccc2nn[nH]c2c1.C(=O)(C(F)CC1CCC1)N C#CC1(C(=O)NCCC2CC(F)C2)CCN(C(=O)C(C)C(C)CC)CC1 c1(CC(=O)N)ccc(Cl)cc1.C1(CC=C)(C(=O)NC2CC(C)C2)CCCC1 c1(C(=O)NCC(c2ccccc2)CNC(c2c(C)nc[nH]2)=O)snc(O)c1Cl C(=O)(CC1CCc2ccccc21)NC(CC=C)CNC(c1cnn(CC)c1F)=O O=C(NNc1ccc(I)cc1)C(=O)NCCC1CCN(Cc2ccccc2)CC1 C1(C)(C(=O)N)COC(C)CO1.Cc1oc(C2CC2)nc1C(N1CCCCC1C)=O CC(CC(N)=O)C(=O)NC1CC2(C1)CN(C(C13CCC(CC1)CO3)=O)C2 C1CC(C)(C)CN1C(=O)CC1CCC(C)CC1.Cc1ccn(C(C)C(=O)N)n1.C Cc1cc(C)c(C(N2CCCC2(C)CNC(C2CCC(C)O2)=O)=O)o1 n1(C(C)C)nc(C2CC2)nc1-c1cc(-c2ccccc2)on1.C(C)(C)C N1(C(c2ccc(=N)[nH]c2)=O)CC(NC(c2cncc(C(F)F)c2)=O)CC(O)C1 Cc1ccc(C=CC(N2CC(CCCCNC(=O)C(=O)N)C2)=O)cc1.C1CC1 N1(C(C=C2CCN(C(C(C)Cc3ccccn3)=O)CC2)=O)CCCC2NCCC12 N1(C(c2c(CCCC)ocn2)=O)CCCC(CC)(NC(c2nnn(C)c2N)=O)C1 N1(C(C(C2CCOCC2)C)=O)CCOC(CC(=O)NCCN2CCCNC2=O)C1 c1(C(=O)NCC2(F)CCC(CNC(C(C)(C)CO)=O)C2)ccn2ccsc12 CC1CN(C(c2cc(CO)[nH]n2)=O)CC1CC(N1CCC1C1CCCCC1)=O CC1(CNC(=O)Cc2ccc(Br)s2)CCN(C(=O)C(C2CC2)C2CC2)C1 N1(C(c2c(C)non2)=O)CC2C(C(=O)NCCc3ncon3)C2C1 CCC(C)(O)C(=O)N1CCC(C)(CCNC(c2cc(C)on2)=O)C1 c1(C(=O)NCC2(NC(c3c(C)ocn3)=O)CCCC2)cc2cc[nH]c2cn1 C1(NC(C(C=CCCC)O)=O)CCCN(C(c2n[nH]cc2Br)=O)C1C C1(C(=O)NCC(CC)NC(=O)CCc2ccoc2)CCn2nccc2C1 C12(NC(=O)CCCF)CCCC1N(C(=O)CCc1ncc[nH]1)CC2 N1(C(c2cc(C)nnc2)=O)CCC12CN(C(=O)Cc1cccc(Cl)c1Cl)C2 S(=O)(=O)(c1cccc(=NC2COC3(CCCOC3)C2)[nH]1)NCC1CCC(C)CC1 C1(CNC(C2C(CC)C2)=O)CN(C(=O)C)C(C)(C)C1.c1ccc(O)cc1 c1(OCC)nc2ccc(C(N3CCC(NC(=O)CC(C)SC)C(O)C3)=O)cc2[nH]1 Cc1ccc(C(=O)NCCN(CCO)C(C2C(C)C2C)=O)c(O)c1.CCO CCC(C)(C(=O)NCCO)C(N)=O.c1(C(N2CCC2)=O)cnc(C(F)F)nc1 N1(C(C(CCSC)OC)=O)CCC(C2CC2)(NC(=O)CSc2nccn2C)C1 c1(OC)cc(C(=O)NC2CC(F)CN(C(C3(OC)CCOCC3)=O)C2)c(Cl)cn1 O=C(CC(Cc1cccs1)NC1CC1)N1CC2C(CO)C2C1 c1(C(C(=O)NC)N(C2CCS(=O)(=O)CC2)CC(=O)OC)cc(OC)ccc1Br CN1CCN(C(C23CC(F)(C2)C3)=O)C(C)C1.c1(C=O)cn[nH]c1.C1CCC1.N C(=O)(C1=CCC(C)(C)CC1)NC(C)C(CO)NC(c1cc(O)cc(Cl)c1Cl)=O C1(NC(C(C(C)NC(c2n(CC)ncc2)=O)C)=O)CC(=O)NC(=O)C1 Cc1cc(=NC2CCN(C(C)C)C2)[nH]c(=NCc2ccc(F)c3c2CCC3)[nH]1 N1(C(COCCOCCOC)=O)CC2CC1C2C.C(=O)(C1=NOCC1)N Cc1cc(C(=O)NCCCOCCN(C(=O)Cc2cnsc2)C)c(C)o1 CP(C)(=O)c1ccc(C(=O)NC2CC23CCC3)cc1 C1(C)(NC(CC(C)OC)=O)CCN(C(c2ccnn2C2CCC2)=O)C1 O=C1CCc2cc(C(=O)NCC3CCCC3NC(c3ccsn3)=O)c(F)cc2N1 c1(N(C(C(=O)NC2CC2)c2cccs2)CC2CCC2)ccccc1 Cc1nc(=N)[nH]cc1C(=O)N(C1CCCN(C(=O)CC2(C)CC2(Cl)Cl)CC1)C C1(C(N(c2ccccc2)CCC#N)=O)COCCN(C(=O)CSc2ccccc2)C1 CC1NC(=O)OC12CN(C(C1CN(C(=O)C(F)(F)C(F)F)CCO1)=O)C2 n1(CCC)nc(C)cc1C(=O)N.C1(O)(CC)CCN(C(c2c[nH]c(=N)s2)=O)C1 N1(C(c2ccc(C(F)F)o2)=O)CCCC2C1CCCN2C(=O)CCc1cnn[nH]1 c1(C(C(=O)NC)N(C)CC2CCC(C)CC2)cc(F)ccc1Cl C12(CNC(C=CCC)=O)CC3CC(CC(C3)C1)C2.n1(CC=O)ccnc1C C(=O)(C(C)CN(C)C(c1cccn1C(C)C)=O)NCC1(CCC)CC1 CC1CN(C(C2CCCCO2)=O)CCN1C(=O)CC1CCNC1=O CC(C)(C=O)OCC(F)(F)F.C1(C2(C=O)CC2)CCCO1.CCC1CC1.N c1(C(N2CCN(C)CC2)C(=O)NCCC2CC2)nc(Br)ccc1F Cc1cc(=NCC2OCCO2)[nH]c(=NCC2(C)CC2(C)C)[nH]1 CC1=C(C(=O)NC(C)C(C)NC(c2ccc3occc3c2)=O)SCCO1 C(CC(=O)N(C1CCC1)C)C(F)(F)F.C(CCC)(CCC)=CC(=O)N.C=CC=C C12(NC(C3CCCOCC3)=O)CCCCC1CN(C(=O)CCn1ccnc1)C2 N1(C(C(OCC)OCC)=O)C2CCC1C(C(=O)NC13CC(C)(C1)C3)C2 Cc1ccc(C(C)CC(=O)NC2CCN(C(c3cnc(CN)n3C)=O)CC2)cc1 C1CCNCC1(C)C.N1(CCNC(C(=O)NC(C2CCC2)C)=O)CCCCC1.N C(=O)(CC(O)C(C)C)N1CC(NC(c2cc(CCC)on2)=O)C(F)C1 CC1CC(C(F)F)n2ncc(C(N3CCC(NC(C45CCC(C4)C5)=O)C3)=O)c2N1 C1(CNC(CCCC=C)=O)(NC(c2csnc2C)=O)CC2CCC1C2 N1(C2CCC(NC(CC(N)=O)=O)C2)CCC(C(=O)Nc2ccc(Cl)nc2)CC1 c1(C(C)N(C)C)cn(CC=O)nn1.C1(C)CN(C(=O)CN2CCC(C)C2)C1.N C1(C=O)CC(S(C)(=O)=O)C1.C1(NC(C2(c3cccs3)C(C)C2)=O)CCCC1 C=C(C)C(C)(O)C(=O)N1CCCC(N(C(=O)CCc2nc(C)cs2)C)C1 CC1OCCN(C(C2CN(C)C2)=O)C1C(=O)NCCN1C(=O)CNC1=O CC1(C(=O)NCc2cccc(NC(c3sc(Cl)cc3Cl)=O)c2)CCCCO1 N1(C(c2cc(F)c(N)c(F)c2)=O)CC2CCC(C1)C(NC(C13CC4CC1C3C4)=O)C2 c1(C(N(C)CC2CCCC(NC(C3CC(OC)C3)=O)C2)=O)cc2cccn2cn1 c1(OC)cc(C(=O)NC2CCOCC2NC(C2(CO)CCCC2)=O)nc(C)c1 S(=O)(=O)(c1cccnc1)N1CCCN(C(c2cn(C3CCCC3)nn2)=O)CC1 C(=O)(CC1OCc2ncccc21)N1CC(C(C)NC(c2cc(F)cc(N)c2F)=O)C1 c1(N2CCN(CC(C)O)C(C)C2)nc(=NCC2CC23CCC3)[nH]c2c1COCC2 N1(C(CSc2c(C)cccc2)=O)CC=C(CNC(C2CCNC(=O)C2)=O)CC1 CCCC(CNC(c1cc(CO)[nH]n1)=O)C(=O)N1CCCC(OCC)C1 C(CCS(C)(=O)=O)(C(=O)N(C)CC)OC.C1(S(C)(=O)=O)(C=O)CCCC1.N c1(SCC(=O)NC(CN(C(C2CC(OC)C2)=O)CC)C)ccc(C)cc1 C1(C(=O)NC(C(C)C)C)CC(=O)CN1C(=O)Cc1cnnn1C CC1=NNC(=O)C1CC(=O)NCCC(C)NC(=O)CC1CCC(=O)N1 C(=O)C(C)CC(N)=O.C(=O)(CCC(=O)N1CCC(C(C)(C)C)C1)N(C(C)C)C.N Cc1nn(C)c(C(F)(F)F)c1C(N1CC(S(=O)(=O)N2CCN(C)CC2)C1)=O O=NN1CCCCC1C(=O)NCCC1CN(C(C2CC3CCC(C2)O3)=O)C1 N1(C(=O)OC(C)(C)C)CCC(NC(c2csc(Nc3ccccc3I)n2)=O)CC1 c1(C(=O)NC2CN(C(C=NOC)=O)C3C2C3)nnn2c1CCCCC2 c1(CC)ccc(-c2nc(CCc3ccc(Cl)cc3)n(Cc3ccncc3)n2)cc1 N#Cc1ccc(S(=O)(=O)NCCCc2nnc(C(F)F)o2)cc1 CCCCCCCC(F)C(=O)N1CC(C2(NC(=O)CCc3cncs3)CC2)C1 N1(C(CSCC)=O)CCC(NC(c2c[nH]c(Br)c2)=O)C(CO)C1 C1(CNC(CCOCC(C)C)=O)C2CN(C(=O)C=CS(C)=O)CC12 c1(C(N2C(C)C(=O)NCC2)=O)n[nH]c2cccc(-c3cccc4c3OCCO4)c12 C12(CNC(COC)=O)CN(C(C3CCCOC3)=O)CC(F)(C1)C2 CC(C)(C)C(C(=O)NCC1(C)CCCN(C(=O)CC(F)(F)F)C1)C1CCC1 c1(C(N(C(C2(C)CC2)C)C)=O)ccc(CNC(C2CC=CCO2)=O)cn1 c1(CC)cnn(CC(=O)NC(COC)CNC(=O)CC2CSCCO2)c1 Cc1cc(Br)c(C(=O)Oc2ccc(F)cc2)cc1F.N12CCN(CC1)C(=O)CCC2 CCC(C)C(O)C(C)C(=O)N1CCC(C)C(N(C(=O)C=CC=C(Cl)Cl)C)C1 C1(N(C(C=NOC)=O)C)CCCC2CN(C(C3COCCO3)=O)CC12 c1(C(N(C(C)CNC(C2(C)CCNC2=O)=O)C)=O)cnc2c(Cl)cccn12 CCC(C)(CC(=O)NCC=CCNC(c1cc(OC)ccc1Cl)=O)C(=O)OC C1(N(CC(c2ccccc2)(C)O)C(C2CCC(C)CC2)=O)CCNCC12CC2 C(c1ccc(C)c(C)c1)=CC(N1CC(CC)CCC1)=O.c1(C=O)cnc(S)[nH]1.N C(=O)(C1=NOC2(CCOC2)C1)N1CC(CC=C)(NC(=O)CCC(C)N(C)C)C1 CC1CC(CCNC(=O)CC(=O)NC2CC2)CCN1C(=O)CCC1(C)CC1 Cc1nn(C)c(C(F)(F)F)c1C(N1CCC(CC)C1)=O.C1(C=O)CC(C#N)C1 c1(N2C3CN(C(c4ccccc4O)=O)C(C3)C2)ncc2sccc2n1 c1(C2N(C(c3c(C)cc(C(=O)OCC)o3)=O)CCC2)cn2cccc(C)c2n1 O=C1CC(C(=O)NCCc2n[nH]cc2C(=O)NC)CN1.C1(CCO)CCCC1 C(=O)(C(C#N)CC)NCC1CCC(C(N(CCCC)CCO)=O)C1 C(=O)(N1OC2CC1C(O)C2O)C1CCC(C)N1C(C1CCC(=O)NC1)=O c1(SCC(=O)N(C2CCN(C(c3ccon3)=O)C2)C)nnc2ccccn12 CC(C)(O)C(C)(C)CNC(c1ccoc1C)=O.C1(C=O)CC1.C(N)=O c1(C(N2CCC(O)C2)=O)c(F)cc(Cl)cc1F.C(C(=O)N)NC(=O)OCC=C N1(C(C)=O)CCCCC1C(=O)NC1(CCO)CN(C(=O)CCc2cnccn2)C1 Cc1ncc(Cl)c(C(N2CC(NC(C3(F)CC=CCC3)=O)CC(C)C2)=O)n1 C#CC1(C(=O)N(C(C)CNC(=O)CC2(c3ccccc3)CCC2)C)CCCC1 c1(-c2scc(-c3onc(C4C(C)(C)COC4)n3)n2)ccc2c(c1)OCO2 c1(N(C(=O)Cc2ccoc2)C2CC2)ncnc2c1ncn2CC1CCCCC1 c1(C(N(C2CCN(C(c3cn(CC)nc3C)=O)C2)C)=O)nnn2c1CCC2 N1(c2nnc(SC)s2)CC2CC1CCC2NC(=O)Cc1sc(O)nc1O c1(OCC)ccccc1C(=O)NCC(CC)NC(=O)C(C#N)CC1CC1 C(C(CC)(CC)NC(C1CC12CCC2)=O)NC(c1cn(CC)nn1)=O N1(C(CC(C)O)=O)CC(N(C(=O)CCC2OCCO2)C)C2(CC2)C1 N1(C(C(CC)N(C(=O)C=Cc2cccnc2)C)=O)CCOC(C)C1C CC1CCCC(N(C(=O)CC2CCN(C(C3CC(=O)C34CCC4)=O)C2)C)C1C Cc1cc(F)ccc1NC(=O)C(C1CN(C)CCO1)N(CC(C)(C)C)CCC#N [nH]1cc(S(C)(=O)=O)cn1.Cc1cc(CO)ccc1C(=O)NCCn1ccnn1.C c1(C(C)NC(c2cn(CCNC(c3cc(=N)[nH][nH]3)=O)cn2)=O)ccccc1F C1(C(=O)NC2CCCN(C(=O)CC3(O)CCC3)CC2)CCCc2ccccc2C1 N1(C(c2ccc(C)c(Cl)c2)C(=O)NCC2CC2)CC2CCC1C(O)C2O c1(C=O)cnc2sccn12.Cc1cc(CCCC(=O)NCC2CC2C)c(C)s1.N Cc1sc(Cl)nc1C(N1CCC(C(C)NC(=O)C(F)CC2CCCCC2)CC1)=O N1(C(C(C)OC2CCCC2)=O)CCC2(CCCN(C(=O)C(F)C(F)(F)F)C2)C1 Cc1c(F)ccc(C(N2CCCC2CNC(=O)CCCC2CC2C)=O)c1N N1(C(c2ccc(C)n2C)=O)CCN(C(c2ccc(N(C)C)cc2)=O)C(C(F)F)C1 N1(C(CC(=O)NC)=O)CCCC1(CNC(C1(C)C=CCC1)=O)COC CC1OC2(C(=O)NC3CN(C(=O)Cc4ccccc4O)CCC3O)CCC1CC2 C#CC1CCCN(C(C2CNC(=O)CN2C(=O)C(C)=CC(C)(C)C)=O)CC1 N1(CC(N2CC(C(=O)NCCNC(C3CC(=C)C3)=O)C2)=O)CSCC1=O c1(C=O)c(C)nn(C(C)(C)C)c1C.n1(CC=C)cccc1C(=O)N(C)CC.N CC1CN(C(c2nc[nH]c2C(F)(F)F)=O)CCC1NC(c1cnc(O)o1)=O Cc1nc2ccc(C(=O)NC3CC4C3CCN4C(C3CC(C)(O)C3)=O)cc2s1 Cc1nc(CCCNC(=O)CCCc2ccc(C3CC3)cc2)sc1C C1(N(C(=O)CN2CC=CC2)CCOCC)CCCN1C(=O)Cc1cccs1 C1(C(=O)NCCC(C)(C)NC(C(C)OCC#C)=O)OCC2CCCC1C2 C1(CC(=O)NCC2(C(=O)NC3(C(F)F)CCC3)CCCO2)CCCSC1 CC12CN(C(c3ccc(C(F)F)o3)=O)C(C=O)(C1)C2.C(C(N)=O)C1CCCC1 C(C)(C)(C(=O)NC1CC1(C)C)NC(C(=O)NCCOCCCC)=O N1(C(c2cn(C)nc2Cl)=O)CCC2CN(C(=O)C(c3ccnn3C)O)CCC12 CC(C)CC(CNC(=O)CCC(=O)c1cnn(C)c1)NC(=O)CC.CC(F)F.O C1(CNC(C(CC)C)=O)CC(C)CCN1C(=O)CS.c1cc(C)cc(C)c1.C c1(OC)cccc(C(N2CCOCC(CNC(=O)CC3CCCO3)C2)=O)c1OC N1(C(C#CC(C)(C)C)=O)CC2CCC(CNC(C3CC3c3ccco3)=O)(C2)C1 c1(OC)c[nH]c(C(=O)NC)cc1=O.C12CC(C1)C(C)O2.C1(C=O)COCCO1 c1(CC(=O)NCCC(C)NC(C)=O)ccccc1C1CC1 N1(C(c2c(C#C)c[nH]n2)=O)CC2(CCC2NC(=O)CN(C)C(C)=O)C1 c1(C(=O)Nc2ccc(Cl)nc2)c(Cl)ccc2c[nH]nc12 N1(C(Cc2cccc(C)c2C)=O)CCC(C2CC2)(NC(c2ccoc2)=O)C1 N1(C(C2(OCC)CCC2)=O)CC2(CCN(C(c3nc(C)oc3C)=O)C2)C1 c1(NC(CCNC(CC(C)OC)=O)C)cc(C)c([N+](=O)[O-])cc1F CC(C)CCCCCC(=O)N1CC(C)(NC(C2CCCCC2C)=O)C1 N1(C(C2CN(C)C(=O)N2)=O)CC2(C1)CN(C(=O)C(C1CCCO1)C1CC1)CCO2 Cc1coc(C(N2CCC2(C)CC(=O)NC2CC(CO)(CO)C2)=O)c1 C(CN=c1[nH]nco1)C1CC(NC(C2C(C)C2)=O)C1 c1(SC)ncc(CN2CC(NC(C3CCS(=O)(=O)C3)=O)C2)c(Cl)n1 c1(C(=O)NCC2N(C(CCc3nccc(C)c3)=O)CCC2)cccc2c1CCN2 C(=O)(C1COc2ccc(F)cc21)N(C1CN(C(C23CCC(CC2)OC3)=O)C1)C CC(CCC(=O)NCCCCN(C)C1CC1)NC(=O)CC1CC=CC1 O=C(N1CC(n2cc(C3CCOC3)nn2)CO1)c1cn(CC(F)(F)F)nn1 C1(C(N2CCC(C(=O)NCCNC(C)=O)C2)=O)COc2ccccc2O1 C(=O)(C(F)CC(C)(C)C)NCC=CC(=O)NCc1cnn(C)c1O C=CCN=C(NCC(CO)CC=C)NCc1ncccc1C(=O)OCC c1(C(=O)NCC(CC=C)NC(=O)C(C)(C)OC)cccc(Cl)c1[N+](=O)[O-] c1(C(=O)NCC(CC=C)NC(c2cnc(S)[nH]2)=O)ccc2c(c1)C(C)(C)CN2 N1(CC)C(=S)NC(c2cc(C)cc(Br)n2)C(C(=O)Nc2cccc(Cl)c2)=C1C n1(CC=O)nc(C)c(Cl)c1C.C1(OC)CCN(C(=O)C=CC=C(Cl)Cl)C1.C c1(C(=O)NCc2cc(C(N(CCC(O)CO)C)=O)n[nH]2)cc2occc2[nH]1 c1(CC(=O)N(C2CC(NC(C3C(C=C)CC3)=O)C2)C)c[nH]c2cc(OC)ccc12 C1(NC(C#CC(C)C)=O)CC2CCC(C1)N2Cc1ccn(-c2ccccc2)n1 Cn1ccc2cc(C(=O)NC3CN(C(C4CC(C)(F)C4)=O)CC34CC4)ccc12 C1(CC)CCCCN1C(C1CCC(C(N)=O)CC1)=O.c1(OC)cc(C(=O)N)on1 N1(C(C2CC(C)CC(C)C2)=O)CC2CC(C1)CN(C(=O)C(C)(C)N(C)C)C2 C12(C(=O)NC34C(CN(C(C5CCCC(=O)O5)=O)C3)CC4)CCC(CO)(CC1)CC2 C1(NC(C=Cc2cn(C)nn2)=O)CC2CC1N(C(=O)CNS(N)(=O)=O)C2 c1(OC)ccc(NC(C2CCC3(CC3)N2C(C2(Cl)CCCCC2)=O)=O)c(O)c1 C(=O)(C(C)C(CC)CC)N(CCCNC(c1cnn(CCCC)c1C)=O)C(C)C C(=O)(CCCC(C)(C)NC(=O)C(C)OCC(C)C)NCC=C C(=O)(CCC(=O)N1CC(CO)(NC(c2cncc(Br)c2)=O)C1)NC C#Cc1ccc(F)cc1C(=O)NCCC1CCCN1C(=O)COc1ccsn1 C1(C(=O)NCC(C)(C)NC(c2c(CC)ocn2)=O)Cc2ccccc2C1C c1(NC(C)=O)cc(C(=O)N)ccc1C.C1CN(C)CCN1C(=O)C.C1CC1.C C1(NC(CCSCC)=O)CN(C(C2(CC)CCC(O)CC2)=O)CCC1(C)C c1(OC)ccc2cc(-c3nc(C4CC4C)nn3Cc3cccc(C)n3)sc2c1F C1(C2CCCN(C(C3CCC=CCC3)=O)C2)(NC(C(CC(C)(C)C)OC)=O)CC1 C(=O)(C1CCCc2ncccc21)C(=O)Nc1c(C(=O)OCC)n(C)cn1 CN1CC2CC2(NC(=O)CCNC(=O)Cc2cccc(F)c2)C1 N1(C(C2C(CC)CCO2)=O)CCCC2(C1)CN(C(C1CC1C#N)=O)C2 C(=O)(C(CC(C)C)N1CCC(C(O)C(N)=O)CC1)NCCOC.C(C)(C)C.O CC(CN=c1cc[nH]cc1S(=O)(=O)NCc1cccnc1Cl)N1CCCC1 N(C(=NCc1cccc(OC)c1)NCC(C(F)(F)F)OC1CCC1)C(C=C)C C(=O)(C1CSc2ccccc21)NCC1CCCCN(C(c2c(Cl)cn(C)n2)=O)C1 C(CCCC(C)C)(C(=O)NCCC#N)N1C(COC)CCC(C(=O)OC)C1 Cc1ccnc(C(=O)NC2CC2NC(c2cnc(C(C)C)nc2)=O)c1 Cc1cn(C)nc1CNc1nccc(N(C)Cc2nnc(C)n2C)n1 C1(C(N2CC3C(NC(c4c(C)sc(O)n4)=O)(C3)C2)=O)CC1C1CCCCC1 c1(SCC)cnc(O)c(C(=O)NC2CCN(C(=O)Cn3c(C)ccc3C)C2)c1 N1(C(c2c(C)c[nH]n2)=O)C(C(=O)NCC2(F)CCOC2)CC2CCCC12 c1(CSC)cc(C(=O)NCC(CC)NC(c2ccc3c(c2)CC3)=O)ccc1F C(CCC1CC1)(C(=O)N)NC(CC1CC(OC)C1)=O.CCC(C(C)C)N(C)C N1(C(C2C(=C)C2)=O)CCC(C(C)C(=O)NOCCC(F)(F)F)CC1 C1(NC(c2c(C)nc(C)o2)=O)CCCCCN(C(C23CCCC2(C(N)=O)C3)=O)C1 N1(C(c2cnc(OC)s2)=O)CC(C)C2(CCC2)C1.C1(C=O)CCCC(=O)N1C.N C(=O)(C(C)(C)C)NCC.C1(C(=O)N)CSCN1C(=O)C=CC1CCOC1 N1(C(N)=O)CCCC(NC(=O)NCC(C(F)(F)F)N2CCOCC2)C1 C=CCC(CC)C(=O)NC1(C(=O)NCC23CCC(CO2)C3)CSC1 C(Cc1ccccc1)(C(=O)NCCN(C(=O)COCCOC)C)OC C1(C(C(N2CC(CC=C)(NC(=O)CN(C)C3CC3)C2)=O)C)CCCCCC1 Cn1nc(CC(=O)NC2CCC(CNC(=O)C3CC3)C2)c2ccccc2c1=O N1(C(C(=O)NCCSC)C(C2CCC(F)(F)CC2)C)CC(C)Cc2ccccc21 C(=O)(C(C)(C)CCOC)N1CC(C(=O)NCCOCCCC#C)C(CCC)C1 c1(CC)ncoc1C(N1CCC(CC(=O)NCCS(=O)(=O)NC)C1)=O C(C)(C)(CC(=O)N1CCCC(CF)C1)N(C(CCSC)=O)C C(=O)(C(CC)CCOC)NC1(C(N2C(CC=C)CCCC2)=O)CCCCC1 c1(OCC#C)ccc(C=O)cc1.c1(C(N(C(C)C)C)=O)ccnc(C2CC2)c1.N c1(SC)cccc(C(=O)NCCCC(C)NC(=O)Cc2ccc(C(F)F)cc2)c1 CC1(C(=O)NCc2ccnn2C(C)(C)C)CN(C(=O)C)C1.C1(C)CCC1 N1(C(c2ccc(I)cc2)C(=O)NCCOC)C(C)CN(c2ccccc2)CC1C CC1(C)C(C)(C)C1(F)C(N1CCN(C(=O)C2=NOCC2)C(CC(F)F)C1)=O C1(CNC(C2(CC)CCCC2)=O)CN(C(=O)Cc2ccc(F)cc2)CCO1 C1(C(=O)NC2(CNC(c3csnc3Cl)=O)CCOCC2)CC2C=CC1CC2 N1(C(c2ccc(CC)[nH]2)=O)CC(CNC(=O)C(F)Cc2ccccc2)C(C)C1 c1(CNC)nc(C)c(CNc2cc(Oc3ccccc3)ncn2)o1 c1(C(=O)NC(C2CCN(C(C3CC(F)(CO)C3)=O)C2)C)ncc[nH]c1=O c1(OC)cccc(CN2CCOCC2C(=O)NC(C)C)c1.C1C(=O)N1 c1(C(=O)NCC(CC)NC(=O)C=C(Cl)Cl)ccc(OCc2nccs2)cc1 C1(CCNC(C2(O)CC(F)(F)C2)=O)CCCCN1C(=O)C=CBr C1(N(C(c2ccc[nH]2)=O)CC)CCN(C(c2cc(C(N)=O)ccn2)=O)CC1 S(=O)(=O)(c1cnn2ccc(N3CC4CCC4(C)C3)nc12)NCCCOC CC1(C)NC(=O)CC1C(N1CC(F)(C)C1)=O.C(=O)(C(F)CC1CCOC1)N C1(NC(C(C2(O)CCC2)NC(Cc2c(C)cccn2)=O)=O)CCCC2(CC1)CC2 C1(C(N(CCCNC(=O)CC(C)(C)C2CC2)CC)=O)CCCC2(CC2)C1 Cc1nc(C(N2CCCCC2CC)=O)c(C)n1C1CC1.c1(C(=O)N)cc(F)c[nH]1 C12(NC(CCN(C)CC)=O)CCC(CC1)N(C(c1ccc(CF)cc1)=O)C2 CC1=C(C(=O)NCC2COCC2NC(=O)CC(C)C2CCCC2)CCCO1 N1(C(CC(C(C)C)O)=O)CC2CCN(C(c3ccc(C(N)=O)cn3)=O)CC(C2)C1 C1(NC(=O)CC23CC(C2)C3)CCN(C(=O)Cc2ccsn2)CC1F CN1N=C(C(=O)N2CC3C(NC(c4ccc5nnn(C)c5c4)=O)C3C2)CCC1=O C1(NC(C(COC)O)=O)CCC2CC1CN2C(=O)CCCS(N)(=O)=O C1(C(C)C)C2CN(C(=NCCF)NCc3ccc(-n4ccnn4)cc3)CC12 CC(O)(CC(=O)NC1CCC1CNC(c1cnc2ccncc2c1)=O)C(F)(F)F CC1(C)CCn2cc(CNC(c3cccc(Cn4cnnc4)c3)=O)nc21 C12(NC(C3N(C=O)CCC3)=O)CC3CCC(C1C2)N3C(=O)CSc1nncs1 C1(CCOC)CN(C(=O)C(c2ccc(Cl)s2)C)CCN1C(c1ccn(C)c1)=O C1(C(=O)NC(CCCCNC(c2c(C)onc2)=O)CO)CN2CC3CC2(CO1)C3 c1(-n2c(C(c3ncco3)Nc3cn(CCF)nc3)nnn2)ccc(F)cc1 C1(NC(CS(C)(=O)=O)=O)CCCN(C(c2cocn2)=O)CCC1 C1(C)(C(=O)NCC(C)N(C(c2ccn(C)c2)=O)CC)CC=CCO1 c1(OC)ccc(F)c(C(N2CCCCC2CNC(=O)C=O)=O)n1.CCC(N)=O c1(OC)cc(NC(C2(N)CC2)=O)cnc1Cl.c1cccnc1-c1ccc(F)cc1.C CCC(C)(CNC(c1ccnn1CC1CCC1)=O)NC(=O)CN1CCCC1 N1(C(C2C(COC)C2)=O)CCC(NC(c2cn(CCOC)nn2)=O)C1C N1(C(c2c(CC)[nH]nc2Cl)=O)CC2(CC(NC(=O)C(F)C(F)(F)F)CO2)C1 Cc1ccc(C(=O)NC(C)C(C)(C)NC(=O)CC2CCC(=O)N2C)c(C)c1 C(=O)(C(O)C(F)(F)F)NCC1(CCCNC(C2C(C)OCC2)=O)CCCC1 C1(C(=O)NC(CC)CNC(=O)CN(C)C(c2ccoc2)=O)CCCCN1C C1(C(N(CCC#C)C(C)(C)C)=O)(C(=O)OC)C=CCC1 c1(CCC(=O)N(C(CCNC(C2(C(C)C)CCC2)=O)C)C)cc(Cl)sc1Cl c1(C(=O)NCC2N(C(CCC3OCC(C)(C)C3)=O)CC2)cc[nH]c2nccc1-2 c1(CC(=O)N)cnc2ncccn12.CC(Cc1cnc[nH]1)C(=O)NC1CCC1C c1(C(C)C)nc(NCC(C)Cc2cccs2)cc(N2C3CCCC2CC3)n1 CC1(C)CCN(C(c2ccc(F)c(N)c2)=O)C1CNC(=O)Cn1cnnn1 c1(C(=O)NC(CCNC(c2cn(CC)nn2)=O)C)c(C(F)(F)F)coc1C C(CCC1CCC1)(C(=O)N)NC(CC1(OCC)CCC1)=O.C1(F)CC1.C C1(C(=O)OCC)CCN(C(=O)CCc2cc3ccccc3o2)CC1C1CC1 Cc1cc(C)n(CC(=O)NCCC2(O)CN(C(=O)C(C)(C)CC3CC3)C2)n1 N1(C(C23CCC(OC)C2C3)=O)CC(C(=O)N)CCC1(C)C.c1(CCC)cnc[nH]1 c1(N2CCC(=CCNC(CC(C(F)(F)F)OC)=O)CC2)ncc2cnn(C)c2n1 C(C)(C(=O)NNC(=O)c1cc(S(N)(=O)=O)ccc1N)(c1ccccc1F)OC C(C)(CCCCNC(c1nc(C(C)C)oc1C)=O)NC(C(C)OC)=O Cc1nc(Cl)ccc1C(N1CCC(CNC(=O)C2=COCCO2)CC1C)=O Cc1cccc2c(C(=O)Nc3ccc(-c4ccc([N+](=O)[O-])cc4Cl)cc3)n[nH]c12 N1(C(C(CC#C)(C)C)=O)CC2(CCN(C(c3csc(C4CCOCC4)n3)=O)C2)C1 Cc1cnc2ccccc2c1C(=O)NCCCN(C(=O)C(C)(C)C)C1CC1 CC1CC(N=c2nc[nH]n3cccc23)CN1C(c1cc2c(cn1)CCCC2)=O Cc1ccc2c(C(=O)NCC3CN(C(=O)Cn4cccn4)CC3O)c[nH]c2c1 C(=O)(C(C(C)(C)CC)OCCO)NC(CC)CN(C)C(c1ccc(OC)cc1)=O CCCC(C)(O)C(=O)NC1CN(C(c2ccc(F)c(C(F)(F)F)c2)=O)CC1(C)C C(C(CCC)C(=O)NCC=CC(C)(C)C)NC(C(CSC)C)=O c1(OC)cc(C(=O)NC(C)CCNC(C2CC2[N+](=O)[O-])=O)cnc1O c1(C(=O)NC2CC3CC(NC(C=COCC)=O)CC32)cnc2ccccn2c1=O CCCCC(C)C(=O)NC1CCN(C(c2sc(C)cc2Cl)=O)C1 C1(CNC(CN(C)C(c2ccc(Br)s2)=O)=O)CCN(c2ccncc2)CC1 N1(c2nc(C)nc(Cl)c2)C2CCC1CC(CNC(=O)CSc1ccccn1)C2 O=C(C1=CC(O)CCC1)NC1CCCCN(C(c2ccnc(Cl)c2O)=O)C1 c1(C(N2CCC(N(C(=O)CCC3CCC3)CCC)C2)=O)coc2c1C(=O)NCC2 c1(C(=O)NCC(CNC(=O)CC2CCCCC(=O)N2)O)ccc(F)c(F)c1F CN=c1[nH]c(C(=O)NC(C)(C)CCNC(C2(C)CC3CC3C2)=O)cs1 N1(C(c2cocn2)=O)CC2(CCC(=O)NC2)C1.C1(C(=O)OC)CC1C(=O)N C1(NC(=O)Nc2c(SCCCC)cccc2)(CCCCC)CCNCC1 CC1CN(c2nnc(C#N)s2)CCC1NC(c1snnc1C1CC1)=O CCCCC(=O)NC1CN(C(C23CC(CF)(CO2)C3)=O)C1.C(C)(C)C.C=O Cc1cc(Br)cc(Cl)c1NC(N1CC(C)CC1C(N1CC(F)(F)CC1C#N)=O)=O CC(C)CCC(=O)NC(C)CCNC(c1ccccc1Nc1cccs1)=O CC1CN(C(c2cnco2)=O)CC1NC(=O)C(C)(O)C1CC1 C1(CCNC(Cc2cn(CC)nc2)=O)CCCN(C(c2ccc(Cl)[nH]2)=O)CC1 CN1CCC(CC(N2CC3C(CN(C(=O)CC4CC5(CCC5)C4)C)C3C2)=O)CC1 N1(C(Cc2n(C)ncc2)=O)CC2CCC(C1)C2NC(=O)CC(O)C1CCCC1 c1(C(=O)NC2C(NC(C3CC(C)C3)=O)C2)scnc1Cl CCCCCCC(F)C(=O)NCCCCC(C)NC(c1ncc(F)cc1F)=O C1CN(C(c2ccccc2C2CC2)=O)CC1(F)F.c1(C(=O)N)coc(C(F)F)c1 N1(C(c2ccc(C#C)cc2)=O)CCC2(C(=O)N(C3CC34CC(O)C4)CC)CCCC12 CN1CCCCC(NC(C2CC(=O)C23CCCC3)=O)C1=O Cc1n[nH]cc1C(=O)NCC(C)N(C)Cc1cn(Cc2cccs2)nn1 Cc1cnnc(O)c1C(=O)NC1CC(CNC(c2ccn(CCF)n2)=O)C1 N1(C(C2(CC)CC2)=O)CCC(CCNC(c2cnc(C(C)C)[nH]2)=O)CC1 C(=O)(CCN=c1[nH]c2ccccc2s1)N1CCC(CNC(C(F)=CCC)=O)CC1 C(=O)(CCCCN1CCCCC1)NCC(CC)(C)NC(c1ccn(C2CC2)n1)=O c1(C(=O)NC2(C)CCC2)ccc(O)c(C(N)=O)c1.C(=O)(C(F)n1cccn1)N c1(C(=O)NC2(CCN(C)C)CC2)cc(-c2cnn(C)c2)nc2ccccc12 CC1CN(C(c2cnn3ccncc23)=O)CCC1N=c1[nH]c2c(F)cccc2o1 c1(C(=O)NC2C=CCN(C(c3c(CC)nns3)=O)C2)ccc(F)cc1F CC(C)C(CNC(c1cc(Cl)ns1)=O)C(=O)NCC1=CCCOC1 C1CN(C(=O)Cn2cccnc2=O)C(C)(C)C1.c1(C(C)C)occc1C(=O)N.C C1(CC)CCCC1C(=O)N(CCCNC(c1cccn1C)=O)C.c1ccccc1 C(=O)(C1=C(Cl)CCC1)NC(c1ccccc1)C(C)NC(=O)CCN(C)CCO CC1CN(C(C2(C)CCCO2)=O)CC1N(C)C C1(C)(NC(C(OC)OC)=O)CN(C(=O)CCc2nc(C)cs2)C1 CC1CN(C(=O)C=Cc2ccc(C(F)(F)F)cc2)CCC1N(C)C c1(-c2onc(C(=O)NCc3cn(CCN4CC(C)C4)nn3)n2)cccc(F)c1 C1(NC(C2CCC23CCC3)=O)CC2(CCN(C(c3ccnnc3)=O)C2)C1 CCC(C(=O)NC1CCCCC1N(C)C(c1cc2c(s1)CCC2)=O)C(C)C CN1CCC(N(C(=O)C(=O)NCc2ccns2)C)C1=O C(=O)(C(C)(C)C1CCN(C(C2CC(=O)CS2)=O)C1)N(CC(=O)N(C)C)C C1(NC(Cc2cc(C)on2)=O)CCN(C(c2cc(Cl)ccn2)=O)C2CC12 C(C1=CCN(C(c2cn(CC(F)F)cn2)=O)CC1)NC(C1(C)CCN(C)C1)=O Cc1cc(S(=O)(=O)N(C2CCCCC2C)CC(F)F)ccn1 c1(CC)cc(C(=O)NC2CC(NC(C3(O)CC3(C)C)=O)C2)n(C)n1 C1(CNC(CN(C(C)=O)C)=O)C2CC1N(C(=O)Cn1nc(C)cc1C)C2 C1(C)(C(=O)Nc2c(C)noc2C)CCCN(CCc2ccccc2Cl)C1 c1(Cc2nnn(C(COC)(COC)C(=O)O)n2)c(OC)ccc(OC)c1[N+](=O)[O-] C(=O)(CCCC#CC)NCC(CC=C)NC(c1cc(NC(C)=O)ccc1F)=O C(=O)(N=c1[nH]nc(CC(F)(F)F)s1)C1CC(C)N1.c12cccc(n1)OCC2 N1(C(C=C(C)C(C)(C)C)=O)CC(O)CC1CNC(=O)CCCN(C)C N1(C(C=CC)=O)CCOC(CCNC(c2cnn(C)c2SC)=O)C1 N1(C(C2CC(CC)(CC)C2)=O)CCOC(CNC(=O)C(CC)N(C)C)C1.S N1(C(C(CC)SC)=O)CCN(C)CC1CNC(c1coc(C#N)c1)=O c1(C(N2CC(C)C(CNC(c3cncc(F)c3)=O)C2)=O)cc2sccc2n1C N1(C(C2CC(OC)C(OC)C2)=O)CCCC(F)(CNC(=O)CC(C)SC)CC1 CN1CCn2ncc(C(=O)NCc3ccc4nnnn4c3)c21 C1(CNC(C(C)NC(=O)NC)=O)CN(C(C2CC2(F)Cl)=O)CC1(F)C C#CCCC(O)CCNC(=O)COC1CN(C(=O)CC(CN(C)C)CC)C1 N1(C(c2c(C)cc[nH]2)=O)CC2CC(NC(=O)CCCNC(=O)C3CC3)CC2C1 N1(C(C(CC#C)O)=O)CC(C)(C)OCC1CNC(=O)Cc1cccc(SC)c1 c1(C(N(CCN(C(c2cnco2)=O)CC)CC)=O)cc([N+](=O)[O-])ccn1 c1(CN(CC(Cc2ccc(OC)cc2)O)C=O)cc(C)ccc1Br N1(C(CC2ON=C(CC)C2)=O)CC(F)(F)CC1C(=O)NCC(CC(C)C)N(C)C Cc1cccn2c(C(N3CCS(=O)(=O)C(CCNC(=O)CC(C)C)C3)=O)cnc12 C1(NC(C2CCCN(CC)C2)=O)CCC2(CC1)CC2NC(=O)CC(C)(C)O C1(NC(c2n(C)ccc2)=O)CN(C(=O)C2=CCCC2)CC2CCCC12 c1(C(=O)NC2(CNC(CC3(C)CC3)=O)CC2)csc(C2CCCO2)n1 C12(NC(c3c(CC)nc(Cl)cc3)=O)CCCN(C1)S(=O)(=O)C2 C1(CC)C(C(=O)NCCOCC(=O)N(c2ccc(C)cc2)C)CCN1C C1(CC(=O)NCCCCOC)C(=O)N(C)N=C1C.c1(C=O)csc(=N)[nH]1.N c1(CNC2C(C)CCNC2)cccc2c1CCO2 N1(C(Cc2ccc(C)o2)=O)CCN(C(C2CCC(CCO)CC2)=O)CC1C1CC1 C1(COC)CC(O)CN1C(=O)C(C1CCN(C(C2(C#N)CC2)=O)CC1)C N1(C(=O)NCCCCC(=C)C)CCC(Oc2ccc(CC)cc2)C12CCC2 C12CCC(CC1)C2(C)C.CC1CCCC(C(=O)NCCc2n[nH]cc2C(=O)N)C1 C1(C)(C(=O)NCCCCC(C)NC(c2cnc(C)nc2C)=O)CCCNS1(=O)=O CC1CC2(CC(C(=O)OCC(C)(O)C)C2)CN1C(N)=O.C(C)(C)C.C=O C12(C(=O)NC(CC)CNC(C3CC=C(C)CC3)=O)CCC(CC1)CC2 C(N=c1cc(C(N)=O)nc[nH]1)C1CCN(C(C(c2c(C)cccc2)C)=O)C1 c1(C(N2C(CCC(=O)NC3CC3)CCCC2)=O)ccc([N+](=O)[O-])o1 N1(C(CCN(C(C)=O)C)=O)CCC(N(CCO)Cc2cc(C)nn2C)CC1 C(=O)(CCC1=CCCCC1)N1CC(n2cc(C3C(C)C=C(C)CC3)nn2)C1 N1(C(C(C)(C)C(N)=O)=O)CCC(C2(NC(C3CC3c3cccs3)=O)CC2)CC1 c1(C2(CNCCO)CC2)cnc2ccsc2c1 C12(NC(C(CSC)OC)=O)CC1CN(C(=O)CCOC1CC1)C2 c1(C(N2CC(C(C)NC(C(CNC(C)=O)(C)C)=O)C2)=O)[nH]c2ccccc2c1Cl C1(CNC(C(CCOC)C)=O)CC2COCC2N1C(=O)C=Cc1cncn1C c1(NC(C2CC(C(=O)OC)C2)=O)ccc(NC(C)=O)nc1 c1(C(C)OCC2CC2)nc(-c2ccnn2C)nn1-c1ccc(Cl)nc1 Cc1nnc2ccc(C(=O)NC(C)C(CO)NC(C3(CO)CCCC3)=O)cn12 C(=O)(C(O)CCCNC(C1C=C(C)CS1)=O)NC(CC(=O)OC)C1CC1 C1(c2nnnn2CCCF)(NCCc2c(C)cncc2)CC(C)(C)OC(C)(C)C1 CCC(C(=O)NCC1CN(C(=O)C#CC2CCCCO2)C1)C(C)(C)CC N1(C(CN(C)CCc2ccccc2)=O)CCC2(NC(C3CCCC3)=O)CC2C1 c1(NC(C(CNC(C=Cc2n(C)cnc2)=O)(C)C)=O)cccc2ccncc12 N1(c2nnc(CC(=O)OCC)s2)CCC(NC(C2C=C2C)=O)C(C)C1 C1(C#N)(C(N2CCC(NC(CCc3n(C)cnc3)=O)C(F)C2)=O)CC12CCCC2 c1(C(=O)NCCC2CN(C(C3N(C)CCC3)=O)C2)csc2cncn12 c1(C(=O)NC(CNC(C2CC(=C)C2)=O)C(C)C(C)C)cc2cc(C)[nH]c2cc1Cl c1(CCC(=O)NC2C3CN(C(c4c(C)ocn4)=O)CC32)c(C)[nH]c2ccccc12 C(N=c1[nH]c(=N)[nH]c(=NCCCNC(=O)C(C)(C)C)[nH]1)C1C(C)COCC1 C(CC(C(=O)N(C)Cc1csnc1C)NC(c1cccnc1O)=O)=CC c1(CC(N2CCC(CN(C(C3CCC(C)O3)=O)C)C2)=O)ccc([N+](=O)[O-])cc1Cl C1(CC(=O)NC2(CO)CN(C(C(c3ccccc3F)C)=O)C2)CCC(F)(F)CC1 c1ccccc1C#N.N1(CC(=O)NC(CN(C(=O)CO)CC)C)CCNC1=O C(N=c1[nH]c(N2CCC(C)(CS(C)(=O)=O)C2)nc2cc[nH]c12)c1c(C)nccc1 C1(CC)C2CN(C(=O)CC3(NC(=O)C(C(C)C)OC)CC3)CC12 c1(C(C(=O)NCC(CNC(C=CC(C)(C)SC)=O)C)=O)cccn1C N1(C(c2ccc(C)cc2)=O)CC2COCCC2(NC(=O)CCc2cnc(C)s2)C1 C1COCC2(CCN(C(=O)CC(=O)N(C)C)C2)O1.C(C(COC)C(=O)N)OC.C c1(C(=O)OC)nccnc1N1CC=CC(NC(=O)C(O)C2CCCC2)C1 c1(CC)nonc1C(=O)NCC1CCCC1NC(C1(C)CC(F)C1)=O Cc1ccc(C#N)c(NC(C2CC2C(=O)NCc2ccccc2[N+](=O)[O-])=O)c1 C(C(C)C)(C(O)C(=O)NC1CC2CC1N(C(=O)CCc1ccccc1O)C2)OC c1(CC)ccc(C)cc1C(N1CCC(CNC(C2CC3CCC3C2)=O)C1)=O C1CC2(C1)CN(C(=O)CC1C=CCC1)C2.c1(C(=O)N)cc(-c2ccccn2)no1 c1(OC)ccc(CCC(=O)NC2CN(C(=O)CCCNC(C)=O)CC2C)cc1F N1(C(C2CC(=C)C2)=O)CCCN(C(c2cnn(CC3CCCCO3)c2)=O)CC1C c1(C=O)ccc(N(C)C)nc1.C1(C(N(CCC)CC)=O)CC(=O)N(CC)C1 N1(C(CC)=O)CCC2(CCN(C(=O)CC3C(CC)C3(F)F)CC2)C(C)C1 C(=O)(Nn1cnn(C)c1=S)c1n[nH]c2c1CN(C(c1c(C)cncc1C)=O)C2 c1(C(C)C(=O)N(CCCCCCNC(c2nn[nH]c2Cl)=O)C)nc(F)ccc1Cl N1(C(C(CSC)O)=O)CCC(CC(N)=O)(NC(c2ncc(Cl)cc2F)=O)CC1 N1(C(C2(C(N(C)C)=O)CC2)=O)CCCC(F)(C(N2CCCC(F)C2)=O)C1 C1(CNC(c2c(OC)nccn2)=O)CC(C)(C)CN1C(=O)CC1CC1.S C1(CC(N2CC(SC)C2)=O)CN(C(C2CC2C(N)=O)=O)CC12CC2 C1CCN(C(C2C3COCC23)=O)C12CCC2.c1(C(=O)NC)cncc(C(F)F)c1 c1(C(N(C(C)CNC(=O)C(O)C(C)(C)C)CC)=O)cc(O)cc(N)c1C c1(CCCC(=O)NCC2CCN(C(=O)CC3(F)CCOCC3)C2)ccccc1Cl C(C)(CC(C)C)NC(c1c(CCC)nco1)=O.c1(CCC(=O)N)cccc(F)c1 c1(CC)ccnc(C(=O)NC2CC(C)(C(N3CCC(O)(C(F)F)C3)=O)C2)c1 C1(CC(=O)NC(C2CN(C(c3ccc[n+]([O-])c3)=O)CCO2)C)CCC(=O)NC1=O c1(C(N2CC(CNC(c3c(OCC)ccs3)=O)C2)=O)cc2ccoc2cn1 Cc1cc(C(=O)NCC2CCCC2C(=O)NC)c(C)nn1.c1ccc(F)cc1 N1(C(c2c(C(C)NC(=O)C(C)O)noc2)=O)CC2(COC(C)(C)C2)C1 N1(CC)CCC(CNC(=O)CC2CCCCC2)CC1.C12(C(=O)N)CSCC1C2 N1(C(CC(=C=C)C)=O)C2CCCC1CN(C(C1CC3(C1)CC1(CC1)C3)=O)C2 C(=O)(CC1=CCCCC1)N1C(CN(C(=O)C=CC(F)F)CC)CCC1 C1(C(=O)OC)(NC(=O)C(C(C)(F)F)c2ccccc2)CCC(F)(F)CC1 n1(CC)nc(C(=O)N(CCNC(=O)CC(C)C2CCCO2)C2CC2)cc1O c1(C(N2CCC(NC(CCC(CC)OC)=O)C2C)=O)ccc2ccccc2n1 CCCCC(C(=O)NCc1ccsc1C(=O)NCCO)C(C)C.CC(F)(F)F Cc1ccc(CC(=O)NC2CC2CNC(=O)C(C)Oc2ccccc2Cl)cc1 C1(C(=O)N)CC2(CCC2O)C1.c1(CC(=O)N(C)CC2(C)CC2)nc[nH]n1 C1(NC(C2CSCCS2)=O)C(CNc2ncnc3scnc23)CCC12CCC2 CN1C(=O)CC(CNC(=O)CONC(C2(C)CNC(=O)N2)=O)C1=O CCCCCC(C)(CC)C(=O)NCC(CNC(=O)CCc1ccccc1F)CO N1(C(C(C)(C)C2(O)CCC2)=O)CCCC(NC(=O)COCCCF)C1 C(=O)(C1=CC2CCCC12)NC(C1(O)CCN(C(C2Cc3ccccc3C2)=O)C1)C C(N=c1[nH]c2c(c(=NCc3ccc(C)nn3)[nH]1)COC2)C1OCCN(CC)C1 C(=O)(C1=CCC2CCC1N2C(C)=O)NC1CCCN(c2c(OC)cccc2)C1=O N1(C(c2cc(C)sc2C)=O)CCCCCC(NC(C23CC(C)C2C3)=O)C1 C(C)(CN=c1nc(-c2ccccc2)nc(N2CCCCCC2)[nH]1)SC c1(C(N(CC(C)NC(C2CC(SC)C2)=O)CC)=O)nc2n(c1Cl)CCCC2 N1(C(CCCCC(CC)C)=O)CCC(C2(O)CC(NC(=O)CC=C(C)C)C2)CC1 n1(CCC(=O)N(CCCNC(=O)CC2CCCC(O)C2)C)ccc2ccccc12 C=CCC(C(=O)N1CC(O)CC1C(N1CCC(CCC)(CO)C1)=O)OC C1(CCO)(NC(C2CC(N(C)C(C3CCSC3)=O)C2)=O)CCCCC1 c1(OC)cc(C(N2CC(C)C(C)C2)=O)ccc1C#N.C1(C(=O)N)CC2(CC2)C1 N1(C(CC(CCC)C)=O)Cc2n[nH]cc2C1C(=O)NCCCc1ncnn1C N1(C(C(C)OCC=C)=O)CC2(CCN(C(c3cc4cscc4s3)=O)C2)C1 N1(C(c2cc(C)sc2C)=O)CCC2(CCC(NC(=O)CS(N)(=O)=O)C2)CC1 CCCCC(CNC(c1cccnc1OC)=O)NC(C1CCC(O)C1)=O O=C(O)C(F)(F)C1CN(C(c2cnnn2C2CC2)=O)C1 C(=O)(C(C)C(C)NC(=O)C(O)CCNC(c1ncoc1C)=O)OC c1(C(=O)NCC(CC)NC(c2nn[nH]c2Cl)=O)cc(Cl)cnc1C C1(C(N2C(C)CC(OC)C2)=O)CCC2(CCC2)C1.C(c1cc[nH]c1)=CC=O.N C(C)(C(C)(C)C(=O)NCCC1CCSC1)NC(COCC(=C)C)=O C(=O)(CCCC(=O)N1CCC(C(=O)N)C(C)C1)OCC.c1ccc2c(c1)CC2.C N1(C(CC2CC(C)(C)C2)=O)CCC2(CCCC2NC(c2cc(N)ccc2Cl)=O)C1 C(=O)(C1=CC2CCCCCCC12)NCC1CN(C(Cc2c(CC)cccc2)=O)C1 C1(NC(c2c(Cl)ncc(OC)c2)=O)CCCC2CN(C(c3csc(Cl)c3)=O)CC12 Cn1ccc(=NNC(=O)C(C)OC(F)(F)F)cc1C(N)=O c1(CNCCc2cc(Br)sc2)ccc2c(c1F)OCCO2 C12(CNC(CC(C)(C)C)=O)CCCC(CN1C(=O)Cc1cc(F)ccc1Cl)C2 C1(C(N2CCNC(c3cn[nH]c3)C2)C(=O)NC2CC2)CC2(C1)C(F)(F)C21CCC1 O=C(C1=CC2CC(C1)CC2O)N1CC(F)(c2cn(CC(F)(F)CO)nn2)C1 C1(CC)CN(C(c2cc(Cl)ns2)=O)CC1C(=O)N(C(C)CCO)C C(=O)(CCCC1CC1)NCC1(C(=O)OC)CC1.c1(C=O)cc(O)ncn1 C1(NC(Cc2ccc(C(=O)OC)s2)=O)CCCC1(C)NC(=O)C#CC(C)C C1(CCNC(c2coc(Br)c2)=O)CSCCN1C(c1ccnnc1O)=O CC(C)(C)CC(=O)NC(Cc1ccccc1)C(C)NC(=O)Cn1cc(Br)cn1 C(=O)(CCCCC(N)=O)N1CC(CCNC(c2cnc(OC)s2)=O)OCC1 C(=O)(CC(C)C(C)(C)NC(=O)C(C)=C(C)C)NC(COCCOC)C S(=O)(=O)(c1cccnc1Cl)N1CCN(C(c2c(Cl)cccc2I)=O)C2C1C2 C=C(CNC(C1(C)CC(C)(C)C1)=O)C(F)(F)F.c1(CC=O)sccc1C CC1(CC(N2CCCC(NC(C3C4COCC34)=O)CC2)=O)Oc2ccccc2O1 c1(CNC(=O)C=C2CCC2)ccc2c(c1)CCC2NC(=O)Cn1nccn1 c1(C(=O)NC(C)C(C)(C)NC(c2nsc3ccccc23)=O)cnn2ccn(C)c12 C=CC(C)(C)CCNC(c1cnc(CNC(C2(OC)CCC2)=O)nc1)=O c1(NC(C2CC(OC)CN2Cc2ncccc2C)=O)cc(O)cc(Cl)c1 Cc1c(F)ccc(Cl)c1C(=O)NCCC1CCCCN1C(c1nc(O)c(C)s1)=O N1(C(C(CC#C)C)=O)CC2CCC(C1)N2C(=O)C=C(C)c1cnn(C)c1 C(C(COC)CC(=O)N1CCC12CN(C(=O)CSc1n[nH]c(C)n1)C2)OC C1(CNC(C(C)(C)OCC)=O)CC2CC1CN2C(C1CCCCNC1=O)=O C1(NC(C2(C)CC2(F)F)=O)CCC(CC(=O)NC2CCCC(C(N)=O)C2)CC1 C(N=c1cc(C)c(C#N)c[nH]1)C1(C)C(OC(C)(C)C)CN(C(=O)OC)C1 C1(NC(CCC=CC(C)C)=O)CCC12CCN(C(=O)CC1(C)CCOCC1)CC2 C(C)(CN=c1[nH]c2ccccc2s1)NC(CC(c1c(C)n[nH]c1C)C)=O c1(CNC(C2(COC)CC(=C)C2)=O)ccc(C)cn1.C1(C=O)C=CCC1 N1(C(=O)CCN2CCCC2=O)CCCC(C2CCN(c3cc(O)nc(O)n3)C2)C1 C1(C(=O)NCc2scc(C(N3C(C(C)O)CC3)=O)c2)(CO)CC(C)(C)C1 CC(CCN(C(CCc1cccc(F)c1)C(=O)NC1COC1)C)C(F)F C(c1ccc(Cl)cc1F)=CC(=O)NC1CCC1.c1(C(=O)N)cnccc1C(F)F C(=O)(C1=CC(C)(C)C1)NC1(C(=O)Nc2cnc(N(C)C)nc2)CSC1 N1(C(CC)=O)CCC(NC(C2CN(c3nnc(C(N)=O)s3)CCO2)=O)CC1 c1(C(CC)CC)cn(CC2CCC2CNC(=O)C)nn1.CC=O.C(C)(C)C CC1(C)CC(CNC(c2n[nH]cc2Cl)=O)CN(C(C2(C)CC(C#N)C2)=O)C1 C(C(C)(C)CC)(c1n(CCCC)nnn1)NCCOCCCOC C(=O)(C(C)(C)S(C)(=O)=O)NC(C)CCC(=O)NCCN1CCOCC1 N1(C(c2c(CC)c[nH]c2)=O)CCCCC1C(C)NC(c1sc(OC)nc1C)=O N1(C(C(CC)CC)=O)CC2CC(NC(=O)COc3ccon3)CC2C1 C(=O)(CC(CC(N)=O)CC(C)C)NCC1N(C(C(Br)=C(C)C)=O)CC(O)C1 c1(C(N2CC3(OCC(N)C3)C2)=O)cc(OC(=O)C(F)(F)F)ccc1[N+](=O)[O-] C(=O)(C1=CC2(CCOC2)C1)NCC(CCNC(c1ccc(N)cn1)=O)O C1(C=O)CCN(S(C)(=O)=O)CC1.c1(CC)nc(C(C)(C)C)no1.CCC(N)=O N1(C(C=CC2(C)COC2)=O)CCC=CC1C(=O)NCC(F)(F)Cl CC1C(NC(C2C3COCC23)=O)CCCN1C(c1cnn(C(C)(C)C)c1Cl)=O C(CC(O)CCO)NC(C1CCN1C(C1CC2(CSC2)C1)=O)=O c1(C(N2CCC(C(C)OC(C)=O)CC2)C(=O)NCCCC)ccc(Cl)c(C)c1 C(=O)(CC(C)(C)C(=O)OCC)N1CCOCC(CNC(C(C(CC)C)O)=O)C1 c1(N2Cc3c(ccc(C)c3)OCC2)nc(=NCC2(CC3CC3)CC2)[nH]c2ccccc12 N1(C(C=CC=CC)=O)CCCCC(NC(=O)C(C)Cc2ccccc2Cl)CC1 Cc1[nH]nc(C(N2CC(C(N)=O)(CNC(c3cc(Cl)cs3)=O)C2)=O)c1O N1(C(C(CC)Oc2ccccc2C)=O)CC2(C1)CN(C(C1(O)CC1)=O)C2 Cc1cncc(CC(=O)NCC(C)(C2CC2)NC(c2cc(C3CCC3)no2)=O)c1 N1(C(C2(C)CCCOC2)=O)C2CCC1CN(C(=O)CCN)C2.[SH](=O)(=O)C(F)(F)F C(=O)CC(CC)C(F)F.C(C)(C)(C)OCC(=O)N(CCCC)CC(N)=O.N C#Cc1ccc(C(=O)NC(C)CC(C)NC(C2(C(F)F)CCC2)=O)c(C)c1 c1(C(=O)NCC(C(C)C)NC(C(C)=O)=O)ccnc(Cl)c1 Cc1ccc(NC(N2CCC(OCCC(C)(C)CO)C2)=O)c(C)c1 C1(C(N(C2CCCN(C(C(CC#C)(C)C)=O)C2)CCF)=O)CCC(N=[N+]=[N-])CC1 C1(C(N2CCC(n3cc(-c4cnsc4)nn3)CC2)=O)CC2CCC1O2 C(CNC(=O)C(=O)NC1CC1)(CC(=O)NC(C)(C)C(F)(F)F)OC C1(NC(C2CC2(F)F)=O)CCN(C(=O)CC=C(Cl)Cl)C12CCCC2 Cc1nn(CC(N2CC(O)(CC)C2)=O)c(=O)o1.c1(C=O)ccn(CC(F)F)n1.N C=CC(CCC)CC(=O)NCC(C)C(=O)NCc1cc(O)ns1 C12(C=O)COC(C1)C2.N1(C(CCOCC#C)=O)CC(O)(C(C)(C)C)C1.N C1(C(=O)OC)(NC(=O)CCC(CN)C(F)(F)F)CC(C)(C)OC(C)(C)C1 Cc1cc(Cl)cc(C(N2CCC(CCNC(C3CC3(Cl)Cl)=O)CC2)=O)c1N N1(C(c2ccc(C)nc2)=O)CC2CCC(C1)N2C(C1CCCC(C2CC2)O1)=O C1(NC(c2c(CCC)onc2C)=O)CC(O)CN(C(c2nnsc2SC)=O)C1 S(=O)(=O)(c1cccnc1NCc1nnc(CO)s1)NCc1c(C)ccs1 C(CC(F)F)(C(=O)NC1C(O)C2CCOC12)N(C(C(C)c1cc[nH]n1)=O)C N1(C(C=C(C)Cl)=O)CC(NC(c2cnc(S)n2C2CC2)=O)CCC1C C1(NC(C2CSCC(=O)N2)=O)CCN(C(=O)CC2CCCC2)CC12CCC2 C1(C2CCCN(C(=O)CC3OCCC3(C)C)C2)(NC(CCC=C)=O)CC1 c1(C(C2CC(C(C)C)C2)NC2(CC(C)(C)C)CC2)nnnn1C1CCCC1 C1(CN2CCC(Oc3ccc(C(=O)O)cc3)CC2)CC2CCCC2O1.c1(C)cnc[nH]1 C1(C(N(CC(C(=O)OC)(F)F)C)=O)CN2CCCN1CC2 c1(C(c2nnnn2C2(C)CC2)NCC2(COC)CC2)ccc(Br)cc1C N1(C(c2c(C)nns2)=O)CCC2CC2(C(N2CC3(CCC(=O)N3)C2)=O)CC1 C1(CNC(C(N2CCN(C(c3ccco3)C)CC2)=O)=O)CCCOC1(C)C C1(C(N2C(C)CCN(C(C3COC(=O)N3C)=O)CC2)=O)Cc2ccccc2N1C c1(OCC=C)ccc(C(=O)NC2CCC2NC(=O)C(C)O)cc1.C(C)C C1(C(N(C(C)C)CC2CCC2)=O)C2CC(O)C(C2)N1C(c1cnn[nH]1)=O CC1=CCC(C)(C(N2CCCC(CNC(=O)CC3CCCCC3O)CC2)=O)CC1 CC(C)CC(O)C(=O)NCC1(NC(c2cc(N(C)C)ccn2)=O)CCCCCC1 O=S(=O)(c1ccc(NCC(F)CO)c(F)c1)NC1COC2(CCOCC2)C1 Cc1cc(C(C2CC2)NC2(c3nnnn3Cc3cccs3)CCOC2C)c(C)s1 c1(CC)cc(C(N2CCC(NC(=O)C(C)C(C)C)C2C(C)C)=O)ccc1F C(=O)(C(C)CC1CCC1)NCC.c1(CC2CN(C(=O)C)C2)n[nH]c(C)n1 c1(N(CC(COC)(C)C)C)nc(=NCCc2cc(C)sc2C)[nH]c2c1SCC2 Cc1ccc(OCC(N2CCCCCC2CNC(C2C(C)C2(F)F)=O)=O)cc1C c1(OCCC)cc(C)ccc1-c1csc(C(=O)NCc2ccc(CO)cc2F)c1 C1(CC)CC(C(=O)NC2(C)CC(C(=O)Nc3cnn(C)c3C)C2)=NO1 NS(=O)(=O)CCCC(=O)NC1CCC(NC(C2CCCN2C(N)=O)=O)CC1 c1(N2CCCC(CC=C)(NC(c3snc(Cl)c3Cl)=O)C2)nccc(S(C)(=O)=O)n1 Cc1c(Br)ccnc1C(N1CC(NC(C2CCC(=O)N2C)=O)C(F)C1)=O C(CC(=O)NC1C=CC(CO)C1)(C(F)(F)F)NC(Cn1c(C)ccc1C)=O C1(NCc2ccc(OC)nc2)C2CCC1CN(C(c1c(Cl)cncc1Cl)=O)C2 N(C1CS(=O)(=O)c2cc([N+](=O)[O-])ccc21)C(CN1CC2(CC(CN)OC2)C1)=O c1(CNc2c(C)nc(-c3ncccn3)s2)ncc(Br)cc1F Cc1oc(C(=O)NC(C)CC(C)Nc2ncc(Br)cn2)cc1CO c1(CN(CC(=O)Nc2ncc(C(C)(C)C)s2)C)ccc(Br)cc1F n1(CCN(CC(=O)NS(C)(=O)=O)C)cc(CCSC2CCOCC2)nn1 N1(S(C(CC)C)(=O)=O)C2CCC1CN(C(c1cc(F)c(Cl)c(Cl)c1)=O)C2 N1(C(c2cccc(C#C)c2)=O)CC2(CC(NC(c3c(C)ncn3OC)=O)CO2)C1 N1(C(CCCC(=C)C)=O)CCC2CCCC12CNC(=O)C1=CC(C)(C)C1 N1(c2n(CCC=C)c(C3CCC=CCC3)nn2)CCc2ccc(C)cc2C1 C1(OC)CCCC(C(N2CCC(CN(C(c3ccno3)=O)C3CC3)CC2)=O)C1 C1(NC(C=C(COC)C)=O)CCN(C(C2CC3(CCC3OC)C2)=O)CC1F C(=O)(C1=CCOCC1)N(C)CC1N(C(Cc2cc(C(=O)OC)sc2)=O)CCOC1 N1(C(CCC#CC)=O)CCN(C(C2CC2COC)=O)C(CC(F)(F)F)C1 S(=O)(=O)(CC(=O)NC1CCC(CNC(c2cc[nH]n2)=O)C1)NC C(CC(C(C)(C)C)NC(=O)COC(F)(F)F)N(C(c1c(C)cc[nH]1)=O)C C1(CC(N2C(CNC(C(=Cc3cccnc3)C)=O)CC2)=O)CCC2(CCC2)O1 CCCCC(CNC(C1(C2CC2)CCC1)=O)NC(=O)C=Cc1cncs1 c1(OC)cncc(C(=O)NCCCSC(c2ccccc2)c2nccs2)c1 N1(C(CSCC#C)=O)CCN(C(c2cc(F)cnc2O)=O)CC1c1cn[nH]c1 N1(C(Cc2cc(C)[nH]n2)=O)CCCC1CNC(=O)CSc1n[nH]c(O)n1.C CC1CN2CCN1C(C(=O)NC1CC3CCC1N(C(C1CCN(C)C1=O)=O)C3)C2 N1(C(C2(C)C(C)OCC2)=O)CCCC2(C1)CN(C(c1cnc(O)o1)=O)C2 Cc1ccc(F)c(C(N2CC3CCC(C2)N3Cc2ncc(Br)cc2Br)=O)c1F c1(C(N(CCCNC(C2(CO)CCC2)=O)CC)=O)ccccc1.[nH]1cncn1 C1(C(=O)NC2CC3N(C(C=NOC)=O)C(CC3)C2)Cc2ccc(C)cc2S1 c1(C(=O)NCCCC(C)NC(=O)C=CS(C)=O)c[nH]c2cccc(C#N)c12 C1(C(=O)NCC2CC(S(C)(=N)=O)C2)CCC2(C1)CC2(F)F CC(C(=O)NCCc1cc(F)cc(Cl)c1)S(C)(=O)=O.c1(C(=O)N)ccnn1C C(=O)(C(CC(F)F)NC(c1cc(O)n(C)n1)=O)NC1CCN(C)C1 C(=O)(CC(C)CC(C)C)NCC1(C)N(C(C(c2ccccc2)OC)=O)CCC1 C1(CCNC(C2CCOCC2)C(=O)OC(C)(C)C)CC2C=CC1C2 c1(OC)cc(C(=O)N(C2CCN(C(c3ccc(C)o3)=O)C2)C)c2ncccc2c1 C12(C(=O)NC(CC#CC)CO)CCC(CN(C(C3(CC(C)C)CC3)=O)C1)C2 C(=O)(CC1OCc2cc(Cl)ccc21)N(C)CC1CCN(C(=O)C=C2CCC2)CC1 Cc1[nH]c(-c2ccccc2)cc1C(=O)NCC(CO)NC(=O)C(C)c1cc[nH]n1 N1(C(COCCC=C)=O)CC2CC(NC(=O)CCC3CCC(=O)N3)CC1C2 c1(NC(C2N(C(c3c(CC)ncs3)=O)C3CCC2C3)=O)nc2ccccc2s1 C(C(F)(F)CNC(C1CCCC1CNC(=O)C=O)=O)OC.C1CC1.N CC(C(=O)Nc1ccc(OCCC2CC2C)cc1)C(=O)OC(C)(C)C C1(C(N2C(CN(C)C(c3nnc(S)n3C)=O)CCC2)=O)CCC(C)(C)CC1 N1(C(CCCCC(C)C)=O)CCCC2(CCN(C(=O)C(C)O)C2)C1 c1(C(=O)NC23CCN(C(c4cnc(Cl)s4)=O)CC2C3)ccc2c(c1)COC2 N1(C(CCCC#C)=O)CCCC2C1CCCN2C(=O)CCn1ccnc1 N1(C(c2cnn(C(C)C)n2)=O)CC2CCCC2(NC(c2cc(Cl)ncc2O)=O)C1 CN1CCC(C#N)(C(=O)NC)CC1.C1CN(C(=O)CN2CCC(C)(O)C2)CC1O C(C)(CC(F)(F)C(F)(F)Br)(c1n(CC)nnn1)NCCCc1ccsc1 C1(CCC(=O)OCC)CCN(C(c2cnc(C(N)=O)cn2)=O)CC1 C1(COC)CN(C(c2ccc(F)c(Cl)c2)=O)CCN1C(C1CC(F)C(=O)N1)=O C1(C(N2CCCC2)=O)C(O)C(=O)N(C)C1C.c1(CC(C)C)c(C(=O)N)cnn1C C1CC1(C)C.CC(C)(C)OC(=O)NC1(CC(=O)N)CC1.C(=O)C.C C=C(F)CN=c1[nH]c(=NC)nc(N2CCN(c3ccc(F)cn3)CC2)[nH]1 c1(C(N2CC3CN(C(Cn4ccc(C)n4)=O)CC32)=O)ccc2[nH]nc(Br)c2c1 c1(C(=O)NCCC(C)Nc2nccc(C)n2)ncc2ccccc2c1O CCC(C)C(C(=O)NCC#CCNC(=O)C=C(Cl)Cl)NS(C)(=O)=O c1(N2CC3C(C(=O)Nc4cc(C#N)cc(Br)c4)C3C2)ncnc2c1CC(=O)N2 CN1C(=O)CCC1(C)CNC(=O)CC1(N(C(=O)C(C)(C)CC#N)C)CC1 N1(C(C2(C)COC(=O)C2)=O)CCCC(NC(c2ccc(Cl)o2)=O)CC1 Cc1ccc(C(=O)CNS(=O)(=O)C2CC2c2cccc(F)c2)cc1.C(C)(C)C C1(C(=O)NCC(CC)C(C)C)CCCCCC1NC(=O)Cc1ccoc1C C1(C(C)NC(C(C)NC(N)=O)=O)CN(C(c2cscc2Cl)=O)CCO1 c1(C(=O)NCC2(C)N(C(C=C(CCC)C)=O)CCC2)n[nH]c2c(=O)n(C)cnc12 C(=O)(C#CC1(C)COC1)N1C(C)CC1C(=O)NCCC1NC(=O)NC1=O N1(C(c2c(C)noc2N)=O)CCC(F)(CNC(=O)CN2CCOCC2)CC1 c1(CC(C(N)=O)NC(C)C(=O)NCCC#N)ccc(O)cc1 C(=O)(C(O)CCC(C)C)NCCCCC(C)NC(Cc1cccc(OC)c1F)=O CCCC(C)CC(=O)NC1CCCCC1CC(N1CC(C)(OC(C)=O)C1)=O C(=O)(C(C)C(F)F)N1CC(O)(C(C(=O)C(Cc2onc(C)n2)=O)F)C1.C1CCC1 CC(C)(C)C(O)C(=O)NC1(CNC(C2CCC(CCO)CC2)=O)CCCCCC1 C(CCCCC(=O)N1CCC(N(C)C(c2cnc(C)cn2)=O)C(C)C1)SC c1(C(N2CC(NC(c3ncn(C)c3)=O)C(O)C2)=O)c(Cl)cc(Cl)c2ncccc12 N1(C(CC(c2ccccc2F)C)=O)C2CCC1C(NC(=O)Cc1ccccc1)C2 CC(CC(C)(C)CO)NC(C1CN(C(C2CCOC(C)(C)C2)=O)CC1C)=O c1(CC(N2C(COC)(C)CCC2)=O)cc(C)cc(F)c1.C(=O)C.CC.N c1(OC)cnnc(-c2nc(-c3cccc(F)c3)nn2Cc2ccncc2)c1 n1(CCO)cnc(C(=O)CN2CCCCC2)c1.O=[SH](=O)CC1CCC1 C(C(CC(C)C)C(=O)N1CC(C(=O)Nc2cc(C)c(O)cc2C)C(F)(F)C1)OC N1(CC(=O)NC)CCCC(C2CCCN(C(c3cnoc3C(C)C)=O)C2)C1 C1(C(=O)NC(COC)CO)(CNC(c2cn(C(C)C)cn2)=O)CCCCO1 c1(CNC(c2c(C)scn2)=O)cccc2c1CN(C(=O)C(C)S(N)(=O)=O)C2 N1(C(CCN(CC)CC)=O)CCC(NC(c2cccc(C3CC3)n2)=O)C(O)C1 Cc1cc(C(=O)NCC2CN(C)CCN2C(C2CC(C#N)C2)=O)cc(Br)c1 CS(=O)(=O)CCC(=O)NC1CCCC1CNC(=O)C(c1ccc(Cl)cc1F)O C1(NC(c2c(C)nc(Br)o2)=O)CCCCCN(C(c2cscn2)=O)C1 N1(C(c2cn(CC)nn2)=O)CC2CCN(C(c3oc(CC4CC4)nc3C)=O)CC12 C1(NC(C2=CC(C)(CC)C2)=O)C(C)CCN(C(c2nc(C)nn2C)=O)C1C Cc1nccc(CCC(=O)N(C2CN(C(=O)C=CBr)CC2F)C)n1 C1(C(N(CC(CN(C(c2c(N)sc(C)c2C)=O)C)O)C)=O)CCc2nn[nH]c2C1 N1(C(C)=O)CCOC(C(N2CCC(C(c3ccc(C)cn3)=O)CC2)=O)C1 C=CCC(CC)C(=O)NC(CNC(c1ccc(-c2ccccc2)nc1)=O)CO c1(C(C)=O)ccc(S(=O)(=O)NCCC2SCCS2)c(OCC(N)=O)c1 C(C(C(=O)N1CC(CC(N)=O)C1)NC(c1cnn(C(C)C)n1)=O)OC(C)C C12(C(CNC(C3C(=C)CC3)=O)NC(c3cc(Br)n[nH]3)=O)CCC(CC1)C2 S(=O)(=O)(c1cccnc1Cl)N1CC(F)CC(C(=O)Nc2cccc3nccn23)C1 C(=O)(C1CCc2snnc21)N1CCC(NC(C(C)(C)N2CCCC2)=O)C1 CC(C)C(C#N)C(=O)NC1CC2CC(NC(c3ccc(C(F)F)cc3)=O)C1C2 C1(C(=O)N)CCCC2(CC2)C1.N1(C(C2(c3ccn(C)n3)CC2)=O)CCCC1(C)C N1(CCC)CCN(C(C2C3CC4C(C3)C24)=O)CC1.c1ccn(C)n1.C(=O)(C)N C=CCCCCCC(=O)NC1(C)CCC(NC(=O)COCCCOC)CC1 N1(C(CC(C)C(F)(F)F)=O)CC2CCC(C1)C(NC(=O)C(C)(C)n1cccn1)C2 c1(-c2nc(-c3ccc(OC)cc3)nn2C2CCCC(C)C2)cccc(OC)c1C Cc1cc(Br)cc(F)c1NC(=O)C(N1CCC(O)(c2cnnn2C)CC1)=O C1(C(N2CCOCC2CC2CCCC2)C(=O)NC2CCOCC2)CC2CCC1O2 C1(CC)CCCCN1CCCNCc1c(C)n[nH]c1C C1(C(N2C(C=C)CCC2)=O)CCN(C(c2cnc(C)o2)=O)CCO1 c1(C(=O)OC)ccccc1S(C)(=O)=NC(=O)C1CCN(C(=O)O)CC1.C(C)(C)C c1(CC(N2C(CCNC(=O)Cc3cnccn3)CSCC2)=O)cc(O)nnc1O C(CC(C)C)(C(=O)O)N(C(c1c(C)noc1C)C(=O)NC)CC=C.C(C)(C)C C1(C(N(CCCCNC(c2nc(Cl)cs2)=O)C)=O)CC2CCC1C2 c1(C(CN(C(C2C(Cl)(C(=O)OCC)C2)=O)C)O)ccccc1Br Cn1nccc1C1=CC2CCC(C1)N2C(=O)NCCc1cnc(C2CC2)nc1 C(C)(C)(CC(=O)NC1(CCCC(=O)NCC(O)C2CC2)CCC1)OC C1(O)(c2ccccc2)CCC1.CC(C(=O)N(CCCN(C(=O)CO)C)C)OC n1(CC)cc(C(N2CCCC(C)C2)=O)c(C)n1.c1(C(=O)N)ocnc1C1CC1 C1(C(=O)NC2CCCCC2)(OC)CS(=O)(=O)C1.c1(CC=O)cncn1C.C N1(C(C(C(C)C)NC(C)=O)=O)CC(NC(c2cnsn2)=O)CC(C)(C)C1 C(C)(C)(CC(=O)N1CCCC(CN(C)C)C1)SC C1(CNC(C2(CC=C)CCOC2)=O)CCC(F)C1.c1(C=O)cc(C)[nH]n1.C c1(C(=O)NCC2CN(C(C(CC)COC)=O)C(C)C2)cc(OC)cc(F)c1 N1(C(C(C2CC2)OCC)=O)CC2CCC2(NC(=O)CCC2CC(C)C2)C1 C1(C(=O)NCC(n2cc(C(CCC)=O)nn2)C)CCCC(=O)N1C n1(CCC(=O)OCC)nnnc1C(c1nccs1)NCCCn1cc(C)cn1 c1(C(N2CCC(NC(C(CC)O)=O)C2)=O)cc(Cl)c2ncccc2c1F c1(C(=O)NCC(CCNC(C(CC)n2cncn2)=O)O)c(F)ccc2ccoc12 N1(C(C(C(=O)OC)C)=O)CCN(C(=O)CCc2ccc(F)cc2Cl)CC(CO)C1 c1(C(C)C(=O)NCCCN(C(=O)C(C)SC(C)C)C2CC2)cnn(C)c1 Cc1nn(CCC(N2CC(F)(F)CC2C)=O)c(C)c1C.C1(C(=O)N)CCC(=O)N1 N1(C(C)=O)CC2CC(C1)N(C(c1cc(C3CCC3)[nH]n1)=O)C2.C(=O)(CO)OC C1(CNC(CCNC(C)=O)=O)CN(C(c2c(C)cncc2F)=O)CCC1C C(=O)(C(C)C(=O)NC(C)C1CCC1)OC.c1(C=O)cc(-c2ccns2)on1.N CC1(C)CCCOC1C(N1CC(C(=O)NCC2OCC3CCC2C3)CC1(C)C)=O C1CC2CC1CN(C(=O)CCC1(C)CCCN1C(C1CC(=C3CC3)C1)=O)C2.C O=C1CCC(Oc2cccc(C(=O)Oc3ccccc3Cl)c2)C(=O)N1 C1(O)(CNC(CC2C(C)(C)OCC2)=O)CCN(C(=O)CC2CSCCO2)CC1 C(C(=O)N=c1nc(C2CCN(C(=O)OC(C)(C)C)CC2)[nH]n1C)N(C)C(N)=O CCC(C)C(O)C(=O)NC1CCCN(C(c2cc(C(F)(F)F)cnc2O)=O)CC1 c1(CC)cccc(CC)c1NC(=O)CC1(CC(=O)OC)CCCC1 C1(C(N2CCC(F)(CNC(C(C)(C)c3ccsc3)=O)C2)=O)CCC(C2CC2)C1 c1(C(=O)NC2C3CN(C(C(CC)(C)O)=O)CC2C3)cc2cc(OC)ccc2cn1 C1(OC)(CNC(C2(C(C)C)CCC2)=O)CN(C(c2ccc(CO)o2)=O)C1 c1(OC)ccc2c(C(=O)N)csc2c1.C1CC2CCC(C1)N2C(=O)C=C(C)C C(CCCCCNC(C1CC1(F)F)=O)N(C)C(c1cc(CCO)on1)=O N1(C(Cc2c(Cl)ccc(OC)c2)=O)CC(CNC(=O)CC(C)O)OC(C)(C)C1 N1(C(c2cn(C)c(=O)cc2)=O)CCC2(CCN(C(=O)CC3CCCSC3)C2)C1 C(=O)(C(C)(C1CC1)N(C)C(c1ccco1)=O)N.CCCCOCC1CC1 N1(C(C2CC(NC(C3C(C(C)C)CCO3)=O)C2)=O)CCC(O)CC12CC2 N1(C(CC(C)C(F)F)=O)CCCC2C1CCN2C(c1cnc(Br)s1)=O C1(C(=O)NCC(C)N(C(c2ccc(OC)cn2)=O)C)NC(=O)OC1(C)C C=CCC(C(=O)N1CC(OCC)C(CNC(c2ncn(C)c2C)=O)C1)C(C)C c1(SCC(=O)NC2CCN(C(C(CCC#C)O)=O)C(C)C2)ccc2c(c1)CCC2 c1(C(=O)NCC(CC(F)(F)F)NC(COCCC#C)=O)cccc2c1OCC2 c1(C=O)nc(O)c2ccccc2c1C.c1(OCC)cc(C(=O)NC(C)C)[nH]n1.N N1(c2nc(C)c(Br)cn2)CC(NC(=O)CC2CCC3CC23)C2(CCOCC2)C1 Cc1[nH]nc2cc(C(=O)NC(C)C(C)(C)C)ccc12.C(c1cc[nH]n1)=CC=O.N C(C(C)CC(=O)NC(C1CCCCC1)CNC(=O)CCc1ccccc1Cl)OC CC#CCCCCNC(=O)C(C)(CO)NC(c1c[nH]nc1Cl)=O C1(C(=O)NC2C(NC(c3ccsc3)=O)C2)C2CCC1(c1cccs1)C2 c1(CC(N2C(CNC(N)=O)CCC2)=O)ccc(Br)cc1 C(C)(C)(C=CC(=O)N(CCNC(=O)C(C)SC)C(C)C)SC C(=O)(NNc1cc(F)c(F)c(F)c1)NCc1ccc(OC)c(C2CC2)c1 O=C1OC2CCN(C(=O)NCCc3noc4ccccc34)CC2O1 Cn1cnnc1CNC(C1COC(CN)C1)=O.c1(CC=O)ccoc1 N1(C(C2(C)CC(=C)C2)=O)CCC(CO)(NC(=O)CCC(=O)c2ccc(C)cc2)C1 N(S(=O)(=O)N(C)C)CC(=O)NC1(C)CN(C(CC2(C=C)CC2)=O)C1 C(=O)(C1=CCCCC1P(C)(C)=O)N1CC(CC=C)(NC(c2cn[nH]c2)=O)C1 C1(C(=O)NC(c2ccn(C)n2)CC)CN(C(C2CC(=O)C2)=O)CC(C)(C)C1 C#Cc1ccc(C(=O)NCC(=O)NCCC2CCSC2)cc1 N1(C(Cc2c(C)ccc(F)c2)=O)CCCC1C1CCCN1C(c1cnsc1C)=O C1(NC(=O)Cn2cnnc2)CCC2CN(C(c3cnc4n3CCC4)=O)CC2C1 N1(C(CC(CC)(F)F)=O)CCC2CC2(C(N2CC(n3cnnc3)C2)=O)CC1 N1(C(N(c2nnc(C)o2)C)=O)CCCCC1c1ccccc1 c1(C(N(C2CCCN(C(C3CC4CC3C4)=O)CC2)C)=O)cc(O)cc(Cl)c1 N1(C(=O)CCN2CCC2)CC2(C1)CN(C(=O)CCc1nncs1)C2 N1(C(C2(SC)CN(C(c3ccccc3O)=O)C2)=O)CC2CCCC(O)C2C1 C1(SCC)CCCCC1N(C(=O)C(=O)NC12COCC(C1)C2)C C1(C(N(C)C)=O)CCCN(C(C2(n3cc(C(C)(O)C(=O)O)nn3)CC2)=O)C1 N1(CC(=O)NCC(C(=O)N(C(C(C)SC)C)C)C)C(=O)CCCC1=O CP(C)(=O)CCC(=O)N1CCCC1c1nc(C(=O)NC)cs1.C1CC(F)(F)CO1 N1(C(C2C(C)CCO2)=O)CCN(C)C(C(=O)NCCC(F)(F)F)C1 C(=O)(C1=CC2CCCC12)N1CC(C(C)NC(c2ccc(C(=O)NC)nc2)=O)C1 C1(C(N2CCC2)=O)CC2(C1)CC(O)C2.C1(C(N(C)C)=O)(C(N)=O)CCC1 C(=O)(C(CC(C)C)N(C(=O)CCC(C)OCCCCC)C)N1CC(OC)C1 C(C)(CN=c1ccc(C#N)c(C(F)(F)F)[nH]1)N(C(c1c(SC)cccn1)=O)C N1(C(c2c(CC)csc2)=O)CC(CNC(=O)C(O)C2CCCC2)CC1C N1(C(C)=O)CCN(C(C2OCCN(C)C2=O)=O)C(C2CCC2)C1.C(=O)(CO)OC C(=O)(CC(C)(C)C)NCC(n1cc(CCCSc2ccccn2)nn1)C C(=O)(CCN(C1CC1)CCC=CC=C)NC(COCC#C)=O c1(CCC)nnc(-c2ccn(C3CCSCC3)n2)o1 c1(CC)n[nH]c(=NC2CN(C(c3ccc4cc(C)cn4c3)=O)CC(C)(C)C2)s1 C(=O)C1CCc2nccn21.C1(CC=C)(CNC(C2CC2C)=O)CC=CC1.N CCCCCC(C(=O)NCC(C(C)(C)C)NC(=O)CC(O)C1CC1)C(C)C N1(C(c2cc(C)[nH]n2)=O)CCCCC(CNC(c2ocnc2C(F)(F)F)=O)CC1 C(=O)(C(CCC(C)(C)C)N1CCCC(CC#N)C1)NCC=C C1(O)(CCNC(CC(=C)C)=O)CCCN(C(c2cncc(N)c2)=O)C1 CCC(CN(C(=O)Cn1ccnc1)C)NC(C1CCSC1)=O C12(NC(=O)COCC3CCC3)CC1CN(C(=O)CN1C(=O)CNC1=O)C2 C1(CC)CN(C(=O)CCN(CC)CC)CCN1C(=O)CCCC1CCCC(=O)N1 c1(COC(COCCOCC)=O)ccccc1OC(F)(F)F.C(C)C=O c1(C=O)cc(C)c(C(F)F)cn1.N1(C(C(=O)NCC)=O)CC(CO)CC1 C(=O)(C(C)(F)C(=O)NCCCCC)OCC.c1(C(C=O)(F)F)ccc(F)cn1 C1(OC)CCC(C(=O)NC2CCCC2NC(=O)CC(O)Cc2ccccc2)CC1 C1(CNC(C2CCCN(C(N3CCCC3)=O)C2)=O)C2CNCC12.C1CCCC1.C c1(C(=O)NCC2C(CNC(C3(C)CCCS3)=O)C2)ccccc1.C1CC1 C12(CNC(C(C)c3cccs3)=O)CCC(NC(=O)C3=CC(C)CC3)(CC1)CO2 C1(CNC(Cc2c(SCC)cccc2)=O)CCN(c2cc(C)ncn2)C1(C)C N1(CC)CCC(N(C(=O)C(C)(C2CCC2)NC(c2cncn2C)=O)C)C1 C1(OC)CN(C(=O)CC2CCC(F)(F)C2)CCC1.n1(CC(=O)N)ncccc1=O c1(CC)cc(C(N2CC3CCC2(CNC(c2csc(C)n2)=O)C3)=O)cc(Cl)n1 Cc1cc(F)ncc1-c1csc(C(=O)Nc2ccc(F)cc2)c1 CC1(C)CCC(CC(=O)NC2CCCC2NC(=O)CCC#N)c2ccccc21 c1(C(=O)NC2CC(NC(C3(C)CC3)=O)C23CCC3)ccnc2[nH]c(O)nc12 CCC(c1ccccc1)=CC(=O)NCC(C)CNC(C1CC(C)(O)C1)=O c1(C(N2CCCC(O)(CNC(C(CC)(C)F)=O)C2)=O)cc2nc(C)ccc2o1 N1(C(c2c(CC)nns2)=O)CCC(C(C)C)CC1.C1(C(C=O)C)CCC(=O)N1.N C1(C)(C(=O)OC)CCC(NS(=O)(=O)OC(C)C)CC1 C12(C(N(C3CCCCC3)C(C)C)=O)COCC1CN(C(=O)CC1C=CCC1)C2 c1(C(=O)NCCC2CCN(C(C3(SC)CCC3)=O)C2)ccc2cc(O)ccc2n1 C1(C(=O)NCCCNC(=O)C(C)(C)C2CCOC2)(OC)CCCC(C)(C)CC1 C1(NC(C(n2cc(C)nc2)(C)C)=O)COC2CN(C(=O)CCc3ccsc3)CC12 N1(C(CC(C(=C)C)OCC)=O)C2CCC1C(F)C(NC(=O)CC(C)(C)SC)C2 C(=O)(C(C(C)(C)O)NC(C1CC=CCC1C)=O)NCc1nccc(OC)n1 O=C(C1Cc2c(Cl)cccc21)NC1COc2cccc(Cl)c21 C1(C#N)(COC)CN(C(=O)CCOC2CN(C(=O)CC3CCCCO3)C2)C1 CC1(C)CC(CNC(=O)CCSC2CCCC2)CN1C(=O)CCc1ccsc1 C1(NC(CC(C)OC)=O)CS(=O)(=O)C12CCN(C(C1(C)CCSCC1)=O)CC2 C1(C(C)C)N(C(=O)CN=S(C)(C)=O)CC12CCN(C(C1CC(=O)N(C)C1)=O)CC2 N1(C(Cc2c(C)con2)=O)CCCCC1CCNC(=O)C(C)c1cncs1 c1(OC)ccc(C(C)C(=O)NCCC2CCCN2C(c2sccc2C)=O)c(C)c1 Cc1ccccc1SCC(=O)N(CCCCNC(c1cnn(C(C)C)c1C)=O)C c1(OC)cccc(C2CC(=O)N(CN(C)CC(c3cccc(C)c3)O)C2)c1 C(=O)(C(O)CC(F)(F)F)N1CCCC(CCNC(Cn2nnc(C)n2)=O)C1 n1(CCC)cc(-c2c[nH]nc2C(=O)O)nn1.C(C(=O)NC(C)(C)C)SCC C1(C(N2CCN(C(c3cc(Cl)c[nH]3)=O)CC2CCO)=O)Cc2ccncc2C1 C12(C(N3C(C(C)NC(=O)CSC4CC4)CCC3)=O)CCOC(C)(C1)C2 C=CC(CCC)CC(=O)NC(C1CC1C(N1CC2COC(=O)C2C1)=O)C c1(C(=O)OC)ccc(CC(=O)NCC2CC2)cc1.c1(CC=O)ccno1.N c1(C2CC(C(=O)NCC(CC)NC(c3ccnn3C(C)C)=O)O2)ccccc1 N1(C(C(C(C)O)(C)C)=O)CCC2(CC(NC(C3CCCC3O)=O)CO2)C1 C12(COC)CC(C(=O)NC3CCN(C(c4cnc(Cl)s4)=O)C3)(CO1)C2.C C1(NC(c2occ(C(=O)OC)c2)=O)CCCC(N(C)C(c2cnn[nH]2)=O)C1 C(=O)(C1CCCc2nccn21)N1CCC(NC(C(C)(C)NC(=O)OC)=O)C1C C12(NC(C=C(C)C)=O)CCCCCC1N(C(c1nn(C)c3ccccc13)=O)CC2 c1(OC)ccnc(C(=O)NCC2(NC(c3sc(C)cc3Br)=O)CCC2)c1 C(c1ccc2c(c1)CCO2)=CC(=O)NCC1CC1.C(=O)CCCC(F)(F)F.C Cc1c(F)ccc(N)c1C(=O)NCC1CCN1C(C1(C)CC(C)(C)C1)=O C=Cc1cc(C(N2CCC(C)(CCNC(C3CCC(=O)N3)=O)CC2)=O)cc(F)c1 C(=O)(C1=CCOCC1)NC(CNC(C(C)OC1CCOC1)=O)C(C)(C)C C(c1ccc(C(F)(F)F)cc1)=CC=O.C1C=CCN(C(C2(F)CC=CC2)=O)C1.N c1(C(N2CCCC(C(C)NC(c3ncoc3C3CC3)=O)C2)=O)ccnc(F)c1Cl C1(NC(=O)NC(c2ccccc2-c2ccccc2)CC)CCC(=O)NC1(C)C CC1(C)CC(CNC(c2cccn2C2CC2)=O)CN(C(=O)Cn2cnnc2)C1 C(=O)(C(F)CC(C)(C)C)N1CCCC(N(C)C(C2CCCC2)=O)CC1 CCC(CC(=O)NC1CC1CNC(C1(C(F)F)CC1)=O)C(C)(C)C N1(C(C(CC#C)(C)NC(c2ccc(O)c(C)c2)=O)=O)CCc2ncccc2C1 CCCC(CC)CC(=O)N1CC2(C1)SCCC2NC(=O)C(N1CCC(O)CC1)C N1(C(c2n(C)cc([N+](=O)[O-])c2)=O)CCCc2c(Cl)cccc21 N1(C(CC(=O)NC)=O)CCC(C)C(CNC(=O)C(=Cc2cnn(C)c2)C)C1 C(=O)(C#CC1(CC)COC1)N1CCC(CCNC(C(COC)OC)=O)CC1 C(CCCCC(=O)NC(CNC(c1ccoc1C)=O)CC(F)(F)F)OCC C(CCC(=O)NCCN(C1CCC1)Cc1ccccc1)C1C(C)C1 C(CNC(=O)CSc1cnn(C)c1)(CC(F)(F)F)NC(C=CCC)=O C1(CNC(CN2C3C(C(C)(C)C)C(C3)C2)=O)CC2CC(=O)C1O2 C(=O)(C(C)(C(C)C)OC)NCC(CC=C)NC(=O)Cc1cccc(F)c1 c1(SC)nc(NC2CC(CNC(C34CCC(CC3)C4)=O)C2)ncc1C N1(C(C2CC(=C)C2)=O)CC2CC(C(=O)NCc3cnc(CC)[nH]3)C(C2)C1 C1(CC(=O)O)(NC(C2CC2c2ccccc2Cl)=O)CCCCC1 C1(C=O)CCC2(CC2)C1.CC(C)COCCCNC(=O)C.c1nccs1.N C(C(O)C(=O)N1CC(N2CC(F)C2)C1)NC(=O)CSCC(F)F C(=O)(C1CCCc2n[nH]cc21)N1CCOCC(F)(CNC(CN(C)C)=O)C1 Cc1nncn1NC(=O)CC1CCCCC1NC(c1cn2ccccc2n1)=O C(=O)(C1Cc2c(Cl)cccc21)NC1CN(C(C(CC=C)(C)C)=O)CC(C)(C)C1 N1(C(c2ccnc(OC)n2)=O)CCC2CC1CN(C(c1cc([N+](=O)[O-])c[nH]1)=O)C2 N1(C(C(CC(C)C)N(C)C)=O)C2CCC1CN(C(c1cc(Cl)cc(F)c1F)=O)C2 C(C(CC(C)C)C(=O)NCC(C(=O)NCCC(=O)N(C)C)C(C)C)OC N1(CC(=O)N(C2CN(C)CCC2O)c2c(C)cccc2)CC(O)CCC1C C1(NC(C=C(C)C(C)C)=O)CC1C1CCN(C(c2ccc(Cl)o2)=O)CC1 N1(C(c2ncccn2)=O)CCC2C1CCCN2C(c1cc(Cl)cc2c1CCC2)=O C(=O)(CCC(=O)NC1CC(CCNC(=O)C=CC=O)C1)NC.C1CC1 Cc1ccccc1CN(C)C(C1CCN1C(=O)CC1CC2CCC1C2)=O c1(C(N(CCC(C)(C)NC(C(C)N2CCC2)=O)C)=O)cc[nH]c2nccc1-2 C(C)(N=c1ccc2c(Br)coc2[nH]1)c1nc(COC)on1 C(C1=CCCC1)NC(c1nnnn1CCCSC)(CC)C1CC1 c1(C(=O)NC2(CCNC(C=C(COC)C)=O)CCC2)cn2ccccc2n1 C1(NC(C(CC#C)C)=O)CCC(C)(CNC(C2CC3CCC2C3)=O)CC1 CCC(C(=O)NC1CCC1NC(=O)Cc1nccn1C)Oc1ccccc1 c1(C(N2CC(F)(CNC(C=C3CCN(C)CC3)=O)C2)=O)cc(Cl)cc(Cl)c1 C(=O)(C1=NN2CCCN=C2N1)N1CCC(C)C(N(C(=O)CC2CNC(=O)C2)C)C1 C=CC1(C(N2CCCC[Si](C)(C)C2)=O)CCN(C(=O)C(O)CSC)C1 O(NC(=O)C(C1CCOC1)NC(c1ncsc1C)=O)CC N1(C(C=Cc2ccc(C)s2)=O)CC2CN(C(C3(C)CCCC(F)(F)C3)=O)CC2C1 CC1c2ccccc2CC1C(=O)NCC1CN(C(c2cnn(CCF)c2)=O)C1 O=C1CN(C(N2CCC(F)C2)=O)C2(CC2)CN1 c1(CNCc2cccc(OCC(=O)OCC)c2)cc(I)ccc1Cl N1(C(CC2CCN(C(c3nc(=N)[nH]cc3)=O)CC2)=O)CC2C(C1)C2(F)F C(=O)(N=c1[nH][nH]cc1I)C1N(C(c2cc(C)cc(Br)c2)=O)CC(C)C1 c1(CC(=O)NCCNC(C(C)c2ccsc2)=O)cc(Br)nn1C CCC(C)CC(C)N(C)C(C1(OC)CCN(C(c2ccncn2)=O)C1)=O C1CC2CCC(C1)N2C(C1CN2CCN1C(C)C2)=O.CC(C(=O)NC)=C1CC1 C1(O)(CNC(CC(C)C)=O)CCCN(C(c2c([N+](=O)[O-])cnn2C)=O)CC1 c1(C(N2C3C(NC(C4CCCO4)=O)CC(C3)C2)=O)cc(F)cc(F)c1Br C(=O)(C(C)CC(N)=O)NC(CCNC(C(C)(C)OC(C)=O)=O)C N1(C(CN2CCN(CC)C(=O)C2=O)=O)CCCC2CN(C(=O)C)CCCC12.C(C)C.O N1(C(c2nc(CC)sc2)=O)CC(NC(c2snnc2C2CC2)=O)CC1(C)C c1(C(N(C2CCC(NC(C=C(C)C3CC3)=O)CC2)C)=O)ncnc2c1cnn2C C1(CNC(CC2(C)CCCO2)=O)CCCCN1C(=O)C(F)Cc1ccccc1 N1(C(C(C(C)=O)(C)C)=O)CCCC2(CCN2C(c2scc(C)c2C)=O)C1 CC(C)(C)CC(O)C(=O)NCC(CNC(=O)Cc1cn2ccccc2n1)CO N1(C(C23CCC(C=O)(C2)CO3)=O)C2CC3CCC2(CS1(=O)=O)C3(C)C.CC.O c1(C(N(CC(CC)NC(c2cc(C#N)on2)=O)CC)=O)cc(C)cc(Cl)c1Cl c1(CNCC(C(C)(C)C)O)ccc(N)c(F)n1 Cc1nc(C2CC2)oc1C(=O)N.C(=O)C[SH](=O)=O.C(C)(C)C.C(C)(C)C CCS(=O)(=O)CC(=O)N(CCC(C(C)C)NC(c1cc2sccc2[nH]1)=O)C C(=O)(C1CCCn2ncnc21)NC1CCC(NC(COCC(=O)OC)=O)C1 c1(C(=O)OC)cccc2c(SCC3CCC3c3nc[nH]n3)cccc12 C(=O)(CCCC(=O)NCCCCC(C)NC(C1(C(F)F)CCCO1)=O)OC C(=O)(C1=NOC(C)(C)C1)NC1C(C)N(C(c2cnn(C3CC3(F)F)c2)=O)CC1 C1(C(=O)NCC(N2CCOCC2)c2cccs2)CC(O)C12CCC2 Cc1cc(Cl)c(C(=O)NC2CCC(C)(CNC(c3nccn3C)=O)C2)cc1F C1(C(=O)Nc2cc(CC)ncc2)CN(Cc2cc(Cl)c(C)cc2O)CC(F)(F)C1 c1(C(=O)NCC(CCCC)NC(C2(CF)CC2)=O)c(C)cc(C)cc1N c1(C(N2CCC(N(C(C(C(C)C)SC)=O)C)C2)=O)ccc(C)c(N)c1 N1(CC(=O)NCCCC(C)=O)CCCC(N(C)C(=O)C2CC2)C1 C1(C(C)(C)C)CCN(C(c2cccc(F)c2)C(=O)Nc2ccccc2)CC1O CCC(O)CC(=O)NC1CN(C(=O)CC2CCC(C(F)(F)F)O2)CC1C c1(C(N2C(c3nc(C)sc3)CCC2)=O)csc2c(C)cccc12 C#CC(C(C)(C)C)NC(C1C=CCCN1C(=O)CN1CC(=O)NC1=O)=O C(=O)(C(C)(C)C(N)=O)N1CCCC(CN(C)C(C2CCOC(=O)CC2)=O)C1 C1(C(=O)NCCCCCN(C(c2ccn(CCC)n2)=O)C)CCCCCN1C N1(CCC)CC(NC(=O)CC2CC(NC(=O)Cc3cnsc3)C2)CC1=O C1(NC(C(CC)(C)CNC(C2CCCN2C(C)C)=O)=O)CCn2ccnc2C1 C(CCC(=O)NCC1CC1CO)NC(C(C)C1CCC1)=O Cc1nn(C)c(C)c1CCCNCC1OCCC1F C1(C)(CC(=O)NC(c2nccn2C)CC)CCN(C(=O)Cn2nccn2)C1 C1(NC(c2cccc(CO)c2)=O)CCN(C(=O)CCC(=O)c2cccs2)CC1O C1(NC(CCOCCC)=O)CC2(CCN(C(c3cnnn3C)=O)CC2)C1 Cc1cc(C(F)(F)F)ncc1C(=O)NCCCCCC.C1(=CC(=O)N)CCCC1 Cc1c(C(=O)NC2CCN(C(=O)CCN3CCN(C)CC3)CC2O)cccc1F c1(C(N(C)CC2CN(C(C(C)c3ccsc3)=O)C2)=O)conc1C1CCC1 C(=O)(CN=S(C)(C)=O)N1C(CNC(C(C=C)O)=O)CC2CC21 C1(C(=O)NC2CC(NC(C3(O)CCSC3)=O)C2)CCOC2(CCOCC2)C1 n1(CCC)nc(C)c(C(=O)NC2CCN(C(C3CC(F)(CO)C3)=O)CC2F)c1C O=S1(=O)CCN(Cc2ccc(-n3cncn3)c(F)c2)C2CCCCN12 c1(CC)cccc(CN(C(C2CC(=O)NC2=O)=O)C2CC2)c1.N12CC1C2 CCCCC(CC)C(=O)NCC(C)N(C(=O)Cc1nc(C2CC2)nn1C)CC c1(OC)cc(C(=O)NC2CCCC(NC(=O)C(O)CC(C)C)C2)cc(Cl)c1 c1(C(=O)Nc2c(OC)ccc(Br)n2)cccc2c1CN(S(=O)(=O)C(F)(F)F)C2 c1(OC)c(C)ccc(C(=O)NC(C)CC)c1F.c1(C(=O)N)cncn1C(C)C N1(C(C(C)=C(C)C)=O)CCC2C(NC(=O)C(c3ccc(Br)s3)C)C12 C=C(CNC(=O)CC(C1CC1)C1CC1)CCNC(=O)C1CC1 c1(C(NC(C)C)=O)cnc2c(c1)COCC2.C1(S(C)(=O)=O)(C=O)CC1.C c1(CC)cc(C(N2CCCCC2CN(C(=O)CCC(F)F)C)=O)c2c(c1)CCO2 C1(CNC(C(C)S)=O)CCCCN1C(=O)C(C)n1ccnn1 n1(CC)ncc(C(=O)N(CCNC(C2CC2c2cccs2)=O)CC)n1.O C(=O)(C1CCCc2nn[nH]c21)NC(C(C)(C)C)CNC(=O)CC1CCNC1=O Cc1cc(C(=O)N(C2CCCC2)CCCNC(c2nccn2C(C)C)=O)ccn1 C1(NC(C(CCC)OC)=O)C2CC(O)C1N(C(c1ccc(OC3CC3)cc1)=O)C2 C(=O)(C(C)(C)CC(C)(C)C)N1CC(C)N(C(C2CCC3(CC2)OCCO3)=O)CC1 N1(C(c2n[nH]cc2Cl)=O)CC2CC1CN2C(C1CC1C(F)(F)F)=O S(=O)(=O)(c1ccc(N2CC3CCC(CO)(C3)C2)nc1)NC(c1ccsc1)C c1(C(C(C)NC(CC=CCC)=O)NC(=O)CCOC2COC2)ccccc1 N1(C(C(CC)(C)CNC(C2(C)CCCC2O)=O)=O)CC2C=CCC(C2)C1 N1(C(C2CCC(C)(C)C2)=O)CCCC2(C1)CN(C(c1ccc(C#N)cc1O)=O)C2 c1(C(N2C(CC)C(C(=O)Nc3cnn(CC)c3C)CC2)=O)ccc(F)cc1F CC1=NOC(C(=O)NCCOCCC(=O)N(CC(C)O)C)C1.C(N)=O N1(C(C2C(OC)C2)=O)C2CCC1CC(O)(CNC(c1ccc(C)nc1)=O)C2 N1(C(CCC(=O)NCC)=O)CCC(NC(=O)CCc2cnn(C)c2C)C(OC)C1 c1(C(N(CCNC(C(C(C=C)C)C)=O)C)=O)c[nH]c2cc(O)ccc12 N1(C(C2(C)CC(NC(c3c(CC)ncs3)=O)C2)=O)CCSC(C)(C)C1 c1(N2CCC(C(C)NC(C3(C)CCC(C)C3(C)C)=O)C2)ccc2nccnc2n1 C1(C(C)NC(CCC)=O)CN(C(=O)C(C2CCCCC2)O)CCO1 CC(C(=O)NCc1nc(C(C)(C)C)cs1)C(C)c1ccc(Cl)cc1 Cc1ccc(-c2ccc3nc(C(=O)N=c4cco[nH]4)cn3c2)c2ccccc12 c1(N(CC(CN(C(C(Cn2ccc(C)n2)C)=O)C)O)C)nc(Cl)c(C#N)s1 CC1CN(C(=O)C(C)(C)c2ccns2)CCN1C(c1ccc(C2CC2)c(F)c1)=O C1(NC(=O)CC2C=CCC2)(C)CCCCCC1.c1(C(=O)N)cc(C2CCC2)no1 C1(CNC(C=CCN(C(c2n[nH]c(C)c2Cl)=O)C)=O)Cc2nccn2C1 N1(C(CCC(CC)OC)=O)CCC(C)N(C(=O)Cc2c(C)cccc2C)CC1 c1(C(=O)NCCNC(C2(F)CCC2)=O)cc2c(cc1Cl)OCCO2 C12(OC)CCC1CN(C(=O)C(CC1CCC1)NC(=O)C=Cc1ccccc1C)C2 c1(C(N2CCC(NC(c3nc(C)c(C)s3)=O)C(C)C2)=O)ccc([N+](=O)[O-])cc1N C1(c2ccc(C(N)=O)o2)CCN(C(=O)NCC2CCCCS2)CC1 c1(C(=O)NCCCN(C)C(C2CC2Cl)=O)ccccc1C1CCC1 C1(OC)(OC)CC2(CCCN(C(c3cn(C)cn3)C(=O)NC3CCOCC3)C2)C1 c1(C(=O)NC(C2CCCN2C(c2ccnn2C)=O)C)ccc(F)cc1Br CC(C)(C)C(O)C(=O)NCc1ocnc1C(=O)NC1CCCC1F c1(OC)ncc(CNC(c2sc(C)nc2C)c2nnnn2CCCF)cc1Br C1(C(=O)NC2COCCN(C(C(C(C)C)(C)O)=O)C2)CCC2CC(C)CN2C1 C(=O)(C1=CC2(CCOC2)C1)NC1C(NC(=O)CCc2cocn2)CCCC1 CC(c1ccsc1)=CC(=O)NC(C)(C)C1CC1.c1(C=O)ccc(C2CC2)nc1 O=C(CN=c1cc[nH]cc1)NCC(CNC(=O)CS(=O)(=O)C(F)F)CO C1(C)(CC)CCC(NC(C2C=CCCN2C(=O)C(C)=C2CCC2)=O)CC1 c1(SCCC(N2CCC(N(C)C(c3nnn(C)n3)=O)C2)=O)ccc(F)cc1 N1(C(C(CC=CC)NC(=O)C(F)C(C)C)=O)CC2C3CCC(C3)C12 c1(C(=O)NC(c2c(C)nc(C)s2)C)nc2ccc(C(F)(F)F)cc2nc1C N1(C(=O)C=CCO)CCN(C(=O)C(O)CF)C2(CCC2)C1 C(=O)(C(CC1CCCCC1)C(C)C)N1CC(CNC(C=NOC)=O)C(O)C1 CCCCCC(C)CC(=O)NCCc1n[nH]cc1C(N1CC(=O)NC(=O)C1C)=O c1(CCC)sc(C(=O)NC(C)C(C)NC(=O)C=C2CCC2)cc1CC C1(NC(C(=C(C)C2CC2)F)=O)CCC12CCC2.c1(C(=O)N)c(C)nc(C)n1O C1(COC)CN(C(=O)CC2=CCCC2)CCN1C(=O)CCNS(C)(=O)=O C=CC1CN(C(c2ccc(C)c(Cl)c2)=O)CC1NC(=O)C=CCO N1(C(C2ON=C(C)C2C)=O)CCC2C(C1)CN2C(=O)CCCn1cncn1 N1(C(CCc2c(C)noc2C)=O)CCC(NC(c2ncc[nH]2)=O)C(CO)CC1 C1(NC(C2(CC#C)CCCCC2)=O)CC2CCC1N2C(c1ccnn1C=C)=O C#CCC(O)C(=O)NC1CC(c2ccccc2)(CNC(=O)CCc2nccs2)C1 c1(C(=O)NCC(CNC(C2C(C)C2)=O)O)cccc2sc(C(F)(F)F)nc12 C1(CNC(=O)COC2CCOC2)CC2CCCC2N1C(=O)Cc1ccccn1 N1(C(c2c(C(C)C)c[nH]c2)=O)CCCC(CC(N2CC(O)CC(O)C2)=O)CC1 N1(c2nnc(CC)o2)CCC(C)C(NC(c2coc(C)n2)=O)C1 c1(C(N2C(CN(C)C)COCC2)=O)cc(-c2ccco2)cn(C)c1=O C#Cc1ccccc1CCNC(=O)C(=O)NC1CC2NCCC12 N1(C(C=CCC(C)(C)NC(c2ccnnc2O)=O)=O)CC2CCC(O)CC2C1 Cc1cc(CC(=O)NC2CCCCC2CNC(=O)CC2CC(F)C2)c(C)s1 N1(C(CC2(C)CC2)=O)Cc2ccccc2C(NC(C2CC3CCC2CC3)=O)C1 C(CC(C)C)(C(=O)N1CCCC1(C)CO)ONC(c1cc(OC)nn1C)=O CCCCCCCCCC=CC(=O)NC1(C)CN(C(=O)CCCN(C)C(C)=O)C1 C1(CC=O)CC2CCC2C1.CC(C)C(C1CCC1)NC(=O)CCC1CCC1.N C(=O)C(C)S(C)(=O)=O.c1(C(C(=O)N)OC(C)=O)ccccc1.C1CCC1.C N1(C(c2c(CNC(C(CC(C)C)N(C)C)=O)noc2)=O)CC2(CNC(=O)N2)C1 c1(N(C)C)nc(Cl)c(C(=O)N)s1.C1CCN(C(C2CC(N3CCCC3)C2)=O)C1.C CCC(C)(CC)C(=O)N1CCN(C(c2cc[nH]c2C2CC2)=O)C(COC)C1 Cc1nn2ncccc2c1C(=O)NC1CC2(C1)CN(C(C1(C)CCC(C)C1)=O)C2 c1(CN2C(C(=O)NCCCOC=C)CC(O)C2)cc(Cl)cc(C#N)c1 C1(C(=O)NCC2(NC(c3cnc(CC)s3)=O)CC2)CC2CCCCC12 C=CCC(CC)C(=O)N1CC(=O)NCC1C(=O)NC(CO)C(C)O C1(CC(=O)N(CCNC(CCC#C)=O)CCc2ccccc2)COCC(C)(C)O1 c1(C(N2C(CNC(c3csc(-c4ccsc4)n3)=O)CCC2)=O)ccnnc1S Nc1c(C(=O)Nc2cc(OCC(F)(F)F)ccc2Cl)ccc(Cl)c1F n1(CC(=O)OC)cnc(C)c1C(=O)N.c1(C=O)n[nH]c(C)c1Cl.C1COCC1 O(NC(=O)C(F)C(C)CNC(=O)Cn1nc(C)nc1C)CCC C1(C)(OC)CC(NC(C2CSCN2C(=O)Cc2cn(C)nc2C)=O)C1(C)C C1(CC(=O)NCCN(C(=O)C(O)CC2CCOCC2)C)Cc2ccccc2O1 c1(C(C(=O)NCC(=C)C)N(CC(=O)NC2CCCC2C)C)cnc(C)cn1 Cc1ccc(O)c(C(N2CCC(O)(CNC(=O)C(F)(F)c3nccn3C)C2)=O)n1 c1(CC)cc(C(=O)NCC(O)C)ccn1.c1(C=O)cccc(OC(F)(F)F)n1.N c1(C(N2CC(OC)C(NC(=O)C(C)CF)C2)=O)cncc(P(C)(C)=O)c1 Cn1cc2cc(C(=O)NCC(C3CC3)NC(c3ccc(=N)[nH]n3)=O)ccc2n1 C12(C(N(C3(CC(=O)N(CCCO)CC#C)CC3)C)=O)CCCC1C2 C1(NC(=O)CC2CCCO2)CC2C(NC(C3(C(F)(F)F)CCCCC3)=O)C2C1 C1(C(N(C2CCCCCC2)CCNC(c2c(C)noc2)=O)=O)CCCC(=O)N1 c1cc(O)nc(O)n1.C1(F)(C(=O)NCC2CC2)CCC1.N12CC(C1)C2=O C1(n2c(C(C3CC3(C)C)NCC(C)C)nnn2)CCCCCC1 C(=O)CCCCC(C)(C)C.CC(C(=O)N)NC(=O)NCC1CCC1.C1CC1 O(P(C)(=O)CNC(C1CCC(CNC(=O)C2=CCCC2)CC1)=O)CC CC1(C)CCC(C(N2CC=CC(NC(C3CC(N4CCCC4)C3)=O)C2)=O)CC1 C1(NC(CCC#C)=O)CCCCN(C(c2cnn(C)c2N)=O)C1 c1(NC(=O)OC)cccc2ccccc12.C1CCCN1C(=O)Cc1cc(C)no1.C Cc1ccc(-n2ncc(-c3noc(C(c4cccnc4)(C)C)n3)c2N)cc1 C1(C)(CNC(C2N(C(=O)OC)CCC2)=O)CCN(C(c2ccccc2)=O)C1 CC1CC2(CC2)CN1CCC(=O)Nc1cccc(Cl)c1 C1(NC(C(CC)C(C)C)=O)CCCC12CN(C(c1cc(C(C)=O)cs1)=O)C2 C1(NC(C2CCC(CC)O2)=O)CC(NC(c2ccc(O)nc2)=O)CC1O c1(C=O)scnc1C(N1CCC1)=O.C(=O)CC.CC(C)C.CC.CCO.N C(=O)(CCCCc1cnn[nH]1)N.n1(C2CN(C(CNC(C)=O)=O)C2)cc(C)nn1 c1(C(C)=O)cc(C(=O)NCC=CCNC(=O)CCc2cc[nH]n2)no1 CC1(N)CCC(NC(N2CCCC2C2CCCC2)=O)CC1 C(=O)(C(CC)C(=O)OC)NC1C(NC(c2n[nH]c(CC)c2Br)=O)C1 C1(NC(c2cc(OC)cc(CC)c2)=O)CCCC12CN(C(=O)CCN1CCC1)C2 n1(CC#C)cnnc1C(N1CCCC1C(=O)NCCOCCC=C)=O C1(NC(C=C(CC)C)=O)CN(C(c2cc(C(C)C)on2)=O)CC2(CCOCC2)C1 c1(C(C(N2CC3CC3(C)C2)=O)O)cccc([N+](=O)[O-])c1.C1(C=O)(CCO)CC1.N C1(C(=O)NC(C)C(O)C(F)F)CC2(CCN1C(=O)CC(C)(C)CN(C)C)CC2 N1(C(C(C(CNC(COCCOC)=O)C)F)=O)CCOc2ccccc21 c1(CN2CCCN(C(c3[nH]cc(C(=O)OCC)c3)=O)CC2)cc(Br)c(F)cc1F C(=O)(C(C)(C)C(=O)NC1CC(C)N(C(=O)CCc2ccc(Br)cn2)C1)OC N1(C(C=CC=CCCCCC)=O)CCCC(C)C1CNC(=O)CC(=O)N.C C(=O)(CCCCCC#N)NC1C(C(N2C(CSC)CCC2)=O)C2CCC1C2 C1(NC(c2csc(CO)n2)=O)CCN(C(=O)CC2CCCCC2)C1 c1(NC(C2(O)CCN(C(C3(C)CC3)=O)C2)=O)cc(O)ccc1[N+](=O)[O-] N1(CC2(c3ccc(Cl)cc3)C(C)C2)CCC(=O)N(CC2CCOCC2(C)C)C1=O CCC(CC(=O)NCC(C)(O)COC)NC(c1ncoc1C(C)C)=O N1(C(C(CC)F)=O)CCOCC12COCCN(C(c1nc(C)c(C)[nH]1)=O)C2 C=CCC(CC)C(=O)N1CC(COC)(NC(c2cc(OC)cc[n+]2[O-])=O)C1 C1(CC)CCN(C(=O)COC2(C)CCC2)C(C(=O)NCCC(C)CCO)C1 C1(CNC(c2ccc(OC)c(N)n2)=O)CN(C(C2CC2C)=O)CC12CCOCC2 c1(CNc2cncc(C(=O)NCc3c(C)ccnc3)c2)ncc(Cl)cc1Cl C1(CNC(c2cncc(C)n2)=O)CC2CCC1N2C(c1cc(F)ccc1C)=O N1(Cc2cc(OC)cc(Br)c2)CCC2(CCCN(C(c3cnn(C)c3Cl)=O)C2)C1 C1(C(N(CC(=O)NCCC2COCC2O)C2CC2)=O)CCCCC(=O)C1 N1(C(C2C(C=C)C2)=O)CC(CNC(=O)CCc2cncc(F)c2)C2(CCC2)C1 Ic1cnc2ccc(Nc3ccn(-c4ccccc4)n3)nn12 CCC(C)C(C(=O)NCC1(F)CC(O)C1)NC(=O)CCOCC1CC1 N1(C(C(COCC)(C)C)=O)CC2CC(C1)C2NC(=O)Cn1cc(C)nn1 C=C(C)CC(C(=O)N)NC(c1ccc(COC)o1)=O.C1CCC2(CC2)CO1.C N1(C(c2cc(C)nc(O)c2)=O)CC(C)C(NC(c2cnn[nH]2)=O)C(C)C1 c1(C(C(=O)NCC2CCOCC2)N(CC=C)C(C)C)nc(Cl)sc1Cl C(C(COC)C(=O)NCC1CC1C)OC.c1(C(=O)N)nc(Br)c(C)s1 C1(C(=O)OCCC2CCNC2=O)CC2CC1C1CC21 Cc1cc(C(N2CC(NC(C3(C)CCCN3C)=O)C(C(F)(F)F)C2)=O)cc(C)c1 C1(NC(c2cc(CCC)c(C)s2)=O)CCN(C(=O)C(C)(O)C2CCC2)CC1F C(=O)(C1=CC2(CCOC2)C1)NC(C(CC)C)C(=O)NCCC(=O)NC(C)C N1(C(Cc2cc(OC)no2)=O)CCC2C(CCCN2C(C2CC(SC)C2)=O)C1 N1(C(c2cn(CCC=C)nn2)=O)CCN(C(C2CCC(F)C2)=O)CC1CCO c1(C(N2C3(C(=O)NCCCc4n(C)ncn4)CC3CC2)=O)cccn2ccnc12 C1(CNC(=O)NCCOCCN=[N+]=[N-])(CO)CC12CCC2 C=Cc1cc(C(=O)NCC2CCN(C(C3(C)COCCO3)=O)CC2O)cc(F)c1 N1(C(C(C)(C)OC(C)C)=O)CCC(C)(C)CC1.C(=O)(C=O)N.CC(F)(F)F N1(C(C(C(=C)Cl)(C)C)=O)CC2C(NC(=O)CC3CC3)CS(=O)(=O)C2C1.C C1(C(=O)NCC(NOCC)=O)CC12CCN(C(C1CCN(C)C1)=O)C2 N1(C(C2(CCCC)CC2)=O)CCC(C(N2CCC(O)(C(N)=O)CC2)=O)C1(C)C CC1(C)CCC(C(N2CC3CC(NC(C4C(C)(C)C4(C)C)=O)C2C3)=O)CO1 c1(CNC(C(CC)CC)=O)ccccc1C=O.N(C1CC1)(CC)CC.O C(=O)(C1=CC2(CCOCC2)C1)NC1C(N(C(C(C(C)C)C)=O)C)CCCC1 C(CC1CC1)(CC(=O)N1CC(N(C)C)C1)NC(CN(CCC#C)C)=O C(CCCC(F)(F)F)NC(C1CCCC1C(c1cnn2c1CCC2)=O)=O N1(C(C2C(C)(C)C2(C)C)=O)CCCC(CCNC(c2nsnc2O)=O)CC1 c1(C(N2CC(CCNC(CC(CC)SC)=O)OCC2)=O)nc2c(s1)COCC2 N1(C(N)=O)CCCC(C(N2CCC(CF)(NC(C3CCCC(CF)C3)=O)C2)=O)C1 C1(CNC(=O)C)CC(O)CN1C(=O)CCc1cc(Cl)cs1.C1CC1(Cl)Cl C(=O)(C1=C(C#N)CCC1)NC1CC(C)(C(N2C(CC#C)CCCC2)=O)C1 C=C(C)CN=C(NCC(C)(C)OC)N1CCC(OCc2ccccc2OC)C1 c1(CNC(C(C2CC=CCC2)C)=O)cncc(Cl)c1 c1(CC)ncncc1C(=O)NCC(C)(O)C.C1(C)(C(=O)N)CCC1C=O C1(NC(C2(CC)CN(C(=O)CCCn3cccn3)C2)=O)CCCCCC1F c1(C(C=O)O)cccc(F)c1.c1(C(C)C)ccc(C(N2CC(OCC)C2)=O)s1.N C(=O)(CCC(F)(F)C(F)F)N1CC(O)(CNC(=O)CCc2cnoc2)C1 N1(C(CC=C)=O)C(C)CN(C(=O)C(C)(C)C(F)F)CC1C c1(C(N(C)CC)=O)ccc(NC(C2(CC)CCC2)=O)nc1 CN=c1[nH]c(=NCCc2nnc3c(=O)[nH]ccn23)[nH]c(=NC2CS(=O)(=O)C2)[nH]1 c1(C(=O)NCC2CCCC2)ccc(O)cc1Cl.n1(C2(C(=O)N)CC2)ccnn1 C1(CC)CCC(O)(C(N2CCC(CN(C)C(C3(OC)CCCC3)=O)CC2)=O)C1 c1(OC)ccccc1C(CNC(=O)CC1CCN(C(C)=O)C1)NC(C)=O N1(C(C2C(C)(CC)C2)=O)CC2(C)CN(C(C3CCCCS3)=O)CC2(C)C1 C1(OC)CC(C(=O)NC2CC(O)(C)C2)CC1.c1(C=O)cnoc1C(C)C N1(C(C(C)(CC2CCC2)OC)=O)CC(CC(=O)O)OC(C)C1 n1(COCC)nnc(C=O)c1N.C1(CC)CN(C(=O)CN2CC(C)C2)CCO1.N CC1CSCCN(C(=O)CC(C(F)F)NC(=O)CCN(C)C)C1 C#Cc1ccc(C(=O)NCC(C2CCCCC2)NC(C2CC(F)C2)=O)nc1 N1(C(C(C)NC=O)=O)CCCC(CN(C)Cc2c[nH]ccc2=N)C1 c1(CC)cc(C(=O)NC(C)C(C)NC(C2(CC(C)C)COC2)=O)on1 c1(C(=O)NC(CCNC(Cc2ccc(C)o2)=O)(C)C)cc(Cl)sc1S(N)(=O)=O Cc1nccc(C(=O)N(C2CCN(C(c3nnn(C(C)C)c3C)=O)C2)C)c1Cl N1(C(CC(=O)OC)=O)C(C(=O)NCc2ccc(O)nc2)CC2CC12 C1(CC(=O)OC)CC(NC(C2CC(NC(C3(SC)CC3)=O)C2)=O)C1 N1(C(C(C)N(CCC)C(c2cnsn2)=O)=O)CCC12CCN(C)C2 CC1(C)CC(NC(=O)CC2CCCN2C(=O)C(N)=O)CCO1 c1cnn2c1CN(C(C1C3CC4C(C3)C14)=O)CC2.c1(C(=O)N)cccc(O)n1.C c1(CC)nccn1C(C)CC(=O)N1CCC(N(C(=O)COCC)CC)C1.O C(=O)(C1=NOC2(CCC2)C1)N(C1CN(C(c2ccc(F)c(F)c2F)=O)CC1F)C C=CC(C)CC(=O)N1CC(=O)CC1C(N1CCN(C2CC2)CC1)=O C1(NC(COCc2ccc(C)cc2)=O)CC12CCCCC2.C(=O)C(F)=C(C)C N1(C(C(C)=C(C)C)=O)CCN(C(c2n[nH]c(C)c2F)=O)C(CC(F)(F)F)C1 CC(C)CC(C(=O)NCCCCCNC(=O)Cc1ccc2nonc2c1)C(C)C C1CN(C(=O)CCc2ccnn2C)CC1C(F)(F)F.Cc1cc(C(=O)NC)sn1 c1(C=O)cncc(S(C)(=O)=O)c1.C(=O)(CCCC(=O)NC(C)C(C)C)OC.N c1(NC)ccc2ncnc(N(C3CC(N)C3)CC)c2n1.c1ncc(C(F)(F)F)[nH]1 Cc1cc(Cl)c(C(=O)NCC2(C)CCCC2)cc1C.c1(CC(=O)N)cccnc1 C1(C(=O)NCC2N(C(C=C)=O)C3C(C2)COC3)CCC2CCCCC2C1 N1(C(C(CC#C)C)=O)CCn2ncc(CN(C(=O)C3=CCCCC3)C)c2C1 Cc1cnc(C(=O)N(C(C)CNC(C2CC(=O)CO2)=O)C)cc1C C(=O)(C#CC1CCCC1)N1C(C(=O)NC(C(CC)C)CO)CC2CC21 n1(CC2CC(NC(=O)C(O)C3CC3)C2)cc(-c2cnc(C3CC3)s2)nn1 CC(C(C)C)NC(c1ccn(-c2ccccc2)n1)=O.n1(CC(=O)N)cc(Cl)cn1 CN1CCC=C(CNC23CCC(CC2NC(=O)OC(C)(C)C)C3)C1 c1(C(CC)NCCNC(C2(C)CC2)=O)cc(C)ccc1OC Cc1coc2c(NC3CC(CC#N)C3)ncnc12 C1(NC(C2(C)CCCCNC2=O)=O)CCC2CN(C(=O)C=CBr)CCC2C1 C(C(CC1CCOCC1)N(C)N1CC2(CCC2)C1c1ccc(F)o1)OC C12(C(N3CC(O)(CC)C3)=O)CCCN(CC1)C2.c1(OC)ccccc1CC(=O)N N1(C(CCNC(NC)=S)=O)CCC2CN(C(=O)Cc3ccc(O)cn3)CC2C1 c1(OC)cc(Br)c(F)cc1NC(=O)C(C)CCCl C1(NC(c2ccc(C)o2)=O)COC2(CCN(C(=O)COc3ccccc3F)C2)C1 C#Cc1ccc(OCC(=O)NC(C)C(CO)NC(c2ncsc2C)=O)cc1 N1(C2CC2)CCC2(CCCN2C(=O)CCS(C)=O)C1.CC1CCN2C1C2=O C1(COC)(C)CCCN1C(=O)CC1COC(=O)N1.C1(C=O)CCCCC1.N N1(C(c2c(C)cco2)=O)CC2CN(C(=O)Cn3nnnc3C)CC2C(F)(F)C1 C1(NC(CC2CC(CC)C2)=O)CS(=O)(=O)CC1.c1(C(=O)N)ncn(C)c1C C(CCCC(=O)NC(C)(C)CC(C)C)N(C(c1cc(OC)ns1)=O)C C1(C(N2CCC(C(F)F)(CNC(=O)CC3CCCO3)C2)=O)OC2CCC1CC2 C1(NC(C(C)C2CC2)=O)CC12CCN(C(=O)CNC=O)CC2 C=CC(CC)CC(=O)N1CCC1C(=O)NCCCc1nc[nH]n1 C(C)(CNC(C1CCC(O)CN1C)=O)(CC(C)C)NC(CCOCC)=O N1(CCOC)CC(C(=O)NCC(C(C)C)NC(=O)CC)CC1=O.C1CC1.O c1(CC)ccc(NC(C2(CNC(C3CCCC(CF)C3)=O)CCOC2)=O)cn1 c1(CC(=O)NC(C)C(C)NC(=O)CCC#N)ccc(C#N)cc1 CC1CN(C(c2csc(C3CCCCC3)c2)=O)CCN1C(=O)CNC(=O)C1CC1 c1(C(=O)N)[nH]c2ccc(F)cc2c1Cl.CC1(C)CC1(C)C(=O)NCCCC1CC1 c1(C(N(C2CCN(C(c3cnn(CC)c3)=O)C2)CCC)=O)ncccc1CC N1(C(C=Cc2cncc(C)c2)=O)CCC2CN(C(=O)CC(F)(F)C(F)F)C2C1 C1(C(=O)N(C(C)C=O)C2CC2)(OC)CC(C)C1.C1CC(CC(N)=O)C1.N CCC(C)CCC(O)CC(=O)NC1CCCC1CNC(C1(c2cccs2)CC1)=O c1(C(=O)NC2C(C)CN(C(c3cc(N)c(Cl)cn3)=O)CC2)cc2cn[nH]c2cn1 C(=O)C1=NOC(C)C1.C1(C(=O)NC(C)C2CC2)(OC)CS(=O)(=O)C1.N C(C(C(=O)NC(C)(C)C(C)NC(C1CC(OC)C1)=O)N(C)C)OC N1(C(c2cnc(=N)[nH]c2)=O)CC(NC(C2(Cl)CC23CCC3)=O)CC2(CCC2)C1 C(=O)(CC(CC=C)NC(=O)C(C)c1cc[nH]n1)NC(CC#C)C(=O)OC CCC(CCCC(=O)NCCCn1cncn1)NC(=O)C(C)C(F)F Cc1c(C(=O)NC(CO)CC)[nH]c2c1C(=O)CCC2.C(=O)(CC(C)P(C)(C)=O)N C1(C(=O)NCc2occ(C)n2)CC12CC(NC(c1cc(C)n(C)n1)=O)C2 C1(C(=O)NCC(F)CO)(CC)CCCN(C(=O)CCN=[N+]=[N-])C1 N1(C(CCSC)=O)CCC2(CC(NC(c3cnn(C(C)(C)C)c3)=O)CO2)C1 C1(NC(C=C(C)C)=O)CCC2(CC1)CC2NC(c1cc(Cl)ccn1)=O CCC(CC)(CCNC(=O)C(C)C(F)F)NC(=O)C(C)CC(C)C c1(OC)c(F)ccc(C(N2CCC(C)CC2)=O)c1F.C1(C=O)CC1C(F)(F)F c1(C(N2CCC(NC(C#CC3(CC)CC3)=O)C(O)C2)=O)ccc2nc(O)oc2c1 N1(C(CC(CC)C)=O)CC2CCCC1(CNC(c1cc(O)nc(O)n1)=O)C2 S(=O)(=O)(c1cccnc1NCC1COCCC1(F)F)N1CCN(CC(C)F)CC1 C(=O)(CC(C)C(F)F)NCC1(OC)CN(C(C(c2cccc(Cl)c2)OC)=O)C1 N1(C(c2cn(CC=C)nn2)=O)CCC2C(CCCN2C(=O)C=Cc2cc[nH]c2)C1 CC1CC(NC(c2ccccn2)=O)CN(C(=O)CN2CCCC2CO)C1 c1(C(=O)NC(CN(C(C(C)c2ncco2)=O)C)C)cc2cc(F)ccc2[nH]1 C1(NC(c2[nH]cc(OC)c(=O)c2)=O)CCOC12CCN(C(C1CSC1)=O)CC2 CN=c1cc(C(N2CCN(C)C(CNC(c3cc(F)cnc3O)=O)C2)=O)cc[nH]1 N1(C(c2cnc(OC)s2)=O)CCCC(C2(NC(c3cccc(F)c3C)=O)CC2)C1 CC1CCC(F)(C(=O)NCC2(F)CN(C(C3CC3)=O)C2)CC1.C1CCC1.C CC(CCCCCO)NC(C1(C)CC2CCC1C2)=O c12ccc(cc1)CNC(=O)NCS2.c1(OC)sccc1C(=O)OC N1(C(c2c(C(C)C)cccc2F)=O)CCN(C(C2CC(CF)C2)=O)CC(O)C1 Cc1nc2cc(CN3CC4CC3C4C(=O)Nc3cncc(Cl)c3C)ccc2s1 CCC(C#N)C(=O)N1CCCCC1CN(C)C(c1cn(C)nc1SC)=O c1(CC(N2CCC(F)C2)=O)cc(F)cc(F)c1.c1(COC)ccoc1C=O.N C(C(COC)C(=O)N(CCCNC(c1ccccc1)=O)CCO)OC.CCO.O C1(C(=O)NCC=C2CCN(C(C(CC=CC)CC)=O)CC2)CCOCC12CCC2 c1(OC2CN(C(C(C)=CC)=O)C2)nc2c(Br)cccn2c1N C(C(C)(C)CC(=O)NCCCN1CCCC1)NC(COCCC=C)=O N1(C(C(C2CCC2)OCC)=O)CCOC(C)C1.C(=O)(C=CSc1ccccc1)N c1(C(=O)N)ncccc1.CCCC.C(=O)CC=C(C)C.C(C)(C)C.C(C)=O N1(C(C2C(NC(c3c(CC)noc3C)=O)CCOC2)=O)CCc2cccnc2C1 CCCS(=O)(=O)CC(=O)NC1(CNC(c2n[nH]c(C)n2)=O)CCC1 N1(C(c2c(CC)[nH]nn2)=O)CC(N(C(=O)C(C)CN(C)C)C)C2(CC2)C1.C CCC(CC)(C(=O)NC1CN(C(c2cc(O)ccc2C)=O)CC1SC)C(C)C CCCCC(O)C(=O)NC1CCC(CNC(=O)COCc2cccnc2)CC1 CCCC(C)(O)CC(=O)NC1CN(C(c2ccc(C(C)(C)C)s2)=O)CC1(C)C c1(OC)cccc(OC)c1C1CC1NC(C1(NCCO)CCCCC1)=O C(=O)(C1=CCS(=O)(=O)C1)NCC1(O)CCN(C(C2CCC(C)(C)CC2)=O)C1 C(=O)(C#Cc1ccccc1Cl)N1CCCC(O)(C(=O)OCC)C1 c1(C(N(C2CCN(C(=O)C#CC3CC3)C2)C)=O)ccc(C(F)(F)F)cc1O C(=O)(C(C)(C)CCF)N1CCC(C(C(=O)NC2C(C=C)COC2)F)C1 c1(CC)cnc(O)c(C(=O)NCc2ccc(N(C)CCO)cc2)c1 c1(CNC(C2(NC(=O)CCC3CCCC3)C(C)CCC2)=O)ccc(O)cc1F c1(C=O)c(F)cc(F)cc1F.c1(C(=O)OC)ncccc1C(=O)NC1CC1.N CC1=C(C(=O)NC2CCN(C(=O)CN3CCOCC3)CC2O)SCCO1 C1(N(C(=O)Cn2cc(Cl)cn2)CC#C)CCN(C(C2CC3(C2)CC3F)=O)CC1 C1(CC(=O)OCC)NC(=O)CN(CC(=O)CC2CC(O)C23CCC3)C1=O.C C1(C(N2CCN(Cc3ncon3)CC2)=O)CCC(O)(c2ccccc2)C1 C(P(=O)(OC(C)C)c1cccc(C)c1)OC(CC=Cc1ccc(C(C)C)cc1)=O CC(F)(F)CCC(=O)NCCN(C1CCCC1)C(c1cnc[nH]1)=O C1(C(=O)NCCSC)CCCC1CNC(c1sccc1CO)=O Cc1cc(CCC(=O)N(C2CC=CCC2)CCO)no1 n1(CCC)cccc1C(N1CC=CC1C(=O)NC(C)Cc1cn[nH]c1)=O N1(C(Cc2scc(C)c2)=O)CCC2C(CCN2C(=O)CCCC(C)(C)C)C1 C12(C(=O)NC3CCC(N(C(c4ccc(C)o4)=O)C)C3)CC(C(F)F)(CO1)C2 O=C(CC(C(F)(F)F)NC(=O)C1=CCCOC1)NCc1cnccn1 N1(C(c2c(C)n(C)cc2)=O)CCN(C(c2csc(Cl)c2)=O)CC1CCO C1(n2cc(-c3ccn(C(C)C)n3)nn2)CN(C(c2cc(C3CC3)on2)=O)CC1C Cc1cccc(O)c1C(=O)NC1CC(CNC(=O)CC2CC3CCC2CC3)C1 C(N=c1nc2c(c[nH]1)ncn2C)C1N(C(c2ccn(CCC)n2)=O)CCCC1C Cc1c2ccc(NCCc3ccc(OCCF)cc3)cc2nn1C c1(C(=O)OC)cc(NC2(CCO)CCOC2)c(N)c(COC)c1 CC1CN(C(c2ncoc2CNC(c2ccc(F)cn2)=O)=O)CCC1O C1(CNC(CSC)CCO)CCCC(F)(F)CC1 C1(CC(=O)NCC(CC)N(C)C)C2CCC(C2)N1C(=O)C(=O)N(C)C O=S(NC(c1cccc(C(F)(F)F)c1)C1CCOCC1)c1ccccc1Cl c1(C(=O)NCCCCCOC)ccc(-c2coc(C)n2)cc1 Cc1c(CC(=O)NCC#CC(=O)Nc2ccsc2)cnn1C N1(C(C2(c3ccnc(F)c3)CCC2)=O)CCC(n2ccnc2)CC1 N1(C(C(C=C)O)=O)CC(=O)NC2CN(C(=O)CCc3cc(OC)no3)CCC12 C1(NC(c2n(C)cc(Cl)c2)=O)CN(C(=O)CSCC(N)=O)CC1(C)C C1(C(=O)NC2C(C)CCN(C(C3(CCC)CCC3)=O)C2)CCc2nnc(C)n2C1 c1(CCCNC(C)C=O)c(C(N2CC(CSCC)NC2=O)=O)ncnc1C.O C1(CC)CN(C(=O)Cc2cnc[nH]2)CCO1.c1(C(=O)N)ccccc1C(F)(F)F C(=O)(C1=CC2CCCC12)NC1COCCN(C(c2c(Cl)nc(N(C)C)s2)=O)C1 c1(C(=O)NCC2CCCC2F)cc(Br)cn2ccnc12 N1(C(c2c(C)onc2Cl)=O)CCC(C)(C)C(NC(c2ccns2)=O)C1 C1(CC(=O)N(CCNC(CCC(C)C)=O)CC)Cn2ccnc2NC1=O.CCO.O c1(C(N2CC(NC(C(C)=C(CC)C)=O)(COC)C2)=O)cc(CO)n(C)n1 C#CCC(O)C(=O)N1CCC(C(C)C(=O)NC2(c3ncc(C)o3)CC2)C1 c1(C2CC(NCC(O)CC3(O)CCOC3)C2)ccccc1Cl c1(CC(N2CCC(CCNC(C3CC34CCC4)=O)C2)=O)ccnc(O)c1 C1(CCNC(CCC(=O)NC)=O)CC(F)(F)CN1C(C1CCCN(C)C1)=O c1(C(N2CCC(CNC(C(C3CC3)OC)=O)CC2)=O)c(N)cc(Cl)cc1Cl C(CCCC(CO)NC(c1nn[nH]c1C(F)(F)F)=O)NC(=O)Cc1cnsc1 c1(CC(=O)NCC2(C(=O)NCc3ccc(Cl)nc3)CC2)ccc(F)cc1O C1(NC(CC=C(C)C)=O)CCCC12CN(C(c1cc(Cl)cc(Cl)c1N)=O)C2 c1(C(N2CC(C(N(CCOCCC#N)CC)=O)C2)=O)c(F)cc(O)cc1F c1(C(=O)NC2CN(C(C3C=CCC3)=O)CC2O)cc2cc(F)cc(F)c2o1 N1(C(C(C)NC(C)=O)=O)CCCC(NC(C2(CS(C)(=O)=O)COC2)=O)C1C Cc1nc(C(=O)NC2C3CC2N(C(c2cc(=O)cc[nH]2)=O)C3)c(C)s1 C(=O)(C1CC(O)c2ccccc21)N1CCC(C)(NC(C(C=C)O)=O)CC1 Cc1cccc(C)c1C(=O)NCC(C)N(C(C)C(=O)NCC(C)C)C CC1CCOCC1C(=O)NCCn1cnc(C(=O)NC2CC(CCF)C2)c1 c1(CC)nocc1C(=O)NCC(C1CC1)NC(C1CC(SC)C1)=O C(=O)(CCCC(C)(F)F)NCC(CC)NC(c1c(CC)ncnc1CC)=O C=CC1(C2(C(N3CCC(NC(=O)C(O)CC)C(O)C3)=O)CCC2)CCC1 c1(C(=O)NC2C(N3CCN(C(COC(C)=O)=O)CC3)CCC2)cc(F)cnc1O C12(CC)CC1CN(C(=O)C(C1CC1)NC(=O)CC1CC(F)(F)C1)C2 C(=O)(CC(C(F)(F)F)NC(C12CCC(CC1F)C2)=O)NC(CC)C(=O)OC c1(C(=O)NC(C)C(CO)NC(c2ocnc2C2CC2)=O)ccc(C2CC2)cc1 n1(CC(=O)NCC(CNC(=O)C(F)C2CC2)OC)ccc2ccccc12 C1(CC)CN(C(C2CC=CCC2)C(=O)NCc2ccco2)CC(=O)N1 C1(C)(CNC(COCCN(C)C)=O)CN(C(=O)CCc2cncn2C)CCO1 c1(N(CCN(C)C)C)nccc(=NC2CCCC2)[nH]1 N1(C(C2(C(F)(F)F)CC(C)(C)C2)=O)CCCN(C(=O)CC2CCCO2)CC1 N1(C(CC(C)O)=O)CCCOC(CCNC(C2(N3CCNC3=O)CC2)=O)C1 c1(OC)c(C(=O)NCC2CC2)cccc1[N+](=O)[O-].n1(CC(=O)N)ccnn1 Cc1nn(C)cc1CC(=O)NC1CC(C(C)NC(C2CCCCN2C)=O)C1 c1(NC(C)=O)ccc(C(N2C(C(=O)NC3(CCO)CCC3)CC3CC23)=O)cc1 n1(CC)nc(C(N2CCC(CC(C)NC(C3(C(F)F)CCC3)=O)CC2)=O)cc1C N1(C(C2(F)CCN(C(CCCOC(C)C)=O)C2)=O)CCCOC(C)C1 n1(CCCC#C)c(N(C(C)CS(C)=O)CC)nnc1CC1CCOCC1 C=CCC(C)C(=O)NCc1nc(C2CCN(C(=O)CCCF)CC2)n[nH]1 N1(C(COCc2cc(C)no2)=O)CC2CC(C)N(C(=O)C(F)C(C)C)C2C1 C(=O)C(C)CCC(C)(C)C.C1(CC#C)(C(=O)NCC2(C)CC2)CCC1.N N1(C(c2c(F)cc(OC)cc2Cl)=O)CCCC2C1CCN2C(=O)CSCCO c1(NC(=O)CC2(NC(=O)Cc3cc(Br)nc(Br)c3)CCC2)cc(C)ccc1F C(=O)(C(C)(C)CNC(=O)CCc1csnn1)N1CCC(CCC)C1 Cc1nnc2n1C(C(=O)N1C3CCC1CN(C(C1(F)CCCOC1)=O)C3)CC2 C1(NC(c2nc(F)ccc2Cl)=O)CC2CN(C(c3ccccn3)=O)CC2C1 N1(C(c2nc(COCC)sc2)=O)CC2(CCCO2)C1.C1(C=O)C2CCC1CC2 N1(C(C2(COC)CCC2)=O)CC2CC2(C(=O)NCC2(Cl)CC2(F)F)C1 C(c1cccc(F)c1)=CCC(=O)OCCC(C)N(C)C Cc1cc(CN2CCC(CNc3ccncn3)CC2)ccc1F N1(C(CC2CC(C)C2)=O)CCC2CN(C(=O)CSCCC(F)(F)F)CC2C1 C1(NC(c2c(C)nc(CC)o2)=O)CN(C(=O)Cc2cnnn2C)CC2(CC2)C1 C1(C)(CCC)CCN(C(=O)CCN(C)C(C2COCC2C(N)=O)=O)C1 Cc1cnc(C(C=O)N(C2CCN(C=O)C2)CC(F)F)o1.C(C)(C)C.C1CC1 n1(CCC)cc(C(=O)NC(C)C(CO)NC(=O)CC)cn1.[SH](=O)(=O)CC.N N1(C(C2CC(C)C2)=O)CCC2CCCC(C1)N2C(c1ccc2cccnc2n1)=O c1(C(=O)N)c(S(N)(=O)=O)ncn1C.N1(C(C2C(=C)CC2)=O)CC2CC2(C)C1 C1(C(=O)NC(C)CCC)(COC)CCCCO1.c1(C(=O)N)nc(=O)n(C)[nH]1 c1(SC)cc(C(N2CC(C(C)(C)O)(C)C2)=O)co1.C(=O)CC.C(C)=O.N c1(CC(=O)NCCN(C(c2cccc(Br)c2)=O)CC)c(C)cc(C)cc1C C(=O)(C(C)(C)CC(=O)NCC1CCC1)OC.c1(C=O)cc(C)cc(C)c1.N CC#CCCCC(=O)NCCN(C(c1ccc(C2CCOC2)s1)=O)C1CC1 c1(NC(CCc2cn(C)nc2C(F)F)=O)cccc2c1CCC2N C(CN=[N+]=[N-])(C=O)N(C)C(c1cc[nH]c1C1CC1)=O.C1CN(C(=O)CCC)C1 c1(CN(C(C)C)C)cn(C)c(=O)n(C)c1=O.N1(CC=O)CC(=O)N(C)C1=O c1(C(N)=O)cccnc1C(=O)NCCc1ccc(C(=O)NCC(O)CO)cc1 c1(NC(C(COCC)NC(c2ccn(C)c(=O)c2)=O)=O)ccc2ccncc2c1 N1(C(c2c(C)cc[nH]2)=O)CCCCC(CNC(C2(N(C)C)CC2)=O)CC1 C(C(C)Cn1cccn1)NC(COC(C)C)=O.C(=O)(CN(C)C(N)=O)N C1(C(N(CC(C)CCl)Cc2cc(C(=O)OC)no2)=O)CN2CCN1CC2.CC=C C12(C(=O)Nc3cccc(I)c3)CCCCC1C2(F)F C=CC(O)C(=O)NC1CCCC1NC(=O)COC1CC1 C1(C(=O)NC2CC(C)N(C(c3ccc(O)cc3F)=O)CC2)CCC2CCCCN12 C1(C(N2CCC(CC3CC3)C2)=O)(COC)CN(C(=O)Cc2ccns2)C1 CCC(CN(C)C)CC(=O)N1CCCC(NC(c2ccc(CSC)cc2)=O)C1C C1(CCC(=O)N(C2CCN(C(=O)COc3ccsc3Cl)C2)CC)CCCCC1 c1(C(N(C2CCCCN(C(c3cnccc3Cl)=O)C2)C)=O)cccc2cncn12 N1(C(C(C(=O)N(C)C)(C)C)=O)CC2C=CC1C(C(=O)N(C1CSC1)C)C2 c1(C(C)=O)cccc(OCC(O)CNCC2(O)CC2)c1 N1(C(C(CC#C)O)=O)CCC2(C1)CN(C(c1cc(F)cc(C#C)c1)=O)CCO2 c1(C(=O)NC(CNC(CCOCC#C)=O)CO)cnc(Br)s1 N1(C(c2ccnc(C)n2)=O)CCc2ccccc2C(N(C)C(C2CC(O)C2)=O)C1 CCCC(C)CCCC(=O)NC12CC1CN(C(c1ccc(OC)c(Cl)c1F)=O)C2 C1(CC(=O)NCc2ccsc2Br)CCCN(Cc2occc2Br)CC1 CCC(C(=O)N1CCC(NC(c2ccc(OC)cn2)=O)C1)C(C)C C(CC(C(=O)NCCCCCCC1CC1)NC(c1cnc[nH]c1=N)=O)=CC CCCCC(C)C(=O)NCC(C)(O)CNC(c1cccc(C2CC2)c1)=O Cc1nsc(N)c1C(=O)N.C1(C=O)CCOC1C(F)(F)F.C1(CC)CC1.C c1(NC(c2c(CNC(C(C3CC3)OC)=O)n[nH]c2)=O)cccc(NC=O)c1 c1(C(=O)NCCN(C)C(c2ccccc2SC(F)F)=O)ccc(Cl)nc1O C(=O)(CP(=O)(C(C)C)C(C)C)N1CCCC1(C)C.c1(CC)nc(C(=O)N)co1 Cc1nn2c(c1O)CN(C(=O)C(=O)NCCc1c(C)cc(Br)c(C)c1C)CC2 C1(C(N2CCN(CC(CN(C)C)O)CC2)=O)CC2CCC1CC2N CCCC(CNC(=O)CCNC(N)=O)C(=O)NCC(O)COC(C)C C1(CCOC)(NC(CCSCCC)=O)CCN(C(=O)CCC(=O)N(C)CC)CC1 CC1(NC(C2C=CCCC2)=O)CCCN(C(c2ccccc2-c2cn[nH]c2)=O)C1 N1(C(CN(C(C2CCC(C#N)CC2)=O)CC)=O)CCN(CC)C(C)C1 C(=O)(C1=CCS(=O)(=O)C1)N.c1(OCC)ccc(C)cc1C(=O)NCCC c1(CC)nc(C(=O)NC2C=CCN(C(C3CC4CC3CO4)=O)C2)c(Br)s1 CC1C2C(CCN2C(c2ccc(F)cc2F)=O)CN1C(c1ccc(CO)s1)=O C1(OC)CCC(C(=O)N(CCNC(=O)Cc2scnc2C)CC2CC2)C1 CC1CN(C(c2ccco2)=O)CC2(CCN(c3nnnn3C)C2)O1 C1(O)(CCNC(CCCOC(C)C)=O)CCCN(C(C2(C(C)C)CC2)=O)C1 Cc1ncnc(C)c1C(=O)NC1CCCCC1NC(=O)CC1(CO)CCOCC1 CC1CN(C(=O)C=Cc2nccs2)CCN1C(=O)CC1C(C)(C)C1(C)C C(C(CC(=O)NCC1CCC=CO1)C1CCC1)NC(Cn1ccc(C)n1)=O C1(CNC(c2c(C)ncn2C)=O)CCN(C(C2CCC(F)(F)C2)=O)C12CCC2 C1(NC(c2ncc(F)cc2F)=O)COCCN(C(=O)COc2ccc(Cl)nc2)C1 C1(C(N2CC(O)(CN(C(=O)C=CI)C)C2)=O)(N(C)C)CCCCC1 C(=O)(C1=NNC(C(F)(F)F)C1)N(C1CC(NC(c2nc(C)oc2)=O)C1)C CCCC(CCCNC(C1(C)CC=CC1)=O)NC(=O)C(C)(C=C)CC c1(NCC2(C(=O)Nc3cnc(SC)nc3)CC2)ccc(C#N)cc1Br C12(NC(=O)C=CCF)CCCCC1CN(C(=O)CCN1CCCS1(=O)=O)C2 c1(C(F)Cc2cccnc2)nc(-c2cccc(Cl)c2)nn1CCC1CCCCC1 c1(C(=O)NCC(CC(C)C)NC(c2nc(C)oc2C)=O)ccc(C#N)c(F)c1 C(=O)(CCC(=O)NCC(C1CC1)NC(=O)Cc1cccc(C)c1)OCC c1(C(=O)NCCN(C(=O)CC)CCC)ccc(NC=O)cc1.C(=O)(C)N c1(C(=O)NC(c2ccccc2)CNC(CCSC)=O)ccsc1C(F)(F)F c1(C(=O)NCCCC=C)ccc2nc(C)nn2c1.C1(CC=O)CCCN1C(C)=O C=CC(CCC)CC(=O)NCCN(C)C(C1CC2CCC1O2)=O C(=O)(C1=CC2CCC(C1)C2)NC1(CO)CCCN(C(c2c(C)c(C#N)[nH]c2)=O)C1 N1(C(c2c(C)[nH]cc2)=O)CCN(C(c2cc(C3CC3)on2)=O)CC1C Cc1ccc(C(=O)NCC2CC(S(C)(=O)=O)C2)cc1-n1nccn1 N1(C(C)C)CCCC1C(=O)NCC1CCN(C(C23COCC2C3)=O)C1 c1(C=O)cc(C)c(Cl)cn1.c1(C(N(CC)CC)=O)cc(C)nn1C1CC1.N c1(C(N(CCCNC(c2cc(CC)[nH]n2)=O)C2CC2)=O)cc(C)ccc1C c1(OC)cc(CO)ccc1NC(c1cc(F)ncc1)=O.C1(C=O)C2COCC12.N c1(C(=O)NC2CC(NC(c3cn(C(C)C)nn3)=O)C2)ccc2nc(O)oc2c1 C1(CC(=O)NCCN(CCOC)C)CN(C(=O)CC(C)F)CC12CC2 C(=O)(C1CCc2cccc(OC)c21)NC(CC=C)CNC(=O)C(C)=C1CCC1 O(NC(=O)C(C)(C)C(N)=O)CC(=O)NC(CC)(C)CC c1(C(N2CC3CN(C(c4c(C)n(C)nc4)=O)C3CC2)=O)cc2c(s1)CN(C)CC2 C1(=CC(=O)NC2CCCN(C(c3nc(C)oc3C)=O)C2)CCOc2ccccc21 c1(NC(C2C(=O)NCCCC2)=O)ccnc(Br)c1[N+](=O)[O-] C12(C(=O)NCCOC(C)=O)CC1CCN2C(=O)Cc1ccsn1 O=C(C1OCCc2c(O)cccc21)N1CCCNC(c2ccccc2C(F)(F)F)C1 N1(C(c2ccc(C(=O)NC)cc2)=O)CC2CN(C(c3cncc(F)c3)=O)CC12 C1(NC(C2(c3ccc(Cl)cc3)CC(=O)C2)=O)CCCCC12CCCC2 c1(C(=O)NCC(N(C(CCCSC)=O)C)C2CC2)c(C)oc(C)c1Br CC1CCc2[nH]nc(C(=O)NC3CCCCN(c4ncnc(Cl)c4Br)C3)c2C1 C1(C(N(C2CCN(C(C3CCOCC3)=O)C2)C)=O)CC(=O)N(C(C)(C)C)C1 N1(C(C(C)CN(C)C(C)=O)=O)CCn2ccnc2C1.C1(=O)C(C)(C)CN1 c1(C(N(CC(CC)NC(c2ccoc2Cl)=O)C)=O)ccc(-c2ccccc2)s1 c1(C(=O)NC(CNC(C(CC)CC(C)C)=O)C(C)C)c(C)oc2nc(Cl)ccc12 C1(N(C(CCSCC(C)C)=O)CCO)CCCN(C(C2CCNC(=O)C2)=O)C1 Cc1cccc(C(C)(C)NC(=O)NCC23CCC2CCN3)c1 N1(C(c2c(C)[nH]c(C#N)c2)=O)CCC2(CC2)CC1C(=O)NC1CCCSC1 N1(C(C)=O)CCN2CCOCC2(C(N2CC(CC(C)(C)C)C2)=O)C1.C(C)(C)C.CC C1(NC(c2c(C)oc(CO)c2)=O)CCN(C(C2CCOC2CC)=O)C12CCCC2 C(=O)(C1=COCC1)NC(CC)CN(C(c1cnc(-c2cccs2)o1)=O)CC C(=O)(C1CCc2c(Cl)cccc21)N1C(CNC(=O)C(O)Cn2cncn2)CCC1 Cc1cc(C(=O)NCC2CCN2C(=O)CCC(=O)c2ccccn2)c(O)nn1 C(=O)(C1=NN(C)C(=O)CC1)N(CC(CN(C(CC=C(C)C)=O)C)O)C c1(C(N(CC(F)F)C)=O)ncc(NC(C2(C)CC2)=O)cn1 N1(C(c2cncc(C#N)c2)=O)C2CCC1CC(CNC(c1cccc(F)c1)=O)C2 S(=O)(=O)(c1ccc(Cl)cc1Cl)Nc1ccc(NC(c2cc(F)ccc2Cl)=O)nc1 c1(C(N2CCNC(C(N3CCC3CO)=O)C2)=O)c(F)ccc(F)c1F Cc1c(CC(N2CC(NC(=O)Cc3nc[nH]n3)C2)=O)cnn1C c1(C(N(CCCNC(=O)CCC2CCCCO2)CC)=O)cnn(C(C)C)c1F Cc1ccc2c(c1)CC(C(N1CCC(C(C)(C)NC(c3cnc(Cl)[nH]3)=O)C1)=O)S2 Cc1noc2nc(=NC(C)c3ccc(S(C)(=O)=O)c(F)c3)[nH]c(O)c12 C(=O)(CCS(=O)(=O)CC(C)C)NC1(COC)CN(Cc2ccccc2C)C1.C C1(CNC(C(c2cnn(C)c2)C)=O)CCN(C(=O)C(=O)N(C)C)C12CC2 CCC(CC)C(C)C(=O)NCC1CCN(C(C2CNC(=O)C2)=O)C(C)C1 CCCCC(C)C(=O)NC(CO)CCCNC(C1(F)CCC1)=O N1(C(CCC=C=C)=O)CCCN(C(=O)CN2CCC2C)CC1C N1(C(Cn2ccc(C)n2)=O)CC2CC1C2NC(c1cnn(C2CCCC2)c1C)=O Cc1cc(C(=O)NC(C)CC(C)C)n(C)n1.c1(C(=O)N)ccc(C2CCC2)nc1 C1(C(=O)NC2CCCN(C(c3sccc3F)=O)C2)CC2CCC(C1)C2O n1(C(C)C)nnc2c(N(CC)C3CC3)ncnc12.C1(CC(=O)N)CCCC(=O)N1 N1(C(CCOCC(C)C)=O)CC2CCC1CC2.C1(C=O)CC(=O)N(C2CC2)C1.N CCCCCCCC(=O)N1CCCC12CN(Cc1cc(C(C)(C)C)ccc1O)C2 C1(C(C)C)CN(C(=O)Cc2c(O)ncnc2O)CCN1C(C1CC12CC2)=O N1(C(CN2CCN(C)CC2)=O)CC(C2(NC(C3CCCCC3(C)C)=O)CC2)C1 C12(NC(=O)C=Cc3cccs3)CCCCCC1N(C(C1CCC(F)C1)=O)CC2 N1(C(c2nc(COCC)sc2)=O)CCOC(CCC)C1.c1(C(=O)N)occc1C C1(C)(CC(=O)NCC(CCC)NC(=O)C=CCN2CCOCC2)CCOCC1 N1(C(=O)CC2(O)CCOC2)CC2CCC(C1)N2C(=O)COc1c(F)cccc1Cl C#CCCCCCCC(=O)N1CCC(CNC(c2cccnc2C)=O)CC1 Cc1nc2cc(C(N3CC4(C3)SCCC4NC(C3CSCCS3)=O)=O)cnc2[nH]1 C(=O)(CS(=O)(=O)c1cnnn1C)Nc1cccc(C(=O)NC)c1C C(CS(=O)(=O)CC(=O)N(CCCCC(N1CCC12CCCSC2)=O)C)OC Cc1[nH]c(=N)nc(O)c1CC(N1CCC(CO)C(NC(=O)CC(O)C(C)C)C1)=O CCC(C(=O)NC(CCCNC(=O)CC1CCC(=O)N1)c1ccccc1)C(C)O N1(C(C2C(CC)N(C(=O)C(C)=CC3CC3)CC2)=O)CCn2nccc21 Cc1ccc(C(N2CCC(N(C(=O)C(O)CC3CC3)C)C2)=O)c([N+](=O)[O-])c1 N1(C(c2c(C#N)nccn2)=O)CCCC2(NC(=O)CSCC(F)(F)F)CCCC12 C1(OC)CC(NC(c2c[nH]c(-c3ccccc3)c2)=O)CN(C(c2cn[nH]c2)=O)C1 N1(C(c2c(C)coc2C2CC2)=O)CCC2C(CCCN2C(=O)C(C)N(C)C)C1 c1(C(=O)NC2CN(S(=O)(=O)c3nccs3)CCC2Cl)ccc(O)c(F)c1F N1(C(C2CN(C)C2)=O)CCC2CN(C(=O)Cc3cccc(Cl)n3)CC12 Nc1cc2[nH]cnc2cc1C(N1CC2CC2(NC(=O)C=CCN2CCCC2)C1)=O N1(C(c2cc(Cl)sc2C)C(=O)NC(CC)(C)C)CC(=O)NCC12CC2 Cc1nc(O)[nH]c1C(=O)NC(CNC(C12CC3CC1C2C3)=O)C(C)(C)C c1(C(N2C(C(C)(C)CNC(=O)C)CCC2)=O)ccc(F)cc1F.[SH](C)(=O)=O c1(C(=O)NC2C(NC(c3ccc(C)nc3N)=O)C2)cc2cccc(C)n2n1 c1(CN(C)CC2CCCCN2C(=O)COCCF)cc(Cl)ccc1F C1(NC(C2C(C)CC2)=O)CCN(C(=O)CNC(=O)C(C)(C)C)CC1(C)C C1(C)(C(=O)NC(c2nccn2C)C(C)C)CCCN(C2CCC(O)CC2)C1 c1(OC)cc(CCNCc2cc(Cl)ccc2C(F)(F)F)ccc1Cl C1(NC(C2CSCCN2Cc2ccc(O)c(Cl)c2)=O)Cc2ccc(Br)cc2C1 C1(C(N2CC(OCC(=O)N(C)CC3CCCCO3)C2)=O)CC(=O)NC1(C)C C1(CC(N2CCN(C(=O)OC(C)(C)C)CC2COO)=O)CCC2(CCCC2)O1 C(=O)(C(C(C)(C)O)NC(=O)CC(C)C)N1CCC(N(C)C)(CC)C1 N1(C(C2CCOC2C(=O)NCC2CC3CCC3C2)=O)Cc2cccc(O)c2C1 c1(NCCP(C)(C)=O)ccc(CNCC2CCC3(CCCOC3)O2)cc1[N+](=O)[O-] N1(CC)C(=O)CCC1CC(=O)NCC(C1CC1)NC(c1c[nH]nc1F)=O C(=O)C(C)(C)CC(C)(C)C.C1(NC(C2(CSC)CCC2)=O)CCCCCC1.N N#Cc1ccc(CS(=O)(=O)Cc2c[nH]nc2C(F)(F)F)cc1 C(=O)C(S(N)(=O)=O)c1ccccc1.c1(C(=O)NCC(CC)C)ccn(C)c1C.N c1(C(=O)NCC(CCCC)NC(c2cc(F)c[nH]2)=O)cccc2c1OCCCO2 Cc1cc(NCCCC(C)(C)NC(=O)CN2CCCC2=O)cc(C#N)c1[N+](=O)[O-] C1(CNC(CCC=CC(C)C)=O)CCCN(C(=O)C(C2CC2)N(C)C)C1 N1(C(c2nc(C)n(C)c2)=O)CC2CCC2(CC(=O)NCC2=CCCC2)C1 C1(C(N2C(C)(CCO)CC2)=O)C2CCC(C2)N1C(C1CCN1C(C)(C)C)=O c1(C=O)cccc2c1CC(=O)N2.C1(CNC(C2(CC)COC2)=O)CCCC1.N N1(C(CC2(OC)CCC2)=O)CC2CCCC(C1)N2C(C1CSCCS1)=O C1CS(=O)(=O)C2CN(C(C3CC4CCC4C3)=O)CC12.O=CCCOC.C1CC1 C1(CNC(=NCCOC)NCC(c2ccnn2C)O)CCN(S(N)(=O)=O)CC1 C1(NC(=NCc2nc(C)oc2)NC2CN(C)CC2O)CCc2ccccc2C1 N1(C(CC(C)(C)O)=O)CCn2nc(CNC(=O)CO)cc2C1.C1CC(F)(F)C1 c1(CC)ccc(C(=O)NCC(C)(O)CNC(=O)CS)o1.c1cccs1.C c1(OCC(=O)NC(CNC(C2N(C(C)=O)CCC2)=O)C)cccc(Cl)c1 N1(C(C(CCCNC(=O)C#CC2CC2)O)=O)CCc2c[nH]nc2C1 C(CCC(C(=O)NC(COC)C1CC1)NC(c1cccc(C)c1F)=O)OC N1(c2nnc(C(=O)OC)s2)CCC2(CCCN2C(C)=O)CC1 C12(NC(CC3(C)CC3)=O)CCCC(NC(c3cn(CCF)nn3)=O)(C1)C2 N1(C(C2(C=C)CCOCC2)=O)CCC2(CCN(C(=O)C(CC)NC(N)=O)C2)C1 N1(C(CCCCC(C)(C)C)=O)CCC2(CCCC2NC(C2CC=CCC2)=O)CC1 CS(=O)(=O)c1ccc(C#N)cc1.c1(C2C(C(=O)O)C2)ccsc1C(F)(F)F c1(NC(C2CCN(C(c3c(OC)c(C)ccc3)=O)C2)=O)ccc(S(N)(=O)=O)cc1 n1(CC)cc(CN2CCCC(NC(C3CCCO3)=O)C2)c2cccnc12 N1(C(C2C=CCN(C(c3n(C=C)ncc3)=O)C2)=O)CCOC(C)(C2CC2)C1 C1(C(NOCCCC=C)=O)CC2C=CC1N(C(c1cc(C)ccc1F)=O)C2 n1(CC=O)ncn(C)c1=O.C1(CC)(C(=O)N(C)CCN(C)C2CC2)CC1 N1(C(C2(C#N)CC(C)C2)=O)CC2CC(NC(=O)C(=O)NC3CC3)C1C2 CC1C(NC(c2cccnc2SC(C)C)=O)CCN1C(c1ccncc1)=O N1(C(CSCC(C)=O)=O)CC(C)(C)OCC1C.c1(CC=O)n[nH]c(C)n1.N c1(OC)cc(-c2nc(NC(=O)C(c3ccc(O)cc3)C)cs2)ccc1F N1(C(=O)Nc2c(C)cccc2)CCN(Cc2cc([N+](=O)[O-])cs2)C(CO)C1 C(=O)(C(O)CCC(F)(F)F)N1C(CNC(CCC=C(C)C)=O)C(C)CC1 C(C(C)CC(=O)NC(c1nc(C(N2CCCC2(CO)CO)=O)co1)C)OC c1(C(N2CCC(N(C(=O)CCCc3sccc3C)CCC)C2)=O)ccncc1F C1(CC(=O)NC2(CC=C)CCCC2)CN(C(=O)CCCC=C)CCO1 c1(CCC(=O)NC(CN(C(c2cc(Br)cn2C)=O)CC)C)ccc(N)cn1 Cc1ccc(C=CC(=O)N(CCC)C2CC2)o1.C1(C=O)CC1(C)C(C)C.N Cc1occ(C(F)(F)F)c1C(N1CCCC(NC(C23CSCC2C3)=O)C1)=O C1(CNC(C2(SCC)CC2)=O)C=CCN1C(c1ccnn1CC)=O c1(C(=O)Nc2c(OC)cc(-c3nn[nH]n3)cc2)ccnc2cccc(C#N)c12 CN1C(=O)C(=O)N(CC(=O)NCCCC2CC2)C1=O.C(=O)C(F)C1CC1.N C(=O)(C(F)(F)CC(C)C)N1CCC(NC(c2ccc(OC)nn2)=O)C(O)C1 c1(C(N2CCC(CCCNC(CSCCC)=O)CC2)=O)ncc(N)nc1C C(=O)CCCCN1CCOCC1.C1(CC(=O)N(C)CC2CC2)COC(=O)N1.C C(c1cnccn1)=CC(=O)NC1CC(CCNC(C(COCC)C)=O)C1 C(=O)(CC(F)(F)C(F)(F)F)NCC(CNC(C=C1CCC(C)CC1)=O)O Cc1cc(CNC(c2cn(C)nc2-c2cnn(C)c2)=O)ccc1C1CC1 C1(NC(c2n(C(C)C)ncn2)=O)CCN(C(=O)C(F)CC2CCCC2)CC1F c1(C=O)ccc(N(C)C)c(F)c1.CC1CCC(C(=O)NC)S1.C12CC(C1)C2 C12(CNC(C3(C(F)(F)F)CC3)=O)CCC(N=c3cncc(Cl)[nH]3)(CC1)CO2 n1(C(C)C)cc(C(N2CCC2C(=O)N(C)Cc2cn(C)cn2)=O)nn1 c1(CNCC2(C)CCCCC2(F)F)nccc2cc(Cl)ccc12 N1(C(CC(C=C)(C)O)=O)CC2(C1)SCCC2NC(c1sc(C2CC2)nc1C)=O CC(C)CC(CC(C)C)(c1nnnn1C1CCOC1)NCc1ncc(Br)s1 C1(O)(C(=O)NC2CCC3CCN(C(C(CC(C)C)O)=O)C32)CC2(CCOCC2)C1 C(=O)(C1=C(C)CCOC1)NC1C=CCC(C(=O)NCC(C(CC)CC)OC)C1 CC1CCN(C(c2cncc(CO)c2)=O)C1C(=O)NCCC(C)c1cn[nH]c1 C12(NC(C3CC(C#C)(O)C3)=O)CC(C)(C1)OC21CCN(C(=O)CCC(C)O)CC1 N1(C(c2c[nH]c(=NCC)s2)=O)CCC2(CC1)CC2NC(=O)C1=CC(O)CCC1 c1(C(N2CC3CN(C(C4(C5CC5)CC4)=O)CCC23)=O)ccc2cccnc2n1 N1(C(C2(C)CC(C)C2)=O)CCC(C)(NC(c2cccc(CCO)c2)=O)C1 C(N=c1[nH]c(=NCCS(=O)c2ccc(C)cc2)c2[nH]ccc2[nH]1)C1C(CC)C1 C1(CNC(c2c(C(C)C)c[nH]n2)=O)CC(F)CN1C(C1COC(C)C1)=O c1(C(N(CCC(c2cccs2)NC(CSC(C)C)=O)C)=O)cc(Cl)cs1 c1(C(=O)NCC#CCNC(C2C(C)C2)=O)c(F)cc(F)cc1Cl N1(C(c2ccc(C)c(I)c2)C(=O)NCCC)CCN2C(=O)N(C)C(=O)C2C1 C1(C(=O)NCC(CO)NC(=O)Cc2cncnc2)(CC)CC1(F)F C#Cc1cn(C)nc1C(N1CCOC(CC(=O)Nc2ccccc2C2CC2)C1)=O C1(NC(CC2CC(SC)C2)=O)CCN(C(=O)CC2CC2C)CC1 C12(CC)CN(C(=O)CN3CCCNC3=O)C(C)(C1)C2.C(=O)(C)N.CC=O C(=O)(C(F)(CNC(=O)CC1CC2(CC2)C1)C(C)C)NCCC(C(C)C)C C1(C(=O)NCCCC(C)NC(c2ccc(N(C)C)nn2)=O)CCS(=O)CC1 c1(OCC)ccccc1C(N1CC(NC(c2cccc(OC)n2)=O)C(C)C1)=O C(=O)(C(C)CC(=O)NC)OC.C1(C(N2CCC(F)C2)=O)CC(=O)NC(=O)N1 C12(CNC(C34C(CN(C(C(COC)(C)OC)=O)C3)C4)=O)CCC(CC1)OC2 C1(CC)CC(C)CN1C(C1C(O)CCN1C(c1cn(C)c(C)n1)=O)=O C(CC(C(=O)N1CC(C(N)=O)C1)OC)NC(C1CCC(CC)O1)=O N1(C(=O)COc2ccc(-n3cnnn3)cc2)CCCC2(CCO2)CC1 n1(CC)cc(S(=O)(=O)N2CC3CN(C(=O)CCc4ccnc(C)c4)CC3C2)cn1 C1(NC(C(COC)COC)=O)CC(F)CN(C(=O)C(C(C)C)n2cc(C)cn2)C1 c1(CC(N2CCCC(CNC(C3C(C)(C)C3)=O)(C)C2)=O)cccc2c1CCC2 N1(C(C2CCN(C)C2)=O)CCCC12CCN(C(c1cnc(C(F)(F)F)cn1)=O)C2 CCCCC(O)CC(=O)NC(C(=O)NC(CN(C)C)CC)C(C)OC N1(C(c2cc(C(C)C)no2)=O)CC2CCCC2(NC(=O)C#CC2CC2)C1 C(=O)(C(CNC(c1nccc(OC)n1)=O)CCC)NCC(COCC)(F)F N1(C(c2ncn(C)n2)=O)CCCCCC(NC(=O)CC2(CS(C)(=O)=O)CC2)C1 c1(C(=O)OC)ccc(CNC(=O)CC2CCCCC2)[nH]1 c1(N(C(=O)C(C)C(F)(F)F)CCNC(CC(C)F)=O)cc([N+](=O)[O-])sn1 Cc1noc(C)c1C(=O)NCC1CCCC1C(N1CCC1)=O.C(C(N)=O)N Cc1nc(-c2ccc(COC(C3(N)CC(OC)C3)=O)cc2)oc1C Cc1cc(C(=O)NCC2(O)CCCN(C(=O)Cn3ncc(Cl)c3C)C2)cc(O)n1 C1(CC(=O)NCCCC=C)CCCC12NC(=O)NC2=O.n1(CC(=O)N)cnnc1 N1(c2nnc(CCC)s2)CCC2(CC1)CN(C(=O)CC1CSC1)C2 C1(c2ccccc2Cl)(C(=O)NCC(CNC(=O)C(N)=O)OC)CCCCC1 C1(N(C)C)CCCCN(C(=O)C(=O)Nc2cn(C)c(C3CC3)n2)C1 C1(NC(C(CCC)OCC)=O)COCCN(C(=O)COCCc2ccccc2)C1 c1(C=O)c(C)nn(C)c1C.C1(C(=O)N)(COC)CC1(F)F.C(C)C1CC1 O=S(=O)(c1cc(Br)ccc1OC(F)(F)F)Nc1cc(F)cc(F)c1Cl N1(C(c2[nH]c(C)c(C(=O)Nc3ncncc3Cl)c2C)=O)CCc2c(O)n[nH]c2C1 C1(Cn2cc(C3N(C(Cc4nc(C)[nH]n4)=O)CCC3C)nn2)CCn2ccnc2C1 c1(C(=O)NC2CCCN(C(c3ccc(C)nc3)=O)C2)ccc(C#N)cc1F CC1(C(=O)NCC2CCCCN2C(c2cccc(N(C)C)n2)=O)CCSCC1 CC1(C#CC(=O)N2CCOC(CNC(=O)Cc3cnoc3)C2)CCCO1 C=CCCCC(C)(C)CNC(=O)C(C1CC1)N(C)C(c1csc(Cl)n1)=O CC1CN(C(c2cncnc2)=O)CCN1S(=O)(=O)CC1CCCC(F)C1 C(CC(O)C(=O)N(C1(C(=O)NCC(C)(C)C(=O)O)CCC1)CC)SC N1(C(c2c(C(C)(C)C)n[nH]c2)=O)CC(C)OC2(CCC2)C1.C(=O)C.C1CC1.N N1(C(Cc2cc(C)cc(F)c2)=O)CC(C(=O)NC(c2cscn2)C)C2(CCC2)C1 c1(C(N2CC(NC(=O)CC3CCC34CCC4)C3(C2)CC3)=O)ccc2nsnc2c1 c1(COCC)nnc2n1CCN(C(N1CCC1)=O)C2 C1(C(=O)OC)CC=CCN1C(=O)CC1COCCN1C(c1cc(OC)ns1)=O c1(NC(C)=O)cnccc1C(=O)N.n1(CC=O)cc(Cl)c(C)n1.C1CCCC1 C1(NC(c2n(CC)ccn2)=O)CC2CCC1CN2C(c1ncc(N)cc1C)=O Cc1cc(C(=O)NC(CCF)C(=O)NC2CN(C)NC2=O)c(C)[nH]1 CC1CCN(C(=O)C2=CCSC2)C(C(=O)NC(c2ccoc2)C)C1 N1(C(C2(CC)CN(C(=O)C(N=[N+]=[N-])C(C)C)C2)=O)CC2(CCCCCC2)C1 c1(C(=O)NCC(CC)NC(=O)C(C)N=[N+]=[N-])cc(O)nc(O)n1 c1(C=O)sccc1C1CC1.C1(C=O)CC1(C)C(=O)N(CCC)C1CC1.C Cc1cccn2ncc(C(N3C4CCCC3(F)CC4)=O)c12 N1(C(=O)OC(C)(C)C)CC(NC2CCSC2)CCC1C(F)(F)F Cc1n[nH]c(=NCC23CC(CNC(c4cc(C5CC5)ccn4)=O)(CO2)C3)o1 N1(C(C2(C(C)C)CCC2)=O)CCC2(CC(NC(c3cc(F)cc(Cl)c3)=O)CO2)C1 c1(C(N2CCN(CCNC(c3nn(CC)nc3C)=O)CC2)=O)c(C)cccc1N c1(OCC#C)ccccc1CC(=O)N(C(C1CC(O)CN1)=O)C1CC1 C1(NC(c2c(C)cncc2)=O)(CNC(C2CC=CCO2)=O)CC2CCC1CC2 CCCCCC(O)C(=O)N1CC(CN(C)C(C2CCN(CCO)C(=O)C2)=O)C1 N1(C(c2ncc(C)cn2)=O)CC(C)N(C(=O)CCc2csc(=N)[nH]2)CC1C c1(C(=O)NCC(CC)NC(c2cccc3ccoc23)=O)ccc2c(C)noc2c1 C1(F)(C(=O)NC(C2CN(C(C=CC)=O)C2)C)CCCCC1 C1(NC(=O)COc2cccc(F)c2)CC2CC(NC(c3cccnc3O)=O)C1C2 n1(CCC=O)ccnc1C(C)C.CCCCNC(=O)CCN.[SH](=O)(=O)CC C=C1CCC(C(=O)N)CC1.c1ccc(C(N)=O)cn1.C1(F)CN(C(=O)C)C1.C C(=O)CC(CN(C)C)C(F)(F)F.N1(C(C)=O)CCN(C(=O)C)CC1.C#CCO C1(N(C(C(C)OC2CCCCC2)=O)C)CCCN(C(c2cc(C3CC3)[nH]n2)=O)C1 N1(CCC)CC(C(=O)N(CC)C)CC1=O.C1CCCN(C(=O)Cc2cnc[nH]2)C1 c1(C(N2C(C)CCC(NC(C3(CC)CCC3)=O)C2)=O)cc2n(n1)CCCC2=O c1(C[SH](=O)=O)ccccc1.C(C)(CC)NC(C1(CCC)CC1)=O.C(=O)C CC(C)(O)CCN(c1ccccc1)CC1CCC1 C(C(C)(C)C(=O)N1CSCC1C(=O)NCCCc1nncn1C)N(C)C N1(C(c2ccnc(C)n2)=O)CCC2CC2(NC(c2cncnc2)=O)CC1 C1(NC(C2(OC)CCC(C)C2)=O)COC2(C1)CN(C(=O)CCC1CCOCC1)C2 c1(NC(COC(C)C)=O)cc(N(CC(C)(C)C)C)ncn1 c1(OC)cc(N)c(C(N2C3CCC2C(C)C3)=O)cc1F.c1(CC(=O)N)cccs1 C1(CNC(C#CC(=O)N(C)C)=O)CC(C)(C)CCC1NC(=O)CCCCCS c1(C(=O)NCCCCN(C(=O)CCc2cccs2)C)cc(C2(C)CC2)n[nH]1 c1(C(CNC(=O)CO)NC(CC=C(C)C)=O)ccc(F)cc1.C1CCCOC1 c1(C(N2C(CC)CN(C(=O)CCN(C)CC)CC2)=O)cccc2ncsc12 C1(C(C)NC(c2cnn(-c3cccnc3)c2)=O)CN(C(=O)C(C)(C)CF)CCO1 C1(CNC(c2n(CC)cnn2)=O)CCC(C)CC1.n1(CC(=O)N)ncnn1 C1(c2ccccc2)(NC(=O)C=CCO)CCN(C(=O)C(O)C2CCCC2)C1 Cc1cc(C(N2CCC(O)(CCNC(c3nocc3Cl)=O)C2)=O)c(O)nn1 c1(N(C)C(C2CC(=O)CN2C(c2ccc[nH]2)=O)=O)cccc(F)c1F N1(C(Cn2c(C)cc(=O)cc2)=O)CCC2CCN(C(c3cnccn3)=O)C2C1 C(=O)(C1=CC2(CCOCC2)C1)NCC1C(NC(=O)Cc2c[nH]nc2O)CC1 c1(C=O)cc(C#N)c(O)nc1N.C1(CC)CCCCC1C(=O)NCC1CC1.N C(=O)(CCCCNC(=O)CC1CCN(C)C1=O)NCC(C)N(C)C c1(C(=O)NC2CCCN(C(C(C)(C)c3ncco3)=O)C2)ccnc2ccnn12 c1(OC)ccc2c(NC(=O)NCCCc3cncc(F)c3)ccnc2c1 C1(C(=O)NCc2c(C(=O)NC(CCC=C)C3CC3)scc2)CCC(C)CC1 N1(C(CCOC)=O)CCC(CO)(CNC(=O)CNS(=O)(=O)N(C)C)C1 C(=O)(C(C)(C)C(C)(F)F)N1CC(C(C)C)N(C(=O)C(O)Cn2cncn2)CC1 N1(C(c2cccnc2)C(=O)NCC(=C)C)CC2CC3CC2C1C3OCC C1(C=O)CCN(C)S1(=O)=O.n1(C(C)C(=O)NCCCO)cnc(C#N)n1.CC C1(C(N(C(CC#C)C)C)=O)(NC(c2conc2CC)=O)CCOCC1 N1(C(CCC=C)=O)CCCN(C(=O)CN(S(=O)(=O)c2ccccc2)C)CC1C N1(C(CCOCC#C)=O)CC2CC(NC(c3cc(C(F)F)[nH]n3)=O)C(C2)C1 CC1(C)CC=CCN(C(C2C(C3CC3)CCN2C(=O)C=Cc2nccs2)=O)C1 C1(NC(CN(CCC)C(C2CCCN2CC)=O)=O)CC12CCCC2 N1(C(C2CCCN(C(CCCCN(C)C)=O)CC2)=O)CCC(C)(O)C(O)C1 c1(NC(c2nc(-c3c(OC)cccc3)sc2)=O)ccc(Br)c(F)c1F C(=O)(CCC1=CCCCC1)N(CCCCCCNC(C=CC(=O)OCC)=O)C CC1CCN(C(=O)CC(C)(F)F)CC1NC(C1(c2ccccn2)CC1)=O N1(C(C2(CC)CC2)=O)CC2(CC(CC(N3CC(c4nncn4C)C3)=O)C2)C1.CO C1(NC(c2n(CCOC)nnn2)(CC)C2CC2)CC2(CCC2)C12CCC2 CCCC(CCC)NC(C1CCC(C2CC2)N1C(=O)CC(=O)OC)=O C1(OC)CC(NC(c2n[nH]cc2[N+](=O)[O-])=O)CN(C(C2CC(C3CC3)=NO2)=O)C1 C1(CCC)CN(C(c2cc(=O)c(O)c[nH]2)=O)CCN1C(=O)C(C)c1cccs1 O=S(=O)(c1c[nH]ccc1=NCc1c[nH]nc1-c1cccs1)N1CCCCC1 C1(CN(S(C)(=O)=O)C)CCCN(C(=O)NC)C1.C1CCCN(C(N)=O)C1 N1(C(C(c2ccc(C)o2)C)=O)CCCC(N(C)C(C2CCCC(C)(C)C2)=O)CC1 C(=O)(C1=CC(O)CC1)N(c1cccc(C)c1)CC.C1(C=O)C2CN(C)CC12.N C(CN=C(NCc1cccc(N2CC=CC2)c1)NC(C)C)OCC(=C)C N#Cc1n[nH]c(=NC2(CNC(=O)CCn3cc(Cl)cn3)CCCCC2)s1 CC1OC2(CO)CC1(C(=O)N(C1CCN(C(=O)CCCC(F)F)C1)C)C2 CC1CC(C)CN(C(=O)NC(c2ccc(C#N)cc2)c2ccc(Cl)cc2)C1 N1(C(c2n[nH]cc2Cl)=O)CC2CCC1CN2C1CCc2c(Cl)cccc21 N1(c2nnc(-c3cc(C)sc3C)o2)CCC(C)N(C(=O)OC(C)(C)C)CC1 CCCCCC(F)C(=O)NC1CCC(C(=O)NCC(O)CC2CCC2)C1 N1(C(C(CCC)NC(C)=O)=O)CC2CCC(C1)C2CNC(C1CCSCC1)=O C(CNC(c1csnc1C)=O)(CC(F)(F)F)NC(c1ccc(CC)nc1)=O c1(C(=O)NC23CC(C(=O)NCC(=O)N)(C2)C3)ccc(O)nc1.C1CC1 C1(O)(C(=O)NC2C(CNC(c3ccc(C(C)=O)[nH]3)=O)COC2)CCCCCC1 N1(C(C(C2(O)CCC2)NC(c2nccc(C#C)c2)=O)=O)CCC(C=C)(CO)CC1 C1(C(C)NC(c2cncnc2)=O)C2CN(C(c3nn(C)nc3Br)=O)CC12 N1(C(C2(CC)CCCC2)=O)CCCC(O)(CCNC(=O)CC(C)C2CCCC2)C1 C(=O)(CCC(CC)CCC)NCC1CCCN(C(C(CC)=CC)=O)C1 C1(N(CC(C)C)C(=O)Cc2ccoc2)CCN(C(=O)COc2cccnc2)C1 N1(C(C(=O)C2CC2)=O)CCCC2(CC(C(=O)N3CCCOC(CO)C3)=NO2)C1 C1(C(C)C)CCN(C(=O)CCc2cn[nH]c2)C(CNC(C2CC(CF)C2)=O)C1 N1(C(C(C)CF)=O)CCC2(CCCN2C(c2cncs2)=O)C1 N1(C(c2ccc(C(CC)C)cc2)C(=O)Nc2ccccc2)CCCC2(CC2)C1 C1(CNC(c2cn(CCOC)nn2)=O)(O)CCN(C(=O)CC(C)(C)O)CC1 c1(C(N(C(c2cc(Cl)c(Br)[nH]2)=O)C2CC2)=O)ccn2c1CCCC2 N#Cc1ccc(C(=O)NCC(O)CC(=O)NCc2csnn2)cc1 C(CCCC(C)(C)C(=O)NNC(=O)C(CC)C(F)(F)F)NC(C1C(C#C)C1)=O c1(C(=O)NC2C(NC(=O)Cc3cc(Cl)ccc3O)C2)n[nH]c2c1CCCC2 C1(NC(CCOC2CCN(C)CC2)=O)CCN(C(=O)CC2OCCO2)CC(O)C1 c1(C(=O)NC2CC(C)(NC(=O)COC3CCC3)C2)ccccc1.C(CF)O C#Cc1ccc(C(N2CCC(N(C)C(C3CC3C)=O)C3(CC3)C2)=O)cc1C CCCCCCCNC(N1CCC(CNC(c2nc(C)c(C)s2)=O)C1)=O N1(Cc2cccc(C(N)=O)c2)CCC(=O)N(CCCOC2CCCCCC2)C1=O C(=O)(CCCC(=O)OC)NCc1c(C(=O)NC2C(CCCC)CCC2)con1 N1(C(C(COCC)NC(=O)C(C)C(C)CNC)=O)CC(O)C(O)C12CCC2 Cc1cncc(C(N2CC(O)(C(C)NC(=O)CCC3CCCCN3C)C2)=O)n1 C(C(C)(C)C(=O)N(CCC(=O)NC1(C)CCCC1C)CC1CC1)SC c1(CC)nnc(CN(C2CC2)CC)o1.C12CCCC1C(=O)NC2=O Cc1cc(C(=O)N(C)CC2C3CN(C(C4(C)CCCS4)=O)CC23)sc1Cl Cc1cccc(F)c1CC(=O)NC1CCCC1NC(C1(C(C)C)CC1)=O c12ccccc1C(c1nnnn1CC(F)F)N2.C(C)C(C)(C)C.[SH](C)(=O)=O c1(C(=O)NCCC(C)NC(=O)C(F)(F)c2ccccc2)ccc(Cl)c(N)c1Cl N1(C(C(C(C)NC(=O)CCCCCN(C)C)C)=O)CCCC(C2(C)CC2)C1 N1(C(C(CC)=CC)=O)CC(C(=O)N(CC(C)C(=O)OC)C)C2(CCC2)C1 N1(C(CC(C)SC)=O)CC(NC(c2cccc(-c3nnco3)c2)=O)C(N=[N+]=[N-])C1 N1(C(C2C(C)CC(=O)N2)=O)CCn2nc(C)cc2C1.C(c1cccs1)=CC(=O)N C1(C)(C(=O)NCC2C(C(=O)NC(CC#C)CO)CCO2)CCCC1O CC1CCC(Cl)=C(C(=O)NC(C)(C)CC)C1.C1(CC=O)COC2(CCC2)CO1.N c1(CC)nc(C)c(C(=O)N(CC(C)NC(=O)CCC2CC2(Cl)Cl)CC)s1 C1(COC)(NC(=O)CCNS(C)(=O)=O)CCN(c2ccnc(C)n2)CC1 N1(C(C(C)NC(N)=O)=O)CCCC(C2CC2)C1.C1(CC=O)CC2C=CC1CC2.N CC1(c2cn(C3CCC(C(=O)NCCCN4CCOC4=O)C3)nn2)CCOCC1 C1(CNC(CCSC)=O)CCN(C(c2cccc(C(C)C)c2N)=O)CC1C C1(C(=O)NC2CCN(C(C3OCCC3C(F)(F)F)=O)CC2)CCC2(CCC2)CO1 N1(C(c2cc(C)nn2C2CCC2)=O)CCCC(C2(NC(=O)C3=CCCS3)CC2)C1 N1(C(c2n[nH]c(C)c2Cl)=O)CC2CCCCC2(NC(=O)C(c2cnn(C)c2)=O)C1 c1(N2C3C(NC(C(=O)NC(C)C)=O)CC(CC3)C2)ncc([N+](=O)[O-])cc1F CC1(NC(C2(CC(F)F)CCC2)=O)CCN(c2nc(C3CC3)ns2)C1 C(C(CC(=O)NCCc1ccncn1)NC(c1cc[nH]c1C)=O)OC c1(C(=O)OCC)ccc(NC(C)CCNC(c2cc(O)ccc2F)=O)nc1C Cc1c(C(=O)NC2CC(C)C2(C)C)oc2c(F)cccc12.c1(C(=O)N)cc[nH]c1 CCCCN=C(NCC1CCCS(=O)(=O)C1)NCC(CC)Oc1ccccc1 Cc1cc(-c2ccc(C(N3CCOC(C)(C)C3)=O)cc2)c(C)n1-c1cnn(C)c1 CCC(CCC(=O)N1CC2CC1(C(=O)NC)C2)NC(=O)CCC1CC1(F)F N(C1CCCn2cnnc21)C(=O)Cn1ccsc1=O.n1(CCCNC)ccnn1 C1(CCNC(C2(C(C)(C)OC)CC2)=O)CCCN(C(=O)CCCC#N)C1 C1(CNC(CC(CCC)O)=O)CN(C(=O)CC2CCC(=O)NC2=O)CCC1(F)F N1(C(COC(CC)C)=O)CCC(CC(=O)NCCCCC(C)C)C1(C)C Cc1ccc(C(N2CC3C(CNC(=O)Cc4cnsc4)C3C2)=O)cc1[N+](=O)[O-] Cc1ncc(C=CC(=O)N(CCCCN(c2nccnc2F)C)C)s1 N1(C(C(C(=O)OCC)F)=O)CC2CCC1CN2C(=O)C(C)=C(C)CC CC(C)(CS(N)(=O)=O)C(=O)N1CCC(NC(=O)CC2CC2)C(CO)CC1 N1(C(CC=CC)=O)CC(CO)C2(CCN(C(C3CC(C)(C)OC3(C)C)=O)CC2)C1 C1(C)(CC=O)CCS(=O)(=O)N1.N1(C(c2cscn2)=O)CC2CC2C1.CC.N c1(C(CO)NC(=O)NCC2C(C)(C)COC2)ccc(F)c(Br)c1 c1(C(=O)NCC2CCCN(c3nc(C#N)c(Cl)s3)C2)cccc2nc(O)oc12 c1(C(=O)NC(CN(C(C2CC(=C3CCC3)C2)=O)CC)C)ccsn1 c1(C(=O)NCCCCNC(c2c(CC)scn2)=O)ccc(C2CC2(F)F)cc1 N1(C(c2nccc(CC)c2)=O)C(C(=O)Nc2cncc(Cl)c2)CCC12CC2 c1(CNC(=NCCC#C)NCC2CCCNC2=O)cccc2ncccc12 n1(CC)nc(C(N2CCC(N(C(=O)Cc3c[nH]nc3O)C)C2)=O)cc1C1CC1 N1(C(CCOCCOC)=O)CCC(C(C)C(=O)NCC2CC2Cl)C1 C1(C(=O)Nc2cc(C)no2)CC(F)(F)CN1C(c1cnon1)=O c1(CC=O)cc(C)c(Br)c(C)c1.N1(C(C(OC)OC)=O)CC(C)C(C)(C)C1 c1(C(=O)OC)ccnc(NC(C2CC2NCc2cnccc2OC)=O)c1 CC1CC(CNC(=O)CCc2ncccn2)CN(C(c2cc(C#N)c[nH]2)=O)C1 N1(C(c2cc(CC)cc(F)c2)=O)CCN(C(=O)CCCC(C)CC)CC12CCC2 N1(C(C(=O)Nc2ccc(OC)c(OC)c2C)=O)CCC(C2(O)CCOC2)CC1 Cc1cc(C#N)nc(N2CC(NC(c3cc(C4CCCN4C)[nH]n3)=O)C(C)C2)n1 N12CCC(F)(F)C(C1)C2=O.S(=O)(=O)(c1cccs1)N.c1(OC(C)C)ccccn1 N1(C(CC(CC)C(C)C)=O)CC2CCCC(C1)N2C(c1ccnc(OC(C)=O)n1)=O CC(C)CC(C)CNC(c1cc(C(C)(F)F)ccn1)=O.c1(C(=O)N)ccoc1Cl N1(C(c2c(C)cc[nH]2)=O)CC(NC(C2(C(F)F)CCOCC2)=O)CC(C)(C)C1 c1(CCC(=O)NCC(n2cc(C(C)(C)O)nn2)C)cc2ccccc2o1 N1(C(C(C)C(C)O)=O)CCC2(CC(NC(=O)CS(C)(=O)=O)C2)C1 c1(OC)cc(F)c(NC(C2CN(C(c3cccnc3F)=O)CCO2)=O)cc1F C#CCC(O)C(=O)NC(C1CCCN1C(=O)Cc1nnn(C(C)(C)C)n1)C C1(CNC(C2(F)CCOC2)=O)CCN(C(=O)CCCc2nccs2)C1 N1(C(c2ncn(C)n2)=O)CCCC(O)(C(=O)Nc2cnn(CC3CC3)c2)C1 C(C)(C)(CC(=O)N(CC(C)C(=O)NCCc1cn(C)cn1)C)OC Cc1cn2cc(C(=O)NC3CCN(C(=O)COc4cc(C)on4)C3)cc(C)c2n1 S(=O)(=O)(c1ccsc1C(=O)NC1CC1)NC.C12(C(=O)N)CC(C)C1C2 C=C(C)CC(=O)N(CCN(C)C(C1COC(C)C1)=O)C(C)C c1(OC)ccc(C(O)C(=O)NC2CCC(NC(=O)C(C)C3CCCO3)CC2)cc1 c1(C(=O)NCCCN(C(=O)CCOCC(F)F)C)cnc(-c2nccs2)nc1O C1(CC(F)F)CN(c2cc(N3CC=CC3)ncn2)CCO1 C(CC(C(=O)N1CC(C)(NC(C2(COC)CCOCC2)=O)C1)OC)OC C1(C(=O)NC(c2c(C)nns2)C)CC12CCN(CC(=O)NC(C)(C)C)C2 Cc1cc(C)c(C(=O)NCC2CCCCC2)c(O)c1.CC(F)(F)F.C(=O)C.C N1(C(CCSCCCC)=O)CCCC(CNC(=O)C(N2CCC(C)C2)=O)C1 C1(CC)CN(C(=O)Cc2cccnc2O)CCC1CNC(c1[nH]nnc1C)=O N1(C(C(C=C=C)C)=O)CCN(C(c2cc(C3CC3)ccn2)=O)CC1CF C1(Cl)(C(=O)NCCCN(C(C2CC(=C)C2)=O)C(C)C)CC1(F)F C(N=c1[nH]c(=NC2CCC3CC2CO3)[nH]c2c1CSC2)c1c(C)nn(C)c1 C(CCC(O)C(=O)NCCn1nncc1C)NC(C1CC(=C)C1)=O C(c1cnc[nH]1)=C(C)C(=O)N1CC(CCCCNC(=O)C(n2nccc2C)C)C1 CCC(C)(C)C(C(=O)NCC1CN(C(=O)Cc2cccc(Cl)c2)CC1O)OC.O CCC(C)C(=O)C(=O)N1CCC(O)C1C(=O)NCc1ccc(OC)cc1 N#CCCCCCC(=O)NCCOCCNC(=O)CCCC1CCC1 CCCCC(CC)C(C(=O)NCC(F)F)N1CCC(O)(CN(C)C)CC1 C(=O)(C(=O)C(C)C)N(CC(=O)N(CC#C)CCOC)C1CC1 c1(C(C)C)ccc(C(N2CC(CNC(c3cnccn3)=O)C(C)C2)=O)nc1 N1(C(C2(n3nc(C)oc3=O)CC2)=O)CCCN(C(N)=O)CC1c1ccccc1 c1(-c2nc(C3S(=O)(=O)CC3)nn2CCN2CCOCC2)cn2ccnc2s1 C12(C(N3CC(C#C)C(O)C3)=O)CCN(C(c3ccnc(C)c3)=O)CCC1C2 C1(NC(c2c(CCC)nco2)=O)CCCCC1NC(=O)C(C(C)O)N(C)C Cc1[nH]c(=N)nc(O)c1CC(=O)NC(C)C(C)(C)C.C1(C=O)CC2CC2C1.N n1(CCCN(CC(=O)NOCc2ccccc2)C(C2C(C)C2)=O)cc(CN)nn1 C(=O)(CC(C)(C)C(F)F)NC1CC(C)(NC(=O)CN2C(=O)CCC2=O)C1 c1(OC)ccc(S(=O)(=O)NC2(C)COC2)cc1.c1(C(=O)N)cc(=O)cco1 C1(CCC(=O)NCC(CNC(CSCC)=O)C)CNC(=O)N1 C(C(C)C(=O)NC1COCC1C(=O)N(CC(c1nn[nH]n1)C)C)OC c1(N(C)C)ccc(C(N2CC=CC2C(=O)NC(c2cccc(Cl)c2)CO)=O)cc1 c1ccc(OC2COC(C3CCC3)C2)cc1.c12nnc(o1)CO2 C(=O)(C1=CCCC(C)(C)C1)NCC(CC)NC(C1CCOCC12CCC2)=O Cc1nc(Cl)ncc1NC(C1CN(C(C2(C)CNC(=O)N2)=O)CC(C)O1)=O c1(CNC2CCCC(C(=O)NCC3CN(C)C3)C2)cccc2ccoc12 Cc1nc(C)c(CNC(=NCC2CC2)NCC(C)(C)CC#N)o1 c1(C2C(C(N(CCC)C(C)C)=O)C2)ccccc1Cl.Cc1conc1C(=O)N c1(NC(C2C(C)N(C(=O)CN3CC4CC4C3)CC2)=O)cc(O)cc(F)c1 C1(C(N(C(CCCC)C)C)=O)CC(O)(C2CCNCC2)C1 C1(NC(C2CCC=CCC2)=O)COC2(C1)CN(C(C13CC1COC31CCC1)=O)C2 c1(C(N(CC(C)NC(C2CCOC2C2CC2)=O)C)=O)c[nH]nc1-c1ccccc1 C1(C)(CNC(C(C)OCCOCC)=O)CCC1C.C(C)(C)C.C=O C1(C(=O)NCCc2cncc(C)n2)CCCCCC1NC(=O)CC(=O)N(C)C N1(C(c2n(C)cc(Br)n2)C(=O)Nc2ccccc2)CCCC2(CC1)CNC(=O)C2 N1(C(COC2CCCC(C)C2)=O)CCN(C(=O)CC(C)(C)C#N)CC2(CC2)C1 c1(N2CC(CCCCNC(Cn3nc(C)oc3=O)=O)C2)ncc(Br)cc1C#N c1(C(N2CC3C(NC(C(CC)CC)=O)(C3)C2)=O)cc(-n2cnnn2)cc(Br)c1 C1(C(=O)NC2(CCCNC(C3C(C)C3)=O)CC2)Cc2nccnc2C1 Cc1ccc(C(=O)C(C)OC(C2CC(c3nn[nH]n3)(N(C)C)C2)=O)cc1F C1(CNC(C=CC=CCC)=O)CN(C(c2sccc2SC)=O)CCC1(F)F C1(C2CCCN2C(=O)C)CC2(C1)CC1(CC1)C2.c1(C2(C)CC2)cc(C=O)[nH]n1 C(C(COC)C(=O)NC(COC)C(=O)NCC(C)C#N)OC Cc1nc(C)c(C(=O)NCC2CCCCC2NC(c2cnn(C)c2C)=O)s1 C1(N(C(=O)C)CC)CCCN(C(=O)CS(=O)(=O)CC)CC1.c1ccc(C)cc1.S C1(CC#C)(C=O)CCN(C(=O)C=C(C)C(C)C)C1.C(C(N)=O)C1CC1.N N1(C(COC)=O)CC2C(CNC(c3cccc(C4CCCOC4)c3)=O)C2C1 CCCCCC(=O)N1CC2CC2(CNC(C2C=C(C)CS2)=O)C1 CCC(CO)(C(=O)NC1C=CC(CC(=O)N(C2CC=CC2)CCO)C1)OC c1(CNC(c2cn(C)nn2)=O)cc(O)nc(C)n1.c1(C=O)cn2ccnc2s1.N N1(C(C(C(C)C)OC)=O)CC2=C(C1)CN(C(=O)CC(c1ccc(F)cc1)C)C2 CC(CC(=O)N1C2CCC1C(C)C(NC(c1cnn(C)c1N)=O)C2)CC(F)(F)F Cc1nn(C)cc1CCC(=O)N(CC(F)F)Cc1ccc(C(=O)C(F)(F)F)cc1 C(=O)(C(F)C(CC)CC)N1C(CNC(C2CCC(CC)O2)=O)CCC1 CC1CN(C(C2(CC3CC3)CC2)=O)CCC1NC(C1CC(=O)N(C)C1)=O N1(C(C(CC#C)C)=O)CCN(C(=O)CN(C)C)C(c2cccc(F)c2)C1 c1(C(=O)NC2CCN(CCNC(C(CCC)OC)=O)CC2)ccn2nncc2c1 C1(O)CCN(C(=O)C)C1.CCC(C=O)NC(=O)OC(C)(C)C.CC(N)=O N1(C(C2C(C)OCC2)=O)CC2CC(NC(=O)Cc3cncnc3O)CC(C2)C1 c1(OC)cc(C(=O)NC(C(=O)N(CCO)CC2CC2)c2cccs2)ccn1 c1(OC)ccc(OC)c(Nc2cccc(CNC(N3CCN(C)CC3)=O)c2)n1 N1(Cc2cc(C)sc2)C2CCC1CN(C(c1cncc(OC)c1)=O)CC2 C1(CNC(C(C)(O)C2CC2)=O)COCCN(C(c2snnc2C2CC2)=O)C1 C1(NC(CN(CCC#C)C)=O)CCN(C(C2CC(C)CC(=O)N2)=O)CC1C c1(C(=O)NCC(CNC(=O)C(O)C2CC2)OC)cnn(CC(C)C)c1 CC1(CO)CC(O)CN1C(C1CCOCC1NC(=O)CC1CC2C=CC1C2)=O C1(NC(C2ON=C(C)C2)=O)CC12CCCCC2.c1(C=O)c(C)coc1C(C)C.N N1(C(C(C)n2cncn2)=O)CCN(C(=O)CN=S(C)(C)=O)CC1C1CCCC1 N1(C(c2c(CC)occ2C)=O)CC2CCCC(NC(c3ccncc3F)=O)C2C1 Cc1oc(C(N2CCCCC(CNC(=O)C)C2)=O)cc1S(C)(=O)=O.C1CC1.O c1(CN2CCN(CC(=O)NCCn3c(C)cc(C)n3)CC2)ncn2ccccc12 CC1COCCN(C(=O)NCC(C)Oc2cc(Cl)ccc2Cl)C1 CC1(C)COCC(C(N2CCCC2CNC(c2ccsc2Cl)=O)=O)O1 N1(C(c2cc(CC)c(C)s2)=O)CC(C)CN(C(c2n[nH]c(C3CC3)n2)=O)C(C)C1 N1(C(CCN(C)CCO)=O)CCCC(C)(C)C1CNC(=O)C(O)C(C)(C)C N1(C(C(CC)(C)O)=O)CCC(O)(CCNC(c2[nH]nc(OC)c2Cl)=O)CC1 C1(N(C(CC(C)c2ccco2)=O)CCO)CCCN(C(c2ccc[n+]([O-])c2)=O)C1 c1(C(=O)NCC2C(NC(c3nccc(C)n3)=O)CCC2)cc([N+](=O)[O-])sn1 C(C(C)(C)CNC(c1cnn(C)c1)=O)NC(C1C(C)(COC)C1)=O C1(C)(C(=O)N)C2CC3CC(C2)CC1C3.C#CCC(C)(C)C(=O)NCC(C)(O)C Cc1ccnc(C(=O)N(CCNC(=O)C(C)NS(C)(=O)=O)C(C)C)n1 c1(CN2CCCC(CC(N3CCCC(C(=O)O)C3)=O)C2)cc2ccncc2s1 C1(NC(c2cc(CC)[nH]n2)=O)CC2(C1)CC(NC(c1ccc(Cl)cn1)=O)C2 C(=O)(C(O)CC(F)F)NC1(C)CN(C(C2COC(=O)O2)=O)C1 CC(C)(C(=O)NCC1(O)CN(C(=O)C(C)(C)N2CCOCC2)C1)C1=CCSCC1 c1cccc(Cl)c1C(F)(F)F.C1(OCC)CCC(NC(=O)C(=O)NC)C1 c1(C(=O)NC23CC(C(=O)NC(C)CC(N)=O)(C2)C3)nccc2cc[nH]c12 n1(CCC(=O)N)ncn(C)c1=O.C1(C(=O)NC(C)CC)(COC)CCCC1 N1(C(C(=O)NCC(C(CC)C)C)=O)CCC2(Cc3ccccc3C2=O)C1 N1(C(c2cc(COC)on2)=O)CC2CCN(C(=O)Cn3cc(C)cn3)CC(C2)C1 c1(C(N2CCCC(NC(C3CCC(=O)N3)=O)(CO)C2)=O)cccc2c1OCC2 N1(C(CCCCCSC)=O)CC2CCCC(CNC(=O)C(C)(C)CCF)C2C1 C1(N(C)C)(C(=O)N(CCCn2cc(C3CCC(=O)CC3)nn2)CCF)CCCCC1 Cc1ccc(C)c(C(=O)NC2CCN(C(=O)CCNC(N)=O)CC2C)c1O CN1CCC(CCNC(=O)NC2CC2(C)C(F)F)C1=O c1(C(N2C(CNC(c3scc(C(N)=O)c3)=O)CCC2)=O)cccc(F)n1 C1(CNC(c2c(OC)ccs2)=O)CC2(CC(NC(C3OCCC3C)=O)C2)C1 c1(OCC(N2C(C3(NC(c4c(C)onc4)=O)CC3)CCC2)=O)ccccn1.C O=C(C1CCc2c[nH]nc21)N1CCN(C(C23CC4CC(CC(C4)O2)C3)=O)CC1 N1(C(C(COC)(F)F)=O)CCOCC1(C)c1cn(CCCCF)nn1 Cc1cccc(C)c1NC(=O)C(C)OC(c1ccccc1C1CCC1)=O N1(C(C(CCN(C)C)NC(=O)C=CC2CC2)=O)CC2CSCC(C2)C1 C1(NC(=O)C2=CCCC2)CC(F)(F)CC1NC(c1[nH]nnc1-c1ccccc1)=O c1(C(N2CC(C)C(C(=O)NOCCO)C2)=O)cnn2cccc2c1 C1(OC)CCN(CCC(=O)NC2CC2CN)CC1 C1(CC(=O)NCCC=CC)CCC(NC(c2cn(C3CC3)cn2)=O)C1 N1(C(C)=O)CCC(NC(=O)CC2CCCCNCC2)c2ccccc21 CC(C)(CCCNC(=O)COC1CCC1)NC(C1CCS1(=O)=O)=O c1(C(=O)NCc2ccc(C(=O)NC(C#C)C(C)C)cc2)cc(C)nc(C)c1 CC1(C)OCCC1NC(C1COCCC1NC(C1(C#N)CCC1)=O)=O Cc1cnn(C)c1C(N1CCCC(N(CCO)C(c2cc[nH]c(=N)c2)=O)C1)=O C1(C(N(CCNC(COCCCOC)=O)C2CC2)=O)CCCN1CC CN1CC(n2cc(CNC3CCCNCC3)nn2)CC1=O C1(C(=O)NC(C(C)SC)C)CC2CN(C(=O)C(C3CCOCC3)=O)CC2C1 c1(OC)cc(C)cc(C(N2CCC(C)(CC)C2)=O)c1C.C1(C(=O)N)CC12CCC2 N1(C(C(=Cc2ccncc2)C)=O)CCC(C2CN(C(=O)CN(C)C(N)=O)C2)CC1 C1(NC(CCOC(C)C)=O)CCN(C(=O)CC2CCCC(=O)N2)C1(C)C c1(NC(C2CCN(C(c3nccc(C)c3)=O)C2)=O)ccc(I)cc1C#N C1(C)(C(N2CC(CCC#C)C2)=O)CN(C(=O)CC(O)C(C)C)CC1C CC(C)C(C(=O)N1CC(Cn2cc(C3CC34CC4)nn2)C1)c1ccc(Cl)cc1 CC1CC(CNC(=NCCNS(C)(=O)=O)NCc2ccccc2)CC(C)O1.C N(C(=NCc1cn(C)nc1CC)NC1CCC1)C(C#C)COCC N1(CCC)CCCC1C(N1CCC1C(=O)NCCC1(O)CCC1)=O N1(C(C(C)(C)NC(C)=O)=O)CCCC2(CCCN2C(C2CCOC2)=O)CC1 c1(OC)ccc(CC#N)nc1.C12CCCCC1NC(=O)CN2 N1(C(C2C3CC(=O)CC32)=O)CCOC2CN(C(=O)C3=CC4(CCOC4)C3)CC12 C(=O)(C1=NOC(CNC(c2nc(C)sc2C)=O)C1)NCC1(SC)CC1 CCC(C)(CO)C(=O)NCC1(F)CC(NC(c2ccnc(Br)c2N)=O)C1 N1(C(c2ccc(C(N)=O)o2)=O)CCC2CCN(C(=O)CC3COCCO3)CC2C1 n1(CCC)cc(CNC(=NCc2cccc(F)c2)NC(C2CCCO2)C)c(C)n1 N1(C(c2[nH]cc(CC)c2)=O)CCCC(O)(CNC(C2C=CC2C=O)=O)C1 c1(C(C(=O)NCCOC)N(C(C=C)C2CC2)C)ccc(OC)nc1C CCCCC(C)C(=O)NC(CC)(CC)CCNC(c1cc(OC)cc(F)c1)=O C1(OC)CC(C)N(C(=O)C(C)N(C)C)C1.C(=O)(C)N.C1CC1.C(C)=O Cc1ccc(C(N2C(C(=O)NCCN3CC=CC3)CC3CC23)=O)c(O)n1 C1(CCC)(NC(=O)C(O)C2CC2)CCN(C(=O)CCS)CC1.c1ccc(C)cc1 Cc1ccnc(-n2nc(CCC(C)C)nc2C(C2CCCC2)N(C)C)c1 CC12CCC(C(=O)NC3COCC3CNC(C3CCCC3)=O)(C1)OC2 Cc1nc(C)c(C(C)NC(=O)C(C2CC3(CCC3)C2)N)[nH]1 C1(C(C)(C)C)CC(C(=O)OCC(=O)NCC2(c3ccccc3)CCCCO2)=NO1 C1(CC(=O)OCC)CCN(C(C2CC3CC3N2)=O)CC1.c1cc(C2CC2)[nH]n1 n1(CC=O)nc2n(c1=O)CCCC2.C(C(O)C(=O)NCC1CC1)=CC.C C(C(F)C=O)NC(=O)OC(C)(C)C.C1CCN(C(=O)C=C2CCC2)C1.N C(C(CC(F)(F)F)NC(=O)C(c1ccccc1Cl)(C)C)NC(C(C)C(F)F)=O C(=O)(C(C)(C)CC(=O)NC1CCCCN(C(c2ccc(C)c(CO)c2)=O)C1)OC C1(NC(C(CCC)=CCC)=O)CC2CCC1C2.C1(CC=O)CCC1.C1CC1.N c1(CNC(c2n(CCCSC)nnn2)(C)CCSC)cccc(Br)c1C C1(N(C(CNS(CC)(=O)=O)=O)C(C)C)CN(C(=O)CC2CCCO2)CC1O c1(C(N2CCC(N(C(C3CCC(=O)N3)=O)CC)C2)=O)cc(O)cc(O)c1 C1(C)(C(N(C(C)CO)C2CC2)=O)CCN(C(=O)CCC2CCC2)C1 C(=O)(C1=CCN(C(=O)C(C2CCCCC2)F)CC1)N(CCCCCC)C C(=O)(C1=CC2(CCOC2)C1)N1C(CC(=O)N(CC(C)(C)C2CCCO2)C)CC1 N1(COCC)C(=O)CCC1C=O.c1cccnc1.C1CC1C=O.C1CC1 N1(C(C)C(N2CCCCC2)=O)CCCC(C(c2ccccc2)N2CCCCC2)C1 c1(CC)cc(NC(c2ccc(NC(C)C)cc2C(=O)NC)=O)cc(C)c1 N1(C(CC(=C)C)=O)CCC2(CCN(C(c3ccc([N+](=O)[O-])cn3)=O)C2)C1 N1(C(C(C(C)(C)C)c2cccc(C)c2)=O)Cc2cnc(C)nc2C1 c1c[nH]nc1.C=C1C(C(=O)NC)C1C=O.C12CC1CNC2=O.C CN1CCC2(CCN(Cc3ccc(-c4ccc(Cl)cc4)o3)CC2)C1 C1(C(N2CCCC(N(C(=O)Cc3cn(C)cn3)C)CC2)=O)CN2CCCN1CC2 c1(C(=O)NC(COCC)C(=O)NCCN2CCCC2=O)ccnc(O)c1 C(=O)(CCC(=O)NCCC(O)CNC(=O)C(C)Sc1ccccc1)NCC n1(CC)cnc2[nH]c(=NC(C)CNC(=O)N(C)C)[nH]c(=NC(C)CCCO)c12 c1(OC)cc(O)ncc1C(=O)NC1CCCC(NC(c2cc(C)ccc2Cl)=O)C1 C(CCN=C(NCC(c1ccncc1)C)N1CCC(NC(N)=O)C1)OCC Cc1ccc2sc(C(=O)NC3CN(C(c4cccc(=S)n4O)=O)CC3C)cc2c1 C1(NC(CC(C(C)(F)F)(C)C)=O)CCS(=O)(=O)C12CN(C(=O)C=CCO)C2 Cc1cc(N)c(C(=O)NC(C)CCNC(c2cnc(C(F)F)s2)=O)cc1F N1(C(c2c(C#N)cccc2)=O)CC2CCCN(C(=O)CCc3ccon3)C2C1 c1(C(N(C2CCCCN(C(=O)CCC3CC3(F)F)C2)C)=O)cnn2c1CCCC2 C(=O)(C(C1(C)CC1)NC(=O)C(F)C1CC1)NCCCN(C)C C1(CNC(c2cncnc2)=O)CCCN1C(C1OCCO1)=O N1(C(C)C)CC(N=c2nc(N3CCOC(CCO)C3)c3c(ncn3C)[nH]2)C1 C(=O)(C(C)S(N)(=O)=O)N(CCOCCCN(C(C(C)(C)SC)=O)C)C C1(c2nnnn2C2CCOCC2)(NC2C(CC)C2)CCCC(n2cc(Cl)cn2)C1 C1(N(C)C(C2CCC3(CC3)C2)=O)CN(C(=O)Cc2cnoc2)CC12CC2 Cc1cccc(CONC(=O)CC2CC2CNC(=O)Cc2cnoc2)n1 C1(NC(=O)CCn2cncn2)CC2CN(C(=O)CCn3ccnc3)CC12 C1(C(=O)NCC2N(CCOC)CCC2)C2CCC(C2)C1(C)C C1(CC=C)(NC(c2ccn(C)n2)=O)CN(C(=O)CC(C)c2ccco2)C1 C(CN=C(NCC(c1cccc(Cl)c1)CO)NC1CCOC(C)(C)C1)OC C1(C(C)C)N(C(=O)C2=CC3CCCC23)CC12CCN(C(c1cn[nH]c1)=O)CC2 N1(C(C(CSC)C)=O)CC(C)CN(C(c2n[nH]cc2C(F)(F)F)=O)C(C)C1 c1(N(C2CN(CC(N)=O)C2)C(=O)Cn2cccn2)ccc(F)cc1 CC1CN(C(=O)C(C)(C)Cc2cnn[nH]2)CC(C)N(C(=O)CC(F)F)C1 C1(C(=O)N(C)CC2(C)CC2)(OC)CC(C)(C)C1.C1(C=O)CCCCS1.N CC1CCC(C)(C(=O)NCC(C)(C)NC(c2ccc(-c3ccncc3)s2)=O)C1 C1(C(C)=O)CCCC(CC(=O)NCC2CSCCN2C(=O)C=Cc2cn[nH]c2)C1 N1(C(C(c2ccc(F)cc2)Oc2ccccc2)=O)CC=CC(NC(=O)CCF)C1 O=S(=O)(c1ccc(N2CCOC3(CCSC3)C2)nc1)NC1CCC(CCO)CC1 c1(CN2C(c3ccc(C)o3)CCCCC2)cc2cnccc2o1 c1(C(N(C)CC2(O)CN(C(COCC(=C)C)=O)C2)=O)ccc2c[nH]nc2c1 C12(CNC(C3N(CCC)CCC3)=O)CCCC1N(C(c1cc(C)nn1C)=O)CC2 C=C(C)CC(C(=O)NCC(C)C1CCC1)NC(C1COC(=O)N1)=O c1(C(=O)N)cnc([N+](=O)[O-])cc1C.c1(SC)cc(C)c(C(=O)N(C(C)C)C)o1 CC1C(NC(c2cncs2)=O)CC2CCC1N2C(C1(C)CC(=O)C1)=O C1(C(N2CC(CC(C)NC(=O)CCc3ccon3)C2)=O)CCCCC1(C)C C1CN(C(=O)CC2(N(C(=O)C=CC)C)CC2)C1.N1CCC1.CCCNC Cc1nc2cc(C(=O)NC3CCN(Cc4cnc(Cl)s4)C(C)C3)ccc2n1C N1(C(=O)OC(C)(C)C)CCC(C(=O)NNC(=O)OCC(F)C2CC2)CC1 N1(C(c2cc(C)ncc2)=O)CCN(C(c2cccc(F)c2Cl)=O)CC(C)(F)C1 Cc1sc2ncnc(N(C)CCN(C)C(c3ccnc4[nH]ncc34)=O)c2c1C c1(C(=O)NCCN(C)C(c2cc3ccsc3n2C)=O)ccc2[nH]c(=N)[nH]c2c1 C1(CNC(c2cnc(CC(C)C)[nH]2)=O)C2CN(C(C3CC(CF)C3)=O)CC12 c1(CNC(C=CC=CCC)=O)nc(C)c(C(=O)N(CC(O)C)C)o1.O N1(C(Cn2c(C)nc(C)n2)=O)CCCCC(CNC(c2csc(CO)n2)=O)CC1 C1(C(N2CCCC(O)(C(=O)OC(C)(C)C)C2)=O)CCC2(CCOCC2)O1 C1(NC(CC(C)CF)=O)CCC(C)N(C(c2cccc(-n3ccnc3O)c2)=O)C1 C1(O)(CCNC(C(Cc2ncn(C)c2)O)=O)CCN(C(=O)C=C2CCSCC2)C1 C1CC2(C1)CS(=O)(=O)C2.Cc1nc(F)ccc1C(N1CCCC(CC(=O)N)C1)=O O=C(CCCCO)NCC1CC(CNC(c2cccc(-n3cncn3)c2)=O)CO1 Cn1nc(C(=O)NCC2(C(N)=O)CN(C(=O)CC(C)(C)C#N)C2)c(Cl)c1Cl C(=O)(CCCCC(F)(F)F)NCC1CN(C(c2c(C)cco2)=O)CC12CC2 c1(-c2cc(C(=O)NCCOCC=C)c3c(c2)[nH]cc3)cc2c(C#N)cccc2[nH]1 N1(C(CCC2C(=O)NC(=O)N2)=O)CCC(N=c2[nH]c3ccccc3s2)CC1 c1(C(C)NC(c2n[nH]c(-c3ccccc3)c2Br)=O)cc(Cc2nn[nH]n2)nn1C C(=O)C(F)(F)c1nccs1.C1(C)(COC)CC1C(N1CC(CCC)C1)=O.N N1(C(=O)CCc2ccon2)CC2CCN(C(c3cncc4sccc34)=O)CC2C1 c1(C(C)NC(C2CC(=O)C2)=O)sccc1C#N C(=O)(C1=CCC(C)CC1)N.C1(C(=O)NCc2cn(C(C)C)nn2)CCC(O)C1 N1(C(=O)OC(C)(C)C)CC(C(=O)N)CCC12CCC2.N1(CC)CCC12CC(O)C2 c1(OC)ccc2c(c1)CCC2C(=O)NC(C)CCCCNC(=O)Cc1cc[nH]n1 C1(NC(C(C)c2ncco2)=O)CCSC12CN(C(c1ccccc1)=O)C2 CCCCC(CC)C(=O)NC(CNC(=O)Cc1cnn2c1CCCC2)CCCC C1(CO)CCCCN(C(=O)CC2(NC(C(CC#C)C3CC3)=O)CCCCC2)C1 C1(C)(CC)CCCN(C(C2CN(C(C3CC=CC3)=O)CC23CC3)=O)C1 C(=O)(C(CNC(=O)C(Cl)Cl)CC1CC1)NC(C)CO C1(C(C)NC(C2C3CCCC23)=O)CCN(C(=O)CC2(N(C)C)CC2)CC1 c1(C(=O)NC2(C3N(C(COC)=O)CCCC3)CC2)cc2c(nn1)CCC2 CC#CCCCC(=O)NCCC1(O)CCN(C(C2CC(=C3CCC3)C2)=O)CC1 N1(CC(=O)NCC(CCNC(CC2C(C)CC2)=O)O)C(=O)CNC1=O N1(C(=O)NC2CCSCC2)CCCC2CN(C(=O)CCCC(F)(F)F)CCC12 c1(CC)cc(C(=O)NCCCC2(C)CCCC2)cc(O)n1.C(=O)C(O)C(C)C c1(CCC)cc(N(C2CCN(C(c3cccnc3Cl)=O)CC2)C)nc(Cl)n1 C(=O)(CC1=CCN(C(=O)C(C)Cn2cccn2)CC1)NCC(COC)(F)F CCCC(CC(=O)NCc1cccc(OC)n1)NC(C1CCCC1CC)=O c1(C(N2C(C(CC)C)CCC2)=O)cc(CNC(c2ccncc2)=O)ccn1 NC(=O)CCCC(=O)NCC1CN(C(c2ocnc2C(F)F)=O)CC1O c1(C(N2CCC(CNC(c3ccn(CC)n3)=O)C2)=O)oc2c(F)cccc2c1C Cc1ncc(C(=O)NCC=CC(N2CCC(N3CCCC3)C2)=O)cn1 Cc1ccnc2c(C(N3CC(NC(C4CC(=O)N4)=O)CC4(CCC4)C3)=O)cnn12 N1(C(C2C(C)C2C)=O)CCC(O)C(NC(c2c[nH]nc2I)=O)C1 C1(C(=O)NC(Cc2ccccc2)CO)CC2(C1)CN(Cc1cc(Cl)ncc1Br)C2 c1(CC)c(C=O)cnn1C(C)(C)C.C1C(C)CCN1C(=O)CC.C(C)=O.N c1(C(=O)N)c[nH]c2ccncc12.CC1CC(C)CN(C(C2(P(C)(C)=O)CC2)=O)C1 C(=O)(CCCC(=O)NCCC1CCN(C(=O)CSc2ccc(Cl)cc2)C1)N(C)C CCC(C)CCC(=O)N1CCC(CNC(c2cscn2)=O)(COC)C1 C1(C(=O)NC)(OCC)CCOCC1.C1C2CN(C(c3n[nH]c(C)c3C)=O)CC12 c1(C(=O)NC(CNC(c2c(CC)con2)=O)CC)cc(C)c(F)cc1N C12CCCC1CN(C(=O)C=Cc1ccccc1)C2.CC1(C)CC2(CC2C(=O)N)C1 C=C(C)C(C)(O)C(=O)NC12CC1CN(C(=O)CNS(=O)(=O)N(C)C)C2 C1(CNC(CCOC(C)=O)=O)CCC(C)N(C(c2nn(C)nc2Br)=O)C1 c1(-c2nnc(COC(C(C(C)C)F)=O)o2)c(F)cccc1F C1(NC(C(C(CC)CC)F)=O)CN(C(=O)CCn2ccnn2)C2(CCOC2)C1 C1(CC(=O)NCC(C)NC(c2cscc2Cl)=O)CCS(=O)(=O)C1 N1(C(CCOCCC)=O)CCSCC1CCNC(C1CC2(CCC2)C1)=O C(C(CNC(C1CCCOC1)=O)C(F)(F)F)NC(c1c(C)nc(C)o1)=O C(=O)(C1=C(C)CCCC1(C)C)NCC1N(C(C(CC)NCC)=O)C2C(C1)C2.C c1(COC2CCN(CC(c3cccc(I)c3)=O)CC2)ccc(F)cc1F C12(CNC(CNC(CC)=O)=O)CCC(CN(C(c3cncn3C)=O)C1)C2 C1(C(N2CC3(CC(NC(c4ccc[n+]([O-])c4)=O)C3)C2)=O)COC2(CCC2)CO1 C12(C(=O)NCCCC)CCN(C1)S(=O)(=O)C2.c1ccccc1.C(=O)CNC N1(C(c2c(CC)noc2)=O)CCN(C)CC1C.C(=O)C(F)(F)F.C(=O)C.N c1(CSC)cc(C(=O)NC2CN(C(c3nccnc3N)=O)CC2F)sc1C C1(N(C(=O)C(F)C2CCC2)C)CCCC2CN(C(=O)Cc3csnn3)CC12 c1(C(C)C)nc(NCc2cc3n(n2)CCC3)cc(N2CCCC(CO)C2)n1 Cc1cc(CNC(C2C=CCN(C(=O)C(c3ccn(C)c3)C)C2)=O)n(C)n1 Cc1ccc(C)c(C=O)c1.c1(C(N(C(C)C2CC2)C)=O)cc(CC(C)C)on1.N c1(C=O)cc(C)c2[nH]nnc2c1.C1(C(=O)N(CC(C)C)C)(OCC)CCOC1.N CC(C)(C(=O)N1CC(O)(CCNC(=O)CC2CCNC2=O)C1)c1cscc1Cl N1(C(c2c(SC)cn(C)n2)=O)CCN(C(=O)CS)C(C(F)F)C1.c1nncn1C N1(C(c2c(C)ccs2)=O)CC2CC(NC(=O)Cc3cccc(F)c3F)C(C2)C1 C1(C(=O)NCCC2CCOC2(C)C)(CC)CCN(C(C2COCCO2)=O)CC1 CN1CCC(CC(=O)NCC2(F)CC(NC(C3(C)CCC3)=O)C2)CC1 c1(C(=O)NCCC2N(C(C(C)C3CCC3)=O)CCSC2)ccc2c(c1F)CCC2 c1(C(C)C)cc(C(=O)NC2CC(C)(NC(=O)C(C)CF)C2)cc(F)c1 c1(C(CC(=O)OC)NC2CCC2C)ccc(Cl)cc1.C(C)(C)C.C=O.N C(=O)(C1=C(C)OCCS1)N1CCCC(N(C(COCCCC#C)=O)CC)C1 c1(C(=O)NC2CN(C(CCC)=O)CC2c2nccn2C)ccc2c(n1)NCC2 N1(C(C)=O)CCOC(CC(=O)N(CC(O)CNC(=O)C=CC(C)(C)C)C)C1 c1(C(=O)O)cc(C(N2CCCC2)=O)n(C)n1.C(=O)C(O)CN1CCCC1.CC C(=O)(N=c1cc(C)n(C2CC2)[nH]1)C1C2CN(C(C(CC=C)C(C)C)=O)CC21 O=C(Nn1cccn1)C(F)C1CCN(C(=O)CC2CC(F)(F)C2)C1 C1(SC)CN(C(c2ncc[nH]c2=O)=O)CC1NC(=O)C(C)n1cncn1 c1(C(=O)NCC(CNC(C2(O)CC2)=O)OC)ccc(C(=O)CF)cc1 N#Cc1ccc(NC2CC(F)(CNC(c3cccc(C(F)F)c3)=O)C2)cn1 c1(C(=O)NCC(C2CCOC2)NC(=O)CCc2ncc[nH]2)cscc1C1CC1 CCCC(CCCNC(c1cc(C)oc1C)=O)NC(c1cc(C)ccc1F)=O C(CCC(F)F)N(C(C)C(=O)N)C(=O)Cc1cnn(C)c1.C(=O)C1CC1 CCC(F)(F)CC(=O)N1CC2(CCN2C(C2CC(C)(C(C)(C)C)C2)=O)C1 C(c1ccncc1)=CC=O.C(C(C)(CO)NC(=O)CNC(=O)C)OC.N C(C)(C(C)(C)C(=O)NCCC(C)C(C)(C)C)NC(C(C)=NOCC#N)=O CC#CCC(C(=O)NC(c1ncc(C)o1)C)NC(=O)C(=O)NCC C1(CC=C)(NC(=O)COC2COC2)CN(C(=O)C(C)(C)n2cccn2)C1 N1(C(COCC=C)=O)C2CCC1C(CNC(c1cc3scnc3[nH]1)=O)C2 N1(C(C(C)SCCCC)=O)CCCC1C(C)(C)CNC(=O)CCN1CCC1 c1(SC)cccc(F)c1C(=O)NCC1C2CN(C(C3CC(O)C3)=O)CC12 c1(C(=O)NCC2CN(C(CCCOCCC)=O)CC2C)ccc(C)cc1O C12(C(=O)NCCN3CCN(C(=O)CSc4ccccc4F)CC3)CCC(CC1)C2 Cn1nc(C(N2CC(OCCNC(=O)Cc3ccc(F)cc3F)C2)=O)ccc1=O C1(CNC(C2CCC=CO2)=O)CC2(CCN(C(=O)C3=CCSC3)CC2)CO1 n1(CC(N2C(CC)C(NC(=O)C(C)C(F)F)CC2)=O)ncc(=O)c2ccccc12 c1(NC(=O)NC(C#C)CC2CCOC2)ccc(C2(OC(C)=O)CCC2)cn1 c1(C(=O)Nc2scc(-c3ccc(OC)cc3CO)n2)nc(O)c2nc[nH]c2n1 c1(COC)ccc(C(=O)N(CC(=O)N(C)C(C)C2CC2)C(C)C)o1 c1(C(=O)NCCCCN(C(C2CC(CC)OCC2)=O)C)ccc(C)c(C)c1Cl C1(C)(CC)NC(=O)N(CC=O)C1=O.C(=O)CC(C)C(F)F.C1CC2(C1)CC2.N c1(-c2ccc(CC)nc2)cnc(OC)c(C(=O)NCC(c2ccccc2)O)c1 N1(C(CC(C)C)=O)CC(O)(C2CCN(C(C3CC3C)=O)CC2)C1 C#Cc1ccc(C(=O)NCc2ncccc2C(=O)NN2C(CC)CCC2)cn1 CN1CCC(C)(C(N2CCN(C(c3nc(Cl)sc3Cl)=O)C(CCO)C2)=O)C1=O C#Cc1ccc(NC(C2CC(O)CN2C(=O)C(c2ccccc2)O)=O)c(C)c1 N1(C(CCc2n(C)ccc2)=O)CC(C2CCCCN(C(=O)CCC3CC3)C2)C1 N1(C(c2ccn(CC)n2)=O)CCN(C(c2ccc(F)cn2)=O)C(C(F)F)C1 C(=O)(CC(Cc1cccs1)NC(c1ccccc1)c1cncs1)NCC(F)F CN1CCC(C(=O)NC2CN(C(C3CC(O)C3)=O)C2)C1 S(=O)(=O)(c1cccc(Cl)c1)NC(C)C=O.C1C2CN(C(=O)CC)CC12.C1CC1 c1(C(N2CCC(C)(NC(C(CCSC)O)=O)C2)=O)ccc2[nH]nc(O)c2c1 N1(C(=O)NCCc2noc3ccccc23)CCc2nnc(O)cc2C1 C1(C(=O)NC)(OC)CCS(=O)(=O)C1.C(=O)CCCn1cccn1.C1CCC1 C1(CC(=O)NCC(CC2CC2)CO)C2CCCC2N1C(C1(F)CC=CCC1)=O C1(NC(c2c(OC)nc(C)cc2)=O)CC2CCC1CN(C(=O)C(C)(C)C(F)F)C2 CN1CCC(CO)(CNC(c2ccncc2)=O)C1.C1(C=O)C2CC(=O)CC12.C N1(C(c2cccc(OC)c2)C(=O)NC2(c3ccccc3)CC2)CCN(C)C(C)C1 C1(C(=O)OCC)CCCN(C=O)C1.C1(CC=O)CCCCC1.C1(=O)CO1.N c1(C(N(CCCN(C)C)CC)=O)nn(C)c(Cl)c1Cl.c1ccc(C=O)[nH]1.CC C(=O)(C(O)C(F)(F)F)NCC(C)(O)CNC(=O)C(c1ccccc1F)(F)F Nc1cc(F)ccc1C(=O)NC1COCCC1NC(=O)Cc1cccnc1 N1(C(C)=O)CC=C(c2cnc3c(C(=O)NC(C)(C)C)c[nH]c3c2)CC1 C1(C(C(=O)NC(C)CN(C)C(C2CCCC2)=O)F)CCCCCC1 C12(NC(C3CC(C)C3)=O)CCC(C)(C1)OC2.c1(C=O)ccnn1C(C)C.N c1(C(N2CCC(N(CC#C)C(C3CN(C(C)C)C3)=O)C2)=O)cnccc1C C=CC1(C(=O)NCC2C3CCCCCC23)CCN(C(=O)C=C(C)CCC)C1 C1(C(N2CCC(C(C(=O)NC(C(C)SC)C)(C)C)C2)=O)CC2CCCC2C1 C1(C(=O)NC(c2cn(C)nn2)C(N2C(C(=O)OC)CC2)=O)COCCC1C C1(NC(c2cnc3n2CCC3)=O)CC12CCN(C(c1scnc1Cl)=O)C2 C12(C(=O)NC(CCNC(C(COC)OC)=O)C)CC3CC1C2C3(F)F Cc1ccc(OC(C)C(=O)Nc2ccc(N3CCCCCC3)nc2)c(Br)c1 N1(C(c2c(CNC(COCCOC)=O)n[nH]c2)=O)CCCC2CCCC12 c1(C(=O)NCCCCN(C(=O)CN(C2CCCC2)C)C)cnc2cnccc2c1 CON(Cc1ccc(Cl)cc1)C(=O)NCc1nccc(C(F)F)n1 C(=O)(C(C)(O)C1CCOCC1)NCCC(C)NC(CNC(=O)NC)=O C1(NC(C(CC)O)=O)CN(C(C2(OC(C)=O)CC2)=O)CCC12CCOCC2 C1(C(NOCC(CC)C)=O)CC2(CCC2)CN1C(C1CC(O)C1)=O c1(OC)cccc(O)c1C(N1CCC(N(C)C(c2sccc2F)=O)CC1)=O c1(CNC(=O)NC2CCN(CC3CC3)C2)cncc(-n2ccnc2)n1 Cc1ncc2c(n1)CCCC2N=c1nc(N2CCCC2)c2c(ncn2C(C)C)[nH]1 C(=O)(CS(=O)(=O)C1CC1)N(C1CCN(C(CCc2cc(C)no2)=O)CC1C)C N1(C(C(N2CCN(C)CC2)C)=O)CCC(CO)C(NC(=O)Cn2ncnn2)C1 c1(C(=O)NC2CCC(O)CN(C(=O)C3=NOCC3)C2)cc2nn[nH]c2cc1F CC1CN(C(c2cccnc2S)=O)CC(C)CN1C(=O)C=Cc1ncco1 CC1COCCC1N(C(=O)CC1CCN1C(=O)CC(O)C1CCCC1)C C1COCCN1C(=O)CCc1cccc(OC(F)F)n1.C(=O)(CC1CC1)N(C)C C1(C(=O)NOCC)(OC)CN(C(c2conc2C2CC2)=O)C1.c1ccccc1.O n1(CC(=O)NCCCC)ccc(C(F)F)n1.c1(C=O)ccc(-c2ccco2)o1.N Cc1ccc(CCC(=O)N(CC(C)(C)NC(c2cc(O)nn2C)=O)C)cc1 N1(C(CN2C(C)CCC2C)=O)CCC2(CCN(C(=O)C#CC3CCC3)CC2)C1 Cc1cc(C(=O)NCC(C)CN(C)C(c2coc(C(F)F)n2)=O)ccc1Cl N1(c2nccc(OCC)n2)CC2CC(NC(=O)CCC=C(C)C)C2C1 N1(C(C(C2CCCCC2)C)=O)CCC(NC(c2ccn(C)c(=O)c2)=O)C(C)(C)C1 N1(C(C=CC(C)NC(CCCOC(C)=O)=O)=O)CCC=C(F)C1 c1cccc(C)c1.CCC(C(=O)N(CC(C)O)CCNC(=O)CCC)N(C)C.O O=C(CCCCn1ccnn1)NCCn1cc(C2CCOC2)nn1 C1(CNC(CCC2N(C)CCC2)=O)COCCN(C(=O)CC2(C#N)CC2)C1 C(=O)(C1CCCc2sccc21)NCCC(C)(C)NC(CCCCCC(C)O)=O c1(C(=O)NCC(CNC(CCNC(COC)=O)=O)CO)cc(F)cnc1O c1(C(N2CCN(C(c3c(CC)n[nH]c3)=O)C(C)C2)=O)cc(C)cc(Cl)c1N CCCCC(CNC(=O)CC1(C)CC1)NC(=O)CC1COCCN1CC Nc1nn2ccccc2c1C(N1CCN(C(c2ccoc2Br)=O)CC(O)C1)=O N#Cc1ccc([N+](=O)[O-])cc1S(=O)(=O)N1C2COCC1CC(O)C2 C(N=c1[nH]c2c(c(=NC3CCC(P(C)(C)=O)C3)[nH]1)CCC2)c1nccc(C)n1 O=C(CC(O)C1CCCC1)NC1CC(O)C1CC(=O)NCCCN1CCOC1=O N1(C(C(CC)(C)CC)=O)CCC2CCC(C1)N2C(c1cc(Cl)cs1)=O C1(NC(c2ccnc(OC)n2)=O)CC2CCC(C1F)N2C(=O)C(C)n1ccnc1 CC(C)CC(C)CC(C)(c1nnnn1CCC1(C)CC1)NCCCCS(C)(=O)=O N#Cc1ccc(CCC(=O)NCC=CCNC(C2(O)CC2)=O)c(F)c1 CC1(C)CC1(C#N)C(N1CCC(N2CCN(C(C34CC(CO3)C4)=O)CC2)CC1)=O C=CCC(CC(=O)N(CC(O)(CC)CC)C)NC(=O)COCCCF Cc1ccccc1CC(C)C(=O)NC1(C)CCN(CC2CCS(=O)(=O)C2)C1 c1(CC)c(Cl)nc[nH]c1=NCC1CC(NC(=O)C(c2cnn(C)c2)O)C1 C1(C(=O)Nc2ncc(C)cc2Br)CC2CCCCC2N1C(C1CC1F)=O CC(CCC(=O)NC(CNC(=O)CCN1CCCCC1)C1CC1)N(C)C c1(NC(=O)NCCCc2nc(-c3ccncc3)no2)cc(Cl)ncn1 c1(OC)ccccc1C(C(=O)N1CC(OCC)C1)OC.C(=O)(C(C)(C)CO)N C1(CC)(NC(=O)CN(C)CCO)CCN(C(=O)CCc2nc(C)no2)CC1 c1(OC2CN(C(CNS(CC)(=O)=O)=O)C2)ccccc1 c1(C(N2C(C(C)NC(C(C)OCC)=O)CCC2)=O)cc(C)c(Cl)c(N)c1 c1(NC(C2C=CCN(C(CN(C(C(C)C)=O)C)=O)C2)=O)ccc2c(c1)COC2 c1(C(=O)NC2CC(NC(C3CC(C)OC3)=O)C2)n[nH]c2c1CN(C)CC2 c1(OC)cccc(F)c1CNc1nc(-c2ccc(CC#N)cc2)cs1 c1(CC)ccc(C(=O)NC2CCN(C(c3cnn(C)c3SC)=O)CC2)c(N)c1 C1(CC(=O)NCCC2CCCN2C(=O)CCSC(F)(F)F)Cc2ccccc2O1 N1(C(c2cnccc2Cl)=O)CCC2CCN(C(c3ccc([N+](=O)[O-])cn3)=O)C2C1 C1(CNC(C=C(CC)CC)=O)CN(C(=O)CCC(C)C#N)C2(CCC2)C1 CN1CCN(C)C(C(=O)NCCC(C)(C)NC(=O)CCCC2CCCO2)C1 c1(CCC)n[nH]c(=NCCC2(OC)CN(C(=O)CC(C)C3CC3)C2)s1 N1(CC(N2C(CN(C(c3cnn[nH]3)=O)CC)CCC2)=O)CCC(O)CC1 C1(F)(C(=O)N)CCOC1C.c1(SC)ccc(C(=O)NCc2csc(C)n2)o1 C1(C)(C(N2CC(F)C2)=O)C(C)(C)C1(C)C.c1(OC)csc(C(=O)N)c1.C N1(C(C(C2CC2)OCC)=O)CC=CC(NC(=O)C=CC(N)=O)C1 C(=O)(CCC(=O)NCC1(C)CCCC1)N(C)C.C1(Cl)(C(=O)N)CC12CCC2 n1(COC)nccc1C(N1CC(CN)C1)=O.C(=O)CC1CC1C(F)(F)F C1(C(N2CC3CC(C2)N3C(=O)CCC2CCCC2)=O)CCC2CCC(=O)N2C1 C#CCCC(C(=O)N1CCC(CC2CCC2)C1)NC(c1ccsc1Cl)=O N1(C(CNS(CC)(=O)=O)=O)CCN(C(C2(C)CC2(Cl)Cl)=O)CC1COC c1(CC)nonc1C(=O)NC1CC(C(C)NC(c2csc(C)c2)=O)C1 C(C(CC(C)C)C(=O)NC(c1ccn(C)n1)(C)C)NC(c1cc(C)c(C)s1)=O c1(CC)nc(CN(c2ccccc2)CCC(O)c2cccs2)cs1 c1(C(=O)NC(CN(C(c2nn(C)cc2Cl)=O)CC)C)cc(=O)c2ccncc2o1 N#Cc1ncccc1-c1ccccc1-c1nccn1CCC12CC(C1)C2 C(=O)(C(C)(C)CC(=O)NCCCC(C)NC(C1(OC)CCC1)=O)OC c1(C(=O)NC2CC(C(=O)Nc3ccc(CO)cc3)CC2O)ccc2cc[nH]c2n1 c1(C(N)=O)cc(F)ccc1NCC1CC1c1csnn1 N1(C(c2scnc2C(F)F)=O)CCCN(C(=O)CCc2cnn[nH]2)CC1 C1(CCNC(C(c2ccco2)NC(C2CC(OC)C2)=O)=O)CCCC2CC12 c1(C(CC(=O)N(C)CCc2cccs2)C(=O)Cc2ccccc2)ccccc1F CCC(C)C(CC(=O)NCC1(O)CCN(C)C1)NC(C1CC(C(C)C)C1)=O N1(C(C(C)CC2CCC2)=O)CCC(NC(=O)COC2CCC2)C1C1CC1 c1(NCCC)cccc(C(N2CC3CC2C3CNC(=O)C(C)(C)CC)=O)c1 n1(CCC)cc(Cl)c(C(=O)NCC=CC(C)C)n1 c1(CNC2C(C(=O)NC(CC(C)C)c3ccccc3)C2)cccc(C=O)c1Br C12(C(=O)NC(c3cn(C)nc3)C(=O)NCC3(Cl)CCC3)CCC(CC1=O)C2 CCCCCC(C)CC(=O)N1CCCCC1CN(C(=O)CCCC(=O)NCC)C c1(C=O)cc([N+](=O)[O-])ccc1.C1(CC(=O)N(C(C)C)CC)CN(C)C1.N Cc1cc(C(=O)NC2(C(N3CCC(n4ccnc4)C3)=O)CCCC2C)cc(F)c1 CN1CCn2nc(C(N3CC(O)CC3CNC(=O)Cc3ccnn3C)=O)cc2C1 C1(CC(=O)O)(C(=O)OC)CCCN(C(=O)C(N)=O)C1 n1(CC)cnc2c(N(C)Cc3c[nH]nc3C)[nH]c(=NCC(C)(C)C(F)(F)F)nc12 c1(C(=O)NCCCNC(Cn2nc(C)c(Cl)c2C)=O)cnc2cccnc2c1 N1(CC)CCOC(CNC(c2occc2C)=O)C1.C1(CC=O)CCN(C)C1 c1(C(=O)NCC(=O)OCC)ccc2c(c1)CN(C(=O)Cn1cccn1)CC2 S(=O)(=O)(c1ccc(NC(C)CC(C)(C)OC)nc1)NCCCCCOC c1(C(=O)NC2CCN(Cc3nnc(C(C)(C)C)o3)C2)cccc(F)c1F N1(C(c2c[nH]c(=NC)o2)=O)CCc2sccc2C1CNC(=O)CC1=CCCC1 n1(-c2n(C)ncc2)nc(C2COc3ccccc32)nc1CCC1CCCOC1 CCCC(C(C)(C)C)NC(C1CCC2(CC2)N1C(=O)C(CO)OC)=O N1(C(CN2CC(C)C2)=O)CC=CC1CNC(C12CCC1C2)=O C1(C)(COC)CN(C(=O)CNC(=O)CNC(c2cn(C)cn2)=O)C1 C1CC12CCN(C(C1CC1C(N)=O)=O)CC2.n1(CC(C)C)ccc(C(=O)N)n1 C(=O)(C1=C2CCCN=C2NN1)N1CC(CNC(CC(CC)CC)=O)CC12CCC2 c1(C(c2onc(C3(C)CC3)n2)NC(C2CCCO2)=O)ccc(F)cc1 c1(C2(C(=O)NCC3CN(C(C(CC)(C)C)=O)CC3O)CCC2)c(F)cccc1Cl C1(C=O)CC2CC1CN(C(=O)CC1CCCC(=O)N1)C2.C=C(C)COCC.N CC(CC1CCCCC1)C(=O)N(CC(C)(C)NC(=O)CC(C)F)C C1(CNC(C(=O)N(C)CCO)=O)CSc2ccccc2O1 c1(CC)cc(N)c(C(=O)NCC(C)NC(=O)C(C2CCC2)OC)c(F)c1 c1(OC)ccc2nc1NCC(=O)N1CCC(C1)O2.C1(OC(C)=O)CCOC1 O=C(CC(F)(F)C(F)F)NC12CCC(C(N3CC(OC(F)F)C3)=O)(CC1)C2 N(C1c2ccccc2CC1NC(C1CCCC1O)=O)C(CCCCC(=O)NC)=O c1(CC(=O)NC2CC(C(=O)Nc3c(C#N)cccc3)C2)ccc2c(c1)CCCO2 Cc1c(Br)csc1S(=O)(=O)N1CCC2(CCCC2)CC1 C12(NC(c3cccc(C)c3F)=O)CCOCC1CN(C(c1ccc(O)nn1)=O)C2 Cn1cnc(-c2ccc(F)cc2)c1NC(=O)C=CC(F)(F)F C1(C(c2n(CC(=C)C)nnn2)(C)NCc2ccns2)CCCCCC1.C(C)(C)O C1(NC(C2CC(CCNC(C(CCC)F)=O)C2)=O)CCC2(CCC2)C1 C(=O)(CC(O)CCSC)NCCC1CN(C(c2cn(CC)nc2)=O)CC1C c1(OC)cccc2[nH]c(CN3CCCC(C)(C(=O)NC)C3)cc12.C1CNC(=O)C1 c1(CCC(=O)NCC2CN(C(COCC)=O)CC2C)ccc(Cl)cc1Cl N1(C(C(C)O)=O)C2CCC1CN(C(C1CCC1)=O)CC2 c1(C(C)(C)C)cc(N)ccc1C(=O)NC1C=CCC1.C(=O)C(O)C(F)(F)F.C c1(C(CC(=O)OC2(C(=O)OC)CCCC2)C)ccc(OC(F)(F)F)cc1 C(CC(O)(C(F)(F)F)c1nc2ccccc2o1)NCc1n(C)c(-c2ccccc2)nn1 C=Cc1ccc(C(N2CC3CCC3(OC)C2)C(=O)NCCC2(C)CC2)cc1 C(=O)(CC(F)(F)F)NCC(=O)N(C(C)C1CC1)C.C(=O)C1=CCCC1.N Cc1ccc(CC(=O)NCC2CC2CNC(c2cc(Br)co2)=O)s1 C1(CC)CN(C(C2(C)CC(C3CC3)=NO2)=O)CCS1(=O)=O.C(CC=O)=CC=C C1(C=O)CC2CCC(C1)C2O.C1(F)(CNC(C(CC)OC)=O)CCC(C)CC1.N C12(NC(CCCC(C)C)=O)CCCC1CN(C(c1cccc(OCCF)c1)=O)C2 C#CCC(C(=O)NCCSC)NC(=O)C(C)OC(C)(C)C Cc1nc(Cl)cc(=NCCC(C)(C)NC(C23CC4CC(C2)CC(C)(C4)C3)=O)[nH]1 CC1=C(C(=O)NC2CC(CNC(c3occc3C)=O)C2(C)C)CCS1(=O)=O c1(COC)cnc(NC(N2CCC2C2CCOC2)=O)cn1 C=CCCCC(C(=O)NC1CCCCCC1CO)NC(c1coc(SC)c1)=O C1(N(C(CCCSC)=O)C)CCN(C(C23COCC(C2)C3)=O)CC1 C1(NC(c2c(C)sc(-c3ccccc3)n2)=O)CC12CCS(=O)(=O)CC2 N1(C(c2ccc(-c3cn(C)nc3)o2)=O)CC2CC(NC(=O)C3=COCC3)CC1C2 Cc1cccc(Br)c1CNC(=O)CC1CCCC1NC(c1cc(=N)[nH][nH]1)=O CC1CN(C(C23CCC(C)(C2)OC3)=O)C(C)CN1C(c1cnc(O)c(F)c1)=O c1(C(N2CCCC2C(C)(C)C)=O)ccc(F)c(Cl)c1F.C1(OC)CC1C=O.N N1(C(CC(C)C)=O)CCCC(C)(C(=O)NC2CC3CCC2O3)C1 N(C(=NCC1CCOC1)NCC1CCN1C1CCCC1)C(C)COc1ccccc1F N1(CC)CCN(CC(=O)NC2(C)CCN(C(=O)C(C)Cn3cccn3)C2)CC1 C=CC1CN(C(C2(CC)CCCCO2)=O)CC1NC(=O)C(O)CCN(C)C C1(C)(CNC(c2cncc(C)n2)=O)CCCN(C(=O)CCc2ncc(C)[nH]2)C1 C1(C(=O)NCC2C3CN(C(C4CCCC4O)=O)CC23)SC2C=CC1CC2 c1(C(=O)NC(CNC(CCc2onc(C)n2)=O)CC(C)C)cc(O)cc(C#N)c1 N1(CCCCCNC(c2n(CC)cnn2)=O)CCN(C(C23CC(F)C2C3)=O)CC1 CCC(CCC(=O)N1CCN(C)CC1C(=O)NCCCOC)OC C1(CNCCCO)(CF)CCNC1 C1(C)(CNC(C2C(c3n(CC)cnn3)C2)=O)CCN(C(c2cn[nH]c2)=O)C1 N1(C(C(C)OC)=O)CCn2ncc(C(=O)NCCc3[nH]cnc3C)c2C1 c1(C(=O)NC(CNC(CCNC(C)=O)=O)C2CCC2)cccc2nc[nH]c12 C(CNC(=O)C(F)CC1CCOC1)(CCNC(=O)CCc1cnoc1)OC c1(C(=O)NC(CC=C)CNC(=O)CN(C)CCO)ccncc1.C(C)(=O)N c1(C(=O)NCCOC2CCN(C(C3CC(C)(C)OC3)=O)C2)ccc2n[nH]cc2c1 C(CCC(=O)N(CCC(=O)N1CC(CS(C)=O)C1)C)N(C)C N1(C(=O)NC2C(CC)CCC2)CCSCC12CCC2 N1(C(CCC(C)C)C)CCC2(CC1)CC2C(=O)NC(c1nc(CSC)on1)C c1(C(C(=O)NCC(CC)NC(=O)C(C)C(F)F)O)cccc(Br)c1 CC(C)(CF)C(=O)N1CCN(C2COCC2NC(=O)CNS(N)(=O)=O)CC1 Cc1nc2c(s1)CN(C(C1CC1NC(c1cc(F)c3cn[nH]c3c1)=O)=O)CC2 Cc1cc(C(C)C)ccc1NC(c1cc(C(C)(C)C)cnc1Cl)=O N1(C(C(CC2CN(C(C3C=CCCC3)=O)C2)F)=O)C2CCC1CC1(CC1)C2 c1(C(N2CC3(C(C(=O)NC(C)CF)C3)C2)=O)ccnc([N+](=O)[O-])c1 N1(C(=O)CCC2CCC2)CC2CC(C1)N(C(c1cc(Cl)on1)=O)C2 C1(CNC(Cc2cnc(C)o2)=O)CC2CCC(C1)N2C(=O)Cc1cnc(C)s1 C=CC1CC(N=c2[nH]c3c(c(=NCc4cnc(C)n4C)[nH]2)CC(C)CC3)C1 c1(C(C)C)nc2cccc(C(=O)NC3CCN(C(=O)CCC(F)F)CC3O)c2[nH]1 c1(N(C)C)ccc(C(=O)NC2CCCC2CNC(c2ccc(O)cn2)=O)cc1 CCCCCCC(CC)C(=O)N1CCC(NC(c2cnnn2C2CC2)=O)C1C CCCCS(=O)(=O)CC(=O)N1CC(C(C)NC(=O)C(c2ccc(CC)cc2)C)C1 c1(-c2n(-c3ccc(CC)cc3)nc(Cn3cncn3)n2)cc(C)c(C)cc1C C1(CNC(c2ccc(OC(C)C)nc2)=O)CC(C)(C)CN1C(=O)C(C)CCO Cc1ccc(C)c(C(=O)NCCC(C)N(C)C(C2CC(C)(C)CCO2)=O)n1 c1(COC)ccccc1NC(=O)COc1ccccc1-c1ccccc1 C1(NC(C2(COC)CC2)=O)C2CC1N(C(=O)Cn1cccnc1=O)C2C N1(c2ncc(C#C)cn2)C2CCC1C(C)C(NC(C1CCCO1)=O)C2 c1(C(N2CCC(CC(C)(C)C)C2)C(=O)N)cnc(C(C)(C)C)s1.C(CC)SC c1(C(=O)NCC(C(C)(C)C)NC(c2ccc[nH]2)=O)ccc2c(n1)NCC2 O(NC(=O)C(CC(C)C)NC(=O)C(CC)C1CCOCC1)CCOC C1(N(c2cc(C)cc(C)n2)S(=O)(=O)CCCN2CCC2)CCCC12CCNCC2 C1(C(N(CCCN(C)C(C2(CCOC)CC2)=O)C)=O)CC2CCC1C2 C(=O)(CCS(=O)(=O)C(F)(F)F)NCCCCN(C(C(C1CCOCC1)OC)=O)C C1(NC(C2CCC3(CCC3)O2)=O)CC2CC1N(C(c1cccc(=O)o1)=O)C2 C(=O)(CC(F)(F)c1ccccc1)NCC#CCNC(C(C)SC)=O c1(C(N2CCCCC(N(C(Cc3cnc(C)o3)=O)C)C2)=O)ccn2cnnc2c1 c1(C(=O)NCC2CCCC(NC(c3cc(Br)co3)=O)C2)cc2c[nH]cnc-2n1 C(=O)(C(O)(C(F)(F)F)C1CC1)NCCC(C)NC(c1c(C)cnnc1O)=O C1(NC(C(OCC)OCC)=O)CC2(C1)CC2C=O.C1(CC)CC1.N C(=O)(CC1=NNC(=O)C1)N(C)CCN(C(=O)Cc1csc(Cl)c1)C c1(C(N(CC)C2CC2)=O)ccc([N+](=O)[O-])cc1O.c1(C(=O)N)cc(Cl)cnn1 N1(C(C(c2ccccc2)C)=O)CCC(NC(=O)CC(C)N2CCCC2)C1 c1(OC)ccc(C(=O)N(C)CCOCCC)nc1.C1(C=O)C2CC2C2CC12.N N1(C(C(C)SC(C)C)=O)CC2CCC(C1)N2C(=O)CCn1cccnc1=O C(=O)(CC(F)(F)CC(=O)N(C(C)CCNC(=O)C(C)C(F)F)C)OC O=C(CCCCN1CCCC1)NC(C(=O)Nc1cnn(CCF)c1)=O c1(-c2cn(C3CC(NC(c4c(C)oc(Br)c4)=O)C3)nn2)cc2ccccc2[nH]1 C1(NC(Cc2ccc(C#C)cc2)=O)CN(C(C2CCCCO2)=O)CCC1(C)C c1(NC)cnccc1C(=O)N(CC(NC=C(C)C)=O)C Cc1nc(-c2ccccc2)oc1C(=O)NC1CC1CNC(=O)CC(C)(F)F c1(C(=O)NC(C(C)C)CNC(=O)C(O)c2ccsc2)ccc[n+]([O-])c1 N1(C(C2COC(=O)O2)=O)CC2=C(C1)CN(C(C1(c3ccccc3Cl)CCC1)=O)C2 C(C)(C)(C(C)CC(=O)NCCNS(N)(=O)=O)NC(C1C(C)N(C)CC1)=O N1(CCC(N2CCC(NC(C(C)(C)n3cccn3)=O)C2)=O)C(=O)C=CC1=O C1(CNC(C2C(C)OCCO2)=O)CC2(CCN(C(=O)Cc3ccn(C)n3)CC2)C1 C(c1cccc(C(F)(F)F)c1)=CC=O.C(C)(C=O)OC.C1(CC)CCCC1.N C12(C(=O)NCC3CC4(CC(NC(=O)C5=CCCCC5)C4)C3)CCOC1CCOC2 c1(C=O)c(F)cccc1Cl.c1(C(C(=O)NCCCC)=O)cn(C)nc1C(F)F.N c1(C(N2C3CC(NC(C4CCN(C(C)=O)C4)=O)(C3)C2)=O)cc(Br)ccc1N Cc1nn[nH]c1C(=O)NCC1(CCNC(=O)CC2CCC3CC23)CC1 C1(C(=O)NC(CCC)C2CC2)CC2CC1CN(C(C1(C(F)(F)F)CC1)=O)C2 C1(O)CCC(C)(C)C1.C(CC1CC1)(CC(=O)N)NC(CCCOCC)=O.C CC1NC(=O)C2=C1N(CCF)C(=O)NC2c1cc(C(C)(C)C)sc1C CCC(CC(=O)NCC1CCN1C(c1ccc(NCC2CCCO2)cc1)=O)S NS(=O)(=O)C1(C(=O)NCC2CCCCN2C(C2CCCC23CCC3)=O)CCCC1 C(N=c1cc[nH]c(=NCCCc2nc(=N)[nH][nH]2)[nH]1)C1(OC)CCC1 c1(C=O)cnc(Cl)c(F)c1N.C1(C(N(C)CC2(C)CC2)=O)CC(F)C1.N CC1(C)CC(O)(C=O)C1.C1CCCCN1CC(=O)N.c1ccc(C(N)=O)cc1.C C(=O)(CC(CC)CC(C)C)N(C(C)C(=O)NCCC(C)OC)CCC c1(NC(C)=O)ccc(S(=O)(=O)N2CCN(C(c3cc(C)cnc3N)=O)CC2)cc1 C1(NC(c2ccc(COC)s2)=O)CC2CCC1N(C(c1cc(OC)ncn1)=O)C2 N1(C(Cc2nc(NC(c3cc(C)cc(C)c3)=O)sc2)=O)CCCC(C)(O)CC1 c1(C(N2CCN(C(CNC(C(C=C)O)=O)=O)CC2)=O)cc2c(Br)cccc2cn1 c1(NC(C(c2ccccc2)OC)C)cc(Br)ccc1Cl C(CC(C(=O)N1CC(C)=C(C)C1)NC(=O)Cc1ccoc1)=CC c1(C(C#N)C(C2CC23CCCOC3)=O)ccc(F)c(C(F)(F)F)c1 n1(CC=C)c(N2CCCC2C2CCOC2)nnc1C1CCCN1CC(C)C C1(N(C(CSc2ccc(C)cc2)=O)C)CCCN(C(=O)C=C2CCN(C)C2)CC1 C(CCC(O)C(=O)N(C)Cc1cc(C)n(C)n1)NC(C=C=C(C)C)=O Cc1ccnnc1C(N1CCC(OCCNC(C2(C#N)CCOC2)=O)C1)=O N1(CC(=O)NC(C2CC2)C)OC(C)(C)CC1=O.C1(C=O)COC(=O)O1.C C1(CC(=O)OCC2CCCC(F)(F)C2)Sc2ccccc2NC1=O Cc1ccc(C(N2CCCCC2=O)Cc2nc(CCOC(C)(C)C)no2)cc1 N1(CCNC(C(C)N(C(C2CCC(CC)O2)=O)CC)=O)CCCCC1C c1(OC)cccc(CC(=O)NC(c2ccc(OC(F)(F)F)cc2)C)c1 CC1CC(NC(c2ccc(CC3CC3)cc2)=O)CN(C(c2cc(CO)[nH]n2)=O)C1 C1(N(C(CSCc2cccc(C)c2)=O)C)CCN(C(C2CC(O)C2)=O)CC12CC2 n1(CC#C)cnnc1C(=O)NCC1(OC)CN(C(c2ccsc2C)=O)C1 CC1=CCCN(C(C23CC(CN2C(=O)CCCN2CCCC2)C3)=O)C1 c12nc(Cl)c3ncn(c3n1)CC(=O)O2.c1(NC(C)=O)ccccc1OC1CCC1 Cc1cc(Cl)c(C(=O)NC(CCN(C)C(C2CCN(C)CC2)=O)C(C)C)cn1 C1(CC=C)(NC(c2cc(COC)[nH]n2)=O)CN(C(C2CC2(F)F)=O)C1.C C1(CNC(C(C)n2cnnn2)=O)CN(C(=O)CCc2ccn(C)c2)CCC1(C)C CC(C(=O)N(CCCNC(c1cnc[nH]1)=O)C1CC1)C(C)(C)C C(=O)(C1=CCC(C)(C)CC1)N.Cc1ccc(CNC(c2[nH]ccc2C)=O)nc1 c1(C(=O)NCC(C2CCOC2)O)cc(-c2cccs2)on1 N1(c2c3ncn(CC(c4cccc(C)c4C)=O)c3ncn2)CC2CCCN(C)C2C1 C(=O)(CCC(C)(C)[N+](=O)[O-])NCC(CC=C)NC(=O)C(=O)Nc1ncc[nH]1 c1(C=O)nc(O)nc(O)c1N.C1(N(C)C)(C(=O)NCC2CCC2)CCCCC1.N c1(N2CC3C(C(=O)Nc4c(C)c(Cl)ccc4)(CC3)C2)ccn2ncc(Br)c2n1 C12(NC(CC=CC(C)(C)C)=O)CCOCC1CN(C(=O)Cn1ccnn1)C2 C(=O)(C1=CC(C)(C)C1)NCCC(C)N(C(=O)CCCCc1ccc(F)cc1)C c1(OC)cc(C2CCN2C(=O)Nc2ccc(SC3CCCC3)cc2)ccc1F CC(CNC(C1(c2cc[nH]n2)CC1)=O)(CO)NC(c1n[nH]c(C2CC2)n1)=O C1(C=O)Cc2cc(F)ccc2O1.C(=O)(C(C)CC(=O)N1CC(OCC)C1)OC.N C1(CC(=O)NC(c2scc(C)n2)C)C2CCCC2N1C(C1C2COCC12)=O C1(CCC(=O)NC(C#C)(C)CC)CCCN(C(=O)C(CC2CCC2)OC)C1 Cc1ccc(Br)c(C(=O)NCC2CC2CNC(C2(C#N)CCCC2)=O)n1 N1(C(C2(OC)CCC2)=O)C2CCC1C(F)C(NC(=O)CS(=O)(=O)CC(C)C)C2 C1(O)(CC(=O)Nc2cc(O)ccc2F)CCN(C(c2c(F)cccc2Cl)=O)CC1 C=C(C)CC(C)C(=O)NC1CC(C)CN(C(c2conc2C)=O)C1 N1(CC(=O)N(CC(C)C)CC#C)CCN(C(C2CCCCC2OC)=O)CC1 c1(C(N2CCCC(c3nncs3)C2)C(=O)NCCC)ccc2ccc(Br)cc2c1 N1(C(CCC(C)CN(C)C)=O)Cc2n[nH]cc2C1C(=O)NCc1cn(C)cn1 N12CCC3C(CC13)NC2=O.C1(CSC)CCC(COC)CC1 C12(NC(c3c(OC)n(C)nc3)=O)CCOC(C1)C2.C(C(C)C)=CC=O.C N12CC3(CCCC3)C1C2.Cc1nc(Br)ccc1CNC(=O)OC(C)(C)C N1(C(C2(C)CCN(C)C2)=O)CCC2CN(C(c3cc4sccc4s3)=O)CC2C1 n1(CCC(=O)N(CC(C)NC(=O)C(C)(O)C(C)(C)C)C)ncc2c1CCCC2 Cc1c[nH]c(C)c1CCC(=O)NC1CC(C(N2CCOCC2)=O)C1 c1(C(=O)NCC2N(CC)CC(C)(C)C2)cc(S(N)(=O)=O)cc(F)c1Cl N1(C(CCNC)=O)CC2(CC2C(=O)NCCO)C1 C1(NC(C(C)(C)C(N)=O)=O)CCC(O)CN(C(=O)CCc2ccc(N)c(F)c2)C1 C1(NC(c2ccc(Cl)cc2)=O)CCN(C(=O)CCc2cocn2)CC12CCC2 C12(NC(C=CC(CC)=CC)=O)CCCC1N(C(=O)C#CC(C)(C)C)CCC2 c1(CC(=O)NC2C(NC(C(C(=C)C)(C)O)=O)CC2)ccc([N+](=O)[O-])cc1 C1(OC)CCC2(C(N3CC(C)(C)C3C3CCN(C(C)=O)CC3)=O)CCC12 C1(CNC(C2C(=C)C2)=O)CC(O)CN1C(C1CCN1S(C)(=O)=O)=O CCC(C(=O)NCC(C(C)C)NC(=O)CCc1nccn1C)Oc1ccccc1 C(N=c1cc(C)[nH]c(=NCc2cccc(-n3ccnc3)c2)[nH]1)C1C(CCC)C1 C#CCC(C(=O)N(C1CCCC1)CC#CC)NC(C1CCCC(CF)C1)=O C(C(C(F)(F)F)N1CCN(c2nncs2)CC1)NC(C(CC)n1cncn1)=O c1(CN(CC(=O)OC)C(=O)CC2CCCOC2)c[nH]nn1.C1CCC(=O)N1 C1(C(N2CCC(NC(C(N3CCNC3=O)C)=O)C2)=O)COCCC1(F)F C1(COC)(C)CCCN1C(=O)Cn1ncc(Cl)c1C.C(=O)(CC(F)(F)F)N C(=O)(CC(=O)N(CC(C)C(=O)N(CCOCCOC)CC)C)NCC c1(OC)c(C)cnc(CCNC(=O)C(=O)NCc2ccc3c[nH]nc3c2)c1C c1(C(=O)NCC(N2CCN(C(C3(C)CC=CCO3)=O)CC2)C)cc(=O)cc[nH]1 c1(C(C(=O)NCC(C)CN(C)C(C2CCS2(=O)=O)=O)O)ccnn1C Cc1cc(C(=O)NCc2ccc(C(=O)NC3CCC3C)s2)nnc1C C(=O)(C(O)CCC(F)(F)F)NC1(C)C(NC(c2c(CC)ccs2)=O)CCC1 C(C(C(C)(C)C)NC(C1CCC(C)(C)C1)=O)NC(C(C)Cc1ccco1)=O C(=O)(C(C)C(F)(F)F)N1C2CN(C2)CC(=O)N(C)CCC1.c1cccnc1.CC N(C(=NCc1ccco1)N1CCc2sc(Cl)cc2C1)C1CC(C)(OC)C1(C)C C1(N(C)C)CCN(CCC2CC2(C)C)CC1 C12(CC3CCCN(NC(C4(CC)COC4)=O)C3)CC3CC(CC(C3)C1)C2 c1(C(N(C2CN(C(C3CN(CC(F)(F)F)C3)=O)C2)C)=O)cnc(N)c(Cl)c1 c1(N2CC3(N(C(=O)C(Cl)=CCl)CCCC3)C2)ncnc2sc3ccccc3c12 C1(CC)CN(C(=O)CC2C=CS(=O)(=O)C2)CCN1C(=O)CCC1CC1.CO C1(C(N(CCOC)Cc2nn(C(C)C)cc2Cl)=O)CCc2nc[nH]c2C1 c1(C(=O)NC(C)CCCNC(=O)C=CCO)ccnc(OCC(F)(F)F)c1 C(C)(CNC(=O)C)(CO)NC(CC1CC(C)C1)=O.c1(C(=O)N)ccccn1 C#CCCN=C(NCCc1ccccc1Br)NC1CCSC1C C(CN=c1[nH]c2c(c(=NCCC3(C)CC3(Cl)Cl)[nH]1)COC2)OC(N(C)CC)=O C(=O)(C(C)(C)C(C)(C)C)N1C2CC(CNC(CCN(C)CC)=O)C1CC2 CCCC(CCCNC(c1cc(C(C)(C)C)no1)=O)NC(=O)CC(C)SC C(C(=O)NC(C)(C)C)(C1=NOC2CC12)N1CCC(O)(C(=O)OCC)C1 C1(NC(C2=C(C)OCC2)=O)CCCC12CN(C(=O)CCOc1ccccc1)C2 C1(C(=O)NCc2cc(N3CCN(C)CC3)ncc2)CC(=O)N(C)C1c1cccs1 CS(=O)(=O)CCC(=O)N1CCN(C(c2cccnc2)=O)CC1C1CC1 C1(C(=O)NC(C(=O)OC)C2CC2)CC2C=CC1N(C(=O)C(F)F)C2 Nc1cc(C(=O)NC2CC(CCn3cc(-c4cncc(F)c4)nn3)C2)cc(F)c1 N1(C(C(C=C)(C)CC)=O)CC2CC(NC(C34CCCCC3OCC4)=O)CC2C1 CCCCC(O)C(=O)NCC(C(C)C)NC(=O)CCc1ccc(O)nc1 N1(C(COC(C)=O)=O)CC(C(N2CC(F)(CO)C2)=O)C(F)(F)C1 C(=O)C(C)P(C)(C)=O.Cc1cc(C(=O)N)c(C(F)(F)F)o1.C1CCCCC1.C C1(CC(=O)NCc2c(C)ccnc2)C2CCC1CN(c1ncnc3occc13)C2 c1(C(c2nnnn2C2CCC(C(N)=O)C2)NCCOCCC=C)sncc1Br CC1CC(C(N2CC(NC(c3ccc[nH]3)=O)C2)=O)CC(C)C1 C1(CC(=O)NC(c2ccc(Br)cc2)C)CC(O)CN1CC1CCOCC1 N1(C(C2=CC(C)C2)=O)CCC(C2CC(NC(c3ocnc3C3CCC3)=O)C2)CC1 C1CCC2CN(C(C3(C(C)(C)O)CCC3)=O)CC12.C(CC(=O)NC)OC(C)C C(N=c1[nH]c(C)cc(=NC2CCN3CCCC23)[nH]1)c1c(OC)cc(F)cc1 CC1C(NC(c2ccc3nc(O)[nH]c3n2)=O)CC2CCC1N2C(=O)C(F)(F)CO Cc1ncc(CNC(c2ccn(-c3cccc(Br)c3)n2)=O)c(N(C)C)n1 C(CCN=C(NCc1ccco1)NC(c1ccc(Cl)cn1)C)SC C(=O)(CCCCCNC(N)=O)NCCCCC(C)NC(c1scc(C)c1)=O C1(Nc2snc(CCOC)n2)CCN(C(C2CCCC(=O)N2C)=O)CC1C C1(NC(C2CN(C(C)=O)C2)=O)CC2CC1N(C(C1CC3CCC1CC3)=O)C2 Cn1nccc1CCC(=O)NCC=CC.C1(C)(C=O)CC(C(F)(F)F)C1.N c1(C(=O)NC2CCNC2)ccccc1-c1ccccc1F Cc1ccc(C)c(C(N2CCCC2C2(O)CN(C(=O)C3=CCC3)C2)=O)c1 C1(C)(C(N(C(CC)C)C)=O)CC12CCN(C(c1ccc3nc(C)[nH]c3c1)=O)CC2 C(=O)(C(C)CCC(C)(C)C)NCC1N(C(C(c2cccc(C)c2)=O)=O)CCC1 c1(CC(c2ccccc2)C=C)nc(-c2cncc(F)c2)nn1CCCN(C)C C(C)(C)(CC(=O)N1CCSCC1C)N(C(c1c(C(C)C)n[nH]c1)=O)C C(=O)(C1=CCN(C)C1)N1C(CC(=O)NC)CC(O)C1.c1(C2CC2)cc[nH]n1.C C1(C(N2CC(C)(NC(C(C(=O)OC)C)=O)C2)=O)CCc2ncsc2C1 N(C(=NCc1ccco1)NCc1ccc(Cl)cc1)CCNC1C(C(F)(F)F)C1 c1(C(C2(C)CCCS2)NCc2ncn(C(C)C)c2)ccccc1F C(=O)(CCCC(F)F)NC(C)CNC(=O)Cc1cccc(F)c1 c1(CC=O)ccc(C(F)(F)F)cc1.CC1CCC(C(=O)N(CCC)C2CC2)C1 c1(CN2CCC(N(C(c3ccc(OC)nn3)=O)C)C2)ccc(O)cc1O C12(NC(C3N(CC#C)CCC3)=O)CCCC1N(C(C1CCCC(C)C1)=O)CCC2 Cc1cnncc1C(=O)NCC1CN(C(=O)CCCOC2CCOCC2)CCO1 c1(OC)cc(C(=O)N(C2CC3CCC(C2)N3C(=O)CC2CC2C)C)cc(F)c1F C=CCC(C)C(=O)NCC(C1CCN(C(c2ccc(O)nc2)=O)CC1)(C)O N1(C(c2cc(Cl)ns2)=O)CCC2(CC(C(N3CCOCC3C3CCC3)=O)C2)C1 S(=O)(=O)(c1cc(Cl)c(F)cc1Cl)NC(c1ccc(Cl)c(Cl)c1)C Cc1nc(C)c(C(=O)NC2CC3C(NC(c4coc(Cl)n4)=O)C3C2)nc1C c1(C(N2CC3C(NC(c4cc(C)nc(O)n4)=O)(C3)C2)=O)cccn2c(C)nnc12 N1(C(CC=CC=C)=O)CCC(CC)C1C(=O)NCC1(O)CC(CO)C1 c1(C(=O)NCCN(C(C(c2ccc(F)cc2)CC)=O)C)cc(F)n(C)n1 C1(NC(C(C2CCOCC2)C)=O)CN(C(=O)CC2(O)COC(C)(C)C2)CC1(C)C c1(NC(C2N(Cc3ccc(OC)c(OC)c3)CCCC2)=O)cccc(F)c1C#N C1(C(=O)NC2C(NC(C=CCOC)=O)CCC2)CCc2ccc(OC)cc2C1 C1(CN(C)Cc2cccc(OC)c2)CCN(C(=O)OC(C)(C)C)CC1(F)F c1(NC(C2C(NC(c3c(O)cccc3O)=O)CCC2)=O)ccc2ccncc2c1 N1(C(c2cn(C)c(=O)cc2)=O)CC2(CC(NC(C3CC3c3cnc[nH]3)=O)CO2)C1 N1(c2nccc(SC)n2)CCC2(CCC2)C(CNC(c2coc3c2CSC3)=O)C1 c1(C(=O)NC(CC=C)CNC(c2cncc(Cl)c2)=O)cccc2ncsc12 C=CCC(CC=C)C(=O)N1CCCC(CCCCNC(C2CC23CC3)=O)C1 N1(C(c2ccc(CC)o2)=O)CCC(F)(C(=O)NCC2CCCN2C)C1 C1(NC(c2csc(S)n2)=O)CCC2(CC1)CN(C(c1n[nH]c3c1CSCC3)=O)C2 c1(OC)cncc(C(=O)NCC2CC2)n1.c1(C2C(=O)C=C2)ccccc1 CCC(C(=O)NCCCN(C(=O)CCc1cncnc1)CCO)OC N1(C(=O)Nc2ccc(OC(F)F)cc2)CCOC(CN2CCCC2c2ncco2)C1 C(=O)(CC(O)CNC(C1CC1)=O)NCCCC(=O)NC.C(C)(C)(C)O CCCN=c1[nH]c(N2CCC(CCN)CC2)nc2c1CCCC2 CCCC(CCCNC(C1CCN(C)C1C)=O)NC(=O)Cc1ccc(O)nc1 c1nc2ccccc2[nH]1.C(=O)CC1CC1.C(C(=O)NC(C)C)=CC=CC C1(CN(C(CCC)=O)C)CN(C(c2ccc(OC(F)(F)F)c(Cl)c2)=O)CC12CC2 CC1CCn2cc(C(N3CC(CNc4cnc(F)cn4)C3)=O)nc2C1 c1(C(=O)NCCCCCCNC(C(C)CC2CC2)=O)cc([N+](=O)[O-])c(N)cc1F C1(C(=O)NCC(C2CCC2)NC(C2(C(C)C)CCCO2)=O)CC2C=CC1CC2 c1(OC)ccc2[nH]c(=NCC3CCC(CO)O3)[nH]c(=NCC(Cl)Cl)c2c1 c1(C(=O)NCCCN(C(=O)C(C)(C)c2ncco2)CC)ccc(O)cc1C C1(C2CCN(C(C34CC(F)(C3)C4)=O)C2)CC1.N1(CCC)CCCC(C(=O)N)C1 C1(NC(C2(C=C)CC2)=O)CCCC(NC(c2cc(C3CCCN3C)[nH]n2)=O)C1 c1(CC(=O)NCC2C(NC(C(C)(C)SC)=O)COC2)c[nH]c2cccnc12 C(=O)(CC(=O)NCC(F)CNC(=O)CC(C)n1cccn1)OCC C1(CNC(C(c2ccc(Cl)cc2)C)=O)CCC(C)CC1.n1(CC=O)nccn1.N Cc1ccc(CC(=O)NC2CC(C)(NC(=O)C(O)Cn3cncn3)C2)c(Cl)n1 N1(C(C=C(CC)C)=O)CCOC(CNC(=O)Cc2cc(CC)on2)C1 CC(C)(O)C(F)C(=O)N.CC(C(F)(F)F)N1CCN(C(=O)CCC2(O)CC2)CC1 CC1OC2CCC1(C(=O)NCCCCCn1cc(C3(CC#N)CC3)nn1)C2 C1(NC(C(C)NC(C)=O)=O)CCCN(C(=O)CC2CCC(=O)N2)C1 N1(C(C2CC(OCC)C2)=O)CCN(C(=O)CCc2csc(C)n2)C(CC)C1.O C1(F)(CNC(C2N(CCC)CCC2)=O)CCN(C(c2cc[nH]c2C)=O)C1 c1(C(=O)NCCC(CC)(C)NC(=O)C(COC)OC)ccc(OC)cc1O NC1CCC2CCN(Cc3ccccc3-c3ccc(OC(F)(F)F)cc3)C12 S(=O)(=O)(c1ccc(NC(CC2CC2)CO)c(C#N)c1)NCC(CC)CC(C)C C#CCCN=C(NCC1CN(C)CCO1)NC(c1ccc2c(c1)CCO2)C Cc1nc2cc(C(=O)NC(C)CN(C)C(C3(C)CC(O)CN3C)=O)[nH]c2s1 CC1CN(CC(=O)Nc2ccnc(O)c2Br)CCC1CO N1(C(=O)CC2CC3CCC2CC3)CC2CCN(C(C3CC(O)(C(F)F)C3)=O)CC12 C1(NC(c2ccc(CCC)[nH]2)=O)CN(C(c2cc(C)n(C)n2)=O)CC12CC2 C1(NC(C(CC)(C)O)=O)CC(O)CN(C(=O)C=Cc2scnc2C)C1 C1(N(C(C2C(C(=O)OC)CC2)=O)C)CN(C(=O)C=C(C)C(F)F)CC1O C1(COC)(NC(=O)CC2CSCCS2)CCN(C(=O)CCc2cncn2C)CC1 C(=O)(C1=NN(C)C(=O)CC1)N1CCC(C(C)NC(c2c(C)nc(Br)cc2)=O)CC1 CCCCC(O)C(=O)NCC1(CN(C)C(c2cccc(Cl)c2C)=O)CC1 C1(C(N2CC3CCCN(C(=O)Cc4ccsc4)C3C2)=O)COc2ccccc2C1 c1(CC(=O)NC2CC(n3cc(CCC(F)(F)F)nn3)C2)ccc(C(=O)O)cc1 c1(CC2(C(=O)NCC)CCC2)nccc(=NCc2cc(C)cc(Cl)c2)[nH]1 Cc1ccc2nc(C(=O)NCC3CCCN3C(=O)C(F)n3ccnc3)ccc2c1 c1(C(C=O)(F)F)cccc(Cl)c1.C1CC(O)C1.O=C(CC1(CO)CC1)NC N(C1CCCc2ccc(C(C)(C)C)cc21)C(c1ccc(C=CC(=O)OC)cc1)=O c1(OC)cccc2c1C(C(=O)N1CC3CN(C(C)=O)CC3C1)CC2 Cc1[nH]cc([N+](=O)[O-])c(=O)c1C(=O)N(C)CCNC(=O)CCOC(C)C N12Cc3[nH]nc(c3C1)C(=O)NC(C)C2=O.C(CCOCC)OC.CCO.CC N1(C(C(n2cc3ccccc3n2)C)=O)CCc2nnccc2C1 N#Cc1cc(S(=O)(=O)N2CCOCC23CCN(C(c2ccno2)=O)C3)ccc1Br N1(C(c2cc3ncccc3o2)=O)CCC12CCCN(C(C13CC(F)(C1)C3)=O)C2 Cc1ccc(NCCC=CBr)cc1OCc1ccccc1 c1(OCC)cccc(C(N2CC(C)C2)=O)c1.N1(CC(=O)N)CCN(C)CC1 c1(OC(C)C)cc(CNC(C2CCCN2C(=O)C(C)O)=O)ccn1 N1(C(C(CC)SC)=O)CCCC2(NC(c3ccc(F)c(OC)c3)=O)CC2C1 O(NC(=O)C(C)(C)C(=O)N(C)C)C(C(CC(C)C)CNC(C1CC1C)=O)=O Cc1ccc(C(=O)NC2CCCC2NC(C2CCN(C)C2)=O)c(Br)c1F N1(C(C23CSCC2C3)=O)CCC2(CC1)CC2c1cn(Cc2ncccn2)nn1 c1(C(N(C2CCN(C(=O)CCCc3nccs3)C2)CC#C)=O)csc(O)n1 Cc1cn2cccc(C(=O)NC(C3CCCN3C(C3CCO3)=O)C)c2n1 O(N1CCN(C(C2CCCN(CC(F)F)C2)=O)CC1)CC N1(C(C(c2n(C)ncc2)NC(c2sccc2Cl)=O)=O)CC(O)C(O)C1(C)C C1(CNC(NC(C)C)=NCCCCl)COC2(CCOCC2)O1.C1(C#N)CC1 C1CC2(CCCC2)C1.Cn1ncc(CNC(=O)CSC(F)(F)F)c1C(=O)N c1(C(N(C(CNC(CN(C)CC)=O)C2CC2)C)=O)cncc(N2CCCC2)n1 C1(N2CC(C(=O)NC(CC)CNC(c3occc3C)=O)C2)CCN(C)CC1 c12ccc(cc1)c(=O)n2C(=O)CC.N1(C=O)CCOCC1.N1(CCO)CC=CC1 c1(CC)nc(Br)sc1C(=O)N(C)CCN(C)C(C1(CC(=O)OC)CC1)=O N1(C(CCC(=C)Cl)=O)CCC(CCNC(c2c(OC)ccnc2OC)=O)CC1C CC(CC1CCC1)C(=O)N(C(C)CNC(c1cnoc1-c1ccccc1)=O)C C1(C(N2CCCC2)C(=O)NCCOCC)CC2(C1)OCCO2.C1CCCC1.C c1(CC)cc(C(=O)NCC2CCC2NC(c2ccsn2)=O)c(Br)s1 N1(C(c2n[nH]c(C)c2C)=O)CCCC(CO)(NC(=O)CCc2nncs2)C1 c1(C(CCO)NC(=O)NC2C=CCC2)ccccn1 OCC(CNC(c1ccccc1)C(F)F)C(F)(F)F Cc1cc(C(=O)NCC23CCC(CN2C(c2oc(C)nc2C)=O)C3)c(O)nn1 c1(C=O)ccc(N(C)C)cc1F.C1(C)(CC)CCC(C(=O)NC2CCC2)O1.C C(=O)(C(CCC1CCC1)NC(c1cncc(N)c1)=O)N1CC(OC(CC)=O)C1 c1(SC)cc(C(=O)NCC2CN(C(c3nccnc3N)=O)CCO2)oc1C CC1=C(C(=O)N2CCN(C(=O)C)CC2)CCO1.C1(CCC(=O)N)CC(C)(C)CO1 N1(C(c2cnc(=N)[nH]c2)=O)CCCN(C(C2CCCC(F)C2)=O)CC1 c1(OC)cc(OCC(=O)NC2(CNC(=O)CC(C)C)CCC2)ccc1.S c1(C(N2CCCC(O)(CCNC(c3c(C)snc3)=O)C2)=O)cc2cn[nH]c2cn1 C(=O)(C1CCCc2n[nH]cc21)NCC1(OC)CCN(C(C2CCOC2)=O)CC1 C(=O)(C(O)C(C)(C)C)N1CC(OC)C(NC(=O)C(C)S(C)(=O)=O)C1 C1(C)(NC(C(C)OC)=O)CCN(C(=O)C(C(C)C)n2ccc(C)c2)CC1 C1CCCN(C(C2(C)CC(C)(C)C2)=O)C1.c1(CCCCC)ccc(C(=O)NC)o1 S(=O)(=O)(c1cnn2ccc(N3CCC(O)C(F)C3)nc12)NCC1(CC)CC1 C1CN(C(c2cscc2C(F)F)=O)CCC1C.C1(C(=O)NC)(COC)CC1 c1(C(N2CC(C)C(C(=O)N(c3nnco3)C)CC2)=O)cc2c(s1)CCCC2 c1(C(=O)NC(CC)(C)CNC(=O)Cn2ncnn2)cc(Cl)c(C)cc1Br C1(CC(=O)N(CCCC=C)C)CN(C(=O)C(C)CC(=O)OCC)CCC1C C1(CF)CCCC1N=c1[nH]c(N2CCC3(CCSCC3)CC2)nc2cc[nH]c12 C1(C(N(C2CCN(C(C3(OC)CCSCC3)=O)CC2)CC)=O)Cc2nccn2C1 C#Cc1ccc(C)c(NC(=O)CC23CCC2CN(C(=O)CNC=O)C3)c1.O C1CC2CC(C1)N(C(=O)CN1C(=O)CNC1=O)C2.Cc1nc(O)ccc1C(=O)N N1(C(C(N2CCOCC2)C)=O)C(C(=O)NC(C)CC(C)C(F)F)CCC12CC2 c1(C(N2CCC(F)(CNC(c3nccc(CC)c3)=O)C2)=O)cn2ccsc2n1 CC1CCC(Cc2ccccc2)CN1C(CCC1OCCO1)C(=O)NC1(C)CC1 CC1=C(C(=O)N2CCCC2CCCNC(=O)CCc2nc(C)cs2)CCS1(=O)=O c1(C(C(=O)OC)NC2CCC(N3CCOCC3)C2)ccncc1C CN1CC2CC1CN(C(CC1CCCCO1)C(=O)NCCCF)C2 c1(C(=O)NCC(CC)Nc2ncc(Br)c(C)n2)cnc2[nH]c(O)nc2c1 N1(C(c2c(F)ccc(C)c2)=O)CCC2CCC(NC(=O)CC3CCCCO3)C12 c1(C(=O)NC(C)CN(C(=O)Cc2cncnc2)C)ccccc1.C(=O)N(C)C CC1CN(C(c2ccc(C(F)(F)F)cc2Cl)C(=O)NC2CCOCC2)CC(C)O1 Cc1cccc(C)c1C(N1CCC(N(C(=O)CC2OC(C)(C)OC2=O)C)C1)=O C1(C(N(C(C)C2CC2)CC)=O)CC12CCCOC2 C1(C(=O)NCC)CN(Cc2cccnc2N(C)C)CCC1O N1(C(=O)C=Cc2cnccn2)CCC2(CCN(C(C3CCCOCC3)=O)C2)C1 c1(OCCOC)ccc(C(=O)NCCC2CCC2)cc1.C1(C=O)CCCN1C C(CC(F)(F)F)(c1ccc(Br)cc1)NC(=O)NC(COC)C(C)C C1(c2nnnn2Cc2ccco2)(SCCC)CCC(C(=O)OCC)CC1 C1(C(N(CC#C)CCOC)=O)CC=CCN1C(c1cc(CCC)on1)=O C(C)(CO)(C(=O)NCCC(C)(C)NC(=O)CCCC#N)NC(C)=O C(CCC(N)=O)(C(=O)NC1COCC1NC(C1(c2ncco2)CC1)=O)N(C)C C1(CNC(C2COCCO2)=O)CCC2(CN(C(c3nnc(O)cc3O)=O)C2)O1 CC1CC(=O)NC1C(=O)NCCCCNC(c1cnn(CCF)c1)=O C=C(Cl)CCC(=O)NC1CCC(CNC(c2cccc(=O)o2)=O)C1 C(=O)(NN1CCCC1C(=O)NOCC1CC1)C1(OC)CCC(C)C1 CCCC(O)C(CO)NC(c1ccc(CNC(C2(N(C)C)CC2)=O)o1)=O C(=O)C(F)(C)C(C)C.c1(COC)ncc[nH]1.C1(C=O)CC1C(C)(F)F.C N1(C(CCCCC)=O)CC2(NC(=O)Cn3ncc(O)nc3=O)CCC1C2 CC(CC(=O)NC1(c2ccco2)CC1)C(C)(C)NC(C1CN2CCC1C2)=O C1(CCCC)CCC(C(N2CCCC2)=O)CC1.C(=O)(C(C)C(C)C)N(C1CC1)C c1(C(=O)Nc2cc(-c3ccc(F)s3)cs2)cccnc1Cl N1(CC)CC(C)OC1=O.N1(CC(N2CCC2)=O)CCNC(=O)C1.C(=O)(C)N C(=O)(CC(C)(C)NC(c1cscc1Cl)=O)NC(c1cn(C)nn1)(C)C C=CCCCC(=O)NCCNC(c1[nH]c(C)cc1C)=O c1(C(=O)OC)ncc(C(=O)NC(CO)C(C)NC(c2[nH]cnc2C)=O)s1 c1(C(C(=O)N(C2CCCCC2)CCOC)C)cccc(CN(C)C)c1 O=C(C1=CN2CCN=C2C=C1)NC(c1ccc(Br)cc1)C1CCC1 C(C(C)(O)C(=O)NCC1CCOC1)OC.c1(C=O)cc(-c2ccc(Cl)s2)on1 Cc1cc(=O)oc(C)c1C=O.C1CN(C(C2CC2C(C)O)=O)CC(C)(C)O1.N c1(C(N2CC(N(C(c3c(C)nn(C)c3Cl)=O)C)C2)=O)cc2n(n1)CC(C)NC2=O C(=O)(C1=CCC(C)CC1)N1C(CNC(c2cnn(CC)c2Cl)=O)C(C)CCC1 N1(C(C(C=C)(F)F)=O)CCC(C2CCCN(C(=O)Cc3ccc(SC)cc3)C2)C1 CCCCCC(C)CC(=O)N1CCC(C(=O)NC2CCOCC2)C1(C)C c1(CC)cc(C(=O)N(CCCNC(c2coc(C)n2)=O)CCO)cc2c[nH]nc12 C(CC(C(=O)NOCC)NC(=O)C=CCN1CCC1)OCC C1(C(N2CC(NC(c3ccco3)=O)C(CC3CC3)C2)=O)CN2CCN1CC2.C CC1CN(C(C2CCC(=O)CC2C)=O)CCC1NC(c1ccn(C(F)F)n1)=O C1(C(=O)NC(CC=CC)C(=O)N2CC(C)(C)C2C2CC2)CCC2(CC1)CC2 c1(C(=O)NC2(C)CN(C(C(CC)(C)C#N)=O)C2)ccc(S(C)=O)cc1 N1(C(C(CC=C)OC)=O)CCCC(NC(=O)CC=C(C)C)C1CC C1(CC)CN(C(C2CCCC(C)(C)C2)=O)CCN1C(=O)CSc1c(C)n[nH]c1C c1(OC)ccc(C(C)NC(C)C)c(Cl)c1.C(C)(C)SC C(CC(C)(O)CNC(C1CCN(C)C1)=O)OC.c1(CC=O)c(C)n[nH]c1C.N N1(C(c2ccc(C)cn2)=O)CC2CC(C1)N2C(=O)C(C)NC(=O)C1CC1 C(=O)(C(C)(C)CO)NCC(C)NC(=O)CC1CCCCN1C C=CC(O)(C(=O)NCCC1(O)CCCN(C(=O)Cc2ccco2)C1)C(F)(F)F N1(C(c2ccc(C)c(C)c2)=O)CC(CO)C2(C1)CN(Cc1ccc(F)c(I)c1)C2 CCC(C)C(C(N)=O)NC(=O)C(CC(F)F)NC(c1ccnc(CO)c1)=O C(=O)(C#CC1(C)CC1)N1CCC(CC=C)(NC(C2(c3ccccc3C)CC2)=O)C1 N1(C(CC2CCCC(NC(=O)CCOC3CC3)C2)=O)CC2(CCOC2)C1 Cc1ccc(-c2ncc(C(=O)NC(CNC(C3CCCOC3)=O)CO)s2)cc1C CCCCCC(F)C(=O)NC(CNC(C1(C(F)(F)F)CCC(OC)C1)=O)CC C(=O)(C1=C(Cl)CCOC1)NC1(C)CCCN(C(Cc2ncc(C)s2)=O)C1 N1(C(c2c(CC)[nH]cc2)=O)CCC(CC)C1CNC(=O)CC1CC1 CC1CCN(C(=O)CC2CC3CCC2C3)CCN1C(=O)CNC(N1CCCC1)=O CP(C)(=O)c1ccc(C(=O)NC2CCCCN(C(c3cnc[nH]c3=N)=O)CC2)o1 C1(NC(C(OC)OC)=O)CC(CO)N(C(c2cncc(C(C)(F)F)c2)=O)C1 c1(CC)cc(C(=O)NC(CNC(C2(OC)CCSC2)=O)CC(C)C)ccc1F N1(C(COCCC=C)=O)Cc2ccccc2C(NC(c2cc(O)nc(O)n2)=O)C1 C(C(=O)NCCCn1cnnn1)(C(C)(C)C)NC(c1ccn(CCC)n1)=O CC(C)C(O)C(=O)NC(C)(C)C(C)NC(c1ncn(C)n1)=O CC1(C)CCCC1C(=O)NCCOCCC.c1(CC=O)ccn(C(F)F)n1 C12(C=O)CCOC(C)(C1)C2.C1(OC)CC(CC=O)C1(C)C.C12CC(C1)C2.N Cc1ccc2[nH]c(C(=O)NCC3C=CC(NC(C4(C)CSC4)=O)C3)cc2c1 C1(N2CC(Oc3ccccn3)C2)C2CCCC1NC2 c1(SC)nc2ncnc(N3CCC(C)(C)C(CNC(c4ccn(C)n4)=O)C3)c2s1 S(=O)(=O)(c1ccc([N+](=O)[O-])c(F)c1)N1C(C)c2ccsc2CC1 C1(C)(CNC(C2C3CN(C(c4c(CC)c[nH]n4)=O)C2C3)=O)CCN(C)CC1 c1(C(=O)NC(CCN(C(CN2CCC(C)C2)=O)C)C(C)C)c[nH]c2ncccc12 Cc1cc(=O)c(C(N2CCC(CNC(=O)CN3CCCC3)C2)=O)cn1C c1(C(N2CC(NC(c3c(C)coc3)=O)CC(C)(C)C2)=O)n[nH]c2cc(Cl)ccc12 C1(C(=O)Nc2c(CC)cc(O)cc2)CCC(F)(F)CC1F C1(C)CCCC1.Cc1ncsc1C(=O)NC.C1(CS(C)(=O)=O)(C=O)CCC1 Cc1ccc(C(=O)NC2COCC2NC(=O)Cc2ccsc2)cc1C C(=O)(C(C)(C)CS(C)(=O)=O)N.C1(NC(C(C)Cc2ccccc2)=O)CCCCC1 C1(O)(CNC(CN2CCN(C)CC2)=O)CCCN(C(C2CCCCS2(=O)=O)=O)C1 c1(OC)c(Br)ccc(C(N2CC(C)(C(=O)Nc3cc(C)ccc3C)C2)=O)c1F C1(CCC(=O)NC(CSC)C)CCCCN(C(c2c[nH]nc2[N+](=O)[O-])=O)C1 C(=O)(CCS(=O)(=O)C(F)(F)F)N1CCC(F)C1.O=C(C1=CS(=O)CCC1)NC C(=O)(C(F)C(F)(F)F)NC1CCC(CC(=O)NC2CN(C(C)(C)C)C2)C1 C1(CNC(C(CC(=C)C)C)=O)CN(C(c2cc(O)nn2C)=O)C2(CCC2)C1 C(C(C(=O)N1CCCC1C(=O)N(CCC(O)CO)C)N(C)C)OC CCC(F)(F)CC(=O)NCC1CCN(CC(=O)NCCOc2ccccc2)C1 CC1(CNC(C2(C)CCCS2)=O)COCCN(C(c2sccc2Cl)=O)C1 Cc1cc(C)c(C(=O)NC2CCC(F)(CN)C2)cc1C C1(NCCN(CCC(F)(F)F)CC=C)CCCC1S(C)(=O)=O c1(CC(=O)N(C2CCN(C(=O)C#CC3(C)CC3)C2)C)ncn2c1CCCC2 C(C1=CCN(C(c2cnn(CCF)c2)=O)CC1)NC(C(C)(C)CO)=O C1(C(=O)NCC2(NC(=O)CCc3ccon3)CCCC2)CCc2nc[nH]c2C1 C(=O)(CCS(N)(=O)=O)N1CCN(C(C)C(N2CCCC2CO)=O)CC1 c1(NC(C2CC(NC(c3cccc(OC)c3O)=O)C2)=O)ccc(I)cc1[N+](=O)[O-] c1(CCC(N2CCN(C(c3n(CC)ccc3)=O)CC2C)=O)n[nH]c2ccccc12 Cc1nccn1C(C)C(=O)N(CCC(=O)NCc1nncs1)CC1CC1 c1(C=O)cc(F)cc2cc[nH]c12.CN1C(=O)CCC1CC(=O)NCC1CCC1.N CC(C(C)(C)CO)NC(=O)CC1CC(F)CN1C(=O)CC1CCCCC1O CC1CN(C(=O)CSc2nncn2C)CCC1NC(=O)C(F)(F)C(O)C1CC1 Cc1ncsc1C(=O)CN(C)Cc1cn(C)cn1 C(=O)(CCCCCS(N)(=O)=O)NC1CC(NC(CC(COC)(C)O)=O)C1 N1(C(C2C(NC(C(CO)NC(N)=O)=O)CC2)=O)CCOC2C(O)CC12 C1(NC(C2CCN(c3ncccn3)C2)=O)C2CC1N(C(c1cncc(F)c1)=O)C2 C=CCCCCCCC(=O)N1CCN(C2CN(C(C3CC3Cl)=O)C2)CC1 N1(C(CSS(C)(=O)=O)=O)CCCC2(CCC2)C1.c1(C=O)ncoc1C(F)(F)F N1(C(C2C(C)C2)=O)CC2CCC(NC(c3cc(C4CC4)[nH]n3)=O)CC2C1 C(C#CC(=O)N(c1ccsc1)C)NC(CC1C(CC)C1)=O c1(C(=O)NC2CCN(C(c3ccc(C)o3)=O)C2C(C)(C)C)snc2ccccc12 C1(NC(C=C(COC)C)=O)CC(C)CN(C(c2cncc(OC)n2)=O)C1 c1(OC)ccc2cc(C(=O)NC3(CN(C)C(C4CCCC4)=O)CC3)sc2c1F S(=O)(=O)(c1ccccn1)N.c1(NC(C2CC2)=O)nc(C(F)(F)F)cc(Cl)n1 C(C)CC(C)(C)C.n1(CCCSCC)nnnc1C(c1ccn(C2CC2)n1)N C(=O)(CCCCCS(N)(=O)=O)NCC1C(C)CCN(C(=O)C(C)N2CCC2)C1 N1(C(CC2N(C)CCC2)=O)CCC2(CC1)CC2NC(C1(S(C)(=O)=O)CC1)=O c1(OC)cc(Br)c(C(=O)NC)cc1F.C1(C(N2CCC2)=O)C2(CC2)C12CC2 N1(C(C2C(OC)CCC2)=O)CCc2c(ncn2C)C12CCN(c1ncnc(=N)[nH]1)C2 c1(C(c2nnn[nH]2)NC(C(=O)NCC)C)sc(Cl)nc1C.c1nnn(C)n1.C c1(CC(=O)N(CC(C(=O)N(CC(=O)OCC)C)C)C)cccnc1Cl C1(C)(CC=O)CCS(=O)(=O)N1.CC1CCN(C(=O)CC2(C#N)CC2)C1.C N1(C(C(CC)CCOC)=O)C2CCC1CC(CNC(C13CC1CNC3=O)=O)C2 c1(CC)ccc(C(=O)NC(CCNC(=O)CCC(C)SC)C(C)C)c(O)c1 N1(CCN(C(C2CCC(C)S2)=O)C)CCN(C(c2cnc(C(C)(C)C)o2)=O)CC1 Cc1cc(C)c(CC(N2CCC(NC(C3(CC(C)C)CC3)=O)C(C)C2)=O)c(C)c1 CC1C(C)CN(C(=O)CC2(C)CCN2C(=O)CC2CCCCC2O)C1C n1(CC(=O)NC(CC)CN(C(=O)C(C2CCCCCC2)O)C)nc(C)n(C)c1=O N1(C(CC2CCC(NC(C3C=C(C)CS3)=O)C2)=O)CC(C(=O)O)CC(O)C1 c1(C(N2CCC(n3cc(C)nn3)CC2)C(=O)NC(CC)C)cc(Cl)sc1Cl C(=O)(C(O)C(C)(C)C)N1CCC(CNC(C2C(c3ccc(C)s3)C2)=O)C1 Cc1c(C(N2CCOCC2C(=O)NCC(O)CC2CCC2)=O)ncn1C N1(C(C2CN(S(C)(=O)=O)C2)=O)CCC2(CCN(C(C3CCCCO3)=O)C2)C1 C(C(=O)N)(C(C)(C)C)NC(C)=O.C1CCOCC1.c1(C=O)[nH]nnc1C1CC1 N1(C(CC2CN(C(C(C(CC)C)=O)=O)CC2C)=O)CC(F)(F)CCC1C c1(C(N2CCC(C)(CC(=O)Nc3c(OC)nccc3)C2)=O)cc(C#N)ccc1C N1(C(Cc2ncsc2)=O)CCN(C(=O)C(C)C#N)C(CC(F)F)C1.CC(=O)NC c1(NC)ccc(C(N2CCCCC2C)=O)c(Cl)c1.C12(C(=O)N)CCCC(C1)OC2 c1(C(C)NC(=O)N(C)CCN2CCCC2)nnc2ccccn12 Cc1cc(C(=O)NCC2(C(=O)NC(C)CC(F)(F)F)CCC2)ncc1N C1(N(C)C(C2CCCC(O)C2)=O)CCCCC1CNC(=O)CC1CCC(O)C1 C12(C=O)CC3CC(C1)C(=O)C(C3)C2.c1(C=O)ccnc(C2CC2)c1.CCC.N Cc1oc(C(=O)NCC(C(C)C)NC(=O)C(C)CF)cc1Br N1(C)CCCCC1.c1(CC)c[nH]c(C(=O)NCCN(C)C(c2csnc2Cl)=O)c1 c1(C(N(CC(C)NC(C=C(C)c2cccs2)=O)C)=O)ccc(C)nc1C1CC1 C1(OC)(CNC(c2cnc(O)s2)=O)CCN(C(=O)C(=O)NCC(F)F)C1 N1(C(C(C=C)(C)CC)=O)CCC(C2CCN(C(=O)C=NOC)C2)CC1 C12(C(=O)NC(C(C)O)C(=O)NCCCOCCCN(C)C)CCCN1CCC2 N1(CC(=O)NCCC2CCC(C)C2)Cc2c(Br)cccc2C1=O C(=O)(C=C1SCC(=O)N1C)NCC(CNC(c1ccc(NC)cn1)=O)O Cc1cc2[nH]c(=O)c(C(=O)N)cn2n1.C1(O)(CC=O)COC(C)(C)C1.C1CC1 Cc1cc(C)cc(C=Cc2nc(C(C3(C)CCCCC3)c3ccccn3)no2)c1 CC(CCO)N(C(=O)C(c1cccs1)NC(=O)C(F)C1CCC1)C CCCCC(CCCC)C(=O)NCC(C)(C1CC1)NC(c1ccc[n+]([O-])c1)=O Cc1nn(CC(F)(F)F)cc1C(=O)NCCC(C)N(C)C(C1CC(Cl)(Cl)C1)=O C1(NC(=NCCN(S(N(C)C)(=O)=O)C)NC2CCCC2)CC(C2CCCCC2)C1 C(=O)(C1=C(Cl)CCCC1)NC1CN(C(Cc2c(C)cccc2)=O)CC(O)C1 N#CC1(CNC(N2CCC(=C(F)F)CC2)=O)CCS(=O)(=O)CC1 N1(C(C(CC)NC(C)=O)=O)CCCCCC1C(=O)NC(c1cscn1)CO C(CC(=O)N1CC2CCCC2C1)(C(F)F)NC(c1c(CC)occ1)=O c1(C(N2CC(OC)C(NC(C3CC(=O)N(OC)C3)=O)C2)=O)nnc(Cl)cc1N C(=O)(C(O)CC(C)(C)C)N(CCCCNC(=O)C(c1cccc(Cl)c1)(F)F)C N1(CC)CCN(C(C)(C)CNC(=O)NC2CCOC(C(C)C)C2)CC1 N1(C(CC(C=C)CCC)=O)CCC2CCC(C1)N2C(c1cnc(CC)o1)=O CC(C)CCCC(C)NC(=O)C(CN(C)C)N(C(=O)Cc1ccoc1)CCCO C(=O)(C1=CCN(C(C2(Cl)CCCCC2)=O)CC1)NCC(C)(O)CO c1(CNC(CN(C(c2ccc(O)cc2)=O)CC)=O)nc(C)c(C)[nH]1 c1(-c2cccc3c2cno3)cc2cccc(Cl)c2[nH]1 C1(C(N(C2CCCC2)CC#C)=O)CCN(C(=O)CNC(=O)CC)C1 c1(C(N2CCN(C(C(C(C)C)OC)=O)CC2C)=O)ccc2c(c1)COC(C)(C)O2 C(=O)(CCS(N)(=O)=O)N(C)CC1CCCCC1.N1(CC(=O)N)CC2CCC1C2 C12(NC(C(CC)(C)CNC(c3ncc(C)cc3F)=O)=O)CCC(CC1)C2(C)C CC1(C)C(NC(C2C3CN(C(=O)CCCCC4CC4)CC23)=O)CC1(F)F C(C)(C(=O)NC1CCCN(C(=O)CCCN(C)C(C)C)C1)(C(C)C)OC C(C(CN=c1[nH]c2ccc(F)cc2s1)C(F)(F)F)NC(C#CC1(C)CCCO1)=O c1(C(=O)NC23CN(C(C(C)C)=O)C(C2)C3)ccc(=O)n(-c2cccc(Cl)c2)c1 c1(C(=O)NC(C(C)NC(c2cccc(F)c2)=O)C)cncc(-c2ccccn2)c1 C1(OC)CCN(C(C2CC(F)CCN2C(c2ccc(Cl)o2)=O)=O)C12CCC2 CC1(C=CC(=O)NC2CN(C(c3ccc(C(C)(C)C)[nH]3)=O)C2)COC1 c1(CNC(c2cn(C)nc2Cl)c2n(C(CC)(C)C)nnn2)cccc(Br)c1Cl C(=O)(CCC(=O)NCC(CO)NC(=O)CCc1ccoc1)OCC C1(CCC)CN(C(c2cncc(C(N)=O)c2)=O)CCN1C(=O)CC1OCCO1 N1(C(c2cncc(CC)c2)=O)CCC2(C(=O)N(C3CC3)C3CC3)CCCC12 N1(C(CC(C)(C)F)=O)C2CCC1CC(NC(c1c[nH]c(C(F)(F)F)c1)=O)C2 C=CC1(C(c2nnnn2C2CCC2)Nc2ccc(C(=O)OC)cc2C)CCOCC1 C(C(O)CC(F)(F)F)NC(C1N(C(c2c(C)csc2)=O)CC(C)C1)=O C1(C(N(CC(C2CC2)OC)C)=O)C2CC1N(C(c1cc(Cl)cs1)=O)C2 Cn1cc(C(=O)NCC(CO)NC(c2ccccc2CC(C)(C)C)=O)cc1Br N1(C(C(C(CC)CC)C)=O)CC2CCC1C1CN(C(c3ccsc3OC)=O)CC21 C1(C(C)C)(C(=O)NCCC2COCCO2)CCN(C(=O)CCc2nncs2)C1 C1CN(C(C23CC(F)(C2)C3)=O)CC1C1CC1.c1(C(C)C)ccc(F)c(C=O)c1.N C1(C)(CNC(c2c(CC)cco2)=O)CCCC1.c1(CC(=O)N)ccccc1 Cc1nsc(C(=O)NCC#CCNC(c2cc(C(F)(F)F)n[nH]2)=O)c1N c1(NC(C(=O)NC(C)C(C)n2cncn2)=O)cc(Cl)ccc1-n1cccn1 Cc1cccc(C(C)N(C2CCOCC2)C(N2CC(C)(O)C2)=O)c1C C1(CNC(=O)NC2N(c3cn(C)nc3)CCC2)CC2C=CC1CC2 c1(C(c2n(C(CC)(C)C)nnn2)NCC(C(C)C)OC)cc(Br)nn1C N1(C(C2C(CC)C2)=O)CC2(CCC(CNC(C3CC4CC4C3)=O)O2)C1 c1(NC(C2C3CN(C(c4ccc(F)cc4I)=O)CC23)=O)ccc2c(c1)CCO2 CC1CN(C(=O)C(=O)NC(Cc2nn[nH]n2)C(F)(F)F)CCN1 C1(NC(C(=O)OC)(C)c2cccs2)CCN(CCCc2ccccc2)CC1 C1(CC)CCOCCN1C(=O)COC1CC(NC(=O)C2=C(C)CCC2)C1 Cc1cnn(CCCC(=O)NC2CCC(N(C(=O)C(C)C)C)C2)c1 N1(C(CCN(CCC)C)=O)CCCC2(CC(NC(=O)C(c3ccncc3)C)C2)C1 Cc1cc(CC(N2CC(N3CCN(C(c4c(C)csc4Cl)=O)CC3)C2)=O)n(C)n1 C1(C(=O)NC(C)CN(C)C(C2CSCN2C)=O)COCC1(C)C C1(N(C)C)CCCC(C(=O)NCC(C)(C)CNC(=O)C2=CCCC2)C1 Cc1cn2c(n1)CC(C(N1CCOC(CCNC(c3ccsc3)=O)C1)=O)CC2 N1(C(CC(C)(C)OC)=O)CC(C)C(C)(C(=O)NCC2(C#N)CCC2)C1 c1(C=O)cc2cc(F)ccc2o1.C1(CNC(=O)CC2(C(F)F)CC2)CCCC1 c1(N(C)C)ncccc1C(=O)NCC1CCN(C(=O)C(N)=O)CC1 Cc1nc(NC2CN(C(=O)C=Cc3ccccn3)CC2(C)C)ncc1Br c1(OCC)ccc(C(N2CCCC2CC2COCCN2C)=O)cc1 N1(C(CC2CCC(=O)O2)=O)CCN(C(c2cc(Br)no2)=O)C2CCC12 C12(C(=O)NCCSCC=C)CC1CCN2C(=O)C(C)(CO)OC N1(C(c2c(C#C)c[nH]n2)=O)CCC(NC(c2ccccc2CC)=O)CC(C)(C)C1 N1(C(=O)Nc2cc(C(C)C)[nH]n2)CC(C(=O)O)C2(C1)CN(C(=O)C1CC1)C2 C1(NC(CCC=C)=O)CC(NC(=O)C(c2cccnc2)N(C)C)CC1O N1(C(c2nc(CCCC)sc2)=O)CCCC(NC(=O)COCCCF)C(F)C1 CCCCCCCCN(C(=O)CC1CC2(CC2)CN1C(c1ncncc1Cl)=O)C c1(C(N(CCCCNC(=O)CC2CC(C)(C)CO2)C)=O)n[nH]c2c1CCCC2 C12(CC)CCC1CN(C(C1CCC1)=O)C2.Cn1cc(OCC=O)cn1.C1CC1.N N1(C(Cc2nccc(OC)n2)=O)C2CCC1(c1cn(CC(=O)O)nn1)CC2 CCC(CC)(CO)C(=O)NC1CCCC(N(C(=O)Cc2cccc(OC)c2)C)C1 N1(C(C(c2ccccc2)OC(C)C)=O)CCCC1CNC(c1ccn(C)c1)=O CC(C)(CCNC(C1CCCOCC1)=O)C(=O)NC1(CCF)CC1 CCC(CC(=O)N1CC(C)(C)C1)NC(C1CCNC(=O)C1)=O N1(C2C(C)SCC2)CC(NCCO)OC(C)(C)C1 CC1(NC(=O)C(F)C2CCC2)CCN(c2cncc(Cl)n2)CC1 CCC(C)(O)C(=O)NC(C)CN(C)C(c1ccc(OC(C)=O)cc1)=O C1(NC(C(n2c(C)ncc2)C)=O)CC2CCC1N2C(=O)CSc1cccnc1 c1(C(=O)NCCOC2CN(C(C(C=C)O)=O)C2)cc(Br)cc2nn[nH]c12 c1(C(=O)NCC(CC)NC(C23CC(F)(C2)C3)=O)ccc(-c2ccccc2)s1 C1(NC(c2cc(OC)no2)=O)CCC2CCN(c3nnc(C(C)(C)CC)o3)C1C2 C1(C=O)CCN(C)C(=O)C1.c1(CC(C)C)cc(C(=O)N)n[nH]1.CC(C)C1CC1 CC1(NC(C2CC2C(C)(F)F)=O)CC(NC(c2cc(CO)on2)=O)C1 n1(C(C)C(=O)NC(CNC(c2cccnn2)=O)C2CC2)cnc2c(N)ncnc12 c1(C(N(CC(CO)(CO)NC(C2C(C)OCC2)=O)C)=O)cncc2sccc12 C(=O)(C1CCCc2nc(C)[nH]c21)NC(CCCNC(C1(CC)CCC1)=O)C N1(C(CC)=O)CCN(C(C(=O)NC2CCCC2)c2cccs2)CC1 c1(CC)cc(C)nc(O)c1.C1(C(=O)N)(OC)CCN(CCc2n[nH]c(=N)s2)CC1 N1(C(c2cc(OC)no2)=O)CCC(NC(=O)CN2CCOCC2)C2(CCC2)C1 C(=O)(CCC(CC)CC)NC(C1CCOC1)CNC(Cc1ccn(CC)n1)=O C1(CNC(CC2CCN(C)CC2)=O)CCN(C(c2c[nH]c(C(N)=O)c2)=O)CC1O C1(C(=O)N)COc2c(cc(Cl)cc2[N+](=O)[O-])C1.C1(C(=O)NCC)CC1[N+](=O)[O-] c1(CN(CCC)CCC)cc(C(=O)NC2CCCN2C(=O)C(F)OC)no1 C(C(=O)N1CCOC(C(=O)NCc2ccncc2)C1)(C(C)C)SCC N1(C(C2N(C(c3scnc3Cl)=O)CCN(C)C2)=O)CCCC2OCCC2C1 c1(C(N2C3CN(C(C=C(C)C4CC4)=O)C(C3)CC2)=O)cc2n(c1)CCCNC2=O c1(NC(COC2(C)CN(C(C3(CC#C)CC3)=O)C2)=O)ccc(C)c(O)c1 C1(NC(C=C(CC)CC)=O)CCCN(C(c2cccn3nnnc23)=O)CCC1 c1(OC)ncc(C)cc1C(=O)NCC(CNC(C1CCCCS1)=O)OC CCC(CCCC(=O)NCC(C)Cn1cccn1)NC(=O)Cn1ncccc1=O NS(=O)(=O)C1(C(=O)NC(CNC(c2ccncc2)=O)C2CCC2)CC1.C C(=O)(CCC(CC)CCC)NCC1CN(C(C(C=C)CC)=O)C(C)(C)C1 N1(C(C(CC)Sc2ccccc2)=O)CC2CN(C(c3ncc(C)s3)=O)C2C1 N1(C(c2cccc(C)c2F)=O)CCC2(C=C(C(=O)NC(C3(O)CCC3)C)C2)C1 CC(C)CCCC(=O)N1CCN(Cc2ccc(OC(F)(F)F)c(F)c2)C2CC12 C#CCCC(O)CCNS(=O)(=O)N(C)CC C(=O)(C1=CC2CCCCCCC12)N1CCC(N(C(C23CC(C)(C2)C3)=O)CCO)CC1 n1(CC(N2CC(C(C)NC(C3(CF)CCC3)=O)C2)=O)ccc(O)nc1=O C12(C(=O)NC3(CNC(C=C(CC)C)=O)CCCCC3C)CCC(C)(CC1)CO2 C1(NC(CCCN(C)C(C2(C#N)CC2(C)C)=O)=O)CCCC(O)CC1 C(=O)(C1=C(CC)OCCS1)N1C(CNC(CC(C(C)C)OCC)=O)CC(O)C1 C(CO)(CCCCNC(c1cccc(N2CCOC2=O)c1)=O)NC(CN(C)C)=O c1(CNC(C2C(=C)C2)=O)cccc(CNC(c2ccn(CC)c2C)=O)c1 CC#CCCCC(=O)NCCC1CCCN1C(=O)C=CCO CC1CC(NC(c2c[nH]c(Br)c2)=O)CN(C(c2sccc2Cl)=O)C1 C(=O)(NNC(=O)c1cc(-c2ccc(C(F)(F)F)cc2)on1)N(C)C c1(C(N2CCC(CCC(=O)NC(CC#CC)C)C2)=O)cnccc1C#N C1(C(=O)NC(COC(C)C)C)CC(C)CN1C(C1CCN(C)C1)=O c1(CC(N2C(CNC(c3ccncc3Br)=O)CCC2)=O)cccc(F)c1F N1(CC)CCOCC1C(N1CCC1C)=O.c1(C(=O)N)sc(-c2ncccn2)nc1C c1(C(=O)NCC2CCC(C(N)=O)O2)cc(Cl)c2ncccc2c1F c1(C(N2C(CN(C(CNC(CC)=O)=O)C)CCC2)=O)ccnc(C)c1Cl CC(Cn1ccnc1)CN=c1cc(Cl)nc(C2CCCO2)[nH]1 C1(C(=O)NC(C2CCCCC2)C#C)CN(C(C2CCOC2C)=O)CC12CC2 C1(C(=O)NCC(C2(O)CN(C(C=CCCC)=O)C2)(C)C)CCOC(C)(C)C1 c1(C=O)cc2c(O)ccc(F)c2[nH]1.C1(CC#C)(C(=O)NC)CCCC1.C1CC1 Cc1ccc(C(=O)NCC2CCCN(S(=O)(=O)C(C)C)CC2)c([N+](=O)[O-])c1 c1(NC(c2ncc(-c3cccc(S(C)=O)c3)nc2)=O)ccc(Br)c2ccncc12 C1(C(=O)NCC(CNC(c2cnc(N(C)C)c(Cl)c2)=O)F)CCOC2(CCC2)C1 C(=O)(C1CCCn2cncc21)NC(C1(CNC(C(CC)CC)=O)CC1)C C(=O)(C(C)(C)C(C)NC(c1ccn(COC)n1)=O)N1CC(=C)C1 N1(C(C2C(NC(C3CC4(C3)CC(O)C4)=O)CC=CC2)=O)CCC(C2CC2)C1 N1(C(C(C)(C)c2cscn2)=O)CCN(C(=O)C=C2CCOCC2)C(C2CCC2)C1 Nc1cc(C(N2CCC(NC(c3cnc(O)o3)=O)C(F)C2)=O)c2c(c1)OCCO2 c1(C(N2CC(NC(c3scc(C)c3Cl)=O)C3C2C3)=O)cccc(S(C)(=O)=O)c1 c1(NC(N2CCC(c3nccc(C)n3)CC2)=O)cccc2occc12 C1(CC(=O)NCC2CCN2C(c2ncncc2Cl)=O)NC(=O)NC1=O c1(C(=O)NC(CCOC)CNC(=O)CCc2cc(Cl)cs2)cc(C)ccc1N N1(C(CN(C2CC2)CC)=O)CCC(NC(=O)CC2C=CCCC2)C(CO)C1 CCC(CNC(=O)C(C(C)C)NC(c1ccc(CO)nc1)=O)C(C)C C12(CNC(CCCN(C(C)C)C)=O)CCC(CN(C(c3cnc(Cl)s3)=O)C1)C2 C=CCC(CC)C(=O)NCC1CCN(C(=O)C(CCSC)N(C)C)CC1 CCCCC(C)CCC(=O)NC1CC=CCC1C(=O)NCC(c1ccnn1C)O c1(CC(C)C)cc(C(=O)NCC2CC2)no1.C(=O)(CC(C)C1CCCCC1)N CC1(C)CCCN1C(=O)CC1(O)CCCC1.n1(CC=O)cnc([N+](=O)[O-])c1.C C(=O)(CC1=CCN(C)CC1)NC(C)C(C)(C)NC(=O)CCn1ccc(O)nc1=O C1(C(=O)NCC2CN(C(CCOCC)=O)C2)CCC2(C1)CC2(F)F c1(C(C(=O)NCC(CC)(C)NC(=O)C#CC(C)(C)C)(F)F)cc(Cl)ccc1Cl N(C1CCOc2ccc(Cl)cc21)C(=O)NC(C1CCC1)C1CCC1 CN1C(=O)CCC(C(=O)NC2(CF)CCN(C(=O)CC3CCOC3(C)C)C2)C1=O C(=O)(C(C)(O)C(F)(F)F)NCc1cc(C(N2CCC(C(C)O)CC2)=O)sc1 n1(CC(=O)NCC(C)(O)C)nc2c(n1)CCCC2.c1(C=O)nnc(O)nc1O.N C1(C(=O)NCc2c(C)n3c(n2)scc3)COC2(CCN(c3ncccn3)CC2)C1 C1(NC(c2c(C)nn(C)c2)=O)CCC(C)N(C(=O)C(C)n2ccnc2)C1 c1(NC(C2CCC(c3ccc(F)cc3)C2)=O)c(F)cc(F)c(F)c1F N1(C(C(CC#C)NC(c2occc2COC)=O)=O)CCCC(F)CC1 CCCC(C(=O)N1CCC(CCNC(=O)C(Cc2ccccc2)OC)C1)OC c1(C(=O)NC(CCNC(CCC(=C)C)=O)(C)C)cc(Cl)c([N+](=O)[O-])cc1F Cc1cnn(C)c1CC(=O)NCC(CO)NC(=O)C(c1cccc(Cl)c1)C c1(C(=O)NCC2C(C(N3C(C)CCC3(C)C)=O)CCC2)ccn2cncc2c1 C12CCCC1N(C(=O)CNS(N)(=O)=O)CCC2.C(C(=O)N)=CC=CC.C C(=O)(C(C)(C)c1ccccn1)N1CC(C(C)NC(C2CC2CF)=O)C1 N1(C(C(CC)n2cccn2)=O)CC(NC(=O)CC2CCS(=O)(=O)CC2)CC1(C)C CC(C)CCC(F)C(=O)NC(C(=O)NC1CCC(F)(F)CC1)C1CCC1 C(C(CC(C)C)C(=O)NCc1ccnn1C)NC(c1c(C)nc(CC)o1)=O.O c1(N(CCCC=C)CC(C)C)ccc2cc(F)cc([N+](=O)[O-])c2n1 C1(NC(c2c(C)[nH]nc2)=O)CN(C(=O)C(C)Cc2cccc(Cl)c2)CCC1O C1(C(N2CC3C(CNC(=O)Cc4csc(Cl)n4)C3C2)=O)CC2(C1)CC21CC1 c1(C(=O)N)cc(F)c(F)cc1O.CC1(C)CCCN1C(c1ccn(C(F)F)n1)=O c1(C(N2CC3C(C(N=c4n(C)[nH]cn4)=O)(C3)C2)=O)ccc2cnoc2c1 C1(CC(=O)NC(C)CCNC(=O)CCNC(=O)CO)C=NN(C)C1=O c1(CC(=O)NC(C(=O)N(C(C=C)C)C)CC2CCC2)cn(C)nc1C c1(OC)cccc2c1OCC2NC(=O)NC1CCC(C(C)(C)C)CC1 C1(CC(=O)NCCCCNC(=O)Cc2cnn(C(F)F)c2)CC2COCC12 CCC(O)CC(=O)N1CCCC1CCC(=O)NCc1nnc(O)o1 C(CCCCC(=O)N(C)CC1CCN(C(=O)COCc2ccnn2C)CC1)SC c1(CC(=O)N(C2CCCC2)CCNC(C2(C)CCCOC2)=O)cccc(O)c1F Cc1cc(NC2CC3CCC2(NC(c2cocn2)=O)C3)nc(C(C)C)n1 C(CCCC(C)NC(c1n[nH]c(C)c1F)=O)NC(C(COCC)C)=O C12(C(=O)NCC3(C)CC(NC(CN(C)C)=O)C3)CCCCC1CCCC2 CCC(CN(C)C)CC(=O)NCC(C)(C1CC1)NC(c1cnsc1)=O c1(C(=O)NC2(C)CC(C(=O)OC)C2)cccnc1.C1(F)(C=O)CCOCC1.C C1(C(N(CCN(C(=O)CNC(c2ccccn2)=O)C)C)=O)CCCCN1C N1(C(C(CCC)OCC)=O)CCOCC2(COCCN2C(=O)CCOC)C1 c1(C(N2C(C(C)NC(=O)CC(C)C(F)F)CCC2)=O)cccc2ncsc12 C1(CN(c2ncccc2C#N)Cc2c(F)cncc2F)CC2CCCCCC2C1 C1(n2cc(C3(C(=O)OCC)CC3)nn2)CN(Cc2snc(C)c2Cl)CC1C c1(CC(CC)NC(N2CCC(F)(CSc3ccc(C)cc3)C2)=O)ccc(Cl)cc1 C1(C(=O)NCc2nc(C)c(Br)s2)CC2(CCS(=O)(=O)CC2)CN1 Cn1nc(C(F)(F)F)nc1CNC(C1CNCCOC1)=O c1(NC(N(CC(C)C)CC(C)C)=O)ccc(F)c(Cl)c1 C1(C(NOCCCC=C)=O)(CF)CCN(C(C2C=CCC2)=O)C1 c1(NC2(C(F)(F)F)CCN(C(=O)OCC)CC2)nccn(C)c1=O C1(NC(C2(CCNC(C(CCOC)OC)=O)CCCC2)=O)CCc2nncn2C1 c1(C(=O)N)ccnc(Cl)c1O.Cc1cccc(CCNC(=O)COC2CC2)c1 N1(C(c2ccn(CC)c(=O)c2)=O)CCC(NC(=O)C(C)C(C)COC)C12CCC2 c1(NC(C)CNC(c2conc2C2CCCC2)=O)ncc(Br)cc1C#N CCCCCCCC(=O)N(CC(C)O)CCNC(c1ccncc1Br)=O c1(COC)nc(NCC2(OC)CC2)cc(=NC(C)C2CCC2)[nH]1 C(C)(C(C)C(=O)NC(C)C(O)C(F)F)NC(c1n(CC#C)ccc1)=O Cc1cnc(C(=O)NCCCC(O)C(=O)NCc2sc(C)cc2C)c(F)c1 C1(C(=O)NCC(C2(O)CN(C(CNC(C)=O)=O)C2)(C)C)CN(C)CCO1 c1(C(=O)NCC(CC)(CC)NC(=O)C(C)C2CC2)ccnc2c(Cl)c(C)ccc12 Cc1cc(C(N2CCC(CNC(=O)C(C)C(F)F)CC2C)=O)ccc1O CCC(CC)C(C(=O)N1CCCC(C)C1CN=c1ccnc(C(C)(C)C)[nH]1)OC c1(C(C)=O)ccccc1C(=O)NC(C1CCCCN1C(=O)CO)C.c1ccon1 CC1(C)COC(C(N2CC(F)CC2CNC(=O)CN2CCC(CO)CC2)=O)C1 Cc1ccncc1C(=O)NCC1CCCN1C(c1cccn1C(C)C)=O C(=O)(CCC(=O)c1cnn(C)c1)NC(CNC(C1CC(O)(CC#C)C1)=O)CC CC1(C#N)CCN(C(=O)CC2CN(C(c3cc4occc4[nH]3)=O)CC23CC3)C1 N1(C(Cc2c(C)cco2)=O)CC2CC2C1.C(=O)(C(C1CCC1)C1CCC1)N(C)C O=S(=O)(c1ccc(NCCCCCCCO)c(Br)c1)N1CCSC12CCCCC2 CC1SCCN(C(C2CCC(NC(=O)CCc3nc[nH]n3)C2)=O)C1C c1(C(=O)NCCN(C(=O)Cc2cncnc2)C(C)C)cc([N+](=O)[O-])n[nH]1 C12(c3cn(C4CCN(C(C(CCC)N(C)C)=O)C4)nn3)CCC(OC)(CC1)C2 C1(C(=O)NC2CC(C(=O)NC(C)CO)CC2O)(CC)CCCC1O C1(CNC(C2CC(OC)C2)=O)CC(NC(=O)CCc2ncc[nH]2)C12CCC2 CC1CCCN(C(=O)Cc2csc(-c3ccoc3)n2)C1CNC(=O)C(N)=O c1(-c2ccc(OC(C)(C)C)cc2)cn2ccsc2n1.C1C(=O)OCCN1 C1(CCC)(C(=O)OCCc2coc(C)n2)CCCN1Cc1ccccc1 CC1COCCN1Cc1cn(C2CN(C(N)=O)C2)nn1.C12CCCN(C1)C2=O N1(C(C2C(C)CC(=O)NC2)=O)CC=C(CC(=O)N2CCC(O)(CCC)C2)CC1.CC Cc1ccc2c(CCNC(=O)CC3CCCC4(CNC4)O3)c[nH]c2c1 c1(C(N2CC3C(C3)C2)=O)coc(S(C)(=O)=O)c1.CC1(C(=O)N)CC=CCC1.C N#Cc1c(F)cc(CN2CCCC(CC(N3CC4CCC3C4)=O)C2)cc1F c1(C(=O)NC2CC(O)CN(C(=O)COC)C2)nc2n(c1Br)CCC2.C1CC1 C(c1ccc(CC(C)C)cc1)=CC(=O)NC(CC(C)C)CNC(=O)CC(C)F N1(C(C2=C(C)OCCS2)=O)CCCC(C2CCCN(C(=O)C(=O)N(C)C)C2)C1 Cc1cc(NC(=O)CCN(C(c2ccoc2C(C)C)=O)C(C)C)cc(C)c1O c1(C(=O)NC2C(NC(c3cc(CCO)on3)=O)COC2)cc2oc(Br)cc2[nH]1 c1(C2C(NC(=O)NC3CCN(c4ccccc4)C3)CCO2)ccc(O)nc1 CC(C)CCC(=O)NC1CC(C)(NC(=O)C(C)ONC(=O)OC(C)(C)C)C1 [N-]=[N+]=NCCCC(=O)N1CCC(NC(C2CC2(F)Cl)=O)CC1 Cc1sc(C(=O)NC(C2CN(C(C3CC3C(C)C)=O)C2)C)c(Br)c1C C1(NC(c2c(CCC)n[nH]c2)=O)CCN(CCCCOCC)C(C)C1 Cc1cc(N)c(C(=O)NC(C2CN(C(c3ncoc3C)=O)CCO2)C)cc1C N1(C(c2cc(N)c(F)cc2)=O)CCC2(NC(c3ccccc3Cl)=O)CCCC12 c1cc([N+](=O)[O-])ccc1C=O.C1(CC=O)CC(C)(C)CO1.C(C)CC.CC.S C1(CCNC(c2nncc(OC)c2)=O)CCN(C(c2cnc(C)o2)=O)C(C)C1 C(=O)(C(C(C)C)C(C)C)N(CCCNC(=O)COc1ccccc1O)CC c1(C(=O)NC(CCNC(CSCC=C)=O)C)nn(C(C)C)nc1Br c1(CC)cccc(C)c1CNC(=O)Nc1cccc(CS(=O)(=O)C(C)C)c1 N1(C(C(CO)N(C)C)=O)CCC(C(N2CC(CO)C3(CC3)C2)=O)C12CCC2 C(=O)(CCC(=O)NC(C)(C)CO)NCCC.C(c1cnc(C)s1)=CC=O.N N1CCN(C(c2ccc(=O)oc2)=O)CC1.CC(C(=O)NC1CC1)OC1CCCC1 N1(C(CNC(C(=Cc2cn[nH]c2)C)=O)=O)CCN(C)C(C(C)C)C1 Cc1cc(C(=O)NCCCN(CCCC)C)n(C)n1.C1(C=O)CC1C(F)F.N C#CCC(CC(=O)NCC1CCCC1N(C)C)NC(=O)C(O)C=CC N1(C(C2CCC(=O)C2)=O)C2CCC1C1CC1(NC(=O)Cc1sc(O)nc1O)C2 C1(CC)CN(C(C2(C)COC2)=O)CCO1.n1(CCC)ccnc1C(F)(F)C(=O)N c1(C=O)cc([N+](=O)[O-])c(N)cc1F.C(C(C=O)NC(C)=O)OC.CC(C)C.N C1(C(N2CCC2CO)=O)CCCN1C(c1ccc(Cl)s1)=O.c12cn(nn1)C2 N1(C(C2C3CN(C(=O)Cc4cscn4)CC32)=O)CCCC(F)CC1 C1(C(N(CC(C)NC(c2c(C(C)(C)C)nsc2N)=O)C)=O)CC2CCC1O2 C(=O)(C(F)(F)C(F)(F)F)NC1(C)C(C)CN(CCN(C)Cc2ccccc2)C1 CCCS(=O)(=O)C(C)C(=O)N1CC(C)(C)OCC1CNC(C1CC(F)C1)=O C1CCCC2CC12.C(=O)(C(C)N(C)C)N(C)C.C1(C=O)C(C(F)F)C1(C)C c1(CC)ccccc1-n1nc(COCc2c(C)n[nH]c2C)nc1CC(C)C C1(C(=O)NCCCC)C(CO)=C(C)C1C.c1(C(=O)N)cn(C)nc1C1CCC1 N1(C(c2cc(C)oc2)=O)CCCC(N(C(=O)CCc2ncc(F)cn2)CCO)C1 c1(SC)cn(C)nc1C(=O)NC1CCCC1C.C1(CC(=O)N)CCCCN1C CC(CC(=O)N1CC(N(C)C(c2cc(=N)[nH]cc2Br)=O)C1)C(C)(C)C CCC(CCCC(=O)N1CC=CC1CF)NC(c1ccc(F)cc1F)=O C1(CCCCCNC(CC2C(C)C2)=O)CCN(C(=O)CN(S(C)(=O)=O)C)CC1 N1(C(C(c2ccn(C)n2)C)=O)CC2(CCN(C(=O)Cc3cncn3C)C2)C1 N1(C(CCCOC(C)C)=O)CCC(NC(=O)CCN(c2ccncc2)C)CC1C c1(CC)nc(Cl)nc(N2CCC(C3CC3)(C)C2)c1Cl.C1(CC(=O)N)CC2CC2C1 C1(O)(CC)CCN(C(c2cccc(=O)o2)=O)CC1.N(C)(S(N)(=O)=O)CC=O CC1CN(c2ccc(Cl)c(F)c2)CCN1N1CCCC(O)(c2ccccc2)C1 n1(CCOC)nccc1C(=O)N(CCC(C)NC(C1C=CCC1)=O)C O=C(C(CC1CCOCC1)NC(C1CC1Cl)=O)NCCC1CCSC1 c1(OCCNC(=O)Nc2cc3cc(O)ccc3[nH]2)cccc2c1OCCO2 Brc1ccc(-c2ccc(NCCc3cccs3)s2)cc1 C(C(C)(C)C#CC(=O)NC(CO)C(C)C)NC(c1cc(COC)on1)=O C1(C)(C(=O)NC2C(C(N(C)Cc3cccnn3)=O)COC2)COC(=O)N1 c1(NC(C(N2CC(COC)OCC2)CC)=O)ccc(Cl)c(F)c1 N1(C(COCC=C)=O)CCN(C(=O)C)CC1.C1(CC(=O)N)CC(C)(C)CO1 Cc1ccc(C(=O)NCC(C)N(C(=O)C)C)c(N)c1Br.C(C)(C)C.C(=O)N C(=O)(C(=O)N=c1ccn(CC#N)[nH]1)NC(c1cc(Br)cc(C)c1O)C c1(N(CC(C)NC(c2c([N+](=O)[O-])cnn2C)=O)C)ncc(C#N)cc1Br C1(NC(=O)C2CC2)CCC2CN(C(=O)Cc3ccn(C(F)F)n3)CCC2C1 Cc1nn2cccnc2c1CN(c1ccnc(N(C)CCN2CCOCC2)n1)C C(=O)(CC(C)(C)CC(F)F)N(C)CCN(C)C(C1CCCN1C(N)=O)=O C(=O)(C(F)CC(C)C)NC1CC(NC(c2ccc(OCC)cc2)=O)C1 N1(C(CN(C)C(=O)Oc2sccc2Br)=O)CCOC(C)(c2nn[nH]n2)C1 C#CCCCCCCC(=O)NC1CN(C(=O)CC(=O)OCC)CC12CC2 C1(CCC)(NC(=O)C(CC)n2nccc2C)CCN(C(=O)CCc2ccoc2)CC1 N1(C(CSc2ccn(C)n2)=O)CCC2CC(NC(=O)C=CS(C)(=O)=O)CCC2C1 CCCC(CCC)C(=O)NC1CC(NCc2cn(C)nc2C)C12CCC2 C(N=c1[nH]c2ccc(Cl)cc2s1)C1(NC(=O)C2=CC3(CCOC3)C2)COC1 C(=O)(CCCC(=O)C1CC1)N(C(C(=O)NC(COC)C)C1CC1)C Cc1nc(CCC(=O)NC(CNC(=O)C(C)(C)c2ccsc2)CC(C)C)[nH]c1C N1(C(C(C=CC)O)=O)CCCC(C2CCN(C(=O)CC(C)n3cccn3)CC2)C1 Cc1cccc2cc(C(=O)NCC3(C)CCN(C(=O)C=C(Cl)Cl)C3)nn12 C1(C(=O)NCc2ccc(C)s2)CN(C(c2cnsc2C)=O)CC1(F)F CCCCCCC(CC)C(=O)NC1CN(C(=O)Cc2ccc(Cl)c(C)c2)CC1C Cc1cn2c(=O)c(NC(=O)C(C)C(F)(F)F)cnc2s1 CC(C)CS(=O)(=O)CCC(=O)N(C)CCN1CCN(C(C23CC(F)C2C3)=O)CC1 CN1CCN(C(C2(CCNC(C3CCC(C)(O)CC3)=O)CC2)=O)CC(O)C1 C1(NC(CCCC)=O)CN(C(=O)C(CC)c2ccccc2)Cc2nccn2C1 C#CCC(C)(CC)C(=O)NCC(CC(C)C)NC(c1ncn2ccccc12)=O C1(CC)(NC(=O)CN2CCC(C)(C)C2)CCN(C(C2(F)CC2)=O)CC1 CC1C(NC(C2(O)COC2)=O)CCCN1C(c1ccc(Cl)c(N)c1)=O C(=O)(C1=NOCC1)N(C1CCN(C(c2cnn(C)c2COC)=O)C1)CCC N1(C(c2nc(C)c(Br)cc2)=O)CCC(NC(c2ccc(O)cc2O)=O)C(C)(C)C1 C1(CC(=O)N)CCOCC1(C)C.c1(CC)nocc1C(=O)NC1(CC)CCC1 N1(C(C=C(COC)C)=O)CC2CC1(C(N1CCC(C(C)OC)CC1)=O)C2 c1(N2CCC(N(C(c3cc4ccsc4s3)=O)CC)C2)ncnc2cccnc12 C(=O)(C1=COCCO1)NCC1(F)CC(NC(Cc2ccc(C(C)C)cc2)=O)C1 c1(C(=O)NC2(CNC(=O)CC(Cl)Cl)CCOC2)nc[nH]c2ncnc1-2 n1(CC)cnc2[nH]c(=NC3CC(F)(F)C3)nc(N(C)CC3CCCCO3)c12 CC1CC(CNC(c2n[nH]cc2-c2ccncc2)=O)CN1C(=O)Cn1cnnc1 C(C(=O)N1OC2CCC1C2)(C(C)OC)NC(C(CC=C)(F)F)=O CC(C)C(O)CNC(=O)CC1(NC(=O)Cc2cnn(C)c2)CC1 C1(C(=O)NC(C)(C)CC(=O)N2CCCC(CCO)C2)CC12CCOCC2 c1(OC)ccc(F)c(C(=O)NC2(C)CN(C(c3cnn(C)c3C)=O)C2)c1 c1(C(=O)N)cccc[n+]1[O-].CCCCN(C(C1CC(N(CC)CC)C1)=O)CC C1(CNC(c2cnc(C(F)(F)F)s2)=O)CN(C(=O)CC2CC2)C2CC12 N1(C(C2(COC)CC=CC2)=O)CC2CC(C(N3CCCC(F)(F)C3)=O)C(C2)C1 CC1C(NC(c2ccn3ccccc23)=O)C(C)CCN1C(C1CCOC1)=O c1(OC)cc(N)ccc1C(=O)NC1CN(C(=O)C(C)(C)C(N)=O)CC1(C)C c1(-c2cc(C(N(CCCNC(C3CC(C)(O)C3)=O)C)=O)on2)cccc(F)c1 C1(CN(C2C=CCCC2)Cc2cccs2)CC12CCCCC2 N1(C(C2N(CC(C)C)CCC2)=O)CCN(C(=O)CC2CCOC2=O)C2(CC2)C1 Cc1ncc(C(=O)NC23CCC(CC2n2cc(C(O)C(C)C)nn2)C3)c(C)n1 N1(C(CC2(C)N(C(CC(C)C)=O)CC2)=O)CCC(N=[N+]=[N-])C1 N1(C(C=CCC)=O)CCN(C(c2ccc(C)c(C)n2)=O)CC1CC(F)F c1(C(=O)NCC2CCCCN(C(C3(CC)CC3(F)F)=O)C2)cccc2c1COC2 c1(C(N(CC(O)CNC(C2Cc3nncn3C2)=O)C)=O)n[nH]c2c1CSCC2 C1(C)(C(=O)NCCOCCC(=O)N(C(c2cc(C)on2)C)C)CCNC1=O c1(OC)c(C(=O)NCCOCCN(C)C(C2CCSC2)=O)cnn1C Cc1c(C(=O)NCC2CC(C)N(C(=O)C)C2)cnn1C1CCOCC1.C1CC1 N1(C(C2CCCC(C)C2)=O)CCC2CN(S(=O)(=O)C3CC3)CCC12 C(=O)(C(C(C)C)n1cncn1)NCC1CC(NC(C(C)=C(CC)C)=O)C1 CC(C)(C)C(C(=O)NC1(C)CCN(C(c2cnsn2)=O)C1)C1CCC1 C12(C(=O)NCC3(F)CCN(C(C4(CF)CC4)=O)C3)CCCC(CO1)C2 c1(N2CCC(C)(CC)C2)ncnc(NCc2cc(-c3ccco3)on2)c1C C1(C=O)CC12CCC2.C1CC(=O)N(C(C)C)C1.Cc1ocnc1CC(=O)NC C1(C(=O)NCC2C=CC(NC(Cc3c(C)scc3)=O)C2)CCc2nncn2CC1 C12(CNC(CCCN(C)C)=O)CC3CC(CC(C3)C1NC(=O)C(C)(F)F)C2 Cc1cn2c(n1)CC(C(=O)NC1CN(c3nc(Cl)c(C#N)s3)CC(C)(C)C1)CC2 Cc1[nH]nc(C(=O)NC(CCNC(C23CCCCC2C3)=O)C(C)C)c1O C12(C(=O)NCCOC)CCN(C(c3cc(C)ccc3C)=O)CC1C2 Cc1cc(F)cc(C)c1C(=O)NCCC1(O)CCN(C(=O)C(C)(O)C(C)C)C1 Cc1nc(C(F)(F)F)ccc1C(N1CCCC(CCC(F)(F)F)C1)C(=O)NC1CC1 C12CC(CO1)C2.c1(C(C)(C)C)ncc(C(=O)N)[nH]1.C(C=C(Cl)Cl)=CC=O N1(C(c2c(C)onc2)=O)CCCC(C2CCCCN2C(=O)CSS(C)(=O)=O)C1 c1(C(=O)NCCCOCCNC(CCc2cc(C)[nH]n2)=O)nn(C)cc1Cl CC(C)CCN=C(NCC1(OC)CCCS(=O)(=O)C1)NC1CC1C1CCCCC1 C=CCC(CC)C(=O)N(CCCNC(=O)C(O)CC(C)C)CC1CCCC1 C1(NC(c2c(COC)noc2)=O)CCCCC1.C(=O)CCC(=O)N(C)C(C)C N1(C(C2(N(C)C)CC2)=O)CC2CCC(NC(c3nccc(N)c3Cl)=O)(C2)C1 C1(NC(c2cnsn2)=O)(CO)CCCN(C(=O)C2=COCC2)C1 c1(C(C)NCc2ncn(-c3ccccc3)n2)ccncc1Cl c1(OCCCC)ccc(C=NOCC(=O)OCC)cc1Oc1cc(F)ccc1F Cc1nn(C)c2c(N(CC(C)(C)S(C)(=O)=O)C)nc(=NCc3ccsc3)[nH]c12 c1(COC)ccc(C(=O)NC2CC(CCn3cc(C(C)(C)F)nn3)C2)cc1 N#Cc1ccc(Cl)c(C(N2CC3CC2C3NC(=O)Cn2nc(Cl)ccc2=O)=O)c1 C1(C(=O)NCC2C=CCN2C(=O)CC2CCC=CCC2)CC2CC1CC21CC1 C1(NC(c2ccccc2Br)c2n(CCCSCC)nnn2)C2CCC(F)(F)C12 C(=O)(CC(C)P(C)(C)=O)NCC(C)CNC(C12CC(F)(C1)C2)=O C1(CC)(NC(=O)CCNS(C)(=O)=O)CCCN(C(=O)CC)C1.C1COC1 Cc1ccc(C2=NOC(CNC(N3CCCC(F)(CN(C)C)C3)=O)C2)cc1 C1(C(N(CC)CC)=O)CN2CC3CC2(CO1)C3 N1(C(C)=O)CC2(C1)CN(C(c1ccc(CNC(C3CC(F)C3)=O)o1)=O)C2 N1(C(c2cc(CC)no2)=O)CC2CC(C)N(C(=O)CCCOC(C)=O)C2C1 n1(CC(=O)NC2CCC(CNC(c3ccc(C(F)F)o3)=O)C2)cnnc1O Cc1cc(N)ccc1C(=O)NCC1CC1NC(=O)CC1CC(F)C1 c1(COC)ccc(C(=O)NCC2C=CCN2C(=O)COC(F)(F)F)s1 C(=O)(CCCCC1CCCCC1)NCC(C)NC(CN(S(CC)(=O)=O)C)=O c1(NCC(c2ccc(C)cn2)(C)C)nccc(=NCC(C)C(C)C)[nH]1 C(=O)(CCCC(=O)N(CCCNC(=O)C(O)C(F)(F)F)CC)OCC Cc1oc2ccccc2c1CC(N1CCCCCC(NC(c2cnc[nH]2)=O)C1)=O c1(NCC(COC)(C)C)ccc(S(=O)(=O)NCc2ccc(Cl)cc2F)cc1F c1(NC(=O)NC2CCSC2)ccc(-n2ccnc2O)cc1 CCCC(C(=O)NC(C1(C(=O)O)CC1)=O)NC(=O)Cn1cc(CO)nn1 CCCCCCC(=O)N1CCCC(C)C1CCNC(c1cc(OC)ncc1Cl)=O C1(N(C(c2n[nH]c(C3CC3)c2)=O)C)CN(C(=O)C(O)C2CCC2)CC12CC2.CC C1(NC(c2cn(CC)nc2)=O)C2CC1N(C(=O)C(O)C(C)C)C2 c1(OC)cc(C)cc(C(=O)NC(C)C(C)C)c1O.C1(C)(C(=O)N)C=CCCC1 CC(C(=O)OCc1ccccc1)S(N)(=O)=O.C12CC(C1)CCOC2=O C1(CNC(C(Cc2cnc[nH]2)NC(CC)=O)=O)COCC(=O)N1C c12cnc(F)cc1C(=O)N2.C(=O)(C#CC(=O)O)NCCCOCC CC1CC(C)CC(S(=O)(=O)N2CCN(Cc3cscn3)CC2)C1 S(=O)(=O)(c1ccc(C(N2CC(CO)(C)C2)=O)cc1)NCC.c1cccc(C)c1 C(CNC(c1onc(C)c1C)=O)(CC(F)(F)F)NC(c1cc(C)on1)=O N1(C(c2ccc(CO)o2)=O)CCN(C(c2cncn2C(F)(F)F)=O)C(CO)C1 C1(C(=O)NC(C(=O)NC2(CC=C)CC2)C)CNC(=O)C1 N1(C(C2C(C(=O)OC)C2)=O)CCCC(C)(C)C1.C(=O)CC=CC(C)(C)C Cc1ccc(F)c(C(=O)NC2CCC(C(=O)N)OC2)c1.c1cnn(C(F)(F)F)c1 c1(C(=O)NC2C(NC(=O)C#CC3CC3)CCOC2)cccc2nonc12 C(=O)(CCC(C)(F)F)N1CCC(C(C)NC=O)C1.c1cn(-c2ccccc2)cn1.C C1(NC(c2nc(CC)sc2)=O)(CO)CCCN(C(=O)Cn2nc(C)oc2=O)C1 c1(COC2CC(C(=O)NCc3ccc(C)cc3)C2)nc(Cl)ccc1F CCC(C(=O)N1CC(CC(C)NC(=O)C(C)NC(C)(C)C)C1)NC(N)=O c1(SCC)cccc(C(=O)NC2CCC2CNC(C2(O)CCCC2)=O)c1 N12CC3CC1(C3)C2.C1(C(=O)O)CC(F)(c2cn(CC(F)(F)CO)nn2)C1 Cc1cc(Cl)c(C(=O)NC2CN(C(c3cc(F)cs3)=O)CC2C)cc1F c1(C=O)cnn(C(C)C)c1N.c1(C(C)NC(C(Br)=C(C)C)=O)ccccc1F.N C(C(CC(C)C)C(=O)NCc1ccsc1)NC(C(C)(C1(C)CC1)OC)=O C(=O)(C(F)(F)C(F)F)NC(C1CCN(C(c2[nH]cc(-c3nc(C)sc3)c2)=O)C1)C c1(C(=O)NCCN(C(C2C(CC)OCCC2)=O)C)nc(Cl)c(Cl)c(N)c1Cl c1(OC)cccc(C(=O)NCC23CC(C2)C3)c1Cl.C(=O)CCCn1ccnc1 CC1(C)CC(O)(CC(=O)NC2CC(CCNC(c3ncc[nH]c3=O)=O)C2)CO1 C1(NC(CC(COC)COC)=O)CC1C1CCN(C(c2cc(C#N)cs2)=O)CC1 N1(C(c2c(N(C)C)cccn2)=O)CC2(CCCCN2C(=O)C=CS(C)=O)C1 Cc1cc(F)c(CC(=O)NCC2CCN(C(C3CCCCS3)=O)CC2)cc1F Cc1cc(C)n(C(C)C(=O)NC2CCN(C(=O)C(C)(C)F)C2)n1 N1(C(CCC2CCC(=O)C2)=O)CCC2CC12C(N1CCCCC1)=O c1(C(N2CC(NC(=O)CC3CC=CC3)C(C3CC3)C2)=O)ccc2c(n1)CCCC2 C#CCCCC(=O)N(CCNC(=O)CC1CC2CCC1C2)Cc1ccc(Cl)nc1 O=S(=O)(c1ccc(Br)cc1NC1CC1)N1CCCC(OCC(F)F)C1 C1(c2cc(C(C(F)(F)F)(F)F)ncc2)CC12CCCc1ccccc12 c1(CC=O)ccccc1.c1(COC)cc[nH]c1C(=O)NCC1(F)CCC1 C=C1CCC(C(N2CC3CC3C2C(=O)NCC2SCCS2)=O)CC1 N1(C(C=CCCC)=O)CC(N(C)C(c2ccsc2Cl)=O)C2(CC2)C1 C1(NC(c2ccc(=N)[nH]c2)=O)CC2CCC(C1)N2C(=O)C#CC1CCOC1 N1(C(c2c(C)cn(C(C)C)c2)=O)CCC2C(CCCN2C(C2CC(C)(C)C2)=O)C1 C1(NC(c2occ(C)c2C)=O)CC2(CCN(C(C3CC(=C4CC4)C3)=O)C2)C1 C1(N(C(=O)C=Cc2cc[nH]n2)C)CCN(C(=O)CCC(=O)N(C)C)CC12CC2 C(c1cccc(F)c1)=CC(=O)NCCCN(C(=O)CCc1cc[nH]n1)CC n1(CC(C)C)[nH]c(CC(N2CC(NC(=O)CCC3(C)N=N3)CC2C)=O)cc1=O c1(C(=O)NCC2CC(NC(C(CC)F)=O)C2)cc(O)c2nc(C)n(C)c2c1 O(CP(C)(C)=O)CC(=O)N(CCC(C)NC(=O)C(c1ccccc1)F)C C(=O)(C(F)(F)C(C)O)N1CCC(OC)(CNC(=O)CS(C)(=O)=O)C1 c1(C(=O)NC2(COC)CN(C(C3(CC=C)CCOC3)=O)C2)sc(C)nc1C Cc1ccc(C(=O)NC2CC(C)C2(C)C)c(C)n1.c1(C=O)ncoc1C(C)C Cc1[nH]c(C)c(C(N2CCC(CC(N3CC(CC(F)(F)F)C3)=O)C2)=O)c1C C1(C(=O)NCc2ccc(O)nc2)CC2CC(C1)N(CCN1CCCC1=O)C2.C CC1(CNC(C2CCN(c3nc(=N)[nH][nH]3)CC2)=O)CSCCO1 c1(C(=O)NC2C3CC2N(C(c2cnc(Br)s2)=O)C3)ccc2occc2n1 N1(C(C(C)=C(C)C)=O)CCCC(C(C)NC(c2csc(Cl)n2)=O)C1 Cc1snnc1C(=O)N(C)CCNC(c1ccc(C(C)(C)C)[nH]1)=O C1(C(N2CCC(CC=C)C2)=O)CCCCCCN1C(=O)CCC1CC(C)C1 C1(CCOC)(NC(=O)C2=CCC2)CCN(C(=O)CC2CCN(C)CC2)C1 S(=O)(=O)(C1C2CCCCC12)NC(c1ccc(F)cc1Br)CC(=O)O C=CC(C)CC(=O)NCCCCN(CCCNC(c1coc(Br)c1)=O)C C1(C(N2CC(C(C)NC(C(CCOC)OC)=O)C2)=O)CC2(CCO1)CC2 c1(C(CCNC(=O)NC(c2nnc(C)s2)C)O)ccc(Cl)c(Cl)c1 c1(C(=O)NC2C(CNC(CC(=O)N(C)C)=O)C2)c(Cl)oc2ccccc12 c1c(C(=O)N(C(C)C2CC2)C)cccc1Cl.C(=O)(C(C)C)N(CC=O)C.C c1(-c2cn(CC(C)NC(c3ccon3)=O)nn2)cccc(C2CC2)c1 C=CC(CCC)CC(=O)N1CCN(C)C(C(=O)N(C)CC2(CO)CCC2)C1 CC1CCC(C(=O)NCC23CC(F)(C2)C3)N(C(=O)Cc2cc[nH]n2)C1 n1(CC)nc(CNC(=O)CC2CCC(N)CC2)cc1C CCC(CC)CCCC(=O)NC1CN(Cc2csc(N3CCCCC3)n2)CC1C C1(NC(C=C(C)CN2CCOCC2)=O)CCCC1.C1(C(=O)N)(C(N)=O)CC1 C1(CNC(c2onc(C)c2C)=O)C(O)C(O)CN1C(=O)CCc1ccn(C)n1 C1(C(=O)NC2(CCOC)CCOC2)C2CC(C(O)C2O)S1(=O)=O C(=O)(CC(C)(O)COC)NC(CNC(c1cnc(CC)s1)=O)(C)CO c1(C(N(CCN(C(c2cc(SC)oc2C)=O)C)C)=O)c(F)cc(N)cc1F c1(C(N(C(CNC(c2nonc2N)=O)C2CC2)C)=O)c[nH]c(=O)cn1 CC1=CCC(C(N2CCC(CCC(=O)N(C(C)CC(C)C)C)C2)=O)CC1 C1(CNC(c2cnncc2O)=O)CC2(CO1)CN(C(c1cccc(Cl)n1)=O)C2 c1(CN(c2cnn(C)c2)C(c2c(C)coc2C(C)(C)C)=O)c(OC)cccc1C c1(N2CC(CN(C(c3cc(C)cc(F)c3)=O)C)OCC2)ncnc2cccnc12 c1(C(=O)NCCC(C)CCNC(C2CC23CCOCC3)=O)cnc2ccsc2c1 c1(CC)ccc(C(N2CC(NC(=O)CN3CCS(=O)CC3)C(C)C2)=O)nc1 C1(NC(C(CN(C)C)c2ccccc2)=O)C2CC1N(C(=O)CCn1cnnn1)C2 C1(C)(OC)CC2CC1CC2NC(=O)N(C(C)C)Cc1ccsc1 C(C(C(=O)NCCC(C)NC(C1(c2ccno2)CCC1)=O)OC)OC c12nc(Cl)c(s1)C(C(=O)NC(C)C)N2C(C)C.c1ccccc1.CC(=O)N CC(C)CC(C(=O)N1CCC(O)(CN(C)C)C1)N(C(=O)C(C)n1ccnn1)C N1(C(c2nc(Cl)cs2)=O)CCCC(C2CCCN2C(=O)C)C1.C1CC(F)(F)C1.O Cc1oc(C(C)(C)C)cc1C(N1C2CN(Cc3cc(C)n(C)n3)CC12)=O C1(C(=O)NCC2C(CC)CCN2C(=O)C(=O)N(C)C)CC2CCC1CC2 c1(CN2CCC(C(C)C(=O)NC(=S)Nc3cccc(Br)c3)CC2)cc(O)ncc1Br c1(C(=O)NCC2C(NC(=O)Cn3cccn3)C2)ccc(C2CC2)cn1 CCN=c1cc(C(=O)NCC(C2CC2)N(C(=O)C2=CCSC2)C)cc[nH]1 c1(C(=O)NCC(C)N(C)C(C2CN(C)C2)=O)cc2c(s1)CCC(C)(C)C2 c1(C(=O)NCc2cccc(NC)c2)ncc(Br)cc1F C1(NC(CCN(C(=O)CN2CCCCC2=O)CC)=O)CC(=O)NC1=O O=CCO.C(C(F)F)C1(C(=O)N(CC2(CO)CC2)C)CC1.C1CC1 Cc1nnc2n1CC(C(=O)NCCOC1CN(C(c3coc(Br)n3)=O)C1)CC2 CCCCCCC(C(=O)NC1CC(F)(F)C1)N(C)CC1(OC)CCCC1 c1(C(=O)OC(c2ncc(C(C)(C)C)o2)C)cc2c(s1)CCSC2 c1(CC)cc(C(N2CCCC(N(C)C(C3CCN(C4CC4)CC3)=O)C2)=O)sc1C C1(OCC(=O)N(C)CC)CCN(C(=O)CNS(N)(=O)=O)C1.c1ccoc1 C1(NC(C(CC)N(C)C)=O)CC2CCC(C1C)N2C(c1ccc(O)cc1O)=O C(=O)(C#CC1(C)CCCO1)N1CCCC(CCNC(Cc2cc(CC)no2)=O)C1 CC(C)CC(C)C(=O)NC1CCN(C(C2(CF)CC2)=O)CC1O C(=O)(C1CCCc2nncn21)NC1CCC(NC(CCc2n(C)cnn2)=O)CC1 C1(CC)CCCCC1NC(C1(CNC(c2nsnc2O)=O)CCCCC1)=O C(=O)(C1CCCc2nc[nH]c21)NCC(C(C)C)C.c1(C(=O)N)cc(C(N)=O)[nH]n1 C1(C(N2CCC(C(c3ccccc3)C)C2)=O)CCC2(CCNCC2)C1 c1(OC)cc(C(=O)NCc2cc(O)c(O)c(F)c2)c2ccccc2c1 c1(C(=O)NCC2C(C(N(C)Cc3ccccn3)=O)CCC2)cc(O)ncc1F N1(C(C=CC)=O)CCC2CN(Cc3ccc(OC)c(Br)n3)CC12 CN1CCCCC1CCC(=O)NCC(O)CCNC(=O)CCc1ccc(F)cc1 c1(C(N2CC3C(C2)N3c2nccc(N3CCCC3)n2)=O)cccc(I)c1O c1(CCNC(COC)(C(C)C)c2nnnn2C2CCOC2)cc(Br)ccc1OC Cc1cc(C(=O)NC2CN(C(=O)C(O)CN(C)C)C2)c(C)c(C)c1 C1(C(=O)NCCC(=C)CNC(=O)C(C)CCN(C)C)CCCC(=O)C1 c1(C(=O)NC2CN(C(c3c(Cl)cn(C)n3)=O)C2)cc(Br)ccc1O c1(C(=O)NC(C)CNC(=O)C(C)Cc2ccc(F)cc2F)ccc2cncn2c1 N1(C(CCn2ncc(C)c2)=O)CCCC(NC(=O)CCc2cnoc2)CC1 N1(S(C)(=O)=O)CCC(C(=O)NCC2CCCCC2)CC1.c1(C=O)cccs1.C C12(C(N3CC4C(CNC(CCCC#N)=O)C4C3)=O)CCCC(=O)N1CCC2 C#Cc1ccnc(C(=O)NCC2CCN2C(=O)Cc2ccn(CCOC)n2)c1 c1(C(N2C(CNC(C3C(C)(C)C3)=O)CCCCC2)=O)ccc(C#N)c(O)c1 c1(NC(=O)OCC#C)cc(N(C)C(=O)OC(C)(C)C)ccn1 C1(NC(C(C=CCCC)O)=O)CCC(O)CN(C(=O)CN(C)C(C)C)C1 N1(C(c2c(C)cnnc2)=O)CCC(C)C(NC(=O)C[SH](=O)=O)C1.C(C)(C)(C)N c1(NC(CNC(C(C=C)O)=O)C(C)C)ncnc2c1nnn2C1CC1 c1(C(N2C(CCNC(c3nccs3)=O)CCCC2)=O)cc(F)cc2cc[nH]c12 C1(NC(CC=C(C)C)=O)CC(C(=O)N(CC(C)C#N)C2CC2)C1(C)C N1(C(CC2(NC(c3c(C#C)c[nH]n3)=O)CCCCC2)=O)CCN(C)C(=O)C1 C(=O)(C(C)S(C)(=O)=O)N1C2C(NC(COCC)=O)C(C2)C1 N1(C(C2N(C(CC(CCC)C)=O)CC2)=O)CC(=O)N(C)C(C)C1 c1(C(N2CC(COC)N(Cc3cnccn3)CC2)=O)ccc([N+](=O)[O-])c(C)c1 c1(C(=O)NCC(C)(CNC(C2CC(C)CO2)=O)OC)cccc(Cl)c1 C1(NC(C=Cc2n(CC)ccn2)=O)CC(O)CN(C(C23CC2COC3(C)C)=O)C1 C1(C)(CC=O)CCCCC1.C=CC1(CC(=O)NCC2(O)CC(C)C2)CCC1 N1(C(C=C(C)C)=O)CCC(c2ccc(F)cc2)C(CC)C1.c1(CC=O)csc(Br)c1 CCCC(C(=O)NCCCOC)N1CCC(C(=O)N(c2ccccc2)C)CC1 O=C1NC(C(=O)NCC2(NC(=O)CC3CC3(Cl)Cl)CCC2)CO1 Cc1cnn(C)c1C(N1CCCCC1)=O.N1(CC=CC(=O)N(C)C)CCCCC1 c1(NC2C(C)(C)C(NC(c3cnc4cc[nH]c4c3)=O)C2)ncc([N+](=O)[O-])cc1Br c1(-c2nnco2)ccc(Cl)cc1Cl.C(=O)(C(C)CC1CC(F)(F)C1)N(C(C)C)C C1(NC(C(C)CC(N)=O)=O)CN(C(c2cocn2)=O)CC2(CCC2)C1 c1(NCC2N(C(C)=O)CCC2)[nH]c(=NCc2cccnc2C)nc2sccc12 C12(C(=O)NCC(CNC(C(N3CCOCC3)C)=O)O)CC(F)(C1)C2 CC1CN(C(C2C3CC4C(C3NC(=O)CCN(C)CCO)C24)=O)CC(=O)N1 Cc1ccncc1C(C)(C)C=O.C1(C(N(CC(C)(C)C)C)=O)CCC(C)(C)O1.N C(=O)(CC(C)O)N1CC(F)C1.C(C)(C=O)=CN(C)C.C(C)(C)C.C=O.N Cc1nccnc1C(=O)NC1(CO)CCN(C(c2csc(C3CCCO3)n2)=O)C1 C1(OC)CCC(C)(C(N2CC(C(N3CCC(OC4CCC4)C3)=O)C2)=O)CC1 n1(CC)cnc2nc(N3CCC=C(C)C3)nc(NCCc3c(Cl)cncc3Cl)c12 C1(NC(c2n(CC)cc(Cl)c2)=O)CC2CCC1CC2.c1(C(=O)N)ccnc(O)c1 Cc1cc2cc(C(N3CCC(C)(CNC(=O)C(C)O)C3)=O)oc2cc1C Cc1nc(C(=O)NC2CCN(C(=O)CCN3CCCCCC3)C2)nn1C N1(C(c2c(NC)scn2)=O)CCN(C)C(CNC(C2CCCN2C)=O)C1 c1(OC)cnc(F)cc1C(=O)NCC1C(C)CCCN1C(c1cncnc1)=O c1(CSC)ccc(C(N2CCN(C(=O)CCC3CCCN3C)CC2)=O)cc1 S(=O)(=O)(c1c[nH]ccc1=NCC1CCC(C)(C)CC1)N(C)Cc1ccccc1 c1(C(=O)N)cc2cccc(Cl)c2[nH]1.C1(CCOC)CCN(C(C2CC2(F)F)=O)C1 C1(C(=O)NCC(CO)OC)CCN(C(=O)CN2C(=O)CNC2=O)C1C c1(OC)nc(C(=O)N(CCCN(C)C(C2CC2C)=O)C)ncc1F C1(NC(C(C)C)=O)CCCN(C(=O)NC(c2ccccc2)c2ccccc2)CC1 c1(OCCOC)ncc(C(=O)NCCc2ccc(C)s2)cn1 CC1(C)OCC(N=c2[nH]c(=NCC3(C)CSCCO3)[nH]c3cc[nH]c23)C1 N#CC1(C(N2CC3CCC2C(NC(C2CCSCC2)=O)C3)=O)CC2C=CC1C2 N#Cc1ccc(C=CC(=O)NCC(CNC(C2CCCCO2)=O)CO)cc1 C1(N2C(COC)CCC2)CCN(C(=O)C(C(C)C)c2ccccc2)CC1 C=CCCC(C(=O)NCC(COC)C(C)C)NC(c1csc(=N)[nH]1)=O c1(NC(C2(C)CN(C(C3CCCN(C)C3)=O)C2)=O)cc(Br)cc(F)c1C#N C1(C(=O)NC(CN(c2c(C(=O)OC)cncc2)C)C)CC12CCOCC2 C(=O)(C#CC1CCOCC1)N(CC(C)N(C(C(=O)Nc1cccc(C)c1)=O)C)C c1(C(=O)NCc2cccc(CNC(=O)CCN3CCC3)c2)cc(Cl)ccc1O C1(NC(c2n(C)cc(Cl)c2)=O)CC(CNC(c2sccc2C)=O)C12CCC2 c1(N2CCC(NC(C3CC(=O)N(C4CC4)C3)=O)C(O)C2)ncc2cccnc2n1 N1(C(C(=O)Nc2cc(OC)c(Cl)cc2)=O)CCc2[nH]nc(C(F)F)c2C1 N1(C(CSCCCC)=O)CCN(C(c2ccc(CNC(C)=O)s2)=O)CC(O)C1 C(=O)(CCN=C(NCC(=O)NC(C)C)NCc1ncccc1Cl)NC(C)C c1(C(=O)NCC2CCC(C)CN2C(=O)CCF)ccc2cnnn2c1 N1(C(CCC2C(C)C2)=O)CCC2CC12CN(CCCCn1ccnc1)C(C)(C)C c1(C(=O)NC2C(CNC(C(n3ccc(C)n3)C)=O)C2)onc(Br)c1C N1(C(C(NOC)=O)=O)CC(NC(c2cnn(C)c(=O)c2)=O)C(C2CC2)C1 N1(CC)CCN(CC(=O)N)C(=O)C1=O.C1(CC=O)CC2(CCC2)C1.C(C)CC N1(C(Cc2ncsc2)=O)CCC(O)(CC)C1.C(=O)CCN(S(C)(=O)=O)C.C c1(C(N(CCCNC(=O)CN=S(C)(C)=O)CC)=O)cc2c(Cl)cccc2nc1C N1(C(Cc2scc(C)c2)=O)CC(CNC(C2CC2CN(C)C)=O)C(O)C1 N1(C(c2c(C)nc[nH]2)=O)CCCCC(NC(c2cnoc2-c2ccccc2)=O)C1 C1(N(C)C)CC(C(N2CC(OCCC(=O)NC3CCC(O)CC3)C2)=O)C1(C)C C1(NC(Cc2cn(CC)nn2)=O)CCC(C)N(C(c2coc(C)c2)=O)C1 N1(C(c2cccs2)=O)CCC2C(CCCN2C(c2cccc(O)c2Cl)=O)C1 c1(C(C)=O)cc(C(N2CC(NC(=O)C(C)CC3CCC3)CC(F)C2)=O)ccc1O c1(CNCC2(NC(c3cc(F)nc(F)c3)=O)COC2)cc(F)c(F)cc1Cl CCCC(CCCNC(C1CC(SC)C1)=O)NC(=O)CC(F)F N1(C(C=C(CC)C)=O)CCC2(CC1)OCCC2NC(C1CC=CCC1)=O C=CC(C)(O)CC(=O)N1CCC(N(C)C(c2cc(OC)ccc2OC)=O)C1 C(CC(C)C)(c1ccccc1)NC(COCCOCC)=O.c1nc(O)sc1C.N C1(C(=O)NCC(C)(CO)NC(CCOCCC)=O)CCc2nc(C)sc2C1 CC(c1cnn(C)c1)=CC(N1CCC(NC(C2CCCOC2C)=O)C1(C)C)=O c1(NC(C2C(OCC)C2C)=O)cccc(NC(=O)Cc2ccccc2)c1.S C1(NC(CN(C2CC2)CC)=O)CCN(C(C2CN(C)CCN2C)=O)C(C)C1 c1(C2(C(=O)NC3CC(C)C3)CC2)cc(F)cc(Cl)c1.C(=O)(C(Cl)=CCl)N C1(NC(c2cn(C)nc2C2CCC2)=O)COC2(C1)CN(C(=O)C#CC1(C)CC1)C2 N1(C(C(C)SCC)=O)CCOC(C)(C)C1.c1(C=O)cn(C(C)(C)C)cn1.C Cc1ncc(Cl)cc1C(=O)NC1(CF)CCN(C(=O)Cc2cnn(C)c2)C1 N1(C(c2c(CC)nn(C)c2)=O)CCN(C(=O)C(C)N2CCC2)C(CC(=O)NC)C1 c1(C(c2nnnn2C)NC2C(C)(CC)C2)c[nH]nn1.c1ccnn1C.C1CC1 N1(C(c2ncn(C(C)C)c2)=O)CC2C(CNC(=O)C(F)=CC3CC3)C2C1 N1(C(c2n(CCC)ncc2)=O)CCN(C(C2CC2(C)C(F)F)=O)CC1C1CCC1 N1(C(=O)OCC)CCC(NCCOCCC)C1.C(=O)CCc1nncs1.N CCCC(C)CCCC(=O)N1CCN(C(=O)CC(C)(C)O)C(C2CC2)C1.C C(C1CCc2ncnn21)N1CCCC(NC(=O)CCc2ccccc2)C1 CC1CN(CCNC(=O)CC2COCCN2)CC(C2CC2)O1 c1(C(N2CC(CC)N(C(=O)Cc3cnns3)CC2)=O)cc2c(C)ccc(C)c2[nH]1 c1(C(=O)N(CC(N2CCC(OC)CC2)=O)CC(C)C)cc([N+](=O)[O-])c[nH]1 c1(C(=O)OC)cccc2c1NCCN(C(=O)NCC(C)(C)c1cccs1)C2 Cc1ccc(Br)nc1CNC(c1ccc(F)cc1)CC(=O)N1CCC(CO)C1 C1(CNC(CC(C)C(=O)c2cccc(F)c2)=O)CCc2c[nH]nc2C1 N1(NCC(C)OCCC)CCC(NC(C2CCN(C)C2=O)=O)CC1 N1(C(CCNC(COC)=O)=O)CC2C(c3cn(CC4CCCO4)nn3)C2C1 c1(C(=O)NC(C(=O)OC)C2CC2)ncn2cc(-c3cc(C)[nH]n3)sc12 c1(CN(C)C(=O)NC2CCCC2CCCF)ccc(OC(C)(C)C)nc1 C(=O)(CC(F)(F)F)NCC(CNC(CCNC(=O)NC)=O)O.C(=O)C n1(CC)cccc1C(N1CC(O)(C(F)C(=O)NCC(c2cnc[nH]2)C)C1)=O CCC(CC)C(F)C(=O)N1CCCC1CN(C(=O)C(=O)NC(C)C)C N1(Cc2ccc(C)[nH]2)CCC2(CC(C(=O)Nc3ccc(O)cc3O)=NO2)C1 C(=O)(C(C)(C)n1ccc(C2CC2)n1)N1CCC1.CC(C=O)OCC1CC1.N c1(C(=O)NCCC(C)N(C)C(c2cccc(Cl)c2N)=O)cccn2nccc12 C1(CC=C)(C(=O)NC2CC(CC)C2)CCCCC1.C1(C=O)CCS(=O)(=O)C1 CN1N=C(CC(=O)NCC2(C(=O)NCC(O)CF)CCC2)CC1=O CC1CCC(C(=O)NCC(C2CC2)NC(=O)Cc2cccs2)O1 C1(N(c2nc(C)c(C)s2)C(c2cc(C)[nH]c2)=O)CCNCCC1C C=CCN=c1[nH]cc(C(=O)N(C)CCN(C)C(c2ccc(CC(N)=O)cc2)=O)s1 c1(C(=O)Nc2ccc(C(C)=O)cc2)cccc(OC)c1OC(C)C Cc1cncnc1N1CC(NC(=O)CC2(C(F)(F)F)CC2)CC1C C1(NC(C2(C#C)CCCC2)=O)COC2C(NC(c3c(C)ncnc3O)=O)COC12 N1(C(c2c(SCC)cccc2)=O)CCCC(O)(CNC(=O)CCC(C)CC)C1 C(=O)(CCC=O)NC1CCC1.c1(C(=O)OC)csc(CC(C)C)n1.CC(C)C.N C1(NC(CCc2onc(CC)n2)=O)CC2CC1N(C(=O)Cc1sc(S)nc1C)C2 Cc1cccc(C(=O)NCC(=O)NC2CC(N(C)C(C3C(C)C3C)=O)C2)c1 CCC(CCOC)C(=O)N1CCOCC(NC(C2CCCN2CC(C)C)=O)C1 CCCC(CNC(=O)COCCC(C)C)C(=O)NOCC=C(C)C C1(CNC(CCCCC)=O)CC(CC)CN(C(=O)COc2ccc(F)cc2F)C1 CC1CN(C(=O)Cc2cocn2)CC(C)N(C(c2cc(C(N)=O)ccc2F)=O)C1 O=C1NCCCn2nc(C(N3CCC4COC4C3)=O)cc21 C=C(Cl)CCC(=O)N(CCC(=O)NCC1CC(C(C)C)C1)CC C12(C(=O)NC3(C=C)CCC3)CC(CN1C(=O)CCCNCC)C2 C(=O)(C(CNC(=O)CC1CCC1)N(C)C)N(CC#CC)CC#C CN1CCC(C(=O)NC2CN(C(c3nc(Cl)c(Cl)s3)=O)CC2(C)C)CC1=O c1(OC)ncc(C(=O)NC(C)C(C)NC(c2cccn2C)=O)cc1Br C1(CC(=O)N)CC=CCN1C.c1(C(C)NC(=O)CCC2CC2)nn(C)cc1O N1(C(CC2CCCC(C)C2)=O)CC(NC(=O)CNC(=O)OC)CC(C)(C)C1 C1(NC(C2C(C)OC(=O)N2)=O)CCN(C(C2CCCC2O)=O)CC1(C)C N1(C(C2CCC(C)S2)=O)CC=C(CNC(c2cnoc2C2CCOCC2)=O)CC1 c1(C(=O)NC23CCN(C(C=C(C)C)=O)CC2C3)nn(C)c2c1COCC2 C(C)(C(=O)N(CCC(=O)NCC(C)O)CC)OCC=C C(CCN(C)C(C1CNC(=O)N1)=O)C(C)C.C(C(=O)N)(OCC)OCC N12CC(C(C)(C)C1)CNC2=O.C#CC1CCC(OCC)C1.C(C)(C)C c1(C(=O)NCCN(C(=O)CCC2CC2C)CCC)cnc(SC)nc1 c1(SC)cc(C(N2CCCC(C)(NC(=O)Cc3nc[nH]n3)C2)=O)ccc1[N+](=O)[O-] c1(C(=O)OCC)cn2c(n1)CCC(N(C(=O)CC1CCNCCC1(F)F)C)C2 CC1CCCC(C)C1SCC(=O)NC(c1nccc(C(F)(F)F)n1)C c1(C(=O)N)cccc(S(=O)(=O)C(F)F)c1.C(=O)(CC1(C)CC1)N(C)CC C1(CNC(C2C(C)(C)CO2)=O)CN(C(C2CCOCC2)=O)CCO1 O=S(=O)(c1cc(F)ccc1F)N1CC2C(C1)N2Cc1c[nH]c2nccc(Br)c12 C#CCCCC(C)C(=O)NC1CC=C(C(=O)NCCC(CC)CO)C1 C(=O)(CCC(=O)NCC1CC(NC(=O)C(C(C)C)OCC)C1)OCC C1(CCNC(C2(C)CCCCO2)=O)CC(F)(F)CN1C(c1ccco1)=O C1(OC)CC2(C1)CC(C(=O)NCCNC(=O)C=Cc1ccccn1)C2 N1(C(Cc2c(C)non2)=O)CCC(C2N(C(=O)CC(=O)N(C)C)CC2(C)C)CC1 CC1CN(C(C2CC3C(C2)C3(C)C)=O)CCC1CNC(c1cnc(O)nc1O)=O N1(C(C(CCC)OC)=O)CC(C2CCCN(C(c3csc(CO)n3)=O)C2)C1 CON(CCC(=O)NCC(C)(F)F)C(=O)C1CC1OC(C)=O CC(C)C(C)CC(=O)NC1CCN(C(=O)COc2ccn(C)n2)C1 c1(C(=O)N)cnc(Cl)cc1N.c1(SC(C)C(=O)NC2CC2C)ccc(Cl)cc1 C(C(=O)NCCCCCCNC(C1SCC=C1C)=O)(C(C)C)SCC CN1CC(C(N2CCC(C(=O)NCCC3(C)CCOCC3)C(O)C2)=O)CCC1=O N1(C(c2cnc(OCC)s2)=O)CCCC(N(C)C(c2nccc(C)n2)=O)CC1 C(CC1=CCN(C(C2CCC(F)C2)=O)CC1)NC(c1ccc(OC)cc1Cl)=O C(=O)(C(=O)N=c1cc(C)o[nH]1)NC(CC1CCN(C(C(COC)(C)O)=O)CC1)C c1(C(N2CCC(F)(F)C2)=O)nccn2nccc12.C1(C(=O)N)CC12CC(O)C2.C c1(C(=O)N)ccc([N+](=O)[O-])cn1.C1(CCC(=O)N(CCCC)C)NC(=O)NC1=O C(C1CCc2nccn21)NC(CC(CCC)NC(c1sc(F)cc1C)=O)=O C1(NC(c2ccc(CCC)[nH]2)=O)C2CN(C(c3cc(OCC)no3)=O)CC12 c1(OC)cc(OC)cc(C(=O)OCC(C2CCNC(C)(C)C2)=O)c1 N1(C(c2c(C)nn[nH]2)=O)CC2CCC1C2NC(c1nn(C)cc1Br)=O N1(C(CC2OCC(C)(C)OC2)=O)CC2(CCC(CNC(c3cscc3Cl)=O)O2)C1 N1(C(CCc2cnn(C)n2)=O)CC(NC(C2COC(C)(C)O2)=O)CC(C)(C)C1 C(C(C)(C)CNC(c1ccsc1)=O)N(C(C1C(C)C1(F)F)=O)CC C(=O)(CC(C)(C)F)NCC(c1ccccc1)NC(C1(N(C)C)CCCC1)=O c1(C(=O)N)ccc(N)c(Cl)n1.C1(CNC(C2C(OCC)C2)=O)CCC1 Cn1ncc2c(=O)n(CC(=O)NC3CCCC3NC(c3coc(Cl)c3)=O)cnc12 N1(CC)C2CCC1CC(NC(=O)CCCc1nc(C)no1)C2 C#Cc1cccc(C(=O)NC2CC(C)C2)c1F.c1(C(=O)N)ccoc1CC(N)=O c1(C(=O)NCCC(=O)N(C)C)ccc(N2CCN(C(C3CCC3O)=O)CC2)nc1 C(=O)(C(CC1C=CCC1)N(CC)C(c1coc(Br)n1)C)NCCCOC.O c1(C(=O)NCCN2CCN(C(C=C3CCC(C)C3)=O)CC2)c(OC)cccc1Cl CN1CCC2CN(c3nnc(C45CC=CCN4CCC5)n3C)CCC12 Cc1nc2ncnn2cc1C(N1CC(CC(N)=O)OC(C)(C)C1)=O C(=O)(CCCCC(C)C)NCC1CC(CNC(CCc2occ(C)c2)=O)OC1 C(=O)(C(=O)C(C)(C)CC)N1C(C(=O)N)C(C)(C)CC1.n1(CC=C)cc(C)nn1 C(CC(C(C)(C)C)NC(=O)CC1CC1(Cl)Cl)N(C)C(C1(C(F)F)CC1)=O C1(NC(C2(COC)CC=CCC2)=O)CN(C(=O)C(F)=CCCF)CCC1CO C1(C(=O)N)CCCCC(=O)N1.CC(CNC(C1(CC(F)(F)F)CCC1)=O)CO c1(OCC)ccc(C(=O)N)cn1.C(C1CCCN1C)=CC(N1CC(CC)C1)=O c1(C(=O)NC2CN(C(C=CSC)=O)CC(C)C2)cn2c(n1)CCCC2 c1(CNC(C2C(NC(c3sccc3I)=O)CCC2)=O)cnc2[nH]ccc2c1 Cc1cc(C(N2CC(C(N3C(C)CCCC3C)=O)CC(F)C2)=O)ccc1Cl C12(C(=O)NCC(C)C(=O)NCC(c3cnc[nH]3)C)CC(C#N)(C1)C2 C1(C(=O)NC(CNC(CC=C(C)C)=O)C2CC2)Cc2cc(Cl)ccc2O1 c1(CNC2CCCN(Cc3c(C(C)C)nco3)C2)ccc2n[nH]cc2c1 N1(C(Cc2nnc(C)s2)=O)CCN(CC2(NC(C3CC=CCC3)=O)CC2)CC1 CN1N=CC(CC(=O)N(CCCNC(c2cnc(C3CC3)o2)=O)C)C1=O C(=O)(C(CC(C)C)N(C)C)N1CCC(CCNC(Cn2c(CCC)ncc2)=O)C1 CCCC(CCCNC(=O)CN1CCCCCC1)N=c1[nH]c(Cl)ncc1Br c1(OC)ccc(Br)c(C)c1C(=O)NC1CCCC12CN(C(c1snnc1C)=O)C2 Cc1nc(CN=C(NC(C)C)NCC(C)(C)C)[nH]c1C C(CC(=O)NC(CNC(=O)CCc1cnco1)C1CCC1)OCC(C)C c1(CN(C2C(C)OCC2)C=O)nc(C(F)F)nc(=N)[nH]1 C(CCCC(=O)NCc1ccccc1C)NC(C1(COC)CC1C)=O C(=O)(C(CC1CC1)NC(=O)CC1(O)CCC1)N(C(C)CC1CC1)C c1(C(=O)NC2CCCC2Cc2ccc([N+](=O)[O-])cc2)cccn2nncc12 c1(C(N2CCC(C(F)(F)F)C2)=O)ccc2c(c1)COC2.CS(=O)CCC(=O)NC c1(C(=O)NCC2C(NC(C=C(C)c3ccsc3)=O)CCC2)sc2cncn2c1C c1(OC)ccc2c(c1)CCCC2c1noc(C(CS(C)(=O)=O)C(=O)OC)n1 C(C(C)CC(=O)NCCCOCC(F)F)NC(c1c(CC)c[nH]n1)=O c1(CN2C(C(=O)Nc3ncc(F)cc3F)CC(O)C2)c(F)cc(I)cc1F C(=O)(CCCCCC(C)(C)C)NC1C(NC(c2cnn3ccc(C)nc32)=O)C1 CC(=O)CCCC(=O)N1CCC(C)(CNC(=O)CCO)C1.c1ccc(F)c(Cl)c1 C1(COC)(C)CCN(C(=O)C(O)CN(C)C)CC1.C1(C=O)CC(C)CO1.N C1(CC(=O)OC)CN(C(=O)C(C)(C)OCCCl)C2COCC2O1 c1(C(N(C2C3CN(C(=O)Cn4cnnc4)CC23)C)=O)cncc(-n2ccnc2)n1 C(CC(C)(C)C)(C(=O)NCC(O)CO)NC(COCCCC)=O C1(CNC(CCC(=C)Br)=O)CCC(F)(CNC(C2(C)CCCO2)=O)CC1 N1(C(c2ccc(SC)cc2)=O)CCC(O)C(NC(=O)CC2CC23CC3)C1 c1(C(=O)NC2(C)CCCN(C(=O)CC3C=CCC3)C2)ccn2ccnc2n1 N1(C(CCCC(=O)O)c2ccccc2)CCCC2C(O)CC12 C=C(C)C(C)(C)C(=O)NCCN(C(=O)COc1ccc(Cl)nc1)CCC CCC(CCC(=O)Nc1cccc(OC)c1)NC(=O)C=CC1(C)COC1 CC1(C)CCN(C(C2COCCO2)=O)C1CC(=O)NCCC1(O)CCCC1 C(=O)(C1CCc2ccccc21)NCC(CC)N(C(=O)C(C)C(O)C(C)C)C c1(C(=O)NC2CN(C(CC3(CS(C)(=O)=O)CC3)=O)C2)ccc(Cl)nc1 C1(NC(CC2N(C(C(=Cc3cn[nH]c3)C)=O)CC2)=O)CCCN(O)C1=O c1(OC)cc(CN=C(NCC2CC3CCC3C2)NC2CCS(=O)(=O)C2)cc(Cl)c1 Cc1cccc(NC(=O)C(=O)N(CCCNC(=O)Cn2[nH]cnc2=N)C)c1 N1(C(c2cccc(CC)n2)=O)CCC(NC(=O)CCc2ncc[nH]2)C(CO)CC1 O=C(C(C1=NOCC1)N1CCC(c2cccc(O)c2)CC1)NC1CCOC1 N1(C(C(C2CCCOC2)OC)=O)CCOCC1CN(C)C(c1cc(Cl)c(Cl)[nH]1)=O CC1=C(C(=O)N2C(C)CC3CN(C(=O)C(C(C)O)N(C)C)CC23)C(=O)OC1(C)C c1(NC)ccc(C(N2CCOC(CCNC(=O)Cc3nnc(S)n3C)C2)=O)nc1 C=CCCCC(C)NC(=O)C(CC1CCCC1)NC(=O)COC C1(C(=O)NC2C(NC(C(C(CC)O)C)=O)CCC2)CCc2c(nnn2C)C1 c1(CC(=O)N(CC)CC)c(C)[nH]c2ccc(F)cc12.C1(C=O)C(C)C1(F)F C(=O)(C(O)C(F)(F)F)NCc1c(C(=O)NC(c2ncccc2F)C)con1 C1(NC(CCC(=C)C)=O)CCOC12CCN(C(C1(CCF)CC1)=O)CC2 c1(C(=O)NC2CCCC(NC(c3cncs3)=O)C2)cnc2occc2c1 C(C)(CC(C)NC(c1ncoc1CC)=O)NC(CCC)=O Cc1nc(C(=O)NCCC2CSCCN2C(C2CNC(=O)O2)=O)c2ccnc-2[nH]1 C1(OCC)CCCC(NC(=O)NCC(Cc2cccc(Br)c2)CC)C1 C1(NC(Cc2nc(CC)sc2)=O)CCCN(C(=O)C(CO)N(C)C)CC1 C1(CC(=O)NCC(C(C)(C)C)NC(C(CCCC)O)=O)CC2CCC(C1)N2C C1(C=O)CC2CCC2C1.CC1OCCC1N(C(=O)Cc1ccnn1C)C(N)=O.N C1(C(=O)NC(CC)CC(=O)NCc2nncn2C)CC(C2CC2)=NO1 N12CCC3C(CC13)C2=O.N1(C(=O)OC(C)(C)C)CCC2CC12CC(=O)OC CC(C)(C(=O)N)C(F)(F)F.C1(O)(CC)CCCN(C(C23CCCC2C3(F)F)=O)C1 C=CCC(C)(C(=O)NC1CN(C(c2cc(CO)c(C)o2)=O)CCC1C)N(C)C C(=O)(C(O)CC(N)=O)N(CC(=O)NCC(C)CN(C)C)CCC N1(C(C2CCC(=O)O2)=O)CCCC2CN(C(c3cc(Cl)ns3)=O)CC12 c1(OC)cc(N(C)C(c2c[nH]nc2-c2ccnn2C)=O)ccc1C(=O)O N1(C(COCC)=O)CC2(CC2)CC1CNC(=O)C1=CCN(C)C1 C1(NC(C(C)(C)Oc2ccccc2)=O)CCC(C)CC1.C(=O)CCC1CCC1.N Cc1cc(C(N2CCN(C(C3CCCS3(=O)=O)=O)C(C(F)F)C2)=O)cc(C)n1 C1(CC(=O)NC2(C)CN(C(c3ccc(Cl)c(O)c3)=O)C2)CN2CCC1CC2 C1(C(=O)NCC2(C)CCC2)SC2C=CC1CC2.c1(CC(=O)N)ccnc(O)c1 c1(C(N2CCC2)=O)cccc(-c2ccccc2)c1.C(=O)(C=CC=O)OCC.N c1(C(=O)OC)ccc(Br)cc1Cn1cc(C2CNCCN2C)nn1 N1(C(=O)OC(C)(C)C)CC2CCC1C(C(=O)NCCC1CCOCC1)C2 Cc1nn(C)cc1CCC(=O)NCCC(C(C)C)NC(=O)CCc1nc(=N)[nH][nH]1 N1(C(=O)Nc2c(C)n(C3CCC3)nc2)CCCC2(CCC(O)C2)C1 N(C1CCCc2n[nH]cc21)C(CNC(c1cnc(CC)o1)=O)=O C1(C(=O)NCC(CN(C(=O)C(F)(F)c2cscn2)C)O)COCC(C)(C)O1 C1(CC)(CC)CN(C(C2CCN(C(=O)CCc3nncn3C)CCO2)=O)CCO1 C1(C(=O)NCC2N(C(C(C)OCC(C)C)=O)CCC2)CCCCCS1(=O)=O C1(NC(C2CCC(O)C2)=O)C=CCC(C(N2CCCC2CC2CC2)=O)C1 CCCCC(O)C(=O)NC1CCCC1C(=O)Nc1cc(-c2ccccc2)ns1 C1(NC(c2c[nH]c(=N)o2)=O)COCCC1C(=O)NCC1CC1C1CC1 N1(C(c2cc(C(C)C)[nH]n2)=O)CCCCCC1CNC(=O)CC1C(C)C1(F)F Cc1c(C(=O)NCCN(C(=O)CC(C)n2cccn2)C)cnn1CC1CCCC1 Cc1cn2cc(C(=O)NC(C3CCN(C(=O)CCS)C3)(C)C)ccc2n1.C(C)C C1(C(=O)NCC2(NC(c3n(C)c(S)nn3)=O)CCCCC2)CCN2CCOCC12 CC1(NC(C2CC3CC2CO3)=O)CCCN(C(=O)Cc2cccnc2Br)C1 C(=O)(CC(C)C(C)(C)NC(C1COCC1C(N)=O)=O)N1C(C)CNC(=O)C1 C(=O)(CCn1cncn1)NCC(C1CCCC1)C.C(=O)(C(C)(C)c1ccno1)N CC1CCC(C)(C(=O)NC(C)CCNC(c2ncccc2O)=O)CC1 C(=O)(C(CCC)C(=O)OC)N1CC(NC(CCC)=O)C(CO)CC1 Cc1nc(C)n(CCC(=O)NCC(C)NC(c2sncc2Br)=O)n1 c1(C(=O)NC(C2CCCN2C(=O)COCC2CCCCO2)C)ccnnc1O C1(O)(C(C)NC(c2c(C)nns2)=O)CCN(C(=O)C(C(C)C)n2cncn2)CC1 C1(OC)COC2(CCN(C(=O)O)CC2)C1.c12cnc3n1CCN(C3)C2=O.C(C)(C)C C1(C(N2CC(CNC(C3(C#C)CC3)=O)OCCC2)=O)Cc2cc(C)ccc2O1 C1(NC(=O)NC(C)Cc2ccncc2)CC2CCC(C1)C2(F)F c1(NC(CCC=C)C)ncnc(N2CCCC(NC(c3ccccn3)=O)C2)c1C C1(C(=O)NC2CCC(C)N(C(c3cc4n(n3)CCO4)=O)C2)CC2CCCCN2C1 C1(CNC(CCS(C)=O)=O)CN(C(c2ncnc3sccc23)=O)CC(C)(C)O1 c1(C(=O)NC(CCNC(CCOC(C)=O)=O)(C)C)c[nH]cc(Cl)c1=O C1(CNC(C(C)(C)C(N)=O)=O)CC2CCC(C1)N2C(=O)CC1CC1 N1(C(c2cc(SC)c(C)o2)=O)CC2CCC(C1)C(NC(C1CCNC1=O)=O)C2 c1(C(N(CCCNC(Cn2c(=O)sc(C)c2C)=O)C)=O)ccc2c[nH]nc2n1 C1(C(=O)NCCOCC(=O)OC)OCCC1.c1(CCC=O)nccn1C.N C(C(=O)NC1CC(C)(NC(=O)CN2CCSCC2)C1)(C(C)(C)C)SC Cc1cc(C(C)C)ccc1Br.c12ccc(cc1)N(C)C(C1CCCOC1)C(=O)N2 N1(C(c2ncc(C)c(C)c2)=O)CCN(C(=O)C=CCN2CCCC2)CC(C)(F)C1 C1(NC(C(CO)OC)=O)CN(C(c2cccc(O)n2)=O)CC1C C1(NC(CN(C(C(C)C)=O)C)=O)CCCN(C(=O)CSc2nc[nH]n2)CC1 Cc1nc2c([nH]1)C(C=O)CCC2.C1(C(F)(F)F)(C(N(CC)C)=O)CC(C)(C)C1 N1(C(c2ccc(F)cc2)C)CC=C(c2ccc(O)cc2)CC1 C(=O)(CCC(C)NC(C1C=CCC1)=O)NCCCOCCOC C1(C(=O)NCc2c(OC)ccnc2)CC2CC(C1)CS(=O)(=O)C2 c1(C(N2C(C)(C(=O)Nc3cn(CC)nc3C)CC2)=O)ccccc1[N+](=O)[O-].C C1(COC)(NC(=O)CCCN(C)C)CCN(C(=O)CC2CCN(C)C2=O)C1 C12(C(=O)N)CCCC(C)(C1)OC2.Cc1noc(C)c1CC(C)C(=O)N1CC(C)C1 CC(C)CC(C(=O)NCCC1CCN(C(c2ncccc2Cl)=O)C1)C(C)C C(=O)(C(O)C(C)(C)C)N1CC(C(N2CC(OCCCCC)C2)=O)(COC)C1 Cc1ccc2[nH]c(C(N3CCC(N(C(=O)C(C)S)CCO)CC3)=O)cc2c1 N1(C(c2ccc(NC)cc2)=O)Cc2ccccc2C1C(=O)NCC(O)CO c1(NC(C2CC(OC)CN2C(=O)Nc2c(C)cccc2Br)=O)cccc(F)c1F C1(NC(C(C=C)(F)F)=O)CCCN(C(c2c[nH]c(=N)nc2CC)=O)C1C N1(c2cc(CO)cc(OC(C)C)c2)C(=O)C2CCCCCN2C1=O c1(C(N2CCC(=C(C#N)C(=O)NCCCF)CC2)=O)cc2ncccc2o1 CC1CN(C(=O)CCc2nncn2C)CCCN1C(=O)Cc1ccsn1 C1(CNC(c2nn[nH]c2Cl)=O)CN(C(=O)CC2CCCS2(=O)=O)CCCO1 CC1(C(N2CCC2CNC(c2cc(-c3ccncc3)ccn2)=O)=O)CC(C#N)C1 N1(C(CC(CC)CC)=O)CCCC2CCN(C(c3ccc([N+](=O)[O-])cn3)=O)CC12 CC(F)(F)C(C)(C)C(=O)NCC1CC1C(=O)NCCCc1cn[nH]c1 C(=O)(C1=CCCN(C(C2C3CCC(F)(F)C23)=O)C1)N(CC(C)(C)CO)C O=C(CSCC(C1CCC1)C1CCC1)N.C1(F)CC1.C(=O)CC1CC1 Nc1c(C(=O)NCC(O)CNC(=O)CC2CCCC(=O)N2)ccc2cccnc12 C1(O)(C(N)=O)CCN(N2CCCCC2c2ncc(Br)cn2)C1 Cc1[nH][nH]c2ncnc(=NC(=O)Nc3c(Br)cc(F)cc3[N+](=O)[O-])c1-2 CC1(C)CCC1(C)NC(c1c[nH]nc1-n1cnnn1)=O Cc1cc(Br)cnc1CN1CCNCC1C(N1CCC(C(C)(C)O)CC1)=O c1(C(c2n(CC=C)nnn2)NC(C)CCO)cc(OC)ccc1OC.C1CCC1.C c1(C(N2CC3CC2CN3Cc2c(F)cncc2F)=O)ccc2[nH]c(=O)ccc2c1 N1(CC(N2CCC(CNC(C=C(C)C)=O)CC2)=O)C(=O)C(=O)N(C)C1=O N1(C(c2c(COC)cco2)=O)C(C(=O)NCC(C)CCCO)CCC12CC2 C1(NC(c2nc(C)n(C)n2)=O)CC2CN(C(=O)C(C3CCOCC3)C)CC12 C1(C(=O)N(C2CCC2C)C)(CC)CCCN1C(c1ccc(C(F)F)o1)=O NS(=O)(=O)CC(=O)NC1CCCC(NC(C2(c3cccnc3)CCCCC2)=O)C1 C(=O)(CC(C)C(=O)N(CCCNC(c1cc(C)ncn1)=O)C)OC c1(CNC(C(Cn2cncn2)NC(C=CCC)=O)=O)cc(O)ccc1C C12(NC(CCOCCCOC)=O)CCC(C1)N(C(=O)CCc1cn(C)nn1)C2 C1(CNC(C(C)Oc2cccnc2)=O)CCN(C(=O)C(F)C2CCC2)CC1C N1(C(COCCCC#C)=O)CCCC2(C1)CN(C(C1CCCC(F)C1)=O)C2 c1(C(N2CCC(CN(C)C(c3snnc3C3CC3)=O)CC2)=O)csc2nnsc12 C1(CC(=O)N(CCCCCNC(C(CN(C)C)O)=O)C)CCCS(=O)(=O)C1 c1(CC)cnccc1C(N1CCC(NC(=O)CCCN2CCOCC2)C1)=O C1(CC)CN(C(=O)CCOc2ccc(C)cc2)CCC1.c1(CC(=O)N)cc[nH]n1 c1(C(N2CC(C)CCC2)=O)c(N)cccc1[N+](=O)[O-].C1(OCC)CC1C(=O)N N1(C(c2n(CC)ccn2)=O)CC2CC(NC(c3c(Cl)c(C)nn3C)=O)CC1C2 N1(C(C2C(C)CCC2)=O)CCN(C(c2sccc2-n2ccnn2)=O)CC12CC2 c1(C(N2CC3CN(C(c4nccc5occc45)=O)C3C2)=O)cc(F)ccc1[N+](=O)[O-] c1ccc(C)cc1C.c1(CC(=O)NC(CN(C(=O)C)CC)C)cncc(O)c1 C(=O)(C(O)C1=CCCCC1)N1CC(C(C)(C)O)C1.CC(C(=O)NC)C(F)(F)F C1(NC(C(C)CC2CCCC2)=O)CCCN(C(C2CCCC(F)(F)C2)=O)CC1 C1(CC)(CC)CC(C(N2CCC(CN(C(=O)C=C(Cl)Cl)C)C2)=O)C1 c1(C(=O)NC(C)C(C)(C)NC(c2cn3cnnc3cn2)=O)nc2ncccn2n1 c1(C(=O)NCC(CN(C(=O)CP(C)(C)=O)C)(C)C)cccc2oncc12 c1(C(N(CCC(C(C)C)NC(C(F)OC)=O)C)=O)cccc2oc(C)cc12 C(C(C)(C)C(=O)NC1CCCCC1NC(=O)CCn1ccnn1)SC CC1CCC(NC(C2(CC(F)(F)F)CC2)=O)CN1C(=O)CC1COCCO1 CON=C(C(=O)NC(C)CC1CN(C(c2cc3sccc3s2)=O)C1)c1ccco1 C=C=C(C)CC(=O)N1CC(CNC(c2ccccc2-c2cn[nH]c2)=O)(OC)C1 C(=O)(CCC(C)(C)[N+](=O)[O-])N.c1(CSC)cc(C(=O)NC2CCC2)ccc1F C(CC(=O)N(CC)C(C)C)(C(F)(F)F)OC.c1(C=O)cc(F)c(O)c(Cl)c1 C(CCCCCC(=O)N1CC(C)OC(C)(C)C1)NC(C(COC)C)=O C1(NC(CCc2ccc(C)cc2)=O)CCN(C(c2ccnc(F)c2Cl)=O)CC1F Cc1ccc(C(C)C(=O)NC(C2CCCC2)CNC(=O)C(c2ccncc2)C)s1 C(=O)(CC1=CCCC1)N1C(CC)C(C(=O)Nc2ccccc2CCO)CC1 C12(C(N(CC(=O)OCC)CC=C)=O)CC1CCN2C(C1SCC=C1C)=O C(CC(=O)NCC1CSC1)(C(F)F)NC(CCC(C)SC)=O C1(NC(C(c2ccc(Cl)cc2)CC)=O)CCN(C(=O)Cc2ccoc2)CC1O C1(CC(=O)N)CCCC(C)(C)O1.c1(CC)cccc(C(N2CCCCC2C)=O)n1 N1(C(CCSCC(C)C)=O)CCC(O)C(N(C)C(c2coc(C(F)F)c2)=O)C1 N1(C(C2(C)CC(=C)C2)=O)CC(C(=O)NCC2CCCCCC2)CCC1(C)C c1(CNC(N(C2CCC(CC)CC2)C)=O)ccc(CO)c(C)c1 C1(C)(CNC(CN(C)C2CC2)=O)CCCN1C(=O)Cc1n[nH]cc1Br N1(C(c2cc(C(C)C)nn2C)=O)CCCC(CO)(NC(c2[nH]cnc2C#N)=O)C1 C1(N(C(c2nccc(C)c2)=O)C)CCN(C(=O)CCC2CCCN2C)CC12CC2 N1(C(C2C(C(C)(C)C)C2)=O)CCC2C(C1)CN2C(=O)C(c1ccc(Cl)cc1F)O C1(C)(C=O)C2CN(C=O)CC12.CCCCCCOC(C)(C)C.C(C)(C)C Cn1[nH]c(=NC(=O)CC(C)(C)NC(C2CCCC23CCC3)=O)cc1C(N)=O C1(NC(CC=C)=O)CC(C)CN(C(=O)Cn2cc(C(C)O)nn2)C1 Cc1cc(S(=O)(=O)NC(C2CCCCN2C(c2cnc(Br)o2)=O)=O)ccc1Cl c1(OC)nccc(-n2cccn2)c1CNC(C)CC1(O)CCC1 C1(CC(N2CCCC(C(C)NC(=O)C3=CCCOC3)C2)=O)Cc2ccccc2N1 n1(CC)nc(C(N2CC(C)C(C(F)(F)F)C2)=O)cc1O.C(=O)CC.CC(F)F Nc1ccc(F)c(C(=O)NCC2CCC2NC(c2cnc3sccn23)=O)c1 c1(C(N2CCC(N)(COC)C2)=O)nn(C)cc1S(N)(=O)=O Cc1cc(C(N2CCN(C(=O)C(C)C)C(C(C)C)C2)=O)c(N)c(F)c1 CC1CN2CCN1C(C(N1CC(NC(C3CN(C)C3)=O)C(O)C1)=O)C2 C1(NC(c2c(C)sc(O)n2)=O)CCCCCC1NC(=O)C(O)c1ccsc1 c1(C(=O)NCC2N(C(C(c3ccccc3)OC)=O)CCCC2)cncc(F)c1C C1(OC)CC(NC(=O)C(n2nc(C)cc2C)C)CN(C(C2CC(F)(C)C2)=O)C1 CCC(CC(=O)NC1C=CC(CO)C1)N(C)C(C1COC(=O)N1)=O CN1C(=O)NCC1C(N1CCOC(CCNC(=O)CCC2CCOCC2)C1)=O C1(CC(=O)NCC(C)NC(c2ccn(C3CCCCC3)n2)=O)CCCCCC1 N1(C(c2[nH]c(=NC)sc2)=O)CC2OCC(NC(=O)CC3(O)CCC3)C2C1 c1(OC)ccc(S(=O)(=O)N2CCC(C(=O)NC3CCc4n[nH]cc4C3)C2)cc1F CC(C)CC(CNC(=O)CC1CC(=O)C1)C(=O)N1CCC(C)C1CO C12(NC(C(C)OC)=O)CCCC1N(C(=O)Cc1c[nH]c3cc(F)ccc13)CCC2 C(=O)(C1COc2ccc(F)cc21)NCCN(C(c1ccnn1CC)=O)CC c1(C(=O)NC2COCC2O)cncnc1-c1ccc(-c2cc[nH]n2)cc1 C1(NC(C2(C)CCN(C(c3n(CC)ccn3)=O)CC2)=O)CCCCN(C)C1=O c1(CNC(=O)NCCN2CC(=O)OCC2)c(Br)cc(F)c(F)c1F C(C(C(=O)O)NC(C1(CN)CCOC1)=O)SCC N1(C(C(CC)(F)C(=O)OC)=O)CCC(S(C)(=O)=O)C1.c1(CC=O)cccnc1.N N1(C(C(C)O)=O)CC2OCC(C(=O)NCCCN3CCSCC3)C2C1 Cn1cc(Cl)cc1C(=O)NCC1(NC(=O)CC2OCCC2(C)C)CCCCC1 CC1C(NC(C2CCC(NC(N)=O)CC2)=O)CCCN1C(c1ccc(O)nn1)=O C1(c2cn(CC(CC)C)nn2)N(C(c2cn(CC)nn2)=O)CC12CCOCC2 C1(OC)CN(C(c2ccc(C#N)o2)=O)CCC1NC(=O)CCc1nccs1 C1CCC12CCC2.C(C)(CO)(C=O)OC.C12(C=O)CC(c3ccccc3)(C1)C2.N c1(C(=O)NC23CC(C(N4CCCC4C)=O)(C2)C3)cc(O)ncc1F.C1CC1 C12(CNC(COC3CCN(C(C(C)OCCCC)=O)C3)=O)CC(CCO1)C2 N1(C(C2CCC(=O)O2)=O)CCC(NC(c2ccc(C(F)F)s2)=O)C(O)C1 C=CCC(C(=O)NC(CCNC(=O)Cn1cncn1)C(C)C)OC CCCC(CNC(c1c(C)ccnc1C)=O)C(=O)NCC(CC)(CC)CO c1(C(=O)NC(C2CN(C(=O)C(CO)NC(N)=O)CCO2)C)cc(Cl)ccc1O c1(C(N2CCC(NC(COCCC)=O)(CF)C2)=O)ccc2c(c1)C(=O)OCC2 C1(CNC(c2nc(COC)oc2)=O)C(C2CC2)CCN1c1cc(Cl)ncn1 C(=O)(CCCCC(N)=O)N1C(C(C)C)CN(C(=O)COCCF)CC1 Cc1c(CC(=O)NC(C)CCCNC(C2CCCCCC2)=O)oc2ccccc12 C(=O)(C1(C)CCc2ccccc21)Nc1cccc(C2CCN(C)C2)c1 c1(C=O)ccc(C)cc1O.C1(OCC)CC2(C1)CC2.C1(C=O)CCN(C)C1.N c1cc(O)c(F)cc1F.CC(C)(O)C(F)C(=O)N1CCC(O)C12CC2 Cc1csc2ncc(C(N3CC(NC(=O)C(C)CO)C4(CCC4)C3)=O)c(=O)n12 N1(C(CCC(CC)NC(=O)C(C)(C)CCF)=O)C2CCC1CC(CO)C2 c1(C(=O)NS(CC)(=O)=O)ccc(CS(C)(=O)=O)cc1F c1(C(C)=O)cc(C(=O)NC2CCC2)oc1C.c1(C=O)cc(C(C)(C)C)no1.N N1(C(CSCC)=O)CC(NC(=O)C(C(C)C)NC(C)=O)C(C2CC2)C1 c1(C(=O)NCC2(O)CCN(C(CC(C(=O)OC)C)=O)CC2)nc2ncccn2n1 c1(C=O)cn(C)c(=O)n1C.C(C)(CO)(C(=O)NC)NC(C)=O.C1CCCC1 CCC(F)(C(=O)OC)C(=O)N1CCOCC(NC(c2ccnc3ccsc23)=O)C1 c1(C(N(CCC)C)=O)cc(F)ccc1S(C)(=O)=O.C1(C=O)(COC)CC1 C12(C(=O)N)CC(C)(CCO1)C2.Cc1cnncc1C(=O)N(C)CC1CCCCC1 C(=O)(CCC(C)(C)O)NCCCN(CCCNC(=O)C(C)(C)n1cccn1)C C1(NC(c2cnsn2)=O)CCN(C(c2nc[nH]c3ncnc2-3)=O)C12CCCC2 c1(N(C)CC2CCCN2C(c2cccc(S(C)=O)c2)=O)ncnc2c1nnn2C c1(C(=O)NC(c2ccccc2)CCO)ncnc2c1OCCO2 C1(NC(c2ccc(C)cn2)=O)CC=C(C(=O)N2CC=CC2CF)C1 N1(C(C2(CC)CCC2)=O)CC2(C)CCC1CC2.c1(C(=O)N)ccc(C)c(F)c1N C(=O)(CC1=CCN(C(c2nccc(C)c2N)=O)CC1)NCC1(SC)CCC1 c1(C(N2C(C3CCN(C(C4C(C)=C4)=O)CC3)CCC2)=O)cccn2nnnc12 Nc1cc(Cl)ccc1C(=O)NC1CC(NC(=O)CC2CC(F)(F)C2)C1 CC(O)(CC(F)F)C(=O)N1CCC(C)(CNC(=O)CCn2ccnc2)C1 c1(C(N(C)CC2CCCCN2C(=O)CSC(F)F)=O)coc2ccc(Cl)cc12 C(C)(C(=O)NCC1(NC(C2CC2OC)=O)CC1)OCCC=C Cc1cc(-c2ccoc2)c2sc(=NC3CC3c3ccsc3)[nH]c2n1 C(CCC(=O)N)N(C(C)=O)CC.C(=O)(C(O)C)N1CCC1.C(C)(C)C.C O=C(CC1=NNC(=O)C1)NC1CN(C(c2ccc(OC(F)F)cc2)=O)CC2CC12 N1(C(C(=O)NCC2OCC(C)(C)C2)=O)CCN2C(=O)CCC2C1 C1(C(=O)NCCCC(=O)N(C)C)CN(C(=O)C(O)c2ccco2)CC12CCC2 C12(NC(c3c(OC)ccc(C)c3)=O)CCN(C(C3(SC)CC3)=O)CCC1C2 C12(C=O)CC3CC(CC(C3)C1)C2.n1(C(C)C)cncc1C(=O)N.CC(C)(C)C c1(C(=O)NCc2occ(C(N(C3COCC3(C)C)C)=O)c2)cnc(S)nc1 C1(C(N2CCCCC2)=O)CC2(CCC2)CO1.c1(C(=O)NCCO)cc(O)ncn1 C(C(=O)NCCCNC(=O)CCC1CC1(F)F)(c1ccccc1)=C(C)C C(c1ccccc1C#N)=CC(N1CC(NC(c2[nH]c(CC)c(Cl)n2)=O)C(F)C1)=O CC1(C)CN(N2CCCC2C(N)=O)C1CS(=O)(=O)c1ccccc1 N1(C(c2cnn(CC)n2)=O)CCCC2(NC(C3CC34CCOC(C)C4)=O)CC2C1 C1(NC(c2c(CC=C)cccc2)=O)CC2(C1)CN(C(C1CCC(OC)C1)=O)C2 N(C(=NCCc1cnc(C)cn1)NC1CCC(N2CCCCC2)CC1)C(C=C)C C12(C(=O)NCCC3CC3)CCCCC1OCC2.C12(C=O)CCC(CC1=O)C2.C C1(N(C(CCC=C)=O)CCC)CCN(C(=O)C(n2nc(C)cc2C)C)CC1 C1(CNC(CC(C)OC)=O)CN(C(=O)C=Cc2cnc[nH]2)C2(CCC2)C1 c1(N(C(C(=O)NC)C)CC2CCCN2C)ccc(N(C)C)cc1OC C(=O)(C#CC1CCCCC1)N1C(C2(Nc3ccc(C#N)nc3)CC2)CCCC1 Cc1cc(C(=O)NC2CCC2)n(C2CC2)n1.n1(CC=O)ccc(C(=O)O)n1 C1(C(=O)NCCCC(C)NC(c2cnco2)=O)CCCN(C(=O)N(C)C)C1 N1(C(C(CC)(C)CC)=O)CCC2CCN(C(=O)CCC3(C#N)CCC3)CC2C1 C(=O)(C#CC1CCOC1)N(CCCC(=O)N(C1CCCCCC1O)C)C C1C2CC3CN(C(c4cc(F)cc(Cl)c4N)=O)C1C3C2.C(C=O)NC(=O)OC.N N1(C(Cc2scc(C)c2)=O)CCC2CCC(C1)N2C(c1ccc(N(C)C)cn1)=O N1(C(C#CC(C)(C)C)=O)CCCN(C(c2cc(Cl)cc(=O)[nH]2)=O)CC1CO C1(C(=O)NCc2ncc(C)[nH]2)CC(NC(C2CC3(CSC3)C2)=O)C12CCC2 Cc1cc(C)c(C(N2CC3CCC2CN3C(=O)CC2CC3C=CC2C3)=O)c(C)n1 C1(C(=O)NCCN(CCCC)C)CCN(C(=O)C(C)=C2CC2)C1CC CC1CCc2[nH]c(=NCC3(F)CC3)[nH]c(=NCC3(C)CCOC3)c2C1 C1(CCCC)(C(=O)NC(CNC(c2csc(Br)n2)=O)C2CC2)CCCC1 C#Cc1ccc(C(=O)NC2CC(C)(CNC(=O)C=CC)C2)cc1Cl CCCC(C(=O)OCC)NCc1ccc(C(=O)OC)cn1 Cc1nc(C2CC2)nc(C)c1C(=O)NC1CN(C(=O)Cn2cnnc2O)CC1C c1(COC)ccccc1-n1cc(CC(O)C(=O)N(C2(C(=O)O)CC2)C)nn1 c1(N2CCC(N(C(COC)=O)C)CC2)ccc([N+](=O)[O-])c(SC)c1 CCC(CCC(=O)NC1CC2(C1)CC2C(=O)Nc1c(C)cccc1C)OC c1(C(=O)NC2(CO)CN(C(C3CC(OC)C34CCC4)=O)C2)cnc2sccc2c1 c1(CCC(c2ccc(-c3ccc(F)nc3F)s2)=O)cnc2sccc2c1 Cc1ncc(C(N2CCOC(C(C)NC(=O)C(F)=C3CCC3)C2)=O)c(=N)[nH]1 C12(N(C)C(C3CCC3)=O)CCC1CN(C(c1cc(C)n(C(C)(C)C)n1)=O)C2 C1(NC(C2CCSCC2)=O)CC(CO)N(C(=O)CC2(N3CCCC3)COC2)C1 [N-]=[N+]=NCC(F)(F)CCC(=O)NCC1CCN(C(c2csc(CO)n2)=O)C12CC2 C1(F)(CNC(CCCC(C)C)=O)COCCN(C(c2cc(Cl)c(F)cc2O)=O)C1 N1(C(=O)Nc2ccc(C)cc2)CC2CN(C(=O)C(F)(F)Cl)CC12 N1(C(c2c(C)nc(N3CCCC3)cc2)=O)CC(C)(C)CCC1CO C=C(CNC(c1csc(Cl)c1)=O)CCNC(C1CCC(CC)C1)=O O=C(C1=CCCN(C(C2(Cl)CC2(F)F)=O)C1)NC12CCCCC1C2 C1(C(N(CCC)CC)=O)CCCC2C1C2(F)F.O=CCC1(C(F)(F)F)CC1 S(=O)(=O)(c1ccc(-c2ccco2)s1)C1CCCN(c2cc(C)c(Br)cc2)C1=O C1(NC(N2CCN(C(C(=O)OCC)C)CC2)=O)CCCC12CCCCC2 CCCC(C(C)CC)(c1nnnn1CC1CC1)NCC1CC1c1ccoc1 c1(C(N2CC(NC(C(CCC)OCC)=O)C2)=O)ccc2c(c1)NCC2 C1(CNC(C(CC)(F)F)=O)(NC(c2ncccc2CO)=O)CCCCC1C N1(C(Cc2c(C)n[nH]c2)=O)CCN(C(c2coc(Br)n2)=O)C2CC12 C1(NC(C(C)(C)N(C)C)=O)CC2CCC1N(C(=O)C=CBr)C2 C(C(C(=O)NC(C)(C)C(N)=O)C(C)C)NC(C1C(CCC)C1)=O c1(C(=O)C2CC2)cn2cc(C=CC(=O)Nc3ccc4c(n3)CCC4=O)ccc2n1 C1(CCCNC(C(CO)NC(C(C)C)=O)=O)CCN(C(=O)C)CC1.C(=O)N C12(CNC(=O)CCC3CCOC3)CC(NC(C3CC3F)=O)(C1)C2 C1(NC(CCOc2ccc(C)cc2)=O)CCSC12CN(C(C1(C)CC1(Cl)Cl)=O)C2 C1(C(=O)NC(c2nccs2)C)CN(C(=O)Cc2nccn2C)CCO1 C(C(=O)Nc1cnn(C(F)F)c1)(C(C)CC)NC(COC(CC)CC)=O N1(C(c2c(OC)c(Cl)sc2)=O)CC2(CCCC2NC(=O)CCC(C)SC)C1 C12(C(=O)NC)CC1CN(C(=O)CN(CCOC)C(c1ccoc1C)=O)C2 c1(CCC(=O)NC2CN(C(Cc3cc(C)ns3)=O)CC2C)ccc(C(=O)O)nc1 N1(C(CN(C)C)=O)CCc2c(ncn2C)C12CCN(C(=O)CN=S(C)(C)=O)C2 N1(C(CCCCCn2cc(CCC(N)=O)nn2)=O)CC2CCC(C(=O)O)(C2)C1 c1(C(=O)NC(c2cn(Cc3cccs3)nn2)CCC)coc2c(C)cc(Br)cc12 N1(C(c2n(C)ccc2)=O)CCN(C(=O)CC23CC(C2)C3)C(CCO)C1 c1(N(CCS(=O)(=O)NC)C)nc(NCC2N(C)CCCC2(C)C)nc2scnc12 C(CCOCCO)(C(=O)N(C1CC2(CC2)C1)C)NC(C=CC=CC)=O C=CC(C)(O)C(=O)NCC1(C(N)=O)CN(c2nccc(C(=O)OC)n2)C1 Cc1cc(C(N2CCCC2CN(C)C(c2cnc(Br)s2)=O)=O)ncn1 C1(NC(C2N(C(=O)C=Cc3ccc[nH]3)CCC(CC)C2)=O)CC2CC1CC2(C)O C1(CC)C(C(=O)NC(C)(C)C)CCN1Cc1nnc(C2CC2)n1C1CC1 c1(C(=O)NCCCOCCC2CCCO2)ccccc1F N1(C(c2sc(C)c(Br)c2)C(=O)NCCC#N)CCOCC(C)C1 N1(C(c2cc(C)[nH]c2C)=O)CC2CC(C(=O)NCC(c3cn(C)cn3)O)C(C2)C1 C#CCC(C(=O)NCC(F)(F)Cl)NC(c1c[nH]c(=S)cn1)=O C(CCC(C)CC(=O)NC1CC(NC(c2cn(C)c(=O)cc2C)=O)C1)=C(C)C c1(CNC(=O)Nc2ccc(I)cc2Cl)ccc2[nH]ccc(=O)c2c1 C=C(C)CCC(=O)NC12CC1CN(C(=O)C(C1CCCC1)OCC)C2 c1(C(=O)NC2CCN(C(CSCCC)=O)CCC2CO)c[nH]c2ccc(F)cc12 C1(CCNc2c(C(=O)OC)[nH]cc2)C(C)CCCN1C(=O)CNC(C)=O C1(NC(CCCNC(C)=O)=O)CCCN(C(=O)CC2CNC(=O)C2)C1 C(=O)(CCCCCC(C)C)N1CC(O)C1.CC(C(F)(F)C(F)(F)F)=CC(=O)NC N1(C(C(CC)CC)=O)CCN(C(=O)CC(C)C2CC2)CCC1C C=CCCC(C)(C)C(=O)NCC(C)CN(C)C(c1cn(CCCC#N)nn1)=O c1(OC(C)C(=O)NCC(C)(C)CCNC(=O)C(C)(C)CO)ccc(F)cc1 C12(NC(C34CC(C)C3C4)=O)CCC1CN(C(=O)Cn1ncnn1)C2 N1(C(c2cc(Br)n[nH]2)=O)CC2(CCN2C(C2CC3(CC3)CO2)=O)C1 c1(NC(=O)NC(C(=O)OC)Cc2cncs2)cccc(Br)c1I CCC(C)(CO)C(=O)N(CC(C)CNC(c1cncc(Br)c1C)=O)C O=C1CC2C(C(N3CCCC(CNC(C45CCCC4C5)=O)C3)=O)C2C1 N1(C(c2c(OC)c(Cl)ncc2)=O)CC2(CCCC2)C1.C1(C=O)C(C)(C)C1(F)F.N C12(C(=O)NCc3cc(C)cc(C)n3)CC(CCO1)N(C(C1CC(C)CCO1)=O)C2 N(C(=NCCC1CS(=O)(=O)C1)N1CCCC(CC(N)=O)C1)C(C)C C(=O)(CC(C(C)C)NC(=O)CC)NCC1(CCC)CC1.CCN(C)C.O Cc1noc(C(N2CCC(NC(C3(F)C4CCCC34)=O)CC2)=O)c1C C1(NC(CC(=C)Br)=O)CN(C(c2cc(N)ccc2C)=O)CCC1C O=C1NC2CN(C(C3CC4(CCN(C(c5ccnc(O)c5)=O)C4)C3)=O)CC2O1 c1(SCC)nc(C)c(CC(=O)NC2(CF)CCN(C(C3CCOC3C)=O)C2)s1 Cc1cc(C(N2CC(OCC(=O)N(C3CCOC3)C3CC3)C2)=O)c[nH]1 N1(C(CCc2n(CC)ccn2)=O)CCC(O)(C(=O)Nc2cc(O)ccn2)CC1 c1(NC)cncc(C(N2CCC(CC(=O)NCCC(C)O)C2)=O)c1 C1(C(=O)NCC(C2CCCCC2)NC(CC2(N(C)C)CC2)=O)CC12CCCC2 C1(CCOC)(NC(c2c[nH]nc2F)=O)CCN(C(c2ccsc2)=O)C1 CC1(C)C(NC(=O)COC2CC2)CC1CNC(=O)COCCCF C1(C#N)(CC(N2CC(C)C(C)C2)=O)CCCCC1.c1(C=O)ccc([N+](=O)[O-])o1.N c1(CC(=O)NCC(C)N(C(C=C(CCC)C)=O)CC)cccc(C)c1Br c1(C(=O)OCC)cc(C(=O)Nc2ncc(CC)s2)ccc1.C(=O)CC#N.N C(=O)(C(C(C)CC)N(C(=O)C(C1CC1)C1CC1)C)N(C(C=C)C1CC1)C c1(C(=O)NC2CCN(C(c3cnc(C)[nH]3)=O)CC2)cc(F)c(F)c(F)c1F C1(OC)CCC2(C(N3CCC(NC(C4CCCCS4)=O)C3)=O)CC12 C1(C(N(CCCc2ccccc2)C)=O)CC(O)CN1C(C1(C(N)=O)CC1)=O c1(CC=O)cc(Cl)cc2c1OCC2.C(C)(C(C)C)NC(C1CC(CC)C1)=O.N N1(C(C(C)CC2CCCC2)C(=O)NCC2CCOC2)CC2(C)CN(C)CC2(C)C1 C1(CNC(=NCC=C)NCC(C)N(c2ccccc2)C)OC(=O)CC12CCC2 c1(CC)cccc(F)c1NC(C1CC1C(=O)NC1(C(=O)N)CCC1)=O N1(C(C2(C3CCC3)CC2(F)F)=O)CCCCC(N=c2[nH]ccn3nnnc23)C1 CC(C)(C)CC(O)CC(=O)NCC1(NC(C2COC(=O)C2)=O)CCOCC1 c1(C(c2n(CCOC)nnn2)NCCCSC(F)F)cc(C)nn1CCF N1(C(Cc2c(C)ccc(C)c2)=O)CC2CC1CN(C(c1ccccc1C#N)=O)C2 C(CCC(C)C)(C(=O)N)NC(C)=O.c1ccc(C)c(C)n1.C1CCCN1C=O.C c1(CN2CC(NC(c3csc(Br)c3)=O)C(F)(F)C2)c(Cl)cc(Br)cc1Cl c1(C(=O)NCC2(O)CN(C(c3cnn(C)c3F)=O)C2)cncc2c1CCNC2=O C12(C(N(CC(CC)NC(c3ccc(C)c(N)c3)=O)C)=O)CCCC(=O)N1CCC2 c1(CC)cc(Br)ccc1CC(N1CC(c2cc(C(=O)OC)ncn2)C1)=O c1(C(=O)N)cnc2cc(C)ccc2c1.Cc1ccc(C(=O)NCC2CC2)c(Cl)c1 CC1COC2(C1)CN(C(=O)C(Cc1ccoc1)NC(c1ccc(F)s1)=O)C2 C(=O)(C(C)(C)C(=O)N(C)C)N1CC(NC(C(CC)NC)=O)(COC)C1 CC(F)(F)C(C(=O)NC1CCC(NC(c2n[nH]cc2Cl)=O)C1)c1ccccc1 N1(C(c2c(C)ocn2)=O)CCC(C(=O)NCCCCCCF)CC1C N1(C(=O)NCCn2c(C)nnc2)CC2CCC(C1)C21OCCO1 C1(NCCCC=C)(CO)CCC(c2nnnn2CCOC2CC2)C1 CC(C)C(C(=O)N(C)CCN1CCN(C(c2cccc(F)c2)=O)CC1)C(C)C C1(O)(CC(=O)Nc2cccc(F)c2C(F)F)CCN(Cc2cnc(Cl)nc2)CC1 n1(CC)nnc(C)c1C(=O)NC1COCCC1NC(C1C2CCCCC12)=O C(=O)(CCOC1CCCC1)NCC(=O)NC1(CCC=C)CC1 Cc1cc(O)ccc1C(N1CC(CN(C)C(C2CC3(C2)CC3(F)F)=O)C1)=O c1(C(=O)NC2CCN(C(c3cnc(OC)nc3C)=O)C2)cc2c(nn1)OCCS2 c1(CNC(=O)CSC(F)(F)F)ccc(-n2cc(C3CC=CCC3)nn2)cc1 C1(CC(=O)NCC=CCNC(c2n[nH]c(C3CC3)n2)=O)CCC1C1CC1 N1(C(CCC)=O)CCC2CN(C(c3nc(SC)n4ccccc34)=O)CC2CC1 CCC(C)C(C(=O)N(C)CC1CCCCC1)N(C)C(c1cc(C#N)cs1)=O C12(NC(CCOC)=O)CCC(CN(C(c3csc(-c4cnccn4)n3)=O)C1)C2 c1ccccc1F.C1(C(CNC(=O)CS)NC(COC(CC)C)=O)CCCCC1 CCC(C(=O)O)C(=O)NCC1CCC1NC(=O)C(c1ccc(Cl)nc1)(C)C c1(CN(CC(O)CN(C)C(C2CCN(C)C2)=O)C)cc2c(cc1Cl)OCCO2 C#CCC(CC#C)C(=O)N1CCCC(N(C(=O)C(F)C(F)(F)F)C)C1 c1(C(CNC(C2CCN(Cc3cc(=O)cco3)C2)=O)O)ccccc1Cl C1(C(C)NC(CCc2onc(C)n2)=O)CCCN(C(=O)C(C)(C)N(C)C)C1 Cc1nc(C=CC(N2CCC(NC(C3(C(F)F)CC3)=O)C(O)C2)=O)[nH]c1C C(=O)(CC(F)(F)C(C)(F)F)N1C(C)CC(C)C1.c1(C=O)ccn(C(C)(C)C)n1 N1(C(C(C)=CC2CC2)=O)CCCC(NC(=O)C(C(C)C)c2ccc(F)cc2)CC1 N1(C(c2cnc(C(C)OC)s2)=O)C2CCCC1CN(C(C1C(C#N)C1(C)C)=O)C2 c1(C(N2C(CNC(CCC(C)(F)F)=O)CCCCC2)=O)cc2nc[nH]c2cn1 c1(CC)nc(=N)[nH]cc1C(=O)N.C1CCCCN(C(=O)CC2NC(=O)NC2=O)C1 n1(-c2cn(C)nc2)cc(C#CC(C)(C)NC(c2ncoc2Br)=O)nn1 C1CN(C(=O)C=Cc2ccncc2)C2CC12.c1(C=O)cn(CC(F)(F)F)nn1.N N1(C(CC(C)N(C)C)=O)CCC(F)(F)C(CNC(C2C3CC4C(C3)C24)=O)C1 C(=O)(C1=CC(C)(C)C1)NCC(C(C)C)NC(C1CC2C(C1)C2(F)F)=O Cc1nc2ccccn2c1C(N1CC2(CCCC2NC(=O)CCCCC#N)C1)=O Cc1cccc(CCC(N2CCC(CN(C(=O)CC3CC4(CC4)C3)C)C2)=O)n1 c1(C(=O)NC2CCC(C(N3CCC(C)(O)C3)=O)C2)cc(Br)cnc1Cl C12(c3nnnn3CCCF)CSC(C1)C2.C1(OCC)CCN(CC(F)(F)F)C1 CC1CCN(C(c2c[nH]nc2Cl)=O)CC1CC(=O)NCCC1OCCC1C C1(C)(C(=O)Nc2ccc(CC(=O)NC)nc2)CCN(Cc2ccccc2Cl)CC1 N1(C(C(COC)C)=O)CCCC(C(=O)NCCc2nnc(C)n2C)CC1 N1(C(C(C(C)O)N(C)C)=O)CC(C2CC2C=O)C1.C(CC1CC1)CC1CC1 C(=O)(C1=C(Cl)CCC1)NCC1(C)CCCC1.C1(c2ccon2)(CC=O)CCC1 C1(NC(c2cccc(O)n2)=O)CCC2(CC1)CN(C(C1(O)CCC1)=O)C2 Cc1cncc(C)c1C(N1CCC(O)(CN(C)C(c2ccoc2Cl)=O)C1)=O c1(CC)ncccc1NC(C1CCC(NC(c2ccc(C3CC3)o2)=O)C1)=O c1(C(=O)NC2CCC(NCc3cccc(OC)c3C)C2)cccc([N+](=O)[O-])c1 c1(NC2(CNC(C=C(C)C)=O)CCCC2)nn2cc(C)nc2s1 Cc1cc(Cl)c2c(c1)CCCN2C(c1ccc2oc(O)nc2c1)=O C1(CCNC(c2c(CC)con2)=O)COCCN1C(=O)C.c1ccc(O)cc1.O c1(NCC(CNC(c2c(C)ncn2C)=O)C)c(Cl)cc([N+](=O)[O-])cc1Cl c1(C(=O)NCc2c(CNC(C(C)OC)=O)cccc2)c(C)cc(F)cc1C N1(C(CCCC#C)=O)CCN(C(=O)C(F)CC2CCCCC2)CC(O)C1 C1(C(CC)NC(=O)C=C(C)I)CCC2CC12 C1CC2CCC1N2C(C1CC1C(F)(F)F)=O.c1(OC)cccc(CCC(=O)N)c1 CCC1=C(C(=O)NC2CS(=O)(=O)CC2NC(c2snnc2CC)=O)SCCO1 C12(NC(=O)Cc3cccnc3)CCCC1N(C(=O)CSCc1ccccc1)CC2 c1(OC)cc(C(N2CC(CO)C2)=O)c(Cl)cn1.c1(C(C(=O)N)F)ccc(F)cc1 C(=O)(CCCC(F)(F)C(F)(F)F)NC1CN(C(CS(N)(=O)=O)=O)CC1O c1(CNC(C(N2CCC(C)C2)=O)=O)ccccc1.C1(C=O)CC2(CC2)CO1.C N1(C(=O)Nc2ccc(NC(C)=O)cc2)CCCC2C(O)CC12 C(C(CNC(=O)CC(F)(F)Cl)S(C)(=O)=O)NC(C1CCN(C)C1)=O C1(CCC#C)CCCN1C(C12CC(C1)C2)=O.C(=O)(CCCN(C)C(C)=O)N Cc1ccc2c(C(=O)NC3CC3CNC(c3occ(C)c3C)=O)n[nH]c2c1 N1(C(CNC(CCC(C)C)=O)=O)CC2(CC2)CC1C(=O)N(C1CC(F)(F)C1)C c1(OC)ccc(C(=O)N)c(C)n1.C1C2CCC(C2)N1C(=O)C=O.C1CC1.C N1(C(c2n(C=C)nnc2)=O)CCC(F)(CNC(c2ccc(C3CC3)nn2)=O)CC1 C1(CC(N2CC(F)(C(=O)NCC(C)OCC#C)C2)=O)CCCC(C)C1 c1(C(C(=O)N(C(C)CNC(c2c[nH]nc2[N+](=O)[O-])=O)C)=O)ccc(F)c(F)c1F C1(C(=O)OCC)C2CC(CN(C(=O)CCC(N)=O)C2)N1C(=O)C#CC1CC1 C1(NC(c2nc(CC)oc2)=O)CC2CCC1N(C(C1CCC3(C1)N=N3)=O)C2 C(=O)(C#CC(=O)N(C)C)NC(c1ccccc1)C.C1(O)(C=O)CC1(C)C.C C1(C(=O)NC2C(CNC(=O)CCn3cccn3)C2)CC(=O)c2ccccc2C1 C=CC(CC)CC(=O)N1CCC(N(C(C)C(=O)Nc2ccc(F)cc2)C)CC1 C(CC(C)C(=O)NCCC1CCCN1C(c1cnc(Cl)n1C)=O)=CC c1(C(N2C(CNC(c3cn(C)nc3O)=O)CC2)=O)ccn2nccc2n1 C(C1=NOC2CN(C(=O)C=Cc3ccc(F)c(Cl)c3)CC12)NC(c1cnco1)=O C1(NC(C(C)(C)NC(=O)C(F)(F)F)=O)CCCCN(C(c2nccnc2N)=O)C1 CC(=O)C(C)CC(C)C(=O)N=c1[nH][nH]c(=Nc2cnn(C(F)F)c2)cc1C C(=O)(CC(C)CC(C)(C)C)N1CC(C(C)(C)O)C1.CC(C(=O)N)C(F)(F)F.C C(=O)(C(C)(O)C(C)C)NCC(CCOC)NC(C1COCCN1C=O)=O c1(CC(=O)NCC2C(O)C(O)CN2C(c2cc[nH]n2)=O)ccc2ccncc2c1 C1(C(=O)NC(COCC)(C)C)CN(C(=O)CC(C)C(C)C)CC1(F)F N1(C(=O)OC)C2CCC1C(C(=O)NCCCCn1ccnc1C)C2 C(C(COC)C(=O)NCCC1CCC1)OC.c1(C(=O)N)csnc1C1CC1 c1(C(N(C)CC2CC23CC(O)C3)=O)ccc(=NCCNc2ccccc2)[nH]c1 N1(C(Cc2c(C)cccc2)=O)CC2N(C(c3cn(C(C)C)cn3)=O)CCC2(C)C1 CC1(C)CN(C(c2cc(=O)cc[nH]2)=O)CC1NC(C1COC(=O)O1)=O c1(C(=O)NCC2(NC(C3(F)CCOC3)=O)CCCC2)ccc(O)c(Cl)c1 C(=O)(C1=CC2C=CC1C2)NC(C(=O)NCc1cccc(C)c1)CC1CC1 C1(CC(=O)N(CCNC(c2ccc(C(C)=O)cn2)=O)C)COC(C)(C)CO1 CC1CCN(C(=O)COCCCN(C)C)C1C(=O)NCCCCCCO C(=O)(C1CCCn2nccc21)NC1C2CN(C(c3n(C)ncc3Br)=O)CC21 N1(C(C(C(=O)OC)C)=O)CCC(C2(C(NCP(C)(C)=O)=O)CCOCC2)CC1 S(=O)(=O)(c1c[nH]ccc1=NCc1ccc(F)c(F)c1)NC1C(CCC)C1 C1(CNC(C2N(CCC)CCC2)=O)CC2CC2N1C(c1ccn(CCF)n1)=O C=CC(CC(=O)N1CC(O)(CCNC(C2(C)CC2(F)F)=O)C1)c1ccccc1 N1(CC(=O)N(C(=O)C(c2ccncc2)C)CC(C)C)CCOCC1 c1(N(C)Cc2c(C)cncc2)nc(N(CCC#N)C)nc2c1CSC2 C(=O)(C(COCC)CC)NC(c1occ(C(=O)NC(C#C)C)n1)C C1(NC(c2ccc(CCNC(N)=O)cc2)=O)CCCN(C2CC2)C1=O c1(NCC2(C(=O)OC)CCCO2)ccc2ccccc2c1.C1C(=O)O1 c1(NC(C=C(CNC(C(COC)OC)=O)C)=O)cnc(F)c(C)c1 c1(CNC(N2CCC(c3nc(C)on3)C2)=O)n[nH]c2ccc(Cl)cc12 C1(NC(c2cc(OC)ncn2)=O)CC=C(C(=O)N(C)Cc2ncco2)C1 N1(C(c2c(Cl)cn(CC)n2)=O)CCC(NC(c2ccn(C3CC3)n2)=O)CC1.C N1(C(C2(C#C)CCCC2)=O)CC(C)C(C)(CNC(=O)C(CC(C)C)N(C)C)C1 C(=O)(C1Cc2ccccc21)NC(CN(C(c1c(COC)ncs1)=O)C)C CC1(C)CC(C(=O)N2CCCCC2C2CCN(C(=O)CCn3cccn3)C2)=NO1 O=S(=O)(c1cnc(-c2ccccc2)o1)NC1CCC2(CCC2)C1 c1(C2CCCN(C(=O)NC(C)CS(C)(=O)=O)C2)nc2c(s1)CCCC2 N1(C(C(c2ccco2)NC(C(C)OC(C)=O)=O)=O)CCN(C(=O)CO)CC1 C(=O)(C1CCCc2c(O)cccc21)NC1CC(C)(NC(CC2(C)CC2(Cl)Cl)=O)C1 N1(C(C(CC=C)CC)=O)CCn2c(CNC(=O)CCC(=C)Cl)nnc2C1 C(=O)C(O)C(F)(F)F.n1(CCC)cc(C)nn1.C(=O)CC=CC(C)(C)C.N S(=O)(=O)(c1ccccc1C(F)(F)F)N1CCN(C(c2c(C)nc[nH]2)=O)C(C)C1 C(C(O)C(=O)N(CCCNC(c1ccnn1C(C)C)=O)CC)=CCCC C1(NC(=O)C(F)OC(F)(F)F)CCC2CN(C(c3ccoc3Br)=O)CC2C1 N1(C(C(OC)OC)=O)CC(C)(CNC(C2(C)CCC(=O)NC2)=O)CC1(C)C C1(C(=O)NC2CCN(S(CCCC)(=O)=O)CC2)CCc2nc(C)cn2C1 C1(C)(CC)CCC(C(N2CC(F)CC2CNC(c2c[nH]ccc2=O)=O)=O)O1 CN1CCC(CC(N2CC(NC(=O)CC3CCN(C4CC4)C3)C(CO)C2)=O)C1=O C(=O)(C1CCSc2ccccc21)N1CC(CCNC(C2CC2C)=O)(OC)C1 N1(C(C2C(C(C)C)CCC2)=O)CCCC(NC(=O)C(C2(O)CCOCC2)(F)F)C1 N1(C(C)C(=O)NC2CCN(C(C3CCOC3)=O)C2)CCN(C)CC1 c1(SCCC)ccc(C(N2CCN(C(C)(C)C)CC2)=O)cc1 C1(NC(C(F)=CCC)=O)CC(CNC(=O)CC(C)(C)OC)C(O)C1 C1(C(N2CCC(O)(Cn3cc(-c4cc(C)sc4)nn3)C2)=O)COCC2(CCC2)O1 Cc1nnc(N2CCN(c3nnc(-c4ccccc4)n3C)CC2)c2ccccc12 C(CCC(O)C(=O)N1CCCC1c1ncc[nH]1)NC(=O)CC1CC(F)C1 c1(C(c2nnnn2C)NCc2c(C)n(C)nc2)ccc(F)c(F)c1Br CC#CCC(C(=O)N1CC(O)CCO1)NC(=O)CC(CC)CC(C)C C1(N(C(C(CCOC)C)=O)C)CN(C(c2c[nH]cc2C)=O)CC12CC2 N1(C(C2(CC)CCCC2)=O)CCC(NC(=O)C(C(C)C)n2cncn2)CC1 c1(CC)nn(C)c(CC)c1S(=O)(=O)N1CCC(c2ccccc2OC)C1 c1(CN(C)C)ccc(C(=O)NCCNC(C2CC2c2cccs2)=O)[nH]1 C1(NC(c2ccoc2)=O)COC2(CCCN(C(c3onc4c3CCCC4)=O)C2)C1 C1(O)(C(=O)NCc2n(CCOC)cnc2)CCCCC1 C(=O)(CCP(C)(C)=O)NC1C(N(C(c2cc(C(C)C)[nH]n2)=O)C)CCCC1 Cc1nnc(N(C2(CC(F)F)CCC2)C)n1CC1CCS(=O)(=O)C1 N1(C(c2c(C)cc(CO)o2)=O)CCC2(C)CCCC12.C1(C=O)CC1C(F)(F)F c1(C(=O)NC(C)(C)CNC(=O)Cc2cn[nH]c2)cc(C(F)(F)F)cnc1O N1(C(C2C(CNC(CC=CC=C)=O)CCC2)=O)CC2(CCNC(=O)O2)C1 c1(CNCCCCCN(CC)CC)ccc([N+](=O)[O-])cc1Cl N1(C(CSCC)=O)CCCC(CN(C2CCCC2C)c2ccccc2)C1 C1(NC(c2ccc(OCC)nc2)=O)CS(=O)(=O)CC1NC(C)=O C1(CC=O)CCCCCC1(F)F.c1(CC)onc(C)c1C(=O)NC1CCC1C C(=O)(C(N=[N+]=[N-])C(C)C)N1CC(OC)C(NC(C2(n3cccn3)CC2)=O)CC1 N1(S(C(CC)C)(=O)=O)CCC(Nc2ncncc2I)C(O)C1 c1(CC(N2CC3CCC3(C(F)(F)F)C2)=O)cncc2ccccc12 N1(C(C(CCC)NC(N2CCCC2Cc2ccccn2)=O)=O)CCS(=O)(=O)CC1 CCC(C(=O)OC)C(=O)N(CCC(C)NC(=O)CCCCc1ccc(C)cc1)C n1(C(C)C)cc(C(N2CC(CNC(=O)Cc3cnnn3C)CC2C)=O)ccc1=O C1(NC(C(C)OC)=O)CCC(CCNC(C2CCCSC2)=O)C1 c1(C2(C(=O)NCC(C(F)F)n3cccn3)CCC2)ccc(O)nc1 N1(Cc2cn(C3CC(NC(c4[nH]cc(C#N)c4)=O)C3)nn2)CCS(=O)(=O)CC1 c1(OC)cccn2ncc(C(=O)NCC(C)NC(=O)CC3CCCOCC3)c12 C1(C)(NC(C2(NC(C(CC=CC)CC)=O)CCC2)=O)CCCC(C)(C)C1 N1(C(c2c(C(=O)OC)c[nH]n2)=O)CC(NC(=O)C(O)CF)C(C)C1 CC#CCC(C(=O)NC(C)Cc1ccnn1C)NC(c1cc(O)nn1C)=O c1(CC(=O)NCC(CC=C)NC(c2cnc(OC)s2)=O)cn2ccccc2n1 C(=O)(C(CC(C)(C)C)OC)N(C(C)C(=O)NC1CCCC(C)(C)C1)CCC C1(C(=O)NC(C(=O)NCCCCCOC)Cc2cc[nH]n2)CC(C)(C)CCO1 C1(C)(CC)CCN(c2nnc(CCc3cccnc3OC)n2CC)CC1 C1(C(=O)N(C)OC)(NC(CCCOCC)=O)CC12CCC2 N1(C(C2C(CC)CCC2)=O)CCCC12CCN(C(c1cnc3c(c1)COC3)=O)C2 N1(C(C(CN(C(C(C)N2CCCC2)=O)C)(C)C)=O)CCNC(=O)CC1 c1(C(N)=O)cc(-c2nc(NC(=O)Cn3nc(O)ccc3=O)cs2)ccc1O C1(C)(CC)CC(C(=O)NCC(C)CC(C)C)CCO1.C1(O)(CC=O)CCC1.N C(=O)C1=C2CCN=C2NC=C1.c1(CC(C)C)cc(C(=O)NCCC2CC2)n[nH]1 c1(C(C(=O)NC2CC(CCNC(C3(C)CC(F)C3)=O)C2)O)ccccc1Cl N1(C(C(c2cccnc2)C)=O)CCCC12CCCN(C(=O)CN=S(C)(C)=O)C2 Cc1cccnc1-c1cn(CCC2CN(C(c3cc(C(N)=O)cs3)=O)C2)nn1 N1(C(c2ccc(C)s2)=O)CCCC12CCN(C(c1cc(S(N)(=O)=O)oc1C)=O)C2 C1(C(=O)NCCCCCNC(C2(C)CCCN2C)=O)(CC)CCC(O)CC1 c1(C(=O)NC2CN(C(COc3c(OC)cccc3)=O)CC2O)c[nH]cc(C)c1=O c1(CNc2c(C(=O)NCCCN3CCCC3)cc(F)nc2)cccc(C=O)c1Br c1(C(=O)NC2CCN(C(C3CCCS3)=O)CC2O)ccc2c(c1)COCC2 c1(C(=O)NCC(C)N(C)C(c2cnc[nH]2)=O)ncsc1Br N1(C(c2c(C)nc(C(C)N(C)C)o2)=O)CC2CCC(CO)(C2)C1 CN=c1[nH]c(=NCC2CCN(C)C2)[nH]c(=NC2CCCN(CC3CC3)C2)[nH]1 C(C(=O)NC12CCC(NC(C3CCN(C)C3C)=O)(CC1)C2)(C(C)(C)C)OC c1(CC)nnc2cc(NC3C4CC3CN(C(C3C=C3C)=O)C4)ncn12 C1(C(=O)Nc2cc(OC)nc(=N)[nH]2)CCC([N+](=O)[O-])CC1 C1(NC(C(C)OCC)=O)C2CCC1CN(C(=O)CN(C)C1CC1)C2 c1(COCC(CC(F)(F)F)O)c(Cc2ccccc2)cccc1F N1(C(CCSC)=O)C2CCC1CC(N(C(=O)C=Cc1ccc(C)s1)C)C2 c1(NC(C2(CC)CCCCC2)=O)ccc2ccccc2c1 c1(C(=O)NC2C(CC=C)CCC2)oc(C)nc1C.C1(C)(C(=O)N)CCNC1=O c1(N2C(CNC(c3c(C)nc(Br)s3)=O)CC(F)C2)ncnc2ccc(Br)cc12 C1(C(=O)NCC(CNC(c2n(CCC)ncc2)=O)OC)Cc2cccnc2C1 N1(C(C2N(C(c3cc(C)c(F)cc3)=O)C3C(C2)C3)=O)CC2OCC(F)(F)C2C1 N1(C(C2(C)CC(NC(C3CCSCC3)=O)C2)=O)CCOC2(CC2)C1 c1(OC)ccc(CC(C(=O)O)NC(=O)CN(C)C(C)=O)cc1OC C(=O)(C(C)(C)CC(C)C)NCCn1ncc(C(=O)Nc2cc(C)sc2)c1 c1(C(C(=O)NCC(C2CCCC2)NC(C2CCCCO2)=O)O)ccc(F)c(Cl)c1 C(=O)(C1=CCC(NC(C2(CC=C)CCOC2)=O)C1)NCC1(C#C)CCCC1 C1(NC(c2nc(COC)sc2)=O)C2CN(C(=O)CCc3cnc(C)s3)CC12 N1(C(C2CC(C)(CC)C2)=O)C2CCC(C2)C1CC(=O)NCc1cscc1C c1(CN(C(=O)NC2C(C(N(C)C)=O)C2)C)ccc(-c2ccccc2)cc1 N1(CCNC(c2n(CC)ccc2)=O)CCCN(C(c2c(C)cncc2C)=O)CC1 N1(C(CC)=O)CCCC1C(C)(C)C.C1(C=O)CC(N(C)C)C1.CC.CC.O N1(C(c2c(CC)c(C)sc2)=O)CCC2CCC(NC(c3cc(CF)on3)=O)C12 c1(C(C(=O)OC)N(C)CC2CCNCC2)cccnc1 N1(C(CNS(NC)(=O)=O)=O)CCC2(CCCCC2NC(=O)COC(C)C)C1 c1(C(N2CCC(C(C)O)C2)=O)c[nH]c2c(-c3ccc(O)cc3C(=O)O)cccc12 S(=O)(=O)(c1cccnc1Cl)N1CC(NC(C2N(C)CCCC2)=O)C(F)(F)C1 c1(CC(=O)NC2(CCNC(c3cnn(CCF)c3)=O)CC2)ccc(Cl)cc1Cl c1(CNc2c(C)n(C3CCOC3)nc2)c(O)cc(F)cc1F CCC(CC(F)F)C(=O)N1CCC(NC(c2cc(O)n(C)n2)=O)C(F)C1 C1(C(=O)NC2(C)CC(NC(C(C=CC)O)=O)C2)CCCCC1C(F)(F)F CC1CC(O)CCN(C(=O)CN(C(=O)C=CC(=O)N(C)C)C2CC2)C1 c1(C(=O)NC2CCC(C)N(C(C3CCCSS3)=O)C2)ncnc2ccsc12 C1(C(=O)OC)CC2OCCN(C(=O)C(c3ccccc3C)C)C2C1 c1(CSCC(N2CCCC(N3CCCCC3=O)C2)=O)cccc(F)c1C(F)(F)F CCCCCC(O)C(=O)N1CCN(C2CN(C(C3CCC(C)C3)=O)C2)CC1 C=CCCC(C(=O)N1CCCC(N2CCC2)C1)NCC(O)C(=O)OC CP1(=O)CCC(Nc2ccc(CN3CCCCCC3)cc2)CC1 c1(OC)c(C(=O)NC2(c3cnnn3CC)CCCO2)sc(C)c1Br C(=O)(C(CCSC)NC(=O)CC1CSCCO1)NCC1N(CC)CC1 CC(C)(C)C(CO)NC(c1cncc(CNC(c2csc(C#N)c2)=O)c1)=O c1(C(N2CCC(C(C)C)C2)=O)ccc2c(c1)CC2.C1(OC)(OC)CCC1C=O c1(C(N2CCC(=Cc3cccs3)CC2)=O)nc(Br)n2ccccc12 C1(NC(C(CC)OC2CCCC2)=O)CCN(C(=O)CCc2nnc(S)n2C)CC1 c1(OC)cc(C)sc1C(c1nnnn1C)NC.C1(O)CCC1 N1(C(C2C(C)(C)C(=O)C2)=O)CCCC2(CCN(CC34CCC(N=[N+]=[N-])C3C4)C2)C1 N1(C(c2c(COC)cc[nH]2)=O)CC2CN(C(=O)CC(C)(C)CC(F)F)CC(C1)O2 N#Cc1ccc2[nH]c(-c3csc(=NCCc4ccc(Br)s4)[nH]3)cc2c1 C1(C(N2CCC(CCCO)CC2)=O)CC2OCCC2N(C(=O)NCCCl)C1 C(CCC)(CC(=O)NCCC1CCCN1C)NC(C(CC)=CC)=O N1(CC(=O)Nc2nc[nH]n2)CC2CC(CN3CC(O)C3)CC(C2)C1 N1(C(CSC)=O)CCc2nc[nH]c2C12CCN(C(C1CC(F)C1)=O)C2 C1(C(=O)NC2(C)CN(C(c3c(O)cc(C)nn3)=O)C2)COc2ccccc2O1 c1(CC)cccc(C(N2CC(C(=O)NCC(C)(F)F)(CC)C2)=O)c1 C1(C(=O)N)CCC2(CCC2)CO1.c1(-n2cc(CC(=O)OCC)nn2)ccccc1 N1(C(C(CCSC)NC(C2CC3(CCC3=O)C2)=O)=O)CCC2(CC(F)C2)C1 N1(C(CCCOC)=O)CCC(C)(C)C1CC(=O)NC1CC1c1ccsc1 C1(OCC)CC2(C1)CC2NC(=O)C(C)CNC(=O)CC1CCCCC1 c1(NCC)ccc(C)cc1C=O.C1(=O)C(CC2CCC2)NC2CC(C2)N1 C1(NC(c2c(C)n3c(s2)ncc3)=O)CN(C(=O)CCS(C)(=O)=O)CC1S(C)(=O)=O C(=O)(C(CC(C)C)OC)NCC(C1CC1)NC(c1nc(CC)oc1C)=O C1(CNC(CC(CC)OC)=O)CC2(CC2)CN1C(c1cc(CO)c(C)o1)=O C1(C)(CNC(C2C(C(=O)OC)C2)=O)CCN(C(c2ccnnc2)=O)C1 n1(CC(N2CCC(NC(CCOCCC)=O)C2)=O)cc(Cl)c(O)nc1=O CC1(C)C(CNC(C2CC2C2CCC2)=O)CCN1C(C1CCSCC1)=O c1(C(N(C2CN(C(=O)C=Cc3cccs3)C2)C)=O)ccc(P(C)(C)=O)o1 N1(C(c2ccc(OC)cc2)=O)C2CCC1CC(N(C)C(C1CC1(C)C)=O)C2 N1(C(C(OC)OC)=O)CC(CNC(=O)CC2COC(C)(C)CO2)CC1(C)C C1(NC(CC(C)F)=O)CC(C(=O)NC(CCO)C2CC2)=CC1O N1(C(c2c(CC)noc2)=O)CC2(CCN(C(c3nc(C)c(C)[nH]c3=O)=O)C2)C1 N1(CC(CC)OC)CCCC(NC(c2ccnc(NC(C)=O)c2)=O)C1C C(C1c2ccsc2CCN1C(C1CCNC1=O)=O)NC(c1cnc(O)c(F)c1)=O c1(N(C(C)=O)C)ccccc1C(=O)NC1CCC1.c1(CC=O)cn(C)nn1.N C1(CC)CC(c2nnnn2CCCF)(NCc2cnccc2C(C)C)CCO1 C12(C(=O)N)CCC(n3cc(-c4cscc4)nn3)(CC1)C2.CC1CC1C(F)(F)F C(c1ccccc1)=CC(=O)NCC(C)C.c1(C=O)ccc(SC(F)(F)F)o1.N N1(CC(=O)N(CCCC)CCCC)CCCCCC1Cc1ccccc1F N1(c2cc(CC)ncn2)CCN(C)CC1CNC(C1(OC)CCCCCC1)=O CS(=O)(=O)C1(c2nn[nH]n2)CN(C(c2c[nH]ccc2=O)=O)C1 N1(C(CCC(=O)c2ccc[nH]2)=O)CCC2(CCN(C(=O)CC3CC3(Cl)Cl)CC2)C1 C1(CC)CN(C(c2nnccc2C)=O)CC1C(=O)N(C(C)CCO)C c1(C(=O)NCC#CC(=O)OCC)c(C(F)(F)F)ccc(F)c1F C1(NCc2c(C)cc([N+](=O)[O-])cc2)CCc2ccc(O)cc2C1 C1(NC(c2cnnc(O)c2)=O)CC2(CCCCN2C(=O)C2=COCCO2)C1 C1(NC(C2C(C)OCCO2)=O)CCCCN(C(=O)Cc2cccnc2Cl)C1 c1(C(N(C2CCN(C(c3cncc(OC)n3)=O)C2)C)=O)cncc(N)c1C C(=O)(CC1COc2cc(O)ccc21)N1CCCN(C(c2c(C)csc2)=O)C(C)C1 C1(CC#C)(C(=O)NCCOCC(F)F)CCN(C(c2ncsc2C)=O)C1 c1(C(=O)NC2(C3CN(C(c4cccc(C)c4)=O)C3)CC2)ccc([N+](=O)[O-])cc1N c1(NC(CC2N(Cc3cnc(CC)s3)CCOC2)=O)cc(OC)c(F)c(F)c1 O=C(C1=C(F)CN(C(C2CCCC(O)C2)=O)CC1)NCCSC(F)F C1(Nc2nccc(OCCC)n2)CC2CCC(C1)N2C(C1CC12CC(O)C2)=O c1(C2C(C(=O)NCC3(O)CC(NC(C(F)OC)=O)C3)C2)ccccc1C c1(C(=O)NCC2OCCN(C(c3c(C)noc3)=O)C2)c(Br)ccnc1Cl C1(C(=O)NCCC(C=C)C)CCN(C(=O)CCc2cnco2)CC1O c1(C(=O)NC(C(C(C)C)NC(c2ccc(C#C)cc2)=O)C)cn2ccnc2cn1 c1(CC(=O)NC2CCN(C(c3sccc3C3CC3)=O)C2)c(F)cccc1F C1(NC(c2cc3scnc3[nH]2)=O)CC12CCN(C(=O)C=CC1CCC1)CC2 c1(C(N2CC(O)(C(C)NC(C(C)S(C)(=O)=O)=O)C2)=O)cnc2ncccc2c1 C1(NC(C2(CC)CCCC2)=O)CN(C(C2CC2c2ccc(C)nc2)=O)CCC1C O=C(CS(=O)C(F)(F)F)NCC1CCN1C(c1cncc(-n2cnnn2)c1)=O c1(C(=O)NC(CNC(C(C)OCOC)=O)C)csnc1C C1(C(N(CCCNC(C2(CCO)CC2)=O)CC)=O)CCCC2(CCOC2)O1 n1(CC)cc(C(=O)NCCC(C)N(C)C(C2CC(OC3CC3)C2)=O)cn1 C(=O)(C(C)(C)CC(=O)N1CCCCC(N(C(=O)CC2CC(F)C2)C)C1)OC C1(C(=O)NC(CCC=C)C2CC2)CC=CCN1C(C1CCCO1)=O C1(O)(C(C)NC(CC2CCC(C)C2)=O)CCN(C(C23CC4CC2C3C4)=O)CC1 Cc1ccc(-n2nc(-c3ccc(Cl)cn3)nc2CC2C(C)C2(F)F)c(C)c1 C1(C(=O)NC(c2ccc(C)s2)C)CC1C1CN(C(=O)CCC2CCCC2)C1 CC(C)(C)CC(F)C(=O)N1C(C(N2CCCC2(C)CO)=O)CCC12CC2 C1(C)(C=O)CCCN(C(C2CC3(C2)CC3(F)F)=O)C1.n1(CC)nnnc1C.N c1(Nc2ccc(NC(c3cnccn3)=O)cn2)nccc(C(F)F)c1Br C1(C#N)(C=O)CC(F)(F)C1.Cc1nscc1CN(C)C(c1occc1C)=O N(C1CCCc2cc(COC)ccc21)C(N1CC(OC(=O)NCC)C1)=O c1(CN(CCNC(C2(C)CC2Br)=O)CC)ccc(Cl)cc1 C1(C)(C(=O)OC)CCN(C(=O)C(CNC(C2CCC(C)(C)C2)=O)C)C1.S c1(C(=O)NCCC(C(C)C)NC(C=CC)=O)ccc(S(=O)(=O)CC)cc1 C1(NC(C(CC)(C)O)=O)C2CCCC1CC(NC(=O)C=Cc1cccnc1)C2 N1(C(c2cnc(Cl)s2)C(=O)NCCC)CC(C)c2ccccc21 C#Cc1ccc(C(=O)NCC(C)N(C)C(c2ccccc2)=O)c(F)c1.C(C)=O.N c1(C(N2CCCC(CCCCNC(C(C(C)C)O)=O)C2)=O)cnc2n1CCCC2 NS(=O)(=O)c1ccc(CCC(=O)N2CCCC2)cc1.C1(C(=O)O)CC(=O)N1 Cc1ccc(Cl)c(C(=O)NCC=CCNC(=O)CSC2CCCCO2)c1O N1(C(C2CC(C)OCC2)=O)CCC2CN(C(=O)CN(S(C)(=O)=O)C)C2C1 Cc1cc(C(=O)NCC(CO)NC(C2CC(OC(C)(C)C)C2)=O)c(O)nn1 C#Cc1cc(F)c(C(N2CCC(N(C(c3ccc(Cl)o3)=O)CC)CC2)=O)c(F)c1 N1(C(c2n(C)cc(NC(c3ccc(O)cc3O)=O)c2)=O)CCN2C(=O)CCC2C1 C1(NC(c2cncc(C)c2)=O)CN(C(=O)CC2CCC(C)(O)CC2)CCC1C C1(NC(c2c(C)nccn2)=O)CCC(C)N(C(=O)C(O)CN(C)C)C1 N1(C(CC2N(C(C(CC=C)C)=O)CC2)=O)C2CCC1CC(F)C2 C(=O)(C=CS(C)=O)NCC1(OC)CN(C(c2ccccc2C)=O)C1 N1(C(C2N(CC)C(=O)CC2)=O)CCC2(CCCN2C(c2ccc(N)c(Cl)c2)=O)C1 c1(C(=O)NCC(CNC(c2ccc(C)c(CO)c2)=O)O)csc2c1CCC(C)C2 N1(C(=O)NC(Cn2c(C)cc(C)n2)C)CC2(C1)OC(=O)NC2=O c1(CC(=O)OC)ccccc1.N1(C(=O)N)CCC(C)(N(C)CC)C1.C(C)=O C(=O)C1=NOC2COCC12.N1(CC(=O)N(CCC)C(C)C)OC(C)(C)CC1=O.N N1(C(C2(CC)COC2)=O)CC2(CCN(C(=O)CC(c3cccc(F)c3)C)C2)C1 c1(OC)ccc(NC(c2ncccc2-c2ccc(SC)cc2)=O)cc1Br c1(N(C)C)ccncc1-c1cn(CCCN(CCO)C(C2CC2Cl)=O)nn1 CCCCC(C)C(=O)NCC(O)CC(=O)NC(C(N)=O)C(C)O C1(CCOC)CN(C(c2c(C)ccn2C)=O)CCN1C(=O)Cc1ccsc1 O=C1CCC2CC12C(=O)NOC1COC1 CON(CCC(=O)NC1(C)CCOC1C)C(=O)C1(OC)CCCC1 N1(CC(CCOC)C)CCC(=O)N(CCc2sccc2Br)C1=O N1(C(C2(OCC)CCSC2)=O)CCC(F)C1.c1(C=O)cccnc1OC(F)F.N C1(CN=C(NC2CCN(CC)C2)NCC2CCC2)OCCOC1(C)C N1(C(Cn2ncc(C)c2)=O)CCC(F)(CNC(C2CCC(C(C)(C)C)O2)=O)C1 N1(C(c2ncccc2N2CCOCC2)=O)CC2CCCN(C(=O)C(O)CCl)C2C1 O=C1NC(CC(=O)N2CCN(C(c3cscn3)=O)CC(O)C2)c2ccccc21 N1(C(C2CCC(C)O2)=O)CCC(N2CCN(Cc3ncc(C(F)F)o3)CC2)CC1 C(=O)(C1CCc2ccccc21)N(C1CCCN(C(=O)C2=CCCCO2)CC1)C N1(C(c2nc(CC)oc2)=O)CC=CC(NC(C2(Br)CC23CCC3)=O)C1 c1(CC(=O)N(C2CCN(C(=O)CN3CCCCC3)C2)C)cc(F)c(F)cc1F C(=O)(C#CC1CCCCO1)N1CCN(c2ncc(C)c(O)n2)CC1 c1(C(=O)NCC2(CNC(C3CC3)=O)CCC2)cnoc1C1CC1.C C1(CC(=O)OC)CCC(NS(=O)(=O)CC2CC(=O)C2)C1 C1(NC(C(COC)(C)C)=O)CN(C(c2cccc(C3CCOC3)c2)=O)CCC1C c1(CNC2(CC(=O)N(C3CCC3)CC)CCC2)ccc2c(c1)OCCN2C Cc1nc(Cl)ccc1C(=O)NC1CC(NCC2(C)OCCO2)C1 N1(C(c2cc(COC)oc2C)=O)CCC(NC(=O)C(C)C#N)C(C)(C)C1 N1(C(c2nc(CC)oc2C)=O)CC(C)CC(C)C1.N1(CCC(=O)N)CCOC1=O C1(CNC(c2ccc(CO)cc2F)=O)COCCN(C(=O)C2=CCOCC2)C1 c1(C(=O)NC2CC(C)N(C(=O)Cc3cnn(C)c3)C2)nc2ccccc2[nH]1 c1(CC)c(I)c(C(N2CC3(CC3C(=O)Nc3nccs3)C2)=O)nn1C Cc1cnc(N2C3CCC2CC2(CC2)C3)c(S(=O)(=O)N2CCC(CF)C2)c1 C(C)(c1ccccc1C)=CC=O.C1(C(=O)OC)COCC1C(=O)N.CC(O)C C(CCCC(=O)NC(C1CC(NC(=O)C(c2ccncc2C)C)C1)C)OC N1(CC)CCOC(C(=O)NCCNC(=O)Cn2nc(C(C)=O)cc2C)C1 c1(C(=O)NC2CC3CN(C(C(CC)(C)CO)=O)C2C3)ccnc2c1cnn2C N1(C(=O)Cc2ccns2)CCC2CN(C(=O)Nc3cccc(Br)c3)CC2C1 c1(N2CC(OC)(CNC(=O)CC(C3CC3)C3CC3)C2)ncc(C#N)cc1C CC1(C)C(CNC(=O)CC2CCOC2)CCN1C(=O)CCCCF C1(C(N2C(CNC(c3ccc4ncnn4c3)=O)C=CC2)=O)Cc2cccnc2C1 c1(CNC(C2(CN)CC(F)(F)C2)=O)ccc2cc(Br)ccc2n1 C1(C(N(CC)CC)=O)CS(=O)(=O)C1.c1(C=O)cn(CF)cn1.CCO C1(NC(C2CC23CCC3)=O)CCCCN(C(c2ccnnc2)=O)CC1 C1(NC(C2CC(N(C)C(C3CCOC3=O)=O)C2)=O)CC2(CCCCO2)C1 C1(NC(c2ncn(CC)c2)=O)C2CC3C(C2)C13C(=O)NCCCOC N1(C(C2CCN(CC)CC2)=O)CC2CN(C(=O)CSc3cccs3)CC12 N1(C(C2(C#N)CCC2)=O)CCC(O)(CNC(C2CCOC2C(F)(F)F)=O)C1 Cc1nscc1C(N1CCCC1CCNC(=O)C(=O)Nc1ncc[nH]1)=O C1(NC(C(CC)(C)C)=O)COC2CN(C(=O)CC=CC(C)(C)C)CC12 C(N=c1[nH]c(=NCc2cc[nH]n2)[nH]c2c1CC(C)CC2)c1cc(C)c(CO)cc1 C1(OCC)CCCCCC1NC(=O)C(C)=NC(CC(=O)NC1CC1)=O N1(C(C2C(C)C2)=O)CC2(CCN(C(c3ccc(O)cc3)=O)C2)C1 N1(C(CC(COC)C)=O)Cc2n[nH]cc2C1C(=O)NCCc1ccnn1C c1(C(=O)NCC2CCC(NC(Cc3cc(C)no3)=O)C2)ccc(C)cc1N=[N+]=[N-] C(c1ccccc1Cl)=C(C)C(N1CC2CC(NC(=O)CP(C)(C)=O)C1C2)=O C1(N(C(Cc2c(C)ccs2)=O)C2CC2C)CC2(CNC2)C1 C1(CNC(C2(N(C)C)CCCCC2)=O)CC12CCN(C(=O)CC1=CCCC1)CC2 N1(C(c2c(CC)cccn2)=O)CC(C)(C(=O)NC(C)CC(C)(C)CO)CC1(C)C c1(OC)cc(F)c(F)cc1C(=O)NCC(C)(C(C)C)NC(C1SCCS1)=O N1(C(c2nc(CC)sc2)=O)CCN(C(C2CCCCC2)=O)C(c2ccnn2C)C1 c1(C(=O)NC2CCC2CNC(=O)C(F)C(F)(F)F)nccn2c(Br)cnc12 CCC(CC(=O)NC1CCC1NC(=O)CC1(O)CCC1)C=O.C(C)(C)C.O Cc1cc(F)cc(C)c1CNC12CC(C(=O)N)(C1)C2.c1cnc(Br)c(Cl)n1 N1(C(C2(C)C(CC)CCC2)=O)CC2(CCCN(C(=O)COC)C2)C1 C1(NC(c2csc(CC(F)F)n2)=O)CC(O)CN(C(c2ccc(O)nc2Cl)=O)C1 N1(CC)CC(C(N2CCCC(F)(CNC(=O)C=C(C)Cl)C2)=O)CCC1=O C1(OCC)CCC(NC(c2ccsn2)=O)CC1N c1(CNC(COC)(C)C)cc(-c2ccccc2)cs1 C1(C(N2CCCC(NC(CN(CC)CC)=O)C2)=O)Cc2cccc(C)c2O1 c1(COc2c(C(=O)OCC)cccc2)ccc(COCC)nc1C c1(OC)cc(C)nc(NC2(CO)CCCN(C(=O)CN(C)CCOC)C2)n1 C(=O)(CCCC(C)C)N(C1(CC(=O)N(CCC(=O)NC)C)CC1)C C1(OCC#C)CCN(C(=O)Nc2ccc(-n3cc(C4CC4)nn3)cc2)CC1 C(=O)(CC(C)(C)CC(F)(F)F)N1C(C)CCC(NC(c2cnn(C3CC3)c2)=O)C1 C1(NC(c2coc3c2COC3)=O)CCCCCCC1NC(C1CCCCS1)=O CCC(CC)C(=O)N1CC(CCCCNC(=O)CCSc2n[nH]c(C)n2)C1 CN=c1cc(C(=O)NC23CC(C2)C3)cc[nH]1.c1(C=O)ccc(C(C)(C)C)cc1 C(=O)(CCC(C)(C)O)NCCc1nc(-c2ccc(C)cc2)sc1 c1(C(=O)N)ccnc(N2CCOCC2)n1.C1CCN1C(C1CC(C(F)F)C1)=O.C C1(C)(CC(N2CC(N(C(CC3CCCC3)=O)C)C(O)C2)=O)CCS(=O)(=O)N1.C C1(CC)CN(C(c2ccc(C(C)(C)C)cc2)C(=O)NC(C)C)CC(C)O1 CC(CCC(=O)N(C1CCN(C(=O)CCC(F)F)C1)C)N(C)C N1(Cc2nc(C)oc2)CC2(CN(C(=O)Cc3cccc(Cl)c3)CCO2)C1 c1(CC(=O)NCCCC(C)NC(=O)C(C)n2cncn2)cc(Cl)ccc1O N1(C(C(=O)NC(c2cccnn2)C)=O)CC2CC3CCCN3C2C1 C1(C)(C(=O)NC(C=C)CO)CC(O)CN1C(=O)C=C(CC)CC C12(C(N(C3CN(CC4CCC4n4ccnc4)C3)C)=O)CC3CC(CC(C3)C1)C2 C(CCC(O)C(=O)NC1CN2CCCC1C2)NC(CC1N(C)CCCC1)=O c1(C(=O)Nc2ncc(C(C)=O)nc2)cc(-c2cc(C)ccc2F)cc2c[nH]nc12 N1(C(CCSC)=O)CCc2nn(C)c(C(=O)O)c2C1 c1(CNC(=O)C(c2cccc(Br)c2)=O)cccc(Br)c1-n1cc(-c2cc[nH]n2)nn1 C#CC1(C)CCN(C(C2C(CNC(C3(C#N)CC3)=O)C2(C)C)=O)CC1 c1(C(N2CC(c3ccc(F)cc3)CC2C)C(=O)NC)nn(C)nc1C n1(-c2ccc(C(=O)NCCCCNC(C3CC3Cl)=O)cc2)cnc2ccccc12 O=C(C(F)C1CCCC1)NCC1CC(NC(C2(C3CCCO3)CC2)=O)C1 CCCCC(=O)C(=O)NCC(C)N(C(=O)C(=O)NCC(F)F)C C1(C(=O)NC(COCC)C)CCCN(C(=O)C#CC2CCC2)CC1 c1(C(=O)NC(C2N(C(CCCCCCC)=O)CCC2)C)cccc2c1OCC2C N1(Cc2c(OC)cccc2)CC2(CC(C(=O)NCc3c(F)cncc3Br)C2)C1 C1(C)CCN(C(c2cnc(N(C)C)nc2)=O)C1.N1(C(C)C)CCCC1C(=O)N.C C1(NC(C=C(C)C2CC2)=O)CC2CN(C(c3cscn3)=O)CC12 CC(CC(=O)NC1CC(CNC(=O)CCOC2CC2)C1)N(C)C C#CCCC(C(=O)NCc1nn(C)cc1CO)NC(C1CCCCNC1=O)=O c1(CC(=O)NC2C=CC(CNC(c3ccncc3O)=O)C2)cccc(O)c1F N1(CCC)CCC(c2sccc2C)CC1.c1(-c2[nH]ccn2)ccc(F)cn1 C1(CNC(C(C)NC(c2cc(C3CC3)no2)=O)=O)CNC(=O)O1 c1(C(=O)Nc2c(O)cccc2Br)ccc2c(c1)CCN(Cc1cncnc1)C2 c1(C(N2CC(CNC(C(C)=C(C)C)=O)C(C)C2)=O)ccc(Br)cc1F c1(CNC2CCN(C(=O)C=CCO)C2)ccc(OC(F)(F)F)cc1 N1(CCCC(=O)N2CC(NC(C(N3CC(SC)C3)=O)=O)C2)C(=O)CNC1=O C1(OC)CC(CNC(=O)NCCC(O)C(OC)OC)C12CCCO2 C1(C(C)C)(C(N2CCC(CNc3nc(-c4ccccc4)ns3)C2)=O)CNC(=O)C1 c1(OC)cccc(Cl)c1C(=O)N.C1CCCN1C(=O)CC1C(C)C1(F)F.C N(C(=NC)N1CCC2C(C(=O)OC)CCCC2C1)CCCCOCC n1(CC)c(CNC(N2CCC(C(c3ccccc3)C)C2)=O)cnc1C N1(C(C2(CC#C)CC2)=O)CCOC(CC)C1.c1(C=O)cn(C(C)(C)C)cn1.N C1(N(CCNC(C)=O)C(c2cnc(C)c(Cl)c2Br)=O)CC2C=CC1C21CC1 C1(CCC=O)Cc2ccccc2NC1=O.C12(NC(C3(C=C)CC3)=O)CC(C1)C2.N C1(C(C)C)CC(C(=O)NC2(C)CCN(C(C)C(=O)NC(N)=O)C2)CCO1 C1(CC)CC(C(=O)NC(C(=O)N(C)CC2CC(O)C2)c2ccco2)C1 CC1CN(C(=O)Cc2cc(C3CC3)on2)CC(C)N(c2ncnc(=N)[nH]2)C1 C(c1ccc(Cl)cc1)=CC(N1CC(NC(CC2ON=C(C)C2)=O)(CO)C1)=O C1(CC)C(C(=O)N(C)CC2(N(C)C)CC2)CCCN1C(c1ccncc1Cl)=O c1(NC(C2CCN(C(c3cncnc3)=O)C2)=O)cc(CO)ccc1Br C1(C(=O)NCC(F)Cl)(CC)CCN(C(c2cnc(Cl)s2)=O)CC1 C(=O)(CC(C)(C)CC)N1C(C2(C(N(C(CC(CC)C)C)C)=O)CC2)CCC1 C1(NC(=O)CC2CCCC(O)C2)C2CC1CN(C(C1(C(F)F)CCOCC1)=O)C2 CCC(C)CC(=O)N1CCCCC1CCC1CCCN1C(C12CSCC1C2)=O CCC(C)C(O)C(=O)N1CC(NC(C2CCCS2)=O)C2(CC2)C1 S(=O)(=O)(c1ccc(CBr)cc1)NC1CN(C(Cc2ccc(C)cc2)=O)CC1C#N N1(C(C2(CC)CCC2)=O)CCC(C)C(CC(N2CC(OCCO)C2)=O)C1 c1(OC)cnc(C(N2CC(CC(N3CC(OC)CC3CO)=O)(OC)C2)=O)cn1 Cc1ccc(Br)c(C(=O)NC2CC2(c2ccccc2Br)F)c1F C(CCCCC(=O)N(C)CC1CCN(C(=O)Cc2cc(C)cs2)C1)(OC)OC CC(C)(C(O)C(F)F)NC(c1[nH]ccc1CNC(C1CC1(Cl)Cl)=O)=O Cn1nc(C(=O)NCC2CN(C(c3cnn(CCO)c3)=O)CCO2)cc1Cl N1(C(CCCC(=O)NCC)=O)CCC2(CCCN(c3ncc4ncnc-4[nH]3)C2)C1 C1(NC(c2ccc(SC)s2)=O)CCCN(C(C2CCC(C(N)=O)O2)=O)C1 Cc1cc(C(N2CC(F)(F)CC2C(N2CC(CO)C(C)(C)C2)=O)=O)nnc1O Cc1cc(C(=O)NCCCCNC(C2C3CCCC23)=O)nn1C(C)C1CC1 c1(C(=O)NCC2CCC=CO2)ccnc(CNC(C2(F)CCC2)=O)c1 c1(Cn2cc(C(=O)NCCCN(C(C(C)SCC)=O)C)nn2)ccccc1 CN1CC(C(=O)NCC(CNC(c2ccncc2)=O)S(C)(=O)=O)CCC1=O.C C(=O)(CCC(CC)CC)N(C1CN(C(c2ccc(C#C)nc2)=O)CC1O)C c1(CNc2cn(C)c(C(N3CC4COCC4C3)=O)c2)cc(F)cc(Br)c1F CCCC(C)C(=O)NC1CCC(CNC(c2ccncc2OC(C)C)=O)CC1 N1(C(Cc2cccc(C(C)C)c2)=O)CCN(C(=O)C2=COCC2)C2COCC12 C1(C(=O)NC(C2CN(C(c3ccc(O)cc3)=O)C2)C)CC2(C1)CC21CCC1 N1(C(c2nn(CC)nc2C)=O)CC2CCC(NC(=O)CC=C(Cl)Cl)CC2C1 C(CN=c1[nH]nc(C2CC2)o1)N1CCN(C(C(CC)F)=O)CC1 C1(C(C)C)CN(C(=O)CCC(C)NC(c2ncccc2N)=O)CCN1C Cc1n[nH]cc1CC(=O)NCC1C=CCN1C(=O)C.c1(CC)ccc(Cl)s1.O c1(N2CCC(NC(C3(CCOC)CC3)=O)C2)ccnc(C)n1 O=C(C1CCc2nccn21)NC(c1ccc(F)cc1F)CNC(C1(O)CC1)=O N1(C(c2ccc(CC)cc2)=O)CCOCC(CNC(=O)CCNC(=O)N)C1 C(CC(C)(C)C(=O)NC1CC(CCNC(=O)CCCCC2CC2)C1)OC CC1(C)CCC(C(=O)NC2C=CCN(C(=O)Cc3cccnc3Br)C2)C1 Cc1cc(C(N2CC3CC2CC3NC(C2CC(F)(F)C2)=O)=O)cc(=O)n1C N1(C(C=CC(CC)C)=O)CC2CCC2(CC(=O)N(CC(C)(C)O)C)C1 C(=O)(CC(CC)CCCC)N1CCC(O)(CCNC(CC(C=C)C)=O)CC1 CC1CN(C(=O)COC(C)(C)C)CCC1N(C)C(C1C2CC3C(C2)C13)=O c1(C(=O)N)ccc2c(c1)C=CCC2.CCCN(C(=O)CSCCN(C)C)C c1(C(N(CC(O)CNC(=O)CCCc2nccs2)C)=O)ccn2ccsc12 S(=O)(=O)(c1cnccc1CCc1ccccc1)N(CC(COCC)C)C S(=O)(=O)(c1ccc(Cl)cn1)N1CC(C)C(Nc2ncnc3cc[nH]c23)C1 c1(C(=O)NCC(C2CC2)NC(C(C)(C)C2CC2)=O)cn2c(n1)COCC2 C12(C(=O)NCCN3CCN(C(CCC(=C)Cl)=O)CC3)CCC(C)(CO1)C2 Cc1cnc(C(=O)NC2C=CC(CNC(C3(F)CC=CCC3)=O)C2)c(Br)c1 n1(CCC(=O)NCCCN(C(c2ccc(OC)s2)=O)C)ccc(O)nc1=O C1(NC(C(C)SC(F)(F)F)=O)CCSC12CN(C(c1nnc3ccccn13)=O)C2 C1(C2CCN(C(=O)C=CCF)CC2)(NC(c2cc(Cl)ncc2F)=O)CCC1 c1(C(C(=O)NCC2CCCO2)N(CCCC#C)C)cc(I)n(C)n1 c1(C(N2CC(C)CC(NC(C(C(C)C)N(C)C)=O)C2)=O)cn2ncccc2n1 C1(CNC(=O)Nc2c(C(C(C)C)O)cccn2)CCCCS1(=O)=O CC1CN(C(c2conc2CNC(=O)CCN(C)C)=O)CC(C)C1O C(=O)(C(C)CC(F)(F)F)N(C(CNc1c(C(=O)OCC)cccn1)C)C N1(C(Cc2scc(C)c2)=O)CCC(NC(c2nn(C(F)F)cc2Cl)=O)C12CC2 C#Cc1ccc(OCC(=O)NCC(C)NC(=O)C(F)CC(C)C)cc1 N1(C(c2scc(OC)c2)=O)CC2CC(NC(=O)CN3CCCC3)CC1C2 N1(C(c2cc(=N)[nH]cc2)=O)CCC(NC(=O)CCCCCO)C(CO)CC1 C1(CC)CN(C(=O)CCN(C(=O)CCC2CC2)CCO)CC12CC2 N1(C(CC=CC=C)=O)CCC(OCCNC(c2coc(C(C)=O)c2)=O)C1 C1(NC(c2ncc(C)nc2)=O)CN(C(C2CN(CC(F)(F)F)C2)=O)C2(CCC2)C1 C(c1ccc2c(c1)OCO2)=CC(N1CC(NC(CC(=C)C)=O)CC2(C1)CC2)=O CC1=NOC2(C1)CC(C(N1CCN(C(=O)COC3CCCOC3)CC13CC3)=O)C2 C1(C(N2CC3CCN(C(C4Cc5nccn5C4)=O)C3C2)=O)CC2(CCOCC2)C1 c1(CC(=O)NCC(CNC(C=C(C)c2ccsc2)=O)O)noc(C)c1C#N c1(NC(=O)NC(C2CS(=O)(=O)C2)C)nc(CC(F)(F)F)cs1 C(C=O)C(C)C.C(C(CC(=O)N(C1CC1)C(C)C1CC1)C1CCC1)OCC C(C(CC(C)C)C(=O)NCC(c1ncc[nH]1)C)NC(c1c(C)oc(Cl)n1)=O C(C(CO)C(F)(F)F)NC(CCCNC(C(CC)C#N)=O)=O C1(CC(=O)N)CCC(=O)NC1=O.C1(C(N(CC(O)C)C)=O)CC2(CCC2)CO1 c1(C=O)ccc(OCF)cc1.C(=O)(CCO)NCC(CNC(=O)C=CCF)F N1(C(C=C(C)C(C)C)=O)CCCC(CNC(C2CCC(=O)N2)=O)CC1 C12(CC)CCC1CN(C(=O)CC1(C)CCC1)C2.C1(C(=O)N)(OCC)CC1 CCC(C)C(C(=O)NC1COC(C)(C)C1)NS(C)(=O)=O c1(C(=O)NCC(CCCC)NC(c2cc(O)cnn2)=O)cc(S(N)(=O)=O)co1 c1(C(N2CCC(F)(C(=O)NC(CC)C(=O)NC)C2)=O)ccc(O)c(F)c1 C1(N(C(c2c(C)cc(Cl)cc2)=O)C)CCN(C(C2CCSCC2)=O)CC12CC2 C1(CNC(CCc2ncn(C)c2)=O)CCCCN(C(=O)CN2CCCC2)C1 Cc1cc(=O)n(CCC(=O)NC2CN(C(=O)C3=CC(C)CC3)CC2O)cn1 n1(CC)ncc(NC(=O)C(N)C(C)F)c1C(=O)OC C(=O)(C(C)(C)CC(=O)N1CC(O)(c2cn(CC3CC4CC4C3)nn2)C1)OC C(=O)(C(CO)c1ccccc1)NCC1N(C(C(N)=O)=O)CC1 c1(C(=O)N)csc2c(O)ccnc12.C=C(Cl)C(C)(C)C(=O)NC1CCCCC1C C1(COC)CCCN(C(C2(C)CCN(C(=O)CCc3cncs3)C2)=O)C1 N1(C(C(C)=C(CC)C)=O)CCSCC1CCNC(c1nc(C2CC2)no1)=O C1(N(C(C(COCC)C)=O)CC)CCN(C(c2cncc(C)n2)=O)CC1 C1(NC(c2c(C)[nH]nc2Br)=O)CN(C(=O)Cc2ccccc2)CC(C)(C)C1 C(C(C(=O)NCC(c1cccnc1)O)NC(=O)C(O)COCC)OCC C1(C)(Cn2c(N(CCCCC=C)C)nnc2CC2CC2)CCS(=O)(=O)CC1 C(=O)C(C)CCC(C)(C)C.C1(COCC(=O)N(C(C)C)CC)CCCC1 c1(C(N2CC(CN(C)C)(CO)C2)=O)ccc(C(F)(F)F)c2c1OCCO2 CCCCCCC(=O)NC(C(=O)NCC(c1cnn(C)c1)C)C1(C)CC1 CC1(C)CCN(C(=O)CC2OCCCO2)C1CC(=O)NC(CO)C(F)(F)F C1(CC)CN(C(C2CC(=O)N(CC)C2)=O)CC1C(=O)N(CCCO)C CCCN=c1nc(N2CC(CO)C3(CCOCC3)C2)c2cccc(F)c2[nH]1 c1(C(N2CCC(C)(C(=O)Nc3cccc(F)n3)C2)=O)ccc2nccn2c1 Cc1nccc(=NCC(C)(C)NC(=O)CCC2CCC(=O)NC2)[nH]1 c1(C(=O)NCCN2CCC(Nc3cc(C)ncn3)CC2)cc2scc(C)c2[nH]1 Cc1ccc(CC(=O)N(C)CCOCCN(C)C(C2CCCS2)=O)cc1 N12CC(F)(F)CC1C2=O.Cn1nncc1-c1nn[nH]n1.C1(CC)CCCC1 C=CCC(C(=O)NC1(C2CCCN2C(c2cc[nH]c2)=O)CC1)C(C)(C)C c1(C(C)NC(C2CC(CC)C2)=O)c(F)cc(F)cc1F Cc1n[nH]cc1CC(=O)NC1COCC1CC1CC1.C1(CC=O)CSCCS1.N CCCCCCCCCC(O)C(=O)NCC1(CO)CN(C(=O)CCNC(N)=O)C1 C=CC1(C(N2CCCC(CO)C2C)=O)CCN(C(C2CCCC(=O)C2)=O)CC1 Cc1ocnc1C(N1CC=CC1C(=O)NCC(=O)OC(C)C)=O CN1Cc2ccc(C(=O)NC3CCN(c4cc(Cl)c(O)nn4)CC3F)cc2C1 c1(CN2CCC(C(=O)Nc3nccc(C(N)=O)c3)C2)ccc([N+](=O)[O-])cn1 Cc1cccc(OCC(=O)NC2CCN(C(c3ccc(Cl)cc3)=O)C2C(C)C)c1 N1(C(N(CCC)CCc2ccccc2F)=O)C(=O)NC2(CCCCC2C)C1=O C(C)(C)(CCC(=O)NCCCN1CCC1)NC(Cc1c(C)cnn1C)=O c1(NC(C2N(C(c3c(C)cnnc3)=O)CC(F)(F)C2)=O)ccnc(O)c1[N+](=O)[O-] c1(C(=O)NCC(CNC(=O)C=Cc2cnc[nH]2)F)cc2n(c1)CCCC2 CCCCC(C(=O)NC1COCC1N=[N+]=[N-])NC(c1ccc(CC)nc1)=O N1(C(C(=O)NCCCOCCOC)=O)CCC(CS(C)(=O)=O)CC1 N1(C(C2(COC)C=CCC2)=O)CCCC(CO)C1.c1(C(=O)N)cnc2sccn12 CC1(C)COC(C(=O)NC2CCC(CC(=O)NCC3CSC3)CC2)C1 C(=O)(CCC(=O)c1ccc(Cl)cn1)NCC1N(C(CNC=O)=O)CC1 C(=O)(C(CCCO)c1ccccc1)N1CCC(CCOC)(NC(COCC)=O)C1 C1(CNC(CCCCNC(C2COCC(C)O2)=O)=O)CC2(C1)CC(O)C2 C1(NC(C2CC2F)=O)C2CC3CN(C(=O)CC4(O)CCCCC4)C1C3C2 C(CNC(C12CCC1CC2)=O)(C(C)C)NC(COCCC)=O N1(C(C(CC=CCC)C)=O)CCN(C(=O)CCC2CCCC2)CCC1C C(=O)(C1=CCCCO1)N1CCCC(CNC(C(c2n(C)ccn2)(F)F)=O)C1 C(=O)(CCCCCC(C)C)N1CCN(C(C(C)NC(C)=O)=O)C(C)C1 N1(C(CCN(C(C)=O)C)=O)CCCN(c2nccc(S(C)(=O)=O)n2)CC1C C#Cc1cc(NC(=O)C=CCN(C(=O)C(C)N(CC)CC)C)cc(F)c1 CC1CC(NC(c2cccc(-c3ccoc3)c2)=O)CN1C(=O)Cn1ncnn1 C#CCC(C)(C(=O)N1CCC(CC(C)C)C1)NC(c1ccn(CCF)n1)=O C(C(CC(C)C)C(=O)N1CCC(CNC(=O)CCCN=[N+]=[N-])C12CC2)OC c1(C(=O)NC(C(C)NC(CCCCSC)=O)C(C)C)cnc2c(c1)ncn2C S(=O)(=O)(c1cccc(Br)c1F)N1C(C(N2CCC(C)(C)CC2)=O)CCCC1 C(=O)(CCC(F)(F)F)N(CCCNC(C1CC2C(C1)C2(C)C)=O)CCC.O c1(CC)nc(C)c(C(=O)N(CC(C)O)CCNC(=O)Cc2cc[nH]n2)o1 C1(C(=O)OC)CCCCCN1C(=O)CCCn1cc(Cc2cccc(F)c2C)nn1 C(=O)(CC(C)(F)F)NCC1(O)CCN(C(C(C)C)=O)C1.C(C)(C)C.C=O N(C(=NCc1ccc(N(C)C)cc1)NC1C(C)(C)C1(C)C)C1CCC(SC)C1 C(=O)(C(O)CC(F)(F)F)NCC(c1ccccc1)NC(=O)CCc1cncnc1 C(=O)(C(C)(C)CCCO)NCC(CCCC)NC(c1cnoc1CC)=O c1(-c2ccc(C#N)cc2F)cc(C(N2CCCC(O)CC2)=O)c2cn[nH]c2c1 c1(N2CCC(n3c(OC)ncn3)CC2)nc(-c2ccccc2F)ccc1Br c1(C(N2CCC(NC(C(C3CCCCO3)C)=O)(CF)C2)=O)ccnc2c1CCO2 CC1(C)OCCC1C(=O)NC1CCOC1C(N1CC(CO)(CF)C1)=O C1(CNC(c2c(C(=O)OC)coc2)=O)CN(C(=O)C=CS(C)=O)CCO1 c1(CNC(C(CCC)OC)=O)cc2n(n1)CCN(C(=O)C(CCO)N(C)C)C2 N1(C(c2c(C)c[nH]c2)=O)CC(NC(c2cc(CO)n(C)n2)=O)C2(CCC2)C1 C1(N(C(CCN(CCCCC)C)=O)C)CN(C(=O)Cc2coc(C)n2)CCC1C C1CCCCC1O.c1ccc(Cl)cc1.C1(C(=O)NC2(CS)CC2)CN(C=O)C1 C1(NC(C(C)=CC)=O)CCN(c2cnc(C(=O)OC)cn2)CC1(C)C c1(-n2c(-c3cc(CC(C)C)c[nH]3)nc(CCC)n2)ccc2ccccc2c1 C1(NC(c2c(CC)n(CC)nn2)=O)CCN(C(c2cccc(C)c2)=O)CC1CC c1(C(=O)OC)cc(Br)c2ncc(CN3CCC(c4c(C)[nH]c5ccccc45)C3)n2c1 c1(C(=O)NC2CCCCN(C(=O)CCC3CCCO3)C2)ccc2ccsc2c1 N1(C(c2ccc(C3(C)CC3)cc2)=O)CC2CN(C(C3(F)CCOC3)=O)CC2(C)C1 C1CN(C(C23CC2CCC3(F)F)=O)CC12CC2.C(c1cccs1)=CC(=O)NC.C C1(C(=O)Nc2cnc(OC)nc2C)CN(C(=O)C=Cc2ccoc2)CCC1(F)F c1(CNC(c2n(CCOC)nnn2)C(C)(C)SC)cccc(N(C)C)c1 C1(N(C(C(CC(=C)C)C)=O)C)CC2CCC(C1)N2C(c1cn(C)nc1C)=O CC1Cc2cc(CC(=O)NC34CC(NC(=O)CN(C)C)(C3)C4)ccc2O1 c1(CC(=O)NCCCNC(C2ON=C(C)C2)=O)nc(-c2ccco2)oc1C C1(NC(C(C)SC)=O)CCC(CCNC(=O)Cc2ccn(C(C)C)n2)C1 N1(C2CCC(NC(C=C(CCC)C)=O)C2)CCN(C(c2cc(Cl)n(C)n2)=O)CC1 C(=O)(C(CCCOC)NC(c1ncc(F)cn1)=O)N1CC(C)(CC=C)C1 C(=O)(C(CCC(C)C)NC(C1CCOCC1)=O)N1CC(OCC(=O)NC)C1 CN1CCC(C(N2CC(NC(c3cc(Cl)ccc3O)=O)C(C)C2)=O)CC1=O C1(NC(Cn2c(=N)nc[nH]2)=O)CN(C(=O)COC2CC=CC2)C2(CCOC2)C1 n1(CC)nc(C(F)(F)F)cc1C(N1CCC(CC=O)C1)=O.[SH](=O)(=O)C(C)C c1(OC)ccc(CCC(=O)NC2(CCO)CN(C(c3ncccc3C)=O)C2)cn1 C1(C(=O)NCCCNC(c2cnn(C)n2)=O)CCC2(CC1)CC2(F)F Cc1oc(C#N)cc1C(N1CCC(O)(CN(C)C(c2cc3cscc3s2)=O)C1)=O N1(C(CC2C(C)(C)C2)=O)CCN(C(=O)COC2CCC2)CC(C)(F)C1 c1(OC)cccc(C)c1NC(=O)CC1CCCN(CC(=O)NCC2CC2)C1 C1(C(N2C(C(=O)NCCSC(C)C)(CC)CCC2)=O)CC(C)(C)CN1C C1(NCc2cccc(SC)c2C)CCC2CC1CN2C(=O)OC(C)(C)C C1(C(N2CC=CC2)=O)CN2CCCN1CC2.C1(OC)CC2(C1)CC(C(=O)N)C2.C c1(C(=O)NC(C)CCCNC(C2CSCCS2)=O)ccc(Cl)cc1Cl C1(C(N2CC3(CCC3)C2)=O)CCN(C(C2CCC(CO)CC2)=O)C12CC2 Cc1ccc(CC(N2CCC(C(=O)Nc3cc(NC(C)C)n(C)c3)CC2)=O)cc1 N1(C(Cc2c(COC)cccc2)=O)CCC12CN(C(=O)C(C)SC(F)(F)F)C2 c1(C(=O)NC2C3(CN(C(C(CC(C)C)O)=O)C3)CC2)cc2n(n1)CCCNC2=O CC(C)C(F)(CNC(=O)COCC(F)F)C(=O)N.CCC=O.C(C)(C)C CC(C)C(C(=O)NC1CC2CC1N(C(=O)C(C)Oc1ccc(F)cc1)C2)C(C)C CCC(C#N)(CNC(=O)C(=O)Nc1ccccc1COC)CC c1(NCC(c2ccc(OCC(=O)N)cc2)NC(C)=O)ccccc1P(C)(C)=O C1(N2CCN(c3cccc(C)c3)CC2)CC2CC(C1)N(C(c1cncn1C)=O)C2 C1(C(N2CCC2CNC(=O)Cc2ccon2)=O)(OC)CCCCC1 CC(CC(=O)N1CCCC(C2(NC(=O)Cc3cn(C)nn3)CC2)C1)CC(F)(F)F N(C1CN(C(=O)C(F)C(F)(F)F)CCc2ccccc21)C(c1ccnnc1)=O Cc1ncn(O)c1C(=O)Nc1cccc(C(=O)NC2CC2)c1 n1(CCC)c(C)cc(C=CC(=O)NC2CCCN(C(=O)CC3CCCO3)C2)c1C N1(C(Cc2nc(C)[nH]n2)=O)CC2CCC(Nc3ncnc4c3COC4)C2C1 N1(C(C2CCC(=C)CC2)=O)CCC(C2CC2)C1CNC(c1ccnnc1)=O N1(C(c2cc(CC)n(C)n2)=O)C2CCC1C(C)C(NC(C1(OC)CCSC1)=O)C2 N1(C(C(C2CC2)OC)=O)CC(C)(NC(=O)C=CCN2CCOCC2)C1 C#Cc1ccc(CNCc2cncc(C(=O)Nc3cnc(C)c(C)c3)c2)cc1 N1(C(C2CC2C2CCCC2)=O)CCCC2(CCCN2C(C2C3CCC2CC3)=O)C1 Cc1cn(C(C)(C)C(=O)N2CCC(NC(c3nc(C4CC4)cs3)=O)C2)cn1 C1(C(N2CCC(C)(C)C2)=O)(OC)CCS(=O)(=O)C1.c1(C=O)nc(F)ccc1Cl C1(CNC(COCCCOC)=O)CCCN(C(C2CCS(=O)(=O)N2)=O)CC1 N1(C(Cc2c(C)noc2Cl)=O)CC(C2(NC(=O)CC3CC(=O)C3)CC2)C1 C(C1=CCCOC1)N(C(C(COC(C)C)NC(C1CCCC(O)C1)=O)=O)C CC(C)C(CNC(C1(CF)CC1)=O)C(C)C N1(CCC(=O)NC(CC(C)NC(C2(CC3CC3)CC2)=O)C)CCC(O)CC1 Cc1ccc2c(=NCC(C)(C)Cc3ccccc3)[nH]c(=NC3CSC3)[nH]c2c1 N1(C(CCCSC)=O)CC(NC(c2[nH]cc(C)c2C)=O)C(F)C1 C1(CC(=O)NC2(C(=O)NC)CC2)CCCN(C(C2CCSC(C)C2)=O)CC1 C(C1=NOC2COCC12)NC(C1(NC(C2CCCCC2F)=O)CSC1)=O c1(C(N(CC(CN(C)Cc2cncc(Br)c2)O)C)=O)ccc(F)cc1Cl N(C(=NCc1cc(Br)ccn1)N1CCCC(CC(N)=O)C1)C(CC)C C1(O)(CC)CCCN(C(=O)C=Cc2cnc[nH]2)C1.c1(SC)nccnc1C(=O)N N1(C(CC(CC)CC)=O)CC2CCCN(C(c3ccc(C(C)(C)C)nc3)=O)C2C1 n1(CC(=O)NCC(O)CNC(=O)C#CC2CCCCO2)ncn2cccc2c1=O N1(C(CC(=O)NCC#C)=O)CCN(C(c2cnnn2C=C)=O)CC1C(C)C C1(NC(=O)COCCF)CCOC(C2CCN(C(c3ccon3)=O)CC2)C1 C#CC1(C(=O)Nc2cccc(O)c2)CCN(C(C2CC=CCC2)=O)C1 c1(C(N2CC=CC(NC(C(C(C)(C)C)N(C)C)=O)C2)=O)ccn2nccc2n1 CC1=C(C(=O)Nc2cccc(OC(C)(C)C)c2)CN(C=O)C1.C(C)(C)C.O C(CC(=O)N1CC2CCC1(CNC(c1cncnc1)=O)CC2)(C(F)(F)F)OC N1(C(c2c(C)nc(C)s2)=O)CCC=C(C(=O)N(C2(C)CC2)C)C1 C(CNC(C1(C(N)=O)CC1)=O)(CC(=O)N)OC.c1(CC)noc(=O)n1C C1(CS(C)(=O)=O)(C(N(CC(CNC(CC=C=C)=O)(C)C)C)=O)CCOCC1 Cc1cc(CC(N2CCC23CN(C(C2CCCNC2=O)=O)C3)=O)cc(C)c1 C1(OC)CNC(C)(C(N2CCN(C(C3CCCO3)=O)CC2)=O)C1 CCC(CNC(c1cnn(CC(C)C)c1)=O)N=c1ccnc(COC)[nH]1 c1(NCc2c(C)nn(C)c2C)ccc(S(=O)(=O)N)cc1Cl.c1ccc(Cl)cn1.C C1(F)(C(N2CC(NC(C(C)O)=O)C(C)C2)=O)CCCC=C1F O=C(C1=COCCC1)NC1CN(C(c2cncc(NC3CCC3)c2)=O)CC1O C=C(Cl)CC(C(=O)NCc1ccncc1CC)NC(=O)CC(=O)OC C(=O)(C(=O)CC1CC1)NC(C)CN(C(=O)CC1CCCO1)C CC1CC(CCNC(=O)CCC(F)F)CCN1C(c1ncc(F)cc1F)=O c1(C(=O)OC)ccn(CC(=O)N(CCC)C)n1.C1(C=O)CCC(N(C)C)C1 C1(CC)CCN(C(c2cnc(O)c(F)c2)=O)C(C(=O)NCCC2CCCOC2)C1 C1(C(=O)NCC2OCCN(C(C(C(C)O)C)=O)C2)COc2c(F)cc(F)cc2C1 c1(NC(CC)=O)ccc(C(C)NC(=O)Cc2cccc(OC(F)(F)F)c2)cc1 C(=O)(CN=S(C)(C)=O)NC(C1CCN(C(C(CC)SC)=O)C1)C C1(c2c(C)n(C)nc2)C(C(=O)NC(C)C(=O)N(C)C)CC(=O)N1C C(CC(C(C)C)NC(c1ccnc(C(N)=O)c1)=O)N(C(C)=O)C N1(C(c2c(OCC)cccn2)=O)C2CCC1C(NC(c1c(Cl)cnn1C)=O)C2 N1(C(Cc2c(C)n[nH]c2)=O)CC(C)C(F)(F)C1.c1(CCC=O)cc(C)n(C)n1.N c1(C=O)cn(CC(O)CC)nn1.CC(C)C1CC1.C1(C(=O)N)(OCC)CC1 Cc1cc2c(cc1C)N(CCOc1cccc(F)c1)CC2 C1(NC(CN(CC#C)C(C2CC(C#N)C2)=O)=O)CCCN(C(C)CC)C1 N1(C(C(CC)N(C)C)=O)CC(CNC(c2c(F)cccc2Cl)=O)C(C)(C)C1 c1(C(=O)NCCOCCC)cnn(C2CC2(F)F)c1.c1(C(=O)N)cnc[nH]1 c1(C(=O)N)ccccc1.CC1CCSC1C(N1CC(F)(C)C1)=O.CCN(C)C C1(NC(CSCC)=O)COC2C(NC(c3cnc(C(C)=O)s3)=O)COC12 C1(NC(CCc2cnn(C)n2)=O)CC2(CCN(C(=O)C(F)C(F)(F)F)CC2)C1 N1(C(C(c2cccs2)SC)=O)CC2CC2(C(F)(F)F)C1.C(=O)C(O)C(F)(F)F c1(C(=O)NCC2N(C(CCCNC(C)=O)=O)CCN(C)C2)cnc2ccsc2c1 c1(C(N2CCC(Cn3cc(CCOC(C)=O)nn3)C2)=O)cc2cc(Cl)sc2[nH]1 CC1CN(C(=O)CC(F)(F)F)CC1C(=O)N(C)CCN1CCOCC1 C1(NC(C(CO)NC(c2cc(C)c(C)[nH]2)=O)=O)CCC(F)(F)CC1 C(=O)(C(C(C)C)n1cnnc1)N(C(C)C1CC1)C.C1(C=O)CC=CC1.CO.C Cc1nn(CCO)cc1C(=O)NC1CC(N(C)C(C2CC(C)(C)CO2)=O)C1 c1(NC(=O)NC2CS(=O)(=O)CC2N2CCCC2)ccc2c(c1)CNC2=O c1(CC(C)NC(C(C)N(C)C)=O)ccc(C)cc1.N(S(N)(=O)=O)CC=O c1(OC)cc(C2(C(=O)NCC(C)N(C(=O)C(C)c3ccsc3)C)CC2)ccc1C N1(C(CSC(C)C)=O)CCCC2(CCCN2C(=O)CC2=CCCC2)C1 N1(C(CCC#CC)=O)CC(NC(C2CCN(c3ccccc3)C2=O)=O)CC(F)C1 C1(c2nc(C)on2)CN(C(c2cc(C(C)C)ccn2)C(=O)NC2COC2)CCO1 N1(C(c2c(C)cc(OC)cc2C)=O)CCC(C2CC2NC(=O)C(Cl)=CCl)CC1 C1(N(c2cc(OC)c(Br)cc2)C(C2CCC2)=O)CCC2(CC1)CNC2 CN1CCC2CCN(C(=O)C(C3(C)CC3)NC(=O)C(O)Cn3cncn3)C2C1 c1(N(C(c2cnc(CC)[nH]2)C(=O)NCCC#N)C)cccc(C#N)c1 CC1CNc2ccc(C(N3CC(NC(C4CCCO4)=O)C(C)C3)=O)cc21 c1(C(N(C)CCNC(C2CSCC(=O)N2)=O)=O)cnc(O)c(F)c1 Cn1ccn2ncc(C(N3CC(C)(C)CC3CNC(=O)CCCC3CC3)=O)c12 CC1C(C(=O)NCCC)=NOC1C.c1(CC(=O)N(CC)C)ccnn1C.C(N)=O c1(CN(S(C)(=O)=O)Cc2ccccc2Br)cc(Br)cc(I)c1O N1(C(Cn2ncc(C#C)c2)=O)CC(C(=O)NOCC(C)O)CC1(C)C C(=O)(C(C)CC(C)C)NCC(CN(C(c1cn(CC=C)nc1)=O)C)C O=C(CCCC1CCCO1)NC(CC1CCC1)C(=O)N1CC(N2CC(F)C2)C1 CS(=O)(=O)c1ccc(C(=O)NC2CN(C(C3(C4CCC4)CCC3)=O)CCC2O)[nH]1 CC1CCc2ccccc2C1NC(=O)Cc1ccc(F)c(C(=O)O)c1 N1(C(C2CC(=O)N(CC(F)(F)F)C2)=O)CC(O)C(O)CC12CNC2 C12(CNC(CCC)=O)CC(C1)C(C)O2.c1(C=O)cccc(N2CCNC2=O)c1.N CC1OC2(CNC(C3(C#N)CCCC3)=O)CC1C2.C1(C=O)CCC2(CCC2)C1 C1(C(=O)NCC2C(NC(=O)CN3CCCCCC3)C2)COc2ccc(O)cc2O1 c1(C(=O)NC(C)CCNC(C2CC3(CCC3)C2)=O)cc(OC(F)F)cc(F)c1 c1(C(=O)N)cc2cccc(C)c2o1.c1(CC)sc(=N)[nH]c1C(N1CCC2CC12)=O C(=O)(N=c1[nH]c(OC)ncc1F)C1N(C(c2cn(COC)nc2)=O)CC(O)C1 CCC(C(=O)NC(CCF)C(=O)NC1CCCCCCC1)C(F)(F)F N1(C(c2[nH]c(=NCC)sc2)=O)CC(C)(C)OCC1CNC(=O)Cn1nccc1C CN1CCn2ncc(C(=O)N(CCCNC(=O)Cc3c[nH]nc3O)CCO)c21 C1(CC(=O)N(CC(=C)C)CC)Cn2nc3ccccc3c2NC1=O C12(NC(c3cc(CC)oc3C)=O)CCCN(C(C3COC4COCC34)=O)CC1C2 N1(C(c2c(C)csc2)=O)CCCC(C2CC2NC(c2cnn(C3CC3)c2)=O)C1 C(=O)(C1COCc2ccccc21)NC1(C)CN(C(c2cnc(C(F)(F)F)s2)=O)C1 CC(C)(CC(F)C(=O)NC1CN2CCC1CC2)NC(c1ccn(C2CC2)n1)=O Cc1cncc(CC(=O)N(CCC(C)NC(c2oc(C3CC3)cc2C)=O)C)c1 N1(C(CCOC(C)C)=O)CC(CO)C2(C1)CN(C(C1CC3(CCC3O)C1)=O)C2 c1(-c2nc(C)oc2)ccc(NC(=O)CC2COCC(C)O2)cc1 c1(C(=O)NC2CC(C)NC2)cncn(C)c1=O c1(C(=O)OC)nc2c(s1)CCN(CCCCN=[N+]=[N-])C2 N(C(=NCC1CCNC(=O)C1)NC1CCN(c2ncccc2F)C1)C(C)C1CC1 C1(CNC(CC(=O)NCC)=O)CCN(C(c2csc(COC)c2)=O)CC1C c1(C(=O)NC(CN(C)C(C2(C3CCCO3)CC2)=O)(C)C)cc2ccccc2nc1O C1(C(=O)NCCN(CC(C)O)C(=O)C)CC2CCC(C1)C2.CC(N)=O.S c1(C2CCN(C(c3ccc(C4(CC)CC4)cc3)=O)CC2)ncc(Cl)cc1F Cc1ccc(C(=O)NCC2CC2(F)F)cc1O.C(=O)CC=CC(C)(C)C.C C1(CC(=O)N(CCOCC)CC)CCCCC1.C(=O)(CCC)N.C(N)=O CCC(CNC(C1CCOCCN1C(=O)CCC(C)CN(C)C)=O)C(C)(F)F N1(C(CNC(CC)=O)=O)CCOC(C(C)NC(c2ncccc2CC)=O)C1 C(=O)(C1CSc2ccccc21)N1C(C)C(NC(=O)CC#N)CCC1 C#Cc1cccc(CCC(=O)NCC(C)(C2CCC2)NC(=O)C(=O)NCC)c1 C1(c2nnc(C)o2)CCN(C2CCNCC2)CC1 CS(=O)c1ccc(C(N2CCC(Cc3cccc(F)c3)C2)=O)cc1 Oc1c(CNC(c2ccc(Cl)c(Cl)c2)CCC(F)(F)F)c(Br)cc(F)c1F Cc1ncccc1C(C)NC(C1(NC(=O)C(C)C2CCCO2)CCCC1)=O C(CO)(CCCCNC(=O)C(=O)Nc1ccc(F)c(Cl)c1)NC(CCC(=C)C)=O C=CCC(CC=C)C(=O)NCC1CN(C(=O)C=CC2CC2)CC1(F)CO C(C)(C)(C(=O)N(CCOCCO)CC)NC(C(C)N)=O c1(C(N2CC(CNC(CC=C=C)=O)N(C)CC2)=O)ccc(C)c(Br)c1N c1(CC)cc(NC(=O)C2=NOC(C)C2)cc(F)c1.C(=O)(C(O)C(C)(C)C)N C(C(C)(CC)NC(=O)CCC1CCC1)NC(C=CC(CC)C)=O C(=O)C(C)S(C)(=O)=O.C1(CC(=O)OCC)(C(N2CCC2)=O)CCCC1 c1(OC)cc(C(=O)NCc2n[nH]cc2C(=O)NCCC(N)=O)[nH]n1 c12cccc(c1)C(=O)N2.C(=O)(C(=O)N1CC(CCO)C1)NC(C)C C=CC(C)(C)CC(=O)NC(Cc1ccoc1)C(=O)NC1CC2(CCC2)C1OC C#Cc1cc(C(N2CCC(C)(NC(=O)Cc3nnc(C)o3)CC2)=O)ccc1C C1(NC(COC)=O)CC(C(F)F)(NC(=O)C(F)(F)Oc2ccccc2)C1 N1(CCNC(=NCC)NCc2ccccc2C)CCCc2ccccc21 C12(C(N(CC(C3CCN(C(=O)CSC(F)F)CC3)F)C)=O)CCC(N=[N+]=[N-])C1C2 Cc1cc(=N)[nH]cc1C(N1C2CCC1C(NC(=O)C(C)(C)C(N)=O)C2)=O C1(C(=O)OC)CC1C1CCN(Cc2ccc(OC)c(SC)c2)C1 CC1CN(C(=O)CN(S(C)(=O)=O)C)CC1NC(=O)COC1CCCC1 c1(C(=O)NCC#CCNC(=O)CCSc2ccoc2)cc(-c2cccnc2)no1 CC1(C)CCC(CNC(c2cccc(CO)c2)=O)(NC(c2ccc[nH]2)=O)CC1 N1(C(c2nc(C)oc2)=O)CC(C)N(C(C2CC2c2ccncc2F)=O)CC1C Cc1cc(N2CCC(NC(=O)C(C)OCC3CC3)C2C)c(Br)cc1[N+](=O)[O-] c1(CC(=O)N(CCCN(C)C(C2CSCCO2)=O)C)c(O)ncnc1O C1(C(N(CCCC)Cc2cc(Br)ccn2)=O)CCC(C(=O)OC)CC1 N1(C(C(c2cnn(C)c2)OC)=O)CCCC(NC(C2(F)CC=CC2)=O)CC1 c1(OC(C)(C)C)ccc(OC(c2ccccc2OCC(F)(F)F)=O)cc1 C(=O)(C1SCc2cccnc21)N(C(CCNC(c1c(CC)[nH]cc1)=O)C)C c1(CC(C)C(=O)NCCC(=O)C(C2CCCCC2)O)cccc(Cl)c1.CCC.CC C1(CNC(c2c(C)ccs2)=O)CC2CCC(C1)N2C(=O)CNc1nccs1 Cc1ccccc1CC(=O)NCC1C=CC(NC(=O)Cn2cncn2)C1 C=CCCCCCC(=O)N1CCN(C(c2nn(C)cc2C#C)=O)CC1C1CCC1 c1(CC(=O)N(C)CC2CN(C(=O)C#CC(=O)N(C)C)C2)c[nH]c2cnccc12 C1(CNC(C(C)=C(C)C)=O)CCN(C(=O)CC2CC(F)(F)C2)CC1(F)F C1(O)(C(N2CCC(CNC(C(C)C3CCC3)=O)C(C)C2)=O)CCCC(C)(C)C1 C(=O)(C1=CCN(C(=O)CCCC(=O)OCC)C1)N(CCCC)CC N1(C(C=CC)=O)CCCC(O)(CCNC(c2cc(C3CCC3)[nH]n2)=O)C1 C1(O)(CC(=O)NCCC2CN(C(c3ncn(CC)n3)=O)C2)CCOCC1 C1(N(C)C(c2nnsc2C(F)F)=O)CCCN(C(c2ccns2)=O)CC1 C1(C(=O)NC(CCCC)CNC(=O)CC2CC(CC)C2)CC2CCC(C1)N2C CCC(C(C)(F)F)NC(=O)C(C)(C1CCC1)NC(C1CCCC1OC)=O n1(CCC)cc(C(c2nnnn2Cc2ccco2)NC(C)CCSC)cn1 C12CCC(C1)N(C(=O)C(O)Cc1cnc[nH]1)C2.CCS(=O)(=O)N1CC(C=O)C1 C1(NC(C(C)n2cnnn2)=O)CN(C(=O)CCC(C)(C)C#N)CC(F)(F)C1 C1(CF)CC(=O)C1.C(C(O)CCO)NC(CCN(C)CC(=O)O)=O C=C1CCN(C(=O)CCC(CC)SC)C(C(=O)NCCC(C)(C)F)C1 C(c1ccccc1C)=CC(=O)NC1CCCN(CCOCC)C1 Cc1cc(NC(=O)Nc2ccc(N(C)C)nn2)c(C)cc1Br C1(C(=O)NCC(c2c(OC)ccc(OC)c2)O)Cc2cccc(Cl)c2C(=O)O1 c1(C(=O)NC(C(=O)NC2CC(C(C)C)OC2)CO)cccc(F)c1N C(=O)(C(O)CC(F)(F)F)N(CCNC(C(C)(C)C(F)F)=O)CC1CC1 C1(NC(C(CCC)(C)CC)=O)CCC2(CC1)CN(C(=O)CC1OCCO1)C2 C(=O)(CC(CC)C(C)(C)C)NCC(CNC(c1c(C)cc(CC)o1)=O)(C)O CC(C)(C)[Si](C)(C)OCCN(CCO)C(c1cc(-c2cccc(Cl)c2)[nH]n1)=O CCCC(C)(CCC)C(=O)N(CC(O)CNC(C1CC(n2cccn2)C1)=O)C C1(NC(c2c(CNC(C)=O)ocn2)=O)CC12CC(OC1CCOC1)C2 CCC(CC(=O)NC1CCC(NC(=O)CCCOC)CC1)SC N1(C(C2(NC(C(CSC)OC)=O)CC2(C)C)=O)CCC(C)(C#N)C1 C(CC(O)CC(=O)NCC1CCCN1C(c1ccc(C2CCOC2)cc1)=O)SC N1(C(C(CC)=CC)=O)CCN(C(=O)C(n2ccccc2=O)C)CC1C1CCCC1 c1(-c2n(CC)ncc2)nc2c(s1)CC(C(=O)NC(C)C)CC2.c1cc(C)cs1.C C(=O)(C(C)(C)C(O)C(C)C)NCC(N(C(CC=CC)=O)C)C1CC1 CCS(=O)CC(=O)N1CCCC(NC(=O)CCC(N)=O)C1 c1(CN2CCC(n3nccc3N)C2)ccccc1N1CCCC1.N1(C(=O)C)CCCCC1.O Cc1ccc2occ(C(=O)NC3CC(C)(C)C3)c2c1.C1(C(=O)N)CC12CCCC2 C1(NC(C(CC)(C)C)=O)CCN(C(c2cccc(C(N)=O)n2)=O)CC1O C1(CCOC)CCN(C(=O)C(CO)NC(c2cc(Cl)n[nH]2)=O)C1 c1(C(=O)NC(CN(C(C2C(OC)CCC2)=O)C)C)nccc(Cl)c1F C1(C(=O)NC(CC=C)CNC(=O)CN(C2CC2)CC)CCOC(C)(C)C1 C1(F)(C(=O)OC)CN(C(=O)CCN(C(=O)C(=O)N(C)C)C(C)C)C1 c1(CNC2C(C(=O)Nc3c(C(=O)OC)cccn3)C2)cnc(OC)cc1C C(C(=O)NC(C)CC(C)(C)O)(C(C)C)NC(CN(CC)CC)=O N1(C(c2csc(C)c2C2CC2)=O)CC2CN(C(C3(N(C)C)CCCC3)=O)CC2C1 C1(NC(C(C2CCOC2)NC(C2CC(C)(C)C2)=O)=O)CCC(=O)NC1 Cc1occc1C(=O)NCC(CNC(c1cc(C2CC2)[nH]n1)=O)CO N1(C(c2c(C(=O)OC)noc2C)=O)CCCC2(CC(C(=O)OC)=NO2)C1 Cc1csc(C(=O)NCC2CCCCC2)c1C.c1(C=O)cc(C(F)(F)F)c[nH]1.N c1(C=O)cccc(F)c1O.C1(CNC(C(C)OCCN(C)C)=O)CCCC1.N c1(OC)ccc2[nH]nc(C(N3CCCC(CO)(NC(c4ccns4)=O)C3)=O)c2c1 C1(CC(N2CCN(CCF)CC2)=O)COCCN1C(=O)C1=CCCC1 C=CCC(CNC(c1cnn(C(F)F)c1)=O)NC(C1(CCOC)CC1)=O c1(C(=O)NC2C(NC(c3c(CN(C)C)ccs3)=O)CCCC2)ncncc1C#N c1(C(N(C(C(=O)NCCNCC)C)C)=O)cccc(Cl)c1F C#Cc1cccc(OCC(=O)NC2COCCC2)c1.C1(C#N)(C(=O)N)CC1(C)C N1(C(C2CC(=O)NC2)=O)CC2CCN(C(=O)C3=CCCOC3)C(C2)C1 C1(C)(COC)CCCN(C(=O)CC2(C)CCN2C(c2oc(C)cc2C)=O)C1 c1(CC(N2C(CN(C(=O)CCF)C)CC(F)C2)=O)ccc2c(c1)CCO2 c1(CC(C#C)N(C)C(c2cnn(CC3CCOC3)c2)=O)ccc(C)cc1 c1(OC)ccc(N(C(=O)CNCCC(C)C)C(C)C)c(OC)c1 n1(CCCC)nnnc1C(CCC1CCCCC1)NC(C)COCC C1(NC(C2CCS(=O)(=O)C2)=O)CC2CCC1N2C(c1cccc(F)c1)=O c1(CC)ccc(C)nc1C(N1CCSC(COC)C1)C(=O)Nc1ccc(F)cc1 C(C(COC)C(=O)NC1CC2(C1)CC2)OC.c1(C=O)ccc(C2CCOC2)s1 N1(C(C(C)=C2CC2)=O)CC(C)(C(=O)NCc2ccc(Cl)cc2)CC1(C)C C1(CCC(N2CCC(N(C(=O)C3=CCSC3)CC3CC3)CC2)=O)CC2CCC1C2 C1(CC)CN(C(c2coc(CNC(C3CCCCC3O)=O)n2)=O)CCN1C C1(C(=O)NCCN(C(=O)CC2CN3CCC2CC3)C)CN(S(N)(=O)=O)C1 N1(C(C(C)(N(C(CN2C(C)CCC2)=O)C)C2CC2)=O)CCC(O)(C(N)=O)CC1 N1(C(C(CC#C)O)=O)CCN(C(c2ccn(CCC)n2)=O)C2(CCC2)C1 C1(C(C)NC(c2cn(CCO)nn2)=O)CN(C(=O)CCCCF)CCO1 CC1(C)COCC(NC(=O)Nc2cc(-n3cnnn3)ccc2F)C1 n1(CC(N2CCC(=CCNC(C(CC)(C)C)=O)CC2)=O)ncn2cccc2c1=O N1(C(=O)CN2C(=O)CCC2=O)CC2CCN(C(C3C=CCS3)=O)CC2C1 C1(C(=O)NCCc2cccc(C)c2)CC(S(N)(=O)=O)C1.c1(C=O)cnsc1.N c1(C(=O)NC2C(CC(=O)NC3(CC)CCOCC3)CCC2)cc(C)nnc1O C(CS(C)(=O)=O)N(CC)Cc1nn[nH]n1.C1(=O)NCO1 c1(CC(N2C(C(=O)NCc3cnc(Cl)s3)CCC2)=O)cccc(F)c1I C(=O)(C(F)CC1CN(C(C2CN(C(C)C)C2)=O)C1)NCCNC(CC)=O CC1(C)CCC(C(=O)NCC2CCOC2)C1.c1(C=O)cc(-c2ccoc2)[nH]n1.N C(C(C(=O)N1CCC1c1ccccc1)C(C)(C)C)NC(c1nc(C)sc1C)=O C1(C(=O)NCC(CC=C)NC(c2cn(C)nc2C(C)C)=O)CNC(=O)N1C C1(NC(=O)CCCOC2CCOCC2)CC(N=c2[nH]c(Cl)ncc2C(F)(F)F)C1 N1(Cc2n(CC)ncc2)CCc2c1ccc1[nH]c(C(=O)Nc3ccns3)cc21 c1(CC)ncc(C(=O)NCc2cc(C(=O)NC3(CC)COC3)ccn2)cn1 CC1CN(C(=O)C=CCNC(=O)CCC2CC2C)CCC1O S(=O)(=O)(c1cc(Cl)ccc1OC)NC(C(CC)C)C(=O)N1CCS(=O)C(C)C1 C1(NC(c2cnc(C(C)(C)C)o2)=O)COCCN(c2cc(Cl)c(O)nn2)C1 c1(C(=O)NC(CCCNC(C2(COC)CCCO2)=O)C)ccc(Cl)c(Cl)c1O C(=O)(C(O)CCC(C)C)NC(CCC)C(O)C(=O)N1CCN(C(C)=O)CC1 CN1CCn2ncc(NC(c3csc(Br)c3)c3nnnn3C3CCOC3)c2C1 C1(N(C(C(C)NC(CC)(C)C)=O)CCO)CCN(C(=O)C(CCO)N(C)C)CC1 C1(C2CCCC2)(C(N2CCN(CCC)CC2)=O)CCC1.C1(C)(CC)CC1C(=O)N c1(C(=O)NCc2ccc(C(=O)NC(C#C)(CC)CC)cc2)ccc2c(c1)CC2 n1(CCC)nc(C)c(C(=O)NC(CO)C(C)NC(=O)CN(C)C)c1C Cc1ccncc1CC(=O)NCC1CC1C(N1CCCC1CCO)=O CC1=C(C(=O)NC(C2CN(C(c3cnc(O)c(F)c3)=O)CCO2)C)CCC1 Cc1ncc(C(=O)N(C2CCN(C(=O)CCN3CCCC3=O)C2)C)cc1N C1(C=O)CCN(C)C1.C1(C=O)CC(=C2CC2)C1.C(=O)(NC)NCC.N Cc1cc(C(N2CC3C(CNC(C4(C)CCCC4)=O)C3C2)=O)cc(O)n1 CC12CC(C(=O)NCCCCCn3cc(C4(CO)CC4)nn3)(C1)C1(CCC1)O2 Cc1nc2c(C(N3CC(NC(c4cscc4C)=O)C(C)C3)=O)cccc2o1 Cc1cc(N)c(F)c(C(N2CCC(F)(C)C2)=O)c1F.C(=O)C(C(C)O)N(C)C.N C=CCCC(C)(C)C(=O)N(CCCNC(=O)C#CC1(C)CC1)CC C(=O)(N=c1ccn(C(C)C(=O)OC)[nH]1)NC(C(=O)OCCC)Cc1ccsc1 CC(CC(=O)NC1CCCC1NC(C1CC(c2ccccc2)C1)=O)P(C)(C)=O C(C)(CCC(=O)N1CCCC(CNC(c2cnc(CC(C)(C)C)s2)=O)C1)SC C(CO)(CCC(C)C)NC(CCOC1CN(C(c2cc(COC)[nH]n2)=O)C1)=O c1(N(C2CCN(C(c3ccc(C(F)(F)F)[nH]3)=O)C2)C)ccc(C(N)=O)cc1 C1(NC(CC(=C)Br)=O)(CO)CCCN(C(=O)Cc2cc(CC)nn2C)C1 C(=O)(C1=CCC(C)CC1)N1CC(C(C)NC(c2cnc(CC(C)C)s2)=O)C1 Cc1cn2c(CC(=O)NC3CC(NC(=O)Cc4cnoc4)C(O)C3)csc2n1 C12(NC(CSc3cccc(C)c3)=O)CCCN(C(=O)Cc3n[nH]c(C)n3)C1C2 C(CC1=CCN(CC(=O)NC2CCCC2)CC1)NC(C1C(C)OCC1)=O C1(C#N)(C(=O)NCc2scc(C(N(C(CO)CO)CC)=O)c2)CCCC1 n1(CCCCC(=O)NCC(C)N(C(C(CSC)O)=O)C)cnc2c(N)ncnc12 CCC(C)CC(C)C(=O)N(C)CCN(C)C(c1ccc(OC)nc1)=O CCCC(C)C(=O)N1C(C(=O)Nc2cc(N(C)C)ncn2)CC2CC12 C12(NC(CCc3n(C)ncc3)=O)CCCN(C(=O)CCCC(F)(F)F)CC1C2 CC(CC(=O)NCC(C1CCC1)NC(=O)Cc1cnn(C)c1)C1CCCC1 N1(CC=CC(=O)NC(C2CN(c3cnc(F)cn3)C2)C)CCc2ccccc21 CN1CCN(N(CC2CC2)Cc2ccccc2)CC12CCC2 C(C)(N=c1[nH]c(N2CCN(CC(=O)N(C)C)CC2)nc(=N)[nH]1)c1cnc(C)s1 C1(NC(Cc2cc(OC)no2)=O)CN(C(=O)CCCN(C)C(C)C)CCC1CO C1(C(=O)NC2C(NC(Cc3cc(C)[nH]n3)=O)CCC2)CCCCC(C)(C)C1 c1(C(=O)N)ccc2nn(C)cc2c1.C(=O)(C(C)(C)c1cnsc1)N(CCC)CC C1(NC(C2(OC)CCOC2)=O)CN(C(c2ccc(Cl)c(F)c2N)=O)CC2(CC2)C1 c1(OC)nccc(C(=O)NC2CN(C(c3cc(-c4ccco4)on3)=O)CC2O)n1 c1(C(=O)NC(C2CN(C(C3CC3C3CCCCC3)=O)C2)C)coc2ccccc12 C1(c2nnnn2C2COC2)(NC(CC)COC(C)C)CCCC(F)(F)CC1 CC(C)CCNC(=O)Cn1ccnn1.C1(C(=O)N)CCN(c2nc(=N)[nH][nH]2)C1 N1(C(Cc2ccn(C)c2)=O)CCOC(C2CN(C(C3(F)CC=CCC3)=O)C2)C1 N1(C(C2(C)CC(O)CN2C(=O)CN2CCOCC2)=O)CCC2C(=O)NCC2C1 C(=O)(CC(COC)COC)N(CCC(C)NC(CCCC#C)=O)C C1(C(=O)NCCC(C)C)CCCCC1C(N)=O.c1(C(=O)N)cccc(CCO)c1 c1(COC)ccc(C(=O)NCC(C)N(C)C(c2coc(C3CC3)n2)=O)o1 c1(C(=O)NC(C)CCNC(c2ncn(C)n2)=O)ccccc1SC(F)(F)F CCCCCCCCCNC(c1nnnn1CCC)(CC)C1CC1 C1(c2ccccc2)(NC(C(F)=C(C)C)=O)CCN(C(=O)C2=C(Cl)CC2)CC1 Cc1cc(N)c(C(=O)NCC2CN(C(C3(C)CC3(C)C)=O)CC2(C)C)cc1F c1(C(c2nnnn2CCSC)NCC(C(=O)NC)C)ccc2ccccc2n1 c1(OC(C)C(N2CCC(C)C2c2cn(CCN(C)C)nn2)=O)cccc(C#N)c1 N1(C(C2CCCC(C#N)C2)=O)CCC=C(C(=O)NCC2(CO)CCCC2)C1 c1(C(=O)NCC2CCN(C(CCSCC)=O)C23CC3)cncc2ncccc12 N1(C(c2cc(OCC)no2)=O)CCCN(C(c2ccc(F)cc2F)=O)C(CO)C1 C1(C)(C(=O)NCCCn2cc(-c3nc(C)sc3)nn2)COC(=O)OC1 c1(NCCNC(CC)=O)[nH]c(=NCCCc2cnn[nH]2)nc2scnc12 C1CC2(CCN(C(=O)C(C)(C)F)C2)C1.C(c1cccs1)=CC(=O)NC(CCC)C c1(C(=O)NC(CNC(CC(CC)OC)=O)(C)CC)ncn2c1CCCCC2 N1(C(=O)NCCC2CC=CC2)CCC(C(F)(F)F)C2(CCOCC2)C1 C(=O)(CC(C)(C)C(F)(F)F)NCC(CNC(C(c1n(C)cnc1)O)=O)O C1(C(N(CC(CN(C(C2C(=C)C2)=O)C)O)C)=O)CC(=O)CC12CCC2 Cc1c(C(=O)NC2C3CN(C(=O)C=Cc4ccco4)CC23)oc2c1C(=O)CCC2 C=C(CNC(c1cnc(CC(C)C)s1)=O)CCNC(C1CC1=C)=O c1(C(=O)NC2C3CN(C(c4cc(C(C)C)[nH]n4)=O)CC32)ccc2ncccc2c1 Cc1cc(C(=O)NC2CC(C)(C(=O)N(CC(C)C)CCO)C2)cnn1 C(C)(CCCC(=O)Nc1cncc(Cl)c1)NC(C1C(CC)C1)=O C12(C(=O)NCC(CN(C(C3C(C=C)C3)=O)C)C)CCN(CC1)S(=O)(=O)C2 CCCC(C(O)C(=O)N1CCC2(CCOC2)C1)NC(=O)CCCCN(C)C C#Cc1ccc(C(=O)NC(c2cccnc2)C(=O)N2CCC2)o1 C(=O)(C1CCc2nccn21)N(CCCNC(C(C)(F)c1ccccc1)=O)C1CC1 c1(C2N(C(C=CCN(C(CCN(C)CCO)=O)C)=O)CC2)ccccc1 c1(C(=O)NC2(CNC(C(c3c(C)nn(C)c3)C)=O)CC2)ccn2c1CCCC2 N1(C(C2(C)CC2(F)Cl)=O)CCC(NC(=O)C=Cc2ccccn2)C(F)C1 c1(C(=O)NC2C(CNC(C3CC(=O)N3)=O)CCC2)cnc2c(c1)CCOC2 C1(SC)COCC1N=c1[nH]c(=NCCN2CCC2)c2c(F)cccc2[nH]1 N1(C(c2cn(C)c(=O)cn2)=O)CC2(CCC2)CC1C(=O)NCC(F)C1CCC1 c1(C(=O)NC2CC(CNC(CCC(=C)C)=O)C2)[nH]c2cc(Cl)cc(Cl)c2c1C C1(c2nnc(NC3CC(=O)NC3=O)n2CC2CCCO2)CCC2(CCC2)O1 S(=O)(=O)(c1cccc(Cl)n1)N1CC(CC(=O)Nc2cn(C)nc2C(F)F)C1 c1(C(=O)NC(CNC(c2c(CC)cno2)=O)C(C)C)c(Cl)ccc(F)c1F Cc1cc(C(=O)NOCc2cn(Cc3cnc(Cl)cn3)nn2)sc1Cl c1(C(N(C2CCN(C(=O)CC3CNC(=O)C3)C2)C)=O)cccc2c1CC(=O)N2 C(=O)(C(O)C(C)(C)C)NCC1(CNC(CCc2cc(C)no2)=O)CC1 C1(N(C(C=CCN(CC#C)C)=O)C)CN(C(=O)CC(C)C(C)C)CC12CC2 c1(C(=O)NC2C=CCN(C(CC=C=C)=O)C2)cc([N+](=O)[O-])cc(Br)c1C N1(C(C(CC)(C)C)=O)CCC(C2CC2)(CNC(c2ccccn2)=O)C1.C(C)=O CC1(NC(C2CNC(=O)CN2C(=O)Cn2cccn2)=O)CC2(CCC2)C1 C(C(F)(F)CO)NC(C(C1CCCCC1)NC(c1nocc1Cl)=O)=O N1(C(CSC(C)C)=O)CC(NC(=O)Cn2cncn2)C(C)(C)C1 N1(C(=O)NCc2nc(-c3ccccn3)cs2)C2CCC1C(O)C(O)C2 C1(N(C(COCC)=O)C)CN(C(c2cc(C3CC3)cc(F)c2)=O)CCC1C Cc1cccn2ncc(C(=O)NCC3CCCN3C(c3ncc(Br)cn3)=O)c12 c1(C(=O)NC2CCC(CCNC(CNC(CC)=O)=O)C2)cnc[nH]c1=N c1(N2CCCC(CNC(C(n3cc(C)nc3)(C)C)=O)C2)ncnc2ccsc12 c1(C(=O)NCC(CC)NC(c2cnc(N(C)C)s2)=O)ccc2c(c1)COB2O N1(C(c2cc(Cl)ncc2Cl)C(=O)NC)Cc2cnn(-c3ncccn3)c2C1 c1(C(=O)NCCCCNC(C2C(C=C)C2)=O)ccc(C2CC2)o1 N1(C(C(CC)Oc2ccccc2)=O)CCCC12CCN(C(=O)C(C)(C)SC)C2 C12(CC(N3CC4(CSC4)C3)=O)CCC1CN(C(=O)C(O)Cn1cncn1)C2 CC(C)CC(C(=O)N(CCCN(C)C(c1cnc(C(C)O)s1)=O)C)C(C)C N1(C(C(COC)(C)OC)=O)CC2OCCN(C(=O)CN3CCCNC3=O)C2C1 C1(C(N(CCN(C(=O)C=CC2CCCO2)C)C)=O)CC12CCCC2 N1(C(c2ccc(Cl)c(F)c2O)=O)CCC2CCCC(C1)N2c1nnc(C2CC2)s1 C1(c2n(-c3cccc(F)c3)nc(Cc3ccncc3)n2)CCCC2(CCC2)C1 C1(C(=O)NC(CC#C)(C)C)CC12CC(NC(=O)C(C)C)C2 CCCC(C(=O)NCC(c1ccccc1F)NC(c1cn(C)cn1)=O)OCC c1(N(CC(C)CO)C)nc(NC2CCCN(C)CC2)c2ncsc2n1 c1(C(=O)NS(=O)(=O)CC2CCOCC2)cccc2[nH]c(CO)nc12 C12(CNC(c3cc(C)[nH]n3)=O)CCCN(C(c3cc(F)ccc3C)=O)C1C2 C1(NC(C(C2CCOCC2)OC)=O)(C)CCCCC1.C1(C(=O)N)C(C)C1(F)F Cc1cc(CNC(c2n[nH]cc2C(F)(F)F)=O)on1 C(=O)(CS(=O)(=O)C1CCCC1)NCC1C2CN(c3nc(SC)nc(C)c3)CC21 C1CCC2(CCC2)O1.C1(OC)CC(C=O)N(C(C2CC(=C3CCC3)C2)=O)C1.N N1(C(C(CCC)C(C)C)=O)CCN(c2nc(CC)nc(C)c2OC)CC(C)(F)C1 C1CC2(C1)CC21CCC1.C(CC(F)F)(C(=O)N)N(C(=O)Cn1cnc(=N)[nH]1)C C12(CC)CN(C(=O)CCC(C)CN(C)C)C(C1)C2.c1(CC=O)ccnn1C.C C1(C)(OC)CCCN(C(=O)C(C)(C)CCCNC(=O)CC(C)C(F)F)CC1 C(=O)(CCCC(C)C1CC1)N(CC#CC)C.C(=O)(C(C)N=[N+]=[N-])NCC CC#CCC(C)NC(=O)COC1(C)CN(C(=O)C(C)(F)c2ccon2)C1 C(=O)(CCP(C)(C)=O)N(C(C(=O)NC(C=C)(C)CC)CC)C C(=O)(C#CC(C)(C)O)N1CC2C(NC(c3c(C)con3)=O)(C2)C1 C(C(C)CC(=O)NC(CO)C(O)c1cccnc1)NC(C)=O c1(CC(=O)NCCCCOC)sc(S)nc1C.C1(C(=O)N)CCC1.C(C)=O N1(S(C(C)C)(=O)=O)CC2CCC(C1)C2NCc1ccc(Cl)cn1 N1(C(CN(C(C(C)C2CCC2)=O)C)=O)CCN(C(=O)CC2CC2(Cl)Cl)CC1 c1(COC)nc(C)c(C(=O)NCc2cccnc2)s1.c1(C=O)ccsn1.C c1(C(=O)NCC2(NC(c3c(C)cn(C)n3)=O)CC2)ccc2[nH]nc(Cl)c2c1 C1(N(C(=O)CC2CC2C(F)(F)F)C)CCCCC1.c1(C=O)nnn(C)c1N.N C1(C(=O)NCCN(C)C(c2ccncc2)=O)CC2CCCC(C1)C2.C(C)(C)C CC1(C)CN(Cc2cccc(Br)c2F)CCC1NC(c1ccn2ccnc2c1)=O CC(C)CCCCC(=O)NCC1(C2CC2)CCN(C(c2ccc(C#N)o2)=O)C1 Cc1cc2occ(C(=O)NCCC(C)NC(=O)Cc3cccnc3O)c2cc1C c1(CC)cncc(C(=O)N(CC(CC)NC(=O)C=CCN(C)C)C)c1 C(=O)(C(C(=O)NCC(C)NC(=O)C(F)(F)c1nccn1C)OC)OC C1CN(C(c2ccc(N(C)C)cn2)=O)CC(C)(C)C1.c1(OC)cc(C(=O)N)on1 N1(C(C2(C(=O)NC)CC2)=O)CC2CCC2(C(=O)NCC2(C)CCOC2)C1 c1(-c2ccc(C(N(CC(CNC(C(C=C)(C)O)=O)O)C)=O)o2)cccc(F)c1C N1(C(CCOC(C)C)=O)CCOCC1CNC(c1cncc(C(N)=O)c1)=O C1(C(=O)NCC2C(C(=O)NCC3(OCC)CC3)C2)CC1(C)C c1(C(=O)NC(C2CN(C(=O)C(C)(Cl)Cl)C2)C)ccc2c(c1)OCCO2 N1(C(C(COC)C)=O)CC2(CCC(NC(=O)C(C)(C)NC(C)=O)C2)C1 Cc1cc(CNc2ncn(Cc3ccc(Br)cc3)n2)cc(C)c1C c1(CC(C)C)ccc(F)c(F)c1.C=CCC(CC=O)NC=O.C(C)(C)C.O C1(C(=O)NCC(C(=O)NC)O)CCCCC1.c1(C(=O)N)cn(C2CC2)cn1 c1(NC(CC2N(C(=O)Nc3cc(CC)n(C)n3)CCC2)=O)cc(Cl)cc(Cl)c1Br c1(N2CCCC(CCCCC)C2)ccncc1S(=O)(=O)N(C1(CO)CCOC1)C C=C(C)CC(C(=O)N1CC2CC2C1)NC(c1cccnc1NC)=O c1(C(=O)NC(CN(CC(COCCOC)O)C)C)c(OC)ccc(Br)c1C Cc1cc(F)ccc1CC(N1CC(NC(c2cc(N)ccn2)=O)CC1C)=O N1(C(C=C(C)c2ccsc2)=O)CC2CC(NC(c3sncc3C)=O)C1C2 n1(CC(=C)C)nc(-c2cnn(C)c2)nc1C(C)Cc1ccc(C)o1 C(C(C)CC(C)C)(c1nnnn1CCCF)NCc1nnc(CC)s1 c1(NC(=O)COC)cc(C(=O)NC(CCNC(CC)=O)C)ccc1C C(=O)(C(C)C(C)(C)C)NCc1nc(C(CC)O)nn1-c1ccccc1 CC1(C(N2CCCC(NC(=O)CCc3cscn3)C(F)C2)=O)CC(C2CC2)=NO1 Cc1ccccc1OCC(=O)NCC(C)(C)NC(=O)CNS(C)(=O)=O c1(C(N2CCCC(C)(CNC(C3(OC)CCOC3)=O)C2)=O)cnc2[nH]cncc1-2 C1(C(=O)NCCCCNC(CC2CCN(C)C2=O)=O)CCn2nccc2C1 N1(CC(=O)NCCN(CCC)C(c2cnc(OC)s2)=O)CCNC(=O)C1 N1(C(CSCC#C)=O)CC2CC3CC2C1C3NC(c1ncoc1C1CC1)=O N1(S(CC(C)NC(=O)OCc2ccccc2)(=O)=O)CCC2(COCCO2)C1 C1(C(C)C)CN(C(c2cc(O)nn2C)=O)CCC1NC(=O)CS(N)(=O)=O C1(NC(C2CC23CCCC3)=O)CCN(C(C2(C(O)C(F)(F)F)CCC2)=O)CC1 c1(CCC(N2C3CC(C2)C3)=O)cc(F)ccc1F.CN1CCC(=CC(=O)N)C1.C N1(CCn2c(CCN(CC)CC)nnc2N2CCOCC2)CC(C)OC(C)C1 C1(C(=O)NCC(C)N(C(=O)CCc2ccon2)C)CCCN(C)C1 c1(CCC(c2nnnn2C)NCC(=C)CC)ccc(OC)c(OC)c1 C(=O)(CCCCCO)N(CCN(C(c1n(CC)nnc1)=O)C)C(C)C CN1CCN(c2ccnc(NC3CCOC(c4ccncc4)C3)n2)CCC1=O CC1CCOC1CC(=O)NCCN(C(=O)COCP(C)(C)=O)CCOC N1(CC(=O)NC(c2ccccc2)C(C)C)CCN(CC(=O)OC(C)(C)C)CC1 c1(C(N2CC3CN(C(c4cc(Cl)nc(Cl)c4)=O)CC3C2)=O)ccc2c(n1)CCC2 C1(NC(=O)CCOC2COC2)CCCCCC1NC(c1cnc(O)s1)=O c1(C(N2CCC(C)C2)=O)nc2cc(F)ccc2s1.C(C)(C(=O)NC)(C1CC1)OC N1(C(=O)CO)CCC2CCC(C1)N2C(=O)Cc1ccc(OC(F)(F)F)cc1 C(=O)(C(C)(C)CC(=O)N(C(C)CNC(=O)C=Cc1ccccc1Cl)C)OC C(CC(C(=O)NCc1nc[nH]n1)NC(c1[nH]nnc1C)=O)SC c1(Cn2cc(C3N(C(C(CC)C#N)=O)CCCC3)nn2)cc(Cl)ccc1F c1(CCC(=O)NC(CNC(C23CC(CO2)C3)=O)C2CC2)sccc1Cl C1(NC(C(C)=C(C)C)=O)COC2C(NC(=O)C(c3ccccc3F)C)COC12 c1(OCC=C)cccnc1C(=O)NCCCC(C)NC(=O)C(C)CO C(=O)(CCC(C)NC(c1ccc(CO)o1)=O)N1CCC(NC(CC)=O)C1 C(N=c1[nH]c2ccccc2o1)C1(CNC(=O)CCCc2ccc(F)c(F)c2)CC1 c1(C(=O)NCC(C)CNC(=O)CCNS(C)(=O)=O)noc2ncccc12 N1(C(COCCC=C)=O)CC2(CCN(C(=O)C=CC3CCOC3)CC2)CC1C c1(C(N2C(CNC(C3(c4cc(C)[nH]n4)CC3)=O)CCC2)=O)cc(C)cnc1Cl C1(NC(C2(COC)CCCC2)=O)(C)CCCCC1.C12CCCCC1CC(=O)N2 CCC(C(=O)N1CC(C)CC1C(N1CC(N2CCOC2=O)C1)=O)C(F)(F)F N1(C(c2c(CNC(c3ccc(C)o3)=O)noc2)=O)CCCC(C)C1CCO CC1CN(C(=O)C(O)C2CCCC2)CCN1C(=O)CC1CCOC1 c1(C(C(=O)NC2CCC(NC(=O)NC(C)C)CC2)O)ccc(Cl)c(F)c1 C(=O)(C(C)C(C)(C)C)N.N1(C(c2ccc(C(=O)OC)s2)=O)CCOC(CC)C1 C(N=c1ccnc(NCCC2CCCC2)[nH]1)C1CCC(NC(CCSC)=O)C1 C1(NC(c2c(C)c(Cl)ncc2)=O)CN(C(=O)CSc2nc[nH]n2)CCC1(F)F N1(C(c2cnc(CC)s2)=O)CCCCC1CN(C)C(C1CC2(CC2)CO1)=O c1(OC)ccc(CN2CCC(c3cn(-c4ccc(N)cn4)nn3)C2)nc1Br C(=O)(C1CCC(=O)c2ccccc21)NC(CNC(c1c(OCC)cccc1)=O)C C1(NC(N2CC(NC(C3CN(C4CCCCC4)C3)=O)C2)=O)CCCCCC1(F)F C1(OCC(C)C)CCN(Cc2cncc(F)c2)CC1 c1(C(=O)NC2(CC=C)CN(C(c3cnc(S)n3C)=O)C2)ccc(C)c(F)n1 C#CCCC(C(=O)NCc1ccc(CC)cn1)NC(c1ccc(C#C)cn1)=O C(=O)(C(C)(C)CC(=O)N1CCOCC(C)C1)OCC.C(=O)C(F)CC1CC1.C C1(C(CN(CCC)CC23CC2CCN3)=O)CC(C)(F)C1 C1(NC(c2nccc(OC)c2N)=O)CC2CC(NC(C3CNC(=O)C3)=O)CC2C1 c1(CC(C)C(=O)NCCNC(C2CC2F)=O)cnc2ccccc2n1.C1CC1.C Cc1cnc(C(N2CC3CC(C2)C3NC(c2sccc2C(F)F)=O)=O)c(C)c1 C1(C(N2CCC(O)(C(C)NC(C=C(CCC)C)=O)C2)=O)CCC([N+](=O)[O-])CC1 CCCCCCC(C)C(=O)NCC1CN(C(=O)C(C)N2CCC2)CC1C N1(C(CSc2c(C)cccc2)=O)CCN(C(=O)COC(=O)CO)CC(C)C1 C1(C(=O)NC2CC(OCC)C2)CC2(CC(NC(C3CCCC3)=O)C2)C1 N1(C(CCC)=O)CC=CC(NC(C2CCC2)=O)C1.C(C)(C)C.C=O.C(N)=O c1(NC(c2ccc(Cc3ccccc3)cc2)=O)cccc2c1CCS2(=O)=O N1(C(C(CC)n2cccn2)=O)CC2CC(C1)N2C(=O)C(C)(C)C(C)C c1(C(=O)NCC2C(NC(CCSCC)=O)C2)nnc(O)c2ccccc12 c1(C=O)ccc2c(c1)C(=O)OC2.C12(CC)CCC1CN(C(=O)C=CCO)C2.N c1(C(C)C)ccc(C(=O)NC2CCN(C(C34CC(F)C3C4)=O)C2)cn1 C1(NC(C2CCN(C(c3c(C)n(C)nc3)=O)C2)=O)CC2CC1C(O)C2O Cn1nc(C(=O)NCc2c[nH]c3ccc(C(C)(C)C)cc23)c2c1CNCC2 c1(CC)ncnc(CC)c1C(=O)N(CC(C)C)C.c1(C(C=O)C)nc(C)cs1.N C1(c2nnnn2CCCSC)(NCCCC(CC)O)CCC2COC1O2 CC1(NC(C2CCC2n2cccn2)=O)CCN(C(C2(C)CC2(F)F)=O)CC1 c1(OCC#C)ncccc1C(=O)NCCCCCNC(C1(C)COC1)=O N1(C(c2ccc(C)[nH]2)=O)CC(C(=O)NCc2c(C)cccc2C)C(F)(F)C1 c1(C(N2CC(C)C(NC(=O)C(C)(C)C3CC3)CC2)=O)cnc2ccncc2c1 CCCC(C(=O)OC)C(=O)N1CCCC(NC(C2CC2(Cl)Cl)=O)C1C c1(SC(C)(C)C)ccccc1C=C(C#N)C(=O)N(O)Cc1ccccc1 c1(OC)ccn2ncc(-c3nc(-c4cccs4)nn3C3CCSC3)c2c1 C1(CC)CCOCC1.C(S(C)(=O)=O)C1(CC=O)CC1.CC1CC1CC(=O)N Cc1ccccc1C(C(C)NC(=O)COc1cccnc1)NC(c1ccsn1)=O C1(C=O)CNC(=O)CC1(C)C.C12CC(C1)C2.C1(OCC)C(C(=O)N)C1C N1(C(CCCCC=C)C(=O)NCCC2(C)CC2)CCN2C(=O)OCC2(C)C1 C12(NC(c3cc(C)ncc3)=O)CCC(CNC(=O)CCN3CCC3)(C1)OC2 c1(C(N(C2CCN(C(C3CC(OC(F)F)C3)=O)CC2)C)=O)ccnc(C2CC2)n1 C1(CC(=O)N)CN(C(=O)C=Cc2cscn2)CCO1.c1(C(N)=O)nc(C)no1 C1(CC(C)NC(C2(F)CCCOC2)=O)CCN(C(=O)CCCCNC(N)=O)CC1 N1(Cc2c(C)cc(F)cc2)CC2CN(C(c3occc3Br)=O)CC2C1 c1(C(N2CCCC(NC(c3cn(C4CC4)nn3)=O)CC2)=O)cccc2nccn12 c1(C=O)c(N)sc(C)c1C.N1(CCC)CCCC(C(=O)NC(C)(C)C2CC2)C1 C(C1=CCN(C(=O)Cc2ccc(F)cc2F)CC1)NC(C1CC12CCCOC2)=O N1(C(C2CC(F)C2)=O)CCC2(CCCN2C(C2CCC3(C2)N=N3)=O)CC1 C(Cn1cc(CCC=C(C)C)nn1)(CC(C)C)NC(Cc1ccn(CC)n1)=O c1(CC)[nH]nc(C(=O)NCC(=C2CN(C(c3ncccc3N)=O)C2)F)c1[N+](=O)[O-] C=CC(C)(CCOC)C(=O)NC1CC(NC(=O)CC2CC(F)C2)C1 C(=O)(C1CCCc2cncn21)N1CC(C)N(C(c2nc(Cl)c(Cl)s2)=O)CCC1 N1(C(C=C(CC)CC)=O)CCC(N=[N+]=[N-])(C(=O)NCCC(C)C(F)F)C1 Nc1cc(C(N2CC3CC(NC(C4CCCCC(=O)N4)=O)C2C3)=O)cc(O)c1Cl C1(CCC)CCC(CNCc2ccc(-c3csc(C=O)c3)cc2)CC1 C(=O)(C1CCC(=O)c2cccn21)N1C(C(C)NC(=O)CCC(C)(C)F)CCC1 Cc1nscc1C(=O)NCCC1(C(=O)Nc2sccc2CN(C)C)CC1 c1(C(COC(CC(c2ccc(F)cc2F)C)=O)=O)cc(F)ccc1N n1(CC)cc(CC(=O)NC2C=CC(CC(N3CC(CC(C)C)C3)=O)C2)cn1 C=CCCC(C)(C)C(=O)OCC(=O)NCc1ccc(I)cc1Cl N1(C(=O)CN2CSCC2=O)CCC2(CCCN2C(C2CC23CCCCC3)=O)CC1 c1(C(=O)NC2(CF)CCN(C(C(C(C)C)SC)=O)C2)ccc(F)c(C(C)C)c1 C1(NC(C2(c3n(C)ncc3)CC2)=O)C2CN(C(=O)C(=O)NC3CC3)CC12 c1(-n2cc(C(NC)=O)nn2)ccc(C)cc1.C(CSC)(C(=O)N)OC.C1CC1 N1(CC2CCc3c(cn(C)n3)C2)CCC(O)(C2(C(=O)O)CCC2)CC1 N1(C(C2C(C)CC2)=O)CC(C2(NC(c3ccc(N4CCCC4)cc3)=O)CC2)C1 S(=O)(=O)(c1c[nH]ccc1=NC1C=CCC1)NCCP(C)(C)=O c1(CC)ccc(C(=O)NC2CC(CC(=O)NC3CSC(C)C3)C2)o1 C1(C(N2CC3=C(CN(C(c4c(C)nsc4)=O)C3)C2)=O)CC12CCC(F)(F)CC2 C1(CC(=O)NCc2c(C)scc2)CC2(C1)CN(C(C1(F)CCOC1C)=O)C2 CC(Cc1ccccc1)C(=O)NC12CC(C(=O)NCC3(O)CCC3)(C1)C2 N1(C(c2cccc(C)n2)=O)CCN(C(=O)CCCc2ccncc2)CC(C)(F)C1 C1(C(=O)NCC(C)NC(=O)CCc2nnc(C3CC3)o2)CCN(C)C1 C1CC2(C1)CN(C(=O)Cc1cc(C)cc(C)c1)C2.Cc1cnc(CN)s1.C=O C1(NC(=O)CC2CCCCC2O)CC(CNC(C2(CCO)CC2)=O)C12CCC2 c1(NCC(COC)C)ncc(S(=O)(=O)NCCC2(C)CC2(Cl)Cl)cc1Cl C(=O)(CCC(C)C)N1CCC(CCC(=O)NC(CC)CC)C1 CCC(C)(C#N)C(=O)N1CCC(NC(c2cnsc2)=O)C(CO)C1 Cc1cc(C(=O)NC(C)CCCCNC(=O)C(C)O)cc2nn[nH]c12.C1CC1.C Cc1cc(-c2nc(C(=O)NC3CC3CNC(c3cncs3)=O)co2)ccn1 c1(-c2ccn(CC(=O)NC3COCCOC3)n2)ccccc1Cl c1(-c2n(-c3c(C)cccc3C)nc(-c3ccsc3)n2)cccc2nc(O)n(C)c12 C1(N(C)C)CCC(C(=O)NCC2CC(O)(Cn3cc(C4CC4)nn3)C2)CC1 C1(C(=O)NC(CC)COC)CC(C)CCN1C(c1cc[nH]n1)=O c1(CC)ccc(CC(=O)NC2(CNC(c3ccc(C)nn3)=O)CC2)cc1F C12(NC(C3CC(OC)C3)=O)COC(CNC(=O)CC)(C1)C2.C(C)=O C1(NC(=O)NC2(COC)CCCSC2)CCC=CCCC1 c1(C(CNC(=O)NC(CCC)C2CC2)N(C)C)cccc(OC)c1 Cc1nc(O)ccc1C(N1CC(=O)NCC1C(=O)N(CC(F)Cl)C)=O C1(CNC(=O)N)(CO)CC2CCC1CC2.C1CCN(C2CC2)CC1c1nn[nH]n1 CC1C(C(=O)N(C(C(N)=O)C2CC2)C)CCCN1C(C1CCSC1)=O c1(CCC)ccc(CC(=O)N(CC(C)NC(C2(C)COCCO2)=O)C)cc1 N1(C(c2cnc(C(C)C)[nH]2)=O)CCN(C(C2CCC(C)(O)CC2)=O)C2CCCC12 c1(C(=O)NC2CCCN(c3ncnc(CC)c3F)C2)cnc2ccccn2c1=O N(C(=NCC(C)C)N1CCC(c2ncccc2C)C1)CCOC(c1ccccc1)C c1(C(N(C2CCCN(C(C3CC(=O)N3)=O)C2)CCO)=O)cc(Cl)nc(Cl)c1 Cc1ccc2nc(C)c(C(=O)NC3CC(C)(NC(C4C(C)CC4C)=O)C3)cc2c1 Cc1ccc(C(=O)NC2CC3CCC2N(C(C2CCCOC2)=O)C3)c(=O)n1C CC1(C)CCC(CNC(=O)CC2CC2)OC1.C1(C)(C=O)CC(F)(F)C1.C C1(COC)(CNC(=O)C(C)(O)C2CCC2)CN(C(C2CCC2)=O)C1.O C(=O)(C#CC1CCCCO1)NCCCNC(c1ccnc(C)c1Cl)=O c1(C(C(=O)N(C(C)CO)C2CC2)NC(CSCCC)=O)ccnn1C C(=O)(CC1OCCc2ccccc21)N1CC(NC(C2OCCN(C(C)C)C2)=O)C1 C1(C)(CC=O)CC(F)(F)C1.c1(C(C)C)ncsc1C=O.CC(C)C1CCC1.N N1(C(C2CN(C(C(C)N=[N+]=[N-])=O)CC2C2CC2)=O)CCCC(O)(C2CC2)C1 N1(C(C2C3CCC2(c2ccco2)C3)=O)CC2CCC(C1)N2C(c1ccsn1)=O c1(C(N(C)CC2N(C(C(CC)CN(C)C)=O)CC(F)C2)=O)ccc(O)cc1Cl c1(OC)cccc(C)c1C(=O)N(C)CC1CC(F)CN1C(C1CCCOCC1)=O c1(OCCC(=C)C)cccc(NC(c2nnc(S)n2C)=O)c1 N1(C(CCC(=O)OCC)=O)CCN(C=O)C(C)C1.c1cccc(C(C)(F)F)c1.N C#Cc1nccc(=NCc2cccnc2-n2cccn2)[nH]1 N1(C(COCC)=O)CCCCCC1C(=O)NCCCCc1ncc[nH]1 N1(C(CC(CC)NC(=O)CC2CCCC2)=O)CC(CO)C2(CC2)C1 C(C)(C)C=O.C1(O)(CC)CN(C(=O)CN(C)C(N)=O)C1.C=O.CC.N C(C(F)(F)CO)NC(C(C1CN(C(=O)CCSC)C1)OC)=O N1(C(c2nncn2C)C(=O)NC)CC2CC(Nc3ccccc3OC)CC1C2 C1(CCC)CN(C(c2nc(Cl)oc2C)=O)CC1C(=O)NCCC1CCCO1 O=C(CC1=CCCCC1)NCC1(F)CCN(C(C23CCC(CO)(CC2)C3)=O)C1 N#Cc1ccc(CC(=O)NC23CCN(C(=O)CSc4ccccn4)CC2C3)cn1 c1(COCCNc2cc(NCC)ncn2)cc(C)c(OC)c(C)c1 S(=O)(=O)(c1ccc([N+](=O)[O-])cc1)N1CCCC(C#N)(C(=O)OCC)C1 C1(NC(C=CCOC)=O)CN(C(c2ccc(=O)n(C3CC3)c2)=O)CCC1.C c1(C(=O)NCC2C(CNC(C(C=C)C)=O)C2(F)F)cc(C)sc1N C1(C(=O)OC)C2CC2CN1C(=O)Cc1cn(C)nn1.c1(C(=O)N)scnc1Cl c1(-c2n(C)ncc2)ccc(NC(c2cc(C(F)(F)F)ccn2)=O)nc1 C(=O)(C(CCC1CCC1)NC(c1cc(CO)oc1C)=O)NC(COC)C(C)C N1(C(Cc2ccc(C(C)C)cc2)=O)CC2CC(NC(c3csc(O)n3)=O)C(C2)C1 c1(C(=O)NC2C(C(C)(C)C)N(C(C3CC3C)=O)CC2)ccc2c(c1)CCCS2 C(=O)(C(O)C(C)C)OC1(CNC(CC2C(OC)CC2)=O)CCOC1 c1(CNC(C(c2cnnn2C)C)=O)ocnc1C(=O)NCCO.C1CCCCC1 N1(C(CCc2ccc(C)s2)=O)CCn2cc(C(=O)Nc3cccnc3Br)nc2C1 Cc1ccc(C(c2nnnn2CC2CCOC2)NCc2cncnc2)c(F)c1F CS(=O)(=O)C1(C(=O)NC2CC2NC(=O)CCC2CCOCC2)CC1 N1(C(C(CCN(C)C)O)=O)CCOCC(NC(=O)COc2cncc(Cl)n2)C1 C(CC(C(=O)Nc1cn(CC)nc1C)NC(=O)CCCOC)OCC C1(C(=O)NC2(CO)CCOCC2)COCCN(C(=O)COCc2ccccc2)C1 C1(CNC(C2(CC)CC2)=O)CN(C(c2ccc(C)nn2)=O)CCC12CCOC2 N1(C(C(CCC)N(C)C)=O)CC(NC(=O)C=Cc2ccco2)CC2(CC2)C1 c1(CN2CCC(CC(=O)Nc3c(CC)cc(O)cc3)C2)cccc2c1CCCC2 C1(C=O)Cc2cccnc2C1.c1(COC)nn(C)c(Cl)c1C(=O)NC1CCC1 C1(C(C(=O)NC2CC2)N(C2CCC2)CCC)CCOC1c1ccccc1 CC1(C)CCC(CNC(c2onc3c2CCCC3)=O)N(C(=O)Cn2ccnn2)C1 N1(C(CN(CCOC)C)=O)CCN2CCN(C(C3(CO)CC(C)(C)C3)=O)CC2C1 c1(C(N(CC(C)C)C(C)C)=O)cc(Br)ccc1[N+](=O)[O-].C(=O)CN(C)C.N c1(CC(=O)NCCN(C(C(CC)(C)C#N)=O)C)c[nH]c2ccc(F)cc12 S(=O)(=O)(C1CCc2ccccc21)N1CC(CC(C)(C)C)C(C(=O)O)C1 c1(C(=O)NCCC(CNC(=O)CC2(O)CCC2)O)cc(Cl)ccc1[N+](=O)[O-] C1(C(NOCC(C)C)=O)CN(C(C2CCCCN2C)=O)CCN1C Cc1cnc(C(N2CCC(NC(c3cc(Cl)n(C)n3)=O)CC2C2CC2)=O)cc1Cl C1CCCCN1C(C1CCC(O)CC1)=O.N(C(C(=O)NC)=Cc1cccs1)C(C)=O N1(C(CCC(C)SC)=O)CCN(C(=O)C(C)OC2CCCCCC2)CC1C(C)C C1(NC(Cn2c(C)cc(C)n2)=O)CCCN(CCN2CCN(C(C)C)CC2)C1C C1(C(=O)NCC(C)NC(C2(OC(C)C)CC2)=O)(SC)CC1 c1(C(N2CC(COC)N(C(c3csnn3)=O)CC2)=O)cc2ccc(F)c(F)c2o1 CCCC(C)CC(=O)NC(CC1CC1)C(=O)NCc1coc(C)n1 CS(=O)(=O)C1CN(C(=O)C(=O)NC(C2CCCO2)CO)C2(CCOCC2)C1 C1(CNC(C(C)(C)C2CCOCC2)=O)CN(C(=O)C=CCO)CC1O c1(C(=O)NCCNC(C2C(CC)CCC2)=O)ccc(C)c2c1CCCN2 c1(OCC)ccc(OCCC(=O)N(CCC)C)cc1.C1(C)(C(=O)N)CCCCC1 C1(C)(C(N(CCN(C(C)=O)CC)C)=O)CCC(=O)CC1.Cc1n[nH]c(C)c1 C(C(CC(C)C)C(=O)NCCC12CC(CCO1)C2)NC(c1c(C)csc1)=O C1(NC(c2c(CC)c[nH]n2)=O)(CO)CCCN(C(C2(C#N)CCOC2)=O)C1 c1(C(N2C(C)CN(CC3CCC(C(F)(F)F)O3)CC2)=O)c[nH]c2cccnc12 c1(OC)cc(C(N2CC(NC(C3(CSC)CC3)=O)CC(C)C2)=O)cc(Cl)n1 C1(CNC(C2N(C(C(n3ccc(C)n3)C)=O)CC2)=O)CC(C)(C)CO1 C#CCC(C)(CC)C(=O)N1CC(NC(c2cc(F)ccc2OCC)=O)C(O)C1 C1(C(N2C(CNC(CCN3CCN(C)CC3)=O)C=CC2)=O)OCCOC1(C)C C1(CN(C(CC=CC)=O)CC)C(C2CC2)CCN1C(=O)C=CC(C)C C(c1cccnc1)=CC(=O)NCC1CCN(C(c2cc(C(F)F)no2)=O)C1.C c1(-c2nnc(C)o2)cccc(C(=O)NCC2(O)CCN(C(c3csnn3)=O)C2)c1 C1(N(C)C(C2CC(n3cnnc3)C2)=O)CCCN(C(C2SCCCS2)=O)C1 N1(C(c2ccc(C)s2)=O)Cc2[nH]nc(NC(=O)CSc3n[nH]c(O)n3)c2C1 N1(C(C2(CCC=C)CN(C(=O)C(CC)n3ccnc3)C2)=O)CCC(C)(C#N)C1 c1(C(N2CCC(N(C(C(CC)OCC)=O)C)CC2)=O)cc(OC)cc(OC)c1Cl CCC(C(=O)N1CC(O)CC1(C)C(=O)NCCN1CC2CC2C1)C(C)C c1(CC=O)cccc(C)c1C.n1(CC(=O)N(CCC)CC)ncc(C#N)c1N.N N#Cc1ccc(C(=O)NCC2(F)CCC(NC(=O)C(c3cccnc3)O)C2)o1 C1(C(C)C)CN(C(C2(O)CCCCCC2)=O)CCCN1C(=O)CC1(O)CCCC1 C1(CC(=O)NCCN(C(=O)C(F)=CC2CC2)C2CC2)CCC(O)C1 C1(NC(C2CC(C#C)(O)C2)=O)CC=C(C(=O)NOC2CCC(O)C2O)C1 N1(C(C(CC(F)F)NC(=O)C(F)OC(F)(F)F)=O)CCOCC2(CC2)C1 c1(C(=O)NCCN(C(=O)C(F)(F)c2ccnn2C)C)cnc(O)c([N+](=O)[O-])c1 C1(NC(C(CC)NC(C)=O)=O)CCN(C(c2n[nH]c3c2CCSC3)=O)C12CCC2 Cn1cc(C=CC(N2CCC2CC(=O)NCC2(Cl)CCC2)=O)nn1 N1(c2ncc(C(N)=O)nc2)CCC2(CC1)CC(NC(=O)OC)CCO2 C1(CNC(=NCC=C)NCc2cccnc2OC)CCC2(CCCOC2)O1 C=CCC(CC)C(=O)NC(CN(C)C(c1cn(CCOC)nc1C)=O)(CO)CO C12(C(=O)NCCCCCC#C)CCC(CC1)N(C(=O)CCCC1CC1C)C2 N1(C(C)C)C(=O)CCC1C(N1CCCC1C(C)NC(c1cncnc1)=O)=O C(=O)(C(C)CC(C)(C)C)NC1C(CC(=O)N(C2CCN(C)C2)CC)C(O)C1 c12ccc(cc1)S(=O)(=O)NC2.C1(c2nc(CC)[nH]n2)CN(CC)CCO1 c1(C(=O)NCC2(NC(CC3(C)CC3F)=O)CCC2)ccc2cnccc2c1 CC(C)C1=NOC(C(=O)NCC2=CCCN(C(C3CCC4(CC4)C3)=O)C2)C1 Cc1nn(C)c(Br)c1C(=O)NC(C)CN(C)C(C1CC2CC2C1)=O CCCC(CC(=O)N(C)C[Si](C)(C)C)NC(=O)CC1CSC1 c1(C(C(=O)NC)N(CC(C)Cc2ccc(F)cc2)C)cccc(OC)c1 C=CCC(CC(C)C)C(=O)N1CC(C(=O)NC(C)C(CC)CC)CC12CCC2 Cc1ccc(-c2nc(-c3cc[nH]n3)nn2CC(C)C2CC2)cc1Cl C(=O)(CCN(OC(C)C)C(=O)CCc1ccccc1)NCCOC C12(C(=O)N)CCCC1CCN2C(=O)CC1CC(N(C)C)C1.C=CCCC1CC1 C1(CCNC(COCCCOC)=O)CCN(C(c2ccc(C)cn2)=O)CC1 c1(C(N2C(CC)C(C(N3CCOC4CC34)=O)CC2)=O)ccc2cc[nH]c2c1 C1(NC(C(C)=CC)=O)CCC2(CC1)CC(NC(c1c(C)nn(C)c1F)=O)C2 N1(C(c2cnn(CC)c2C)=O)CCCC(O)C1.c1(C(=O)N)ccc(C(F)(F)F)o1 c1(OC)cc(F)cc(C(=O)N(C)CCNC(=O)C(C)C)c1N.[SH](C)(=O)=O Cc1nc(SCC2CC2)sc1C(=O)N(C)C(C)C.C1CCCCC1.C(=O)C S(=O)(=O)(c1cc(Br)ccc1C(=O)OC)NCC1CCCN(C(C=C)=O)C1 Cc1cc(C(N2CC3C(C2)N3C(c2ccc(F)cc2Br)=O)=O)ccc1I S(=O)(=O)(CC(=O)NCC(C1CCOC1)NC(c1cc(Cl)sc1Cl)=O)NC N1(C(C2N(C(c3[nH]cc(C)c3)=O)C3C(C2)C3)=O)CC2CC1C(F)(F)C2 C=CCC(CNC(C1CCC1=C)=O)NC(=O)CCN1CCC1 N1(c2scc(C)n2)CCCC(C(=O)NC2(CC)CC2)C1.C(=O)CC(C)N(C)C.N N1(C(C(CC2CN(C(CC3C(C)OCC3)=O)C2)F)=O)CCN2CCC1C2 Cc1onc(Br)c1C(=O)NCCCC(C)NC(C1COCCO1)=O C1(NC(=O)CCc2ncc[nH]2)CCN(C(c2n[nH]cc2[N+](=O)[O-])=O)C12CCCC2 N1(C(c2cc(C)[nH]n2)=O)CC2CN(C(c3nsc4c(Cl)cccc34)=O)CC2(C)C1 c1(NC(N2CCC(F)(C(=O)NC)C2)=O)c(C)nc2ccccc2c1C N1(C(=O)C=Cc2cscn2)CC2CC(NC(C3(CO)CCCO3)=O)C1C2 N1(C(c2ccc(NC(C)=O)cn2)=O)CC2CC(NC(C3CCOCC3)=O)CC2C1 N1(C(c2ccc(CCCC)o2)=O)CC2CC(NC(c3ccsc3OC)=O)CC1C2 c1(CN2CC3(CC(C(=O)OC)C3)C2)nc(O)c2cnn(C)c2n1 N1(C(CC(C)C(F)F)=O)CCC(C2(NC(C3CCC(=O)O3)=O)CCC2)CC1 C(C(C)C(F)(F)F)NC(CCC1(C)N(C(C)=O)CCC1)=O.c1(C(=O)N)cccnc1 N1(C(C2CN(C(CSCCC(C)C)=O)CC23CC3)=O)CCc2ncccc2C1 N1(C(CCCC)=O)CCC(CNC(=O)CCCCCNC(C)=O)C1(C)C C=CCC(C(=O)OC)NC(C1CC1C(C)NC(C1(Cl)CCCCC1)=O)=O C=CCCCCCCCC(=O)NCC1CCN(C(=O)Cc2ccc(C)cc2)CC1 N1(C(c2c(C)ccc(O)c2)=O)CC(C)OC(C)(C)C1.C1(CC(=O)N)CC1(C)C c1cncc(C(=O)N(CCN(C(=O)C(n2cc(C)cn2)C)C)C(C)C)c1.CC c1(C=O)ccc(C)nc1C.C#CC(CC1CCCC1)NC(=O)CO.C(C)(C)C C(CC(=O)N(CC(F)(F)CO)C)(C(F)(F)F)NC(C(CCC)NC(C)=O)=O C1(C)(CCNC(C(C)SC(C)C)=O)CCN(C(C)C(N2CCCCC2C)=O)C1 Cc1cccc(C(N2CCCCC2C(C)C)C(=O)NCc2ccc(F)cc2)c1Br C1(CCNC(C2C(C(C)O)C2)=O)CCCN(C(c2ccncc2)=O)C1.C(CO)O c1(NC(C)=O)cc(Br)ccc1C(=O)OCC1(O)CC2CC1C2 N1(C(c2c(C)scn2)=O)CCC2(CC1)CN(C(=O)CC1CCSCC1)CCO2 c1(CC)nccnc1C(=O)NC1CCOCC1C(=O)NC(CO)C(F)(F)F C(CCC(O)C(=O)NC(c1cnn(C)c1)(C)C)NC(C1CC=C(C)CC1)=O c1(-c2cnc(CS(CC)(=O)=O)nc2)ccc(OC)cc1OC(C)C N1(C(C2C(C(=O)OC)C2)=O)CCCC1CNC(C1(Br)C(C)C1C)=O C(c1cccnc1)=CC(=O)N(CCC(=O)NCCCCO)CC#C N1(C(c2cnc(CC)s2)=O)CCCC1(C)C(=O)NCCC1CCCOC1 N1(CC)CCOC(CNC(C2CC(NC(=O)C(C)(F)F)CCO2)=O)C1 c1(-c2n(C)nc(-c3ccccc3)c2)cccc(F)c1C(N)=O C(=O)(C1=C(SC)CCCC1)NCCN(C(c1cc(F)c(F)c(O)c1F)=O)CC CC1(NC(=O)C(O)P(C)(C)=O)CCCN(C(c2cnc(C(F)F)nc2)=O)C1 C(CCC)(C(=O)N1CC(F)CC1C(=O)NCc1cnc(C)o1)=CCC c1(CNC(=O)NCC(c2ccccc2)OC)c(F)cc(Cl)cc1F C1(C(N(C(CCNC(C(C2CCOC2)OCC)=O)C)C)=O)COCCO1 CC1CN(C(=O)NC(c2ccccc2)CN2CCCS2(=O)=O)C(C)CO1 c1(C(N2CCOCC(CNC(C3(CC)CCC3)=O)C2)=O)cccc2c1CCC2=O c1(CCC)nc(C)c(C(=O)NC(C)CCNC(c2c[nH]c(=N)s2)=O)s1 c1(CCN)cncc(C2CC2)c1.N1(CCNCCCl)CCCC1 c1(C=O)ccc(=O)n(C(C)C)c1.c1(CC)ccc(C=O)o1.C(C)C1CCC1.N CON(CCC(=O)NCCC(N)=O)C(=O)c1nc[nH]n1 CC1CCC(NC(c2n[nH]c3c2CCC3)=O)CN1C(=O)CSc1nnnn1C Oc1ncc(OC(F)F)cc1C(=O)OCC(N1CCOCC1)c1ccco1 C(=O)(C#CC1(C)CC1)NC(C(C)C)CNC(=O)CC1C=CCC1 c1(C(=O)NCCn2ccc(=O)cc2)cc2cccc(Br)c2cn1 CCC(C)(C)C(O)C(=O)NC1CCN(C(C2(F)CCC(F)(F)CC2)=O)CC1 N1(C(c2ccc(C(C)=O)o2)=O)CCOCC(NC(c2ncc(Cl)cc2F)=O)C1 C1(C)(CNC(CC2CC(C)(C)C2)=O)CN(Cc2cc(Cl)ccc2Cl)CCO1 C1(C(N(CCN(C(C2C(C#C)C2)=O)C)C)=O)CCCC(N=c2cncc[nH]2)C1 Cc1nc[nH]c1C(N1CCC(NC(=O)CCc2nnc(C(C)C)o2)C1)=O c1(OC)ccc2[nH]cc(C(N3CC(NC(c4cnc(O)[nH]4)=O)C(O)C3)=O)c2c1 c1(C(N2C(C(=O)Nc3cccc(C(C)=O)c3)CCC2)=O)ccnc(N(C)C)c1Cl c1(CC)[nH][nH]c(=NC(=O)C2CC2c2ccncc2)c1C C(=O)C(C)CCC(C)(C)C.c1(CC)c(C(=O)NCC2C=CCC2)cccc1C.N C(=O)(CCCCCCC(=O)O)N(CC)Cc1ccc(-n2cc(CSC)nn2)cc1 N1(C(c2c(C)scn2)=O)CCC(C)C1c1cn(CCSc2ccccc2F)nn1 C1(n2cc(C(CC)(C)C)nn2)(C(N2CC3CC2C3C(=O)O)=O)CCOCC1 C1(C(=O)NCCCN(C(=O)C(O)CC(F)(F)F)C)CS(=O)(=O)CC12CCC2 C1(CNC(c2cccc(F)c2Cl)=O)CN(C(C2CCCS(=O)(=O)C2)=O)CCCO1 N1(C(c2cc(C(C)=O)on2)=O)CC2CCC1C(NC(c1ocnc1C)=O)C2 c1(CN2C(C)(C(=O)NCc3cnn(C4CC4)c3)CC2)cc(O)cc(Br)c1 N1(CC(N2CCC(C(N3CCC(COC)CC3)=O)C2)=O)CCS(=O)(=O)CC1 c1(OC)cncc(C(=O)N(CC(C)CNC(c2ccsc2Br)=O)C)n1 C12(NC(C3CCCN(CC)C3)=O)CCCN(C(=O)Cc3nncn3C)CC1C2 C1(C(N(C2C3CN(C(=O)CCc4ccccn4)CC23)C)=O)Cc2ccncc2C1 C(=O)(C(C)(CC)CO)NCCC(CNC(CC(CC)C)=O)(C)C C1(C(=O)NCC(C(=O)NCC(COCC)(C)C)(C)C)CC2CCCC2C1 c1(C(=O)NCCCC)cc(F)cc(S(N)(=O)=O)c1.c1(C(=O)N)cccc(N)n1 C1(C(=O)NCC2(C(=O)NCc3n(C)cnn3)CC2)CN2CCC1CC2 C(CC1=CCN(C(=O)C(C)C2CC2)CC1)NC(C=Cc1ccc(C)o1)=O N1(C(C(C)CSc2ccccc2)=O)CC=CC(NC(=O)C(N)=O)C1 C1(NC(C(c2ccccn2)C)=O)CC2(CCN(C(=O)C(C)(O)C3CCC3)C2)C1 c1(OC)c(Cl)ccc(C(=O)N(C2CCCN(C(=O)C(=O)N(C)C)C2)C)c1F c1(C(=O)NCC2CN(C(C(C(C)C)C)=O)C(C)(C)C2)cc2c(cn1)NC(=O)CO2 CC1CN(C(C2CCC(CNC(=O)Cc3ccnn3C)C2)=O)CC(C)(C)C1 c1(C(=O)NCC(CCOC)NC(=O)C#CC2(CC)CC2)cnc2[nH]nnc2c1 C1(NC(C(c2cn(C)nn2)N(CCCC(O)CO)C)=O)CC2CCC1C2 C1(C)(CC)CC(NC(C2(N(C)C)CCCC2)=O)CN1C(=O)CCC(C)(C)C C1(C=O)CC2(C1)CS(=O)(=O)C2.c1(C=O)cc(C(F)(F)F)c[nH]1.CCCC.N C(=O)(C(O)CC(N)=O)NC(C)(C)CCNC(C1(C(F)(F)F)CC1)=O CCC(C)(C)C(O)C(=O)N1CCCN(C(c2ccnc(OC)n2)=O)CC1C c1(N2CC(C)C(NC(C3COC(C)(C)C3)=O)C2)ncnc2c([N+](=O)[O-])cccc12 C#Cc1ccc(NC(c2ccc(CNC(c3cc(OC)nn3C)=O)s2)=O)cn1 CN1CCOC(C(=O)NC2(CO)CCN(C(=O)CCn3cnnn3)C2)C1=O Cc1nsc(C)c1C(=O)NCCOCCCN(C(=O)Cn1nnnc1C)C C1(NC(C(C)(C)OCCC)=O)CCCN(C(=O)C(=Cc2ccncc2)C)C1 C1(CCNC(CCC2(C)N=N2)=O)CSCCN1C(c1nnn(C(C)(C)C)n1)=O N1(C(C2CCN(C(=O)NC)C2)=O)CCCN(C(c2cc(N)ccc2Cl)=O)CCC1 c1(CC(=O)NCC2CCC(C)CC2)cccc(O)c1.c1(C(=O)N)nc(Cl)cs1 Cc1c(C(=O)NC)c(C(F)(F)F)nn1C.C1COCCN1C(C1(F)CCOC1)=O c1(NCCC(=O)OC)ccccc1C1CC1(F)F.C12CCC(CC1)NC2C C=CC(CC)CC(=O)N(C(C)(C(=O)NCCOCCO)C1CC1)C c1(OC)ccc(CNc2ccsc2C(N2CCOCC2C(C)C)=O)cc1Cl c1(C(=O)NC2CCCCN(C(C(C)C(F)F)=O)C2)c(O)ccc2ccccc12 N1(C(C(C=C)CC)=O)CC23CCCC2(C1)CN(C(C1CC12CCOC2)=O)C3 C1(C)(CNC(c2n(CC)nnn2)(C)CNC(C)=O)CCC2(CC1)CC2 [nH]1nc(C2CC2)cc1C(N1CCCC(N(C(=O)CC2CCC(=O)O2)C)C1)=O.C C1(NC(C(C)Cc2ccncc2)=O)CN(C(=O)COC(F)F)CC1N(C)C CC(CCc1cnn(C)c1)N=c1nc2c(cnn2C)c(NCC(F)F)[nH]1 c1(OC)cc(C(=O)NNC(=O)C2CC2C(=O)O)ccc1C1CC1 c1(N2CCC(C)(NC(c3c(C)nn[nH]3)=O)C2)ccc(C#N)nc1 N1(C(COCC)=O)CCN(C(c2cccc(C)c2Br)=O)C(CC(F)F)C1 c1(CC)ccc(CNC(C2CCCN2C(=O)CC2COC(=O)C2)=O)nc1.C CC1(CNC(c2ccc(Cl)cc2)=O)CCCN1C(=O)CCn1cccc1 C1(NC(CN(C)C)=O)CN(C(c2csc(C(C)(F)F)n2)=O)CC12CCC2 C(=O)(CCC(C)(C)[N+](=O)[O-])N(CC(C)NC(c1ocnc1C1CC1)=O)CC c1(C=O)cc2n(n1)CCCCO2.S(=O)(=O)(CC(=O)NCC)NCC.CC.O c1(OC)cc(N2CCN(CC)CC2)nc(C(F)(F)F)n1.C(=O)(C(O)C(C)(C)C)N c1(CC)c[nH]c(C(=O)NC2CC(CNC(C3(C)CCCS3)=O)C2)c1 c1(C(=O)NCC2CCCC(CNC(CCC(C)OC)=O)C2)ncc(C)cc1C N1(C(C2CC(=C)C2)=O)CCC2(CCCC2NC(=O)COCCC(C)C)C1 C1(O)(C(C(N2CCC(OC)C2)=O)NC(c2nocc2C(C)C)=O)CCCCC1 C(c1nc(C)c(C)[nH]1)=CC(=O)NC(CCNC(C(C=CC)O)=O)C Cn1cnc(C(=O)NC2CCC(NC(C3(C)CCCC3)=O)C2)cc1=O C1(C(=O)Nc2c(C(=O)OC)cc(Cl)cn2)CC1C1CC(F)(F)C1 N1(C(=O)CCOc2ccccc2)CCC2(CO)CN(C(=O)C3=CCCC3)CC2C1 C1(NC(C2C(C=C)C2)=O)CCN(C(=O)CC2(C)OCCO2)C1(C)C C(=O)(CCCC(C)C)N(CC(CC)NC(C1(CC)CCC(O)CC1)=O)CC C1(NC(c2c(Cl)nc(OC)s2)=O)CCN(C(=O)COC(F)(F)F)CC1C N1(C(C(Cc2ccccc2)NC)=O)CCC(O)(c2ccc(Cl)cc2)CC1 CC(=NO)C1CC(C(=O)NCC)C1(C)C.N1(CC(=O)N)C(=O)CN(C)C1=O N1(C(c2scc(C)c2C)=O)CCN(C(=O)C(C)n2cnnn2)CC1C(C)C N1(C(c2ccc(C)[nH]2)=O)CC=C(CNC(C2COC3COCC23)=O)CC1 C=CCC(C)C(=O)N1CCN(CCCNC(=O)C(CC)=CCCC)CC1 C(=O)(C(C)CC(C)C)NCC(CNC(Cn1cc(C(=O)OC)nn1)=O)(C)O C1(N(C)C)CN(C(=O)NCCc2ccccc2F)CC1O Cc1cc(CC(=O)N(C2CCCC2)CCNC(C2CC2C)=O)sn1 N1(c2cc(Nc3ccc(N)cc3)nc(C)n2)CCc2ncc(C)n2CC1 c1(OC)ccc(C(C)C)cc1C(=O)NC1CCC1.c1(C(=O)N)cc(Br)ccn1 C(=O)(C1=Cc2ccccc2OC=C1)NCCCN(C(CN(C)C(N)=O)=O)C N#Cc1cc(C(=O)NC2CC(NC(C3C4CCC3(c3cscn3)C4)=O)C2)no1 c1(CC(N2C(CCNC(c3ccncc3)=O)COCC2)=O)cc(F)ccc1Cl c1(OC)ccnc(C(=O)N(CCCCCNC(c2cc(Cl)ns2)=O)C)c1 Cc1nn(CC(=O)NC(CNC(=O)CN2CCC(C(N)=O)CC2)CO)cc1Cl C1(NC(c2c(OC)c(=O)cco2)=O)CCSC12CN(C(=O)Cn1ncnn1)C2 C(C)(CC(=O)NCCCCCc1cn(Cc2ccc(Br)s2)nn1)OC c1(OC)ccc(C(=O)NC2CCC(NC(c3ccncn3)=O)CC2)c(Cl)c1 C(=O)(C1=CCCOCC1)N1C(CC(=O)NC(C)CN=[N+]=[N-])C(C)(C)CC1 C1(NC(c2c(C)nc[nH]2)=O)CN(C(c2ccc(C(F)(F)F)cc2)=O)CC1C1CC1 c1(CC(=O)NCC(C)(C2CC2)NC(Cc2c(C)con2)=O)ccc(C)cc1 C(=O)(C(F)C(F)(F)C(F)(F)F)NCCCNC(C(CC)Oc1ccccc1C)=O Cc1cc(C(N)=O)cc(C(=O)NC(CO)CC)c1.c1(CC=O)cn(C)nc1C.N Cc1cnccc1CNC(=O)C(=O)NCCCn1ccnn1 c1(NC(C)=O)scc(C(N)=O)c1NC(=O)CCC1(C#N)CNC1 C1(C(=O)NC2CCN(C(c3ccc(C(C)(C)C)[nH]3)=O)C2)CC2(CC2)CO1 c1(CNC2CC(CC(=O)Nc3cc(Br)cnc3O)C2)ccnc(Cl)c1Br c1(NC(=O)NC(C2CCOCC2)C)ccccc1NCC(F)(F)F CC1(C)CC2(CO1)CN(Cc1cn(CC(N3CCSCC3)=O)nn1)C2 CCCC(C(c1nnnn1CCSC)NC1(c2ccccc2F)CC1)OC N1(C(Cn2c(C)csc2=O)=O)CC(F)(F)CC1.C12(C=O)CCOC(C)(C1)C2.C C(=O)(C1=COc2ccccc2O1)Nc1ccc(CC#N)c(Cl)c1 Cc1cc2c(cc1O)CCN(C(=O)CN(S(=O)(=O)c1ccc(F)cc1)C)C2 NCC1CN(C(C2COCCC2c2ccc(F)cc2)=O)Cc2ccccc21 c1(C(=O)NC2(C)CN(C(=O)CC3CCCOC3)C2)ccc(-c2cnccn2)cn1 Nc1cc(F)cc(F)c1C(=O)NC1CC1.c1(C2C(F)(C=O)C2)ccccc1.N CC1(C)CCOC1CNC(C1(F)CCN(C(C2COCC2C(N)=O)=O)C1)=O N1(C(c2ccc(C)cc2F)=O)CCN(C(=O)C(C)OC2CCCC2)CC2(CC2)C1 c1(OC)cnc(Cl)[nH]c1=NC1CC(CNC(C2CN(C)C(=O)N2)=O)C1 N(C(=NCC1COC(C)(C)C1)NCc1ccco1)C1CC(OC(C)C)C1 CC(C)C(=O)C(=O)N(CCC(=O)N(C(CO)C1CC1)C)CCCO N1(C(c2cc(C(=O)OCC)n[nH]2)=O)CC(NC(=O)C(O)CC)C(C)(C)C1 C1(CNC(c2n(C(C)C)ccc2)=O)CCCN(C(c2cccc(N)c2)=O)C1 C1(C(=O)NCC(CO)NC(c2ccccc2F)=O)Cc2nncn2C1 C1(C)(C(N(C2CCCN(C(C)=O)C2)CCO)=O)CCN(c2ccccc2)CC1 C(N=c1ccn(CCO)c(O)n1)c1n(-c2ccc(N(C3CC3)C)cc2)ncc1 C1CCC(=O)N1C(c1ccc(C(F)(F)F)o1)=O.c1(C(=O)OC)ccccc1I CC1=C(C(=O)NCC2(F)CCN(C(C3CCCSC3)=O)CC2)SCCO1 CC1CC(C(=O)NCC2CCC(NC(c3cncc(Cl)c3)=O)CC2)=NO1 N1(c2n(CCN(S(CC)(=O)=O)C)nnn2)CCC(C(c2ccco2)O)CC1 C=CC(C)(CCOC)C(=O)N1CCC(C)(C)C(C)C1.C(=O)C(F)CC1CC1.N c1(C(C(=O)NC(C)(C)CO)N(C)C)cccc(Cl)c1 CC1(C)CCCC(C(=O)NCC2CN(C(c3ccc(CO)nc3)=O)C2)O1 c1(C(N2CC(OC)C(NC(=O)C3=CCCC3)C2)=O)nc(Cl)ccc1N Cc1nn(C(C)C)cc1CNCC1CCCCC1 N1(S(=O)(=O)C2CC2)CCC2(CCN(S(=O)(=O)c3ccc(F)cc3F)CC2)C1 c1(CN2CCC(NC(=O)Nc3c(C)c(F)ccc3)CC2)cccc2c1OCC2 C1(C(=O)NCCN(CCCCCC)C(=O)C(C)=CC2CC2)CCN2CCOCC12 C1(CC(N2CCCC(N(C(=O)C(c3cccnc3)O)C)C2)=O)COC(C)(C)CO1 N(C1CCCc2cnccc21)C(C(Br)=C(C)C)=O CN1CC2CN(S(=O)(=O)NCC#N)CC2C1=O CN1CCC(C(=O)N(CCCNC(=O)CCC2NC(=O)NC2=O)C)S1(=O)=O C(=O)(CCC(=O)N1CCCC(CC(=O)NC(c2ncc[nH]2)C)C1)NCCC C1(CNC(c2n(CC)cnn2)=O)C2CN(C(c3cocc3C)=O)CC12 C1CN(C(C2CCCC2)=O)C2(CCC2)C1.C(C(=O)N)SCCOC.C(C)=O c1(CNC(=O)Cc2cscn2)ccc(C(N2CCCC(OC3CC3)C2)=O)cn1 C1(C2CCN(c3nccc(CO)n3)C2)(NC(C2C(C)CCC2)=O)CC1 C1(NC(C(=O)N(CCCNS(C)(=O)=O)C)=O)CCCC12CCCO2 c1(C(N2C(C)C(NC(=O)C(=O)NCCC(N)=O)CCC2)=O)ncn2c1CCCC2 C1(C(N2CCC(N(C)C(c3nnn(C)c3N)=O)C2)=O)COc2ccccc2C1 N1(C(c2nc(C(C)C)oc2)=O)CC2CC2(C(N2CCC(CO)CC2)=O)C1 C=C=CC(C)C(=O)N1CCC(CCNC(=O)CCCC2CC2)C1 C1(NC(=O)CCn2cnnn2)CC2(C1)CC(CNC(C1C3COCC13)=O)C2 C1(C(N(CCOCC(=C)C)CCC)=O)CCOC(C(C)(C)C)C1 O(NC(=O)C(CCCC)NC(C12CSCC1C2)=O)CCOCCOC C1(C(N2CC3CC3(C(=O)NCc3cnc(Br)s3)C2)=O)CCc2ccccc2C1O c1(C(=O)O)ccc(F)c2c1CCN(C(=O)Cc1ccc(F)nc1)C2 N1(CC)C(=S)NC(c2ccc(Cl)c3c2CCC3)C2=C1CCNC2=O Cc1nonc1CC(=O)NC(C)CCN(C(=O)C(Cc1ccsc1)NC=O)C N12CC3=C(C(=NC(=O)C(=O)C14CC4)NN3)C2.C=C(C=O)C(F)(F)F.N1CCCC1.C C(CC(C)C(=O)N(C(C)C)C)=CCC.c1(CC(=O)N)cc(-c2ccccc2)on1 c1(C(=O)NCC(CN(C(C(C)=C2CC2)=O)C)O)cc2c(cnn2C)nc1O c1(C(N(CCCNC(C2(C3CC3)CC2)=O)C)=O)c[nH]cc(Br)c1=N c1(C(C)C)ncncc1NC(c1cccnc1CNC(C1CCCN1C)=O)=O C1(NC(C(C)(N(C(C(=O)N(C)C)=O)C)C2CC2)=O)CCC(N=[N+]=[N-])CC1 c1(C(=O)NC(CN(C(c2c(C)snn2)=O)C)C)cc2ccc(Cl)cc2o1 C1(C(=O)NC2(C)CCCN(C(c3ccc(CO)cc3)=O)C2)Cc2ccccc2S1 O(NC(=O)C#CC1CCOC1)C(C(=O)NCCc1c(C)n[nH]c1)CC(C)C C12(NC(c3cc(Cl)c[nH]3)=O)CC1CN(C(=O)COCC1(F)CC1)C2 c1(C(N2C(CCNC(c3ncnc(O)c3Cl)=O)CCC2)=O)cccc2[nH]ccc12 N1(C(C(CCOC)OC)=O)CC(NC(c2cc(C3CC3)cs2)=O)CC12CCCC2 N1(c2nnc(-c3ncc(OC(C)(C)C)o3)n2C2CC2)CC(C2CC2)C2(CCC2)C1 N1(C(CSCC)=O)CCC(F)(F)C(CNC(C2CC2c2ccccn2)=O)C1 CCC(C)CCCC(=O)NCc1ccnc(C(=O)NOC(C)C)c1 C1(N(C(CS(CC)=O)=O)C)CCC2(CC1)CCN(C(c1cnns1)=O)C2 C(=O)(CCCCNC(C1CC(O)C(F)C1)=O)N(c1cnn(C)c1)CC C(c1cccc([N+](=O)[O-])c1)=C(C(N1CCCC2(CC2)C1)C(=O)NCCOC)C C1(NC(c2c(SC)nn(C)c2)=O)CN(C(=O)CCc2nc[nH]n2)C2(CCOC2)C1 c1(C(=O)NCC2C(C(=O)NC(COC)CO)CC2)c[nH]c2ncccc12 C=CC1(C(=O)NC2CC(O)C(F)C2)CCN(C(c2cc(Cl)no2)=O)C1 Cc1ccc(Cl)c(C(=O)NC2C3CC2N(C(C2CCCN2C(N)=O)=O)C3)c1 C1(NC(C2(CC)CCOC2)=O)CN(C(=O)CCC(F)(F)F)C(CC)(CC)C1 Cc1cc(C)c(C=CC(N2CC(NC(c3cn(C)cn3)=O)C3CC3C2)=O)cc1C c1(C(C)C(=O)N(C2CN(C(=O)CC3CCOCC3)CC2O)C)ccc(F)c(Cl)c1 C1(CNC(CC(=C)C)=O)CCCCN(C(=O)C=Cc2ccccc2OC(F)F)C1 C(C)(CC1CC1)(C(=O)NOC1CCOC1)NC(CC(=O)N(C)C)=O C1(CNC(=O)C(F)=CC2CC2)CC2COCC2N1C(=O)CCC(=O)c1cccs1 C1(NC(CCCCNC(=O)CCC2CC2)=O)CC1C1CCCC1 N1(C(C(C(=C)C)(C)C)=O)CCCC2(CCC(NC(=O)C=Cc3ccncn3)C2)C1 C1(c2nnnn2C(C)C)(NC(c2cc(C)on2)C)CCC2(CCCC2)C1 c1(CC)cc(N)c(C(=O)NC)cc1F.C1(C)CCCN1C(=O)CCc1ccon1 C=CCC(C)(CC=C)NC(C1CC(C)N1C(c1cc(C#N)n(C)n1)=O)=O c1(C(C(=O)N(C(CNC(CCC=C)=O)C)CC)C)noc2ccccc12 C(=O)(C(F)(F)CC(C)C)N1CCCC(CCNC(c2cnc(C)o2)=O)C1 N1(C(c2c(C)nc(C)s2)=O)CCN(C(=O)C#CC(C)(C)C)CC(C)C1 C1C=CCC1.c1(C=O)cscc1C1CC1.CCS(=O)(=O)N(CC(=O)NC)C N1(C(Cn2ccc(C)n2)=O)CCCC(C2CC2NC(C2COC(C)(C)C2)=O)C1 C(=O)(C(C)(C)OC1CCOC1)NCCC(C)N(C(=O)Cn1cncn1)C CCC(C)C(CC(=O)NC(c1n[nH]c(CO)n1)C)NC(c1ncn(C)c1C)=O N1(C(C2C(C)OCC2)=O)CCC(CNC(=O)CC2CN3CCN2CC3)C1(C)C CC1(C)CC(NC(C23CCCN(CC2)C3)=O)CN1C(c1cc(CF)on1)=O N1(C(c2ccc(CC)cc2)C)CC2(C1)OCC(O)C2O CC(CS(C)=O)C(=O)NCCCC(C)(C)NC(c1cnc(O)c(Cl)c1)=O C(=O)(CCC(C)(C)F)N1C(C(=O)NCC(CCOC)O)CSCC1 C1(NC(CCSC)=O)CCC(C(=O)NCCN(C)C(C2CCCO2)C)CC1 C1(CCN2CCN(C(c3ccc(N(C)CC)cc3)C)CC2)CCN(C)C(=O)O1 CC1=C(C(=O)NC2CC2NC(c2cnc3n2CCCC3)=O)SCCO1 Cc1cc(C(=O)N(C2CN(C(=O)C(O)CC(F)F)C2)C)cc(C)c1OC(F)F c1(CCC)cc(C(=O)N)sc1C.C1(C(N(CC)C2CC2)=O)CCC(CCCC)O1 C1(CC)CN(C(c2ccnc(CO)c2)=O)CCN1C(c1ccc(OC)nc1F)=O N1(CC)CCN(C(C2CC(NC(=O)CCCC#N)C23CCC3)=O)CC1=O Cc1oc2ccccc2c1C(=O)NC1CCCN(C(=O)C(O)CCC(C)C)CC1 O=C1CC(C(=O)N2CCOC(CCNC(C3(C(F)(F)F)CCC3)=O)C2)=NN1 C(c1cccc(C)c1)=CC(=O)N(CCC(=O)NC(CCC)C(=O)N(C)C)C c1(C(=O)NCC2(C)CCC(NC(C(CCCC)O)=O)CC2)cccc2c1CCN2 C(=O)(C(O)C(C)CC)NCC1(C(=O)NCCc2ccccn2)CC(=C)C1 CC(CC(C)(C)C)C(=O)NCCC1CN(C(=O)Cc2ncncc2Cl)C1 c1(C(C)=O)cncc(C(N2CCC(C)C2c2cn(-c3ncc(F)cn3)nn2)=O)c1 c1(C(N2CC(CCC)N(C(c3ccns3)=O)CC2)=O)cc(C)c(F)cc1F c1(NC2(C(=O)NC(C3CN(C(C)=O)C3)C)CCOC2)cncc(F)c1 N1(C(c2c(COC)ccs2)=O)CC2CC(O)C1C2NC(c1ccc(C)cc1)=O N1(C(C2CC(C(C)C)C2)=O)CCC2C(NC(=O)CCn3cc(Cl)cn3)C12 C1(NC(C(C)OCC=C)=O)CCCN(C(=O)C(C2(O)CCOCC2)(F)F)C1.C c1ccc(O)cc1.c1(NC2C(C(=O)N(C(C)(C)CO)C3CC3)C2)ccccc1 c12ccc(cn1)[nH]c2=O.N1(CC)CCCCC1CCC(=O)NC1CCC(C)CC1 Cc1cc(CCC(=O)N2CC(n3cc(C4CCCO4)nn3)C2)cc(C)c1 N1(C(CC(C)SC)=O)CCC(CN(C)C(c2sccc2OC(F)F)=O)CC1 c1(C(=O)OC)ccc(C(F)(F)F)nc1.C1CCCCN1C(=O)C(C)=C1CC1.N N1(CC(N2C(CNC(C(CC)n3cncn3)=O)CCC2)=O)CCCS1(=O)=O Cc1[nH]ccc1C(=O)N(CCN(CCCN(C)C)C(C1CCC1)=O)CC N1(Cc2n(C)ncc2)CCC2C(CCCN2C(c2cc(F)cc3ccoc23)=O)C1 n1(CC)ncc2cc(C(=O)NC3CC3)cnc12.c1(C(NC)=O)c(Cl)cnn1C.C C1(C(=O)NCc2nc[nH]n2)C2CC1N(C(C1CC(F)(F)C1)=O)C2 C1(C(N(CCN(C(=O)Cc2ccnn2C)C)C)=O)OCC2CCCCC12 N1(C(=O)C=Cc2ccc(-n3ccnc3)cc2)CCN(C(c2ccoc2)=O)C2CC12 N1(C(c2ccsc2)=O)CC2(C1)CN(C(c1occc1-c1ccccc1)=O)C2 N1(C(Cn2cc(COCC(OCC)OC)nn2)=O)CCc2c(nnn2C)C1 CC1(C)C(NC(C2CC2c2ccccc2)=O)CCN1C(c1cccnc1O)=O N1(C(CSC(C)(C)C)=O)CCC2CCN(C(c3ccn(C(C)(C)C)n3)=O)C2C1 c1(C(C=O)(C)F)ccc(F)cc1.c1(COC)nocc1C(N1CC(CC)C1)=O C1(CNC(c2n(CC)ncn2)=O)CN(C(C2CCOC(C)C2)=O)CC1(C)C c1(OC=O)cccc(Cl)c1.c1(C(N(C2CC2)CC)=O)ccc(CO)cc1 c1(C(N(CCCNC(C2C(CC)CCO2)=O)C)=O)ncnc2cc[nH]c12 C1(C(C#C)NC(=O)C)CCOCC1.C1CN(C(=O)CC2CC2)C1.C(N)=O C1(NC(C(C)=C2CCC2)=O)CC(C2CCN(C(=O)CSC(C)C)CC2)C1 c1(OC)ccc(CN2CCCC2C)cc1C(=O)O.c1(C=O)c(Cl)cncc1Cl.N C(C(C(=O)N(C1CCC1)CCO)NC(C1CC1C#N)=O)OCC O=S(=O)(c1ncc[nH]1)N1CCN(C2CCCCCC2)CC1 c1(NC(=O)Nc2c(C(=O)NCCC(CC)CO)nccc2)c(Cl)c(C)nn1C C1(CNC(CSCCNC(C2CCOC2C2CC2)=O)=O)C2COCC12 Cc1ncc(Cl)c(C(N2CCCN(C(C3(C(F)F)CCCCC3)=O)CC2)=O)n1 n1(CC)nc(C(=O)NCC2CCN2C(=O)CN(C)C2CC2)c2c1CCOC2 CN1CC(=O)Nc2cc(C(=O)NCC(O)CCNC(=O)CC(C)(C)O)ccc21 N1(C(CCc2cc(C)no2)=O)CCC(O)C1C(=O)NC(c1nc[nH]n1)C1CC1 c1(OC)ccc(C(=O)NCCN2CCN(C(C3CC(C)C3)=O)CC2)cc1Br c1(NC(C)=O)ccc(C(N2CCCC2CCC(=O)Nc2cn(C)nc2C)=O)cn1 N1(C(C2(C#C)CC2)=O)CCN(C(C2CC2C2CC2)=O)CC(C)(C)C1 c1(CC)noc(CC)c1CC=O.C1(CCC)CCN(C(=O)C(O)C2CC2)CC1.N c1(C(=O)NCC(CNC(C(CC=C)C)=O)O)oc2ccccc2c1CO c1(CCC(=O)NCCOCCN(c2ncc(Br)cn2)C)nc2cccnc2[nH]1 C(=O)(CCCCCCNC(=O)C(C)n1ccnn1)NCCC(C(C)C)O C1CCCCN1C(=O)C=Cc1ccn(C)c1.C(C(O)C(=O)N(CC)C)=CC c1(CCC)cccc(C(=O)NC2(CF)CCN(C(C3CCC3(OC)O)=O)C2)c1 N1(CC(=O)NC)CCS(=O)(=O)CC1.N1(C(Cc2c(C)nsc2)=O)CC(F)CC1.C c1(C(=O)CN2CCC(O)(c3ccc(Br)cc3)C2)ccc([N+](=O)[O-])cc1 C1(O)(CCNC(c2n(C)ccn2)=O)CCCN(C(c2ccc(C(N)=O)nc2)=O)C1 c1(C(N(C2CN(C(c3nccc(OC)c3)=O)C2)C)=O)ccc(C)c(O)n1 C=Cn1nccc1C(=O)NC(C)C(C)NC(c1sccc1-c1ccc(F)cc1)=O Cc1cccc(C)c1C(=O)N(CC(C)NC(c1ncoc1CCC(F)(F)F)=O)C C(CC(C(=O)Nn1cnc2ccccc12)NC(=O)C(O)C1CCC1)N(C)C C(C)(CO)(C(=O)NCC=CC)NC(C)=O.C1(C(C)C)(C=O)CC1.N CCC(C)(O)C(=O)N1CCN(C(C23CC(c4ccccc4)(C2)C3)=O)CC1 c1(NC(CC(CNC(C(C)=CC(C)(C)C)=O)C2CCC2)=O)cccc2cnccc12 C1(CCC)CN(C(=O)C(C)(C)c2ncco2)CCN1C(=O)COC(C)CC C1(C(=O)NC(CC)CO)CCN(C(=O)C(CC2CC2)OC)CC1 c1(C(=O)NC2(CC)CC2)cc2cccc(Cl)c2[nH]1.C1(C2CC2)(C=O)CC=CC1 CC(C)CC(C)(C)C(=O)NCC(O)CNC(C1CCC=CO1)=O c1(OC)ccccc1OCC(=O)N(C)CCNC(C1CC(C)(C)CO1)=O C1(O)(CCNC(CC(C)c2ccco2)=O)CCN(C(=O)C(F)n2cccn2)CC1 c1(C(N(CCC)C)=O)ccnc(NC(N)=O)c1.N1(CC=O)C(=O)CCC1=O CC1CC(CC(N2CCOC(C)C2)=O)CN1C(c1ccsc1Cl)=O C1(N(C)C(c2cnoc2)=O)CCCCN(C(=O)COc2cccc(Br)c2)C1 C1(C)(C(=O)NC2CCCN(C(COCCC)=O)C2)CCCCCC1 c1(CC)cc(C(=O)Nc2cccnc2C(=O)Nc2nccnc2C)n(C)n1 N1(C(C(=O)NCC(F)F)=O)CCCC(NC(=O)C(F)(F)CC2CC2)C(F)C1 C1(CNC(CCn2nc(C)c(Br)c2)=O)CC2(CCN(S(C)(=O)=O)CC2)CO1 C1(C(=O)NC(C(=O)OC)C)CCCN(C(c2cc3n(n2)CCO3)=O)CC1 N1(C(C2NC(=O)C(F)C2)=O)CC(O)CC2CN(C(C3CCCCC3)=O)CCC12 C(=O)C(C)(C)CN(C(=O)CC12CCCC1C2)C.C1(COC)(C)CC1.N c1(C(=O)NCC(CC)NC(C2N(CCC)CCC2)=O)cc(O)ccc1[N+](=O)[O-] C1(C(=O)NC(C(C)O)C(=O)N(C)Cc2cccs2)CCCCNC1=O C(CC(C)CC)(C(=O)N(C1CC2(CCC2)C1)C)NC(c1cc(CC)sn1)=O c1(C(N2CC3=C(C2)CN(C(C2C=CCCC2)=O)C3)=O)cc2c(nc1O)CCOC2 CS(=O)(=O)c1ccccc1CS(=O)(=O)Nc1ccc(Cl)s1 c1(C(=O)NCCC2CCN(C(C3CC3Cl)=O)CC2)ccc(C(F)F)cc1F N1(C(C2C(C(C)(F)F)C2)=O)CC(C2CCN(C(c3cnn4c3CCC4)=O)CC2)C1 CC1CC(=O)NC(C(N2CC(CN3CCN(C(c4ccco4)=O)CC3)C2)=O)C1 c1(C(C)C)cc(C(=O)NC2CC(CO)N(C(C3CC(O)C3)=O)C2)cc(F)c1 N1(C(c2cnc(C(C)(C)C)nc2)=O)C2CCCC1CN(C(C1CCCCO1)=O)C2 C1(C(=O)NC2(CC=C)CN(C(=O)C(C)(C)CO)C2)Cc2ccccc2S1 Cc1cc(-c2nc(C3CCCO3)nn2CCCO)c(C)cn1 CCCC(O)C(=O)N1CCCCC1CCNC(c1cc(O)n(C)n1)=O C1(CCN(C(C2CC(O)(CC#C)C2)=O)C)CCCCN1C(c1sc(C)cc1C)=O c1(N(C(c2c(CC)cccn2)C(=O)NCC2CCOC2)C)ccc2c(c1)OCO2 n1(CCOC)c(=S)n(CN(C)Cc2ccc(F)cc2F)c2ccccc12 c1(C(N2C3CN(C(C(CCCC)C)=O)CC2CC3)=O)cnn2c(C)cc(C)nc12 CC(CC1CC1)C(=O)NCC1CC(C(=O)NC2CC2c2cncs2)C1 c1(NC(C(C)C)=O)ccc(N2CCN(CC3CC3c3ccc(F)cc3)CC2)nc1 c1(N2CC(CC)N(C)CC2)[nH]c(=NCc2ccc(C)cc2Br)nc2ncn(C)c12 C1(CO)CCC(c2nnnn2CC(F)F)CC1.Cn1cc(C)c(O)n1.C(C)(C)CF.N c1(C(N(C)CC2CCCC(NC(CC=C=C)=O)C2)=O)ccc2c(c1)CN(C)CC2 C1(C(N)=O)CCC(C(=O)NCCCCC2CCCN(C(=O)C3=CCOC3)C2)CC1 Cc1ccc(C(=O)NC2CCC(N(C(=O)CCc3nccn3C)C)CC2)nc1F Cc1ncc(C=CC(N2CCC(C)(CCNC(=O)CC(Cl)Cl)C2)=O)s1 C1(C(=O)OC)CC2(CCC2NCCc2ccc(Br)cn2)C1 C(CCC(O)C(=O)N(C)CC1CCCS1)NC(C1(COC)CCCO1)=O C1(C)(NC(c2c(C)cc(C)s2)=O)CCC(NC(c2ccsc2Cl)=O)CC1 c1(CC)nc(C(=O)NCc2ccc(C(=O)N)cc2)c(C)o1.C1CCCC1C.C CC(O)CCCCCC(=O)N1CCC(C)N(C(=O)C=CC2CCOCC2)CC1 c1(C(=O)NCCNC(=O)CN2CCCS2(=O)=O)cc(F)cc2nccnc12 N1(C(CN(C2CCCC2)C)=O)CC(O)CCC1C(=O)NC1(CF)CCC1 C(=O)(C(CN(C)C)C(C)C)N(C1(CC=O)CC1)C.C(CC)N(C(C)C)C.N N1(C(Cn2ncc(C#C)c2)=O)CCN(C(=O)C(O)CCc2ccccc2)C2CC12 c1(C(CC)NCc2cn(C(C)CCCO)nn2)cc(-c2ccccc2)n(C)n1 N1(C(c2ccc(OCC)cc2)=O)CC2CC1CN2C(c1ccnn1C(C)CC)=O c1(OCC)cccc2c1CCC2NC(=O)C(=O)NCC(N1CCN(C)CC1)C c1(CC(=O)N(CCCNC(c2c(CC)occ2C)=O)C)ccc(O)c(O)c1 c1(C(=O)NCc2cn(C3CCCCNC3=O)nn2)cccn2cnnc12 C1(C(F)(F)F)(NC(N2CCCCC(N(C)C)C2)=O)CCc2ccccc21 CC1(C#CC(=O)N2CCCc3[nH]nc(CO)c32)CCCO1 N1(C(C(c2n(C)ccn2)(F)F)=O)C2CCC1CN(C(C1CC13CCC3)=O)CC2 c1(N2CC(CC)N(C(=O)Cc3ccc(O)cn3)CC2)nc(C)ncc1C#N N1(CC)CCN(CC(=O)NC2CC(CNC(=O)C(C3CCOCC3)O)C2)CC1 C(C(CC(C)C)C(=O)O)NCc1ncc(NC)cn1 C1(NC(C(C(=O)OCC)OC)=O)CCN(C(C2(OC)CCCCC2)=O)CC1.C C1(CC(=O)N(CC(C)C)CC#C)C2CCCC2N1C(c1cncnc1)=O Cc1ccc(Br)cc1C(N1CCC(NC(=O)C(CO)N(C)C)C1C)=O N1(C(C2C(C)=CCC=C2)=O)CCC(C#N)(NC(c2ccc(CCO)cc2)=O)C1 c1(N2CC3(CN(C(c4coc5c4COC5)=O)C3)C2)nc2cc(Cl)ccc2s1 C1(C(=O)NC(COC)C)COCCN(C(c2oc(C)cc2C)=O)C1 c1(C(N2C3CCC2CC3)=O)ccc(S(N)(=O)=O)cc1.C1(OCC)CC1C=O CC(N=c1[nH]c(=NCc2ccc(Cl)cc2N)c2[nH]ccc2[nH]1)c1ccncc1 C=CC(CC)C(=O)NCC1C(C)C1(F)F.c1(C(=O)N)noc(C2CC2)c1C n1(CC(N2CC(CCNC(C(COC)(C)OC)=O)C2)=O)ncc(O)nc1=O CC(C(=O)NC1(CNC(c2ccc(Cl)cn2)=O)CCOC1)C1=CCCC1 c1(CC)nn(C2CC2)cc1C(=O)N(CC(C)NC(C1CCCCC1)=O)CC N1(C(CC2N(C)CCC2)=O)CC2(CCN(C(=O)COC3CCCC3)CC2)C1 N1(C(CCNC(=O)CO)=O)CC(NC(C2CN=C3N=CNN3C2)=O)CC12CCC2 C12(NC(CCCCC)=O)COCCC1CN(C(c1cnc3ccnn3c1O)=O)C2 c1(C(C(=O)NCCCSC)N(CCCCC#C)C)ccc(F)cn1 c1(CC)ccc(C(N2CCC(CF)(NC(=O)C(C)CO)C2)=O)c(O)c1 c1(C(=O)NC2CCC(NC(C(C)=C3CCC3)=O)CC2)cc2cc(F)c(Cl)cc2[nH]1 c1(OC)cccc(OC)c1CC(=O)NC1CC1.c1(CC=O)ncc(Cl)n1C.C C1(NC(COCC(=O)NC)=O)CCN(C(=O)CCc2ccco2)C1C c1(CC)ccccc1F.C1C(C=O)C1(C)C.C1(CC(=O)NC)(COC)CC1 C1(C(N2CC3CC=CCC3C2)=O)N(C(C2CCCS2)=O)CC12CCCC2 c1(C(=O)NC(C)CNC(C2CCCN2C)=O)ccc(Nc2nccn2C)cc1 c1(OC)ccc(C(=O)NC(c2cccc(C)c2)CNC(=O)C(O)C(F)F)cc1 CC(=NOCC#N)C(=O)NCCC(=O)N(C)CCc1cnccn1 N1(C(CC(=C)Br)=O)CCCN(C(c2ccc[n+]([O-])c2)=O)C(C(C)C)C1 CON(C(=O)C1CC12CCN(C(=O)CSc1cn[nH]c1)CC2)C1CCOCC1 C(=O)(C#CC1(C)CCCO1)NCC1N(C(c2cccc(SCC)c2)=O)CCCC1 C(=O)CC(C)C(F)(F)F.C(C(CO)NC(=O)COC)OC c1(CNCC(=O)NCCCC)c(C)cc(OC)cc1C.c12nc(n[nH]1)S2 C(=O)(CCCCC(C)(C)OC)NCC1C(NC(c2cc(OC)ns2)=O)C1 C1(N(C(c2c(C)c[nH]n2)=O)C)CCCC(NC(c2ncccc2C2CC2)=O)C1 C1(CC)CCC(CNC(=O)COC(C)(C)CNC(=O)CC(C)F)C1 CC1CN(C(=O)C(=O)Nc2ccc(Oc3ccc(Cl)cn3)cc2)CC1C(F)(F)F N1(C(C2N(C(C)=O)CC(O)C2)=O)CCN(C(=O)C2=CC(O)CCC2)CC(C)(C)C1 C(C1Cc2ccccc21)NC(=O)CCC1CCCCN1C(c1ccccn1)=O Cc1nc(C)c(CC(=O)NCCC(O)CNC(=O)C(n2nccc2C)C)s1 N1(C(C23OCC(C)(C2)C3)=O)CCC(CNC(=O)CCC2CC2)C(F)(F)C1 CC1(C)CC(CNC(C2CCCN2N=O)=O)N(C(=O)C(=O)N)C1.c1ccccc1 C(C)(C(O)C(=O)N(C)CCN1CCN(C(=O)CCCC2CCCC2)CC1)OC c1(SC)ccc(C(C)NC(=O)CC2CCCCC2)cc1.C12CCC(CC1)NC2=O N1(Cc2scc(CC)n2)CCc2ccc(F)c(C(=O)O)c2C1 C1(CC=C)(NC(=O)CC2CCN(C(C3CC3(C)C(F)F)=O)C2)CCCCC1 N(C1c2ccccc2CC1NC(=O)CCS(C)=O)C(C(C)CSC(F)(F)F)=O Cn1c(C(=O)NC2CCOC2C2CCN(C(=O)C(C)(C)C)CC2)cnc1O c1(C(=O)NC2CN(C(=O)CCCn3ccnc3)CC2F)ccc(Cl)nc1Cl N1(C(c2c(C)ncnc2C)=O)CCOC2(CCN(CC3CC(F)(F)C3)CC2)C1 CN1CC(=O)N(CC(=O)NCCCCC2CN(C(c3ccn4ccsc34)=O)C2)C1=O C1(C=O)CSCC(=O)N1.Cn1cc(-c2nc(C(=O)NCC=CC)co2)cn1.N Cc1cccnc1CC(=O)NC1COCCC1NC(=O)C(O)CN1CCCC1 C(=O)(C1CC(=O)Nc2ncn(C)c21)N1C(CNC(C2C(C#C)C2)=O)CCCC1 c1(OC)ccc(C(=O)NCC(=O)NC2CC(NC(N)=O)C2)nc1 N1(C(CSCC#C)=O)CC2CC2C1C(=O)NCCc1cnn(C)c1 C1(NC(c2cc(C(C)C)[nH]n2)=O)CC=C(C(=O)NCC2COCC2(C)C)C1 C(=O)(C1=CCCCCC1)N1C(CN(C(c2c(C)nns2)=O)C)CCCC1 N1(C(C2C(C(C)NC(c3ccc(F)s3)=O)C2)=O)CC(C)CCCC1C N1(C(C2CC(=C)C2)=O)CCCC(Cc2cn(C(C)C(=O)N3CCCC3)nn2)C1 C12(NC(CC(CC)(F)F)=O)CCCN(C(=O)C=Cc3cn(C)nn3)CC1C2 c1(NC(CC2(OC)CN(C(=O)CC3CCOCC3)C2)=O)ccc(Cl)cc1 Cc1nnc(SCC(=O)N(Cc2ccco2)CC2CCCCO2)o1 Cc1ccc2sc(N3CCC(NC(c4ccc(F)c(F)c4)=O)C(O)C3)nc2c1C C(C1=NOC2CCCC12)NC(CC1CCC(NC(C2(C)CC(C)(C)C2)=O)C1)=O C1(NC(Cc2c(C)cco2)=O)CCC(NC(c2cccc(C3COC3)c2)=O)CC1 c1(OCC)c(C(N2CC=CC(NC(c3cn(C)nc3C)=O)C2)=O)cccc1F N1(C(c2c(C)ccc(C)c2)=O)CCCC(C)(C)C1.C(=O)CCN(S(C)(=O)=O)C N1(C(CS(N)(=O)=O)=O)CC2CCCC(NC(=O)CCN3CCC(O)CC3)C2C1 c1(C(N2C3(CNC(C(C)=CC)=O)CCCC3CC2)=O)ccc2nnn(C)c2n1 c1(C(N(C2CCC(NC(=O)C=Cc3cn(C)cn3)C2)C)=O)cncc2nc[nH]c12 C1(NC(C2(C)CCNC2=O)=O)CCN(C(=O)Cn2nnc(=N)[nH]2)CC12CCC2 N1(Cc2c(C)cccc2Br)CCC2(CN(C(=O)CN(CCO)CCO)C2)C1 C(=O)(C(C)S(C)(=O)=O)N1C(CNC(c2cccc(C)n2)=O)CC(OC)C1 C1(OCC)CC(NC(=O)CS(=O)(=O)C(C)(C)C)C12CCOCC2 C1(CNC(c2ccccc2NC(C)=O)c2n(CC)nnn2)CCC=CCCC1 c1(C(N(C2CN(C(C(C)C(F)(F)F)=O)C2)C)=O)nccc2c1[nH]c1ccccc21 C(=O)(CCCC(F)(F)F)N1CC(F)(CNC(C2CC3C=CC2C3)=O)C1 N1(C(C(C=C)(C)CC)=O)CCN(C(=O)CCN(C)CCC)CC(CO)C1 C1(C(=O)NC(C(=O)N(CC(CC=C)(F)F)C)(C)CSC)CCC2(CCC2)O1 N1(C(CCOC)=O)CCCC(C)(C)C1CNC(c1cc(CO)ccc1Cl)=O C1(CC=C)(NC(c2ccc(CC)o2)=O)CC2CCC(C1)N2c1ncnc(Cl)c1Br C1(NC(C2(c3ccccc3)CC(C)C2)=O)COCCN(C(C2CCCS2)=O)C1 C1COC(C)(C)CN1C(c1cccc([N+](=O)[O-])c1)=O.Cc1cc(C(=O)NC)no1 c1(C(C(C)NC(=O)NCC2CCC2)O)ccc(F)c(F)c1.c1nnn(C)n1.N N1(C(CC)=O)CCC(C2CCCN(C(C3CC4(C3)CC4F)=O)C2)CC1 CC1C(NC(C23CC(F)(C2)C3)=O)CCCN1C(=O)COC1CCCC1 N1(C(C(N2C(CC)CCC2)=O)=O)CCC2(NC(c3coc(SC)c3)=O)CCCC12 C1(CC(=O)NC2C(C)CN(C(=O)Cc3cn(C)nc3Cl)C2)CC(O)C12CCC2 C1(CC)CN(C(=O)C(c2ccco2)NC(=O)CCc2ccn(C)n2)CCO1 N1(CCCOc2ccc(OC)cc2)CC2CCC2(N2CCN(C)CC2)C1 N1(C(CCCc2onc(C)n2)=O)CC2CC(C1)CN(C(C1(C)CC3CC3C1)=O)C2 c1(C(=O)NC(CCN(C(C2ON=C(C)C2)=O)C)C)ccccc1.O(C(F)(F)F)C c1(-c2ccc(C)c(F)c2C)ccnc2ccc(C(N3CCCC(O)C3C)=O)cc12 N1(C(C(N)=O)=O)CCC2(CC1)CC2CNC(=O)CO.c1nc(O)nc(O)n1 CN1CCCC1C=CC(=O)NC1(CO)CN(C(C2OCCC2C(F)(F)F)=O)C1 C1(CNC(CN(c2ccccc2)C)=O)CCN(C(c2ccn(C)n2)=O)CC1 CCCCC(C)C(C(=O)NCCOCc1ccccc1)N(C1CCOC1(C)C)C c1(C(c2nnnn2C2COC2)NCC(CC)CC(C)C)c(Cl)ccc(Br)c1F c1(C(N2C3CN(C(C4C(OC)C4)=O)C(CC3)C2)=O)ccnc2ccccc12 CCC(O)CN(C(=O)C=CCN(C(=O)CN1CC=CC1)C)CC C(=O)(C1CCCc2nc(C)[nH]c21)N1CC(C2CN(C(c3c(C)con3)=O)C2)C1 c1(C(N(C)CC2CCCN(C(C(COC)C)=O)C2)=O)c(O)ccc(Cl)c1F N1(C(C(C)c2cccs2)=O)CCc2c(C(N3CCC(F)(C(=O)O)C3)=O)cccc2C1 CC1=C(C(=O)NCC2(O)CCCN(C(C3CC3c3ccco3)=O)C2)CCO1 C1(O)CCN(C(=O)C(F)OC(F)(F)F)CC1.Cc1cc(C(C)(C)C(=O)N)cs1.C Cc1nc(C(=O)NCCC(O)CNC(c2cc(Cl)ns2)=O)nn1-c1ccccc1 c1(C(=O)NCC2N(C(C=CCC)=O)CC(O)C2)ccc(CO)cc1F Cc1ccc2c(c1)C(C)(NC(=O)Nc1ccc(Cl)cc1F)CC2 N1(C(C2CCCN(C(=O)CN3C(=O)CCC3=O)C2)=O)CCc2ncccc21 C(=O)(C(CC)C(F)(F)F)NC(CN(C(c1c(C)nc(CC)s1)=O)CC)C C1(C)(CNC(c2c(CC)cccn2)=O)CCN(C(=O)CC2CCCC2)CC1 N1(C(c2c(C)ccn2C)=O)CCC2CN(C(c3csc(S)n3)=O)CC2C1 c1(CN(CC(O)C)C)cc(C(F)(F)F)cc(O)n1.c1(CCC=O)ccccn1.N C(=O)(C(C)(CSC)NC(C1CCC(=O)O1)=O)NCCNC(=O)OC C(C)(C(C(=O)NC1CCCCC1)N(C)C)OC.c1(C=O)cnn(CC(F)F)n1.N c1(CC(N2CC3C(NC(=O)Cc4ccno4)(C3)C2)=O)cccc2ccoc12 C1CC(O)CN(C(c2ccc(=O)n(C(C)C)c2)=O)C1.C1(CCC)(C(=O)N)CC1 S(=O)(=O)(CCC(=O)NCC(C)(C)CC)NC.C(=O)(C(C)Cc1ccccc1)N C1(C(=O)NC(COC)(C)C(N)=O)CN(C(=O)Cn2cncn2)CC1C1CC1 c1(C(N(C2CN(C(C(C)OC)=O)C2)C)=O)cc([N+](=O)[O-])c(F)cc1N C1(O)(c2cn(CC)nn2)CC2CCC1C2.C(=O)(CC(C)C)NCCSCC.O n1(CCC=O)ccc2ccccc12.C1(OCC(=O)NC2CC2C)CC=CC1.N C1(C(=O)NCC2CC(NC(=O)COc3ccccn3)C2)CCc2ccccc2O1 c1(OC)cncc(C(=O)NCC(C2CC2)NC(C2(C#N)CCCO2)=O)c1 Cc1c[nH]c(C(=O)NCCOCCNC(C2(F)CCOC2C)=O)cc1=O C(=O)(C(C)C(C)C(C)(C)C)N.C12(NC(CSCCOC)=O)CC(C1)C2 N1(C(CN2C(=O)CCC2)=O)CC(NC(=O)CSC2CC2)CC12CCCCC2 C(C1=CCN(C(C2CC3CCC2C3)=O)CC1)NC(CC(C)c1ccco1)=O Cc1nn(C)c2c(NC(C)Cn3ccnc3)nc(N3CCN(C)CC(C)C3)nc12 N1(C(=O)C(O)CC(F)F)CCCC2C1CCN2C(c1nocc1Cl)=O N1(C(C2(CC#C)CC2)=O)CC(CNC(=O)CCC(C)N(C)C)C2(CC2)C1 CCCS(=O)(=O)CC(=O)NC1CN(C(=O)Cc2cn(C)nc2Cl)CCC1C c1(C(N2CC(O)(CN(C(C(CC=CC)C)=O)C)C2)=O)cnc2n1CCS2 N1(c2ccc(C(=O)OC)cn2)CC2(CN(C(C3(C)CC(F)C3)=O)CC2CO)C1 c1(CCCCNC(C2CCCN2C(c2cccs2)=O)=O)cn(C2CCCC2)nn1 c1(C(=O)NCC=CCNC(CC(C(C)C)C)=O)c(N)ccc(Br)c1F c1(C(N2CC(NC(c3n[nH]c(C)c3C)=O)CC2(C)C)=O)cnn2c1CCCC2C C1(N(C(=O)CC(Cl)Cl)CC)CCC(NC(=O)CN2CCCOC2=O)CC1 c1(CC(N2CC(N(C)C(C3CC3[N+](=O)[O-])=O)C2)=O)ccnnc1O c1(C(=O)NCc2n[nH]c(N)c2C#N)ccc(C(F)(F)F)c(F)c1.c1ccncn1 N1(C(c2c(OC)nsc2)=O)CCCC(C)(C)C1.C1(C)(C=O)CC(=O)N(C)C1.C N1(C(C=CCN(C)CC)=O)CCCC1CC.c1(CC=O)csc(CC)n1.N C#Cc1cnc(C(=O)N(CCC)C)c(C)c1.c1(C(=O)N)c(C)[nH]c(C(C)=O)c1C N1(C(C(C2CN(C(C3CCCCC3O)=O)C2)OC)=O)CC2(CCOC2=O)C1 N1(C(c2c(C)[nH]cc2)=O)CCC2(CC1)CN(C(C1C=CCC1)=O)CC(C)O2 C(=O)(C(C)(O)C(F)(F)F)N1CC2C(C(N3CCCN(C(C)=O)CC3)=O)C2C1 N1(C(=O)CN2CSCCSC2)CCC(C2CCOC2)C1 C1(C(=O)NCCNC(C=Cc2cncc(C)c2)=O)CCc2nnc(C)n2C1 C(=O)(C(F)(CNCC)C(C)C)N1CCC(CC(N(OCC)CC)=O)(C)C1 C1(O)(CC)CCN(C(c2c[nH]nc2C)=O)CC1.C1(C(=O)N)CC1C=O.C#CC CC1(C)CCCN(C(=O)C=CCN2CCCC2)C1C(=O)N.CC(O)C(C)(C)O C(=O)(C(O)C1=CCCCC1)N1CCC(C#C)(C(=O)NC2(CC(=O)OC)CC2)CC1 Nc1cc(C(=O)NCC2CCN2C(c2ccc(F)s2)=O)cc(O)c1 CCCCCCCN(C(=O)C(C1CCN(C(c2cnc(Cl)n2C)=O)C1)C)C Cc1nc2c(o1)CCCC2CC(=O)NCC(C)CN(C(=O)C(C)(C)O)C c1(OC)cccc(-c2cnc(C(=O)NCC34CC(CC3C(=O)O)C4)o2)c1 O(N1CCC(CC(=O)NCCCCNC(=O)COC(C)CC)CC1)CC N1(C(c2cnc(CCC)s2)C(=O)NCCCOC)CCC(C)(F)CC1 c1(C(N(CC2N(C(CC3(C=C)CCC3)=O)CCCC2)CC)=O)cc(O)ccc1F c1(C(N2CC(NC(C(C(C)C)NC=O)=O)C2)=O)cccc2c1CCO2 c1(N(C2CCN(C(Cc3cn(CC)nc3C)=O)C2)C)cc(C)nc2nc(C)nn12 C(=O)(C(C(C)(C)C)NC(c1occc1CC)=O)NC(C1CCOCC1)C#C C(CCC1CC1)(C(=O)NC1(CCCF)CC1)NC(C1C(C(C)C)C1)=O C#CCCC(C(=O)Nc1csnc1C)NC(=O)C1=NOC(C)C1 C1(NC(c2cc(Cl)on2)=O)CCN(c2ncc(Br)c(O)n2)C12CCC2 C(=O)(C1=C(C)OCCS1)N1CCC(C(C)NC(C(CC)CC)=O)C1 CN1CCN(C(c2ccc(OC(F)F)nc2)=O)C(CN(C)C)C1 c1(C(=O)NC2C(C)CN(C(c3ccoc3Br)=O)CC2)cc(O)cc([N+](=O)[O-])c1 Cc1nc(C)n(CCC(=O)NCCOCCNC(C2CCSC(C)C2)=O)n1 c12ccc-1cc2.CC1(C(=O)NC2CCN(C(c3coc(CO)c3)=O)C2)CCCO1 C(=O)(CC(O)CNC(=O)Cn1cc(Cl)cn1)NCCSCC=C C#CCCCCCC(=O)N1CCCC1C(C)(C)C(N1CC(OC)C1(C)C)=O C12(NC(CCC=C)=O)CCCC1CN(C(=O)CN1CCCC1)C2 c1(NC(c2c(CC)cccc2)=O)ccc2nc(C3(C(F)(F)F)CC3)[nH]c2c1 CCCCC(C(=O)NCC(C)(C)NC(C1CC1C=O)=O)C(C)C.C(C)(C)C Cc1nccnc1C(N1CCC(NC(=O)C(N2CCCCC2=O)C)C1C1CC1)=O c1(C(N2CC=CC(NC(C3CC4CCC3C4)=O)C2)=O)ccc2cc[nH]c2c1 N1(Cc2c(C)cc(-c3ncco3)cc2)CCC(C)(C)CC(C)(C)C1 C(CCCCNC(=O)Cn1cc(C2CCN(CC)C2)nn1)N(c1ccccc1)C c1(C(=O)NC2OCCN(C(=O)NCc3ccc(OC)cc3)C2)ccc(Br)nc1F C1(NC(C=C2CCC(C)C2)=O)CCC12CCN(C(=O)C(C)(C)n1cccn1)CC2 c1(C(C)C)ccc(O)cc1C(=O)NC1CN(C(C2CS(=O)(=O)CCO2)=O)C1 C1(NC(CCC=C(C)C)=O)CC2CCCC(C1)N2C(c1cccc2[nH]ncc12)=O C1(CCC)CN(C(c2cc(C(=O)OC)co2)=O)CCN1C(=O)C(C)SC(C)C c1(CNC(=O)Nc2c(C)ccnc2)ccc2oc(O)nc2c1 C(=O)(C(C)(C)C)NC(C)C(=O)NC1CN(C(=O)CC2(C)CC2)C1 C1(CC)CCCN1C(=O)C(O)CNC(=O)C(C1CCCCC1)F N1(C(Cc2c(OC)ccc(C(F)(F)F)c2)=O)CCCC2(CCCC2O)C1 N1(C(C(C(C)C)NC(c2cncc(CO)c2)=O)=O)CC2CCC(C1)N2C NS(=O)(=O)N1CCC(CNCc2csc(C(F)(F)F)n2)CC1 c1(CN(C(=O)CC2CC(OCC)C2(C)C)CCC)ncc(Br)cc1C#N Fc1ccc2sc(NCCN3C(=O)CCC3=O)nc2c1 CCCC(CCCNC(C1CC1c1ccc(F)nc1)=O)NC(C1CC=CC1)=O CCCCC(C)C(C)(c1nnnn1C1COC1)NC1CCCC1C#N c1(C(=O)NCC(CC=C)NC(=O)CCCCC)cnc(C(C)C)nc1C c1(C(=O)NCC(C)(C2CC2)NC(CCN(C)CC)=O)c(C)nc(C)n1O Nc1c(C(=O)NC(CNC(C23CC4CC2C3C4)=O)C2CC2)nc(O)nc1O N1(C(C)=O)CCC(NC(=O)Cc2ccc(C)nc2Cl)C(C)C1 C1(c2nnc(C)o2)CCCN(C(c2nnc(C)s2)C(=O)NC2(C)CC2)C1 Cc1ccc2oc(=NCC3CCCN(C(=O)COc4cccnc4)C3)[nH]c2c1 C1(CCNC(C2C(C)(C)CO2)=O)CSCCN1C(=O)COCCCF C1(CCC)CN(C(=O)Cc2cc(Cl)ccc2O)CCN1C(=O)COCC(C)C N1(CC(C2COCCO2)(C)O)C(=O)NC(C2CC(F)(F)C2)C1=O N1(C(C(=O)NC)C)CCC(N(C)C(C23CC(C)C2C3)=O)CC1 N1(C(Cc2n(C)ncc2)=O)CCC2CC(NC(C3(C)CCNC3=O)=O)CCC2C1 c1(C(N2CCC2CNC(C2(Cl)CC2(F)F)=O)=O)coc(C2CCC2)n1 C1(COC)CN(C(C2(n3nccn3)CC2)=O)CCN1C(C1(C)COCCO1)=O C1(CC=O)(C(F)(F)F)CCC(=O)NC1.C(=O)C(C)(C)C(F)F.C=CCCC.N C1(C(=O)N)CNC(=O)CC12CCC2.n1(CC(=O)NCC2CC2C)cnnc1 N1(C(COC(C)C)=O)CCCCC1C(C)(C)CNC(c1cnn(CCO)c1N)=O Cc1ccc2oc(C(=O)NCC(C3CC3)N(C(=O)Cc3cn[nH]c3)C)cc2c1 c1(NC(C2C3CC2N(C(c2c(F)cccc2Br)=O)C3)=O)cnc(Br)c(Cl)n1 Cc1sc(Cl)nc1C(=O)NC1CC2(C1)CC2NC(=O)CCCc1nncn1C C1(C(=O)Nc2c(C)csc2)CCC(C)N(C(=O)CC2CCCN(C)C2)C1 C1(C(N2C(C)(C)CCC2)=O)CC12CCc1ccccc12.C(C=C(Cl)Cl)=CC(=O)N C1(C(N2C(CC)CN(C(=O)C(CO)N(C)C)CC2)=O)CCC2CC1C2(C)C c1(C(N2CC(CNC(CCOC(C)C)=O)C(O)C2)=O)cnc2ccnn2c1N Cc1cc(C(=O)NC2CCN(C(C3CC3C(F)F)=O)C2(C)C)nc2ccccc12 c1(NC(C2C3CN(C(C=Cc4cnc(C)s4)=O)CC32)=O)cc(F)c(C)cn1 N1(C(C(CC(C)C)C)=O)CCC2(CCCCN(C(C3CCC(C)(C)C3)=O)C2)C1 c1(C(=O)NCC(CN(C(CC=CC=C)=O)C)C)nn(C)cc1Br c1(C(=O)NCC2(F)CCCN(C(C(C)(C)C)=O)C2)ncnc2c1CCCC2 Cc1c(C(=O)NCC2CCCN2C(=O)Cc2cnnn2C)cnn1C1CC1 C(=O)(CC(C(F)(F)F)n1cccn1)N1CCN(CCNC(C(COC)C)=O)CC1 Cc1ccc(C(=O)NC2CCCC(N(C(=O)Cc3nc(C)sc3C)C)C2)c(C)c1 c1(C(N2C(C(NOC)=O)CCC2=O)=O)cc(Cl)c(Br)c(Cl)c1[N+](=O)[O-] N1(c2cc(NC(c3ncc(C)s3)C)ncn2)CCSC2(CCOCC2)C1 c1(C(=O)OC)cc(C)cc(CO)c1NC(N1CC2COCC2C1)=O c1(CC(C)C(N2CCC(C(N3CCC3(C)C(=O)O)=O)CC2)=O)ccc(O)cc1 c1(CN(C(=O)NCCC(C)F)CCOC)ccc(Br)cc1 N1(Cc2cn(-c3nccc(CC)n3)nn2)CC(C)C(N)C(C)C1.c1(C)ccccc1 N1(C(CC2CC(=O)C2)=O)CC2(CCCCN(C(C3CCCCN3C(=O)O)=O)C2)C1 CC1CC(NC(=O)Cn2ncc(O)nc2=O)CCN1C(=O)CC(=O)NC1CC1 C(C)(CO)(CC(F)(F)F)NC(CCCn1cc(CCN(CC)CC)nn1)=O C(=O)(C1=Cc2ccccc2C1O)N1CC(O)CC(NC(=O)Cc2ccc(Cl)s2)C1 Cc1cc(N2CCOCC2)ccc1NC(=O)NCC1COCC(C)O1 C1(NC(C=CC(CC)C)=O)CC2(C1)CC2C(N1CCC(O)(C(C)C)C1)=O C(C)(CO)(C(=O)N1OC2CCC1CC2)NC(C1C(C)CCOC1)=O Cc1cc(C(N2CCN(C(=O)C3=NNC(=O)C3)CC2C(C)C)=O)cc(O)n1 c1(C(=O)NCCCCN(C(C2C(OCC)C2)=O)C)cnc(-c2ccccc2)o1 C1(CNC(C(C2CCCC2)OC)=O)CCCN1C(=O)C(F)(F)c1ccccc1 C1(C)(C(N(C2CC(C(=O)NC3CC3)C2)C)=O)CC(F)C1.c1cnnn1C.C N1(C(C2(C)CCOCC2)=O)CCC2C1CCN2C(c1cc(F)ccc1O)=O C1(CCCC)CN(C(=O)C(C)(C)OCC)CCN1C(=O)C(c1ccc(Cl)s1)C C1(NC(c2cc(C)ncn2)=O)CCC2(CCN(C(c3nocc3Cl)=O)CC2)C1 C(=O)(C(CCF)NC(C1CC2CCC2C1)=O)N1CCC(CSC)C1 c1(C(N2CCC(C)(NC(c3c(C)ccnc3)=O)C2)=O)ccc2cccnc2c1O Cc1ccnc(C(=O)NC2CCC2NC(C2CCCN2c2ccccc2)=O)c1 c1(CNCC2C(O)CCC2)ccc2occc2c1 N1(C(=O)CC2CCC2)CCN(C(C2CC=CCO2)=O)CC(O)C1 C1(C(=O)NC(COC)COC)CC(C)CN1C(c1cnccc1C)=O CC(CCNC(=O)CC1CCC1)NC(=O)CC1CSC1 CC1(NC(C2CSCN2S(=O)(=O)CC2CCOC2)=O)CC(F)(F)C1 C1(NC(c2ccc(OC)nc2C)=O)CC2CCC1CN2C(=O)COCC(C)C S(=O)(=O)(CC(=O)N(C1CC(NC(=O)CC23CC(C2)C3)C1)C)NCC c1(C(N2CCOC(c3nc(C(F)(F)F)cs3)C2)=O)c(F)cc(C(F)(F)F)cc1F C1(C(N(CC(C(C)C)OC)C)=O)N(C(c2ccsc2C)=O)CC12CCCC2 C1(CN(C(CCC=C(C)C)=O)C)CCCCN1C(C1CC1(C)Br)=O C1(C)(CC(=O)NCCCOCCNC(C(C)SC)=O)CC1(F)F C(C(N=c1[nH]c(=NCC(C)(C)C(C)(F)F)[nH]c2c1CCC2)c1ccnn1C)OC C(=O)(C1=NOC2COCC12)N1CC2(CNC(C(CC#C)O)=O)CC1(CO)C2 Cc1cnc(C(=O)NC2CCN(C(c3ccc(F)cc3Cl)=O)C2)cc1C C(CC(C)C)(C(=O)NCCOCC1CCC1)NC(C(C)OC)=O Cc1cccc2c(=O)n(CCC(N3CCC(NC(C4(F)CCC4)=O)C3)=O)cnc12 c1(C(=O)OC)cc(C#N)ncc1NC(c1cc(C)cc(C)c1)CN(C)C N1(C(CC2N(C(C(CCCCC)F)=O)CCCC2)=O)CCC2(COC(=O)N2)C1 C1(O)(C(=O)NCC(=O)N)CCCCCC1.C12(CC1)C(=O)NC2.C1CC1 c1(C(=O)NC(C(N2CC(N(C(C)C)C)C2)=O)C)ccnc(CO)c1 Cc1c(C(=O)NCC2(C)CN(C(c3ncc(F)cc3F)=O)C2)cccc1O c1(C(=O)NCCC(CNC(c2ccc(OC)s2)=O)OC)c(C)nc(C)n1O Cc1c(Br)sc(C(=O)NC23CC2CN(C(=O)C(O)CC2CC2)C3)c1C C(CCC)(C(O)C(=O)N1CCOC(C#N)C1)NC(C(C(=C)C)(C)C)=O Cc1nc2ccccc2n1CCC(=O)NC(C)CNC(C1CCC(C)C1)=O c1(OC)cc(C(=O)NCC(C)NC(C23CCC(O)C2CC3)=O)ccc1F Cn1nnc(=NC(CNC(C2(C)CC2Br)=O)c2ccc(N(C)C)cc2)[nH]1 C1(O)(CC(N2C(CN(C(C(C)SCC)=O)C)CCC2)=O)CCCCC1 O=C(CS(=O)CCC(F)(F)F)NCCNC(=O)C(F)(F)CCc1ccccc1 c1(C(=O)NC2C(OC)CN(C(C3CC(CF)C3)=O)C2)cc2c(O)cccc2n1C C1(CNC(NCC(=C)Cl)=NCCc2ccccn2)CCCC2(CCC2)O1 c1(OC)c(Cl)cccc1NNC(=O)C(=O)c1cccc[n+]1[O-] C(=O)(N=c1nc(C2CC2)[nH]s1)NCCC1C(c2ccc(OC)cc2)C1 C1(C(N(CCC)C)=O)CCCCS1(=O)=O.C1(O)(C(=O)N)CCN(C(N)=O)CC1 c1(CNC(C(COC(C)C)NC(=O)C2=CC(C)C2)=O)cc2ccccc2[nH]1 c1(N(C2CCNC2)C(c2ccc(F)c(I)c2)=O)ncc2cccc(O)c2n1 C1(NC(c2nnsc2C(F)F)=O)CCCN(C(=O)CSc2ccccn2)C1 c1(C(N(CC(=O)N(C2CC2C)C)CC)=O)ncc2ccccn12 C(=O)(C(C)C(O)CC)N1CCC(NC(C(C)SCC)=O)C1 C1(O)(CNC(C2N(C)CC(O)C2)=O)CCCN(C(=O)C=Cc2cccn2C)CC1 N1(C(c2cc(C)c(O)nc2)=O)CC2CC3CC2C1C3NC(=O)C(C)CC1CCC1 Cc1cnc(NC2CN(C(C3CCCN3C(c3nnn(C)n3)=O)=O)CC2C)nc1 N1(C(C2N(C(CNC(C)=O)=O)CCC2C2CC2)=O)CC2CCC(C1)C(=O)N2 n1(CC)cnc(C(=O)N(C2CCN(C(c3conc3C(C)(C)C)=O)C2)C)n1 C(CCCCC(=O)N1CCOC(C(=O)N(CC(C)C(=O)NC)C)C1)OCC Cc1ccc(F)c(C(N2CCC2(C)CC(=O)NCCCC2CCCCO2)=O)n1 C1(C(=O)NCCC(C=C)C)N(C(=O)CC2(O)CCCC2)CC12CCCC2 CC1=C(C(=O)N2CC(N(C(=O)Cc3cnns3)C)C2)Cc2ccccc2O1 C1(CC)(NC(C2CC2F)=O)CCCN(C(=O)CCCc2ccccc2Cl)C1 N1(C(CC(C)F)=O)CC2CCN(C(=O)CCC3CCCO3)CC(C2)C1 N1(C(c2c(C)nsc2)=O)CCN(C(=O)CC2CN3CCC2CC3)CC1CF N1(C(CN(CC)CC)=O)CC(C2C(=O)N2)C1.c1(NC)cn[nH]c1.OC C1(CNC(Cc2c(C)ccnc2)=O)CCN(C(C2CC(O)CN2)=O)CC1(F)F C12CCCC(CN1C(c1cn(C)nc1Cl)=O)C2.CC1=NNC(=O)C1CC(=O)N.C C1(C(=O)NCc2cn(CC(N3CC(=C)C3)=O)nn2)CC(O)CN1C Cc1nn(C)c(F)c1C(=O)NC1COCC1NC(c1ccccn1)=O c1(C(=O)NCC2CN(Cc3occc3Br)CCO2)cc(I)c(O)c(I)c1 c1(CC)occc1C(=O)NCC(C)(C1CCC1)NC(=O)C=Cc1cscn1 C(=O)(C(C)CCCOC)NC(CNC(c1sc(CC)c(C)c1)=O)CCOC C1(C(N(CCC)C)=O)CC=CCC1C(F)(F)F.C(c1ccccn1)=CC(=O)N C1(CNC(c2cn(CC=C)nn2)=O)CCCN(C(=O)CN2CCCOC2=O)CC1 C1(CC)CC(C)(C)CN1CC(O)COC(c1cccs1)C CC1C(NC(=O)C(c2cccc(Cl)c2)O)CCN1C(=O)C=C1CCC1 N1(C(c2cnc(C)nc2C)=O)CC2CS(=O)(=O)CC2(NC(C2CN(C)C2)=O)C1 N1(C(CC(C)SC)=O)CCC2(CCN(C(c3cccc(C)c3[N+](=O)[O-])=O)C2)C1 CC1CC(C(F)(F)F)CN1C(c1nccn1-c1ccccc1)=O C1(CNC(c2c(C)csc2)=O)CN(C(=O)C(F)(F)CC2CCCO2)CCN1C CC1(C)CC=C(C(=O)NC2C3CCN(C(=O)Cn4cnc5c4CCCC5)C23)CC1 c1(C(N2CCC(N(C(CCC(=O)NC)=O)CCO)CC2)=O)nn(C)c(C)c1Br c1(C(=O)NC(C(C)NC(=O)CCCF)C)ccc(Sc2ccc(F)cc2)c(Cl)c1 N1(C(CCN(CCC)C)=O)CCCCC1C(C)(C)CNC(c1ocnc1CC)=O C1(CNC(c2cnns2)=O)CCC(NC(C2CC(=C3CCC3)C2)=O)CC1 CC1CC(C(N2CCCC2C2(NC(=O)C=CC(F)(F)F)CC2)=O)CCN1C C1(NC(C(F)=CC)=O)CC(C)N(C(c2nncs2)=O)C1 Cc1cc(=O)oc(C)c1C(N1CC2(NC(=O)C#CC3CCOC3)CCC1CC2)=O c1(C(N2C(CC)CN(C(=O)C3CC3)CC2)=O)cc(C(F)(F)F)cc(Cl)c1F.CO c1(NC(C2(COC)CN(C(C3(C)CC=CCC3)=O)C2)=O)nc(C)c(C)s1 C1(NC(CNS(CC)(=O)=O)=O)CCC2CN(C(=O)CN3C(C)CCC3C)CC2C1 N1(C(C2C3CCC2(c2ccco2)C3)=O)CC2(CCC(COC3CCOC3)O2)C1 C1(N2CCN(C(=O)NCC(CC)(CC)CC)CC2)CC(C)(C)OC1(C)C N1(C(c2c(C)nn[nH]2)=O)CCC2CN(C(C3(C)CC(C(F)(F)F)C3)=O)CC12 N1(C(c2c(C)nc(C)o2)=O)CCCC(C2CCN(C(c3ccccc3F)C)C2)C1 CC1=NOC(C(=O)NCCCNC(c2ccnn2-c2cccnc2)=O)C1 CCC(CC)(C(=O)NCC1(OC)CN(C(=O)C(n2cc(C)cn2)C)C1)OC C(=O)(C(C)(C)CC(=O)N)OC.N1(C(C(C2CCC2)F)=O)CCCC1CCC(C)C CCCC(C(=O)OC)C(=O)NC1(C(N2CCC23CCCC3)=O)CCC1 c1(C(=O)NCC2(O)CCN(C(C(CC=CC)C)=O)C2)c(Cl)nn(C)c1Cl C12(CNC(C3CCN(C(=O)C(F)OC(F)(F)F)C3)=O)CCC(CC1)OC2.C Cc1csnc1C(N1CC(CO)(NC(C2CC(F)(F)C2)=O)C1)=O C1(NC(c2ccc(CSCC)cc2)=O)CCC2CCN(C(=O)C3=CCSC3)C12 C(C1=NOC2CN(C(=O)Cc3cnns3)CC12)NC(c1nc(COC)sc1)=O CCCC(C(=O)NC1CC(F)(C)C1)N(C)C.C(CCC=C(C)C)=CC=O C1(C(=O)Nc2ccc(N)c(Cl)n2)CCCC12CN(C(=O)Nc1cncc(Br)c1)C2 C(C)(CCC(=O)NC1(C2CCCN2C(c2cccnn2)=O)CC1)SC C1(C(N(C2CN(C(=O)CCOC3CCCOC3)C2)C)=O)CC2(CCC2)CO1 C=CC(CC)C(=O)NC(C(=O)NC(C)Cn1cc(C)cn1)C1(O)CCC1 c1(CNC(C(C)(C)NS(C)(=O)=O)=O)ccccc1C.C(=O)C=C(Cl)Cl C1(NC(C(C)Cn2cncn2)=O)CC2(CCN(C(C3CCCC3)=O)CC2)C1 C(=O)(C1CCc2nccn21)NC(C(=O)NCCc1n(CC)cnn1)CC(F)F Cc1cc([N+](=O)[O-])ccc1C(=O)NC1(CNC(=O)C2=CCCOC2)CCC1 c1(OC)cc(O)c(C(=O)NC2CC3CC2N(C(=O)C2=C(C)CCC2)C3)c(F)c1 C(C(C)(C)C(=O)NCCCCC1CC1)N(C(CC1CCC(C)C1)=O)C C1(C(=O)NCCCCNC(C(CCC)O)=O)CCC(=O)N(C)C1 N1(C(C(C(C)C)C)=O)CCC2(CCOCC2)C(NC(=O)CN(C)C(C)C)C1 C12(c3cn(C(C(=O)N(C4CCCCC4)C)C)nn3)CC3CC(CC(C3)C1)C2 C12(CNC(C(C)OCC(C)C)=O)CN(C(=O)CC)CC1CCO2.C1CC1.O c1(C(N2CCCCC(NC(c3ccn(C)c(=O)c3)=O)C2)=O)nccn2nccc12 C1(N(C(=O)CC2(CC(=O)OC)CCCC2)CC)CCN(CC(F)(F)F)C1 C(=O)(C#CC1(C)CC1)NC(CCNC(CCCCN(C)C)=O)Cc1ccccc1 CCCCCCCCN(C)C(C1C2CC2CN1C(C1CCCC(=O)N1)=O)=O C=CC(O)(C(=O)NC1CC(CCNC(c2ncn(CC)n2)=O)C1)C(F)(F)F C1(C(=O)NCCc2ccc(C)s2)CN(C(c2nocc2C)=O)CC12CC2 c1(OC)ncc(C(=O)NCC23CC(CN2C(=O)C(C)c2ccsc2)C3)cc1Cl c1(-c2ccn(C)n2)ccc(F)cc1Cl.c1(CC(=O)OCC)ccc(CN)s1.C CC(C)(CO)CCCc1nc(-c2ccc(N)cn2)nn1CCc1ccncc1 C1(NC(C2(N(C(C(C)NC(N)=O)=O)C)CC2)=O)CCc2n[nH]cc2C1 Cc1nccc(Cl)c1C(=O)NCCc1cccc(Cl)c1.C(=O)(CCN1CCC1)N C[S+](C)CCC(O)C(=O)NCC1(O)CN(C(C2CC2c2ccccn2)=O)C1 Cc1cc(F)ccc1CC(=O)NC1CC(C)N(C(c2cc(C3(C)CC3)n[nH]2)=O)C1 C1(CNC(c2c(C(N)=O)cccc2)=O)CCCN(C(c2ncc(F)cn2)=O)CC1 c1(C(c2nnnn2CCSC)NCCC)nn(CC)nc1Br C1(CNC(c2cnn(C3CC3)c2)=O)CCCCN(C(C2CC2F)=O)CC1 C(CNC(=O)Cn1ncnn1)(CCNC(c1sccc1F)=O)OC C1(CNC(C(CC)n2cccn2)=O)CC2(CO1)CN(C(=O)CN(C)CC)C2.O N1(C(c2cncc(C)c2)=O)CCOC2CCN(C(c3ccsn3)=O)CC12 CCCCC(CC)C(=O)N(C(C)CNC(=O)Cn1cnc([N+](=O)[O-])c1)CC c1(C(N2C(C)CC(NC(=O)CCCn3cccn3)CC2)=O)csc2c1CCCC2 Cc1ccc(C)c(CC(=O)NCC(C2CC2)NC(c2cc(F)cnc2O)=O)c1 C1(CC(=O)N)CC(=O)NC(=O)C1.N1(C(C(c2cn(C)nc2)=O)=O)CCC2CC12 Cc1nc2ccc(C(=O)NCC3CCC3NC(=O)CC(F)(F)C(C)C)cn2n1 c1(OC)cc2c(cc1OC)N(Cc1ccccc1C=O)CC2 N1(C(COCCC)=O)CC2C(C(N3CCC(CC)C3C)=O)C2C1 N1(C(C2C(C)N(C(C3CC(F)C(=O)N3)=O)CC2)=O)CC2COCC2(C)C1 Cc1cc(C(=O)NCCC(O)CNC(c2cnccc2C)=O)c(Cl)cc1N CC(CCCNC(=O)CC1(CS(C)(=O)=O)CC1)NC(C1C2COCC12)=O S(=O)(=O)(c1ccc(N2CCC(CF)C2)c(Br)c1)NCC(CC)(C)CO C1(N(C(c2c(CC)nc[nH]2)=O)C)CN(C(=O)C(C)=CC2CC2)CC1F CC1(C(N2CC(NC(c3ccn(C4CCC4)n3)=O)C(O)C2)=O)CCC(O)CC1 C(=O)(C(C)(F)F)N(CC(O)CNC(=O)Cn1cnnc1)C [SH](=O)(=O)c1c(C)cccc1Cl.n1(CC(=O)OC)nc(C(F)F)cc1C.C=O C1(C(=O)NC2(CO)CN(C(Cc3scc(C(=O)OC)c3)=O)C2)CCN(C)CC1 Cc1ccc(CC(=O)N(C)CC2CCCCN2C(=O)C(C)N2CCC2)cc1 CCC(CC)C(=O)NCC1CCC(NC(=O)CCOCC(F)(F)C(F)F)C1 N1(C(=O)C2=COCCO2)CCC2(CC(NC(C3(c4ccc(Cl)cc4)CC3)=O)C2)C1 N1(C(c2ccnn2C)=O)CC(N(C)C)CC1(C)C.CCCC(C(=O)NC)N(C)C Cc1ccc(C(=O)NC2CCCCC2(F)F)cc1[N+](=O)[O-] Cc1cccc(C(N2CCC(NC(C34CC(C(C)C)(C3)C4)=O)C(C)C2)=O)c1N N1(C(CNS(N(C)C)(=O)=O)=O)CC2CC(NC(=O)Cn3ncnn3)C1C2 C1(CNC(C(n2cc(CC3(O)COC3)nn2)C)=O)(CO)COC(CO)C1 c1(C(N2CC(NC(=O)C=CC(F)(F)F)CC(C)C2)=O)ccc2ncsc2c1 c1(NC(C2(SCC)CC2)=O)nnn2ccccc12 C1(N(C(C=CC=CC)=O)C)CCCN(C(=O)CS)CC1.c1(CC)ccccc1 c1(C(N2CC(O)(CCNC(C(C(C)C)O)=O)C2)=O)cccc(N)c1C(F)F C1(C2CN(C(=O)OC(C)(C)C)C2)CC(=O)N(NS(=O)(=O)CCCCC#N)C1 N1(C(c2cc(C)on2)=O)CCC(C)C(CNC(c2coc(Cl)c2)=O)C1 c1(C(=O)OC(C(C)C)CN(C)C)ccc(S(=O)CC#N)cc1 C(C)(CNC(C1CSC1)=O)(CC(C)C)NC(CCc1cccc(C)c1)=O Cc1ccc(C(=O)NC2CCCC23CN(C(=O)C=CS(C)=O)C3)c2ccccc12 c1(CNC2C(c3c(C)c(Br)ccc3)C2)c(C(F)(F)F)nn2ccccc12 CC1CN(C(=O)CO)CC(CCNC(c2cc(C3CCC3)nn2C)=O)O1 N1(C(CCCCN(C)C)=O)CC(NC(C2CC(F)(CO)C2)=O)C2(CC2)C1 N1(C(CCCOCC=C)=O)CCC(N=[N+]=[N-])(C(=O)NC2CN3CCCC2C3)C1 C(=O)(CC1=CCCCC1)NCCCNCc1cccc(NC(C)=O)c1 C12(C(=O)NC(c3onc(C)n3)C)CCC(CN(C(c3ccc(C#N)cn3)=O)C1)C2 C(=O)(CC(C)CC(C)(C)C)N1C2CC(NC(Cc3c(C)cnn3C)=O)C(CC2)C1 Cn1cc(NC(=O)CN(C(=O)Cc2cc[nH]n2)C2CCC2)c(Cl)n1 N1(CCNC(c2cccc(O)n2)=O)CCN(C(C2CC3(CCO3)C2)=O)CC1 C1(CNC(CSCC#C)=O)CC12CCN(C(C1(N(C)C)CCCCC1)=O)CC2 C1(C(=O)NC2(CNC(=O)CC3CCOC3)CCC2)C=CCCC1.CCCC c1(NCC2CN(C(C(C)O)=O)CC2(C)C)ncnc2sc3c(c12)CCCC3 C(=O)(C(C)(C)CCC#N)NC(c1cccc(C)c1)CNC(=O)Cc1ccccc1 c1(C(=O)NC2CCC(NC(C(CC)O)=O)C2)cnc(Br)c(N)n1 N1(C(=O)C=Cc2ccsc2)CC2CC2(NC(C2(F)CC=CC2)=O)C1 N1(C(Cc2c(F)ccc(C)c2)=O)CCN(C(c2ncoc2C)=O)CC(O)C1 N1(C(C=COCC)=O)CCC(CO)(NC(c2cccc(OC(F)(F)F)c2)=O)C1 C(=O)(C1CSc2ccccc21)N1CC(Nc2nc(C)n3c(c2)nnc3)C1 CC(=NO)C1CC(C=O)C1(C)C.C1CC2CC(C1)N(C(=O)C=C1CCCC1)C2.N c1(C2(C(=O)NC(C)CCNC(=O)CCCC(N)=O)CCC2)cccc([N+](=O)[O-])c1 c1(CCC)ncc(C(=O)NCC2CC(C)CO2)s1.C1(CC=O)OCCCO1.N c1(C(N2CC3C(NC(c4cc(C)ns4)=O)(C3)C2)=O)c(N)cc(Cl)cc1Cl Cc1cnc(Br)c(NC(N2CCCCC2C2CCCCC2O)=O)c1 c1(C(=O)NC2CCC(NC(c3c(C)cccc3N)=O)C2)cc2c(s1)CCCCC2 C1(C(=O)NC2CN(C(C3CC(C4CC4)=NO3)=O)CC2F)CCCCC12OCCO2 C1(CC)CCN(C(=O)CCN(C)CCO)C(C(=O)N)C1.C1CCOC(C)(C)C1.C N1(C(CC(CC)C2CC2)=O)CC2CN(c3ccccc3)CC2C1.c1cccc(C)c1 CCCS(=O)(=O)CC(=O)N1CC(N2CCN(C(=O)CCc3cnoc3)CC2)C1 C(c1cccc(Cl)c1)=CC(N1C(CCNC(C(CC)=CC)=O)CCC1)=O.O C1(C(=O)NCCC(CC)(C)O)N(C(=O)CCc2ccnn2C)CCC1(C)C c1(C(N2C(C)CC(NC(C3CCN(CC#C)CC3)=O)C2)=O)ccc(N)c(N)c1 C=CCC(C)(C)CC(=O)NCC(CO)NC(c1ccnn1C(F)F)=O N1(C(CSCCC)=O)CC(C(=O)NCc2ncoc2CC)C(CCC)C1 c1(C(C(C)NC(=O)NCCC2CNC(=O)C2)O)ccc(F)c(F)c1 CC1(C)CC=C(C(=O)N2CCC3(CC(C(=O)NCc4ccsc4)C3)C2)CC1 N1(C(Cc2c(C)scc2)=O)CCC(C)C(NC(=O)CCc2nnc(C3CC3)o2)C1C N1(C(c2ccc(C)c(F)n2)=O)Cc2c(ccc(F)c2Br)C(C)(C)C1 c1(C(N2CC(NC(=O)C(C)COC)CC(OC)C2)=O)ccc2[nH]ccc2c1 c1(C(NC)=O)ccc(C(F)(F)F)nc1.N1(C(C2C(CC(C)C)C2)=O)CCCC1 c1(C(N2CC(C(=O)NCCOCCOC)C(C)C2)=O)cn2ccccc2n1 c1(CC)cccc(C(=O)NCC(CO)NC(C2CN(C(=O)NC)CCO2)=O)c1N c1(OC)ccc(NC(=O)C(N2CC(OC)C(OC)C2)c2ccn(C)c2)cc1 c1(CN2CCC3(C(=O)OC)C(C2)C3(F)F)cc2cc(Cl)cnc2[nH]1 Cc1cncc(C)c1C(N1CCC(C(C)NC(c2cc(CO)oc2C)=O)CC1)=O N1(C(c2ccc(OC)cc2C)=O)C2CCC1CC(CCNC(c1cnco1)=O)C2 N1(C(C(CN(C)C)NC(C2CC3CC(=O)C2O3)=O)=O)CCC(C2CCC2)C1 C1(C)(C(=O)N)CCCO1.C1(C(N(CCC)CC)=O)C(c2ccncc2)C1(C)C C1(CNC(C(C#C)(C)C)=O)CC2(CCN(C(=O)CCS(C)(=O)=O)CC2)CO1 C1(NC(=O)Cn2cc(Cl)cn2)CCC(O)CN(C(c2ccc(Cl)c(O)c2)=O)C1 c1(C(=O)NC(C2CCCN2C(=O)CCS(C)=O)C)cn2ccsc2n1 N1(C(CN(C(C)=O)C)=O)CCOCC(C)C1.C1(C=O)(C(F)F)CC(F)(F)C1.N c1(C(=O)NC(Cn2cc(CNC(C)=O)nn2)C)c[nH]c2cccc(F)c12 C1(OC)CC(CCNC(c2cc(C)oc2C)=O)N(C(=O)CN(C)C2CC2)C1 N1(C(C(=O)NCC2(CC(C)C)CCC2)=O)CCc2sc(CN)nc2C1 N1(C(C(CSC)C)=O)CCC(C)C(C(=O)N(CC(N)=O)CC(N)=O)C1 C(=O)(CC1=CCCCC1)NC1CCN(C(CCSCCC)=O)C1(C)C c1(NC(c2cc(OC)c(F)cc2)c2nnnn2C)cccc2c1CCC2 c1(C(=O)NCC(CN(C(=O)CCc2cccnc2)C)O)ccc(C2CC2)s1 c1(OC)cccc(CN2CCN(c3ccccn3)CC2)c1O.C12CCN(CC1)C2 c1(C(CC)SCc2nn(C)cc2Br)cccc([N+](=O)[O-])c1 CC1C(NC(C2CCS(=O)(=O)N2)=O)CCCN1C(c1nc(C2CC2)cs1)=O Cc1ccnc2c(C(N3CC(CNC(=O)C(F)=CCCF)CC3C)=O)cccc12 c1(CC)ccc(C(N2CC3(CCC3NC(=O)CCCn3cncn3)C2)=O)c(Cl)c1 N(C(=NC1CC1)N1CCCC(Oc2ccccc2OC)C1)C1CC(C#C)C1 c1(C(=O)NC2C(CNC(c3cnc(C)[nH]3)=O)C2)nc2ncc(Br)cc2[nH]1 c1(OC)ccccc1OCC(=O)N.c1(C(C=O)C)c(C)noc1C.CC=CC C(N=c1[nH]nc(C(F)F)o1)C1CCC(NC(=O)OC(C)(C)C)CC1 N1(C(c2n(C)ncc2CNC(C2C=CCCC2)=O)=O)CCCC2CC1C2(C)C C1(C(=O)NC(c2c[nH]ccc2=O)C)CC2(CCN1C(c1sccc1C#N)=O)CC2 C1(NC(C2C(C)CCCC2)=O)(C)CCC(F)(F)CC1.C(=O)(CCc1csnn1)N CCCCCC(F)C(=O)N1CCC(N(C(=O)CNc2cccnc2)CC2CC2)C1 N1(C(CCc2cc(C)[nH]n2)=O)CC2C(NC(=O)CC3CCOC(C(C)C)C3)C2C1 c1(NC=O)ccc(C(=O)NC(CCCNC2CCC2)c2ccccc2)cc1 c1(OC)cc(C(=O)NCC2CCC2)cc(F)n1.c1(CCC=O)cc(C)sc1C N1(C(CC(=O)OC)=O)CC2COCCC2(NC(c2ccc3nc(S)[nH]c3c2)=O)C1 C1(NC(C(C)NC(CC)=O)=O)CCCC(CNC(c2cnn(CC)n2)=O)C1 N1(C(CC2CCCN(C(c3c(C)csn3)=O)C2)=O)CCCOC(C(C)C)C1 N1(C(C)=O)CC2CCC1CN2CCO.Cc1cccnn1 N1(C(C(C2CCC(F)(F)CC2)OC)=O)CCCC(C#N)(c2ccccn2)C1 CC1CN(C(C2(n3cccn3)CC2)=O)CCC1N(C)C(C1CC(Cl)(Cl)C1)=O c1(C(=O)NC(CN(C(C(C)S(N)(=O)=O)=O)C)C)ccnc2c1CCO2 C1(NC(=O)COCc2ccncc2)CCCC(NC(c2cc(O)ncn2)=O)C1 N1(C(c2cc(OC)no2)=O)CCC2(CC1)OCCC2NC(=O)C1=C(Cl)CC1 c1(CN(c2c(C)cccc2C)C(N2CCSCC2C#N)=O)cc(Cl)c(Br)cc1F c1(C(=O)NC2C(NC(C=Cc3cncc(C)c3)=O)C2)cc(Br)c2n[nH]cc2c1 c1(NC(C2CC(NC(c3cc(O)c(O)cc3O)=O)C2)=O)ccn2ccnc2c1 c1(CC)cc(NC(=O)C(O)CNC(=O)C(C)(C)CF)ccc1F C1(N(C(C=COCC)=O)C)CN(C(=O)CSc2ccccc2C)CCC1O Cc1cc(F)c2cc(C(=O)NC3CC(CNC(C4CCCSC4)=O)C3)[nH]c2c1 N1(C(Cc2n(C)ccn2)=O)CCC2CCN(C(=O)CN3CCOCC3=O)CC2C1 CCCC(CCCNC(=O)C(O)CSC)NC(C12CC(C)(C1)C2)=O c1(C(=O)NC(C2CN(C(C=C(CCC)CCC)=O)C2)C)ccc2cc(C)cn2c1 Cc1cc(C(=O)N(C2CN(C(c3ccccc3O)=O)C2)C)cnc1C C(=O)(CCP(C)(C)=O)NCCOCCNC(C(C)(C)C1CCOC1)=O N1(C(C(c2ccc(C)cc2)C2CC2)=O)CC2CC(NC(c3cncs3)=O)CC2C1 Cc1cc(C(=O)NC(CNC(C2COCCO2)=O)C2CCC2)c(N)cc1F N1(C(=O)NCC(=O)OCC)CCCCC1.C1(C(=O)N)CN(C=O)CCO1 C1(CCNC(C(CC)F)=O)CCN(C(=O)Cn2cc([N+](=O)[O-])cn2)CCC1(F)F N1(C(CC2(C=C)CN(C(c3c[nH]nc3C3CC3)=O)C2)=O)CCC2(CCOC2)C1 C1(C(N2C(C)CC(NC(CCC(C)C)=O)C2)=O)CN(CP(C)(C)=O)C1 C1(C(N2CCC(C(C(=O)NC3C(SC)COC3)(C)C)C2)=O)CCC(C)=C(C)C1 C(=O)(CC1OCCc2ccsc21)NC1C(NC(=O)C=Cc2cccc(F)c2)C1 Cn1cnc(C(=O)NCC(C)(CO)NC(=O)CCC2(C)CC2(F)F)c1 N(C1c2ccccc2CC1NC(C1CCC(F)C1)=O)C(c1cnc(CC)s1)=O c1(C(N2CC(F)CC2C)C(=O)NC)cc(Br)ccc1OC C1(NC(CC)=O)CCCC(C(=O)NCC#CC#CCO)C1 c1(CC(=O)NCC2CN(C(c3ncccc3O)=O)C2)ccc(Cl)c2cccnc12 c1(C(CCC2N(C(CCn3ccc(C)n3)=O)CCC2)=O)cnccc1C c1(CNC(C(C(C)O)NC(C2CCC3CC3CC2)=O)=O)ccc2c(c1)CCO2 c1(C(=O)NCCC(C)NC(C(c2ccccc2F)OC)=O)ccc(C)c(N)c1 c1(C(N(C)C)=O)cc2c(s1)CCC2.C1CN(C(C2CC2c2cccs2)=O)CCO1 C1(CNC(COCc2c(C)ncs2)=O)C(C)CCN1C(c1cnn[nH]1)=O N1(C(c2nnn(C)n2)=O)CC2COCCC2(NC(=O)CCOc2cccnc2)C1 Cc1[nH]c(=N)nc(O)c1CCC(=O)OCc1cnc(-c2cccs2)o1 C(=O)(CC(O)CCCCC)NC(CC#C)(C)C(=O)NC1CCCC1O C1(NC(Cc2c(C)noc2)=O)(CO)CCCN(C(c2cc(Cl)ns2)=O)C1 C1(NC(c2c(OCC=C)cccn2)=O)CCN(C(C2CC2O)=O)CC12CCC2 c1(CC)ccc(C)c(C(=O)NC23CC(C(N4CCC(C)(O)C4)=O)(C2)C3)c1 Cc1cc(NC(C2CCC(C)N(C(=O)CC3CCCCC3)C2)=O)cc(CO)c1 CC(C)S(=O)(=O)CC(=O)N(C1CN(C(c2cc(O)ncc2F)=O)CC1(C)C)C c1(C(N(CC(C)O)CC)=O)cc(CNC(c2ccn(CCF)n2)=O)ccn1 N1(C(CSCCC)=O)CC(CCNC(c2ccccc2-n2cnnn2)=O)C(C)C1 Cc1nc(Cl)ccc1C(=O)NC1CC(C)N(C(=O)CC(C)n2ccnc2)C1 Cc1cccc(C)c1CC(=O)NC1CCCCC1NC(=O)C(F)C1CCC1 c1(CC(N2CCC(NC(C3(F)CCC(F)(F)CC3)=O)C2)=O)ccc2nonc2c1 C(=O)(C(C)(C)CCC#N)NCC(C)NC(=O)CCNC(c1cccnc1)=O c1(C(C)=O)c(C)[nH]c(C(N2CC(NC(C3C4CCCC34)=O)CC(C)C2)=O)c1C N1(C(C2C(C)C2)=O)C2CCCC1CN(C(=O)CCC(C)(C)F)C2 N1(C(c2cnoc2)=O)CCCC2(CCN(C(C3CC4CCCC(C3)C4=O)=O)C2)C1 C(=O)(C1=CCCN(C(=O)C2CC2)C1)NC1(C(=O)O)CC(OC)C1(C)C C=C(C)CC(C(=O)NC1(C(=O)NCC(N2CCCCC2)C)CC1(C)C)OC C1(C(=O)NCC2(C)CCN(C(=O)C3CC3)CC2)CCn2c(cnc2Br)C1 Cc1[nH]c2cc(Br)ccc2c1C(=O)N(C)CCNC(=O)CCc1ncco1 C1(C(C)(C)C)CCCC(CNC(N2CCN(C(=O)Cc3nc[nH]n3)CC2)=O)CC1 C1(CNC(c2c(CC)nc[nH]2)=O)CN(C(c2nc(C)no2)=O)CC(C)(C)O1 C1(C)(OC)CC(NC(C2CC(F)CCN2C(C2CC3CCC2CC3)=O)=O)C1(C)C C1(NC(CC(=O)OCC)=O)CCCCC1CNC(=O)C=CC1CCOC1 C(C(=O)N1CCC(N(C)C)CC1)(C(C)C)NC(Cn1ncc(CC)c1)=O N1(C(c2c(C#N)csc2)=O)CCC2CCC(NC(=O)CC3C=CCC3)C1C2 C1(C)(C(=O)NCc2c(C)nc(C)o2)CC(O)CN1C(=O)CC1CCSC1 c1(C(=O)N)cc(=O)n(C)c2ccccc12.C1(C=O)CC(C)=NO1.C(C)(C)OC C1(CC=C)(C(=O)NCC2(O)CC(C=O)C2)CCOC1.c1(CCC)ccccc1 S(=O)(=O)(c1ccc2c(c1)OCO2)N1C(CNC(CNC(N)=O)=O)COCC1 C1(C2CC2)(NC(c2c(OC)nsc2)=O)CCN(C(c2ncc(F)cc2F)=O)C1 c1(OC)cc(C(=O)NCC(C)NC(=O)C(C(C)C)n2cnnn2)cnc1OC C1(C(=O)NCCC=CCOC)(NC(C2CC2Cl)=O)CC(CO)C1 c1(C(N2CC(CNC(c3ccccc3)=O)C3C2C3)=O)ccnc2c(F)cccc12 c1(OC)cc(C(=O)NC(c2ccccc2)C)sc1Cl.C12(C=O)CC(C)C1C2.C N1(C(C(C)NC(C2COC2)=O)=O)CC=CC(NC(=O)CC23CC(C2)C3)C1 C=C(CNC(c1cnn(C)c1)=O)CCNC(c1cc(CCSC)on1)=O n1(CCC(=O)N(C)Cc2cnn[nH]2)cc(C2CC23CC3)nn1 c1(N(CC(CNC(C)=O)(C)C)C)nc(NCc2c(C)n[nH]c2C)c2ncsc2n1 c1(C(N2CCN(C(C(C)=C(C)C)=O)CC2C2CC2)=O)cc(C)c2nc(C)cn2n1 c1(C(=O)NC(c2cccc(C)c2)CNC(CC=C)=O)sc(S(N)(=O)=O)cc1C n1(CC)ncc2cc(C(=O)OC(C)C(=O)NCc3ccco3)c(C)nc12 C(c1ccc(Cl)s1)=CC(=O)NC1(CO)CN(C(c2n(CCCC)ncc2)=O)C1 Cc1nc(CC(=O)N(CC(O)CNC(c2nc(Br)c[nH]2)=O)C)n[nH]1 c1(C(N2CCC(C(C)NC(c3csc(C(F)F)n3)=O)C2)=O)nn(C)cc1Cl CC1=C(C(=O)N2CCC(=CCNC(=O)C(F)Cc3ccccc3)CC2)CCO1 C1(C(=O)N)CC2(CCOCC2)C1.c1(C(=O)NCC(C)CO)ccc(C2CC2)cc1 c1(C(N2CCC(NC(c3nnc(O)cc3O)=O)C(F)C2)=O)c[nH]c2cnccc12 CN1CCC(F)(C(N2CC3(CNC(C4(C)CCC4)=O)CCC2C3)=O)CC1 c1nc(O)c2c(n1)CCC2.C1(C(N(CCCC)CCO)=O)CC2CC2N1C(=O)N C(=O)CN=c1[nH]c(C)cs1.c1(CC)nnsc1C(=O)NCC1CC(F)(C)C1 C1(CNC(C2(C#C)CC2)=O)CCCCC1NC(=O)CO.c1nc(C)no1 c1(C(=O)NC2C(NC(C(C)SCCCC)=O)CCC2)nnn(CC)c1CCC C1Cc2ccccc2C1NC(=O)CCC1CCN(C)C1.C1(SC)CC(C(=O)N)C1.C N1(C(c2c(C)cc(C)o2)=O)CCCC2C1CCN2C(=O)CC1(C)CC1(Cl)Cl c1(C(=O)NCC=CCNC(CC(C)F)=O)cccc(Cl)c1C(F)(F)F c1ccc(Cl)c(F)c1.C1(CC)CSCCN1C(=O)C.CC(C)(C)C=CC(=O)N c1(CN2CC(O)(CNC(Cc3cccc(C)c3)=O)C2)ccc(C)c(Br)c1 C(=O)(CCCC1CC1)N(C1CCCC1)CCOC.C(=O)(C(C)c1ccco1)N CCCC(C=O)C(=O)NCC1(OCC(=O)NCC2CCCOC2)CCCC1 C1(C(=O)NCC2C(CC)CC2)CCCCC1CNC(c1cnn[nH]1)=O c1(CNC(C2(C)CCN(C3CCN(CCF)C3=O)C2)=O)ccc(F)c(F)c1 C1(c2n(CCCCCC)nnn2)(NC2CCN(C3CC3)C2=O)CCOCCC1C C1(CNC(C2CCN(C)C(=O)C2)=O)N(C(c2ccc(C#N)s2)=O)CCCC1(C)C N1(C(C(C2CCCN(C(CCOC)=O)C2)C)=O)CCN2C(=O)OCC2C1 c1(C(N2CCC(N(C(C(CC)OCC)=O)CC)C2)=O)c(OC)cnnc1OC CS(=O)(=O)C1CCCCC1C(=O)NCc1cn2c(n1)COCC2 CCC(CCCC(=O)N(C)CC1(C)CCCC1)NC(c1snc(C)c1N)=O C=CCCCCCCCCC(=O)N1CCCC1CNC(=O)C=CC(C)=O CC1CN(CCO)CCN1C(c1ccc(C2CCCCC2)cc1)=O c1(C(=O)NCC(CC)NC(c2cccc(C#N)c2C)=O)[nH]c2c(c1C)CCCC2 N1(C(c2cccc(C#C)c2)=O)CC2CCCC2(C(=O)NC(c2cccs2)(C)C)C1 c1(NC(C2CC2NCc2ccc(Cl)cn2)=O)ncc(C(F)(F)F)cc1Cl C(=O)(C1=CC2C=CC1C2)NCC(C)(C(C)C)NC(CC(CC)CN(C)C)=O N1(C(CN(C(CC2CC(=C)C2)=O)CC)=O)CCN(C(c2ccncc2Cl)=O)CC1 N1(C(CC2(NC(C(C(CC)C)N(C)C)=O)CCC2)=O)CCC2(C1)CC2(F)F n1(CC)cncc1CNC(=O)CC1CCN(C(C)C(=O)NC(C)C)C1 C1(OC)CCC2(C(=O)NCCCCCN(C)C(C3(C)CCN(C)C3=O)=O)CCC12 C1(O)(CN(C(COCCC#C)=O)C)CCN(C(=O)CC(C)COC)CC1 c1(C(C(=O)N(C)CC2N(C(Cc3ncc(C)o3)=O)CCC2)C)ccc(F)cc1 N1(CC=O)CCC(N(C)C)CC1.c1(C(N(CC(O)C)C)=O)sccc1C1CC1 c1(C(N(C(C)CNC(=O)CSc2nnnn2C)C)=O)nc(Cl)ccc1N c1(COC)nccc(N2CCC(C(C)NC(c3nc(C)sc3C)=O)C2)n1 c1(C(=O)NCCCC(C)NC(c2cn3c(n2)SCC3)=O)cc2n(n1)CCCN2 Cc1nc(C(=O)NCC(C)C(C)C)c(C(F)F)[nH]1.C(=O)(CCCN1CCCC1)N C(=O)(N=c1cc[nH]cc1F)C1(C)CN(C(C2(C(=O)OCC)CC2)=O)C1 C#CCCCC(C)C(=O)NCC(C(C)(C)C)NC(=O)Cc1cccc(C2CC2)c1 CC(C)(C)CCNC(c1cc[nH]c1C1CC1)=O.C1(C(C(=O)N)O)CCCCCC1 c1(C(=O)NCC2N(C(c3c(Cl)cn(C)n3)=O)CCC2)cc2c(cn1)CCCC2 c1(C(=O)N)cc2nnn(C)c2s1.c1(NC(C)=O)cccc(C(=O)N(CCC)C)n1 CC(C)C(C)CC.c1(CC=O)nc(=N)[nH][nH]1.C1(C(C)(C)C)(C(=O)N)CCC1 C(CC(C)C(=O)N1CCCC1C(C)(C)C(N1CC(C(N)=O)C(C)C1)=O)=CC C1(CCNC(CSC)=O)CC(F)(F)CN1C(=O)C(F)n1ccnc1 CCC(C)CCC(=O)NC1CC2(C1)CC(NC(=O)C(C)(C)C1CCOC1)C2 C1(O)(C(CNC(C)=O)C)CCN(C(c2cn(C3CCOC3)cn2)=O)C1 N1(C(Cc2c(C)cccn2)=O)CC(C)C(C)(C(=O)NC2(C(F)(F)F)CC2)C1 CC1CC(C(N2CCN(CCNC(=O)CCC3CCCOC3)CC2)=O)CCC1=O S(=O)(=O)(c1ccc(NCc2cnc(N(C)C)nc2)c(Br)c1)NC1C(C)CCC1 C1(C)(NC(C2CN(C(CC(CC)O)=O)CC2(C)C)=O)CCC2(CC1)CC2 CC(CF)C(=O)NCC(C)(O)CNC(c1csc(-c2ccco2)n1)=O Cc1ccc(Br)c(CC(=O)NC2CCN(C(C3C4CCOCC34)=O)CC2)c1 N1(C(CCc2n(C)cnn2)=O)CC2(CCN2C(C2CC2c2nccn2C)=O)C1 c1(C(=O)NCC2C(NC(C3(N=[N+]=[N-])CC3)=O)C2)cncc([N+](=O)[O-])c1 C(CCCC(=O)NC1(C)CC(C)C1)N(C(C(n1c(C)ncc1)C)=O)C C1(CC(=O)NC2C(Cc3c(C)cccc3)CCC2)COCC2(CCNCC2)O1 C1(C(=O)OC)CN(C(=O)CCc2ccc[nH]2)CC12CN(C(C1CC1C1CC1)=O)C2 Cc1c(C(=O)NCCCCN(C(=O)Cc2ccccc2Cl)C)oc2ccccc12 CCC(CCC(=O)N1CCCC(CN(C)C(c2c(C)ncnc2C)=O)C1)OC Cc1cccc(C)c1NC(=O)CCCCCN(C(=O)C(n1nccc1C)C)C CN1CCC(C)(C(=O)NC2CCCCC2)C1=O.C1(CC(=O)N)(N(C)C)COC1 N1(C(c2csc(C)c2C)C(=O)NCCCC)CCCC(CCO)CC1 CCC#CCN=c1ccc(Br)c(S(=O)(=O)NCC2(C)CC3CC3C2)[nH]1 CN1CC2CCN(C(C3OCCC3NC(=O)CCN=[N+]=[N-])=O)C2C1 C(CN=c1cccc(S(=O)(=O)N(C2(C)CCOC2)CC(F)F)[nH]1)(C(C)(C)C)N(C)C CS(=O)(=O)c1ccc(CNC(c2cccc3cnccc23)=O)cc1 C(C(C(=O)NCC1CCN(C(C)=O)C1)NC(C1CCOCC1)=O)SCC N1(C(c2c(C)cns2)=O)CCC2CN(C(c3nn(C(F)F)cc3Cl)=O)CC2C1 c1(-c2nc(CCCCCC)nn2C(C)C)cc(C)cc(F)c1 C1(C)(C(=O)NC(CCCNC(c2c(C)noc2C)=O)C)CCNC(=O)C1 C1(C(=O)NCC(C)N(C(=O)Cc2ccsc2Br)C)CN2CCC1CC2 C1(CC)CN(C(=O)C(C(C)(C)C)n2cnnc2O)CC2(CCCOC2)O1 N1(C(c2cc(C)c(I)cc2)=O)CC(CNC(=O)C(F)(F)F)CCC1(C)C c1(CC)cccc(F)c1.C1(C(=O)N)CC1C=O.C(=O)(C)N(CC)CC c1(C=O)ccc(F)c2ccccc12.C(CC)(C(C)C)NC(C1(OCC)CC1)=O C1CN(C(c2cccc(N)n2)=O)CC1(F)F.c1(CSC)ccc(C(=O)N)cc1.C C(=O)(CCCCC(=O)N1CC2CC(NC(c3c(Cl)cccc3Cl)=O)CC1C2)OC C12(CNC(CCN(C)CC)=O)CCC(CC1)N2C(=O)CC1CCC2CC12 C1(C(N2C3C(NC(=O)Cn4ncc(Br)n4)C(C3)C2)=O)CCc2cnnn2C1 C(C)(CCC(=O)NCC(N1CC2C(C(=O)NCCOC)C2C1)=O)OC N1(C(C(C)(C2CC2)OC)=O)CCOC(CN(C(=O)Cc2cscn2)C)C1 N1(C(C2C(C)C2)=O)CCc2cc(CC(=O)Nc3cccnc3C(F)(F)F)ccc21 C(CC(C)(C)C)(C(=O)N1CCCC1C)NC(CN(CCOC)C)=O N1(C(Cc2ncc(C)s2)=O)C2CCCC1CC(NC(=O)CC1CCCS(=O)(=O)C1)C2 C1(C(N2CC(C(C)NC(c3c(C)nsc3N)=O)C2)=O)CCC(C)NC1=O C12(CNC(C(CN(C)C)NC(C(CC#C)O)=O)=O)CC=CC(C1)OC2 c1ncc(C(F)(F)F)cc1Cl.C1(CCNC(C)=O)(CNC(=O)N)CCCC1 c1(CNC(c2c(N)ccc(SC(F)(F)F)c2)=O)cc2c(s1)CCOC2 C1(CC=C)CCN(C(=O)CCc2ccn(C)n2)C1.c1(CCC(=O)N)cnn(C)c1 N1(C(c2nc(C)oc2)=O)CC(C)CCC1CNC(=O)C=Cc1cncn1C c1(C(=O)NC2C(NC(C(c3ccc(C)cc3)C3CC3)=O)C2)ccc(C)nc1N C1C2CN(C(C3CC3c3cn[nH]c3)=O)CC12.c1(OC)cc(CCC(=O)N)on1.C C1(CNC(CC=CCC)=O)CN(C(C2CCS(=O)(=O)N2)=O)CCCO1 c1(CC(=O)NC(CC(=O)NC)c2ccccc2)cccc(N2CCCC2=O)c1 N1(C(CNC(C(CC)C)=O)=O)CCCC(N(C(=O)C2=CCC2)C)C1 C1(NC(C)=O)CN(C(=O)CC(c2ccccc2)N2CCCC2)CCC1CO C1(C(N2CCOCC2)C(=O)NCc2ccsc2CNC2CC2)CC12CCOC2 C1(C(=O)NC2(CN(C(CCSC)=O)C)CC2)CCCC(C)(C)O1 CON(CCC(=O)N1CC(N(C)OC)C1)C(=O)CCS(C)(=O)=O C1(C(N2C(CNC(CC(C)(C)C#N)=O)CCC2)=O)CC(c2cccc(F)c2)=NO1 C1(NC(=O)NC2(c3ccc(Br)cc3)CCC2)COc2ccc(F)cc2C1 C(C(C(=O)NC1CC1NC(=O)COc1cccnc1)N(C)C)OC C12(COCC)COC(C(=O)NC3CCC3)(C1)C2.C1(C=O)CC(C)CO1 N1(C(CCN(CC)CC)=O)CCN(C(C2CNC(=O)C2)=O)CC1CC.C(C)C C1(CNC(CCC#C)=O)COCCN(C(C2(c3cncc(Br)c3)CC2)=O)C1 C(=O)(C1=NOC2(CCC2)C1)N1CC(O)(CNC(CCc2scc(C)c2)=O)C1 c1(CC)cc(F)c(C(=O)NC2CC3CC2N(C(c2nc(C)oc2C)=O)C3)c(F)c1 CCC(C(=O)NC1CCCC1(C)CNC(=O)CC(C)N(C)C)C(C)C c1(CN(C(=O)C(C2CCOC2)NC(=O)CO)CC)cncs1.C(C)C C1(NC(C(CO)OC)=O)CCC2(CC1)CN(C(=O)CCC1(C#N)CCC1)C2 C1(OC(C)C)CCCN(C(C2CCC(CNC(=O)CN=[N+]=[N-])C2)=O)C1 N1(C(C2C(OCC)CC2)=O)CCC(C)N(C(C2CC(SC)C2)=O)CC1 C1(C(=O)NC(c2ccccc2)CO)C2CCCC2CN1C(c1ccc(CO)s1)=O C12N(CC1(C)C)C(=O)c1ccc(cc1)OC2.n1(C(CC)C)cc(CSC)nn1.O C(c1cn(CC(C)NC(=O)CN2C(C)CCC2C)nn1)=CC C1(O)(CN(C)C(c2cc(Cl)ns2)=O)CCN(C(=O)CC2(CO)CC2)C1 C1(c2onc(-c3ccc(OC)c(Br)c3)n2)CC2(CCOCC2)CCO1 CCCC(CCCNC(c1n[nH]cc1CC)=O)NC(=O)CC1CC2(CCC2)CO1 N1(C(CSCCC)=O)C2CCC(C2)C1CC(N1CCOCC1C(F)F)=O c1(C(N2CC3C(CNC(C(CC)(C)F)=O)(C3)C2)=O)cc2cc(Cl)ccc2n1C N1(C(COC(C)C)=O)CCC(C)(CNC(c2cc(N)ccc2Cl)=O)CC1 C(=O)(C(CCCCCCCC1CC1)N1CCC(F)(C(=O)OC)C1)NCCC C1(NC(C2CC(C)C2)=O)C2COCC1CN(C(=O)CCN1CCCCCC1)C2 Cc1cc(F)c(C(=O)NCC(C)CO)c(Cl)c1.c1(C(=O)N)coc(C(N)=O)c1 C12CCCC1N(C(C1CCS(=O)(=O)CC1)=O)CC2.Cc1cn(C)cc1C(=O)N.C CC1=C(Br)CCN(C(=NCCCCl)NCc2nnc(CO)s2)C1 C1(C)(NC(c2cncc(C(C)C)c2)=O)CCC(NC(C2CSCCS2)=O)CC1 c1(NC(C2(O)CCN(C(C(CC)CC)=O)C2)=O)ccc(Cl)nc1Cl Cc1cc(CN2CC3COCC3(C(N3CC(C)OC(C)C3)=O)C2)c(O)c(C)c1 C=CCCCCC(=O)N1CC(F)CC1CNC(c1cccc(CC#N)c1)=O c1(C(=O)NCC2CC(NC(CCCC=C)=O)C2)ccc(F)c2occc12 N1(C(c2c(C)coc2)=O)CCCCCC(NC(=O)COc2cn[nH]c2)C1 c1(CC(N2CC(C(C)(C)O)C2)=O)ccc(C)c(Cl)c1.C(C=O)(C1CC1)OC c1(C(N2CCCC(N(C(C(F)=CCC)=O)CCF)C2)=O)ccc(C)c(C)c1Cl C1(CNC(C#CC(C)C)=O)CN(C)CCN1c1cc(Cl)nc(C2CC2)n1 N1(C(C2(F)CCC2)=O)CC2CC1CN2c1nccc(OCC2CCOCC2)n1 C12(NC(CCN(CC)CC)=O)CCCC1CN(C(c1c[nH]cc1Br)=O)C2 C(C(C)CC(=O)NCCCC(CO)NC(C1CC(OC)C1)=O)OC c1(CC)n[nH]c(=NCC=CCNC(c2cc3c(nn2)CCC3)=O)s1 N1(C(C(=O)NCC(C)(C)OCCNC(C(CC)O)=O)C)CCCCCC1 Cc1nnc(CCC(=O)NCCC2CCCN2C(=O)CC2(C)CCC2)n1C N1(C(=O)C=CC2CCCCC2)CCC2(CC1)CCN2C(c1cc(Cl)cc(I)c1)=O N1(C(C2(OC)CCC(C)C2)=O)CC2(C1)CN(C(=O)C(F)=CC1CC1)C2 c1(C(N2CCC(NC(=O)CC3CC3(Cl)Cl)C23CC3)=O)coc2c1CS(=O)(=O)C2 C(C)(CCN=c1[nH]cc2ccnc-2[nH]1)NC(C(CC)Sc1ccccc1)=O c1(CC(=O)NC(CC)C(F)(F)F)cccc2c1CCC2 CCC(CCOC)C(=O)N1CC(CNC(c2cccc(C)c2O)=O)C2(CC2)C1 c1(C(=O)NC(CNC(CCCN(C(=O)OC)C)=O)C)cccnc1C(F)F C(=O)(C1CCSc2ccccc21)NC1C(O)CCN(C(C(C)=C2CCCC2)=O)C1 c1(OC)cc(C(=O)NCC2CCC2NC(C2CC2C2CC2)=O)cc(Cl)n1 N1(C(=O)Cc2ccc(Cl)cn2)CCN(Cc2ccc(Cl)o2)C2CC12 C(=O)(C1=C(C#N)CCC1)N1C(C(=O)NCC(C)OC(F)F)C(C)CC1 C1(N(C)C(C2CC3(CCC3)CO2)=O)CCCN(C(C23CCCC2(CF)C3)=O)CC1 C1(NC(CCN(C)CC)=O)CN(C(=O)C(C)OCC(F)(F)F)CC12CC2 N1(C(C(c2ccnn2C)C)=O)CCC(NC(c2csnn2)=O)C12CCCC2 CCCCCCCC(=O)N(C)CC1CN(C(c2ccc(CO)cn2)=O)CC12CC2 C=C(C)CN=C(NCc1csc(COc2ccccc2F)n1)NC1CCSC1 O=C1CC(C(=O)N2CCC23CN(C(c2cnn(CCO)c2)=O)C3)=NN1 c1(C(=O)NC2CCN(CC(C)(C)C)C2)cc(C(F)(F)F)nc2c1CCCC2 Cc1nonc1CC(=O)NC(C)CNC(c1cc(I)on1)=O C1(C2CN(C(C3(CO)CCCC3)=O)C2)(NC(CC(c2cccc(F)c2)C)=O)CC1 C1(CC(=O)N(C)CC2CCN(C(CSCCC(C)C)=O)C2)CCC12CCC2 N1(C(=O)NCCOc2ccc(CC)cc2)CC2CC(N=c3ccnc(CO)[nH]3)C2C1 c1(C(N(CC(CC)NC(=O)Cc2ncsc2Cl)CC)=O)nocc1Cl C(=O)(N=c1nc[nH]n2cccc12)c1c(-c2cc(C)cc(C)c2)ncs1 C1(NC(c2c(C)nc(CC)o2)=O)CC(O)CN(C(c2cn(C)nn2)=O)C1 C1(SCC(=O)N)CCCCO1.n1(CCC=O)cc(CC(c2ccccn2)O)nn1 c1(C(N(CC(=O)N(C)CC2CC2(F)F)CCC)=O)cnnc(O)c1 C1(CC(N2C(C)(CCC)CC2)=O)CC2(C1)CN(C(=O)CC1CCCCC1)C2.C N1(C(C2C(=C)C2)=O)CCC2(CCCN(C(c3cc(Br)c([N+](=O)[O-])[nH]3)=O)C2)C1 N1(C(=O)CC2CCC2)CC2CN(C(c3c(Cl)cccc3I)=O)CC2C1 c1(OC)ccc(-c2cn(CC(F)CCNC(=O)C=C3CCC3)nn2)nn1 Cc1c(C(=O)NCCNC(=O)COC2CCCC(C)C2)ncn1C CCCC(CCC)C(=O)NC1CCC(C(=O)NCC23CCC(CC2)OC3)CC1 c1(C(C(=O)NCCC)(C)C)ccc2c(c1)OCO2.C12(C=O)CCC(F)C1CC2.N C1(C(N2CC(CC(=O)NCC3CN4CCN3CC4)OCC2)=O)CN2CCC1CC2 N1(C(CC(C)C2CC2)=O)CCC(CF)(NC(=O)Cc2ccc(Br)cn2)C1 N1(C(C(COC(C)C)(C)C)=O)CCC2OCCN(C(c3cccc(Cl)c3)=O)C2C1 C(=O)(CC1OCCc2ccccc21)NCC1(O)CN(C(CC(CCC)(C)C)=O)C1 CC1CCNCC1CNC(C1CCC1CS(N)(=O)=O)=O C1(N(CCN)CC2CC2)CCN(C(c2cnn(C3CCC3)c2)=O)CC1 c1(C(=O)NC(CNC(CC2CC(CC)C2)=O)(C)C2CCC2)cc(C#N)c[nH]1 N1(C(C(C)OC)=O)CCCC1CN(C)C(C1CC(C(C)C)C1)=O CC(C)(CN=c1[nH]c2c(c(=NCC3CCOCC3(C)C)[nH]1)SCC2)n1cccn1 C1(CCC)CN(C(=O)OCC(F)(F)C(F)F)CC1NCCOC(C)(C)C CCC(CC)(CO)C(=O)NC1CCCC(C(=O)NCC(C)(C)COC)CC1 c1(NCCC(CC)(C)C)[nH]c(=NC2CC(C)N(C3CC3)C2)nc2sccc12 Cn1nc(C(=O)N(CC(N2CC(O)CC(O)C2)=O)C2CCC2)ccc1=O C1(NC(c2cc(COC)no2)=O)C2CCN(C(=O)C(C)C3CCC3)C12 c1(C(N2CCCC2C=O)C(=O)N)ccc(C2CCC2)nc1.C(C)(C)C.C=CC N(C(=NCCC1CC=CCC1)NCC1CC1)CCc1c(OC)cccc1 c1(CC)nn(C)cc1NC(C1CC(CNC(=O)C2=C(C)CC2)C1)=O C1(NC(C(C)O)=O)CCC(F)(CNC(c2cnc(N(C)C)nc2)=O)C1 N1(C(C(=O)NCCCC)C)CCC2(CC1)OCCC2C(=O)OCC CP(C)(=O)C(CCSc1ccccc1)NS(=O)(=O)C1CC1(C)C N1(C(C(CC)OC)=O)CCC2(CC1)CC(NC(=O)Cn1ncc(O)nc1=O)CO2 c1(-n2c(CNC(CCCC#C)c3ccccc3)nnn2)ccc2c(c1)CCC2 c1(C(N(C(C)CN(C)C(c2ccnc(C3CC3)n2)=O)C)=O)cc2c[nH]cnc-2n1 C1CCCCN(C(c2ccnc(C)n2)=O)C1.N1(C(C)=O)C(=O)CCC1C(=O)NC C1(NC(c2ccnn2C2CC2(F)F)=O)CN(C(C2CC2)=O)CC2(CC2)C1.C CCC(COc1ccc(F)cc1)N=c1[nH]c(=N)[nH]c(=NCC2(CN(C)C)CC2)[nH]1 N1(C(Cc2cc(C)no2)=O)Cc2ccccc2C(CNC(C2(N=[N+]=[N-])CC2)=O)C1 c1(C(=O)NC2CC(OC)CN(C(c3cccnn3)=O)C2)cccc2ccoc12 N1(C(C2=CCN(C(c3cncc(C)c3)=O)C2)=O)Cc2cc(O)nnc2C1 c1(C(N2CCC(CNC(C3(CCCC)CC3)=O)C(C)C2)=O)c(C)cc(C)nc1O C(=O)(C1=CC2(CCN(C(=O)C(C)O)C2)C1)NCCC=CC=C C=CC(CC)C(=O)NCc1cc(C(=O)NCCC2(C)N=N2)n[nH]1 Cc1csc(=O)n1CC(N1CCCC(CN(C)C(C2C3CCN2CC3)=O)C1)=O C1(NC(C(C2CCC(=O)N2)C)=O)CCC(C=O)CC1.c1(C(=O)N)snc(O)c1Cl Cc1nc(C(c2ccccc2)OC(F)F)c2c(C)csc2n1 N1(C(c2n(CC(C)C)ncc2)=O)CC2CCN(C(c3cccc(=O)o3)=O)C(C2)C1 C=C(C)C(C)(C)C(=O)NC1CN(C(c2cc(Cl)ncc2NC)=O)CC1C C(C)(C)(C(=O)NCCCC(=O)NCC#CC1CC1)SC C1(NC(C(CC)N(C)C)=O)CC2COCC(C1)C2NC(=O)Cc1cncn1C c1(C(=O)NC2CN(C(C3CCN(C(CC)=O)C3)=O)C2)ccc(=O)n(CC)n1 C(C(C)C(F)C(=O)NCCC(C)(C)CC=C)NC(C(C=C=C)C)=O C1(C(=O)NCCCOCCCC)CCC2(CN(Cc3ccncc3F)C2)O1 N1(C(CSCCC)=O)CC(C2CCCN(C(=O)Cc3c(C)nc(O)nc3C)C2)C1 N1(C(C2CN(C(N)=O)C2)=O)CCN(C(=O)CS(N)(=O)=O)CC1C1CC1 c1(C(=O)NC2(CCN(C)C)CC2)ccc(Cl)c(Cl)c1N c1(C(=O)NCC(c2cccc(Cl)c2)NC(CS(CC)=O)=O)cccn2nccc12 C1(COC)(CNC(c2ccncc2Cl)=O)CCCN1C(=O)CN1CCCCCC1 C1(CNC(CCCN(C)C)=O)CC2CCCC2N1C(C1CC(CF)C1)=O C1(C(=O)NC2CN(C(C3CC(C)C3(C)C)=O)C2)CCC2(CC1)CC(N(C)C)C2 Cn1cc(C2CC2C(=O)NCC(O)CC)cn1.c1(C2(C(=O)N)CC2)ccno1 N1(CC=C)CCC(NC(=O)C(CC2CCC2)NC(c2cc(F)c[nH]2)=O)CC1 N1(C(c2cccc(SC)c2)COC)CC(C)(C)c2cccc(C(F)(F)F)c21 n1(C(CC)C)cc(S(=O)(=O)N(C)C)cn1.N12CCOC(C1)C(=O)C2 c1(C(=O)OC)ccc(O)c(NC(C2C=CCN2C(C2CC(=O)C2)=O)=O)c1 C#Cc1cnn(C)c1C(=O)NC1CCC(C(=O)NC2C(O)C3CCOC23)CC1 N1(C(COCCC)=O)CC(C(=O)NC(C)(C)CCF)C(C)(C)C1 N1(C(C2=C(C)OCC2)=O)CCC(C2(NC(C3CN(C(N)=O)C3)=O)CC2)CC1 C1(NC(C(N(C)C)C2CC2)=O)C2CN(C(=O)CCCN3CCCC3)CC12 C(N=c1ccc(Br)n[nH]1)c1c(C)nn(CCO)c1 N1(C(C(C)Cn2cccn2)=O)CCC2C(NC(c3cc(C4CCC4)[nH]n3)=O)CC12 C1(CC(=O)NC2C(C(N3CCC(C(C)C)C3)=O)OCC2)CCCC(C)O1 c1(CC)ccc(C)cc1C(=O)NCCCN(C)C(c1cc[nH]n1)=O c1(C(=O)NC(CNC(C2N(C(C(C)C)=O)CCC2)=O)CO)ccc2nncn2c1 N1(C(c2cc(N)cc(F)c2)=O)CC2(C1)SCCC2.C1(CC(=O)N)CC(=O)NC1=O C(C)(C(CC(=O)NC1CCCC(O)CC1)NC(=O)C=CC(=O)N(C)C)OC N1(C(c2nnc(-c3c(CC)cccc3)s2)=O)CC2(c3ccccc3)CC1CCO2 Cc1[nH]nc(C(=O)NCCN2CCN(C(=O)CCC(=O)OC(C)(C)C)CC2)c1Cl Cc1ccc(Br)c(NC(c2ccc(CCC(=O)Nc3ccc(O)c(C)c3)[nH]2)=O)c1 c1(CC(=O)NCCC2CC(NC(CCNC(=O)NC)=O)C2)ccccc1 C1(COC)(NC(c2nnnn2CC(F)F)C2CC2(Br)Br)CC=CC1 C1(C(N2CC(OC)(C)C2)=O)CC(=C(F)F)C1.C1(C(=O)N)CC1C(C)C C1(C(N2C3CC(CN(C(c4ccnc(F)c4)=O)C3)C2)=O)C2Sc3ccccc3C12 N1(C(c2c(C)ncn2C)=O)CC2CCC2(NC(c2ccc[n+]([O-])c2)=O)C1 c1(C(=O)NCCC2N(C(C3OCCC(C)C3)=O)CCC2)cc2cccnn2c1 c1(NCc2ccc(C(=O)OC)[nH]2)cc(C(C)C)c(F)cc1C CCCCC(C(=O)NCc1nnc(O)n1C)NC(=O)COC(C)=O N1(C(C2C(C)(CC)C2)=O)CC(NC(=O)CSC(C)C)C(CO)C1 c1(C(=O)NC(C(=O)N(CC(F)(F)CO)C)C2CCCC2)ccn2ccccc12 S1(=O)(=O)c2c(OC)cc(cc2)O1.n1(CCOC)cc(CNCCO)cn1.O C1(C(=O)NCC(CC=C)NC(=O)COC)CCCN(C(C2CCN2C)=O)C1 N1(C(C2C(CNC(c3nc(C)n(C)c3)=O)C2)=O)CC(C)OC(C)(C)C1 C=CC(C)(C)CC(=O)N1CCC(OCC(=O)NCC(CO)CC(C)C)C1 C(=O)(CC1=CCOCC1)NC1C(NC(CCCOC)=O)CC(F)(F)C1 C(=O)(CCCCCC#N)N1C(C(=O)NCCN(C2CC2)CC)C2CC2C1 CC(C)(C)CC(=O)NC12CC(NC(c3coc(C4CCCC4)n3)=O)(C1)C2 C1(NC(c2cc(C)on2)=O)CN(C(c2cc[n+]([O-])cc2)=O)CCC1C N1(C(COCCCC#C)=O)CC(CCNC(c2c(C)ccnc2C)=O)OC(C)C1 C1(C(=O)NCCCCCC(=O)OC)CC12CCN(Cc1ccc(Br)s1)CC2 C1(C(=O)NC2CCC(CNC(C3(C=C)CC3)=O)CC2)COc2cc(F)ccc2O1 C(=O)(C(F)CCC(C)(C)C)N.C(=O)(C(C)CNC(=O)CCC1CCC1)OC C1(C2CCC2)(C(N(CC(C)(C)C)C)=O)CC1(F)F.Cc1ccc(N)c(C=O)c1.N C(=O)(C(CCC)C(C)C)NC(C(=O)N(C1CCCC1)CC=C)CC1CC1 N(C(=NCCCCl)NC1CCN(C(=O)C(C)C)CC1)CC(CC(C)C)C c1(NC(C(CCSC)NC(C2CCCC(=O)N2C)=O)=O)ccc([N+](=O)[O-])cc1 C1(CCNC(C=Cc2cn(C)nn2)=O)CN(C(c2ccnc(S)c2)=O)CCCO1 c1(C(N2CCN(C(=O)OC(C)(C)C)CC23CC3)=O)nc(O)c2ccccc2n1 C1(NC(CCCOCC)=O)CC(NC(C23CC(CO)(C2)C3)=O)CC1O C=C=CCN=c1[nH]c(=NCCCN2CC(C)CC(C)C2)c2cccc(F)c2[nH]1 Cn1ncc(Br)c1CN1CC(NC(=O)Cc2ncccn2)C(O)C1 C1CC2(C1)CN(C(c1cc(C(F)F)cs1)=O)C2.c1(CC)cc(CC(=O)N)on1 Cc1onc(C2CC2)c1C(N1CC(NC(=O)CCc2ccc(Cl)s2)C(O)C1)=O C=C(Br)CCC(=O)N1CC=CC1CNC(=O)C(C)(C)n1cnnn1 c1(C(C(=O)NCCCSCC)N(CC(F)Cl)C)cc(Cl)cc(Cl)c1 C1(C(=O)NCC2(NC(C3N(C=O)CCC3)=O)CC2)CCC2(CCC2)CO1 c1(C(N2CC(O)(CN(C(C(F)=C(C)C)=O)C)C2)=O)n[nH]c2c1CCCC2 CC(C)CCC(O)C(=O)N1CCC(C)(NC(C2(F)CCOC2)=O)C1 C1(NC(C(C)CC(C)(F)F)=O)CC1C1CCN(C(=O)CCc2cnn(C)c2)CC1 CCCCC(F)C(=O)N1CCN(C)C(C(=O)NC2CC(CO)C3CC23)C1 C1(NC(C2CCCN(C(C3(C#N)CC3)=O)C2)=O)CCCCC1(F)F CC1(C)CN(C(=O)C(N2CCCC(C(c3ccccc3)O)C2)=O)CC(C)(C)C1 C1(NC(c2n(CCC)nc(C)c2)=O)CCC12CN(C(c1cn(C)nc1O)=O)C2 c1(N2CC(CC(=O)NC)OCC2)nc2cc[nH]c2c(=NC(C)c2cn(C)nn2)[nH]1 Cc1nccc(C(N2CCC=CC2C(=O)N(C2CC3(CC3)C2)C)=O)c1C c1(NC(CNC(Cc2cnc(C)s2)=O)(C)C)ncnc2sc3c(c12)CCC(C)C3 c1(C(N2CC3C(N(C(CC(C)C)=O)C)C3C2)=O)cc(N=S(C)(C)=O)ccn1.CO N1(C(c2cccc(C(N)=O)c2)=O)CCC2C(NC(C3CC4CC4C3)=O)CC12 CCCC(C(=O)N1C2CCC1C(C)C2)S(N)(=O)=O.C1(C(=O)N)CN(C(C)C)C1 N1(CCNC(C2CC23CC3)=O)CCCC(OCC(F)F)C1 CC(O)C(F)(F)C(=O)NC1CCC(NC(C2(O)CC2)=O)C1 C#Cc1c[nH]nc1C(=O)NCC1(F)CCC1.C(=O)C(C)(C)Cc1ccccc1 CCC(CC)(CO)C(=O)N1CCC(C)C(NC(C2(c3cccc(Cl)n3)CC2)=O)C1 C1(NC(CCCCCNC(CC(C)F)=O)=O)CC(C)N(C)CC1C c1(NCc2c(C)onc2)ncnc2c(Cl)cccc12 O=C(C1=CSCS1)NCC1CCN1C(=O)COc1cccc(OC(F)F)c1 C(c1ccccc1)=C(OC)C(N1CCOC(CNC(=O)COC2CCOC2)C1)=O C1(C(N(CC(CC)NC(=O)CCCOC(C)=O)C)=O)CCCCCC1 Cc1cc(C(=O)NCC23CC(NC(C4(C)CCOCC4)=O)(C2)C3)c(C)o1 C(C(COC)CC(=O)NC(C(=O)NCC(c1nccs1)C)C(C)C)OC c1(C(N(CC(C)CNC(=O)C(F)C2CC2)C)=O)snc(Cl)c1Cl C1(CCNC(c2c(CC)onc2)=O)CN(C(=O)CCN2CCOC2=O)CCCO1 N1(C(C(C=C)O)=O)CC(=O)NC2CN(C(=O)C(c3ccc(Cl)cc3)(C)C)CCC12 c1(CC(=O)N)n[nH]c2ccccc12.CC1(C)NC(=O)CC1C(N1CC(CO)C1)=O c1(NC(=O)NCC(C(OCC)OCC)O)cc(Cl)ccc1Cl C1CC(C)N(C(=O)C(CC)=CCCC)C1.C1(CC(=O)N)(C(=O)OCC)CC1 c1(C(N2C(C)(C(=O)OC)CC(F)(F)C2)=O)cc2c(Cl)c(Br)ccc2s1 N1(C(C2CC(OC)C2)=O)CCC(CNC(=O)CCC2CCCOC2)C(O)C1 c1(CN(C)C(c2cc(-c3ccsc3)n[nH]2)=O)cncc(Cl)c1 Cc1ccc(C(C)NC(=O)C(C)N(C)CCN(C)CCO)s1 C=CCCN=C(NCc1ccnn1C)NCC1CCC2(C1)CC2(F)F c1(CN2C(C(=O)Nc3ncc(Br)c(O)n3)CCC2)c(F)ccc(Cl)c1F N1(C(CC(C)C2CC2)=O)CC2CN(C(C3C4CCC(=O)C34)=O)CC2C1 CC1(C)C2CN(C(c3sccc3Cl)=O)C(C(=O)Nc3cccc(C(N)=O)c3)C12 Cc1nn(C)c(Br)c1C(N1CC2(CC(NC(=O)C=CC3CCCO3)C2)C1)=O C12(C(=O)NC(CCC=C)C)C(NC(C3CC4(C3)CC43CC3)=O)C3CC1C2C3 c1(-c2cn(C(C)CNC(=O)COCCCF)nn2)cn2ccccc2n1 c1(C(=O)NC(CNC(c2c(CC)nc(C)n2C)=O)C)nnc2n1CCCC2 c1(C(N(C2CCN(C(COC(CC)C)=O)CC2)CCO)=O)cccn2nnnc12 C1(N(C(c2cc(C)sc2)=O)C)CN(C(=O)C(C2CCOCC2)C)CCC1C Nc1ccc(C(N2CC(O)CC2CNC(c2sccc2C(F)F)=O)=O)cc1F C1(C(=O)NCCN(C(CC=CCC)=O)C)CCC(C)CC1 NC(=O)CC(O)C(=O)NC1CN(C(=O)CSCc2ccncc2)CC1O n1(C(C)C)ncc(Br)c1C(N1CCCC(N(C(=O)C(CO)N(C)C)C)C1)=O c1(CCC)ccc(C(=O)CCC(=O)NC(C)(COCC)CO)cc1 C(=O)(C1Cc2ccc(F)cc21)NC1CCN(C(c2n(C)c(Cl)cn2)=O)CC1(C)C c1(C(=O)NC(C2CN(C(=O)CCCc3ccc(N)cc3)C2)C)occ2c1CCOC2 C1(CC(C(=O)NC2CCN(c3cccc(Br)c3)C2=O)N(C)C)CCCCCC1 C1(NC(=O)C=CC2CC2)CN(C(=O)C(O)C2CC2)CC2(CC2)C1 N1(C(CCNC(COC)=O)=O)CCC(C)C1.c1(C=O)cc(C(C)(F)F)on1.C CCCCCCCCCCC(=O)NC12COCC1CN(C(=O)C(C)OCCC)C2 C(=O)(C(C(C)O)N(C)C)NCC(C1CC1)NC(c1c(CCC)n[nH]c1)=O Cc1nc(C)c(F)c(=NCC2CN(C(=O)C(F)n3cccn3)C2)[nH]1 C1CCC(C(N)=O)CC1.C1(CC(=O)NCC(C)(C)OCC=O)CSCCO1.N N1(C(C(C)OCCOC)=O)CCC12CN(C(=O)Cc1cccnc1C)C2 Cc1cc(C(N2CCSCC2C(=O)NCC2CCOCC2(C)C)=O)nnc1O C(CCC(N)=O)(C(=O)NC1CCN(CCNC(C2CCN(C)C2)=O)CC1)N(C)C N1(C(C(C(C)(C)F)(C)F)=O)CCC2(CCCCN(C(=O)C(N)=O)C2)C1 c1(C(=O)OC)cc(C(NC2=COCC2)c2nnnn2-c2ccccc2)oc1C C1(c2ncc(C)s2)CCCCN1C(=O)Cc1ccoc1C c1ccccc1.CCC(C)C(=O)NCC1(O)CN(C(=O)COC2CCCC2)C1 N1(C(C2(OC)CCSC2)=O)CCC2CCC(NC(c3cnnc(O)c3)=O)C1C2 N1(C(C2CC=C(C)CC2)=O)CCC2(CC1)CN(C(=O)C(O)(C(F)(F)F)C1CC1)C2 CC(F)CN=c1[nH]c(=NCCOCC(F)(F)F)[nH]c2ccsc12 C1(CNC(=O)CO)CN(C(c2cnc(COc3ccc(Cl)cc3)o2)=O)CCO1 N1(C(CC2(C=C)CN(C(C3CNC(=O)C3)=O)C2)=O)CCc2nccnc2C1 C1(NC(C(C)OCOC)=O)CN(C(=O)C(CC(C)C)n2cccc2)CCC1CO CN1CCC2CCN(C(C3CC(NC(=O)C#CC4CCCCC4)C34CCC4)=O)C2C1 CCC(C(=O)NCc1c[nH]nc1C1CCN(C(C2(F)CC2)=O)C1)c1cccnc1 N1(C(CCC(=C)Cl)=O)CC(=O)NC2CN(C(=O)C(CC)CCOC)CCC12 N1(C(C)=O)CCCCC1CC(=O)N(C1CC(NC(=O)C=CC2CCOCC2)C1)C C1(CN(C(CSCCC)=O)C)CCCC1NC(=O)C(=Cc1ccco1)C C(=O)(CC(C)(C)C1CC1)N1C(Cn2cc(C3(COC)COC3)nn2)CC1 c1(-c2cc(C(=O)NC(C3CCN(C(C4CCO4)=O)CC3)C)n[nH]2)ccccc1O N1(C(=O)CSc2cccc(Cl)n2)CC2CCCC(C(=O)O)(C2)C1 N1(C(C(CC(=C)C)NC(=O)CN2CC(=O)NC2=O)=O)CCCC(F)(F)CC1 C(=O)(CCCCCF)NCC(C)NC(=O)Cc1cccc(OC(C)C#N)c1 C1(CC(=O)N(C(C)C(=O)N(c2cnsc2)CC)CCC)CCSCC1 N1(C(C)=O)CCCC(N=c2nc3c(ncn3C)c(NCC3(OCCO)CCC3)[nH]2)C1 C1(CCC)CCCCC1NC(=O)NC(C)Cc1cn(C)cn1 N1(C(C(COCC)C)=O)CCC2(C)CCCC12.c1(C(=O)N)c(O)nnc(C)c1C C1(CC(=O)N(CCOC)CCOC)CCN(C(=O)CCC2CCCC2)CC1 c1(C(N2CC(CN(C(c3ccc(CC)[nH]3)=O)C)OCC2)=O)cc(O)cnc1N Cc1cc(C(=O)NC2CC2NC(=O)Cn2cnc([N+](=O)[O-])n2)c(F)cc1Cl N1(CC(=O)NCCC2CC2)CC(CC(=O)ON)C1 c1(OC)cc(C(N2CCCCC2C)=O)c(Cl)cn1.C1(C)(CC=O)CC1(F)F.N CCC(C(=O)N1CC=C(C)C1)NC(C1CCN1CC)=O c1(NC(N2CC3CN(C(Cc4cn(C)nc4)=O)CC32)=O)cccc([N+](=O)[O-])c1 c1(C(=O)NCCCCCN(C(=O)C(C)(C)F)C)cc2c(Cl)cccc2s1 N1(C(Cc2ccc(C)o2)=O)CCCN(C(=O)Cc2ccns2)C(CO)C1 C1(C)(C(N(C)C)=O)CCCN(C(c2cc(C)nc(O)c2)=O)C1.N1(CC)CCCC1 CCCCC(C)CCC(=O)N1CC(NC(c2ccn3ccnc3n2)=O)CC1(C)C C(=O)(C#CC1CCCCO1)NCC(CNC(c1ncc(OCC)cc1Cl)=O)CO C1(CNC(C(CC)O)=O)CN(C(=O)C(=O)NCCC(N)=O)C2(CCOCC2)C1 c1(N(CC)C)cc2ccccc2c(=O)o1.C(=O)(CNCC(=O)NCC)N(C)C N#Cc1c(N2CC3(CN(C(=O)Cc4ccc([N+](=O)[O-])cc4)C3)C2)cccc1F C1(C(=O)NC2(C(C)O)CC2)CC(F)CCN1C(=O)CC1CC=CC1 CCC(CC(=O)NCc1cn(CCOC2CCSCC2)nn1)C(C)(C)C N1(C(C(C)C)=O)CCC(C(c2ccccc2)O)CC1.n1(CCN)nnc(CC(=O)O)n1 N1(C(C)=O)CCC2(CC(NC(=O)CON=C3CCCCCC3)C2)C1 CCCC(C(O)C(=O)NCC(N)=O)NC(=O)CCCn1ccnn1 C1(C(N(C2CCN(C(=O)CC3COCCO3)CC2)CC)=O)CCN(C2CC2)C1=O c1(CN(C)Cc2ccnn2C)ccccc1CNC(c1nccn1C)=O C1(C(=O)NC(C)C(=O)NCCC2CCCC3CC23)C2C3CCC(C3)C12 c1(C(N2CC(NC(c3ccc(=N)[nH]c3)=O)C2)=O)cc(Cl)c2cc(Cl)ccc2n1 N1(Cc2csc(C)c2C)CCOC(C#N)C1.C12CCCN1C(=O)c1csc2n1 c1nnc2nc(C)cc(C)n12.C1(C(OCC)OCC)CC(F)CN1C=O.C c1(C(=O)NC2C(NC(CCC=C(C)C)=O)COC2)nc(-c2cnn(C)c2)oc1C Cc1sc(C(=O)NC2CC(CNC(=O)CCN(CC(F)(F)F)C)C2)nc1O Cc1ccccc1C1CC1NC(C12CSCC1C2)=O.C1(=O)CCN1C(C)C C(CCCC(=O)NCC1CCCC1NC(=O)CC1CN(C(C)=O)CCO1)OC C1(CNC(=O)CC(F)(F)F)CC2(C1)CN(C(c1cc(O)no1)=O)C2 C(=O)(C(CC(C)C)OC)NCCN(CC(C)O)C(c1noc(CC)c1C)=O CC(C)C(C(=O)NCc1cc(C(=O)N(C(C)C(C)(C)C)C)n[nH]1)N(C)C N1(c2snc(C(=O)OC)n2)CCC(NC(c2cnn(C(C)C)c2)=O)C(CO)CC1 C(=O)(CC1=NNC(=O)C1)NCCc1ccc(CNC(CC(C)C(F)F)=O)cc1 C(=O)(CCCCCCCCCn1cc(C(C)NC)nn1)NC(CCSC)=O c1(C(=O)NC2(CCC)CCC2)cc(CNC(c2ccccc2)=O)[nH]n1 C1(NC(c2occc2F)=O)CN(C(c2ccoc2)=O)CC2(CCOCC2)C1 C(N=C(NC(CF)CF)NCc1ccco1)c1cnc(C)s1 N1(C(Cc2cn(C)nn2)=O)CC2CCN(Cc3ccc(C(F)(F)F)nc3)CC2C1 C1(NC(c2cc(SC)oc2)=O)CN(c2ncc(C(C)(C)O)cn2)CC1(C)C c1(C(N2CCC3C(C2)CN3C(=O)CCCn2ccnc2)=O)ccc2ncnn2n1 c1(N2CCN(C(c3nc(OCC)oc3)=O)CC2CCO)ncn(C)c(=O)c1Br CCC(CC1CCCCC1)C(=O)NC1CCC1NC(c1cnn(C)c1C)=O C1(C(C)NC(c2cc(CC)no2)=O)CCCN(C(C23CC(C)(C2)C3)=O)C1 Cc1nnccc1C(=O)N(C(C)CNC(c1n[nH]c(C)c1Cl)=O)C c1(NC(=O)NCCC2CC(C)N(C)CC2)cc(C(F)(F)F)ccc1[N+](=O)[O-] CCCCCCC(=O)NC1CCC(CNC(c2conc2C(C)C)=O)C1 c1(CC(=O)NCCN(C)C(C2CCCS2)=O)cccc(C2CCC2)c1 Cc1cc(C(N2CC(C)(CC(=O)NCc3ccnc(Br)c3)C2)=O)nn1C(F)F c1(C(N2CC(F)(C(N(CCCC)CCCC)=O)C2)=O)c[nH]c2cccc(C)c12 C1(NC(C(CCC)C)=O)CCN(C(c2ccc3c(n2)CCOC3)=O)CC(C)(C)C1 C1(NC(C(CC(C)C)O)=O)CC2CCCC(C1)N2C(C1CCC(C(N)=O)O1)=O N1(C(CC(C=C)CC)=O)CC2(C1)CN(C(C1CC3(CC3)C1)=O)CC2CO C1(C)(CNC(C2CC(CC)C2)=O)COCCN(C(=O)CCC(F)(F)F)C1 CC1CC(NC(=O)C2=CCOCC2)CN(C(c2cc(C3CC3)on2)=O)C1 C(=O)(CC(C)(C)CC(=O)OC)NC1CN(C(C(CCC)C)=O)C1 C(C(C)(O)C(=O)NCCCNC(c1ncncc1Cl)=O)OC C1(OCC)CCCC1NC(=O)CONC(c1nc[nH]n1)=O C(=O)(C#CC(C)(C)C)N(C(C)CN(C(=O)CC1CCCCC1O)C)C CC1C(NC(c2cccnc2)=O)CCN1C(c1cccc(-c2ccncc2)c1)=O c1(N2CCN(C(=O)NC(C(=O)OC(C)(C)C)CCF)CC2)cncc2nnnn12 N1(C(C2C3(CCN(C(C4(CC=O)CC4)=O)C3)C2)=O)CC2(CCC2)CC1C.C C1(C(N(C)C)=O)(Cc2ccccc2)CN(CCNC(=O)NC2CN2C)C1 c1(C(=O)OC2CC(OCC)C2(CC)CC)c(C)cccc1C c1(CC)sc(C(=O)NC2CC(NC(c3cnoc3-c3cccs3)=O)C2)cc1C C1(C=O)CC(C2CC2)=NO1.c1(CNC(C2CCCCC2)=O)ccc(F)nc1.C Cc1cccc(C)c1C(N1CCC(C)C(CNC(c2sc(=N)[nH]c2C)=O)C1)=O c1(C(N2CC(NC(c3n[nH]c(CC)c3Cl)=O)C3(C2)CC3)=O)c(F)cc(F)cc1F C1(C(N2CCOCC2c2cn(-c3ncc(Br)s3)nn2)=O)OCC2CCC1C2 C1(CC(C)C)OCCCC1N(C=O)CCCN(c1ccc(Cl)cc1)CC(C)C C(=O)(C(C1CCC1)NC(=O)COC1CCCC1)NCCNC(C)=O O=C(C1=CCC(NC(c2ccc(CO)cc2)=O)C1)NC(Cc1ccco1)CO c1(OC)cccc(C(=O)NCCC(C)(C)CNC(c2cccc(F)c2)=O)c1 C(=O)(CCCCCF)NCC(CC)(C)NC(=O)CC1CC(=O)C1 CCCCCCC(=O)NCC(C)CC(=O)NC(C)CN(C)C(C)C C1(NC(c2nn(CC)c(O)c2)=O)CC(C)CN(C(c2cnoc2C)=O)C1 C1CCC(F)(F)CC1.N1(C(C2CC(SC)C2)=O)CC(NC(=O)CO)C(F)C1 C(=O)(C1CCc2c[nH]nc21)NC1CN(C(c2c(CC)[nH]cc2)=O)CC1(C)C Cc1nc(C(=O)N(CC(C)CNC(=O)CO)C)cn1C(F)F.c1nccn1C c1(-c2nnc(-c3[nH]cc(Br)c3)o2)ccc(-c2ccccc2)cc1 C1(C(CNC(CCC(CC)c2nn[nH]n2)=O)OC)C2CC3CC(C2)CC1C3 C1(OC)CC(CNC(=O)Cn2cccn2)N(C(=O)Cc2ncoc2C)C1 C1(N(C)C(c2ccco2)=O)CCCC(C(=O)NC(C)(C)C)C1 C1(O)CCCN(C(=O)CC2CC23CC3)C1.c1(C(N(C)C)=O)ccc(O)c(F)c1 c1(C(=O)NCCNC(C2CC3(CCC3)C2)=O)cc2c(Cl)c(Cl)ccc2[nH]1.C c1(NC(C2CC23CCN(Cc2cc(Br)cnc2Cl)C3)=O)cnc2[nH]ncc2c1 c1(C(N2CCC(C)C(NC(c3nc(Cl)c(Cl)s3)=O)C2)=O)cccc2c1ccn2C C(CCCCC(=O)NCC1CCCCN1C(c1ncc(OC)nc1OC)=O)OC C12(CCNC(C(C=C)(C)C)=O)CCC1CN(C(c1snnc1C(C)C)=O)C2 c1cc(C(F)(F)F)c(C)cc1Br.C(=O)(CC)CCN(CC)CC.C(C)=O.N C1(NC(CCOC2CN(C(C3C(C(N)=O)C3)=O)C2)=O)CCOC(C2CC2)C1 c1(CC)cnc(Cl)[nH]c1=NCC(c1ccccc1)NC(=O)Cn1nnc(C)n1 C1(NC(c2ccc(Cl)c(I)c2)=O)CCCCN(C(C2CC(O)C2)=O)C1 CN1N=C(C(=O)N2CC(O)(CCNC(c3n[nH]cc3Cl)=O)C2)CCC1=O N1(C(=O)Nc2cccc(CF)c2)CCCCC(C2CCOCC2)C1 C1(C(N(CCNC(C(COC)(C)O)=O)C)=O)CCN(S(=O)(=O)N(C)C)C1 c1(C(N2CC(NC(C34CC(F)C3C4)=O)CC(F)C2)=O)ccc2ccsc2c1 C1(CC)CC(C(=O)N(C2CCN(C(c3ccc4c(c3)CC4)=O)CC2)C)CC(=O)N1 CC1CN(C(=O)CC2CCN(S(=O)(=O)CCc3ccncc3)C2)CCO1 C1(NC(=O)NCC2CCN(C(CC)C)C2)CC2(CNC(=O)N2)C1 C(=O)(C1=CCCC1(C)C)NC(CNC(CCCC(=C)C)=O)(C)C1CCC1 N(C)(C1CS(=O)(=O)c2ccccc21)C(c1ncc(C)cc1Cl)C(=O)NCCCF C(=O)(CS(=O)(=O)C1CC1)N(C1CCN(C(C2CC(=C(F)F)C2)=O)CC1)CC Cc1cccc2c(C(N3CC(NC(=O)C4=CCCS4)CC4(CCC4)C3)=O)cnn12 c1(C(=O)NCC(CNC(C(CCC)OCC)=O)OC)ccc(N)c(SC)c1 C#CCCCC(=O)NC1(COC)CCCNC1 C1(CC=C)(NC(C2(c3ccccn3)CC2)=O)CCN(C(=O)C(C)C#N)C1 c1ccc(Cl)c(F)c1.O=C1CN(C(=O)OCC2CC(O)CN2C(=O)N)CCN1 C(=O)(CCCCCC#N)NCC1CCCCN(C(CCc2onc(CC)n2)=O)C1 c1(C(=O)NC2(CN(C(c3c(C)cnn3C)=O)C)CC2)csc2ccc(F)cc12 c1(C(N2CCC(N(C(c3ocnc3C)=O)CC)C2)=O)ccc(C#N)[nH]1 C1(C(=O)OC(CCOC)C(C)(C)C)COC2COCC2O1 C1(C(=O)NC(C)CN(C)CCSc2nncn2C)CC1C1CCCC1 Cc1nc2c([nH]1)CC(C(=O)NC1CC(C)C(O)C1)CC2.C(=O)C(C)(C)C(C)C Cc1cc(CO)on1.C1(C(=O)O)CC(C(=O)NC(=O)CC2CC(=O)C2)C1 N1(C(C(C)SC(C)C)=O)CC(C(N2CCC2C2CCCC2)=O)C(C)C1 C(=O)(CCC(C(=O)OC(C)(C)C)NC(c1nnc2ccccn12)=O)OC C1(CN(C)C(c2cc(Cl)cnc2O)=O)CCCN(C(C2(n3cnnn3)CC2)=O)CC1 c1(CNC(=O)NCCNC(c2cccs2)=O)cc2cccnc2o1 N1(C(c2cncs2)=O)CC2CN(C(=O)COc3ccc(Cl)c(Cl)c3)C2C1 C1(OC)CN(C(=O)C(C2(O)CN(C(C3CCC(=O)N3)=O)C2)F)C2(CCC2)C1 Cc1cc(CC(c2ccc(Br)cc2F)NC(N2CCOC(=O)C2)=O)cc(C)c1 N1(C(C)=O)CCCCC1C(=O)NC1CCN(C(=O)C(c2ccc(F)cc2)CC)C1 N1(C(c2c(C)nncc2)=O)CCN(C(=O)CCN2CCN(C)CC2)C(C)C1C C#Cc1ccc(NC(=O)CC2CCC(NC(c3ccncc3)=O)CC2)cc1 c1c(Cl)cccc1[N+](=O)[O-].N1(C(C2C(C)C2)=O)CC(NC(=O)C)C1.C(=O)N C(=O)(CCCCCF)NC1CCC(N(C(=O)CNC(C2CCC2)=O)C)CC1 N1(C(c2cc(CNC(C3N(C=O)CCC3)=O)[nH]n2)=O)CCCC2CCCCC12 C1(NC(C2(OC)CCSC2)=O)C=CCN(C(=O)C(Cc2ccccc2)OC)C1 C1(NC(c2cn(C3CCC3)nn2)=O)CC2CC1CN(C(c1c[nH]c(Br)c1)=O)C2 N1(C(C=CCCC)=O)CC2(CC(CNC(=O)C(F)(F)COC)C2)C1 N1(C(CCSCCC)=O)CCCCC12CN(C(C1(C(C)C)COC1)=O)C2 C#Cc1cc(F)ccc1CN1CC(C(=O)Nc2ncc(F)cc2O)CC(F)C1 c1(NCC)ccc(Cl)cc1C(=O)NCC1CC1.C(=O)C=CS(C)(=O)=O N1(C(C(C)(C)n2cccn2)=O)CCCC(CNC(C2CC(C3CC3)C2)=O)C1 C1(CNC(C(C=CCCC)O)=O)COCCN1C(c1cc(C2CC2)on1)=O Cc1cc(F)ccc1-n1nc(CO)nc1C1C2CN(C(=O)OC(C)(C)C)C12 C(=O)(C(F)(CC)C(=O)OC)NC1C(C=C)CN(C(=O)CCc2ccccc2)C1 Cc1nc(Cl)cc(=NCC2C(C)CCCN2C(=O)C(O)C2CCC2)[nH]1 c1(CC)ccc(C(=O)NCCCCC(=O)NC(c2nn(C)cc2O)C)nc1 N1(C(C2(NC(C)=O)CCCCC2)=O)CCC(NC(=O)CCCCN(C)C)C(C)C1 O=C(C#CC1CCCCC1)NC1CC2CC1N(C(c1cc(=O)cc[nH]1)=O)C2 C1(NC(CCC(=O)N(C)C)=O)CC2CC(C1)N(c1cc(C(N)=O)ncn1)C2 Cc1ccccc1NC(=O)CN1CC(N(C(=O)CCc2ccc(Br)nc2)C)C1 C12(C(=O)NC(c3c[nH]ccc3=O)C)CC1CCN2C(=O)CCc1cnoc1 C(C(=O)N1CCCC(NC(c2nccc(C(F)(F)F)n2)=O)C1)(C(C)C)OC C1(=O)C(CC(C)C)O1.c1(CC)cccc(NC(=O)CN2CCN(CC)CC2)c1 N1(C(C(=C)F)=O)CC2CCCC(C1)N2C(c1nn(C)cc1Cl)=O C(CC(=O)Nc1cnn(CC2CC2)c1)(C(F)F)NC(CN1CCC(C)C1)=O N1(C(C(C)O)=O)CCC2(CCC(NC(=O)CC3CC4(CCC4)CO3)CC2)CC1 c1(C(=O)NC(CNC(CCCCC(=O)NC)=O)C)cncc(S(N)(=O)=O)c1 CN=C(NCC1CCCN1S(C)(=O)=O)N1CCCC(S(C)(=O)=O)C1 N1(C(CCOCCC)=O)CCC(C)(CNC(=O)CCn2ccnc2)C1 C1(NC(=O)CCSc2ccccc2F)CC2CCCCN2C1 C1(C(=O)NCC2(OC)CN(C(=O)CC3(C)CC3)C2)CC2CCC1O2 C1(NC(CN(C)CCO)=O)CC2CCC1CN(C(C1CCC3CCC1O3)=O)C2 C(=O)(CC1=CCN(C)CC1)N1C(CN(C(=O)CCNC(=O)CO)C)COCC1 CC1CC(NC(=O)C(C)(C)N(C)C)CN(C(c2cn3ccnc3s2)=O)C1 c1(SC)cnn(C)c1C(=O)NC1CCCCC1.c1(C=O)cnc(C2CC2)o1.C c1(C(=O)NCCC2CC(NC(C(C)N(C)C)=O)C2)ccc(Cl)c(F)c1 S(=O)(=O)(c1ccc(N2CCOCC3(CCC3)C2)nc1)N1C(C(C)O)CCCC1 Cc1cc(F)ccc1C(=O)NCCNC(c1cncn1C)=O C(=O)(C(C)(C)CF)N1CC(CCCCNC(C(=O)NC(C)C)=O)C1 C(=O)(CCC1=CCCCC1)NC(C)CNC(=O)CN1CCn2nccc21 c1(C(C)C)ccc(CC(N2CCC(N3CCC(O)C3)C(C)CC2)=O)cc1[N+](=O)[O-] C1(C(=O)NC(CC=CC)CO)CC(=O)CN1C(c1ccc(C2CC2)cc1)=O Cc1cccc2c1OC(CNC(c1ccnn1-c1nc3ccccc3s1)=O)C2 CC1=C(C(=O)N2CC3CC2(C(=O)Nc2cc(C)cc(C)c2)C3)CCCC1 CC1(C)C(=O)CC1C(N1CCC(NC(=O)C(C2CC2)C2CC2)C1)=O.C c1(NC(N(C)CC2CCOCC2)=O)cn(-c2ccccc2)nc1C(C)(C)C C(=O)(C1=CC2(CCOCC2)C1)NC1CC(C)N(c2ccnc(C#N)n2)CC1 N1(C(c2ncc(C)cn2)=O)CCC(CNC(=O)CC2(O)CCCN(C)C2)C1(C)C N1(C(c2c(CC)occ2)=O)CCOC(CCCNC(c2ccsc2)=O)C1 c1(C(=O)Nc2cnn(C3CC3)c2)cc2c(s1)CCN(Cc1cnc(Br)s1)C2 C(=O)(CC(C)CCC=C(C)C)NC(CCCC)CNC(=O)CCn1cc(Cl)cn1 C12CCC(CC1)CO2.CC(CC1CCC1)C(=O)NC.C(=O)CCC1CC1(F)F C1(NC(CCC(C)N(C)C)=O)CC2CCC1CN2C(C1(C)CSC1)=O C1(CNC(c2cnsn2)=O)COCCN(C(C2(Br)CC23CCC3)=O)C1 C1(CCC)CN(C(C2NC(=O)C3CCC23)=O)CCN1C(=O)Cn1ncn(C)c1=O N1(C(C2(CC)CCOC2)=O)CCOC(C(=O)N)C1.CCN(C(C)C)C(C)C C1(CNC(c2cc(CC)n(C)n2)=O)CN(C(c2n[nH]c(C)c2F)=O)CCC1C C1(NC(c2cccc3nn[nH]c23)=O)COC2(CCN(C(C3(Cl)CC3)=O)CC2)C1 C1(CC=C)(NC(=O)C(F)CC)CCN(C(C2CN(C(N)=O)C2)=O)C1 C1(O)(CNC(=O)CCc2csc(-c3ccco3)n2)CCN(C(=O)C2=CCSC2)C1 N1(C(c2cnccn2)=O)CC(C(N2CCCC2c2ccc(Cl)s2)=O)CC(F)C1 C1(NC(CCc2cc(C)no2)=O)CN(C(C2CCCO2)=O)CC1C CC1(CNC(=O)Cc2cccc(F)c2)CCCN(C(C2C3CCC(=O)C23)=O)C1 C1(NC(C(C)SCC)=O)CCC(C)N(C(=O)CC(C)(C)c2ccccc2)C1 C(=O)(C1CCCc2scnc21)NC1CCN(C(C(CCSC)N(C)C)=O)C1C C=CCCCC(C)NC(C1CCC1CNC(c1ncsc1CC)=O)=O CC(=O)CCC(=O)N1CCC(C(=O)Nc2cn(C)nc2O)O1 C1(NC(CC(CNC(C2CC3CCC3C2)=O)OC)=O)CCCCN(C)C1=O c1(C(N(C(c2ccccc2)C)CC2CC2)=O)cc2cncc(Br)c2s1 C(=O)(CCCCC(C)(C)C)N.c1(CCC)nnsc1C(=O)NC1(C(F)F)CCC1 c1(CNC(C2C(C)CC2)=O)ccsc1C(N1CC=CC1CF)=O N1(C(CC(C)C(F)F)=O)CC(C(=O)NC(C)(C)C(C)(C)CO)CC(C)(C)C1 c1(C(=O)NC2C(SC)CN(C(=O)Cn3cncn3)C2)csc2cncn12 c1(C(C)C)[nH]nc2ncc(C(=O)N=S(C)(=O)CCNC(=O)O)cc12.C(C)(C)C CCCC(C(=O)N(C)Cc1cccc(CNC(=O)CC)c1)C(C)C.C(N)=O.N C1(C(N2CC(CC(C)NC(c3sccc3Cl)=O)C2)=O)OCCC1c1ccccc1 n1(CCCOC)nc(C(=O)N(C)CCNC(C2(C)CC2Br)=O)ccc1=O C(=O)(C1CC(=O)Nc2ncccc21)N1C(C2(NC(CC(C)SC)=O)CC2)CCC1 C1(CNC(C(C)OC)=O)CCN(C(=O)C=CCO)CC1C.c1ccccc1 C1(NC(CN(C)C)=O)CC2(CCC(C)OC2)C1.c1(C(=O)N)cc2n(c1)CCSC2 c1(N(C2CCCN(C(C3(COC)CCC3)=O)C2)C)ncc(C#N)cc1F N1(c2cc(NCC(CC)Oc3ccccc3C)ncn2)CCC(C)C(F)(F)C1 C(c1ccccc1C#N)=CC(N1CCC(O)(C(C)NC(CCC(C)O)=O)C1)=O C(=O)(CCCC(C)(C)NC(=O)Cc1cccnc1)NC(C(C)(C1CC1)OC)C C(C1CCOC1)=CC(N1C(CC(=O)NCCC23CC(CO2)C3)CC1)=O c1(CCN2C(C(O)C(F)(F)F)CCC2)ccc(OCC(F)(F)F)cc1 c1(CC(N2C(CNC(C3CCC(=O)N3)=O)CCCCC2)=O)ccc([N+](=O)[O-])cc1 C=CCC(C(=O)N)NC(C)=O.c1(CC=O)cnn(C(C)C)c1.CC=CC C1(C(=O)NC(CNC(C2CC23CC3)=O)C2CC2)(COC)CCCO1 Cc1nc(N(C(C)CCNC(=O)CSCCN(C)C)C)[nH]c(=N)n1 C1(OC)CC2CCC1CC2C(=O)NCC1(OC)CN(C(c2nocc2Cl)=O)C1 N1(C(C2NC(=O)OCC2)=O)CCN(C(c2cccs2)=O)C(CC(F)(F)F)C1 C1(C(N(C)CCNC(C2C3(CC3)C23CC3)=O)=O)OCC2CCCC1C2 C1(NC(Cc2ccc(C)s2)=O)COC2(C1)CN(CC1CCCO1)C2 C(c1cnccn1)=CC(=O)N(CCCNC(C1CSC(C(F)(F)F)C1)=O)C N1(C(C23OC(C)C(C2)C3)=O)CCC(NC(=O)Cn2cnnn2)CC(C)(C)C1 N1(C(CSCC)=O)CCN(C(c2nc(-c3ccccc3)ncc2Cl)=O)C(CF)C1 CC1CN(C(c2ncccc2N)=O)CC1NC(=O)Cc1ccnc(Br)c1 C1(CCNC(C(C)OCCC=C)=O)CCCCN1C(c1noc(C2CC2)n1)=O C(=O)(CCCCCC#N)N1C(CC(=O)NC(C)C(=O)N(C)C)CC1 Cc1ncc(CCC(=O)NCC(C)(C)OCC)c(O)n1.C(=O)(CC(C)C(C)C)N c1(CC)cc(C(=O)NCCOCC(=O)NCCP(C)(C)=O)n[nH]1 C1(CC(C)C)OCCCC1NC(c1ccccc1NC(N)=O)=O CC1CN(C(=O)CC2CCOC2)CC1C(=O)NOCC1CC1 Nc1ccc(C(=O)NC2(CO)CCCN(C(c3cscn3)=O)C2)nc1Cl C(=O)(C1=NOC(CNC(C2CCC(O)C2)=O)C1)NCC(C(CC)C)C N1(C(C(n2cc(-c3cnsc3)nn2)C)=O)C2CCC1CC(c1ccnn1C)C2 N1(CC2CN(C(C(CC)O)=O)C2)CCN(C(c2cncnc2C2CC2)=O)CC1 N1(C(C(C)CO)=O)CC2CCC1C1CN(C(c3cc4cc(F)ccc4o3)=O)CC21 c1(C(N(CC(C)NC(C2CCCN2C)=O)CC)=O)cc(C)n(C(F)F)n1 C1(NC(C(C)(C)C2CCOCC2)=O)CCc2c[nH]nc2C1 n1(CC(N2CC(C)C(NC(C3C=CCCC3)=O)C2)=O)ccc2cc(Br)ccc12 C(=O)(C1CCc2cccc(O)c21)N1CCC(NC(c2cc(OC)c(C)cc2)=O)C1 C1(NC(=O)OCC(N2CCCCC2)=O)CCC2CN(C(=O)CC)CC12.C(C)=O CCCC(CCCNC(=O)Cc1nocc1C)N=c1[nH]nc(C(C)C)o1 Cc1ncc(S(N)(=O)=O)cc1C(N1CCC(Cc2nn[nH]n2)C1)=O c1(CC)ccc(NC(=O)C(C)N(C(=O)CC2CC(C)(C)CO2)C)c(F)c1 N1(C(c2c(C)scn2)=O)CCC(CCCNC(c2ccc(CCO)cc2)=O)CC1 C(CC(C)C)(C(=O)N=c1cc(C)n(CC=O)[nH]1)NCc1nc(O)cc(CC)n1.O C1(CC(=O)N(C(CCOCCOC)=O)Cc2cccnc2)CCCCCCC1 C1(NC(C(C2CN(C(C(C3CC3)SC)=O)C2)O)=O)CCC(F)(F)C1 N1(C(c2c(SC)scc2)=O)CCN(C(C2CC(=O)NC(C)C2)=O)CCC1C C1(C(=O)NC(c2nc(C)no2)CC)CN(C(c2cccc(Cl)c2)=O)CC1CC C#CC12CC(CN1C(c1cnc(C3CC3)[nH]1)C(=O)NCc1ccccc1C)C2 C1(C(N2CCC(C3COCCO3)CC2)C(=O)NC)CCN(C)C(C)C1 N1(C(c2c(CC)nn(C)c2)=O)CCN(C)CC1.C12(C=O)CC(C(F)F)(C1)C2 C1(NC(C2CCN(C(C3(F)CC=CCC3)=O)C2)=O)C2CCC1CC2 C1(CC#C)(Nc2cc(NCC)ncn2)CCN(C=O)CC1.C(C)(C)(C)O.C c1(C(N2CCN(C(CC(CC)SC)=O)C(C)C2)=O)nn2cccnc2c1Cl C1(C(C)C)(C(=O)N)CNC(=O)C1.C1(CC)CCCC1.C(c1ccoc1)=CC=O CC1(C#CC(=O)NC2CCCN(C(=O)CCCC(F)(F)CO)C2)CCCO1 CC1CCCC(NC(=O)C#CCNC(=O)C(c2cnn(C)c2)=O)C1 N1(C(CN(C)C(N)=O)=O)CCN(C(c2ccc(C#N)[nH]2)=O)C2CCCC2(C)C1 C1(CN(C(C2C(=C)C2)=O)C)CCCN1C(=O)CCCN1CCCC1 C(=O)(C(C)(C)C(F)(F)F)N1C(C)CCC(NC(=O)Cc2csc(=N)[nH]2)C1 C1(OC)CN(C(c2ccc(C3CC3)o2)=O)CC1C(=O)NCCCn1ccnc1C C#Cc1ccc(Cl)c(C(=O)NCC(C(C)C(C)C)NC(=O)C=CCF)c1 O=C(CN=c1[nH]c(-c2ccccn2)cs1)OCc1ccc(Cl)cc1 C1(OC)CN(C(C2(NC(c3ncc(F)cc3C)=O)CSC2)=O)CC12CC2 C1(NC(C(C)CN(C)C)=O)CCC(C)N(C(c2ncccn2)=O)C1 N1(C(C(c2ccccc2F)C)=O)C2CCC1CN(C(=O)CCC#N)CC2 N1(C(c2[nH]cc(CC)c2)=O)CCC2(CCC2)C(CNC(=O)Cn2nccn2)C1 c1(C=O)ccn2ncnc2c1.C(=O)C(C)S(C)(=O)=O.CC1CN(C(=O)C)CC1.N C1(C(N2C(c3ccc(OCC)cc3)CCC2)=O)CC2(CCC2)CCO1 N=c1cc(C(=O)NCC2(F)CCC2)cc[nH]1.c1(C=O)ccc(C(F)(F)F)[nH]1 O=C(CCC1=CCCCC1)NC1CCCC(C(=O)N(CCO)C2CC2)C1 c1(CC)cn2cc(C(=O)NC3CCCC3NC(C3CC3(C)C)=O)cc(F)c2n1 N1(C(c2cc(Cl)cc(C)c2N)=O)CCOC2(CCCN(C(C3(C)CC3)=O)C2)C1 c1(OC(CNC(CCCOCC)=O)(F)F)ccc(F)cc1F N1(C(c2cc(C#N)oc2)=O)CCC2(CC1)CN(C(=O)CCC(F)F)C2 N1(C(=O)NCC2(C(=O)OC)CCC2)CC(F)(C(F)(F)F)C1 N1(C(CCSc2c(C)ccc(C)c2)=O)CCC(C2CN(C(C3CC3C)=O)C2)CC1 C#CCCCCCC(=O)NC(C)(CNC(c1nc(O)nc(O)c1F)=O)CC C1(C(N2CC(C(C)C)C2)=O)CCC(CNC(=O)CC(C)n2cccc2)O1 C1(C(C)C)CN(C(=O)C(O)CC2CCC2)CCN1C(=O)CC1C=CCC1 N1(C(C(CC)c2ccccc2)=O)CCN(C(C2CCS(=O)(=O)C2)=O)CC1 CCC(CC(C)C)C(=O)NCC1C2CN(C(=O)C(C)c3ccco3)CC12 CC(C(=O)NCC1(F)CN(C(c2c(C(F)(F)F)cnn2C)=O)C1)C(C)O C1CN(C(=O)C=C2CCOCC2)CC2(CC2)C1.c1(C=O)nn[nH]c1C(F)(F)F c1ccc(C#N)cc1.N1(C(C)=O)CCN(C(=O)C(C)O)CC1.C=CCC(C)NCC C(CCN(C)C(C1CC(=O)N1)=O)(C(C)C)NC(c1cc(OC)n[nH]1)=O c12ccncc1S(=O)(=O)NC2C.CCCCCC(O)CN.C(=O)N(C)C C#Cc1ccc(CC(N2CC(N(C(=O)C=Cc3ccco3)C)C3(CC3)C2)=O)cc1 N1(C(C=CSC)=O)CCC2(NC(c3ccnc(C4CC4)c3)=O)CC2C1 c1(C(=O)NCC2(COC)CN(C(C3(C)CC3)=O)C2)snc(OC)c1Br N1(C(c2cc(C)n(C)n2)=O)CCCCC(C(N2CCSC(C)(C)C2)=O)C1 CC(C)CC(C(=O)NCC1(C)CCC1)C(N)=O.C1(CC(=O)N)CCOC1=O CC(CC(N)=O)C(=O)N1CCC(C)(NC(c2cc(O)nc(C3CC3)n2)=O)CC1 c1(C(N(CC(CNC(C(F)=CCC)=O)C)C)=O)cnc(N(C)C)s1 c1(CC)nnc(C)cc1C(N1CC(NC(=O)CCNC(N)=O)C(F)C1)=O Cc1nc(C(=O)N(C)CC2CN(C(C3COC4COCC34)=O)C2)c(=O)[nH]c1C CCC(CC(=O)NCc1cc(C)c(C)o1)NC(=O)C(C)Cn1cccn1 c1(OC)cc(N)c(C(=O)NC(C)(C)CCC)cc1F.N1(CC=O)CCCC1=O.N C1(NC(CNC(C)=O)=O)C(C)CCC12CCC2.n1(CCCC=O)nc(C)cc1C c1(CS(N2CCC(OCCCCCc3ccccc3)C2)(=O)=O)ncsc1Br N1(C(C(F)=C)=O)CCC(C)(NC(=O)C(c2ccc(F)cc2)C)C1.CCI c1(N2C(C3CCN(C(C45CC(F)(C4)C5)=O)C3)CCC2)ccc2c(n1)CCC2=O.C C1(NC(C(C)CNC(c2cnncc2O)=O)=O)CCN(C)CC1C N1(C(c2c(C)cco2)=O)CCN(C(=O)CN(C)C(=O)N)CC1.C1CNC(=O)N1C C1(C(=O)NCCCN(C(c2cnc3[nH]cnc3c2)=O)CC)CCn2nnnc2C1 N1(C(c2csc(O)n2)=O)CC2(C1)CN(C(C1CC3(CCO1)CC3)=O)CC2CO c1(NCC(C)C(C)O)ccc(S(=O)(=O)N2CCC3(CCS(=O)(=O)C3)C2)cc1C#N O(NC(=O)C1(NC(=O)C=CCC2(N3CCCC3)CC2)CC1C)CC(=C)Cl C1(C(=O)N)CCC2(CN(CC(=O)N)C2)O1.C1(C(=O)NC)CCC1.C1CC1 N1(C(C(C)(N(C)C(c2cnn(C(F)F)c2)=O)C2CC2)=O)CCC12CC(CO)C2 N1(C(CCN(CCC)C)=O)CCC2(CC1)CCN(c1nc(CC)cc(C)n1)CC2 C1(CC)CCCN(C(C2CC2CCOC)=O)C1C(=O)NCc1ocnc1C C1(C2CC2)(C(N(C)CC2(O)CCOC2)=O)CN(C(c2cccc(=O)o2)=O)C1 C(=O)(CCCCCN(C)C)N(C)CC1C2CN(C(Cn3c(C)ccc3C)=O)CC21 C1(CNC(C(CC)(C)F)=O)CCCN(C(c2ccnc(N(C)C)c2)=O)CC1 N1(C(c2cc(N(C)C)nc(Cl)c2)=O)CCN(C(=O)CCN2CCC2)C2COCC12 c1(C(=O)NCC(CC(N2C(C)CC3(CC3)C2)=O)OC)cccn2cncc12 c1(C=O)cc(O)nc(O)n1.c1(OC)csc(C(=O)NCC2(F)CCC2)c1.C c1(C(N(CCN(C(C2OCCOC2C)=O)CC)CC)=O)cc2cc(Cl)cnc2[nH]1 c1(C(=O)NCC(C)(C)NC(c2cc(C)no2)=O)ccc([N+](=O)[O-])cc1 c1(C(=O)NC(C2CCOC2)CNC(C(F)=CC)=O)cc2c(Cl)ccnc2s1 C12(C(=O)NCC(CNC(C(C)(O)C3CC3)=O)O)CCC(C(F)F)(CC1)C2 C1(C(=O)NCC(C)CCO)CC12CCN(C(=O)Cc1cnsc1)CC2 c1(CNC(CCS(C)=O)=O)nnc2n1CCN(C(=O)C1=C(Cl)CCC1)C2 CC1(CNC(c2cnnc(O)c2)=O)CN(C(C2(C)CSC2)=O)CCO1 n1(CC(N2CCCC2)=O)c(O)nc2ccccc12.O=C1NC(C(=O)NC)C2CC12 CCCCC(C)C(=O)NC(C(=O)NCCCOCC(C)C)c1cccs1 c1(C(CC(=O)NC2CCC(NC(c3n(C)nnc3)=O)CC2)O)cc(Cl)cc(Cl)c1 CCCCCC(O)C(=O)N1CC(=O)NC(CNC(=O)CSCC)C1 C(=O)(C(C)(CC)C(=O)NC1COCC1)OCC.c1(C=O)cnc2[nH]ncc2c1.N N1(C(c2ccc(-c3cn(CC(CC)O)nn3)cc2)=O)CCC(C)=C(Br)C1 C(=O)(CC(C)(C)C(F)(F)F)NC(CN(C(c1cc2nn[nH]c2cc1F)=O)CC)C C(=O)(CCCC(C)CC)N1C(C(=O)NCC(CC)(C)C)C(C)CC1 C=C(Cl)CC(C(=O)NC(C1CCOC1)CO)NC(c1sccc1C#N)=O CCC(CC(=O)NC1CC1NC(=O)CCc1cc(C)cs1)OC O(NC(=O)CC1(NC(=O)CC2CC=CCC2)CCC1)C(C)(C)C n1(C(C)C)cc(C(=O)N(CCC#N)CC2CC2)ccc1=O Cc1ccc(C)c(NC(=O)C2=CCC(NC(C3(C#N)CC(=O)C3)=O)C2)c1 C12(NC(c3cnn(C)c3Br)=O)CCOC(CNC(C3CCC3)=O)(C1)C2 c1(C(N2CCC(C)C2CNC(=O)CCc2ncc[nH]2)=O)ncc(F)cc1F C(C(F)(F)C(C)(C)C)NC(=O)Nc1ccc(-c2n(C)cnn2)cn1 CC(CNC(C1CC(F)(F)C1)=O)CC(=O)NOCC(N)=O c1(CSC)ccc(C(=O)NC)cc1.C1CN(C(c2nc(C)c(C)[nH]2)=O)CC1C c1(C(C2CCSC2)CCNCCCCn2cncn2)nnnn1C1CCCC1 c1(C(C(=O)NCCC)N(C(c2ccc(Cl)cc2)CC)C)c(C)ncn1C c1(C(=O)Nc2c(SCC(C)C#N)cccc2)ccc(=O)n2c1COCC2 N1(C(CN2C(C)CC2)=O)CCN(C(=O)CCc2cnccn2)C(c2cn[nH]c2)C1 c1(C(N(CCNC(c2cocc2C)=O)CC)=O)c(S(N)(=O)=O)ncn1C C1(NC(c2ccccc2O)=O)CCN(Cc2cc(Br)ccc2F)CC1F Brc1cc(NCc2c[nH]nc2-c2ccc(Br)cc2)cc2cn[nH]c12 c1(CC(=O)N(C2CCCC2)CCNC(CCCC2C(C)C2)=O)cncc(Br)c1 N1(C(CN(CC(C)(C)C)C(C)=O)=O)CCOC(c2cn(CCCO)nn2)C1 Cc1cc(C(=O)NC2CCC(C)N(C(c3cccn(O)c3=O)=O)C2)c(O)nc1C N1(C(CC=CCC)=O)CC(F)(F)CC1C(=O)NCc1ccc(F)cc1Br N1(C(c2c(C)n[nH]c2)=O)CCCC(CCNC(c2ncnc(C)c2C)=O)CC1 CC(C)(O)C(F)C(=O)N1CCOCC1CNC(N)=O Cc1noc(C(F)(F)F)c1C(N1CC(NC(C2CCCC(=O)N2)=O)C(O)C1)=O C(=O)(CC(C)(C)n1cc(-c2ccc(F)cc2)nn1)NCc1ccn(C)n1 CC1CN(C(=O)CNS(=O)(=O)C2CC2)CC1CNC(c1cccnc1)=O c1(C(C)C)ccc(C(N2CC(CNC(N)=O)C(C)C2)=O)c(O)n1 N1(C(CC2(C)CCC2)=O)CCCC2(CCN(C(=O)C(C)(O)C(F)(F)F)CC2)C1 C1CC2CC1CC21CC1.c1(CNC(=O)CC2CC3CC3C2)ccc(C(=O)N)nc1 C(CCCCN(C)C(C1CCN(CC(F)(F)F)C1)=O)NC(C=C(C)C1CC1)=O CCCC(CCC)C(=O)NCC1(C)CCCN(C(=O)C(CC)C(F)(F)F)C1 N1(C(C(CC)(C)C)=O)CC2CN(C(=O)CC3CCN(OC)CC3)CC(C1)O2 C(C1c2ccsc2CCN1C(=O)CC1(C)CC(F)(F)C1)NC(CCN(C)CC)=O c1(N(CCOC)C)nc(N2CCC3(CCN(C)C3=O)C2)nc2c1CCCCCC2 c1(C(=O)Nc2ccc(OC)cn2)cc2c(-c3ccc(N(C)C)nc3)cncc2s1 Cc1cc(CC(=O)NC2CN(C(C3CCOC3c3ccncc3)=O)C2)c(C)s1 n1(CCOC)nccc1C(=O)NCCCN(C)Cc1ccc(Br)s1 CN1CCOC(C(N2CCC(CO)(NC(=O)C3=CCOC3)CC2)=O)C1=O C1(C(=O)NCC(C2(O)CN(C(C3C(C)=CCS3)=O)C2)(C)C)Cc2nccn2C1 c1(C=O)nn(C)c(C)c1[N+](=O)[O-].c1(NC)cncc(C(=O)NCC(C)(O)C)c1 Cc1ncc(C(=O)N(CC(O)CN(CC(=O)NCC(C)(C)C)C)C)c(C)n1 C(=O)(CCC(=O)N1CCC(NC(=O)Cc2nc(C)sc2Br)C1)NC N1(C(c2cn(C(C)C)nc2)=O)CC2CCCCN2CC1CNC(=O)C(F)(F)CO N1(C(C=Cc2cccc(OC(C)C)c2)=O)CC(N=c2cc(Cl)c(O)n[nH]2)CC1C Cc1ccc(-n2cc(-c3c(Cl)cccc3Cl)nn2)c(F)c1Br CC(C)CC(C(=O)N1CC2CC2C1C(=O)NC1CCOCC1F)C(C)C C(=O)(C(=O)CC(C)CC)N1CC(CC(=O)NC2CC(C#C)C2)C(C)C1 Cc1cc(NNC(=O)C(C)n2ccc(C3CC3)n2)ncc1Br N1(C(C(C)(C)N(C)C)=O)CCN(C(C23CCCN(CC2)S3(=O)=O)=O)CC(C)(F)C1 c1(C(=O)NCC(CC)NC(=O)C(C)C(F)(F)F)cc(OC)cc(C)c1 c1(C(=O)NC2C(C)(C)C(C)C2)cc(=O)cc(Cl)[nH]1.c1(C=O)ccc(O)nc1Cl c1(CNC(=O)N(C2CCCO2)Cc2ccc(Cl)cn2)cccc(F)c1 c1(C(=O)NCC(O)CNC(C2CC(F)C2)=O)cccc2c1CCC2 N1(CCC)C(=O)NC2(CCc3c(C(F)(F)F)cccc32)C1=O CC(C)C(C)CC(=O)N1CC(CC(N2CCC3(CC3)C2)=O)CC1(C)C C1(CNC(C(C)OCCC=C)=O)CC2(CC2)CN1C(=O)Cc1ccoc1C Cc1c[nH]c(C(=O)NCC(c2ccccc2)NC(C2(c3ccnn3C)CC2)=O)c1 C(=O)(CC(CC)OC)NC(C(=O)NC1(C#C)CC1)C1(O)CCC1 N1(C(c2cnns2)=O)CCN(C(=O)Cc2cc(O)nc(O)n2)C(CO)C1 N1(C(=O)CC2CC2)CCCC(C(N2CCC(c3ncc[nH]3)C2)=O)C1 C(=O)C1=CCC(C)CC1.c1(NCC(C)C)ncccc1C(=O)N.CCC1CC1 c1(-c2c(CNC)cccc2)ccc2cc(C(N3CCC(C)(O)C3)=O)[nH]c2n1 NS(=O)(=O)c1c[nH]c(C(N2CCOCC(F)(CNC(C3(F)CC3)=O)C2)=O)c1 C1(NC(C2C3N(C(Cc4c(C)n(C)cn4)=O)C(CC3)C2)=O)CCOC2(CCC2)C1 O=C1NC2CCN(C(=O)C(=O)NC3CC4CNCC34)CC2O1 C1(CNC(C2CC(=C)C2)=O)COCC1.c1(C=O)cc(-c2ccn(C)n2)on1.N C(=O)(C1CCCc2c[nH]nc21)NC(CC)CN(C)C(c1ncc2[nH]ncc2n1)=O c1(OCC(N2CCC(CNC(CCC3C(C)C3)=O)CC2)=O)ccc(Cl)c(Cl)c1 C1(NC(C(C2CC2)OC)=O)CN(C(c2ccn(-c3cccc(Cl)c3)n2)=O)CC1C C=CCC(CC)C(=O)NCCCCC(=O)NC(C12CCC(CO1)C2)C c1(C(N(CCNC(=O)CCn2ccnc2)Cc2ccccc2)=O)cncc(F)c1 C(N(C)N1CC2(CCN2S(C)(=O)=O)C1)c1cccc(C(=O)NC)c1 C(=O)(C(F)CC(C)C)N(CCNC(C(CC)Cc1cccc(Br)c1)=O)CC c1(OC)ccc(C=CC(=O)NC2CCN(C(=O)CCCC(F)F)CC2F)cc1 C1(CC(=O)NC2CN(C(=O)CCCCN3CCCC3)CC2F)NC(=O)NC1=O CCC(CC)CCCC(=O)NCCNC(c1cnc(N2CCOCC2)nc1)=O C1(N(C(C(C)=CC)=O)C)CCN(C(=O)Cn2ccnn2)C1 c1(C(CC(C)C)NC(C2(CC(C)C)CCC2)=O)cccc(C(F)(F)F)c1 S(=O)(=O)(c1[nH]c(=NC(CO)c2ccccc2)ccc1Br)NCC1(S(C)=O)CC1 CC1(C)CCOC(C(=O)NCCCN(C)CCOc2ccccc2)C1 CCC(C)C(O)CC(=O)N1CCCCC1CNC(C12CCC(CC1)O2)=O c1(C(N(CCC(=O)NC(COC)COC)C2CCC2)=O)cc(O)nc(O)n1 O=C(C1=C2CCCN=C2NN1)NCC(F)CNC(c1ccc2nccn2n1)=O C1CCCCC1.c1(C=O)c(C)coc1C(C)(C)C.C(C)(C(=O)N)OCCC#C C(=O)(C1CCCc2ncnn21)NCC1C(C)CCCN1C(c1ccns1)=O c1(C(c2n(CCC)nnn2)NCc2nc(C)c(C)o2)cc(Cl)nc(Cl)c1 C#CC1(C(N2CCC3(CC2)N=N3)=O)CCN(C(=O)C(C)OCC(C)C)C1 C1(CC)CN(C(=O)CNC(=O)C(F)(F)F)CCC1NC(C1CC1F)=O c1(C=O)cc(Cl)ccc1C(C)C.C1(C(N(CCC)CC)=O)CCC(=O)N1C.N CC1CN(C(=O)OC(C)(C)C)CC(C(=O)N)O1.c1(CC)cccc(C(F)F)c1 C1(C)(NC(CCN(C)CC)=O)CCN(C(=O)C(c2cc(F)cc(F)c2)O)CC1 C#Cc1cn(C)nc1C(=O)N(CC(O)CNC(=O)CSCCCC)C c1(CC)ccc(CCC(=O)N(CC(C)N(C)C(C2CCCSC2)=O)C)cc1 N1(C(=O)Cc2cccnc2)CCN(C(=O)COc2cccc(F)c2F)C(C2CC2)C1 C1(CC(=O)NCCN(C(Cn2c(C(C)C)ncc2)=O)C)CCCN(C)C1 C1(N(C(=O)C(C)C2CC2)CCCC)CCN(C(=O)CC2CS(=O)(=O)C2)CC1 N1(C(=O)NC2(COC(C)(C)C)CC2)CCc2cnoc2C1 c1(C(=O)NCC(CCCC)NC(=O)C(C)CCOC)cc2sc(=O)n(C)c2s1 CC1CC2CN(C(=O)COCCCF)CC2N1C(c1ccc(Cl)c(O)c1)=O N1(C(C(C2CN(C(CN(C(=O)OC)C)=O)C2)O)=O)Cc2cc(O)nnc2C1 C(CN=C(NCC1CCCSCC1)NC1CC2CCC1O2)OC C1(CCC)(NC(C2C(CCC)C2)=O)CCN(C(=O)C(c2cnn(C)c2)O)CC1 c1(C(N(CC(C)NC(C23CC(F)C2C3)=O)CC)=O)onc2c1CCCC2 CC1=C(C(=O)NCC2CC3(CO2)CN(c2cc(=O)n(C)c(=O)n2C)C3)CCCC1 C12(NC(c3ccccc3)=O)CCCC1CN(C(c1cnc3[nH]ncc3c1)=O)C2 c1(NC(C2N(Cc3cnc(N(C)C)nc3)CCSC2)=O)ccc(I)cc1I C(=O)(C(=O)N=c1cc(C)o[nH]1)N(CCNC(CCC)=O)CCOCCO CCCC(CNC(c1cnc(C)cn1)=O)C(=O)NCC1(n2nccn2)CC1 C(=O)(CC(C)C(=O)N)OC.c1(C(N2CCC2)=O)ccccc1CCC(F)(F)F.C c1(C(N2CCC(NC(C(C)(C)c3cccs3)=O)C2)=O)cccc2nn[nH]c12 N1(c2snc(C(=O)OC)n2)CCN(C(=O)C2CC2)CC1 C1(OC)CC(CNC(=O)C(C)N(C(=O)C(C)NC(N)=O)C)C1 N1(C(C(C(C)C)S)=O)CC2COCC(C1)N2C(c1ccccc1Cl)=O N1(Cc2cccc(N(C)C)c2)CC2(CC(NC(c3cccc(O)c3F)=O)C2)C1 Cc1ccc2c(c1)C(Nc1ccc(S(=O)(=O)N3CSCC3C)cc1Br)CO2 CC(C)C(CC1CCCC1)C=O.c1(C(N(CC)CCC)=O)cocc1C(N)=O CC1(C#CC(=O)OCC(c2ccc([N+](=O)[O-])cc2)=O)CCCO1 C1(C(N2CCCCC2)=O)C2C3CCC(C3)C12.C(C(=O)NCC)N(CC)CC C1(CCC)C(C)CCCN1C(c1ccc(C2CCCC2)cc1)C(=O)NC1(C)CC1 C1(CC)CCN(C(=O)C2=NNC(C(F)(F)F)C2)CC1.C(=O)CN(C)C(C)=O Cc1cc(C(C)S(=O)(=O)N(CC(c2ccccc2)C)CCO)cc(C)c1 C#Cc1ccc(C(N2CC(C(=O)Nc3cc(O)cc(F)c3)CC2(C)C)=O)cc1 N1(CCNC(CCOCC)=O)CCN(C(=O)CC(C)(C)C2CC2)CC12CCC2 c1(C(N(C2CCN(C(c3c(C)noc3C)=O)C2)C)=O)cc2c(cc1N)CCCC2 c1(C(N2CCSC(CC)C2)C(=O)NCC(=C)C)cccc(COC)c1 N1(C(CC2(N(C)C)CCC2)=O)CC(NC(=O)C=Cc2ccnn2C)C(C)(C)C1 c1(N(C(C2CCC2)C)C)nnc(-c2cccnn2)n1CC1CCOC1 c1(C(=O)NC2CC(F)(CNC(C(C)C(F)F)=O)C2)cncc(C#N)c1 N1(C(CCCn2c(C)ncc2)=O)CCC(C(C)NC(C23CC2CNC3=O)=O)CC1 c1(CC)[nH]c(Cl)nc(=NC2CS(=O)(=O)CC2NC(C2C3COCC23)=O)c1C c1(CN2CC(C(N3CC(C)(CO)C(O)CC3)=O)C2)ccc2cccc(Br)c2n1 C12(NC(Cc3n(C(C)C)cnn3)=O)CCCC1N(C(C1CCC1)=O)CCC2 C1(C(N(CCN(C(=O)CC2OCCC2C)C(C)C)C)=O)CC12CCC2 C1(C(N(CC(C)(C)NC(C(N2CCOC2=O)C)=O)C)=O)CCCN(C)C1 C1(C(=O)NC2C(OC)CC2)(NC(C2(C)CC2C(=O)OC)=O)CSC1 c1(C(=O)OC)cc(NC(C2CCCN2Cc2ccc(Cl)nn2)=O)ccn1 S(=O)(=O)(c1nc(N2CCCCC(CO)C2)ccc1Br)N1C(CCC)CCCC1 C1(CC=O)CC(C)(C)OC(C)(C)C1.CC(C)(C)CC(=O)NCC1CCC1.N C1(C(=O)NCCCC(C)NC(c2cnccc2C(F)(F)F)=O)C2CCCOC12 N1(C(c2ccccc2Cn2cc(COCCO)nn2)=O)CC(=O)N2CCCC2C1 Cc1cc(C(N2CCOCC2CN(C)C(c2cc[n+]([O-])cc2)=O)=O)nn1C c1(-n2c(C3CCCN3C(C)=O)nc(CC(CC)C)n2)nc2ccccc2[nH]1 C1(NC(C2(C#C)CCOCC2)=O)COC2(C1)CN(C(C1(CO)CCC1)=O)C2 C(=O)(C1=CC2CCC(C1)C2)N1CCC(C(C(=O)NC(CCC)(C)CC)C)CC1 c1(C(=O)NCC2C(NC(c3nc(C)oc3C)=O)C2)ccc(Cl)c(Cl)c1N N1(C(c2cnc(N(C)C)o2)=O)C2COCC1CN(C(C1(F)CCCC=C1F)=O)C2 c1(N(CCC)CCNC(C2CC2c2ccccc2)=O)nc(Cl)nc2c1SCC2 C1(C(=O)NCC(C)(C)OC)(CC)CCN(C(=O)C(C(C)C)OC)C1 Cc1cc(C(=O)NCCN(C(=O)CCCc2ccccn2)C)c(C)n1NC(N)=O N1(C(C(C)(C)C(F)F)=O)CC2CC(C(=O)NCC3CC34CCC4)CC2C1 C(=O)(CC(C)(C)CC(F)(F)F)NC(C(C)NC(Cn1nc(C)c(C)c1C)=O)C Cc1cc(C(=O)NCC(C)NC(C2COC(C)(C)C2)=O)ccc1[N+](=O)[O-] c1(CN=c2scc(C(N(CCO)CC)=O)[nH]2)cc2ccccc2cn1 O=C1NC2CN(N3CCC(c4nc5ccccc5[nH]4)C3)CC2CO1 c12cccc(n1)-c1cn-2nn1.c1(CC(=O)NCC2(C)CCCO2)ccc(O)cn1 C1(C(=O)NCC(CC=C)NC(c2ccc(C)s2)=O)CC(=O)N(CCC)C1.C c1(CN2CC(C(=O)Nc3c(C)ncc(C)n3)C(O)CC2)c(F)cc(Br)cc1Br N1(C(C2CN(C)CC(C)O2)=O)CC2CC(C1)CN(C(=O)C(O)C1CC1)C2 C1(NC(C(COC)C)=O)CN(C(=O)C(C)(C)OC(C)=O)CC1O N1(C(CC2CCN(C(Cc3c(C)ccnc3)=O)C2)=O)CC2(C1)CC2(F)F C1(NC(c2sc(Cl)cc2Cl)=O)CCCN(C(c2ccc(O)nc2Cl)=O)CC1 c1(C(=O)NCC(C)=CC(=O)NCC(F)Cl)cscn1 O=C(C1=CSCCO1)NCC1CCN(C(c2cn(-c3ccccc3)nn2)=O)CC1 c1(CCNC(c2cn(CCOC)nn2)=O)ccc(OC)c(O)c1 N1(C(C(c2ccccc2F)C)=O)CCCCC1CNC(C1SCCCS1)=O C(=O)(C(CC(F)F)N(C)C(C1CC(N=[N+]=[N-])C1)=O)NC(C)C(=O)NC1CC1 c1(C(N(C(C)CN(C(=O)C=Cc2cscn2)C)C)=O)n[nH]c2c1COC2 Cc1coc(C(=O)N(CCC(C)NC(=O)CSCC2CCCO2)C)c1 C1(NC(C2C(OC)CN(C(=O)CC3CCCCC3)C2)=O)CC2(CCCC2)C1 c1(OC)ncc(C(=O)NC2CCCC(N(C)C(c3coc(C)c3)=O)C2)cc1F c1(-n2c(CCCCC(=C)C)nc(C3CC3)n2)ccc(F)c(Cl)c1 Cc1ccc(F)cc1CN(CCO)C(=O)NCc1ccc(Cl)nc1 C12(NC(c3c(CC)cc(Cl)cc3)=O)CCCC1N(C(=O)Cc1cc(C)no1)CC2 N1(C(CNC(=O)CC2CCC(C(F)F)CC2)=O)CCN(C(c2ccon2)=O)CC1 C(C1=NOC2CCCC12)NC(C1(NC(C=CC(C)C)=O)CC(F)C1)=O c1(OC)ccccc1C=CC(=O)NCCNC(c1cc(-n2cccn2)ccn1)=O C1(NC(c2n(C=C)ncc2)=O)COC2(CCCN(C(c3ncc(C)cc3F)=O)C2)C1 C1(SC)CCN(C(C2(CNC(=O)C=CC=O)CCCC2)=O)CC1.C1CC1 C(=O)(CC(C(F)(F)F)O)NC1C(C=C)CN(C(=O)COCC2CCCC2)C1 N1(C(c2cc(OC)n(C)n2)=O)C(C)CN(C(=O)C(C)CC(F)F)CC1C C(=O)(CCCC(F)(F)F)NC1CC(C)N(C(c2cnc3occc3c2)=O)C1 N1(C(c2c(C)oc(C3CC3)n2)=O)CCN(C(=O)CSc2n[nH]c(=N)s2)CC1.C N1(C(C2CC(CC)NC(=O)C2)=O)CCN(C(c2ncccc2F)=O)CC(CO)C1 c1(-c2ccc(NC(C3CC(C)OC(C)C3)=O)c(Cl)c2)nc2ccccc2[nH]1 CCCCC(CC)CC(=O)NCC1CC1NC(c1cc(C#N)ccc1N)=O C(CCC(O)C(=O)N1CC(C(C)(C)O)C1)NC(COC1CCCC(C)C1)=O c1(C(=O)OC)cc(NC(c2cnn(-c3ccc(Cl)cc3)c2)=O)c(N)c(Br)c1 c1(C(=O)NC2CC(NC(c3cn(CC)nn3)=O)C2)cc2c(nn1)CCOC2 C1(C(=O)NCC(C(=O)N(CC(=O)OC)C)O)CC2CCCC2C1 N1(C(c2c(C(=O)OC)nn(C)c2)=O)CCN(Cc2ccc(F)cc2)C(=O)C1 Cn1cc(SCCc2cn(CCCCNC(=O)CC3CCC3(F)F)nn2)cn1 C(=O)(C1=C2CCN=C2NC=C1)N.C1(C)(CNC(COCCC#C)=O)CCC1 N1(C(N2CCC(n3c(C(=O)OC)ncn3)C2)=O)CCOC(C)(c2ccccc2)C1 c1(OCC)oc(C)nc1C(N1CCC(F)(CNC(c2cn[nH]c2)=O)C1)=O C1(CC#C)(C(=O)N(C)Cc2nc[nH]n2)CCN(C(=O)CSC)C1 N1(CC(CCCCC)=O)CCOCC1C1CCCO1 C1(CC=C)(C(=O)N(C)CCOCCCO)CCN(C(c2cncnc2)=O)C1 N1(C(C2C(CC)CCO2)=O)C2CCC(C(=O)NCCc3ncnn3C)C1CC2 C1(C2CN(C(C3CCCN3N=O)=O)C2)(NC(c2ccc(C(C)(C)C)nc2)=O)CC1 N1(C(C(CCCC)F)=O)CC(C(=O)NC(C)C(=O)N(C)CC)C2(CCC2)C1 Cn1cc2c(n1)CCCC2C(=O)NCCCNC(C12CC3CC1C2C3O)=O CCCCCC(C)CC(=O)N1CCCC(O)(CCNC(=O)Cn2cnnn2)C1 C1(CCNC(C2(C)CC2)=O)CN(C(=O)CC23CCCC2C3)CCO1 c1(C(=O)NCC(CN(C(=O)Cc2csc(-c3ccsc3)n2)C)O)ccncc1O c1(C(=O)NC2(CC=C)CN(C(=O)CCN(C)C(C)=O)C2)nc(C)oc1C Cc1sc(C(N2CC3OCCN(C(C4CCC(C)C4)=O)C3C2)=O)cc1S(N)(=O)=O C(C(CO)CC(C)C)NC(C(CC)N(C(=O)COc1ccn(C)n1)C)=O n1(C(CC)CC)ncc(C(=O)NC2(C)CN(C(c3ccn(C)c3)=O)C2)c1C C1(CC(=O)NC(C(C)NC(Cc2cnc(C)[nH]2)=O)(C)C)CC(C)(C)OC1=O Cc1cnncc1C(=O)NC1(c2ccccc2)CCN(C(C2C(C)C2(F)F)=O)C1 N1(C(CN2CC(=O)N(C)C2=O)=O)CCN(C(C2CC2C2CCC2)=O)CC12CCC2 c1(C(N2CCCC2)=O)cc(C)c(C)c(F)c1.c1(CC)cc(C(=O)N(C)C)nn1C N1(C(C(CC)n2ccc(C3CC3)n2)=O)CCN(C(C2(CCF)CC2)=O)CC1C CCC(C)(CNC(C1CC1(C)C)=O)C(=O)NCC(Cl)Cl Cc1ccc(NC(=O)Nc2cccn3ncnc23)cc1-c1ncco1 c1(C(N(CC(C)NC(=O)C#CC(C)(C)O)CC)=O)cnc2ccccc2n1 N1(C(C2C3(CCN(C(C(=Cc4ccco4)C)=O)C3)C2)=O)CC2(CCOC2=O)C1 N1(C(c2cc(CSC)on2)=O)CCC(O)(CN(C)C(C2CCCCS2)=O)C1 C1(C(=O)NCCc2onc(CC)n2)(CF)CCN(C(c2csc(C)c2)=O)C1 c1(CC(c2ccc(C(=O)NC(CCOC)(C)C)cc2)=O)c[nH]c2cccc(Cl)c12 Cc1nccc(=NCC2CCCCC2NC(C2(CCc3ccccc3)CC2)=O)[nH]1 c1(CCNC(C(=O)NCC2(OC)CCCCC2)=O)c[nH]c2nccc(C)c12 N1(C(CN(C(C)C)C)=O)CC(O)CC1(C)C(=O)N(C)CCn1ccnc1 c1(C(=O)OCC)cccc(CC(=O)OC(c2csc(CC(C)C)n2)C)c1 C(=O)(C1CCCCc2ccccc21)N1CCC(NC(CC2(OC)CC2)=O)C12CC2 c1(OC)cnccc1C(=O)NC1CC(CO)N(C(c2ccccc2O)=O)C1 c1(CC)csc(C(N2CC(OCCNC(=O)C(c3ccn(C)n3)C)C2)=O)c1 c1cccc(Cl)c1.C1(CC)CCCC1C(=O)N.c1(C(NCC)=O)cn(C)cn1 C(=O)(CCC1=NNC(=O)CC1)N1CCC(N(C(C2(C)CCC(O)CC2)=O)CC)C1 C1(CC=C)(NC(c2cc(CCO)on2)=O)CCN(C(c2sc(OC)nc2Cl)=O)C1 C(=O)(C(CNC(c1nc(Cl)oc1C)=O)C(C)C)N(CC(C)N(C(C)=O)C)C C1(NC(c2cn(CC(F)F)cn2)=O)CN(C(=O)CCc2ccco2)CC1C1CC1 N1(C(C2C(NC(c3ccc(-c4ccccc4)s3)=O)C2)=O)CCCC(O)C1 Cc1cc2[nH]c(C(=O)NCC34CN(C(c5ccccn5)=O)CC(F)(C3)C4)cc2o1 Cc1cccn2cc(C(=O)NCC3CN(C(=O)C(F)C(F)(F)F)CCO3)nc12 c1(N(C(=O)NC2CN(C)CC2(F)F)CCO)ccc2c(c1)CCC2=O C#CCCCC(C)C(=O)N(C)CC=CC(N1CCC(CO)(OC)C1)=O CC(C)(CC(F)F)C(=O)NC12CCC(CC1F)C2.C12CCN(C1)CCCNC2=O N1(c2nnc(CCC)s2)CC2CC1(CNC(C1C(c3ccccc3)C1C)=O)C2 c1(CNc2ccc(-c3cc(CO)ncc3)cc2)cc(=N)[nH]c2ccc(Br)cc12 c1(C(C)C)cnc(O)c(C=O)c1.C1(CN(C(C)C2CC2)C)C2CC3C(C2)C13 C1(C)(CNC(C(F)OC)=O)CCN(C(=O)CCC2CC2C)CC1 c1(C(N2CC(O)(CNC(Cc3c(C)cc(O)cc3)=O)C2)=O)cc2ncccn2n1 CCCCCC(O)CC(=O)NC(Cc1cn[nH]c1)C(=O)N(CC(O)(CC)CC)C C1(O)(C(=O)N)CCCC(C)CC1.C(C(C)(C)C(=O)N1CCC(C)C1)NC(C)=O CCCC(C)(O)C(=O)N1CC(NC(=O)CC2(c3ccccc3)CCC2)CC(F)C1 c1(NC(C2CSCCN2C(=O)Cc2ccc(F)c(Br)c2)=O)nc2cccnc2s1 C1(CC(=O)N)CCN(C(C2CC(C)CC(=O)N2)=O)CC1O.C1(COC)CCC1 c1(CN2CC(CNC(=O)Cc3cnc[nH]3)C2)nccc(OCC(F)(F)F)n1 N1(C(COCCCC)=O)CCC2CCC12CNC(c1nc(C)sc1C)=O c1(C(C)C(=O)NCC(O)Cc2cccc(Cl)c2)noc2ccccc12 c1(C(=O)NC(COC)CC(N2CCOC(C)CC2)=O)c[nH]nc1[N+](=O)[O-] N1(C(CC2(OC)CCCCC2)=O)CC(C)CC1(C)C.C(=O)(CC(C)CN(C)C)N C1(NC(C(n2cnc(C#N)n2)C)=O)C2CC1CN(C(C1CN3CCC1CC3)=O)C2 c1(C(=O)NC2(CCNC(C3CC(C)(O)C3)=O)CCCC2)cc2cnccc2[nH]1 c1(CC)ccccc1OCCC(=O)N(CCCCNC(c1cc(C#N)c[nH]1)=O)C N1(C(C2C(=C)C2)=O)CCC(NC(c2cccn3nccc23)=O)CC(O)C1 Cc1cccc(CN(C)C(C2(C)C=CCN2C(c2ccccc2Cl)=O)=O)c1 C1(C2CN(C(c3c[nH]nc3C3CC3)=O)C2)(NC(c2cc(C)ncc2)=O)CC1 Cc1nc2ccccn2c1C(=O)NC(C)CN(C)C(C12CC1COC21CCC1)=O C1(CC=C)(C(=O)NCC(C)(O)CNC(=O)CC2CC2)CCCC1 CC(CCc1ccc(F)cc1)C(=O)N1CC(n2cc(CO)nn2)C1 C1(CNC(CN(C(C)=O)C)=O)CN(C(=O)C(=Cc2cscn2)F)CCO1 O=S(=O)(c1cnc(N2CCC(c3ccco3)C2)c(Cl)c1)NCC1(Br)CC1(F)F CN1CCN(C)C(CNC(N2CCC(C)(c3nn[nH]n3)C2)=O)C1 N1(C(C2CC=C(C)CC2)=O)CCC2CC(NC(C3CN(C)CCO3)=O)CCC2C1 CC1CN(C(=O)C)CC1n1cc(CCCN(C)C)nn1.N1(C)CCCC1.C1CC1 c1(-c2cn(CC(=O)NC3CN(CC(F)(F)F)C3)nn2)ccncc1F C1(C(=O)NCCCN(C(c2c(OC)ccs2)=O)C)CC(C)(C)CO1 C(C(C)(C)CNC(c1ccnn1CC)=O)N(C(=O)Cc1c[nH]nc1)CC c1(-n2cc(CC3CCN(C(CC(C)OC)=O)C3)nn2)cccc(F)c1 CC(=Cn1ccnn1)C(=O)NCCCCCNC(C1C2CCC(=O)C12)=O N1(C(COC)=O)CCN(C(c2cc(C)sc2-n2cccc2)=O)C(CC2CC2)C1 C1(C(=O)NCCCN2CC=CC2)CCN(C(=O)C(O)Cc2cnc[nH]2)CC1 Cc1[nH]nc(CN2CC(CC(C)NC(C3(C4CCCCO4)CC3)=O)C2)c1Cl N1(C(C2ON=C(C)C2)=O)CCC(Nc2nc(-n3cccn3)cc(C)n2)C(C)C1 c1(C(N(CC(=O)NCCCc2cc[nH]n2)CCOC)=O)ccccc1C N1(C(C=CC=CCCCCC)=O)CCN(C(c2cnc(S)n2C)=O)CC(C)(F)C1 c1(CC(=O)NC2(COC)CN(C(=O)CN3CCSCC3)C2)cn(C)nc1Cl Cc1cccc(CC(N2CCC(C)(CC(N3CCCCC3CN(C)C)=O)C2)=O)n1 N1(C(C2(C)CCSCC2)=O)CCCC(O)(CCNC(=O)CC2CCNC(=O)C2)C1 c1(CC)cc(C(=O)N(CCC(C)NC(=O)C=CC2CCCN2C)C)ccn1 C(=O)(N(CCC(=O)NCC(C)CC1CC1)OC)c1c(CC)nns1 N1(CCCC)CCCC(C(=O)N(CC)Cc2cnc(O)n2CC)C1 Cc1ccc(C(=O)NC(C)Cn2cc(C)nn2)c(N)n1.C(=O)(CCS(C)=O)N C1(O)(CC(=O)Nc2c(OC)ccnc2)CCN(Cc2ccc(Br)c(F)c2)CC1 CC1CN(C)C(=O)CN1C(C1C=CC(NC(c2ccc[nH]2)=O)C1)=O C1(C#CC(=O)NC(C2CCN(C(c3nc(Cl)sc3Cl)=O)C2)C)(CC)COC1 N1(C(C2(C3(C)CC3)CC2)=O)CCN(C(C23CC(F)(C2)C3)=O)CC(C)(F)C1 Cc1cccc(Cl)c1-c1cn(C2CCCN(C(=O)CC3(O)CCOC3)CC2)nn1 C(=O)(CC(O)CNC(=O)Cc1cnnn1C)N1CC=C(C)C1 C(c1nc2ccccc2s1)=CC(N1C2CCN(C(c3c(C)nn[nH]3)=O)C(C2)C1)=O N1(C(COC)=O)CCC2(CCCN(C(=O)Cc3c(F)cc(F)cc3F)C2)CC1 N(C(=NCCC(C)C)NC1CC(O)C1(C)C)CC(C)(CO)OC C1(C(=O)NCCOC(C)C)CCCCCC1NC(C12CCCC1C2(F)F)=O C1(CC(=O)N(CC(CO)(CO)NC(C2C(C)C2C)=O)C)CCCNC(=O)C1 C1(C(=O)NCC(N2CCN(C(c3cnn[nH]3)=O)CC2)=O)C2C3CCC(C3)C12 c1(NCC(COC)OC)cc(Br)ccc1S(=O)(=O)NC12CCCN(CCC1)C2 N1(C(C23CCC(OC)C2C3)=O)CC2(CC(C=O)CO2)C1.CC(C(C)C)C(C)C.N c1(C(N(C(C)CNC(C2CC(C)(F)C2)=O)C)=O)cc2ccc(Br)cc2cn1 N1(Cc2ccc(NC(C)=O)cc2)CCCCC(C(=O)Nc2nccc(NC)n2)C1 C1(C(=O)OC)CCN(CC(=O)N(C)CCc2cccs2)C12CCC2 Cc1cc(C(N2CC(F)(C(=O)NCc3ccc(F)c(F)c3)C2)=O)cc(F)c1 N1(C(CCN(CCC)C)=O)CC(N(C(=O)C=Cc2ccccc2)C)C(F)C1 CCCS(=O)(=O)CC(=O)N1CCC1CNC(C1CCN1C(C)(C)C)=O C1(C(=O)N)CCc2nc(O)[nH]c2C1.C1(NC(C2(C(N)=O)CC2)=O)CCC(O)C1 C1(NC(C=CC)=O)CCSC12CN(C(C1CCCN1N=O)=O)C2 c1(OC)ncc(C=CC(N2CCC(C(C)(O)CNC(=O)CCCF)CC2)=O)cn1 N1(C(c2ccc(CSC)o2)=O)CCC(C2CCN(C(c3ccc(C#N)[nH]3)=O)C2)C1 C12(NC(c3cc(C(C)=O)sc3)=O)CCCC1(F)CN(C(=O)C=CC(C)C)C2 c1(N(CCOCCNC(C(c2cccnc2)C)=O)C)ncc2c(ncn2C)n1 C1(NC(C(C(C)(C)O)NC(c2noc(CC)c2C)=O)=O)CC2C=CCC(C1)C2 n1(CC(=O)NCCC(C)N(C(C(COC)OC)=O)C)nc2n(c1=O)CCCCC2 N1(C(CC=C)=O)CCC(O)(C(C)NC(=O)CS(=O)(=O)N2CCOCC2)CC1 C(=O)(C(C)C(N)c1ccccc1)NC(c1nnc(COC(C)C)s1)C C(=O)(C(Cc1cncs1)NC(=O)CCCc1nc[nH]n1)OC c1(SC)nc(N2CCCC(CCNC(=O)CC3CCC(F)(F)C3)CC2)ncc1C C1(NC(c2ccnc(O)c2)=O)(CO)CCCN(C(c2cc(O)ccc2F)=O)C1 C1(C(=O)Nc2ccc(CCC)cc2)CCCCCN1C(c1cnc(Cl)n1C)=O N1(C(C2(CC(C)C)CC2)=O)CCC(O)(C(C)C)C1.c1(C=O)cnn(CC)c1 C(=O)(C1CCCc2scnc21)NC1C2(CN(C(C(F)=CCC)=O)C2)SCC1 C1(C(N2CC(O)(CNC(CS(=O)(=O)N(C)C)=O)C2)=O)CCCC12OCCO2 c1(CCC(=O)NC2CCN(C(C(C)OCCC#C)=O)C2)ccc(Cl)c(F)c1.C c1(CC(=O)NC2(C)CN(C(c3cnc(SC)s3)=O)C2)nc([N+](=O)[O-])n[nH]1 C1(NC(C2(C)CCC2)=O)CCN(Cc2ccccc2-c2cccnc2)CC1F C(=O)(C1=CC2(CCOC2)C1)NCCCC(C)NC(C1CS(=O)(=O)C1)=O N1(C(c2cc(C)oc2)=O)CC2(CC2CNC(=O)OC(C)(C)C)C1 c1(C(=O)NC2CCCN(C(c3cc(C(C)C)no3)=O)C2)cc(Cl)cc2c1CCC2 C(=O)(C(C)CCCC(C)C)NC(CNC(CCC)=O)CO Cc1cnc(NCc2nnnn2CC2CC2)c(S(=O)(=O)N2CSC(C)C2)c1 c1(OC)cc(-c2nc(COc3ccc(F)cc3)nn2C(C)CC)cc(OC)n1 C1(CNC(C(CCC)(C)C)=O)CC2(CCC2)CN1C(=O)C=CC1CCCO1 C1(OC)CC2(CCC(C(=O)NC(C)CNC(C3(C)CC3C)=O)CC2)C1 C1(C(=O)NCC(CC)CO)CC2(CCC2)CN1C(=O)Cc1c(C)n[nH]c1C c1(CC(=O)NCC2N(C(C(CC=C)C)=O)CC(F)C2)cccc2nonc12 N1(C(C2N(C(COC(CC)C)=O)CCC(C)C2)=O)Cc2nncn2C(C)C1 c1(C(CNC(=O)CC2CC(C)=NO2)NC(COC)=O)ccc(C)cc1 N1(C(c2nc(OC)oc2)=O)CCC(NC(=O)CCc2cccnc2C)C(F)C1 C(CS(=O)(=O)CC(=O)NCC(C)(O)CNC(c1cn(CCO)nn1)=O)OC Cc1cccc(Cl)c1C(=O)NC1CCC(C)CC1.C(=O)(C=O)N.CC(F)(F)F C(C)(c1ccccc1)=CC(=O)NC(C(CO)NC(C(C)OC)=O)C C1(C)(C(=O)NCCC(C)F)CCN(C(c2cn(C)cc2C(F)(F)F)=O)CC1 C1(C(N2CC(OC)C2)=O)CCCCCN1C(=O)C(C(C)O)N(C)C N1(C(C(CCC)F)=O)CCC(C(=O)NCC(c2cnc[nH]2)C)C(C)C1 CCCCC(C(=O)N1CCC(C)(O)CC1)NC(c1[nH]nnc1C)=O C1(C(N(C2CCN(C(C3CCC(C)CC3)=O)C2)CC#C)=O)CC(C)C1(C)C N1(C(C2C(C)CN(C)C2)=O)CC2(C1)CN(C(=O)C=Cc1cnn(C)c1)CCO2 Cc1ccc(Cl)cc1C(=O)NCCn1cc(C)nn1.C(=O)C(C)C(C)(C)C.N C1(C(=O)NC(C2CCCC2)CC)CCOCCN1C(=O)CC1CCCC2CC12 c1(C(=O)N)noc(C2CCCCC2)n1.C1(CNC(=O)OC(C)(C)C)COC1 C1(NC(C2CC(OCC)C2)=O)CCN(C(=O)C(C)(C)CO)CCC1CO C(=O)(CC1=CCOCC1)N1CCN(CC2(NC(C(CCC)C)=O)CC2)CC1 N1(CCNC(=O)CC2OCCO2)CCN(C(=O)C)CC1.c1csc(C(F)F)n1.N CC1OC2CCC1(C(=O)NC1CCC(NC(=O)COCCF)CC1)C2 C(=O)(CC(F)(F)C(F)(F)F)N1CCCC(N(C)C(C2(C)CC2)=O)CC1 N1(C(CCOC(C)=O)=O)CCC2(CC2)CC1C(=O)NC(C)CCn1cncn1 N1(C(c2c(C(C)NC(C3(CC)CCCC3)=O)noc2)=O)CC2CCCC2C1 c1(C(N2CCC(C)(C)CC2)=O)ccc(F)c(F)c1F.C1(C(=O)N)CCC1C(F)F C(C(C)(C)C)N(C(=O)C(C)CN1CCCCC1)CC.c1(C=O)cc(Cl)no1.N Nc1cccc([N+](=O)[O-])c1C(=O)NCC1CCCC1.c1(C=O)cccc(F)c1.N N1(C(c2cc(C(C)=O)c(F)cc2)=O)CCCC(C2CC2NC(C2(O)CCC2)=O)C1 C1(C(N2CC(C(C(=O)NOCc3ccc(O)cc3)OC)C2)=O)CC2(CCO1)CC2 C1(C(N(CC(=O)N(C)CC2(CC)CC2)C(C)C)=O)CCCC12CCC2 C1(C(N2CC(N(C=O)C)C2)=O)CSCN1C(=O)C.C=O.C1CC1.CC.N N1(C(CN2C(C)CCC2)=O)CCC(=CCNC(c2cccc(N(C)C)c2)=O)CC1 CC1(C)CN(C(=O)COC2CN(C(C3(C)CC(C#N)C3)=O)C2)C1C1CC1 C1(C(N2CCN(C(c3cnn(C4COC4)c3)=O)CC2)=O)CC2CCCN(C1)C2 C1(OCCC)CCCN(C(=O)CC2COCCN2C(C23CSCC2C3)=O)C1 c1(OCC)c(Br)cc(CN2CCC2C(=O)N)cc1Br.c1(C(C)O)ccc(O)cc1 C1(C(=O)NCc2cccc(OC)c2)N(C(=O)C(C)C(O)C(C)C)CCCC1(C)C C12(CNC(N3CC4CC(c5ccccc5)C4C3)=O)CCC(CC1)OC2 N1(C(C2=CC(C)(C)C2)=O)CC2(CC(NC(=O)C(C)(C)c3ccns3)CO2)C1 C(=O)(C1CCC(=O)c2cccn21)N1CCC(NC(C2CC(C)(C)C2)=O)CC(O)C1 c1(C(=O)NCC2N(C(C=CCCC(C)C)=O)CCCC2)nn2c(c1Br)CCC2 C1(C(N2CCN(C3CCN(C(C4C(=C)C4)=O)C3)CC2)=O)CC12CCCCC2 Cc1nn(CCO)c(C)c1C(=O)NCC1CC2CCC1N2C(C1CC=CC1)=O C(=O)(C(F)(F)c1csc(Cl)c1)NCC(c1ccccc1)CNC(C=C(C)C)=O N1(CC(=O)NCCn2cc(C(N3C(C(C)O)CC3)=O)nc2)CCC(F)CC1 c1(CN(C2CC2c2cnn(C)c2)CCNC(C)=O)ccc(Cl)cc1 c1(C(=O)NCC2(O)CN(C(C(COC)OC)=O)C2)ccc2n[nH]cc2c1 N1(C(Cc2c(C)ccnc2)=O)CCCC(CO)(NC(=O)CCCC(F)F)C1 c1(C(=O)NC2CCN(C(c3ccn(CC)c3C)=O)C2CO)ccc(F)cc1OC c1(NCC(C)(C)NC(C(CC)CC)=O)ncc(C)cc1C(=O)OC C1(CC=C)(C(=O)NC2CCOCC2OC)CCN(C(=O)C(C)=CCC)C1 C1(NC(c2ccc(N3CCC3)nc2)=O)CCC2(CC1)CCN(Cc1cnsc1)C2 N1(C(c2c(C)scn2)C(=O)NCc2ccc(Cl)cc2)CCCC2C1CCN2C c1(OC)cc(F)ccc1C(=O)NC1C2CCN(C(c3nccc(Br)c3C)=O)C12 N1(C(=O)NCC2CSC2)CCCC1C1CCCCC1 Cc1c[nH]c2ncnc(N(C3C4CNCC34)C(c3ccc(Cl)c4cc[nH]c34)=O)c12 c1(C(=O)NCC2CCCN(c3nnn(C)n3)C2)ccc2cc[nH]c2n1 N1(C(C(CN(C)C)NC(=O)CC2OCCCO2)=O)CCCC(O)CC1 C1(NC(=O)CCn2ccnc2)CC(C(F)F)(NC(c2ccoc2)=O)C1 c1(CCC(=O)N)ccc2ncsc2c1.c1(OC)ncc(C(=O)NCC2CC2)s1 C(N=c1nc(N2CCC3(CC2)CC3)c2cc(OC)ccc2[nH]1)c1ccc(CC)s1 CCCCCCC(C)C(=O)N1CC2C(NC(c3ccc(C)cc3OC)=O)C2C1 C1(NC(c2cc(C)oc2C)=O)COC2(CCN(C(c3cnns3)=O)C2)C1 c1(C(=O)NC2CCCN(Cc3cn(CC(C)C)nc3)C2C)ccc2nc[nH]c2c1 CC1CC(CC(=O)NCC(F)(F)CC2CC2)CN1C(c1cscc1Cl)=O C1(CC)(NC(c2ccc(C)s2)=O)CCN(C(C2CC(C)CC(C)C2)=O)CC1 N1(C(CN(c2ccnn2C)C)=O)CCN(C(=O)C(O)C(F)F)C(C2CC2)C1 N1(C(c2cncc(OCC(F)F)c2)=O)CCN(C(=O)C(Cl)=CCl)C(C(F)F)C1 C1(C(=O)NCC2(CCNC(=O)Cc3cnc[nH]3)CC2)CC2(CC2)CO1 C(=O)(CCS(C)(=O)=O)N1CCC(NC(CCC2CCCN(C)C2)=O)(CF)C1 c1(C(=O)NC(C)CNC(c2cc(F)c(O)c(F)c2)=O)cccc(C=C(F)F)c1 CN1Cc2ccc(C(N3CCN(C(c4cccc(Cl)c4Cl)=O)C4CC34)=O)cc2C1 C12(CN(C(CNS(C)(=O)=O)=O)CC3CCCC3)CCC(C#N)(CC1)C2 C1CN(C(=O)CC2CCCN2C)C2(CCOCC2)C1.C1(OC)CC(C(=O)NC)C1 C1(CSc2nnc(CC)n2-c2cccc(C(C)=O)c2)CC2CCC1O2 c1(CNC(CCSC)=O)ccc(C)c(F)c1.c1(C(=O)N)coc(C(C)C)n1 c1(OCC)ccccc1NC(C1(C(C)C)CCCN1C(c1ncncc1Cl)=O)=O C1(N(CCC(=O)NCC(CC=C)NC(C2CC3C=CC2O3)=O)C)CCCCCC1 N1(C(CC(C=C)CC)=O)CCOC2CCN(C(c3ccc(O)cn3)=O)CC12 C(CN=c1cccn[nH]1)N(C(C(n1cc(C2CC=CCC2)nn1)C)=O)CC(F)F C1(C(=O)NC2CC(C)CCC2O)(CC)CCCN(C(C2CC=CC2)=O)C1 C1(CCCC)CN(C(c2nnn(C(C)(C)C)n2)=O)CCN1C(=O)C(O)COC C1(NC(c2cnn(C)n2)=O)CCN(C(=O)CC2C=CCCC2)CC1F C(=O)(CCCCN(C)C)N(CCOc1ccc(C(F)(F)F)cc1)CC Cc1ccc(C(=O)NC2CCC(C)N(C(C3CC4(CSC4)C3)=O)C2)cc1O C1(CC(=O)N)C=CS(=O)(=O)C1.C1(NC(=O)Cc2cnns2)(C)CCCC1 CCC(C(=O)NCC1CCN(C(=O)C(Br)=C(C)C)CC1)C(C)(F)F C(CCC(F)(F)F)NC(C=Cc1c(C)ncs1)=O.C1(C(=O)N)(C(C)C)CCCO1 C12(C(=O)NC3CC(NC(CCN(CCC)C)=O)CC3O)CCCC(CO1)C2 Cc1[nH]c2ccccc2c1C(=O)N(C)CC1CCCN1C(C1CC(C)CO1)=O CC1CCN(C(=O)C=CC2CC2)C(C)C1NC(c1ccc(CO)c(F)c1)=O c1(C(=O)N)ccccc1.CCC(C(=O)N1CC(C(N)=O)(C)C1)SC.CC(N)=O n1(CC)c(=N)[nH]c2cc(C(=O)N(C(C)CNC(c3occc3F)=O)C)ccc12 N1(C(Cc2c(C)nsc2)=O)CCC(O)(C(C)NC(c2cnn3ccsc23)=O)CC1 C1(NC(c2cccc(OC)c2)=O)CN(C(=O)CC2CC(O)C23CCC3)CCC1O C12(NC(C(C)=CC)=O)CCC(CN(C(c3csc(C(C)=O)n3)=O)C1)C2 Cn1nnc(Br)c1C(=O)NC1CCCCC1CNC(=O)C(C)(C)O C1CCN(C(C2CC(=C3CCC3)C2)=O)C1(C)C.C(C)(C)(C=O)OC(C)=O.N C(=O)(CC(C)CC(C)C)N1C(C(=O)NCCCOC=C)CC=CC1 c1(NC2(c3n(CCCOC)ccn3)CC3COCC23)csc(=NC2CC2)[nH]1 c1(CN(C(=O)CC)C)cccc(C)c1.C(C1CCCO1)=CC=O.C1CC1.N CCCCS(=O)(=O)CC(=O)NC1CC2CCC1(Nc1ncc3c(n1)CCCC3)C2 C1(C(=O)OC)CCC(C)N(C(c2c(Br)cnn2CC(F)F)=O)C1 C(=O)(C1=CCN(C(C2CC(=O)C23CCC3)=O)CC1)NC(CCOC)C(N)=O c1(-n2c(CC)c(NC(=O)C=O)cn2)ccc(NC(C2SCCC2C)=O)c(C)c1 N1(C(CC=CCC)=O)CCN(C(c2coc(Br)c2)=O)CC1CCC C1(NC(C2C(C3C(C)C3)C2)=O)CC2CCC(C1)N2C(=O)C(O)Cc1cnc[nH]1 c1(C(N2CC(NC(C3(CC#C)CCCC3)=O)C(C)CC2)=O)cnc2[nH]ccnc1-2 C1(O)(CN(C(=O)CCOC2CCOC2)C)CCCN(C(=O)CS(C)(=O)=O)C1 N1(C(=O)N)CC2(CC2)CC1C(N1CCC(C#N)C1)=O.c1(OCC)ccccc1 N1(C(CC2(C)CCCCC2)=O)CC2(CCN(C(=O)CC3CN4CCN3CC4)C2)C1 CC(CCO)C(=O)NC(C)C(C)NC(=O)C(C)NC(N)=O N1(C(=O)NCC2(N(C)C)CCCCCC2)CC2CSCC(C2)C1 Cc1cc2ncnc(N3CCCCC3CNC(C3CCn4ccnc4C3)=O)c2[nH]1 C(C1(C)Cc2ccccc21)NC(c1n(C)nnn1)CCc1ccc(SC)cc1F Cc1nsc(NC2CC2)c1C(=O)NCC(F)CNC(=O)CCCN(C)C c1(NC(=O)NC2C(C#C)CCCC2)cc(F)c(N2CCOCC2)cc1F N1(C(CC2CC(C)N(C(=O)CC3CCSC3)C2)=O)CCN(C)C(CO)C1 c1(NS(CC)(=O)=O)cccc(C(N2CCC(n3nnnc3C(F)(F)F)CC2)=O)c1 C1(NC(=O)CCCc2cnccn2)CN(C(=O)Cc2nc[nH]n2)C2(CCCC2)C1 N1(C(c2ccc(C)cc2N)=O)CCC(NC(c2csnn2)=O)C(CO)CC1 C(=O)(CS(=O)C(F)(F)F)N(CCCN(C)C(C1(CF)CC(F)(F)C1)=O)C Cc1ccc(-c2csc(N(C(=O)C(C)SC(F)(F)F)C3CCCC3)n2)cc1 C1(C)CC(C)(C)OC1=O.CC1(C)CCC(C(N2C3CCC(C3)C2C=O)=O)CO1.N C(CC(C)(C)C(=O)NCC1COCCN(C(C2CSCCS2)=O)C1)OC C=C(CNC(C1CCCN(C(=O)OC(C)(C)C)CC1)=O)c1ccc(F)cc1F CN=c1[nH]nc(CC(=O)NC(C2CN(C(=O)CCCOC(C)C)CCO2)C)s1 N1(C(=O)CCCOC2CCCC2)CC2CCN(C(c3cc(F)cnc3O)=O)C2C1 Cc1cnc(N)c(C(=O)NC2CCCC2NC(c2cc(C(C)C)[nH]n2)=O)c1 N1(C(C)=O)CCOC2(CCN(C(C3CCN(Cc4cccnc4)CC3)=O)C2)C1 c1(C(=O)NCCC(=C)CNC(=O)Cc2c[nH]nc2O)cccc2nc(C)[nH]c12 N1(C(C(c2ccnn2C)C)=O)CCCCC(NC(c2cc(=O)cc(Cl)[nH]2)=O)C1 C1(CNC(CCC(C)CN(C)C)=O)CN(C(=O)C2CC2)CCC12CCOC2 CCC(C(=O)N1CC(CNC(C2(CF)CC2)=O)(OC)C1)n1cncn1 N1(C(C2(CC)CCC2)=O)CCC(CN(C)CC2(C)CCC2)C1 O(NC(=O)CC(C(F)(F)F)NC(=O)C1=NN(C)C(=O)CC1)CC(=C)C N1(C(C23CCC(COC(C)=O)(CC2)O3)=O)CC2(CCC(F)(F)CC2)C1 N1(C(c2c(OC)ccc(C)c2)=O)CCCC2C1CCCN2C(c1coc(C)n1)=O Cc1c(C(=O)N(C(C)CCNC(=O)CCN2CCOCC2)C)sc2ccccc12 c1(C(=O)NCCOCCN(C(CC(=O)NCC)=O)C)c(F)cccc1F N1(CC=C)CCN(C(=O)CC2CCN(C(=O)CC3COCCO3)C2)CC1=O C#Cc1ccc(C(=O)NCC2CC3CC3N2C(=O)Cc2cccc(O)c2)cc1C S(=O)(=O)(c1ccc(C#N)c(NCCn2cnnc2)c1)N1CCC(C)CC1C(C)C Cc1oc(CNC(=O)Cc2ccc(OC3CCC3)cc2)cc1C(=O)O Cc1ccccc1CCC(=O)NC1(CO)CN(C(=O)CC2CC2C)C1 Cc1cc(C(N2C3CCC2C(CNC(=O)Cn2cncn2)C3)=O)cc(C)c1Br Cc1ccccc1OCCC(=O)NC1COCCC1NC(c1ccc(C#N)[nH]1)=O C12(C(=O)NC3(C(=O)NCc4cnc(C)o4)CCCC3C)CCC(CC1)CO2 N1(C(C(C=C)C)=O)CC2(CCC(CNC(=O)COc3cc(C)on3)O2)C1 CC1CN(C)C(C)CC1NC(=O)CC1CCCCC1NC(=O)C1=C(Cl)CCCC1 N1(C(c2ccc(N(C)CC)nc2)=O)CCC(C)(CNC(=O)CCCCSC)CC1 C=Cn1ncc(C(N2CCOC(C(=O)NCC3(C)CCN(C)C3)CC2)=O)c1N c1(C(C(=O)NCCOCc2ccccc2)NC(CCCC=C)=O)cc(Br)cc(C)n1 N1(C(c2c(C)n(CC(F)(F)F)nc2)=O)CC2CC(NC(=O)C(C)CC(C)C)C1C2 c1(C(N2CC(CCCNC(c3n(C)c(O)nc3)=O)OCC2)=O)ccc(Cl)c(N)c1 C1(C(=O)N)CC(=O)C12CCC2.N1(C(c2cnccc2)=O)CC(F)(C2CC2)C1.C C1(C=O)CC(F)(F)C1.C1(CNC(=O)CC2(c3ccon3)CC2)COCC1.N C1(C)CN(C(=O)Cn2nnnc2C2CC2)CCO1.N1(C(C)C)CC(C(=O)N)C1 C1(C(=O)NCC(c2cnc[nH]2)C)N(C(c2cnc(S)nc2)=O)CCCC1(C)C C1(C(=O)NCCCCCC)CN(C)CCN(C)C1.C(C(C)(C)C)N(CC(=O)N)C c1(C(=O)NCC(C)NC(=O)CC=C(Cl)Cl)cccc2sncc12 CCCS(=O)(=O)CC(=O)NC1CCN(CCNC(=O)C(O)C2CC2)CC1 c1(C(=O)NCC(C)NC(c2cnn(-c3ccccc3)n2)=O)c(F)ccc(F)c1N N1(C(c2n(C)nc(Br)c2)=O)CCC2(CCN(C(=O)CC3CC34CC4)C2)C1 C(=O)(C(C)(C)C(C)(C)C)NCC(C(C)C)NC(CC1(OC)CCC1)=O C12(C(=O)NCC3(C)N(C(CCC(=O)OCC)=O)CCC3)CCCC1(O)OCC2 N1(C(c2ccc(C#C)cc2OC)=O)CCN(C(=O)CC(C)(C)C=C)C(C)CC1C N1(C(C2CCC(=C)CC2)=O)CC2CN(C(=O)Cc3cccc(OC)c3Br)C2C1 C12(C(N3CCCC3)=O)CC(CN1C(=O)C(CC)N(C)C)C2.CCC(=O)NC C(=O)(C(CCC1CC1)NC(=O)CC1CC1)NCC1(C)C(C)(C)C1 C1(NC(C2C(CCC)C2)=O)CCC(CNC(=O)C(C)CC)CC1 Cc1cc(Cl)ccc1OCCCn1cc(-c2ccccc2C)nn1 c1(CC)c(C(=O)NC(Cn2ccnn2)C(=O)N)cnn1C.C1CCC2(CC2)C1 c1(OC)ccc(CCCC(=O)NCCNC(=O)CC(C)CN(C)C)c(OC)c1 C1CC2CC1OC(=O)N2.c1(CC(=O)NC2CC(C(F)C(=O)N)C2)ccc(F)nc1 N1(C(C)=O)C2CCCC1CN(C(c1ccc3csnc3c1)=O)C2 N(C1CCCc2sccc21)C(c1ccccc1Cl)=O C1(CNC(c2cccc(C3CCC3)c2)=O)CCCCCN1C(C1CCOC1)=O N1(CCC(=O)N(C)C)CCSC(C)(C)C1.C1(C(N2CCCC2)=O)CC2C=CC1C2 Cc1ccc(CC(=O)NCC2CCN(C(=O)C=Cc3ccn(C)c3)C2)cc1Cl c1(C(N2C(CC#N)CN(c3ncc(C4CC4)cn3)CC2)=O)ncnc2occc12 N1(C(C(c2cncc(F)c2)C)=O)CCN(C(=O)CSc2nncn2C)C(CF)C1 C1(NC(CSCCC)=O)CN(C(=O)CC=C(Cl)Cl)CC(C)(C)C1 Cc1nc2c(o1)CCN(C(=O)C(C1CCCCC1)NC(=O)CCC1CC1(F)F)C2 c1cn2c(n1)CCC(NCC1(C3CCCO3)CC1)C2 C1(NC(=O)CCSc2ccc(F)cc2)C2CN(C(=O)C(F)C3CC3)CC12 C1(C(C)C)CCC(C(=O)NC2(CO)CC2)N1C(=O)CCC1CCOC1 n1(CCC)nc(-c2ccsc2)nc1C1CC(=O)N(CC2CCCC2)C1 c1(C(=O)N)cncc(C)c1.n1(CC)ccc(CCNC(C2(CC)CC2)=O)n1 N1(C(C2CN(C(C3(F)C(C)(C)C3(C)C)=O)CC2(F)F)=O)CCc2ncccc2C1 N#Cc1c2c(cn(CC(c3cccs3)NC(=O)CN3CCCC3)c1=O)CCCC2 N(C(=NCCC1CCOC1)NC1CC1)CC1C(C)(C)CCO1 N1(C(=O)CSC(F)F)CCN(C(c2ccc(C3CCCOC3)cc2)=O)C(CF)C1 c1(CN2CC(CC(=O)NCC3(O)CCOCC3)OCC2)cccc(Cl)c1Br C1(C(=O)NC)C=CCC1.C1(C(N(CCC(=O)N)C(C)C)=O)CC12CCC2 n1(CC=O)ncc2cc(C)cnc12.C1(C(N(CCC)CC)=O)CC(C)OC1=O.N N1(C(C(CC(C)C)OC)=O)CCn2c(C(=O)O)cnc2C1C CC1CN(C(=O)OC(C)(C)C)CC1CS.C1(C=O)CC2(C1)CC2F.CC C12CC3CC(C1)CC(C3)C2.CC(C=O)O.C1(CC=O)CC12CC2.C1CC1.C Cc1snnc1C(=O)N(CC(C)O)CCNC(=O)C(C)CC1CCC1 C1(CC(=O)NC(C2CCCN(c3snc(Cl)c3C#N)C2)C)CCCNC(=O)C1 c1(CC)occ(C)c1C(N1CC=CC(C(=O)NC(C)CCC(C)C)C1)=O C1(C(=O)NC2(CSC)CC2)CN(C(=O)CCC(C)OC)CC12CCC2 CN1CCC(CC(=O)NCC2CCCCC2NC(=O)C=C2CCCCC2)CC1 N1(C(c2cn(CC=C)nn2)=O)CCN(CC(=O)NCC2=CCCC2)CC1 C(=O)(C#CC(=O)N(C)C)NCCN(C(=O)CCC1CCCO1)C(C)C Cc1cc(=O)n2nc(COC(c3ccc(F)c4c3CCC4)=O)sc2n1 Cc1cc(C(N2CCC(C)(NC(=O)C=Cc3ccsc3)C2)=O)c(C)[nH]1 C1(OC)(C)CN(C(=O)C)C1.c1(C(C=CC=O)=O)ccccc1.C1CCOC1 c1(NC(=O)Nc2scc(CN3CCC(C)CC3)n2)cccc2c1N(C)CCO2 Cc1[nH]c(C(=O)NCC2C(C)CCN2C(c2ccc(C3CC3)s2)=O)c(C)c1C NC(=O)CC(O)C(=O)NCC1CN(C(=O)Cc2scnc2-c2cccs2)CCO1 CC(C)CCC(O)C(=O)N1CCCC1(C)C(=O)NCC(F)(F)CO Nc1c(C(=O)NCCC2CCN(C(C3CCCC3O)=O)C2)ccc(Cl)c1F Cc1ccc(C(=O)NCCC2CCCCN2c2ccnc3ncnn23)c(F)c1F N1(C(C(CC#C)C)=O)CC2CCC1C(NC(=O)Cc1cnccc1OC)C2 N#CC1(F)CN(C(=O)C(C2(O)CCC2)NC(C2CCC3(CC3)C2)=O)C1 N1(C(Cc2nc(C(C)C)on2)=O)CCC(c2ncc(-c3ccccc3)[nH]2)CC1 N1(C(C2C(C#C)C2(C)C)=O)CCC(C)N(C(c2cc(C)n(CC)n2)=O)CC1 S(=O)(=O)(C1CCOCC1)NC(C1CCC2(C1)CC2C(=O)O)=O N1(C(c2cnc(CC)nc2)=O)CC2(C)CCC1C2.c1(C=O)occc1C(C)C.N C(=O)(N(CCC(=O)NCCCCC#CC)OC)c1ccc(COC)o1 c1(OC)cc(OC)cc(C(=O)NC2CCCC2NC(C2Cc3nccn3C2)=O)c1 N1(C(C2(CNC(c3c[nH]c(=O)cn3)=O)CC=CC2)=O)CCC(F)(F)C1 C12(C(=O)NCc3cc(C(=O)Nc4cn(CC)nc4)on3)CCC(CC1)CC2 C1(NC(C(CC2CCC2)NC(=O)CCc2ccccc2)=O)CCC2(CCCC2)C1 N1(C(c2cc(CC)on2)=O)CC2CC(C1)C2NC(C1CC(F)(F)C1)=O C1(CNC(C(C)C2(O)CCC2)=O)CCCN1C(c1c[nH]cc1Br)=O N1(C(CCC2CCN(C(C(CC(F)F)OC)=O)C2)=O)CC2(CCOCC2)C1 C1(C(=O)NC(COC)COC)CN(C(C2(CF)CCOCC2)=O)CCO1 C1CN(C(=O)Cn2nccc2C)C2CC12.c1(C(=O)OCC)c[nH]cc1C=O.N n1(CC)nnc2c1CCC(C(N1CCCC1CNC(=O)C(C)C1CC1)=O)C2.O c1(CC)oc(C(N2CC(C)(C(=O)NC(C)(C)C)C2)=O)cc1C.C(N)=O.N N1(C(C(C)(C)C)=O)CCC2(CCC2)C(NC(C2CC(=O)NC(=O)N2)=O)C1 C#CC1(O)CCCN(C(c2c[nH]nc2CNC(=O)Cc2cnnn2C)=O)C1 c1(C(=O)NCC2(F)CCN(C(c3ccc(C)cn3)=O)C2)cc(C)nc(O)n1 C(CCC(=O)NCCc1cc(C)on1)(C(C)C)NC(c1nncc(OC)c1)=O C1(C(N2CCC(Cn3cc(C(C)(C)OC)nn3)CC2)=O)CCCC(C)CC1 c1(C(=O)NCC2C3CN(C(C4(CC#C)CC4)=O)CC32)c2ccccc2nn1C c1(C(=O)NCC2C(NC(=O)COC3CCC3)CCC2)ccc(F)cc1 N1(C(c2ncncc2Br)=O)CCC2(NC(C3(F)CCCCC3)=O)CCCC12 Cc1ccc(Br)c(NC(C2CC3CC3N2C(c2ccnc(C(C)C)c2)=O)=O)c1 N1(CC(=O)NCCOCC(=O)NCCc2cnn[nH]2)CCNC1=O N1(C(C2CC2)=O)CCCc2ccccc2C1.c1(OC)ccc(C(=O)O)cc1C(=O)N CN1CCOc2c(-c3nc(C4CCOC4)nn3C3CCSC3)cccc21 C1(CC)C(C(=O)Nc2cccc(C(F)F)c2)CCN1C(c1ccc(O)nc1)=O N1(C(C(C)=C2CCC2)=O)CCC(F)(F)C(CNC(C2CCC3CC3CC2)=O)C1 C1(NC(C2CCCOCC2)=O)CN(C(c2ccc(OC(F)F)cc2)=O)CC1F N1(C(CN(CCC#C)C)=O)CCOCC(CNC(C2CCCC(=O)N2C)=O)C1 C1(C=O)CCC(=O)N(C)C1.c1(OC)cc(C(=O)NC(C)C2CCC2)ncn1.N N1(C(c2c(C)nc(C)o2)=O)CCC(C(=O)N(CCS(C)(=O)=O)C)C(C)(C)C1 C1(C(N2CCC(CCNC(C3CC4(C3)CC(O)C4)=O)C2)=O)CCc2c[nH]nc2C1 C1(NC(c2cnc(CCC)s2)=O)CC(NC(=O)CC)C12CCC2.C1CCCC1.S C(c1cc(C(F)(F)F)ccc1Cl)=CC(N1CCC(OC)(CN)C1)=O CCC(CC(C)CO)N=c1[nH]c(=NCc2nc(C)c(C)[nH]2)[nH]c2ncn(CC)c12 Cc1ccc(C=CC(N2CCC(N(C)C(c3cnc(C)nc3C)=O)CC2)=O)nc1 N1(C(=O)Nc2ccc(C(C)=O)cn2)CCCC2(C)CCCCC12 C(=O)(C#CC1(C)CCCO1)N(CCC(C)NC(C1(C)CSC1)=O)C C(=O)(C(=O)CC(C)C)NCc1ncc(C(N(C2CC(=C)C2)C)=O)cn1 C1(O)(c2cn(CC(=O)NCCS(C(C)(C)C)=O)nn2)CN2CCC1CC2 N1(C(c2ccn(C(C)C)n2)=O)CCN(C(=O)C(C)(C)C2CC2)CC1 C1(CNC(C(CCCCCCC)C)=O)CCCC2(CCN(C(=O)C(N)=O)CC2)O1 c1(NCC(N2C(c3cn(-c4cccc(OC)c4)nn3)CCC2)=O)ccc(Br)cc1F c1(C(=O)NCC(CC(C)C)NC(C(CC)(C)CC)=O)cc(Cl)cc2cccnc12 c1(CC)ccc(C(=O)N(C(C)CNC(C2(Br)CC2)=O)CC)cc1N C(=O)(C1CCCc2ncnn21)NCCCCNC(CC(CN(C)C)O)=O c1(NC(C23C(CN(C(c4cccnc4Br)=O)C2)C3)=O)cccc2c1C(=O)NC2=O C(C(=O)NC1(C(=O)NCCCOC(F)(F)F)CSC1)(C1CCC1)OCC c1(C(=O)NC(CNC(c2c(CC)ncnc2)=O)(C)CO)cccn2c(C)nnc12 C#Cc1cccc(NC(C2(F)CCCN(C(=O)COc3ccccc3Cl)C2)=O)c1 N1(C(C(OC)OC)=O)CCC(CO)(CNC(=O)CCc2ccsc2)C1 CC(C)CCCC(=O)N(CCCCCCC(c1ccccc1)O)CCO N1(C(c2ccc(C(=O)OCC)o2)=O)CCN(C)CC1C.c1(C=O)n[nH]cc1Br C(=O)(CCC(C(C)C)NC(c1coc(N(C)C)n1)=O)NCc1cnc(C)o1 CC1COc2c(C(=O)NC3CCN(C(=O)CC(C)c4cccnc4)C3)cccc21 c1(C(=O)NCC2C(C)CN(C(C3CCCC3(C)C)=O)CC2)ccc2c(c1)CCN2 C1(C(N(CC(CN(C)C)O)C)=O)N(C(=O)C2=CCCC2)CC12CCCC2 Cc1nc2c(o1)CCCC2CC(=O)NC1COCCN(C(=O)C(C)S(N)(=O)=O)C1 CN1CCC(CC(=O)NCC2C3CN(C(=O)CN)CC23)CC1.c1ccc(O)cc1 N1(C(c2cccnc2)C)CCC(NC(c2ncoc2-c2ccc(F)cc2)=O)C1=O C=CCC(CC)C(=O)NCC1CC(O)CN1C(=O)COCCSC c1cccc(Cl)c1.C(=O)CC.C1(CCCCO)(C(=O)NC(COC)C)CC1 Cc1coc(C)c1C(=O)NC1CC(C)N(C(C2CS(=O)(=O)C2)=O)C1 C1(C(N2C(C)CS(=O)CC2)=O)CN(C(C2C3CCC(F)C23)=O)CC(C)(C)C1 N1(C(c2cccc(CCO)c2)=O)CC2(CCN2C(=O)C(Cl)(Cl)Cl)C1 c1(CC)ccc(C(=O)NC2C3CC(NC(=O)Cn4nccc4C)CC23)cn1 c1(-c2c(C(=O)OCC)ccs2)ccc(CNC(=O)C(F)n2ccnc2)cn1 C1(OC)CCN(C(c2csc([N+](=O)[O-])c2)C(=O)NCc2ccccc2Br)C(C)C1 Cc1cc(F)ccc1C(N1CCC(O)(C(=O)NC(c2ccc(Cl)cc2)C)CC1)=O C1(CNC(CC(CC)O)=O)CC2COCC2N1C(=O)C(=O)Nc1cccc(C)c1 N1(C(c2cnc(-n3cccn3)s2)=O)CCCC2(CCN(C(=O)COC(F)F)C2)C1 N1(C(C2(OC)CC2)=O)CCCN(C(c2ccc(C(C)=O)cc2F)=O)CC1C c1(C2CCN(C(=O)NC3(CO)C(C)(C)C3)CC2)ccc(Cl)cc1Br Cc1ncc(C(N2CCC3(C2)CN(C(C2CCC=CCC2)=O)C3)=O)cc1C#N CC12CCC(C(N3CCN(C(=O)CC4(O)CCOC4)CC3CCO)=O)(CO1)C2 CCCC(CC)CC(=O)N1CCC(CNC(=O)C=CCF)C12CCC2 N1(C(c2ncn(CC)n2)=O)CC(C(=O)NCC2(F)CC(O)C2)C(C)(C)C1 C1(COC)(NC(=O)CC(C)C2CC2)CN(C(=O)Cc2ncc(C)s2)C1 C1(NC(CCN(C(CC)CC)C)=O)CC1C1CCN(C(=O)C(C)CO)CC1 N1(C(=O)C2CC2)CC2CC2(C(=O)NCCCc2cn(C3CCC3)nn2)C1 C1(NC(c2c(C(C)C)ncs2)=O)CCN(C(C2COC(=O)O2)=O)CC1F N1(C(C=Cc2n(C)cnc2)=O)CCC(C)(C)C(NC(C2C3COCC23)=O)C1 c1(Oc2ccc(N(C(C3CSC3)C)CC3CC3)cn2)ccccc1F Cc1sc(S(N)(=O)=O)cc1C(=O)N.C1CCCN(C(=O)CN(C)C2CC2)C1C Cc1csc2c(C(N3CCN(C(C4CCC=CO4)=O)C4(CCC4)C3)=O)ncnc12 C1(CNC(CC(CC)OC)=O)CN(C(c2ccc(OC)c(Cl)c2)=O)CCN1C C(=O)(CCC(F)(F)C(F)F)N(C(C)CNC(c1scc2c1CCCC2)=O)C c1(C(N2C(C)CC(NC(C=COCC)=O)C2)=O)ccc2cncn2c1C N1(C(c2c(C)ncnc2O)=O)CC2(CC(NC(C34CC(CO3)C4)=O)CO2)C1 Cc1ccc(Cl)cc1NC(c1nnnn1C(C)C)(C)Cc1nc(O)n[nH]1 C1(CNC(CC(CN(C)C)C(F)F)=O)(CO)CC12CCN(C(=O)CNC=O)CC2 c1(C(N(C)CCN(C)C(C2(C)CCS(=O)(=O)CC2)=O)=O)cnc2ccnn2c1N C1(C(N(C)CCNC(c2ccc(CO)o2)=O)=O)Cc2c[nH]cc2S1(=O)=O Cc1cccc2c1ccn2CC(=O)NC1COC2CN(C(C3CC3F)=O)CC12 C1(C)(C(N2CCCC(C(=O)NCCC(C)C)C2)=O)CCCN(c2ccccn2)C1 C1(C(N2CCC(N(C)C)(CC)C2)=O)CN(C(=O)CC2CCCC2O)CC12CCC2 C1(C(=O)OC)CCCCC1.c1(C=O)coc(N(C)C)n1.C(=O)CC1CCC1.N c1(SC)ccc(Cl)c(C(N2CCC(N(C(=O)C(C)Cc3ccnn3C)C)C2)=O)c1 N1(C(CCC)=O)CCN(C(c2ccccc2COC)=O)CC(F)(F)C1 N1(C(c2c(OC)nsc2)=O)CCC(NC(=O)C(C)Cc2ccncc2)CC1 C1(C(=O)NC2CN(C(c3[nH]c(=NC)sc3)=O)CC2C)CC2(CCC2OC)C1 N(C(=NCc1cccc(F)c1)NCC1(C)CCOC1)C(COC)C CCC(O)C(F)(F)C(=O)NC1CCN(C(c2cnc(CO)nc2C)=O)C(C)C1 C1(NC(C2(C(N(C)C)=O)CC2)=O)CC2CC1N(C(C1(C)CCN(C)C1)=O)C2 N1(C(c2ccc(N)c(C)c2Cl)=O)CCN(C(=O)Cn2cccc2)C2(CCC2)C1 C1(NC(c2cc(C)c(C)nc2)=O)CC2CN(C(C3C(C)(C)OC3(C)C)=O)CC2C1 C(=O)(C(C)(CNC(c1c[nH]c(=S)cn1)=O)CC)N1CCCC(CCC=C)C1 c1(C(C)(C)C)ccccc1CC(=O)NCCNC(c1ccccc1)=O.C(CO)S c1(C(=O)OCC(c2ccc(C(C)C)cc2)=O)ccnc(S(N)(=O)=O)c1 C1(C(N(CCCCC)Cc2ccccc2)=O)CC(C2CCNCC2)CN1 C1(NC(C(COC)O)=O)CCC2CN(C(c3cc(Cl)nnc3Cl)=O)CC2C1 C(=O)(C1=CC2CC=CCC12)NCC1CC(NC(c2ncn(C)c(=O)c2)=O)C1 C1(C(=O)NC(COC)CNc2cc(C(N)=O)ncn2)CC2(CC(=O)N2)C1 N1(C(c2cc(C(C)=O)c(F)cc2)=O)CCC2(C1)CN(C(=O)CCOCC(F)F)C2 c1(C(CN(CC)Cc2ccccc2)C)ccc(C(C)(C)C)cc1 c1(C(=O)NCC(=O)NCC2CC(F)(F)CO2)ccc([N+](=O)[O-])cc1 C(C(C)(C)C#CC(=O)N(CCC(C)C)C)NC(c1c(CC)cccn1)=O C(C(=O)NC1CCCC1)(C1=NOC2COCC12)NC(CC)CC#N N1(C(Cc2cn(C)nc2Cl)=O)CCC(NC(c2cc(Cl)cn2C)=O)C(C)(C)C1 C1(C(N2CCC(CC)C2CNC(C2CSCCS2)=O)=O)CCC([N+](=O)[O-])CC1 CC(C)C(O)CC(=O)NCCCN(c1ccc(C(=O)O)c(C(F)F)n1)C(C)C CCN=c1[nH]c(C(N2CCN(CC(C)(C)NC(c3ccnn3C)=O)CC2)=O)cs1 c1(C(=O)NCCNC(c2n(C)nc(C)c2I)=O)cc2ncccc2[nH]1 C=CC(C)(C)CC(=O)N1CCC(NC(c2ccc(Cl)c(CC)c2)=O)CC1C C1(C(=O)NC2CN(C(C3CC3c3cccs3)=O)CC2O)(OCC)CCSCC1 C1(CC=C)(C(N2CCC(C(C)(C)C)CC2)=O)CCN(C(=O)C(O)CSC)C1 c1(C(=O)NC2(CC(=O)NCCCn3cccn3)CCC2)ccc(F)cc1 N1(CCC=O)CCSC(C)(C)C1.CC1=NOC(CC(=O)NCCC2CCC2)C1.N C(CC)(CCC(=O)N(C(C)CC)C)NC(C(C=C)C)=O CC1CCn2cc(C(=O)OCc3nocc3C(C)(C)C)nc2C1 N1(C(c2ccccc2)=O)CCN(C(=O)Cc2ccn(C)c2)CC1C(C)C.COC C1(C(=O)NCc2ncc(Cl)cn2)CC(F)CN(Cc2ccc(Br)[nH]2)C1 Cc1cc(C(F)(F)F)ncc1C(N1CCC(O)(CC)C1)=O.C(=O)C(C)(C)CO.N C1(CC)CCN(C(C2CC(C)(C)C2)=O)CC1.c1(C(=O)N)scnc1C.C(C)=O C1(C(=O)NC(CC#CC)C)COCCN1C(c1ccc(CCO)cc1)=O C(=O)(C1=CCC(NC(c2ccsn2)=O)C1)NC(CCOC)CO C1(CNC(=O)Cc2cc[nH]n2)CC2(CCN(c3ccnc4ncnn34)C2)CO1 N1(C(C2(OC)CC(C)C2)=O)CC2(CNC(C3CC=CC3)=O)CCC1CC2 C1(C(=O)NCCC2N(C(CSC(C)C)=O)CCCC2)CCC2(CCOCC2)CO1 c1(C(=O)NCC(CN(C(C(F)=C(C)C)=O)C)O)ccc2cccnc2c1F Cc1c(F)cc(CN2CC(CO)(NC(c3cc(Cl)c(F)cc3F)=O)C2)cc1Br c1(CC(=O)NC(C2CCCCO2)C(=O)O)ccc(S(=O)C2CC2)cc1 N1(C(c2c(C)noc2C2CC2)=O)CC2CCC(C1)C(NC(=O)Cn1cnnn1)C2 c1(N(CC(=O)NCC(CC)NC(c2cc(C)c[nH]2)=O)C)ccnc(Cl)n1 C(=O)(CC(F)(F)C(F)F)N1C(C(=O)NC(C(=O)OC)C)CC1 C12(C(=O)NC3CC(CNC(C4(OC)CCCCC4)=O)C3)CCCCC1OCC2 CC(CCC(C)(C)C)Nc1cc(N2C3CCC2COC3)nc(C(F)(F)F)n1 C(=O)(CCC(=O)NN(C)C)NC(CC1CN(C(c2cc(C)c(F)cn2)=O)C1)C n1(CC(=O)NC(CC=C)CNC(C2CC3CCC2O3)=O)ccc2cc(F)ccc12 N1(C(CC)=O)CC(N=[N+]=[N-])CC1C(N1CC(CS(C)=O)C1)=O.C(=O)(NC)N N1(C(C(C)OCC(C)C)=O)CC2CCCC2(NC(c2csc(=N)[nH]2)=O)C1 C=CCC(C(=O)N1CC2(CNC(=O)C3=CCSC3)CC1CCO2)C(C)C c1(C(=O)NC(CCSC)C(N2CCOCC(O)C2)=O)cc(C)cc(O)n1 c1(C(=O)NC(CSCC)C(=O)NCCCCCO)cccc(C#N)c1 C1(NC(C(CCC)N(C)C)=O)(CNC(c2cn(C)ccc2=O)=O)CCCCC1C C(=O)(C(F)(F)C(F)F)N(CC(CC)NC(c1cccc(-c2ccco2)c1)=O)C N1(C(C2CN(C(C(SC)SC)=O)CC2F)=O)C2C=CCC1CC2 c1(C(=O)NCc2nccc(C(=O)NCCCC(=C)C)c2)cn(C)ccc1=O CC(C(=O)N1CC(O)C1)C(F)(F)C(F)F.n1(CC=O)cnc(C(F)(F)F)n1.C c1(C(=O)NC2CN(C(C(CC)NC(C)=O)=O)CC2C)cccc2c1COCC2 c1(C(C)C)ccc(C(=O)N)c(F)c1.C1CC(F)CN1C(=O)CN1CCOC1=O.C N1(C(C(COC)O)=O)C2CCC1CC(N(C)C(C1CCC(=O)N1)=O)C2 C(=O)C(C)(O)C(F)(F)F.Cc1cnc(C(F)(F)F)c(C(=O)N(CC(O)C)C)c1 CC1=C(C(=O)NC2CC3C(NC(=O)C(C#N)C(C)C)C3C2)COCC1 CCCCC(C(=O)N1CCCC1CN=[N+]=[N-])NC(C1CCCCC(=O)C1)=O C(=O)(C(C)CC1CCCC1)N.c1(C=O)[nH]ccc1C.C(C(C)C)N(CC)CC c1(C(=O)NCCCOCCCNC(c2cccc(F)c2)=O)cccc2nonc12 C(=O)(C(O)C(C)(C)C)N1CCC(CCC(=O)Nc2c(C)noc2)C1 CCC(CC)CCC(=O)NC1CC(NC(C2CC(CF)C2)=O)C1 C1(O)(C(C)(C)CN2CC(n3cc(-c4ccccc4)nn3)C2)CCCCC1 C1(CC)(NC(=O)CS)CCCN(C(c2sccc2C(C)C)=O)C1.CC(N)=O CC(C)CC(C(=O)N1CCCC(C(=O)NCC(=O)NCCO)C1C)C(C)C Cc1ccc(C)c(C(=O)NCCNC(=O)CCN2CCCCC2C)c1O C(=O)(CCC(C)(C)F)NCCN(C(Cn1nnc(C)n1)=O)C1CC1 N1(C(c2cnn(CCO)c2)=O)CCCC(c2cn(CCF)nn2)C1 C1(CCOC)(C(=O)N(CCC)C)CCN(C)CC1.c1(CC(=O)N)csc(C)n1 N1(C(C2C(CCC)C2)=O)CCN(C(c2ccc(-c3cnn(C)c3)cn2)=O)CC1C C1CCN(C(C23CC2COC3(C)C)=O)C(C)C1.c1(C(=O)OC)ccc(C=O)o1.N C(=O)(C1=CCC(C)(C)CC1)N1CCN(C(c2cc(OC)cc(C)c2)=O)C2C1CC2 C1(N(C(=O)CN(C(=O)CCc2ncnn2C)CC2CC2)C)CC2CC2C1 c1(C(N2C3CN(C(C(c4ccccc4)=O)=O)C(C3)C2)=O)ccc2c(c1)CCCS2 C(c1ccc(OC)cc1)=CC(=O)NCCCNC(c1nc(CC)sc1)=O c1(-c2nc(C(CC)NC(=O)NCC3(C(=O)O)CC3)on2)ccc(F)cc1 c1(C(C(=O)OC)NC(=O)CC2CCC2O)ccc(CC(C)C)cc1 C1(CCC(=O)NCC(=O)NC)CCCCN(C(c2ccc(CO)s2)=O)C1 Cc1ccnc2[nH]cc(CNC3CCCC(CNC(=O)OC(C)(C)C)C3)c12 c1(CC=O)cccc([N+](=O)[O-])c1.C1(CC)(C(N2CCC2)=O)CCCC1.CCO C(N=C(NCc1ccnc(OC(F)F)c1)NC1CC1C)c1cc(C)oc1 C=CC1CN(C(=O)CC(O)CC)CC1NC(=O)CCc1ncc[nH]1 N1(C(c2ccc(C(C)=O)o2)=O)CCCC12CCN(C(C1CC1c1cccs1)=O)C2 C1(CNC(C(C)OC)=O)CC2CCC1CC2.N1(CC=O)CCC(=O)NC1=O.N C1(NC(C2CCCC2O)=O)CCCCC12CCN(C(=O)Cc1ccc(F)cn1)C2 C(=O)(C(C)CC(N)=O)NC(C(=O)N(CC#C)C)Cn1cccn1 C1(OC2CN(C)C2)CCCCN1C(=O)COC1CC1(F)F C1(C(=O)NCc2nccs2)(OC)CCN(C(=O)CC2CCCO2)C1 c1(C(N2CC(c3nc(C)cc(C(=O)OCC)n3)C2)=O)cc(Cl)nc(Cl)c1C C=C1CCN(C(c2cc[nH]c2)=O)C(C(=O)NCC23CCN(CC2)CC3)C1 CC(C)(C)C(C#N)C(=O)N1CC(NC(c2ccnc3cc[nH]c23)=O)C(O)C1 C1(CC(=O)N(CC)C)CCS(=O)(=O)C1.CC(Cc1cnc[nH]1)C=O.CCC.N n1(CC#C)cccc1C(=O)NCc1cc[nH]c1C(=O)NCC(C)C(C)O N1(C(C(C)SC)=O)CCc2c(C(=O)NCC(=O)NC(C)(C)C)cccc2C1 Cc1ccnc(C)c1C(=O)N(C1(CC(=O)NCC2(C)CCCCCC2)CC1)C C1(NC(CC)=O)CCC(O)CN(C(=O)C(C)SC2CCCC2)C1 C(=O)CC(C)C(F)F.c1(SC)c(C(=O)NCC2CC2)cnn1C.C(N)=O.C S(=O)(=O)(c1c[nH]ccc1=NCCSCCO)NC(C)Cc1ccccn1 c1(OC)ccc(F)c(C(=O)N(C2CN(C(=O)C#CC(=O)N(C)C)C2)C)c1 Cc1ccc(C(=O)N)cc1F.C1(O)(CC(N2CCC3CC32)=O)COC(C)(C)C1.C C(=O)(C1=CC2CCC(C1)C2)N1C(C(=O)NCC2CCCOC2)(CC)CCC1 C1(NC(=O)CN2CCCCC2)CC2(C1)CC2NC(C1CCC(F)(F)C1)=O CN=c1[nH]cc(C(=O)NC2CC3(C2)CC3C(=O)N(C(C)CC(N)=O)C)s1 C1(C(=O)NCCCN(C(C)=O)C)CC12CCN(C(=O)CCCCC#N)CC2 n1(C(C)C)ccc(C(=O)NC(CNC(=O)C(C)(C)c2ccsc2)CO)n1 c1(COCCNC(=O)NCc2cccc(OCF)c2)ccc(Br)cc1 CC1CC=C(c2ccc3nc(CC(N4CCCCC4CCO)=O)sc3c2)CC1 Cc1ccc(=N)[nH]c1C(=O)NC1CC(C)(NC(C)=O)C1 C1(C(=O)NC2(C3CCCCN3C(=O)CC(C)C)CC2)(OC)CCS(=O)(=O)C1 c1(C(N(C2CCN(C(C3CS(=O)(=O)C3)=O)CC2)CCO)=O)[nH]cc2c1CCC2 CCC(C)C(O)C(=O)NCC12CC(NC(=O)CCc3cn(C)nn3)(C1)C2 C1(=CCNC(C2(C(N)=O)CCC2)=O)CCN(C(=O)C(F)C2CCOC2)CC1 CC1CN(C(C2CN(C)C2)=O)CCCN1C(=O)CC#N C1(NC(c2cnco2)=O)CCOCC1C(=O)N(C1CCOC1)CCF c1(C(=O)NC2CN(C(C=COCC)=O)CC2O)cc(C)cc2nc[nH]c12 c1(C(N2C3CCC3CC2)=O)cc(C)cc(F)c1N.C1(C(=O)N)(COC)CCCO1 CC1(C)CC(NC(=O)CCc2ncccn2)CN1C(C1CC2CC2C1)=O C12(CNC(=O)CSc3nc[nH]n3)CCCC1CCN2C(=O)CCn1cnnn1 N1(C(Cc2c(C)cc(C)s2)=O)CCN(C(=O)Cc2cnns2)CC1C C#CCC(CC#C)C(=O)NCC(C1CCCC1)NC(=O)CCC(F)(F)F C(=O)(CCCS(=O)(=O)c1ccccc1)NCCNC(CC1(C=C)CC1)=O C1(CNC(C(C)=C2CCC2)=O)CC2(CO1)CN(C(c1ccn3c1CCCC3)=O)C2 N1(c2c3ccn(C)c3ncn2)CCc2nn(C)c(-c3ccc(C(F)F)cc3)c2C1 c1(NC(CC2OCCN(CC)C2)=O)cc(C)c(C(=O)OC)c(C)c1 N1(C(c2c(C)ncn2O)=O)CC(NC(c2cnc(O)nc2O)=O)CC2(CC2)C1 C1(C(C)(C)CNC(C2CCCS2)=O)CCCCN1C(=O)C(F)=C1CCCC1 C(=O)(C(F)(F)CC)N(CC=CC(NOCC#C)=O)C c1(C(=O)NC(C)C(CO)NC(=O)CSc2ccccc2)coc2c(F)cccc12 N1(C(CC(CC)(C)C)=O)CCC2CN(C(=O)C(n3cc(Br)cn3)C)C2C1 N1(C(C(C)SC(F)(F)F)=O)CCC2CC(NC(=O)CC3(C)CC3)CCC2C1 Cc1cc(CNC(C2CCCCC2(C)NC(=O)CN2CCCC2=O)=O)cnc1F C(=O)(C1=Cc2cc(Cl)ccc2OC1)NCC1C(NC(CCC=CCC=C)=O)C1 c1(OC)ccc(C)cc1C(C)NC(=O)NCCCC(C)O CCCC(C(=O)NC1CC(NC(=O)CCNC(N)=O)C1)N(C)C c1(NCCN(CCCO)C)[nH]c(=NCc2nc(CO)cs2)nc2scnc12 c1(C(N2CCC(C#N)(NC(c3cc(Br)ccn3)=O)C2)=O)cn2ccc(Cl)cc2n1 S(=O)(=O)(c1cc(C)cnc1N(CCCN(C)C)C)NC(CC)C(C)C C1(NC(=O)NC(c2cn(C)nn2)(C)C)CCC(OC(F)(F)F)CC1.c1ncon1 c1(CNCc2n(C)cnc2Br)ccc2cnn(C)c2c1 C(C1C(C(N2CCCC2C2CCN(C(c3cnns3)=O)C2)=O)C1(C)C)=C(C)C C1(C(=O)NC)CCN(C(C2CCCN(C(c3cc(CO)ccn3)=O)C2)=O)C1C CCN=c1ccc(CNC(c2coc(CNC(C)=O)c2)=O)c[nH]1 C1(CNC(CCN(C)CC)=O)CC2CCC1N2C(c1cc(=O)n(C)cn1)=O N1(C(CC2N(C(c3ccc(C#N)s3)=O)CCC2)=O)CC2CC=CCC2C1 C(=O)(C#CC1(C)COC1)NC1(C(=O)NC2C(OC)CCC2)CCSC1 c1(CC)cnoc1C(N1CCC1CNC(=O)C(C)OCOC)=O C1(CC(=O)N(C2CC(Oc3ccccc3)C2(C)C)C)CCCCC(=O)N1 c1(C2OCCN(c3nc(C=Cc4nc(C)sc4)[nH]n3)C2)cccc(Cl)c1Cl c1(CN2C3C(C(=O)NCc4c(C)ccnc4C)CC(C3)C2)ccc(F)c(C#N)c1 C1(C(N2C(CNC(c3n(C)ncc3C(N)=O)=O)CSCC2)=O)CC2CCCC2C1 C(=O)(C1CCCc2nn[nH]c21)NC(C1CN(C(C(C)OCC2CC2)=O)C1)C C1(C(=O)NCCCCNC(=O)CCC2CC2(Cl)Cl)CC2(CCOCC2)C1 C12(C(NOC(C)C)=O)CCC(CN(C(C3(C#N)CC3(C)C)=O)C1)C2 N1(C(c2cc(C)on2)=O)CCC(O)(C(C)C)C1.C(c1ccc(Cl)s1)=CC(=O)N N1(C(CCCNC(=O)OC)=O)CC2CC2(NC(=O)C(c2ccc(F)cc2)F)C1 N1(C(CC(CC)O)=O)CCn2ncc(CNC(C3CC34CCOCC4)=O)c2C1 N1(C(c2c(Cl)nc(N(C)C)s2)=O)CCC2(CO)CN(C(=O)CC(F)F)CC2C1 C(=O)(CC(O)C(C)CC)NCCCCCC(=O)N(CC=C)CCC C1(CC=C)N(CC)CC1(C)C.c12cccnc1Cn1cc(nn1)C1CCN1C2=O C1(CNC(c2c(C)nc[nH]2)=O)C(O)C(O)CN1C(c1cn(C)nc1C)=O c1(N(CC(C)C#N)CC)ccc(Cl)cc1F Cc1cc(C(N2CC(NC(C3CC4OCCC4O3)=O)C2)=O)cc2c1NCCC2 C12(NC(C3CCC(C)N(C(=O)CCC4(C)N=N4)C3)=O)CC1COC21CCC1 C1(C(=O)OCC(C2(C)CC2)O)CC12CCN(C(=O)OC(C)(C)C)C2 c1(C(C)C)nc(NCC2CCC=CCCC2)cc(=NCc2c(F)cccc2Cl)[nH]1 C1(C(N(CCCNC(c2c(C)snn2)=O)CCO)=O)CCC2C1C2(F)F C1(C(=O)NCC2N(C(C3CCC(C)C3)=O)CC(C)(C)C2)CN2CCCN1CC2 C(=O)(CC1COc2ccccc21)N1CCN(C(C)=O)CC1.C123CC(C1)(OC2C)CN3 C(C)(C)(CC(=O)NC1CCN(C2CC2)C1=O)NC(CC1C(C)OCC1)=O O=C(N=c1ccn(C2CN(C(c3ccsn3)=O)C2)[nH]1)c1ccc(S)cc1 C1(NC(c2c(C)c(F)ccc2)=O)CN(C(=O)CC(C)C)CC(C)(C)C1.C(N)(=O)N Cc1ccc(C(N2CCOC(C3CN(C(=O)C(C)C(C)C)C3)C2)=O)nc1O C(=O)(C1=CC(O)CC1)N(C)CC1CCCCO1.C(=O)C(C1CC1)C1CC1.N C(=O)(C(O)CC(C)C)NCC(C)N(C(c1ccc(SC)cc1)=O)CC C(C(C(F)(F)F)c1ccon1)NC(c1ccn(C(C)C2CC2)n1)=O Cc1ccc(C(N2CC(CNC(c3ccccc3SCCO)=O)C2)=O)cc1 C1(C(=O)NCC(C)NC(c2nn(C)c3c2CSCC3)=O)C2Cc3ccccc3C12 N1(CC)CCCN(C(C2CCCCCN2C(=O)CC2(CSC)CC2)=O)CC1 C1(NC(CC(C)N(C(CC(C=C)C)=O)C)=O)COC2(CCC2)C1 C=CCC(CO)C=O.n1(CC(N2CCC2)=O)cc(-c2ccccc2)cn1 C(=O)(C1=NOC(C)C1C)N1CC(C(N(C)Cc2c(C)occ2)=O)C(C(C)C)C1 N1(C(c2c(NC)cnc(Cl)c2)=O)CC2CCC(C1)C(NC(=O)Cc1ccsc1)C2 C1(OC)CCN(c2ncnc(NCCC(=O)NCC(C)C)c2C)CC1C C1(NC(c2c(C(C)C)onc2)=O)COC2(C1)CN(C(C1(C)CC(F)C1)=O)C2 C1(CO)COC2CN(N3CCOC(c4cccc(OC(F)(F)F)c4)C3)CC12 c1(C(=O)NC(COC)CNC(c2csc(C)c2)=O)cccnc1C1CC1 c1(C(NOC(C=C)C)=O)coc(CNC(c2csnc2OC)=O)n1 [N-]=[N+]=Nc1cncc(C(N2CCC(F)(F)C(CNC(C3CCCOC3)=O)C2)=O)c1 c1(CCC(=O)NC2C(NC(COC(CC)C)=O)C2)ncn(C)c1C CC(C)C(C)CNC(c1ccc(C)cc1)=O.C(=O)C(N)=O.C(=O)C1CC1 CCS(=O)(=O)C=CC(=O)NC1(C2CCCN2C(=O)C(C)N2CCC2)CC1 Cc1cc(N)ccc1C(N1CCCCC(NC(=O)COC2CC=CC2)C1)=O c1(OC)c(C(=O)NC2(CNC(C3(F)CCOC3C)=O)CCCC2)cnn1C c1(OCC)cccc(C2(C(=O)NC(C)CN(C)C(C3CCO3)=O)CC2)c1 C1CC2(C1)CC2C=O.C(=O)(COCC(=O)N(C)CCOCC)NC C1(N(CCCCC(=O)O)C)CCCN(C(=O)NCc2cccnc2)CC1 C1(O)(CC)CCN(C(C2C=CC2C=O)=O)C1.C(CCC=O)OCCOC.N C(N=C(NC1CCC1)N(C)CC1(CO)CC2CCC1C2)C1C(=C)C1 CC12CC3CC(CC(=O)NC4C=CCC4)(C1)CC(F)(C3)C2.C(=O)C1CC1.C C(=O)(C1=C(Cl)CCC(C)C1)N1CC(C(C)C)N(C(=O)CS(=O)(=O)N(C)C)CC1 C1(CC(=O)N(C(C)CNC(=O)C=C2CCC2)C)Sc2ccccc2NC1=O C1(C(N2CC(C)C(CNC(=O)C(C)(C)O)C2)=O)C2(CCC2)C12CCC2 CC1(C)CN(C(C(=O)NC2CC(F)(F)C2)C2CC2)CC(CCO)O1 C12(C(N3C(C(=O)N)CCC3)=O)CC1CN(C(=O)Cc1cccc(Cl)c1)C2.CC c1(C(=O)NCC2CCOC2c2ccncc2)noc2c1CCCCC2 c1(C(N2CCC(C(=O)N)C2)=O)cc(O)c(Br)c(O)c1.Cc1cccc(C(N)=O)c1 N1(C(CC)=O)CCN(C(=O)CNC(=O)C(c2ccc(Cl)cc2)C)CC1 N1(C(C=CC=CC)=O)CC2CCN(C(c3csnc3Cl)=O)CC12 C1(C(=O)NCCCn2cc(CNC)nn2)CC(C)S(=O)(=O)C(C)C1 C1(NC(Cc2nc(CC)sc2)=O)CCN(C(C2CSC2)=O)CC1C C(=O)(CS(=O)C(F)(F)F)N.CC(C)CCCNC(c1cnc(C(N)=O)cn1)=O C1(NC(C(CC)CCOC)=O)CCN(C(C2(C)CC2)=O)CCC1CO N1(C(=O)C=Cc2cnc[nH]2)CCN(C(=O)CC2C=CCC2)CC(CO)C1 CS(=O)CCC(=O)NCCOC1CN(C(=O)C(c2cccc(N)c2)O)C1 C(CCC(O)C(=O)N1CC2CC(C)C2C1)NC(Cc1c(C)nsc1)=O C(=O)(N=c1cc2n([nH]1)CCCC2)C1C(NC(C2CN(C(C)=O)C2)=O)CC=CC1 C=CC(C)CC(=O)N(CC(O)CNC(c1ccc(-c2ncc[nH]2)nc1)=O)C C1(CC)(CC)CC(NC(c2ccc(C)c(C)c2)=O)CN1C(=O)CC.C(N)=O C1(CNC(=O)CC2CC3(CC3)C2)COCCN(C(=O)CCc2cccnc2Cl)C1 N1(CC(C)C)CC(C)Oc2cc(C(F)(F)F)ccc21 CC(C(=O)NCc1cn(C2CN(C(c3ccc(Cl)cn3)=O)C2)nn1)C(C)(F)F c1(CNC(CCCNC(COCC(=C)C)=O)=O)ccc(CO)cc1 C1(NC(=O)CCC(F)(F)F)COC2(CCCN(C(c3cc(F)ccc3O)=O)C2)C1 CN1CC23CCCC2(CN(C(C2C4CN(C(=O)C(N)Cc5cnc[nH]5)CC24)=O)C3)C1 C1(COC)CCCCC1.C(=O)(C(C)=C1CCCC1)N(C1(CC=O)CC1)C.N C=CCC(C)(C)CC(=O)N(CC(C)CNC(=O)C(CC)Nc1nc(C)cs1)C C1(NC(=O)C=CC(F)F)CCCC(C(N2CC(O)C(O)C2)=O)CC1 N1(C(C2(CC=C)CN(C(=O)Cn3nnnc3C)C2)=O)CCCC(CO)C1C c1(-c2ccccc2)nc(-c2nccs2)nn1CCc1ccncc1 C(CC)(C(=O)NC(CNC(=O)C=CC1CC1)C1CC1)OCC C1(NC(C(C2CCCCC2)OC)=O)CC(C)CN(C(c2cnc(CN)nc2)=O)C1 C1(CC(=O)N(C(C)C(N2CCC(C)(CC)C2)=O)CC)CCC(=O)N1C N1(C(CCc2cc(C)nc(C)c2)=O)CC2(CCN(C(c3cccnc3)=O)C2)C1 C1(C(=O)NCCOCC(=O)NCC2CCCSC2)CCC2(CC1)CC2 c1(C(=O)NC(CN(C(=O)C(F)CC2CC2)C)(C)C)ccc2c(n1)CCC2 c1nccc(C(F)(F)F)n1.c1(C(=O)NCCC2(CN)CC2)ccc(F)cn1 C1(C(=O)NC2CCN(C(CC(CC)C)=O)CC2)CC2CCCN2C(=O)N1 Cc1ccc2c(C(=O)NC34COCCC3CN(C(C3(C)CCC3)=O)C4)csc2c1 c1(C(N2CCC(N(C(CCC(C)OC)=O)C)C2)=O)cc(Br)n2c1CCC2 S(=O)(=O)(c1cccs1)NC(C)C(=O)N.C1CCCCC1.C(=O)CC1CCC1.C c1(CCNCC(c2cn(C)nn2)C)cccc(C(=O)O)c1.c1coc(C2CC2)n1 c1(C(=O)NC(C2CCN(Cc3cccc(Br)c3F)CC2)C)cc(Cl)cc(Cl)c1F Nc1cc(C(F)(F)F)cnc1C(=O)N.C1C2CCC(C2)N1C(C1CCCSC1)=O C1(C(=O)NC(CC(C)(C)C)c2cccnc2)CC2(CCC2)C12CCC2 Cc1cc(C(N2CCN(C(C3CC4CC3CC4O)=O)CC2C(F)F)=O)cc(F)c1 Cc1ccc(C)c(C(N2CCCCC2CC(=O)NC2(c3nn[nH]n3)CC2)=O)n1 C1(CCNC(c2ccc(OC)o2)=O)CCCN(C(=O)CC2C=CCC2)C1 C=CC(C)(C)CC(=O)N1CC(NC(C2(C(F)(F)F)CC=CCO2)=O)CCC1C N1(C(C2C(C)(C)CO2)=O)CC2CCC1CN2C(=O)CCc1ccc2c(c1)CCO2 N1(C(Cc2c(C)con2)=O)CC(C(=O)NCCc2ccc(F)cc2)C2(CC2)C1 c1(CC(=O)NC(C)CNC(C2CSC2)=O)ccc2c(c1)CCCC2 C1(C)(C(=O)NCCC(C)NC(=O)CC)CCCCCCC1.C(=O)CC(C)(C)C.N c1(N2CCCCC(NC(C(C)C(=O)OC(C)(C)C)=O)C2)ccc(F)cc1[N+](=O)[O-] N1(C(CSC)=O)CC(NC(=O)C(C)(C)COC2CCCC2)CC(O)C1 c1(CC(N2CC=CC2)=O)ccc(-n2cncn2)cc1.Cc1nnnn1CC(=O)NC N1(C(C(C=C)C)=O)CCC(CO)C(NC(=O)COCC(=O)OC)C1 Cc1c(C(=O)NCc2nocc2C(=O)NC(c2cn[nH]c2)C)c[nH]c1C#N C1(NC(c2c(C)cnnc2)=O)CCN(C(=O)CCCn2cccc2)CC1O c1(N2CCC(C3(NC(c4cc(SC)oc4C)=O)CC3)C2)ncc([N+](=O)[O-])cc1F C(=O)(CCC(C)C)NCCCNC(c1c(CC)nnc(C)c1)=O.C(C)=O.N c1(C(=O)NCc2ccc(C)cc2Br)cc2c(Br)csc2[nH]1 C=CCC(C(=O)N1CCCC(CNC(=O)C=CC2CCOCC2)C1)C(C)C N1(C(c2ccc(C)cc2N)=O)CC2(C1)SCCC2.C(c1cnc(C)s1)=CC(=O)N N1(C(C=C(CC)CC)=O)CC2CC(NC(c3cn4ncccc4n3)=O)CC2C1 CC1(C)CC(CC(N2CCCC(NC(=O)Cc3csc(Cl)c3)C2)=O)CC(C)(C)O1 C1(OC)CC(c2nnnn2CC2CCOC2)(NCCc2nncn2C)C1 C(=O)(C(C)CS(C)(=O)=O)NC1CC2(CN(C(C(c3cccnc3)OC)=O)C2)C1 c1nc(C)cc(O)n1.c1(CC)conc1C(N1CC(OCCC(=O)NC)C1)=O CN1CC(C(=O)NC(CC2CC2)CC(=O)NCC2(CCO)CC2)NC1=O C1(CNC(C2(C)COC2)=O)COC(C)(C)CN1C(C1(F)CCOC1)=O C(=O)(CCCS(C)(=O)=O)NC(CC)(C)CNC(=O)CC1C=CCCC1 C=CCC(C)(C)C(=O)N1CC(C(=O)NC(CN(C)C)CC(C)C)OC(C)C1 C1(N(C2CCCC2)C(C2CCCC2OC)=O)CCN(CC(=O)N(C)C)CC1 C1(NC(c2cc(C(F)F)[nH]n2)=O)COCCN(C(C2CCC(F)(F)C2)=O)C1 C12(CNC(c3cnc(OCC)nc3)=O)CCC1CCN2C(C1CC=CC1)=O Cc1nc(CN2CCC(C3CCCCN3C(=O)C(C)CO)C2)c2ccnc-2[nH]1 C1(C(N(CCC(N2CC(C)(CO)C2)=O)C(C)C)=O)CCC(=O)NC1 N1(C(C(C(CC)CC)F)=O)CC(CO)C2(C1)CN(C(=O)CN(C)C(N)=O)C2 N1(C2CCN(C(c3ccc(F)s3)C(=O)NCCSC)C2)CCCOCC1 C(=O)(CS(=O)(=O)NC1CN(C(=O)OC(C)(C)C)C1)OCC c1(C(=O)N)cccc2c1COCC2.C(C(=O)N1CC2CC2(C)C1)(C(C)C)SCC N1(C(C2ON=C(C)C2)=O)CCOC2CN(C(c3cncc4nc(C)[nH]c34)=O)CC12 C(CCC(N)=O)(C(=O)NCCC1(NC(=O)CC2CC=CC2)CC1)N(C)C Cc1cc(CCNC(=O)NC(C)C(c2ccc(Cl)cc2)O)c2cn[nH]c2c1 c1(CC2CCCN(CCCN3CC(=O)N(CC)C3=O)C2)ccc([N+](=O)[O-])cc1 c1(-c2nc(C(C)OCC)nn2C(COC)COC)cc2c(F)cccc2s1 N1(C(C(CC)CC)=O)CCN(C(C2(CN(C)C)CCCC2)=O)CC(O)C1 N1(C(C(CCC)CC)=O)CCN(C(c2c[nH]c(C(=O)OC)c2)=O)CCC1C N1(C(c2sc(CC)c(C)c2)=O)C2CCC1CN(C(c1c(C)cccc1O)=O)C2 C(=O)(CCC(=O)c1ccccn1)N1CC(C)(NC(C(C)Cc2ccccc2)=O)C1 c1(OC)nc(C)cc(=NC2CCCC2C(=O)Nc2ncc(F)cc2F)[nH]1 C(=O)(CCCCC(=O)N(CCC(C)NC(c1ccc2nsnc2c1)=O)C)NC N12CC3CCC1CN3C(=O)C2.c1(N2CC3CC(C)C3C2)cn2cccnc2n1 CC(C)(C)C(CNC(=O)Cc1cccs1)C(=O)NCC1(O)CCCC1(C)C N1(C(CSC)=O)CC(CNC(C2CC3CCCC(C2)C3)=O)CC(C)(C)C1 C(=O)(CCN=c1ccc(C)c[nH]1)N1CCC(CC=C)(NC(C2CCC(C)O2)=O)C1 N1(C(C2(C)CC(O)CN2C(c2ccc(N)cn2)=O)=O)C2CCCC1COC2 C1(CCC(=O)NC(C2CC2C(=O)NC2CC(Cl)(Cl)C2)C)CCCN1C C#CC1(O)CCN(C(C2CCCC(C)C2)C(=O)NCCOC)CC1 N1(C2CN(C(c3cn(C4CCOC4)nn3)=O)C2)CCC(CO)CC1 C1(COC)CN(C(c2nccnc2C(N)=O)=O)CCN1C(c1snnc1C)=O CCS(=O)(=O)c1ccccc1C(N1CCC1CNC(=O)Cc1cnccc1C)=O C1(NC(C(c2ccc(F)c(F)c2)C)=O)CC2CC1N(C(=O)C=CC1CC1)C2 Cc1cccc(C(F)(F)C(=O)N(CCCN(C)Cc2ccco2)C)n1 CN=c1nc(C(N2CC3(CCNC(=O)C#CC(C)(C)C)CCC2C3)=O)cc(C)[nH]1 C1(C(=O)NCC(=C)CCNC(c2cc(C(F)(F)F)n[nH]2)=O)CN(C)CCO1 c1(CC(=O)OC2CC2)oc2ccccc2c1SCCC1COC(=O)N1 CC1C(=O)N(C)CCN1C(C1CCCC(NC(=O)COC2CCCCC2)C1)=O N1(C(C2(N(C)C)CC2)=O)CC2CCN(C(=O)CCCCCNC(N)=O)C2C1 C(=O)(CC(C(F)F)NC(C1CC(C=O)C1)=O)N1CCCC(CC=CC)C1.O C1(C(=O)NC2C(CNC(c3cnc(O)s3)=O)CCC2)CCCC(F)(F)C1 C1(NC(CC2(N(C)C)CC2)=O)(CNC(C2CCCS2)=O)CCOC1 N1(C(c2c(CCC)n(CCO)nc2)=O)CCN(C(C2(O)CC(F)(F)C2)=O)CC1C C#CCC(CC#C)C(=O)N1CCC(C2CCCN2C(C2CN(CC(C)C)C2)=O)C1 N=c1ccc(C(N2CC3(C2)CN(C(=O)CN2CCC(CO)CC2)C3)=O)c(Cl)[nH]1 CN1CCN(CC(=O)NC2CCCC(NC(C3(C4CC4)CCCO3)=O)C2)CC1.OC CC1CN(C(c2ncn(C)n2)=O)CCCN1C(C1(C2CCC2)CC1(F)F)=O C1(CNC(C(COC)NC(=O)Cc2ccnc(F)c2)=O)CCC2(CC2)CO1 Cc1cc(C#N)nc(=NCC2(NC(c3ccc([N+](=O)[O-])c(Br)c3)=O)COC2)[nH]1 C(=O)(C1=CC(O)CCC1)NC1C(NC(C2CC(O)(CC#C)C2)=O)CCCC1 C(C(=O)N1CCC(F)(CNC(c2ccncc2Cl)=O)C1)(C(C)C)OCC C1(CCOC)CN(C(=O)CC2(O)CCC2)CCN1C(c1ccc(Br)o1)=O C1(N(CC)CC2CCCCN2N=O)CCC(N=c2[nH]c3ccc(Br)cc3s2)CC1 C1(CNC(Cn2c(C)nnn2)=O)CCCCN1C(=O)CC1CCCOCC1 C1(NC(c2n(CC)ccn2)=O)CCCCN(c2cc(Cl)nc(CS(C)(=O)=O)n2)C1 N12CCOC(C1)C2=O.C1(C(=O)OC(C)(C)C)CC(F)(C)C1.C(=O)C(N)=O CC1CN(C(C2CC(F)(F)C2)=O)CC2(CCN(C(=O)Cc3cn[nH]c3)C2)O1 Cc1nn(C)cc1CC1COCC1.C12(C=O)CC(n3cc(C4CC4)nn3)C1C2.N C1(C(N2CC3C(C)C3C2)=O)CC12CCN(C(=O)CC1CC(C)(C)CO1)CC2 C1(NC(N2C(C)C2=O)=O)CCCN(CC)CC1.c1(CC2CCCN2)scnc1C c1(C(N2CCCC(N(C(C(C)=C(CC)C)=O)C)C2)=O)cnc2nc(C)oc2c1 c1(C(N(CC(CNC(C(CCC)CC)=O)O)C)=O)cc2ccsc2c(O)n1 N1(S(CCCCC)(=O)=O)CCN(C(=O)NC2C3CC4C(C3)C24)CCC12CCC2 c1(C(N2CCOCC(CO)C2)C(=O)NCC(=C)C)cccc2cncn12 Cc1cc(C(=O)NCC2CC2NC(c2ccc(C(N)=O)nn2)=O)cn1C N(C)(C1CN(C(C2CC(C)C2)=O)CCc2ccccc21)C(Cc1cnc(C)s1)=O C1(Cn2cc(CN3C(=O)CCC3)nn2)CC12CCSCC2 C1(F)(C(=O)NCC(C)CC2CC2)CCCN(C(=O)CCC(C)(C)F)C1 N1(c2nc(CC)nc(C)c2)CCCC2CN(C(C3CCNC3=O)=O)CCC12 C(CO)(CCCCNC(C1(C)CNC(=O)C1)=O)NC(CCC=CC(C)C)=O N1(C(CN(S(CC)(=O)=O)C)=O)CCC2CCN(C(c3ncc(C)cc3C)=O)CC12 C1(C)(NC(C(CC(C)C)NC(C2CCC(C)(C)CC2)=O)=O)CCC(=O)NC1=O c1(C(=O)NC2(COC)CCN(C(c3ccsc3C)=O)C2)cccc(C)c1Cl C1(NC(C(C)SCCCC)=O)C=CCC1.c1(CC=O)nocc1C(C)C.C Cn1c2c(ccc1=O)C(NC(C)(C)CN1CCN(Cc3cn[nH]c3)CC1)CCC2 N(C(=NCc1ccc(-n2ccnn2)cc1)N1CCC(CC)C1)C1CC(OCC)C1 C1(CC(N2CCCC(Cc3nccs3)C2)=O)CC2OCCC2O1 N1(C(C2(c3cc(C)c(N)c(C)c3)CC2)=O)CCc2c(ncn2C)C1C C(C#CCCO)NC(C(C1CCOC1)NC(=O)CN1CCNC1=O)=O C(CC(CC)C(=O)NC1CCCN(C(C2(OC)CCOCC2)=O)C1)=CC N1(S(=O)(=O)Cc2ccc(Br)cc2)CCC2OCCCC2C1 C(=O)(CN1C(=O)COc2ccccc21)N1CCC(O)(C(N2CC3CC3C2)=O)CC1 C1(O)(CNC(c2ccc(C(CC)=O)cc2)=O)CCN(C(=O)C(O)C(F)F)CC1 C(C(C)C(=O)Nn1cnnc1C)N(C(c1ccc(OC)cc1)=O)C N1(C(Cc2cn(C)nc2)=O)CC2(CCNC(C3CCS(=O)(=O)C3)=O)CCC1C2 C=CC1(CC(N2CC(CC3CC3)C2)=O)CN(C(=O)CN(C2CCC2)C)C1 N1(C(c2c(C)c[nH]c2)=O)CCC(NCc2cnc(C(=O)O)nc2)CC1 C1(n2ccnn2)CCCN(C(=O)CCn2cncn2)C1.C(C(=O)NC)SCC=C C(C(=O)NC(C1CCN(C(=O)Cc2cnc(C)s2)CC1)C)(C(C)C)OCC C12(CN(C)C(C3CC3c3ccc(F)c(F)c3)=O)CC3CC(CC(C3)C1)C2 c1(NC(C)=O)ccc(NC(=O)CCC2CCCCN2C)c(O)c1 c12cnn3c(O)cc(nc13)CNC2=O.N1(CC)CC2CC(N)C2C1 c1(CC)cc(C(N2CC3CC3C2)=O)nn1C.n1(CC(=O)N)cnc(C(N)=O)n1 C(CN=c1[nH]c(N(C)Cc2cc(Cl)ccc2Cl)nc(=N)[nH]1)OC(CC)C c1(OC)cccc(C(=O)NCC2CCCCN2C(c2cncc(OC)c2)=O)c1C c1(C(N(CCOCCCN(C(=O)CCC2CCOC2)C)C)=O)cn2ccsc2n1 N1(C(C2C(C(N)=O)C2)=O)CCN(CCCNC(c2cnc(Cl)cn2)=O)CC1 C1(CC=C)COCC1NC(=O)C(CNC(=O)CC1(O)CCCC1)N(C)C C1(CCOC)(NC(C)=O)CCN(C(=O)C(c2ccccn2)C)CC1 Cc1nc(NC(=O)Nc2cnn3c2NCC3)nc(Cl)c1C CCCC(C(O)C(=O)NCCOCCOC)NC(C1CC(CC)(CC)C1)=O C1(NC(c2n(C)cnc2)=O)CC(NCc2nccs2)C12CCC2 C1(CC(=O)NCC2CC2CC(=O)NCC2CCCC2CF)CCC(O)C1 C(c1ccc(C)cc1)=CCC(=O)N.CC1=CCC(C(=O)NC(C)C2CC2)CC1 C1(CNC(=O)Cn2cnnn2)CC(C(=O)N2CCCC(F)C2)=NO1 c1(C(=O)NC23CC2CN(C(=O)CCOC2CCCOC2)C3)cccn2nnnc12 N1(C2CCN(CC=C)C2=O)CC(NC(=O)Cn2c(C)c(C)sc2=O)C(C)(C)C1 N1(C(C(C)(C)OC)=O)CC(NC(=O)C(C)Cc2ccc(F)cc2)C(O)C1 c1(C(=O)NCC2(O)CC(NC(CC3(C)CCC3)=O)C2)cc2scc(Cl)c2[nH]1 CC1C(NC(C2CCCC2C)=O)CCCN1C(=O)C(O)CC1CCCCC1 S(=O)(=O)(CC(=O)NCC(C1CC1)N(C(=O)CC1(OC)CC1)C)N(C)C CC1(C)CC(C(=O)NCCC(=O)NCc2ccoc2)CCO1 CCCCC(C)C(=O)NCC(CCOC)NC(=O)C(c1ccc(F)c(F)c1)O C(c1nccs1)=CC(=O)NCc1cn(CCC)nn1.c1(C=O)c[nH]c(=N)o1 N1(C(CC(=C)C)=O)CC(NC(c2cn(CC)nc2C2CC2)=O)C(C)C1 C1(C(=O)NCC(CC=C)NC(C2OCCC2C)=O)CN(C)CC(C)O1 C12(NC(CSCC(N)=O)=O)CCC1CN(C(c1csc(-c3ccco3)n1)=O)C2 Cc1c(Cl)sc(Cl)c1C(=O)NCCCCNC(C1CCOC(C(C)C)C1)=O n1(CC(N2CCN(C(COCCCCC)=O)CC2)=O)cnc2cc(C)ccc12 N1(C(c2ccc(C#C)cc2)=O)CCCN(C(C2CC3CCC2O3)=O)CCC1 C1(CNC(C2(C(C)C)CC2)=O)CC12CCN(Cc1ccc(F)cc1)CC2 C(=O)(C1=CCC(NC(=O)C(C)(C)OCCC)C1)N1CCCC(CCCC)C1 O=S(=O)(c1c[nH]ccc1=NC(CO)C1CC1)NCCN1CCC2CCCCC2C1 CCCCC(CNC(C1(CC)CCOCC1)=O)NC(=O)CSC.c1ccccn1 N1(C(C2(CNC(c3nc(CC)oc3)=O)CC2)=O)CCc2ccccc2C1 C1(OC)C(NC(C2CCC(NC(=O)C(F)(F)C3CC3)CC2)=O)CC12CCC2 CCC(C(=O)N1CC(O)(CNC(=O)C=CC=C(Cl)Cl)C1)NC(C)=O C1(C(CNC(c2cn(C)nn2)=O)O)CCN(C(=O)CCCN2CCCC2)CC1 C1(CNC(c2c(CC)nc[nH]2)=O)CCN(C(c2ccc(CO)o2)=O)CC1O N(C(=NCC1CCOC1)NCc1cncn1C)CC(C1CCC1)OC N1(C(c2[nH]c(=NC)sc2)=O)CC=C(CNC(=O)C(C)C(C)n2cccn2)CC1 n1(CC#C)nc(CN2CCC(NC)C2c2ccccc2)oc1=O c1(CN(C(c2ccc(COCC)o2)=O)C)ccc(F)c(F)c1 N1(C(C23CCC(CC)C2C3)=O)CCC2(C=C(C(=O)N3CCC4(CCSCC4)C3)C2)C1 N1(C(C(C)C2CC2)=O)CCCC1CC(=O)NCCOCc1ccccc1 c1(C(N2CCCC2C)C(=O)NC)ccc(C2CC2)nn1.C(=O)N=S(C)(C)=O C(=O)(C1CCCn2cncc21)N1CCC(N(C(=O)C(C)(C)C(N)=O)C)CC1 C1(OC)CCCN(C(C2C3CC2CN(C(=O)OC(C)(C)C)C3)=O)CC1 CC1CCCCC1CNC(C1(NC(c2cccn2C)=O)CC1C)=O C1(NC(Cn2c(C)ncc2)=O)CCN(C(c2cnc(C3CC3)[nH]2)=O)CC1C N1(C(C2CC(C#C)(O)C2)=O)CCC2(CCC2NC(c2ccc(Br)s2)=O)CC1 c1(C(N2CC(F)(CNC(c3c(C)scn3)=O)C2)=O)c(O)cccc1F C(=O)(C1=CCCCO1)NCC(C1N(C(CC2CCCN(C)C2)=O)CCCC1)(C)C C(C(CC(=O)N(C)C)C(F)(F)F)N1C(C)C(C(F)(F)F)NCC1 c1(SCC(=O)NC2CCN(C(CC3CCN(C)C3=O)=O)C2)nnc2ccccn12 C12(NC(C(CN(C(CCC=C=C)=O)C)C)=O)CC1COC2(C)C c1(C(=O)NC(C)CN(C)C(c2ccc(F)c(O)c2F)=O)cc2cc(Cl)ccc2s1 C1(c2n(CCOCC)nnn2)(NCC2C3COCC23)COC2(CCC2)C1 C1(CNC(C2(OCC)CC2)=O)CN(C(=O)Cc2cncs2)CC1O c1(N(C)C)nc2ccc(N(C)C(C3CC3(C)C)=O)cc2[nH]1 C=CC1CN(C(=O)CC2CC2)CC1NC(=O)CCC1CCOC1 c1(N(C2CCCC2)C(c2cccc(-c3c(CC)cccn3)c2)=O)ccc(C)cc1F C=CCCCNC(=O)C(=O)NCCOC.N1(CC=O)CCC(C=O)C1.N N1(C(=O)C(F)F)CCC2CCC(C1)N2C(c1cccnc1S)=O CC(CCNC(=O)C(C)O)CC.c1(C=O)ccccc1-n1cncn1.C(C)(C)C C1(N(CC(c2n(C)ncc2)O)C(=O)C=CC)CCC(=O)NC1.N1CCC1.C c1(OC)ccc(OC)c(C(=O)NCC2CCCC(C)C2)c1.C(=O)(C(F)F)N C(=O)(CC(C)(C)C(F)F)NCCCCCC(=O)Nc1ccc(C#C)nc1 c1(C(=O)NCCC2(NC(C(C)OCC)=O)CC2)cnccn1 C1CN(C(=O)C(F)=C2CCC2)CCN1C(c1cc(-c2ccco2)c[nH]1)=O.COC C(=O)(C1CCCn2cc(C)nc21)NCCN(C(C1CC(F)C1)=O)CC n1(CC(=O)OC)ccc2ccc(NC(=O)Nc3ncccc3S(C)(=O)=O)cc12 C(=O)(CC(O)CNC(=O)C(C)N1CCCC1)NCC1(OC)CC1 CCCC(C)(C)C(=O)NCc1cc(C(=O)NC(C)CN(CCO)C)co1 c1(C(N2C(C)CC(CC(=O)NCC3CCC3(F)F)C2)=O)cccc(F)c1O c1(C(N2CCC(C3CC3)(NC(CC(C=C)C)=O)C2)=O)ccc([N+](=O)[O-])c(O)c1 c1(CCC(=O)NCCCC(C)NC(=O)CC(C)O)ccc2[nH]ccc2c1 N1(C(c2nc(CC)oc2)=O)CCCC(CN(C)C(C2C(C=O)C2(C)C)=O)C1 Cc1ccc(C(=O)NC23CCN(C(=O)CCc4scnc4C)CC2C3)cc1C C1(CC(=O)NCC2C(COC)C2)CCCCN1C(C12CC(C1)C2)=O C1(C(C)(C)NC(C(c2cncnc2)C)=O)CCN(C(c2ccc(C(N)=O)o2)=O)C1 CN1N=C(CC(=O)NC2CC(CNC(C3COC4(CO)CC3C4)=O)C2)CC1=O C1(C(N2CCN(C(CNC(=O)NC)=O)C(C)C2)=O)CCc2cn(C)nc2C1 Cc1coc(C=CC(=O)NCC(c2cccc(Cl)c2)NC(c2cnco2)=O)n1 c12ccc(Br)cc1NC(=O)CS2.C1(NC(C)=O)CCCCC1.c1ccccc1.O C1(C2CCN(C(C3CCCS(=O)(=O)C3)=O)CC2)CC1.C(C(F)(F)F)OCC=O N1(C(C(N(C(=O)CO)C)C2CC2)=O)CCCC2C(=O)NCC12.C1(C)CCOCC1 C1(N(C(=O)C(C2CC2)SC)CC)CCCN(C(=O)C=C2CCN(C)C2)C1 CCC(CC)CCC(=O)NCC1CCC2CN(C(=O)CSCCN(C)C)CC12 N1(C(c2cc(OC)cc(F)c2)=O)CC2CC(NC(=O)C)C(C2)C1.C(C)=O.O C(=O)(C1=CNC2=NCCC2=C1)NC1(C)CCN(C(c2ccc(C)nn2)=O)C1 c1(CNC(c2cccc(N)n2)=O)nnc2n1CCN(C(C1CCCCS1)=O)C2 c1(C=O)cc[n+]([O-])cc1.C(=O)(C(C1CCC1)C1CCC1)N(CC)C1CC1.N N1(C(c2nc(COC)[nH]n2)=O)CC(C)(C)CC1.c1(C=O)cc(C)cc(F)c1.C Cc1c(C(N2CC(NC(C3CC(C)CO3)=O)CC2C)=O)cnn1CC(F)F C1(C(=O)NCC(CN(C)C)O)(CNC(=O)CC2CC(F)C2)CCCO1 C1(CCNC(=O)CCC2CCN(C(C3C4(CC4)C34CC4)=O)C2)CCCC2CC12 C1(CC)CN(C(=O)CCOC2CCC2)CCC1NC(=O)CCc1cc[nH]n1 C1(NC(C(C)=CC)=O)CC2C1CCN2C=O.c1(C=O)ccccc1.C(C)C N1(C(c2c(C)nns2)=O)CCN(C(=O)C(F)(F)C(F)F)CC1CC(F)(F)F C1(NC(c2c(CC)con2)=O)CCN(C(=O)CCCc2cccc(Cl)c2)CC1O Cc1cc(C(=O)NCC2CCN(C(=O)CCOCC(F)F)C(C)C2)nc(C)c1 c1(CN2C(C(=O)NCc3c(C)cccc3)CNCC2)cc(F)c(O)c(Br)c1 Cc1cc(C(N2CCCCC(C(N3CC(CN(C)C)C3)=O)C2)=O)ncc1N c1(C(=O)NCC2(C)N(C(c3n[nH]c(C)c3Cl)=O)CCC2)sc2cncn2c1C c1(C(N(C2CCCN(C(C3(C#N)CC3)=O)C2)CC)=O)ccc(C)nc1C C#CCCCC(=O)NC(C)CC(C)NC(=O)CCc1ccsc1Cl CC1CCC2(CC2)N(C(=O)COC2CCN(C(C34CCC(CC3)C4)=O)C2)C1 CC(C)C(O)CC(=O)NCC(C)(C)CCNC(C1CC(=O)NC1(C)C)=O C1(C(N2CCCC(c3cn(Cc4cc(C)on4)nn3)C2)=O)CC2(CC2)CN1C N1(C(c2cc(SCC)ncc2)=O)CCCC(C)C1.c1(C=O)cn(C2CC2)cn1.N C1(C(C)C)CN(S(=O)(=O)Cc2c(F)cccc2F)CCCN1Cc1ccccc1 C(=O)(C(C)CS(C)(=O)=O)N1CC(CC)N(C(c2cc(Br)ccn2)=O)CC1 C(=O)(CCN(OC)C(=O)c1c[nH]c(=O)cn1)NC(c1n(CC)ncc1)C C1(CC#N)CC(=O)NCCN1Cc1csc(N)c1 Cc1cccc(C(=O)NNC(=O)C2(c3ccccc3C)CCCC2)c1 C1(N(C)C(c2cnc(=N)[nH]c2)=O)CCCCN(C(=O)COc2cncc(Cl)n2)C1 N1(C(CNC)=O)CCC2(CCOCC2)C(C(=O)NC)C1.c12nnc3n1CC2CC3 CC1CC(NC(=O)CC2(C)CC2)CN(C(=O)CC2(O)CCC2)C1 CC1CCc2ncc(C(N3CC(C)(NC(C4CCCSC4)=O)C3)=O)n2C1 c1(CC2N(C(c3nscc3C(F)F)=O)CCC2)c(F)cccc1Br c1(C(N(CCNC(Cn2cc(C(=O)OC)nn2)=O)C)=O)cc(O)ccc1O CN1CCN(C(=O)C=CCNC(=O)C2=COCCC2)C2CC12 C(=O)(CS(=O)(=O)C1CCCC1)N(CCC)CC.C1(CC=O)C(C)C1(F)F.N Cc1nn(C)cc1C1=NOC(C(=O)NCC2(C)CCN(C(c3ccsn3)=O)C2)C1 N1(C(CC(C)(C)C(F)F)=O)CCCC2CN(C(c3ccc(Cl)c(F)c3F)=O)CC12 n1(CC)nc(C)c(C(=O)NC2CN(C(=O)C(C)(C(C)C)OC)CC3CC23)c1Cl c1(C(=O)NC2CN(C(C3CC(CSC)C3)=O)C2)cc(F)ccc1N C1(C(C)C)CN(C(c2cc(F)n[nH]2)=O)CCN1C(c1ccnc(C2CC2)c1)=O N1(CC(=O)NCC2COCCN2C(C2CC3CCC2O3)=O)CCCCS1(=O)=O N1(C(C2(C)CC(C#N)C2)=O)CC2(C1)SCCC2NC(C1CCCCO1)=O CCCCC(C)(F)C(=O)N1CCOC(CC(=O)NC2CC2C2CCCCC2)C1 c1(C(=O)NCC2(C)CCCN2C(c2ccc(F)o2)=O)cnc2ccnn2c1O Cc1sc(C(=O)NCC(C)CNC(c2cc[nH]c(=N)c2)=O)nc1O N1(C(c2cccnn2)=O)CCOC(C(c2cn(Cc3ccccc3Br)nn2)=O)C1 CC(C)C1=NOC(C)(C(=O)NCCC(C)NC(c2ccccc2)=O)C1.C(CO)O C(=O)(C1CNC(=O)c2ccnn21)NCCC.C1(C=O)CC(C)(C)OC(C)(C)C1.N Cc1cc(N2CC3CC(NC(c4ccn(CC(C)C)n4)=O)C3C2)nc(CO)n1 C1(CC(=O)NC23C(NC(=O)CCC4CC4)CC(CC2)C3)CCn2cncc2C1 C1(CNC(CCCOCC)=O)CCC2(CCC2)CN1C(=O)C(F)C1CC1 C1(C(=O)NCCCN(CCC)C(C2CC2(F)F)=O)OCC2CCCC12 C1(C(=O)NC(C2CCN(C(C(C)OCC=C)=O)C2)C)CCC(CC)CC1 S(=O)(=O)(c1cccs1)Oc1ncc(NC(CNc2ccc(CC)cc2)=O)c(C)n1 N1(C(C2N(C=O)CCC2)=O)CCOCCC1C(=O)NC(c1ncc[nH]1)CO N1(C(c2ccc(CC)[nH]2)=O)CCOCC(NC(=O)NCCC(=O)OC)C1 CCC(C)C(O)C(=O)NCC12CC1CN(C(=O)C(F)(F)c1csc(Cl)c1)C2 Cc1cnn(C(C)C)c1NC(N1CCN(C2(C#N)CCCC2)CC1)=O N1(C(c2snc(C)c2N)=O)CC2CC(NC(C3CCC4(CC3)N=N4)=O)CC1C2 C=CC(O)C(=O)N(CCCCN(C(=O)CC1(C)CC1(Cl)Cl)C)C c1(C(N2CC(NC(c3nc(C4CC4)cs3)=O)C3C2C3)=O)cc(F)cnc1O c1(CC=O)ccc(C)c(F)c1.C1(C(=O)NC2CCCC2O)(CC)CCNC1=O.N N1(C(C2(COC)CCCC2)=O)CC2C(NC(c3oc(Br)cc3C)=O)C2C1 C1(O)(CCNC(C(c2ccc(C)cc2)O)=O)CCCN(C(c2sccc2F)=O)C1 C1(CNC(C(C)N(C)C)=O)Cc2ccccc2CN1C(c1nc(Cl)ccc1F)=O C1(CC=C)(C(N2CCC(C(C)NC(c3ccoc3)=O)C2)=O)CC=CC1 n1(CCCC(=O)N(C)C)cc(N=c2[nH]c3ccc(Br)cc3s2)cn1 c1(C(=O)NC2CCC(N(C(Cc3c(C)non3)=O)C)C2)cccc(C#N)c1 C(=O)(C1=CCCS1)N(c1c(C(N2CCCC2C2CCCOC2)=O)n[nH]c1)CCO c1(OC)ccc(Br)c(NCc2ccc(COC)o2)c1.c1cccs1 C1(NC(c2cn(C)nn2)=O)CCCN(C(=O)CN2CCC(O)CC2)C1 C(c1cccc(CO)c1)=CC(N1C(CNC(=O)C(O)C2CCC2)CCC1)=O C1(C(=O)NC(CC#CC)CO)CCN(C(=O)Cc2ccc(O)cc2)C(CC)C1 C1(N)(C(N(C)CC2COC(=O)N2)=O)CCOCC1(C)C N1(C(C(C(=C)Cl)(C)C)=O)CC(NC(=O)C(CC)SC)C2(CCC2)C1 N1(C(Cc2c(C)n[nH]c2C)=O)CCCC2C1CCN2C(C1CCCCS1)=O C(C(=O)NC1CC(CCOC)N(C(c2[nH]ccc2)=O)C1)(C(C)C)OCC.C c1(OCC(=O)NCC(C)(C)NC(C2CC(F)(F)C2)=O)ccc(Cl)cc1 c1(OCC)ccc(CCC(=O)N(CC(C)N(C)C(C2CC2CO)=O)C)cc1 N1(C(C(CC(C)C)OC)=O)CC(C(N2CC3(CCC3)CC2C)=O)C2(CCC2)C1 c1(NC2C3(CC(OCC)C3)C2)cc(C(F)(F)F)cc(C)c1OC N1(C(CCc2n(C)ncc2)=O)CCC(C)(C)CC1C(=O)NCC1CC1(Cl)Cl C1(C(C#C)C)CCN(C(=O)CC(C)(C)NC(c2ccnc(C)n2)=O)CC1 c1(CN2CCC(NC(c3nn(C)c(Cl)c3)=O)CC2)ccc(S(=O)(=O)C(F)F)cc1 C=CCC(C)(C)CC(=O)N1CCCC(F)(C(=O)NCC2CC(=C3CC3)C2)C1 c1(NC(CNC(C(c2ccccc2)N(CC)CC)=O)=O)ccc2c(c1)CCO2 C(C)(CC1=CCCCC1)NC(C(CCOC)NC(=O)CC(Cl)Cl)=O N1(C(c2cc(C#N)[nH]c2)=O)CCN(C(=O)CCCc2nccs2)C(CO)C1 CC1(C(N2CCC(NC(=O)C(F)CC3CCC3)C2)=O)CCOCC1 c1(OC)ccc(CN2CCC(C)(C(=O)NC3CCS(=O)(=O)C3)C2)cc1OC N1(C(C2N(S(CCC)(=O)=O)CCC2)=O)CCC(C)N(C(=O)CSC2CC2)CC1 C(N=c1[nH]c(Cl)nc(C2CC2)c1F)C1CN(C(C=Cc2nc(C)c(C)[nH]2)=O)C1 C(=O)(CC(C)(C)C)NCC1OCCN(C(COC(C)C)=O)C1.C(C)(C)C.O c1(C(=O)NCCN(C(c2ccc(C#C)c(F)c2)=O)C)cn(CC)c2ccccc12 C1(C(=O)NCCn2cnc(C)c2C)CC1C1CN(C(=O)CC2CCOC2C)C1 c1(CN(C)C(C2COCCO2)=O)cnn2c1CN(C(=O)Cc1cnn(C)n1)CC2 C(C)(CNC(c1nocc1C)=O)(C(C)C)NC(c1cn(CCCC)nn1)=O.C c1(C(=O)NC2CC(C(N3CC(COC)OCC3)=O)C2)cc(=O)nc2cccnn12 c1(CN2CCC3CCC(C(=O)NCC4C(=C)CC4)C32)cn2ccc(C)cc2n1 C1(C(N2CC(CNC(c3scc(C)c3Cl)=O)C2)=O)CC(=O)N(C)C(=O)N1 C1(NC(c2c(C#C)cn(C)n2)=O)CCC(O)CN(C(C2CCCS2)=O)C1 Cc1cc(C(=O)NC2CCC(NC(C3C=CCC3)=O)CC2)c([N+](=O)[O-])c(O)n1 N1(C(C(CC=C)(F)F)=O)CCC2CC2(C(=O)NCCC(C)(C)COC)CC1 C1(O)(CNC(c2cccc3c[nH]nc23)=O)CCCN(C(=O)CO)CC1.C1CCC1 C1(NC(=O)CCNC(c2ccsc2)=O)CC2CC1N(C(C1CC13CC3)=O)C2 N(C(=NCCN1CCOCC1)NCc1ncnn1C)C1C(C)C1 CC(CC(C)(C)C)C(=O)NCCCCNC(=O)CCc1nc(-c2ncccn2)no1 C1(CC(=O)NC2(CCC(N3CCC(C(C)(C)O)C3)=O)CCC2)CC2C=CC1O2 C1(C=O)Cc2cc(Cl)ccc2C(=O)O1.C12CC(C1)C2.CC(C)(C)OC(=O)N c1(NC(C2C(C)(C)C2)=O)ccc2c(c1)CN(C(c1cc(Br)cnc1Br)=O)CC2 C(C(=O)NCC(C1CCCC1)NC(=O)Cc1ccns1)(C(C)(C)C)SC C1(C(N(C)CCNC(C2COCCO2)=O)=O)Sc2ccccc2NC1=O C1(NC2CCC(CC)C2)C=C(c2ccccc2)CCC1 C(C)(c1ccc(C(F)(F)F)cc1)=CC(=O)N.C(CC(=O)N1CCC1)OCC C(=O)(C(O)CC(F)F)NCC(CC)NC(C1(Cc2cccnc2)CC1)=O c1(C(N(CCNC(c2ccc(OCC)nc2)=O)C)=O)cc(C)c(C)nc1O C(C(O)CC(C)(C)C)NC(CONC(C1(CC)CCNC1=O)=O)=O N1(C)C(=O)c2ccccc2C1=O.C1(C(=O)NCCNCCNC)CCCO1 N1(C(C2C(C)C2C)=O)CCN(C(=O)C(c2cncn2C)O)CC1C N1(C(c2cc(C)cc(F)c2)=O)CC2CCCCC2(NC(C2CC2C(C)(C)C)=O)C1 c1(CN=C(NC(C)C2CC2)NC(CF)CF)ccc([N+](=O)[O-])cc1 CC1C(NC(=O)Cc2cnc(C3CC3)[nH]2)CCCN1C(c1cc(O)n(C)n1)=O C1(NC(c2cc(C)ns2)=O)CN(C(c2ccncc2C)=O)CC1C c1(C(=O)NC(CC(C)NC(C=CSC)=O)C)ccc2c(c1)S(=O)(=O)NC2 C(=O)(CC(CN(C)C)C(F)F)N(CCCNC(CC(CCC)O)=O)C C(C(C(=O)NCC(C)OC(F)F)NC(c1cc(N(C)CC)on1)=O)OCC Cc1cc(F)cc(C)c1C(=O)NC1CC(C)C1.c1(CC=O)cn(C)nc1C.N C1(NC(CC(C)SC)=O)CC(C(=O)NCCc2cnc(C)o2)CC1O CN1CCC(C(N2CC(N(C(=O)CC3SC(=N)NC3=O)C)C2)=O)S1(=O)=O N1(C(C(C)c2ccsc2)=O)CCCN(C(=O)C2=CCSC2)C(CO)C1 C1(NC(=O)NCc2nc(C(C)C)sc2)CCN(C)C(=O)C1 c1(C(N2CC(NC(C=COCC)=O)C(C)CC2)=O)c(OC)cc(OC)cc1N N1(Cc2cc(OC)ncc2)CCC2(NC(=O)CCc3cncc(C)c3)CCCC12 C1(NC(C=Cc2cnc(C)s2)=O)CC(C)CN(C(C2(C)CC(C#N)C2)=O)C1 C1(CNC(C=NOC)=O)CCCC(NC(c2ncoc2-c2ccc(F)cc2)=O)C1 c1(C(=O)NCC2CC(CNC(CC(=O)OC)=O)OC2)ccnc(Cl)c1 c1(CC)c(C(=O)NC2CCC(N(C(=O)CCSc3ccccn3)C)C2)ccn1C c1(C(N2CCC(NC(c3ccc(C(C)C)o3)=O)CC2)=O)cc(F)c2[nH]nnc2c1 C1CCCCN(C(C2(CC(C)C)CC2)=O)C1.n1(CC)nc(C=O)cc1C(C)C.N c1(CNC(CCN(C(C2CC3(CCC3)CO2)=O)CC)=O)cccc(C)c1O C(=O)(C(C)CC(C)(C)C)NCC(CC(C)C)NC(C(CC)c1ccccc1)=O C1(C(N(C)CCc2ccccn2)=O)CCN(C(C2(C)C=CCC2)=O)CCO1 c1(C(=O)NC(C(C)NC(C(c2c(OC)cccc2)O)=O)CO)ccc(C)cc1F N1(C(C=CC)=O)Cc2ccccc2C(NC(=O)CCC(=O)N2CCOCC2)C1 CC(C)C(C)(O)C(=O)N1CC(O)(CCNC(c2n[nH]c(C(C)C)c2Br)=O)C1 C1(C(=O)NCc2ccccc2N2CCC(O)C2)CCC2C(C1)C2(F)F c1(C(=O)NCC23C(CN(C(c4c(CC)n[nH]c4)=O)C2)C3)snc2ccccc12 N1(C(=O)CCn2cccn2)CC2CCC2(C(N2CCN(CC(=O)O)C(=O)C2)=O)C1 C1(C(N2C3C(C(N(C4CCCCC4(F)F)C)=O)C(C3)C2)=O)CCCCC(=O)N1 c1(OC)cc(N)c(C=O)cc1OC(F)F.C(=O)(CP(C)(C)=O)N1CC(CC)C1 c1(CCC(=O)N(CC(O)CN(C)C(C2COCCOC2)=O)C)ccccc1C#N C1(CCCCCNC(c2cc(Br)ccn2)=O)CCN(C(C2CC2F)=O)CC1 CC(C)(C#N)CCCC(=O)N1CC(CNC(C2CC(n3ccnc3)C2)=O)C1 C1(NC(C(C)=CC)=O)CCC12CCOCC2.c1(CC(=O)N)ccc(C)c(F)c1 C1(CC(=O)OC)Cc2ccccc2CN1N1CCC(c2cccc(OC)c2)CC1 C(=O)C(O)C(F)(F)F.c1(C(=O)OC)oc(C(N2CCCC2C(C)C)=O)cc1C CCC(C(=O)N1CCCC(C)(CNC(c2cnn(CC)c2)=O)C1)C(C)O c1(OC)ccc(C(C)SCC(=O)Nc2ccc(-n3ccnc3)nc2)cc1 c1(C(=O)NCC(CO)NC(C(c2cccc(C)c2)C)=O)n[nH]c2cccnc12 C1(CN(C(CCOCCC)=O)C)CCN(C(c2ccnn2CC(C)C)=O)CC1 N1(C(CC2CC(C)C2)=O)C(CNC(c2[nH]nc3ncccc23)=O)CC2CCCC12 c1(OC)ccc(C(=O)NC2CN(C(C3(C4CCC4)CC3)=O)CCC2C)c(C)c1 N1(C(C)C(=O)NCC(O)CCNC(=O)C(F)F)CCC(O)CC1.c1cnn(C)c1 C1CN(C(=O)C)C2(CCC2)C1.c1ccc(C(N)=O)cc1.C=C1CCC1C(=O)N c1(C(=O)NC23CN(C(C(F)=CC)=O)C(CC2)C3)cnc2ccccc2c1 c1(C(N2C(CNC(c3n(C)c(S)nc3)=O)CCC2)=O)ncc(C(F)(F)F)cc1O N1(C(c2occ(C)c2C)=O)CCN(C(=O)CCCCOc2ccccc2)C2CC12 C1(c2n(CCC)nnn2)(NCc2c(Cl)sc(Cl)c2Cl)CCCC(SC)C1 C1(C)(CN(C)C(=O)OC2CCOC2)CCCO1 c1(C(C=O)O)cc(F)c(F)cc1F.CNS(=O)(=O)NCC(=O)NC1CC1C CCC(CN=c1cc(C)[nH]c(=NCc2cc3ccccc3s2)[nH]1)N(C)C N(C(=NCc1cccs1)NCC1(OC(F)F)CCSC1)C1C(C)(C)SC1 c1(C(C)OCC)nc(-c2cc(C(C)CC)no2)n(CCF)n1 C(CCC(C)C(=O)NCC(C)(O)CNC(=O)C=CC(=O)N(C)C)OC N1(CCOC)CCCC1C1CCCCN1C(c1ccc(C(F)(F)F)cc1)=O N1(C(CC(C(C)C)O)=O)CCC2CCN(C(=O)CCC(CF)CF)CC12 Cc1cc(=O)ccn1CC(=O)N(C)CCC1CCCCN1C(=O)CCC(F)(F)F C(=O)(CC(CC)CC)NC(C(=O)NCc1nc(CC)oc1)CCF C1(C)(CC)CC(C(N2CCC(C)(CNC(C3CC3(F)F)=O)C2)=O)CCO1 N1(C(C2C(C)CN2C(=O)CSC2CC2)=O)CCCCC1CC(N)=O C1(C(N2CC(OC)C2)=O)CN(C(=O)Cn2cc(Cl)cn2)CC1(F)F.CC(=O)N c1(CNC(C(CC)NC(=O)COC2CCCC2)=O)ccnc(F)c1F c1(C(=O)NC)ccccc1NC(C12CC1CN(c1ncc(I)cn1)C2)=O c1(C(C)C)ccnc(NC(N2CCCC2c2cn(C)nc2C(F)F)=O)c1 C1(C)CCN(C(C2(O)CC2)=O)C1.N1(C(=O)OC(C)(C)C)CCC(CC=O)C1 CCC(C)CCCCC(=O)N1CCN(C(c2cncnc2)=O)CC2(CC2)C1 N1(C(C2C(c3nc(C)[nH]n3)C2(C)C)=O)CC(CNC(=O)C(C)(F)F)CCC1C CC1(CNC(=O)COC2CC=CC2)CCN(C(c2csc(CO)n2)=O)C1 N1(c2ccnc(COC)n2)CC23CCCC2(C1)CN(C)C3 c1(C(N2C3(CN(C(C(C(C=C)C)C)=O)C3)CC2)=O)ccc2nc(S)oc2c1 N1(C(c2n[nH]c(CC)c2F)=O)CCC2(CCN(C(c3ocnc3C)=O)C2)C1 N1(C(c2cc(CC)no2)=O)CCC(CNC(=O)CSCCC#N)C(C)C1 N1(C(CC=CCC)=O)CCN(C(c2cc(C)nn2CC)=O)C2CCCCC12 C1(C(=O)NCC2(C)CC=CCC2)CCC(C)(C)N(C(=O)C)C1.C1CCCCC1.O Cc1cc(C)c(C(N2CCC3(NC(c4nn(C)cc4C)=O)CC3C2)=O)c(=O)o1 C1CCC(C)N(C(=O)C)C1.c1ccc(C)cc1C.C(C=CC(=O)N)(CC)=CC C1(NC(c2c(COC)ncs2)=O)CCN(C(c2cncc(OC)n2)=O)C12CCC2 N1(C(C(=O)OC)C)CC2(CC(CNS(=O)(=O)NC(=O)CSC)=NO2)C1 CS(=O)(=O)CCCC(=O)NCCC1CN(C(c2ccn3ncnc3c2)=O)C1 Cc1nc(=N)[nH]c(=NCC(C2CCCCC2)NC(=O)CC2CCCC(C)C2)[nH]1 N1(C(c2ncn(C)c2)=O)CCC2(CCS(=O)(=O)CC2)C1.C(=O)(CCP(C)(C)=O)N O(NC(=O)C(Cc1ccoc1)NC(c1c[nH]c(=N)o1)=O)C(C=C)C N1(C(C(C(C)C)N2CCCC2=O)=O)CC2CCC2(CNC(c2cnsc2)=O)C1 N1(C(CC2NC(=O)OC2)=O)CC2=C(C1)CN(C(c1ccoc1Br)=O)C2 c1(OCCCC)cccc(OC(c2ccc(-n3cncn3)nc2)=O)c1 CC1COC(C)(C)CN1C(=O)C(C1CC1)N(C(=O)C=CC1CCCCC1)C C1(C)(C(=O)Nc2ncn(-c3ccn(C)n3)c2)CCCC(F)(F)C1 CC(CC(F)F)C(=O)N1CC(C(C)Nc2nccc(OC3CCOCC3)n2)C1 c1(OC)ccc2cc(C(N3CCC4(CC(C(=O)N(C)CC#N)C4)C3)=O)ccc2c1 CC(C(C)(C)CO)NC(=O)CC(C1CC1)NC(=O)Cc1cncn1C c1(C(N2C(C3CCN(C(c4cnn[nH]4)=O)CC3)CCC2)=O)ccc2ocnc2c1 C1(NC(c2c(CC)cccn2)=O)CCN(C(=O)Cc2cnc[nH]2)CCC1CO CP(C)(=O)c1cnc(C(=O)NC2(CO)CCN(C(=O)CC3C=CCC3)C2)cn1 C(=O)(CCN(OC)C(=O)c1cnnn1CC)NC(C#C)(C)C1CCOC1 N1(C(C23CN(C(c4occ(C)c4)=O)C(C2)CO3)=O)CCN(C)C(C)(C)C1 C(CN=C(NCCc1cccs1)NC1CCOCC1)C1(O)CCCOC1 c1(C(=O)NCCCCCCNC(C2CCCSC2)=O)ncnc2c1CCCC2 N1(C(C(C(=O)NC(C)C)C)=O)CC(C)(C)CC1CC(=O)N.CCC(O)C(F)F C1(CC(=O)NC2CC(NC(c3ccc(N)c(Cl)n3)=O)C2)CSc2ccccc2O1 C1(NC(c2c(COC)ncs2)=O)CCOC(C)C1.c1(C=O)cn(C)nc1.N C1(CNC(=O)NOCCO)CCCC(C(F)(F)F)O1 C(C(C)(C)CNC(C1(C2CCCN2C(=O)C(CO)SC)CC1)=O)SC C1(CC#C)CN(C(=O)C=CC2CCCN2C(=O)C(CC)CC)CCO1 N1(Cc2cn(CC3CN(C(C(C)C)=O)C3)nn2)CCCCCC1=O.C1C(=O)N1C C1(C(=O)OC)CCC(C(=O)NCC(C)N(C)C(C2COC(C)C2)=O)CC1 C1(CNC(c2c[nH]nc2Br)=O)CCC2(CN(C(C3CCOC3)=O)C2)O1 c1(OCCNC(COC(c2c(C)cco2)=O)=O)cccc(Br)c1 Cc1ccnc(C)c1C(=O)NC1C2CC1CN(C(=O)CSc1nccn1C)C2 c1(C2(C(N3CCC(NC(C(c4ccncc4)C)=O)C3)=O)CC2)ncccc1F C1(CC(=O)N(CCN(C(=O)CC2(O)CC2)CC)CC)CCCCC1.O c1(C(=O)NCC2(O)CN(C(C(C)SC)=O)C2)ccc(F)c(O)c1F Cc1cc(-n2cc(C(C)(C)NC(=O)C(C3CCS(=O)(=O)CC3)F)nn2)ccc1Cl C(C(C)(C)C#CC(=O)NCC(O)C(N)=O)NC(C(C)=C(C)C)=O C(=O)(C1=NNC(C(F)(F)F)C1)NCCCNC(C(CCC)C)=O C1(NC(CC(C)F)=O)CCC(O)CN(C(=O)CC2CC(=O)C2)C1 c1(C(N(CC(C)N(C(=O)C)C)C)=O)ccc(C(C)(C)C)cc1N.CC(F)(F)F C(=O)(C(C)C(F)(F)C(F)F)NCCCCN(C(C1C(COC)C1)=O)C C1(NC(C(=O)NCC(F)F)=O)CN(C(c2cccc3sccc23)=O)C2(CCC2)C1 Cc1cc(NC2CCCC(NC(=O)C(c3cscn3)N(C)C)C2)n2ncnc2n1 C(=O)(C1=C(Cl)CCC1)NCc1c(C(=O)NC2CC(C(C)C)OCC2)c[nH]n1 N1(C(C)=O)CCCCC1C(=O)NC1CCN(Cc2cn(CCO)nn2)CC1 C1(C(=O)NC(c2ccccn2)CCC)CCN(C2CCCCC2O)CC1 Cc1cc(F)ccc1NC(C(c1cnc(C)c(C)c1)N(CCCF)C)=O CC(C)(CC#N)C=O.c1(CN(C(C2OCCC2)=O)C)ccccc1.C(C)(C)C N1(C(c2ccc(CC)[nH]2)=O)CC2CCC1C(CNC(=O)C(C)(C)CC(F)F)C2 N1(C(=O)CC2(O)CCOCC2)CCC2CC(C1)CN(C(c1cnc(O)o1)=O)C2 N1(C(C2CCN(C)C2)=O)C(CNC(c2cn(C3CC3)nn2)=O)CC2CCCCC12 c1(CC(N2CCCC2c2cn(C3COCC3O)nn2)=O)c(Br)sc2ccccc12 N1(C(C2CCC(=O)N2)C)CC(NC(C2CC23CC3)=O)CC2(CCOCC2)C1 C(=O)(N=c1[nH]n(C)c(=O)n(C)c1=O)NC(c1ccc(Cl)s1)C C12(CNC(=O)C(F)=CC3CC3)CCCC1CCN2C(c1ncncc1Cl)=O Cc1cc2c(C(N3CC(NC(c4cnn(C)c4C)=O)CC3(C)C)=O)cccc2o1 C1(NC(C2CCC(CC)CC2)=O)CCSC12CN(C(=O)Cc1scnc1C)C2 O=C(C(O)C(F)(F)F)NCC1(O)CCN(C(c2ccoc2C(F)(F)F)=O)C1 C=CCC(CC(=O)NC(c1ccc(C)s1)C)NC(=O)C(O)CC1CCCC1 CCC(C)C(O)C(=O)Nc1ccc(NC(c2cc(C)c(C)o2)=O)nc1 Cc1cccc(OCC(=O)NCC(C)(C)C)c1C.N1(CC(=O)N)CCN(C)CC1 c1(C2(O)CC(C(=O)N)C2)cccc(Cl)c1.C1(C(=O)NCCCO)(CC)CCC1 N1(C(c2ccn(C)c(=O)c2)C(=O)NCCOCC)CCOC2(CCSC2)C1 C1(N(C(c2n(CC)ccn2)=O)C)CN(C(=O)CC2CCC3CC23)CC1(C)C c1(C2C(C(=O)N)C2)ccc(F)c(Cl)c1.C#CC(C)(C)C(=O)N(CCCC(C)C)C c1(C(C(N2CC(O)C2)=O)O)ccc(Cl)c(Cl)c1.Cc1cc(C)c(C(=O)NC)o1 C(=O)(C(C)C(C)S(C)(=O)=O)N.N1(C(c2cc(=NC)[nH]cc2)=O)CCCC(C)(C)C1 C1(C(=O)NCC(C)NC(c2c(C)nc(C)[nH]2)=O)CCc2ncnn2C1 C(CO)(CCCNC(C1CCS(=O)(=O)C1)=O)NC(CCc1n(C)cnc1)=O c1(C(=O)NCC(CN(C(CCCC)=O)C)O)cc(C(F)(F)F)[nH]c1C C(C(CC(F)(F)F)NC(c1cncc(F)c1Cl)=O)NC(CC(C)OC)=O N1(C(c2c(C)cns2)=O)CCN(C(C2COC(C)C2)=O)CC12CC2 C1(O)(C(=O)NC(C2OCCN(C(COC)=O)C2)C)CN2CCC1CC2 c1(C(=O)OC)ccc(N2CCC(NC(=O)CC(C)C)C(O)C2)nc1C.C(C)=O.N Cc1nccn1CC(=O)NC(CNC(=O)C(C)(C)c1cc[nH]n1)C(C)C N1(C(C2C(C)(C)C2)=O)CCN(C(=O)CC(C)(C)C2CCCC2)CC(C(=O)N)C1 C1(NC(C(C)OCC=C)=O)CCC(F)C1.c1(C=O)cc(C(C)(C)C)[nH]c1C C1(C(=O)NCC(CN(C)C(C2(F)CCC2)=O)O)CCOC(C)(C)C1 c1(OC)ccc(C(c2cscc2Br)NCCc2ccc(CO)cc2)cc1 n1(CCC(C)C)cc(NC(=O)NC)nn1.C1(N(CC)C)CCCCC1.C1CCC1.C CC1CN(C(=O)C(C2CCOCC2)F)CC1Nc1ncnc(C(C)(C)C)n1 CCC(C)(COC)C(=O)N1CC(C(C)NC(c2csc(-c3ccoc3)n2)=O)C1 C12(NC(c3c(COC)ncs3)=O)CCC1CN(C(c1cnc(C)nc1C)=O)C2 C1(NC(C(C=C)O)=O)CC(NC(=O)Cc2ccno2)C(O)C1 c1(C(=O)NC(CNC(C(C)NC(C)=O)=O)CO)[nH]c(-c2cccnc2)nc1C n1(CCCC)nccc1C(=O)N(C(C)CNC(c1cocc1C)=O)CC CCC(C)(C)CCCC(=O)NNc1cc(C(F)(F)F)ccc1F c1(C(=O)NC(C)CN(C(=O)CCc2nc(C3CC3)no2)C)cncc(O)c1Cl N1(C(C)=O)CCC(C2CCN(C(=O)CCOC3CCC3)C2)CC1 C=CC1(C(N2CCC(NC(C)=O)C2)=O)CCN(C(=O)C(F)F)CC1 C1(NC(C(=O)Nc2cccc(-n3cnnc3)c2)=O)CC2CCCCCC2C1.C1(C)CC1 N1(C(C2(CC)CC2)=O)CC(NC(c2ncsc2NC)=O)C(C(F)(F)F)C1 C(C(F)C(=O)N(CCN(C(=O)Cc1cc[nH]c1)C)C(C)C)N(CC)CC n1(CC)cnc2c(NCC3CSCCO3)[nH]c(=NC3CC4CC5C(C4)C35)nc12 CC(CCC(C)(C)C)C(=O)N1CCCC(CO)(CNC(c2ccsc2)=O)C1 C(=O)(C1=CC2(CN(C(c3cocc3C(N)=O)=O)C2)OC1)NC(CC)(C)CC C(=O)(C(C)(CC)C(F)F)NCCCOCCNC(COCCC=C)=O c1(N2CCCC(C(=O)Nc3cccnc3)C2)ncnc2c1ccn2C1CC1 c1(CC(=O)N)cnc(O)nc1O.C1(CC(=O)N(CC)CC)CCC(F)(F)C1 c1(C(=O)N(c2ccn3nccc3c2)C2CC3CC2CN3)ccc([N+](=O)[O-])cc1O c1(CC)cc(C(=O)N)cc(C)c1.C1(C(C)C)CCCN1C(=O)CC1CCOCC1 C1(C2CCCN(C(c3cnsc3)=O)C2)(NC(=O)CC(F)(F)c2ccccc2)CC1 C1(C(N2CCC(C)(CNC(CC3CC(=C)C3)=O)C2)=O)CCC(C)(CC)CC1 c1(NC(N2C(C(=O)O)C3CCC2C3)=O)ccc2c(c1)NC(=O)NC2 CC1COC(C(=O)NCCCCNC(C2CC(O)C2)=O)c2ccccc21 c1(C=O)c(O)nnc(C)c1C.C1(OC)CC(CC(=O)NC2CC(C)C2)C1(C)C c1(C(=O)NCC2C(NC(CC3C(C)(C)COCC3)=O)C2)nc2ccccc2[nH]1 c1(C(C=O)O)ccccc1.C1(F)(C(=O)OC)CC1C(=O)NCC1CCC1 N1(C(c2cc(C)on2)=O)CCCC2CN(C(=O)CC3(C)CCCC3)CC12 C(C(C)CC(=O)N1CC(NC(c2ccc(COC)s2)=O)C(C)C1)OC CC1(C)CC(C(=O)NOCC2CNC(=O)CO2)CN(C(c2ncccc2N)=O)C1 c1(C(=O)NCC2C(NC(c3ccc(C)s3)=O)CCCC2)nn(C)c(C)c1N C(=O)(CCC(C(C)C)NC(=O)C=C=C(C)C)N(C(CCCC)C)C CCC(CNC(C1CC(=O)C12CCC2)=O)(CC)C(=O)N(C)CC1(O)CCOC1 n1(CC(N2CC(NC(c3c(SC)csc3)=O)C3(C2)CC3)=O)ccc2ccccc12 c1(C(N)=O)cc(NC(=O)Cn2cnc(-c3ccccc3)cc2=O)cc(F)c1Cl C(=O)(C(C)(C)CCCNC(=O)CC(C)C(F)(F)F)N1C(C=C)CCC1 C(=O)(C(CCC)CCC)N1C(CNC(c2cn(CCC)nc2)=O)CCC(C)C1 C(Cc1ccco1)(C(=O)N1CC(CCO)C1)NC(CCOCC#C)=O c1(OC)ccc(F)cc1C(=O)NC1CCN(C(c2cnn(C)c2C#N)=O)CC1O C#CCCCCCC(=O)N1CCC(CNC(=O)CSCCNCC)C1(C)C.C N1(CC(C2CCC(C)CC2)CC)CC2CC1CCC2NC(C1COCCN1C)=O N1(CCOC)CCC(N=c2[nH]c(=NCc3ncc(C)o3)[nH]c3ncn(C)c23)C1 CC1CC(NC(=O)C)CCN1C(c1[nH]cnc1C#N)=O.C(=O)CCC1CCCC1.N CC(=O)CCCC(C)C(=O)NC(C)C(=O)N(C)CCO Cc1ccc(N)c(C(=O)NCC(C)(CC(C)C)NC(=O)CC2CCC(=O)N2)c1 c1(C(C(=O)NCC)N(CCCCCC)CCCCCC)cccc2ccncc12 CS(=O)(=O)C1(C(=O)NCCCC(CO)NC(C2CC=CCO2)=O)CCCC1 O=C(N=c1[nH]ccc2cnccc12)NCC1CC2CCC2C1 N1(C(C(N2CCNC2=O)C)=O)CC(F)(CNC(C2CC(F)(F)C2)=O)C1 C1(Cl)(C(=O)NC2CN(C(=O)CCc3cnn(-c4ccccc4)c3)C2)CC12CCC2 N1(C(c2cc(C)sn2)=O)CCOC2(CCCN(C(C3C(C#N)C3(C)C)=O)C2)C1 C(=O)(CCCC(F)(F)F)NCC1(C(=O)Nc2cc(C)c(Cl)nc2)CC(C)(C)C1 C1(C(C)NC(c2c(Cl)csc2Cl)=O)CCCN(C(C23CC4CC2C3C4)=O)C1 C(CS(=O)(=O)c1ccccn1)NC(C(=O)NCC1CCNC12CCOCC2)=O N1(C(c2n(CC)ccc2)=O)CCC2C(C1)CN2C(=O)C(F)C(C)(C)O n1(CC)ncc(C(=O)NCC2CCN2C(=O)CCCn2nc(C)nc2C)c1.C N(C1CN(C(=O)C=C(C)c2cccnc2)Cc2ccccc21)C(C(C)=CC)=O C1(C(=O)NCCCCCCF)(NC(Cn2ncn(C)c2=O)=O)CCC(C)(C)C1 C1(NC(C2CCC(NC(c3nccc(OC)c3)=O)C2)=O)CC2CC1CC2CO C1(CNC(=O)CCc2cocn2)CC(F)CN1C(c1cc(F)c[nH]1)=O N1(c2cc(OC)ncn2)CC2CC(NC(c3cnccc3Cl)=O)CC2C1 c1(C(=O)NC(CCCNC(C2CC(C)C(=O)CC2)=O)C)c[nH]c2cc(F)ccc12 c1(C(N2CCN(C(C=CC=C)=O)CC2C(C)C)=O)ccc(C(C)(F)F)nc1O.C CC1(C(=O)NCC(CC2CCC(F)(F)CC2)CO)CC(C2CC2)=NO1 c1(CC(N2CC(CCNC(=O)C)(OC)C2)=O)cn2ccsc2n1.C1CCOC1 CC(CCN=c1[nH]ccc(C#N)c1[N+](=O)[O-])NC(C1(C)CC1C(F)(F)F)=O N1(C(c2cc(CC)n(C)n2)=O)CC2OCC(NC(=O)C(C)(CC)OC)C2C1 c1(C(=O)NC(c2ccc(C)cc2)CO)cc(C)c2n[nH]cc2c1 C1(CC)CCN(C(C2CC2C(C)(C)C)=O)C1C.c1(C(=O)N)c[nH]c(C)c1 N1(C(CCC(C)OC)=O)C2CCC(C2)C1C.c1(C(=O)N)c(C(C)C)cccc1F C1(N(C(=O)COCCCOC)CCC)CCN(C(=O)CCN2CCOCC2)CC1 CC(C(CO)NC(=O)CC1CC2(CC2)C1)NC(c1cnn(CCF)c1)=O c1(C(=O)NC2(CF)CCN(C(=O)CO)C2)cccc2nc[nH]c12.c1nccs1.C c1(C(=O)NC(CCOCC)C)oc(CNC(c2cccs2)=O)cc1C c1(C(=O)OC)cc(OCC2CCN(c3cccc(Cl)c3)C2)ccc1C N1(C(c2nc(CCC)oc2)=O)CCC(C(C)NC(=O)Cc2scnc2C)CC1 C1(C(=O)NCCC(C)N(C)C(C2CCN(C)CC2)=O)CCC(F)CC1 c1(C(=O)Nc2ccc(C(=O)OCC3CCC3)cc2)cccc2c1CCCC2 Cc1csc(CCNC(=O)CCC2(C)CN(C(=O)CNC=O)C2)n1 c1(-c2ccn(CCOC)n2)nc(-c2ccc(N)cc2)nn1C1CCSC1 C12(C(=O)NC(C3CCN(C(C(C)=C4CCC4)=O)CC3)(C)C)CC1COC21CCC1 C(C)(C(O)C(=O)NC(C)(C)CCNC(c1cnc(C2CC2)nc1)=O)SC N1(C(C2CCCC(C)(C)C2)=O)CC(C)(C)OC2(C1)CN(C(C1CC13CC3)=O)C2 CCC(C)CCCC(=O)N(C1CCN(C(c2cn(C)nc2C(F)(F)F)=O)C1)CC C1(S(C)(=O)=O)(C=O)CCOCC1.C(C)(C)C(C)C.CCC(C=O)NC(C)=O N1(C(c2c(CC)cccc2)=O)CC2CC1CC2NC(c1cccs1)=O c1(C(=O)NC)cccc(C(=O)O)c1.n12nccc1NC(=O)C2C CCCC(C)C(=O)Nc1cccc(CNC(=O)C(C)Cc2cnco2)c1 N1(C(COCCCC)=O)CCC(C2CC2)(C)C1.c1(C(C(=O)N)C)ccc(F)cc1 N1(C(c2cc(C)c(C)[nH]2)=O)CCC(NC(C23CCCC(C2)OC3)=O)CC(O)C1 C(C)(CCCCNC(=O)Cn1cnc(=N)[nH]1)NC(c1nc(C)oc1)=O c1(CC)ccc(C(=O)NC(C)CCCNC(c2cnnc(O)c2)=O)c(Cl)c1 C12CCCCC1(C)NC2=O.C1(NC(=O)OC(C)(C)C)CC(O)C(F)C1 C1(CNC(c2cc(CC)[nH]n2)=O)CCCCCN1C(=O)CCCc1ccncc1 C1(C)CC(F)(F)CN1C(=O)CNS(N)(=O)=O.C(C(C)C(=O)N)OCC CC(C)C(C)(C)C(=O)NCC1CN(CC#N)CCCO1 c1(C(=O)OC)cc(NC(CC2CCCCO2)CO)cc(Br)n1 C1(CC(N2C(C)(C)CCC2C(=O)N(C)C)=O)CC2(CCNCC2)CO1 C1(C(C)C(=O)N2CCC2CF)CCN(C(c2cc[nH]n2)=O)C1 N1(C(CSCC(=O)NC(C)(C)C)=O)CC(S(C)(=O)=O)CC12CCOCC2 C1(CNC(c2ccc(C#C)o2)=O)CN(C(=O)C(CCC)N(C)C)C(C)(C)C1 c1(OC)cc(C(=O)NC2CC3(C2)CN(C(c2ccncc2OC)=O)C3)ccc1C c1(C(N2CC(Nc3cccc(OC)c3)C2)=O)cc(S(=O)(=O)N(C)C)cn1C.O c1(CNC)ccccc1-c1cccnc1C(N1CCC(SC)CC1)=O C(=O)(C1=CCCCCC1)NC1C(NC(CN2CCC(C)(O)C2)=O)CC1 CC(C)(C)C#CC(=O)N1CCOC(CC(=O)NC(CCO)C2CCC2)C1 CN1CCC(NC(=O)NCc2cc(C(=O)OC)n[nH]2)(CO)CC1 c1(C(=O)NCCC2CCN(C(CC(CC)C)=O)C2)cc(F)cc(Cl)c1O S(=O)(=O)(CC(=O)N1CCC(C(C)NC(=O)Cc2cccc(C)c2)CC1)NC c1(C(N2CCC(n3cnnn3)CC2)=O)cc(Cn2cncn2)ccc1O C12(NC(c3c(C)cnnc3)=O)CCCCC1CN(C(=O)CC=C(Cl)Cl)C2 c1(CC)c(C(=O)N(CC(C)NC(C2(NC(N)=O)CC2)=O)C)nnn1C C1(CC)COCCN(C(C2(CO)CCN(C(c3cc(C)ncc3C)=O)C2)=O)C1 N1(c2ccnc(SC)n2)CCC2(CN(C(C3CC3C3CCCC3)=O)CC(C)O2)C1 C1(C(N2CCCN(C(=O)Cn3cnc([N+](=O)[O-])c3)CC2)=O)COCCC1(F)F Cc1ccc(Br)c(Cn2cc(C3CCC3C(=O)N)nn2)n1.C1C(F)(F)C12CCC2 C=Cn1cc(C(N2CCCC(N(C(C3CCOCC3)=O)CC)CC2)=O)c(C)n1 C1CCCC(C)C1.C(c1ccco1)=C(C)C(=O)NC1(C)CC(NC(=O)C)C1.O Cc1ncsc1-c1cn(CCNC(C2CC2c2cccnc2)=O)nn1 C1(C(=O)NCC)CCN(C(C2(F)CN(C(=O)C(Cl)Cl)C2)=O)CC1 C(=O)(C#CC1CCCO1)N(CCC(c1cccs1)NC(c1n[nH]c(C)c1C)=O)C C1(NC(C(C)NC(C)=O)=O)CC(F)CN(C(=O)CCCCCNC(N)=O)C1 N1(C(c2cncc(OCC)c2)=O)CCN(C(C2CC23CC(C)(C)C3)=O)CC1C N1(C(c2c(CC)ncs2)=O)CCCCC(C(=O)NCCCCS(C)=O)C1 C(=O)(C(C)CCCC(C)C)NCCOCC(=O)NC(CC#C)CC(=O)OC c1(C(CC)NCCCc2ncco2)ccc(C)c(OC)c1 C(CO)(CC(F)(F)F)NC(C(C)(CO)NC(c1cn(C)nc1)=O)=O Cc1cc(-n2nc(-c3nc[nH]n3)nc2C(C)OCc2ccc(F)cc2)cc(C)c1 CN1CC=CCC1CC(N1CCCC1C(C)C)=O.N1(CC(=O)N)C(=O)CCC1=O CC(C)CCC(C(=O)N1CCC1CN=[N+]=[N-])NC(=O)CCc1ccccn1 c1(CCC(=O)NC2CC(O)(CNC(CCC3N(C)CCC3)=O)C2)ccccc1F c1(C(=O)NC2CCC(NC(=O)COCC3CCCO3)CC2)[nH]cc2c1CCCC2 n1(CCC)cc(C(=O)NC(CNC(c2cc(C)c[nH]2)=O)CCOC)nn1 N(C(=NCC1CN(C(=O)OC(C)(C)C)C1)NCC1CCOC1)C(C=C)C.O Cc1c(C(=O)NCC=CCNC(=O)CC2OCCOC2(C)C)nc2sccn12 N1(C(C=CC(C)NC(=O)CCc2nncnc2O)=O)CCN(CCOC#N)CC1 C1(CC)C(C(N2CC=CC(OC)C2)=O)CCCN1C(c1c[nH]c(C(N)=O)c1)=O N1(C(CCn2c(C)ccc2C)=O)CCCN(C(=O)C(F)OC(F)(F)F)CC1C CC(CN(C)C)CC(=O)NC(c1ccc(C(F)(F)F)cc1)C(F)(F)F c1(CN2C(C(N3CCC(N(C(C)=O)C)C3)=O)CC3CC32)cncc2ccccc12 N1(C(C2N(C)CCC2)=O)CCC(C)(NC(c2ccc(C(N)=O)cc2)=O)CC1 c1(NC(C)=O)ccsc1C(=O)NC(C)CN(C)C(c1ccccc1)=O c1(C(c2cccs2)NCC(=O)NC)cc(OC)c2c(c1)OCCO2 CC1(NC(=O)Cc2cccc(Cl)c2F)CCCN(C(C2CCS(=O)(=O)C2)=O)C1 CC1(O)CCCCC1C1CCCN1C(=O)NCCCN1CCCCC1 C1(NC(C2(COC)C=CCC2)=O)CCCCC1.C(=O)C.[SH](C)(=O)=O.C C(=O)(C(N)CC1CC(F)(F)C1)NC(c1nc(C(C)(C)C)no1)CC Cc1cnc(Cl)c(S(=O)(=O)NCC2CCCN2Cc2csc3ccccc23)c1 N1(C(C(C)(C)c2cncs2)=O)CCOC(C)(CNC(=O)CSS(C)(=O)=O)C1 C1(C(=O)OC(c2ccc(Cl)cc2C(F)(F)F)C)CCCCCC1(F)F Cc1cc(C)nc(CNC(=O)CC2(C)CC2)n1.C1(C=O)CCC(=O)N1C.N C#Cc1ccccc1CC(=O)NCCC1CN(C(=O)C=CCO)CC(C)O1 C=CCC(CNC(=O)C(C)n1cccc1)C(=O)N1CC2CCCCC12 n1(CC#C)c(C(=O)NC2CN(C(c3ncsc3Br)=O)C2)cc2ccccc12 CC1(C)CN(c2ncc(O)cn2)CCC1NC(c1ccc(OC(F)F)cc1F)=O N1(C(c2c(CC(C)C)cccc2)=O)CC2CCC(C1)N2c1nc2ccccc2o1 C1(C(N(C2CN(C(=O)Cc3cncc(O)c3)C2)C)=O)C(F)(F)C12CC2 C1(CCC)CCN(C(=O)C)CC1.C1(CC=O)CC(O)C1(C)C.CCN(C)C.S C1(C(=O)NCC2N(C(C(CC#C)C)=O)CCN(C)C2)CC2CC(C1)CC(F)(F)C2 CC(C)C(CCC(=O)N(C)CC1COC(=O)N1)NC(c1ccccc1C#N)=O C1(C(=O)N)CC2(C1)CC21CC1.C1(CC)C(C)CCN1C(=O)CCC1CCCC1 N1(CCC)CC(CNC(=O)CN2CC(C(c3ccc(F)cc3)=O)C2)CC1=O C(C(C)CC(=O)NCCOC1CCN(C(c2ccsc2C)=O)C1)OC N1(C(CCc2c(C)ncs2)=O)CCC2C(C1)CN2C(C1CC2(C1)CC2(F)F)=O C12(C(N3CC4C(NC(c5ccc(OC)c(N)n5)=O)C4C3)=O)OCCCC1C2(F)F N1(C(C(CNC(C2(OC)CCCOC2)=O)C(C)(C)C)=O)CCc2oc(C)nc2C1 C1(C(=O)Nc2c(C)nsc2)CN(C(=O)CC2CC=CCC2)CCC1(C)C c1(C(=O)NC2C(C)N(C(=O)Cc3nncs3)CCC2)ccc2[nH]ccc2n1 c1(N(CCC)C)ccc(C(=O)NCC(C)CNC(c2coc(C)c2)=O)cc1 C1(F)CN(C(C2C3CCCC23)=O)C1.c1(C(C(=O)N)NC(C)=O)ccccc1.C Cc1ccc(C(O)CNC(=O)C(Cc2cn(C3CC(O)C3)nn2)N(C)C)s1 c1(C(N2C(C(C)(C)CNC(C3CCC=CCC3)=O)CCC2)=O)cc2occc2s1 C1(N(C)C)CCC(NC(=O)CC2(N(C)C(C3CC=CC3)=O)CC2)C1 CC(O)CCCCCC(=O)N1CCC(NC(=O)Cc2cc(F)cc(Cl)c2)C(O)C1 CC1(C)C2CN(C(=O)CC3CN(C(=O)CC(F)(F)F)CC34CC4)CC12 N1(C(C=C(C)C)=O)CCC(CCNC(=O)Cc2cc(F)ccc2F)C(F)(F)C1 c1ccc(C)o1.C1(C(COC)(C)NC(=O)C(=O)NC2CC2)CC(F)(F)C1 c1(CN(C(c2c(C)cc(F)cc2)C(=O)NC(C)C)C)ccc2c(c1)OCCO2 c1(N(CC(N2CCOCC2)=O)C)nc(=NCc2ncc[nH]2)[nH]c2c1SCC2 C1(C(N(C)Cc2ccc(O)cc2)=O)CC2CCC(C1)N2C(=O)CC1COCC1O CC(C(=O)C(F)(F)F)N(C)Cc1ccc(C(=O)OC(C)(C)C)cn1 c1(C(N2CCC(Nc3cccc(C(C)NC(C)=O)c3)C2)=O)c(N)cc(C)cc1F N#Cc1ccc(CC(N2CCC(O)C(C(=O)Nc3ccnc(C(N)=O)c3)C2)=O)cc1 C1(CNC(c2ccn3nnnc3c2)=O)CN(C(C23CCC2C3)=O)CC12CCC2 C12(C(N(CC(C)NC(=O)CCCCCC(C)O)C)=O)CCCC(=O)N1CCC2 c1(SCC)ccc(C(C)NCCC(C)C)cc1 C(C(CC(C)C)NC(=O)CC1(C)CCOC1)NC(C=C(C)C1CC1)=O Cc1cc(Cl)ncc1CC(=O)NCC12CC1CN(C(=O)CCCC1CCC1)C2 C1(C(=O)NCC(C)(C)NC(c2cnc(-c3ccco3)s2)=O)CC2CCCCN2C1 c1(NC(CCC2N(Cc3cncc(C)c3)CCC2)=O)cnc(F)c(C)c1 c1(C(c2n(CCC)nnn2)NCC(C)C(C)C)ccc(CC)cc1 c1cccc(C(N2CCOCC2C(N)=O)=O)n1.c1(C(C)C)oncc1C(=O)NC N1(C(CCc2ccc(C)c(C)c2)=O)CC2CC1CN(C(c1cnc(S)nc1)=O)C2 CC1COCCCN1C(C1CCN(C(C2(F)CCCCC2)=O)CC1)=O CC1(NC(c2cn(C(F)(F)CO)nn2)=O)CCN(C(C2CCC=CCC2)=O)CC1 c1(C(N2CCCCC(SCC)C2)=O)cccn2[nH]c(=N)nc12 c1(CC(=O)NC)ccccc1NC(=O)Cn1ccnc1.C1CCC(C2CC2)O1 C1(OC)CCCC(CC(=O)NC(C)CC(C)NC(=O)CN2CC(=O)NC2=O)C1 N1(S(CCCOC(C)C(=O)O)(=O)=O)CC(O)CC1c1ccccc1 Cc1nsc(NC2CC2)c1C(=O)NCCC.N(C)(S(N)(=O)=O)CC=O C(CCCNC(=O)C(C)(C)C1CCC1)OC.c1(C(=O)N)cnn(CC(F)F)c1 N1(c2cc(C)[nH]n2)CCN(N2CC3CC2C(F)(F)C3)CC1 N1(C(C(CC)(C#N)CC)=O)CCC2(CCCN2C(=O)C=Cc2nc(C)co2)C1 N(C1CCCSc2ccc(Br)cc21)C(N(OC)C)=O C(=O)(CC(C)C(=O)NC1(CF)CN(C(c2cnc(-c3ccccc3)s2)=O)C1)OC N1(C(C(=O)NCC(=C)C)C2CCCC2)CCCC(N2CCOCC2)C1 C(C(=O)N1CCCCCO1)OC1CCN(C(c2cnn(C(C)C)n2)=O)CC1 c1(CN2CC(CNC(=O)CCC3CCC3)OCC2)ccc(N2CCCC2)cc1Cl N1(C(C2(COC)CCOC2)=O)CCN(C(=O)C(C)(C)c2cncs2)C(C)C1 CC(CCCCNC(=O)CCc1ccccc1O)NC(=O)C(O)CCN(C)C c1(OC)ccc(C2CCN(c3nnnn3Cc3cc(Cl)c(Cl)s3)CC2)cc1 c1(C(N2CCN(C(C(CC#C)C3CC3)=O)C(C)C2)=O)cnn2c1OCCCC2 c1(C(N2C(CCC)CN(C(=O)Cc3cn[nH]c3)CC2)=O)nc2ccccn2c1F c1(C(=O)NC2CC(C)N(C(=O)CCCC(F)(F)F)C2)cncc([N+](=O)[O-])c1 c1(CN2C3C(C(N(CC)Cc4ccc(Cl)cc4)=O)C(C3)C2)cnc(O)nc1O C=C(Cl)CN=c1nc2c(ncn2CCOC)c(NCc2cc(C)nc(C)c2)[nH]1 c1(C(=O)NC2(CCNC(c3n(C=C)nnc3)=O)CCCC2)nc(C)ccc1C n1(CC=O)nnc2ccccc12.C=C(C)C(C)(C)C(=O)NC(C)CC(F)(F)F.N CCCCC(O)C(=O)NC12COC(C1)C(NC(C1CN(S(N)(=O)=O)C1)=O)C2 c1(CC)cc(C(N2CC(CCNC(=O)CN3CCCCC3)C2)=O)cc(F)c1 C1(C(=O)NCCN(C2CCCCC2)C(C2C(C)(C)CC2)=O)CCCC(=O)O1 C(=O)(CCCCC(=O)N1CCC(C2(NC(=O)C3=CCOCC3)CC2)C1)NC c1(C(=O)NCC#CC(=O)NCC2ON=C(C)C2)cc(F)n(C)n1 C(C(CC)(CC)C(N)=O)NC(C(C1CCOC1)NC(C(CC)OCC)=O)=O c1(C(N2CC3(C(C(=O)Nc4c(C)ccnc4Br)C3)C2)=O)cccc2cn(C)nc12 N#Cc1ccc(-c2ocnc2C(=O)N(C2CCN(C(=O)C3CC3)CC2)CCO)cc1 C(=O)(CC1OC(=O)c2ccccc21)N(CCCNC(C1C=CC=CC=C1)=O)CC N1(C(Cc2c(OC)ccc(Br)c2)=O)CCC=C(C(=O)NC(C2CCC2)C)C1 N1(c2c(C)c(NC3CN4CCC3CC4)ncn2)CCn2c(C3CC3)nnc2C1 C(C(C(=O)NC1(C)CC1)NC(C1CC(O)C1)=O)OC C(=O)CC(C)(CC)C=O.C1(NC(C2(COC)CCC2)=O)CC(C(F)F)C1 C#CC1CC2(CC(C(N3CCN(C(c4ccnc(S)c4)=O)C(C)C3)=O)C2)C1 C1CCCCN1C(=O)Cc1cc[nH]c(=N)c1.C1(C(N(CC)C)=O)CCCN1N=O Cc1ccc(C#N)c(NC(c2ccc(-c3ccccc3N(C)C)c(C)n2)=O)c1 C1(C(N2CC3(CN(C(C(CCC)OC)=O)C3)C2)=O)CCc2nc(CC)ncc2C1 C(=O)(CCCCN=[N+]=[N-])NCCC(CNC(C(C)NC=O)=O)(C)C N12CCN(CC1)CC1(CC1)C2=O.C1(C(=O)Nc2cnns2)(OC)CCSC1 C#Cc1cccc(C(=O)NC(C(=O)Nc2ccc(C)cc2CO)C2CC2)c1 Cc1cccc(F)c1C(N1CCCC1CNC(C1(n2cccn2)CCC1)=O)=O C12CC3(CC3)CN1C2=O.CC1CCN(CC(N2CCC(OC3CC3)C2)=O)C1 CC1(C)OCCC1(O)C(=O)N1CCC(C(=O)NCCC2COCCO2)O1 c1(C=O)cc2ccccc2cc1.C(F)(C(=O)NCC1CC1)=CC.CC#N.C c1(C(=O)NCC(CCCC)NC(c2ccc(F)cc2OC)=O)c[nH]cc(C)c1=O C1(C2CCN(C(C3CC3c3ccsc3)=O)CC2)(NC(C2CCN(C)C2)=O)CCC1 C=CCC(CC(=O)NCc1cn(CC=C)nn1)NC(C1(C(C)=O)CC1)=O N1(C(c2c(C)cnn2C)=O)CC(NC(=O)CCCc2nccs2)CC(C)C1 CC1CCN(C(c2ccc(C3CC3)c(F)c2)=O)C(C)C1.c1(C(=O)N)cc(Cl)ns1 C=C1CC2(C1)CN(C(C1CN(C(=O)C(CC)CCOC)CCN1C)=O)C2 c1(C(N2CC(C(N(CCC(=O)O)C)=O)C3(C2)CC3)=O)cc(C#N)ccc1N.CC c1(CN2CCN(Cc3ccc(OCC)c(OC)c3)CC2)cc(=O)n2ccsc2n1 C1(CNC(Cc2cc(C)on2)=O)C2CC1N(C(=O)Cn1cccn1)C2 C1(CNC(C(C)c2ccsc2)=O)CCCCN(C(c2ccc[nH]2)=O)C1 N1(C(C(COC)C)=O)CCCC(C(=O)NCCc2cncc(C)n2)C1 N1(C(C(C(=O)OC)(C)C)=O)CCCC(NC(=O)C(c2nc(C)cs2)C)CCC1 c1(CC(=O)N(c2ncc(-c3ccccc3)cn2)CC2CCNC2)ccc(F)cc1 c1(C(N2CC(O)C2)=O)ccc2oc(S)nc2c1.Cn1cc(C(=O)C(=O)NC)cn1 C(c1ccccc1OC(F)F)=CC(=O)NC1CCCN(C(CC=C)=O)C1 N1(C(c2ccc(CC)cc2)=O)CC2CCC1CN(C(=O)C(O)C(C)C)C2 N1(C(c2c(C)cn(C)n2)=O)CCN(C(C2(CC(F)(F)F)CC2)=O)CC12CCC2 O=C(CCCCN1CCCC1)NCc1csc(C(=O)NCCC2CC2)c1 C1(CC(=O)NC2CCN(C(c3c(C)cccn3)=O)CC2F)CCn2cncc2C1 Cn1cc(CNC(=O)C=CCNC(c2cscn2)=O)ccc1=O c1(C(=O)NC2(C)CCCN(C(c3ccc(SC)cc3)=O)C2)cc(C)c(C)nc1C c1(C(=O)NCCOCCCNC(c2ccnn2CC(F)F)=O)ccncc1 c1(NC(=O)NCCCCc2ccc(Br)cc2)cccc(CC(F)(F)F)c1 O=C(CN=c1cc[nH]cc1)N1CCC(CF)(NC(C23CCCC2C3(F)F)=O)C1 N1(C(CNC(CC)=O)=O)CC2CC(NC(c3c(Br)noc3C)=O)C1C2 Cc1ncc(NC(=O)C(C)CC2CC2)c(C)c1C.C(=O)CCC(C)(C)N(C)C.N CC1(C)CC(F)(F)CCC1C(N1CCN(C(C23CCC(C2)C3)=O)CC1CO)=O N1(C(C2(C(C)(F)F)CC2)=O)CC2CCN(C(=O)C(c3ccc(Cl)cc3)CO)C2C1 c1(NC(C)=O)cccnc1C(N1CC(NC(C2CCCCS2)=O)CC1C)=O c1(N2C(C)C(NC(=O)COCC3CCCO3)CCC2)ccc2nccnc2n1 N1(C(C(C)SCCCC)=O)CCOCC(CNC(C2CCC(N(C)C)CC2)=O)C1 C1(NC(C(CO)N(C)C)=O)CC2CN(C(C3(C)COC(=O)C3)=O)CC2C1 N1(C(=O)OC)CC2CCC1C(C(=O)NCCCCCC)C2.C(=O)(CC1CCC1)N CC1Cc2cc(C(=O)NC(C)CN(C(=O)CC3CCCO3)C)ccc2O1 C1(CN(C(=O)C2=C(Cl)CC2)C)CCCC(NC(=O)CCCn2cncn2)C1 C(=O)(C(C)CC(C)C(C)=O)N(CC(=O)NCC(CC)(CC)OC)CCOC C(C(C)(C)C(=O)NC1CCN(C(c2cnnn2-c2ccccc2Cl)=O)C1)OCC C(=O)(CC(F)(F)C(F)(F)F)N1CCC(C)(C)C1.c1(COC)c(C=O)cnn1C.N N1(C(CC2CCC(=O)NC2=O)=O)CC2CCOC2(CNC(=O)Cc2cc[nH]c2)C1 C(=O)(C(C)(C)CCC#N)N(CCCNC(=O)CCc1cccnc1Br)CC N1(C(=O)Nc2ccc(OC)cc2)CCC(CN(C(=O)CCC(C)C)C)(OC)CC1 N1(C(C2=C(C)S(=O)(=O)CC2)=O)CCC(NC(=O)Cc2c[nH]nc2C)CC(C)(C)C1 C1(NC(C(CC#C)(C)C)=O)CCN(C(=O)Cc2cccc3nsnc23)CC1(C)C N1(C(C2C(OCC)C2)=O)CC2(CCCC2)C1.c1(CC=O)c(C)ncnc1C.N Cc1ccc(C(=O)NCC(C)(O)CNC(=O)CCCc2ccccc2)c(O)c1C c1(C(N(CC(C)C)C(c2sccc2C#N)=O)=O)nc2ccc(Br)cn2n1 N1(Cc2cnc(CC)s2)CC2C(C1)N2C(c1cccc(Cl)c1)=O CC1CCC(NC(=O)CC2(CO)CCOCC2)CN1C(c1nc(=O)cc(N)[nH]1)=O N1(C(C2CC(C)C2)=O)CCC2CN(C(c3cnc4c(Cl)cccn34)=O)CCC12 CC1N(C(C2CCCCN(C(=O)Cn3ccccc3=O)C2)=O)CCCC1(C)C CC1(CCCN)NC(=O)NC1=O.n1(C2CCC2)cc(CCc2nn[nH]n2)nn1 c1(C(N(C(C(=O)NC(C(=O)OCC)C)CC)C)=O)cc2n(n1)CCC2 Cc1cc(NNC(=O)NCc2nc(-c3ccccc3)cs2)n2ncnc2n1 c1(C(N2CC(NC(CC(=O)N(C)C)=O)C(O)C2)=O)nn(C)c2c1CCC2 C1(C(N2CCCC2)=O)CCn2cc(C)nc2C1.c1(OC)nn(C)cc1C(=O)NC C1(CC(=O)N(C2CC(O)C2)CC)CCN(C(=O)CCCC2CCCO2)C1 CCCCCCC(C)CC(=O)NCCCNC(c1cc(O)ccc1C)=O CC1(C)CN(C(c2cc(CO)ccn2)=O)CC2(CN(C(C3CC3[N+](=O)[O-])=O)C2)O1 CN=c1ccc(C(N2CC3C(CC(N4CCC(OCC5CC5)C4)=O)C3C2)=O)c[nH]1 C=CCCCC(=O)N1CCC(C)(C(=O)NCCn2cccn2)C1 C1(NC(CC(=O)NCC2CC2)=O)CC2CCC1N2C(C1CC=CCO1)=O Cc1cnnc(O)c1C(=O)NCC(c1ccc(F)cc1)NC(C1CC1C)=O CC1(C)CC2CCCN(C(=O)C=C3CCC3)C12.C1(CC(=O)N)CC2(CC2)C1 c1(C(N(C(CNC(c2ncccn2)=O)C2CC2)C)=O)cccc(F)c1F C1(O)(CN(C)C(C2(C)CCCO2)=O)CCCN(C(C2CCS(=O)CC2)=O)C1 Cc1[nH]nc(C(=O)NCC2(CNC(C3CCC(C)C3)=O)CCCCC2)c1C CC1(C)C2CCC(C2)C1C=O.c1(CC=O)cc[nH]c1.C1(CC)(C=O)CC1.N N1(C(c2n(CC#C)ccc2)=O)CC(NC(c2cocc2C)=O)CC12CCOCC2 c1(C=O)cc(C2CC2)nn1C.C(C)(C)C=O.C(C)CO.CCCNC(=O)N c1(NC(CC2(C)CN(N3CCN(CC(F)F)CC3)C2)=O)ccncc1[N+](=O)[O-] C(=O)(C(N=[N+]=[N-])C(C)C)N(CC(=O)NC1(c2nc(C)no2)CC1)CC#C C1(N(C(C2CCN(C(C)=O)C2)=O)CC2(C)CCCC2)CC2CNC1C2 CCCCN=C(NCCCN1CCOCC1)NCCNC12CCCCC1C2(F)F CC1CN(C(=O)Cn2cnnc2)CCC1CNC(C12CC(C)(C1)OC2C)=O N1(C(C(=O)NCCOC)=O)CC2CN(Cc3ccc(C(F)(F)F)cc3Cl)C2C1 N1(C(Cc2c(C)scc2)=O)CCC2(CCN(C(C3CC4(CSC4)C3)=O)CC2)C1 C1(NC(CCC(C)SC)=O)CN(C(=O)CSCc2csc(=N)[nH]2)CCC1O N1(C(C2CC(OC)C23CCC3)=O)CC2=C(C1)CN(C(C1CS(=O)(=O)C1)=O)C2 C1(CNC(CC(c2cccc(F)c2)C)=O)CC2(CC2)CN1C(c1ccncc1)=O N1(C(C(=O)NCCOC)=O)CC2CCC1CN2C(c1cc(CS)ccc1F)=O c1(C(NC2CCN(C(C3OCC3(C)C)=O)CC2)=O)ccccc1C(C)(C)C.CC Cc1ncc(Cl)cc1C(N1CCN(C(c2cc(C3(O)COC3)on2)=O)CC1)=O C(=O)(C(C)(C)C1=CCSCC1)N(CC(CC)NC(C1CCC1)=O)C.C(C)=O.N c1(C(=O)NCC(C)NC(C2(C)CC2)=O)ccc(Br)cc1F CCCCCCC(C)C(=O)NCC(CCOC)NC(c1cc(C)c(Cl)cc1F)=O CCCC(C(=O)N1CC(NC(=O)CC2CCCCO2)C2CCCC12)C(C)C CC(C)(O)C(C(=O)NCc1ccnc(F)c1)NC(=O)CC1CC2CC2C1 c1(C(=O)NCCN(C(CC(CC)C(C)C)=O)CC(C)O)ncnc2c1CCCC2 C1(O)(CNC(c2n(C)ncc2N)=O)CCN(C(C2CC2(C)Br)=O)CC1 c1(CNC(C2(CCNC(C(C)(C)C)=O)CCC2)=O)cncc(F)c1 Cc1cnc(NC2CN(C(C3CC4CC4CC3C)=O)CC2(C)C)nc1O Cc1nc(SCCNCC(c2ccnn2C)O)n[nH]1.C1CS1 C1(C(=O)NCCOCCN(C(=O)C=CC2CCC2)C)CCCCC1C1CC1 c1(C(NOCC(=O)OC)=O)cc(C)c(Br)c(Cl)c1 C1(C)CCOCC1.c1(CNC(C2C(C(=O)OC)C2)=O)nccs1.C(=O)C C1(C)(C(=O)NCC(C)C2CC2)CC2CCC1CC21OCCO1.C(=O)CNC=O.N c1c([N+](=O)[O-])c(C)n[nH]1.c1cccc(C)c1.c1(C(=O)OCC)nc(C)no1.N C1(NC(C2(CC#C)CC2)=O)CC2CCC(C1)N2C(c1cc(C)[nH]n1)=O c1(N2CC3CC(NC(C=CCC)=O)CC3C2)nc(C)nc2sc(C)c(C)c12 C1(CC(=O)NOCC=CCl)CC2(CC2)CN1C(C1CCCC12CCC2)=O n1(CCSCCCC2C(C)=[SH]CC2)c(-c2ccncc2)nc2c(C)cccc2c1=S c1(CC)sc(C(C)NC(=O)NCC(c2ccc(OC)nc2)(C)C)cc1C Cc1cncc(C(N2CC(N(C)C(c3c[nH]cc(Cl)c3=O)=O)C3(CC3)C2)=O)c1C Cc1nn(C)c(C)c1CC(N1CCC12CN(C(C1COCCN1C=O)=O)C2)=O N1(C(C(C2CCOCC2)C)=O)CC(NC(=O)CS(N)(=O)=O)C2(CC2)C1 C1(C(=O)NC2C(C(N(CC(C)O)CCF)=O)CC2)CCCC(=O)CC1 C1(CNC(c2ccc(C)[nH]2)=O)CN(C(=O)C(C)Sc2nncn2C)CC1C c1(NC(C2SCCN(C(C=C(C)C)=O)C2)=O)cccc(Cl)c1[N+](=O)[O-] N1(C(c2c(S(C)=O)cccc2)=O)CC23CCCCC2(C1)CN(C(=O)CNC=O)C3 N1(C(CCNC(=O)CO)=O)CC2CN(Cc3cc(Cl)c(Cl)s3)CC2C1 N1(C(C=CC(CC)C)=O)CCCC(O)(CNC(c2c[nH]nc2[N+](=O)[O-])=O)C1 C(=O)(CCC(C)(C)F)N1C(CNC(C(C)(C)SC)=O)COCC1 N1(CCCCCNC(CCCN(C)C)=O)CCC(NC(=O)COCCCF)CC1 CC1CC(CCNC(C2CN3CCC2CC3)=O)CCN1C(=O)CC(F)F N1(C(CCCC#C)=O)CC2CC(CNC(=O)C(C)Sc3ccccn3)CC1C2 c1(C=O)cnc(F)c(F)c1.N1(C(c2cnc(C(C)=O)s2)=O)CCC(O)(CC)C1.N Cc1sc(=O)n(CC(=O)NCC23CC2CN(C(=O)C=C(Cl)Cl)C3)c1C C1(C#N)(C(N(CCOCCNC(C(CC=C)OC)=O)C)=O)CC12CCCC2 C1(CC(=O)NCC2CN(C(=O)Cc3cccnc3O)C2)CCc2ccccc2C1 C1(CNC(Cc2c(C)occ2)=O)CCN(C(=O)CN2C(=O)CCCC2=O)CC1O C1(CC)CN(C(=O)C=Cc2cccc(O)c2)CCN1Cc1cc(Br)c(C)s1 N1(C(C2CC(CNC(=O)Cc3nncs3)C2)=O)CCN2CC(O)CC2C1 C1(NC(COc2ccc(C)cc2C)=O)CC2CCC(C1)N2C(=O)C(C)S C1(NC(c2cnn(CC)n2)=O)CCCN(C(c2cocn2)=O)C1.C(C)(C)C.C c1(C(=O)NCCN(C)CCO)ccc(Cl)cc1.C1CCN1CCn1cnnn1 N1(C(c2cc(C3CC3)cc(F)c2)=O)CC2CCN(C(=O)Cc3cc[nH]n3)C2C1 C1(NC(Cn2cc(CNC(c3c(C)n(C)cn3)=O)nn2)=O)CC(=O)NC(=O)C1 CC(C)C(C(=O)NCCC1CCCN(C(=O)CCc2ccccn2)C1)NC(N)=O C1(CNC(COCCCC)=O)C2CCC(C2)N1C(C1CCC(=O)NC1)=O CCC(CC(=O)NOCCCO)NC(=O)CC1(O)CCOC1 N1(C(c2[nH]cc(C)c2)=O)CCN(C(=O)C=Cc2cn(C)cn2)C2CCC12 c1(CNC(Cc2cc(C)no2)=O)ccc(CNC(=O)C(c2cncn2C)O)cc1 N1(C(c2c(CNC(CCC=C(C)C)=O)cc[nH]2)=O)CCN(C(=O)CO)CC1 Cc1nccnc1C(=O)NCC(C)(C)OCC(=O)NC1CCC1O c1(C(=O)NC(C2CCCCC2)CNC(C2CCC2)=O)c(O)cc(F)cc1F.C C1(CCNC(c2ccco2)=O)CCN(C(C2(C(F)F)CC2)=O)C1.C1CCC1 C1(NC(CCOCC#C)=O)CCC(CCNC(=O)C(F)(F)c2cncs2)C1 c1(CC)cnoc1C(=O)NC(CNC(=O)CC1(O)CCC1)C1CCC1 N1(C(C(CCC)C)=O)CCC(NC(c2ccc(C)s2)=O)CC1C C(C)(CC(C)C)NC(C1C(C(=O)OC)C1)=O.c1(CC=O)cc(C)no1.N Cn1cnc2[nH]c(C(N3CC(O)(CNC(=O)C4=NNC(=O)C4)C3)=O)cc12 C1(CC(=O)NCC#CC(F)(F)F)(NC(=O)C=CCN2CCC2)CCCCC1 N1(C(c2ncnc(OC)c2F)=O)CC2CCN(C(=O)CCc3cnccn3)CC12 c1(CC)nc(C)c(CC(=O)N(CC(C)NC(c2nccc(Cl)c2O)=O)C)c(C)n1 N1(C(c2cc(CC)no2)C(=O)NCCC#N)CCC(C(N)=O)CC1 CC(C)C1=CCC(NC(C2(F)CN(C(=O)C3=CCSC3)C2)=O)CC1 N1(C(c2c(C)coc2C)=O)CCC(NC(C2C3CCCCCCC23)=O)C12CCC2 N1(C(C(CCC)c2ccccc2)=O)CCCCC(N(C(=O)C2=C(C)OCC2)C)C1 c1(C(N2CC(Cn3cc(-c4cnsc4)nn3)C2)=O)c(Cl)ccc2cccnc12 C1(C)CCCCC1(C)C.N1(C(COCC(=O)OC)=O)CCC(C(C)(C)C=O)C1 C(=O)(C(C(C)O)NC(c1ccnc(O)c1)=O)N(CCC(=O)OC)C N1(Cc2n(CC)cnn2)CCC(N=c2[nH]c(Cl)ncc2C(N)=O)C(C)C1 C1(NC(C(C)NC(=O)NC)=O)CC(C)(NC(=O)C(C)CN(C)C)C1 C1(NC(CC(CC)C2CCC2)=O)CC2CN(C(=O)CC(C)C(F)F)CC2C1 N1(C(=O)COC(F)(F)F)CCCN(C(C2(n3cc(C(=O)O)cn3)CC2)=O)CCC1 c1(CNC(C2C3CN(C(C4ON=C(CC)C4)=O)CC32)=O)c(C)cccc1F C1CN(C(c2ccc(C)c(Cl)c2)=O)C(C)(C)C1.c1(CC)nc(C(=O)N)c(N)s1 c1(NC(c2ccnc(CNCC3CC4C=CC3C4)c2)=O)cc2cccnc2[nH]1.C C(=O)(CC(F)(F)C(F)F)N1CC2C(N(C)C(c3c(Cl)csc3Cl)=O)C2C1 C1(NC(CCC2CCC(=O)N2)=O)CCCC12CN(C(C13CC1C3)=O)C2 C1(CC(=O)NCc2cccnn2)C2CN(C(=O)C=CC3CCOC3)CC12 c1(C(N2CCC(C)N(C(C3CCCS3)=O)CC2)=O)ccc2oc(O)nc2c1 C1(C2(NC(COC(CC)CC)=O)CC2)CCN(C(=O)CCc2csc(C)n2)C1 CC1(C)CC(NC(c2cccnn2)=O)CN(C(C2CC(CF)C2)=O)C1 CCC(CCC(=O)NCC1CN(C(c2ccc(OC)nc2Cl)=O)CCO1)OC C1(C(=O)NCC2CCC3(CC3)CO2)CCC(O)CN1C(=O)C(F)=CC1CC1 n1(CCC(=O)NC)nc(C2CC2(C)C)nc1Cc1ccc(N(C)C)s1 Cc1nc(N2CCC3(CCCCC3NC(C3CC3(F)F)=O)C2)c2scc(C)c2n1 c1(OC)ccccc1C(=O)N.C(C)(C=O)N(CCC)C1CC1.CC.C(C)C c1(CC(N2CCC(C)(CC)C2)=O)ccc(F)cc1F.Cc1[nH][nH]c(=N)c1C(=O)N N1(C(C2CN(CC)C(=O)C2)=O)CC(C(=O)NC2CCOC2)C(F)C1 N1(C(C(C)C(F)F)=O)CCCC(O)(CNC(C2(n3cnnn3)CCCCC2)=O)C1 C1CC2COCC2N1C(=O)C(C)C.C(CC(=O)N)NC(C)=O.[SH](C)(=O)=O.C C1(NC(c2c(C)nc(C)[nH]2)=O)CCCN(C(c2sc(C#N)cc2Cl)=O)C1C c1(CC(N2CCC(O)(CC)C2)=O)ccc2ccccc2c1.C(=O)(C1=C(Cl)CCC1)N c1(-n2c(C3CCC(C)O3)nc(CCCSCC)n2)cc(F)c(Br)cc1C N1(C(C2(OC(C)C)CCOC2)=O)CC2(C1)CN(C(=O)C(O)C(F)F)CCO2 C1(CC)CN(C(=O)C(Br)=C(C)C)CCC1NC(C1CC2(CCOC2)C1)=O C12(OC)CC(C1)N(CC(=O)NCC(=O)NC1CCCCC1)C2 c1(OC)cc2ccccc2cc1C(=O)N(CCCNC(C1(C#N)CC1C)=O)C C1(C(N(CC(C(=O)OC)C)C)=O)CCN(C(=O)CCCC2CCC2)C1C c1(C(=O)NC2CC3CN(C(C4C(OC)C4)=O)CC3C2)cn2cc[nH]c(=O)c2n1 c1(NC(C2N(C(CCCOCCC)=O)CC(O)C2)=O)ccc(C)c(O)c1C C(C)(C)(C(=O)NOC1CCC1)C1CCCN(C(c2nc(C)oc2)=O)C1 C1(C)(C(=O)NCC2CCCN(C(C=C(C)C(C)(C)C)=O)C2)CCCNC1=O CC(C(=O)N=c1ccn(-c2ccc(Cl)cc2C#N)[nH]1)n1cnnn1 C1(NC(c2ccoc2)=O)CC2CC1CN(C(C13CCCCC1C3(F)F)=O)C2 C(C(C)(O)CC(=O)N1CC(C)C2(CC2)C1)OC.c1(C=O)ncsc1C(C)C.N C(=O)(CN=[N+]=[N-])NCC(CSc1ccccc1)OCC C1(NC(C2CC2(F)Cl)=O)CC2(C1)CN(C(c1ccc(C3CC3)cn1)=O)C2 CCCCS(=O)(=O)CC(=O)NC(CO)C(C)NC(c1cn2cc(C)ccc2n1)=O c1(CC(C)C)cc(C(=O)NC2CC(NC(=O)C(C)(O)C(C)C)C2)cc(O)n1 C(=O)(CCCCCCC(=O)N1CCCN(C(C2(C)CCC(=O)N2)=O)CC1C)OC Cc1nc(C)c(C(N2CCCC2CNC(c2c[nH]nn2)=O)=O)[nH]1.c1cccs1.C N1(C(c2cn(CC(C)C)nc2)=O)C2CCC1CN(C(c1cnn[nH]1)=O)CC2 C1(NC(=O)CCc2ccccc2Br)CCS(=O)(=O)C1 C(=O)(C(C)c1cc[nH]n1)NCC(C1CCC1)NC(C=CC=CCC)=O N1(C(c2cccc(N)c2C(F)F)=O)CCCC(C2CC2NC(c2cnc[nH]2)=O)C1 N1(C(Cc2cc(C)on2)=O)CCC(CNC(=O)CCC2CC2)C(C)C1 C1(CC=C)(NC(=O)C(C)(C)C2CCCO2)CCN(C(=O)CN2CCC2)C1 N1(C(C(CO)N(C)C)=O)CC2CC(NC(c3cncc(C(F)(F)F)n3)=O)C1C2 N1(C(C(CCC)C)=O)CCC(C)(C)C1CNC(C1(C(F)(F)F)CCCC1)=O C1(C(=O)NCCC2(O)CN(C(C3CCCNS3(=O)=O)=O)C2)Cc2cccnc2C1 N1(C(C(C(C)C)=O)=O)CCC(C(N2CC3CC(F)CC3C2)=O)C(C)(C)C1 c1(C(N(C2CCN(CCOC(C)(C)C)C2)CCC)=O)cc(O)cc(=O)o1 Nc1ccc(C(=O)NCC2CCCCC2)c(F)c1.c1(C=O)n[nH]cc1C1CC1.N C1(C(=O)NC23CC2CN(C(=O)COc2ccccc2)C3)C2CCC(F)(F)C12 N1(C(c2ccc(-n3cncn3)c(F)c2)C(=O)NCC2CC2)CCN2CCC1CC2 c1(C(N2CC(O)(CNC(C(=Cc3cnc[nH]3)C)=O)C2)=O)c(C)cccc1O C1(C(=O)NCCCOCC(C)C)(NC(C2CCC(=O)O2)=O)CC1(C)C C1(CC(=O)N(CC(C)C(F)(F)F)C)CCCCN(C(=O)COc2ccsc2)C1 N1(C(c2ccc(Cl)c(C)c2O)=O)CCCC(C2(NC(c3cnns3)=O)CC2)C1 C(C1=CCCN(C(C2CC3(CCC3)CO2)=O)C1)NC(CC1N(C)CCCC1)=O N1(C(C(C)CC2CCC2)=O)C(CNC(=O)CCSc2ccccc2)CC2CC12 N1(C(CC(C=C)C)=O)CCC(NC(=O)C(C)(C)OC(C)C)C1(C)C N1(C(C(C(C)(C)C)OC)=O)CC2CCC1CN2C(=O)CCC1CCCO1 C1(NC(CC2N(C)CCC2)=O)CCC2(CC1)CC(C(=O)NCC(C)(C)C)C2 C1(C(=O)NC2CN(C(C3(C)CCNC(=O)C3)=O)CC2F)CCC2(CCC2)CC1 N1(C(C(CSC)(C)C)=O)CC2(CC(NC(c3ncccc3C3CC3)=O)CO2)C1 C12(NC(C(CCSC)O)=O)CCOCC1CN(C(c1cc[nH]c3nccc1-3)=O)C2 Cn1nc(Br)c2c(NC(=O)Cc3ccc(F)c(F)c3F)cccc12 C1(NC(c2cc(C)ns2)=O)CN(C(=O)C2=C(Cl)CCC(C)C2)Cc2nccn2C1 Cc1scc(C(=O)NC2(C)CC(NC(C3CC3C)=O)C2)c1C.c1ccccc1 CCCC(CCC)C(=O)N1CCC(OCCNC(c2cnsn2)=O)C1 C1(O)(CCNC(Cc2cn(C)nc2)=O)CCCN(C(c2ccsc2Cl)=O)C1 Cc1cc(C(=O)NCC2(C(=O)N(C)CCOCCO)CC2)n[nH]1 CCC(C#N)C(=O)Nc1ccc(C2CCN(Cc3ccccc3)CC2)cn1 Cn1nc(C(=O)NC2CC3C(NC(=O)CC4CC(C)(C)CO4)C3C2)cc1.C c1(C(N(CCNC(C2(C)CC=CCO2)=O)CC)=O)cc(F)c(Br)cc1N C1(NC(c2cc(OC)ncc2)=O)CN(C(=O)CCn2nc(C)cc2C)CC1C#N C(CCCCCC(=O)N1CCN(C(=O)Cc2cnns2)CC1CCO)SC CCC(CN(C)C)CC(=O)NC1CC(F)(F)CC1.c1(CC=O)cccc(F)c1.N C(=O)(C(F)(F)C(O)C1CC1)NCCCCN(CCCNC(CC=C)=O)C CCS(=O)(=O)c1ccccc1C(C(=O)N)NC(=O)OC(C)(C)C.C1COC1 CC(c1ccsc1)=CC(=O)NC(C)(CNC(c1nocc1C)=O)C1CC1 c1(N2CCC(N(C)CC)C2)ccc(S(=O)(=O)N(C)Cc2ccccc2F)cc1Cl N#Cc1ccc(=NCC2CC(CNC(=O)CC3CCOCC3)CO2)[nH]n1 N1(C(=O)C=CI)CCCC2(CCN(C(c3occc3Br)=O)CC2)C1 C1(NC(C(CCF)NC(=O)CC2NC(=O)NC2=O)=O)CC2CC1C(O)C2O C(=O)(C(F)CC(C)(C)NC(=O)CCC(C)=O)NC1CCC(OC)CC1 N1(C(c2n(C=C)ncc2)=O)CC(C)C(NC(=O)CCCc2cccnc2)C(C)C1 Cc1ccc(C(N2CCC(O)(CNC(c3cc(C4CCC4)[nH]n3)=O)C2)=O)cc1F N1(C(C2(C)CC2)=O)CCC(NC(C2CCCN2C=O)=O)C(CO)CC1 C1(CC(=O)NCC2(C(N3CC(C(CC)CC)C3)=O)CC2)CCC(C)CO1 CN1CCC(C(=O)NC2(C)CN(C(c3ncn(C(C)(C)C)n3)=O)C2)C1=O N1(C(C2C(CCC)CCC2)=O)CC2(CCCCN(C(=O)CS(N)(=O)=O)C2)C1 C1(CC)CCCN(C(c2ccc(N)c(N)n2)=O)C1.C1(C=O)CCCS(=O)(=O)C1.N c1(CNC(=O)CCc2ccc(C(N(C(C)(C)C)C)=O)s2)cccc(Cl)c1 c1(C(=O)NCC(N2CCC(OC)CC2)=O)cnn2c1OCC2 N1(C(C(C(CC)CC)F)=O)CCC2(C1)CN(C(=O)CCC1(C)CC1(F)F)CCO2 N1(C(C2C(C)(C)CC2)C(=O)NCC2CC2)CCC(CC2CC2)C(F)(F)CC1 n1(C(C)(C)C)nccc1S(=O)(=O)NC1CCN(c2cnccc2C(=O)O)C1 C1(O)CN(C(c2cccn2C2CC2)=O)C1.C(=O)(C(C)(C)c1cccs1)NC.C c1(CC(=O)NCC2CCN(C(C3CCCC(O)C3)=O)CC2)ncn2c1CCC2 N1(C(COC(CC)C)=O)CC2CCC1CN2C(c1ccc(CC(C)(C)C)cc1)=O C12CC(CO1)C2.C1(CC=O)CCCOCC1.CC(C(=O)N)OCC1CC1.C C1(O)(CNC(CC2(NC(CC3CCC(=O)C3)=O)CCC2)=O)CCCOC1 CC(C(=O)NCCC1(O)CCCN(C(c2c(N)cccc2F)=O)C1)C(C)(F)F CC1CN(C(c2cn(C)cn2)=O)CC1CNC(c1cscc1-c1ccccc1)=O N1(C(C2N(C(=O)OC(C)(C)C)CCC2)C(=O)NCCF)CCCC1C#N.CCC#N CC(C)C(F)C(=O)N(C1CN(C=O)C1)C1CC1(F)F.C(C)(C)C.CC=O.N c1(C(=O)OC)ccc2c(c1)CN(C(=O)C(=O)NCc1ccc(N)c(I)c1)CC2 C1(CC(=O)NCC=CCNC(CC=C)=O)CC(OC)C1(C)C C(=O)(C(CO)NC(C1CCCN1C(N)=O)=O)NC(C)CCN1CCCC1 c1(C(N2C(CN(C(C(C)SCC)=O)CC)CCCC2)=O)cn2ccnc2cn1 CCC(O)C(F)(F)C(=O)NC1CC(CNC(c2cc(F)cc(N)c2N)=O)C1 c1(CCC(=O)NCC(C2CCCCC2)OCC)ccc(N2CCOCC2)cc1 Cc1ccc(CC(=O)NCCO)c(Cl)c1.c1(C(N(CC)C)=O)cc(C#N)ccn1 C1(NC(=O)CC2CCOC2)CCCCC1C(=O)NCC1CCCCC1 C1(C(=O)NCc2nc(C)c(C)s2)CCCCCC1NC(=O)CC1CCOC1 CC1CC(NC(=O)CCC(C)(C)C)CN(C(C2(N3CCOCC3)CCC2)=O)C1 C1(NC(CC(C)C)=O)CN(C(=O)COC2CCCC(C)C2)CCC12CCC2 CC1CC(NC(=O)CN2CCS(=O)CC2)CN(C(=O)CCC2CCOCC2)C1 Cc1c(C(C)NC(N2CCC(C(F)(F)F)(OC(C)C)C2)=O)cccc1F C1(CNC(CC(CC)SC)=O)CCN(C(=O)CN2CCC(C)(C)C2)C12CC2 c1(CC)ccc(O)c(NC(C2CCCCC2C)=O)c1.C(=O)(CC1CCC1)N N1(C(c2c(N)n(CCO)nc2)=O)CC2CN(C(C34CCC3CC4)=O)CC2C1 C(=O)(CCC(C)(C)C(=O)N1CCCC(C)C1)OC.C1(C(=O)N)CCOC1C1CC1 N1(C(CCC=CC)=O)CC=CC(C(=O)NCC2CCN(CC)C2)C1 C1(OC)CC(CNC(C2(SC)CN(C(c3nc[nH]n3)=O)C2)=O)C1(C)C C(=O)C(C)(C)C1CCOC1.c1(CC(=O)N(CCOC)CC)ncc(C)s1.N Cc1ccc(CCC(=O)NCC(C)C(=O)N2CCC2C(C)C)o1 C1(NC(COCCC)=O)CCC(CC(=O)NOC2CCCCC2)C1 c1(OCC)nccc(C(N2CCCCC2CCN(C)C(C2CCN2C)=O)=O)c1F C1(NC(C=C(C)C(F)F)=O)CN(C(C2(C(F)(F)F)CCC2)=O)CC1C c1(C(N2CCCC(NC(=O)C(F)C3CC3)CC2)=O)cc2ccccc2nc1O c1(COc2ccc(C(N3CC4(CCOC4)C3)=O)cc2)cc(F)cc(F)c1 C1(NC2C(c3ccc(OC)nc3)C2)CC2(CCN(C(=O)C(O)C3CCCC3)C2)C1 c1(CCC=C)ccc(C(=O)NC(C)C(C)NC(c2ccc(O)cn2)=O)cc1 CC1CN(C(=O)C(C(C)O)NC(=O)C2CC2)CC1.C(=O)CC.CCN(C)C c1(C(N2CC(Cn3cc(C4CCC4)nn3)C2)=O)ccc(-c2ccccn2)s1 c1(OC)cccc(N(C(=O)C=C(Br)Br)C)c1C N1(C(C(C)OCC)=O)CCN(C(c2c(C)ncn(C)c2=O)=O)CC12CCC2 c1(C(=O)NC2CC(NC(C3C(CCOC)C3)=O)C2)cc(CC(C)C)c[nH]1 CCCC(CC1CCCC1)C(=O)NCC(C(C)(C)C)NC(=O)Cc1cnc(C)o1 N1(C(CCC(=O)OC)=O)CCC(C)C(NC(c2occc2C2CC2)=O)C1 CC(C(=O)NCC(C1CCN(C(=O)Cc2ccc(O)cn2)CC1)C)C(F)F C(=O)(CC(O)CNC(=O)CCCC1CC1)OC.C1(C(C(=O)N)O)CCCCC1 c1(CC(=O)NC2CC3C2CCN3C(=O)CC2(O)CCC2)nc([N+](=O)[O-])n[nH]1 CC1CCN(C(c2coc(Cl)c2)=O)CCN1C(=O)CC1CC2(CCC2)CO1 c1(NC(CN(CC(F)(F)F)C)(C)CO)ccc(Cl)nc1 N1(C(CNC(CC)=O)=O)CCCCC1CCNC(c1ncn(CC)n1)=O C(=O)(CC=C(Cl)Cl)NCC1CC(NC(C2C(C(C)=O)C2(C)C)=O)C1 N1(C(C2C(=O)NCC2)=O)CCC(C2CCN(C(c3ccc(CO)nc3)=O)C2)CC1 C1(NC(c2cc(CC)[nH]n2)=O)CN(C(=O)C(CO)NC(N)=O)CC12CC2 Cc1sc(O)nc1C=O.c1(CC(=O)N(CC)C2CC2)scnc1-c1cccs1 C(=O)(NN1CCCC1C(N1CCCCCC1CO)=O)c1ccc(C#C)cc1 N1(C(CSCC)=O)CCN(C(C2CN(C3CCC3)C2)=O)CC12CC2 CC1(C)CCCC1(C)NC(C1(CCNC(C2CNC(=O)C2)=O)CCC1)=O Nc1cccc(C(=O)NC2CCCCC2CNC(=O)C(F)n2cccn2)c1F c1(OC)ncccc1C(=O)NCCC1COCCN1C(c1cc(Cl)ccn1)=O C(=O)CCCCc1cnn[nH]1.C1(NC(=O)CC2CN(CC(F)(F)F)C2)COCC1.N C1(CCC=C)CCCN(C(c2coc(CNC(=O)CN3CCOCC3)c2)=O)C1 N1(C(C(C)C2CCCO2)=O)CCC2(C1)CN(C(c1coc3c1CCCC3)=O)C2 c1(C(N2CCC(N(C(C=CCN)=O)C)C2)=O)n[nH]c(C)c1C(C)=O.CC C12(CN(Cc3ccc(C)cc3)Cc3scnc3C)CC=CC(C1)OC2 c1(C(N2C(CNC(C3CCCS(=O)(=O)C3)=O)CCCC2)=O)cn2cnnc2cn1 N1(C(c2c(C)[nH]cc2)=O)CCCC2C1CCCN2C(c1ccc(S(N)(=O)=O)s1)=O CC1(C)CC(C(=O)NC2(CCCNC(=O)C=Cc3ccoc3)CC2)C1 N1(C(C2N(C)CCOC2)=O)CCC(C)(C)C1CNC(C1(N(C)C)CC1)=O CC(C)(C(=O)NC)C(N)=O.C1CC2CC2N1C(c1cc(-c2cccnc2)no1)=O N1(C(c2[nH]c(=NC)sc2)=O)CCC(NC(C2CC2c2ccoc2C)=O)CC(O)C1 N1(C(C(CC)CC)=O)CCC(C)C(CNC(=O)C=Cc2ccnn2C)C1 c1(OC)ccc(C(=O)NCc2ccc(C(N3CCCCC3)=O)cc2)cc1.C1CC1 C(=O)(C(F)CC(C)(C)NC(=O)CCN=[N+]=[N-])N(c1ccccc1)C Cc1cc(C(=O)N(C2CCC(NC(=O)CC3CCCSC3)C2)C)cnc1C C(=O)(C(C)P(C)(C)=O)N1CCCC(CN(C(c2cc(OC)nn2C)=O)C)C1 c1(N)cc(C2CC2)ccc1C.C[IH](=O)CCN(CCO)C(=O)NCC c1(C(C(=O)OC)OC(=O)CCCCNC(c2ccccc2)=O)ccccc1I c1(C=O)cc(F)c(F)c(O)c1F.c1(CCC(=O)N(C)C)ccc(Cl)s1.C1CC1 CS(C)(=O)=NCC(=O)N1CC(NC(C2CC(=O)N2)=O)C1 C1(C(=O)NCCC2CCN(C(=O)C3=CCCOC3)C2)CCc2nnc(O)cc2C1 c1(C(=O)NC2CC2NC(c2cccc(F)c2O)=O)cc2cc(Cl)ccc2[nH]1 CC(CN(C)C)CCC(=O)NC1CCCC1CC(=O)N(C1CCSCC1)C Cc1ccc(C=CC(N2CC(C)N(C(=O)CN3CCSCC3)CC2C)=O)cc1Cl C1(C)(CNC(COCCC(C)C)=O)CN(C(C2C=CCC2)=O)CC1C c1(C(N(CCNC(C(C(C)C)SC)=O)C2CC2)=O)n[nH]c2ccc(C)cc12 c1(-c2c(-c3n(Cc4c(SC)nn(C)c4)ccn3)csc2)ccnc2[nH]ncc12 N1(C(C(C(C)C)C)=O)CCN(C(=O)Cc2cnc[nH]2)CC(O)C1 c1(NC2COC(C)(C)OC2)ccc(S(=O)(=O)N2CCCCCCCC2)c(Br)c1 c1(C(CC)(C)CNCc2nc(-c3ccccn3)no2)cccc(C)n1 C(=O)(C(O)CCC(C)C)NC(CC(=C)Cl)C(=O)NC1C2CCCC1CC2 C12(NC(CCC#C)=O)CCCC1CN(C(C1COC(=O)O1)=O)C2 Cc1cccc2cccc(CN3CC(Nc4ncc(I)cn4)C(C)C3)c12 CCCCCC(F)C(=O)N1CCC2CCCC12C(N1CC(O)C(F)C1)=O C12(CNC(=O)NC3CCN(C(=O)NCC)CC3)CCCC1C2(F)F c1(CC)ccc(C(N2CCCC(N(C)C(C3CC3(F)F)=O)CC2)=O)c(C)n1 N1(C(c2nn[nH]c2Cl)=O)CC2(CCN(C(C34CCC(CF)(C3)OC4)=O)C2)C1 CCCCC(C)CCC(=O)N1CCC(C(C)NC(=O)CC(O)CCCCC)CC1 C(=O)(C#CC1CCCO1)N1CCC(O)(CCNC(c2c(C)n(C3CC3)nc2)=O)C1 n1(CC(=O)NC(CN(C(=O)C(F)CC2CC2)CC)C)cc(F)ccc1=O n1(CC)nccc1C(C(=O)NC1CC1)N(CCC#N)C1CC1.c1cscn1.C N1(CC(=O)NC2CCC(NC(=O)COCC3CCC3)C2)CCOCC1 C#CC1(C(N2CCOCC2CCC)=O)CCN(C(c2sncc2C)=O)CC1 CC1(C)CC(C(N2CCC3(CCC3)C2)=O)CC(C)(C)C1.C(=O)(C(O)C1CCC1)N C1(CC(=O)NC(C)C(CO)NC(=O)CN2CCCC2=O)OCCCC1(C)C N1(C(C2C3(CCN(C(c4cc(C)cc(O)c4)=O)C3)C2)=O)Cc2cncnc2C1 C1(CN(c2ccnc(NCC(C)OC(C)(C)C)n2)C)CCn2ccnc2C1 c1(CNC(=O)NC2COCC2n2cccn2)cc(Cl)cnc1Cl Cc1ccc(Cl)c(C(=O)NC(C)CCC)c1.C(=O)C(CC1CC1)CC1CC1.N CC1CN(C(=O)NC2(c3cc(Br)ccc3F)CC2)CC(c2ccsc2)O1 N1(C(C2CCCSC2)C(=O)NCCC(=O)OCC)CCC2(CCOCC2)C1 C1(OC)(CN(C(=O)CCCn2cc(CC(C(=O)O)C3CC3)nn2)C)CCSC1 C(=O)(C1=NNC(=O)CC1)N1C(CCNC(c2cc(C)cc(F)c2)=O)CCC1 c1(C(=O)NC2(CNC(C(C)C3CCCC3)=O)CCCC2)cccc(C2CC2)c1Cl CC(C)(CO)CCc1cn(CCCNC(C2CCCOC2)=O)nn1 CCCCCC(O)C(=O)N1CCC(C(C)(C)CNC(=O)CC(C)SC)CC1 CC1(C)CC(C(=O)NC(CNC(C2(C#N)CC2)=O)CO)CCO1 C1(c2cn(C(C(=O)NCCCN(C(C)C)C)C)nn2)CC2(CCC2)C1 C1(NC(C2(C(C)(C)O)CCC2)=O)CCOCC1C(=O)NCC(Cl)Cl C1(C(N2CCC(O)(C3CC3)CC2)=O)CCN(C(=O)Cc2cn[nH]c2)O1 c1(CCNC(C2C(CCC)C2)=O)ccc(F)cc1F.c1(CC(=O)N)cc[nH]n1 CC1CCN(C(C2CCCC3CC23)=O)CC1CNC(=O)CCC(N)=O c1(C(N2CC3CCC2C(NC(C2(C(F)F)CC2)=O)C3)=O)ccc2c(c1)CCCO2 C1(C(=O)NCC(CC=C)NC(c2ccc(Br)o2)=O)CC2C=CCC(C1)C2 C1(C)(C(N(C)CC2(O)CN(C(c3c(OC)csc3)=O)C2)=O)CC=CCO1 N1(C(C(CC)C)=O)Cc2occ(C(=O)NC(C)Cc3cnc[nH]3)c2C1 C1(C(=O)N(C)OC)(CC#C)CCN(C(=O)Cc2n[nH]c(C)n2)C1 c1(OC)cccc(C)c1C(N1CC(NC(=O)Cc2nc(C)sc2C)C(F)C1)=O CC1CN(C(c2cn(C)nc2C(C)(C)C)=O)CCCN1C(c1nccnc1N)=O N1(C(CCSCC)=O)CCCC1C1CCN(C(=O)COc2ccccc2)C1 C1(C(N2C(C)(C(=O)OC)C2)=O)CN(C(=O)CCS(C)=O)CC1(C)C C1(CNC(CCSC)=O)CCN(C(C2CCCC(CF)C2)=O)C1C1CC1 N1(C(C2CCN(CC)C2)=O)CC2(CNC(c3ncc(C)cc3F)=O)CCC1CC2 Cc1cc(=NCc2ccc(F)cc2F)[nH]c(N2CCC=C(F)C2)n1 C1(C=O)C2C3CCC(C3)C12.C1(C(=O)NC)CC(C(F)(F)F)C1.C1CC1 C(C1CN(C(c2n[nH]cc2C)=O)Cc2ccccc21)NC(C(CCC)C)=O C(=O)(C(C)CN(C)C(C1CC(O)C1)=O)NCCSCC=C N1(C(C=CCCC)=O)CCC(C)(C)C1CNC(c1nccn1C)=O C(=O)(C(O)CCCNC(C1CC2CCC1CC2)=O)NC(C)C(O)C(F)F C(CC)(CCCC(=O)NC(CCC)C(F)(F)F)NC(CCCCC)=O N1(C(CC(CC)OC)=O)CCOC(C(=O)NCCc2cccs2)CC1 CC(CF)CC(=O)NCC(=O)NC1CCN(CC2CCCN2CC(F)(F)F)CC1 C1(N(C(c2cn(C)nn2)=O)CCO)CCN(CC2(c3ccc(F)cc3)CC2)CC1 N1(C(CCCOC)=O)CC(C)CN(C(=O)Cc2c(C)cc(OC)cc2C)C(C)C1 c1(NC(C2C(C(=O)NC3(C(=O)OC)CCCC3)C2)=O)cc(Cl)n(C)n1 C1(C(N2CC(OC)C2)=O)CN(C)C(=O)CCO1.c1(C=O)cc(=O)cc(Cl)[nH]1.C CC1C(NC(=O)CCc2cccnc2F)CCCN1C(=O)C(C)S(C)(=O)=O C1(CC(=O)NC(CC(C)C)C)CCN(C(=O)CCCOC(C)(C)C)C1(C)C N1(C(C(c2scc(C)n2)C)=O)CCCCC(N(C(=O)Cc2cscn2)C)C1 c1(C(=O)NCC23CCC2CN(C(C2CC=CCC2)=O)C3)c[nH]c2cccc(F)c12 C(=O)(C1=CCCCO1)NC(C(N1CC(C(CC)C)C1)=O)C1CCC1 C1(C(=O)Nc2cc(C)nn2C)CCCC12CCN(c1ccnc(N3CCCC3)n1)C2 N1(C(C(CNC(c2c(C)cn(C)c2)=O)C)=O)CCC(O)CC12CC2 C1(C(=O)NCC2CC(C)C2)(SCC)CCC1.C1(CC=O)CN(C)C1 c1(C(=O)N)ccc(C(C)(F)F)nc1C.c1(C(N(C(C)C)CC)=O)ccccn1 N(C1c2ccccc2CC1(C)C)CC(c1cc(C)n(CCc2cccs2)c1C)=O N1(C(C2ON=C(CC)C2)=O)CC2(C1)OC1(C)CC2(NC(C2CCCC2C)=O)C1 C1(C(=O)NCC2CC(C)SCC2)COc2cc(F)ccc2C1 Cc1nc(C(=O)NC2CC(CC)C2)c(C)n1C1CC1.c1(C(=O)N)ccnnc1 c1(CC)cc(F)ccc1COCC1CCCO1.C12(CC1)C(=O)OC2 C1(CC(=O)NCCC2(O)CN(C(CNC(N)=O)=O)C2)NC(=O)NC1=O N1(C(CS(CC)(=O)=O)=O)CC(NC(=O)Cc2nncn2C)C2CCCCC12 c1(C(=O)NC2C(C)(C)CN(C(C3CC4(C3)CC4F)=O)C2)ccc(Cl)c(N)c1Cl C1(CC=C)(C(=O)NCc2nn[nH]n2)CCN(C(c2ccc(OC)nc2)=O)C1 c1(C(N2CC(C)CC(NC(CCOCC)=O)C2)=O)cnc2ccnn2c1 N1(C(C(COC)NC(=O)C(O)C(C)(C)C)=O)CCC12CC(C)(CO)C2 c1(C(=O)NCC(CNC(c2n(CCCC)ncc2)=O)F)c(F)cc(O)cc1F N1(C(C2CCCN(C(C(C)=C(C)C)=O)C2)=O)CC2CC(N(C)C)CC1C2 Cc1ccc(C(=O)NC2(C)CC(NC(c3ccccc3)=O)C2)cc1.C(C)(C)C c1(C(=O)NC2CC(CNC(C3C(C#C)C3)=O)C2)cc2c(C)c(Cl)ccc2[nH]1 CC(C)CC(C)(O)C(=O)N1CC2(CCC(CNC(=O)CCCC3CCC3)O2)C1 C1(NC(c2c(C)cncc2)=O)CC2CC(C1)N(C(c1[nH]ccc1C1CC1)=O)C2 c1(C(N2CC(NC(CS(C)(=O)=O)=O)C3(C2)CCC3)=O)noc2ccc(Cl)cc12 N1(C(c2cccc(SC)n2)=O)CC(CNC(c2cnns2)=O)C2(CCOCC2)C1 CCC(F)(CNC(C1CC2CC2N1C(c1cn(C(C)C)nn1)=O)=O)CC N1(C(CNC(=O)CC2CCCC2)=O)CCC2(C1)CN(C(C1COC(=O)N1)=O)C2 C(=O)(C(C)(C)CC(=O)NC1(C)CCN(C(=O)C(CSC)OC)C1)OCC Cn1c(C(F)(F)C(=O)NCc2ccc([N+](=O)[O-])cc2F)nc2ccccc12 c1(C(CC)C)ccc(C(=O)NCCNC(=O)C(C)CSC)c(O)n1 CC1(C(=O)NCCNC(=O)COC2CCCCC2)CCC(=O)N1 c1(OC)ccc(C(=O)N(CC(O)CNC(C23CCC(CC2)C3)=O)C)cc1 c1(C(=O)NCC(CNC(C2CCC(CC)O2)=O)C)c[nH]c2cccc(C#N)c12 c1(CC)ccc(C(N2CC(OC)CC2CNC(c2n[nH]c(C)n2)=O)=O)cc1F N1(C(c2ccc(C(C)C)cc2)=O)CC2CCCC2(Nc2ncnc(=N)[nH]2)C1 CCC(CC(=O)N1CC2CN(C(c3nnn(C)c3N)=O)CC2C1)CC(F)(F)F N1(C(CCC2C(C)(C)C2)=O)CC(NC(=O)C2=CSCS2)CC2(CCC2)C1 c1(CC(=O)NC2CN(C(CC3(OC)CCC3)=O)CC2C)ccc2[nH]ccc2c1 C1(NC(C=CC)=O)CN(c2ncnc3c2ncn3C)CC12CCOCC2 c1(OC)cc2c(cc1-c1n(CCN3CC4CCC3CC4)ccn1)OC(C)C2 C1(NC(Cc2cc(C)sc2)=O)CCC2CN(C(c3ccoc3Cl)=O)CCC2C1 Cc1cc(S(C)(=O)=O)ccc1C(N1CC(F)CC1C(=O)NCC(F)F)=O C(=O)(C1CCc2c[nH]nc21)NCC(CC(C)C)NC(c1ncc(C(F)F)s1)=O C(=O)(C1=CCN(C(C2(CSC)CC2)=O)CC1)NCC1CCN(CC)C1 C1CS(=O)(=O)C12CCN(C(=O)CCSC(F)(F)F)CC2.C1(C(=O)N)C=CCC1 N1(C(COCCC(C)C)=O)C2CCC1CC(CC)C2.C(=O)CC1(C(F)F)CC1 c1(C(N2CCC(CCC(=O)N(CC)CC3CCCO3)C2)=O)ncc(F)cc1F C1(C(N2CC(CC)(OC)C2)=O)CCN(C(C2CC(C)=NO2)=O)CC1O c1(CC)ccc(C(c2ccccc2)CNC(c2nnn(C)c2C)CC)cc1 c1(C(=O)OC2CC3(C(C(=O)OC)C3)C2)ccc2cccc([N+](=O)[O-])c2n1 C(=O)(C(O)C1CCC1)NCCN(CCC)C(C1(C)CCC1)=O C1(NC(=O)CNS(=O)(=O)C2CC2)COC2(C1)CN(C(=O)CO)C2 c1(C(C)NC(c2n(CCOC)nnn2)CCC2CCC2)ccc2ccccc2c1 C1(CC(=O)NC2C3CN(C(C(CCC)O)=O)C2C3)CC2CCC(C1)N2C n1(CC(=O)NCCOCCNC(=O)Cc2cccs2)cnc(Br)n1 Cc1ccc(Cc2nc(-c3ncnc(C(C)C)c3F)no2)c(C)c1 C=C(Cl)CC(C(=O)N1CCC(NC(=O)CC)C1)NC(=O)CCCCSC N1(CC)CCN(C(c2sncc2C)C(=O)Nc2cccc(OC)c2)CC1 c1(C(=O)NC2C(NC(C(C)NS(CC)(=O)=O)=O)CCC2)cc(C)[nH]c1C Cn1c(-c2cn(CC3CCCN3C(C3CCC(F)C3)=O)nn2)nc2ccccc12 N1(C(CN(C2CCCCC2)C(C)=O)=O)CC2(CCCN(C(C3(C)CC3F)=O)C2)C1 Cc1ccc(O)cc1CCCC(N1CC2CC1CN2C(=O)COCCN(C)C)=O CC1(CNC(C2CCCCN2N=O)=O)CN(C(=O)COCCN(C)C)CCO1 C1(NC(c2ccon2)=O)CC2(C1)CN(C(C1CCC(=O)N(C3CC3)C1)=O)C2 C=CC(C)(O)CC(=O)NC1CCN(C(c2cnnn2-c2ccccc2CC)=O)C1 c1(CN(CC(=O)NC)C2CC2)ccc(NC(c2ccccc2)=O)nc1 N1(C(CCOCC(C)C)=O)CCC(NC(C2CCNC(=O)C2)=O)C1C c1(C(=O)NC(C2CN(C(c3n(C=C)ncc3)=O)C2)C)cc(Cl)ncc1Cl N1(C(C(c2cccc(Cl)c2)C)=O)CCC2(CC1)CN(C(C1CCCN1N=O)=O)C2 N1(C(CCC)C)CC(C(N2CC(Nc3nccc(C(C)=O)n3)C(O)C2)=O)CC1=O N1(C(CCC(=O)N(C)C)=O)CCCC2C1CCN2C(=O)CC1(C)CCCO1 c1(C(=O)OC)ccc(C(=O)NC2(C)CCC2)c(O)n1.c1(C(=O)N)ccco1 N1(C(=O)COc2ccccc2Cl)CCC(O)(c2cn(-c3ccccc3)nn2)CC1 N1(C(C(CC)C#N)=O)CCC(F)(F)C(CNC(=O)C=C(C)c2ccsc2)C1 CCC(Cc1ccc(N)cc1)C(=O)N(CCNC(=O)CN(C)C)CC C(=O)(CC(C)C(F)(F)F)N1C(C(N2CCCC(C#C)C2)=O)C=CC1 C12(NC(CCCC(=C)C)=O)CCCCC1N(C(c1cnc(Cl)cc1N)=O)CC2 CC(O)(C(=O)N1CCC(C(=O)NCC2(N3CCOC3=O)CC2)C1)C(F)(F)F C=CCC(CNC(=O)CNC(C1CC1C)=O)C(=O)NCc1ncccc1Cl c1(C(=O)NC(c2ccccc2)CNC(C(N)=O)=O)ccc(F)cc1C(F)F n1(C2CN(C(c3c(OC)c(C)sc3)=O)C2)cnc(C(=O)OC)cc1=O N1(C(C2C(C)OCCC2)=O)CCCCC(CNC(c2cc(Cl)cn2C)=O)C1 c1(C(=O)NCC(C2CCC2)NC(CNC(CC)=O)=O)csnc1Br Cc1nnc2n1CC(C(=O)NC1CCN(C(=O)CC(C)c3ccco3)C1(C)C)C2 c1(C(N(CCC)CCNC(C2(C)C=CCC2)=O)=O)cccc2ncn(C)c12 c1(OC)cc(Br)c(CN2CCCC2(C)C(=O)Nc2ccccn2)cc1OC C1(C(=O)NCCCOCCNC(C(CC#C)C)=O)CCCC(C(N)=O)CC1 N1(C(C(C)N(C(=O)C(C)CC)CC)=O)CCC(C(C)NC(CC)=O)CC1 Cn1nnc(C=CC(=O)NCCNC(C2CC23CC(O)C3)=O)n1 C=C=CCC(=O)NC(CN(C(=O)C(CC)=Cc1cn[nH]c1)C)CC c1(C(N(CCCC)C)=O)cncc(S(N)(=O)=O)c1.C1(C=O)CCCN1C(N)=O CCCCCCCCC(=O)N1CCC(CCNC(=O)CC(O)C(C)C)C(F)(F)C1 Cn1c(C(=O)NCC2CCN(C(c3cc(C#N)n(C)n3)=O)C2)cc2sccc12 C1(NC(c2cnc(Cl)s2)=O)CCOCC1C(=O)NCc1ccncn1 N1(CCNC(C(C)CC2CCCC2)=O)CCCN(C(=O)CN2CCCC2)CC1 N1(C(CC=C(C)C)=O)CCCC2CN(C(c3cc(CC(C)C)on3)=O)CCCC12 c1(C(=O)NC2CC(C)(CNC(CCC=C)=O)C2)cncc(C(F)(F)F)c1.O N1(C(C(C)N(CCCC=O)CC)=O)Cc2ccccc2C1.C(C)(C)C.C=O.N CCCCCCCCCC(O)C(=O)Nc1ccc(SC(F)(F)F)c(OC)c1 N1(Cc2ccc(COC)o2)C(C(N2CCC3(C2)CC3(F)F)=O)CC2CCCCC12 C(=O)(N1CC(C)(O)CO1)C12CCN(C(C(CC)=CC)=O)CC1C2 N1(C(c2c(C)nc(=N)[nH]c2)=O)C2CCC1C(C)C(NC(=O)COCCO)C2 Cc1cc(C(N2CC3CC2(C)C3)=O)n(C2CCC2)n1.C1(C)(C(=O)N)C=CCC1 C1(NC(Cc2cc(C)on2)=O)CCC(NC(c2sc(F)cc2Br)=O)CC1 C1(C(=O)N)CCc2ncnn2C1.c1(OC)ccc(CCNC(=O)C(C)(C)F)cc1 N1(C(C2CC(NC(CC3(CCCC)CC3)=O)C2)=O)CCCC1CCC C1(NC(C2CCC3CC3CC2)=O)CCCCC12CCN(C(C1CC1F)=O)C2 N1(C(c2cc(C)cc(C)n2)=O)CCCC2(NC(=O)COC3(C)CCCC3)CC2C1 C1(C(=O)OCC(C2CCC2)OC)CCn2nnnc2C1 C1CN(C(C2(O)CC2(C)C)=O)C1.c1ccco1.C(=O)C.C(C)(OC)OC c1(C(=O)NCC(C)CN(C(=O)CN2CC=CC2)C)n[nH]c2c1CC(C)(C)C2 c1(C(=O)NC2CCC(CC(=O)NC(C(C)O)(C)C)CC2)ccccc1C#N C1(C(=O)NCCC(C(C)C)NC(CNC(CC)=O)=O)CCc2ccnn2C1 C(=O)(CS(=O)(=O)CCO)NC(CNC(c1cc(N)c(Cl)cc1)=O)CO CCC(C)CC(C)CONC(c1ccsc1I)=O N1(C(C2C(c3ccn(C)c3)C2)=O)CC(OC)C(NC(C2(C)CCCS2)=O)C1 C1(C(=O)NC2C(C)CCC2)Cc2nccnc2CN1C(=O)C(C)CN CC(C)C(CO)C(=O)N1CCCC(C)(CNC(=O)C(C)(C)C2CCC2)C1 c1(C(=O)NCC=C)ccc(C(=O)N)cc1.CCC(C)N(C(=O)C=CCF)C C(C)(CO)(C(=O)N1CC(C(C)CC)C1)NC(CCC#C)=O C(=O)CCC(C)(C)N(C)C.C(=O)(C#CC(=O)N1CCCC1C(C)(C)C)N(C)C.N OC1CN(Cc2ccccc2)CCC1Nc1ncnc(Cl)c1Br c1(OC)cnc(C(=O)N)nc1.C12CC(C(F)(F)F)(C1)C2.C1(C=O)CCCO1 CC(C)CC(O)CC(=O)N1CCCCCC(NC(C2(C#N)CCOCC2)=O)C1 c1(OC)cccc(C(=O)NC2CC(C)(NC(=O)COC3CCCCC3)C2)c1 c1(NC(N(C)Cc2cnc(-c3ccccc3)[nH]2)=O)nc(F)c(F)cc1F CC(CC(=O)N1CCCC1C(C)NC(C1(n2cncn2)CC1)=O)c1ccccc1 c1(C(=O)NC2CC(CCNC(c3c(C)ccnn3)=O)C2)c(N)ccc(Br)c1F N1(C(c2c(CC)nc(C)nc2)=O)CC2COCC(C1)C2NC(C1CCCC1C)=O N1(C(Cn2c(C)cnc2)=O)CCC(NC(=O)C(C)c2cccs2)C12CCC2 [nH]1nnc(C)c1C=O.c1(C(N(CCC)C(C)C)=O)ccc(C(N)=O)cn1.C c1(N2C(CN(C(Cc3cccc(C)c3)=O)C)CCC2)ncnc2c1cnn2C C1(C)(NC(CC(C)C2CC2)=O)CCN(C(c2nocc2Cl)=O)C1 c1(CC(=O)NC(c2ccccc2)C(=O)N2CC(n3cccn3)C2)cccc(Cl)c1 Cc1ccc(C(C(C)(C)C)N(C)CC2COC2)cc1 N1(c2nccc(C(=O)OC)n2)C2CC1CN(Cc1cc(C)ccc1OC(F)F)C2 S(=O)(=O)(c1ccc(Br)cc1NCCOC1CCC1)NCCc1ncn(C)c1Br N1(C2C(C)(C)CC2)CCC(NC(=O)C(C2CCOCC2)N)CC1 C1(C(=O)NC(C)(C)C(F)(F)F)CCCN1NC(=O)CCn1cccc1 c1(C(=O)NC(CC(C)NC(c2ccc(C(C)=O)cc2)=O)C)cc(C)nc(C)n1 c1(C(=O)NCC(C2CCOC2)NC(Cn2ccc(C)c2)=O)ccnc2c1CCC2 C(=O)C1=C(Cl)CCCC1.Cc1nc(C2CC2)sc1C(=O)NCC1CCCCC1.N CN1C(=O)CCC1C(N1CCOCC1CC(=O)NCCc1ccnc(O)c1)=O CCC(C)(CNC(c1ccc(OC)nc1)=O)C(=O)N1CCC(CSC)C1 N1(C(c2n(C)cnc2I)C(=O)NCC2CCCO2)CCCC(F)(CO)C1 C1(C(=O)O)(CC)CCN(CCCCCCCF)CC1 c1(C(C)C)ccc2c(c1)C(NC(=O)NC(C)(C)CF)CCO2 N1(C(C=CC)=O)CCC12CCCN(C(c1cccc(OC(C)=O)c1C)=O)C2 C(C)(CO)(C(F)F)N(C(C(CNC(C)=O)c1ccccc1)=O)c1cccs1 N1(CC)CC(NC(=O)C(CNC(c2coc(O)n2)=O)N(C)C)CC1=O.C C=CC(CC)CC(=O)N1CCCC1CN(C(=O)CC(=O)NC)C C(=O)(CC(CC)C(C)(C)C)NC1CCN(C(c2cnc(CC)nc2O)=O)C1 CC(CN(C(=O)CCCC1CCCC1)C)C(=O)NCCCN1CCC1 N1CCCN(C(c2cn(C)nc2)C(=O)Nc2ccc(F)cc2)CC1.CC(O)CO N1(C(c2[nH]cc(C)c2)=O)CC2CN(C(c3cc(Br)c(C)o3)=O)CC2C1CO c1(N(C)CC2CCC(O)C2)ccnc(N2CCC(N3CC(F)(F)C3)CC2)n1 C(=O)(C1=NOC(C)C1)NCC(C)=CC(N1CCOCC1C(F)F)=O N1(C(C(CC)NC(C)=O)=O)CCCC2(C1)CN(Cc1ccncc1F)CCO2 c1(CNCC2(O)CCC(C)CC2)ccccc1S(=O)(=O)N1CCNC(=O)C1 Cc1cc(CC(=O)NC2CC(NC(C3CC4C=CC3C4)=O)CC2O)ccc1F C(=O)(C#CC1CCCCC1)N(CC(C)O)CCNC(C1(C)CC=CCO1)=O CC1CC(C(N2CCC(C)(C)C2C(=O)N(C)Cc2cccnn2)=O)CC(C)C1 C1(N(C(=O)C)C)COCCN(C(=O)C(C2CC2)CC)C1.C(C)(C)C.C=O Cc1nc(-c2nc[nH]n2)sc1C(=O)NCC1(C)CC1.C1(C(=O)N)CCCO1 C1(C2CCOCC2)(C(=O)NC(CNC(COCC#C)=O)(C)CC)CC1(F)F C(=O)(CCCC(=O)NC(C1CCOC1)CNC(c1n[nH]cc1Br)=O)OC c1(N(C)C)cccc(N2CCN(C(c3c[nH]cc3-c3ccccc3)=O)CC2)c1 C1(C(=O)NC(C(C)C)C(=O)N(C2CCCC(O)C2)C)CC2(CCC2O)C1 C1(c2nnnn2C(C)(C)C)(NC2(CC=C)CC=CC2)COC2(COC2)C1 C1(OC)CC(C)N(C(C2C(CN=[N+]=[N-])C2(C)C)=O)C1.c1(C=O)nnn(C)c1C C1(C(=O)OCCCn2nccn2)Cc2cc(F)ccc2C(=O)O1 C1(N(C(=O)Cc2ccc(C(N)=O)s2)C)CCN(C(C2CC23CC3(F)F)=O)CC1 C=C(C)CCCC(=O)N(C)CC1CCCN(C(=O)C(C)SC(F)(F)F)C1 c1(C(=O)NCC2(NC(C3C(OC)CC3)=O)CCC2)sc(C)nc1Br S(=O)(=O)(c1cccnc1N1CCCC(O)C1)NC(c1cc(F)ccc1F)CCC C1(CC)(CNC(C2(CNC(c3conc3C)=O)CCCCC2)=O)CCCCO1 c1(N(C2(C(=O)N)CC2)C)nc(O)c2c(ncn2C)n1.c1ccccc1.C1CC1.C n1(CC(=O)NCCNC(Cc2c(C)n[nH]c2C)=O)ncc(=O)c2ccccc12 C(CC)(C(=O)N1CC(NC(c2csnc2Br)=O)C1)=CCCC N1(CC)CCOCC1CC(=O)NCC1CC(O)CN1C(=O)CCc1nc[nH]n1 CC(C)(N=[N+]=[N-])C(=O)NC1CCC1NC(=O)C1=C(Cl)CCC1 c1(C(N(CCCNC(=O)C=C2CCOCC2)C2CC2)=O)c[nH]cc(Cl)c1=O CC(C)(C(=O)NC1CC(C)(NC(C2CC(F)(CO)C2)=O)C1)c1cscn1 CCC(CC(C)C)C(=O)NCCC(C)(C)CNC(=O)C(C(C)C)SC c1(C(=O)NC2C(CNC(C(C)CF)=O)C2)ccc(Cl)c(N2CCCC2)n1 N1(C(c2occ(C)c2C)=O)CC2(CCCN(C(c3cncc(F)c3Cl)=O)C2)C1 C1(C(=O)NCC(C)CNC(C2(C#N)CC=CC2)=O)CN2CCC1CC2 N1(C(c2c(CCC)nco2)=O)CCC(N=[N+]=[N-])(C(=O)NCC(C)OC(F)F)C1 c1(C(N(C2CN(C(c3c(CC)nns3)=O)CC2O)C)=O)c[nH]c2nc(Cl)ccc12 c1(C(N2CCN(C(C3CCCC(C(N)=O)CC3)=O)CC2)=O)ccc2c[nH]nc2c1 C(=O)(C(F)(F)CCS)OCCOCc1c(C)n(C)nc1.c1cc(N)cc(F)c1 CON=C(C(=O)NCC1CCN(C(=O)CC2CC(C)OC2C)CC1)c1ccco1 C1(COCC)CCCN(C(=O)CCC2CC(NC(=O)C(=O)NOC)C2)C1 C1(C)(C(N(CCC(C)O)C)=O)CN(C(=O)CC2CCCCO2)CC1C C1(C(=O)NCC=C)CN(C(c2cc(C)nc(C)n2)=O)CC(C)O1 C#CCCCCC(=O)N1CCCC(N(C(=O)CCc2cc[nH]n2)CCF)C1 N1(C(C(=O)N(C)C)=O)CCCC2(C1)CN(c1nc(C3CC3)ns1)CCO2 Cc1nsc(C)c1NC(C1(CCNC(=O)C=C2CCC2)CCCC1)=O c1(C(=O)OC)ccc(C(=O)NCC)s1.C1(C=O)CC1C(N)=O.CC.O CON(Cc1ccc(C)o1)C(=O)CSC1CN(C(C2(C#N)CCC2)=O)C1 CCC(C(=O)NC1(CNC(=O)CC)CCOC1)NC(C)=O.C(C)(=O)O Cc1cnc(C(=O)NCCC2CCCN(C(C3C4CCC34)=O)C2)nc1 CC1CN(C(=O)CC2(COC(F)(F)F)CC2)CCN1C(C1CCC(C)C1)=O C1(CCNC(C(COC)O)=O)CSCCN1C(=O)CC(O)C1CCCC1 C1(N(C(C(CC)n2ccnc2)=O)CC(C)C)CCN(C(=O)Cc2ccco2)CC1 C#CCC(C(=O)N(C)C(C)C1CC1)NC(=O)CN1CCNC(=O)C1 CC1CN(c2ccc(C(F)(F)F)cc2)CC(C)N(S(=O)(=O)c2cccnc2)C1 C1(C2CC2)C(=O)N(C)CC(=O)N1.C1(CC)CC1CC(=O)NC(C)(C)C c1(OC)ccc(C(N2CCCCC2CCNC(C2CC2C2CC2)=O)=O)cc1F c1(C(=O)NC(CCC)CO)ccc(=O)n(CC(=O)NC(C)C)c1 N1(C(c2ncn(CC)c2)=O)CC(NC(=O)C(C)(Cl)Cl)C(C)(C)C1 C(N=c1nc(O)c2c(ncn2C)[nH]1)C1C(NC(C(CCCC)C)=O)CCC1 Cc1nc(C(=O)NCC(C2CCCC2)NC(=O)C(C)n2ccnn2)cs1 C(=O)(CCC(C(C)C)NC(C1CCCCC(=O)N1)=O)NCc1cc(C)no1 N1(C(c2c(OC)csc2)=O)CCOC(CC(=O)Nc2cncc(SC)c2)C1 c1(C(=O)NC(C(C)NC(CN(C(C)=O)C)=O)CO)cc2c(C)cccc2[nH]1 Cc1c(Cl)ccnc1C(=O)NC1CN(C(=O)CCc2sccc2Br)C1 c1(-c2ccc(N3CCN(C(=O)CCc4ncc[nH]4)CC3)nc2)cccnc1Cl c1(OC)ccc(C)cc1C(=O)NC1CN(C(C2C3CCC2CC3)=O)CC1F N1(C(C)=O)CC(NC(c2nc(C)c(C)nc2C)=O)CC12CCC2 C(C(CNC(c1ccc(SC(F)(F)F)cc1F)=O)C(F)(F)F)NC(COC)=O N1(C(c2c(CC)nc(=N)[nH]c2)=O)CC(C)CN(C(=O)C(O)C2CCC2)CC1C CC(C)C(CN(C)C)C(=O)NCC(O)CN(C(=O)C(c1cccc(F)c1)F)C CC(=O)CCN=C(NCC(C)C)N1CCN(Cc2ccc3c(c2)CCO3)CC1 c1(C(=O)NC2CN(C(c3c(CC)c(C)sc3)=O)CC2O)cc2n(n1)CCO2 C1(C(N(CCCCN(C(=O)CC2CCCO2)C)C)=O)CCC2(CCC2)O1 c1(C(N2CC(CC(N3CCC4CC34C)=O)(OC)C2)=O)ncc2ccccn12 N1(C(c2ccn(CC)n2)=O)CC(NC(=O)CO)CC12CCOC2.CCN(C)C N1(C(c2c(C)[nH]cc2)=O)CCC(CNC(=O)CN2CCCNC2=O)C12CC2 C=C(CNC(=O)C(C)CF)CCNC(=O)C=C(C)Cl N1(C(=O)CCc2cccc(F)c2)CC2CCCN(C(=O)C#CC3CCOC3)C2C1 c1(COC)cc(C(=O)N)n(C)c1.C1(CC)CCCN1C(=O)C.c1nccn1C C1(NC(C2CC(OCC)C2)=O)CCC(C(=O)N(CC(F)F)C)CC1 C=Cn1nncc1C(=O)NCC1CC(NC(=O)Cn2ccc(C)n2)C1(C)C c1(C(=O)NCCCCC(C)NC(c2c(C)coc2)=O)ccc(Br)cc1C#N C12(C(=O)Nc3cc(C(C)C)no3)CCN(C(c3ccnc(O)c3)=O)CC1C2 C1(c2c(C(=O)OC)cn(C)n2)CN(S(=O)(=O)N2CC3CCC2C3)C1 n1(CCCC)cc(CN2CCCC2CN2CCSCC2)c(C)n1 C12(C(=O)NCC(CC)NC(c3ncn(C)c3C)=O)CCCC1(C(N)=O)C2 C1(NC(CC2C(C)(C)CCO2)=O)CCC(O)CN(C(=O)CC(F)(F)Cl)C1 C1(CNC(c2cncc(CC)c2)=O)CC2CCC1N(C(C1CC(OC)C1)=O)C2 c1(C(C2CC2)NC(CN(C)CC)=O)cc(C=O)no1.c1(C(C)O)ccncc1 c1cccc[n+]1[O-].C1(OC)CC(C(=O)NCCC2(NC(=O)CS)CCC2)C1 N1(C(c2c(NCC)cccn2)=O)CC2CC(NC(=O)C3=COCCO3)C1C2 Cc1cnc2c(C(=O)N(C)CCN(C)C(c3cc(C)c(Cl)cc3F)=O)cnn2c1 c1(CC)nc(C)ccc1NC(=O)CCCNC(=O)C(C)=C1CCCC1 N1(C(c2ccc(CS(=O)(=O)Cc3ccsc3)cc2Cl)=O)CCCC(C2CCC2)CC1 CCC(C)C(O)CC(=O)N(C)CC=CC(N1CCC(OCCF)C1)=O N1(C(Cn2c(C(F)(F)F)cc(C)n2)=O)CCOC2CS(=O)(=O)CC12 C1(c2n(C(C)(C)C)nnn2)(NCCCC2CCC2)CCN2CCCC2C1 c1(N2CC=C(CCNC(C(CCC)OC)=O)CC2)nc2ccc(F)cc2o1 N1(CCn2cc(C(CCC)=O)nn2)Cc2cnc(C(=O)OC)nc2C1 C(N=c1[nH]c(=NCCNS(C)(=O)=O)[nH]c2c1CSC2)c1cc(C)c(C2CC2)cc1 c1(C(=O)NCC2C(CNC(c3cocn3)=O)C2)cnoc1-c1cccs1 Cc1cc(F)ccc1CC(N1CC(CC(C)NC(C23CCC(CC2)O3)=O)C1)=O N1(C(C=C=C(C)C)=O)CC(C)N(C(=O)CN2CCCCC2C)CC1C C(=O)(C1=CC2CCCCCC12)N(C(CNC(c1cn(CC)nc1C)=O)C)C Cc1cc(C)c(NC(=O)C(Cc2ccco2)NC(=O)C(CO)N(C)C)cc1O N(C1CCCc2ccoc21)C(C(CCOC)NC(C1C=CC1C(=O)OC)=O)=O c1(C(=O)NC2CCN(C(CC=C=C)=O)C(C)C2)cc2cc(OC)ccc2n1C N1(C(c2c(OCC)scc2)=O)CCCC1(C)C.c1(C=O)cn(C2CC2)cn1.N S(=O)(=O)(c1cc(C(N2CCCC(C)(NC(=O)CC(C)F)C2)=O)co1)NC C1(C(=O)NCC(CC)NC(=O)CCC(C)OC)CCC(=O)N1C C(=O)(C(C)(C)CS(C)(=O)=O)N.C1(C(N2CC(OC)CC2)=O)CN2CCCN1CC2 C1(C(N2CC3CC3(C(=O)OCC)C2)C(=O)NCC)C2CCC(F)(F)C12 C1(CNC(C2(C)CNC(=O)C2)=O)CCC2(CCN(C(=O)C3=CCCS3)CC2)CO1 C1(C(C)C(=O)NCCc2cscn2)CCN(C(C2(n3cccn3)CC2)=O)C1 N1(C(C(COC(C)=O)C)=O)CCCC1(C)CCC(=O)NCc1nnc(O)n1C C(C(=O)N(C)OCc1ccccc1)(C1(C)CC1)NC(C1CCN(CC)C1)=O O(P(C)(=O)CNC(=O)CCNC(C1CCO1)=O)CC c1(C(=O)NCCC(C)Nc2nccc(OCCC)n2)cnc2n1CCCC2C N1(C(c2cnn(CCC)c2C)=O)CCC(NC(c2nnc(O)nc2O)=O)C(C)C1 c1(OC)nc(C(=O)NCC(C)(C)C(O)C2CCC2)ncc1F C=CC(C)(O)CC(=O)NC1(CCCC(N2CCC(C)(C)C2)=O)CCC1 N1(C(CC#N)=O)CC=CC1CNC(c1ccsc1I)=O C(=O)(CCCC(F)F)N1CCC(NC(CC2C(=O)NC(=N)S2)=O)C1 C12(NC(=O)C(C3CCCCC3)=O)CCN(C(c3ccc(Cl)o3)=O)CC1C2 Cc1cccc(F)c1CC(=O)NC1CN(C(c2ccc(O)c(Cl)n2)=O)CCC1C c1(CCC(N2CCCC(C(N3CCCCC3C(=O)O)=O)CC2)=O)cc(F)ccc1Br C1(NC(C(C)NC(C)=O)=O)CC2(C1)CN(C(=O)Cc1ccnnc1O)C2 Cc1nc(C)n(CC(=O)NC2CCC(C(=O)NC(C)C=O)C2)n1.C(N)=O.N C1(NC(C2CC2C2CC2)=O)CN(C(=O)Cc2ccc(Cl)cc2)C2(CCOCC2)C1 C(=O)(C(C)C(F)(F)F)NCC(CC=C)NC(c1cc(C)sn1)=O C#Cc1ccc(F)cc1C(=O)N.C12(C(N3CC(O)(CC)C3)=O)COC(CCO1)C2 c1(OC)cc(C(N2CC(NC(C3(CS)CCC3)=O)C(F)(F)C2)=O)ccc1C c1(C(=O)NC(C2(O)CN(C(C(C)(C)SC)=O)C2)C)cc(C)c(F)c(C)c1 C(C#Cc1ccccc1)N1CCCC(NC(C2CCC(C)(C)O2)=O)C1 c1(N2CCC(NCCOC)CC2)nnc(C2CC2)cc1C(F)(F)F Cc1cc(C(=O)NCC=CC(=O)NCC(C)(C)C(C)(C)C)c[nH]c1=N N1(C(C2(SC)CC2)=O)CCC(C2CCCN(C(C34COCC(C3)C4)=O)C2)C1 C(=O)(CCC(=O)N)NCCC.C1(C(N)=O)CN(C(C2(O)CCSC2)=O)C1.C C(N=c1cc(Cl)nc[nH]1)C1C(NC(c2ncnc3ccsc23)=O)CCC1 C1(CNC(C(c2ccccc2)NC(C2CC(=C)C2)=O)=O)COCC1(C)C OCC(CN=c1[nH]c(=NCc2cnn[nH]2)[nH]c2c1CSC2)c1ccc(F)cc1 C1(CNC(Cc2c(C)cc(F)cc2)=O)CC2CCCC(C1)N2C(=O)C=CCO c1(OC)ccc(-c2cnn(CC(N3CC[Si](C)(C)C3)=O)c2)cc1 O(NC(=O)CCN(CCCO)C(C1CC(n2cnnc2)C1)=O)CCOC c1(NCCc2ccc(NC(CC)=O)cc2)cc(Br)c(C)cc1S(N)(=O)=O Cn1ncc(C(=O)NC2CCC(CCNC(=O)C(F)(F)CC3CC3)C2)c1Cl CC1CCOC(C(=O)NCCC2CCN(C(C3(n4ccnc4)CCCC3)=O)C2)C1 c1(C(N2CCN(C(C3=C(C)OCC3)=O)CC2C)=O)ccc(C)c2c1CCC2 c1(C2CN(C(=O)OC(C)(C)C)C2)n[nH]c(=Nc2cnn(C)c2C2CC2)o1 C1(CNC(C(F)=CC)=O)CN(C(C2CC(Cl)(Cl)C2)=O)CCC12CCC2 c1(CN(C(=O)C)C)ccccc1CNC(C1C2CCCCC12)=O.C(N)=O C1(C(=O)NCCC=C)COC2CN(C(c3c[nH]c(C)c3)=O)CC12 C(=O)(C1=C(C)N(C)c2ncnn2C1)N1CCC(OC)(CNC(=O)CCSC)C1 CCC(CC(=O)NC1CC(CCC(=O)N(C)Cc2ncc[nH]2)C1)CC(C)C [nH]1ccc2ccccc12.Cc1ccnc(N2CCCC(N3CCNCC3)C2)n1 N1(C(CC=CCCCCC)=O)CCC2CN(C(=O)COc3cc(C)on3)CC12 Cc1ccc(OCCC(=O)Nc2ccccc2CNCCC(C)C(C)C)c(C)c1 C(=O)(C(C)(F)C(=O)N(CC)CC)OCC.C1(C)(C=O)CCCS1(=O)=O C1(SC)CCCCC1N=c1[nH]c2c(c(=NCc3c(C)coc3C)[nH]1)COC2 c1(NC(=O)NCCNC(c2ccccc2)C)cc(N(C)C)n(C)n1 C(C(C(=O)N1CCC(N2CCC2)C1)NC(c1ccsc1C)=O)OCC c1(OC)ccc(F)c(Br)c1C(=O)N(CCCNC(C1OCC1(C)C)=O)C C(=O)(C(C)CC(C)(C)C)N1C(CNC(c2c(C)n(C)cn2)=O)CC(F)C1 c1(C(C(N2CCCC(N(C(=O)CCP(C)(C)=O)C)C2)=O)O)cccc([N+](=O)[O-])c1 N1(C(C=C(C)C(C)(C)C)=O)CC2CC1CC2C.C(=O)C(C)(C)c1cccnc1.N C1(N(C(C(=Cc2ccco2)C)=O)C)CN(C(c2ccccc2Br)=O)CC1(C)C C1(C(=O)NC(C2CCCC2)CC)CCN(C(C2CCC(C)(CC)O2)=O)CC1(C)C c1(C(NCC)=O)c2c(nn1C)CCSC2.C1(C=O)CC(=O)N(C)C(=O)N1.CC C1(CCNC(C(c2n(C)ncc2)NC(=O)C(F)F)=O)CCCC1(C)C C1(NC(c2c(CC)scn2)=O)CCN(C(=O)C(CC)CCOC)CC1C C1(C(=O)NCCN(C(=O)CO)CC)CCC(C(=O)OC)O1.C1CC1 C(N=c1[nH]c2cccc(OCC(F)(F)F)c2s1)C1(NC(C(CC)C)=O)COC1 Cc1cccc(S(=O)(=O)N2CC3CN(c4ncnc5c4ccn5C)CC23)c1 c1(CC)cc(C(=O)NC(COC(F)F)C2CC2)nn1CCO N1(C(C(CN(C)C)N(C)C)=O)CCN(CCNC(C2(C#N)CCCO2)=O)CC1 C1(CC(=O)NCCn2ccc(C(=O)NC(C)CCn3cncn3)c2)CCCOC1 C=C(C)CC(C)C(=O)NC1(c2ccccc2)CCN(C(=O)Cc2n[nH]c(C)n2)C1 Cc1ccsc1-c1cn(C2CCC(C(=O)NCCCCN(C)C(C)C)C2)nn1 C(=O)(C1CCCc2sccc21)NCCCC(CCC)NC(c1ccncc1O)=O C1(NC(C2(CC)CN(C(COCC)=O)C2)=O)CC(C)(C)OC1=O Cc1ncc(N)cc1C(=O)NCC(C)S(C)(=O)=O.C1(C(=O)N)CCN(C)CC1 C1(CC(=O)NC(CSCC)C(=O)N2CCSCC2)CCCCN1C Cc1ccc(CC(=O)NCC2(C(N)=O)CN(C(c3n[nH]cc3C)=O)C2)s1 N1(C(C2(C)CN(C(=O)Cc3ccccc3I)C2)=O)CCc2n[nH]cc2C1 c1(CNC(C(C)=C(C)C)=O)cn(C2CCN(C(=O)CC)C2)nn1.CC(N)=O C1(CC(C)F)CCN(C(c2cnc(Cc3ccccc3)s2)=O)CC1 CC1C(=O)N(CC(=O)NCC(O)C)C(=O)C1C.c1csc(=N)[nH]1.C(=O)(C)N c1(OC)cc(C(=O)OC(C)(C)C)ccc1CSC.C12CCC1C(=O)N2 Cc1ccc(C(=O)NC2C=CC(CC(=O)N(C3(CCO)CC3)C)C2)cn1 c1(C(=O)NC2CCN(C(C3(SC)CCC3)=O)CC2C)cc(Cl)cc(F)c1N c1(C(=O)NCC2CCN(C(c3cc(CC)nn3C)=O)CC2)cccc2c1OCC2 C12(CCC)CC(C(=O)NCC(C)CNC(C3CC3C(N)=O)=O)(C1)C2 C(C(=O)NCC)(C(C)C1CCC1)N(C1CC(O)C1)C.C1CCOC1 Cc1cccnc1C=CC(=O)NC1CC(O)CN(C(=O)C(C)C)C1.[SH](C)(=O)=O N1(C(Cc2c(C)ccs2)=O)CCN(C(c2ccsc2Cl)=O)C(CO)C1 N1(CCCOC)CC2(CN(C(c3ccc(C(C)C)cn3)=O)CCO2)C1 c1(C(N(CCCN(C(c2cc(C(C)=O)sc2)=O)C)C)=O)cnn2c1C(C)CCC2 N1(C(C2(N(C(C(C)SC)=O)C)CC2)=O)C2CCCC1CC2 Cc1ncccc1CNC1CCC(CNC(=O)CCc2cnn(C)c2)CC1 C12(NC(c3c(C)n(C4CCOC4)nn3)=O)COC(C1)CC2.c1(C(=O)N)cnsn1 N1(C(CCCCC)=O)CCCCC(CNC(c2ccc(O)nc2Cl)=O)C1 N1(C(CN(C(=O)CC(C)(C)OC)CC#C)=O)CCC(C#CC)CC1 c1(-c2c(C)cc(O)cc2)cnc2c(C(=O)Nc3cnn4ccccc34)cccn12 C(=O)(CCCC(F)(F)F)NCC1C(C(NOCC=C(C)C)=O)CCO1 C1(COCn2cc(CCCC)nn2)CCN(C(=O)CCc2nc(C)c(C)o2)CC1 c1(C(=O)NC2C(NC(COCCOC)=O)C2)c(N)cncc1Br N1(C(c2ccco2)=O)CC2CC1CN2C(=O)CC(O)CN(C)C.N(CC)CC c1(C(=O)NC23C(CN(C(CC4N(CC)CCC4)=O)C2)C3)ccc(=O)n(CCF)n1 C12(C(N(C3CCCC3)CC)=O)COC(C1)C2.C1(C(C=O)O)CC(F)(F)C1.N c1(C(=O)NC2CC3(C2)CN(C(=O)CC2CCCOC2)C3)ccc2cccnn12 c1(OCC)c(C)cccc1C.c12ccc(cc1)-c1sccc1NC(=O)C(NC)C2 C1(CC)CN(C(=O)C(=O)c2ccco2)CCO1.C12CCN(CC1)C(=O)C2 C1(NC(C(SC)SC)=O)CN(C(=O)C(C)Cc2c(C)noc2C)CC1(C)C C1(C(=O)NCC=CC)CN(C(=O)C=Cc2cocn2)CCC1(C)C C1(C)(NC(C2C(OC)C2)=O)CCN(C(=O)C#CC(=O)N(C)C)C1 c1(-c2nc(C3CCOC3)no2)cn[nH]c1.C(=O)(COCC)NCC.C(=O)N c1(C(=O)NC2CCCN(C(=O)C)C2)c(O)cc(F)cc1F.c1(C=O)cccs1.N C1(NC(CCc2cn(C)nn2)=O)CCOCC1C(N1C(CO)CCC1CO)=O C(CC(C(=O)NCCN1CC2CC2C1)NC(=O)Cc1cccs1)OCC N1(C(C2N(C(C(OC)OC)=O)CC(F)(F)C2)=O)CCN(C)C2(CC2)C1 C=CC(C)(C)CC(=O)N1C2CCC1C(NC(c1ccnc(S)c1)=O)C2 C1(C)(C(=O)NC(C)CC(=O)NCc2nncs2)CCC2CC2C1 C=CC1(C(=O)NC2CCCC(O)C2)CCN(C(c2cccc(NC)n2)=O)C1 CC1CN(C(=O)CCOCCNC(C2(C)CCC3CC3C2)=O)C(C)CCO1 c1(C(=O)NCC(CC=C)NC(C2(C=C)CCC2)=O)ccc(OC)c2cn[nH]c12 CC1CCCc2c(C(N3CC4(CCCC4NC(=O)CO)C3)=O)cnn21 c1(C(=O)NCC(C(C)(C)C)NC(C23CC2COC3(C)C)=O)cccc(N)c1O N1(C(CNC(C)=O)=O)CCCC1C(C)(C)CNC(=O)CCCC1CCOCC1 c1(C(N(CCC(C(C)C)NC(CCCCC)=O)C)=O)n[nH]c2cc(C)ccc12 Cn1nc([N+](=O)[O-])cc1C(N1CCCC(CC)C1)=O.C(=O)(C(C)(O)C1CCC1)N C1(NC(C=C(COC)C)=O)CCN(C(=O)CCCO)C(C)C1.[SH](=O)(=O)CC.N Sc1ccc2c(c1)C(N=c1nc3sccc3c(NCC3CCOCC3C)[nH]1)CC2 N1(C(C)C)C2CCC1CNC2.c1(C2(N3CCOCC3)CC2)ccc(C2CCOC2)s1 c1(C(N(C(C(=O)NCC(C)CO)C)C2CC2)=O)nccc2cc[nH]c12 N1(C(c2c(C)cco2)=O)CCC(C)CC1CNC(C1(C(F)F)CCC1)=O C(=O)(C1CCCc2ncnn21)NCC(=O)Nc1ccccc1 c1cn(C)c2ccccc12.c1(OCCOC)ccccc1C=CC(=O)NCCO N1(CCNC(CN(C(c2nocc2C)=O)CC)=O)CCOCC1C [N-]=[N+]=NCCCCCNC(C1C2CCC(C2)C1)=O.C1(CC(=O)N)CCC(=O)CC1 Cc1nc(C(N2CC3CC3(NC(c3cnncc3O)=O)C2)=O)cc(O)n1 c1(C(=O)NC(CNC(C(C)(C)c2ccns2)=O)C2CC2)cccc2c1OCCC2 c1(N(C)C)ccc(C(=O)NC2CC(C(F)F)C2)nc1.C1(C=O)CNC(=O)N1.N c1(CC(=O)NCC2C3CN(C(CC(C=C)CC)=O)CC2C3)c(C)cc(C)cc1C Cc1ccsc1CC(=O)N(CCNC(=O)C(C)c1ccco1)C(C)C Cc1csc2c(C(=O)NC3(CO)CN(C(=O)CC4CC4C)C3)ncnc12 C(CC(C)C(=O)NC(C)(C)C(C)C)=CCC.C(C1CC1)(C1CC1)=CC=O Cc1oc(C)nc1C(N1CC(C(N)=O)C1)=O.c1(C(=O)N)coc(C(C)C)n1 N1(C(C2CC(=O)NC2)=O)CC2(CO)CC1(C(=O)NCC(O)CCO)C2 CC1(C#N)CCC(c2nnnn2Cc2ccco2)(NC(CF)CF)CC1 C(=O)(CCCn1cc(C(C)(C)OC)nn1)NCC=C=C C=C=CC(C)C(=O)N1CCC(C)C1CNC(c1cnc(C(C)C)o1)=O c1(N2CCC(N(CC(CC)=O)C)C2)[nH]c(=N)nc2c1cnn2C C(=O)(C(C)C(C)n1cccn1)NCCN(CCOC)C(c1nc[nH]n1)=O N1(C(c2c(COC)scc2)=O)CCOC(CCCNC(=O)C2=CCC2)C1 N1(C(CCC(=O)N(C(C)C)C)=O)CCN(C(C2C=CCCC2)=O)CC1CC(F)F C(=O)(C(CNC(=O)C(C)(C)CO)CC1CCCC1)N(C1CC2CCC1O2)C Cc1c(Cl)nc(NC(=O)CCC2CCCN2C(c2ccncc2)=O)nc1Cl N1(C(C2CC(C)OC2)=O)C2CCC1CN(C(=O)CCc1cccc(C(F)F)c1)C2 Cc1ccc(C2CC2CC(=O)N(CC(F)(F)CN(C)C)C)cc1 c1(OC)cnc(C)[nH]c1=NC(C)C1CCN(C(c2ccc([N+](=O)[O-])n2C)=O)C1 CCC(C)CCC(=O)N1CC(CNC(=O)C(O)c2cnc[nH]2)(OC)C1 CC1CCCC(NC(=O)C(C)(C)C2CCCN2C(c2ccn(C(F)F)n2)=O)C1C C12(NC(c3cnc(=N)[nH]c3)=O)CCOCC1CN(C(C1CC3(CSC3)C1)=O)C2 C12(CC(=O)N(CC)CC)CNC(=O)C(C1)C2.c1(C=O)cc(C)co1.CO C=C(C)C(CC(=O)N1CCC(C)C1c1cn(C2CCCC2)nn1)OCC CC(C)CC(CNC(=O)C(O)CC1CCCCC1)NC(=O)C(C1CCCCC1)O c1(C(=O)N)c(Br)cnn1C.n1(CCOC)ccc(C(=O)NCCC2CC2)n1 N1(C(C=Cc2ncc(C)[nH]2)=O)CC2CC(C)N(C(c3ccc(O)nn3)=O)C2C1 C1(CNC(C(C)CO)=O)CCCCN1C(=O)Cc1cnn(C)c1 C(CN=c1[nH]cncc1I)N(C(C(C(CC)O)C)=O)C N1(C(CN(C(COC)=O)C)=O)CC(C)CN(C(=O)C(c2nc(C)cs2)C)CC1C c1(CSC)cc(CN(C=O)Cc2ccccc2-c2cccs2)ccc1OC C1(n2cc(CN)nn2)CCCN(C(C2CCN(CCO)CC2)=O)C1 C1(C(C)C)CCN(C(=NCCCSc2ccc(F)cc2)NCc2ccnn2C)C1 c1(C(N2CCN(CCCNC(CC(C)CF)=O)CC2)=O)ccc2c(c1)CCC2=O CCC(CC)CC(=O)NCC1CCC1NC(=O)Cc1cncc(C)c1 C1(OCCNC(c2cc(C)on2)=O)CCN(C(=O)Cc2ccon2)CC1 c1(SC)cncc(NC(c2c(Cl)cnn2C)c2nnnn2CC2CCOC2)c1 C1(CN(C(=O)CCC2(C)CC2)C)CCCC(NC(=O)CC)C1.c1ccccc1 N(C(=NCCC1(C)CC1(F)Cl)NCCF)CC(N1CCN(C)CC1)C Cc1ccc(C(=O)NCC(C)NC(=O)CC2COC(C)(C)CO2)c2c1CCC2 C(=O)(C(CCC1CCCCC1)N(C)Cc1cccc(O)c1)NC(C)C C(=O)C1CCSc2ccccc21.CC(C)(C)C=CC(=O)NCC1(CC)CC1.N N1(C(CN2C(C)CCC2)=O)CC(C(=O)NC2(CCO)CCCC2)C(C)(C)C1 c1(C(C2CCC(C)C2)N(C2CCNCC2)CC(C)C)nc(-c2cccnc2)no1 N1(C(c2[nH]cc(CC)c2)=O)CCC(C)(C)C1C.C(=O)(CCCc1ccncc1)N c1(C(N(CC(C)CNC(=O)CNS(=O)(=O)N(C)C)C)=O)cc(O)ccc1F c1(C(=O)NCC(CCOC)NC(c2cccc[n+]2[O-])=O)cccc2nonc12 c1(C(=O)NC2(c3noc(-c4ccco4)n3)CCC2)ccc2[nH]nc(Br)c2c1 n1(CC)c(C)cc(C(=O)NC(C2CN(C(C3CCOCC3)=O)C2)C)c1C N1(C(C(C)(C)OCC)=O)CCN(C(c2csc(NC(C)=O)n2)=O)C(C)C1 CC(C)CCNC(=O)C(C)Cn1cccn1.c1(C(=O)N)ccnn1C1CCCC1 Cc1ccc(NC(=O)C(CN=[N+]=[N-])NC(=O)CCn2cccc2)c(O)n1 N(C1CCCn2nccc21)C(C(=O)N(CCCCCC)C)=O c1(C(=O)NCCC2CCN(C(=O)CC3=CCCC3)C2)n[nH]c2c1COCC2 c1(NC2CCCC(SC(C)(C)C)C2)ccc(P(C)(C)=O)cn1 c1(OC)c(C(=O)NC2CCN(C(=O)C3=CCCCO3)CC2C)occc1=O N1(C(C(C=C)OC)=O)CC2CC1CN2C(=O)COCc1nccs1 c1(C(=O)NC2C(NC(C(C)(C3CC3)OC)=O)CC2)cnc2n1CCCC2 c1(C(=O)NCC(C2CC2)(OC)OC)ccc(C=O)o1 C1(C)(CC)C=C(C(=O)N2CCCC(NC(=O)Cn3cnc(Br)c3)C2)C1 C(C1=CCCN(C(C2(C)CCCCCC2)=O)C1)NC(c1nnn(C)c1C(F)F)=O Cc1ccnnc1C(=O)N(C(C)C(=O)NCCC1CC1C1CC1)C N1(C(C(C)(C)C2CCC2)=O)CCC2(CCCCN(C(C3CCC(C)CC3)=O)C2)C1 N1(C(c2cccc(OCC#C)c2)=O)CC2CCC1CN2C(=O)CSC Cc1nc(C)n(O)c1C(N1CCCC(NC(c2cccc(Cl)c2O)=O)C1)=O c1(C(N2CC(F)CC(NC(c3cccc(C)n3)=O)C2)=O)ccnc2nc(C)nn12 C(N=c1[nH]c(N(C)Cc2cccc(Cl)n2)nc(=N)[nH]1)C1N(C)CCCC1 c1(N2CCC(N(C(=O)C=Cc3nccs3)C)C2)ncnc2c1CCCC2 C1(C(N(C(C(N2CC(C=C)(O)C2)=O)C)C)=O)CN2CCN1CC2 C1(C(=O)OCC)CN(C(=O)CCC(=O)NCC2(SC)CCCCC2)CC1(C)C C12(C(N3CCC(N(C)C(C4CCCC5(CC5)C4)=O)C3)=O)CC(C1)OC2(C)C.C C1(NC(C2(Br)C(C)(C)C2)=O)CN(C(=O)C(N)=O)CC2(CCC2)C1 C1(CC)CCCC1(C)C(=O)NC(C1CN(C(c2cnccc2OC)=O)C1)C c1(C(N(CCN(C(C)C)C(c2ccc[nH]2)=O)C)=O)cc2c(nc1N)CCC2 C1(C=O)(C(F)F)CCCO1.CC(C)(C)OC(=O)NCC(=O)N.C1CC1 C1(C2CCN(C(C3(C)CC=CCO3)=O)C2)(NC(c2cc(CCC)n(C)n2)=O)CC1 c1(CC)cc(NC(=O)C(=O)N(C2CCC2)CC2CC2)c(C)o1 C(=O)(C(=O)C(C)C)NCC(CC=C)NC(=O)CN(C1CCCC1)C N1(c2cc(C(=O)OC)ncn2)CC2(CN(C(=O)CC3CCCC3)CC2CO)C1 c1(C(=O)NCC(=C)CCNC(C2CCOCC2)=O)ccc(OC(C)C)nn1 C1(CC(=O)NCCN(C(=O)Cn2nc(C)oc2=O)CC)CCC(=O)N1C c1(CC(N2CC(CC=C)(NC(=O)CC(C)CF)C2)=O)c(C)nn(CC)c1C C12CCC(CC1)N(C(c1scnc1C1CC1)=O)C2.CC(C(=O)NC)c1ccsc1 C(c1ccc(F)cc1)=CC(N1C2CN(C(c3c(C)nc(Cl)s3)=O)CC21)=O C=CCCCCC(=O)NCC1CN(C(=O)C(c2cccnc2)O)CCCO1 c1(C(=O)NC(CN(C(C2N(C)CCOC2)=O)C)(CO)CO)cn(C)c(=O)nc1O CC(CS(C)=O)C(=O)NC1CC(C)(NC(c2cncc(Cl)c2)=O)C1 N1(CC2C(C(F)F)CC2)CCC2(CCCN(Cc3nccc(Cl)c3F)C2)C1 C1(CN(C(=O)Cc2ncoc2C)CC)CCCN(C(=O)C(C)CCN(C)C)C1 N1(C(c2nc(CC)sc2)=O)CC(F)(F)CC1.C1(CC=O)(N(C)C)CCCC1.C N1(C(C2C(OC)(OC)CC2)=O)CCC(CCC(=O)NCC2CNC(=O)O2)CC1 CCCC(CC(C)C)C(=O)N1CC2C(CNC(c3cc(O)ncn3)=O)C2C1 C=CCC(CC=C)C(=O)NC1CC2CCC1C(NC(c1cccc(F)c1)=O)C2 C1(C(N(CC)CC2CCCCC2)=O)CC(F)CN1C(=O)C(F)n1ccnc1 c1(N2CCC(CN(C)C)C2)nc(N2CCC(C)(C(=O)NO)CC2)nc2c1CSC2 c1(CC)ccccc1CC(=O)NCC(O)CNC(=O)CC(c1ccc(C)cc1)C c1(C(=O)NCC(CNC(CCOCCC)=O)O)ccc(F)cc1C#N C1(C2CN(C(=O)OC(C)(C)C)C2)NC(=O)CCC1.C1(C=O)CCCC(=O)C1.O C1(C(=O)NC(c2cccc(Br)c2)C)CCC2COC1O2 N1(C(C(=Cc2ccco2)C)=O)CCC(CCNC(C2SC3C=CC2C3)=O)CC1 C1(CCNC(=O)CCc2ccncn2)CN(C(=O)CSC(F)(F)F)CCO1 N1(C(C2CC(C)C2)=O)CCC(C(CO)NC(c2ncccc2F)=O)CC1 N1(C(c2ccc(C)cc2N)=O)CC2(CCCN(C(C3CCC3C(F)(F)F)=O)C2)C1 CS(=O)c1nc(NCC(CO)C2CCOC2)c(Br)c(Cl)n1 N1(C(C2ON=C(C)C2)=O)CC(C)OC2(CCN(C(=O)C(C)(F)F)CC2)C1 c1(C=O)nc(C)c(C)nc1C.n1(CC)nc(C(=O)NCCC)cc1C(F)(F)F C12(CNC(c3c(CC)scc3)=O)CC(CN1C(=O)C(C)c1ccco1)C2 N1(C(CCC(=O)OCC)=O)CC(C2(NC(=O)CC3CC=CCC3)CC2)C1 CC(c1ccccc1C)=CC(=O)NC1CCC1NC(=O)C(C)C#N C1(C)(NC(c2n(CC)nnn2)C(C)(C)N2CCOCC2)CC(C)(C)CC(C)(C)C1 C1(C(N(C(CC(=O)OC)C)C)=O)CCCN(C(C2CC2(C)C(F)F)=O)C1C N1(C(c2coc(C(C)(C)C)n2)C(=O)NC(CC)(C)C)CCCC(N(C)C)C1 C1(CC)CCC(C(=O)NC(C)(C)CCCNC(C2CC3(CSC3)C2)=O)CC1 N1(C(CCN(CCCCC)CC)=O)CCC(NC(c2cn(C)c(O)n2)=O)C12CC2 C1(C(=O)OC)CN(C(c2cccs2)C(=O)NC)CC(=O)N1.C1CC1.C1CC1 N1(C(C(C)OCCC(C)C)=O)CC2CC(NC(C34CCC(CC3)CC4)=O)CC1C2 CCC(F)C(=O)N(CCNC(C1CC1(C(C)C)CC)=O)C1CC1 c1(C(=O)NCC2N(C(C(C)c3cccs3)=O)CCOC2)cc(C(C)C)ccc1O c1(C(N2CCN(C(CNC(C3CCC(C)C3)=O)=O)CC2)=O)ccc2c[nH]nc2c1 c1(OC)ccc2[nH]c(=NCC(C)CO)[nH]c(=NC3CCCSCC3)c2c1 c1(OC)ccc(C(N)=O)cc1C(N1CCN(C(=O)Cc2cnsc2)C2CC12)=O C1(C(C)NC(C(=O)NCC2(CO)CC2)C2CC2C)CCc2nccn2C1 C1CC(C)CC(C)C1.c1(Cn2cc(CCC(=O)OC)nn2)ccc(C(=O)N)cc1 Cc1nc(NC(C)CCNC(=O)CCc2ccc(C3CC3C)o2)c(C)c(Cl)n1 S(=O)(=O)(C1CCN(C(=O)Cc2cccc(CC(=O)OC)c2)CC1)NC N1(C(c2cc(C)ns2)=O)CCCC2CN(C(C3Cc4cccnc4C3)=O)CCC12 C1(CNC(COC)=O)CN(C(=O)CCc2c(C)n[nH]c2C)CCN1C c1(C(=O)NC2CC(C)N(C(=O)CCc3cnco3)C2)ccc2c(c1)NC(=O)C2=O C1(NC(C2C=CCC2)=O)CCN(C(=O)CCC2CCC(O)CC2)CC1O c1(C(N2CCN(C(CSC)=O)CC(C)(F)C2)=O)cccc2c1oc(=O)n2C C(=O)(CCCCCNC(C1(CC=O)CC1)=O)OC.n1(CC)nc(O)ccc1=O.N c1(OCC=C)cccnc1C(=O)NC(C1CCN(C(c2cccnc2O)=O)C1)C C1(CCF)(NC(C(C)c2ncco2)=O)CCN(C(=O)CNC(N)=O)CC1 C1(C#N)(SC)CN(C(=O)CC2(C)CCN2C(=O)CSc2cn[nH]c2)C1 CC1(C)CCCN2C(=O)CONC(=O)C1CCN(C(C)(C)C)C2CC N1(C(C(CC(N)=O)O)=O)CCC2(CCCN(C(c3ncsc3C3CC3)=O)C2)CC1 C1(CC(=O)NC2CC2CNC(c2cnn(C3CCOC3)n2)=O)COCCO1 c1(C(=O)NC(CNC(c2c(CC)nccn2)=O)CO)ncsc1S(N)(=O)=O C12(C(=O)NC3CCN(C)CC3)CC(CN(C(C3CN(C(N)=O)C3)=O)C1)C2 c1(C(=O)NCCCNC(c2cccc(Cl)c2Cl)=O)cc2n(n1)CC(F)C2 c1(N2CCC(NC(c3sc(C)c(O)n3)=O)CC2C)ncc2ccsc2n1 c1(C(=O)NC2CCN(C(C(CC)C)=O)C2C)ccc(N)cc1S(N)(=O)=O c1(OC)cc(C(=O)NC2CN(C(C3CC3c3cccnc3)=O)CC2F)c(F)cn1 C1(C(=O)NC)(C(=O)NC(C)CNC(=O)C(C)SC)CCC1 Cn1cccc1C(=O)C(=O)NCC1(NC(c2ccc(Br)o2)=O)CCC1 N1(C(CC2C(C)CCCC2)=O)CC2(CC(NC(C3(n4cncn4)CC3)=O)C2)C1 c1(C(N2C(CNC(C3(CC=C)CC3)=O)C(C)CC2)=O)cc(O)cc(=O)o1 c1(NCC)ccc(Cl)cc1C(=O)NC.C1(F)(C(N2CCCC2)=O)CCOCC1 CC1CN(C(C2CCC(C)(C)CC2)=O)CC2(CCN(c3cc(=O)n(C)cn3)C2)O1 N1(C(C=CCN(C)CC)=O)CC2CCCCC2C1.C1(CC=O)CC2C=CC1C2.N C1(CC)CCC1.CC(C)(C)C(N)=O.CC=O.C1(C=O)CC1.C(=O)(O)N C1(NC(=O)C2=CCC2)CCCC12CCN(C(c1cc(C(F)F)nc(O)c1)=O)CC2 N1(C(N=c2[nH]nc(Cc3ccc(OC)cc3)s2)=O)CCC(O)C2CCCCC12 Cc1ccc(C(=O)NC(C(=O)Nc2ccc(C3CC3)nc2)C(C)C)nc1O N1(C(C(C)NC(C)=O)=O)CCC(NC(C2CCOC2)=O)C(C)C1 C1(OC)CCCN(C(C2(NC(c3cnn(C(C)C)n3)=O)CSC2)=O)CC1 c1(C(N2C3(CN(C(C(C)OC)=O)C3)CC2)=O)ccc(F)c(F)c1N C(N=c1nc(N2CCC(N(C)C)C(C)C2)c2sccc2[nH]1)c1cc(Br)cc(C)n1 C#CC1(CNC(=O)CCC(C)(C)NC(C2CC(=O)NC2(C)C)=O)CCOCC1 c1(C=O)cc(C)sc1N.CCS(=O)(=O)NCCNC(=O)C.C(=O)(C)N c1(C(N2C(CC(N3C4CCC3CC4)=O)CCC2)=O)n[nH]c2c1CCCC2 C(c1cnc(O)nc1O)=CC(N1CCC(NC(C2CC(=O)C2)=O)(CO)C1)=O c1(C(N(CCN(C(c2cn(C(C)C)nn2)=O)C)C)=O)cc2ncc(Br)cn2n1 C(=O)(C(CC)CCC)NC(CC=CC)C(=O)NCC1(C)CC(O)C1 C(C(C)(N)C(=O)N(CC(OC)OC)Cc1cccc(F)c1)OCC N1(c2ncc(OC(C)C)cn2)CCC(NC(=O)C=Cc2cc(OC)ns2)C(O)C1 C(=O)(C(C(C)(C)C)n1ccnn1)NC(CC=C)CNC(=O)C=C(C)CCC C=CC(CC)CC(=O)N1CCCC(OCc2cn(CCN(C)C)nn2)C1 C1(=O)CCOCCN1.CCCCC(C#C)NC(=O)CC.CCC.C(C)=O C1CC(C)(C)CN1C(c1nnn(C)n1)=O.n1(CC(C)C)nccc1C(=O)N.C [SH](=O)(=O)c1ccc2c(c1)CCC2.c1(C(=O)NC2COC2)cnc(Cl)c(Br)c1.C N1(C(c2cnc3n2CCC3)C(=O)NCSc2ccccc2)CC2CNS(=O)(=O)C2C1 c1(CC(C)C(=O)N2CCCC2CCNC(C2CCC2)=O)ccccc1Cl c1(OC)cc(F)c(F)cc1NNC(=O)CC1C2CNCC12 N1(C(C(c2ccc(N)cc2)O)=O)CCCCC(NC(C2CCC3CC3C2)=O)C1 c1(C(N2C(CN(C)C(C3CCNC3=O)=O)CC(F)C2)=O)cn2c(n1)COCC2 C1(C(N2C(C)CCC(NC(c3cncc(CO)c3)=O)C2)=O)CCC2(CCCC2)C1 c1(NCCCC)ccc(C(=O)NC2CC(NC(=O)CCCC)C2)cc1.C(C)=O C1(C(N(CCCCN(C(C(CC)COC)=O)C)C)=O)CCS(=O)(=O)C1(C)C C(=O)(C(=O)CC)N(C(C)C(=O)N1CC(OCCOC)C1)CCC C1(CC)CN(C(c2cnc(O)n2C)=O)CCN1C(c1cn[nH]c1)=O Cc1nccc(Cl)c1C(N1CC(CCNC(=O)CSc2cccs2)C1)=O C12(C(=O)N)CCCCC1C2Cl.c1(OC)ccc(-c2n[nH]cn2)cc1 C1(C(N2CCN(c3c(C)n[nH]c3C)CC2)CC)CC(C)CC(C)(C)C1 Cc1onc(CC(N2CCC(NC(C3CC(F)(CO)C3)=O)C(CO)C2)=O)c1C#N N1(CC)CCCC1C(=O)N(CC(C)(C)NC(c1ccncn1)=O)C n1(CCC#C)c(N(C2CCS(=O)(=O)C2)CCC)nnc1-c1ccc(OC)cn1 c1(C(C2CCNC2)OC)cnc2n1CCCC2Cn1cc(-c2ncccc2N)nn1 c1(N(C)Cc2cccc(C)n2)nccc(=NCC(=O)N(C)Cc2ccoc2C)[nH]1 c1(OC)ncc(C(=O)NCC2CCN(C(=O)CCNC(C)=O)CC2C)cc1C CC1(C)CC(C(=O)NC2(CNC(=O)C(C3(O)CCCC3)F)CC2)O1 C(CC1=CCN(C(c2cc(C3CC3)ns2)=O)CC1)NC(C1(C)CCC(=O)N1)=O Brc1ncccc1C(c1nnnn1C1CCCCC1)NCCC1CCCO1 C1(CC(=O)NCC2(O)CN(C(CC(=O)OC)=O)C2)CCCC1(F)F C(=O)(C(F)CC1CCCC1)NC(CCN(C(COCC)=O)C)C CC(CC(C)(C)CNC(=O)OC(C)(C)C)C(=O)OCCCCCCO Cc1c(C(=O)NC2(CF)CN(C(=O)CC3CC4CC4C3)C2)ccn1C N1(C(C(C)=C2CC2)=O)CCC2(CCC2)C(NC(=O)Cn2ccc(C)n2)C1 Cc1cc(C(=O)NC2CCN(C(=O)CCn3cccn3)C(C)C2)ncc1C(F)F c1(CC(=O)N(CC(=O)NCCCOCCCC)CC)cccc(F)c1 CC1(C)CN(C(=O)CS(N)(=O)=O)CCN(C(C2CC(OC(F)(F)F)C2)=O)C1 c1(NC2C(NC(C(CCC)C)=O)CS(=O)(=O)C2)nn2cc(C)nc2s1 C(c1ccc(C#N)cc1)=CC(=O)N.C1(C(=O)NC2CCCC2)(OC)CCOC1 c1ccc(F)c(OC(F)F)c1.C1(C(=O)NC(=O)N)CC(F)CN1CCF.CC n1(CC)nc(C)cc1C(=O)NC.C1CC(C)N(C(c2cn(CCF)nn2)=O)C1 c1(CNC(c2n(CCC(=O)OCC)nnn2)(C)COC)cncc(Cl)c1 CC1COC(C(N2CC(CO)(NC(=O)C(O)Cc3cnc[nH]3)C2)=O)C1 C1(NC(c2ccc(C)n2C)=O)(CNC(c2cc(C(F)F)on2)=O)CCCCC1C C1(C(=O)NCC2(C)CCN(C)C2)C2CCCC2CN1C(=O)CCCCN=[N+]=[N-] Cc1cnc(C)c(C(N2CCOC(C(C)NC(=O)CN(C)C)C2)=O)c1 CC1CC(CNC(c2cccnc2CO)=O)CN1C(c1cnncc1O)=O c1(OC)ccccc1CC(N1CC(C)C2CC12)=O.c1(C=O)c[nH]nc1C(C)C.N CS(=O)c1nc2ccc(NC(c3c(Cl)oc4ccccc34)=O)cc2[nH]1 N1(C(Cc2cc(C)n(C)n2)=O)CCC2C(C(=O)NC3CCOCC3(C)C)C2C1 Cc1ccn(CC(=O)NC(C)C=CC(=O)NCC(F)C2CCC2)c1 Cc1cc(F)ccc1CC(=O)NC1CCCC(NC(=O)CC2CC23CC3)C1 n1(CC(=O)OC(C)(C)C)cc(C(N2CCC2CF)=O)nn1 N1(C(C2(CC)CCCCO2)=O)CCC(CNC(=O)C(=O)N(C)C)C(F)(F)C1 C(=O)(C(C)CCCOC)N1CCC(OCC(N2CC(CCC#C)C2)=O)C1 N1(C(CC(CN(C)C)O)=O)CC2OCC(NCC3C4CCC3(c3ccco3)C4)C2C1 C(CC(=O)N1CC(C)(C)C1C(C)C)(C(F)F)NC(c1c(OC)noc1C)=O CC1CC(C#N)(C(N2CC(CN(C)C(c3coc(Cl)c3)=O)C2)=O)C1 c1(OC)cc(NC(C2CCCC(NC(c3cccc(Cl)c3Cl)=O)C2)=O)cc(Br)c1 C(C(CCOC)NC(=O)Cc1nc(C)no1)NC(CC1C(CC)C1)=O c1(CC)cc(F)ccc1CC(=O)N(CC(C)N(C(=O)C=Cc1ncco1)C)C C(=O)(C1=C(C)CCCC1(C)C)N1CC(CNC(C(CCC)NC(C)=O)=O)C(C)C1 n1(C(F)F)ncc2c1CC(Nc1ncccc1OCc1ccc(Br)cc1)CC2 C(C(=O)NCCNC(=O)Cn1nnnc1C)(C(C)(C)C)c1cccc(C)c1 N1(C(CSCCN(C)C)=O)CC2CC2(NC(c2cnc(-n3cccn3)cn2)=O)C1 c1(NC(N(C2CCCCC2)C(C)(C)C)=O)sc(Cl)cc1Br C1(O)(C(C)(C)CNC(C2CC2(Cl)Cl)=O)CCN(C(C2CCCNC2=O)=O)CC1 c1(C2N(C(=O)NCCCCn3cnnc3)CCOC2)ccc(F)cc1F c1(OC)cnnc(C(=O)NC(C)CC2CN(C(C3CCCN3C=O)=O)C2)c1 c1(CC)c(C(=O)NC2(C)CC(C(=O)NC(C3CCOC3)CC)C2)nnn1C N1(C(=O)CC2CC3CCC2O3)CCCN(CCNC(C2(Br)CC2)=O)CC1 C1(C(=O)N)CCc2nn[nH]c2C1.C1(CC(=O)NC(C2(C)CC2)C)CC=CC1 C#CC1(C(N2CCCC(C(C)NC(c3sccc3OC)=O)C2)=O)CCCC1 C(N=c1nc(O)c2ccccc2[nH]1)C1CCN(C(=O)CC2CCCCC2O)C1 C1(C(C)C(=O)NC2CN(C(=O)Cn3cnnn3)C2)CCC(C)CC1 Cc1ccc(C)c(CC(N2CCC(N(C)C(C3(CC4CC4)CC3)=O)C2)=O)c1 c1(CNc2nc(COC)nc(N(C)CC3CCCC3)c2)cc2ccccc2o1 O=C(CCCCCO)NC1CC1CNC(C1CCC(C(F)F)CC1)=O Nc1cc2c(cc1C(N1CCN(c3ncc(Cl)cn3)CC1)=O)CCC2 C1(C(=O)N)C(Cl)(Cl)C12CC2.C(CCCC)N(C(CNC(=O)OCC)=O)C CC1COCCC1NC(C1(F)CCN(C(C2CCCC2)=O)C1)=O C#CCC(C(=O)NCCCC=C)NC(=O)CC1CSCCO1 c1(C(=O)NCC(C)(C2CC2)NC(C2CCSC2)=O)c(F)c(N)cc(Cl)c1F C1(CS(C)(=O)=O)CCCCN1C(CC(N)C(F)(F)F)=O C(C1CCc2ccccc21)NC(=O)CCn1cc(-c2ccc(CO)cn2)nn1 C1(CNC(c2ccc(OC)cc2)=O)CN(C(C2(OC)CC2)=O)CC(C)(C)O1 C1(NC(C(CC#C)C)=O)CC2CCC(C1)N2C(c1ccc(F)cc1OC)=O C1(NC(CCC)=O)CCC(CNC(=O)CCc2nc(C3CCCCC3)no2)C1 c1(C(=O)NCC(C)NC(C2N(CC)CC2)=O)csc(C(C)(C)C)c1 c1(N)ncnc2c1ncn2C1CC1.c1(NC(C23CC(C2)C3)=O)cccc(Br)c1O C1(c2n(C(COC)C)nc(-c3ccncc3)n2)CC12CCOc1ccccc12 Cc1ccc(C(=O)NCC2(C)CC(NC(c3ccncc3N)=O)C2)n1C C1(C(N(CC(CC)NC(C2CCC2CF)=O)CC)=O)CCCN1C(C)=O C1(OC)CN(C(C2CCC(=O)O2)=O)CC1NC(=O)Cc1ncccc1C C1CCC2(CCCCC2)O1.C(C(C(=O)NC)n1cc(CCN(C)C)nn1)OCC c1(C(N2CC(O)(CNC(C3(F)CCOC3)=O)C2)=O)cc(C(F)(F)F)n[nH]1 N1(c2cc(OC)ncn2)CCC(NC(c2cn(C)nc2C(C)C)=O)CC1C N1(C(COC)=O)CCC(C2CC(NC(=O)C(C)CC3CCC3)CCO2)CC1 c1(OC(C)C)cc(F)ccc1C(=O)NC1CC(CC)C1.C1(C=O)CCC1.N C1CC2(CO1)CN(C(c1ccc(O)cc1C)=O)C2.C(C(=O)N)=CCN(C)CC CCCC(CC(=O)N1CCCC1C(O)CO)NC(=O)CN1CCCC1C c1(C(=O)NC(CN(C(C=CC)=O)C)Cc2ccccc2)nc(C)ccc1F CC1C(NC(=O)CCC2CCCCO2)CCCN1C(=O)Cn1cc(CO)nn1 N1(C(C)=O)CC(CNC(c2cn3cc[nH]c(=O)c3n2)=O)CC12CCOCC2 c1(CC)[nH]c(C(=O)NCCC2CCN(C(C3(CO)CCCO3)=O)C2)nc1Cl C1(NC(C(C)OC(C)(C)C)=O)CN(C(=O)Cc2nccn2C)CC1F C1(C)(C(N2CC3CC3C2)=O)CCC2CC2C1.C1(C(F)F)(OC)CC(C=O)C1.N C(=O)(CCc1cn[nH]c1)NCCC(C)N(CCC)C.C(=O)C(F)n1ccnc1.N CC1CN(C(c2cc(-c3ccco3)nn2-c2ccccc2)=O)Cc2ccccc21 c1(CC)[nH]ccc1C(=O)NCC1CCC1.c1(C=O)c[nH]nc1C1CCOC1.N c1(C(N(C)CC2C(C)C2)=O)c[nH]nc1CCNC(C1CNC(=O)C1)=O c1(CC(=O)NCC(CNC(C2CC(O)(CC#C)C2)=O)C)cccc(F)c1 C(=O)(C(C)C(C)(F)F)NC(CN(C(c1nn(C(CC)CC)c(C)c1)=O)CC)C C=CCC(CC)C(=O)N1CCC1C(N1CC(OC(=O)NC)C1)=O C(=O)C(C)(C)S(C)(=O)=O.c1(CCC)ccccc1.C(C=C(Cl)Cl)=CC=O N1(CC)CCCCCC1.C1CCN(CC)C1.n12cc(nn1)N(CC(F)F)C(=O)C2C c1(OC)c(CN(C)CC2(C)C3CCCCC23)cc(Cl)cc1Br C(C1CCCCc2ccccc21)NC(c1ncoc1Br)=O N1(C(C2=NOC(C)C2)=O)CCC(C2CC2)C1.C(c1ccc([N+](=O)[O-])s1)=CC=O.N N1(C(CC2N(CC)CCC2)=O)CCC(O)(CCNC(=O)CCOC(C)C)C1 CC1CCCC(C)N1C(=O)C(=O)NCC1CCCC(C(F)(F)F)C1 C1(C(N2C(C)CC2)=O)CNC(=O)CN1C(=O)CC1(O)CCCOC1 C12(C(N(C3CC(OCC)C3)C)=O)CC1CN(C(C1(CCCF)CC1)=O)C2 Cn1c(I)cc2c(NC3(C)CCC(NC(=O)OC(C)(C)C)CC3)ncnc12 N1(C(C(CC)CCOC)=O)CCCC12CCN(C(C1CCC1(C)C)=O)C2 CC1CCN(C(=O)CCn2cccc2)CC1NC(c1cnc(Cl)s1)=O c1(COC)ccccc1C=O.N12CCC(C1C)NC(=O)C2C1CCC(F)C1.O N1(c2cc(C)nc(Cl)n2)CCCC1C1CCCCN1C(=O)CCS(N)(=O)=O C(=O)(C(=O)C(C)(C)C)NC1(C)CCN(C(C2CCN(CC(C)C)C2)=O)C1 C(=O)(C(CC)(CC)CO)N1CCC(CC=C)(NC(=O)C(N2CCCCCC2)C)C1 c1(C(N(C)CC2CCC(CNC(C(C)C)=O)CC2)=O)ccc(O)cc1[N+](=O)[O-] C#Cc1ccc(F)c(CNCC2(C)CCCOC2)c1 c1(CC)ccc(C(N2CC3C(NC(=O)C(C)(O)CC)C3C2)=O)cc1OC c1(OC)ccc(CN2CCN(CC(=O)NC3CC(O)CN3)CC2)c(O)c1OC C1CCN(C(=O)C(C)(C)c2cncnc2)CC1C.C(C)(C)(C(=O)N)OC(C)=O.C n1(CC)ncc(C(=O)NC2CCCC2NC(c2cnc(-c3cccnc3)s2)=O)n1 c1(NC(C2CCN(C(Cc3ccc(OC)c(C)c3)=O)C2)=O)ccc2nn[nH]c2c1 c1(-c2cn(C3C(C(=O)NC4(C(CC)=O)CC4)CCC3)nn2)cn2ccccc2n1 n1(CC(N2CCCCC23COC3)=O)nc(C(F)(F)F)c2c1CCOC2 C(C1=Cc2ccccc2OC1)N1CCCC(C(=O)NCC(C)(C)OC)C1 c1(OC)cc(C)sc1C(=O)NC.C1C(C)CCN1C(=O)C=Cc1cscn1 N1(C(C2(OC)CCSC2)=O)CC=C(CCNC(c2ccc(Cl)[nH]2)=O)CC1 CC1C(C(=O)NC(C)CC(C)(C)C)CCN1C(=O)C=Cc1cc[nH]c1 C1(NC(Cc2c(C)cccn2)=O)CC(NC(C2CC=CC2)=O)C12CCC2 N1(C(c2c(OC)c(Cl)sc2)=O)CC2(CCN(C(=O)CN3CC(C)(OC)C3)C2)C1 N1(C(c2n(C(C)C)ncn2)=O)CC(C)C(C)C1.C(=O)(CC=O)N.CC(F)(F)F C1(C(C)(C)O)CCN(C(=O)Cc2c(C)n[nH]c2C)CC1.C(C)(C=O)OCC=C.N O=C(C1=CCCC1)NCC1(C(=O)NC(C2CCC2)C2CC2)CCCO1 c1(NC(C(C)C)C(C)NC(=O)C=CC2CCOC2)ncc(Cl)cc1[N+](=O)[O-] c1(C(=O)NC(C2(O)CCCN(C(=O)CC3(C)CC3)C2)C)ncc2n1CCCC2 N1(C(C(C)N(C(=O)CN2CCCC2C)C)=O)CC=C(CO)CC1 C(=O)(C#CC(C)(C)CNC(=O)Cc1cnns1)NCc1ccc(C)c(C)c1 C1(C(=O)N)CC2(CCOC2)C1.Cc1csc(=O)n1CC(N1CC(OCC)C1)=O CC(C)CC(C(=O)NCC1(C)CCCC1)N1CCCC1=O.C(=O)C=CS(C)=O.N N1(C(c2c(C)onc2CO)=O)CCCC(CO)(Nc2ncnc(Cl)c2F)C1 C1(CNC(C(N2CCC(O)CC2)C)=O)CN(C(=O)CC2C=CCC2)CCN1C C12(NC(c3nc(CCC)sc3)=O)CCCC1N(C(=O)CCCOCC)CC2 c1(C(NCCNC(=O)CCc2ccc(F)nc2)=O)csc2cncn12.C1CC1.C C1(NC(c2cc(CNC(=O)C#CC3CCCC3)no2)=O)C2Cc3ccccc3C12 C1(F)(C(N2C(c3cn(CCCC(=O)OCC)nn3)CC2)=O)CCOCC1 c1(CC)ccc([N+](=O)[O-])cc1C(=O)N(CC(C)NC(c1cc(C)ccc1C)=O)C C(Cc1ccccc1)(C(=O)NCCC1(NC(c2coc(C)n2)=O)CC1)OC c1(C(=O)NCCN(C(CCOCCOCC)=O)C)nc(OC)c(Br)s1 C1(NC(C2CC=CCC2)=O)C=CCN(C(c2nc(Br)c[nH]2)=O)C1 c1(OC)cccc(CCc2nc(-c3ccnc(Cl)c3)nn2Cc2cnn(C)c2)c1 C1(C(=O)NCCN(C(C(CCC=C)(C)C)=O)C)C2CC3CC(C2)CC1C3 Cc1cc(C)cc(S(=O)(=O)NC2(CNC(c3cc(C)ccc3Cl)=O)COC2)c1 n1(CCC(=O)NC2C(NC(c3ccc(C)cn3)=O)C2)ccc2cccnc12 N1(C(COCCCC)=O)CC(NC(=O)C=CI)C(CC2CC2)C1 C1(NC(CNC(CC(C)C)=O)=O)CCCN(C(=O)Cc2ccc(Br)cc2)C1 c1(C(=O)NC(C2CCN(C(C3(C#C)CC3)=O)C2)C)cccc2c1nnn2C N1(C(c2cccc(Cl)c2)=O)CC2CCCC2(C(=O)Nc2ccccc2C2CC2)C1 C(=O)(CCCC(C)(F)F)NCC1(C)CCN(C(CN(C(C)C)C)=O)C1 C=CC(C)(O)CC(=O)NCC(C(=O)Nc1cccc(C(C)=O)c1)C(C)C C(c1cccnc1)=C(C(N1CC(NC(c2ccc(SC)s2)=O)(CO)C1)=O)C Cc1ncc(Cl)c(C(N2CC(NC(c3ccc(Cl)c(F)c3)=O)C(C(F)F)C2)=O)n1 Cc1ncc(NC2CCN(Cc3cnn(C(=O)OCC(C)(C)C)c3)CC2)cc1F CC(C)CC(C)C(=O)NC1CC(OCC(=O)NCC2CCCCS2)C1 Cc1nc2c(s1)CN(C(=O)CC1CCCN1C(c1ccc(Br)cc1)=O)CC2 Cc1cc(C(=O)O)ccc1C(=O)N(C1CCN(C(C2CC(C=O)C2)=O)CC1)C c1(CC(=O)NCC(C)=CC(=O)N(CC(C)C)CCO)ccc(O)cn1 C(=O)(CC(F)(F)CS(C)(=O)=O)NCCCCN(C(=O)C(c1ccccc1)O)C c1(C(N2CC(NC(C3C4COCC34)=O)C(O)C2)=O)cc(C(F)(F)F)ccc1Cl C1(N(C(c2csc(C)c2N)=O)C)CN(C(=O)CC(O)C2CCCC2)CC1(C)C c1(CN2C(C(=O)Nc3c(C)noc3C)C(O)CC2)c(Br)cc(Br)c(O)c1Br N1(C(C(C)OCCC=C)=O)CCC(C2CCCN(C(C3CC4C=CC3C4)=O)C2)C1 c1(-c2cc(C(N=c3[nH]nc(CC)s3)=O)c(=O)n(C)c2)c(Cl)c[nH]c2nccc1-2 c1(CC(=O)NCC2(C)N(C(c3cccc(C)c3)=O)CCC2)ccc(C)c(C)c1 c1(CC(=O)N)csc2ccccc12.c1(CCC)cc(C(=O)NCC2CC2)no1 N1(C(C=C)=O)CCCCC1C1CCN(C(=O)C(CC)N(C)C)C1 n1(CC)nc(C(C)C)cc1C(=O)NC1CCC1NS(=O)(=O)CC(=O)N c1ccc(Cl)c(Cl)c1.c1(CCN(C(=O)CN2CCCCC2)C)ccc(C(=O)N)s1 c1(C=O)cn2nc(C)cc2[nH]c1=O.c1(C(=O)NCCCC)ccc(S(N)(=O)=O)o1 c1(CC)ncsc1C(=O)NC(C1CCN(C(=O)CN2CCC2)C1)(C)C c1(CN2CC(CNC(c3noc(C)c3C)=O)C2)c(O)cc(Cl)cc1Cl C1(NC(c2cnoc2C2CCC2)=O)CCN(C(c2cnco2)=O)CC12CCC2 C1(NC(C2CC(Cn3cc(C)nn3)C2)=O)CC2(CCC2)CO1.C1(O)CCSC1 c1(C(N(CCC)CCNC(=O)C(F)C(C)(C)O)=O)cc(F)c(N)cc1F c1(N2CCC(NC(=O)CN3CCCS3(=O)=O)C(O)C2)nc2cccc(Br)c2o1 Cc1cccc(C(O)C(=O)NCC(C2CC2)NC(=O)C(C)c2cc[nH]n2)c1F N1(C(c2ccc(C#N)s2)=O)CC23CCCC2(C1)CN(C(C1C=CC=CC=C1)=O)C3 Cc1ccc(CC(=O)NC2CCOCC2NC(C2CCCN2C(C)C)=O)cc1F Cc1cccn2c(CC(=O)NCC=C3CCN(C(=O)C4=COCC4)CC3)cnc12 C1(S(C)(=O)=O)(C(N(C)Cc2n(C(C)C)ccn2)=O)COC(=O)C1 Cc1n[nH]cc1C(=O)N(C)CC1CN(C(=O)C(C)COc2ccccc2)C1 c1(N(CCC)CCNC(=O)CCSC(F)(F)F)cc(O)nc(=O)n1C c1(C(C(=O)NCCCC)N(C(C)C(=O)OCC)C)cc(C(N)=O)n(C)n1 c1(C(=O)NC2CCCN(C(CS(CC)=O)=O)C2)coc(=O)c2ccccc12 C(=O)(CS(N)(=O)=O)N(CC(O)Cn1nnc(-c2ccco2)n1)C c1(OC)ccccc1C(=O)NC.c1(CCN2CCC2)ccc(CC(C)(C)C)cc1 Cn1cnc2ccc(C(N3CC(C(=O)Nc4cc(Br)ccc4CO)C3)=O)cc12 c1(OC)cccc(F)c1CN1CCCC(CO)(NC(C2CCNC2=O)=O)C1 C1(NC(c2cc(C)n(C(C)C)n2)=O)CCC2CN(C(=O)Cc3cnoc3)CC2C1 CC1CN(C(=O)CCN2CCCC2=O)CC1NC(=O)CNC(N1CCCC1)=O C1(NC(c2c(C)scn2)=O)COC2(C1)CN(C(=O)CC)C2.C(C)(C)C.CC.O C1(C(=O)N)CCCCN(C)C1=O.N1(CCC)CCCC(C(=O)NCCC2CC2)C1 N1(C(C=Cc2ccc(C)nc2)=O)CC2OCCN(C(C3CC3(Cl)Cl)=O)C2C1 c1(C(=O)NC23CC(C(=O)Nc4nc(C)c(Cl)cc4)(C2)C3)[nH]nc2ccncc12 C1(C)(COC)CCCN1C(c1coc(CC)n1)=O.C1(CC=O)CCC(=O)C1 C1(C(=O)N)CC2(C1)CC2(F)F.C1(C=O)CCN(S(=O)(=O)CC)CC1.CCCC C1(OCC#C)CCN(C(=O)C(O)CNC(C2CC2(C)C(F)F)=O)C1 c1(C(N2CCC(CN(C(=O)C#CC(C)(C)C)C)C2)=O)cc2cccc(O)c2n1C C(CC(C(=O)N(C)Cc1nncn1C)NC(=O)C=CC1CCCN1C)=CC C1(C(N2CCN(C(Cc3c(C)scc3)=O)CC(O)C2)=O)Cc2ccc(F)cc2O1 C(=O)(C(O)CCN(C)C)NC1(CCNC(CC(C)N(C)C)=O)CCC1 C1(CNC(c2n[nH]c(C)c2Br)=O)CN(C(=O)C(O)CC(F)F)C(C)(C)C1 CCCC(C(=O)N(CC)CC1CCN(C(=O)CCOc2cccc(F)c2)C1)NC O(C=CC(=O)N(C(C)CNC(=O)CCc1nc(-c2nc[nH]n2)no1)CC)CC c1(C(=O)NCC(CC)NC(=O)CCc2cnc(C)s2)c(C)oc(C)c1C CC1(C)CC(NC(=O)C(C2(C)CC2)NC(C2CCS(=O)CC2)=O)CCO1 C1(C(N(C2CCN(C(C=C(C)C)=O)C2)CC2CC2)=O)CC2CCC1O2 c1(C(=O)NCC(c2ccccc2)NC(C2C3CCN2CC3)=O)ccc(O)cc1Cl c1(C(N2CC(C(=O)Nc3cc(O)c(O)c(O)c3)C2)=O)ccc(Br)c2cccnc12 C1(C(N(c2ccccc2)CC)=O)CCC2CCC1N2C(C1C2CCC(C2)C1C)=O C1(C=O)CC2C(C1)C2(C)C.C(C)(C)(C)NC(CC1(OCC)CC1)=O.N C1(CCNC(C(c2cccnc2)OC)=O)CCCN(C(=O)C(O)CN(C)C)C1 c1(NCc2c(OC)nccc2C)ccc([SH](=O)=O)cc1Br.C(C)CC1CC1.N N1(C(C(=O)Nc2c(C)cccc2)C)CCC2(C1)OCc1ccccc12 C(=O)(C1CCOc2ccccc21)NCC(CNC(=O)CCS(C)=O)OC C(C(O)CC(=O)N1OC2CCC1CC2)NC(CCN(C)CC)=O C1(CNC(c2c(C)ncnc2)=O)CN(C(c2cnoc2)=O)CCC12CCC2 CC#CCC(C(=O)Nc1cc(Cl)ccc1O)NC(C1CS(=O)(=O)C1)=O c1(C(N2C3CC(NC(COCCCC)=O)(C3)C2)=O)nc2ccccc2cc1C C1(C(=O)NCC2(c3ccccc3)CCC2)CCN=C2NNC=C12 C1(C(=O)NCCCN(C)C(c2ncsc2C2CC2)=O)CS(=O)(=O)CCO1 Cc1ccc(C(N2CC=CC(NC(=O)Cc3cnsc3)C2)=O)c(C(C)C)n1 C1(C(N2CC(NC(CCC)=O)C3(CC2)CCC3)=O)CCc2ncnc(C)c2C1 C1(C(N2CCC23CCC3)=O)(NC(C(CN(C)C)O)=O)CCCC1C c1(OC)ccc(CC(=O)NCC2(C)CCCN2C(c2cccnn2)=O)cc1O C12(CC(=O)N(CCC(C)(C)O)C)CCC1CN(C(C1C=CCS1)=O)C2 [SH](=O)(=O)CC=O.c1(C(N2CC(C(N)=O)C2)=O)ccc(O)cc1.CC(C)(C)N C1(NC(CCn2ncc(C)c2)=O)C2CC3CN(C(=O)C(C)NC(N)=O)C1C3C2 N1(C(c2cc(C)sc2C)=O)CCCC(C)(NC(=O)C=CCO)C1 Nc1ccc(C(N2CCCCC2CNC(=O)COCC2CC2)=O)nc1N Cc1ccc(CNC(=O)C(C)C(C)NC(=O)C2=COCC2)c(O)n1 C=Cc1ccc(C(N2CCC(OCC(=O)N(CC(F)F)CCO)C2)=O)cc1 C(=O)(CCCC(=O)N(C1C2CN(C(c3cc(C(C)C)on3)=O)CC12)C)OC Cc1noc(Cl)c1CC(N1CCOCC1CCNC(=O)CC(F)(F)F)=O CCCC(CNC(=O)CCc1ccccn1)C(=O)N(CC(F)F)C1CCC1 c1(-c2nc(C(CC)CC)nn2-c2nc(C)c(C)nc2C)ccnc2c1cnn2C c1(C(=O)NCCCN(C(CC(CC)O)=O)C)cc(Cl)c(OC)c(Cl)c1 N1(C(C(C)(C)c2csc(C3CC3)n2)=O)CCN(C(c2ccco2)=O)C2(CC2)C1 c1(C(=O)NCC2C=CCN2C(c2cccc(Cl)c2O)=O)ccc2cnoc2c1 N#Cc1cccc(CC(N2CC3(CCN3C(=O)CC3CC(C(F)F)C3)C2)=O)c1 N1(C(CCc2ccc(N)cn2)=O)CC2CCCC(C1)N2C(=O)Cn1ccnn1 c1(NC(N2CCN(c3ccc(C)c(S)c3)CC2)=O)ccc2c(n1)CCC2 C1(OC)CCCC1C(=O)NCCCN(C(=O)C(O)Cc1cnc[nH]1)CCO C1(CC)CSCCN1C(=O)Cc1cc(C)[nH]n1.C1(OC)(OC)CCC1C(=O)N C1(c2cn(-c3c(C)cccn3)nn2)CON(C(=O)CCc2c(C)cccc2C)C1 c1(NC(C2CN(c3nc(OC)c(F)cn3)CC(F)C2)=O)noc2ccc(Br)cc12 C1(NC(Cc2cc(C)sc2)=O)CC2CCC1C(NC(=O)C1=CCCCC1)C2 C1(C(=O)NCCCC(C)NC(c2cnc(C3CCOC3)s2)=O)CCC(C)(C)OC1 Cc1nc(-c2ccc(-c3nccn3CC)s2)cc(O)n1.c1(C)cc(C)c(C)nn1 c1(C(N2CCC(Cc3nccn3C)CC2)C(=O)NC)sc(Br)nc1Cl Cc1nn(C)c(Cl)c1C(=O)N(CCC(C)NC(c1[nH]ccc1-c1cccs1)=O)C CC1CN(C(C2(C)COCCO2)=O)CCC1C(=O)NCc1cnc[nH]1 N1(C(c2c(C)cco2)=O)CCC2(NC(c3ccc(OC(C)C)cn3)=O)CC2C1 c1(N2CCC(SC)C2)ncnc2c1ncn2CC1(CO)CCC1 N1(C(C(CO)N(C)C)=O)CC(NC(=O)C(c2ccc(C#N)cc2)O)CC(C)(C)C1 C1(CC)CN(C(=O)Cn2cc(C3COCC3O)nn2)CCN1C Cn1ccc(=O)cc1C(=O)Nc1ccc(C(=O)NCC2(O)CCC2)cn1 C1(C(=O)NC2Cn3c(C)nnc3CC2)CC12CCCc1ccccc12 C1(C(=O)NC(C2CCCCC2)CNC(C2C(C)C2C)=O)C(C(F)F)C1(C)C C1(C(N2C(CCC#C)CCC2)=O)COCCN1C(C1C2CC(=O)CC12)=O C1(C(=O)NCC(=O)NCCO)(CC)CCCN1C(c1cnc(NC)nc1)=O C1(C(=O)NC(C)C(F)F)(CC)CCN(C(=O)CS(C)(=O)=O)CC1 C1(O)(CC(=O)N(C(C(=O)N(C(C)C2CC2)C)(C)C2CC2)C)CCCCC1 N1(C(c2nc(CCCC)sc2)=O)CC2CC(C1)N(C(=O)CSCCC(C)C)C2 c1(C(=O)NC2(C)CC(NC(c3scc(OC)c3)=O)C2)c[nH]c(=O)cn1 n1(CC)cc(CCNC(c2cc(CNC(C3CC3C)=O)on2)=O)cn1 C(=O)(CCC(C)c1ccccc1)NCC1N(C(Cc2cc(OC)no2)=O)CC1 c1(C(C(=O)NC(C)(C)C)N(C(C(=O)NC)C)C)ncccc1OC CC(C)CC(=O)NC1(COC)CCC1.c1(CC)ccco1.C(=O)C.C=O.N N1(c2cccc(C)c2)CCN(C(c2cc(O)nc(C3CC3)n2)=O)CC1C N1(C(c2c(CC(C)C)onc2)=O)C2CCC1CN(C(=O)CC1CC1(C)C)C2 CN1CCc2[nH]nc(C(N3CCC(NC(c4cn(C)c(O)n4)=O)C34CC4)=O)c2C1 CC(CCNC(=O)C=Cc1ccoc1)CCNC(=O)Cn1cnnn1 CC1CN(C(=O)CSc2ccsc2[N+](=O)[O-])CCC1C.c1(CC=O)ccon1.N C1(NC(c2cc(Cl)ccn2)=O)CN(C(c2cc[nH]c2C2CCCC2)=O)CCC1F C1(NC(C(C)CF)=O)CC(C)N(C(=O)CCCCc2cccc(O)c2)C1 C1(C(c2n(CC(=C)C)nnn2)Nc2ccc(C)nc2)CCCC12CCOCC2 c1(C(=O)NC2C3CCN(C(=O)Cc4cnc[nH]4)C23)noc2cc(Br)ccc12 CC1CN(C)CC(C(=O)NC(C2CCCN2C(=O)C)(C)C)O1.CC(C)(C)C.O C12(NC(Cc3c(C)cccc3Cl)=O)CCCC1N(C(=O)C1CC1)CCC2 Cc1cc(NC(C2(C#N)CC2C)=O)ccc1NC(c1csc(C(C)C)n1)=O c1(OC)ccc(CC(=O)NCC(CO)NC(C2C=CCC2)=O)cc1[N+](=O)[O-] CC1(C)CCCN(C(c2cnnn2C2CC2)=O)C1C(N1CCC(OCCO)C1)=O C1(C(=O)NC)CCCCN1C(=O)CCN(C(=O)C(C)CC1CC1)C C1(C(=O)NC(C(CO)SC)C)CNC2CCN1C2 C=CCCC(CC)(c1nnnn1C(C)(C)C)NCc1ccn(CC(F)F)n1 c1(CN(C(CC)C(=O)O)CCC)cc(C)c(OCCNC2CCCO2)cc1C C1(CC(=O)NC2(C3CCCO3)CC2)C2CCCC2N1C(=O)Cn1ccccc1=O Cc1cccc(C(C)NC(=O)C(c2cccnc2)N(C)C)c1C c1(CC)nnc(C(=O)NCC(C)(C2CC2)NC(c2csc(C)c2)=O)s1 C1CC2(CCC2)C1.c1(C=O)ccc(C2(C)CC2)cc1.C(C)(C)(C(=O)N)SC O=C1CC(NC(=NCC2CCCC2)NCC(F)F)CN1Cc1ccc(Cl)cc1 C12(C(=O)NC3C(C(=O)NC)CCC3)CCN(C(c3ncn(C)c3C)=O)CCC1C2 C1(NC(c2nccc(C#C)c2)=O)CCC2(CC1)CN(C(=O)CCC(=C)Cl)CCO2 N1(C(C2CC(=O)N(CC(F)(F)F)C2)=O)CC2CC(NC(C3(F)CC3)=O)CC1C2 CCC(C)(C#N)C(=O)NCC1(C)CCCN1C(c1ccn(CC(F)F)n1)=O C(=O)(CCC(=O)N1CCCCCC1)NCC(C)N(C(=O)CCCNC(N)=O)C C1(=O)CC(C(C)OC)NC(=O)C2(CC2)N1C1CC1.C(C(=O)OC)OC C1(NC(c2nc(C)oc2)=O)C=CCN(C(c2ccccc2)=O)C1 C1(C(=O)NC2C(NC(CC(C)(C)C)=O)CCOC2)CC2(CC(OC(F)F)C2)C1 N1(C(c2cn(CC)nc2)=O)CC2(C)CC1(C(N1CC(O)CC1C(N)=O)=O)C2 c1(C(=O)NC2CC(C)(NC(CCC(CC)OC)=O)C2)cc(S(N)(=O)=O)cnc1C C#CCC(C(=O)N(CCO)CCOC)NC(c1ocnc1COC)=O C1(NC(=O)NC2CC3(CCCCC3)C2)CC2CS(=O)(=O)CC2C1 N1(C(C2SCCN(C(c3c(Br)ccc(C)c3)=O)C2)=O)CCn2cnnc2C1 C1(C(=O)NCCN(c2nccc(I)n2)CCO)CN(C(=O)C2CC2)CCC1O CC1CN(C(C2C3C4CCC(C4)C23)=O)CCN1C(C1CCCN1C1CCCC1)=O C1(c2c(CC)nccc2)C(C(=O)N2CCC(C)CC2)=C(CC)N(C)C(=O)N1C C1(O)(C(=O)NCCCN(C(C2CS(=O)(=O)C2)=O)CC)CN2CCC1CC2 CN1CCC(CC(N2CCC(OCCNC(=O)C(F)(F)CO)C2)=O)CC1 c1(OC)ccc2cc(C(=O)NC3CC(NC(=O)C(F)CC4CC4)C3)[nH]c2n1 N1(C(C2CCCN2C(c2cc(=O)cco2)=O)=O)CC2COCC2C1 Cc1ccc(CC23CC(CCN2C(=O)OC(C)(C)C)C3)c(Cl)c1 N1(C(CCC=C)=O)CC23CCCCC2(C1)CN(C(=O)CNc1ccccn1)C3 CC1CCN(C(=O)C(F)C2CCC2)CCN1C(=O)Cc1ccc(C(F)F)cc1 C1(C(=O)NC(CC=C)CNC(c2cn[nH]c2)=O)CCc2nccn2C1 C1(O)(CCNC(c2cc(CC)sn2)=O)CCCN(C(=O)Cc2cccs2)C1 c1(CC)n[nH]c(CC)c1CC(=O)NC1C2CC1N(C(C1CCC1OC)=O)C2 C1(C)(OCC)CN(C(c2occc2C)=O)C1.C(=O)(C(C)=C1CCCC1)N c1cn(-c2ccccc2)nc1C(C)(C)C.c1(C(N(CCOC)C)=O)sncc1C c1(C(=O)N)coc2c(Cl)cccc12.C1(C(=O)NC2CCC2)(COC)CCOC1 CC1c2c[nH]nc2CCC1C(N1CC2(CC(NC(=O)Cc3nc(=N)[nH][nH]3)C2)C1)=O C1(OC)CC(C(=O)NCc2ccc(C(=O)NC3CCOC3)nc2)C12CCC2 CCC(CC)C(F)C(=O)NCC(C)CC(=O)N(C1CCCC(C)(C)C1)C c1(C(C)OCC)nc(-c2cc(C)sc2C)n(CC2CCCOC2)n1 N1(C(C(C(=O)OCC)OC)=O)CCN(C(=O)CCc2cccc(C)c2)CC(O)C1 CCCCCCC(C)C(=O)NCC12CC(CO1)N(C(=O)C(O)CC)C2 C(=O)(C(C)(C)C(C)NC(C1CC(O)CN1C)=O)NC1CN(CC)C1 C1CC2CCC(C1)N2C(c1cn(C)c(=O)n1C)=O.C(C(=O)N)(C1CCC1)OC N1(C(CC2CC(C)C(C)CC2)=O)CC2CCC(C1)C(NC(C1C3CCCC13)=O)C2 c1ccccn1.c1(C(=O)N)ccnc(O)c1.C12CC(C=O)(C1)C2.CC(F)(F)F Cc1ccc(CCC(N2CCC(N(C)C(C3(C)CCCS3)=O)CC2)=O)cc1 C1CC2CN(C(c3ccn(C)c3)=O)CC12.C1(C(=O)OC)CCC(C(=O)N)O1.C C1(OC)CC(NC(=O)CCc2ccon2)CN(C(=O)C=Cc2ccc(Cl)cc2)C1 CC1C2CCC(C2)C1C(=O)NC(C(N1CC(C)(C)C1)=O)c1cccs1 N1(C(c2cnn(CC)n2)=O)CCCC(C)(NC(=O)CC2CCCCC2)C1 c1(CC)ccccc1C(N1CCC(N(C)C)CC1)C(=O)NCC1CCCO1 O=C1Nc2ccc(C(=O)NC3CCN(C(=O)CCN4CCCCC4)C3)cc2C1=O c1(C(=O)NCC(C)(C2CC2)NC(c2n(C)ccc2)=O)sc(F)cc1Cl CC(C)CCCC(C)C(=O)NC1(C)CCN(C(c2ccc(C#N)c(F)c2)=O)C1 Cc1sc(C)c(C(=O)NCCOCCCNC(=O)CN2CC3CC3C2)c1C Cc1cc(C(N2CC(C)C(C)C2)=O)ncc1C(N)=O.c1(CC(=O)N)ccns1 C(c1cccc(F)c1)=C(C(N1CCC(O)(CNC(C=COCC)=O)C1)=O)C.O c1(CC=O)ccc2ncccc2c1.C(=O)(C(C)(F)C(=O)NCC1CCC1)OC N1(C(C2CCC(C)CC2)=O)CC2C3CCC(C2C1)N(C(C1CC(O)CN1C)=O)C3 N1(C(CC(CC)O)=O)CC2CC(NC(=O)CC(C)n3ccnc3)CC1C2 C1(N(C)C(c2cccnc2Cl)=O)CCCN(C(c2cnc3n2CCS3)=O)CC1 C1(CCC(=O)N(CCC(=O)NC(C)(C)CON)CCO)CCCCO1 C12(C(=O)NCCNC(c3ncc(OC)nc3)=O)CCC(CC1)CC2 Cc1nc(C(N2CCOC(CNC(C3CC(F)(F)C3)=O)C2)=O)c2ccccn12 N1(CC)CCC(C(=O)NC2CCCC2)CC1.C1(C=O)CC(C(F)(F)F)CO1.C N1(C(c2csc(C3CC3)n2)=O)CCOC(c2ncno2)C1 CCCC(C(O)C(=O)N1CCCCC1C1CC1)NC(C1CC(=O)CC(=O)N1)=O O=C1CC(CC(=O)NCC2CC(NC(=O)C)CC2O)C(=O)N1.c1cccnc1 c1(CC(=O)OCC)nc(Nc2cccc(-c3ncnn3C)c2)sc1C C1(NC(C2CC(CC)C2)=O)CCC12CCN(C(c1ccco1)=O)CC2 C1(OC(C)C)(CN(C)C(C2CCCN2c2cnccn2)=O)CCOC1 c1(OC)cc(N)c(C=O)cc1F.C1(C(N(C(C)C)C)=O)CC(N2CC(O)C2)C1.N c1(C(=O)NCC(CCOC)NC(=O)C#CC2CCCO2)cccc2oc(O)nc12 CC1(C)CN(C(c2[nH]ncc2C#N)=O)CCC1NC(c1cccnc1O)=O n1(C2(CC(=O)NCCCN(C(c3cnsn3)=O)C3CC3)CC2)cncn1 c1(C(=O)N)ccn2cnnc2c1.N1(CCOC)CC(C(=O)NCC(O)C)CC1=O C12(CC)CN(C(=O)CC(C)F)C(C)(C1)C2.n1(CCC=O)cc([N+](=O)[O-])cn1 C1(C(=O)O)CCC2(CC(NC(c3ccccc3Oc3ccccc3)=O)C2)O1 N1(C(C=C(CCC)C)=O)CCC2(NC(c3ccc(-c4cn[nH]c4)cc3)=O)CC2C1 c1(NC(=O)NCCc2scc(C)c2)cccc(C(F)F)c1F C(=O)(CC1C(=O)Nc2ccccc21)N.C(=O)(CC1CCC1)N(CCOC)CC C(CC(C)(C)C)(C(=O)N1CCN(C(C2CC3CC(=O)C2O3)=O)CC(C)C1)OC c1(-c2nn(-c3cnc(C)s3)c(-c3nc4ncccn4n3)n2)cc2ccccc2o1 Cc1cc(C(=O)NCCN(C)C(C2(C)CC=CCC2)=O)sc1Br c1(C(N2CCC(C)C2CNC(C2SCCS2)=O)=O)nnc2ccccc2n1 C1(C(=O)NC(COC)C(C)C)(NC(=O)C(F)=CC2CC2)CCC(C)(C)C1 c1(C(=O)NC2(C(=O)NC(C)CC(F)(F)F)CC(CO)C2)ccc2c(c1)CC2 N1(C(C(CC(=C)C)C)=O)CCC2(C1)CN(C(=O)CN1CC(C)(OC)C1)C2 N1(C(CC(C=C)C)=O)CC2(C1)CN(C(=O)CC(=C)Br)Cc1ccccc1O2 C1(C(N(CCN(C(=O)CNC(c2cnn(C)c2)=O)C)C)=O)COCCN1C CCCCC(C)C(=O)N1CCCC(F)(CNC(c2nn(CCC)cc2Cl)=O)C1 CCCC(C(=O)NCCCCCC1CC1)NC(=O)C(=O)N(C)C C1(NC(CCCOCC)=O)CC2CC1CN(C(=O)C(CC)(CC)CC)C2 CC1(C(N2CC(O)(C)C2)=O)CC(C2CC2)=NO1.C1(C=O)CNC(=O)CC1(C)C c1(C(=O)NC2CN(C(c3n(C)ncc3)=O)C(C)(C)C2)c(F)ccc(F)c1N C1(C)(CC(N2CC(NC(C3C(CC)CCC3)=O)(CO)C2)=O)CCCCC1 C12(CCNC(CC(=C=C)C)=O)CCC1CN(C(C1CC(SC)C1)=O)C2 C(=O)(C1=NOCC1)NCC(CC)NC(C1C(C)CN1C=O)=O.C(C)(C)C Cc1nc(C)c(C(=O)NCC(C)(CO)NC(=O)Cc2cnc(C)o2)o1 C(F)(F)(C(=O)N1CC(C(N)=O)C1)C1(OC)CCC1.C1CCOC1.C(=O)C.C O=C(CCCN1CCCC1)NCc1n[nH]cc1C(=O)NCCC1CCCO1 O=C1Cc2ccc(C(N3CCCC3CNC(c3nccnc3Cl)=O)=O)cc2N1 C1(NC(c2n(CC)nc(C)c2)=O)CCCCCC1.C12(C(=O)N)CC(C)(C1)C2 c1(C(=O)NC2CCCC(NC(C(COC)(C)C)=O)C2)cnc(OC)c(C)c1 CCC(C)C(=O)N1CC(N(C)C(c2ccc(CC(C)(C)O)s2)=O)C1 c1(C(=O)NCC(C)(C(C)C)NC(CCC(C)OCC)=O)cc2ccccn2n1 C1(C(=O)NC(c2cn(-c3cccc(C(=O)OCC)c3)nn2)C)OCC2CCCC12 C1(C(N2CC(CCNC(C(C=CCCC)O)=O)C2)=O)OCCN(C)C1=O C12(CNC(C(C)(C)C3CC3)=O)COC(C)(C1)C2.C(=O)CCc1cn[nH]c1 c1(CC=Cc2cc[nH]c2)ccc(F)c(F)c1.N1(C(C2CC2)=O)CC(O)C1 C1CC2(C1)CN(C(C1CCCNC1)=O)C2.C(C=CC(=O)NC)(CC)=CC CN1CCC(C(=O)N(C)CC2CC(F)CN2C(c2ccc(O)nc2)=O)CC1 c1(C(=O)NC2C(CNC(c3c(N)cccn3)=O)C2)ccnc2cc(Cl)ccc12 CC1=C(C(=O)NCC2(C)CCN(C(=O)C(C)n3cnnn3)C2)COCC1 Cc1cc(C)c(C(N2CCC(C(C)NC(C3CCCC(=O)C3)=O)C2)=O)s1 C1(CC=C)(CNC2CCC(C(=O)OC)CC2)CCOCC1 C(=O)(CCCCC(F)F)NCC1CN(C(CCC2CCN(C)CC2)=O)C1 N1(CCCNC(C2CC2C2CC2)=O)CCN(C(C2(O)COC2)=O)CC1 C(C(C(=O)N1CC(C(=O)NC)C1)C(C)(C)C)NC(C(CC)OC)=O.C(C)=O Cn1nc(C(N2C(CNC(=O)C(F)n3cccn3)CC3CC23)=O)cc1O S(=O)(=O)(CCCCCl)N1C(C(N(CCCCO)CCCC)=O)C(O)CC1 c1(CNC(c2ccc(C)cc2)c2nnnn2C)ccc(C)c(F)c1F C1(NC(CCCOCC=C)=O)CCC12CCCN(C(=O)CCC(=O)NCC)C2 C1(NC(CCSCCCC)=O)CCC2CN(C(=O)Cc3ccn(C)n3)CCC2C1 c1(NC(C)=O)cccc(C(N2CCN(C(C34CC(C)(C3)C4)=O)CC2)=O)n1 C1(NC(CN(C)C(C2CCCC(=O)N2C)=O)=O)CC12CCCCC2 CN1CCCCC1CC(=O)NC(C)(C)CCCNC(C1CCC(=O)C1)=O C1(CC(=O)NC2CCN(CCC)CC2)CC2(CC2)CN1C(C1CCCSC1C)=O C12(C(=O)NC3CC(C)(CNC(CCCCC)=O)C3)CCCCC1C2(F)F N1(C(C(CSC)O)=O)CC2(CNC(C3CCCCC3)=O)CC1CCO2 S(=O)(=O)(c1cccnc1NC1CC(O)C12CCC2)NC1CCC([N+](=O)[O-])CC1 c1(C(N2CC(CC)N(C(C3CCC(=O)O3)=O)CC2)=O)cnc2ccccc2c1 Cc1cc(CC(N2CCC(NC(=O)C=Cc3ccco3)C(CO)C2)=O)ccc1F N1(C(C(C=C)CC)=O)CCCC(C(=O)NCC2(CCO)CCC2)C1CC C1(O)(CC=C)CCN(N(C)Cc2cc(F)c(F)c(F)c2)C1 N1(C(c2ccc(C)o2)=O)CCC2(NC(=O)COc3ccon3)CCCC12 C(CN=c1[nH]c(=NC2CCCC2N(C)C)[nH]c2cc[nH]c12)C1CCN(C)C1=O c1(C(=O)NCCOC2CCN(C(c3c(C)nccn3)=O)C2)cccc2nncn12 c1(C(N2C(C(N)=O)CC2)=O)c(-c2ccc(F)cc2)csc1C(=O)O C1(NC(C(C)C2CC2)=O)CN(C(c2cn(-c3cccc(CO)c3)nn2)=O)CC1O c1(NCC)ccc(S(N)(=O)=O)cc1C(=O)OCC1CCCC(C)(C)O1 C1(C(N2C(C=C)CCCC2)=O)CC2C=CC1CCC2 c1(SCC)nc(C(N2CCC(CNC(c3cn[nH]c3)=O)C2)=O)cc(=N)[nH]1 C(=O)(CCC(O)C(C)(C)C)N1CC(C(C)NC(c2cccc(SC)n2)=O)OCC1 C1(C)(CCC(=O)N(C2CCCC2O)CC)CN(C(=O)C=CCNC)C1.C c1(NC(C(C2CCN(C(C=CC=CCC)=O)C2)C)=O)cc(OC)cc(C)c1 C1(CC)CCCCN1C(=O)C(C(C)C)NC(=O)Cc1cccc(F)c1 CC(CCCCNC(c1n[nH]cc1Cl)=O)NC(=O)C(C(C)O)NC(=O)C1CC1 N1(C(c2cc(CC)nn2C)=O)CCC(NC(=O)Cn2cnnn2)C2CC12 NC1CCC(CN(CCC(O)c2cccs2)Cc2ccccc2)CC1 c1(C(=O)NC2C(OC)CN(C(C3C(C)C3C)=O)C2)cc2cc(C)ccc2o1 CN1CCC(c2cn(CCOCCNC(C3(C)COCCO3)=O)nn2)CC1 Cc1ccc2nc(Cl)c(CN3CC(C(=O)N=c4[nH][nH]c5cccnc45)C3)cc2c1 N1(C(c2cc(C)c(C#N)[nH]2)=O)CC(C)N(C(=O)CC(C)C)CC1C c1(C(=O)NC2C(OC)CN(C(c3ccccc3)=O)C2)cc2c(ccn2C)[nH]1 CN1CC2(CC(NC(=O)C=CC3CCCN3C(c3cnc(O)c(F)c3)=O)C2)C1 N1(C(C2(CNC(CCCC)=O)CCCC2)=O)CC2CCC2(OC)C1 Cn1cc(CNCc2cc[nH]c(=N)c2)c2ncccc2c1=O CC(C)C1=NOC(C(=O)NCC2CCC2)C1.c1(C=O)nn[nH]c1C(F)(F)F C1(NC(C=NOC)=O)CC(F)(F)CC1NC(c1ccc(Br)cc1)=O C1(C(=O)O)(NC(CCc2c(C)ncs2)=O)CCCN(C(=O)C(C)SC(F)(F)F)C1 c1(C(=O)NCCNC(C2(O)CC3CCC2C3)=O)cc2c(Br)coc2cn1 c1(CNC(CCC2CCN(C(c3cc(OC)n[nH]3)=O)C2)=O)cc(C)c(C)s1 Cc1nn(C)c2sc(C(N3CCC(CO)C(C)C3)=O)cc12 C1CC2(C1)CS(=O)(=O)C2.c1(OC)ccc(-n2nnnc2Cc2cn[nH]c2)cc1.N c1(C(C)C)nc2n(n1)CCCC2NCc1cccnc1O C(=O)(N1CC(O)C(O)CO1)C1(CNC(C2C=CCS2)=O)CCCC1 Cc1cccc(C)c1CC(N1CCCC1CC)=O.C(=O)(C(C)C)N.[SH](C)(=O)=O C(CCCC(C)(C)NC(=O)C(C)CC#N)NC(C1N(CC)CCCC1)=O c1(C(N2C(CNC(CC=C(C)C)=O)CN(C)CC2)=O)cc2cccc(Cl)c2o1 n1(CC)nc(C(=O)NCC=CC)cc1C.c1(C=O)c(C(F)(F)F)cnn1C C1(C(N2CC(CCCNC(CCC(C)OC)=O)OCC2)=O)SC2C=CC1CC2 N1(Cc2nc(C)sc2-c2ccccc2)CC=C(CCNC(=O)C(F)C(C)C)CC1 CC(C)C(C(=O)NC1C(C(=O)NC2CCOC23CCOC3)C1(C)C)C(C)C CCCC(O)CC(=O)N1CCN(C(c2cnc(C)[nH]2)=O)C(CCOC)C1 Cc1ccc(C(=O)NC(C2CCCN2C(c2cnc3n2CCS3)=O)(C)C)cc1Cl Cc1ccc(C=CC(N2CCCC3(CNC(=O)C(F)(F)C(F)F)CC23)=O)cc1 c1(C(N2CC3CN(C(c4cccc(F)c4Cl)=O)C3C2)=O)[nH]nc2ccncc12 Cc1ccc(=NCCC(=O)N2CCOC(C(C)NC(=O)CC(=O)N(C)C)C2)[nH]c1 Cc1[nH][nH]c(=NC(=O)c2ccc(CCC(=O)Nc3c(F)cc(F)cc3Br)[nH]2)c1Cl CC(C)CC(C)CC(C)C(=O)Nc1ccc(NC(=O)C2CC2)cc1 N1(C(C2(COC)C=CCN2C(=O)CC2CCCC2)=O)CCOC2COCC2C1 c1(C(=O)NC(CC(C)NC(CCSCC(C)C)=O)C)ccc2nc(O)[nH]c2n1 c1(CCC(=O)NCCNC(c2ccnn(C)c2=O)=O)ccccc1[N+](=O)[O-] c1(NC(C2CCCN2)C)nc(N2CCC3(CCOC3)C2)nc2sccc12 C1(NC(c2cc(COC)no2)=O)COCCC1NC(=O)C.c1ccccc1.O N1(C(C2CC(=C)C2)=O)CCC2(NC(C34CCC(CO)(CC3)CC4)=O)CCCC12 c1(C(N(C2CCN(C(c3cn(CCC)nn3)=O)C2)CC)=O)ccnc(OC)c1 Cc1cc(C(=O)N)c(N)c(Cl)n1.C1CN(C(c2scc(C)c2C)=O)C(C)(C)C1.C c1(CC)ncc(Br)cc1C(=O)NCC1CCCCN1C(C1CN(C)C1)=O c1(C(C)C)nn(-c2ccccc2)cc1COC(=O)C=C(C)c1cccs1 c1(NC2(COC)CCOCC2)ncc2c(C)cn(C)c2n1.C12(CCOCC1)NC2 C(=O)(C(O)CN(C)C)N(CC(C)CNC(=O)CO)C.n1(CC)cncn1 c1(C(N2CC(NC(c3cc(C(F)F)cs3)=O)C(O)C2)=O)cccc2c1SCCC2 CCC(CC)CCC(=O)N1CC2CCC2(CC(N2CC(COC)(CC)C2)=O)C1 N1(C(C(CCC)NC(N)=O)=O)CCN(C(c2cnc3n2CCC3)=O)CC1CO C(=O)(C(CCC1OCCO1)N(C(C)C(=O)OC(C)(C)C)C)NC(CC)C Cc1[nH]nc2c1CC(C(N1CCCC(CO)(NC(=O)C(F)=CC3CC3)C1)=O)CC2 C1(NC(c2cc(CC)ncc2)=O)CCN(C(=O)Cc2ncc(C)s2)CC(C)(C)C1 C1(C(=O)NCC(C)C(=O)NCCF)CCCC(CF)C1 C(CC(C)C)(C(=O)NCCc1cccnc1F)NC(C(C)N(C(C)=O)C)=O C(=O)(C(C(C)(C)C)N1CCCC1=O)N(C1C(C)CCNC1)c1ccccc1 Cc1ccc(-c2nc(-c3c(I)n[nH]c3C)no2)cc1C N#Cc1cc(NC(c2cscc2Br)=O)ccc1Cl Cc1ccc(C=CC(=O)NC(C)CC(C)C)o1.C(=O)(CCCN1CCOC1=O)N CCC(CC)C(C)C(=O)NCC1CC1NC(c1cc(Cl)c(F)cc1F)=O c1(C(=O)NCc2cc(C)sc2)ccnc(C2CC2)c1.C12(CC1)C(=O)NC2 CCC(CC)C(=O)NC1CCC1NC(=O)CCc1nncn1C N1(C(Cn2c(C)ncc2)=O)CCC(O)(CC)C1.C(F)(F)C(F)(F)F.C(=O)(C)N C(C)(CCCC(=O)NCCC(=O)N(C)C)NC(CC(CC)O)=O c1(C(N2C3CC(NC(=O)CC4CCOCC4)C2CC3)=O)coc2cccc(O)c12 c1(NC(C(N2CCSCC2)C)=O)nc(Cn2cc(Br)cn2)cs1 c1(OC(F)(F)F)cccc(CNc2ncc(C(F)(F)F)[nH]2)c1 c1(C(N(CCOCCC(=O)NC(CCC)C2CCCC2)C)=O)ncsc1C C(CC)(C(=O)N=c1[nH]n2cccnc2c1Cl)N(CCN(C)C)CC c1(C(N2CCC3(CCCN(C(=O)C(F)F)C3)C2)=O)c2c(cc3c1CCC3)CCC2 C(=O)(C1CCCc2c[nH]nc21)N1CC(NC(c2c(COC)ncs2)=O)(CF)C1 c1(C(N2C3C(NC(C4CCN(C)C4=O)=O)CC(C3)C2)=O)cccc2sccc12 N1(CC2CN(C(c3cc(C(C)(C)C)no3)=O)C2)CCN(C(=O)CC2CC2)CC1 N1(C(C2C(OC)(OC)CC2)=O)CC=CC1(C)C(=O)NC1CC(C)OC1=O c1(C(=O)NC(C2(O)CN(C(C3C(OC)C3)=O)C2)C)ccc(Br)c(C)c1F Cc1cc(Br)cc(C(N2CCN(C(=O)CC(C)NC(N)=O)C(CO)C2)=O)c1N C1(C(=O)NCc2nnc(COC)o2)C2CC(C(O)C2O)S1(=O)=O Cc1ncccc1C(=O)NCc1csc(CN(C)C)n1 n1(CC(=O)NCC23C(CN(C(CC=C=C)=O)C2)CC3)ncc2ncccc12 N1(C(C(C(C)C)OC)=O)CC(C)C(C)(CNC(c2cncn(C)c2=O)=O)C1 c1(NC(CNC(C(C=CCCC)O)=O)C(C)C)cc(SC(C)C)nc(C)n1 C1(NC(c2ccc(OC)c(C)c2)=O)CC2CC(C1)N(C(c1ccccc1)C)C2 CCCCCC(O)C(=O)N1CCCCC1CCCNC(=O)CSC c1(C(=O)NC)cccc2c1CCOC2.C1(C=O)CC(C(F)(F)F)CO1.C1CCC1 C=CC(CC)C(=O)NC1(CCC(=O)N(C)CC2CCCCC2O)CCC1 C1(NC(CN(CCC)C)=O)COCC1C(=O)NC(c1cscn1)C C1(C(=O)NC2CCC(NC(C3CC4CCC3O4)=O)C2)(OCC)CCCCCC1 N1(C(C(C2CCC2)OC)=O)CC(NC(c2cnc[nH]2)=O)CC12CCCCC2 C1(NC(C(C)C2CCC2)=O)CC2CN(C(c3csc4ccccc34)=O)CC2C1 c1(OC)ccccc1NC(=O)C(C)CO.C1(COC(C)C=O)COCC(C)O1 C12(C(N3C(C(=O)NCC4CCCCC4O)COCC3)=O)CCCN1CCC2 N1(C(C2(C)N(C(CCCOC(C)(C)C)=O)CC(O)C2)=O)C2C=CCC1CCC2 N1(C(C=CC=CCC)=O)CC2(NC(=O)C=Cc3csc(C)n3)CCC1CC2 C1(CNC(C(C)SCC)=O)CN(C)CCN1C(C1CS(=O)(=O)C1)=O N1(C(C2CC3CCC(C2)C3)=O)CC2CCC(C1)C2.C(=O)(C(F)(F)c1cncs1)N C(C)(CC(C)C)NC(C=C(C)C(C)C)=O.c1(C(=O)N)ccc(N2CCCC2)nn1 N1(C(C(C(C)C)OC)=O)CCC(F)(F)C(CNC(=O)C2=COCCO2)C1 C1(O)(CN(C(C(C)CC2CC2)=O)C)CCCN(C(=O)CCC2CCCCC2)C1 C(=O)(CC(F)(F)C(F)(F)F)NC1CCCCN(C(c2ccc(CN(C)C)[nH]2)=O)C1 C1(CCOC)(NC(c2cccn2C)=O)CCN(C(=O)CCC2CCCN2C)C1 C1(C)(C(N(CC(C)C)CC(=O)NCC2CCCS2)=O)CCCCC1C N1(C(C(C)OCC)=O)CCC(F)(C(=O)NC(c2cccc(C)n2)C)C1 C(=O)(C(C)(C)C(F)c1ccccc1)NCC(C)(C)NC(c1cnn(C)c1F)=O C(=O)(C1CCCc2nncn21)N1CCOCC(CNC(C2(CCCC)CC2)=O)C1 O=C(CC(F)(F)C(F)F)NC1CC2(C1)CC2NC(C1Cc2cccnc2C1)=O c1(C(=O)NCC2(OC)CN(C(C3CCC(O)CN3C)=O)C2)cnc2c[nH]nc2c1 N1(C(C2CCN(C(=O)CCc3ccco3)C2)=O)CC2CCC(CC2)C1 c1(C(N(CCCN(C(CC2(CC(=O)OC)CC2)=O)C)C)=O)ncccc1Br C(=O)(C(C)N1C(=O)COc2ccccc21)N(CC=C)C CCC(c1ccccc1)=CC(=O)NC1CCCCCC1NC(C1CCCC1)=O c1(C(C)C)noc(CCC)n1.C1(CC=O)CN(C(C2(n3nccn3)CC2)=O)C1.N N1(C(C(C)=C(CC)C)=O)CC(CNC(c2cnncc2OC)=O)N2CCC1C2 C1(NC(CCCN=[N+]=[N-])=O)CCC2CCN(C(=O)COCCCF)C1C2 CCCCC(F)C(=O)N1CCCC(NC(C2OCCC2(C)C)=O)CC1 Cc1ccc(O)c(C(=O)NCC2CC(C)N(C(=O)CCC)C2)n1.[SH](C)(=O)=O c1(C(N2CCC(N(C(C3C4CC4C4CC34)=O)CC)CC2)=O)ccc(F)c(O)c1 N1(C(CC(C)(C)OC)=O)CCC(C)(C)C(CNC(=O)C(C)C2CCCC2)C1 c1(OC)nscc1C(=O)NC1CC(C(=O)NC2CC(C(C)(C)C)C2)C1 C1(C(=O)NCc2oc(C)c(C(N3CCC4CC34C)=O)n2)CN2CCC1CC2 Cc1cc2c(Br)ccc(-c3c(N)ncn3C)c2o1 C1(O)(CN(C(c2c(C)cc(C)o2)=O)C)CCCN(C(=O)C(F)C2CCCC2)C1 C(=O)(CC1OCCc2ccccc21)N(CCCNC(C(CC#C)O)=O)C1CC1 c1(C(=O)NC(C(C)NC(c2nc(Br)c[nH]2)=O)(C)C)cc(O)nc(O)n1 c1(CC(=O)NC(C(C(C)C)C)CNC(c2scnc2Cl)=O)cnc2n1CCOC2 C#CC1(C(=O)NC(CO)CCCCNC(c2ccn(C)c2)=O)CCOCC1 c1(C(N2C(CNC(CC(COC)(C)O)=O)CCCC2)=O)ccnc2ccncc12 C(=O)(C(C)CC1CCCCC1)NCCN(C(C1C(CC)C1)=O)CCOC C12(CNC(C)=O)CCCC1CCN2C(=O)Cc1ccc(Cl)c(C(F)(F)F)c1 Cc1ccc(C(=O)NC2CCCCC2C)c(C)n1.c1(C=O)cnc(N(C)C)o1.N C1(C(=O)NCCOCCNC(c2ncccc2Br)=O)CC2CCCC(C1)C2 CCC(C)CC(C(=O)N(CC(C)(CC)OC)C)NC(=O)CC1(N(C)C)CCC1 N1(C(Cc2c(C)nsc2)=O)CC(F)CC1CNC(c1cn[nH]c1)=O C12(C(N(CC(CC)O)CC)=O)CC(NC(=O)C(N3CCCCC3)C)(C1)C2 c1(OC)cncc(C(=O)NCC(CCNC(=O)Cc2c(C)n[nH]c2C)OC)c1 c1(SCC(=O)NCC2(O)CCN(C(CCCSC)=O)CC2)nc2ccccc2s1 C1(C(N2C(C(=O)OC)C(C)(C)C2)=O)COC2(C1)CN(C(C1CC(O)C1)=O)C2 C=CCCCC(C(=O)NC(C)Cc1cn[nH]c1)NC(c1cnn(CC)c1)=O c1(C(=O)NC2(CF)CCN(C(C(C=C)(C)O)=O)C2)cc2nccc(C(F)F)n2n1 C(CCN=c1cc(Cl)nc(C2CCOCC2)[nH]1)NC(CCC(=O)N(C)C)=O CC(C)(CNC(=O)CCCCCF)CC(=O)N1CC(F)(CF)C1 C1(CNC(C(C)c2ncco2)=O)CCCN(C(=O)Cc2cnco2)C1 C1(c2nnc(C)o2)CCCCN1CCCOCC(F)(F)F c1(C(N(C(C)C)CCNC(c2sncc2Br)=O)=O)cccc2c1OCC2 C(CC(=O)NCCOCCNC(=O)C(O)c1ccco1)=CC C1(OC)(OC)CC(C)(C(=O)NC2CCC2)C1.N1(C(C=O)C)CCCCC1=O.C Cc1cc(C(N2CCC(C)C2)=O)c(O)c(C)n1.c1(C(=O)N)ccnc(N(C)C)c1 N1(C(C(CC#C)C2CC2)=O)Cc2n[nH]cc2C1C(=O)NCc1ncsn1 c1(-n2ncc(C(N3CCCCC3)=O)n2)ccc(Cl)cc1.O=C(CSC1CC1)N.C c1(NC(C2N(C(C(C)(CO)CO)=O)CC(F)(F)C2)=O)ccc(F)c(F)c1Br N1(C(CCC(=C)Br)=O)CC(C(=O)OCC)OC2COCC12 N1(C(C2CCC(C)O2)=O)CCCCC1CNC(C1(n2cnnn2)CCOCC1)=O C(N=c1[nH]c(=N)[nH]c(=NC2CC(CCO)C2)[nH]1)c1cc(C)nc(O)c1 N1(C(c2ccc(CC)c(C)c2)C(=O)NCCC)CCN2C(CNS2(=O)=O)C1 CC1CN(C(C2(CO)CCCCO2)=O)CCN(C(=O)C(C)NC(N)=O)C1 C1(OC)CC2CC(NC(C34CC3CCN4C(C3CC(CF)C3)=O)=O)CC12 N1(C(C(CCC)N(C)C)=O)CC2(CCN2C(=O)CSc2nnnn2C2CC2)C1 Cc1nc(NC(c2ccc(C(C)(C)C)[nH]2)=O)sc1C(=O)NCC1CCC1 C=CC(CC)CC(=O)N1CCCC1C(C)NC(c1cn(C)nc1C1CCCC1)=O C(=O)(CCCC(=O)N1CCC2(CC2NC(=O)CN(C)C(C)=O)C1)NCC c1(C(=O)NC(CCOC)CNC(=O)C(O)c2ccsc2)ccc(F)c(F)c1 C1(NC(CSCC#C)=O)CC12CC(NC(C1(NC(N)=O)CC1)=O)C2 c1(C(N2CCC(NC(=O)CCC3CCCC3)C23CC3)=O)ccc(F)c(F)c1F c1(C(=O)NCC(CO)NC(Cc2cncc(C)c2)=O)coc2c1C(=O)NCCC2 c1(NC(CCC(=C)Br)=O)ccc(NC(C23CCCC2OCC3)=O)c(C)c1 c1(C(=O)NC2CC3CC2N(C(=O)C2=CCCOC2)C3)cccc(C#CCO)c1 Cn1nnc2c1CC(C(=O)NC1CCC1CNC(=O)CC=C(Cl)Cl)CC2 C(=O)(C1=C(Cl)CCC(C)C1)N(CCN(C(c1c(CSC)cccn1)=O)C)C C=C(CNC(=O)C(=O)NC1CC1)CCNC(C1CC1(F)F)=O C1(NC(Cc2ccc(C)s2)=O)CC2CC1CN2C(=O)CCC(=O)N(C)C N1(CC(=O)N(C)CC)CCC(C2CCCN(C(=O)CC(C3CC3)C3CC3)C2)C1 C1(CNC(C=CCCC=C(C)C)=O)CCN(C(C2(C(N)=O)CCC2)=O)C1 Cc1cc(CC(=O)NCC(C2CCCC2)NC(C2CCC(C)O2)=O)n[nH]1 c1(OC)c(CN2CCC(CC(N3CCC(C)(O)C3)=O)C2)cccc1F c1(C(=O)OC)cc([N+](=O)[O-])ccc1NC1C(C)CCCC1C C1(C(=O)NCCSCC(=O)NCC(C(=O)OC)O)CCCC(C)CC1 CCCC(C(=O)NC(CCC1CC1)C(=O)N(C)C)OCC.C12CCC(CC1)C2 Cc1ccc(-n2cc(C3(NC(=O)C(F)CC4CC4)CCC3)nn2)c(F)c1 N(C(=NCc1ccc(Br)cc1)NCc1cnccc1Cl)C(COC)C NC(CC(=O)NCc1nc(C2CCCO2)n[nH]1)C(F)(F)F c1(C(=O)OC)cc(C)c(C)cc1NCc1ccc(OC)cn1 c1(N(C2CCCCNC2)C(C)C)ncccc1NC(N1CCCC1)=O.C(C)(C)C.O N1(C(c2cscn2)=O)CCN(C(C2CCN(C3CCSC3)CC2)=O)C(C(F)F)C1 C12(C(N(C)CCOCCNC(=O)Cc3ncc[nH]3)=O)CSCC1C2(F)F C1(C(=O)NC(CNC(c2c(SC)ccs2)=O)C2CCC2)CCn2nncc2C1 c1(C(N2CCC(N(CCC)C(C3CC3CC)=O)CC2)=O)ccc(C)c(OC)c1F C1(CCNCC(C)CCO)CCC(c2nnnn2C)(Nc2ccccc2)C1 CCC(CCC(=O)N1CCC(CC(F)F)C1)NC(=O)CC(O)CC C(=O)(N=S(C)(=O)C1CCCC(O)C1)c1c(C)occ1C(F)(F)F N1(C(c2cc(C)ns2)=O)CC2CCN(C(c3nccc4c[nH]nc34)=O)C2C1 C1(C(=O)NC(C23CCC(CO2)C3)C)CN(C(=O)C(C2CCCCC2)C)CC(C)O1 C1(CC(=O)NCC(CN(C(C2CC(=C)C2)=O)C)(C)C)CCCC(C)(C)C1 c1(C(N2CC(NC(C(CC=C)C)=O)CC(C)(C)C2)=O)ncnc2c(C)csc12 C(=O)(C1=NOC2COCC12)NCC1(CNC(C(C=C)(F)F)=O)CCOCC1 C1(C=O)CCCCC1C(F)(F)F.C1(CC)CN(C(C2CS(=O)(=O)C2)=O)C1 C1(C(=O)NCCC2(O)CN(C(=O)CCC3CCCC3)C2)CC12CC2(F)F N1(C(CCN(C)C)=O)CC2(CC2)CC1CNC(C1CCOC1)=O N1(C(CC(C)(C)C)=O)CCC(NC(C2CN3CCN2CC3)=O)CC1C1CC1 N1(C(C2ON=C(CC)C2)=O)CC2(CO)CC1(C(=O)Nc1ccccc1CO)C2 N1(C(C(C)SC)=O)CCC2(CCOCC2)C(NC(c2ccn3ccccc23)=O)C1 Cc1ccc(NC(C2CCN(C(C3CCCC(C)C3)=O)CC2)=O)cn1 c1(C(=O)N)cccc(C)c1N.N1(C(C2(OCC)CCC2)=O)CCC(C(F)F)C1 c1(N2CCCC(CCC=C)C2)cc(NCc2nnc3n2CCC3)nc(C)n1 Cc1c(NC(C2CC3CC3N2C(=O)C(C)(F)F)=O)cccc1C#N C1(N(C)C(c2n[nH]cc2Cl)=O)CC2CCC(C1)N2C(=O)C(C)(F)C(C)(C)F CCCC(O)C(=O)N(CC(C)NC(C1CCCN(C)C1)=O)C CC(C)C(CCN(C(=O)CC(F)F)C)NC(=O)Cc1csc(-c2cccnc2)n1 C1(n2cc(CCOC)nn2)CCC(C)(C)N(C(c2nc(Br)cn2C)=O)C1 C(=O)(CC1=CCOCC1)NC1C(CO)CCN(C(CNC(=O)CC2CCCC2)=O)C1 C#Cc1cccc(C(N2CC(O)(c3cn(CC4CC(F)(F)CO4)nn3)C2)=O)n1 Cc1[nH]c2ccc(C(N3CCN(C(=O)CC4CC4)C(CF)C3)=O)cc2c1C C1(CC(=O)NC(CN(C(c2cnc(CC)s2)=O)C)(C)C)CCOC(CC)C1 n1(CC(=C)C)nnnc1C(CC1CCCO1)NCc1cc(C(C)(F)F)on1 C1(NC(COC(C)C)=O)CCC(NC(=O)C=CCN2CCCC2)CC1 Cc1nc2n(c(=O)c1CCNC(C1CCSCN1)=O)CCCC2 N1(C(CC=CC=C)=O)CCCC2(NC(c3cc(C4CCC4)[nH]n3)=O)CC2C1 c1(Cc2cn(C(C)C(=O)NN3CCNC(=O)C3)nn2)cn2ncccc2n1 C1(NC(=O)CCc2cccs2)CN(C(C2(CC(F)F)CC2)=O)Cc2ccnn2C1 c1(C(=O)NCCN(CCCC)C(C)CC)cnc(CC)s1 C1(CN(C(=O)C(C2CCOCC2)=O)C)CCN(C(=O)CCS(C)=O)CC1 C=Cn1nccc1C(=O)NC(C1CCN(C(c2cnc(C(C)C)[nH]2)=O)C1)C C(C)(CCC(=O)NC(CN1CCCC1)CO)OC.C1(C=O)C2(CC2)C12CC2.N C1(CC(=O)NC2CCCN(C(c3ccc(Cl)c(F)c3)=O)CC2)CCCCC1(F)F C=CC(C)(CC)C(=O)N1CC(NC(=O)CCc2cc[nH]n2)C(n2cccn2)C1 N1(C(CC(CC)CC)=O)CCCC2(NC(c3ccnc(C)n3)=O)CC2C1 CCS(=O)(=O)CC(=O)NC1CC(CCNC(=O)C=CC=C(Cl)Cl)C1 c1(C(=O)NC(COC)CC(=O)NCC(F)(F)Cl)cccc(F)c1O C1(C(=O)Nc2c(OC)ncc(F)c2)CC2OCCC2N(C(=O)C(=O)C2CC2)C1 C1(NC(c2c(C)ccc(F)c2)=O)CC12CCC(NC(C1(F)CCCOC1)=O)CC2 N1(C(Cc2c(C)cccn2)=O)CCN(C(C23CCC(C)(C2)OC3)=O)C(CCO)C1 CCCCCCC(F)C(=O)N1CCN(C(c2noc(C3CC3)c2C)=O)CC1CC C(C(C)CCC#N)N(C)Cc1c(CC)noc1 CCC(C)CCC(=O)NCC(C)(C)OCCNC(C1C(C)C1(F)F)=O c1(NCCCN(C(=O)C(C2CCCCC2)O)C)ncnc(Cl)c1F N1(C(CC(C)c2ccco2)=O)CCN(C(=O)CCn2ccnn2)CC1CF C1(C(N(C(CNC(=O)Cc2cscn2)C2CC2)C)=O)COc2ccccc2C1 CCC(C)C(C)C(=O)N1CC(NC(=O)C(c2ccccc2F)F)C(CO)C1 N1(C(C23C(C(N)=O)(CCC2)C3)=O)CC2CCC(C1)N2C(c1cc(F)cc(Cl)c1)=O Cc1ncn2ccc(C(N3CCCC3CN(C)C(c3csc(Cl)c3)=O)=O)cc12 C(=O)(CCCCNC(=O)CC12CCCC1C2)N1C(CCC(=O)NC)CCC1 C1(NC(c2cccnn2)=O)CN(C(c2cnc(Br)s2)=O)CC12CCC2 Cc1n[nH]cc1C(=O)NCC1CCC(C(=O)NC2(C(C)O)CC2)O1 N1(Cc2cn(CC(N)=O)nn2)CCN(C(c2cncc(-n3ccnc3)n2)=O)CC1 C(CC(C)C(=O)NCCCCCNC(C1CCCN1N=O)=O)=CCC c1(C(=O)NC(CN(C(=O)Cc2csc(C)c2)CC)C)cn(C)[nH]c1=N c1(CN2CCN(CC(=O)Nc3c(OC)nccn3)CC2)ncccc1C#N C=C(C)CCC(=O)NCC1(F)CCC(NC(=O)C=CC)C1.C(C)(C)C C12(OC)CCC(C(=O)NC3CC4CC3CN4C(c3ncc[nH]c3=O)=O)(CC1)CC2 C(=O)(C(=O)C(C)CC)N1CCC(NC(c2ccc(CCC)cc2)=O)(CF)C1 Cc1ccc2snc(C(=O)NCC3CN(C(C4CCCS4(=O)=O)=O)CC3C)c2c1 Cc1cncc(CC(=O)NC2CC(Cn3cc(-c4ncccn4)nn3)C2)n1 C1(C(C)=O)CC(C(N2CC(CCCCNC(=O)CSC(=N)N)C2)=O)C1(C)C C1(NC(C(CC=C)C)=O)C2CCCC1CC(NC(=O)COC(CC)CC)C2 c1(C(=O)NCC(n2cc(-c3ccon3)nn2)C)ccc(OCC(F)F)cc1 c1(C(=O)NC2CC2C)ccc2c(c1)CCCS2.c1(C=O)cc(C(F)F)ccn1 C(=O)(CCS(=O)(=O)c1ccccc1)N1CC2CC(NC(c3cc(O)no3)=O)C2C1 CCCC(N(C)N1CCC2(COC(=O)N2)C1)C1CCC1 C(=O)(C(C)(C)C1=CCSCC1)NC1CN(C(c2cncc(C)n2)=O)C1 N1(C(C(C)n2ccnc2)=O)CC2(CCN(C(C3Cc4ccccc4S3)=O)CC2)C1 C1(C(N(C)CC2CC(F)CN2C(C2COCCO2)=O)=O)CCC(F)(F)CC1 c1(C(N(C(C(CC)C)C(=O)NCC2(COC)CC2)C)=O)n[nH]c2ccccc12 C1(CCC(=O)NCC(COCC)O)CCCCN(C(=O)Cc2cc(C)on2)C1 N(S(=O)(=O)N1CCC(O)C1)(CCC)CC1CCCCCC1 CC1CN(C(=O)C(C)(C2CC2)N(C(=O)Cc2ccoc2)C)C(C)C1C c1(C(N2CC=CC(NC(c3c(C)nc(CCC)o3)=O)C2)=O)c(C)ccc(Cl)c1N N1(C(c2nc(C)oc2)=O)CCCC(CNC(c2nnn(C)c2C)=O)C1 c1(C(=O)NC2C(NC(c3cc(C4CC4)ccn3)=O)COC2)cnn2c1OCC2 N1(C(CCC=CC(C)C)=O)CC(NC(C2CCCC2C(C)C)=O)C2(CCC2)C1 c1(CNC(c2cnn(CF)c2)=O)cccc(-n2cc(CC3CCCCO3)nn2)c1 C(C)(C)(CC(=O)N(CCC(=O)NC1CC1)C)N(C(Cn1c(C)nnn1)=O)C C1(O)(CNC(c2ncsc2Br)=O)CCCN(C(C2CC(=C3CC3)C2)=O)C1 CC1CN(C(=O)CC(C)P(C)(C)=O)CCCN1C(c1ccc(SC(F)(F)F)s1)=O N1(C(CC2(C=C)CC2)=O)CCC(NC(=O)C(CC)CC=CC)C12CC2 C1(C(N2C(C)CCC2)=O)CN2CCN1C(C)C2.Cc1cc(C2(C(=O)N)CC2)on1 C(c1ccccn1)=C(C)C(N1CCCC1CN(C)C(C1(C2CCCO2)CC1)=O)=O C1(NC(=O)CC2CC(F)C2)CN(C(=O)CCc2ccon2)CC12CCOCC2 C1(NC(CSCCN(C)C)=O)CN(C(=O)CCc2cnc(O)[nH]2)CC12CC2 n1(C(COC)CC(C)C)c(-c2ccc(Cl)cc2Cl)csc1=Nc1cc(C)cc(C)c1 C1(CO)CC(NC(c2cc(CC)on2)c2nnnn2CCC2CC2)C12CCC2 N1(C(c2cc(C)[nH]c2)=O)CC2CCC2(CC(=O)NC2CC3CC3C2)C1 Cc1ccn2ncc(C(=O)NC3CC3NC(c3cccnc3O)=O)c2c1 c1(C(=O)OC)ccc2c(n1)CCN(C(C13CCC1CN(C(=O)C(F)Cl)C3)=O)C2 N1(C(CSC)=O)CCOC(C(C)NC(c2ncsc2-c2ccccn2)=O)C1 CC1COCC(C(=O)NCCC2CN(C(=O)Cn3cccnc3=O)C2)O1 N1(C(CC2C(CC)C2)=O)CCC(CNC(c2nc(C3CC3)cs2)=O)C1 C(=O)(C1=NOC(C)C1)NCC1(NC(C(CCSC)O)=O)CC1 N1(C(Cn2ncc(C#N)c2)=O)CCC2(C=C(C(=O)NCCC(N)=O)C2)C1 CC(C)C(O)C(C)C(=O)N1CCC(C(C)(C)CNC(=O)CC2CCOCC2)CC1 C1(NC(c2n(CC)c(O)nc2)=O)CC(OC)CN(C(c2cc(C(C)C)no2)=O)C1 C1(CNC(Cc2c(C(C)C)con2)=O)(NC(C2CCCCC2O)=O)CCCCC1 C1(NC(Cc2nc(C(C)OCC)sc2)=O)CC2(C1)CCC2.C(=O)C1=CCC1 c1(NC(c2nccc(C)c2)c2nnnn2C2CC(F)(F)C2)cc(Br)c(F)cc1C C1(C2CCN(C(C3CCNC3=O)=O)CC2)(NC(C(CC)COC)=O)CC1 N1(C(C(C)(C)OCC)=O)CCOCC(C)(C)C1.C(=O)C(CC(C)C)N(C)C.N C#CCC(C)(CC)C(=O)N1CC(NC(=O)CSc2ccccc2C)C(F)C1 N1(C(C(CC)(C)CO)=O)CCOC2(C1)CN(C(c1sc3nccnc3c1N)=O)C2 C1(C(N(CCC)CCO)=O)C=CCN(C(=O)C=Cc2cn(C)nn2)C1 C1(C(=O)NC(C(C)C)CCO)CCCC12CCN(C(c1ccc(C3CC3)cc1)=O)C2 C=CCCC(C(=O)NCC1(C)CCCCC1)NC(C1CCC#CO1)=O N1(C(C2(OC)CCC2)=O)CCCC2(CC(NC(=O)C(O)C(C)C)C2)C1 c1(CNC(=O)CCC2CCCN2C(C2CC(O)C2)=O)ncccc1F C1(CNC)CCN(C(C)CN2CCCCC2)CC1 CC1=C(CNC(c2ccc(CNC(N)=O)cc2)=O)S(=O)(=O)CCO1 C(CN=c1[nH]c(Cl)ncc1[N+](=O)[O-])(CC(C)C)NC(c1cc(CC)nn1C)=O CC(CCCOc1cccnc1)N(C(=O)Cn1nccc1N)C1CC1 c1(SC)ncc(C(=O)Nc2cccc(OCc3ccccc3)c2)cn1 N1(C(CONC(C2C(C)CCOC2)=O)=O)CC2(CO)CC2(CO)C1 CCCCC(C(=O)N(CC)CC)NC(N)=O.n1(C(CC(=O)N)C)nc(C)cc1C C(=O)(C1=CCN(C(C2CCC(=O)N2)=O)CC1)NCC1(C#N)CC1 Cc1cc(C)c(CC(N2CCCC(NC(=O)Cn3cccn3)CC2)=O)c(O)n1 C1(C(N(CCCC)C(C)CC)=O)CCCCC1C.n1(CCC=O)ccc(C)n1.N C1(CNC(C=CC)=O)N(C(=O)C(c2cccnc2)OC)CCCC1(C)C Cc1cc(C(=O)N(CCCN(CC(=O)NCC2CCCC2)C)C)ccn1 N(C1c2ccccc2CC1O)C(C1CSCCN1Cc1cccc([N+](=O)[O-])c1)=O c1(NC(=O)NC(CC2CC2)CC2CC2)ncnc(O)c1I n1(CC)ncc(C(=O)NC2CCC(N(C(=O)C=C3CCCC3)C)C2)n1 C1(N(C)C(c2cc(=O)c(Br)c[nH]2)=O)CCCN(C(=O)CSC2CC2)CC1 C(=O)(C(C)(O)C(C)C)N1CC(CNC(c2c(CC)scn2)=O)C(C)C1 N1(C(C(C)(F)F)=O)CCOC(CCNC(c2coc(Sc3ncccn3)n2)=O)C1 C(=O)(CC(C)N(C(=O)COCCNC(C1CCSCC1)=O)C)NC Cc1c(C(=O)NC2CC(C)(NC(=O)CC3CC=CCN3C)C2)cnc2ncnn12 N1(C(c2ccc(C#C)cc2)=O)CCC2(C(N3CCOC(C#C)C3)=O)CCCC12 CC1CN(C(c2cc(C#N)cs2)=O)CC(C)N(C(=O)COc2cnc(Cl)cn2)C1 C1(NC(CN(CCC)C)=O)CN(C(=O)CN2CCCCC2=O)CCC1C(F)(F)F C(=O)CC(C)(C)CN(C)C.C1(C(=O)NC(C2CCC2)C)(CO)CCCO1.N C(CN(C)C)(C(=O)NC1(C(O)CO)CC1)NC(CNC(CCC)=O)=O C1(NC(C(c2ccccn2)C)=O)CN(C(=O)C(C)C(F)(F)F)CC12CCC2 N(C1CC2(CN(C(c3cccc(=O)o3)=O)C2)n2ccnc21)C(c1ccccn1)=O C1(C=O)CC(C)CN(C(=O)CC(C)(C)CN(C)C)C1.C(=O)CC1CC1.CO c1(C(N(c2ccc(O)cc2)CC)=O)cc(=O)c(OC)co1 c1(CC)c(C(N2CC(O)(C(C)NC(=O)C(CC)C)C2)=O)nnn1CC C1(NC(C=C(CC)C)=O)CCN(C(=O)Cc2cccc(Br)c2)CCC1(F)F C1(C)(CNC(COCCOC)=O)COCCN(C(c2nnc3ccccn23)=O)C1 C(=O)(C1CCc2nccn21)N(CCNC(CC(c1c(C)n[nH]c1C)C)=O)C Nc1cc(C(N2CCOCC(NC(=O)C#CC(=O)O)C2)=O)nc2ccccc12 N1(C(c2nnn(C)c2N)=O)CCN(C(C2CCCO2)=O)CC2(C)CCCC12 CC(C)CC(CC(C)C)C(=O)NCC1CC(NC(=O)CCc2cscn2)C1 CN1CC(=O)Nc2cc(C(=O)OCC3CC34CCCCC4)cnc21 CC(C)C(C(=O)NCC(C)CNC(C1CCN(S(C)(=O)=O)CC1)=O)C(C)C Cc1[nH]c(C)c(C(N2CCC(C)(CNC(=O)C(C)Cc3cccnc3)C2)=O)c1C C1(C(N2CC(C#C)(C(NC[Si](C)(C)C)=O)C2)=O)CCCCNC1=O C(=O)(CCC1=CCCCC1)NC1CC(C(=O)NC(C=C)C)C12CCC2 C1(C(N(CC2=CCCOC2)C)=O)CN2CCCC1CC2 C1(NC(c2c(C(C)C)noc2)=O)CC(C)C(O)C1.C1(CC(F)F)(C=O)CC1 CON(CCC(=O)N(C)CC1CCCOC1)C(=O)c1oc(C)cc1C C1(NC(C(CCC)=CCC)=O)CC2CN(C(c3ccccc3CC(C)C)=O)CC12 C#CC1(O)CCCN(C(N2C(C(CNC(C)(C)C)(C)C)CCC2)=O)C1 N1(CC)CCOCC1COC(c1cocc1C(=O)Oc1ccccc1OC)=O N1(C(C=Cc2c(C#N)cccc2)=O)CCCC12CCN(C(=O)CCC1CCC1)C2 C(CC(=O)NO)N(C(COC1(C)CCC1)=O)C(=O)Cc1ccccc1 CCC(CO)(C(=O)N1CC(C(C(=O)NC(c2ncc(F)cn2)C)OC)C1)OC c1(N(C2CCN(CC)CC2)CCC2CNCCO2)nc(N2CCCC2)cc(C)n1 C1(C(CO)NC(CCCSC)=O)CCN(C(=O)Cc2c(C)noc2Cl)CC1 C1(c2cn(CCC=C)nn2)CCCN(Cc2ccc(-c3cn(CC)nn3)cc2)C1 Cc1nn(C)c(Cl)c1C(=O)NCC(CO)NC(=O)C(C)(F)CC1CCCC1 C1(COC)CN(C(c2cnc(CC3CC3)s2)=O)CCN1C(=O)CC1CC1 CCC(CO)(C(=O)NCC1(CO)CN(C(C2CC3(CCC3)C2)=O)C1)OC c1(OC)cncc(C(=O)N(CC)C(C)C)n1.C1(C=O)CCCN1CC(F)F.N C1(NC(C(CC2CN(C(c3c(C)cc(F)s3)=O)C2)F)=O)CCCCC12CC2 C1(C(=O)NC2CC(CC(=O)Nc3c(OC)nccc3)C2)CCCC2(CC2)C1 C12(NC(CCC(C)(F)F)=O)CCOCC1CN(C(=O)CSCc1cccnc1)C2 c1(C(=O)NCC(CC=C)NC(C2CCOC(C)(C)C2)=O)cc2nccn2c(O)n1 c1(C(N(C2CCCCC2NC(=O)CCCF)C)=O)ccc(N)c(Cl)n1 CCC(C)(C)C(O)C(=O)N1CC2CCC(CNC(c3cccc(SC)c3)=O)C2C1 c1(C=O)cc(Cl)cc(Cl)c1O.C(CCC(C)C)NC(C1(CCN(C)C)CC1)=O.N Cn1nc(C(=O)NC2CCCC(NC(=O)CNC=O)CC2)c2ccccc2c1=O C(CC#C)(CC(F)(F)F)NC(=O)NC1(C(=O)OC)CCNCC1 C1(OCC(=O)NC2C(C)CN(C(=O)CC3CCC3)C2)C#CCCCCC1 N1(CCNC(C2CC2C(F)F)=O)CCN(C(=O)CCO)CC1.C1CCCO1 CCCC(C)(C)CC(=O)NC(CNC(c1cccc(OC2CCCC2)c1)=O)CO c1(N2CC(C)C(CNC(C3CC(=O)N(C)C3)=O)CC2)nc2ccc(Cl)cc2s1 c1(SC)cccc(NC(C2CCN(C(=O)Cc3ccc(F)cc3)CC2)=O)c1 C(=O)(CCCC(C)CC)N1CC(C(=O)OC)CC(NC(CNC(CCC)=O)=O)C1 C1(CC)(CNC(c2cn(-c3cccnc3)nn2)=O)CCCC1 N1(C(c2ccc(OC)s2)=O)CC2CC2(NC(=O)CC2CCSCC2)C1 C1(NC(C=CC)=O)CC2CCC(C1F)N2C(=O)Cn1cccn1 C1(CNC(c2ccon2)=O)CN(C(c2cnc3[nH]nnc3c2)=O)CCC1(F)F C1CC(F)CN1C(c1ccc(F)cc1)=O.C1(C(F)(F)F)(C(NC)=O)CCC1.C c1(SCCNC(N2CC(CCC)C2)=O)cc(C)ccc1C C1(c2nnnn2CCCF)(Nc2cc(C)c(Cl)s2)CCN(C)CC1 c1(C(N(C(C)CNC(c2cccnc2F)=O)C)=O)nc2c(s1)COCC2 C1(CN(C(C)C)C)CN(C(=O)C(C)c2ccsc2)CCCO1 N1(C(c2c(NC)nc(C)cc2)=O)CC(NC(=O)C(F)C2CCCC2)CC(F)(F)C1 C(C)(CO)(CS(C)(=O)=O)NC(c1ccc(C(C)(C)OC)cc1)=O CC1CCN(C(=O)CCc2cnco2)CC1N(C(=O)CCCc1n[nH]c(=N)s1)C Cc1ccc(C(=O)NCC2(CNC(=O)CO)CCCC2)o1.C1CCCOC1 Cn1nc(CNC(=O)NCC2CC23CC3(F)F)cc1C#N N1(C(C(C2CCCCC2)(C2CC2)NC(C)=O)=O)CCc2cc(O)ccc2C1 N1(C(C2CN(C(CCC)C)C(=O)C2)=O)CCC(CC)(NC(c2cnsn2)=O)CC1 c1(NC(=O)C(=O)NC2CN3CCC2C3)ccc(OCC(F)(F)F)c(F)c1 C1(C(=O)NC2CC(N(C(c3c(C)nn(CCO)c3)=O)C)C2)CCCC2(CCC2)C1 Cc1cnc(C(=O)NC2CCN(C(C3CCCC(CF)C3)=O)CC2O)cc1Cl c1(NC(N2CCN(C(C3CC=CCC3C(F)(F)F)=O)CC2)=O)c(Br)ccnc1Br Cc1ccc(C(=O)NC(C)C(C)(C)C)c(F)c1F.C1(C=O)CCN(C)C(C)C1.N N1(C(C(C)OCCN(C)C)=O)CCCCC(O)C1.C1(C=O)C2CC3C(C2)C13.N C1(NC(C(C)c2cccs2)=O)CC2CCC1N2C(c1cc(Cl)cs1)=O c1(N2CC(CCC)OCC2)nc(NC(c2ccnn2C)C)c2cnn(C)c2n1 CN=c1[nH]c(=NCc2cccc(Br)c2F)[nH]c(=NC(C)COC)[nH]1 C12(C(=O)NCC(C3CCC3)NC(Cn3nnc(=N)[nH]3)=O)COCC1C2(F)F c1(C(N(CCCOC)C)=O)cccc(-n2cc(C(N3CCOC3=O)(C)C)nn2)c1 C(=O)(CC(C)C(F)F)N1CC(COC)(C)C1.C1(C#N)(C(=O)N)CC(C)C1 N1(C(=O)CCC2CCCO2)CCC2C(NC(C3CC(CF)C3)=O)C2C1 Cc1cncnc1C(=O)NCCC1CCN(C(c2cc(C)n(C(C)C)n2)=O)C1 c1(C(N(CCN(C(C(F)=CC)=O)C(C)C)C)=O)cn(C2CC2)nn1 C1(C)(CNC(C(COC)C)=O)CCCN(c2nc(Cl)c(C(=O)OC)s2)C1 C#CCC(C)C(=O)N1CCC1CNC(C1CC(O)(C(F)(F)F)C1)=O Cc1nc(C(=O)NCC2(F)CN(C(C3CCOC3(C)C)=O)C2)n(C)n1 N1(C(c2cc(CC)no2)=O)CC(OC)CCC1.c1(CC=O)cnc(C2CC2)[nH]1.N N1(C(C(C)S(C)(=O)=O)=O)CCN(C(c2cn(C)nc2C2CCC2)=O)C2(CCC2)C1 CCC(C)C(=O)N1CCCC1CCCNC(=O)C(C)NC(=O)C(C)(C)C C1(CNC(c2cc(C)nnc2)=O)CN(C(c2cc(CO)oc2C)=O)CCN1C N(C(=NCCC(C)C)NCc1cnc(C)cn1)CC1CCN(S(CC)(=O)=O)CC1 N1(C(CCSC)=O)CCOC(C(=O)N(C2CC3(CCC3)C2)C)CC1 C(=O)(C(C)(C)C(N)=O)N(C1CCCN(C(C2CSCN2CC2CCC2)=O)C1)C N1(C(c2c(C(C)=O)ccs2)=O)CCCN(C(C2CCCCO2)=O)CCC1 C(CCF)(C(=O)NCC(CO)C(C)C)NC(c1n(CCC)ccc1)=O c1(C(=O)NCC2(C)CCN(C(C(CC3CC3)OC)=O)C2)[nH]nc2cnccc12 CC1CN(C)CC1NC(=O)C(C)(C)CNC(=O)CCN=[N+]=[N-] Cc1cccc(C(N)C(N2CCN(C(C)C(=O)Nc3cccc(C)c3)CC2)=O)c1 c1(C=O)ccccc1CCC.N1(C(C(=O)NCCOCCCC)=O)CCC1.C n1(CC)nnc2c(NCC3CN(C(=O)C(C)=C4CCC4)CC3C)ncnc12 N1(CC)CCCCC1C(=O)NC1CCC(N(C)C(C2C=CCS2)=O)CC1 c1(NCC(CN(C(C(C(C)C)NS(C)(=O)=O)=O)C)O)ncnc2[nH]c(Cl)cc12 C(=O)(C(C)(C)CCC#N)NCC(C(C)C)NC(=O)C=CSc1nc[nH]n1 N1(C(=O)Nc2cccc(OCC)c2)CCN(C(c2ccccc2)=O)CC(F)(F)C1 c1(OC)ccccc1CC(N1CC2CC2(C(=O)NCC2(Br)CCC2)C1)=O C(CCS(=O)(=O)c1cccc(C)c1)NC(=O)NC1CCN(CCC)C1 Cc1onc(-c2cccc(F)c2)c1C(=O)NCC(C)CO.C(=O)(CCC1CC1)N c1(OC)cc(C#N)ccc1OCC(=O)NCCCO.C1(C=O)CC(F)C(=O)N1 c1(SC(C(N2C(C3(C(=O)N)CC3)CCC2)=O)CC=C)ccc2nn[nH]c2n1 Cn1cnc2cnc(NC3CC(NC(C4CNC(=O)N4)=O)C3(C)C)nc12 N1(C(c2c(C)onc2CO)=O)CC(n2cc(CCc3nn[nH]n3)nn2)CC(C)C1 CC1CCc2[nH]c(=NCC(=O)N3CCOCC3)[nH]c(=NCC(F)(F)C(F)F)c2C1 N1(C(CCCN(C(C)=O)C)=O)CCC(C)(CNC(=O)COC2CCCCC2)C1 N1(C(C2CC(OC)(OC)C2)=O)CCC2(CC2NC(=O)Cc2cc[nH]n2)C1 C1(C2(O)CN(C(C3(O)CC3)=O)C2)(CNC(C2CCc3cncn3C2)=O)CC1 C1(CNC(c2ccc(Cl)cc2)CO)C(O)C2CNCC12 C(=O)(C(C(C)C)NC=O)N(C1(C(N(CCOC)C)=O)CC1)C c1(C=O)cc(=O)c2ccc(Cl)cc2o1.CC1CC1CC(=O)NCC1(C)CC1 c1(C(=O)NC(C(=O)OCC)c2ccoc2)nc(S(C)(=O)=O)n2ccccc12 c1(CC)cc(C(=O)NC2CCC2NC(C2(C)CSC2)=O)nn1C C1(=CC(=O)N(C)CC2CCCC(NC(C(C)NC=O)=O)C2)CN2CCC1CC2 C(CCC(C)(C)C(=O)NCC(C1CCC1)NC(c1cncc(F)c1)=O)OC.O C1(C(N2C(CN(C)C(c3cc4c([nH]3)CCC4)=O)CCC2)=O)CCCC2(CC2)C1 Cc1cc(F)cc(C)c1C=O.C1CN(C(=O)C=CC=O)C(C)(C)C1.C1CC1 CCC(CC(=O)NC1CC(CNC(=O)C)C1)C(C)C.c1cc(F)cc(Cl)c1.O C#CCCCC(C)C(=O)N(C1CC2CCC(C1)N2C(=O)C(C)(F)F)C C1(NC(N2CC3CCC3C2)=O)C2CCOC2C12CCCC2 c1(CC)cc2c(N3CCC(C)(NC(=O)C(C4CC4)OC)C3)nc(C)nc2s1 Cc1ccccc1CN1CCOCC1C.N12CCCC(C1)NC(=O)C2=O c1(C(=O)NCC2CC(NC(C3OCC(C)C3)=O)C2)coc2cc(F)ccc12 c1(C2C(C(NCCNC(c3occc3Cl)=O)=O)C2)ccc(C)c(C)c1.CC C1(N(C(COCCCCC)=O)C)CN(C(=O)CC2(C(F)(F)F)CCC2)CC1O C1CCn2nnnc2C1.c1(OC)nn(C)cc1C(=O)NC(C)(C(=O)N)C1CCC1 C1(C(N2C(C)CCC2)=O)CCCS(=O)(=O)C1.Cc1cc(C)c(CC(=O)NC)s1 N(C1CCC(NC(C23CCC(C)(CO2)C3)=O)c2ccccc21)C(C(=O)N(C)C)=O c1(OC)ccc(C=CC(=O)NC)cc1F.C1CN(C(=O)C)CCC1C.C(C)=O C1(C(=O)NCc2c(C)cnn2C)CCC(C)(C)C1.n1(CC=O)cnnc1O.N C12(NC(c3c(C)nc(CO)s3)=O)CCCN(C(=O)COC(C)(C)C)C1C2 O=C1CCC(N2CCC(NC(=O)NC3CC4CCC(C3)N4)CC2)C2(CCC2)N1 N1(c2ncnc3ncn(C)c32)C2C=CC1c1ccccc12 C1(COC(c2ccc(C(F)(F)F)c(O)n2)=O)CCC2COCCC2O1 N1(C(C)=O)CC2(CCC2)CC1C(=O)NC1CC(CF)C1 N1(S(Cc2cccc(C)c2)(=O)=O)Cc2ccc(CN3CC(C)OCC3C)cc2C1 c1(C(=O)NC(CC(C)NC(CCCOCC)=O)C)ccc2nccnc2c1 C(=O)(CC(C)(C)CNC(c1cn(C)c(=O)cn1)=O)NC(C#C)CC Cc1cc(CC2CCC(NN(c3cc(N(C)C)ncn3)C)CC2)n(C)n1 C(C)(C(C)(C)C(=O)NCC(C)(C)C(C)(F)F)NC(CC(COC)C)=O c1(N2CCC(C)SCC2)nc(NCC(=O)N(C)C)c2c(ncn2C)n1 N1(C(C2N(C(CC(C)C3CC3)=O)CCSC2)=O)CCC12CCCSC2 C1(CNC(=O)CCc2cccs2)CN(C(c2ncc(F)cc2F)=O)CC12CC2 c1(CC(=O)NCC(CN(C(CCOCC(C)C)=O)C)O)cccc(F)c1O C12(C(=O)NC(CC#C)CO)CCCC1CCN2C(=O)CC(C)(C)OC N1(C(C(=Cc2ncn(C)c2)F)=O)CCC(NC(=O)CCF)C(CO)C1 c1(N(CC)CC)cc(NC(C2CC(C)(C)CCC2O)=O)ccc1[N+](=O)[O-] c1(C(N2CC(F)(CNC(CC3CC(OC)C3)=O)C2)=O)ccccc1.CC.O C1(CC(=O)NCC2(OCC)CC2)C2CN(C(=O)C(C)N(C)C)CC12 N1(C(c2c(C)cc(F)cc2)=O)CCN(Cc2c(C)nn(C3CC3)c2Cl)CC12CC2 C1CCS(=O)(=O)C12CN(c1ncccc1S(C)(=O)=O)C2.C(CC(=O)N)NC(C)=O N1(C(C(C2CC2)SC)=O)CCC(OCC(=O)N(C)Cc2cc(C)on2)C1 N1(C(c2c(Br)ccc(C#C)c2)=O)CCCC(C2CCC2)CC1 C(C)(C)(CC(=O)NC(C1CCN(C(=O)CC2(O)CCOC2)CC1)CO)SC N1(C(c2c(C)c(Br)no2)=O)CC(NC(=O)Cc2cncn2C)CCC1C C(C(=O)O)(C(=O)NCCCC(C)NC(c1nc(Br)c[nH]1)=O)OC.C(C)(C)C C#CCC(CC#C)C(=O)NC(c1ccccc1)CNC(C12CCC(CC1)OC2)=O C(=O)(C1=CCCCC1)N1CCC(C(N2CCC(O)(CC)C2)=O)(OC)C1 N1(C(=O)C(N2CCC(c3ccco3)C2)=O)CCCCC1 N1(C(c2n(C)cc(Cl)c2)=O)CCCC2(CC(NC(C3(C)CCC3)=O)CO2)C1 N1(C(C(C)NC(c2ccco2)=O)=O)CCCC2(NC(=O)C3=COCCO3)CC2C1 C1(C(=O)NCCC(Cc2ccccc2)NC(C2(C)CCC2)=O)CCC2(CC2)C1 N1(C(CC2N(C(Cc3c(C)n[nH]c3C)=O)CCC2)=O)CC2CC=CC1C2 c1(NCCNC(C)=O)ccc(S(=O)(=O)NC2COC3(CCC3)OC2)c(Br)c1 c1(C2C(NC(C(C3CC3)NC(C)=O)=O)C2)ccc(OC(F)F)cc1 c1(COCC)nc(C)cc(=NC(C)C2CCN(C(=O)C(C)C3CCOC3)C2)[nH]1 c1(OC)ccc(C(N2CCN(C(C3CC34CCC4)=O)C(C3CC3)C2)=O)c(Cl)c1 c1(C(N2C(C(=O)Nc3cc(Cl)ccc3F)CC(O)C2)=O)c[nH]c2ccc(Br)cc12 N1(C(C2CN(C)C(=O)N2)=O)CCN(C(C2CC(F)C2)=O)C(CO)C1 c1(C(N2CCCC(N(C(CSCC=C)=O)C)C2)=O)ncc(Br)cc1O Cc1[nH]c(C(=O)N(CCCNC(C2CCCC23CC3)=O)C)c(C)c1[N+](=O)[O-] C1(C(N2CCC(C(=O)NOCCOC)(CC#C)C2)=O)CC(C)(C)CCO1 c1(C(=O)OCC)cc(S(=O)(=O)N2CCC(C#N)C2)ccc1F.C1(C=O)CC1F c1(OC)cc(Cl)c(Br)cc1NC(=O)CN1CC(O)(c2ncnn2C)C1 C(=O)(C1CCSc2ccccc21)NC(C(C)NC(=O)C(F)(F)CN(C)C)CO CCCCCC(C)CC(=O)NCCC(C)(CC)NC(C12CC(F)(C1)C2)=O C1(C(=O)NCC2(C)CC23CCC3)Cc2cccnc2C1.C1(C=O)CCCCS1.N Cc1nc(F)ccc1CNC(=O)C(Cc1cn[nH]c1)NC(=O)C#CC(C)C C1(NC(C2N(C(C3C(OC)(OC)CC3)=O)CC=C2)=O)CC12CCCCC2 C(=O)(CCS(C)(=O)=O)NCC1(C=O)CC(=C)C1.c1(CC)ccc(C)cn1.N C1(C=O)CC(F)(F)CN1C(c1ccco1)=O.C(=O)(C)N(C1CC1)CC.N C1(NC(c2c(CNC(C(C(C)(C)C)OC)=O)ocn2)=O)CCn2nnnc2C1 C1(C(=O)NCC(C)CNC(=O)CN2CCOCC2)CCC(C2CC2)C1 c1(OCC)ccc(C(C)N(C)C(C2CN(Cc3cc(SC)oc3C)C2)=O)cc1 C1(NC(c2cnn(CCO)c2)=O)CCC2CCN(C(=O)CSC3CCCOC3)C12 CN1CCC2C(CCN2C(C2CC2c2cn(C)c3ccccc23)=O)C1 N1(C(CSC(C)C)=O)CC(C)(C)OC2(C1)CN(C(=O)C=C1CCN(C)CC1)C2 c1(NC2CCCN(C(=O)CC3CCCOCC3)C2)ccn2ccnc2n1 CCC(CCCC(=O)N1CCC=C(F)C1)NC(=O)COCC1CC1 C1(C(=O)NC)CCN(C(=O)C(CCC2CC2)NC(=O)CCn2ccnn2)C1C CC(C(F)C(=O)NC1CCN(c2ncccn2)CC1)C(F)(F)F c1(C(N2CCCC(C3(C)COC(=O)N3)C2)=O)cccc2c(I)n[nH]c12 C(C)(CCC(=O)NC1(C)CC(NC(=O)CCC2CC2(Cl)Cl)C1)OC CC1=CC(NC(C2CC(=O)CN2C(c2n[nH]cc2Cl)=O)=O)CCC1 N1(C(=O)Cc2ccccn2)CCC2(CC1)CCN2C(=O)C=Cc1cccc(O)c1 C12(COCC)CC(C=O)(CO1)C2.C1CN(C(=O)CCC2(C)CC2)CC1 c1(CC(=O)NC2CC(NC(=O)Cc3ccns3)C2)ccccc1[N+](=O)[O-] C1N(C(C2CC=C(C)CC2)=O)CCCC1(C)C.c1(C(C)=O)cc(C(=O)NC)cs1 N1(C(C(c2cc(C)sc2)(C)C)=O)CC2(CC(NC(=O)Cc3nccn3C)CO2)C1 N1(C(CC2C(C)C2)=O)CCCC2(NC(c3cccc(F)c3)=O)CC2C1 C12(NC(=O)C=Cc3ccc(Cl)s3)CCC(C1)N(C(=O)Cc1ccc(O)nc1)C2 CCS(=O)(=O)c1nc2ccc(NS(=O)(=O)c3cc([N+](=O)[O-])ccc3Cl)cc2s1 C1(CC(N2CC(=C(C)F)C2)=O)CCCC1C.C1(C(=O)OC)(C(=O)N)CC1C Cc1ccc(C(c2nc(-c3nccs3)nn2CC2CCCO2)C(C)C)cc1 c1(OC(C)C(=O)Nc2ccnn2CC(F)(F)F)ccc(Cl)nc1 C(=O)(C(C)(C)CC(F)(F)F)NCC(C)(Cn1cccn1)OC N1(C(c2ccc(C(C)=O)cn2)C(=O)NCCCC2CC2)CCCC(C)CC1 C1(C(=O)NCC(CNC(C2(COC)CCCC2)=O)OC)COCCN1C=O C1(NC(C=COCC)=O)CCC2CN(C(c3cc(Cl)cn3CC)=O)CC2C1 n1(CC)cnc2c(N(CCC(C)(C)C)C)nc(N3CCC(COC)(OC)C3)nc12 CCCCC(O)C(C)C(=O)NCC1CC1CC(N1CCCC2(CCOC2)C1)=O C(N=c1[nH]cnc(C)c1OC)C1CCC(NC(C(CCCOC)C)=O)CC1 C1(C(C(=O)NC2CC2)N(CCCC(=O)OCC)CC(=C)C)CC2C=CC1C2 C1(C#CC(=O)N2CC=C(C(=O)NCC3(C)CC(C)=NO3)CC2)(CC)COC1 C(=O)(C1=COCCO1)N(CCCCCCNC(C(C(C)C)OCC(C)C)=O)C C(c1cc(F)cc(F)c1)=CC(=O)NC1CC1C.C1(C=O)CCCCS1(=O)=O c1(CC)cc(C(C(=O)NCC(F)F)N(CC(F)F)Cc2ccccc2)n(C)n1 N1(C(=O)CC2CCN(Cc3cccc(F)c3I)CC2)Cc2ccncc2C1 c1(COC)nc(-c2ccn(CCF)n2)n(C2CCS(=O)(=O)C2)n1 c1(C(=O)NC2CC(CNC(C(COC)C)=O)C2)cc([N+](=O)[O-])nn1C Cc1ncc(C(=O)NCc2cc(C(=O)NC3COCC3C)on2)cn1 CCC(C)(CO)C(=O)N1CC2CCC2(NC(c2ccc(OC)c(C)c2)=O)C1 N1(C(=O)Cc2cc[nH]n2)CCOC2(CCC(NC(C3(CO)CC3)=O)CC2)C1 N1(C(c2c[nH]c3ccc(C#N)cc32)=O)CCCC(C2CNC(=O)C2)C1 CC1CCCN(C(C2OCCO2)=O)C1CCNC(=O)CCn1ccccc1=O c1(C(=O)NC(CNC(c2c(C)cc(O)nc2)=O)C)c[nH]c(C)c(Br)c1=O c1(CN(CC(C)Cn2cccn2)C=O)ccnn1Cc1ccccc1 C1(C2CCCN(C(=O)Cc3cncnc3)C2)(NC(C2CC23CCOCC3)=O)CC1 C(C(C)C(=O)NC1(CO)CN(C(C2CN(CC(F)(F)F)C2)=O)C1)OC C(=O)(CCC(C)CN(C)C)N(CC)CC.c1(C=O)csc(-c2ccncc2)n1.N C(=O)(C(C(C)C)O)NC(C1CCCCC1)CNC(C=C(CC)C)=O.CC(C)C C1(NC(c2cc(OC)n[nH]2)=O)(CO)CCN(C(=O)C(C)CO)CC1 C12(C=O)CCC(C#N)(CC1)CC2.C#CCC(C)(C)C(=O)NCCC1(C)CC1 CC1(CNC(=O)CCN(C)CCO)CCN(C(=O)Cc2ccccc2Cl)CC1 CC1(NC(c2cnc(Cc3ccc(F)cc3)nc2O)=O)CCN(C2CC2)CC1 n1(CCC(=O)OCC)nnnc1C(CC1CCCCO1)NCC1CCC1C C1(C(N2CC(C)(CO)C(O)CC2)=O)COC2(CCN(C(C3CCC3)=O)CC2)C1 C(=O)(C1=CCCOCC1)N1CCC2(C(C(N(C3CCOC3)CC#C)=O)C2)C1 N1(C(C(C)SCCCC)=O)CC(NC(C2CC(F)(F)C2)=O)C(C(F)F)C1 C1(C(N2CCC(N(C)C(=O)NCc3n[nH]c(=N)s3)CC2)=O)Cc2ccccc2O1 C1(NC(c2cn(C(C)C)nc2)=O)CN(C(=O)C=Cc2nnn(C)n2)CCC1(C)C c1(-n2cc(CNCC3(C(=O)O)CC(=C)C3)nc2)cc(C)ccc1OC C1(O)(CCNC(C(C)NC=O)=O)CCN(C(=O)CC2CCC(O)C2)C1 C1(NC(CCc2ccn(C)c2)=O)C=CCC(C(N2CC(CO)C(O)C2)=O)C1 CC(CNC(=O)CCC1CCCN1C(c1ccc(CO)o1)=O)S(N)(=O)=O c1(C(N2CCC(C)(CNC(C(COC)COC)=O)C2)=O)cc2ccccc2s1 Cc1cc(C(N2CCOC(C)(CNC(c3cc(C)sc3C)=O)C2)=O)nc(O)n1 C1(CNC(C(CC)SC)=O)CC(C(=O)NCC2(O)CCN(C)C2)=NO1 C#CCC(C)(C(=O)N=c1cc(SC)n(C)[nH]1)NC(=O)C(O)C(C)(C)CC C1(C(=O)NCC(CC(=O)NC(C)C(F)(F)F)O)CCC(C)(C)CC1 N1(C(CCC2N(C(C(C)CO)=O)CCCC2)=O)CCCC(C2CC2)CC1 c1(C=O)c(C(C)C)nn(C)c1Cl.c1(CCC)nsc(N)c1C(=O)NC1CCC1 Cc1cn2c(n1)CC(C(=O)N(CC(O)C)C)C2.c1(C(=O)N)cn(C(C)C)nc1C c1(CC(=O)N)cncc2ccccc12.c1(OC)cc(C(N2CC(F)(C)C2)=O)on1 C(=O)(C(C#N)C(C)(C)C)NC1CCN(CCCNC(C2N(C)CC(O)C2)=O)C1 C(=O)(C1CCCc2n[nH]cc21)NCCc1cccc(C)c1C C(c1ccccc1)=C(C)C(=O)N(CCNC(=O)CC1CC(C)=NO1)C(C)C c1(NC(C)=O)cccc(C(=O)N(CC(C)C)C)c1C.C1(CC(=O)N)CCCCC1 c1(C(=O)NCCC(C)NC(C(CC)CC)=O)ccc(C#N)c(F)c1Br c1(C(CC)O)nnc(N(C)CC2(O)CCOC2)n1CCOCc1ccccc1 Cc1cccc(F)c1NC(=O)CC1CCN(C(c2ncc(Cl)cc2Br)=O)C1 CCC(C)C(O)C(=O)NC1CC(CCn2cc(C3(O)CCC3)nn2)C1 N1(C(CC=C=C)=O)CC(NC(=O)Cc2ccc3sccc3c2)CC2(CC2)C1 C1(NC(=O)CCCN2CCCCC2)CC2CN(C(=O)C=CCO)CC2C1 C12(C(=O)NC3C(NC(C4CC(=C)C4)=O)C3)CC3CC(CC(C3)O1)C2 c1(C(=O)NC(CNC(c2c(C)c[nH]n2)=O)C2CC2)cccc(-n2cncn2)c1 C1CCN(C(=O)CC2CC=CCN2C)C(C)C1.C(CC(=O)NC)NC(=O)NC C12(NC(Cc3nnc(C)s3)=O)CCCC1N(C(=O)CN(c1ccncc1)C)CC2 N1(C(C23CC(NC(C(C)C(F)(F)F)=O)C(OC2)C3)=O)CC2CSCC2(C)C1 c1(N(CCC#N)C)nc2ccccc2nc1NC1CC(F)(F)C1 c1(OC)cncnc1C(N1CC(NC(C2OCCO2)=O)CC1C)=O Cc1csc2ncc(C(=O)NC(C)CCCNC(C3CCN(C)C3)=O)n12 C#Cc1cnn(C)c1C(=O)NCC1CCN1C(C1(CO)CCOCC1)=O C1(C)(C(=O)NCC(N2CCCC2)C)CCCN1C(=O)C1=CCSC1 c1(C(=O)OC)cnc(N2CCC(C(=O)NCC(=O)NCC3CC3)C2)nc1 C1(N(C(CCCOC(CCC)=O)=O)C)CCCC(N(C)C(C2=C=C=NC=C2)=O)C1 N1(C(c2cc(C)[nH]n2)C(=O)NCCC2(C)CC2)CCOCC1C C#CCC(C(=O)NC1(CCOC)CC1)NC(c1cc(C(C)C)no1)=O c1(CN2CC(C(=O)Nc3c(C(=O)OCC)n[nH]c3)C2)ccc(OC)cc1Br C(=O)(C1CCCc2cncn21)NCC1OCCN(C(C2CC(C)=C(C)CC2)=O)C1 N1(C(C)C(=O)NC2CC2)CCCN(C(=O)C(C)(N)CF)CC1 C(=O)(C1CCc2snnc21)NCC(CCC)NC(C1(C)CCCOC1)=O C1(NC(c2c(CC)cno2)=O)CC(C(=O)NCCCN(C)C)C12CCC2 c1(C(=O)OC)c[nH]c(=NCCC2CCCO2)cc1C(=O)OC c1(CC(CC)NC(C)(CCN2CCCCC2)c2nnnn2C)cccc(C)c1 C1(CN(C(=O)CCN2CCCC2)C)CCN(C(=O)CN(c2ncccn2)C)CC1 C1(C(=O)NC(COC)C(=O)NCCOC2CC2)CC(O)C(F)C1 C1(NC(CN(C)C)=O)CC2CC(C1)CN(C(=O)CCC1CCCC1)C2 N1(C(c2cc(C)n(C)n2)=O)CC2CCC(C1)C2NC(=O)C(O)CC(C)C C#Cc1cc(F)cnc1NC(C1CCCC(NCc2c[nH]ccc2=N)C1)=O c1(C(=O)NCC(C2CCOC2)NC(c2cc(C)nn2C)=O)cccc2ccnn12 c1(C(N(CC(C)NC(c2c(C)cco2)=O)C)=O)ccc(S(C)(=O)=O)s1 CC1CN(C(=O)C(C)Sc2ccccc2)CCN(C(c2nccnc2N)=O)C1 C1(SC)CN(c2nc(CC(F)(F)F)no2)CC1n1cc(C(C)(C)O)nn1 c1(C(N2CCCC(N(C(CCC(=C)C)=O)CC)C2)=O)cnc2c(c1)COC2 C1(CC(=O)NCC(CNC(C(C)=CC)=O)C)(OC)CCOCC1 C12(NC(CCCOC)=O)CCCN(C(=O)CSc3ccc(C)c(C)c3)C1C2 c1(C(N2CCC(CCNC(C3(C#N)CCC3)=O)C2)=O)cnc(O)c(Br)c1 C1(O)(C(=O)NCC(CNC(C2C(OC)CCC2)=O)(C)C)CC(F)(F)C1 C(CCCC(F)(F)F)NC(CC1CCC(NC(=O)CC2CC2CF)C1)=O C1(NC(c2cccc(C)c2)=O)CCC2(C1)CN(C(c1ccnc(C)n1)=O)C2 C(=O)(CCCCNC(C1CSCC(=O)N1)=O)N1C(C(=O)OC)CC1C C1(C(=O)NCCC2(OC)CN(C(C=CCOC)=O)C2)CCCCC1(C)C Cn1c(C(=O)NC2CC(NC(c3cc(Cl)cc(Cl)c3)=O)C2)cc2sccc12 N1(C(C(C)O)=O)CC2(C1)CN(C(c1cc3c([nH]1)CCC(C)C3)=O)CCO2 N1(c2n(C)ccn2)CCCN(C(=O)NC2(c3nccc(O)n3)CCC2)CC1 c1(SC)cc(C(=O)NCC2CCCN(C(C3CC(C)(O)C3)=O)CC2)ccc1F C#CCC(CC(F)F)NC(=O)C(C)(C)CN(C)C(c1cc(C)[nH]c1C)=O C1(OCC)CCCCC1NC(=O)CCCCN(C)C(c1coc(C)c1)=O N#Cc1cc(S(=O)(=O)N2CC3CCC3C2)ccc1N1CCN(CCCO)CC1 CCC(C)(C)C(O)C(=O)NC1CN(C(=O)C(C)(C)CN(C)C)CC1(C)C.NC C1(C)(NC(CCC(C)NC(c2cc(=O)cc[nH]2)=O)=O)CC2(CCC2)C1 c1(CC(=O)NC(CN(C(=O)Cc2cnsc2)CC)C)c(C)nn(CC)c1C C(=O)(CCC(C)(C)NC(C1CCC(=O)N(C)C1)=O)N(C(C(=O)OC)C)C C1(NC(c2cccc(Cl)c2F)=O)CCC2CCN(C(=O)CCC[N+](=O)[O-])C1C2 c1(C(=O)NCCNC(C(C(C=C)C)C)=O)cc2cc(Br)cc(C)c2o1 C1(C(=O)NCCCN(C(C)C)C(C2CNC(=O)C2)=O)CCCC(N(C)C)C1 c1(C(N2CCC(C(C)C)(C(=O)O)CC2)=O)cc(F)cc(Br)c1Cl C1(N(C(C=CSC)=O)C)CCCN(C(C2(COC)CCCCO2)=O)CC1 C1(NC(Cc2c(C)noc2)=O)CCN(C(C2(C)CC=CCO2)=O)CCC1(F)F Cc1cn(C)nc1C(=O)NCC1(SC)CN(C(c2n[nH]cc2Cl)=O)C1 O=C(CC(F)(F)C(F)F)NC1CC(F)CN(C(=O)C=Cc2cccs2)C1 CC1(C)CN(C(=O)C(=O)NCC(F)F)CCC1NC(c1ncc[nH]1)=O C=CCC(C(=O)NCCc1ccn(CC)n1)NC(C1CC(F)C1)=O CCC(C)C(C(=O)N1CC(F)(F)C1)N(C)C(c1ccoc1Cl)=O C1(C)(C(N2C(CN(C(CCCOC(C)C)=O)C)CCC2)=O)CCCNS1(=O)=O N1(S(CC=C)(=O)=O)CC(C(=O)NC(c2ccccc2)C(=O)OC)CC(F)C1 C(N=c1[nH]c2c(c(=NC(C)c3cccc4cc[nH]c34)[nH]1)COC2)C1(OC)CCC1 N1(C(c2nc(C)n(C)n2)=O)C2CCCC1CN(C(c1cnco1)=O)C2 c1(C(c2nnnn2C2(C)CC2)NC(CC)(C)COC)cccc(C(C)C)c1.O C(=O)(C(C)(C)NC(c1ccccc1)C(=O)OC(C)C)NC CCCCCCCC(=O)N1C2CCC1CN(C(c1cc([N+](=O)[O-])oc1C)=O)C2 Nc1cnc(Br)cc1C(N1CC(Cc2ccccc2Cl)C1)=O N1(C(C2C(C=C)CC2)=O)CCN(C(=O)Cc2ccc(F)cc2C)C2CCCC12 c1(C(=O)NCCCCC(C)NC(C2(C=C)CC2)=O)cc(C(F)(F)F)ccc1C C1(C(N(C)CCC2CCN(C(=O)C#CC3CC3)CC2)=O)CCC(S(N)(=O)=O)CC1 C(=O)(CC(C1CCCC1)NCC(O)COCCOC)OC C1(C2CC2)(NC(C2C(NC(C3C(C)CC(=O)CC3)=O)CCO2)=O)CCOCC1 CC1(CCO)CCN(C(=O)CCC2CCCN(C(=O)CCn3cccc3)C2)C1 Cc1cc(F)cnc1C(=O)NC(C)(C)CN(C(=O)CCn1cccn1)C CC(CN1CCCCC1)N=c1[nH]c2c(c(=NCC3(C)CC4CC4C3)[nH]1)CCC2 C12(NC(C=Cc3ccc(C)cn3)=O)CCCC1N(C(=O)C=C1CCSCC1)CC2 CN1CC=C(CCNC(C2COCCN(C(C3CCC(C)(C)OC3)=O)C2)=O)CC1 O=S(=O)(c1[nH]c(=NCC2COCCO2)ccc1Br)N1CCCC(c2cnco2)C1 CC1(C)CC(C(N2CC(CCCCNC(c3cnnc(Cl)c3)=O)C2)=O)CCO1 c1(OC)ccccc1CC(=O)NCC1CC(F)(C)C1.c1(C=O)cscc1.N c1(NC(C)C(=O)NCC)cc(F)c(C=O)c(F)c1.C1CC1.CC.C(N)=O c1(C(=O)NCCCCN(C(=O)CCC2CCCN2C)C)ccc(C2CC2)c(Cl)c1 c1(CC)ncc(Br)cc1C(=O)NCCC1CN(C(c2cnco2)=O)CCO1 n1(CCC)nc(C)cc1C(=O)NCC(O)CNC(=O)CC1CC(F)C1 N#Cc1ccc(C(C2CC2)NC(=O)C(N)CC2CCCCO2)cc1 C1(F)(CNC(c2c(C)ocn2)=O)CCCN(C(=O)CC2CCSC2)CC1 C(=O)(C(C)(C)C(=O)NCCCC)OCC.C1(n2ccnc2)(C=O)CCCC1.N C1(CCNC(C=CSC)=O)CC(F)(F)CN1C(c1ccnc(C(C)C)n1)=O N1(C(CC2C(C)(C)COC2)=O)CCC2CN(C(=O)CN3CCCC3=O)CCC2C1 CC1CCN(C(=O)C(O)C2CC2)CC1CNC(c1cc(C2CC2)on1)=O C(=O)(CN=c1cc[nH]cc1)NC1CC2CC(NC(C3CCN(C)C3)=O)CC2C1 c1(C(=O)NC(C)CNC(C2CN(C)C(=O)N2)=O)cc(P(C)(C)=O)cs1 c1(C(=O)NC2C(CC)N(C(=O)Cn3cncn3)CC2)cc2cc(Cl)c(Cl)cc2[nH]1 N1(C(CC(=O)OC)=O)CCC(C)(CNC(C2(O)CCSC2)=O)C1 C(=O)(C1CCCn2ccnc21)NC1CCC(CN=c2[nH]nc(CCOC)s2)CC1 CCC(c1ccccc1)=CC(=O)NC1CCC(F)C1.S(S(C)(=O)=O)CC=O.C c1(C(c2n(CC=C)nnn2)Nc2ccc(C3CC3)cc2)cc(C2CC2)cc(C)c1 Cc1ncc2n1CC(C(N1CC3(C1)CN(C(=O)CCCC(C)O)C3)=O)CC2 N1(C(c2c(OC)c(C)sc2)=O)CC2(CC(NC(=O)CCc3ncc[nH]3)CO2)C1 C1(C(N2C(C3CC3)CCCC2)=O)CCCS(=O)(=O)C1.c1(C(=O)N)coc(Cl)c1 c1(OC)ncc(C(=O)NC(C)CCC)cc1C(F)(F)F.c1(CC=O)cccs1 c1(C(=O)NC(CC)CNC(=O)Cc2ccon2)cc(C)c(CO)cn1 Cc1nc2c(s1)CCCC2C(=O)NCC(C)CNC(C1(c2ccccn2)CC1)=O Cc1scc(C(=O)NC(CNC(C2C3CCCC23)=O)C2CC2)c1C C(CN=c1cc(C)nc(SC)[nH]1)N(C(CC1C(OCC)COCC1)=O)C1CC1 C1(CNC(CCc2cn(C)nc2)=O)CC12CCN(C(=O)Cc1cccnc1)C2 N1(C(C2N(C(CCC)=O)CCCC2)=O)CCN(C(C2CC2F)=O)C(C(C)C)C1 C(=O)(CC(C)(C)C(=O)N)OC.C1CCN(C(=O)C(C2CCCCC2)N(C)C)C1 N1(Cc2nnc(CC)o2)CCC2(CC1)CC2(C)C(=O)NCC(C)(C)OC C1(OC)CCC2(C(=O)NCc3c[nH]nc3C=O)CC12.C1(CCO)CN(C)C1 N#Cc1cnc2ccccc2c1N1CC(=C(F)CNC(c2cnsn2)=O)C1 CC(F)(F)CC(=O)NC1CCCC(NC(=O)C=CC2CCC2)C1 C1(CNC(C2CC2(F)Cl)=O)CC(F)CN1C(=O)CCCc1nccs1 c1(NCC(F)F)[nH]c(=NCC(CCC(F)(F)F)c2ccccc2)nc2sccc12 C1(NC(C2CC2C2CCCC2)=O)CC2CCC1N(C(=O)CC1CCCCCC1)C2 c1(CC(N2CC(=C(C)F)C2)=O)ccc([N+](=O)[O-])cc1.C1(C=O)CCC(F)C1.N Cc1cnc(C(=O)NC(C)CNC(=O)Cc2occc2C)cc1C#N c1(NCC(c2cnn(C)c2)OC)ncccc1S(=O)(=O)N(C(C)CC1CC1)C CCCC(C(=O)NCC1C(C)C1(F)F)OC.c1(C(=O)N)c[nH]nc1C(F)F c1(C(=O)NCC2CCC2)ccc2c(c1)NCC2.c1(C=O)cc2c(s1)CCC2.N c1(C(N2CC(CC=C)(NC(C3CCNC3=O)=O)C2)=O)c([N+](=O)[O-])cnn1C C1(OCC)CC(CC(=O)N(CC(O)CN(C(=O)C(O)C2CCC2)C)C)C1 c1(CC(=O)NCCN(C(=O)Cn2nc(C)oc2=O)CC)cc(C)ccc1F C1(NC(c2ccnc(Cl)c2)=O)CC2CN(C(c3cc(C(F)F)[nH]n3)=O)CC2C1 c1(C(C(=O)NCCCC)N(C2CC(O)C2)C)cccc(-c2ccncc2)c1 CCC(C)CC(C)C(=O)N1CCC(N(C(=O)CC(CC)C2CC2)CC2CCC2)CC1 c1(C(=O)NC2CC(C)(NC(c3cnc(S)[nH]3)=O)C2)cccc(Cl)c1O C1(NCCN(C(CCCc2onc(C)n2)=O)C2CCSC2=O)CCCS(=O)(=O)N1 C1(CNC(C2(CC)CCCN2C=O)=O)CC(=O)NC1(C)C.C(C)(C)C.O c1(C(N2CC3CC(NC(C4(O)CCSCC4)=O)CC2C3)=O)scc2c1OCCO2 N1(C(C)C)CCN(C(=O)CC2CN(C(c3ccc(C4CC4)cc3)=O)C2)CC1 C12(C(=O)N)CCCC1CS(=O)(=O)C2.CN=c1[nH]cc(C(N2CCC(C)CC2)=O)o1 C1(F)(C(N2CCCC(OCC)C2)=O)CCCN(C(c2sccc2CO)=O)C1 CNS(=O)(=O)NCC(N1CC(CNC(C2CC2C(N)=O)=O)(O)C1)=O C1(NC(C(CCCC)C)=O)C2CC3CN(C(=O)Cc4ccccc4F)C1C3C2 C1(C(N2C(CC)CCCC2)=O)CCCCC(C)(C)C1.C1(C(=O)N)(COC)CC1 C12(NC(=O)Cn3cccn3)COC(C1)C(NC(c1cccc(F)c1F)=O)C2 C1(N(C(CC(CC)C2CCC2)=O)C)CCC2CN(C(C3OCCC3CC)=O)CC12 Cn1cnc2c(N(c3ccc(=N)[nH]c3)C(c3cc4cc[nH]c4cn3)=O)ncnc12 C(=O)(C(F)C(F)(F)F)N(CC(=O)Nc1ccncn1)CC#C CN1CC2C(C(=O)NC(C(=O)NOCC(O)C(C)(C)C)c3cnn(C)c3)C2C1 C=C(C)CC(C)C(=O)N1CCC1CNC(=O)CCc1cccc(C#N)c1 C1(CC(=O)N(CCCC)CC)CC(C)(C)CN1C(c1cn(C)c(C)n1)=O.O c1(C(N2CC(NC(C3C(COC)C3)=O)C(C)C2)=O)cc(N)ccc1Br C12(C(=O)NC)CCC(F)(CC1)C2.c1cccc(Cl)c1.C1C=CCN1C(=O)C c1(CNC(CC(C)F)=O)nc2c(s1)CCN(C(c1ccnc3ncnn13)=O)C2 C1(C(=O)NCc2c(C)cc(F)nc2)CC2CC1CN(C(c1scnc1C)=O)C2 C(=O)(C1=NN(c2ccccc2)C(=O)C(C)N1)N1CCC(OCC)C1C C1(OCC(N2CCC(N(C(=O)C=C(C)C(F)F)CC)C2)=O)CCOCC1 C(=O)(CCC(C)(F)F)N(C(C)CNC(C1(C(=O)N(C)C)CC1)=O)C c1(C=O)cnc2[nH]ccc2n1.N1(C(C(C2CC2)OC)=O)CC(C(C)(C)O)(C)C1 c1(C(C)NC(=O)Cc2cccc(Cl)c2)ccccc1Cl.C1(C=O)CN(C)C1.CC C1(O)(CC)CCN(C(=O)C=Cc2cccnc2)C1.c1(C(N)=O)ccc(C=O)[nH]1.N C(C#N)(C(=O)NCC(C)N(C(=O)CCc1cnn(C)c1)C)=C(C)C CC(C)(CC(F)(F)F)C(=O)N1CC(NC(C2(CCF)CC2)=O)C2CCCCC12 C1(C(N(C(c2ccc(Cl)cc2)COC)C)=O)CCC2(CCNCC2)C1 C1(C(=O)NCCC(C)(C)NC(C(COC)N(C)C)=O)CCC(=O)NC1 C(CC)(C(C)C)N(C(CCC)=O)C(=O)C(C1CCOCC1)N(C)Cc1ccnn1C C1(C(N(CCCn2cc(-c3cnc(C)s3)nn2)C)=O)Cc2nccn2C1 N1(C(c2cncnc2C2CC2)=O)CC(C2CCCCN(C(C3(Br)CC3)=O)C2)C1 N1(C(C2(c3cc(OC)c(O)cc3)CC2)=O)CCC2(CC1)OCCC2C#N N1(C(C2CC(C)SCC2)=O)CC(NC(c2cccc(F)c2)=O)Cc2ccccc21 C(Cl)(c1ccccc1F)=CC(C(=O)OCC)N(C)Cc1ccnn1C CCC(F)(F)C(C)(C)C(=O)NCc1cccnc1C.c1nc[nH]n1.C(=O)C.N c1(OC)cc(C)c(C(N2CCN(C(C3(Cl)CC3(C)C)=O)CC2CF)=O)cc1O N1(C(C2CCC(OC)C2)=O)CCCN(C(=O)C2=CCCOC2)CCC1 C1(C(=O)NCC(CO)NC(c2c(CCC)nsc2N)=O)Cc2ccccc2O1 C(CCC(C(=O)NC(C)CF)NC(C1CCSCC1)=O)OC C1(NCC(C)(C)NCc2cn(CC(N)=O)nn2)CCCCC1n1cccn1 N1(C(c2c(OCC)ccs2)=O)CCN(C(C2CCCC2(F)F)=O)C(C)C1 n1(CC=C)nnnc1C(c1cc(Cc2ccccc2)on1)NC1CCC=C1Br C1(CC)CCCCC1C(=O)NCC(C(C)(C)C)NC(=O)C(F)C1CCCC1 C1(CC(N2C(CC(=O)N(c3ccc(O)cc3)CC)CC2)=O)CC(=O)NC1=O C(=O)(CC(C)(C(F)F)N(C)C)N1CCN(C(c2c(COC)ncs2)=O)CC1C N1(C(CC(CC)C(C)C)=O)CCC2(CC1)OCCC2NC(C1COC(C)(C)C1)=O CN1CCc2nc(C(N3CCCC(NC(=O)Cc4c[nH]nc4O)C3)=O)sc2C1 N1(C(C(C)(C)c2cnsc2)=O)CCC2(CNC(C3CNC(=O)N3)=O)CCCC12 Cc1nc2ccnn2c(C)c1C(=O)N(C)CCNC(=O)CC1=CSC2=NCCN12 N1(C(C(C(C)C)SC)=O)CC2CCN(C(=O)C(C)=C(C)C)C(C2)C1 c1(C(N2CCCC2)=O)cc(F)ccc1Cl.C1(OC)CC2(C(=O)NCCO)CC12 C1(C(=O)NC(CNC(=O)CSc2cn[nH]c2)C2CC2)COC2COCC12 N1(C(C(=O)NCCCSCC)CC2CCC2)CC(O)CC2(CCCC2)C1 c1(C(=O)NCC(=O)Nc2c(OCC)cc(C)cc2)nccc2c[nH]nc12 Cc1ccccc1C(c1ccccn1)NC(C1CCC1c1ccccn1)=O N1(S(C)(=O)=O)CCC(CC(=O)NCCC2CC2)CC1.c1(C=O)ncccc1Cl.N N1(CC=O)C(=O)C(=O)N(C)C1=O.C1(CC=O)CC2CC2C1.CC(C)C.CN c12ccc(s1)[nH]c2=O.C(C)(C(=O)NC1CC1NC(C)=O)NC(C)=O CCC(CC(=O)N1CC(O)CC1CC)N(C(=O)Cc1cn(CC)nn1)C c1(C(=O)NC(CCOC)CNC(=O)CC(C)OC)ccc(OC)nc1Br c1(C(=O)NC2CC(NC(C3CCC(C)(C)C3)=O)C2)cccc2[nH]ncc12 c1(CC)onc(C(N2CC(NC(=O)C(CC)NC(C)=O)C(C)C2)=O)c1C C(=O)(C#CC1CCCCC1)N(C1CN(C(c2ccc(=N)[nH]n2)=O)CC1F)C CCC(C)(C)CC(=O)NC(c1ccccc1F)CNC(c1cn2c(n1)CCC2)=O c1(OC)cc(F)c(C(=O)NC2CC(F)CN(C(=O)CC(C)(C)C)C2)c(F)c1 CC1CCN(C(c2coc(Br)c2)=O)C(CNC(c2c[nH]c(C#N)c2)=O)C1 N1(C(CC2C(C)(C)C2)=O)CCC(O)(CNC(C2CC3(CCC3)C2)=O)CC1 c1(NC(=O)CC2CCC(OCc3cn(CC(F)(F)CO)nn3)C2)ncccc1Br c1(OC)cc[n+]([O-])c(C(N2CCOCC(CNC(C3C4CCCOC34)=O)C2)=O)c1 CCC(C)(C)C(C)NC(=O)C(c1ccoc1)NC(=O)CN1CC=CC1 C1(NC(Cc2c(C)n(C)cn2)=O)C(C)CN(C(c2ncncc2Cl)=O)CC1C N1(C(C(C)N2CCC2)=O)CC2(C1)CN(C(c1cnn(-c3ccccc3)c1F)=O)C2 N1(C(C(=O)c2ccco2)=O)CCOC2(COCCN(C(c3ccco3)=O)C2)C1 c1(C(N2CCCC(CNC(c3cc(C(C)=O)[nH]n3)=O)C2)=O)cnn2c1CCCC2 N1(C(C(=O)NC2CCC2)C2CC2c2cccc(F)c2)CC2OCCC2(CO)C1 c1(CC)nccn1C(C)CC(=O)NCCC(O)C.c1(C=O)nccn1C(C)C.N C1(C(=O)NCC(C)O)CC(F)(F)CN1Cc1cccc(OCCBr)c1Br c1(NC(C2CC(O)CCN2c2ncnc3cc[nH]c23)=O)ccc(O)cc1[N+](=O)[O-] N1(C(c2ccc(C(=O)OC)o2)=O)CC2OCCC2C1.C(=O)C(O)CCN(C)C.N C1(CCC(=O)N(C2CC(C#N)C2)C)CCCCN1.c1(NC(C)(C)C)cn[nH]c1 c1(N(CC=C)C)nc(N2CCN(CCOC)CC2)nc2cc(C)ccc12 c1(CCN(C(=O)NC(C#C)C)C)ccc(OC)c(OC)c1 N1(C(C2CC(=C3CC3)C2)=O)CCC2CCCC12C(=O)NC(CCO)C(F)F c1(C(N2CC3CNCC(C2)O3)=O)cc(F)c2nc(C3CCOC3)cn2c1 CCCCC(O)C(=O)NCC1C=CC(NC(c2c(C(F)(F)F)coc2C)=O)C1 C(C(=O)N(C(C)CCNC(=O)CC(=O)NC1CC1)C)(C(C)C)OC N1(C(COCCCC(C)C)=O)CCN(C(=O)CN(C)S(=O)(=O)N(C)C)CC1C c1(C(C)C)cccc(C(=O)NCC(O)CN(C(=O)CC2COCC2(C)C)C)n1 N1(c2n(C)ncc2)CCCN(C(C23CC(C(F)(F)F)(CN2)C3)=O)CC1 c1(OCC)ccc(OC(C)C(=O)NC2CCCC2N)cc1 C#Cc1ccnc(C(=O)NCC(O)CN(C(=O)C(S(C)(=O)=O)C2CC2)C)c1 c1(C(N2C3CC(NC(CC(C)N(C)C)=O)C2CC3)=O)ccnc2ccsc12 C(C)(CC(C)C(F)F)(c1n(CCC)nnn1)NCc1ncnn1-c1ccccc1 CCCCC(O)CNC(c1ccccc1-n1cc(-c2ncc(Br)cn2)nn1)=O N1(C(C(CCNC(=O)COC2CCC2)OC)=O)CCC(C)CC1C(N)=O c1(C(=O)NCCC(C)(C)NC(C2C=C(C)CS2)=O)ncccc1O C1(CNC(C2N(N=O)CCC2)=O)CN(C(=O)CC2=CCCCC2)CCC12CCC2 N1(C(C2CCC(C)O2)=O)CC2(C1)CN(C(C1C(C)(C)OC1(C)C)=O)C2 C1(C(=O)NCc2ccc(S)cc2)(COC)CCN(C(=O)C2=CCCSC2)CC1 C1(c2ccccc2)(COC)CN(C(=O)CNC)CCO1.c1ccccc1.C(C)=O.C CN1CCC(N(C(C2CCCN(C(=O)C(F)OC(F)(F)F)C2)=O)C2CC2)CC1 C1(CC)(NC(=O)C(F)C2CCC2)CCN(C(c2cn(C)nc2C)=O)CC1 C1(NC(CCCCCN(C)C)=O)CCCC2CN(C(C3C4CC5C(C4)C35)=O)CC12 c1(C(c2nc(-c3ccc(C)c(F)c3)nn2CC2CC2)C)ccc2ccccc2n1 c1(C(=O)NC2CCN(C(c3coc(C(F)F)n3)=O)C2)cc2ccncc2c(O)n1 C1(N=c2[nH]nc(C(F)F)s2)(CCC)CCN(C(C2CCCOCC2)=O)CC1 N1(C(c2n(C(C)C)cnc2)=O)CC2(C1)CN(C(=O)Cc1cccnc1)C2 c1(C(=O)NC2CN(C(CCCSC)=O)C(C)(C)C2)cn(C)c(=O)nc1O N1(C(C(C)OCOC)=O)CCN(C(=O)Cc2cocn2)C(CC(F)F)C1 C(=O)(CC(C)(C)CC(=O)NC(C)(C)CC)OC.c1(C(=O)N)cnn2cnnc2c1 N1(C(c2c(C(C)C)nco2)=O)CCC(C(=O)N(CCC2=CCCCC2)C)=C(F)C1 C(F)(C(=O)NC(C(=O)NC1(CCCCO)CC1)C1CCCC1)=C(C)C C1(NC(c2c(C)cns2)=O)CN(C(c2nc(C(C)C)no2)=O)C2CCCCC12 Cc1cc(C(=O)NC23CC(C2)N(C(=O)Cc2cccc(F)c2)C3)cc(C)c1N CS(=O)(=O)CCCC(=O)NC1(CNC(c2ccno2)=O)CCOCC1 c1(OC)cc(C)c(C(=O)NC2CCCCC2NC(=O)Cn2cnccc2=O)cn1 C1CC2(C1)CC(C#N)C2.C(C(C)C(C)C(=O)NCCC1(C=O)CC1)OC.N C1(NC(C(=O)NCCOC)=O)CC(C(N2CCC(C)(C)C2)=O)C12CCC2 c1(C(=O)OCC)n[nH]c(=NC2C3CC2CN(C(c2cccc(CO)c2)=O)C3)s1 N1(C(C2(C)CCCO2)=O)CCOC2(C1)CN(C(=O)Cc1cccc3nsnc13)C2 N1(C(CCNC(C(C2CCOC2)OC)=O)=O)CC(CO)C(C)(C)C1 CC(O)CCCN(C)C(C1CCN1C(c1cnn(C(F)F)c1)=O)=O CCC(C)C(CC(=O)NC(C)C(=O)N(C)CC)NC(=O)C(C)CC(=O)OC c1(CC)nn(C)c(N2CC3CCC2C(NC(=O)C=Cc2cncs2)C3)c1[N+](=O)[O-] C1(C(N(C2(CO)CC2)C)=O)CN(C(=O)CC2CCC2)CCO1 N1(C(CNC(CCC)=O)=O)CCC(NC(c2csc(C(C)=O)c2)=O)C1C c1(C(=O)NC2CCN(C(c3ccc(C)o3)=O)CC2C)ccc2c(c1)OC(C)(C)C2 N1(C(CN(C(C(C)C)=O)C)=O)CCC(C(C)C=O)C1.C(C1CCCC1)=CC=C CCCC(CC(C)C)C(=O)NCC(CNC(c1cc(C)[nH]c1C)=O)C(F)(F)F N1(C(CC=CC)=O)CC2CCC2(CNC(C2(c3ccc(O)nc3)CCC2)=O)C1 N1(C(C(C2CCN(C(c3cc(C)cc(O)c3)=O)C2)(C)C)=O)CC(=O)NC2(CC2)C1 N1(C(c2cc(C)[nH]c2C)=O)CC2(CCNC(c3ccccc3)=O)CCC1CC2 Cc1cc(C(N2CCC(C(=O)NCC(C)Cn3cccn3)C2)=O)sc1C N1(CCOC)CC2(CCC2)C1c1nc(-c2cccc(OC(F)(F)F)c2)no1 C=CCCC(C(=O)NC1COCCC1(F)F)NC(c1cc(C(C)C)[nH]n1)=O N1(C(=O)OC(C)(C)C)CCC2CN(C(=O)C=CCCc3ccccc3)CCC2C1 C1(NC(CN(C(=O)Cn2ncn(C)c2=O)C)=O)CC2(CCC2)C1O Cc1cc(C(N2CCC(NC(=O)Cc3nc[nH]n3)C(F)C2)=O)cc(O)n1 C12(NC(CCCC#C)=O)CCCN(C(c3cc(N)c(F)cn3)=O)CC1C2 C12(CC(=O)Nc3c(C)nn(C)c3)CC3CC(CC(C3)C1)C2 C(C(C)(C)C(=O)NCc1nc(=O)o[nH]1)N(C)C(c1ccc(F)cn1)=O Cc1[nH]nc2ccc(C(N3CCC(C(C)NC(C4C(C)C4C)=O)C3)=O)cc12 c1(NC(c2c(NC(C3(C)CCCCC3)=O)cccn2)=O)c(O)cccc1Cl C1(CNC(C2CCOCC2)=O)CC2(CC(NC(C34CCCCC3C4)=O)C2)C1 Cc1[nH]nc2cc(C(=O)NCC3CCC4COCCC4O3)ccc12 C1(C(=O)NC(C2(O)CN(C(=O)C)C2)C)CC12CCCC2.c1ccc(F)cn1.O c1(N2CCC(OC(C3C(C(=O)OC)C3)=O)C2)nc(Cl)ncc1C1OCCO1 C1(CC(N2CCCC(CC)C2)=O)CC(C)(C)C(=O)N1.C=Cn1nccc1C=O.N N1(C(C(C)OCC)=O)CC2(CCC2NC(=O)Cc2cc(F)cc(Br)c2)C1 C(N=c1[nH]c(=NC2CCn3cncc3C2)c2sccc2[nH]1)c1nc(C)c(C)o1 c1(NC2C(C)CN(C(c3cc4occc4s3)=O)C2)ncnc2c1CCO2 c1(OCC)ccccc1C(=O)NC1CN(C(c2ccc(C3CC3)cn2)=O)CC1F C(=O)(C(F)(CC)C(=O)OC)N1CCC(NC(CC(CC)CN(C)C)=O)CC1 C(=O)(C(F)CC(C)C)N1CCC(OCCNC(c2c(CC)occ2)=O)C1 O=S1(=O)CCC2(CCCN(CC3CC3C3CCCO3)C2)C1 C1(C(N2CCC(CN(C(c3c(CCC)n[nH]c3)=O)C)C2)=O)C2CCN1CC2 c1(OC)cc(C(O)C(N2CCCC(F)C2)=O)c(F)cc1O.C(=O)C=CC(C)C.N n1(CC(=O)NC(C2CN(C(C3(N(C)C)CCC3)=O)C2)C)ncc(O)nc1=O C1CN(C(c2cn(C(C)(C)C)cn2)=O)CC1O.C(C(=O)N)OCCOCC C1(CC(N2C(C(C)O)CCC2)=O)C2CN(C(=O)Cn3cnnc3O)CC12 CN1CCN(C(=O)C=Cc2cccc(Cl)c2)CC1CNC(=O)Cc1ccco1 c1(OC)ccc(C(N2CC(O)(CC)C2)=O)nc1.c1(C=O)c(C2CC2)cnn1C.N C(=O)(C1=C(F)CN(C(=O)CC2(CN)CCC2)CC1)NC(C1CCOCC1)C N1(C(c2cc(Br)sn2)=O)CCCCC1Cc1cn(CC2CCCOC2)nn1 N1(C(C2CC(C#N)C2)=O)CC2(C1)CN(C(=O)C1=CS(=O)CCC1)CCO2 c1(N2CC(C)N(C(c3cc(I)ccc3F)=O)CC2)ncc2c(Cl)cccc2n1 C(=O)(C(C(=O)NC1(C)CN(C(C2CCCN2C=O)=O)C1)OC)OC N1(C(C(C(C)C)(C)O)=O)CCCCC12CN(C(=O)C(CO)c1ccccc1)C2 c1(N2CCC(NC(=O)NCCSC)C2)ccc(C)cc1 c1(C(=O)NC(C2OCCN(C(CCNC(C)=O)=O)C2)C)ccn2c(O)nnc2c1 N1(C(CCC#C)=O)CC2CC2(CNC(=O)CC(C)NC(N)=O)C1 c1(C(c2n(CCCC(=O)OCC)nnn2)N)cc(C)nc(Cl)c1.C1C=CCCC1 C1(C(=O)NC(CSC)(C)C)CC(C)N1C(c1cc(C)c[nH]1)=O N1(C(C2COC2)=O)CC(Cn2cc(CSCCO)nn2)C(C(F)(F)F)C1 C1(CCC2N(C(CC3CC(=C)C3)=O)CCC2)CCCCN1C(c1cnco1)=O C1(NC(C(CC)OC)=O)CCCN(C(=O)C(C)CO)C1CC c1(CCC(=O)NCCCc2nnc(C)s2)c(C)noc1Cl Cc1cccc(N)c1C(=O)NC1CCCCC1NC(C1CCCC(C)(C)O1)=O C1(NC(C(CC)NC(N)=O)=O)COC2CN(C(=O)CN3CCC(F)CC3)CC12 c1(C(=O)NC(C=C)(C)C)cn(CCNC(c2ccnn2CC)=O)cn1 CCC(CC)(CCNC(C12CSCC1C2)=O)NC(C1CCCCC1(F)F)=O c1(CNC(CC2C(CC)C2)=O)ccc(CNC(=O)C(F)OC)cc1 c1(CC)ccc(C(N2CCC(C3CCOCC3)(CN)C2)=O)cc1S(C)(=O)=O c1(CC(C)C)n[nH]c(=NCC(C2CC2)NC(=O)C(c2ccccc2F)(F)F)s1 c1(OC)c(C(=O)N(C2CCN(C(c3ccnn3C3CC3)=O)C2)C)cccc1F CCC(F)(F)CC(=O)NCCOCCCNC(=O)CC1(O)CCOC1 C1(C(=O)OC)N(C(c2cnc(-c3ccc([N+](=O)[O-])cc3)s2)=O)CCOC12CCC2 C1(CC)CN(C(c2ccnn2CC(F)(F)F)=O)CCN1C(C1C2CCC1CC2)=O C(=O)(C1=C(c2ccccc2F)CCC1)N1CCC(C(=O)OC)CC1.c12cn(nn1)C2 Cn1nc(C(=O)NC(C)(C)CNC(=O)CCCc2ncco2)c2c1CCC2 N1(C(COCCC#C)=O)C2CCC1CC(CNC(C1(C)CC=CCO1)=O)C2 N1(C(CCN(C(=O)CC2CCCC(C)C2)C(C)C)=O)CCC(C#N)CC1 Cc1oc(C)c(C(=O)NC2CCC(NC(c3cnn(C)n3)=O)CC2)c1C c1(NC(C2CCN(C(C(CC)=O)=O)C2)=O)cccc(C2(C#N)CC2)c1 C1(C(N2CCN(c3c(Br)cnc(OC)n3)C(C)C2)=O)CCC2(CC1)CC(O)C2 c1(CNC(N(CC)Cc2cccc(Cl)c2)=O)ccc2c(c1)CCO2 Cc1cc(C(N2CCC(C)(NC(=O)C=CC3CCCO3)C2)=O)c(N)c(Cl)c1 N1(C(CNC(C=C)=O)=O)CCC(O)CC1C(=O)NCc1ccc(Cl)c(C)c1 CC1(NC(=O)Cc2cc(Cl)cc(Cl)c2)CCCN(C(=O)CCC(N)=O)C1 N1(C(c2c(OCC)c(F)ccc2)=O)CCN(C(=O)C(C)C)CC1CF C1(NC(c2cc(C#N)no2)=O)CC2CC(NC(=O)C(O)Cc3ccccc3)C1C2 c1(CC(N2CCC(C(C)NC(C(C(C)C)CO)=O)CC2)=O)ccn2cncc2c1 c1(C(=O)OCC)c[nH]ccc1=NCC(C)N(C)C(c1cc2cc(F)ccc2[nH]1)=O C(c1cccc2ccccc12)=CC(=O)N(CC)C1CC1.C(CC(C)C(=O)N)OC CC1(C)C2CCC1(C(=O)NCC(c1ccc(Cl)cc1)CO)C2 c1(C(N2C(CCNC(C(N)=O)=O)COCC2)=O)ccc(F)c(CC2CCC2)c1 N1(C(CC(C)SC)=O)CCCCC2(CCN(C(c3ccc(F)o3)=O)C2)C1 N1(C(C=C(CCC)C)=O)CC(C(=O)NC2CC(OCC)C2)CC1(C)C C1(NC(C2(c3ccc(C)cc3)CC2)=O)(C)CCC(F)(F)CC1.C(=O)C(C)O.N c1(CC)cc(C(=O)OC)cc(C(C(=O)NC)N(CCC(C)C)CC(C)C)c1 CC(C(=O)NCCOCCCN(C)C(c1ccsc1)=O)C1CCOC1 N1(C(c2cccc(OC)c2)=O)CC(CNC(C23CCC(CC2)OC3)=O)CCC1C N1(C(CCCC(=C)C)=O)CCc2ccccc2C1CNC(=O)Cc1csc(C)n1 N1(C(C(CC(C)C)C)=O)CC2(C)CN(C(c3ccnn3CC3CC3)=O)CC2(C)C1 C1(CNC(CSCCNC(C(C)=C(C)C)=O)=O)CCC2CC12 C1(NC(C(CN(C)C)NC(C2C3CC(=O)CC23)=O)=O)C(O)C2CCOC12 Cc1c(-c2nc(C3CC3)nn2CC2CCCO2)[nH]c2c(Cl)cccc12 C1(NC(C(CC)CCOC)=O)CCSC12CN(C(C1(CO)CCCO1)=O)C2 N1(C(C(C)n2cccn2)=O)CC2C(NC(=O)Cc3ccc(Cl)cn3)C2C1 C1(O)(CC(=O)N(CC(CN(C(C2C(C=C)CC2)=O)C)O)C)CCCCC1 N1(C(c2[nH]cc(CC)c2)=O)CCC2(CCC2)C(CNC(=O)CC)C1.C=O.N C1(NC(C2C(C)CN(C)C2)=O)CC2(C1)CC(NC(C1(C#N)CCC1)=O)C2 C1(NC(C2CC(=O)NC(=O)N2)=O)CN(C(c2coc(Cl)c2)=O)CC2CCCC12 C(=O)(CC(C(F)(F)F)NC(C1CCC2(CCC2)O1)=O)NCc1nc(C)sc1 C1(CNC(C2CCCC(F)C2)=O)CN(c2cc(-c3cccs3)ncn2)CCO1 C1(NC(CCCOC)=O)C2CC1N(C(=O)CC(C)F)C2 N1(C(C(CSC)O)=O)CC(C)N(C(=O)CC2C=CS(=O)(=O)C2)CC1C C(CC(O)C(=O)N(CC(F)F)CCO)NC(C(CC)=CC)=O N1(C(C=C(CC)CC)=O)CCC2CCN(C(C3(c4ccno4)CC3)=O)CC2C1 c1(OCC#C)ncccc1C(=O)NCCCC(C)NC(c1nnc(C)s1)=O C(=O)(N(CCC(=O)N1CC(CO)C(C)(C)C1)OC)c1cnc(OC)s1 N1(C(C(C)C2CC2)=O)C2CCC1CN(C(=O)C(C)(C)c1cnco1)C2 c1(C(C)(C)C)nc(=NC2COC3(CCN(C(c4nc(Cl)cs4)=O)CC3)C2)s[nH]1 C1(C(=O)NCC(F)CO)(CC)CCN(C(C2C3CC4C(C3)C24)=O)CC1 C12(C(=O)NC3(CN(C(c4cn(CCC)nc4)=O)C)CC3)CC1COC2(C)C C(=O)(C1=C(Cl)CCCC1)NCCC.N1(CC=O)CC(C(F)(F)F)CCC1=O.C CCCCCC(C(=O)N1CCC(NC(=O)CC(C)(C)C(F)(F)F)C(C)C1)C(C)C C1(CNC(CCNC(N)=O)=O)CCN(C(c2n[nH]c3cccnc23)=O)CC1(F)F C1(N(C(=O)CCC2(C)CC2(F)F)C)CCCN(C(=O)CC(C)(C)O)CC1 C1(C2CCN(C(=O)Cc3ccccc3F)C2)(NC(=O)OC(C)(C)C)CC1 c1(C(=O)NCC2CCC(NC(C3CC(OC)C3)=O)C2)ncc(C)cn1 C1(NC(CSCCOC)=O)Cc2ccccc2C1NC(=O)CCC.C(C)(C)C.S C1(CNC(C2CC(OC)C2)=O)CN(C(=O)CCC=CC(C)C)CCC1(C)C N1(C(c2c(OC)csc2)C(=O)NCCSC)CCOC2(CCOC2C)C1 C1(NC(c2c(C)cc(Br)cc2F)=O)CC(=O)c2ccccc2O1 CCCC(C(=O)NCCCN(C)C(c1ccc(C(C)(C)C)cn1)=O)S(N)(=O)=O C1(CC(=O)NCC(CO)NC(c2ccc(-c3ccccc3)o2)=O)CCCC1O C(=O)C1=CS(=O)CCC1.C1CCC(C)(O)CC1.CC(C)(CNC(=O)CS)C c1(CNC(CC(C)NC(c2cnn(C(C)C)n2)=O)=O)ccn(C)c(=O)c1 C1(C(=O)N)CN(C(=O)CC2CC3(CC3)CO2)CC(C)O1.C(C)(CC(C)C)OC C(=O)C1=CCC2(COC2)OC1.c1(CC(C)NC(COC(C)C)=O)ccccc1.N c1(C=O)csc2ccc(C)cc12.C1(CNC(CC2(OC)CCC2)=O)CCCC1.N C1(C(=O)NC2CN(C)CC2O)CCC2(CC1)CNC(=O)C2 C(c1ccccc1Cl)=CC(=O)NC1CC(F)CN(C(=O)C=Cc2cn[nH]c2)C1 C(CN=c1[nH]cnc2c1COC2)C1CCC(NC(C(C)CC(N)=O)=O)C1 Cc1ccc(C(=O)NC2(C)CC(C(=O)N(CC(F)(F)CO)C)C2)cc1 CN1CC2C(C(=O)NCCCCCCNC(C3(CCCF)CC3)=O)C2C1 C1(C=O)CCc2nc(C(F)(F)F)cn2C1.CC(C)CC(C)CNC(=O)C(C)O.N C(=O)(C1OCCc2ccc(Br)cc21)OC(COC(C)C)C c1(CNC=O)ccccc1F.C1(CCN)CC=CC1 CC(CN(C)C)CC(=O)N1CC=CC(C(=O)N(C)CC2CCOCC2)C1 c1(OC)cc(C)ccc1NC(=O)C(C)(C1CC1)N(C(=O)CCn1ccnc1)C C1(CNC(C2CC(C)C2)=O)CN(C(C23CCC(CC2F)C3)=O)CCC12CCC2 C(CCC)(C(=O)NCC(C1CCN(C(=O)CCC(C)OC)CC1)C)=CCC C1(CC(=O)NCC(CO)N(C)C)CCN(C(C2CCSCC2)=O)C1 c1(NC2(c3ccc(OC)nc3)CC2)nc(Cl)nc2c(F)cccc12 C(=O)(CP(C)(C)=O)NCCCN(C(c1c(OC)c[nH]n1)=O)C N1(C(CN(C(=O)OC)C)=O)CCC2(CC2)C1.c1(C=O)c(C(F)F)n[nH]c1C.C C1(NC(Cc2c(C)nn(C)c2)=O)CCCC12CCN(C(=O)C1=CC(C)CC1)CC2 CC1CCCN(C(C2CCCC2)=O)C1CNC(c1cc(C(F)(F)F)ns1)=O c1(CC(C)NC(=O)C(=O)NCCn2cc(-c3cccnc3)cn2)ccc(Br)s1 C1(NC(c2n(C)cnc2)=O)CCC2(CCN(C(c3cccn4ccnc34)=O)C2)C1 C1COC(C)(C)CN1C(c1cc(C(N)=O)co1)=O.C=C1CC(C(=O)NC)C1 C=CC(C)(CCOC)C(=O)N1CCC(C)(NC(c2ccc(=O)n(C)n2)=O)CC1 C(=O)(C1=CSCS1)NCC1OCC(CNC(C(C)Cc2ccccc2)=O)C1 c1(C(=O)NC(CNC(C2CC(OCC)C2)=O)CO)cccc(CC)c1 C1(C(=O)NC(C2CC2)C)CC1CO.C(=O)(C=CC1CC1)NC C1(C)(NC(COCCN(C)C)=O)CCN(C(=O)CC(=O)N)C1.CC(F)(F)F N1(C(c2c(SC)cccn2)=O)CCN(C(=O)C(C)C(F)(F)F)C2CS(=O)(=O)CC12 C(=O)(CC(C)(C)CC(F)F)N1CCC(NC(Cc2c(OC)ccnc2)=O)C1 c1(C(N2CCC(N(C(C34CCCC3CC4)=O)CC)CC2)=O)cnc(OC)cc1C C1(C(=O)Nc2c(C)nccc2)CN(C(C2(C)CNC(=O)N2)=O)CC1(F)F C1(C(N2CCC(Nc3cc(O)nc(C)n3)C2)=O)(CC)CCC(O)CC1 c1(C(N(C)CC2CCCC2)=O)cc2c(s1)CCC2.c1(C=O)cn(C(F)F)cn1 C(=O)(C(O)C(C)(C)CC)N1CC(NC(c2cnc(CC)[nH]2)=O)C(O)C1 C=CCCN=C(NCC(C)C)NCC1C=CCCCC1 N1(C(C(C2(C)CC2)NC(C2CCC(CO)CC2)=O)=O)CCC2(CSC2)C1 CN1CCN(C(c2cnnc(O)c2)=O)C(CNC(c2cc(Cl)cc(Cl)c2)=O)C1 Cc1cc(=NCC(C)F)[nH]c(=NCc2nc(C)c(C)nc2C)[nH]1 CC(C)(O)C(C(=O)NCc1cccc(CO)c1)NC(c1cc(O)cs1)=O c1(C(=O)NC2(COC)CCN(C(C3CCOC3C)=O)C2)ccc2nonc2c1 c1(NC(N2CC(CC)OC(C)C2)=O)cccc2c1C(C)OC2=O C1(C(N2CCOC(CCNC(c3ccc(C)cc3)=O)C2)=O)(OC)CCCOC1 CC1(C)CCCCC1NC(c1cccnc1CNC(C1CCOCC1(C)C)=O)=O N1(C(C=CCC)=O)CCC(C(=O)NCCNC(c2cc(C)sn2)=O)CC1 C1(C(=O)NC(C)CN(C)C(C2CC2C)=O)(SC)CC1 C1(NC(C2C(C)OCC2)=O)CC2C(NC(C3(C)CSC3)=O)C2C1 N1(C(C)=O)CCOC(C(=O)NCC(CO)NC(c2cccc(C(N)=O)n2)=O)C1 O=C(N=c1cc(C2CCCCC2)[nH][nH]1)C1(CC(F)F)CCCO1 C(CC(C)(C)C(=O)N1CCC(C)(OCC)C1)NC(C(CC#C)O)=O C1(C(N(C(C)(C)C)CC=O)=O)CC12CCN(C(c1cnc(C(F)F)s1)=O)CC2 N1(C(C(C)OCC=C)=O)C2CCC(C2)C1C(=O)N.C1CC2(C1)CC(O)C2 C1(CC(=O)N(C2C(OC)COC2)C)CC(C)(C)CN1C(=O)CCc1cccs1 c1(CC=O)cnc(C2CC2)[nH]1.C(C)(C(=O)NCCCOCC)=C(C)C.N C1(CNC(C2CC(N(C)C)C2)=O)CC2CCC1N2C(C1CCC(C)(C)C1)=O c1(CN(c2ncnc(=N)[nH]2)C)cccc(CNC(C2SCCCS2)=O)c1 C(CNC(C1SCC=C1C)=O)(CC(=O)NC1(C)CCSC1)OC c1(C(=O)NC2C(NC(c3c(COC)cccn3)=O)COC2)ncn2c1CCCC2 C1(C(=O)NCCC2CC=CCC2)CC2(CCN1C(=O)CC1=CCOCC1)CC2 c1(C(=O)NCC2CC(C)N(C(=O)CCC)C2)cc2ccc(F)cc2[nH]1.C(N)=O.N N1(C(CNC(C)=O)=O)CC2CC(NC(=O)CCN3CCC(O)CC3)CC2C1 C(=O)(C(CC)CCOC)N(C1CC(NC(c2cc(CCC)oc2C)=O)C1)C N1(C(=O)Cn2ccnn2)CC2CCN(C(c3cc(=O)cc(Cl)[nH]3)=O)CC(C2)C1 c1(C(N2CC(CCCCNC(=O)C(O)C3CC3)C2)=O)sc(Cl)cc1Cl Cn1ncc2c1CC(C(=O)NCCC1CCCN(C(C3(C)CCCC3)=O)C1)CC2 C#Cc1cnn(CC(=O)NC(C)(C)CC=CC(N2CCC2C2CCCC2)=O)c1 CN1CC(C)(C=O)CCC1=O.C(=O)C=CC.C(C)(C)C.CCN(C)C=O N1(C(CC(CNC(C2CC(O)(CC#C)C2)=O)OC)=O)CCOCC(F)(F)C1 c1(NCc2cncc(C#N)c2)sc2c(c1C(=O)Nc1nc(CO)cs1)CCCC2 CC1CC(C)N(C(=O)Nc2ccccc2)C(C)C1.C12(CC1)CN(C)C2 C=C=CCCC(=O)NC1(C2CCCCN2C(c2cnc(C(N)=O)s2)=O)CC1 c1(C(CNC(N(CC)Cc2ccncc2)=O)O)ccc(F)cc1F N1(C(CN(CC)CC)=O)CC2(CC(C)C2)C1.C12(C=O)CCC(F)(CC1)C2 C(=O)C(F)(F)C(F)(F)C(F)F.N1(C(C(C)OC(C)(C)C)=O)CC=C(CC)CC1 C(=O)(C(COC)CC(C)C)N1C(C(N2C(CC)(CC)CC2)=O)CC(F)C1 C1(NC(C(F)OC)=O)CCCCC12CCN(C(=O)COC(F)F)C2 N1(C(C(C)(F)F)=O)CC2CC2(CNC(c2ccccc2C2CC2)=O)C1 N1(C(C2COCCN(C(CC(C)N3CCCC3)=O)C2)=O)C2CCC1CN(C)C2 N1(C(CSS(C)(=O)=O)=O)CC=C(C(=O)N2CCCC(CN=[N+]=[N-])C2)C1 C1(NC(c2cc(CC)no2)=O)C(C)(C)C(NC(c2oncc2C)=O)C1(C)C C=C(C)CC(C(=O)NC(C)CC1(O)CCC1)NC(=O)C(C)CSC Cc1ccc(Br)cc1C(=O)NC(CO)C(C)NC(c1ccc(O)nc1)=O C1(C)(NC(CCN(C(=O)CC2CCCCN2C)CC)=O)CCC(C)=C(C)C1 O=C(CC1OCCc2ccccc21)NC1(C2CCN(C(c3cc[nH]n3)=O)C2)CC1 C(=O)(C(C(F)(F)F)(C1CC1)Nc1ccccc1)OCC.c1ccc(Cl)cc1C.O C1CN(C(c2c[nH]nc2-c2ccoc2)=O)CCO1.C1(C)(CC)CC1C(=O)NC.C c1(C(N2CCC(CO)C2)=O)cc(-c2cncc(CO)c2)cnc1Cl C1(F)(CNC(Cc2cnc(C)[nH]2)=O)CCN(C(C2CCC(C)(C)C2)=O)C1 N1(C(C(=O)NC2CC(COC)C2)=O)CCC(Cc2nncn2C)(CO)CC1 C12COCCC1CN(C(=O)CS(=O)(=O)C1CC1)C2.C(C(C)(C)C)N(CC(=O)N)C N1(C(C2(SC)CCC2)=O)CC2(CC(NC(C3CCSC(C)C3)=O)CO2)C1 Fc1ccc(Cl)cc1N(CCI)Cc1ccnn1C1CC1(F)F C1(C=O)CCC(=O)N(CC(F)(F)F)C1.C1(F)(C(N2CC(CC)C2)=O)CCCC1 C1(CCNC(c2ccc[nH]2)=O)CCCCN1C(=O)COC(F)F N1(C(c2c(-c3cn(C)nc3)cco2)=O)CCN(C(C2CC(OC(F)F)C2)=O)CC1 C1(OC)C(C)(C)CN(C(CCc2ccsc2)C(=O)NC2CC2)C1(C)C c1(C(=O)NCCCC(C)NC(C2CC(F)(F)C2)=O)nc2ccccc2[nH]1 C=C(C)C(C)(C)C(=O)NCC1C=CCN1C(=O)CCN1CCCCC1=O C1(C(=O)NC(CNC(c2cc(CC)c(O)cc2)=O)C)CCC2(CCC2)CC1 C=C1COCCN(C(=O)CC2CCCCN2C(c2cc(C)c(O)nn2)=O)C1 Cc1nn(CC(=O)NCCC(C)NC(C2(c3ccc(Cl)s3)CC2)=O)cc1Cl C1(OC)CCC(N(C)C(C2OCCC2NC(=O)CC2CCCCO2)=O)CC1 CC1(C)CC(CC(N2CC(NC(=O)C(F)(F)CC3CC3)C(F)C2)=O)CO1 c1(OC)ccc(CN2CCC(CC(=O)Nc3ccnc(F)c3F)CC2)c(C)c1C N1(C(=O)NC(CC)C)CCC2(CC1)CC(=O)N(C)C2 CCCC(C)(O)C(=O)NC1CCCCC1C1CCCN1C(=O)CCCC(=O)NC C1(C)(NC(C2C(C=C)C2)=O)CCCN(C(=O)COc2ccc(Cl)cc2F)C1 N1(C(C(C)(C)OC)=O)CC2(C=C(C(=O)NCC3CCC4(CC4)C3)CO2)C1 C1(NC(C2C(C)CCO2)=O)CCCC12CN(C(c1ccccc1[N+](=O)[O-])=O)C2 C(=O)(C1CCc2nccn21)NC1CCC(NC(C=CC(C)(C)SC)=O)CC1 N1(C(CCC)=O)CCC(NC(=NCC2CCCO2)NCC2CCOC2C)CC1 N1(C(c2cccc(C)n2)=O)CCC(CO)(NC(=O)Cc2ccc(Cl)s2)CC1 N1(C(C=C(CC)CC)=O)CC(NC(=O)C(CC)CCOC)C2(CC2)C1 c1(C(C)=O)cc(C(=O)NCC2CC(C)CO2)ccc1C.c1(C=O)coc(O)n1 N1(C(=O)C2=CCC2)CCN(C(=O)CCc2ccc(F)cc2)C(C(F)F)C1 C(=O)(C(C)(C)CC=C)N1C(C(N(CC(CCC=C)O)C)=O)CC(O)C1 c1(C(N2CC(NC(C(C)C)=O)C3C2CCCC3)=O)ccc2c(c1)CCCC2=O Cc1nc(CC(=O)NCC23CC2CN(C(c2cc(CCO)on2)=O)C3)c(C)s1 c1(N(C)C)cccc(S(=O)(=O)N2CCC(C)(C)C2C(=O)O)c1 N1(C(C=CC)=O)CCC(NC(c2cc(Br)cnc2S)=O)C2(CCC2)C1 c1(OC)cc(Br)cc(C(=O)NC23CC(NC)(C2)C3)c1.c1ccc(Cl)cc1Cl CC1=C(C)OCCS1(=O)=O.C(C(C)(CCO)Nc1nnnn1-c1ccccc1Cl)OC CC(CS(C)=O)C(=O)N1CC=C(C)CC1.C(c1ccco1)=CC=O.C(=O)(C)N C1(CC(N2CCOCC2)=O)CCCN(C(c2cncc(C(=O)O)c2)=O)C1 CC1CCCC(CNC(=O)NCC2(n3nccn3)CC2)N1 C(=O)(CC1=CCCCC1)N1CCC1.c1(C(=O)NCC)cnc(Cl)c(C2CC2)c1.O C(=O)(C(C)(C)C(=O)NCC1CCCCCC1)NC.c1(C=O)cc2n(c1)CCC2 N1(C(c2coc(Br)n2)C(=O)NCC(=C)C)CCSC2CCCC12 C1(COC(CC2C(OC)CC2)=O)CCCC(C)(C)CC1 C12(C(N(CCCN(C)C(c3sc(F)cc3Cl)=O)C)=O)CC3CC(CC1C3)C2 N1(C(CCNC(C2CCOCC2)=O)=O)CCC2C(NC(C3CC34CCC4)=O)C12 C(=O)(C(C(C)C)n1cncn1)N1CC(N(C(=O)Cc2nccn2C)CCC)C1 N1(C(C)=O)CCCC(C=O)CC1.CC(F)(F)C(C)(C)C.CC(C)(C)OC(=O)N C1(C(=O)Oc2ccc(OC(C)C)cc2)CCc2nc(C3CC3)ncc2C1 Cc1ccc(C)cc1O.c1(CS(N2CC3(C(C(=O)N)C3)C2)(=O)=O)ccc(F)cc1F C#CCC(CC(=O)NC(CO)C1(C)CC1)NC(c1ccccc1O)=O C1(N(C(=O)CC2(C=O)CC2)CCC2CC2)CCCC1.CC(C)C.CC=O Cc1c[nH]c(C#N)nc1=NC1CCCC(NC(=O)CC(C)(C)O)C1 Cc1cccc(CCNC(C2CN(C(=O)C)C2)=O)c1.c1ccsc1.C(N)=O.N CCC(CC)N=c1[nH]c(NCC2CN(C)C2c2ccccc2)nc2cccc(F)c12 c1(OC)cc2c(cc1OC)CC(C)(C=O)C2.C(C)C(=O)O.C(=O)CC(C)C.N C1(NC(c2cnn(CC)c2C)=O)CCCN(C(=O)CCc2cnc(O)[nH]2)C1C C1(C2CCN(c3ncnc4c3COC4)CC2)(NC(C2CCCC(OC)C2)=O)CC1 c1(C(=O)NCCC(=O)NCC=C=C)cc(O)nc(O)n1 C#Cc1ccc(C(=O)NCC2CCC2NC(=O)C(C)(C)C#C)cc1Cl C(=O)(CCCCCCn1cc(CCCC#N)nn1)N1CCC(C)C1(C)C C=C(Cl)CC(C(=O)NC(CN(C)C)CO)NC(=O)CCCn1cccn1 CC(O)C(F)(F)C(=O)N(CCCNC(C1(C)CCC(=O)NC1)=O)C C1(CC(=O)NCCCCCF)(OC)CN(C(c2ccc(CO)o2)=O)C1 N1(C(c2c(C)nc(C)s2)=O)CCC(CO)(CNC(=O)CCO)CC1.C1COC1 C1(CNC(C2NC(=O)C(F)C2)=O)CCCCCN1C(=O)CC1=CCCC1 c1(C(=O)NCCC(C)NC(c2cccnc2Cl)=O)c(C2CCC2)cnn1C C1(CC)CN(C(=O)Cc2ccns2)CCC1CNC(c1cc(O)cnc1Cl)=O C(C1c2ccccc2CCN1C(c1cn(C)nn1)=O)NC(C=NOC)=O Cc1c(Br)ccc(C(N2CCCC2c2ccccc2F)=O)c1F c1(CC(=O)NC2CC(NC(C(C)C(F)(F)F)=O)C2)c(F)ccc(Br)c1F C(=O)(C1=C(C)S(=O)(=O)CC1)N(CC)CC.C1(C(=O)N)C2CCC(F)C12 c1(OC)c(C(N2CCC(C)(NC(=O)C(F)OC)CC2)=O)c(C)nn1C c1(C(=O)NCCN(C(CCC(=C)Cl)=O)CCO)cc(F)c(COC)cc1N c1(CC)ccc(O)c(NC(=O)C(O)CNC(C2(O)CCCCC2)=O)c1 CC(C)CC(c1ccccc1)NC(c1sccc1NCc1ccccn1)=O c1(CC)ccc(C(N2CC=CC2CNC(=O)Cc2nc[nH]n2)=O)cc1 C1(C(N(C2CCCC2)CC=C)=O)C2CN(C(=O)C(C)CC3CCCC3)CC12 Cc1cccc(-n2cc(CN3CCCC(CNC(=O)C(C)C(C)C)C3)nn2)c1 c1(NC(C(C)OC(C2CC2[N+](=O)[O-])=O)=O)sc(Cc2ccccn2)cc1C#N CC1(NC(c2csc(-c3ccoc3)n2)=O)CCN(C(=O)CCC(F)F)C1 CC(C)CC(CNC(=O)C1=CC(C)C1)NC(c1nocc1Cl)=O c1(C2(NC(C3CCN(c4cn(C)nc4)CC3)=O)CC2)nccc2ccccc12 N1(C(c2cc(CC)on2)=O)CC2C(C1C(=O)Nc1cccc(C)c1Cl)C2(C)C N1(C(C(C)OCC)=O)CCCCC2(CCN(C(=O)Cc3ccc(F)c(F)c3)C2)C1 c1(CC)cc(CC(=O)NC2(C)CC(NC(C3CCN(C)C3)=O)C2)on1 C1(N(C(c2c(C)nn[nH]2)=O)C)CCN(C(=O)CN2C(=O)CNC2=O)CC1C c1(C(N2CCN(C(C(CC)(C)F)=O)CC2CO)=O)ccnc2[nH]cnc12 N1(C(C(C)NC(C)=O)=O)CCN(C(=O)C(O)c2ccsc2)CC12CC2 C1(CNC(c2c(C)n[nH]c2)=O)CC2CCC1N2C(c1n[nH]c2c1COC2)=O c1(SC)cccc(F)c1C(=O)N(CC(C)N(C(=O)CC(C)(C)C)C)C C(=O)(CC(C)(O)C(F)(F)F)NC(C(C)CC(=O)OCc1ccccc1)(C)C C(=O)CC(O)CC.n1(CC)cc(Cl)cc1C(N1CC(C(=O)NCC)C1)=O.N C(=O)(CC(COC)COC)NC(CCC)CNC(C1CNC(=O)O1)=O Cc1ccc(Br)c2c1C(NC(=O)CCCOCC)CC2.c1(O)cccnc1.N1CC1 N1(C(COCCOCC#C)=O)CCC(C)(C)C1C=O.c1(CCO)nncn1C CC(C(CO)NC(c1ncnn1C1CCOCC1)=O)NC(=O)C1CC1 c1(-c2cn(CC(=O)NCCCOCC3CC3)nn2)cc(Cl)cc(Cl)c1Cl c1(C(c2nnnn2CCOC)NC2CCC(C)(CC)CC2)ccc(Cl)c(Cl)c1C Cc1cc(NC(=O)NC2CCCC2C(=O)NCCc2ccncc2)cc(C)c1Br N1(C(C2C(OCC)C2)=O)CC(F)(F)CC1CC.C(=O)C(C)C1(C)CC1 N1(C(c2cccc(C)c2C)=O)CC(C)CN(C(=O)CCCc2cccs2)CC1C Cc1ccc2sc(=NC3CCCN(C(=O)CNC(=O)C(C)(C)C)C3)[nH]c2c1 Cc1c[nH]c2cc(C(N3CC(CC(=O)Nc4cnccc4[N+](=O)[O-])C3)=O)ccc12 Cc1cc(=NCC2CN(C(=O)CCc3cn[nH]c3)C2)[nH]c(-c2cccc(F)c2)n1 CCC(C)CC(C(=O)N1CC(OCC(F)F)C1)NC(=O)CCc1ccccn1 N1(C(C(CCCC)CC)=O)CC2(C=C(C(=O)NC(C)(C)CCCC)CO2)C1 C1(C#N)(C(=O)NC(C2CCNCC2)C(=O)OC)CCOC1 C(N=c1ccnc(NC2CC3CCCCCC23)[nH]1)c1cccc(C)n1 C1(NC(c2ccc(C(C)C)nc2)=O)CC(C)CN(C(=O)C(C2CC2)N(C)C)C1 Cc1nn(C(C)C)cc1C(N1CC(O)C1)=O.C(=O)(CC)NC.CC(F)(F)F.C C#Cc1cccc(NC(=O)Nc2cncc(I)n2)c1C#N C1(C)(CNC(C2CCC(NC(COC(C)(C)C)=O)C2)=O)CCCCC1O c1(CC=O)c(C)nn(C(C)C)c1C.c1(C(C)=O)c[nH]c(C(=O)N)c1.C(C)CO C12(C(=O)OC)CCCC1CN(C(=O)C(=O)NCc1ccc3c[nH]nc3c1)C2 C1(COC)CN(C(c2nccnc2Br)=O)CCN1C(c1ccc(F)cc1I)=O N1(C(C2CC(C)(CC)OCC2)=O)CC2CCC(C1)C(NC(=O)C(C)O)C2 N1(C(CCc2c(C)nn(C)c2)=O)CCC2CCCC12CNC(=O)COC(F)(F)F C1(C(=O)NCCCN(C(=O)CCc2nncn2C)C(C)C)CCC12CCOCC2 FC1(F)CCC2CN(c3nc(-c4ccccc4)cs3)CCC2C1 C1(NC(C2CC2C2CCC2)=O)CCCN(C(c2cccnc2OCCO)=O)CC1 CCCC(C)(CC)C(=O)NC1CC2CCC1CC2NC(=O)CC1CCCCCC1 C12CCC(CC1)N2C(=O)C(C)(c1ccccc1)N(C)C.C(F)(C(=O)N)OC.C Cc1sc(Nc2cnc(Cl)nc2)c(-c2csc(C(=O)NC(C)C)c2)c1C N1(C(C2CCC(CC)CC2)=O)CC2(CCC(C)O2)C1.C1(C=O)C=CC=CC=C1.N N1(C(c2nc(CC)oc2)=O)C(C(=O)NCC(N2CCCC2)=O)CCC12CC2 C1(NC(C2N(Cc3c(C)cc(C#N)cc3)CC2)=O)Cc2ccc(Br)cc2C1 CC(C)(C)C(CO)C(=O)NC1(C)CC(NC(c2cscc2C(F)F)=O)C1 C1(C)(n2cc(COC(C(C)(C)C#N)=O)nn2)CCC(F)(F)CC1 c1(C(=O)NCCCC(C)NC(c2ncc(C)c(Cl)c2)=O)c(N)cccc1[N+](=O)[O-] N1(C(C(C2CCN(C(CC(COC)C)=O)C2)(C)C)=O)CC2C3CCC(O3)C2C1 C(=O)(CCCS(N)(=O)=O)NCC(C(C)(C)C)NC(C12CCC(F)C1CC2)=O c1(OC)ccc2c(=NC(C)c3n[nH]c(C)n3)[nH]c(=NCC3(C(C)C)CC3)[nH]c2c1 c1(C(N(CC(CC)NC(C2CC2[N+](=O)[O-])=O)C)=O)nc(C)sc1C Cc1[nH]c(-c2ccco2)nc(=O)c1C(=O)NCCC.C1(C)(CC=O)CCCC1.N N1(C(c2nc(CC)on2)C(=O)NCCC#N)CCC(S(=O)(=O)N(C)C)C1 C12(CNC(C3(C)CC3F)=O)CC(CO1)C2.c1(C=O)conc1-c1ccccc1 CC1CCCC=C1C(=O)N1CCC(C(=O)NC2CCC2(C)C)C1 CON(CCO)C(=O)C(F)(CNC(=O)CCc1conc1C)C(C)C c1cccc(Br)c1.C1(C)CCOC1.CC(C)CCNC(=O)CN(C)CCOC.C c1(C(N2C(CNC(c3ccc(F)s3)=O)CC(OC)C2)=O)cccn2nnnc12 C1(CNC(CCCCN(C)C(C2(C)CC2)=O)=O)CC(O)C12CCC2.C1CCC1 N1(C(C(CC#C)(C)NC(c2[nH]ccc2C)=O)=O)Cc2cccnc2C1 N#Cc1cccc(C2(NC(=O)NCC3(n4cccn4)CCOCC3)CCOC2)c1 C1(C(=O)N(C(C)C(=O)OC)C2CC2)(NC(CCNC(C)=O)=O)CCSC1 C1(C(N2CC(c3n(C)ncc3)C2)=O)CNCCN1C(c1cccc(CO)n1)=O C1(OC)CCC2(CCN(C(C3CCCCN3C(=O)CC3NC(=O)NC3=O)=O)C2)C1 Cc1oc(Br)cc1C(=O)NCC1C2CC1N(C(=O)CCc1ccncc1)C2 N1(C(=O)Cc2cccc(O)c2)CCN(C(=O)CC2CC2)C(C2CC2)C1 C1(OCC(C)CNC(=O)C(F)(F)Oc2cccc(Br)c2)CCN(C)CC1 C1(C)(C=O)CCCS1(=O)=O.C1(C(=O)N)(OCC)CCOCC1.CC(C)(C)C N1(C(C(C)Sc2nc(C)[nH]n2)=O)CCCN(C(c2cccc(N(C)C)c2)=O)CC1 CCC(C)(CN=c1[nH]c(=NCC2COC(C)(C)CO2)[nH]c2cc[nH]c12)OC c1(C(=O)NCc2n(C=C)ncc2)ccc(NC(C)=O)c(Cl)c1 C(=O)(N=c1[nH]c(S(C)=O)ncc1Br)OCC1N(Cc2ccc(OCC)cc2)CCC1 C1(N(C(=O)C(F)n2ccnc2)C)CCCC(NC(=O)CCc2ncc[nH]2)C1 c1(N2CCCC(NC(c3c(OC)ccnc3)=O)C2)nc(Cl)nc2sccc12 C1(CNC(C2CCCC2)=O)CCC12CCN(C(C1CCC3(CCC3)O1)=O)CC2 N1(C(CC=C=C)=O)CCC(C(C)(C)C)(CNC(c2ccnn2C)=O)C1 CCCCC(=O)C(=O)N1CC(NC(c2cn(C)nc2OC)=O)CC(C)C1 C(=O)(CC(O)CNC(c1ncncc1N)=O)NC(CC)C(N)=O CC(C)CCCCC(=O)NCCCCN(C)C(c1cc(-n2cccn2)ccn1)=O N1(C(c2ccn(C)n2)=O)CCC2(C(=O)NOCCCO)CC2C1 C(C)(C(C(=O)NCc1ccc[n+]([O-])c1)NC(c1cc(Cl)cn1C)=O)OC N1(C(c2c(COC)n(C)nc2)=O)CC2(CNC(=O)CO2)C1 N1(C(CSCC#C)=O)CCCC(C)(C)C1C.c1(C=O)cc(C2CCC2)[nH]n1.N C(=O)(C1=CC(C)(C)C1)NCC(CNC(C1=NN(CC)CC1)=O)OC C1(C(N2CCC(C(N3CCC(C)(N(C)CC)C3)=O)(CC)C2)=O)CCCC(=O)N1C Cc1c(C(=O)NC2CC2)cnn1C(C)C(C)(C)O.C1(C)(CC=O)CCCO1 C1(C(=O)OC)C2CCC(O2)C1C(=O)NCCCCC.C(=O)(CSC(F)F)N C12(C(N(CCC(C)NC(C3CN(S(N)(=O)=O)C3)=O)C)=O)CCN(CC1)CC2 C12(CNC(c3cscc3F)=O)CCC(C1)N(C(=O)CCN1CCCC1=O)C2 N1(C(c2cn(CC)nc2)=O)CCC(CNC(=O)CC(C)N(C)C)C(O)C1 CCC1=NOC(C(=O)NCC(C)(CO)NC(c2cnc(O)s2)=O)C1 CC(C)CC(C(=O)N1CCN(C(c2cn(C3COC3)nn2)=O)CC1CO)C(C)C N1(C(C(CNC(C)=O)(C)C)=O)C2CCC1C(C)CC2.C(=O)(C(F)n1cccn1)N N(C1c2ccccc2B(O)CS1(=O)=O)C(=O)NC1C(C)(C)CCCC1(C)C C(=O)(CCCCC(C)CC)NC(CC(=C)C)C(=O)N(C1CC(C)CC(C)C1)C N1(C(C2COC(=O)O2)=O)CCOC2(CCCN(C(C3CCCS3)=O)C2)C1 CC1CN(C(c2ccc([N+](=O)[O-])s2)=O)c2ccccc2N(CCO)C1 c1(CCC)[nH]ccc1C(=O)NCCCOCCNC(C1CC1F)=O c1(C(=O)NC(C)CNC(=O)C(c2ccccc2)=O)ccc(CC(N)=O)cc1 N1(C(C(C2(C)CC2)NC(CC(C=C)(C)C)=O)=O)CCC2(CCOC2=O)C1 N1(C(c2cnn(C)c2F)=O)CCC2(CCCN2C(c2cc3ncccc3o2)=O)C1 N1(C(COCCOC)=O)CCC(C2CN(C(c3nscc3Br)=O)C2)CC1 N1(C(CNC(C(n2cc3ccccc3n2)C)=O)=O)Cc2ccccc2C1 C1(C(c2ccc(C)nc2)N(CCOC)C)CCCCN1C(=O)OC(C)(C)C Cc1cc(C(N2CCC(CNC(=O)C(C)(C)C3CCCO3)C2)=O)c(Cl)cn1 N1(C(c2cnc(CC)s2)=O)CCC(C)(C)C1CC(N1CCC(CCO)C1)=O C=CCC(C)C(=O)N1CCCC(N(C(=O)CCN2CCC(O)CC2)CCF)C1 C1(C(=O)NC(c2ccn(C)n2)C)CC(C)(C)CCN1C(c1cnns1)=O C(c1c(Cl)cccc1Cl)=C(C(=O)NCCCCCN(C(C(CC)(C)OC)=O)C)C N1(C(c2[nH]cc(C)c2C)=O)CCC(C(=O)N2CC=C(CO)CC2)=C(F)C1 C(=O)(C#CC1(C)CCCO1)NC1(C(=O)N)CCN(C)C1.C1(C)CC(F)(F)C1.C C(=O)(CC(C)C(=O)OC)NC(C(=O)NCC1N(CC)CC1)CCC1CC1 c1c(Br)cc(F)cc1[N+](=O)[O-].c1(CC)cc(C=O)n[nH]1.C12CC(C=O)(C1)C2.N CCC(C(=O)NC(c1nocc1C(=O)NCC1(F)CCC1)C)C(C)C c1(C(N2CC(C)N(C(C3(C)CCCO3)=O)CC2)=O)ccc2sc(O)nc2c1 c1(C(=O)N)ccc(C(C)C)c(F)c1.C(C)(CCC)NC(C(C)OCC=C)=O CC1(C(=O)NCC2(O)CN(C(c3ccc(O)cc3F)=O)C2)CCOC12CC2(F)F C(=O)C(C(C)C)C(C)C.C1(OC)CN(C)C(C)(C(=O)N)C1.C1(F)CCC1.C C1(C(=O)NC2CC(CNC(C3CC(OC)C3)=O)C2)CCC(C)(C)CO1 c1(N(C23CCC(N)(CC2)C3)C(c2ccn(CC)n2)=O)ncnc2c1CCC2 C1(C(N2C(CCN(C(=O)CN3CC4CC4C3)C)CCCC2)=O)CC2(CCC2)CO1 C1(CCCNC(=O)CC2CSCCS2)CCCCN1C(c1ccccn1)=O C(=O)(CC1OB(O)c2ccccc21)N1CC2CC(CNC(CCC=CC)=O)C2C1 N1(C(C(C)N(C)C)=O)C2CCC1(CNC(=O)C(c1ccc(Cl)cc1)O)CC2 c1(OC)ccc(C)cc1CC(=O)NC1COCCN(Cc2cc(Br)ncc2F)C1 C1(NC(=O)C#CC2CC2)CCC2CN(C(=O)C3=CCCCO3)CC2C1 N1(C(CC2(N(C)C)COC2)=O)CC2(CC(C(=O)Nc3cnc(F)nc3)CO2)C1 C(=O)(CCCCCn1cc(C2CC23CC3)nn1)NCc1cccc(CCC)c1 CCC(C(=O)N1CC(NC(C2C(C(C)=O)C2(C)C)=O)C1)c1ccccc1 CC1OCCN(C(c2ccc(C(=O)NCCCO)cc2)=O)C1C C1(C(=O)NCc2c(C)noc2C)CCC2(CN(Cc3cccc4c3OCO4)C2)O1 C1(NC(C2(NC(=O)CC3CC4C=CC3C4)CCSC2)=O)CCC2(CCC2)C1 c1csc(C=O)c1.C(=O)(C(CC)OCC)N(CCC(=O)NC(CC)C)CC C(=O)(CS(=O)(=O)c1ccccc1C)NCCC1CC(NC(C(CC#C)O)=O)C1 C1(N(C(CC=CC=C)=O)C)CCN(C(C2CCC(COC)C2)=O)CC1 N1(C(=O)CSC(F)(F)F)CCCC2C(CCCN2C(=O)CCn2ccnc2)C1 N1(C(C2(F)CN(C(=O)Cc3ccsn3)C2)=O)C(CO)CCC1CO c1(C(=O)N)nc(C)[nH]c2nccc1-2.C1(CC)CCCC1C(=O)N(CCC)CCO c1(C(N2C(C)CC(NC(=O)CN(C)C)C2)=O)cc2cc[nH]c2cn1 C1(CCC)CN(C(C2CC(=O)CCO2)=O)CC1C(=O)N(C)CCC1CCCC1 C(=O)(CCCN=c1nccc[nH]1)N(C)CC1CCCN1C(=O)CCOCC1CC1 C1(C)(C)C(OC)C(=O)O1.c1(NC(C(C)OC)=O)cccc(C)c1 c1(CNC(C=C(CCC)C)=O)cn(CCC)nn1.c1(CCC=O)ncc(C)[nH]1.N C=CC1(C(=O)NC2CCCC2NC(=O)C=Cc2cc[nH]n2)CCCC1 N1(C(=O)NC)CCC(C=O)CC1.c1(C=O)cnc(C(C)(C)C)o1.CC(C)C.N Cn1ncc(=NC(=O)c2csc(NC(c3ccccc3C3CC3)=O)n2)[nH]1 c1(CC(N2CC(NC(C(=O)NCCCC)=O)(CO)C2)=O)c(C)noc1C c1(C(=O)NC(c2ncc[nH]2)CC)cccc(C2COC2)c1 C1(C(=O)NC2CC(C)(NC(=O)CC3CCC(C4CC4)O3)C2)C=CC=CC=C1 Cc1ccc(OCC(=O)N(C2CCN(C(=O)CCC3(C)CC3)C2)C)cc1 N#Cc1ccc(NC(C2CCCC2NC(=O)Cc2cccc(Cl)c2)=O)c(C#N)c1 N1(C(C(C)CO)=O)CCN(C(=O)C(C)n2cccn2)CC(C)(F)C1 c1(C(=O)NCCCN(C(c2cc(C)c(C(F)F)cn2)=O)C)c[nH]c(C)c(Cl)c1=O C1(C(=O)NCC2(C(C)(C)O)CN(C(C3OCCO3)=O)C2)CCC12CCCO2 c1(CN(C(=O)C=O)CC)cncc(C(=O)NCC2CC23CC3(F)F)c1 C1(O)(CC#C)CC(C(=O)NCC(C(=O)N(C)Cc2ncnn2C)OC)C1 c1(C(N2CCC(C(C)O)C2)C(=O)NC)ccc(F)c(OC)c1 C12(C(N(CCOCCCNC(Cn3c(C)ncc3)=O)C)=O)CCCCC1OCC2 N1(C(COCc2cc(C)on2)=O)CCOCC(NC(c2cnoc2C2CC2)=O)C1 N1(Cc2c(C)cccc2O)CC(C)CC(F)(F)C1.C1(CC(=O)N)CC2CCC1C2 CCC(CC(F)(F)F)C(=O)NCC(C(C)C)NC(c1cnc(C(F)(F)F)cn1)=O C(=O)(C1=CS(=O)(=O)CCC1)NC(C1CCCN1C(c1n[nH]c2c1CCC2)=O)C N1(C(c2cn(CCNC(c3ccc(F)c(F)c3)=O)nn2)=O)CCC2CCCCC12 N1(C(C2CCCSC2)C(=O)NCC(F)F)CCOC(C2CCCO2)C1 C1(CNC(N2CCCC2C2CCOCC2)=O)CC2C=CC1C2 C1(C(N(C2CC(CO)C2)C)=O)COCCC1NC(c1cncc(Cl)c1)=O N1(C(C=C(CC)C)=O)CCN(C(=O)C(C(C)C)n2ccnc2)C(CCO)C1 c1(C(=O)NCC2(CN)CC3(CCC3)C2)c(Cl)ccc2ccncc12 O=S(CCN=C(NCC1CCC1)NCC1CCC2(CC1)CC2)c1ccccc1F c1(OC)ccc(C(N2CC(CNC(c3csnc3O)=O)C(C)C2)=O)c(C)c1 c1(CCC(=O)N)ccc(F)c(F)c1.C(C(O)C(=O)N(C)CCOCCC)SC O=C(C(CC1COCCO1)C(F)(F)F)OCC(C1CNCCC12CCC2)=O O=C(C1=C(Cl)CCCC1)NC1CN(C(=O)Cc2cc(O)nc(O)n2)C2(CCC2)C1 C1(CC(=O)N(CCN(C)C)C)CCN(C(c2ccnc(CO)c2)=O)C1(C)C C1(C)(CNC(c2c(CC)occ2)=O)CCCC1NC(c1sc(O)nc1C)=O CC(C)CCCC(C)C(=O)N(CC(CO)(CO)NC(C1CCCN1C)=O)C c1(C=O)ccccc1.C1(CNC(C(C)OCC#C)=O)CCCN1C(=O)C C=C=CC(C)C(=O)NC1(CCCNC(c2c(C3CC3)noc2C)=O)CC1 c1(C(=O)NCCCCC(C)NC(=O)CCC2CCCOC2)cccn2ncnc12 C1(CCNC(CCNC(=O)C=CCl)=O)CCCN(C(C2CC(F)(F)C2)=O)C1.C Cc1ccc2c(C(N3CCSCC3CCNC(C3(C)CCCO3)=O)=O)n[nH]c2c1 C1(CC(N2C3C(NC(CCC(C)(C)C)=O)CC(C3)C2)=O)Cc2cc(F)ccc2O1 CC1COCC1(c1nnnn1C1CCCC1)NC1CCS(=O)CC1 c1(C(=O)OCC)cc(N2CCC(C)(NC(C3CCCCC3C)=O)C2)nc(C)n1 c1(C(c2n(CCSC)nnn2)NC(c2nnc(C)s2)C)ccc(Br)cc1F C12(CNC(C(C)(C)OC)=O)CCCCC1CN(C(=O)COc1ccsn1)C2 N1(C(C2N(C)CCCCC2)=O)CCN(C(=O)Cc2cccnc2Cl)CC(O)C1 c1(OC)ccc(OCCC(=O)N)cc1.C12CC1CN(C(C13CSCC1C3)=O)C2.C O=C(CC(O)C1CCCC1)NCC1(O)CN(C(C2CC(OC(F)F)C2)=O)C1 c1(OC)cc(C(N2CC(NC(=O)C(C#N)C(C)C)C2)=O)cnc1OC Cc1cccc(Oc2ccc(NC(=O)CN3CCCC3C)cc2)n1 c1(-c2nc(-c3ccnc(CC(C)SC)n3)on2)ccc(Br)c(F)c1 C(=O)(C(CNC(C1CCN(C)CC1)=O)CC(C)C)NC1CCN(CC)C1 CCC(C#N)(CC)C(=O)N(CC(O)CN(C(=O)C(C)(C)CC1CC1)C)C N1(C(C(C)C2CCOC2)=O)CC2(NC(=O)CCC(=O)N3CCOCC3)CC1C2 c1(C(=O)NCC(CC(C)C)NC(c2n[nH]cc2Br)=O)ncc(Cl)nc1Cl C1(Cc2nnn[nH]2)CCC(F)(F)CC1.N12CC1CC2=O.CCC c1(CC(=O)NCC2COCC2NC(=O)CN2CCOCC2)cc(F)ccc1F c1(C(N2CC(CNC(C3(CO)CCCO3)=O)C(O)C2)=O)cc2ncccc2o1 CCC(C)CC(=O)N1CCCC1(C)CNC(=O)CSCC(N1CCOCC1)=O c1(C(=O)NCC2C(NC(=O)C3=COCCO3)C2)cc(Cl)c(F)cc1F c1(C(=O)NC(C(C)NC(C(C)=CC2CC2)=O)C)cc2cc(C)[nH]c2cc1Cl n1(CC=O)c(=O)c(=O)[nH]c2ccccc12.C1CCCCC1.C(C(=O)NC)=CC CC1(C)CCN(c2nnc(C3CCCCC3)n2CC2CCCC(F)(F)C2)CC1 C1(OC)CC2(CCN(C(C3CN(C(=O)C4=COCC4)CC3OC)=O)C2)C1 C1(C(=O)NC(CCN(C)C)C(=O)NC[Si](C)(C)C)CCCCC1(C)C C(=O)(CCCC(C)(F)F)N1C(C)CCC(NC(c2ccnn2C)=O)C1 C1(C(N2C3CC(C3)C2)=O)CCOC(C)(C)C1.c1(CC)nc(C)c(C(=O)N)s1.C N#Cc1ccncc1C(=O)NC(CC1CCC1)C(N1CC2CC1CS2)=O C1(C2CCN(C(c3cnsc3)=O)CC2)(NC(c2c(SCC)n(C)cc2)=O)CCC1 c1(CC(C(=O)NCCCN(C(=O)Cc2ccnc(O)c2)C)O)cccc(Cl)c1 C12(C(=O)OC)CCCC1(C(=O)OCC1CC(=O)C1)C2 c1(OC)ncc(Cl)c(C)c1C=O.C1CN(C(=O)CC2CC23CC3)CC12CCC2.N N1(C(CCN(C(C2C(C)C2)=O)C2CC2)=O)CCCC2(C=CCO2)C1 c1(C=O)ccc(F)c(O)c1.C(C)(C)(C=O)NC(=O)NCC.C1C=CCC1 C(=O)(C1=NN2CCC(C)N=C2N1)NCC(C)NC(c1c(C#C)c[nH]n1)=O c1(CN2CCC3CC23)nc(N(C2CCNC2)C)nc(-c2ccncc2)n1 C(CC(C(=O)N(C)CCOCCO)NC(=O)Cc1cc[nH]n1)OCC C(CCCC(C)NC(=O)CN1CCCNC1=O)NC(c1c(C)nc[nH]1)=O C(=O)(CCC(F)(F)F)N(C1CN(C(C2CCC(CCO)CC2)=O)CC1O)C C1(C(=O)NC2(CCCNC(c3csc(-c4nc[nH]n4)n3)=O)CC2)CCCCS1 c1(C(N2CC(C(=O)NCC(COCC)C)C(CC)C2)=O)nc(C)ccc1C c1(OC)cccnc1C(=O)NC1CN(C(=O)CSc2nnc(S)s2)CC1O O=C1NC(=O)C2(CC(C(N3CCCCC(NC(=O)Cc4cnc[nH]4)C3)=O)C2)N1 N1(C(C(CC)(C)O)=O)CCCC(F)(CNC(C2CC3C(C2)C3(C)C)=O)C1 c1(C(N2C(CNC(C=CCC)=O)COC(C)(C)C2)=O)cc2nc[nH]c2cc1F C1(C(N2CCN(C(=O)OC)CC2)=O)(NC(C(CC)C)=O)CCN(C)C1 C1(C(=O)N(C)CC2CCCCC2)(OC)CS(=O)(=O)C1.C(=O)C.C(N)=O c1(OC)cccc(C(=O)NCCCCC(C)NC(C2CC(CF)C2)=O)c1 N1(C(CCC(C)SC)=O)CC(CNC(=O)CC(C)(F)F)OC2(CCC2)C1 c1ccnc2[nH]ccc12.c1(C=O)nnnn1CC(F)F.O=C(C1CC1)NC.CC C1(C(N2CC(O)(CNC(C3N(C)C(=O)CC3)=O)C2)=O)CCc2ccccc2C1 c1(C(=O)NC2CCC(NC(C(CC#C)O)=O)C2)cnn2ccc(OC)cc12 C(C1(C)OCCc2sccc21)NC(=NCCC1(C)CC1)NCC1(C2CCC2)CC1 C1(C(=O)NCCC2CC(NC(c3cnn(C4CC4)c3Cl)=O)C2)CCCNC1=O CC(O)C(C)(C)C(=O)NC1C=CCN(C(=O)CCC2CCCCN2C)C1 S(=O)(=O)(c1c(Br)cccc1Cl)N1C(CCC(=O)Nc2c(NC)nccc2)CCC1 C(=O)(CCCC(=O)Nc1c(C)nn(C)c1OC)N1C(C(N)=O)CC(=C)C1 c1(C(=O)NC2CN(C(CCCC=C)=O)C(CO)C2)c(Cl)ccc(Cl)c1OC CC1=C(C)CC(C)(C(=O)NCC2CCN(C(=O)Cc3[nH]cnc3C)CC2)CC1 C(C(=O)Nc1cccs1)(C1=CCC2CC1C2(C)C)N(CC(=O)NC)CC=C C(C)(CCC(=O)NC1CC(OCC(=O)N(CC(C)OC)C(C)C)C1)OC N1(C(CCCC)=O)CCC2(CC1)CCN(C(=O)C(F)(F)C(F)F)C2 N1(c2cc(C)nc(NC(CC(N)=O)C3CC3)n2)CCc2nc(CO)sc2C1 c1(NC)cc(=NCCCCCCNC(c2ccon2)=O)nc(-c2ccncc2)[nH]1 Cc1oc2ccc(NC(=O)C(=O)NCCN3CCC(O)CC3)cc2c1C C1(NC(COCCCOC)=O)CCC(C(N2CC(C)(O)C2)=O)CC1 C1(CN(C)CC)CCN(C(=O)CCN(C(C2SCC=C2C)=O)C(C)C)C1 C1(NC(C(C)C)=O)CC(C)C1.C(=O)(C(O)C1CN(C=O)C1)N.C(C)(C)C N1(C(C(COC)OC)=O)CCCCC1C1CCN(C(C2CC(F)CN2C)=O)C1 c1(C(=O)OC)cscc1CC(=O)NCC1(O)CN(C(=O)C=C(Cl)Cl)C1 c1(C=O)n[nH]cc1[N+](=O)[O-].N1(C(C2C(CC)CCC2)=O)CCN(CC2CC2)CC1 Cc1ccc(C(F)(F)C(N2CCOC(C(C)NC(C3CNC(=O)C3)=O)C2)=O)cc1 C(C1=NOC2CCCC12)NC(C(Cc1cc[nH]n1)NC(CN(C)CC)=O)=O c1(C(C)NC(CCN2CCC(CC(C)CO)CC2)=O)cccc2ccccc12 c1(CNC(CCSCCC)=O)ccc(CC)cc1.C(=O)(CC(C)n1cccc1)N Cc1cc(N(C)Cc2ccccc2Cl)nc(NCc2cn(C)cn2)n1 C(CC(C)(C)C(=O)N1C(C(=O)NCCCc2ccccc2)CC1C)SC c1(C(N2CCCC(F)(C)C2)=O)cc2cccnn2c1.C12(C(=O)N)C=CC(CC1)C2 c1(C(=O)NCC(CC)(C)NC(c2cc(C)ccc2OC)=O)cn2cccnc2n1 c1(CC(C)OC)nc(-c2c[nH]c(-c3ccc(F)cc3)c2)n(C23CC(C2)C3)n1 c1(-c2nnn(CC(N3CCC(NC(CC(=C)C)=O)C3)=O)n2)ccc(C#N)cc1 S(=O)(=O)(C=Cc1ccccc1)N1CCN(C(C(c2ccccc2F)C)=O)CC1 c1(CCC(=O)NC(C(C)NC(c2[nH]cc(C)c2)=O)(C)C)ccnc2ccccc12 C(=O)(CC(C)NC(=O)CCOCCC)N(C(C)C)C.C12(C(=O)N)CC1C2 C(CC=CC)(C(=O)N(C1CCC(F)(F)C1)C)NC(CC1CC(=C)C1)=O Cc1[nH]c(C(C)(C)C)cc1C(=O)NC1CCC1.C(C1CCCN1C)=CC=O.N c1(CC(=O)NC2CC2F)cc(NC(N2CCCC2c2ccc(Br)cc2)=O)ccn1 C(=O)(C(C)(C)C(O)CC)N(CC(CC)NC(c1cc(NS(C)=O)ccc1F)=O)C C(=O)(CC1=CCCCC1)NC1CCC(C(=O)NC(C23CCC(CO2)C3)C)C1 C(=O)(C(C)(O)C(C)C)NCC(c1ccc(CC)cc1)N(C)C c1(C(=O)NCC2N(C(C(C)N(CC(F)(F)F)C)=O)CCC2)cc2c[nH]cnc-2n1 c1(OCC)ncnc2c1CN(C(C1(CCc3ccc(F)cc3)CCC1)=O)CC2 c1(C(=O)NC2C(NC(=O)C=Cc3ccc[nH]3)CCCC2)cc(Cl)cc2c1OCC2 C1(NC(c2nnc(C)s2)=O)CCCCN(C(c2cccc(F)c2C)=O)C1 CC#CCCC(=O)N(C)CC1CCC(CNC(=O)C(O)Cn2cncn2)CC1 C1(C=O)CCCCC1.CNS(=O)(=O)NCC(=O)N.C1(F)CCC1.C(C)=O.C C1(NC(C=CC(=O)N(C)C)=O)CCN(C(c2ccccc2O)=O)CC1O C(=O)(C(O)CCC(C)C)N1CCC(NC(c2c(CC)oc(C)c2)=O)(CO)CC1 N(C1CC(C)n2ccnc21)C(c1cc(CNC(C2CCN(OC)CC2)=O)sc1)=O NS(=O)(=O)c1ccc(CC(=O)NCC2(C)CC2)s1.C(=O)C.CCC#N.N N1(C(CC(C)c2ccco2)=O)CC=C(C(=O)N(CCCC(O)CO)C)CC1 c1(C(CNC(C2CSCN2C(=O)CC2CC2)=O)O)cc(F)cc(Cl)c1 CCCCCCn1nnnc1C(c1cc(C(C)(C)C)on1)NC1CC(C)C1 Cc1cc(C(=O)NCC(C)(C)NC(=O)C)c(C)o1.c1(C(=O)N)ccccn1 CC(C)C(C)C.c1(C=O)cnn(C)c1C(F)(F)F.c1(C=O)cc(=O)cc[nH]1.N C1(OC)CC(CC(N2CC(O)(CCNC(=O)CCn3cnnn3)C2)=O)C1(C)C N1(C(c2n(CC)ncn2)=O)CC(NC(=O)Cc2ccccc2Cl)CC(C)(C)C1 N1(C(c2cccc(C)c2)=O)CCC(Nc2ncnc(C)c2F)C(C)C1 c1(N2C(=O)CC(C(N3CCC3C3CCC3)=O)C2)ccc(F)c(F)c1F n1(CC(=O)N)ncccc1=O.c1(C(C)NC(CC2CC(CC)C2)=O)ccccc1 C1(C(C)C)CC(CC(=O)NC23CC(NC(C4CCCCO4)=O)(C2)C3)CCO1 C1(CCNC(=O)C(=O)NCC(F)(F)F)CCCN1C(C1CC=CCC1)=O c1(C(N2C(C=C)CCCC2)C(=O)NCCOC)ccc(OC)c([N+](=O)[O-])c1 CC(CC(=O)NC1CC(C)(NC(=O)C=Cc2cccc(O)c2)C1)C(F)F c1(C(=O)N)nc2c(s1)CN(C)CC2.CCC(C(=O)NCC1CC1)C1CCOCC1 C1(C2CCCCC2)CCC(O)CC1.C1(C(=O)OCC)(CNC=O)CCCC1.N c1(C(N2CCCC(C(N)=O)C2)C(=O)NCC)ccc(OC)c(C)n1 N1(C(C(C(C)(C)C)O)=O)CCCC2(C1)CN(C(c1cn3c(n1)CCCC3)=O)C2 N1(C(c2ccc(C(N(CCC(C)O)C)=O)cc2)=O)CCC2(CC(=O)NC2=O)C1 N1(C(c2ccn(C3CCC3)n2)=O)CC(CO)C2(C1)CN(c1ncc(Cl)c(O)n1)C2 c1(CNC(C(c2c(CC)cncc2)N2CCC3CC23)=O)cccc(Cl)c1C Cc1cccc2c1OC(C(N1CCN(c3ncccc3C#N)CC1C)=O)C2 C12(CNC(c3c(C)n(C)cn3)=O)CCC(CC1)CN2C(=O)C=CC1CC1 C1(NC(CC2N(C)CCC2)=O)CCN(C(=O)Cc2ccc(F)nc2)CC1O C(=O)(C1=CCCCCC1)N1CCC(F)(CNC(C(C)Nc2ncccn2)=O)C1 c1(NC(=O)CC2CCC2)cccc(CNC(C2CCCC(F)C2)=O)c1 n1(C(C)C)ncc2c(O)nc(N3CCC(NC(=O)OC(C)(C)C)C3)nc12 C1(CN(C)C(c2cc(Cl)c[nH]2)=O)CCCC(NC(=O)C(CO)N(C)C)C1 n1(CCC)cccc1C(=O)NC(CO)C(C)NC(c1ccsc1OC)=O C(=O)(C1CCc2nccn21)N1CCC(C)(C)C1CC(=O)NCC1CC(O)C(O)C1 C1(C(N2CC(CC)(NC(=O)CCc3cc(C)no3)C2)=O)CCCCC(=O)N1 N1(C(CP(C)(C)=O)=O)CCC2CCN(C(c3ccc(CSC(F)F)o3)=O)C2C1 N1(C(COc2scc(C)c2)=O)CCN(C(=O)COC2CC=CC2)C(C)C1 C1(NC(c2nccc(CC)c2)=O)CC2CC1N(C(=O)C=C(C)c1ccco1)C2 C1(CNC(C(Cc2ccco2)NC(c2c(C)ccs2)=O)=O)CCCN(C)C1 c1ccc2c(C(N3CCC(F)(F)C(F)C3)=O)ncn2c1.C(C)(C(=O)N)NC(C)=O C(=O)(CCCC(C)NC(c1ccc(CC#N)cc1)=O)NCCCCCC c1(C=O)ncoc1-c1cccs1.C(C(=O)NCC=O)N(C)C(N)=O.C1CC1 c1(C=O)cc(C(C)C)[nH]c1C(C)C.C(C(C)(C)C)NC(C1CC1)=O.C Cc1cc(C(=O)NC2COC(C(C)C)C2)cc([N+](=O)[O-])c1Cl N1(C(c2n(CC#C)cnn2)=O)CC(C)C(C)(C(N2CCCCCCC2)=O)C1 CN1CCCC(NC(c2ccccc2CN2CCSCC2)=O)CC1 c1(CC)nc(C)c(CC(N2CCCC(NC(=O)CC3(C)CC3)CC2)=O)c(C)n1 C1(C(=O)NC2(C)CC(NC(=O)Cn3cnc(=N)[nH]3)C2)CCC2CCC12 C1(N(C(COC)=O)C)CN(C(=O)Cc2ccc(O)cc2)C2CC12.c1cc(C)cs1 C1(CC#C)(C(=O)NCC(C2CC2)N(C(=O)Cc2cncn2C)C)CCCCC1 c1(C(N2CCCC2)=O)sc(C(C)C)nc1C.C=C1CC(C(F)(F)F)(C(=O)N)C1 N1(C(C2(CCC=C)CN(C(=O)C(C)CC)C2)=O)CCCC(C)(C#N)C1 Cc1ccc(O)cc1C(N1CCC(F)(C(=O)NC(C)C(C)F)C1)=O c1(C(=O)NC2C(CNC(=O)C=Cc3ncco3)C2)cccc2sccc12 C1(C(N2C(CCNC(c3cccc(O)n3)=O)COCC2)=O)CCc2cnnn2C1 N1(C(C2C(C(=O)OC)C2)=O)CCCC2CCCCC12.C12(C(=O)N)CC(CO1)C2 C1(C(=O)N)CCCCC1.C1(C)(C(=O)NCCC)CCCC1.C(C)(C)C.C=O N1(C(c2n(CCC)ccc2)=O)CCC(N(C)C(C2(COCC)CCC2)=O)CC1 C(N=c1[nH]c(N2CCC(C)(CC3CC3)CC2)nc2cccnc12)c1ccn(C)n1 C1(C(=O)NC(c2cnn[nH]2)C)CC(NC(C2CCCC2F)=O)C(O)C1 C1(CCC(=O)OC)CCC(C)N(C(=O)NCCCCCC(C)C)C1 c1(C(N(CC(N)=O)C)=O)cc(S(=O)(=O)NC2CC2)c[nH]1 C1(NC(CCCOCC)=O)CCCCCC1C(=O)N(CCS(=O)CC)CC c1(C(=O)NCC2N(C(C3N(C)C(=O)NC3)=O)CC=C2)cnc(O)n(C)c1=O C(CC(C)(C)CC(=O)N1CCC(O)(CNC(C2CCC(C)(C)OC2)=O)CC1)OC N1(C(CN2CCN(CC)CC2)=O)CC(CNC(=O)Cn2nccc2C)CCC1C N1(C(C(C)OCC)=O)CCCC(NC(C2(CF)COC2)=O)C1 c1(C(N2CCC3(CC(NC(CC)=O)C3)CC2)=O)cc(=O)c2ccc(Cl)cc2o1 c1(C(N2CC(NC(CN(C(C)C)C)=O)C3C(C2)C3)=O)cccc2ncnn12 N1(C(c2cc(C)ns2)=O)CC(NC(=O)C(c2ccc(F)cn2)(F)F)CC1C N1(C(C2CCC(CC#N)CC2)=O)CC2CC(NC(=O)CN3CC4CC4C3)CC1C2 CC(C)C(=O)CCc1cccc(NC(C2CSC(c3ccccc3)C2)=O)c1 CC1=CCC=CC1C(N1CCC1C(N1CCCC(Br)C1)=O)=O C=CC1(C(N2CCC(C)CC2C)=O)CCN(C(C2C3CCCOC23)=O)C1 C(=O)(C1=C(Cl)CCOC1)N1C(C)CCC(NC(c2ccc(C3CC3)cn2)=O)C1 C1(C)(C(N2CCCCC2)=O)CCCNC1=O.CN1C(=O)CCC1C(=O)NCCO c1(NC(=O)COC2CC(NC(C34CCCC3C4)=O)C2)cccc(F)c1O n1(CN(CC)Cc2cc(-c3cc(F)ccc3C)n[nH]2)nc(C)c(CN)c1C N1(C(CCC(=O)N(C(C)C)C)=O)CCC2(NC(c3ccc(O)nc3)=O)CCCC12 N1(C(c2c(CC)[nH]cc2)=O)CC2(NC(c3occc3C)=O)CC1C2 C(=O)(C1=CS(=O)CCC1)NC1(C)CN(C(c2cccc3c2OCC3)=O)C1 N1(C(c2cncc(C(=O)OC)c2)=O)CC=C(C)CC1.C1(C(=O)N)CC12CCCC2 CC1CN(C(=O)COc2ccon2)CCC1NC(c1cncc(F)n1)=O C(CC)(C(=O)NC1CCN(CCCNC(=O)C)C1)OCC.C1(C)CCCC1 C1(NC(=O)CCCc2ccsc2)C=CCN(C(=O)C(c2cccc(Cl)c2)(F)F)C1 N(C(=NCCF)N(C)Cc1ccc(Br)cc1C)Cc1c(CC)n(C)nc1 c1(OC)cccc(C(F)(F)C(=O)N(CC(C)(C)C)C)n1.C(=O)(C)N.C(C)C Clc1nc(NC2CC3CC4CC(C3)C2C4)c2[nH]ccc2n1 Cc1cc2c(C(=O)NC3CN(C(=O)COCC(F)F)CC3C3CC3)cccc2o1 N1(C(Cn2ccc(C(=O)OC)n2)=O)CCCOC(CNC(=O)C(C)C(C)O)C1 N1(C(C(COC)OC)=O)CC(=O)CC1C(N1CC(CO)C1(C)C)=O c1(C(N2C(C)(CNC(=O)CCCF)CCC2)=O)ccc2c(=O)cc[nH]c2c1 C1(C(N2CCCC(CNC(C3C=CCC3)=O)C2)=O)CCCCCCC1 C1(N(C(CCOCC)=O)CCO)CCN(C(=O)C(CC)Sc2ccccc2)C1 N1(C(c2cc(CC)on2)=O)CCC(O)C(NC(c2c(Cl)cccc2Cl)=O)C1 CC1(C)C(NC(C2(NC(c3ccc(O)cc3)=O)CSC2)=O)CC1(F)F C(N=c1[nH]c(=NCc2cncc(Br)c2)[nH]c2c1COC2)C1(OC)CCCSC1 c1(CNC(c2nc(CC(C)C)sc2-c2ccccc2)=O)nc2c(s1)CCC2(C)C C1(NC(CSS(C)(=O)=O)=O)CCN(C(c2ccc3snnc3c2)=O)CC12CCC2 N1(C(c2n3cc(C)sc3nc2C)=O)CCCC(C2CCN(C(=O)C3=CCC3)C2)C1 c1(C(N(C2CCCN(C(c3cc(Cl)ns3)=O)C2)CC)=O)n[nH]c2c1COCC2 C1(NC(c2cc(C)nnc2)=O)CC2CCC1N2C(=O)C=Cc1ccccc1F C=CCC(C)(C(=O)N1CCCCC1CNC(=O)C=CC1CC1)N(C)C C(=O)(NNC(=O)C(C)C1CCN(C(C)C)C1)c1nnc(-c2cncc(C)c2)o1 CCC(CC)C(=O)NCC(c1ccc(C)cc1)NC(C1CC(OC(F)F)C1)=O N1(C(c2cncc(OC)n2)=O)CC2CCCC2(NC(=O)CC2CCC=CCC2)C1 C1(C(C)C)CC(CC(=O)NCC23CC(CN2c2cc(C4CC4)ncn2)C3)CCO1 C1(O)(C(=O)NCCCC(C)C)CCC(C)(C)CC1.C(c1cnc[nH]1)=CC(=O)N N1(C(C2(C#C)CC2)=O)CC2(CCCN(C(=O)C(C)(C(C)C)NC(=O)C)C2)C1 CC(C)C(N=c1cc(Cl)c(O)n[nH]1)CNC(c1ccnc(CO)c1)=O c1(C(=O)NC(C2(O)CCN(C(c3n[nH]c(C)c3N)=O)C2)C)cc(O)cc(O)n1 C1(C(=O)NC2C(CC(=O)NCc3scc(C)c3)CCCC2)CCC(=O)CC1C N1(CC(=O)OC)CCC(C)(C)CC12CNC2 CC1C(NC(c2scnc2C(F)F)=O)CCCN1C(=O)CCn1cccc1 CCCCCC(O)C(C)C(=O)NC1CN(C(C2CC(F)(F)C2)=O)CC1OC C1(C2CCN(c3nc4cc(Cl)ccc4s3)CC2)(NC(C(C)N2CCC2)=O)CC1 C1(CNC(c2ccc(C3CCOC3)s2)=O)CCCCN1C(=O)C=C1CC1 C1(C(=O)NC2CCC(NC(CCCC)=O)C2)Cc2cc(Br)ccc2O1 n1(CC)nc(C(=O)NCC2(C)CCN(C(=O)Cc3ccnnc3O)C2)cc1C C1(CNC(C2(C(N)=O)CC2)=O)CN(C(=O)C#CC2CCOC2)C2CCCCC12 N1(C(c2cn(CCNC(CC(C)OC)=O)nc2)=O)CCC2CC12C C1(C(N(CCCNC(c2sc(Cl)cc2Cl)=O)C2CC2)=O)C(F)(F)C12CC2 Cc1cn2c(n1)CCC(C(=O)NCCCCC(C)NC(=O)C(C)C1CCOC1)C2 C1(N(C)CC)CCN(C(=O)C(C)(C)CNC(=O)Cc2cnc(C)s2)CC1 C1(C(=O)NCC(CC(F)(F)F)NC(c2c(C)nn(C)c2)=O)CCCCC12CCC2 c1(C(=O)NC2(COC)CN(C(=O)C(C)(C)CF)C2)ccc(C=O)cc1.N c1(CCC(=O)N(C(CNC(C(CC)C)=O)C2CC2)C)nc2ccccc2oc1=O Cn1nc2c(c1C(N1CC(NC(C3CC3c3ccncc3F)=O)C1)=O)COCC2 N1(C(=O)CC(F)(F)F)CCC2(CCCCN(C(c3csnc3Cl)=O)C2)C1 C1(C(=O)OCC)CCCN(C(c2ccccc2-n2ccnn2)=O)C1.[SH](C)(=O)=O C#CCC(C)(C(=O)NC(C)C(=O)NC)NC(=O)CC(O)C(C)C CS(=O)(=O)c1ccc(C(=O)NC2CN(C(C34CCC3C4)=O)CCC23CCC3)cc1 C1(C(C)NC(c2csc(CO)n2)=O)CN(C(C2CC2C(F)F)=O)CCO1 C1(CNC(C2(CCOC)CC2)=O)CCCC(NC(C2CCCCC2C)=O)C1 C(=O)(C1=COCCO1)NC1(C)CN(C(CCc2cnc(C3(C)CC3)o2)=O)C1 C(=O)(C(CC(=C)Cl)NC(=O)CCC)NCC(=O)NCC#C.C(N)=O.N c1(C(=O)Nc2cc(C)c(-n3ccnc3)cc2)c(F)cc(Cl)cc1Br C12(C(N3CC(F)(CNC(CCC(C)OC)=O)C3)=O)CCCC(C1)OC2 N1(C(C(C)CN2CCCCC2)=O)CCCC2C1CCN2C(=O)C=C1CC1 c1(C(C(=O)NC)N(C2CC2)CC2CCOC2)c(Cl)nc(Cl)n1C Cc1ccc(=O)n(CC(=O)N(CCNC(=O)C2CC2)C2CC2)c1 C1(C(=O)NC(C(=O)OCCC)C)CN(C(C2CC=C(C)CC2)=O)CC12CC2 C1(C(N(C(C)CNC(=O)CCOC2CCC2)CC)=O)CCC(=O)N1 C(C(C)(C)CC(=O)N(C1CCC(C)C1)C)NC(C(C)(C)NC(=O)OC)=O C=CCCCC(=O)NCC1(C(=O)NC(c2cnn(C)c2C)C)CC=CC1 N1(CC(=O)NCCC(C)NC(C2C(C)CCC2)=O)CCCCC(=O)C1=O CC(C)(C)C=CCC(=O)NCCCCNC(=O)CCOCC1CCCO1 CC(C(=O)N1CC(N(C)C)C2(CC2)C1)C(F)(F)C(F)F.C1C2CC3C(C2=O)C13 C1(CC)CN(C(C2CCCN2S(C)(=O)=O)=O)C1.c1(CC=O)cnsc1.CO c1(CC)nccnc1C(=O)NCCC1CCCCN1C(=O)C.c1n[nH]c(C)n1.S N1(C(C(C)=C2CC2)=O)CCCN(C(=O)C(C2CCOCC2)C)C(C(C)C)C1 N1(C(C=NOC)=O)CCN(C(c2cnn[nH]2)=O)CC(CO)C1 C(=O)(CCC(C)(C)C)N(C1CCC(NC(C2C(C(=O)OC)CC2)=O)CC1)C CCCCC(O)CC(=O)NCC12CC(C1)C(C)(C)O2.C(=O)(C=O)N.C1CC1 C1(N(C(c2cnn(CC(F)F)n2)=O)CC)CCN(C(=O)C(O)CCSC)CC1 Cc1ccc2[nH]cc(CCC(N3CCN(C(C4CCC4C(N)=O)=O)CC3)=O)c2c1 N1(C(c2c(C(C)C)con2)=O)CCC(C)N(C(c2cc(F)n[nH]2)=O)CC1 c1(SCC(=O)NC2CC3CCC2N3C(C2(CCF)CC2)=O)nc2ccccc2s1 c1(CC(=O)N)coc2c(F)c(F)ccc12.C(C)(C)(CC(=O)N(C(C)C)C)SC c1(CCC#N)cn(CCNC(c2nn[nH]c2C(=O)O)=O)nn1 N1(C(c2c(C)sc(O)n2)=O)CCC2(CC2NC(=O)CN2CCC(F)(F)C2)C1 C1(C(N2C(CC)C(C(N3CCOCC3)=O)CC2)=O)CC(=O)NC(=O)N1 c1(C(=O)NC2C(C)(OC(C)C)C2)nnc(-c2ccnn2C)o1 C1(CNC(CC2(OCC)CC2)=O)CCCCCN1C(=O)CCC(C)C C=CCC(C)C(=O)N1CCC(CCCNC(=O)C=Cc2nnc(C(C)C)o2)CC1 CCC(C(=O)NC)NC(=O)C(C)CNC(C1CC1[N+](=O)[O-])=O Cn1c(COCC(N2CCC(N(C)C(c3ccc(O)nc3)=O)C2)=O)nnc1S CN1CCC(C)(CNC(C2CCC(NC(C3(C)CC4CC4C3)=O)C2)=O)CC1 N1(C(C2CC(NC(CSC)=O)C2)=O)CC(S(C)(=N)=O)C1 c1(C(N(CCCNC(=O)Cn2cncn2)CC)=O)ccc([N+](=O)[O-])c(N)c1 N(C1COc2c(Cl)cccc21)C(=O)NC1(C#C)COC1 C12CCC(CC1)N2C(c1ccccc1C1(C)CC1)=O.C(C(=O)N)(C(C)C)OC C#CC1(N(C)C)CN(C(=O)C(C)CN(C(=O)C(C)N2CCCC2)C)C1 N1(C(c2nc(C(C)OC)sc2)=O)CCC(CC(=O)OC)C(F)(F)CC1 C1(C(C)NCCC(O)C2CCCC2)OCCC1(C)C C(C(C)C)(C(O)C(=O)NCC(C)NC(c1cc(Cl)no1)=O)OC N1(CC(=O)NCC)CC2CC1CN2C(=O)CCC(C)Nc1nc(CC)oc1C C1(F)(CNC(C(c2cncc(F)c2)C)=O)CCCN(C(=O)CCC(F)(F)F)C1 C(=O)(CC(C)(C)CC)N1C(CCNC(C(CC=C)NC(C)=O)=O)CCC1 C1(C(=O)Nc2ccc(Cl)nc2Br)C2CCC(C2)C1NC(C1CC1Cl)=O C1(NC(C(CN=[N+]=[N-])NC(C(COCC)C)=O)=O)CCCCCC1(C)C C1(O)(C(=O)OC)CCCN(C(C2CCCN(CC3CCS(=O)(=O)CC3)CC2)=O)C1 C(CC(=O)NCC(C)(C1CCC1)NC(=O)C(F)=CCCF)SC c1(C=O)cc(C)ccc1C.c1(CC(=O)N(C)CC2(OC)CCC2)ccnn1C.N N1(C(c2c(CC)nns2)=O)CCN(C2CCC(NC(=O)C(O)C3CC3)CC2)CC1 C1(CCOC)(NC(=O)Cc2ccco2)CCN(C(c2cc(C)ccc2O)=O)CC1 c1(C(=O)NC(CC)CNC(=O)CCc2ccsc2)ccnn1C(C)C c1(C(N2CC(O)CC2CO)C(=O)NC(C(=O)OC)C)ncccc1Br c1(CC#N)cccc(C(=O)NC2CC2CNC(C2CCCO2)=O)c1 c1(C=O)cc2scc(C)c2[nH]1.Cc1nc(CC(C)C)oc1C(=O)NCC1CC1 Cc1cccc(C(N2CC(F)(CNC(C3(C)C=CCCC3)=O)C2)=O)n1 CC(C1CCCCC1)=CC(=O)NCCC1CCCCN1C(=O)C(C)CN(C)C CN1CC2(CCN(c3nc(NCCOC(=N)O)c4ncn(C)c4n3)C2)CC1=O c1(NC(=O)NC2C(=C)COC2)ccc2oc(COC)nc2c1 N1(C(c2ccc(OC)cn2)=O)CCC(NC(=O)CCCCCF)C12CC2 c1(C(=O)NC(CNC(c2cc(OC)cc(Br)n2)=O)C)cc(F)cc(F)c1O C1(C(=O)NCCC2CC(NC(C3CCNC3=O)=O)C2)CCS(=O)(=O)CC1 c1(C(C2CC2)OC(c2occ(C)c2C)=O)c(F)c(F)c(F)c(F)c1F N1(CC(C)C)CCCC1C(=O)NCCCCNC(C1(O)CCSC1)=O C1(F)(CNC(c2nnsc2C2CC2)=O)CCN(C(c2ccns2)=O)CC1 C(=O)(CCC(=O)N1CCC(NC(=O)C(C)(C)SC)C1Cc1ccccc1)OC C(=O)(CCC(C)(C)N(C)C)N(C1CC(C(NOCC=C(C)C)=O)CC1O)C C1(C(=O)N)(C(F)F)CCCCC1.c1(C(=O)NCCC2CCC2)ccc(F)cn1 C1(C(=O)NCc2cn(CCNC(c3cc(Cl)no3)=O)nn2)CC2COCC12 C(CCNC(c1nsnc1O)=O)(C(C)C)NC(C(CC1CC1)OC)=O n1(CC)cc(C(=O)NCC2CC(F)CN2C(=O)CCn2cnnn2)c(C)n1 c1(C(N2CCCC(NC(CCC=C)=O)C2C)=O)cnn2ccnc(C)c12 c1(C(=O)NC(CC)CNC(=O)C2=CCOC2)ccc2c(=O)n3c(nc2c1)CCC3 C12(CNC(C(C)c3ccsc3)=O)CC(CO1)C2.C(c1cccs1)=CC=O.C CC1(CNC(=O)CC(F)(F)c2ccccc2)CN(C(c2ccc(Cl)o2)=O)CCO1 N1(C(CN(CCOC)C)=O)CCC2(C1)CN(C(c1nncn1C)=O)CC(C)O2 C1(CC=O)CCS(=O)(=O)CC1.c1cccc(Cl)c1.C(CN(CC)CC)OC CC1CCN(C(=O)CC2CN(C(=O)CC3(C)CCC3)C(C)(C)C2)CC1O CCC1=CCN(C(=O)CCC(N)=O)CC1.CC(O)C(C=O)NC(=O)O.C(C)(C)C c1(SC(c2snc(C(=O)OC)n2)=O)c(Br)nc2n1CCCC2 C(C(C(=O)NC1COCC1F)C(C)(C)C)NC(C(C)=C1CC1)=O C1(NC(C2CCCCC2CNC(C2CCC(O)C2)=O)=O)CC2CCCCCC12 c1(C(N(C(C(CC)C)C(=O)NC2CC2(C)C(F)F)C)=O)c[nH]c2ccncc12 C(=O)(C(O)P(C)(C)=O)NCC(C)N(C(CN(C)Cc1nnc(C)n1C)=O)C C(CC1CCCc2ccccc21)(C(=O)NC1(C)CC1)N(CC(F)Br)C c1(C(c2ccco2)NC2CN(C(C)=O)C2)nnnn1C(C)(C)C N1(C(C2(C(=O)OC)CC2)=O)CC(NC(=O)C(C(C)C)SC)CC2(CCC2)C1 C(=O)(C1=NOC2(CCOC2)C1)N1C(CNC(c2cn(C)nc2Cl)=O)CC1 CC(N=c1[nH]c2c(c(=NCC3(CO)CC(F)(F)C3)[nH]1)CCC2)c1cnc[nH]1 C1(C)(NC(C(C)SCC)=O)CN(C(=O)CCn2cc(C)cn2)C1 c1(C(N2C(C(=O)Nc3nc(C)c(Cl)s3)CC3CC32)=O)ccc(OC(F)F)c(Cl)c1 c1(C(=O)NC(CC)CN(C(=O)CC(C)OC)CC)n[nH]c2ccc(C)cc12 C1(NC(CC(C)c2cccnc2)=O)CCN(C(=O)CCCCC2CC2)CC1F C=CC(COC)NC(=O)CC1CC(NC(C)=O)C1.C(=O)C.CC(=C)C C1(C(=O)NCCC(=O)NC2CC(CN(C)C)C2)CC=CCO1 c1(C=O)coc(C(C)(C)C)n1.C(C)(C(=O)NCC1CC1)SCCCC.C c1(C(=O)NCCC(C)CCNC(C2CCC(=O)NC2)=O)csc2ccc(F)cc12 N1(C(C2N(C(C(n3ncc(C)c3)C)=O)CSC2)=O)CCCCC1CF Cc1cc(C(=O)NC2CCC3C4C=CC(C4)C23)c2cnn(C(C)C)c2n1 C1(C(=O)NCCN(CCOC)C(c2scc(C)c2C)=O)CCC(C)(C)O1 n1(CC=C)cc(C(=O)NCCN(C)C(c2ncsc2-c2ccccc2)=O)cn1 C(=O)(CCCCCCNC(c1cc(C)c(C)[nH]1)=O)N(CCC#C)CCO c1(NCCNC)cccc([SH](=O)=O)c1.c1ccccc1.C1(C(=O)N)CC1(F)F Cn1ncc(C(=O)NC(CC2CC2)C(=O)N2CCC2C2CCCC2)cc1=O C12(C(N(C3CC(NC(COCCCOC)=O)C3)C)=O)CCC(N=[N+]=[N-])C1C2 C1(NC(c2c(C)nc(CCC)s2)=O)CC(O)CN(C(c2scnc2C)=O)C1 Cc1cc(N2CCC(C)(CNC(=O)CC(C)C(C)C)CC2)c(F)cc1[N+](=O)[O-] N1(C(C2C(C)(NC(C(C=C)OC)=O)CCCC2)=O)C2C=CCC1CCC2 C1(C(=O)NCC2N(C(Cc3c(C)ccs3)=O)CC2)CCCCN1C(=O)CC(C)C C1(NC(C(C)OCC=C)=O)CN(C(c2occc2CC)=O)CC2(CCC2)C1 C(=O)(C#CC1CCCCC1)NCCNC(CC1C(C)(C)C(O)C1)=O CC1CCc2c(C(=O)NC3CCN(Cc4cccc(F)c4I)CC3F)n[nH]c21 C1(C=O)C=CC=CC=C1.C1(C(=O)NCCOCCN(C)C)CCC1C.N C1(NC(C(C)c2cccs2)=O)CCC12CCN(C(=O)CC1(C)CC1)CC2 C(C(=O)N1CC(O)(C)C1)(C(C)(C)C)SCC.C1(C=O)CC(C)(C)C1.N c1(OCCC)ccccc1C(=O)N(C1CCCN(C(=O)CO)C1)CC N1(C(C(CCC)C)=O)CC(CNC(c2ccnc(Cl)c2)=O)OC(C)(C)C1 C12(C(N(CC(C)C(C)(C)C)C)=O)CCCC1CCN2C(=O)CC(C)(F)F N1(C(C(C)OCCCC)=O)CCCC(C(=O)N(C2CC2)Cc2ccoc2)CC1 N1(C(CNC(C(C)(C)C)=O)=O)CCCCC(C2CN(C(=O)C(C)(C)C(N)=O)C2)C1 c1(CNC(c2ccc(OC)c(OC)c2F)c2nnnn2C)cccc2c1CCOC2 CC1(C(=O)NC(Cn2cccn2)C(N2CCOC(CF)C2)=O)CNC(=O)N1 N1(C(CSCC)=O)CCN(CCNC(=O)C(F)(F)C=Cc2ccccc2)CC1 c1(OC)ccc(C(N2CC3CC2C3NC(=O)C)=O)cc1.C1(C=O)CC1C.N N1(C(C23C(C)OC(CO)(C2)C3)=O)CC2(CCN(C(=O)CCCCCF)C2)C1 c1(CC(=O)N)cn(C)c2ccccc12.C1(CC=C)CN(C(C2CCC(C)C2)=O)C1 N1(C(C(C)=CC2CC2)=O)CC(NC(=O)Cc2cc(C)nn2C)C2(CCOCC2)C1 C(C(CC(F)(F)F)NC(c1cc(F)ccc1N)=O)NC(CCOC)=O c1(C(N2C(C(=O)NCC=C)CCC2)C(=O)NC2CCOC2)nc(F)ccc1Br C(=O)(C1=CCCN(Cc2ccsc2Br)C1)N(c1cn[nH]c1)C N1(C(C2(CC=C)CCCN2C(=O)CCn2cnnn2)=O)CCCC2COCC12 C=C(C)C(CC(=O)NC(CC(=O)Nc1cnc(Cl)nc1C)C(C)OC)OCC C(=O)(CC(C)CC(F)(F)F)NC1CCN(C(c2cc(OC)cc(CC)c2)=O)C1 Cc1nc(CNC2CCC(C(=O)N(C)Cc3ccc(Br)cc3)C2)sc1Br n1(CC(N2CCC(C3N(C(CCCCOC)=O)CCC3)C2)=O)cc([N+](=O)[O-])cn1 c1(C(=O)NC(CNC(c2cccc(CC)c2F)=O)C)c(N)ccc(F)c1C C12(C=O)CCCCC(=O)N1CCC2.C1(C(=O)NCCCC)C2CC3C(C2=O)C13.N C1(C(N2C(CN(C(CCCCCOC)=O)C)COCC2)=O)CCCC12OCCO2 c1(C=O)cc(F)c(C(F)(F)F)c(F)c1.N#Cc1csc(C(=O)NC(C)CO)c1 N1(C=O)CCCCC1.c1(C(N(C)CC)=O)ccc(C=O)[nH]1.C1CC1.C=O.N c1(C(C(=O)NCCCC)N(C2CSC2)C)cc(Cl)nc(Cl)c1F C(CNC(C1(C2CC2)CC1)=O)(CC(F)(F)F)NC(C(C)(C)c1cc[nH]n1)=O C(=O)(C1=C(C#N)CCC1)NC(c1ccc(OC)cc1)CNC(CC(C)OC)=O C1(CNC(c2n3cc(C)sc3nc2)=O)CN(C(=O)C(C)CN(C)C)CCC1(C)C C(N=c1cc(C)c(S(=O)(=O)NC(C)C2CC2)c[nH]1)C1(S(CC)(=O)=O)CC1 C(=O)CC(C)C.C(C(C(=O)N)NC(C)=O)OC.c1ccccc1.C1CCC1.C Cc1cc(C(N2CCC(O)C(C(=O)Nc3ccccc3Cl)C2)=O)cnc1F c1(C(=O)OC)ccc(NC2CC(NC(=O)CCC3(O)CCC3)C2(C)C)nc1 c1(OC)cc(NC(C2CC2)=O)ccc1C(C)=O.c1(CC=O)c(C)n[nH]c1C C(CC1=CCN(C(=O)CC(F)(F)F)CC1)NC(=O)Cc1ccccc1C(F)(F)F C1(C)(C(N(CCN(C(C2CCC(CC)O2)=O)C)C)=O)CCCC1(F)F c1(OC)c(C(=O)N(CCCN(C)C(C2(C#N)CC2C)=O)C)cccc1C(F)F C1(C)(CNC(C(C)(C)SC)=O)CCCN(C(c2cc(C)ccc2C)=O)C1 c1(OCC)ncc(C(=O)NC2CC(C)N(C(c3occc3F)=O)C2)cc1Cl C1(C(N(CCNC(=O)Cc2cnoc2)C2CC2)=O)COC2(CCC2)CO1 C1(CNC(c2cnn(CC3CCOC3)c2)=O)C2CN(C(=O)C(Cl)=CCl)CC12 c1(CC)c[nH]cc1C(=O)NC(C)CCNC(=O)CC(C)n1ccc(C)n1 c1(C(N2CC(NC(c3cnc(O)c(Br)c3)=O)C2)=O)cc(F)cc2cnccc12 N1(C(c2c(OC)cc(C)s2)=O)CCCCC(CNC(=O)CC(C)C2CC2)C1 C1(C=O)(COC)C=CCN1C(c1ccc(C#N)[nH]1)=O.C1CC(=O)N(O)C1.N c1(C(=O)NCCN(C(=O)CN2CCCCCC2)C)ccc2ccccc2c1 c1(C(=O)NC(CC)CNC(=O)CCc2cnn(C)c2C)cc(C)cc(Cl)n1 Cc1nn2ncccc2c1C(N1CC(C)(NC(C2CC3(CC3)CO2)=O)C1)=O c1(C(=O)NCCN(C(c2csnn2)=O)CC)ccc(S(=O)CC#N)cc1 C1(C(=O)NC(C2CCN(c3nc(CC4CC4)ns3)C2)C)CCCCC1C C(N=c1[nH]c2c(C)cccc2o1)C1N(C(CCC=C)=O)CCC1 C1(C(=O)NC(C2CCN(c3cncc(C#N)n3)C2)C)Cc2nccnc2C1 S(=O)(=O)(c1c[nH]c(=NCC2CC(CF)C2)cc1C)NC1CCCC(C=C)C1 c1(C(=O)NC2(CO)CCN(C(C(N3CCOCC3)C)=O)C2)ccc2nn[nH]c2n1 C12(CCCNC1)CC(=O)N2C.C1(CNS(C)(=O)=O)CCCS1(=O)=O N1(C(C2COCCN(C(C3CCN(C)CC3)=O)C2)=O)CCC12CCCSC2 Cc1cc(C)c(CNC(C2CC(C)C2)=O)c(O)n1.c1(C(C=O)O)cncn1C C1(C)(C(N(c2ccccc2O)C)=O)CC(O)CN1C(=O)CC1CC2CCC1O2 c1(C(N(CCN(C(C2CC(C(C)C)C2)=O)C)C)=O)ccc(Cl)c(N)c1 C1(C)(C(=O)NC2CCC(CCC)CC2)CN(C(=O)C(CC)SC)C(C)(C)C1 c1(-c2c(CC)cccc2)cccc2cc(C(N3CCC4(CCCOC4)C3)=O)[nH]c12 Cc1nnc2cc(NC3CC(NC(=O)C(c4cscn4)N(C)C)C3)ncn12 C1(C(=O)NCc2c(C)scc2)CCCCCN1C(=O)CCc1ccccn1 CCCC(CCCNC(c1ccc([N+](=O)[O-])s1)=O)NC(=O)CCS(C)=O Cc1cc(C(N2CCC(F)(CNC(=O)C=CBr)C2)=O)ncc1Cl C1(C(C)NC(Cc2cn(CC)nn2)=O)CCCCN1C(=O)CCc1cnc(O)[nH]1 N1(CC)CCc2cc(C3CC3)ccc21.c12cc(N)c(c(F)c1)c(=O)[nH]2 c1(C(C)C)nccc(=NCC(C)NC(c2cc(C3CC3)nc3ccccc23)=O)[nH]1 C1(CC)CN(C(=O)C(O)C2CCCC2)CCC1NC(C1(C#N)CCSCC1)=O Cn1c(C(=O)NC2(CO)CN(Cc3cncnc3)C2)cccc1=O C1(NC(C(n2cc(-c3ccncc3)nn2)C)=O)CCCC12CC2 C1(C(N2C(CNC(c3ccc(C4CC4)nc3)=O)C=CC2)=O)CCC2CCC1O2 c1(OC)ccc(C(N2CCN(C(c3ccc(CF)cc3)=O)C3CC23)=O)cc1O C(=O)(C#CC1CCOC1)N1CCN(C(CSCCC#N)=O)C(CO)C1 N1(C(CCOCC(C)C)=O)CCC(C(=O)N(C2CCCC(C)(C)C2)C)CC1(C)C N1(C(C)C)CCCC(C(=O)NCC2(F)CN(C(c3cc(CCO)on3)=O)C2)C1 CCC(CCC(=O)O)NC(CC)CC.S1(=O)(=O)CCCN1 C1(C(=O)N)CC12CCCCC2.C1(C(N(CC(C2CC2)OC)C)=O)CC12CCC2 c12nnc3c(ccc(C(F)(F)F)n13)C(=O)N2C.c1(N(C)CC)ncc[nH]1 c1(C(=O)NCC(CNC(CCc2onc(CC)n2)=O)O)n[nH]c2ccc(O)cc12 N1(C(C2C(C)CCC2)=O)CCN(C(C2CC2c2ccc(F)nc2)=O)CC(O)C1 CC1CC(=O)NC1C(=O)NCCNC(c1cc(SC(F)(F)F)c[nH]1)=O CC1(C)CN(C(=O)CCc2nccs2)C(CNC(C2CCOC(C)(C)C2)=O)CO1 C1(C(N2CC=CC2)=O)CC2CC(O)C(C1)C2.C1(N(CC(=O)NC)C)CCCC1 CP(C)(=O)C(O)C(=O)NCC1CC(F)(CNC(c2csc(Cl)c2)=O)C1 n1(CCCOC)c(N2CCOC(C(C)C)C2)nnc1C1(C#N)CCCC1 O=C1c2cccnc2CCC1CC(=O)NCc1cccc(Nc2ccccc2F)c1 C1(F)(C(=O)NCCC#C)CCN(C(=O)C(C)OCC)CC1 C1(CC(=O)NCCC(N)=O)CCCN1C(=O)C(F)CC1CCOC1.C(=O)CO CCCC(C)(C)C(=O)N1CC(NC(c2ccccc2C(C)C)=O)C(F)(F)C1 c1(C(=O)OCc2c(OC)ncc(C)c2)cnc2ccccn12 Cc1oc(Cl)nc1C(=O)NC(C)CCCCNC(c1cnn(C)c1F)=O CCCCCCC(C)C(=O)NC1CCCC1NC(c1cccc[n+]1[O-])=O C1(OCC)(OC)CCC(C=O)C1.c1n[nH]c(C)n1.C1(N)CC1.CC(=O)C NS(=O)(=O)c1ccc(C(N2CC3CCC2CN3C(c2csc(O)n2)=O)=O)c(Cl)c1 N(C1CN(C(=O)CCCCCF)CCc2ccccc21)C(=O)Cc1ccco1 N1(C(CN(CCC)C)=O)CCC(CNC(c2ccccc2CN(C)C)=O)CC1 c1(C(=O)NC2(C)CCN(C(C(N3CC(C)C3)C)=O)CC2)cccc2cccnc12 C1(NC(C2N(C(Cn3c(C)ncc3)=O)CCC(O)C2)=O)CCOC2(CCC2)C1 CC(C(C)(C)C(=O)NOC1CCOC1)NC(C1CCOCC1(C)C)=O C1(NC(c2c(OC)scc2)=O)CCCC12CN(C(=O)C1=NOCC1)C2 N1(C(CNC(C2C(C)C2)=O)=O)CCCC(CC(=O)NOCCc2ccccc2)C1 C1(NC(C(C)NC(CC)=O)=O)CN(C(c2cn(C)nc2C)=O)CC1(C)C N1(C(c2c(C)cc(OC)c(Br)c2)=O)CC2(C1)CN(C(=O)C(C)CO)CCO2 c1(C(=O)OC)cc(CO)c(O)c(C=O)c1.C1CC1.C(=O)CN(C)CCO.N C(c1ccc(Cl)nc1)=CC(N1C(C2CCN(C(c3cn(C)nn3)=O)C2)CCC1)=O c1(C(=O)NCC(CC)NC(=O)CSC(C)(C)C)cnoc1C(C)C c1(CNC(=O)NC(c2ccc(Br)cc2)CN(C)C)ccc([N+](=O)[O-])cc1 CC(C)(C(=O)NCc1ccsc1S)c1cncs1 N1(C(c2c(C)non2)=O)CCC(C(=O)N(CCCO)C)CC1C C1(O)CCCN(C(=O)CC2CCCC2)C1.C(C)(C(=O)NC)(c1cccs1)N(C)C N1(C(C(C)(C)OCCC)=O)CC2C(N(C(=O)CSc3nc[nH]n3)C)C2C1 CCCCC(C)N(C(=O)C(C)NC(c1cc(C(N)=O)c[nH]1)=O)C N1(C(C(CNC(c2ncccn2)=O)N(C)C)=O)CCC2CN(C)CC2C1 N1(C(Cc2c(C)ccs2)=O)CCC(C2CCCN(C(c3cnncc3C)=O)C2)C1 Cc1cccn2cc(CC(=O)NC3CN(C(C4CCC(=O)O4)=O)C(C)(C)C3)nc12 C(C(=O)NCCS)(C(C)(C)C)NC(C1CC(OC)CN1)=O.c1ccccc1 C=C(C)CC(C(=O)NC(C1CCN(C(=O)C(O)CN(C)C)C1)(C)C)OC c1(C=O)cc2nc(F)ccc2o1.CCCCN(C(=O)CNC(=O)C1CC1)C.N N1(C(=O)Cn2cccc2)CC(S(=O)(=O)N2CCN(C(=O)C(F)CCCC)CC2)C1 Cc1cc(Cl)c(C(=O)NCC2CCN2C(C2(c3cnccc3C)CC2)=O)s1 c1cn(C)nc1.N1(C(CCN(C)CC)=O)CCC(OCC(=O)N)C1.C1CC1.C C1(NC(CC(CC)SC)=O)CC2CCC1(NC(c1csc(C#N)c1)=O)C2 N1(C(CC2(OC)CN(C(c3cc(CCC)[nH]n3)=O)C2)=O)CC(S(N)(=O)=O)C1 C1(=CC(=O)NC(C2CCCCC2)CNC(C2CC3(CC3)C2)=O)CCCCC1 C(=O)(C1=CCCN(C(C2CC(=O)C23CCC3)=O)C1)NCC1CC(SC)C1 N1(C(CC2N(C(C3C(C)(C)C3C#N)=O)CC2)=O)CCOCC2(CCC2)C1 C1(C2CCN(C(c3cc(O)nc(O)n3)=O)C2)(NC(=O)CCn2cncn2)CC1 c1(C(N2CCN(C(CC3CC(CC)C3)=O)C(C)C2)=O)cccc2oc(C)nc12 C1(NC(C=C(C)c2ccsc2)=O)CC(NC(c2ccc(C)c(C)n2)=O)C12CCC2 c1(C(N2CCC(NC(C3CC(F)C3)=O)C(O)C2)=O)ccc(Cl)c(F)c1 N1(C(C2(CSC)CC2)=O)CC(C(=O)NCCCC(O)CO)C(C)(C)C1 C1(OC)CCC2(CCN(C(C34CC3CN(C(c3ncnc(C)c3C)=O)C4)=O)C2)C1 c1(C(=O)OCC)cccnc1NC(C1CCN1C(C1(C)COC1)=O)=O C1(NC(CNS(NC)(=O)=O)=O)CCC(C)(C)C1.C(c1cscn1)=C(C=O)F c1(OC)ccc(C(C)C(=O)N(CCC)C2CC2)cc1.C1(CC=O)CCC2CC12 c1(OC)ccc(C(N)C(N2CCCC2C(N(C)Cc2cccc(F)c2)=O)=O)cc1 C1(SCCNC(CCCSC)=O)CCCC2(CN(C(=O)C)C2)O1.CCC(C)C.N N1(C(C2(C(C)=O)CC2)=O)CCCC(CCn2cc(-c3cn(C)cn3)nn2)CC1 C1(C(=O)NC2CCC(C(=O)N(C)Cc3cccs3)C2)(OCC)CCOCC1 N1(C(C(C)(C)OCC)=O)CCC2CCN(C(c3nnc(C)cc3O)=O)CC2C1 c1(C(=O)OC)ccncc1-c1cn(Cc2ccncc2Br)nn1 C(=O)(CC(Cc1ccccc1)C(F)(F)F)N.C(C(C)(C)C)NC(C(F)OC)=O Cc1nc(O)[nH]c1C(N1CC(O)CC1CNC(C1CC1C(F)F)=O)=O C1(C(N(CC(C)SC)C)=O)CCC2(CC2)N1C(C1CC1(F)F)=O N1(CC)CCCCC1C(=O)NC(C1CN(C(=O)CC(F)(F)c2ccccc2)C1)C C1CN(C(=O)C(C)CN(C)C)CC2(CC2)C1.Cc1ccc(C(C)C)c(C=O)c1.N n1(C(C)C(=O)N(CCNC(=O)CC2CCOC2)C2CC2)cc(Cl)cn1 N1(C(C(CCO)N(C)C)=O)CCCC(c2ccccc2)(NC(=O)COC2CC2)C1 Cc1c(C(=O)NC2CCN(C(c3cnsn3)=O)CC2C)oc2cc(Cl)ccc12 c1(C(C)C)ccc(Cl)cc1C(=O)NC1CCCCC1NC(C1CCC(=O)O1)=O C(=O)(CC1=NNC(=O)C1)N1CC(NC(c2cc(C)[nH]c2C)=O)C2C1C2.C1CC1 C1(NC(c2cccc(OCC)c2)=O)CC(O)CN(C(=O)CCSC(F)(F)F)C1 C#Cc1c[nH]nc1C(=O)NC(C)CCN(C)C(C1CC1C)=O C1(C(=O)NCC)(CC)CCCNS1(=O)=O.C(=O)C(C)(C)C.C(=O)(CC)N C1(NC(Cn2cc(C(C)O)nn2)=O)COCCN(C(=O)CC(F)(F)Cl)C1 c1(C(C=O)(F)F)ccc(C)cc1.C1CCCC1.C(CC(=O)N)NC(=O)NC.C Cc1ccc(C(N2CCN(C(C3CCC(C)(C)O3)=O)CC2CF)=O)c2c1CCC2 C12(C(=O)NCCCCCC)CC(C)(CN1C(=O)Cc1ncccc1C)C2 C#Cc1ccc(OC)c(C(=O)N(CC(C)NC(c2ccccc2C(C)=O)=O)C)c1 c1(C(=O)NCC2(C(N3C(C)CC3CO)=O)CC=CC2)cc(CO)n(C)n1 C(=O)(CC1OCCc2ccsc21)Nc1cc(C(=O)OC2CCCC2)c(F)cc1 O=C(NNc1ccc(C(F)(F)F)cc1)NCC1CCC12CCCO2 N1(C(CCC(CC)C)=O)CC(NC(=O)CC2CN3CCC2CC3)CC2(CC2)C1 Cc1cn2c(n1)CC(C(N1CCOCC1)=O)CC2.C(=O)(C1=CCC1)N(C1CC1)C C1(C(=O)N)C(C2CC2)CCN1C(c1cc(O)cc(=O)o1)=O.Cn1c(C)nnc1O C(=O)(C(C)CC(C)(C)C)NC1C(O)CCN(C(C23C(C)OC(CC2)C3)=O)C1 N1(C(C2C(C)(C)C2(C)C)=O)CC2CN(C(=O)C=CC3CCCO3)CC2(C)C1 CC1CN(C(=O)C(F)(F)c2ccncc2)CC(CCNC(=O)C2=CCCC2)O1 C(CCNC=O)(C(=O)O)NC(C1CC(NC(=O)OC(C)(C)C)C1)=O N#Cc1cc(CN2CCCC(C(=O)NCc3ccccn3)CC2)ccc1Br C1(NC(CNC(CC)=O)=O)CC2CC1N(C(=O)CCCn1cccc1)C2 Cn1cc(C(N2CCC(C)(C)C(C)C2)=O)c(=O)n(C)c1=O.c1(C=O)ccoc1.N N1(C(C(=O)N(CCc2ccccn2)CC)=O)CCN(C2CCC2)CC1(C)C c1(CN(C(CC)=O)C)ccccc1CNC(c1cccc(-n2cnnn2)c1)=O N1(C(C(c2n(C)ncc2)O)=O)CC2CCC2(CC(=O)NCc2cccc(O)c2)C1 C1(C(=O)NCC2(C(=O)NCCCn3cccn3)CC2)CCCC12CCC2 C1(C(N(C2CCN(C(=O)C(=C3CCCCC3)F)C2)CCO)=O)CCC(F)(F)CC1 CCS(=O)(=O)CCCNC(C(C)CC1CCCC1)c1nnnn1C1CC(F)(F)C1 CCC(C)C(CC(=O)NC1CCCCCC1(C)C)NC(C1C=CCCC1)=O CCC(C)C(O)C(C)C(=O)N1CC(C(N2CCC2C(=O)N(C)C)=O)(CC)C1 C(C(=O)N1CC2CC1C2)(C(C)(C)C)OC.c1(C(=O)N)cc(C(C)C)nc(O)c1 C1(OC)CCN(C(c2cc(C(F)(F)F)ccc2N)=O)CC1(C)C c1(OC)ccccc1OCC(=O)NCCCC.c1(C(=O)N)ccc(C2CC2)nc1 c1(SC)ncccc1C(=O)NCc1ccon1.C1(CC=O)OCCC1(C)C.C c1(CC(=O)NCC2CCCC2)cn2ccsc2n1.C1(C(F)(F)F)(C=O)CCC1 CC1(C)C2CN(C(C3CC(NC(=O)CC=Cc4ccccc4)CCO3)=O)CC12 C1(CCNS(C)(=O)=O)(NC(N)=O)CCN(C(=O)CC2CCCOC2)C1 N1(C(=O)NCc2ccc(C(=O)OCC)nc2)CCc2c(C(=O)O)n[nH]c2C1 c1(OC)noc(C)c1C(=O)NC1CCOCC1C(=O)NC(C)C CCCCC(O)CCC(=O)NC1CC(CNC(c2ccn3ccccc23)=O)C1 C1(CC=O)CCC(C)(C)C1.C1(C(=O)OC)CC=CC1.c1(C(=O)N)n[nH]cc1 CC1(C)OCCc2cc(C(=O)NC(C(C)(C)C)C(F)(F)F)ccc21 C(=O)(C(C=C)CC)Nc1cc(C(N2C(COCC#C)CCC2)=O)sc1 C1(NC(COCCCC#C)=O)CCC(N(C)C(C2OCC2(C)C)=O)CC1 C1(O)(CC)CCN(C(=O)CC(O)CNC(=O)C(O)CN(C)C)CC1 c1(C(N2CCN(C(C3C(CC)C3)=O)C(C)C2)=O)noc2ccc(Cl)cc12 C(=O)(CCCCC(C)(C)C)Nc1c(-n2cc(C(=C)C)nn2)cccc1 c1(C(=O)NC2C(CNC(C(C(CC)C)O)=O)CC2)ccc2oc(O)nc2c1 CCCCCCC(C)C(=O)NCCCCC(=O)NC1(C(O)CO)CCC1 N1(C(Cc2n(C)cnn2)=O)CCC(NC(c2cccc(OC(F)F)c2)=O)C(O)C1 c1(C(=O)OCC)ccc(OCCCNC(c2cocc2C)=O)cc1 C1(C(=O)NCCc2cccc(C)n2)COCCN(C(=O)C(C)(C)n2cccn2)C1 C12(CNC(=O)NC3C(OC)CC3)CCCC1C2 C1(C(=O)NCCc2cccc(O)c2)CC2C=CC1N(C(=O)CO)C2.CC(F)F C(CCNC(=O)Cn1cnc(C#N)n1)(C(=O)N(C)CC1(O)CCCC1)OC c1(C=O)ccc(C2(C)CC2)cc1.C(C)(C)(C(=O)NCC1(F)CCC1)SC Cc1ccc(C(N2CCCCC(NC(C3CC(C)(O)C3)=O)C2)=O)cc1C c1(OC(C)C)cccc(C(=O)N(C2CCCN(Cc3cnn(C)n3)C2)CC)c1F c1(C(=O)NC2CC3(CN(C(C(CC)COC)=O)C3)OC2)cccc(P(C)(C)=O)c1 Cc1cccc(O)c1.C(=O)(CC)NCCN(CC)C.[SH](C)(=O)=O.C(N)=O C1(CCOC)(NC(=O)C)CCN(C(=O)C(C)C2CCCC2)C1.c1ccncc1.S c1(NC(c2c(F)cc(OC)c(OC)c2)=O)c(C)oc(C)c1S(N)(=O)=O c1(NCC2C(P(C)(C)=O)CCC2)[nH]c(=NCc2ccnnc2)nc2scnc12 c1(C(=O)NC2CCCN(C(c3c(C)occ3)=O)C2)ccc2cnsc2c1 c1(C(=O)NC(CNC(C2(COC)CCCC2)=O)CO)cc2ccccc2cc1C c1(OC)cc(F)ccc1CC(=O)NCCC1(O)CCN(C(=O)COC(F)F)C1 c1(OCC2N(C(c3ccc(F)cc3)=O)CCC2)cc(Br)ccc1[N+](=O)[O-] C(C(O)CC(=O)N(C1CCC1C)C)NC(CC1CN(C(C)=O)C1)=O c1(C(N(CC(N2CCOCC2C2(C)CC2)=O)C)=O)cnn2c1CCC2 C(=O)(CCCS(N)(=O)=O)N1CC(COC)C1.c1(C=O)nc(C(C)C)sc1N.C N1(C(C2CCC(=C)CC2)=O)CCC2(CC1)CN(C(=O)CC1CCC1)CCO2 C(=O)(C(C(C)(C)C)c1ccc(OCc2ccnnc2C)cc1)OCC c1(Cc2cnc(NCC(CNCC)(C)C)s2)cc(Cl)ccc1OC c1(C(N2CC(NC(C(C(CC)C)N(C)C)=O)C2)=O)c(F)cc(OC)cc1Cl Cc1nc2ncccc2cc1C(N1CC(NC(=O)CC(F)F)C(O)C1)=O C1(CC(=O)NC(CO)C(=O)NCC2C3COCC23)CCCC12CC2 C1(NC(COCCSC)=O)CCC(NC(=O)C(C)c2cc[nH]n2)CC1 c1(-c2nc(C(C)OC)nn2-c2ccc(F)c(F)c2)ccc2c(n1)CCCC2 C(=O)(CC1=NNC(=O)C1)N(C(CCN(CC(N)=O)C(N)=O)=O)C1CCCC1 c1(SCc2ccc(-c3cn(CC(C)C(=O)O)nn3)cc2)cc(Cl)nnc1Cl N1(C(C(C)(C2CC2)NC(C)=O)=O)CCCC(n2cc(-c3cn(C)nc3C)nn2)C1 N1(C(CCSC)=O)CCC(O)C(C(=O)Nc2cc(Cl)ccc2F)C1 Cc1nn(CC(N2CCC(N(C)C(c3[nH]cnc3C)=O)C2)=O)c(=O)o1 N1(C(C(CC)COC)=O)CC2(C1)CCCS2(=O)=O.c1(C=O)cnn(C(F)F)c1.N c1(OC)ccc(OCC(N2CCC(NC(=O)C(C(C)C)OC)C2)=O)cc1 c1(C=O)ccc(F)c(F)c1F.CC1(C)C(C)(C(N2CC3CC3(C)C2)=O)C1(C)C N1(C(C=C(C)Cl)=O)CCC(C2(O)CCN(C(c3ccc4nonc4c3)=O)C2)CC1 N1(C(C2CC(NC)C2)=O)CCC(C)(C)C(C(N2CCOC(C3CC3)C2)=O)C1.CC N1(C(c2cccc(OC)c2C)=O)CCC2(C)CN(C(C3CCCC(F)C3)=O)CC12 C12(C(=O)NCC(C)CN(C(=O)CCC3CCCO3)C)COCC(C1)C2 c1(CC)cc(C(N2CCOC(CCCNC(=O)C(O)CC)C2)=O)c(C)o1 c1(NC(c2nc(-c3cc(C)nnc3)sc2C)=O)c(F)ccc(Cl)c1F CC1CCN(C(C2CCOC2C)=O)CCN1c1ncc(Br)cn1 c1(C(=O)OCC(=O)NC(c2cccc(Br)c2)C#C)cc(C#N)ccn1 C1(CNC(Cc2ccc(C(N)=O)cc2)=O)CCCC2CN(C(=O)C3CC3)CC12 O(NC(=O)C(F)CC(C)(C)NC(=O)CC1CCCC1)CCC(C)O C(=O)(CC1CCc2ccc(O)cc21)NCC1N(C(CCCCC)=O)CCC1 C(CCC(=O)N1CC=C(N)N1)C1OCC(C)C1 c1(C(=O)NC2C(CNC(C(C)NC(=O)NC)=O)CC2)sc(C)cc1 C1(CNC(C=C2CCN(C)C2)=O)CN(C(C2CCC(C)(C)CC2)=O)CCC1(F)F Cc1cc(O)nc(C)c1C(=O)N(CCC)C1CC1.CC(F)(F)F.C(=O)(C)N O=C1NCC(NC(C2CC(O)CN2C(=O)CC2CCCC(=O)N2)=O)CO1 CCC(CC)C(F)C(=O)N1CCC(O)(CCNC(C2CC(OC)C2)=O)C1 C(=O)(C1CCc2cc(F)ccc21)NCCN(C)CC1CCC1 C(C)(C)(CCCNC(C1CCCC(OC)C1)=O)NC(C=CCC)=O c1(OC)cc(F)c(C(N2CCCCC2CNC(C2CC2CF)=O)=O)c(Cl)c1 c1(C(=O)NC)n[nH]c2c1CN(C(c1ccc(Cl)cn1)=O)C2.CC(C)C1CC1 N1(C(C(C)NC(c2ccoc2)=O)=O)CCCN(C(=O)C=Cc2cocn2)CC1 S(=O)(=O)(CCCC1CCOCC1)Nc1c(C(=O)NC)noc1 c1(C(=O)NC2C(O)C3CCOC23)ccc(F)c2c1CNC2 CCC(C)(CC(=O)N1CCC2C(NC(=O)C(C)(C)C3CCOC3)C2C1)C(=O)OC C1CN(C(=O)C(O)CC2CCCCC2)CCO1.c1(SCC(=O)NC)n[nH]c(O)n1 CCCCCC(C)CC(=O)N1CC(C(F)Cn2cc(C3(C)CCCCC3)nn2)C1 Cc1cccc(CC(=O)NCC2CC2NC(c2cc(-c3ccccc3)on2)=O)c1 CC1(C(N2CCC(CCNC(C3CN4CCN3CC4)=O)CC2)=O)COC(=O)OC1 c1(C(NNC(=O)NCC2(C)CCCC(=O)N2)=O)ccc2c(c1)OCCO2 C(CN=c1nc(N2CC3C(C2)C3(F)F)c2c([nH]1)CCCCCC2)(C(C)C)OCC N1(C(C2C(CC)C2)=O)CCC(O)(C)C1.c1(CC=O)cccnc1C(F)F.N Cc1c(C(=O)N(C2CCN(C(C3CC3C(N)=O)=O)CC2)C)oc2ccc(Cl)cc12 C1(C(N2C(CNC(=O)Cc3cnccc3Cl)CCC2)=O)CCn2c(O)nnc2C1 C1CC(C)CN(C(=O)C(C)(C)c2csc(C)c2)C1.c1(OC)cc(C)sc1C=O.N c1(CN2CCC(NC(C3(C(F)(F)F)CC3)=O)C2)cc(O)ccc1[N+](=O)[O-] c1(C(=O)NC2CCN(C(c3ccc(C)c(C)n3)=O)CC2O)ccc2ccoc2c1 C(C)(C(C)S(C)(=O)=O)NC(c1cc(C)c(C)o1)=O C(CO)(CCCCNC(C1CC=CCC1)=O)NC(c1cn(CCF)nn1)=O C(=O)(C(C#N)C(C)(C)C)NC1CCN(C(c2c(SC)cccc2F)=O)CC1C c1(NC(C2CCCN(C(=O)CCc3ccccn3)C2)=O)ccc(O)c(F)c1 C1(CNC(C(CCCOC)C)=O)CN(C(c2cccc(C)c2N)=O)CCC1(F)F N1(C(C2C(C=C)C2)=O)CCC(F)(CNC(=O)CCO)CC1.c1cccc(C)c1 c1(C(=O)OC)ccc(OC)c(CCN2CC(F)(CN(C)CCOC)C2)c1 C(CCCCCNC(C1(C)CCCC1)=O)NC(C(C)N(C)Cc1ccccc1)=O C(=O)(C(C)C(O)C(C)C)NCC(CC)NC(c1c(OC)ccc(CC)c1)=O c1(OC)ccc(F)cc1-c1cnc(N2CCC(C(=O)NC3CSC3)CC2)nc1 c1(CCC(=O)NCCN(C(=O)Cc2nnnn2C)C(C)C)ccc(CO)cc1 CC(C)C(C)C(CNC(=O)CCCN=[N+]=[N-])NC(c1cc(Br)nn1C)=O Cc1ccccc1-n1nnnc1C(CC(C)C)NCCCCOC(C)(C)C N1(C(c2c(C)nn(C)c2)=O)CCC(C2CCN(C(=O)Cc3cnn(C)n3)CC2)C1 C1(NC(=O)NC(c2c(C)cccc2)CF)CCCCCCC1 C1(OC)CCC2(CCN(C(C3(NC(=O)CCCc4ncco4)CCCC3)=O)C2)C1 C1(C)(C(N2CCC(C)(CC)C2)=O)CC=C(C)CC1.C(C(=O)N)OCCSC N1(C(CC)=O)CC(NC(c2snc(Cl)c2Cl)=O)CC(C)C1 N1(C(C(C)OCCOC)=O)CCCC2(C1)CN(C(c1c[nH]cc(C)c1=O)=O)C2 Cc1cc(=NC(=O)COC(C2CC(C)N(C(=O)CCCn3cccn3)C2)=O)[nH]o1 CC(C)(CC=CC(=O)NCc1nn[nH]n1)NC(=O)C=CC1CCC1 C1(CC=O)OCCC1(C)C.C1(C(=O)OCC)(C(=O)NCCC)CCCC1.N N1(C(CSC)=O)CCN(C(=O)C(C)NC(C)C)C(c2ccncc2)C1 C#CC(C1CCc2ccccc21)NC(=O)NCc1n[nH]c(C)n1 C1(C(N2CCC(c3cn(CCC=C=C)nn3)CC2)=O)CC2CCC1NC2=O CS(=O)(=O)c1cscc1C(=O)N.C1(F)CCN(C(C2CC2C(N)=O)=O)C1 c1(C=O)cccn(C)c1=O.C1CCCCC1.C(C=O)N(CC)CC.C(C)(C)C.N C(=O)(CS(=O)(=O)CCO)N(C1CCN(C(c2c(C)csc2C)=O)CC1)C C=CC1CN(C(=O)Cc2cccc(F)c2)CC1CNC(=O)CC1CC2CC2C1 N1(C(C(C(C)C)OC)=O)CCC2(CC(C(=O)Nc3cc(Cl)nnc3Cl)=NO2)C1 C1(O)(CN)CCN(S(=O)(=O)CC#N)C1.c12cnn(c1)C1CN(C1)C2=O N1(C(Cn2nnc(=N)[nH]2)=O)CCCC1C1CCCN1C(c1ccoc1)=O C(=O)(CC(C(F)(F)F)n1ccnc1)N.C(c1cncs1)=CC(=O)NCC(C)C c1(C(=O)NC2CCN(C(CSCCCC)=O)C2)ccc(C(=O)OC)cc1F C1(NC(CCN(CC=C)C(c2ccc(CC)o2)=O)=O)CCC(C)C1 C1(CNC(CCN(C)CC)=O)CN(C(=O)C(O)C2CCC2)CCO1 N1(C(c2n(C)nc(C(F)F)c2)=O)CC2CCC1CN2C(c1ccc(N)cc1F)=O N1(C(C2CCC(CC)O2)=O)CCN(C(=O)CCc2ncc(C)[nH]2)CC12CC2 C(CCC(N)=O)(C(=O)NCC(C)(C)C1CC1)n1cc(C(CCC)N(C)C)nn1 CC(C)C(CNC(=O)C(=O)NCCCCCO)Nc1ccccc1 C1(CCCC)CCN(C(C2(C)CC(F)(F)C2)=O)CC1.C1(CC(=O)N)(OC)CCC1 CC1OC2(C)CC1(C(N1CCC(NC(C3C(F)(F)C34CC4)=O)C1)=O)C2 C1(NC(CCN(CCCCC)C)=O)CN(C(=O)CC2CCOC2)CC1SC C1CCCC2(CN(C(c3cc(C(N)=O)c[nH]3)=O)C2)O1.Cn1ccc(C(=O)N)c1.C n1(CC(=O)N(C)Cc2c(OC)cccc2OC)cnc2sccc2c1=O C12CCCCN1C(=O)c1nc(cs1)C2.c1(C(C)OCC)cncc(OC(F)F)c1 c1(-c2cn(C(C3CC3(C)C)CC)nn2)cccc(OC(F)(F)F)c1 c1(SC(C(N2CCC(O)(C(N(CC)CC)=O)C2)=O)(C)C)cc(Br)ccc1O NS(=O)(=O)CCCC(=O)N1CC(NC(=O)CSCc2ccccc2)C2CC12 N1(CC(C)(C)NC(Cc2cnc(C)s2)=O)CCN(C(=O)Cc2nc[nH]n2)CC1 CCCCC(CNC(=O)C(N1CCOCC1)C)NC(c1cn(C)c(C(F)F)n1)=O C1(C(=O)NC(C(C)SC)C)CC(C)CN1C(c1cc(=N)[nH][nH]1)=O C123CCC(CN(C1)Cc1cn(nn1)C1(CC1)C(=O)N2)C3.C=C(C)COC c1(C(=O)NCC#CCNC(c2c(CC)ncnc2)=O)cc(C(F)F)ccc1F C1(C(=O)N)CCN(C(c2cc(O)nc(O)n2)=O)C12CC2.NC(=O)CC1CCCC1 c1(N(C)C)ccc(F)cc1-c1ccc(CNC(=O)Cc2c(F)cccc2Cl)cn1 C(=O)(C1=CCOCC1)NCC(CNC(C1(C(F)F)CCCCC1)=O)OC C1(C(=O)Oc2cccc(C(=O)OC(C)(C)C)c2)CC2(CCOC2)CO1 N1(C(c2c(C)cc[nH]2)=O)CC2CC3CC2C1C3NC(=O)CN1CCC1C S(=O)(=O)(c1ccc(C(=O)N)cc1)NCC.C(=O)CCn1ccnn1.C1CC1 c1(-c2c(C(N3CCC(NC(c4n(C)cnc4)=O)C3)=O)c[nH]c2)ccc(F)cc1 C1(NC(c2c(OC)csc2)=O)CCOC(C)C1.C12(C=O)CC(C)(CO1)C2.N Cc1cc(C(=O)NC2CC(C)CN(Cc3ccc(C)c(Cl)c3Cl)C2)c(F)c(F)c1 N1(C(CONC(CC2CC(OC)C2)=O)=O)CC(C)CCC12CC2 N1(C(c2c(C)[nH][nH]c2=N)=O)CC2ON=C(CNC(C3CC3)=O)C2C1.C(C)C c1(OC)cccc(-n2cc(CC(O)C(=O)NC(C)C(=O)N(C)C)nn2)c1 C1(CC(=O)NCC(C2CCOCC2)NC(C2CCCCC2)=O)COCCO1 C#CCC(C)(C(=O)NC1(COCC)CC1)NC(=O)CC1CC1C1CC1 C1(C)(C(=O)NCC(=C)C(F)(F)F)CC(O)CN1C(=O)Cn1cc(C)cn1 N1(CCNC(C2N(C(Cc3cn(CC)nn3)=O)CC2)=O)C(=O)CCC1=O O=c1c(CN2CCc3sc(CO)nc3C2)cnc2n1CCS2 c1(NC(=O)CC(C(F)F)NC(=O)COC2CCCC2)cccn2nccc12 C1(NC(CCCC=C)=O)CCCC12CCN(C(c1cocc1Br)=O)C2 N1(Cc2cn(CCC(=O)NC)nn2)CCOC(c2nnc(C)o2)C1 N1(C(c2cc(CC)[nH]n2)=O)CCCC1(C)C(=O)Nc1cn[nH]c1 Cc1ccc(C)c(CN=c2ccc(NC(c3cccc4nc[nH]c34)=O)c[nH]2)c1O c1(CC)oc(C)cc1C(=O)NCCCC(=O)NCCc1c[nH]nc1O C(=O)(CC(O)CC(C)(C)C)N1C(C#C)CN(C(c2[nH]nnc2C)=O)CC1 N1(C(C2CN(C(C(CC)C)=O)CC23CCC3)=O)CC(C)C12CCOCC2 N1(Cc2c(C)noc2)CCC(NC(=O)CC(C)n2ccc(C)n2)C(O)C1 S(=O)(=O)(c1ccccc1)N1C(C=O)CC(O)C1.NC(=O)C(=O)NC.C1CC1 C1(NC)CCC2CN(C(=O)Cn3cc(C(=O)Nc4ccncc4Cl)cn3)CC12 C1CC2(CCN(C(C3(CC(F)F)CC3)=O)CC2)CO1.C1(C(=O)NC)COCCO1 C#CCC(C(=O)OC)NC(=O)C=CCNC(c1cncc(CC)c1)=O C1(C(=O)NCC(CN(C(C(C)(C)SC)=O)C)(C)C)Cc2nc(C)cn2C1 c1(NCC#CCC)cc(NC2CCCN(c3ccccn3)C2)ncn1 c1(C(N(C)CC2N(C(C(C)S(N)(=O)=O)=O)CCOC2)=O)nccn2cnnc12 N1(C(C(CCC)OCC)=O)CCC(C=CC(N2CC(C(=O)NC)C2)=O)CC1 c1(CC(C)OC)nc(C(O)C(C)(C)C)n(-c2ccccc2)n1.C(C)OC C12(C(=O)NC(c3ccc(C)o3)CC)CC1CN(Cc1cncc(F)c1)C2 N1(C(C2OCC(C)(C)OC2)=O)CCC(NC(c2ccc(Cl)s2)=O)C2(CCC2)C1 C1(C(N2CCC(C(C)NC(C(C)NC(CC)=O)=O)C2)=O)CC(=O)C1(C)C c1(NC2C(C)NC(=O)CC2)ccc(S(=O)(=O)N(C)CCc2cccs2)c(Cl)c1 C1(NC(c2cncc(C(F)(F)F)n2)=O)CCN(C(c2cocn2)=O)CC12CCC2 N1(C(CCSC)=O)CC(F)(F)CC1(C)CNC(c1cc(Cl)n(C)n1)=O C(=O)(C(C)CCCC(C)C)NCC1N(C(CC(CC)OC)=O)CC(O)C1 C1(NC(C2CCCC(C)(C)O2)=O)CC2CCC(C1)N2C(c1cc(O)ccc1F)=O C1CCS(=O)(=O)C1.C1(N(C(C)(C)C)C=O)CNC1.CC(C)C.CC=O.C C=C(Br)CCCN.C(C)(C)(C)OC(=O)N(C)CCC1CC1 C(=O)(CC(Cc1ccc(Cl)cc1)NC(=O)C=C(C)c1cccs1)OC CC1CCN(C(c2cccnc2F)=O)C1CNc1nnc(C(F)F)s1 c1(C(N2CCC(c3nncs3)CC2)C(=O)N)ccc(Cl)cn1.C(=O)(CC)OCC N1(C(c2nc(CC)sc2)=O)CCC(C)C(CC(=O)NC2CC3(CCCC3)C2)C1 C1(CNC(CSCCC)=O)CCC2(CCC2)C1NC(C1CCC(C)CC1)=O CC1CC(C(=O)NCCC2CCN(C(C3CC4CCCCC34)=O)CC2)=NO1 N1(C(C2NC(=O)OC2)=O)CCC2CCN(C(c3ccccn3)=O)CC2C1 Cc1cccc(C(=O)NCC2(C)CCN(C(=O)Cc3cscn3)CC2)c1O c1(CC)[nH]nc(C(=O)NC2CCCC2C)c1Cl.n1(C2(C=O)CC2)cncn1.N S(=O)(=O)(c1cccc(=NCCc2c(C)noc2C)[nH]1)CCC1CC(OC)(OC)C1 C(=O)(C(CO)C(C)(C)C)NCCC1(NC(C2ON=C(CC)C2)=O)CC1 C1(CNC(C(C)C#N)=O)CCCCN(C(c2cccc(F)c2)=O)C1 N1(C(C(CCC)C)=O)CCOCC(NC(c2ccccc2-n2cnnn2)=O)C1 c1(NC(C2N(C(c3cc(C)n(C)c3)=O)CC2)=O)cc(Br)cnc1I Cc1cnc(C)c(C(=O)NC2CCCC2NC(=O)Cc2cncn2C)c1 C(=O)(C#CC(C)(C)C)N1CC(C(=O)NCC2(OCC)CC2)OCC1 c1(C(=O)OC)ccc2c(c1)C(NC(=O)CNC(N1CC3CCC1C3)=O)CCC2 C1(C(N2CCC(N(C(C(CC=C)CC)=O)CC)CC2)=O)CCCCC(C)(C)C1 C1(NC(CCc2n(C)ncn2)=O)CC2CC(C1)N(C(c1ccccc1)=O)C2 c1(C(=O)OCCC2SCCS2)occ2c1CCCC2 CCC(C)(F)C(=O)N1CCCC(OCc2cn(CCCN(C)C)nn2)C1 C(=O)(NNc1ccc(COCC)cc1Cl)NC(CC1CCC(=O)N1)C(F)(F)F C1(CCC)CN(C(=O)Cc2cc(C)n(C)n2)CC1C(N1CCC2CC12)=O O(NC(=O)C(C)N(C(c1[nH]ccc1CC)=O)CC)CCC(=C)C C1(NC(c2c(C)sc(Cl)n2)=O)CC2CCC(C1C)N2C(C1CCSC1)=O C1(C)(CNC(C2(CSC)CC2)=O)CCN(C(=O)CC2CCOC2C)CC1 C1(NC(C2CCN(c3nncs3)CC2)=O)CC2CCC1N(CC1(CO)COC1)C2 N(C(=NCc1ccc(Br)s1)NC(C)C)C1CCN(CCOC)C1 c1(C(N2C(CNC(c3c(CSCC)nccc3)=O)CC2)=O)ccccc1Cl N1(C(C(CCCCC)O)=O)CCCC2(CCCN2C(c2ccc(C)c(C)n2)=O)C1 C=C(Cl)C(C)(C)C(=O)NC1CC(NC(c2cccc(Br)c2OC)=O)C1 c1(C(=O)NCC(C)(CNC(c2ccoc2Cl)=O)OC)ncncc1N C(=O)(C(CCC(N)=O)n1cc(CCc2ccccc2)nn1)NC(CC)C C1(C)(C(=O)NCCOCCCNC(c2c(C)con2)=O)OC(C)(C)OC1C CC1(C)CCC(O)(C(=O)NC2CCCN(C(c3cc(N)c(F)cc3F)=O)C2)CC1 CC(C)CCCC(=O)N1CC2CSCC2(C)C1.c1(C=O)ccc2cc[nH]c2c1 N1(C(C(=O)NCCCOCCCC)=O)CCc2nc[nH]c2C1 C(=O)(CC(C)(C)CN(C)C)NC(C(=O)NCC(CC(=O)NC)C)CC.O C=C(Cl)CCC(=O)N(CC(O)CNC(C1CN(C)CC1c1ccccc1)=O)C C1(C(=O)NC(CNC(C(CC)c2ccccc2)=O)C)CCC(C)=C(C)C1 C1(C(N2CCC(C(N3CC(O)(CCC)C3)=O)C2)=O)COCC1(C)C Cc1ccc(SCC(=O)NCCCNC(=O)CCC)cc1.C1(C=O)CCCC1.N c1(Cc2nc(C3CCC(CC#N)CC3)on2)cc(Br)ncc1F C1(NC(CCS(C)=O)=O)CN(C(=O)CCc2cc(F)ccc2F)CC2(CCC2)C1 C1(NC(C2N(C(C(CC)COC)=O)CC(OC)C2)=O)CCCCC1N=[N+]=[N-] c1(C(N(CCCNC(=O)C=Cc2ccco2)C)=O)ccc(-c2cnco2)cc1 C(=O)(C(CC)C(=O)N(CC(C)C(=O)NC1CC2CCCCC12)C)OCC C12CCN(CC1)CC2.C1(NC(C2CC(=O)C2)=O)CC2(C1)CC2C(=O)NC C(C1=CCN(C(=O)C(C)(C)N2CCCC2)CC1)NC(CN1C(C)CCC1C)=O c1(C(N2C(C)CC(NC(c3cn(CC)nc3C)=O)C2)=O)ccc(N)c(C)c1Cl Cc1ccc(C(=O)NC(C2CN(C(c3c(F)cccc3F)=O)C2)C)c(Cl)c1C C1(C(N2CCC(NC(c3ccc(C)cc3Cl)=O)C2)=O)CSC2(C)CCC(=O)N12 c1(CNCc2ccc(N(C3CCCC3)C)cc2)ccc2cn(C)nc2c1 C1(CC(=O)N)COCC2(CCC2)O1.c1(CCC(=O)NCC(C)C)nc(O)n[nH]1 c1(C(N2CCC3(NC(COCC=C)=O)C(C2)C3)=O)cnc2ncccc2c1 C1(CNC(C(C2CC2)OCC)=O)CN(C(=O)Cc2cnoc2)CCC1C C1(C#N)(C(=O)NCCC(C)N(C)C(C23CC(C2)C3)=O)CCCC1 C(=O)(C(F)C(F)(F)F)N1CC2C(NC(Cc3c(C)occ3)=O)(C2)C1 Cc1cccn(CC(N2CCC(OCCNC(=O)C(C)OC(C)C)C2)=O)c1=O C(=O)(N=c1cc(C)nc(Cl)[nH]1)C1N(CCc2ccc(C(=O)OC)cc2)CCC1O C1(N(C(=O)C=C2CCC2)CC)CCN(C(=O)Cc2cnc[nH]2)C1 C1(NC(C2CCCS2)=O)CCCN(C(=O)C(F)(F)CO)C1 C1(C(N2CCS(=O)CC2)=O)CCCC12CCN(S(=O)(=O)c1nccs1)C2 c1(N(C(C2C(CNC(C(C)OCCCC)=O)CC2)=O)C)ccccc1 n1(CCCC)nnnc1C(COC)(C1CCCC1)NC(c1ccnn1COC)C C(=O)(C(C)(O)C)N(C1CCN(C(=O)C(C)CC=Cc2cccs2)C1)CCC.O c1(C(=O)NC2CC3(C(NC(c4c(CC)n[nH]c4)=O)C3)C2)c(C)ncnc1O C12(C(=O)Nc3ccc(CCC)c(I)c3)CCC(NCc3ccccn3)(CC1)CC2 Cc1cc(CNCC2CCCCC2C(N2CC3CCCC3C2)=O)ccc1[N+](=O)[O-] c1(N(CC(C(C)C)OC)C)nc(C)cc(=NCCN2CCc3ccccc3C2)[nH]1 n1(CCC(=O)N(CC(C)NC(C2(OC)CCOC2)=O)C)cnccc1=O c1(C(=O)NCCN(C(=O)Cc2cc(Cl)sc2Cl)CCOC)ccc(O)cn1 C1(N(CC(C)C)C(=O)NCC(F)F)(CNC(=O)NCC)CCCC1 C12(C=O)CCCCC1OCC2.c1(CN(C)CC)cn(CCOCCO)nn1 C(=O)(C1CCc2nccn21)N1CC2CN(C(c3cc(SCC)ncc3)=O)CC2C1 c1(OCC)cc(C)ccc1CNC(=O)NC1COC2(COC)CC1C2 Cc1cc(C(N2CCC3CCC23CNC(c2cc(CO)oc2C)=O)=O)cc(F)c1 N1(C(C(CN(C)C)O)=O)CCN(C(=O)C(F)(F)Sc2cnn(C)c2)CC(O)C1 S(=O)(=O)(c1ccc(NCc2cc(OC)cc(OC)c2)cc1)N1CCCC2CCC12 N1(C(C)=O)CCCCC1CC(=O)NCC1CCCN(C(c2cn(C)[nH]c2=N)=O)C1 c1(OCCN(C(=O)C(C)OC(F)F)CC#C)ccccc1 CCC(CC(=O)NCC(C)CNC(c1cc(COC)oc1C)=O)C(C)C C1CN(C(C2CCN2C(C)(C)C)=O)CC12CC2.C(CC(=O)N)NC(=O)NC N1(C(C(C2CC2)OC)=O)CCC(CO)(CNC(C2CCN(C)C2C)=O)CC1 Cc1ccc(C(=O)NCC(n2cc(COC(C)C)nn2)C)nn1 C(C(=O)NC1CC1)(C(C)C1CCOC1)N1CCC(CCC)C1 CON(CCCO)C(=O)CNC(c1c[nH]nc1[N+](=O)[O-])=O C(=O)(C1=C(Cl)CC1)N1CCC(C(C(=O)NCCC)C)C1 N1(C(c2c(CC)onc2)=O)CCOC2CN(C(=O)Cn3cncn3)CC12 C=CC(CC)CC(=O)N1CCN(C(=O)NC2CC3C(O)CC3O2)CC1 CCCC(C(O)C(=O)NC(C)CN(C)C)NC(=O)C(O)C1CCC1 c1(C(N(CC)C2CC2)=O)cc(F)cc2nc(S)[nH]c12.O=C(C(O)c1ccco1)N C1(CC(=O)Nc2ccc(-n3nccn3)cc2)CC2(C1)CN(C(C1CC(O)C1)=O)C2 C1(NC(c2cn(CCC=C)nn2)=O)CCCCCN(C(c2cnns2)=O)C1 C(C)(CN=c1nc2scnc2c(NCCCC2CCCO2)[nH]1)OCC=C C(=O)(C(CCF)NC(=O)CCCC1CC1C)NCC1(CO)C(C=C)C1 N1(C(c2cn(CCCC)nn2)=O)CCC2(CCCN2C(=O)C2=CCCCCC2)C1 N1(C(C2CCN(C)C2)=O)CC2(CCN(C(C3C=CC(=O)N=N3)=O)CC2)C1 N1(c2nnc(C)s2)CCC(CNC(=O)CN2C(=O)CCC2=O)C(CO)CC1 c1(C(=O)OC)ccc2c(c1)C1(CC1)CN2C(C1(c2ccc(F)cc2Cl)CC1)=O C1CCN(C(C2CC23CC(O)C3)=O)C12CCC2.O=C(COCC1CC1)N.C N1(C(C23C(C)(C)C(CC2)C3)=O)CCC2(C1)CN(C(c1ccon1)=O)C2 C1(C(=O)NC(C=C)(C)C)CC(O)CN1C(=O)CC1CCC(C)(C)C1 n1(CC=O)nnc2ccccc12.CC(C)(C(=O)NCC1(O)CCC1)C1CC1.N C(C)(C)(C(C)CC(=O)N1CCOC(CCO)C1)NC(C(C=C=C)C)=O c1(C(=O)NCC23C(CN(C(c4c(Cl)ccc(C)c4)=O)C2)C3)cccc2ccnn12 n1(CC)nc(C)cc1C(N1CCC(O)(CC)C1)=O.c1(C=O)cc(C2CC2)on1 N1(C(Cn2c(C)ccn2)=O)CCC(C=CC(=O)NC2CCC(CC(C)C)C2)CC1 c1(C(c2nnnn2Cc2cccs2)NC(C)Cc2ccco2)cccc(F)c1Br C1(C(=O)NCCCCCN(C(=O)COc2ccsc2)C)CCC(C2CC2)CC1 Cc1c[nH]nc1C(=O)NCC(CNC(=O)CCC)CO.c1(C(=O)N)ccccc1 c1(C(=O)NCC2C(NC(c3n(C)ncc3)=O)CC2)cnc2ncc(Cl)cn12 Cc1[nH]nc(C(=O)NCCC2(O)CCN(C(c3cnc(C(C)O)s3)=O)C2)c1O C1(NC(C2N(CC)CCOC2)=O)CCSC12CN(C(=O)C(c1ccnn1C)O)C2 C1(C(N2CCC(NC(COC(C)C)=O)C(O)C2)=O)CCn2nnnc2C1 C1(C(=O)NC2CCN(C(C3(C)CCC(=O)N3)=O)C2)CCCCNC1=O C(=O)(C(C)(C)C(O)C(C)C)NC1C2(CCN(C(C=C(C)C(C)C)=O)CC2)C1 N1(C(C2NCC(CC)C2)=O)CC2(CCC(C)(C)O2)C1 N(C(=NCC(F)(F)C(C)(C)C)NC1CC1)Cc1ccc(N(C)C)nc1 Cc1ccc(C(N2CC(C)(NC(c3[nH]c(=N)ccc3C)=O)C2)=O)c(F)c1 CC1(C)CCC2(CC1)CC2C(=O)NCC1CCOC1.C(=O)(COC(F)F)N C#CCC(CC(=O)OC)NC(=O)CCNCC(O)COC(C)C N1(C(C2C(C=C)CC2)=O)CCN(C(=O)C(Br)=C(C)C)CC1CC(C)(C)C c1(C(=O)NCC(CC(C)C)NC(C=CC)=O)cccc2c1C(=O)CC2 C(=O)(C#CC1CCOCC1)N1CC(F)(C(=O)NCC(C)OC(F)F)C1 c1(OC)ccc(NC(=O)CN(S(=O)(=O)Cc2ncccc2OC)C)c(I)c1 c1(OCCC)ccnc(N(CCCCN(C)C(c2cc(C)cnn2)=O)C)n1 Cc1oc([N+](=O)[O-])cc1C(=O)NC1CCCN(C(c2cc(CO)[nH]n2)=O)CC1F N1(C(C(COC)(F)F)=O)CC2(CC(C(N3CCC(NC(C)=O)C3)=O)CO2)C1 n1(CC(=O)NCC(C)(C2CCC2)NC(c2ccsc2)=O)ccccc1=O C1(C(N(CCCNC(c2c(OC)ccs2)=O)CCO)=O)CCCCC1F C#CCC(C(=O)NC)NC(C1(CNC(c2ncncc2OC)=O)CCC1)=O CC1CCN(C(=O)C(N2CCC(N(C)C(C3CC3c3cccs3)=O)CC2)=O)CC1 N1(C(CC(C)(C)O)=O)CCOCC(NC(C2C3CCCCCC23)=O)C1 C1(C(=O)NC2(CO)CN(C(C3CN(OC)C(=O)C3)=O)C2)CCCCCS1(=O)=O C1(C2CC2)(C(=O)NCC2(NC(CC)=O)CC2)CC1 N1(C(Cc2c(C)ocn2)=O)CC=C(CC(=O)NC(Cc2cnc[nH]2)CO)CC1 N1(C(C(C2CCN(C(=O)C(C)C3(O)CCC3)CC2)C)=O)CCCC(C)(N(C)C)C1 C(=O)(C(CO)N(C(=O)CCc1nc(O)n[nH]1)C1CC1)N.C(C)(C)(C)N(C)C N1(C(C(=O)NC)C(C)C2CCOC2)CCC2(CC1)CC(O)C2 CC#CCCC(=O)NCc1ccc(C(C)NC(=O)CC2CCC(C)O2)cc1 C(=O)(CC(F)(F)C(F)F)N1CCC(CN(C)C(C2C3C4CCC(C4)C23)=O)CC1 N1(C(C2(C(C)NC(c3ccc[nH]3)=O)CC2)=O)CC2(CC2)C1 CCC(CCc1ccccc1)NCc1ccnn1CC(F)(F)F N1(C(c2ccc(Cl)cc2)C(=O)NCCCC2CC2)CCC2CCCCC12 C1(C(=O)NC2CN(C(c3ncn(C)n3)=O)CC2O)COc2ccccc2O1 C1(C(=O)NCC(CCCC)NC(C2CCC3(CC2)CC3)=O)CC12CC(F)(F)C2 CCCCC(C)CCC(=O)NCCC(C)NC(c1csc2cncn12)=O C=CC1(CNC(=O)NCCC2(COC)CCCC2)CCC1 C1(N(C)C(c2cnc(C(C)(C)CF)o2)=O)CCCN(C(C2CC(F)(F)C2)=O)CC1 c1(NC(C2(C)CN(C(=O)CN3CC=CC3)C2)=O)ccc2c(c1)OCO2 C(=O)(C1=CCCC1C)NCc1c(C(=O)NCc2c(C)noc2)n(C)nc1 c1(CN2CCC(N(C(C3CC(OCC)C3)=O)C)C2)ccc2n[nH]cc2c1 c1(C(N(CCCNC(c2cnc(O)s2)=O)C)=O)ccc(F)c(O)c1F Cc1ccc(C(F)F)cc1C(=O)NC(C)(C)CNC(=O)Cc1nc[nH]n1 C1(NC(CCCCCC)=O)C2CC3CN(C(=O)Cc4ccnc(F)c4F)C1C3C2 N1(C(CC2(C)CCN(C(c3ccc(C#C)cc3)=O)C2)=O)Cc2c[nH]nc2C(C)C1 N1(C(Cc2cn(C)nc2)=O)CC2(CC(C(=O)NCc3cocn3)CO2)C1 N1(C(C(CC)OCC)=O)CCC(NC(c2ccc(-c3ncn(C)n3)cc2)=O)C1C c1(N2CC(NC(C3CC(=C)C3)=O)C(C)CC2)cc[nH]c(=N)c1[N+](=O)[O-] N1(C(C2(OC)CCN(C(C3CC=C(C)CC3)=O)C2)=O)Cc2c[nH]nc2C1 C(=O)(C1=CC2CC=CCC12)NC(CN(C)C(c1cc(C(N)=O)co1)=O)(C)C C1(C(N2CCC(CN(C(=O)CN3CCCCC3)C)CC2)=O)COc2ccccc2C1 c1(C(N2CCC(C)(NC(=O)CCC3CCCC3)C2)=O)ccc2c(c1)OCO2 N1(C(=O)NC(C#C)CC2CCC2)CC2(CN(C)C(=O)OC)CCC1CC2 C=C(Cl)CC(C(=O)NCC(C)C1CCC1)NC(c1n[nH]cc1Cl)=O n1(CCC)ccc(C(c2nnnn2C)NC(COC)CC)c1 C(=O)(CCCC#N)NCC1CC(C(=O)NC(C)CCc2cn[nH]c2)C1 C1(NC(C(CCCC)CC)=O)CCC12CCN(C(c1cc(O)cs1)=O)CC2 C1(CCNC(C(Br)=C(C)C)=O)CCC(NC(=O)C(C)Cn2cccn2)C1 N1(C(C2(C)CC2Br)=O)CC2(C1)CN(C(c1nc(=N)cc[nH]1)=O)C2 c1(NC(C2CC23CCN(Cc2ncc[nH]2)CC3)=O)cnc2ccccn12 C1(C(N(CC(CC)OC)C)=O)CNC(=O)CN1C(=O)C(CC(C)C)N(C)C N1(C(c2nc(CC)sc2)C(=O)NC)CCOCC1C(=O)OC(C)(C)C c1(C(N2CCC(OCC(=O)OC)CC2)=O)cc(I)cc(Br)c1C C1(C(N2CCC(NC(COC(C)=O)=O)C2C)=O)CCc2ccc(F)cc2O1 O=C1CC(C(=O)NC2CC2NC(=O)CCOC2COC2)CC(=O)N1 N#Cc1cc(C(=O)NC2CCCCCN(C(=O)CC(=O)NC3CC3)C2)cc(O)c1 N1(C(c2c(C)cc(C)c(C)c2)=O)C(C)CC2CN(C(c3c[nH]nc3Cl)=O)CC12 C=C(C)CCC(=O)N(C1CCN(C(c2c(Br)cnn2CC)=O)C1)C C1(CNC(C2N(C)CSC2)=O)CCCCN(c2nnc(C(=O)O)s2)C1 C1(CCC#C)(CC)OCCO1.C12CCC(C1)n1cc(nn1)-c1cnc(s1)NC2=O N1(C(C(C)O)=O)CCN(C(=O)CC=C(Cl)Cl)C(c2ccc(F)cc2)C1 C(=O)(CCCCCC(S(=O)(=O)NNC(=O)c1c[nH]cc1C)OC)OC c1(OC)ccc(C(=O)N)c(F)c1N.C1(F)CCCC1.C(=O)C(F)=CC1CC1.C C1(C=O)CCc2nc(C)cn2C1.C1(F)CCC1.C1(C(=O)OC)CC1C(=O)N N1(C(C=CC(=O)N)=O)CC2(C1)OC1(C)CC2C1.C(=O)CCCCC.CC c1(C(=O)NC2CC3(C(NC(c4c(C)snn4)=O)C3)C2)cccc2c1CCCCC2 C=C(C)CCCC(=O)NC(C)CC1CN(C(C2CNC(=O)N2)=O)C1 N(C1c2ccccc2CC1NC(C1CC(CF)C1)=O)C(c1cc(O)cc(O)n1)=O C1(CCC)CN(C(=O)CCCCOC)CC1C(=O)NCCC1CC(C)(C)CO1 c1(CC)nccnc1CNC(=O)CC1CCCCN1C(c1coc(C)c1)=O C12CCC(CN(C(c3cn4cnnc4cn3)=O)C1)C2.O=C(C=O)NCC1CC1.N c1(C(N2C(CNC(CSC)=O)CCCC2)=O)c(C)c2ccccc2oc1=O Cc1c(CN2CCCC(C(=O)NCC3CC3(F)F)CC2)cccc1Br S(=O)(=O)(c1ccc(Br)c(C(=O)OC)c1)N1C(CC)CCC1C(=O)OC N1(C(CC2(C)CCCO2)=O)CCN(C(c2ccc[nH]2)=O)C(c2cn[nH]c2)C1 c1(C(N2C(C)CC(NC(=O)CCS(C)(=O)=O)CC2)=O)c[nH]c2c(Cl)cccc12 Cc1cnc(N2CC3C(C(=O)Nc4ncccn4)C3C2)nc1C S(=O)(=O)(c1cc(NC(c2cncc3ncc(C)cc23)=O)ccc1Cl)NC N1(C(COCCC=C)=O)CCCN(C(=O)CC2CCCC3(CC3)C2)CC1C C1(C#N)(C(N2CC(CNC(C(C)NC(COC)=O)=O)C2)=O)CCOCC1 C(=O)(CC(COC)COC)N(C(C)C(N1CC(O)CC1C)=O)CCC C1(C(N2CCC(CC)C2)=O)(C(F)F)CC(F)(F)C1.C(C)(C(=O)N)=C(CC)C N1(C(c2cc(C)c(Cl)cc2)=O)CC2CN(C(=O)CCC3CCC(=O)N3)CCC12 Cc1cc(CCNC(=O)NCc2ncc[nH]2)sn1 C(=O)(C1=C(Cl)CCCC1)N1CCN(C(C2(C)CCCS2)=O)CC1c1ccccc1 N1(C(C(CO)OC)=O)CCC2(CC1)CC(C)N(C(c1ccc(=O)n(C)c1)=O)C2 CN1CC(C(N2CCOCC2CNC(=O)C=CC=C(Cl)Cl)=O)CC1=O C1(CNC(CCCNC(N)=O)=O)CC(O)CN1C(=O)CC1CSCCS1 Cc1c(Cl)ccc2sc(=NCCNC(=O)C(C)SC3CCCCC3)[nH]c12 c1(C(N2C(CC)C(NC(=O)C3=CCC3)CC2)=O)cc2ccccc2nc1OC CC1(CNC(C2(C)CC2F)=O)CCN(C(=O)Cc2cccnc2O)CC1 CCC(C)(CNC(=O)C(O)Cc1cn(C)cn1)NC(c1cn[nH]c1)=O N(C1c2ccc(Br)cc2CC1C)CCSc1cccc(C)c1 N1(C(C=C(C)C(C)C)=O)CC(C)N(C(c2cnc(N(C)C)s2)=O)CC1C c1(C(=O)NCCCC=C)cc(C)c(CC)o1.c1(C(=O)N)ccc(-c2cccs2)[nH]1 C1(NC(CCCC=C)=O)CN(C(C2(CO)CCCC2)=O)CCC1CO C1(CCNC(c2cnc(COC)s2)=O)CCCN(C(C2CC(=O)CO2)=O)C1 C1(C(C)C(=O)N2CCC2C)CCN(C(C2(CO)CCOC2)=O)C1 c1(C(=O)NC(C2CCN(C(CC3CC(SC)C3)=O)C2)C)ccc(Cl)cc1N c1(OC)cccc(CNC(c2ccc(-n3cc(C4CCCCO4)nn3)cc2)=O)c1 C1(NC(CCC#C)=O)CN(C(c2oc(C3CC3)nc2C)=O)CCC1CO C(=O)(CC(C)C(C)C(C)C)NCC1(CNC(c2c(C)snc2)=O)CCCCC1 C1(CC(N2C(CC(=O)N(c3csc(Cl)c3)C)CC2)=O)CC2(CCC2)C1 N1(C(=O)C(F)(F)C2CCOC2)CCc2nc(F)ccc21 CC(C)(CCCNC(c1cc(C(N)=O)[nH]n1)=O)NC(=O)CC1CCCO1 Cc1nn(C)cc1C(C)C(=O)NCCNC(c1cnn(C2CC2)c1C)=O N1(C(c2ccc(CC)o2)=O)CC2CC1CCN2C(C1CC(CC)C1)=O CC1CC(C)(C(N2CCC(C(=O)NCCCC3(O)CCC3)C2)=O)C1 c1(C(N2CC(CCNC(C=CC)=O)OC(C)C2)=O)cnc2c(C)c(Cl)ccc2c1 N1(C(CCC(=C)Br)=O)CCN(C(=O)C(C)CC2CC2)C(C)C1 O=C(C#CC1CCOCC1)NCC1(C(=O)N2CCCO2)CCCO1 C1(C(=O)NC(c2nnc(C)o2)C)Cc2c(C)cccc2O1 N1(CCNC(c2c(C)cc(C)s2)=O)CCCN(C(C2CCC(O)CN2C)=O)CC1 c1(C(=O)NC(C(C)NC(CCCn2c(C)ncc2)=O)C)cccc(Cl)c1F C(=O)(C(CC)CCC)NC(C(=O)NCC(C#C)(C)C)c1ccoc1 N1(CC)CCN(C(c2nc(Br)cs2)C(=O)NCCCc2ccccc2C)CC1=O c1(SC)ccc2cc(C(=O)NCC(C)N(C)C(C3CCCN(C)C3)=O)[nH]c2c1 C12(NC(C=C(CC)C)=O)CCCC1N(C(c1cccc(C)c1)=O)CCC2 CC(C(C(=O)Nc1ccccc1Br)N(C)CCC1CC1)C(C)(C)C c1(C(=O)NCC(CC=C)NC(C2CCCN2CC)=O)ccc(Br)c(OC)c1 Cc1cccc(CNC(=O)C(C2CCN(C(=O)CNc3cc(C)on3)C2)F)n1 c1(CC(=O)N(CC(CNC(CCCc2ncc(C)o2)=O)O)C)cc(Cl)cc(Cl)c1 C(=O)(C1=CCCOCC1)NC1C(CC)N(C(c2cccc(CO)c2)=O)CCC1 C1(C2CCOCC2)(C(=O)NC(CC=C)CNC(c2sccc2OC)=O)CC1(F)F C(=O)(CCC(F)(F)C(F)F)N1CC(NC(C2CC2(F)F)=O)CC12CCC2 CCCC(C)N=c1[nH]c(=NC(C)c2cc(OC)ns2)[nH]c2ccccc12 CC1(CNC(=O)C=CC2CCCCCC2)CCN(C(c2csnc2Cl)=O)CC1 Cc1nn(C)c2sc(C(N3CCCC(NC(C4CCC(=O)N4C)=O)C3C)=O)cc12 CC1CN(C(c2cnccc2Cl)=O)CCCN1C(=O)C(O)C(F)F c1(C(=O)NCC(CCCC)NC(=O)CCc2ncc[nH]2)cn2c(C)cccc2n1 c1(OC)ccc(C(N2CC(NC(=O)Cn3c(C)csc3=O)CCC2C)=O)c(C)c1 CCCC(C(=O)NCC(N1CCCC1Cc1cc2nccn2cn1)=O)C(C)C c1n[nH]c(=NC2CC2)o1.N1(C(=O)OC(C)(C)C)CCCC1c1csc(C=O)n1.N N1(C(C2C(COC)C2)=O)CCC(F)(C)CC1.c1ccccc1F.C(=O)(CC)N c1(C(=O)NCCNC(C2N(C(CCC)=O)CCC2)=O)cc2c([nH]1)CCC(C)C2 Cc1cc(C(N2CCC(C(C)NC(=O)C(C)N(C)C)CC2)=O)c2ncccc2c1 N1(C(C2CC(=C)C2)=O)CCC(NC(c2cnccc2Cl)=O)C(OC)C1 C1(NC(CCC(C)OC)=O)CCN(C(=O)C(=Cc2cscn2)F)C(C)C1 C#CC1CCCC1NC(C1CN(C(=O)CC2C=NN(C)C2=O)CCO1)=O C(=O)(C(O)C(CCC)NC(=O)CC(CC)OC)N1CCC(O)(CC#C)CC1 C(=O)(C1c2[nH]cnc2CCN1C(C1CC1c1cccc2ccccc12)=O)OC Cc1ccc([N+](=O)[O-])c(C)c1CN1CCC(n2nnc3c2CCCC3)CC1 c1(C(C(=O)NCC2CCOCC2)N(C)C)cc(C(F)(F)F)cc(F)c1 Cc1nc(F)ccc1NC(=O)CCC1CCN(C(C2CC(=O)N(C)C2)=O)C1 c1(OC)ccc(CCCC(=O)NC2CCCC(NC(C3CCC(O)C3)=O)C2)cc1 C=CC1(O)CCN(C(C2C3CC4C(C3NC(c3nnn(C)c3N)=O)C24)=O)C1 C(CS(C)(=O)=O)N(C)C(c1n[nH]cc1NC(c1cnc(C2CC2)o1)=O)=O C1(CC(=O)Nc2n(C)ncc2I)CCC2(CC1)CCN(C(=O)CC#N)CC2 C1(NC(C(C)(C)C2CCCNC2)=O)CCCCC1CN.c1(CC2CC2)ccco1 CC1(C)C(CC(=O)NCC(C2CCC2)NC(c2ccc(Br)cc2)=O)C1(C)C N1(C(C2CCCN(CC)C2)=O)CCN(C(c2cc(Cl)ccc2O)=O)C(CCO)C1 N1(CCC)CCC(N(C)CCC2CCCCC2CC)CC1 C(=O)(C(O)C(C)(C)C)N(C(c1ccccc1)CNC(CCOC(C)C)=O)C N1(C(CCN(C)CC)=O)CCCC(O)C1.C(=O)(C(F)(F)c1csc(C)c1)N(C)C C1CCN(C2CCN(C)CC2)C1=O.CC(CNC(=O)OCc1ccccc1)C=O N1(C(CC(C)n2ccnc2)=O)CCC(C(N2CCCC2)=O)CC1(C)C c1(CC)ccc(CCC(=O)NCC2CCCCN2C(c2occ(C)c2C)=O)cc1 C1(NC(c2cnco2)=O)C2CCN(C(c3cn(C4CCOCC4)nn3)=O)C12 C(=O)(C(C)(C)NC(=O)CCCNC(=O)CCc1cnn[nH]1)NC CC1CCCn2ncc(C(=O)NCC3(F)CN(C(=O)C(F)C(C)(C)O)C3)c21 c1(C(N2CCC(NC(c3cc(C)ns3)=O)C(F)C2)=O)ncn2ccccc12 c1(C(=O)NC2(CNC(c3c(C)[nH]c(C#N)c3)=O)CC2)cc2ccccc2nn1 C(=O)(C1=NN(C)C(=O)CC1)NCC1CC(NC(c2cc(C)cc(Cl)n2)=O)C1 CC1CCCC(C(=O)NC(C)(C)C2CCC2)C1.c1(C=O)cnc(N(C)C)nc1.N c1(C(N2CCC(CC=C)(NC(=O)Cn3ccnc3CC)C2)=O)cc(C)ccc1O C1(C(=O)NC2CC(C)(CO)C2)C2CC3C(C2NC(c2cc(Cl)n[nH]2)=O)C13 n1(CCC(=O)NC2CN(C(C3(F)CCC3)=O)CC2O)cc[nH]c(=O)c1=O C1(CNC(CS(N)(=O)=O)=O)CC2(CCC2)CN1C(C1CCc2ncnn2C1)=O C1(CN(C(c2csc(CO)n2)=O)CC)CCCN(C(=O)C)C1.C1(C)CCC1 c1(CNCC2N(C(C(n3ncc(C)c3)C)=O)CCOC2)ccc(F)c2ccccc12 C1(CNC(C2C(=C)CC2)=O)N(c2nnc(C(C)C)o2)CCCC1(C)C N1(C(CCC#C)=O)CCCN(C(c2ccc(-n3cncn3)c(N)c2)=O)C(C)C1 CC1CC(C)(C)CN1C(=O)C(Cc1ccco1)NC(C1CC2CC2C1)=O C(=O)(C(CC(C)(C)C)OC)NCCNC(C1OCCN(CC)C1)=O N1(C(C(=O)NCCSC)C2CCSC2)CC2CC1(c1cccs1)C2 N1(C(CC)=O)CCC2C(NC(c3csc(C4CC4)n3)=O)C2CC1 Cc1c(C(=O)NC2(CNC(=O)CC(F)(F)F)CCC2)nnn1C Cc1nn(CCO)c(C)c1C(=O)NC1CS(=O)(=O)CC1.C(=O)CC.C1CC1 C(C(C)(C)C(=O)N1CC2CC1C2)NC(c1c(C)ocn1)=O C1(CNC(C)=O)C(C)CCN1C(c1cccc(CC(F)(F)F)n1)=O Cc1[nH]c2ccc(O)cc2c1C(N1CCC(CF)(NC(C2CCCCS2)=O)C1)=O c1(CNC(=O)Nc2cn(C(C)C)nc2I)cc2cc(Br)ccc2s1 FC1(F)CCC2(CCC(CNC(c3ccccc3Br)CCCO)O2)CC1 C1(c2n(CC)nnn2)(NCCc2cnoc2)CCCCC1CCC#N C(CC(C)CCNC(c1sccc1NS(C)(=O)=O)=O)NC(CCCOC)=O Cn1nc(C(=O)NC2CCN(C(C3(S(N)(=O)=O)CCC3)=O)C2)c(Cl)c1Cl c1(N2CC(OC)(CNC(=O)C(=O)NCC(F)F)C2)nc(Cl)nc(C)c1Cl n1(CC(=O)N(CCCNC(C(C)N(C)C)=O)C)nc(-c2ccccc2)oc1=O N1(C(Cc2[nH]c(=N)sc2)=O)CCCCC(NC(c2ccncc2Cl)=O)C1 N1(C(CC(c2ccccc2Br)C)=O)CCC(CNC(=O)CO)C12CCC2 N1(C(c2c(C)scn2)=O)CC(NC(=O)C=CC)C(C)(C)C1.CCN(C)C C1(C(N2CC3CC2CN3C)=O)(NC(C(CC)=CCCC)=O)CCC(C)(C)C1 C(C(=O)N(C1CCN(C(=O)C=Cc2cnn(C)c2)C1)C)(C(C)(C)C)OC c1(C(N2CCC2)=O)cc([N+](=O)[O-])c[nH]1.CN1CCC(CCNC(=O)C)C1=O.O C=CC(CCC)CC(=O)N1CCCC1Cn1cc(COC(C)C(=O)OC)nn1 C(C(C(F)(F)F)N1CCN(c2ncncc2I)CC1)NC(=O)COC(F)F C1(C(=O)NCCCNC(CNC(=O)OCC=C)=O)CCC(C)O1 C1(C=O)CCCCC1n1cccc1.n1(CC(=O)NCCC2CC2)cc(Cl)cn1.N Cc1nc(C(=O)NCCC2(NC(C3CC34CCCC4)=O)CC2)c2ccccn12 c1(C(=O)NC2CCN(C(=O)CC3CCCO3)C23CC3)cc2cc(Cl)ccc2[nH]1 C1(NC(C(C2CCCC2)OC)=O)CCN(C(=O)CC2(N(C)C)COC2)C1C c1(C2(NC3CCC(CC(C)C)C3)COC2)ccc(F)cc1 c1(N(CC(CN(C(C)=O)C)O)C)cnn(CC(C)C)c1 N1(C(C(C)n2cnnn2)=O)CC(C(=O)NCCCn2nccn2)CCC1(C)C c1(C(N2CCC(F)(CN(C)C(C3CC3)=O)C2)=O)cnn(C)c1-n1cccc1 C(=O)(CCC(F)(F)C(F)(F)F)N1CC(CN(C)C(c2ccncc2)=O)OCC1 CC(CNC(=O)C=Cc1cocn1)C(F)C(=O)NCc1nccc(O)n1 C(C1c2ccsc2CCN1C(=O)CCCC1CCC1)NC(C1ON=C(CC)C1)=O N1(C(C(C)SCC)=O)CCC2(CCC2NC(c2cccc(C)c2)=O)CC1 C12(CNC(C(CC#C)C)=O)CN(C(=O)Cc3ccc(F)c(OC)c3)CC1CCO2 C1(OC)(CNC(c2cc(C)n(CCO)n2)=O)CCN(C(=O)C(C)C#N)CC1 CCC(C)CCC(=O)NCC(C)(O)CNC(=O)Cc1ccc(-n2ccnc2)cc1 N1(C(c2c(C)[nH]nc2Br)=O)C2CCC(C2)C1CNC(=O)CC(=O)N(C)C c1(C(=O)NC2CCN(C(c3c(Cl)cn(C)n3)=O)C2)ccc2oc(S)nc2c1 N1(C(C=C(C)C(C)C)=O)CCC(CO)C(NC(=O)CN2CCC(F)(F)C2)C1 C1(NC(c2c(CC)ncnc2)=O)CCCCCN(C(c2sc(OC)nc2Cl)=O)C1 c1(C(N(CCCN(C(c2cc(CSCC)on2)=O)C)C)=O)ccc(=N)[nH]n1 c1(OC)cc(COCC(=O)N)ccn1.C1(F)CN(C(c2ccco2)=O)C1.C C1(C(=O)NC(CC)C)(CC)CN(C(=O)C(n2nccc2C)C)C1 c1(C(N2CC(C)C(C)C2)=O)ccc([N+](=O)[O-])n1C.c1(C(=O)N)ccc(N)c(O)c1 CC(CC(=O)N1CCC(CC(=O)NCCc2cc[nH]n2)C1(C)C)C(C)(C)C N1(C(c2cn(C)nc2Cl)=O)CCC(NC(c2ccc(O)nn2)=O)C1(C)C C1(CNC(C=CC)=O)C2CN(C(c3cc(C(F)F)no3)=O)CC12 N1(C(C(C)NC(=O)OC)=O)CCC(C(=O)NCC(c2ncc(C)s2)C)C1 C1(C)(NC(c2cc(OCC)no2)=O)CCCCC1.c1(C(=O)N)cn(C)nc1C C=CC1(C(=O)N(CC(O)CF)C)CCN(C(=O)CC2CSCCO2)C1 C1(CC)CN(C(c2occ(C)c2C)=O)CCC1NC(c1cccnn1)=O C1(NC(C(CC)CC)=O)CC2CC1CN2C(c1ccc(Cl)cc1Br)=O C=Cc1ccc(C(=O)NC2CN(C(=O)C(C)(C)CC3CC3)CCC2CO)cc1 C(C1=CCN(C(c2cnc(O)nc2)=O)CC1)NC(c1c(OCC)oc(C)n1)=O C1(C(=O)OCC)CSC(C)N1C(c1nc(-c2ccccc2)cs1)=O c1(OC(C)C)ccc(C(=O)NCCCC)c(Cl)c1.C1(=CC(=O)N)CCOCC1 c1(N2CCN(Cc3c(C(=O)OC)nccc3)CC2)ncc2c(C)cn(C)c2n1 C1(O)(CC(=O)NCCCC2N(C(c3c(C)con3)=O)CCC2)CCOCC1 C(=O)(CC(O)CC)NC(c1ccccc1)C(=O)NCCSCCOC C1(C(=O)Nc2ccc(C)nc2C)CC(C)(C)CCN1C(=O)C(C)C1CCC1 n1(CCC#C)cc(NC(c2ccoc2C)c2nnnn2CCC2(C)CC2)cn1 C1(CC(N2CC(CC)C2)=O)CCC(F)(F)CC1.c1(OC)ccccc1CC(=O)N c1(N2CC(CC(N=c3c(C(=O)OC)no[nH]3)=O)C2)ncnc2ccc(Cl)cc12 C1(NC(Cn2cc(C3CCCC(C)C3)nn2)=O)CCCC2(CCC2)C1 C(C)(C(=O)N=c1ccn(CCF)[nH]1)N(C(CC(C(C)C)O)=O)C.C1CC(O)C1 C1(NC(C(CC)(C)C)=O)CN(C(C2CC(=O)N(CC(C)C)C2)=O)CCC1C N1C(=O)CCNC1=O.C12CCCC1C2(F)F.C(CS(=O)(=O)CC1CC1)C(=O)N O=C(C(F)C1=CCCCC1)NCC1COCCN(C(=O)C=Cc2cnccn2)C1 CCC(CC(=O)N(CC(C)N(C)C(c1ccn(C(C)C)n1)=O)C)C(F)F C(=O)(CCN(OC)C(=O)C12CCC(CC1)CO2)N1CCC(COC(C)=O)C1 C1(NC(CCCCOC)=O)CCSC12CN(C(c1ccc(N)cc1Cl)=O)C2 CC(=O)CCCC(=O)Nc1nnc(C2CCCOC2)s1 C(=O)(C(CC)CCCCC)NCC(=C)CCNC(c1cn(C2CCC2O)nn1)=O N1(C(c2c(CC)cccn2)=O)CCCOC(CNC(=O)C(C)N(C)C(C)=O)C1 N1(CC)CCCC1C(=O)NC(C)C(C)NC(c1ccoc1C1CC1)=O c1(-c2ccc(N(CC)CC)cc2)cccc2c1CN(C(=O)CN(C)C(C)=O)CC2 C(=O)(C1SCc2cccnc21)NC1CN(C(c2c(C)nns2)=O)CC1C N(S(=O)(=O)N=S(=O)(c1ccccc1)C(F)(F)F)C(C1C(C(C)(C)C)C1)=O C1(NC(C2(CC(C)C)CC2)=O)COC2(CCN(C(=O)CCCCC(F)(F)F)C2)C1 c1(CC)conc1CC(=O)NCc1ccsc1C(=O)NCCCOC(=N)O c1(C(N(C2C3CN(C(c4cnc(O)n4C)=O)CC23)C)=O)ccc(C(F)(F)F)cn1 c1(C(C(=O)NC2CC2)N(C2CCC(F)(F)C2)C)cc(Cl)cc(Cl)c1OC C1(C2CCN(C(c3ccnc(-n4cncn4)c3)=O)C2)(NC(CC(C)C)=O)CC1 c1(C(=O)NC(C(=O)OCC)C2CC2)c(-c2ccccc2Cl)noc1C CC1=C(C(=O)NC2CC(CCNC(c3csc(C(F)F)n3)=O)C2)CCO1 CC1CN(C(=O)C=CCNC(c2cccc(=O)n2C)=O)C(C)(C)C1 N1(C(c2cc(COC)on2)=O)CCC2CCC(NC(=O)C3=CCCCO3)C1C2 Cc1ncn(C)c(=O)c1C(=O)NCC1CCC1(C)C.c1(C(=O)N)ccoc1Br C1(CCOC)CCCCC1N=c1c([N+](=O)[O-])c[nH]c2ccc(N(C)C)cc12 C(=O)(C(C(C)C)NC(=O)CN1CCC(C(C#N)C#N)CC1)NC C(C)(C(C(=O)NCc1cnccc1Cl)C(C)C)NC(C1CC(SC)C1)=O CCC(CCOC)C(=O)N(C1CN(C(=O)Cc2coc(C(F)F)n2)C1)C CCCCC(CC)C(=O)NCC(C)(CNC(=O)Cn1nccc1C)OC C#Cc1ccc(C2(C(=O)NC)CC2)cc1.c1(CCC=O)cc(Cl)no1.C1CC1 c1(CCC=O)ccc(C(N)=O)cc1.C=CC1(C(=O)NCC=CC)CCC1.N CC(C)C(C(=O)NCCC(C)N(C)C(c1ccc(C(F)(F)F)[nH]1)=O)n1cnnc1 Cc1cc(=NC2CN(C(=O)C=CC3CCOC3)CC23CCC3)[nH]c(C)c1C#N Cc1cccc(Br)c1C(C(=O)N(C(C)C(F)F)C)NC(C1CCC(F)(F)C1)=O CC(C)(C)C(=O)C(=O)N1CCCC(C)(CNC(c2cnc(Cl)cc2Cl)=O)C1 CC1(C(=O)NC2CCCN(C(c3cc(-c4ccco4)on3)=O)C2)CCC12CCC2 Cc1ccc(O)c(C(=O)NC(C(=O)N2CC(N3CCCCC3)C2)c2ccco2)c1 C(=O)(C(C)(C)C(=O)NC(C)CC(C)C)NC.C1CC(F)(F)C1.C(=O)C.N C=CCCC(C(=O)NCC1OCC2CCC1C2)NC(C1CC12CCCC2)=O N1(C(c2c(CC)nc[nH]2)=O)CCCCC(NC(c2c(C)cccc2Cl)=O)C1 c1(C(N(CC(CC)NC(c2cnc(C)n2C)=O)C)=O)cc(C)nn1CC(F)F CCC(CC)CN=c1nc(NCCc2c[nH]nc2C2CC2)c2c([nH]1)c(C)nn2C C1(C(=O)NC(CNC(CNC(CC)=O)=O)CC(C)C)CCOCC1(C)C C(=O)(C#CC(C)(C)C)NCC1(CO)CCN(C(C2N(C)CCC2)=O)C1 CC1CN(C(c2cc(Br)n[nH]2)=O)CC1NC(c1c[nH]nc1C1CCOCC1)=O C(=O)(CCCCCS(N)(=O)=O)N1CCCC(N(C)C(c2ccc3cnoc3c2)=O)C1 Cc1cccc(C)c1C(=O)NC(=O)C(C)NC1(Cc2ccccc2)CC1 C[S+](C)CCC(O)C(=O)N1CC2C(CNC(c3ncccc3N(C)C)=O)C2C1 C(=O)(C1=CCN(C)C1)NC(CC(=O)NCC1(OC)CCOC1)(C)C N1(C(C(C)OCC#C)=O)CC2CC1CC2C.c1(CC(=O)N)ccc(Cl)cc1F c1(CC(N2CCC(O)C2)=O)ccc(S(=O)(=O)CC)cc1.N1(CC)CCC1C=O.N c1(-c2cccc(OC)c2)ccc2c(CC(=O)Nc3cc(C)nn3C)n[nH]c2c1 c1(C(C)=O)cc(NC(C2CCN(Cc3conc3C)CC2O)=O)ccc1O Cc1ccc(N)c(C(=O)NC2CC(C)(CNC(C3CCCN3N=O)=O)C2)c1 C1(C)(CC)CCCN1C(=O)C.C(=O)C(C)(C)c1ccns1.C=O.C1CC1.N C1(C(N2CCN(Cc3n(CC)nnc3C)CC2)=O)CCCC(C)(C)C1 c1(C(N2C(C)CC(CNC(=O)CCCC(F)(F)F)C2)=O)cccc2nc(S)oc12 Cc1nc(COc2ccc(Cl)nc2)sc1C(=O)OCc1ccccc1 C1(CC)(OC)CN(C(c2nc(C3CC3)cs2)=O)C1.c1(CCC=O)ncnn1C.N C(=O)(C(C)S(=O)(=O)C(C)C)N1C(CCCC)CN(C(=O)Cc2cncs2)CC1 CCCC(C(=O)NCc1cnccn1)NC(C1CCCN1CC)=O N1(C(C(C)SC)=O)CC(NC(C2(c3ccc(F)cn3)CC2)=O)CC(C)C1 c1(OC)cccc2c1CCC2OC(c1cc(Br)cc2c1OCCO2)=O C1(CCNC(CC2(C=C)CC2)=O)CCN(C(c2ccnc(C(C)C)n2)=O)CC1 N(C1CCc2ccc(O)cc21)C(C(=O)Nc1c(C)cc(C)cc1C)C C(CC(=O)N1CCC(N(C(=O)CCOC2CC2)C)C1)(C(C)C)OCC C(=O)(CCCCCC#N)NCCC(C)NC(c1c(C)ncnc1C)=O CN1C(=O)CSC1=CC(=O)Nc1cccc(C(C)(F)F)c1 Cc1ncncc1C(N1CCCCC1CNCC1(C#N)CC1C(F)(F)F)=O Cc1c[nH]ccc1=NC(=O)C1CCN(C(=O)COC(C)(C)C)C1 c1(C(=O)NCC#CCNC(CC2C(C)CCC2)=O)c(O)nnc2c1CCCC2 Cc1cc2c(cc1C)OC(C(=O)NC1CC3(C1)CN(C(c1csc(O)n1)=O)C3)C2 c1(CC)csc(CNC(=O)C(C2CCCC2)NC(=O)CC2CCOC2C)n1 C1(N(C(C)=O)C)CCCC(N(C(=O)COC2(C)CCC2)C)C1 n1(CC)ncn(NC(=O)CC(C)N(C(=O)CC2COC(=O)C2)C)c1=O c1(SC)nc(N2CCCCC2CNC(=O)C(C)n2ccnc2)cc(Cl)n1 N1(C(C(CC)OC)=O)CC=CC(C(=O)NCCc2cocn2)C1 C1(C(=O)NCCCSCC)CCCCN(C(=O)C)C1.C1CN(C(C)=O)C1.N C1(NC(C2ON=C(C)C2)=O)CN(C(c2ncc(C#N)cc2C)=O)C2CCCC12 N1(C(C2CCS2)=O)CCCC(c2ccc(OC)cc2)(COCCO)C1.C(C)C c1(C(N2C(C)CC(NC(CC(CC(C)C)C)=O)C2)=O)cc2cc(Cl)ccc2[nH]1 C(CC(C(=O)NCC(O)CCSC)NC(=O)C(C)c1cc[nH]n1)SC CC1CCN(CC(=O)NCC(=O)NCC(N2CCCCC2)=O)CC1 C1(C#N)(C(N2CC(CCNC(CC=CCC)=O)OCC2)=O)CC2CC2C1 C1(C(=O)NC2CCOCC2)CCN(C(C2CCC(C(F)F)O2)=O)C12CCC2 CCC(CCCC(=O)NCCOC1CCOC1)NC(c1ccc(C)[nH]1)=O CCCCC(CC(=O)NC1CCC2(CC2)C1)NC(=O)CCC1CCC1 C1(NC(c2c(CC)ccs2)=O)CC2CN(C(c3cn(C)nc3O)=O)CC2C1 c1(C(N2C3CC(CNC(C(CC)C)=O)C2CC3)=O)cccc2[nH]ccc12 c1(OCC)nccnc1.C1(C(=O)N)CSCCN1C(c1ccc(C(N)=O)cc1)=O c1(C(C)NC(CNC(C)C(F)F)=O)nc(C(F)(F)F)n[nH]1 C1(NC(c2ccc(C(C)=O)[nH]2)=O)CCCC(N(C(=O)CCc2ccnn2C)C)C1 C12(C(=O)NCC3N(C(=O)COc4ccc(O)cc4)CC3)CCCC1C2(F)F Cn1nc(C(N2CCOCC(O)C2)C(=O)NC2CC2)c2c1CCC(F)(F)C2 c1(CC)ccc(F)c(C(=O)NC2CN(C(C3CC3C(C)(F)F)=O)CC2O)c1 C1(NC(c2nc(N(C)C)oc2)=O)COCCC1NC(C1(CCF)CCC1)=O CCC(C)(C)CCCC(=O)NC1CCC(C)N(C(c2ncc3n2CCCC3)=O)C1 N1(c2n(CCC=C)c(C3(O)CCC3)nn2)CCC2(CC1)C(OC(C)C)CC2O CC1(C)CC(CC#N)(C(=O)Nc2ccc(CC(N)=S)cc2)C1 N1(C(CCCNC(N)=O)=O)CCCC12CCN(C(C1CC1c1ccccn1)=O)C2 c1(C(N2CCN(C(c3cnc(C)o3)=O)C(C)C2)=O)ccc2ncn(C)c2n1 Cc1cc(CO)ncc1C(=O)NCC1CN(C(c2c[nH]nc2C2CC2)=O)CCO1 c1cnn(C)c1C=O.n1(CC)ccc(CC(=O)NC)n1.c1(CC)cnn(C)c1 c1(C(N2CCOC(CNC(C3(CO)COC3)=O)C2)=O)cnc(Cl)cn1 N1(C(CC2OCC(C)(C)OC2)=O)CCC(NC(=O)CC(C)(C)C2CC2)C(C)(C)C1 Cc1ccc(Cl)cc1C(N1CC2CCC2(CNC(C2(C)CC2(F)F)=O)C1)=O C1(CCOC)CN(C(=O)C2=CC(C)(C)C2)CCN1C(c1cncc(OC)c1)=O C(C(CC(C)C)C(=O)NC(c1ccnn1C)C(=O)NCCC1(CO)CCC1)OC C1(N(C(=O)COCC2CC2(C)C)C)CCN(Cc2ccncc2)C1 C1(O)(CNC(c2cncn2C2CC2)=O)CCCN(C(=O)C=CBr)C1 N1(C(C(C)SC)=O)CCC2(CCCN2C(c2ccc3n[nH]cc3n2)=O)CC1 C(=O)(C1=C2CCN=C2NC=C1)NCC1N(C(CC(COC)(C)O)=O)CC(F)C1 C1(CNC(Cn2nnc(=N)[nH]2)=O)CC(F)CN1C(=O)C(=O)Nc1ccccc1 c1(C(=O)N)cc(O)cc(Cl)c1.C(CCCNC(c1[nH]nnc1C1CC1)=O)OC CC(=O)CCCC(=O)N.C12CCC1CN(C(=O)CN(C)C=O)C2.C(C)(C)C.C c1(CN(c2ccc(C3CCCO3)nn2)C)ccc(Br)cc1 c1(CCC(=O)N(CCNC(c2nnn(C)c2C)=O)CC)cccc2cnccc12 CC1CN(C(=O)C(O)CN2CCCC2)CC1CC(N1CCCC1C1CC1)=O c1(OCCC)cccnc1C(N1CCC(COC)(NC(=O)C(O)C)C1)=O.S N1(CCC(=O)NCCC2CCCN2C(c2cnc(Br)s2)=O)CCC(F)C1 CCC(C)CC(C)C(=O)N1CC(N(C)C(c2cccc3c2CCC3)=O)C1 C(=O)(CC(C)(C)C(F)F)N1CC(C#C)OCC1 N1(C(CC(C)C2CC2)=O)CC(NC(=O)C(F)C2CCC2)CC(C)(C)C1 N1(C(CC(CCC)C)=O)CCC2C1CCCN2C(c1sc(CC)nc1C)=O c1(C(=O)Nc2ccc(C(N3CC(C)OCCC3)=O)cn2)cc2cnccc2[nH]1 C1(CCC)CN(C(C2CCCN2C(C)C)=O)CCN1C(c1oc(CO)cc1C)=O CC(C(=O)NCCSCC(=O)NCC1CCCCC1(C)C)S(C)(=O)=O c1(CC)nncn1NC(=O)C1CCN(C(C2CN(C(N)=O)C2)=O)CC1 C1(NC(c2cccnc2)=O)C2CCN(C(C3(C(F)(F)F)CCCC3)=O)CCC12 C=C(Cl)CC(C(=O)NCC1(O)CCC1)NC(=O)C(F)C(F)(F)F C1(NC(C(C)SC)=O)CCCCC1CNC(C1CC(C)(CO)C1)=O C1(C(=O)NCCC2CNCCCO2)C2Cc3c(Br)cccc3C12 c1(NC(C2NCCN(C(c3cc(OC)nn3C)=O)C2)=O)nccc(F)c1F C=CC(CC)C(=O)NC(C(=O)NCC1(CC(C)C)CC1)c1cccs1 C1(NC(COCCC)=O)CN(C(=O)Cc2csc(Cl)c2)CC2(CCC2)C1 C1(C(N(C2CC2)CC2N(C(CN(C(C)=O)C)=O)CCC2)=O)CCCN1C=O C1(NC(=O)OC(C)(C)C)CN(C(c2ccc3c(c2)CC3)=O)CCC1O c1(C(=O)NCC(C)NC(C2C(COC)C2)=O)cccc(C(C)C)c1N S(=O)(=O)(c1cccc2c(Cl)cccc12)N1CCC(OCC(=O)O)C1 Cc1csc(C(N2CC(NC(c3nsnc3O)=O)C(n3ccnn3)C2)=O)c1C CC(O)C(C)(C)C(=O)N1CC(F)(CNC(c2coc(C(F)(F)F)c2)=O)C1 Cc1nc(=NC(CNC(c2c(C)nsc2C)=O)C2CCC2)s[nH]1 N1(C(c2c(C)n(C)nn2)=O)CCC2(CCN(C(C3CC3C3CC3)=O)C2)C1 C(=O)(C1CCc2nccn21)NCC(CN(C(=O)CC1(O)CC1)CC)(C)C C1(CNC(C(C=C)(C)C)=O)CC(C(=O)N2CCC(C)(N(C)C)C2)=NO1 N1(C(c2c(COC)scc2)=O)CC2C(NC(=O)C=C(C)Cl)C2C1 N1(C(C(C(C(C)C)O)(F)F)=O)CC2C3CCC(C2C1)N(C(C1(C)CC1)=O)C3 C#CC1CCC(CNC(c2cnn(-c3ccncc3)c2)=O)CC1 C#Cc1ccc(OCC(=O)NC(C)CCN(C)C(C2(CO)CCC2)=O)cc1.O c1(CCC(=O)NC2(CCCNC(CCCCOCC)=O)CC2)ccccc1C#N C1(C(=O)NCc2c[nH]nc2C2CC2)C=CCN1C(=O)C=CC1CCC1 c1(C(N(C2(C(=O)NC(C3CCOC3C)CC)CC2)C)=O)cccnc1 c1(C(N2CCC23CCCOCC3)C(=O)NCCC2(C)CC2)n[nH]c2cc(F)ccc12 C#CC1(C(=O)NCC(C)N(C)C(c2ccc(Cl)cc2)=O)CCCC1 C#CCCCCCCC(=O)N1CC(CNC(c2cc(F)ccc2F)=O)C(F)(F)C1 C1(C(=O)NCCCN(C(C=C(COC)C)=O)C)(C(C)C)CCCO1 C1(CC)C(NC(c2cn(CCO)nn2)=O)CCN1C(=O)C(CCSC)OC Cc1ccc([N+](=O)[O-])c(NC2CCN(C(=O)CC3(O)CCCC3)C(C)C2)c1 C1(NC(CC(=O)NCC)=O)CCC2CN(C(=O)CC(O)CC)CC2C1 N1(C(C2C(C)(C)C2(F)F)=O)CC2CCN(C(c3ccc(O)cc3)=O)C2C1 C1(CC)C(C(=O)NC(c2ccncc2)C)CCCN1C(c1ccccc1CC)=O C1(c2ccccc2)(C(=O)NCCCNC(C(C)n2ccnc2)=O)CC(F)(F)C1 C1(NC(C2CC(C)OC2)=O)CCN(C(=O)Cc2csc(=N)[nH]2)CCC1CO c1(OC)ccnc(Cl)c1OCC(=O)NC1CCS(=O)(=O)C1 c1(C(=O)NCC(CCCC)NC(c2cscn2)=O)cccn2ncnc12 N1(C(c2cc(N)c(F)cn2)=O)CCCC2(C1)CN(C(c1cscn1)=O)C2 C1(C(N(C2CCN(C(C3CC(C)(C)C3)=O)C2)C)=O)CC2CC(C1)C(=O)N2 c1(C(N2CCC(CNC(C(CC)OCC)=O)C2)=O)cccc(C2CC2)c1Cl S(=O)(=O)(c1ccc(Cl)cc1I)N(C1CCC2CCC1C2)C C1(N(C(c2cccc(F)c2)=O)CC)CCCN(C(c2ccc(O)nc2C)=O)CC1 C1(N(C(CCc2cnc(C)o2)=O)C)CC2CCC(C1)N2C(=O)C(O)CC(C)(C)C C1(NC(Cc2ccn(CC)n2)=O)CCCC2CN(c3nc(CCOC)ns3)CC12 N1(C(=O)NCCc2c(C)ccc(C(=O)O)c2)CC(C)c2ccncc21 c1(CCNC(C(c2cscn2)N(CCC(F)(F)F)CC)=O)cccc(F)c1 CC(CC(=O)Nc1ccc(-n2ccnc2)cn1)C(=O)c1ccc(Cl)cc1 N1(C(c2csc(C)c2N)=O)CCC(C)C(CNC(=O)Cn2ncnn2)C1 c1(C(N2CCC(NC(c3ccc(SC)s3)=O)CC2C)=O)cn2cc[nH]c(=O)c2n1 C1(NC(c2ccnn2C)CC)CCOCC1 C1(C#CC(=O)NCC(C)(C)NC(c2ccnc(C(C)C)n2)=O)(CC)COC1 N1(C(C2N(C)CC(O)C2)=O)CC(C(=O)NC2CN(C)CC2(C)C)CCC1(C)C C1(C(N(CCC)CC)=O)CS(=O)(=O)CC12CC2.c1(C=O)ccc(Cl)nc1O.N N1(C(C(C(C)C)SC)=O)Cc2ccccc2C(Nc2cc3nnc(C)n3cn2)C1 C1(NC(C(C#C)(C)C)=O)CC2CC(NC(c3ccc(Cl)nc3OC)=O)CC2C1 C1(CNC(c2cc(C)no2)=O)CN(C(=O)C(C)C2(O)CCC2)CC(C)(C)O1 C1(NC(C2C(C)(C)C2(F)F)=O)CCN(C(c2ccccc2Cl)=O)C12CC2 c1(C(N(CC)CC)=O)ccc(Cl)cn1.C(C)C=O.CCC.CC.C(N)=O.O O=C(C1=Cc2ccccc2OC1)NCC1CN(C(=O)CCn2ccnc2)CCO1 c1(C(=O)Nc2ccc(C(N3CC(O)C(F)C3)=O)nc2)ccc(O)c2ncccc12 C1(CCNC(C(C=CCCC)O)=O)CCCN(C(=O)CS(=O)(=O)NCC)C1 c1(C(N2CC3C(C(=O)NCCCC(C)O)C3C2)=O)cc2occc2[nH]1 c12cccc(c1)CN(C)C2=O.N1(C(=O)NC23CNCC2C3)CCCCC1=O n1(CCN(C)C)nccc1C(=O)N(C1CCN(C(=O)C(c2ccccc2)O)C1)C c1(C(=O)NC2C(O)CCN(C(CCCC#CC)=O)C2)cc2ccccc2s1 CCN=c1ccc(C(=O)NCC2CN(C)CCN2C(=O)Cc2cn[nH]c2)c[nH]1 N1(C(c2c(C)scn2)=O)CCCC(C)(CNC(=O)C(CC(C)C)N(C)C)C1 C1(C#N)(C(=O)NC2C(CC(=O)N(CC(C)(C)C)CCO)C(O)C2)CCCO1 Cc1nc(C)c(CNC(C2CC(NC(C3CCCC3F)=O)C2(C)C)=O)[nH]1 c1(CC=O)ccc(Cl)c(F)c1.c1(C(N(C(C)C2CC2)C)=O)ccc(O)cn1.N N1(C(CCNC(COC)=O)=O)CCC(C(C)(C)C=O)C1.C1CC(C(C)O)C1.N N#CC1=C(C(=O)NCC(CO)NC(c2cncc(C3CC3)c2)=O)CCC1 N1(C(c2cc(C)sc2C)=O)CCC(N=[N+]=[N-])(C(N2CC3CCCC(C3)C2)=O)C1 CCCCCNC(c1ccc(CNS(C)(=O)=O)o1)=O.C(=O)CCSC.N C1(NC(c2scc(OC)c2)=O)CCC2(CC1)CN(C(=O)CSC(C)C)CCO2 C1(C(=O)NC2CCN(C(COCC(=O)NC)=O)C2C)CC(C)CC(C)(C)C1 c1(NC)ccc(C(F)(F)F)cc1C(=O)NCCCOCC.C(=O)CC(F)F N1(C(c2cccc(C(N)=O)n2)=O)CC2CCC2(CNC(C2CC2(Cl)Cl)=O)C1 Cc1c(C(=O)NCCNC(=O)C(C)Cc2ccccc2)oc2ccc(F)cc12 Cc1ccc(C(=O)NCC(C)CNC(c2nocc2-c2ccccc2)=O)o1 c1(C(N2CCC(C)C(CC(N3CC(CO)(CF)C3)=O)C2)=O)cc2ncccc2[nH]1 CCCC(O)CC(=O)N1CCOCC1CNC(=O)Cc1cccnc1 Cc1cc(F)ccc1N(C1CCC(N(C)C)CC1)C(N1CCN(C)CC1)=O C(=O)(C1Cc2ccc(F)cc21)NC1CC(C)N(C(c2n[nH]c3c2COCC3)=O)C1 C#CCC(C(=O)NC)NC(C12CC1CN(C(=O)CC1OCCO1)C2)=O N1(C(C(Cn2cncn2)NC(C23CCCC2C3)=O)=O)CCCC2CCCCC12 CC1CCN(C(C23CCCC2C3(F)F)=O)CCN1C(c1cnc(C(C)(C)C)[nH]1)=O N1(C(COCCC)=O)CC(CNC(C2CC(F)C2)=O)CC1(C)C Cc1ccc(C(=O)NCC2(NC(=O)Cc3cnns3)CCCCCC2)c(Cl)c1Cl N1(C(C23CC(COC)(OC2)C3)=O)CCCC(O)C1.c1(CC=O)conc1C.C Cn1cnc2c1C(C(=O)NCCCCNC(C1(C(F)F)CCC1)=O)CC(=O)N2 C(CC(C(=O)N(C(CCF)C(=O)O)C1CC1)c1ccccc1)=C(C)C c1(OC)ccnc(CNC(=O)CC)n1.C(=O)(C(C)=C1CCCC1)N(CC)C C(=O)(C(O)CC(F)(F)F)NCC(C)C(=O)NCCOCC(F)F CC1=CCC(C)(C(=O)NCC#CCNC(c2ncccc2C)=O)CC1 CC(C)CC(C(=O)N1CCCCC1C1CCN(C(=O)Cn2cccc2)C1)N(C)C c1(C=O)cc2ncccc2[nH]1.C(=O)(C(C)C(C)C)N(C(C(=O)OC)C)C1CC1 CCC(C)CC(=O)NOC(CC(C)C)C(=O)NCC(C)(COC)CO N1(C(C(C)N(C(C)=O)C)=O)CCC(=CCNC(c2coc(Br)c2)=O)CC1 CN1CC(C(N2CCC(CO)C(NC(=O)C(F)CC3CCOC3)C2)=O)CCC1=O C#CC1(NC(C2(CNC(=O)CN3CCCC3C)CC23CCC3)=O)CCOC1 C(=O)(CCC(F)(F)Cn1cc(CN2CCCC2CO)nn1)N(C(C=C)C)C Cc1c(C(=O)NC2CC3CN(C(=O)CC(C)c4ccncc4)CC23)cncc1Cl N1(C(c2c(C#N)ccs2)=O)CCC2(CC1)CC(NC(=O)CSCC(N)=O)CO2 Cc1cc(Br)cc(C)c1C(N1CC2CN(C(C3CCC(C)O3)=O)C2C1)=O CC1CCCC=C1C(=O)NCC1CC1NC(c1ccc(O)c(F)c1)=O C1(NC(C(=O)OCC)=O)CN(C(c2ccc(F)cc2Cl)=O)CC1C#N c1(C(=O)NC(CC(C)=O)(C)C)ccc(Cl)cc1SC(C1C(C)C1C)=O C1(CC(=O)NCC2CCC=CC2)CN(C(=O)CSc2nc[nH]n2)CCC1C C(=O)(C(C(C)(C)C)c1ccc(C)cc1)N1C(C2(O)CN(C(C(CC)O)=O)C2)CCC1 c1(C(C)C(=O)NCC2CCC2NC(=O)CS)cccc(Cl)c1.C1CC1.C C1(OCCC)CCCN(C(=O)C(C)(C)NC(=O)C(C)COC(C)=O)C1 c1(CC(N2CC(C)N(C(=O)CO)CC2)=O)cccc([N+](=O)[O-])c1.C1(F)CC1.C C1(CCC(=O)NCCC(C)NC(C2(C(=O)NC)CCC2)=O)CCCCO1 C1(C(=O)NC2(C)CN(C(=O)OC)C2)C2CN(C(C3SCC=C3C)=O)CC12 C1(OC)CCCC(C)(C)C1CN=c1ccnc(-c2ccccc2)[nH]1 N1(C(Cc2n(C)ccc2)=O)C2CCC1CC(NC(=O)CCC(N)=O)C2 C#Cc1cc(C(=O)NC2CC(NC(C3CC4CCC3CC4)=O)C(O)C2)ccc1Cl C1(CNC(CCCc2ccc(C)s2)=O)CN(C(c2cccc(=O)o2)=O)C2CC12 C#CCC(C)(C(=O)N(C1CCCCCC1O)C)NC(=O)Cn1cc(CO)nn1 C1N=C2NC(=NCC13CC3)Nc1ccsc12.CC1Cc2ccccc2C1CNO CC1CCC(CNC(C2(CCF)CC2)=O)N(C(=O)CC2CCCCC2)C1 C1(NC(C2CC23CCSCC3)=O)CCN(C(C2CCC2)=O)C12CC2 C1(C)(C=O)CCCC(F)(F)C1.c1(CC(C)C)nc(C(=O)NC(C)CC)cs1.N C=CC1OCCCC1C(N1CC=C(CNC(C2(C)CC(C)=NO2)=O)CC1)=O CCS(=O)(=O)CC(=O)NC(CC1CC1)CC(=O)N1CC(N2CC(O)C2)C1 C1(CC)CCN(C(C2CCN(C)S2(=O)=O)=O)CC1.N1(CC=O)CC2CCC1C2.N N1(C(CC=CC=C)=O)CCOC2CN(C(=O)CSCc3ccc(Cl)s3)CC12 C1(NC(c2n(C)c(S)nn2)=O)CC2CCC(C1F)N2C(c1ncccc1Cl)=O c12ccc(cc1)N1CCN(CC1)C2=O.Cn1ccc(CN)n1.C(=O)C=CC1CC1 N1(C(CCSC)=O)CCCC(F)(CNC(C2CC(C(F)(F)F)C2)=O)C1 Cc1csc2c(C(N3CCOC(CNC(=O)CC(C)CF)C3)=O)cccc12 N1(CC(C)C)CCC(C(=O)NC(C2CCN(C(c3cn(CCO)nn3)=O)C2)C)C1 C1(CNC(C2OCCN(C)C2)=O)CN(C(c2cnoc2C2CC2)=O)CC1(C)C Cc1n[nH]cc1C=CC(=O)NC(C)CCC.c1(C(=O)N)c(C(C)(C)C)nsc1N C1(CC(=O)N)C2CCC(C2)N1C(C1(Cl)CC1(F)F)=O.C1CC2(C1)CC2(F)F C(=O)(C1=C(Cl)CCC1)N1CCN(CCCNC(C(CC)N2CCCC2=O)=O)CC1 n1(CC)ccc(C(=O)NC2CCC2C(=O)NCC(F)(F)CC2CC2)n1 CC1C(NCC(c2nncn2C)C)CCCN1C(=O)OC(C)(C)C C1(C(N2CCN(C(=O)CNC(C3CC3)=O)CC2)=O)(CC)CCC(O)CC1.C N1(C(CC2C(CC)C2)=O)CC(C)(C(=O)NCc2c[nH]nc2C(C)C)C1 c1(C(N2C(CNC(=O)CCc3cccnc3Cl)CC2)=O)ccnc(CC2CC2)n1 N1(C(c2sc(CC)c(C)c2)=O)CC(C)C(C)(CNC(c2cc(Cl)ccn2)=O)C1 Cc1cc(=NC(=O)C(=O)N2CC(NC(c3ccc(C)s3)=O)CC(C)C2)[nH]o1 C(CCCCCC(=O)N1CC(NC(c2ncc(F)cn2)=O)CC(C)C1)SC Cc1cc(O)cc(=O)n1CCC(=O)NCC1CN(C(=O)CCC(N)=O)CC1C c1(C(=O)NC2C(NC(c3n(CCC)ncc3)=O)COC2)cnn2c(C)ccnc12 c1(NC(C(=O)NC(CC)Cn2cncn2)=O)ccccc1C=CC(F)(F)F N1(C(CC=C=C)=O)CCC=C(C(=O)NCC2(C=C)CCC2)C1 n1(CC)cnc2c(NCCC3CC3)nc(Cl)nc12.C(C1CCOCC1)=CC=O.N C(C(C)(O)C(C)CC)NC(C1CC(CNC(C(CC)C#N)=O)OC1)=O C12(C(N(CCCNC(C3(F)CCC3)=O)C)=O)CCC(CC1)CO2 C1(NC(Cc2cc(OC)cc(OC)c2)=O)CN(C(=O)CCSC)C2(CCC2)C1 C1(NC(C=COCC)=O)CN(C(c2cc(C)n(CC)c2C)=O)CC2(CC2)C1 N1(C(CCOC)=O)CCCC1C(C)NC(=O)C(C)(C)c1cncs1 C(=O)(C(CC)NC(C1CCCCC1)C(=O)OC)OCC c1(C(=O)Nc2nnc(C3CC3)s2)c[nH]c2cc(Cl)ccc12 C12(CNC(C3CCC(CCCC)CC3)=O)CC(C1)C(C=O)CO2.c1ccc[nH]1.N n1(CC(N2CC(C)C2)=O)ncc(=O)c2ccccc12.C(C)(C=O)N(C(C)=O)C.N N1(S(CC)(=O)=O)CC2COCC2(C(=O)N(CC(=O)OC)C)C1 C1(C(N2CC3CCC3C2)=O)CCc2nc(C)cn2C1.C1(CC#C)(C(=O)N)CC1.C c1(N(CCOCCN(C)C(C2CC=CCO2)=O)C)ncnc(O)c1Br C12(C=O)CC(C1)S(=O)(=O)C2.Cc1nc(CCC(=O)NCCC(C)CC)oc1C.N N1(C(CC(=C)C)=O)CCCC2(CCN(C(c3cc(C4CC4)on3)=O)C2)C1 n1(CCCC)nc(C(=O)N(CC(C)(C)C)C(C)C)ccc1=O C1(CC(=O)NCCOCC)CCCN(C(C2CCC(=O)N2C)=O)C1 N1(C(N(CC(F)(F)F)C)=O)CCCCC1C(=O)OC(C)(C)C C(c1csnc1C)=CC(=O)N(CC(CC)NC(=O)Cc1cn(C)nc1C)C CC1Cn2nc(C(=O)NCC(C(C)(C)C)NC(C3CC3(F)F)=O)cc2C(=O)N1 C1(NC(C(c2ccco2)NC(CC(C(C)C)O)=O)=O)C2CCC3C(C2)CC13 C(CCC(C)CC(=O)NCCC1(O)CN(C(=O)Cc2ccoc2C)C1)=C(C)C N1(C(Cc2n(C)nc(C3CC3)c2)=O)CCC(NC(C2CCOC2)=O)C(C)(C)C1 N#Cc1ccc2cc(C(N3CCCC(C4CCCCC4)C3)=O)ccc2c1 C1(OC)CC(N=c2nc3sccc3c(N3CC(C)=CC(C)C3)[nH]2)CC1OC C1(NC(c2scc(C)c2C)=O)CCCN2CCSCC12 c1(C(N(CC(=C)C)CC)=O)ccccc1CN1CCCC1=O N1(C(CCn2c(C)nc(C)n2)=O)CCN(C(=O)C(O)CC(F)F)CC1C(C)C N1(C(C(CC)(C)C#N)=O)C2CCCC1CC(NC(c1cc(C(F)(F)F)c[nH]1)=O)C2 C1(C(c2nnnn2C)Nc2ccc(Br)cc2CCO)(OC)CCOC(C)(C)C1 c1(NC(C2CCN2C(=O)C(F)(F)Cl)=O)ccc(Br)c(Cl)c1Cl c1(Cn2c(C)c(C(=O)Oc3cccc(Br)c3)nn2)cccc(F)c1F n1(CCOC(C2(C)CC2C)=O)cnnc1.CC1=CC(=O)NCCOC1 N1(C(C2(C)CCC2)=O)CC(NC(c2cccc(C(F)(F)F)c2F)=O)C(F)(F)C1 C1(CNC(NCC(CC)OC)=NCCCN2CCOCC2)CC2(CO1)CC(F)(F)C2 N1(C(c2ccncc2Cl)C(=O)NCC2CCOC2)CC(C2CC2)C1C1CC1 Cc1cc(C(=O)NC(C)(C)C(C)NC(=O)CC23CCCC2C3)c(C)n1C C1(NC(CCCOC(C)C)=O)CC2(CCCN(C(c3cc(=N)[nH]c(=N)[nH]3)=O)C2)C1 CCCC(O)CC(=O)NC1CCN(C(=O)C(CCCO)c2ccccc2)C1C CCCCCC(C)(CC)C(=O)NCC1CC2(C1)CN(C(c1cnccc1Cl)=O)C2 C1(NC(=O)C=Cc2ccc(C(F)F)o2)CCSC12CN(C(=O)CC1CCC1)C2 C1(CNC(C2CCC=CCC2)=O)CN(C(=O)CN2CCOC2=O)C2CCCC2O1 C(=O)(CC(C)C(F)F)NC1CC(CNC(c2nc(CC)oc2)=O)C(O)C1 c1(NC(C2CC3CCC2N3C(c2ncon2)=O)=O)cc(F)cc(F)c1F N1(C(C(C(C)C)OC)=O)CC2CN(C(c3snc(C)c3Br)=O)CC2(C)C1 C1(CN(C)C(C2CCSC2)=O)C2CN(C(c3ccsc3C#N)=O)CC12 N1(C(CSc2c(C)cccc2)=O)CC2CN(C(=O)Cc3ncccn3)C2C1 N1(C(C(C)=C2CCC2)=O)CCOCC(C(=O)N(C)CC2CN(C)C2)C1 N1(C(C(CC=C)C)=O)CCCC(F)(CNC(=O)CCS(N)(=O)=O)C1 c1(C(=O)NCCC2(NC(C(C)OCC=C)=O)CCC2)cccc2c1ncn2C n1(CCC)nc(C)c(C(=O)NCC(C)CO)c1C.C1(C=O)CCN(C)C(=O)C1.N C1(C(N(C)Cc2cccc(F)c2)=O)CC1C1CN(C(C2CC(SC)C2)=O)C1 N1(C(=O)C#CC2CC2)CCOCC2(COCCN2C(c2cc(C(F)F)[nH]n2)=O)C1 N1(CC(=O)N(CCCNC(C=C(CCC)C)=O)C)CC2CC2C1 N1(C(C2(C#C)CCN(C(c3ccnc(C)c3)=O)C2)=O)CCCOC(C)(C)C1 N1(C(C2CCC(CC)C2)=O)CCC2(CC1)CCC2.c1(C(=O)N)cnnn1C1CC1 N1(C(C2(C)N(C)CCC2)=O)CC2CCCC(NC(=O)Cc3cnoc3)(C2)C1 Cc1nn(C)c(C)c1CN1CCC(NS(=O)(=O)CC#N)C(O)C1 CC12CCC1CN(C(=O)Cn1nc(C(C)(C)C)cc1N)C2 c1(C(C)C)cccc(C(N2CCOCC2CNC(c2cnn(C)n2)=O)=O)c1 Cc1ncccc1CC(=O)NC(C)CCC(=O)N(C)Cc1cccnn1 c1(OC)cccc(C(=O)NCc2cc(-c3ccccc3)n[nH]2)c1N C(CC(C)(C)C(=O)N1CCC(C(=O)NC(C)CC(C)O)CC1)SC C(CC(C(=O)N=c1ccn(CCCO)[nH]1)NC(c1n[nH]c2c1COC2)=O)=CC Cc1c(Cl)ccnc1C(=O)NC1CC(NC(C2CCCCC2C(C)(C)C)=O)C1 c1(CC)ccncc1NC(C1CCC(C(C)C)N1C(C1CC2CC2C1)=O)=O c1(C(N(CCC)C)=O)ccc(F)c(C(F)(F)F)c1F.c1(SC)ocnc1C=O.N C1(Cc2cn(Cc3nc(C)sc3)nn2)CN(C(=O)C(F)(F)CO)CCO1 N1(C(C2(CCC=C)CC2)=O)CCOC2CN(C(=O)C=Cc3ccccc3)CC12 n1(CC)nnc(C(=O)NCC2(OC)CN(C(=O)C(F)C3CCC3)C2)c1C c1(OC)nscc1NC(=O)C(c1cccnc1)NC(c1cccs1)=O CC1CC(CN)CN1CC1CCC(F)(F)C1 CC1CN(C(C2OCC3CCCC23)=O)CCC1CNC(C1CSC1)=O c1(CNC(c2occ(C)c2)=O)nn(C)c2c1CN(C(c1nncn1C)=O)CC2 C1CCCN(C)C1.c1(CNC(C2(COC)CC2)=O)csc(C(=O)NC)c1 c1(C(=O)NCC(C)(CO)NC(C2CCc3ncnn3C2)=O)cc2ccncc2s1 C1(F)(CNC(c2c(CC)ocn2)=O)COCCN(C(=O)C(C)COC)C1 C1(C)(NC(C(C)c2ccsn2)=O)CC(NC(c2cn[nH]c2)=O)C1 C1(C(=O)NC2(CO)CCCN(C(c3ccccc3F)=O)C2)CC2(C1)CC21CCC1 C1(NC)CN(CC2(C)CCCOC2)CC12CC2 C1(O)(C(=O)NC(C(C)NC(C(c2cnn(C)c2)OC)=O)CO)CCCCC1 C12(NC(=O)CCN3CCCC3)CCCN(C(C3(c4ccc(Cl)cc4)CC3)=O)CC1C2 C(C(C)C(F)C(=O)N(OC)C(C)CC)NC(CCC=CCC=C)=O C1(C(N2CCC(O)(CN(C(=O)CCn3ccnc3)C)C2)=O)COCCC1(F)F c1(NCC(C)NC(c2ccc(Cl)nn2)=O)nc2c(cc1Cl)C(=O)OC2 C(CNC(=O)CCc1c(C)n[nH]c1C)(C(C)(C)C)NC(CSCC=C)=O c1(C(=O)NC)ccc(C(=O)NC2CCC(CC)C2)cn1.c1(C=O)csc(Cl)n1 N1(C(C2CCCN(C(C=CC=CCC)=O)C2)=O)CCC(COC)C(C)C1 C(=O)(C1=NOC(C)(C)C1)NC1(C)C(C(=O)NC(C)(C)CF)CCCC1 CC1N=C2NC(=NC3CN(C3)C(=O)NC1C)NC1=C2CCCC1.C(C)(C)(C)OC CC1(CC(=O)NC2(CO)CN(C(c3cccc(F)n3)=O)C2)CCS(=O)(=O)N1 Cc1cc(C(=O)N(CC=O)CC2COC(C)(C)C2)ccc1[N+](=O)[O-].C(C)(C)C c1(C(N2CCN(C(c3c[nH]c(Br)c3)=O)C3CC23)=O)nncc2ccccc12 C1(C(=O)NCCC(=C)CNC(=O)C(C)=CC)CCCC(O)C1 N1(C(c2c(CC)nc[nH]2)=O)CCCC(CCNC(C2CCC(C)(C)CC2)=O)CC1 C1(C(=O)OC)CC12CC(S(=O)(=O)N1CCNC(=O)C1c1ccccc1F)C2 C(C(=O)NC)(C(C)C)NC(c1ccc(CC)cc1)c1nnnn1CC c1(OC)cccc(CC(=O)NC2(CNC(c3cc(C)nn3C)=O)CCOCC2)c1 Cc1nc(C(=O)NCCO)c2ccnc-2[nH]1.C(=O)CS(C)(=O)=O.C(C)(C)C N1(C(c2c(C)ocn2)=O)CC2C(CNC(C3CCC(C)(C)C3)=O)C2C1 N1(C(CCOC)=O)CCCC1C1CCCN1C(c1cnn(C)c1)=O C(=O)(C1CC(C)Cc2c[nH]nc21)NCCC(C)(C)NC(C=C(COC)C)=O C1(OC)CCCC(C(=O)N(C2CC(NC(=O)Cc3cc(C)no3)C2)C)C1 c1(C(N(C2CC(NC(=O)COc3ccc(O)cc3)C2)C)=O)cccc(O)n1 c1(C(=O)NC(CC(C)NC(c2csc(Br)n2)=O)C)n[nH]c2c1NCCC2 O=C(C(O)CCCc1ccccc1)NCCN(C1CCCCC1)C(C1CC(O)C1)=O C=C(CC)CN=c1nc(N2CCCC(CNS(C)(=O)=O)C2)c2c([nH]1)CCS2 O=C1NCCC1CN.N12CCCC1C1(CC1)C2=O.C12CC(CC(F)F)(C1)C2 CC1(O)CCC(C(=O)NCC2CN(C(C3CCS(=O)(=O)CC3)=O)C2)CC1 C1(C(N)=O)(NC(Cc2ccn(C(C)C)n2)=O)C2CC3CC(C2)CC1C3 C1(NC(C2CCC(=C)CC2)=O)CCCN(C(c2cnc(C)nc2)=O)C1CC N1(C(c2cc(C)nn2C)=O)CCC2C(C1)NC(=O)CCN2C(=O)CC(C)C CS(=O)(=O)CCCC(=O)NC1CC2(C1)CCC2.c1(C=O)ccc(C2CC2)cn1.N C=CCC(C)(C)CCNC(=O)C(C(C)C)NC(c1cnccn1)=O C(C1CCCN1C(c1ccc(CO)cc1)=O)=CC(=O)NCC(c1cccnc1)O C(CNC(=O)CC(C1CCC1)C1CCC1)(C(C)C)NC(CCOCC)=O n1(C(C)C)ccc(C(N2CCC(CO)C(NC(c3cc(O)cs3)=O)C2)=O)cc1=O c1(NCC(N2CCCC2C2(CNC(=O)CO)CC2)=O)cncnc1 C1(CNC(CCC)=O)CCN(C(c2cc(C#N)ccc2C)=O)C12CCC2 C1(CC#C)(C(=O)NC2CCC(CNC(C3(C)CC=CC3)=O)C2)CCCO1 C1(C=O)CSCN1C(N)=O.c1(CC(=O)N(C)CC)cnco1.C(C)(C)C.N N12CCCC(C1)CN(C)CCS2(=O)=O.C(=O)(CCCCc1ccccc1O)OC S(=O)(=O)(c1ccc(NCCCc2ccc(F)cc2)c(Cl)c1)N1CC(C)C(C)CC1 c1(C(=O)NCC2C3CN(C(c4cc(C)cc(C)c4)=O)CC32)ccc2ccoc2c1 C1CN(C(=O)C=C(C)c2ccco2)CCC1C(F)(F)F.C(C)(C)(CC=O)OC C(=O)(C(O)C(F)(F)F)N(CC(C)O)CCNC(c1nonc1N)=O c1(OC)cccc(C(N2CCOC(N(c3ccccc3)C(C)=O)C2)=O)c1C CC(=O)CCCC(=O)NCC1CCN(C(c2ncncc2Br)=O)CC1 c1(CN(C2CCCSC2)C)cn(CC(=O)N(C)C)nn1.C12CC(C1)C(=O)N2 CC1c2c[nH]nc2CCC1NC(=O)N(C)Cc1cc2ccccc2n1C Cc1ncc(Cl)c(C(N2CCCN(C(=O)CCCC(C)C)CC2)=O)n1 C(=O)(CC1=CCCCC1)N1C(CNC(C(CSC)OC)=O)C(C)CC1 C(CNC(=O)CC1CCC(C)CC1)(CC(=O)NC1CCOCC1F)OC N1(C(C2(CS(N)(=O)=O)COC2)=O)C2CCC1CNC2.C1CC(C(F)(F)F)C1.C N1(C(c2cnc(CC)[nH]2)=O)CCC(NC(=O)C(=C2CCCCC2)F)CC1C CCC(C(=O)OC)C(=O)N(C)CC1CCCC1NC(C1(F)CCC1)=O N1(CC=O)C(=O)CC(C)(C)C1=O.N1(C(CC)=O)CCCC1CC.CCCCS N1(CC(C)O)CCN(C(c2c[nH]c(C(C)(C)C)n2)=O)CC1 N1(C(CCCOC)=O)CCCC(CCNC(=O)C(c2ccccc2)O)C1 C(=O)C1=C(C)CCC1.c1(COC)nc(CNC(c2[nH]ccc2C)=O)no1 C1(CC(=O)NC(C2CCOC2)C)CCCN(C(=O)CCC2CC(F)(F)C2)CC1 c1(C(=O)OC2C3CN(C(CC)C)CC32)c([N+](=O)[O-])cnn1CC.c1cccc(C)c1 c1(OC(C)C)ccc(C=O)cn1.c1(C(N2CC(O)C2)=O)c[nH]c(C(N)=O)c1.N C1(NC(COCc2nnc(C)s2)=O)CC2CN(C(=O)CN(C)CCO)CC12 Cc1cc(NC(=O)C(F)n2cccn2)ccc1NC(=O)C(C)N1CCC1 C1(NC(CN(CC(C)(C)C)C)=O)CS(=O)(=O)CC1.C1(C=O)CC(O)C1.N N1(C(C(CC2CC2)OC)=O)CCCC(C(=O)NCCC2CCCC3CC23)C1 CC(C)CS(=O)(=O)CC(=O)N.c1(C(N2CC(O)C2)=O)ccn(C)c1CC(=O)O C1(C)(C=O)CCN(C)C1.c1(C(N(CC)Cc2ccccn2)=O)cccnc1.C N1(C(C(C)S(=O)(=O)Cc2ccccc2)=O)CCN2CCOCC2(CO)C1 N1(C(c2cc(C)ncc2C)=O)CC2CCN(C(C3CC3C#N)=O)C2C1 N1(C(C(C)CN)=O)CC(NC(c2nccn2C)=O)C2(COC2)C1 N1(C(c2ccc(CC)[nH]2)=O)CCCC1(C)CNC(=O)CC1CCC(=O)NC1 C12(C(N3C(CCNC(CC4C(C)(C)C4(C)C)=O)CCC3)=O)CC1COC2(C)C CCCC(CC)NC(C1(NC(=O)C(O)CN2CCCC2)CSC1)=O c1(COC2CCN(C(C3CC3Br)=O)C2)ccc(Br)cc1 Cc1sc(Cl)nc1C(=O)NCC1CCN1C(c1cc(C(F)F)[nH]n1)=O C1(NC(C(F)=CC)=O)CCCC12CCN(C(=O)CN(CC=O)C)C2.C(C)C N1(C(c2c(C)scn2)=O)CCC2(CCN(C(=O)C(CO)C(C)(C)C)C2)C1 Cc1nc(C(F)(F)F)c(C(=O)NC(C)CNC(C2CCC(=O)C2)=O)o1 N1(C(C2(SCC)CC2)=O)CC2(C1)CN(C(=O)CC1CCCCC1F)CCO2 C1(NC(c2coc(O)n2)=O)CN(C(=O)Cc2cccnc2)C2(CCCCC2)C1 Cc1ccc(C(N2CC(C(C)NC(=O)CCO)C2)=O)cc1C1CC1.CC(C)C CC1CC(CCNC(c2cnc3n2CCC3)=O)CCN1C(=O)CSC(F)F C(=O)(C#CC1(C)CCCO1)NCc1c(C(=O)NCCC(CCC)O)con1 c1(C2CC(NC(c3n(C)nnn3)C(C)(C)c3ccccc3)C2)ccc(N)cc1 CC(C)(C)CC(O)C(=O)NC1CCCN(C(c2ncc(F)cn2)=O)C1 c1(C(N(CC(C)N(C(c2nc(C)oc2)=O)C)C)=O)cnn2c(C)c(C)ccc12 c1(C(N2C(c3cn(CCCN(C)C)nn3)CCC2)=O)ccc2c[nH]nc2n1 c1(NC(N2CCC3(CCN(C)C3)C2)=O)cc(Cl)ccc1S(C)(=O)=O C1(OC)CC2CCC(C1)N2C(=O)CC12CCC1CN(C(C1(Cl)CC1)=O)C2 N1(CC=O)CCS(=O)CC1.c1(CN(C)C)ccc(C(=O)N)o1.CCC1CC1 N1(C(C2CC3N(C(C(CC(=O)OC)C)=O)C(CC3)C2)=O)CC=CC12CCOCC2 c1(-c2cn(C)nc2)cncc(NC(=O)CC(C2CCCCCC2)N)c1 C1(NC(c2c(C(C)C)ocn2)=O)CCCC(NC(=O)Cc2cccnc2)CC1 c1(CC(=O)NC(C(=O)OC)C(C)=O)ccc2nn(C)cc2c1 C1(NC(CCCOCC)=O)CC(C(=O)NOCC(C)(C)O)CC1O C1(CC=O)CCCCN1C(=O)CC1CC(=O)NC1=O.C(C)(C)(C1CC1)OC C(C(=O)N(C(C)C(C)C)C)(C1CN(C(c2cc[nH]n2)=O)C1)OC N1(C(=O)C(F)F)CC(NC(C2(c3cccnc3)CCCCC2)=O)C(O)C1 C1(CC(=O)N(CC(CC)C)CC)N(C(c2cccn2C)=O)CCC1(C)C N1(C(C2CCN(CC)C2)=O)CCN(C(C2CCCNS2(=O)=O)=O)CC1C C(CC(CNC(=O)C(F)OC(F)(F)F)NC(=O)C(O)c1ccco1)OC C(C)(CNC(C1C=CCC1)=O)(C1CC1)NC(CN(C)C1CC1)=O Cc1cc(C=CC(=O)NCC2CCCN(C(C3CC3F)=O)C2)ccc1F N1(C(CC2(CC(=O)OC)CC2)=O)CCCC(F)(F)C1.C(=O)C(F)(F)C(C)O n1(CCC)ncc(C(=O)N(CCC(C)NC(c2cnn(C)c2CC)=O)C)c1C C#CCCCC(C)C(=O)N1CCCCCC(NC(=O)CCOC(C)C)C1 Cn1c(=O)c2cc(C(=O)NCCNC(c3cccc(F)c3)=O)sc2n(C)c1=O C=CCN=C(NCCc1nc(-c2ccccc2)no1)N1CCC(n2cccn2)C1 c1(C(=O)NCCC(C)N(C(C2CC(OC)C2)=O)C)ccnc2ccccc12 N#CC1C2CC2CN1C(C1CC1C(=O)NCCO)=O.c1(C)ccccc1 CCCC(C)CC(=O)N1CCCC1C(C)NC(c1ccnc(CC(C)C)n1)=O c1(C(=O)NCC(CNC(c2n(CC)cc(Cl)c2)=O)C)cc2c([nH]1)CCC2 Cc1ccc(F)c(C(N2CC3CC2C3NC(c2ccc([N+](=O)[O-])n2C)=O)=O)c1F C(CC(C)(C)C)(C(=O)NC1(C2CCCCO2)CC1)N(C)C.c1cc(C(=O)O)n[nH]1 C#CCC(C(=O)N(C(C)C(C)SC)C)NC(c1cnncc1NC)=O Cc1cc(C(N2CCC(CNC(=O)CCC(N)=O)CC2C)=O)cc([N+](=O)[O-])c1Cl N1(C(c2cccc(C(C)C)n2)=O)CCC2(CCN(C(=O)CCF)C2)C1 C1(C(=O)NCCN(C2CCCC2)C)CCCC1NC(c1csnc1Cl)=O c1(OC)c(CNC(c2cnn(C)c2)=O)ccc2[nH]ccc12 c1(N2CCOCC(=C)C2)nc(N2CCSC(C)CC2)nc2c1CCCCCC2 n1(CC)nncc1C(=O)NC(C(=O)N(C(CO)C(C)C)C)C1(O)CCC1 C1(S(C)(=O)=O)(C(N2CCC(C#C)(O)C2)=O)CC(O)C1 c1(NC)ccc(Cl)c(C(=O)NC23CCN(C(=O)CO)CC2C3)c1.c1cccnc1 n1(CC(=O)N(CCCNC(C2(CF)CC2)=O)CC)ncc(O)nc1=O c1(C(N2CCCC(CNC(C34CCCC3OCC4)=O)CC2)=O)cc(O)cc(=O)o1 C(=O)(C(=O)N=S(C)(C)=O)NC1CCCN(C(=O)CN(C)S(N)(=O)=O)C1 C1(CNC(c2n(CC=C)ccn2)=O)CC(F)CN1C(c1cn[nH]c1)=O N(C1CCc2ccc(F)cc21)c1c(C)c(NCCCN2CCCC2)ncn1 CC1CC1CC(=O)NCC(C1CC1)NC(C1(NC(N)=O)CC1)=O C=C(C)CC(C(=O)N1CC(C(C)O)C1)NC(c1cc(OC)n[nH]1)=O N1(C(c2ccnn2CCF)=O)CCCCC1C1CCN(c2nnc(C3CC3)s2)C1 Cc1nn(C)c2c(NCc3ccoc3)nc(N3CCC(SC(F)(F)F)CC3)nc12 c1(CNC(=O)CC2CC2)ccc(C(N2CCC(C(F)F)C2)=O)nc1 c1(C(=O)NCCNCCO)cccc(-c2ncsc2C(N2CCOCC2)=O)c1 c1(CC)conc1C(c1nnnn1C1CCC1)NCc1cc(OC)no1 CC1CN(C(C2CNC(=O)CN2C(C2CC(=C3CCC3)C2)=O)=O)Cc2c[nH]nc21 CCC(CC)CCCC(=O)NC1CC2CC1N(C(=O)COC1CC1)C2 C1(C)(CC)CCN(C(=O)C(C)NC(=O)CCC2CC2(C)C)CC1 C(N=c1[nH]c2c(c(=NC3CSC3)[nH]1)CSC2)C1(OC)CCCCCCC1 Cc1cc(=O)oc(C)c1C(N1CC(NC(c2sccc2CO)=O)C(O)C1)=O c1(-c2c(C)ncs2)cncc(CN2CCC(CC(=O)O)C2)c1 Cc1ccc(Cl)nc1NC(c1cc(C(C2CCNCC2)(C)C)on1)=O O=C1OCCC1CC(=O)NCCOCC(N1CC(F)(F)C1)=O C1(C(=O)N)CCCC(=O)N1C.CC(C)C(C)CNC(C1(c2nccs2)CC1)=O N1(C(C)C)CC(CNC(c2cc(Br)ccn2)c2nnnn2CC(F)F)CC1=O c1(C(=O)NC2CN(C(CSc3nc(C)[nH]n3)=O)C(C)CC2)ccc(O)c(F)c1F n1(CC)nc(C=O)cc1C.C1(CC)CN(C(=O)C=CCN2CCCC2)CCO1.N c1(C(N(C(=O)CN2CCCN(CCC(=O)O)CC2)C)=O)cccc2c[nH]nc12 c1(C(=O)NCC(CCC)CCO)n[nH]c2c1CN(C(=O)C(C)S(N)(=O)=O)C2 CON1CC(C(N2CCC(O)C(NC(c3ccon3)=O)C2)=O)CC1=O Cc1cc(NC(C2(C)CN(C(c3cnc(C)c(C)c3)=O)C2)=O)ccc1Cl c1(C(N2CCC(C3CCCN3C(c3nncs3)=O)C2)=O)noc2ncccc12 CCC(CCC(=O)NC1CC(NC(=O)COC2CC2)C(O)C1)OC N1(C(c2[nH]cc(CC)c2)=O)CCC(O)C1.c1(C(NC)=O)ccn(CC(F)F)n1.C c1(C(=O)NC(CC(=O)NC(c2ncc(C)[nH]2)CC)C2CC2)ccc(C)cc1C C1(C(=O)N)CCCC(F)(F)C1.c1(CN(C)C)ccsc1C(=O)NCC(C)CO c1(-c2cc(C(=O)NCC(CNC(C3CCC(=O)C3)=O)O)on2)cccc(Cl)c1F c1(OC)c(C(=O)Nc2ccc(Cl)c(N3CCNC3=O)c2)ccc(F)c1F C12(C(=O)NCCNC(C(N3CCC(C)CC3)C(C)C)=O)CCOC1CC(=O)NC2 C1(CCCC)CCC(N=c2cc[nH]cc2S(=O)(=O)NC(c2cc(C)sc2C)C)C1 c1(C=O)sccc1C(C)(C)C.C(C=O)=CC.CCC1CC1.C(C)OC.O CC1CCCCC1(C)NC(=O)NC(CCC(F)(F)F)c1cccnc1 c1(C(=O)NCC(C)(O)C)cc(F)c(F)cc1Cl.C1(C=O)CCC1C(F)(F)F C1(NC(CC(C)(C)NC(=O)CC23CCCC2C3)=O)CCCN2CCCC12 c1(CC(N2CCCC(CCNC(C(CC)(C)O)=O)C2)=O)cccc(C)c1F CN1CCC(C)(C(=O)NC2CCC3CC3C2)CC1 C12(C(=O)Nc3ccc(OCC)nc3)CCN(C(=O)CC(C)(C)C)CCC1C2 C1(S(C)(=O)=O)(C(N2CCCCC2)=O)CC(O)C1.[nH]1cc(C(=O)NC)nn1.CC C1(CC)C(C(=O)NCC2CSC2)CCN1C(c1ccn(C(F)F)n1)=O c1(CCC(=O)N(CCCCNC(C(C)SC(F)(F)F)=O)C)ccn(C)c1 C=C1CC2(C1)CC(C(=O)NCC(C)NC(=O)C(O)Cn1cncn1)C2 CP(C)(=O)C(O)C(=O)NCC(C1CC1)NC(c1cc[nH]c1C1CCCC1)=O C(=O)(C(F)(CNC(=O)CC1CC2CC2C1)C(C)C)N(C)Cc1c(C)nsc1 CC1CC2CN(C(C3(C)CC(O)CN3C(C3CC(N(C)C)C3)=O)=O)CC12 C12(C(N(C3CN(C(C4C(C)C4c4ccccc4)=O)C3)C)=O)CCCC1C2(F)F c1(OC)cc(CN(CC(O)CN(C(=O)Cc2cscc2Br)C)C)on1 C1(C2CC2)CCN(C(c2cccnc2C2CC2)=O)C1.C1(C(=O)NC)C=CCC1 c1(C(N2CCC(C)(OC)CC2)C(=O)NC)cnc(OC)cc1OC c1(OC)cc(CC(=O)N(CCC)C)cc(Cl)c1.C(=O)(C(C)(C)c1ccn(C)n1)N CC1CN(C(=O)CN2CCC(CO)CC2)CCCN1C(=O)C(F)n1cccn1 C1(NC(c2nn(C)c(C#N)c2)=O)CC2(CCN(C(=O)CCC3CC3)C2)C1 N1(C(C=C(C)Cl)=O)CCC2(CC1)CN(C(=O)COCCCF)CC(C)O2 CC1=NOC(C)(C(=O)NC(CNC(=O)CS(=O)(=O)N(C)C)CC(C)C)C1 C(O)(CC(=O)NCC(C)NC(=O)CCc1ccon1)(C(F)(F)F)c1ccc(C)o1 Cc1ncccc1CC(N1CCC(NS(=O)(=O)C2CC2)CC1)=O N1(C(CC(=O)OCC)=O)CCC(NC(c2n[nH]cc2C)=O)C1c1ccccc1 c1(CCCSC)cn(CC2(C)CC2)nn1.C1(C(=O)N)CCN1C(C)(C)C C(=O)(C1=NOC(C)C1)N1C(CNC(CCSCC)=O)COCC1 N1(C(C(c2ccc(C)o2)C)=O)CC2C(CNC(C3CCC3C#N)=O)C2C1 N1(C(c2n(C)ccn2)=O)CC2C(CNC(=O)CCC3CCCO3)C2C1 C1(C(=O)N(c2ccc(C)cc2)c2ccnn2C(C)C)C(C)OCC12CCNCC2 c1(OC)cc(-c2nc(C(=O)Nc3cc(OC)nc(F)c3)cs2)ccc1OC(F)F Cc1ccc(CC(=O)NCC2CCC2NC(C2CNC(=O)N2)=O)s1 N1(C(c2cnnn2C2CC2)=O)CCN(C(C2CCO2)=O)C2CS(=O)(=O)CC12 C1(NC(=O)CCc2nc(C3CC3)no2)CC12CCN(C(=O)C=CCO)CC2 N1(C(CCC)C)CC(C(N2CC(C(C)NC(=O)CC)C2)=O)CC1=O N1(CC)CCOC(CNC(c2cccc(CNC(C)=O)c2)=O)C1 c1(CC(=O)OC)cn(CC(F)(F)CNC(=O)CCC2CC2(F)F)nn1 CC1CCC(O)(C(=O)N(C2CCN(C(=O)C(C)(C)CC#N)C2)CC2CC2)CC1 c1(C(N2C(CC(=O)NC(C3(C(C)(F)F)CC3)=O)CC2)=O)cc(Cl)cs1 Cc1c(C(=O)NC(C)(CO)C(=O)NC2CCC3(CC3)C2)nnn1C CC1CC(C(=O)N(C)Cc2ccncn2)CN(C(c2ccc(C#N)cc2)=O)C1 C1(NC(=O)CP(C)(C)=O)CCCCC12CCN(C(=O)CCc1ccsc1)C2 C1(NC(C2(N(C(=O)CC3COCC3O)C)CC2)=O)CCCC(O)C1 CCCCC(C)(F)C(=O)N(C)CCO.C1(C(N(CC)C)=O)CC1(C)C(F)(F)F c1(NC(C2(NC(=O)Cn3nccn3)C(C)(C)C2)=O)ccccc1CCO Cn1nc(CN2C(C(N3CC4COCC4C3)=O)CC3CC23)c2ccccc12 N1(C(CNS(C)(=O)=O)=O)CCCC(O)(C)C1.C(c1ccncc1)=CC(=O)N C(N=c1nc[nH]cc1C#N)C1CN(C(c2ccc(CSC)o2)=O)C(C)C1 CN1CCN(C(=O)Cc2nc(=N)[nH][nH]2)CC1C(=O)NC1CCNC(=O)C1 C1(F)CCOCC1.N(C(=NC)NC1CC(C(=O)OC(C)(C)C)C1)CCC Cc1cc(F)ncc1C(=O)NCC1C(C)CCCN1C(c1cnncc1O)=O C1(CC(N)=O)(NC(c2c(C)ccs2)=O)CCN(C(c2cc(F)c[nH]2)=O)CC1 C12(NC(c3c(CC)ccs3)=O)CCCC(NC(c3ccoc3Cl)=O)(C1)C2 C1(CC)CN(C(c2ccc(C)cc2SC)=O)CCN1C(c1ccnn1C(C)C)=O C1(NC(c2c(C)cno2)=O)C=CCN(C(C2CC(Cc3ccccc3)C2)=O)C1 CCC(C)C(C(=O)NCC(C)CC(=O)NC1CCC(C)(O)CC1)N(C)C CCCC(C)C(=O)N1CCSC(C(=O)NCc2sccc2Cl)C1 C1(CC)(NC(=O)NC(c2nc(-c3ccncc3)no2)C)CCNC1=O N1(C(C(C)n2cccc2)=O)CCN(C2CN(C(C3CC(=O)N3)=O)C2)CC1 N1(C(Cc2cc(CC)no2)=O)CC2(CCN(C(C3CC3(c3ccccc3)C)=O)C2)C1 C(CCCN=c1[nH]c(=NCc2nncs2)[nH]c2c(F)cc(F)cc12)N(C(C)C)C C1(CNC(c2cccc(C(N)=O)c2)c2n(CCC)nnn2)COC(C)(C)CO1 C(CC(CC)C(=O)NC1COCCN(C(c2ccc[n+]([O-])c2)=O)C1)=CC c1(C(=O)NC(c2cn(CC3CCS(=O)(=O)C3)nn2)C)c(F)ccc2nc[nH]c12 n1(CC=O)ccc(=O)c2ccccc12.CCCCNC(=O)CCOC.C1CC1 c1(CC(N2C(C)CC(NC(c3c(C)nc(O)[nH]3)=O)C2)=O)ccc(O)c(O)c1 C1(C(=O)NCC2CN(C(C(C(C)(C)C)O)=O)C2)CCc2nn[nH]c2C1 Cc1c(C(=O)NCC2CCC2)noc1-c1ccccc1.C1(C=O)C2CCCC12.N c1(CCC(N2CCC(CC)C2)=O)cc(F)ccc1F.C(C(F)(F)F)=CC(=O)N CC1CCCC1(C=O)NC(=O)OC(C)(C)C.C1CCCC(C(F)(F)F)O1.N C1(NC(C(CC#C)(C)C)=O)CC2CCC(C1)N2C(C1CCCCC(C)(C)C1)=O CC1(C)CC(NC(=O)C(N)Cc2ccc([N+](=O)[O-])cc2)CCC1N c1(C(=O)NCCN(C(C2(O)CCCC(C)CC2)=O)C)cc2c(cn1)CCCC2 C1(CNC(C(C)Cc2ccccc2)=O)CCCN(C(=O)CC2CC3(CCC3)C2)C1 Cn1c(N2CCN(CCC(c3ccccc3)NC=O)CC2)nnc1C1CCCC1 O=C(C1=NOC2(CCN(Cc3ccc(C4CC4)cc3)C2)C1)Nc1cncc(F)c1 CC1(C)CN(C(c2ccc(C3CC3)nc2)=O)CCC1NC(C12CCC(C1)OC2)=O c1(CN2CC(c3cnccc3)C2)ccc(C(=O)O)cc1.n12cc(nn1)C2 C1(C(=O)NC2CCC(OC)C2)(NC(=O)C(F)C2CCCC2)CC(F)(F)C1 C1(C(=O)OC)CN(C(C2(CC3(OCC)COC3)CC2)=O)CCS1 c1(C(=O)NC2CN(C(c3n(CC)nc(C(C)C)c3)=O)C2)cc2ccccn2n1 CCCCC(CC)C(=O)NC(C)CCN(C(=O)CCc1ccc(C(N)=O)cc1)C CCCC(O)C(=O)NCC1(O)CN(C(C2CCN(C)CC2)=O)C1 c1(-c2nc(C)[nH]n2)ccc(CNCCN2CC3CC3C2)cc1 C(=O)(C1=CCCCO1)N1CC(CCC)C(C(=O)NCC2CC[Si](C)(C)C2)C1 c1(CCC)nc(C)c(C(=O)NC(CO)C(C)NC(=O)C(F)CC2CCCC2)o1 O=C(CC1COCCN1C(=O)CC1CC2CC2C1)Nn1nnc2c1CCCC2 N1(C(c2ccc(SC)s2)=O)CCN(C(c2csc(C(F)F)n2)=O)C(CO)C1 c1(C(N2CC(O)CCC(NC(C(C)CO)=O)C2)=O)ccc(C2=CCOCC2)cc1 N(C(=NCCF)NCC1(CO)CC12CCOCC2)Cc1c(C)nc(C)s1 c1(C(=O)NC(c2cn(C)cn2)C)cc(CNC(c2nocc2Cl)=O)cs1 C1CN(C(=O)C)CC(C)(C)O1.Cc1nn(C)cc1C(O)C(=O)N.CC(N)=O.C c1(CC(N2CC(O)C(O)C2C)=O)c(F)cccc1F.C(=O)(C(F)(F)C1CC1)N N1(C(c2cn(C)nc2-c2nccs2)=O)CC2(C1)CN(C(C1CS(=O)C1)=O)C2 N1(C(C(C)OC(C)(C)C)=O)CCOC(C)(C)C1.C1(C=O)(N(C)C)CCCC1.C N1(CCC)CCCC(C2CCCCN2C(c2cnn(C)c2CSC)=O)C1 c1(C(=O)NC(CN(C(CC2CC(=C)C2)=O)CC)C)cc(F)c(C)cc1N C1(CC)CCOCCN1C(=O)C(C)=CCNC(C1CCCC(=O)CC1)=O C1(NC(C(C2(C)CC2)NC(CC(C=C)CC)=O)=O)CCN(C)CC1C#N CN1CCN(C(c2scnc2Cl)=O)CC1CNC(c1ccnc(Cl)c1F)=O CC(C)CCCCCC(=O)NC1CC(CNC(=O)CC2CNC(=O)C2)C1 C1(CNC(c2cc(COC)[nH]n2)=O)CCCCC1.c1(C(=O)N)ccc(F)s1 c1(C(=O)NCc2nc(CCC)sc2)c(OC)ccc2cc[nH]c12 C1(NC(c2cnn(CCC)c2Cl)=O)CCC(C)N(C(=O)Cc2cccnc2C)C1 C1(C(N(CC(CCC=C)O)C)=O)CC1C1CN(C(=O)CC(C)CC)C1 c1(CCC(=O)N(C2CCN(C(CC(C=C)C)=O)C2)C)ccc(Br)c(C)c1 C1(CC=C)(NC(c2ccc(CCF)cc2)=O)CCN(C(C2CCCCN2C)=O)C1 CC1CN(C(=O)C(C2(C)CC2)NC(c2cscn2)=O)CCC1O C1(C(N(CC(=O)NCCc2scc(C)n2)C2CCC2)=O)C2CCC(C2)C1C c1(C(=O)OC)csc(-n2cc(C3CC(NC(c4n[nH]cc4Br)=O)C3)nn2)n1 Cc1cccc(C2CCN2C(=O)CCCn2cc(C3CCC(=O)NC3C)nn2)c1Br Cc1cc(C(=O)NCC2CN(C(c3ncsc3C)=O)C3CC23)ccn1 c1(C2(C)CCO2)cccc(C(=O)NC23CC2CN(C(c2cccc(N)c2)=O)C3)c1 C1(C(=O)NCC(C)NC(=O)C(F)=CCCF)CCC(CC2CC2)CC1 N1(C(CN(CCC)C(c2csc(CC)n2)=O)=O)CCCC(C)(O)C1 c1(N2CC(CC)N(Cc3c(F)ccc(Cl)c3F)CC2)[nH]cnc2nc(Br)cc1-2 CC1CC(=O)NC(C(N2CCC(N(C(=O)C=CC3CCCC3)CCO)CC2)=O)C1 Cc1c(CN2CCOC(CNC(=O)CCn3cncn3)C2)ccnc1Cl CCCCC(CC)C(=O)N1CCCC(CC(=O)N(CCCO)CCCO)CC1 C1(NC(c2[nH]cc(C(=O)OC)c2)=O)CCN(C(=O)C(C)=C2CCC2)C(C)C1 N1(C(c2c(C)nsc2)=O)CC2CCN(C(=O)C=C3CCN(C)C3)CC(C2)C1 C1(NC(CCSCC(C)C)=O)CC2CCC1N(C(=O)C(O)CCS(C)=O)C2 N1(C(COC)=O)CC(NC(=O)CCc2c(Cl)cncc2Cl)C(S(C)(=O)=O)C1 CC(C)C(CNC(=O)CN1CCCC1=O)C(=O)N1CC(=O)NCC1C n1(CC)cnc2c(NC3CCSC3)nc(N3CCS(=O)C(C)(C)C3)nc12 Cc1nc2cc(C(N3CCCC3CNC(c3cc[nH]c(=N)c3)=O)=O)cnc2[nH]1 CN(CCCC(=O)NC1CN(C(=O)Cn2cnc(C#N)n2)CC12CC2)N=O c1c(F)cccc1F.C(=O)(C(C)CN(C)C)N(CC(C)NC(=O)C)CC.O N1(CCNC(C2(C)C(C)OCC2)=O)CCCN(C(=O)CN(C)C2CC2)CC1 Cc1ccc(C(N2CCOC(CCNC(C3CC34CCCC4)=O)C2)=O)c(N)c1 N(C1COc2ccccc21)C(=O)CC1CCCN(c2ncc3[nH]ccc3n2)C1 C1(N(C)C(C2CC(O)(C)C2)=O)CC(O)C(O)C1.C(=O)C(C)(C)c1ccno1 C1(C(=O)NCc2ncn(C)c2)C2CN(CC(=O)Nc3ccc(F)cc3)CC12 c1(OC(C(=O)N(C(c2ccc(Cl)cc2)C)CC)C)ccc(Cl)cc1Br c1(CN(C)CC2CCN(C(C(COC)O)=O)C2)c(Cl)cccc1[N+](=O)[O-] c1(OC)cccc(-n2cc(C3CCCCN3C(c3ns[nH]c3=O)=O)nn2)c1 Cc1[nH]nc(C(=O)NC(C)(C)CNC(c2snnc2C(C)C)=O)c1Cl C1(O)(C(N2CC(CC)C(NC(C3CCNC3=O)=O)CC2)=O)CCCC(C)(C)CC1 N1(c2ccnc(S(C)(=O)=O)n2)CCC2C(CCCN2C(c2ccno2)=O)C1 CCC(C)(C)C(C)CC(=O)NC1CN(C(c2c(C)cc(Cl)cc2N)=O)CCC1O c1(C(=O)NC(CNC(=O)CCN2CCCCC2)CO)coc2c(F)cccc12 C1(CNC(COCC)=O)CN(C(=O)Cc2cncc(C)c2)C2CCCCC12 c1(NCC(=C)F)ccc(S(=O)(=O)NCc2noc3c2CCCCC3)cc1Cl C#CCCC(C(=O)N1CC2C(C(N)=O)C2C1)NC(=O)CC1CC(F)C1 c1(CC(=O)NC2CN(C(C3(C=C)CC3)=O)CC2C)coc2cc(C)ccc12 N1(C(c2c(C(=O)OC)cccc2)=O)CC(C)C(C)C1.C(=O)C(C)(O)C(C)C.C C1(NC(CC2C(C=O)C2)=O)CCN(C(=O)Cc2cnc(C)o2)CC1.CC.O C(=O)(C1=Cc2ccc(Cl)cc2OC1)N1CCN(c2cc(C)cc(C)c2)CC1 C1(C(N2CCC(C)(OC)CC2)=O)C2CC(O)C(C2)N1C(=O)C(C)N1CCCC1 c1(C(=O)NCC2CCN(c3nc(C(C)C)cc(C)n3)CC2)[nH]nc([N+](=O)[O-])c1Cl C1(C=O)COC2(C1)CN(C(=O)CN(CCO)CCO)C2.c1ncncc1.CC.O c1(NC2CCN(C(=O)C(F)(F)Oc3ccccc3)C2)ncnc2sccc12 c1(C(=O)NCC(CC)NC(c2cccc3ncoc23)=O)ncnc2c(C)csc12 c1(CC)cccc(C(=O)NC)n1.C1CC(O)CN1C(c1cnc(N(C)C)o1)=O c1(C(=O)NCCC2CC(NC(CC=CCC)=O)C2)cnc2scnc2c1 C12(C(=O)NCC3C(NC(c4c(C)snn4)=O)C3)CCCC(=O)N1CCC2 C(C(=O)NCc1nnn(C)n1)(C(C)CCC=C(C)C)N1CCC(OC)C1 c1(C(=O)NC2C3(CN(C(COCC=C)=O)C3)CC2)c(F)cc(C)cc1Br Cc1nnc2ccc(-c3ccc4c(C(=O)Nc5cnns5)noc4c3)cn12 C1(C)(NC(CC(C)F)=O)CCN(C(C2CCCN2C(=O)OC(C)C)=O)CC1 C(C)(CC(=O)NCCC(C)NC(c1cc(Cl)sc1Cl)=O)OC N1(C(C(C2CC2)NC(CC(C)n2cccn2)=O)=O)CC2CCCC(C1)N2C C1(C(N2CC(C)(COC)C2)=O)CCC12CCC2.c1(C=O)cc(C)c(C)cn1.N c1(C(=O)N)ccn[nH]1.c1(CC=O)nncn1C.C1(OCC)CN(C(=O)C)C1 CCC(CN(C)C)C(=O)N1CCC(OCCNC(C2CC3CCC3C2)=O)C1 O=C(CS(F)(F)(F)(F)F)N1CC2CCC(C1)N2C(c1cnco1)=O C1(C(=O)NCC2(Cl)CC2(F)F)(NC(CCNC(C)=O)=O)CCCC1C C(=O)(CCCN(C)C)NC1C(CSC)CCC1.C1(=CC=O)CCCCC1.N N1(C(c2nc(C)[nH]n2)=O)CC(F)(F)CC1CCNC(C1CCCCCC1)=O c1(C(=O)OCCc2c(C)ccs2)ccc2c(c1)CCN2 CC(CC(=O)N1CC(CO)(NC(C2CC(=O)N(C3CC3)C2)=O)C1)CC(F)(F)F C1(O)(C=O)CCCC(C)(C)C1.CC(C)CCNC(=O)C(C)OC1CCCC1.N C(=O)C1=CC(C)CC1.c1(CCC)ccc(C(=O)NCC(C)Cn2cccn2)[nH]1.N C(=O)(CCCC(F)(F)F)NCC1(C)CCCN(C(Cc2nc(C)[nH]n2)=O)C1 C1(C(=O)NCCC(C(C)C)NC(c2c(C)coc2)=O)CCCCCS1(=O)=O N1(C(CN(C)CC)=O)CCC(NC(C2CC3(CC3)CO2)=O)C(O)C1 Cc1ccccc1C(C)C(N1CCOC(C2(NC(C3CC34CCC4)=O)CC2)C1)=O C1(C(N(CCC)CCNC(c2ccn(CCF)n2)=O)=O)CCC(=O)N(C)C1 C(CCC(=O)N(C)CC1(F)CCC1)(C(C)C)NC(C(CCC)NC(N)=O)=O C1(CCC)(NC(=O)Cc2ccc[nH]2)CCCN(C(=O)CC2CCCC(=O)C2)C1 N1(C(C(CN(C)C)O)=O)CC(F)(F)CC1CNC(=O)Cc1ccc(F)cn1 S(=O)(=O)(c1cccc(N(C)Cc2nc(C(F)F)cs2)n1)NC(C1CCCO1)C N1(CC=O)CCS(=O)(=O)CC1.Cc1cnc(CCC(=O)NCC2CCC2)[nH]1.N C1(C(=O)NCCCN(C(c2c(Cl)cc(C)s2)=O)C(C)C)CC2CCCCN2C1 C1(CC)CN(C(C2(C(C)(C)C)CCC2)=O)CCC1NC(=O)CCCN(C)C C1(NC(C(CC)C2CCOCC2)=O)CCN(C(c2cn(C)cn2)=O)C1(C)C S(=O)(=O)(c1ccc(F)c(C(=O)NC2CCC2)c1)NCC.C(=O)CC#N.C N1(C(c2c(C)ccc(C(C)C)c2)=O)CC(C)N(C(c2coc(Cl)c2)=O)CC1C C1(C(=O)NCCN(C(=O)CCC2CC2(C)C)CCC)CCn2cc(C)nc2C1 CCCCCC(CC)C(=O)N(C1CCCCN(C(c2ccc(O)c(Cl)c2)=O)C1)C N1(C(C2CC(F)CN2C(c2cccc(O)c2)=O)=O)CCc2cnccc2C1 c1(C(N2CCC(CNC(CCCCC)=O)(OC)C2)=O)cn2c(n1)CCCC2C CN1c2ccc(C(N3CCOc4cc(F)ccc4C3)=O)cc2C(C)(C)S1(=O)=O C1(NC(=O)NCC(CC=C)Nc2ccccn2)C2CCC1CC2 N1(C(=O)CCCn2ccnc2)CC(O)CC1CNC(C1(F)CC=CCC1)=O N1(C(C)C)CCCN(C(C2CCN(C(C3CCCN3C=O)=O)CC2)=O)CC1 CC1(C)CCC(CC(N2CC3C(CNC(c4cncc(Cl)c4)=O)C3C2)=O)OC1 c1(OC)cccc(CN(C)C(C2C=CCNC2)=O)c1Cl CC1CCN(C(=O)C(F)F)C1CNC(C1CC1c1ncccc1Br)=O O=C(C1Cc2ccccc21)NC1C2CC1N(C(c1cnn3c1OCC(O)C3)=O)C2 C=CCCN=C(NCc1cccc(CC(F)(F)F)c1)NC1CCOC2(CCC2)C1 C1(OC(C)C)(NC(=O)NC(Cc2ccccn2)CO)CC(C)(C)C1 C(CC(C)C(=O)N(CC(C)(C)NC(=O)CS(N)(=O)=O)C)=CC c1(NC(C)=O)ccc(C(=O)N(C2CCN(C(c3snnc3C)=O)C2)C)cc1F N1(C(COCCCC)=O)C2CCC1CN(C(c1ccn(CC(F)F)n1)=O)C2 CCCC(CC)CC(=O)NCC1CCCCN1C(=O)C(C)c1cccs1 N1(CCc2cn(C)nc2)CCC2(CCN(C(c3cc4n(n3)CCCC4)=O)C2)C1 c1(CCC(=O)NC(CC=C)CNC(=O)C(C)Cc2cnc[nH]2)ccccc1NC C1(CNC(c2cnc(C(C)=O)s2)=O)CCCCC1NC(c1ccc(C)s1)=O N1(C(C(CC=C)C)=O)CCC(CNC(=O)CCc2cc(OC)no2)C1(C)C C=CC1(c2nc(C3CC(=O)N(c4ccccc4)C3)no2)CCCC1 CC1(C)CC(C)CN1C(C1CC=CCC1)=O.C(=O)(C[SH](=O)=O)N.C(C)(C)C C(=O)(CCC=O)OC.C(=O)C.C(=O)CN(C)C(C)=O.C(C)=O.CC.N C12(CNC(c3occ(C)c3C)=O)CN(C(c3sccc3C#N)=O)CC1CCO2 C1(CNC(CN(C(CC(CC)SC)=O)C(C)C)=O)OC(=O)CC1(C)C CC(C)CCCCC(=O)N1CCOC(C)C1C(=O)NCCC1CCCO1 c1(N(C)C)ccc(C(N2CC3C(NC(C4(n5cccn5)CC4)=O)C3C2)=O)cc1F N1(C(c2c(SCC)cccc2)=O)CCC(C)(CNC(C2CC2C)=O)CC1.O c1(C(=O)NC(C2N(C(CC(CC)C)=O)CCC2)C)cc2c(F)ccc(F)c2[nH]1 C12(C(=O)NCC3OCCCN(C(C(CC)F)=O)C3)CCC(C)(C(=O)O1)C2(C)C N1(C(c2cncc(C#C)c2)=O)CCC2CCCC12C(=O)NC1CN2CCCC1C2 C1(NC(c2c(OC)nn(C)c2)=O)CCCC12CN(C(c1cc(Cl)cc(Cl)c1)=O)C2 C1(CC)CN(C(c2ccc(C(C)C)cc2)C(=O)NC2(C)CC2)CCN1C C1(C(=O)OCCOCCOCC(C)C)C2CCC(O2)C1OCCO c1(C(N2CCCC(CCNC(=O)Cc3cnc[nH]3)C2)=O)cnn2cnnc2c1 C12(C(N(C)CCOCC(F)F)=O)CCN(C(c3ccncc3Cl)=O)CCC1C2 CC12CN(C(c3cccc(Cl)c3Cl)=O)CC1CN(C(C1CC1(F)F)=O)C2 N1(C(c2ccc(OCC(F)(F)F)cc2)C(=O)NCCC)CCOC2CCCCC12 N1(C(c2ncc(CC)s2)=O)CCCCCC1c1noc(C)n1 C1(CC)CC(=O)N1.C12(NC(c3scc(OC)c3)=O)COC(COC)(C1)C2 Cn1c(C(=O)NC2(C)CCN(C(C3CC4(C3)CC4(F)F)=O)C2)ccc1[N+](=O)[O-] N1(C(Cc2ccn(C(C)C)n2)=O)CC=C(CCNC(C2CCC(=O)N2)=O)CC1 C1(NC(C(CC#C)O)=O)COC2(C1)CN(C(c1ccncc1)=O)C2.C(C)(C)(C)S c1(NC2(c3n(CCCSC)nnn3)CCC3CCC23)cc(C)c(F)cc1C C(CCCCN(C)C(C1C=CCC1)=O)NC(C(C)N(C)C1CC1)=O N1(C(C2C(OCC)C2)=O)CCC2(CCC(NC(=O)C(C)C3CCCO3)CC2)C1 c1(CCC(=O)NC2CC2NC(c2csc(O)n2)=O)ccc(Cl)nc1 C1(C(N(C(CCNC(c2ccc(NC(C)=O)cc2)=O)C)C)=O)CC2COCC2C1 CCCCC(C(=O)NC1CCN(C(=O)C2=CSCS2)C1(C)C)N1CCCS1(=O)=O N1(c2c(F)cnc(OCC)n2)CCc2c(C(N3C4CCC3COC4)=O)n[nH]c2C1 CC(CN=c1[nH]c2cccc(F)c2s1)N1CCCC(CC(N)=O)C1 Cc1c(C(=O)NCCCN(C)C(C2(C3CCCO3)CCC2)=O)ccn1C1CC1 C1(NC(c2cnn[nH]2)=O)CCC(N2CCN(c3nnc(C(F)F)o3)CC2)CC1 C12CCC(C1)C(=O)N2.c1(OCCC)cncc(CNC(=O)C(=O)N)c1.C C1(NC(c2c(COC)noc2)=O)CN(C(=O)Cc2ccccc2O)CC1C c1(NC(C2CCC(C)N2C(C2CC2C)=O)=O)ccc(O)c([N+](=O)[O-])c1 c1(C(=O)NC2CN(C(c3c(C)cco3)=O)CC(O)C2)cc(Cl)c(Cl)c(Cl)c1 c1(C(N(CCC(=O)NC2CC23CC(O)C3)CC#C)=O)cc(C#N)[nH]c1C c1(C=O)c(C)nn(C)c1C.C(CC(=O)N)SCC(=O)OC.CC(C)C1CC1 C(CC(=O)NCCS)N(CC(N)=O)C(=O)CC1CCN1C(=O)OCCO N1(C(C(C)n2cnnn2)=O)CCC(O)C(N(C)C(c2cnc(N(C)C)nc2)=O)C1 C1(C(=O)NCCCC2CCN(C(Cc3c(C)nc[nH]3)=O)CC2)CCCC(F)(F)C1 CCCCCC=CCC(=O)NC1(CCNC(C2C(C)C2C)=O)CCC1 c1(C(=O)NC(CNC(Cc2nc(CC)sc2)=O)C(C)C)nc(Cl)oc1C C1(CC)CCC(C(=O)N(C)CC2CCCN2C(c2cc(OC)cnn2)=O)CC1 Cc1ccc2oc(C(=O)NC(C)CCN(C)C(c3cc(Cl)no3)=O)cc2n1 C1(NC(CCC(=C)Cl)=O)CC(NC(=O)C(c2ccccc2)SC)C12CCC2 Cc1sc(C(=O)NC2(C)CC(NC(c3ccc(C#N)nc3O)=O)C2)cc1[N+](=O)[O-] C1(CNC(C2(CC=C)CC2)=O)(NC(C2CC(OC)C2)=O)CCCCC1C Cc1ccc2c(c1)CCN(C(=O)CC1CC1c1ccccc1)C2C C1(CC(=O)NCC2CCC(NC(c3cc(C)on3)=O)C2)CCC(F)(F)CC1 C1(NC(C2CC(N(C)C)C2)=O)C(C)(C)CC1(C)C.C(=O)(CC)N.C1CCC1 CC1CN(C(=O)CCN2CCCC2)CC1CCNC(c1nc(Cl)c(Cl)s1)=O CC1CCN(C(=O)C#CC2CC2)CC1CNC(=O)CCn1cc[nH]c(=O)c1=O C#Cc1cc(F)ccc1CNC(=O)Nc1ncc(-c2ccccc2)cn1 c1(OC)cc(C(N2CC(F)(CNC(C3(OC)CCOC3)=O)C2)=O)on1 N1(C(c2cc(C)nc(O)n2)=O)CC(NC(C2C=CCCC2)=O)CC12CCCC2 C1(CNC(C(C)(C)OC)=O)C2CCCC1N(C(c1ccc(N)c(C)c1F)=O)C2 C1(C)(C(N(CCCCCNC(C=CCC)=O)C)=O)CCC(=O)NC1 C1(CNC(c2[nH]nc(OC)c2Cl)=O)COCCN(C(=O)COc2ccccc2)C1 c12ccc(cc1)C(=O)Nc1nc-2cs1.Cn1nnc(CC(=O)N(C)C)n1 c1(C(=O)NC(C(CO)NC(C(=O)NCCOC)=O)C)ccc(CO)nc1 N1(C(c2ccc(OC)nn2)=O)CCN(C(=O)CCCN(C)C)C(C)C1C N1(C(C2CC23CCOC3)=O)CCC2(C1)CN(C(C1CCCC3(CC3)C1)=O)CCO2 c1(C(=O)OC)ccc(NC(C2(F)CN(C(c3csc(C#N)c3)=O)C2)=O)cn1 N1(C(c2cc(C3CC3)ncc2Br)=O)CCC(=C(Br)Br)CC1 O=C(C1=C(Cl)CCC1)N1CCCCC1CNC(C12CCOC1CCOC2)=O C12(CNC(c3c(C)n(CCO)cc3)=O)CCC1CN(C(c1ncccc1Cl)=O)C2 C(C(C)C)(C(O)C(=O)NC(C)C(N1CCOCC1C(C)(C)C)=O)OC Cc1ccc(C)c(C(=O)NC2(C(=O)NC)CCCC2C)n1.C1CCC1.C1CC1 CC(C)(C(=O)N=c1ccc2cnccc2[nH]1)c1ccc(F)cc1 Cc1ccc(OC2CN(C(c3ccc(Cl)cc3SC3CCOCC3)=O)C2)cc1C n1(CC(C)C)[nH]c(CNC(N2CCCC2CC(C2CCC2)O)=O)cc1=O N1(C(c2ccc(N(C)C)cn2)=O)CCOC2CCN(C(=O)Cc3cc[nH]c3)CC12 Cc1cccc(C(C)(O)C(=O)N2CC(O)(C(Cl)(Cl)Cl)C2)n1 CC1CN(C(=O)C#CCNC(C2(n3cnnn3)CC2)=O)CC(C)N1C Cc1onc(C2CC2)c1C(=O)NC1CCC(C)CC1.C(=O)(C(C)N1CCC1)N C1(CNC(C2(SC)CCC2)=O)CC(F)CN1C(=O)CCc1ncc(C)[nH]1 C1(C)(OCC)CN(C(C2(NC(=O)CC3CC3(C)C)CC2)=O)C1 c1(NC)ccccc1C(N1CCCC(CCC=O)C1)=O.N1(C)CCC(C(=O)OC)C1 C(=O)(CCCCC(F)(F)F)NC1C(C)(NC(c2ccnc3ccnn23)=O)CCC1 N1(C(C=C(C)C)=O)CC(CC(=O)NC(c2cnn(C)c2)C)CC1(C)C C(=O)(C1=C(C)CCC1)NCCC1CN(C(C(CC)(O)c2ccccc2)=O)C1 C(CC(F)F)(C(=O)NOCc1cccnc1)NC(CCC(C)CN(C)C)=O c1(OC)ncc(Cl)cc1C(=O)NCC(C)CNC(=O)COC.C1CC1 c1(C(=O)NCC(CC(=O)N2CC3CCC3C2)OC)cccn2nccc12 Cc1c(Cl)ccc(C(N2CC3C(NCc4ncc5ccccn45)C3C2)=O)c1Cl C1(NC(CCOCC)=O)CCC2CCN(C(=O)CC(C)C3CC3)C1C2 N1(C(CCCNC(=O)OC)=O)CC2CN(C(c3cccnn3)=O)CC2(C)C1 Cn1nc(C(N2CCCCC2CNC(=O)COC2CC2(F)F)=O)c(Br)n1 c1(CC=O)c(C)cccc1F.C1(NC(C2C(COC)CCC2)=O)CCCCC1.N n1(C(C)C)ccc(C(=O)NCC2(F)CC(C)C2)cc1=O.C(=O)CC(F)(F)F C1(NC(c2c(C)cc(F)cc2)=O)C2CC(O)C1N(C(=O)C(C)c1cncs1)C2 C12(NC(c3scc(OC)c3)=O)CCCN(C(=O)COC(F)F)CC1C2 c1(OC)cccc(C(N2CCOC(CNC(c3ccc(Cl)cc3O)=O)C2)=O)c1O c1(C(C(=O)NCC(CNC(CCC#CC)=O)F)C)ccc(OC)c(F)c1 C1(O)(CNC(c2ncn(C)c2)=O)CCN(C(=O)CC(O)Cc2ccccc2)C1 C1(O)(CNC(CCN(C(CCC)C)C)=O)CC2CCC(C1)N2C(=O)CCOC C(=O)(C(O)CC(N)=O)NCC(CN(C(C1N(CC)CC1)=O)C)O C1(C(N(C(C)CC(=O)NC(c2ccn(C)n2)C)C)=O)CCCC(O)C1 Cc1sc2ccccc2c1C(=O)NCC1C2CCC(C2)N1C(=O)C(C)C Cc1ccc(=O)n(CC(=O)NCC2CCCC2)c1.C1(C=O)CCOC(C)(C)C1.N C(=O)(CCCC(=O)N1CC2CCC1C2NC(=O)Cn1ncc(Br)n1)N(C)C c1(C(=O)NC2C(NC(c3cc(OC)c(C)cc3)=O)CC2)cnn2c1OCCCC2 C(=O)(C(CNC(c1c(C)nsc1C)=O)CC(C)C)N1CCC(C(=O)OC)C1C c1(C(N2CCCCC(N(C)C(c3ccnc(O)c3)=O)C2)=O)cccc2ncnn12 C1(NC(C(CC)O)=O)CCCCC1C.n1(CC=O)nc(C(F)F)cc1C1CC1 C(CCC(O)CO)NC(C1C(NC(CN2CCC(OC)C2)=O)C1(C)C)=O n1(CC(=O)NC)nc(C)c2cccnc12.C1(CC)CCCC1C(=O)NC1CC1 N1(CC(=O)NCCC2(CNC(CC3CCC(C)C3)=O)CC2)CCCCCC1 C(=O)(CC(C)C(F)F)N1CC(SC)C(NC(=O)CN2CCc3ccccc32)C1 Nc1ccc(Cl)cc1C(N1CCC(O)(CCNC(c2c[nH]ccc2=O)=O)C1)=O N1(C(c2n(CC)nnc2C)=O)CC(NC(=O)C(C)NC(N)=O)CC(C)C1 C1(C(=O)O)CCN(C(=O)C(c2c(F)cccc2F)F)CC1F CCCCCCCCN(C)C(C1C2CCC(C2)N1C(=O)CN(CCCC)CC)=O N1(C(C=CC(C)NC(C2(C)COC(=O)N2)=O)=O)CC2(C1)CC1(CCC1)C2 c1(C(=O)NC2CCN(C(CC(C)(C)O)=O)CC2)c(O)cc(Cl)cc1Cl C1(C(=O)NC(CCCCC)C)CC(C)(C)CCN1C(=O)CS(=O)(=O)CC c1(NC2CC3(CC(C)(C)C3)C2)nc2c(cc1C(=O)O)CNC2 C1(CC(N2CC(C(C)NC(=O)CC3CCCCO3)C2)=O)CCC(=O)NC1 CC(C(O)C(F)F)NC(=O)CCC1CC(NC(c2ccc(C(N)=O)[nH]2)=O)C1 C=CCCC(C(=O)N1CC(CC)CC(C)C1)NC(=O)CC=C(Cl)Cl Cc1csc2ncc(C(=O)N(CCCNC(c3cc[n+]([O-])cc3)=O)C3CC3)n12 CC(C)N=c1[nH]c(N2CCc3c(NS(C)(=O)=O)cccc3C2)nc2c1CCC2 N1(C(C(CCC)O)=O)CCN(C(=O)CCc2ccc(OC)cc2)C2CCC12 CC(=O)CCCC(=O)NCC(C1CCCN1c1ncc(O)cn1)(C)C Cc1nn(C)cc1S(=O)(=O)N1CCCCC(NC(=O)Cc2cccc(Br)c2F)C1 N1(CCNC(N(c2snc(C)n2)C)=O)CCCc2ccccc21 c1(NC(c2ccc(F)c(Br)c2)c2nnnn2C2CCOC2)ccc2nccn2c1 Cc1ccc(C)n1CC(=O)NCC12CC1CN(C(C1(F)CC1)=O)C2 CC(C)CCC(O)C(=O)NCCCOCCN(C(=O)CCCN=[N+]=[N-])C O=C(C1=CCCOCC1)NCCCCCNC(C1(c2ccc(F)cc2Cl)CC1)=O Cc1nc(N(C)C)sc1C(N1CCCC1C(C)C)=O.C1(C=O)CC(=O)N(C)C1 c1(C2C(C(N3CCCC3)=O)C2)cccc(Br)c1.C1(CC#N)(C(=O)N)COC1.C CC1(C)OC2(C(=O)NCCC3CCC(NC(C4CC4Cl)=O)C3)CCC1CC2 CS(=O)C1(CNC(=O)C(=O)NCCCCN2CCCCC2)CCC1 C1(NC(c2cn(CCC)nn2)=O)CC2CC(NC(=O)C(C)n3ccnn3)CC12 C#CC1(C(N2CC(CNC(C3CCO3)=O)C(C)(C)C2)=O)CCCCC1 n1(CC(=O)N(C(C)CC)C)nc(C2CC2)n(C)c1=O.C1(C(=O)N)CC1C1CC1 c1(CN2CCC(C(=O)OC)C2C)cc(Cl)cc(Cl)c1F C(CC(C(=O)N(CCCNC(=O)CC)C(C)C)N(C)C)SC.C(C)(=O)N Cc1cc(O)ccc1CNC(C1C(C)CCN1C(C1CCCCNC1=O)=O)=O C1(CNC(C(CSC)C)=O)(NC(C2CCCN(C(C)C)C2)=O)CCCCC1 C(=O)(CCCC(=O)OC(C)(C)C)NC(C(C)NC(c1ccco1)=O)CO S(=O)(=O)(c1sccc1Br)N(C(c1ccc(C(F)(F)F)cc1)C)C Cc1nc(O)[nH]c1C(=O)NCc1cccc(C(=O)NC)n1.c1ccc(Cl)cn1 c1(C(=O)NC(C(C)NC(CSCCOC)=O)C(C)C)cc(O)cc(C)c1 c1(C(=O)NCCC2CCC(NC(c3cc(C#N)oc3)=O)C2)ccc(Cl)nc1O S(=O)(=O)(CCC(=O)N1CCC2(CC2)C1)NC.c1(C=O)cnc(C(C)(C)C)nc1 N1(Cc2ccc(F)cc2I)CC2CCN(c3ccncn3)CC2C1 c1(C(=O)NCC(O)CCNC(C2CC2(Cl)Cl)=O)cccc2ncnc(O)c12 C1(C(=O)NC2COCC(C)(C)C2)(OC)CCCN(C(=O)CCc2ccncc2)C1 N1(C(C(CCC(=C)C)C)=O)CC2(C1)CN(C(=O)C(C)(C)CC#N)CCO2 n1(CC)nc(C)c(CC(=O)NCCC(O)CNC(=O)CCC(C)SC)c1C CC(CCNC(=O)C(c1ccco1)NC(=O)CS)C(F)(F)F.c1cn[nH]c1 N1(C(C(C=C)(C)C)=O)CC(NC(=O)C=CCN2CCOCC2)C(C)(C)C1 N(C(=NCc1ccc(Br)cc1)NCC1CC(=C2CC2)C1)C1CCC(F)C1 C(=O)(CC(C)C(=O)NCCCC(=O)NCCCCCCCO)OC C(C)(C)(C(C)CC(=O)O)NC(C1CCC(n2cc(C(=C)C)nn2)C1)=O N1(C(c2c(C)csc2)=O)CCC=C(C(=O)N2CC(CO)C(CO)C2)C1 C(=O)(C1CCCc2nncn21)Nc1cccc(CNC(=O)Cn2ccnn2)c1 Cc1noc(N)c1C(=O)N(CC(C)CNC(C1C=CCCC1)=O)C N1(C(c2cnc(CC)nc2O)=O)CCCC2CN(C(=O)CC#N)CCC12 C1(NC(C(C)NC(CN(C(C)C)C)=O)=O)CCC(C)C1 CC1CN(C(=O)CSC(C)C)CC2(CCN(C(=O)CN3CCOCC3=O)C2)O1 CC1CN(CCN2CCC2CSc2cccc(NC(C)(C)C)c2)CC(C)O1 CC1CN(C(=O)CCc2cnn(C)c2)CC(C)C1NC(=O)CC1(O)CCC1 c1(CCNC(C2(C)N(C(C=CCOC)=O)CCC2)=O)c[nH]c2ccc(C)cc12 N1(C(c2cnc(CCCC)s2)=O)C2CCC1(CNC(c1ncc(CC)s1)=O)CC2 C=CCC(CC=C)c1noc(CN2CCCC(C(c3ccccc3)O)C2)n1 Cc1ncc2ccc(C(N3CCC4(CCC(NC(=O)CC(C)(C)C)C4)C3)=O)cn12 C1(CNC(c2ccc(CN=[N+]=[N-])o2)=O)CCCN(C(C2CCOC2)=O)C1 c1(NC(CC2(C)CN(S(=O)(=O)c3cccnc3)C2)=O)ncc2ccccc2n1 C1(C(=O)N(C2CN(C(C3CCCC3(C)C)=O)C2)C)(COC)CC=CCC1 N1(C(C2ON=C(C(=O)OC)C2)=O)CC2CC(NC(=O)CCC3CCCO3)CC2C1 N(C1c2ccccc2CC1NC(=O)CCSC1CCCC1)C(CCOCC)=O c1(C(=O)OCC(C2C(C)CCCC2)=O)c(N)n(C)c(=O)n(C)c1=O c1(C(=O)NC2(C)CCN(C(c3ccco3)=O)CC2)ccc2c(c1)NCCC2=O c1(C(N2CC(F)(C(=O)NCC)C2)=O)cc(Cl)ccc1O.C1CCS(=O)(=O)C1 C1(NC(=O)CC2CSCCS2)CCC(CNC(=O)CCOC2CCCOC2)CC1 c1(CC)c(NC(C2CC23CC(NC(C2(O)CCOCC2)=O)C3)=O)cnn1C c1(NC(CC)C2CC2)cc([SH](=O)=O)ccc1C#N.c1(CC(C)N)c(C)noc1C C1(CC)CN(C(=O)C(c2ccnn2C)NC(=O)CNC=O)CCS1 N1(CCCCCNC(c2nc(Cl)sc2Cl)=O)CCN(c2ncnc(Cl)n2)CC1 CCCCC(C(=O)N1CCC1C(C)O)NC(c1n[nH]c(C)c1C)=O c1(CC(N2CC(N(C(CNS(NC)(=O)=O)=O)C)C(F)C2)=O)coc2ccccc12 N1(C(c2n(C)nc(CNC(=O)CCC3CCC3)c2)=O)CC2COCC2(CO)C1 N1(C(C2(OC)CCCCC2)=O)CC(NC(=O)C(C)Cc2cnc[nH]2)CC(O)C1 c1(OCC)cccc(C(=O)NC2CCCC2)c1.C1(C#N)(C=O)CC(C)C1.C C1(C(=O)NC2(CCNC(=O)CCF)CC2)CCC2CC2CC1 CCC(C)CC(C(=O)N1C2COCC1C2)NC(=O)Cc1ccccn1 C1(C(N2CCC(C(C)NC(c3cc(C(F)(F)F)n[nH]3)=O)C2)=O)CN(C)CCO1 N1(C(C(Cc2ccoc2)NC(=O)CSCC(F)F)=O)CCC(O)(CO)C1 CC(N=c1[nH]c(N2CCC3CCC(C3)C2)nc2c1SCC2)c1ccn(C)n1 c1(N2CCC(N(C(CC3N(C)CC=CC3)=O)C)CC2)cc(Cl)nc(C2(C)CC2)n1 c1(C(C)C(=O)NCCNC(c2cocn2)=O)cccc(Cl)c1 CC1COC2(CCC2)CN1C(=O)CC1CCN(C(=O)C(F)(F)CO)C1 N1(C(COCC=C)=O)CCC(C2CC2)C1.c1(C=O)ccnc(C(F)(F)F)n1.C CC(C)(C#N)CCCC(=O)NCC1CN(C(c2nc(Cl)c(Cl)s2)=O)CCO1 C=Cc1ccc(C(=O)NCC(CC)(CC)NC(=O)C(C)CN(C)CCC)cc1 CS(=O)(=O)C(CNC(=O)C)C.C1(C=O)CCCC(C(N)=O)C1.CC(F)F C(=O)(CCCCC(C)(C)OC)NC1(CO)CN(C(c2cc[nH]c(=NC)c2N)=O)C1 CC(C)C(C)CC(=O)NCC1CC(F)(F)CN1C(=O)CCc1ccsc1 C1(CCNC(CCNC(=O)NC)=O)CSCCN1C(c1ccc(CCO)cc1)=O N1(C(CC(C)SC)=O)CCN(C(c2cc(CO)c(C)o2)=O)C(c2ccccn2)C1 c1(OC)ncc(C)cc1C(N1CCCC(C(=O)Nc2ccc(O)cn2)C1)=O C1(C)(c2cn(C(C(=O)OC)C)nn2)CCCN1C(c1c(C)csc1Cl)=O N(C(=NCCCc1ccccn1)NCc1nc2c(s1)COCC2)C(C)C N1(C(C(=O)NC2C(C(C)C)OCC2)=O)CCN(C(c2cc(Cl)cnn2)=O)CC1 N1(c2c(C)cnc(C)n2)CCC2(CCCCN(C(c3n[nH]c4c3CCC4)=O)C2)C1 N1(C(C(COC)NC(c2cc(CC)[nH]n2)=O)=O)CCN2CCOCC2C1 c1(C(=O)NC2C(C(C)C)N(C(C3CCCSC3)=O)CC2)cc(F)cc2nc[nH]c12 N1(C(c2c(C)occ2)=O)CCCC(C2(NC(c3cc(F)cc(Br)c3)=O)CC2)C1 C#CC(C(C)C)NC(C1(NC(=O)CSc2nc[nH]n2)CCSC1)=O Cc1ccc2n[nH]cc2c1C(=O)NCC1CCN(C(=O)C(F)C(F)(F)F)CC1 N1(C(C(=O)NCC2(C)CCCC(C)(C)C2)=O)CC2CCC(C1)C(N)C2 Cc1cc(C)c(C(N2CCC(C)(C(=O)NCC3CCCSC3)C2)=O)s1 Cc1cc(C)c(CNC(=O)NCCOCCCO)c(C)c1Br N1(C(CC2CC(=C)C2)=O)CCC2(C=C(C(=O)Nc3ccc(Cl)c(C)c3)C2)C1 C1(CCC)(NC(=O)CN2CCS(=O)(=O)CC2)CCCN(C(=O)CC(C)(C)O)C1 N1(C(C2SCCN(Cc3c(C)ccc(C)c3)C2)=O)CCOc2ccccc2C1 N1(C(c2c(C)nsc2)=O)CCC2CC(NC(=O)Cn3ncnn3)CCC2C1 CC1CCC(NC(=O)CC(C)Cc2ccc(Cl)cc2)CN1C(c1cccnn1)=O C1(NC(CN2C(C)CCC2)=O)CC(C(=O)NC(C)(C)CCO)=CC1O N1(C(c2ccc(C)cc2)=O)CCN(C(c2cnc(C)s2)=O)CC1c1ccnn1C C1(C(=O)NCCC(CC)(C)NC(=O)C(F)Cc2ccccc2)CCOCC1(C)C c1(C(=O)NC2(CCCNC(C=C(COC)C)=O)CC2)sc(CO)nc1C c1(C(NCC)=O)ccn(C)c(=O)c1O.C1CCN(C(=O)C(F)CC2CC2)CC1 CCCCC(F)C(=O)NC(CCC1CC1)C(=O)NCC1CCOC1=O CC(C)(CO)C(=O)NCC1CCCCN1C(C1C(C(F)(F)F)C1[N+](=O)[O-])=O C=C(C)CC(C)C(=O)NC1CCC(NC(c2cccn(C(C)(C)C)c2=O)=O)CC1 c1(CC)nn(C)c(Cl)c1C(=O)N(CCCCCCNC(c1c(C)noc1N)=O)C C(c1cnccn1)=CC(=O)NC1CC(C(=O)NC(C(C)c2ccccc2)CO)C1 c1(OC)cc(C(=O)NC)cc(F)n1.C1CCCN(C(=O)Cc2ccc(Cl)cc2)C1 c1(C(N2C(C=CC(=O)NCc3cc(C)[nH]n3)CCC2)=O)cccc(F)c1N C1(C(N2CC(NC(c3cccnn3)=O)C2)=O)CCCCS1(=O)=O n1(CCCC)ncc(C(=O)N(CCCNC(=O)C(C)C2CC2)C)c1C.C(C)=O C(=O)(CC(C)(C)O)NC(C1(CNC(c2cnn[nH]2)=O)CC1)C c1(C(N(CCCCNC(=O)C=CC=C(Cl)Cl)C)=O)cc2sccc2[nH]1 C1(NC(C(=O)NCCOC)=O)COC2CC1C2.C1(C=O)CC(=O)N(C)C1 CC1(C)CCC=C(C(=O)NC)C1.C1CC2CCC1N2C(=O)Cn1cc(C#N)cn1 N1(C(CSC)=O)CC(NC(c2coc(Cl)n2)=O)CC2(CC2)C1 C1(C(=O)N)CC(=O)CN1C(C1(CC)CCC1)=O.C(=O)(C(C)C)OCC C(C(=O)N(CC(=O)NC(C)COCC)C)OCCC CCCC(C(=O)NCC)N(C(CC1C=CCC1)C(=O)NC)C N1(C(CCCC)=O)CC2CCCC2(CNC(=O)CC2CCOCC2)C1 Cc1cccc2[nH]cc(CN3CCCC(NC(c4snc(Cl)c4Cl)=O)C3)c12 CC1OCCCC1C(N1CC(O)(CNC(c2cccnc2O)=O)C1)=O C(=O)(C(C)=Cn1ccnn1)NC1CC2CN(C(c3c(OC)ccc(O)c3)=O)CC21 CC1(O)CCCN(C(=O)C=CCNC(=O)CC2CCCSC2)C1 c1(C(C)(F)F)cncc(C(N2CCN(c3cc(C(F)(F)F)[nH]n3)CC2)=O)c1 N1(C(C(C(C)O)NC(c2c(OC)nccn2)=O)=O)CCOCC(C)C1 N1(CC(=O)NCC2CN(C(=O)C(O)C3CC3)CCO2)CCCCS1(=O)=O C1(NC(C(C)N(C)C)=O)C=CCN(C(c2occc2-c2cnn(C)c2)=O)C1 Cc1nc2cc(C(=O)CN3CC4(CCC4)C3)ccc2n1CC(N1CCCC1)=O CC(Cc1ccccc1)C(=O)NCC1(O)CN(C(=O)C(C)n2cncn2)C1 CC12CC(C=O)(C1)C(C)(C)O2.C1(CC)CSCCN1C(=O)CC1C=CCC1.N Cc1cc(C(=O)NCCCC2(NC(=O)C(c3cnccn3)C)CC2)cc(C)c1 N1(C(CCC=CC)=O)CC(C)N(C(c2cc(O)cc(F)c2F)=O)CC1C C1(C#N)(CNC(C(CO)NC(c2c(C)snn2)=O)=O)CC(C)(C)C1 C(=O)(CC(C(=O)N1CC2(C1)CN(C(=O)C)C2)c1ccccc1)OC.C(N)(=O)N N1(C(CC(C)n2ccnc2)=O)CC2CC2(CNC(=O)C=CC=O)C1.C1CC1 c1(C(=O)NCCC2C(C)CCCN2C(=O)C2=C(Cl)CC2)cccc2c1CCCC2 c1(C(=O)NCC(c2ccccc2F)NC(C(CCC)C)=O)ccc(O)nc1C C(=O)(CCCCNC(=O)CC1CCCN1C)NC(c1cnc[nH]1)C N1(C(C2(NC(CCOC(C)=O)=O)CSC2)=O)CCCC(C)(CO)C1 C(=O)(CCCCCC(C)O)NC(CNC(Cc1scc(C)c1)=O)C1CC1 c1(C(N(C(CCNC(C2(COC)CCCC2)=O)C)C)=O)ccc(OC)cc1N C(=O)(C1=CCCOCC1)N1CCC(CCCCN(C2CCC2(C)C)C(C)=O)CC1 N1(C(C(CSC)O)=O)CC(C2CN(C(=O)C(C)NC(c3ccccc3)=O)C2)C1 C=CCC(C(=O)NC1CCC(CNC(=O)C(C(C)(C)C)OC)C1)C(C)C C=CC(CC)CC(=O)N1CCC(O)(CN(C)C(c2cnc(OC)cc2C)=O)C1 N1(CC(=O)N(C)C)CCN(c2nnc(C3CCCCC3)n2CCC#N)CC1 c1(COC(=O)NC(COC)Cc2ccccc2)nnc2n1CCCCC2 c1(C(C)NCCCCNC(=O)N(C)C)ccc(C(F)F)cc1 N1(C(C2C3CC3C3CC23)=O)CC2CC(C1)CN(C(C1(c3ccno3)CCC1)=O)C2 c1ccc(S(N)(=O)=O)cc1.C1(CC)CCCCN1C(=O)C1=NOCC1.C(=O)C.N C(C(=O)NCC1(NC(=O)Cn2cnnc2)CCCC1)(C(C)C)n1ncc(C)c1 N1(C(C(C)(CO)NC(c2n(CC)ccc2)=O)=O)CC(C)OC(C)(C)C1C C1CC(C)(C)CN1C(=O)CC1CCC(C)(C)O1.c1(OC)ccncc1C(=O)N C(=O)(CC1CCCc2ccccc21)N1CC2(OCC(NC(CC(=O)NC)=O)C2)C1 C1(OC)CC(NC(=O)CS(N)(=O)=O)CN(C(c2c(O)cccc2Cl)=O)C1 C1(CNC(CC2CCN(C(C=CCCC(C)C)=O)C2)=O)CC2C=CC1O2 C1(C(N2CCN(C(CSCC)=O)CC2CC(F)(F)F)=O)CCCC12OCCO2 Cc1nc(C)c(CC(=O)N)s1.C1(C2CC2)(CC(=O)N(CC(C)O)CC)CC1 CC(C)CC(C(=O)NC(c1cn(C)nn1)C(=O)NCCCSC)N(C)C C1(C(N2CC(F)(c3nn[nH]n3)C2)=O)CCCC1C1CC1 CC1(C)C=CC(N=c2[nH]c(-c3cccc(C(F)(F)F)c3)nc3c2CCCCC3)CC1 C1(NC(CC2C(C)CCC2)=O)CCCCN(C(=O)CN(c2ccnc(Cl)n2)C)C1 S(=O)(=O)(c1ncc(F)cn1)NCc1c(C(C)C)c[nH]n1 c1ccc(F)c(Cl)c1.c1(CC)ncc(C(=O)N(CCCCN(C(=O)C)C)C)s1.O c1(SC)ccncc1NC(C1CCCCC1NC(=O)CCc1cc(C)[nH]n1)=O c1(C(N2CCCC(CCNC(c3c(C)snc3)=O)C2)=O)cc([N+](=O)[O-])c[nH]1 Cc1cc(C(=O)NC2CCC(CC(=O)NCC3OCCC3C)C2)ns1 C1(OC)CC(C(=O)NC(CCO)C(C)C)N(C(c2ccc(NC=O)cc2)=O)C1 C1(CC(N2CC(CC)(OC)C2)=O)CC(C)(C)CN1C(c1cc(CO)ccn1)=O N(S(=O)(=O)N1CCN(CC(=O)N)CC1)CC.c1cc(C(F)(F)F)cc([N+](=O)[O-])c1 CON(C)C(=O)C1CCCN1C(=O)COCC1CC1 C1(NC(C(COC)C)=O)CCC12CN(C(=O)CCCCc1cnn[nH]1)C2 CC(C)(CCC(=O)Nc1c[nH]ccc1=O)NC(=O)Cc1cscn1 C1(OC)CN(C(C2(CO)CC(C)(C)C2)=O)CCC1.C(=O)(CCCC)N.C(C)=O c1(N(CCOC)C(C2(c3ccccc3F)CC2)=O)ccc(Cl)cc1[N+](=O)[O-].CO Cc1cc(F)ccc1S(=O)(=O)NC1CN(C(C2(F)CCOCC2)=O)CC1(F)F C(=O)(C(C)P(C)(C)=O)NCC(c1ccccc1)N(C(C=C(C)C1CC1)=O)C CC1CC=C(C(=O)NCC2CC3COCC3N2c2ncnc3ccsc23)CC1 c1(C(=O)NCCC2CN(C(C(C(C)C)OC)=O)CC2C)ccc(Cl)cc1F N1(C(C=CC(C)(C)NC(c2cc(CO)ccn2)=O)=O)CCC(C2CCC2)CC1 c1(COCC)n[nH]c(=NC2CC(NC(C3(COC)CC=CC3)=O)C2)s1 CC(C)C(CNC(=O)C(C1(C)CC1)NC(=O)CNC=O)CO C(=O)(C(C)CCCc1ccccc1)N1CCC(O)(CCNC(C#CC(C)C)=O)C1 N1(C(c2nc(C)sc2C)=O)CC(NC(=O)C2=COCCO2)C2(CCCC2)C1 c1(C(N2CCC(OCCOC)C2)C(=O)NC(C)C)cc(Cl)nc(Cl)c1 N1(C(C(CC)=CC)=O)CCC(CCN(C(=O)C(C(C)O)N(C)C)C)CC1 N1(C(C(=O)N(C2COC(C)(C)C2)C)=O)CCCOC(c2ccc(Br)cc2)C1 C(CC(C(C)C)NC(C1(C)CC1C)=O)NC(Cc1nc(CC)sc1)=O Cc1cccc(-c2ncn(CC(C3(CCl)CCCCC3)=O)n2)n1 c1(C(=O)NC2C(NC(c3c(OC)c(Cl)sc3)=O)COCC2)cccc(F)c1C CS(=O)(=O)c1ccc(C(N2CCC3CC23)=O)s1.c1(C=O)cc(C(N)=O)c[nH]1.C Cc1cccc(C(C)(C)CNC(=O)C(=O)NCc2ccccc2CN)c1 c1(C(=O)NC2CN(C(CCC)=O)CC(O)CC2)cn2cccc(Br)c2n1 Cc1nc2c(F)cccc2cc1C(=O)NCC1CN(C(c2cncc(N)n2)=O)C1 C1(C(=O)NCCCCNC(C2(C)CSC2)=O)CC2OC1C1CC21 N1(C(c2cc(C(C)C)on2)=O)CC(NC(C2(C)CCCCO2)=O)C2CCCCC12 c1(N2CC3C(CC)(C3)C2)nc(NCc2c(Br)nnn2C)c2ccsc2n1 CCC(C)(C)C(=O)C(=O)N1CCSCC1C(=O)NC1CC2(CCCCO2)C1 N1(C(c2cn(CC)nc2C2CC2)=O)CCN(C(c2cc(N)ccn2)=O)CC(O)C1 c1(-n2cc(CN3CCC(O)CC(C)C3)nn2)ccc(S(C)(=O)=O)c(Cl)c1 N1(C(c2nc(OCC)oc2)=O)CCCC(NC(=O)CCC(=O)N2CCOCC2)C1 C1(CC(=O)NCC(CC(=O)NC)C)CC(C)(C)CN1C(c1ccccc1F)=O Cc1ccc(N)cc1C(N1CC2CC1CN2C(C1CCCC(=O)N1)=O)=O CC1CN(C(c2ncn(-c3ccccc3)n2)=O)CC(C)N1C(C1CCCC1)=O Cc1c(C(=O)NS(=O)(=O)CCCOCc2ccccc2)c(C(C)C)nn1C c1(N(C)CC2(SC)CCC2)ccc(S(=O)(=O)N2CC3CSCC(C3)C2)cc1C#N CC12CCCC(C(=O)NC)(CO1)C2.C1CCC(O)C1.C1(=CC=O)CCCCC1 c1(NC(C2N(C(c3cc(C)cc(F)c3)=O)CC=C2)=O)ccc2ncsc2c1Br c1(C(=O)NC2(C)CCN(C(CSCCC)=O)C2)ccc(OC)nc1Cl N1(CC)CCN(CC(=O)NCC(C)CN(C)C(C2CC2F)=O)CC1 c1(CC(=O)NCC2(NC(C3CSC3)=O)CCC2)ccc([N+](=O)[O-])cc1F C12(CNC(c3c(C)nc(C)s3)=O)CCC1CN(C(=O)C(O)Cc1[nH]cnc1C)C2 Cc1c(C(N2CCN(Cc3cccc(-c4nn[nH]n4)c3)CC2)=O)cnn1C(C)C Cc1cccc(C)c1CNCC1CCC1c1ccc(Cl)c(Cl)c1 Cc1ccc(F)c(N)c1C(=O)NCCC(C)(C)C.c1(C(=O)N)nc(Cl)c(Cl)s1 C(=O)(C(F)(F)CC(C)C)N1C2CN(C(C3(CC#C)CCCO3)=O)C(C2)C1 C1(C(=O)NCCCn2nc(-c3cccs3)oc2=O)CC(C2CCC2)=NO1 CC1CCCC(C)CN1C(C1CC(O)CN1C(c1cc(C(N)=O)c[nH]1)=O)=O C1(C(N2C(C(C)C)C(C(=O)NCC(C)(C)C(F)F)CC2)=O)CCC2(CCC2)O1 C(C)(C)(CCCNC(c1cc(Cl)sc1Cl)=O)NC(C(COC)C)=O c1(OC)ncc(C(=O)NC2CCC(CCNC(c3ccncc3Cl)=O)C2)nc1C c1(CNC(CN(CC#C)C(C2CCOC2)=O)=O)cscc1C Cc1ccc(OCC(=O)NC2CC(N(C(=O)Cc3ccccc3C)C)C2)c(C)c1 c1(C(N2CCC3(CC(NC(C(CC)(F)F)=O)C3)C2)=O)cc(F)cc2ccoc12 C(CCSC)(c1nnnn1C(C)C)(C1CC1)NCCCOC=C c1(C(=O)NC2CCCN(C(c3ccon3)=O)CC2F)cc2ccc(F)cc2o1 C1(NC(C2CC(C)C2)=O)CC(NC(=O)Cc2cccs2)C(O)C1 C1(NC(=O)CN2CC=CC2)CCN(C(c2cccc(C3CCOCC3)c2)=O)C12CC2 C1(C(=O)NCc2cc(C)c(C)o2)CN(C)CCN1C(=O)C(C)CN(C)C N1(C(c2cc(OC)n[nH]2)=O)CC(O)CC1C(N1CCCC1C1CCOC1)=O C1(CCC(=O)NCCCNC(=O)CCC2CC2)CCC(O)CC1 CC(N=c1[nH]c2c(c(=NCC3CCC(F)(F)C3)[nH]1)CCC2)c1nccn1C C1(C)(CN(C)C(c2cc(F)c[nH]2)=O)CCCC1NC(c1ccsc1Cl)=O C1CCCCC1.n1(CC=O)cc[n+](C)c1.C1(CCOCC)(C(=O)N)CCC1 C1(C(=O)NCC(CC)NC(=O)Cc2ccncc2Cl)OCCC1(C)C C1(C(=O)NC2CC2NC(c2nc(C)n(C3CC3)n2)=O)(OC)CCCCC1 C#CC1(O)CCN(C(=O)C(CNC(c2[nH]ccc(=O)c2C)=O)N(C)C)CC1 CC(C(=O)N1CCCN(C(C2CN(CC(F)(F)F)C2)=O)CC1)C(C)S(C)(=O)=O N1(C(C(CC)F)=O)CCN(C(c2cn(Cc3ccncc3)nn2)=O)C(C2CC2)C1 O(N=C1CCCCCC1)CC(N1CC2C(NC(CN(CCOC)C)=O)(CC2)C1)=O C1(CNC(=O)NCC2(N(C)C)CCOCC2)CCC2(CO1)CC(O)C2 CN1CCC(C(=O)NCc2nnn(C)c2C(N2CCCC2CF)=O)CC1=O N1(C(CC2(OC)CC2)=O)CCC(NC(c2nc(C(F)(F)F)cs2)=O)C12CCC2 Cc1ccccc1C1=NOC(C(N2CC(C)C3(CC3)C2)=O)C1.C1(F)(C(=O)N)CC1 C1(CNC(=O)Cc2ccno2)(NC(=O)CCC2CCOC2)CCCCC1 C(=O)(CCCC(F)(F)F)N(CCCNC(C1N(C(CC)=O)CSC1)=O)CC C1(CNC(C(C)S(C)(=O)=O)=O)CN(C(=O)C(C)n2cncn2)CCC12CCOC2 C1(C(=O)NCC(C)(C)CC2CC2)(SC)CN(C(=O)CCc2nc[nH]n2)C1 c1(C(N(C)C)=O)cccc(C(=O)NCC2CCC2)c1.c1(C(=O)N)ccoc1Br CCCCCOC1CN(C(=O)C(C)NC(C2(CO)CC2)=O)C1 CC1CCN(c2ccnc(NCc3ncc(-c4ccccc4)o3)n2)CCS1=O c1(C(=O)NCC(CNC(C(CCOC)C)=O)CO)cc2c[nH]cnc-2n1 C1(CC)CN(C)CCN1C(C1CCN(C(c2cnc(OC)s2)=O)CC1O)=O S(=O)(=O)(c1ccc(Br)c(C(=O)N(C)Cc2cnn(CC)c2)c1)NC N1(C(C2(C)CCCN(C)C2)=O)CC2CN(C(C3CC3C3CCCC3)=O)CC(C1)O2 C(=O)(CS(=O)(=O)CCOC)NC(CCCC)C(=O)NC(c1cncs1)C Cc1cccc(C(N2CCCC(CC(=O)NCC3CCC3C)CC2)=O)c1N c1[nH]c(=NC2CCCC2)nc2sccc12.OCCOCCOCCOCCN.C C(=O)(C1Cc2ccc(F)cc21)NCCN(C)C(C1CCC2(CC2)C1)=O N1(C(CC=CC=C)=O)C2CCCC1CN(C(C13CCCC1(C(=O)OC)C3)=O)C2 c1(NCC2C(NC(c3c(C)c[nH]n3)=O)CCC2)cc(C2CC2)nc2ncnn12 C(C)(C(C)NC(=O)C=CC(C)(C)C)NC(CSCCC)=O C=CCC(C)C(=O)NCCCC(CO)NC(c1ccc(OCCOC)nn1)=O CC(C)CC(O)CC(=O)N1CCN(CC(=O)NCC(C2CC2)N(C)C)CC1 C(=O)C(C)(C)C(C)(F)F.CC1CN(C(c2ccc(C(O)CF)cc2)=O)CC1C.N C1(CC(=O)NC(C)C(F)(F)F)CN(C(c2ncccn2)=O)CCO1 C1(NC(C(C)=C2CC2)=O)CCC(NC(C2CCCC2)=O)CC1.c1ccccc1.C C(=O)(C(F)(F)COC)N1CCC(C(C)(C)NC(COC(CC)(C)C)=O)C1 c1(C(N(CCCCNC(c2cnncc2O)=O)C)=O)cc(C(F)(F)F)cc(F)c1 C1(C(N2CC(CCC)OCC2)=O)CN(C(=O)CNc2ncccn2)CC12CC2 c1(NCc2c(Br)cc(C)s2)cc(=NCC(F)(F)Cl)[nH]c(C(F)(F)F)n1 Cc1cccc(C(=O)NCC=CCNC(=O)Cc2csnn2)c1 Cc1cc(C(=O)NCC(C)CN(C)C(C2COC(=O)N2)=O)cn(C)c1=O N1(C(c2c(CNC(CC(C=C)CCC)=O)ccs2)=O)CCC(O)C12CCCC2 c1(C(N2CC(O)(COC(C)=O)C2)=O)cc2n(n1)CC(OC(C)(C)C)CO2 C(=O)(CCCCCNC(N)=O)N1CCCC(C(C)NC(C=C(C)C)=O)C1 C1(CN(C(=O)Nc2cc(C(C)(F)F)c(Cl)cc2)C2CC2)CCC2CNCCC2C1 O=C(CS(=O)(=O)CC(F)(F)F)NC12CC(C1)N(C(=O)Cc1cscn1)C2 C1(NC(C2CCOC2)=O)CCCC(NC(C2C=CCS2)=O)C1 C1(NC(c2c(CC)cccc2)=O)C(C)CN(C(c2cn(C)c(=O)cn2)=O)CC1C Cc1cc(C(=O)NC(C)CCNC(C2CCCC(C)(C)C2)=O)cn(C)c1=O c1(C(=O)NC2C(NC(c3ccnc4c3CCO4)=O)COC2)cc2cccnc2[nH]1 N1(C(C=C(CCC)C)=O)CCC(CCCCNC(=O)Cc2cc(C)on2)CC1 Cc1cccc(C(=O)NC2CCN(C(=O)Cc3cnn(C)c3C(F)F)C2)c1C#N C=CCCCCCCNC(C1CSCCN1C(c1csc(C)n1)=O)=O C(=O)(C1CCCc2ncnn21)N1CC2C(NC(CC(CCC)CCC)=O)(CC2)C1 CC1CC(CNC(=O)CCCCNC(N)=O)CN(C(c2ccc[nH]2)=O)C1 N1(C(CC2CC(OC)C2(C)C)=O)CCC(NC(c2ccc(C)s2)=O)C(C)C1 C1(Nc2ccc(C(C(=O)OCC)(F)F)n2C)CCN2CCC1C2 N1(C(C(C(C)C)C)=O)CC(NC(c2cc(-c3cnccn3)[nH]n2)=O)C2(CCC2)C1 N1(C(Cn2nnc(C)n2)=O)CCCC(CC(=O)N(C2CC2C)C)C1 Cc1nc(C(=O)N)cc(O)n1.c1(C(N2CC(C)C2)=O)cn(C)nc1C(F)(F)F C1(C(=O)NC2C(C)CN(C(=O)Cn3ccccc3=O)C2)CCn2cnnc2C1 Cc1noc(CCC(=O)NCC2CCCC2NC(C2CC(C)(F)C2)=O)n1 N1(C(CN(S(C)(=O)=O)C)=O)CC2CCCC(NC(=O)CC3=CCCCC3)C2C1 N1(C(C2C(C)C2)=O)CCCC1C1(NC(C2OCCC2C(C)C)=O)CC1 C(C1CS(=O)(=O)c2ccccc21)N(C)C(N1CCCC1)=O S(=O)(=O)(c1c[nH]ccc1=NC(Cc1ccc(Cl)cc1)CO)N(CCF)CC C1(NC(C(CC)CC)=O)CN(C(c2ccc(F)cc2I)=O)CC12CC2 C(=O)(C1=CC(C)(CC)C1)NCC(C(=O)NC1(CC)CC1)CC1CC1 CN1C(=O)CSC1=CC(=O)NCC1CCN(C(=O)C(O)C2CC2)CC1(F)F n1(CC)nccc1C=CC(=O)NC1CCCCC1NC(c1cc(C)nn1C)=O C(=O)(NN1CCCC1C(=O)NC1(CO)CCCC1(C)C)C1(CC)CCC1 C1(NC(c2cc(C)no2)=O)CC2CCC1(NC(C1CCCCCC1)=O)C2 n1(C(CC)C)ncc2c(C(=O)NCc3ncc(C)s3)cc(C)nc12 N1(C(C(CC)=CC)=O)C(C(=O)NC2CCCCC2CCO)CC2CCCC12 C1(NC(C2CC(C)C2)=O)C(CNC(=O)CCOCC(F)F)C1(C)C C(CC)(C(=O)NCCCC(C)NC(c1cn(-c2ccn(C)n2)cn1)=O)=CC N1(C(=O)CCn2cnc3ccccc23)CC(O)CC12CCCCCC2 c1(C(=O)Nc2nc(Br)cnc2Cl)cnc2ncc(-c3ccc(CO)nc3)cn12 c1(C(=O)NC(CC=C)CNC(c2cnc(Cl)s2)=O)ccc(CO)cc1F Cn1nc(C(=O)NCC2COCCN2C(=O)CCC2(C)CC2(F)F)cc1C#N C(=O)C(CC(C)C)C(N)=O.Cc1cccc(CN(C(=O)CNC(=O)C)C)c1 Cc1cnc(C(N2CCCC2CCCNC(c2nccc(Cl)c2F)=O)=O)c(F)c1 CC1=C(C(=O)N(C2CN(C(C3(C)CCN(C)CC3)=O)C2)C)C=C2CCCN=C2N1 C1(C)(COCC)CCN(C(=O)Nc2ccncc2)CC1.N1C(=O)CCC1=O.C N1(C2CCN(C(=O)CN3CC=CC3)C2)CCN(C(c2cnc(Cl)s2)=O)CC1 C12(C(=O)NCCC(C)C(C)(C)C)CCC(CN(C(=O)C3=CCCC3)C1)C2 C(CCCCC(=O)NC(c1nn[nH]n1)CC)NC(CSCCCC)=O C=CCC(C)(C)c1noc(CNC(=O)CC(C)C)n1 N(C(=NCCc1nc(C)no1)N1CCOC(C2CCC2)C1)C(C=C)C N1(C(COCCCC#C)=O)CCCC(N(C(=O)CCc2nc(C)c(C)[nH]2)C)C1 c1(OC(C)C)ccc(=NC(=O)NCCCc2nc3ccccc3o2)[nH]n1 S(=O)(=O)(c1cccnc1NCCC1CCCCCC1)N1CCCC(CC)C1 N1(C(C2(NC(c3coc(C4CC4)n3)=O)CSC2)=O)CCc2ccncc2C1 Cc1ccc2sc(N3CC(NC(=O)C(C)O)C4(CCOCC4)C3)nc2c1C C1(CC)CN(C(C23C=CC(CC2)C3)=O)CCC1.C1(C)(CCC=O)CC1(F)F.N C1(NC(c2c(C)cncc2)=O)CC2CC1CN2C(=O)C(C)C C[Si]1(C)CCN(C(C2(C)C=CCN2C(=O)Cc2ccsc2)=O)C1 CC1CC(NC(=O)CCCC2CC2)CN1C(c1ccn(C2CC2(F)F)n1)=O C1CN(C(=O)CCc2ccncc2)CC12CC2.C1(CC(=O)NC)(CSC)CC1.C C1(NC(C(CNC(C2C(C)(C)CCO2)=O)CC2CCCC2)=O)CCCC(F)(F)C1 N1(C(CCCC)=O)CCC2CCCC12C(=O)NC(C)C(C)(C)CC C1(NC(c2cn(CCCC)nn2)=O)CN(C(=O)C=Cc2cn(C)cn2)CC1(C)C C1(CNC(c2cn(C)nn2)=O)CN(C(C2CC23CCCC3)=O)CCC12CCC2 CC1(C)CCC(CO)(NC(C2CCC3(CC3)N2C(c2ccc(=N)[nH]n2)=O)=O)C1 c1(CNCc2cccc(Cl)c2)nnc2n1CCC2 CN1CC(C(N2CCOCC2CN(C(=O)Cc2ccccc2)C)=O)NC1=O N1(C(c2nccc(CC)c2)=O)CCC(C2CC2)C1CNC(c1cnsc1)=O c1(NC(C2OCCN(Cc3cncc(C)c3)C2)=O)cc(Br)c2cc[nH]c2c1 N1(C(C(C)(CO)OC)=O)CCN(C(C2(Cl)CC23CCC3)=O)CC12CC2 C1(NC(c2c(C)con2)=O)C2CC1N(C(c1cn(C)nc1C(F)F)=O)C2 c1(OC)c(F)cc(F)c(NCC2(C)CC2)c1[N+](=O)[O-].C1(C=O)C(C)C1C C1(C(N(C2CC3CC(O)CC3C2)C)=O)CC2CCC(C1)N2C(=O)CC1CCCOC1 C1(NC(COCCC)=O)C2CC3C1C3C2C=O.C1(O)(C(C)C)CCCC1.N N1(C(C(CC)F)=O)CC2CCN(C(=O)Cc3cn4c(C)cncc4n3)CC(C2)C1 NS(=O)(=O)c1cc(C(=O)NC)c(F)cc1Cl.C1CN(C(=O)CC2CC2)CCO1 C(C1=NOC2CC12)(c1n(CCSC)nnn1)NC(C)(C)S(C)(=O)=O C(C(C)(C(C)C)NC(c1ccns1)=O)NC(C(OCC)OCC)=O CC1(CNC(=O)CS)CN(C(C2C3COCC23)=O)CCO1.c1ccc(F)cc1 c1(C(N2CCCC(NC(c3[nH]cc(C#N)c3)=O)(CO)C2)=O)c[nH]c2cccnc12 C1(C(N(CCN=[N+]=[N-])C)=O)C=CCCN1C(=O)CCC1CCC(=O)C1 n1(CC)ccc(C(=O)NC(CC2CCC2)C(=O)NC2(c3cccs3)CC2)n1 C(C(C)(C)C#CC(=O)N1CCC(CC)CC1)NC(CCCCC=C)=O C12(CC(=O)N(C3CCCCC3)C)CCCCC1C2(F)F.C(C(=O)N)SC(C)C.C C1(NC(=O)CC(Cl)Cl)COCCC1C(=O)NCCCSC(F)F N1(C(c2cc(C)nn2C(F)F)=O)CC2(CCC(NC(c3cn[nH]c3)=O)C2)C1 C#CCCCC(=O)N1CCOC(C2CN(C(C3(C#N)CCCO3)=O)C2)C1 c1(C(=O)NC(CNC(CCCC#C)=O)CCCC)ccc(S(=O)(=O)CF)cc1 c1(CCC)cc(C(=O)N(C(C)CCNC(=O)C(C)COC)C)no1 Cc1nccc(C(N2CCC(C(C)NC(c3ccc(C(F)F)cc3)=O)C2)=O)c1O C1(C(=O)NC2CCCC(NC(c3ccc(C)cc3Cl)=O)C2)CCc2nn[nH]c2C1 Cc1cnc(C(N2CCC(O)(C)C2)=O)c(C)c1.c1(CC=O)ccc(F)c(Cl)c1.N C#Cc1ccc(CC(=O)NCCNC(C23CSCC2C3(F)F)=O)c(F)c1 N1(C(C2CCc3c(C)[nH]nc3C2)=O)CCCC2(CCN(C(=O)C#CC(C)C)C2)C1 C1(CCC)CN(C(=O)C(C)OCC)CCN1C(=O)CCC(C)(C)F c1(CC#N)ccc(S(=O)(=O)N2CC3(C2)SCCC3C(=O)O)cc1 CC1(C)OC(=O)NC1C(=O)NC(C1CCOC1)C.c1(C=O)ccc2c(c1)CC2 C1(OC)CCc2ccccc2C1N(C)C(=O)NCCCCCCCN1CCCC1 N1(C(C2C(C)C2)=O)CCC2(C1)CN(C(C1(c3ccc(Br)cc3)CC1)=O)C2 C1(C(N2C(C)(C(=O)NCCc3scc(C)n3)CCC2)=O)CCC2(CCC2)C1 C1(CC)CN(C(=O)CC2(OC)CC2)CCC1N=c1[nH]c2cccc(Br)c2o1 N1(C(Cc2c(C)nc(SC(F)(F)F)cc2)=O)CCn2ncc(SC(F)F)c2C1 c1(OC)nc(NC2CCN(C(=O)C3=CCCC3)CC2C)nc2[nH]cnc12 c1(-c2cn(C(C)C(=O)N(C)Cc3cnn(C)c3)nn2)ccc2ncccc2c1 C#CCCCC(C)C(=O)N(C)CCN(C(=O)C(O)CSc1ccccc1)C C(=O)(CCC(C)(C)C#N)NC1CCC(CN(C(C2CC(C)N(C)CC2)=O)C)CC1 C1(CN(C(c2ccc(F)cc2)CO)C)(CO)CC12CCOCC2 c1(OC)cc(C(N2CCN(C(=O)C=CC(C)C)CC(O)C2)=O)cc2ccoc12 C12(c3nnc(CC(n4ccnc4)C)o3)CCC(CC1)C2(C)C CCC(CC)C(C(=O)NC1CCC(NC(=O)CCOc2cccnc2)CC1)OC N1(C(C(C)NC(COC)=O)=O)CCOC(CC(=O)NC(c2ccsc2)(C)C)C1 C1(C(N2CC(C)N(C(=O)CCc3cnn[nH]3)CC2)=O)CC(c2ccccc2)=NO1 N1(C(c2ccn(C)n2)=O)CC2CS(=O)(=O)CC2C1.C(=O)(CCC(C)(C)[N+](=O)[O-])N C1(C(N2CC(CNC(C3N(C)CCOC3)=O)C2)=O)CCc2[nH]nc(O)c2C1 CC1CCN(C(=O)C(C2CCCCCC2)O)CCN1C(c1cn2c(n1)CCC2)=O C(CC(C(C)(C)C)NC(=O)Cc1c[nH]nc1O)N(C(C(C=C)(F)F)=O)C N1(C(CC2N(C(C(C)Cn3ccnc3)=O)CCOC2)=O)CC(N(C)C)C2(CC2)C1 C12(NC(CCN(C(CCC)C)C)=O)CCCC(NC(c3nocc3C)=O)(C1)C2 C(=O)(CC(C)C1CCCCC1)NCC1C(NC(C2CC(=C)C2)=O)CC1 c1(C(=O)NC2C(C(N3C(C(C)(C)OC)CCC3)=O)OCC2)ccnc(C)c1 C(C)(CO)(CCF)NC(CCN(C(=O)CC1CCC1)C(C)C)=O C(=O)(C(C)CCCC)N1C(CC(N2CC(O)(CCC)C2)=O)CCC1 N1(C(C=CC(C)C)=O)CCC(O)(CCNC(=O)C(F)=CC2CC2)C1 N1(C(CCCNC(C)=O)=O)CC(NC(C2(C)CC(F)(F)C2)=O)C(C)(C)C1 C1(C(N(C2CCOCC2)C)=O)CC12CCN(C(C1CC(O)C1)=O)C2 n1(CC(N2CC(CCNC(C3C(C=C)C3)=O)C2)=O)cc(CN(C)C)nn1 c1(C(=O)NC2CCC(N(C)C(c3ccncc3N)=O)C2)coc2c1CS(=O)(=O)C2 CCCCC(C)CCC(=O)NCC1CN(C(=O)C2=CSCCO2)C1 C(C)(C(=O)NCCCN(C(=O)C)CC1CC1)SC.c1(C=O)ccsc1 C(CCC(C)(C)C(=O)NC(CC(=O)N1CCCOC(C(C)C)C1)CC(C)C)OC C1(CC)CN(Cc2ccc(OC)c(O)c2)CCN1C(=O)Cc1ccc(Br)nc1 S(=O)(=O)(c1cnc(NC(c2cn(C)nn2)C)c(Cl)c1)NC(CC)CC c1(OC)cccc(F)c1C(=O)NC1CCN(C(=O)CC2(C)CCCC2)C1 CCCCCCC(=O)NC1(CNC(c2cnn(C)c2COC)=O)CCCC1 c1(C(N2CC3(C2)CN(C(c2cc(Cl)ccc2F)=O)C3)=O)ccc2[nH]ccc2c1 C(CCCCNC(=O)CC(C)n1cc(Br)cn1)NC(C(C)C1CCC1)=O CC(CC(C)(F)F)C(=O)NCC1COCCN(C(c2cccc(O)c2F)=O)C1 C(=O)(C1=NN(CCO)C(=O)CC1)NCC#CCNC(C(CCS(C)=O)O)=O c1(NC(=O)NCc2cnc(N(C)C)s2)ccccc1F Cn1nnnc1C(c1cncn1C1CC1)NCC1=CCCC1 C1(CNC(=O)OC(C)(C)C)CC12CCC2.c1(C=O)occc1C1CC1.C CCC(C(=O)N(CC(O)CF)C)N(C(=O)C=C(C)C(C)C)C c1(-c2n(CCS(N)(=O)=O)nc(C3CCCO3)n2)noc2c1COCC2 C1(C(=O)NCCN(C)C(C)C)(CC)CCN(C(c2cc(CO)on2)=O)CC1 c1(C(N2CCN(C(c3c(C)nsc3N)=O)CC2)=O)cc2cccnc2[nH]1 N1(C(c2cc(N(C)C)nc(Cl)c2)=O)C2CCC1CC(NC(C1CCC(=O)N1)=O)C2 N1(C(C(CSC)O)=O)CCOCC1CC1CCN(C(c2ccnnc2O)=O)CC1 C1(C=O)CCC(=O)N(C)C1.C1(C(=O)N)CCN(C)C1.c1(CC)nccn1CC C(=O)(CCCCC(F)F)N1CC(CCC)N(C(c2ccc3ccnn3c2)=O)CC1 N(C1CN(C)Cc2ccccc21)C(N(C1C(OC)CC1)C)=O C1(C(N2CC(C)(NC(c3ccc[nH]3)=O)C2)=O)CCCN(C(N)=O)C1 N1(C(C(CCC)O)=O)CCC2(CCN(C(C3CCC(OC(F)F)CC3)=O)C2)C1 CC1OCCCC1C(=O)NCCN1CCN(C(=O)CC2OCCC2(C)C)CC1 C1CC2(CC2)CO1.C1(CC(=O)N(C)CC)CCS(=O)(=O)C1.CCCNC.C C1(NC(CSS(C)(=O)=O)=O)CCN(C(c2cc(C(N)=O)cs2)=O)CC1F C(=O)(C#CC1(C)CC1)N(CC(CN(C(c1cc(CC)no1)=O)C)O)C C1(CC(=O)NCC2N(CC)CCC2)CC2(CC2)CN1C(=O)C.CCCF.O N12CC(C(CC)C1)CNC(=O)C2=O.CCCCC(C)NS(C)(=O)=O C1(CCNC(CCCOCCC)=O)CCCN(C(=O)CC(C)SC)C1 C1(NC(c2cc(N)cc(O)n2)=O)CC2CC(NC(C3CC4CC4C3)=O)CC2C1 C1(CCNC(CCC=CC)=O)CC(F)(F)CN1C(=O)C(c1c(F)cccc1F)C CCC(C(=O)OC)C(C)(F)F.N1(C(c2cn(C3CCCC3)nn2)=O)CCNC(=O)C1 c1(CNC(C(c2ccccc2)NC(c2c(C)c[nH]n2)=O)=O)cnccc1Cl N1(C(C(C)(C)O)=O)CCOC(C(=O)NCc2nccs2)CC1 c1(CNCC2(C(C)(F)F)CCOCC2)cnc2c(C#N)cnn2c1 c1(CC(=O)NC(C)C(CO)NC(=O)CC2CCSCC2)cc(Cl)ccc1Cl CCC(C)C(C(=O)N(C)CCC1CCN(C(=O)Cn2ncccc2=O)CC1)OC c1(C(c2n(Cc3cccc(OC)c3)nnn2)NCC(Cl)Cl)ccc2nsnc2c1 C1(NC(c2cn(C)nn2)=O)CC2(CCC(NC(c3ncccc3F)=O)CC2)C1 C1(NC(C(C)n2ccnc2)=O)CCC(C(=O)NCCCCN=[N+]=[N-])CC1 c1nn2cc1NC(c1nnnn1C1CCOCC1)CC2.C1(O)CCC1.C1CC1 C1(NC(C2(CCC=C)CC2)=O)CN(C(=O)Cc2ccn(C3CCCC3)n2)CC1O C1(C(=O)NC2(CO)CCN(C(C(C)(C)F)=O)C2)CN(CP(C)(C)=O)C1 c1(OC)cc(CNC(=O)Nc2ccccc2Oc2ccncc2)cnc1OC CC(CO)(C(=O)NCC(O)C1CC1)NC(c1ccc(CO)o1)=O c1(N(C(C2CCCNC2)C)Cc2c(Cl)ccc(F)c2F)ncc2ccccc2n1 C1(C(=O)NC(CCCC)CNC(=O)Cc2ccn(C)n2)COC2COCC12 c1(C(N2CC3CC3(C(=O)NC3(c4ccccc4)COC3)C2)=O)cnc2ccoc2c1 C1(CC)CCC(CNC(=O)CCN(C(=O)CC2COC(=O)C2)CC)CC1 CC1(CC(=O)NCCC2(C(=O)NC34CCCCC3C4)CCC2)CCCCC1 C(=O)(C(=O)N=c1cc(C)o[nH]1)NCC1CCCN(c2nc(OC)nc(OC)n2)C1 N1(C(C(C)CNC(C2CC23CCC3)=O)=O)CC(C2CC2(F)F)C1 CN(C)S(=O)(=O)N1CCC(C(=O)NC)C1.C1CCCCN1C(C1CC=CCC1)=O N1(CC(=O)NC2(CCNC(c3c(C)ocn3)=O)CCCC2)CC2C=CC1C2 C1(C2CCN(C(c3cnc(O)s3)=O)C2)(NC(C(COC)C)=O)CC1 Cc1ccc(F)c(C(=O)NC2CC(CNC(C3(O)CCC3)=O)C2)c1O C12(C(N3CCC(C(F)F)C3)=O)CC1COC2(C)C.c1(CC)ncc(C(=O)N)[nH]1 C1(C(=O)NC(C2CCN(C(CC(CC)C)=O)CC2)(C)C)CC2(C1)CC21CC1 C1(C(=O)NC2(C)CCN(C(C(n3cc(C4CC4)nn3)C)=O)C2)(OC)CCCCCC1 c1(C(C)(C)C)nc2ccc(NC(=O)NC(c3ccccc3)(C)CO)cc2s1 C(=O)(CCS(=O)(=O)C1CCCC1)NC1CN(C(C2C(CC)C2)=O)CC(C)(C)C1 c1(CC)ccc(C(=O)NCC=CCNC(C2CC2C)=O)c(N)c1 N1(C(C(CC)(F)F)=O)CCC2(CCCCC2NC(c2occ3c2CCCC3)=O)C1 CC1(C)CCC(CO)N(C(c2c(Cl)cc(Cl)cc2Cl)=O)C1 C12(C(=O)NCC3CN(C(c4c(C)[nH]cc4)=O)C(C)C3)CCC(N=[N+]=[N-])(CC1)C2 N1(C(c2ncn(C(C)C)n2)=O)CCC2(CCC2CNC(=O)C(C)(F)F)CC1 c1(C(=O)NCCNC(C(C)OCOC)=O)cnc2n[nH]c(C)c2c1 C1(N(C(=O)C(CCSC)OC)CC)CCCN(C(C)Cc2cccs2)CC1 Cc1ccc(C(N2CCC(CCC(=O)NC3(CO)CC(O)C3)C2)=O)c(C)n1 N1(CC(=O)N(C2CCN(C(C(C)C)=O)C2)C)C(=O)NC2(CCCCC2)C1=O.CO Cc1c(C(=O)NCCCN(C)C(c2cccc(CO)c2)=O)nn2ccccc12 c1(-c2cccc(N(C)C)c2)ccc2c(c1C(=O)NCc1ccc(C#N)s1)OCO2 C(C)(C(=O)N(C(C)C(=O)NCCCCC1CC1C)C1CC1)OC(C)=O c1(C(=O)NCC#CCNC(CCCOC)=O)csc2ccccc12 C(=O)(CCCCCNC(=O)CC=CC(C)(C)C)NC(C)CC1CCCO1 N1(C(c2ccc(OC)nc2)=O)CC(C)CN(C(c2ncc(C)cc2C)=O)CC1C C1(C(=O)NCCC2N(C(c3c(C)nn(C)n3)=O)CCSC2)CCOC(C)(C)C1 Cc1cc(C(=O)NCc2cc(C(=O)N(C)CC3CC3C)cs2)ccc1F c1(CC)ccc(CC)cc1.c1(CC=O)nnc(C)o1.C(=O)CN(C)C(N)=O N1(C(C(CCCC)O)=O)CCC(C2CN(C(=O)CCC(C)CN(C)C)C2)CC1 Cc1nn(C)c(C)c1CC(C)C(=O)NC1CN(C(c2csnn2)=O)C1 C1(NC(C=C(C)C(C)(C)C)=O)CCN(C(C2C3CC4C(C3)C24)=O)C(C)C1 N1(C(c2c(Cl)cccc2Cl)=O)CCCCCC(NC(C2(F)CC=CCC2)=O)C1 C1(NC(C(CCC)NC(N)=O)=O)CCN(c2nc(C)ns2)CC(C)(C)C1.C1CC1 C1(CN=c2cc(C3CC3)nc[nH]2)(OCCC(F)(F)F)CC2CCC1CC2 N1(C(C(=O)NCC(c2ccccn2)C)=O)CCn2nnnc2C1 C1(C(N2CC(C)(CC)OCC2)=O)CC2(CCN1C(c1ccco1)=O)CC2 C(=O)(C(C)CC(=O)NC1CC(C)C1)OC.c1(C=O)cccc(-n2cccn2)c1.N CC1(C)CC(C)(CNC(=O)C2=CCCCC2)CN1C(=O)CCCC1CC1 C(=O)(CC1CCCc2ccccc21)NCC1CN(C(C(CC)C)=O)C1 c1(NC(C2CCCN2Cc2cccnc2F)=O)cc([N+](=O)[O-])ccc1F N1(C(Cc2cc(C)cc(F)c2)=O)CC2(C1)SCCC2NC(C12CC(C)C1C2)=O C1(OC)(CNC(C2(c3ccncc3)CC2)=O)CN(C(c2cnnn2C)=O)C1 c1(C(=O)NCC2CC3(CN(C(C(C)(CO)OC)=O)C3)C2)cnc2ccccn12 C1(C(N2CCOC(CO)C2)=O)COC2(CCN(Cc3ccnc(Cl)c3Cl)CC2)C1 CC1Oc2ccccc2N(CC(=O)CCOC(=O)CN(C)C)C1=O c1(C(N2CC3C(CNCc4c(O)ccc(C)c4)(C3)C2)=O)cc(Br)cc(Cl)c1F N1(C(C(C)(C)C#N)=O)CCOCC1(C)c1cn(-c2ccc(Cl)nc2)nn1 C1(CNC(c2nc(C(C)=O)sc2)=O)N(C(c2c[nH]c(=N)s2)=O)CCCC1(C)C c1(C(N2CC(NC(c3c[nH]cc3C3CC3)=O)C(F)C2)=O)cccc2[nH]ccc12 N1(C(CC=CCCCCC)=O)CCC2C(CCN2C(C2CC2C(F)(F)F)=O)C1 C1(OC)CCCC1C(=O)NC1(C)CC(NC(=O)C(C)N2CCCC2)C1 N1(C(c2cccc(CC(C)C)c2)=O)CC2CCC1CN(C(=O)CCOC(C)C)C2 C1(C(NOCC(CC)C)=O)CCN(C(=O)CCC2CC2(C)C)C12CC2 CCC(CNC(=O)C(F)(F)c1ccccc1)(CC)NC(C1CC12CC2(F)F)=O CC#CCCCC(=O)N1CC(N(C)C(C2CCC(C(F)(F)F)CC2)=O)C1 N1(C(C(CC2CC2)NC(=O)CCCC2CC2)=O)CC([N+](=O)[O-])C1 CC#CCC(CO)NC(=O)CCN(C(=O)Cn1nccc1C)C1CC1 C#CCCCC(=O)NCCOCCN(C)C(c1oc(CCC)nc1C)=O C(C(=O)N1CCC(CN(C(=O)CC2(N(C)C)CCCCC2)C)C1)(C(C)C)SC c1(NCC(CO)OC)ccc(S(=O)(=O)N2CCCC2C2CC2)cc1F N1(C(C(N)=O)=O)CCCOC(CCNC(c2ncn3c2CCC3)=O)C1 C1(C(=O)NCC2(NC(C3CC(C)OCC3)=O)CC2)CCc2nncn2CC1 C(CS(=O)(=O)CC(=O)NC1CC(CC)C1)OC.C(=O)(CCC)N.C(C)(C)C C1(C(N2CC3(CN(C(C(COC)O)=O)C3)C2)=O)CC2CC(O)CC(C1)C2 N1(C(c2ccncc2F)C(=O)NCCSC)CCSC2CCCC12 C(=O)(C1COc2ccc(Cl)cc21)N(CCNC(=O)C(O)CCSC)CC C1(NC(C(CNC(c2c(CC)noc2)=O)N(C)C)=O)C=CCCC1CO C(=O)(C1=CS(=O)CCC1)NC1COCCN(C(C(C)n2cncn2)=O)C1 C#Cc1ccnc(C(N2CCCCC2C(=O)NCC(O)CCOC)=O)c1 Cc1ccc(C=CC(=O)NCc2ccc(C(=O)NC3(CF)CC3)o2)o1 C1(CNC(C(C)NC(=O)CN=[N+]=[N-])=O)CCS(=O)CC1 c1(C(C(=O)NCCCOC)N(CCC)C)ccc(Cl)cc1C C(CC(O)CC(=O)NCCC1CCCN(C(=O)C(=O)NCC(F)F)CC1)SC N1(C(c2c(C)nn(C)c2)=O)CC2CC(O)C1C2NC(c1ccc2nccn2c1)=O C(CS(=O)(=O)C(F)F)NC(C1CCC(c2onc(-c3cc(C)oc3C)n2)CC1)=O c1(C(N2CCC(C3CCOC3)C2)=O)c(Br)sc2ccccc12 C(=O)(CCCn1ccnn1)NC1(CN(C(C(C)C2CCOC2)=O)C)CC1 NC(=O)CC(O)C(=O)NCCN1CCCN(C(=O)CCN2CCCS2(=O)=O)CC1 c1(OC)ccc(C2CCN(C(c3nnc(SCc4ccccc4)s3)=O)C2)cc1 Cc1cccc2c1OC(C(=O)NC1CC(C)(NC(c3oc(Br)nc3C)=O)C1)C2 c1(C(C)C)[nH]nc(C(=O)NCC#CCNC(=O)C2=CCCS2)c1[N+](=O)[O-] c1(C(N2CC(C(C)NC(COCCCC#C)=O)C2)=O)cncc(NC)n1 CC(C)CC(C(=O)NC12CCC(C1)N(C(=O)CC1CSC1)C2)N(C)C C1(C)(C(=O)NCCC=C)CCCN(C(c2ccc(C)cc2Cl)=O)C1 C12(CNC(c3c(C)oc(CO)c3)=O)CCC1CCN2C(c1csc(C)c1C)=O N1(C(C(CC)OC2CCCCC2)=O)CCC(NC(C2(C)CC(F)(F)C2)=O)C(O)C1 C(CC(C(C)C)NC(c1nccnc1C)=O)N(C(CCNS(CC)(=O)=O)=O)C CC(C)(C)[Si](C)(C)OC(CNC(C#N)C(N)=O)CF c1(NC(C2C3CN(C(C(CC)=O)=O)CC32)=O)c(Cl)cc(F)cc1Cl C1(OC)CC(C(=O)NC(C23CC(CO2)C3)C)N(C(=O)CCn2cnnn2)C1 S(=O)(=O)(c1ccccc1Cl)NCC1CN(S(=O)(=O)C2CC2)CC1(F)F c1(OC)ccc(Cl)cc1C(N1CC(NC(=O)C=Cc2ncco2)CC(C)C1)=O C1(C(N(CC#C)CC#C)=O)CCN(C(C2CCCCC(=O)N2)=O)CCO1 C1(CC)CC(C(=O)Nn2cccn2)CCN1C(C1CCC(CC)CC1)=O N(C1CCCc2c(F)cc(F)cc21)C(c1cc(C)n(C)n1)Cc1ccccc1 C(=O)(C(CC(C)C)C(C)C)N1CC2N(C(C(CC)SC)=O)C(CC2)C1 C(CC(O)C(=O)NCCC1CCCN(c2nccc(OC(C)C)n2)C1)OC Cc1cc(C(N2CC=CC2CNC(=O)CCS(N)(=O)=O)=O)c(C)cn1 c1(C(=O)NC2CCN(C(=O)OC)C2)cnc(C)nc1O.N12CCCC(C1)CC2=O C1(NC(C=CC(N)=O)=O)CCCC12CN(C(=O)CCc1cc3ccccc3o1)C2 c1(OC)cccnc1C(N1CCC(C(C)Nc2ncnc(C(C)(C)C)n2)C1)=O N1(C(c2nccc(CNC(CC(C)n3ccnc3)=O)c2)=O)CC2C=CCC(C2)C1 C1(C(=O)NC(CNC(CC=C(C)C)=O)C(C)C)CC2C=CCC(C1)C2 c1(C(N2CCN(C(=O)CC3CC=CCC3)C(C3CC3)C2)=O)ccc2nncn2c1 c1(C(=O)NCC(CC)NC(c2snnc2C2CC2)=O)ccc(C(C)=O)o1 N1(C(CC2N(C)CCOC2)=O)CC(C2CN(C(=O)Cc3cncnc3)C2)C1 c1(C=O)ccc2c(c1)C=CCC2.N1(C(C(C2CCC2)OCC)=O)CCC(C)C1.N c1(OC)cc(C2CCCN(Cc3cc(C(C)=O)ccc3O)C2)ccc1C c1(CNC(CCC2(NC(c3c(CC)noc3)=O)CCCC2)=O)cc(C)cnc1O C1(CNC(=O)CCc2ccc(Cl)cc2)(CO)CC2C=CC1C2 Cc1ncc(Cl)c(C(=O)NCCC(C(C)C)NC(C2CCCOC2)=O)n1 CC1CC2CN(C(C3CC3(C)C)=O)CC2N1C(C1CCc2nnn(C)c2C1)=O C(C)(CC(C)C#N)c1n(CCCC(=O)OCC)nnn1.C1CC2(C1)CC(C)C2.N C1(NC(CN(C(C2C(=C)C2)=O)CC)=O)CCCN(CCO)C1 N1(C(C(CCSC)O)=O)C2CCC1CC(N(C(=O)C(F)CC(C)(C)C)C)C2 C12CC(C)C1C2.C1CCCN1C(C1(C=O)CCC1)=O.C(C=O)NC(C)=O.N c1(C(=O)N)cccc2nc(C(F)F)sc12.Cc1ccc(C(=O)NC2CC2)c(O)c1 c1(SCC(c2cn(CC)nc2C)=O)cn(C)c2c(C)cccc12 c1ccc(Cl)c(F)c1.C1(O)(C(C)NC(=O)CF)CCN(C(C2(C)CC2)=O)C1 N(C1CCSc2ccc(Cl)cc21)c1c(C)c(F)ccc1 C1(NC(CC=C=C)=O)CCCCC12CCN(C(c1cn(C(C)(C)C)cn1)=O)C2 C=CCC(C)(O)C(=O)N1CCCN(CCNC(=O)CCCC(=O)NCC)CC1 N1(C(c2c(NC)nccc2)=O)CC2CCC(NC(=O)C(F)CC3CCCC3)(C2)C1 C(CCCCC(=O)NCC1CCCCCC1)N(C(=O)CC1CCOC1)C CC1(C)CCN(C(C2CCCCC(=O)C2)=O)C1CC(=O)NC1COCC1N=[N+]=[N-] c1(CCOCC(=O)NCC2CC(F)C2)cc(Cl)ccc1Cl c1(N2CCC(F)(CC)C2)nc(N2CCCC(N(C)C)C2)nc2cc(OC)ccc12 CCC(CNC(=O)C(c1cnn(C)c1)NC(c1cc(F)n(C)n1)=O)C(C)C n1(CCCCC)cc(NC(=O)CONC(=O)CC2CCCO2)nn1 c1(NC(C2C3CCC23c2ccccc2)=O)cccc2c1CN(Cc1ccccc1)C2 C1(C(=O)NC2CC(CCNC(=O)C=C(Cl)Cl)C2)CC12CCC1(CC1)CC2 C1(CC(=O)NCCC(C(C)C)O)C2CCCC2N1C(C1(F)CC=CCC1)=O CCCCCCCCS(=O)(=O)NCC1CNCCC1(C)C CC1CCN(C(C2CC(O)C2)=O)C1C(=O)Nc1ccc[n+]([O-])c1 C(Cc1ccccc1)(CCc1nn[nH]n1)NC(C1(C)CC1F)=O CN(C1c2ccccc2CC1O)C(=O)NCCc1ccncc1Br C1(F)(CNC(CC2(C)CCCO2)=O)CCCN(C(C2COC2)=O)C1 C(=O)(CC(C)(C)C(F)(F)F)NCCOCCCNC(C1OCC(C)C1)=O c1(C(=O)NC(CC=C)CNC(=O)C(C)c2cccs2)cncc(C(C)C)c1 C(C(O)CN=c1ccc(C(F)(F)F)n[nH]1)NC(C1(CC#C)CCCCC1)=O CC(CC(C)NC(C1CCCOC1)=O)NC(c1csc(-c2nc[nH]n2)n1)=O C1(C(N(C(C)C(N2CCCCC2C)=O)CCC)=O)CC(=O)OC1(C)C C1(CNC(CSCC)=O)CCC2(CCC2)CN1C(=O)Cc1n[nH]c(=N)s1 CC1(C(=O)NC2CC23CCC3)CCN(C(=O)CC2CCCC(O)C2)CC1 c1(C(=O)NC(C)C(CO)NC(c2cnsc2)=O)c(Cl)n[nH]c1C1CC1 c1(C(N(CCNC(C(F)=CC)=O)C)=O)ccc(CN(C)C)cc1 C1(CNC(c2c(OC)n[nH]c2)=O)CCCC(NC(=O)Cc2ccccc2)C1 c1(C(N(CC#N)CC)=O)c[nH]c2cccc(C3=CCCCC3)c12 C1(CNC(Cn2c(C)cnc2)=O)CC1C1CCCN(c2nnc(C3CC3)o2)C1 N1(C(c2cc3cccn3cn2)=O)CCCC(C2CN(C(C3CCC4CC34)=O)C2)C1 N1(C(c2ccc(C)c(F)c2N)=O)CCCC12CCN(C(c1cnoc1C)=O)CC2 N1(C(CC2CCN(OC)CC2)=O)CCN(C(c2ccns2)=O)CCC1C c1oc(C)cc1C(N1CCC(C)C1)=O.C1(C=O)CCN(S(C)(=O)=O)CC1.CC c1(-c2ccco2)ccc(Cl)cc1.CC(CC(=O)O)NC(=O)CN(C(=O)CS)C S(=O)(=O)(c1cccc(F)c1)NC1(C#N)CCN(Cc2ccc(Br)c(O)c2)C1 N1(C(C(CC)N(C)C)=O)CCN(C(=O)Cn2cccc(C)c2=O)C2(CC2)C1 Cc1nn(C)c(-n2cncn2)c1C(=O)NCCCCOC(C)C c1(OC)cc(NNC(=O)C2(C)CC2F)ccc1[N+](=O)[O-] CC1CN(C(=O)CCc2cnccn2)CC1CNC(C1OCCCO1)=O C(N=c1[nH]c(=NC2CCCN(CCF)C2)[nH]c2ccsc12)C1(C)CCCC1(F)F C(C)(C)(CCCCNC(c1ccc(Cl)s1)=O)NC(COC(C)=O)=O C1(CNC(c2ccsc2C(F)F)=O)CC2COCC2N1C(c1cccnc1F)=O CC(C)C(C)C(=O)NCC1C2CN(c3nnc(C(C)(C)C)o3)CC12 C1(NC(c2cc(C)cc(C)n2)=O)CS(=O)(=O)C12CCN(C(=O)CC1CC1)CC2 c1(C(N(C2CN(C(c3cncnc3)=O)CC2(C)C)C)=O)cccc2nc(O)[nH]c12 N1(C(C(CSC)O)=O)CCCC12CCCN(C(c1csc(Cl)n1)=O)C2 C1(NC(C=CC)=O)CC(F)CN(C(c2ccc(OCC(F)F)cc2)=O)C1 C1(C(N2CCC2)=O)CCC(CC(F)(F)F)CC1.c1(C(=O)N)cnc(C2CC2)o1 C1(NC(c2nncc(OC)c2)=O)CCC(O)CN(C(c2ccc[n+]([O-])c2)=O)C1 [SH](=O)(=O)c1cccc(C=O)c1.c1(CC=O)cnco1.C(C)C1CC1.CCN C(C(C)(C)CC(=O)N(CC1CC1)OC)NC(c1ccc(C)c(C#N)c1)=O N1(C(c2c(CC)nn[nH]2)=O)CCCCCC(NC(c2conc2C(C)C)=O)C1 N1(C(CNC(CC)=O)=O)CC2CC1CC2NC(=O)C=C1CCC(C)(C)CC1 Cc1nn(C)c(C)c1CC(N1CCC2(CC2)C1)=O.C1(C(=O)N)COC2(CCC2)C1 C(CCCCC(=O)NCC(C)N(C)C(C1CC2(CCCO2)C1)=O)OCC N1(C(C=CS(C)=O)=O)CCCC(C2(NC(c3ccc(C(F)F)cc3Cl)=O)CC2)C1 n1(CC(=O)NC23CCN(C(C(=O)N(C)C)=O)CC2C3)nnc2ccccc2c1=O CCCCC(O)C(C)C(=O)N1CC(CNC(=O)CCN2CCCC2)OC(C)(C)C1 c1(C(=O)NCCN(C(CC(CC)SC)=O)C)ccc2c(c1)C(CC)C(=O)N2 N1(C(C2N(C(C)C)CCCC2)=O)CC2CCC1CN2C(C1CCC2(CC2)C1)=O C12(C(N3C(CNC(Cc4nc(CC)sc4)=O)CCCC3)=O)CCC(F)C1CC2 CC1ON=C(C(=O)N2CC3(CCN3C(=O)CC3CCCNC(=O)C3)C2)C1C CC1(C)COC(=O)C1n1cc(C2CCCN(C(=O)Cn3cnnn3)CC2)nn1 C1(CNC(CC)C(=O)Nc2nc(C)cs2)CCN(C(=O)CNCC)CC1.C c1(C(=O)NC2CN(C(C3(OC)CC(CF)C3)=O)CC2C)cccc2c1CNC2=O C1(C(N(C)CCN(C)C2CC2)=O)CSCCN1C(=O)C(O)CN(C)C N1(C(C(C)(CO)NC(C(C)=C(C)C)=O)=O)CCCC(C)(N(C)C)C1 N1(C(CCOC)=O)CC(=O)NC2CN(C(=O)CCN3CCP(C)(=O)CC3)CCC12 C(C)(N=c1nc(N2CCC(=C(F)F)CC2)c2cc(OC)ccc2[nH]1)C1C(CC)C1 c1(OC)cccc(C(=O)NC2CN(C(c3ncc(C)cn3)=O)CC2SC)n1 C1(OC)CC(OC(C)(C)C)CN(C(=O)NCC2CC3(C2)CC3(F)F)C1 C(=O)(C(CO)C(F)(F)F)NC(C(=O)N1CCC(C(=O)OC)C1)(C)CO C1(CC(N2CC3C(Nc4cc(SC)ncc4)(C3)C2)=O)CCCCC1(F)F c1(-n2cc(CC(=O)N(C3CCN(C(C=CCOC)=O)C3)C)nn2)ccccc1C C(CSC)(C(=O)NC(Cc1cc[nH]n1)C(=O)NC1CCCOC1)OC CC(C)C(O)CC(=O)NCC(C)NC(c1cc(Br)cs1)=O C1(NC(c2ccc(C(F)(F)F)s2)=O)CC(N=c2[nH]ncs2)C12CCC2 Cc1nc(NCC2CCCO2)cc(=NCc2cnccc2C)[nH]1 c1(CC)nn(C2CC2)cc1C(N1CCC(O)(C(C)C)C1)=O.C(=O)C(C)(C)C N1(C(C(CCC)OC)=O)CCN(C(C2(CCF)CCC2)=O)CC(C)(F)C1 C1(C(=O)O)CCC(NCCOc2ncccc2C(F)(F)F)C(O)C1 c1(CN2CCC(F)(C(=O)NC(C(F)(F)F)C3CC3)C2)cccc(F)c1Br C1(C(=O)N)COCCN1C(=O)CSC1CC1.C1CCC(O)CC1 N1(C(CCNC(N)=O)=O)CC2COCC(C1)C2NC(=O)Cc1c(F)cccc1F CC(C)C(O)C(C)(C)CNC(=O)C(=O)Nc1cccc(C(C)N)c1 CCCCC(CNC(c1ccnn1C(C)C)=O)NC(C1CCC(C)CC1)=O C1(C(=O)NCC2CCN(C(=O)C(c3cncnc3)C)C2)(CC)CNC(=O)C1 N1(C(=O)Cc2cnc[nH]2)CC(CNC(C2CC(O)C2)=O)C2(CC2)C1 CC(C)CC(C)CC(=O)NCC1CC1CC(=O)N(CC(C)C#N)C C(=O)(C1=CC2(CCN(C(c3oc(C)cc3C)=O)C2)C1)NCCSCC#C c1(C(N(CC(CC)NC(=O)C(O)C(F)F)C)=O)sc2cccc(F)c2c1Cl C12(OC)CCC(C(=O)N)(CC1)CC2.C1CC2CCCC12.C(=O)C(C)=CC1CC1 C1(C=O)C(C2CC2)C1(F)F.CC1(C)COC(CCC(N2CC(F)CC2C)=O)C1.N c1(C(C)NC(C2CC(N)C2)=O)c(C)cc(C)cc1N.C1(C2CCCO2)CCOC1 CC(CC)CCCC.C1(C=O)(CNC(c2c(CCC)nco2)=O)CC(C)(C)C1.N Cn1nc(Br)c2c(NCC3CC(NC(=O)C)C3)ncnc12.N1(C=O)CCCC1 c1(-n2cc(CN(C(c3ccc(C(N)=O)o3)=O)CCF)nn2)ccccc1N C1(OC)(CNC(c2ccc(CN=[N+]=[N-])cc2)=O)CCN(C(=O)CCC#N)CC1 Cc1cnc(NCc2cnccc2C)c(S(=O)(=O)NCC(N2CCOCC2)C)c1 CN1CC2CC1(C)C2.C1(CC(=O)N)CCCC1.C1(C=O)CC(N(C)CCO)C1 N1(C(CN(c2ccccc2)C(C)=O)=O)CCN(C)C(CNC)C1.c1cnccc1Cl C1(C(=O)NCC(C)(C)N(C)C)COCCC1NC(=O)CC1(C)CCOCC1 c1(C(=O)NC2C(C)CN(C(=O)CN3CC(=O)NC3=O)C2)csc2ccccc12 Cc1cc(Br)cc(Br)c1NC(C1COCCN1C(c1ccc(F)c(F)c1F)=O)=O C1(NC(=O)CCc2ncco2)CCC(CNC(c2ccc(C3CC3)o2)=O)C1 CC1CN(C(=O)Cn2cnnc2O)CC1NC(=O)CC1COC(=O)N1 C1(CNC(CN2C(C)CCC2)=O)CN(C(C2OCCC2(C)C)=O)CC12CC2 N1(C(C2CCCO2)=O)CC(C)(C)OC2(C1)CN(C(C1CC3(CCC3)C1)=O)C2.CC Cc1cc(=NCC(C)C(F)(F)F)[nH]c(=NCCOCC2CCCO2)[nH]1 C1(NC(C23N(C(CCNC(C)=O)=O)CCC2C3)=O)C2C=CC(C2)C1CO N1(C(CC2CN(C)C2)=O)CCCC(NC(=O)C2=COCCC2)C(F)C1 C1(CC(=O)N(C2CN(C(c3ccc[n+]([O-])c3)=O)C2)C)CCc2ccccc2C1 CC1C(NC(=O)C=Cc2cnc[nH]2)CCCN1C(C1CCS(=O)(=O)C1)=O CCC(C)CC(=O)N1CC(F)CC1COC(c1nc(-c2ccc(C)cc2)cs1)=O C1(C)(C=O)CC2CC2C1.C(=O)CC(C1CC1)C1CC1.CCNCC.CC C1(NC(C(C)(C2CCC2)NC(c2cc(C)c(F)cc2)=O)=O)CC2CC1CC21CC1 CC1CCN(C(C2CCCCS2)=O)C(C)C1NC(=O)CSCC1CCCCO1 Cc1ccc(CSCC(N2CC3CC2C3NC(C2CC2(Cl)Cl)=O)=O)cc1 CS(=N)(=O)C1CCN(C(C2CCCCN2O)=O)C1 C1(NC(c2cncc(OC)c2)=O)CN(C(=O)CCc2cnn(C)n2)CCC1CO c1(C(=O)NC(CN(C(c2n(CC#C)ccc2)=O)C)C)c(N)cc(Cl)cc1Cl C1(CC#C)(C(=O)O)CCN(C(=O)Nc2cc(Br)ccc2C(=O)OC)CC1 C1(CC(=O)NC2(CNC(c3ccc(CC)[nH]3)=O)CC2)C(=O)NN=C1C C(=O)(C(C)(CNC(=O)COC(=O)OC)CC)NCCOCC#C C1(CC)C(NC(=O)C=Cc2c(C)coc2C)CCCN1C(=O)CCC(CC)OC C(=O)(CC(C)(C)CC(=O)N1CCCCC(NC(=O)C#CC2CCC2)C1)OC C1(C(C)C(=O)NC2CC(C(C)O)C2)CCN(C(=O)Cc2cn[nH]c2)C1 C1(C(N2C(C(C)NC(c3c(C)noc3)=O)CCC2)=O)CCCN(S(N)(=O)=O)C1 N1(C(=O)CCc2ncc[nH]2)CC2CCC1CN2C(c1cccc2c1OCC2)=O C=CCCCC(C(=O)N1CC(NC(=O)CO)C1)NC(c1ccc2c(c1)CC2)=O N1(C(c2cn(C(C)C)nn2)C(=O)NC(CC)C)CCN(C(=O)N)CC1.C(C)C c1(C(C2CC2)NC(C)C(=O)N(c2ccccc2)C2CCOC2)ccccc1F Cc1c(CNC(C2CSCCN2C(=O)CCCN2CCCC2)=O)nnn1C C1(C2CCN(C)CC2)(C=O)CC1.C1(NC(Cc2nc(C)[nH]n2)=O)CC2(C1)CC2.N CS(=O)(=O)C1CCN(C(C2CSCCN2C(c2cc(Cl)cnc2O)=O)=O)CC1 N1(C(C2CC(C)C2)=O)CC(O)(C(C)NC(c2cc(CO)[nH]n2)=O)C1 c1(C(=O)NC(C)CN(C(=O)CC2CCN(C)C2=O)C)cnn2cnnc2c1 CCC1=NOC(C(=O)NCCCCCNC(c2occc2C(C)C)=O)C1 Cc1oncc1C(=O)NCC=O.C(CCN(C)C(C1CCO1)=O)c1cccs1.N CC1CCC=C1C(=O)NC(C(=O)NCc1nnnn1C)C1CCC1 C=C1CC(C(=O)NC(CC)CO)(CNC(=O)Cc2cn(CC)nn2)C1 C1(C(=O)NC2CCC(CC(=O)N)C2)(CC)CCCN1C(C1CC1C1CCC1)=O N1(C(CN(C(c2c(C)cc[nH]2)=O)C(C)C)=O)CC(C)(C)CCC1C CC1CC(NC(c2sncc2Br)=O)CCN1C(=O)COC(F)(F)F C1CCS(=O)(=O)C12CN(C(c1cc(S(N)(=O)=O)oc1C)=O)C2.C(C)(C=O)=C.C C1(OCC)CCCCC1.c12ccc(cc1)NC(=O)N2.C(C)C(=O)O.C=O.C C(=O)(CC(C)(C)C(F)F)N1CCC(C)(CCNC(c2c(C)ccc(C)n2)=O)C1 c1(C=O)cc(S(C)(=O)=O)cs1.C1(CC)CN(C(=O)CCc2cnc[nH]2)C1.CO N1(C(c2cc(CCC)[nH]n2)=O)CCCCC1CCC(=O)NCc1ccccc1Cl C1(C(=O)NCC2CCN(C(c3nc(N(C)C)oc3)=O)C2)CCCC1C1CC1 Cc1cc(-c2noc(C34CC3COC4(C)C)n2)cc(=O)n1C CC1CC(=O)NCCN1C(=O)COC1CCC1.c1(C(=O)N)cc([N+](=O)[O-])n[nH]1 C1(CNC(C(CCC#C)O)=O)N(C(c2cc(CC(C)C)on2)=O)CCCC1(C)C N1(C(C(C)N=[N+]=[N-])=O)CC2(CO)CC1(C(=O)NCC1CCC=CO1)C2 N1(C(c2c(C)nncc2)=O)CCC2(CCC2CNC(=O)CC(C)(F)F)CC1 c1(CN(C)CC2OCCO2)nc(-c2ccncc2Cl)n(C)n1 CCC(C)C(C(=O)NC(c1ccccc1O)C)N(C(=O)Cc1cn(C)cn1)C C(C(C)C(=O)NC1(C)CC(C(=O)NCC(c2cccs2)C)C1)OC C1(N(C(C2(CCC)CCC2)=O)CC)CCN(C(=O)COC(C)(C)C)C1 CCC(C)C(C(=O)N1CC(C)C(C)C1)NC(C)=O.C(=O)(C(CCO)N(C)C)N C1(C2CC2)(CNC(c2cc(C)[nH]n2)=O)CCN(c2nnc(C#N)s2)C1 O=S1(=O)CCC(NC(=NCc2ccc(Br)cc2)NC23CC(C2)C3)C1 C12CN(CCC1C)C(=O)N(c1ccccc1)CC(=O)N2.c1(OC)ccccc1F CCCC(CCCNC(=O)C(C)(C)CO)NC(=O)C(CC)NC(C)=O C1(N(C(c2ccccc2Cl)C)Cc2cnc(C3CC3)nc2)COC2(CCCCC2)C1 C1(CNC(CC(C)CF)=O)C2CCC(C2)N1C(=O)CN1CC(C)(C)C1 Cc1cc(C=CC(=O)N(C)CC2(C)CCCC2)on1.C(=O)CC.CC(C)C.N C1(CC)CCCC1(C)C(N1CCN(C(=O)CSc2cnccc2NC)CC1)=O N1(C(c2ccc(CSC)o2)=O)CCC(CC)CC1.C1(C=O)CCN(C(C)=O)C1 C1(NC(C(C)OCCC#C)=O)CCCN(C(c2ccc(OC)c(N)c2)=O)C1C N1(C(C2OCC(C)C2)=O)CCC(C2CC2)(CNC(=O)CCS(C)=O)C1 Cc1cccc(C(N2CCCC2(C)C(=O)NC(C(C)C)c2nc[nH]n2)=O)c1C#N N1(C(C(COC)OC)=O)CCn2c(CNC(c3cnc(O)cc3C)=O)nnc2C1 CC1N(C(c2csc(C(C)(C)C)n2)C(=O)NCCC2CC2)CCC1(C)C c1(C=O)cc2cncn2c(O)n1.C1(CC(C)NC(COCC)=O)CCCCC1.N C(=O)(C(CC(C)C)ONC(c1cnc(N)cn1)=O)NC(CC)CO Cc1nc2sccn2c1C(N1CCC(C(C)NC(C2(C)CC2)=O)CC1)=O S(=O)(=O)(c1ccccc1)NCC(C)NC(c1ccc(C)c(C(=O)O)c1)=O Cc1[nH]nc2ncc(C(N3CCN(C(c4coc(Cl)n4)=O)C(C)C3C)=O)cc12 c1(C(N2CC(CCCCNC(C(C(C)OC)O)=O)C2)=O)c(N)cc(C)cc1F C1(CC(=O)N)CCCS(=O)(=O)C1.c1(C(=O)NCCCC)cnn(C(C)C)c1 C1(C(=O)NCC(CC)N(C)C(c2sc(O)nc2C)=O)CCCC(=O)C1 C1CC2(CCC2O)C1.c1(CC)[nH]c(=N)sc1C(N1CCC(C(=O)NC)C1)=O c1(C(=O)NCC(CNC(CC(C)C)=O)(C)C)c(Cl)c2ccc(Cl)cc2n1C C1(C=O)C2CN(C(=O)CCC3CCCN3C(=O)CN3CCC(C)CC3)CC12.CO c1(NC(CCN(CC(C)O)C)=O)ccc(Br)c(F)c1 C1(C(=O)NC2CC(C)(NC(c3c(C)nc[nH]3)=O)C2)CCC(C2CC2)C1 Cc1nc(N2CCC(CC(C)NC(c3nsnc3O)=O)CC2)ccc1[N+](=O)[O-] N1(C(C(=O)NC(C(N)=O)C2CCC2)=O)CCCC(C(N)=O)(N(C)C)C1 c1(C(=O)NCC(CCOC)NC(c2ccnn2CC(F)F)=O)ccnc(C)c1 N1(C(C2(COC)COC2)=O)CCC(NC(=O)CS)C(C)C1.c1cccc[n+]1[O-] N1(C(C(CCC)C)=O)CCC(F)(CNC(c2c(C(F)(F)F)cccc2O)=O)CC1 C(=O)(CCC(=O)N1CCCCC1CNC(=O)CSCCC(F)(F)F)NC c12cccc(n1)C(C)OC1(CCOC1)N(C)C2C(=O)NCCSC.CC NS(=O)(=O)c1cccc(NC(C2CC2N)=O)c1.c1cccc(-c2ccco2)n1.C Cc1ncc(C(=O)NC(CNC(=O)C(C)C2CC2)C(C)C)s1 c1(C(=O)NC2(C3CN(C(c4cc(C)n(C)c4)=O)C3)CC2)[nH]nc2ncccc12 C1(C(N2CC3C(CNC(=O)CC4CC5C=CC4C5)(C3)C2)=O)CN2CCCN1CC2 C1C2CCC(C2)C1C(N1CCC(C)(C)CC1)=O.CC(C)CCOC(C)C(=O)N Cc1ccc2c(c1)SC(C(N1CCCC1C)=O)C2.C1(C=O)CC12CC(C)(C)C2.N N(C1CCNc2cc(F)ccc21)C(C1(C)CCNC1)=O CC(CC(=O)N)C(F)F.C1(C(=O)NOCC=CCCC(O)C(C)C)CC(O)C1 c1(-c2c(C(C)=O)cccc2)nc2c(s1)CN(Cc1c(Br)cccc1[N+](=O)[O-])CC2 N1(C(Cc2nc3scc(C)n3c2)=O)CCN(C(C2CSCCS2)=O)CC2(CC2)C1 C1(NC(C2CCC(=C)CC2)=O)CC2CC(C1)CN(C(c1cn(C)[nH]c1=N)=O)C2 Cn1ncc(C(=O)NCc2ccc(CNC(C3CC(C#N)C3)=O)cc2)c1Br CN1CCC(CC(=O)NCC2(F)CCN(C(C3(F)CC=CC3)=O)C2)C1=O N1(C(c2n(C=C)ncc2)=O)CCOC(C)(CNC(C2CC(=O)N(CC)C2)=O)C1 Cc1scc(NC(=O)NC2CCCN(c3ccccn3)C2)c1C1CC1 CCCCCC(CC)C(=O)N1CC2CC1(C(N1CC(O)CC1C(C)C)=O)C2 N1(C(C(CC)CC(F)(F)F)=O)Cc2ccccc2C(NC(=O)COC(C)=O)C1 CC1CN(C(C2CCN(C3CC3)C2=O)=O)CCCN1C(c1cncc(N)n1)=O c1(C(=O)NCCC2(CNC(C3(C)CC(F)C3)=O)CC2)cc(=O)cc[nH]1 C1(NC(c2c(OC)noc2C)=O)CCCN(C(c2nccnc2C)=O)CC1 C1(CNC(C(=O)N(CC(C)N)CC)=O)CCCCN1 c1(NC)cnncc1C(=O)NCc1ccsc1C=O.N1(CC)CCC(C)C1.N c1(C(N2CCN(C(c3ccc(N4CCCC4)nc3)=O)CC2)=O)cc2occc2[nH]1 C1(C)(CC(N2C(C(C)O)CC2)=O)CCN1C(=O)CN1CC=CC1 c1(CC(=O)NC2CN(C(C=CS(C)=O)=O)CC2O)ccc2c(c1)CCC2 N1(C(C(=O)NC(C)C)=O)CCC2(CCCC2)C1.c1(C=O)c(C(C)C)cnn1C.N N1(C(C2(NC(C3CCN(CC)CC3)=O)CC(O)C2)=O)CC2C(C1)C2(C)C C1(c2cn(CCOC)nn2)CCN(C(=O)C(c2cccc(Cl)c2)(F)F)C12CC2 C1(CC(=O)N(CCNC(C2(F)CCCC2)=O)CC)CCCC(=O)N1 c1(CC(=O)NCC(=O)OCCc2nc(C3CC3)cs2)ccc2c(c1)CCO2 C(=O)(C(C)(F)C(=O)OCC)Nc1cc(N2CCC(=C)CC2)ncn1 CC(=Cn1ccnn1)C(=O)N1CC2CCCC2(NC(c2csc(C(N)=O)n2)=O)C1 C1(C(=O)NCC(CNC(C=CC)=O)(C)C)CC2(C)CCCN2S1(=O)=O CCCC(CCC)C(=O)N1Cc2[nH]nc(C(N3CC(C4CC4)OC(C)C3)=O)c2C1 C(c1cncn1C)=CC(=O)N(C1CCN(C(=O)CC2CCC2(C)C)CC1)C Cn1ncc2c(C(=O)NC3CCC(C)CC3)cc(Br)cc12.C1(C=O)CC(=O)N1.N C(=O)(C1CCc2nccn21)N1CCC(OC)(CNC(=O)C2=C(C)CC2)CC1 N1(C(CNC(C)=O)=O)CCCC1C(=O)N(C1CN(C(=O)C(C)C2CC2)C1)C C1(C(=O)N)(CNC(C2CC3(CC3)C2)=O)CC2(CC2)C1.CC(F)(F)CO c1(C=O)cc2n(c1)CCS(=O)(=O)C2.O=C(C(=O)C(F)(F)F)NCC(O)C.N N1(C(C(CC)NC(C)=O)=O)CCN(C(=O)CCc2cc(C)cc(C)c2)CC1C C1(C(=O)NC(C2N(C(c3c(CC)ncs3)=O)CCC2)(C)C)CC(C2CCC2)C1 C1(CNC(c2cnn(CC)c2Cl)=O)CCN(C(c2cc(Cl)n[nH]2)=O)CC1O C(c1ccccc1Cl)=C(C)C(N1CCCC(C)C1CNC(c1nncs1)=O)=O c1(CC(N2CC(N(c3nc(C)cc(C(=O)NC)n3)C)C2)=O)cn2c(n1)CCCC2 C1(CO)CCC2(CC1)CCN(c1cc(N3CCC(c4nc[nH]n4)C3)ncn1)CC2 N1(C(c2[nH]cc(CC(C)C)c2)=O)CCN(C(=O)C2=CCC2)CC(CO)C1 C1(C(=O)NCCc2cccs2)CC2(CCN(C(C3CCCC3)=O)CC2)CO1 C1(C(=O)NCC2N(C(c3c(C)cc(C)s3)=O)CC2)CCc2ncnc(C)c2C1 C1(CNC(C(C)(c2ccccc2)NC(C)=O)=O)CC2CCCCN2C1 c1(OCc2scc(CN3CC(C(C)(F)F)OCC3)n2)ccc([N+](=O)[O-])cc1 C(N=c1nc2c(c[nH]1)CCCC2)C1OCC(CNC(=O)C=CC2CC2)C1 C(C(C(=O)N1CC(C)C(F)C1)C(C)C)NC(c1cccc(C)c1)=O C1(CC(=O)NCC2(C)CC2(F)F)CCCN(C(=O)CCc2cccs2)C1 c1(CC)ccc(C)cc1C(N1CCN(C(=O)C(CC)CCOC)C(C)C1)=O C1(C=O)COC2(CCC2)C1.c1(C(=O)NC2CC2)ccnc(N2CCOCC2)n1.C c1(C(=O)NC2CC(CNC(c3cc(C)c(Cl)cc3)=O)C2)cc2cc(O)ccc2[nH]1 N1(C(C(CCO)N(C)C)=O)CC(NC(C2(F)CC2)=O)CC1(C)C N1(C(C)=O)CCN(C(C2(C)CCN(C(c3ccc(C(N)=O)cc3)=O)C2)=O)CC1 CC(C)(CNC(=O)CCC1CCCC1)CC(F)F.C1(CC=O)COC(=O)C1.N C1(NC(c2c(C(C)C)cco2)=O)CN(C(c2cc(N)c(Cl)cn2)=O)CCC1C O=S(=O)(c1ccc(NCCOc2ccccc2Br)cc1Cl)N1CC=CC(O)C1 c1(CNC(=O)NCc2cc3cc(F)ccc3[nH]2)cc(Cl)c(Br)cc1F N1(C(C=CC(C)(C)C)=O)CC2CCCC2(C(=O)NC2CCN(C(N)=O)CC2)C1 C12(NC(c3c(C)cc(Br)o3)=O)CCN(C(c3ccncc3F)=O)CCC1C2 N1(C(c2ncc(OC)cn2)=O)CCC(C)N(C(=O)Cc2ccc(Cl)cn2)CC1 c1(C(N(C2CCN(CC)C2)CC)=O)nccc2[nH]ccc12 Cn1nc(C(=O)NCC2(O)CCN(C(=O)Cn3ncc(Br)n3)C2)cc1O CC(C)C(C#N)C(=O)N1CC(O)(C(F)C(N2CCC(F)CC2)=O)C1 N1(C(CCc2cncc(C)c2)=O)CC2(C1)CN(C(=O)CN1CCC(C)C1)CCO2 C(C(C)C)(C(O)C(=O)N1CC2(C(=O)NC3CC(CF)C3)CC1CCO2)OC C=CCCCC(=O)NC(C1CCN(C(=O)CCC2CCOC2)C1)(C)C N1(CCC(=O)NC(C2(C(N(C3CC3)CC)=O)CC2)C)CCCC1=O Cc1scc(C(N2CCCC2CCCNC(=O)C=CC2CC2)=O)c1C c1(NCc2n(CCC)ncn2)[nH]c(=NCC(CC(C)C)NCC)nc2scnc12 CC(c1cccnc1)=CC(=O)NCC1(C)CCN(C(=O)C(C)N(C)C)C1 N1(C(C=C(CC)CC)=O)CC2CC(NC(c3cnccc3Cl)=O)CC2C1 N1C(=O)c2ccccc2C1=O.c1cccc(C2(C(F)(F)F)N=N2)c1.N1(C)CCCC1 c1(OCC)nc(N(C(c2ccc(=O)oc2)=O)CC2CNCCO2)ncc1OC N1(C(C2CC(C)N(C)C2)=O)CCN(C(C2CC3(CC3)C2)=O)C2CCCC12 N1(C(C2CCC(C(N)=O)CC2)=O)CCC(NC(=O)CCc2cn[nH]c2)C(F)C1 C1(COC)CCC(C(=O)NCC(C)(C2CC2)NC(=O)Cc2ccon2)C1 C1(C(N2CCCC(NC(C=C(CC)C)=O)(COC)C2)=O)CN2CCCC2CO1 C1(C(=O)O)CCC(C(=O)O)CN1Cc1c(Cl)cccc1Br N1(C(c2cc(OC)c(N)cc2)=O)CC(C(=O)O)C2(CCC2)C1 c1(OCC(N2CC(C(C)NC(CN3CC(C)C3)=O)OCC2)=O)cccc(C#N)c1 C1(COC)(NC(=O)Cc2cnsc2)CCCN(C(=O)C=Cc2cccs2)C1 c1(OC)ncc(NC(N2CC(N3CCC(O)CC3)C2)=O)cc1C(F)(F)F Cc1cc(C(=O)N(C(C)C(=O)NCCCc2nncs2)C2CC2)nc(C)c1 c1(C(N2C(CCN(C(=O)CC3CC=CC3)C)CCCC2)=O)cccc2nonc12 c1(C(=O)NC(c2cn(C)nn2)C(=O)NCc2ncc(C)[nH]2)ncccc1F N1(C(c2c(OC)cncn2)=O)CC(NC(C2CCN(C)C(=O)C2)=O)CC1(C)C c1(C(N2CCC(CNC(C3(O)COC3)=O)C2)=O)ccc(-n2cccn2)cc1Cl C1(NC(C(C=C)(C)C)=O)CN(C(=O)C(C2CCC2)OC)CC2CCCC12 C(=O)(CCC(C)(C)C)N1C(C)CC(C)C1.c1(C(=O)N)cn(C)nc1C(C)(F)F c1(CNC(N(CC(CC)NC(=O)OC(C)(C)C)C)=O)cc(Cl)sc1C C(CCCC#N)(C(=O)Nc1ccccc1)N1CCC(NC(C)=O)C1 C(=O)(C1=CCCOCC1)N(CC(N1CC(O)(CO)C1)=O)C C=CCC(CC(C)C)C(=O)NCCCNC(C1(C2CCCO2)CCCC1)=O C1(C)(NC(c2ccc(C)cc2)=O)CCCCC1C(=O)NCCc1ccnc(C)n1 C1(NC(C(C2CCCCCC2)C)=O)COC2(CCN(C(C3(C#N)CCC3)=O)C2)C1 c1(CC)c(C(N2CC(N(C)C(c3cc(C)no3)=O)C(F)C2)=O)csc1C C12(CC(=O)NC3(CC=C)CCN(C(C)=O)CC3)CCCCC1C2(F)F N1(C(C(c2nccc(C)c2)(F)F)=O)CC2(CCN2C(c2cc(Cl)cc(Cl)c2)=O)C1 c1(C(=O)NCC2(NC(=O)CCCN3CCCCC3)CC2)cnc2ccccc2n1 N1(C(=O)C(F)=CC2CC2)CCC2CCCN(C(c3ccc(Cl)o3)=O)C2C1 CC(CN=C(NCC1CCC1)N1CCCC(S(=O)(=O)N(C)C)C1)NC1CCC1 N1(C(c2[nH]c(=N)sc2)=O)CCC(NC(=O)CN2CCC(=O)NC2=O)C(F)C1 Cn1nccc1S(C)(=O)=NC(=O)C1=CC(N)CS1(=O)=O.N(CCO)CCO CN(C)NC(=O)CCC(=O)N1CC2CCN(C(C3C(F)(F)C34CC4)=O)CC12 C(C(C)(O)C(=O)NCC1CCC(NC(C2CC(C)OC2C)=O)C1)OC c1(N(CC(=C)Br)C)nc(NCCCCCCO)c2cnn(C(C)C)c2n1 NC1CC(NCc2cn3c(Br)cnc3s2)C12CCOCC2 c1(-c2cccc(C(CC(=O)O)NC(=O)CC(Cl)Cl)c2)ccc(O)c2ccccc12 N1(Cc2cnc(OC)c(Br)c2)CC2(CCC(NC(=O)Cc3cncnc3)CC2)C1 C(=O)(C(CNC(c1nccs1)=O)CC1CCCC1)N(C1CCCC1(F)F)C C1(NC(c2cc(C)oc2)=O)CCN(C(=O)CC2CCCC(C#N)C2)CC12CCC2 C(=O)(CCC(N)CO)N1CCCC(C(N(C(CC)CC)CCC)=O)C1.N(C)C C(=O)(C(C)(C)CNC(c1cn(C(C)C)nn1)=O)NCCCC=CC CC1(C)C(NC(=O)CCC2CCOCC2)CC1N=c1cc[nH]cc1C#N N1(C(c2occ(C)c2)=O)CC(CNC(c2cc(Br)co2)=O)CC1(C)C c1(C=O)cc2n(n1)CC1(CC1)C2.N1(C(CC2(C#N)CC2)=O)CC(O)C(O)C1.C C1(c2nc(COC)on2)CN(C(c2ccn(CCF)n2)C(=O)NC)CCO1 n1(C2(C(=O)Nc3ccccn3)CC2)nccc1C(F)(F)F O=C(C(O)C(F)(F)F)NC1CC(CO)N(C(c2ccc(-c3nc[nH]n3)cc2)=O)C1 C1(C(N2C(C#C)CC2)=O)CC2CC1CN(C(=O)CCc1nc(O)n[nH]1)C2 N1(C(c2c(C)nc(C3CC3)[nH]2)=O)CC=C(C)CC1.C1(C(=O)N)CCC2C1C2(F)F C1(NC(C=C(C)C)=O)COC2(CCCN(C(c3cc([N+](=O)[O-])oc3C)=O)C2)C1 CN1CCC(NC(c2cc(Cl)ccn2)=O)C12CCCN(c1ccnc(CO)n1)C2 C1(C(N2CCN(C(C3(P(C)(C)=O)CC3)=O)CC2)=O)CCCC2(CCOC2)O1 Cc1nocc1CCC(=O)NCC1CC(NC(C2CC3CC3C2)=O)C1 C1(C(=O)NCC2(OC)CN(C(=O)C)C2)CCCCC1CN.c1cnn(C)c1 N1(C(C2C(OC)C2)=O)CC2(CCC2)CC1CNC(c1cccc2ncoc12)=O N1(C(c2c(CC)nc[nH]2)=O)CC2CCN(C(=O)C=Cc3cncnc3O)C2C1 C(=O)(C=CS(F)(F)(F)(F)F)N1CC(O)(CCNC(C(CC)C#N)=O)C1 N1(C(C(OCC)OCC)=O)CCCC(O)(CCNC(=O)C(CC)S)C1.C C1(NC(CCN(CC=C)C(C2CCCC(=O)CC2)=O)=O)CNC(=O)C1(C)C CC1CCN(C(=O)CN(C2CCC2)C)C(CNC(=O)CN2CCN(C)CC2)C1 c1(C(=O)OC)c(C)sc2cc(C(=O)OC(C)CCSC)[nH]c12 N1(C(C2(C)CC(C#N)C2)=O)CCC2(CCN(C(C3COCCC3(F)F)=O)CC2)C1 C(=O)(C1CCNc2ccccc21)N1CCC(NC(c2coc(Br)n2)=O)C(O)C1 C1(C(=O)NCCOC2CCN(C(Cc3cc(C)[nH]n3)=O)C2)Cc2nnc(C)n2C1 N1(C(CC(=O)OCC)=O)CCCC(NC(c2csc(-c3cnn(C)c3)n2)=O)CC1 N1(C(CSCC)=O)CCc2nc[nH]c2C12CCN(C(c1cnn3c1CCC3)=O)C2 C1(C(C(=O)NC2CCS(=O)(=O)C2)N(C2CCCCC2)CC)CC2(CCCO2)C1 S(=O)(=O)(c1cnc(N)c(Cl)c1)NC1CCN(CCC)CC1.c1nc(C)c(C)o1.C C(=O)(C(C)(COC)OC)NC(C1CCN(C(C=CC)=O)C1)C Cc1cc(C(=O)NCCC2CCCN(C(c3c(C)coc3C)=O)C2)[nH]c1C#N N1(C(=O)CSC2CC2)CC2CCN(C(C3CCC3c3nc(S)n[nH]3)=O)CC2C1 C1(CNC(CC2C(C)CC2)=O)CCC(C(N2CC3CCC2C3)=O)CC1 C1(OC)CC2CC1CN(C(=O)C(C)CN(C)C(c1ccnn1CCF)=O)C2 C1(NC(C(CC)OC2CCCCC2)=O)CN(C(c2coc(Br)n2)=O)CC1C N1(C(CCC)=O)CCN(C(c2ccc(SC)cc2)=O)C(CS(C)(=O)=O)C1 C1(Cl)(C(=O)NCCNC(C2(OC)CCOCC2)=O)CC12CCOCC2 CC(C)S(=O)(=O)C(C)C(=O)N(CCC)C.C(=O)(C(O)C(F)(F)c1ccccc1)N C1(NC(C2C(C(=O)OC)CCC2)=O)CCN(C(c2ccc(Cl)nn2)=O)CC(O)C1 c1(C(=O)NC2C=CCN(C(c3c(C)nc(CC)o3)=O)C2)cccc2cccnc12 N#Cc1ccc(C(N2CCOC(c3cn[nH]c3)C2)C(=O)NC2CCC2)nc1 C1(C(N(CCCCCNC(=O)C2=C(Cl)CC2)C)=O)CCc2n[nH]cc2C1 N1(Cc2ncc(C)cc2F)CCc2cccc(-c3ccc4cncnc4c3)c2C1 N1(C(C(C)(C)OC)=O)CCC2CC(C1)CN(C(=O)C(C)N1CCC1)C2 N1(C(C(C)=CC(C)(C)C)=O)CCCCC1C(C)NC(=O)CN1CCOC1=O Cc1onc(Br)c1C(=O)N(CC(C)NC(=O)C(N1C(=O)CCC1=O)C)C C1(C(=O)NC(Cn2ncc(C)c2)C)C2CN(C(C3(CO)CCOC3)=O)CC12 C1(C=O)COCCC1(F)F.C1(CC)(NC(c2cc(C3CC3)[nH]n2)=O)CCCC1.N Cc1cnc2c(C(=O)NC(C3CCCCN3C(C3(F)CCCC3)=O)C)cnn2c1 c1(CC(=O)NC(CC(C)NC(C=CC(C)=O)=O)C)c(C)cc(C)nc1O Cc1cc(CC(=O)N)cc(C)c1.c1(C(N(CC)C2CC2)=O)cn(C(C)C)nn1 c1(OC)ncccc1C(=O)N(CC(C)NC(c1ccc(CC(C)C)nc1)=O)C C1(NC(CCCC=C)=O)COCCN(C(C2(c3ccno3)CC2)=O)C1 CC(C(=O)N1CCC(CNC(=O)CCC2CCCC2)C1(C)C)C1=CCCC1 c1(NC(C(CC)(C)O)=O)ccc(NC(c2cc(OC)cc(Br)c2)=O)c(F)c1 C(=O)(C1CCCc2cncn21)NC(CN(C(c1c(OC)nc(C)nc1)=O)C)C c1(C(N2CC3C(C3)C2)=O)cccc(N)c1C(F)F.CCCCCOCC(=O)N.C C(=O)(C1=C(C)CCOC1)NC(CC(=O)N(CCCCC)CC(N)=O)C N1(C(c2c(C)coc2)=O)CCC2CN(C(c3coc(C4CCCC4)n3)=O)CC2C1 N1(Cc2nnc(CC)o2)C2CCC1CN(C(C1CCS(=O)(=O)C1)=O)CC2 c1(C(=O)NC(C)CC2CCN(C(=O)C3=COCC3)CC2)cnc(O)c2ccsc12 N1(C(c2ccc(CC)nc2)=O)CC(NC(c2ccncc2Cl)=O)CC12CCCC2 c1(C(=O)NCC=CC(=O)NCC=Cc2cocn2)cccnc1 C(C)(C(=O)NC1CCC1)(C(C)C)NC(C)=O.c1(C=O)ccccc1.N(C)C N(C1CCCS(=O)(=O)c2ccccc21)C(CCC=C)C C12(NC(C3CN(C(C)C)C(=O)C3)=O)CCC(CC1F)C2.c12cn(nn1)CCCC2 Cc1ccc(Br)c(CC(=O)NC(C)C2CC2)c1.N1(C2(C(=O)N)CC2)CCCC1 CN1CC2CCCN(C(c3c(Cl)ccc(Br)c3N)=O)C2C1 C(Cc1ccccc1)(C(=O)NCC(C)C)OC.C(=O)(C(O)CC1CCCCC1)N c1(C(C)C)nnc(C=CC(=O)NCC)o1.C(=O)C(C)(C)CN1CCOCC1.N CC1OCCC1C(=O)NCC1(F)CC(C(=O)NC2(c3cccnc3)CC2)C1 N1(C(C2(C)CCC2)=O)CCC2(CCCN(C(c3c(F)cncc3F)=O)C2)CC1 N1(C(c2n(CC)nnc2)=O)CC2CCC(N(C(=O)CC3(O)CCOCC3)C)C2C1 Cc1c(C(=O)NC2CC(O)CN(C(=O)C(C)(C)c3cscn3)C2)cccc1O C1CCC2CN(C(c3coc(C(C)(C)C)n3)=O)CC2C1.C1(OC)CCC1C(=O)N CN1CCCCC1CC(=O)NCc1n[nH]cc1C(=O)NC1COCC1O N1(CC)CC(C(=O)NCC2CN(C(=O)C#CC3CC3)CCCO2)c2ccccc21 N1(C(C=Cc2nc(C)c(C)[nH]2)=O)CCC2CCN(C(=O)CC3CC4CC4C3)CC12 Cc1cc(C)c(C#N)c(NCC(CC(C)C)NC(c2conc2C(C)C)=O)n1 N1(C(Cc2c(C)nc[nH]2)=O)CCC2CN(C(=O)CP(C)(C)=O)CC2CC1 c1ccc(F)cc1.C1(N(C(=O)COCCc2cccs2)C)CCN(C(=O)C)C1 N(C1CCCc2cc(CNC(c3scc(C)c3C)=O)ccc21)C(C=C(C)C)=O N1(C(c2c(C#C)cn(C)n2)=O)CCC(C2CCCN(C(=O)CC3CN(C)C3)C2)C1 C1(C(C)NC(C(C)SCC)=O)CN(C(=O)CCc2ccc(F)cc2)CCO1 C1(NC(CC2CCN(C)C2=O)=O)CCC12CN(C(c1nnc(O)cc1O)=O)C2 c1(C(N2CCC(COC)(NC(=O)CC(F)F)C2)=O)cc(=O)n2nccc2[nH]1 c1(C(=O)NC23C(CN(C(C(C#C)(C)C)=O)C2)CCC3)oc2ccc(C)cc2c1C c1(OC)cc(C(=O)NC2COCCC2)nn1C.C1(CCC(=O)N)NC(=O)NC1=O Cc1cc([N+](=O)[O-])cc([N+](=O)[O-])c1N1CCN(C(=O)C2=CC3(CCNC3)C2)CC1 CCC(O)CCN=c1nc(N2CCC3(CCC3)C2)c2[nH]ccc2[nH]1 CCC(CC)(CCNC(c1ncn(C)c1C)=O)NC(=O)CCC1CC1C c1(C(=O)NCC2C=CCN2C(=O)Cn2cccc2)cccc(C(F)(F)F)c1 c1(C(N2CCC(C(C=O)(C)C)C2)=O)oc(C)cc1C.N1(C(C)=O)CCC(C)C1.N N1(C(c2c(SC)nccn2)=O)CC(NC(c2c[nH]nc2C)=O)C2(CCOCC2)C1 C1(C(NOCCCC#C)=O)CCC(O)CN1C(=O)CCC1CC(C)C1 N1(C(c2c(N)c(F)ncc2)=O)CC2CC(NC(=O)CN3CCCCCC3)CC2C1 c1(C(C)NC(C2CCC2)C2CCC2)nnnn1C1CC1 c1(C(=O)NCC(C)N(C)C(c2nccc(F)c2Cl)=O)ccc2c(=O)cc[nH]c2c1 N1(CC(N2C(CNC(c3cnn(-c4ccccc4)n3)=O)CCC2)=O)CCCC1=O n1(C(C=O)C)cc(CCCC)nn1.C(C)(C)N(C(C)=O)C.C(C)(C)C.C(N)=O N1(C(c2c(SCC)nccn2)=O)CC2CC(C1)C2NC(=O)CC(C)F CCC(F)(F)CC(=O)N1C2CCC(C2)C1CC(=O)NCC1CCCCN1CC c1(-c2cncc(CNC(COc3c(C)cccc3)=O)c2)cnc2c(c1)CC(=O)N2 N1(C(C(C)(C)OC)=O)CCCCC2(CCN(C(=O)Cc3c(F)cncc3Cl)C2)C1 Cc1cnn(CC(=O)NC(C)C(C)NC(c2ccoc2)=O)c(=O)c1 c1(C(=O)NC(CC)CNC(=O)CCCn2cc(C)cn2)ccc2ncccn12 c1(C2C(C(N3CCC(O)C3)=O)C2)ccc(Cl)cc1Cl.C(CC(=O)N)SCCC.C c1ccc(Cl)c(Cl)c1Cl.c1(C(C)(C)C)ccc(Br)c(NC(C2CC(N)C2)=O)c1.C C(C(C)(CC)C(C)O)NC(CC1(NC(CC=CCCCCC)=O)CC1)=O CS(=O)(=O)C1(C(=O)NC2(C3CN(C(=O)C4=C(Cl)CC4)C3)CC2)CCC1 Cc1cccc(-c2nc(C)c(C(=O)NCCOC3CCCCC3C)[nH]2)c1 N1(C(C2C(CCC)CCC2)=O)CC(CNC(=O)C(Cl)=CCl)C(O)C1 C1(O)(CNC(C(F)=CCC)=O)CCN(C(=O)CCc2cnn(C)c2)C1 C(COC)(CC(=O)NCC=CCCOC)NC(CN(CCC)C)=O N1(C(C23N(C(c4c(C)con4)=O)CC(C2)C3)=O)CC(C)(C)OCC1C C1(OCC)CN(C(=O)C(C)C2CCCC2)CC1CNC(=O)C.c1cn[nH]c1 c1(N2CCC(NC(c3ccc(C(F)(F)F)cn3)=O)C2)ncc2cccnc2n1 c1(N(CCNC(CC(C)C)c2nnnn2C)C)cnn2ccn(C)c12 C(=O)(C(C)Cc1cnco1)N(C(CN(C(CCOC(C)=O)=O)C)C)C C(c1ccc[nH]1)=CC(=O)NCC(C)NC(CSCC=C)=O C(c1ccc(F)c(Cl)c1)=CC(=O)N.C1(NC(C2(Cl)C(C)(C)C2)=O)CCCC1O CC1ON=C(C(=O)NC(C)C(C)(C)NC(c2cnc3n2CCS3)=O)C1C N1(C(C(C=C)(C)C)=O)CCOC2(CCN(C(C3(F)CN(C(=O)O)C3)=O)C2)C1.C Cc1c(Br)ccc(NC(C2CC(C)CN2Cc2ccncc2C#N)=O)c1F C(C(CNC(=O)CCN(C(=O)C(C)CC1CC1)CCO)C(C)C)OC N1(C(C(C(C)OC)N(C)C)=O)CC(C(=O)N)CC(C)(C)C1.C1(S(C)=O)CC1 Cc1cc(C)c(C)c(C(=O)NC(CNC(C2CCC(=O)N2)=O)CO)c1C CC(C)(C)C#CC(=O)NCC1(NC(=O)CCC2CCCC(=O)N2)CCCCCC1 C1(NC(c2cc(Cl)ccc2I)=O)CC12CCN(C(C13CCC(CC1)CC3)=O)CC2 N1(C(C2N(C(C(C)=O)=O)CCC2)=O)CCNc2ccc(Cl)cc2C1 C1(C(=O)NCCNC(C(C)O)=O)CCCN(C(=O)C(C)O)C1 C1(C(C)C(=O)N2CC(N3CC(F)C3)C2)CCN(C(c2cn(C)nn2)=O)C1 O=C1NC(C(=O)NCC2CCC2NC(=O)CCOC2CCCCC2)CCO1 CC1CN(C)CC(C(N2CC3(CCC3NC(=O)CCCN3CCCCC3)C2)=O)O1 N1(C(c2cccc(CO)c2)=O)CCN(C(c2c[nH]nc2C(F)F)=O)C(CF)C1 CC(C)CC(C(=O)N(C1CN(C(=O)CCC=CBr)CC1(C)C)C)C(C)C c1(OC)cc(CNC(=O)C(C)=CCNC(=O)CC2(C)CC2)sn1 C1(C)(CNC(C2(CCC)CCC2)=O)CCC(NC(=O)C)C1.CC(C)C.O c1(C(N(C2C(C)CN(C(c3nncs3)=O)CC2)C)=O)ccc2cncn2c1 CC1CN(C(=O)Cc2nc[nH]n2)CC(C)N(C(c2ccc(NC=O)cc2)=O)C1 c1(C(=O)NC(CN(C(=O)Cc2cn(C)nn2)CC)C)ccc(F)cc1 C1CCN(C(C)C)CC1.C1(OC)(OC)CCC1C(=O)NC1CCOC1C=O.N C12(NC(c3[nH]cc(C)c3)=O)CC(C)(C1)OC21CN(C(C2CC(F)(C)C2)=O)C1 c1(OCC(N2CC(C(=O)NCCC#N)OCC2)=O)ccc(F)cc1O Cc1cc(C(=O)NCC2CCCC2NC(C2CCC(=O)N2C)=O)c2occc2c1 C1(N(C(CC)=O)C)CCC(NC(C2CCN2Cc2ccc(C)cc2)=O)CC1 C1(CC(N2C(CNC(CCC=CC)=O)CC2)=O)CCCC(C(F)(F)F)O1 C1(NC(c2ccc(OC(CC)C)cc2)=O)CN(C(=O)C(F)=C2CCC2)CCC1F c1ccc(Cl)cc1F.c1(CC(=O)N(Cc2c(C)noc2C)C)ccc(O)c(F)c1 c1(C(N(CCC)CCC)=O)cccc(NC(c2cc(Cl)ccn2)=O)c1 CCCC#CC(C)(C)NC(C1(CC)CCCN1C(=O)CCC(C)CN(C)C)=O Cc1c(CNC(=O)C(N)CCF)nnn1C CCC(CC)C(C(=O)NC1CN(C(=O)C(C)(C)O)CC1SC)N1CCOCC1 C(=O)(CCCCCCC(=O)O)NC(C1CCC1)C C1(NCCCn2ccnn2)CCN(CC2CC2)CC1 S(=O)(=O)(c1cccnc1)N1C(C(=O)Nc2cc(Cl)ccc2I)CCC1 N1(C(c2c(CC)occ2C)=O)CC=C(CC(=O)N2CCC(C)C2)CC1.N(C)(C)C Cc1cnn(CC(=O)NCCOCC(=O)Nc2cn(C)nc2C#N)c(=O)c1 c1(C(=O)NCC(CC)NC(c2ccnnc2)=O)c[nH]c2c(OC)cc(C)cc2c1=O C12(C(N3CCC(C(F)F)(CO)CC3)=O)CCCCC1C2Br Cc1ccc(NC(Cc2ccccc2)C(O)C(C)C)c(F)c1 C1(C(C)NC(c2n(CC)ncn2)=O)CN(C(c2sccc2COC)=O)CCO1 C1(CNC(C(C)(C)n2cc(Br)cn2)=O)CN(C(C2CC=CCC2)=O)CCO1 c1(C(N(C2CCN(C(=O)C(C3CC3)C)C2)CCC)=O)csc([N+](=O)[O-])c1 C1(CC)CN(C(C2SCCS2)=O)CCC1NC(=O)Cc1c[nH]nc1O C1(N(C(C(c2ccc(C)o2)C)=O)CCO)CCCN(C(=O)CN(C)C(C)C)C1 c1(SCC(=O)NC2CCCN(CCCO)C2)nc2ccccc2[nH]1 C1(NC(C=Cc2ccc(SC)s2)=O)CN(C(=O)CC2COC(=O)C2)CCC1F c1(C(N(C(C)CNC(=O)CCC(F)F)CC)=O)ccc(OC(F)F)nc1Cl C(N=c1[nH]cnc(Cl)c1CC)C1CCC(NC(c2cc(OCC)n[nH]2)=O)C1 C(=O)(N=c1nc(CS(C)(=O)=O)[nH]o1)C1CCN(C(CC)=O)CC1C C1(C(N)=O)CCN(CCC(N2CCCC(NC(c3ccccc3)=O)C2)=O)C1CN C(CC(=O)Nc1cc(O)cc(F)c1)(C(F)(F)F)NC(CC(C=C)CC)=O c1(C(C=O)(C)C)ccccc1Cl.C12CC(C1)C2.C(C)(C(=O)N)OCCOC c1(C(=O)NCC(=O)NC(C(=O)OC)(C)C2CC2)cc2cccnc2[nH]1 C1(CC)CN(C(=O)CCOC)CCC1NC(=O)C=Cc1cccnc1 N1(C(C(C)NC(=O)C(C)(C)C)=O)CCC(C)(CC)C1.C(=O)CCc1cnoc1 C1(CNC(C=Cc2cn(C)nc2)=O)CC2COCC2N1C(=O)C=CBr c1(C(C(F)(F)F)NC(C2CCC(N)CC2)C)cccc(F)c1F Cc1nn(C)c(C(N2CCC(C)(CNC(c3ncc(Br)cn3)=O)C2)=O)c1Cl Cn1cnc(C2CCCN2C(=O)COCC2CCCO2)c1 N1(C(c2c(C)n(C3CCC3)nc2)=O)CC2(CC(NC(=O)C=C3CC3)CO2)C1 Cc1cc(C(N2CCCC2CN(C(=O)Cc2ccc(O)c(O)c2)C)=O)c(O)nn1 Cc1cc2cc(-c3nc(C)c(NC(=O)CCC=CC(C)C)s3)cnc2[nH]1 N1(CC=C)C(=O)NC(c2c(Cl)cccc2Cl)C(C(=O)NC2CC2)=C1C1CC1C C(=O)C(C)S(=O)(=O)CCC.c1(CC)nn(C)cc1C(=O)NCC1CCCC1 N1(C(c2ccno2)=O)CCN(C(=O)C)CC1.C1(CC=O)COC(=O)C1.CC.O C1(CNC(C2CC=CC2)=O)CC2CN(C(c3ccc(F)cc3F)=O)CC12 C1(C(N2CC=CC(NC(CCC3(C)CC3)=O)C2)=O)CC2COCC2C1 Cc1cc(CCNC(c2c(Br)cnn2C)c2nnnn2CCCO)ncn1.C(C)C C(=O)(C(CC1CC1)NC(=O)CC1CCSC1)NC(COCC)C C1CN(C(c2ccns2)=O)C2(CCC2)C1.c1(C(=O)NC)cc(-c2cccs2)on1 N1(C(C(C)N(C(C)=O)C)=O)CCC(C(=O)NCc2ncccc2C)=C(F)C1 C#CC1CN(C(=O)CC(C)(C)CNC(=O)CC2CC=CCC2)CCN1C c1(C(=O)NCCC(=O)N(C2CCCC2)CCNC(C)=O)ccc(C)nc1 CC(C)(C)CCCCNC(C1CCN(C(=O)Cc2ccsn2)CC1)=O c1(C(=O)NC(C)CN(C)C(c2nonc2N)=O)cc2cccnc2s1 c1(OC)ccc2c(c1)C(C)CN(C(C1CCNc3ccccc3C1)=O)CC2 C12(C(=O)NCC3N(C(CCN(C)CC)=O)CCC3)CCCC1OCC2 N1(CC(=O)NCC(=O)NCCn2cc(-c3ccncc3)nn2)CC2CC2C1 c1(C(N2CCCCC(CNC(C(CC)O)=O)C2)=O)sc2nc(C)nc(C)c2c1C Cc1ncc(C(=O)NCC2CC(F)(CNC(C3(F)CCOC3)=O)C2)n1C C(=O)(C(C)C1OCCc2sccc21)N(CCNC(CC)=O)C S(=O)(=O)(c1cnc(NCc2ccnc(C)n2)c(Cl)c1)NC(COC)C(C)C C(=O)(CCCCC(=O)NCC1(C(=O)N(C(C)CO)C)CCCO1)OC C(=O)(C(CNC(c1cc(C)n(CC)n1)=O)C(C)C)NCCOCCC=C C(=O)(C(F)CC(C)C)NCc1cccc(NC(Cc2cc(C)ns2)=O)c1 C(=O)(CS(=O)(=O)NC)NC(CN(C(C1C=CC1C(=O)O)=O)CC)C C1(NC(C(CC)OC)=O)CN(C(c2csc(C)n2)=O)CC12CCCC2 CC1(CC(=O)NC2CC(NC(C3(Br)CC3(C)C)=O)C2)OCCO1 C(N=c1[nH]c2c(c(=NCCCC3CC3(Cl)Cl)[nH]1)CSC2)C1(C(N(C)C)=O)CCC1 Cc1cc(CNC(C2CN(Cc3c(F)cccc3Cl)C2)=O)c(C)n1-c1nccs1 N1(C(CC2CCN(CC(N3C(CO)CC3C)COC)C2)=O)CCCCCC1 Cc1cc(C(=O)NCCCC(O)C(=O)NCC2(C)CCN(C)CC2)cc(F)c1 N1(C(=O)CCn2cnccc2=O)CCN(C(c2ccncc2)=O)C(CO)C1 C1(C(=O)NC(C2(O)CN(C(c3cnccc3Cl)=O)C2)C)C2CCC(F)(F)C12 c1(C(=O)NC2(C)CCCN(C(CCC(C)OC)=O)C2)cc(Cl)cc2c1OCC2 CC(C)(C(=O)NCC1(C)CCCN1C(=O)Cc1ncc(F)cc1F)C(F)F c1(C(=O)Nc2ncc(Br)cc2OCBr)cc2c(-c3cc4sccc4s3)cncc2s1 C1(CCC(C)C)CCCCN1C(c1nnn(C(C)(C)C)n1)=O.CC=O.CC=O.O C1(C(=O)NCC2(C)CCCN(C(C3COCCO3)=O)C2)C2CCC3C(C2)CC13 c1(OC)cccc(OCCC(=O)NCC(O)CCNC(c2c(Cl)noc2C)=O)c1 c1(C(=O)NCC2C(NC(C(c3cc(C)sc3)(C)C)=O)CCC2)c(C)coc1C c1(C(=O)NCC)ccc(-n2ccnc2)cc1.C1CCN(C(C23CCC2C3)=O)C1.O Cc1cc2c(C(N3CC(CNC(=O)Cc4cccnc4)CC3C)=O)cccc2o1 C1(C(N)=O)(OC)CN(C(=O)COC2CCN(C(C3CCOC3)=O)C2)C1 c1(C(=O)NC(CC(C)NC(=O)CN(C)C)C)ccnnc1NC1CC1 C(=O)(C1=C(CN2CCN(CC(F)F)CC2)NC(=O)NC1)OCC.C1C(=O)N1 CCCC(C)(C)C(=O)N1CC(C(=O)Nc2ccc(Cn3cc(C)cn3)cc2)C1 C=CCCC(CC(C)C)C(=O)NCC(CC)NC(=O)C1=CCC1 c1(N2CC(CNC(=O)CC3CC(F)(F)C3)OCC2)ncnc2cccnc12 Cc1c(C(N2CCOC(CNC(c3cc(C(N)=O)c[nH]3)=O)C2)=O)cc(O)cc1N C1(O)(CNC(c2ccc(CCC)[nH]2)=O)CCCN(C(=O)C=CCNC)C1 c1(C(N2CC(F)(CNC(Cc3c(C)nccc3)=O)C2)=O)cnn2c(C)ccnc12 c1(C(N(CCCC)C)=O)ccc2c(c1)nc(C)n2C1CC1.C1(C=O)C=CCC1.N N1(C(C(C)N(C(c2ccc(C)cc2)=O)C2CC2)=O)CC2(CC(CO)CO2)C1 c1(C(=O)NCCN(C(=O)Cn2nnnc2C)CCC)ccc(F)s1 C1(C(N(C2CC2(C)C)C)=O)CC2(CCC2)CN1C(c1cnc(S)nc1)=O C1(C)(C(=O)NCC2CCN(Cc3n(CC)ncn3)C2)CC=C(C)CC1 N1(C(COCC(=O)OC)=O)CCC(C2CC2)(C)C1.C1(C=O)CC2CCC1C2 C1(C(=O)NC(C)CCNC(=O)C(C)Oc2cccnc2)CCCCCN1C N1(C(C(C)C)=O)CCOCC(C)(CNC(c2cn(C)nc2C(F)(F)F)=O)C1 C1(CC)CCCCC1N=c1[nH]c(=NCc2cc(Br)c[nH]2)[nH]c2cc[nH]c12 Cc1cncc(C(N2CCCCC2CNC(=O)C)=O)c1.c1nccn1C(F)F.S n1(C(C(=O)NCCC)C)cc(C(=O)Nc2ccccc2)c2ccccc12.OCC N1(C(=O)NC(c2ccc(C)o2)C)CCC(N=c2cc[nH]cc2Cl)CC1 C1(C(N(CC)CC)=O)CC(C)C1(C)C.C(=O)(C=CC)N.C(C)(C)C N1(CCNC(C(C)SC)=O)CCCN(C(c2ccc(C)cc2C2CC2)=O)CC1 C12(NC(CCOC)=O)CCCN(C(c3cccc(CO)c3)=O)CC1C2 Cc1cncc(C(=O)NC(C2CCCN(C(C3CC(n4cnnc4)C3)=O)C2)C)n1 c1(C(N(CC(C)N(C(=O)CC2CC(F)C2)C)C)=O)ccc(C2CCOC2)s1 c1(NC2CCC(C)C2)ccc(S(=O)(=O)NCC(c2ccccc2Br)(C)C)cn1 c1(N2CCC3(NC(=O)OC3)CC2)nc(Cl)nc2cc(Cl)ccc12 C=CCCC(O)CNC(=O)C(C1CCCN(C(c2ccc(CO)cn2)=O)C1)C N1(CCNC(=O)NCC2(OC)CCC(C(F)F)CC2)CCc2ccccc21 n1(CC(=O)NCC(COC)NC(c2c(CC)cno2)=O)nc(C)nc1C C1(CC(=O)OCC(c2ccc(C)cc2O)=O)CC(C)CC(C)(C)C1 C1(C(=O)OC)CCCC(C(=O)NCCCCNC(=O)Cc2ccon2)CC1.C N1(C(c2[nH]cc(CC(C)C)c2)=O)CCN(C(c2cn(C)cn2)=O)C2COCC12 c1(N2CCC(NC(c3n[nH]c(C)c3Cl)=O)C(O)C2)ncc2ccccc2n1 N1(C(C=C(C)C)=O)CCOC(C(=O)NCCC(C)C(C)C)C1 c1(C(=O)NC(CC(C)NC(=O)CCc2ccncc2)C)cccc(SC#N)c1 c1(C(=O)NC(CC)CN(C)C(c2c(C(C)C)cnn2C)=O)nccc2cc[nH]c12 C1(CNC(C2(NC(N)=O)CC2)=O)CC2CCCC2N1C(C1COCCO1)=O CCCCCCCCC(=O)N(CCC(=O)NCC1CC(O)C12CCC2)CC c1(NC(CN2CC(O)(CNC(c3c(C)c[nH]n3)=O)C2)=O)n[nH]c2cccnc12 C1(CNC(c2cn(C3CCC3)nn2)=O)CN(C(=O)CCC2CC2(Cl)Cl)CC1O C1(CNC(C=CCOC)=O)CC2CCCC2N1C(c1cc(=O)cco1)=O.O C1(C)(OC)CC(NC(C2(F)CC2)=O)C1(C)C.C1(=O)CC=CCN1 C(CC(=O)N1CC(O)(C)C1)(C(F)(F)F)OC.C1(C(=O)N)CN(C)CCN(C)C1 N1(C(C2(CC=C)CCCN2C(=O)C#CC2CC2)=O)CC2CCCC2(CO)C1 N1(C(CCCC#C)=O)CC(CCNC(=O)CN(C(=O)COC)C)OC(C)C1 Cc1noc(C(CO)NC(c2ncoc2CNC(C2CC2(Cl)Cl)=O)=O)n1 N1(C(c2c(C)occ2C(F)(F)F)=O)CC2CC(C1)C2.C(c1cncs1)=CC=O c1(C(=O)NC(C)C(C)F)ccoc1CNC(=O)C(C)(C)C1CCC1 C1(CC)CCCN(CC(=O)NCC2CCCC2NC(c2ccon2)=O)C1 Cc1ccc(C(=O)NC2(CF)CCN(C(=O)C3=NNC(=O)C3)C2)c(O)c1 O=C(CS(=O)(=O)CCO)NCC1CCCCN1C(c1csc(Cl)n1)=O n1(CC=O)c(=O)nc(O)c2ccccc12.C(C(=O)NCC)(C(C)(C)C)SC.N N1(C(C(C)OC2COC2)=O)CCC2(CC(NC(c3cncs3)=O)C2)C1 C1(N=c2[nH]nco2)(CNC(C(CC(C)(C)C)O)=O)CCCC1 CC1(C)CCN(C(=O)COCC2CC2)C1.c1(C=O)cc(C2CCCCC2)on1 c1(C(=O)NCCC2(O)CN(C(c3c(CCC)[nH]cc3)=O)C2)ncn2ccccc12 CC1(C)CC(C(=O)NC2CCC(F)(F)C2)CN1C(c1ccsc1Cl)=O C1(NC(=O)NC(c2ccnn2C)COC)CC(F)(F)C12CCC2 c1(-c2n(CC)c(N(C)C3CC3)nn2)cc(Sc2ccccc2Cl)cc(C2CC2)n1 C(CC(N)=O)(C(=O)NC(C)CO)NC(C(C1CCCC1)OC)=O C1(C(=O)NCCCC#C)C=CCN(C(=O)C(CC)n2ccnc2)C1 C1(N(C(c2c(C)n(C)cn2)=O)C)CN(C(C2CC(C)CC(=O)N2)=O)CC12CC2 N1(C(C2C(=C)CC2)=O)CCN(CCCCCNC(=O)CC2(C)CC2)CC1 N#CC1=C(C(=O)N2CCN(C(c3coc(-c4ccccc4)n3)=O)C3CC23)CCC1 C1(C(=O)NCC(C2CC2)C2CC2)C2CCN(C(c3cnc(S)nc3)=O)CC12 C1(C(N(C(C)CNC(=O)C(C)(C)n2cccn2)C)=O)COCCN1C=O C1(CCCCCNC(C2(C(C)C)COC2)=O)CCN(C(c2ccc(F)o2)=O)CC1 N1(C(C2CC(C)C2)=O)CC2(N(C(=O)CO)CCO)CCC1C2.c1cccc(Cl)c1 C#CCCC(=O)NCC1(CCCNC(=O)CC)CCCC1.C(=O)(CC(C)C)N c1(C(N2CCCC(N(C(=O)CN(C)S(N)(=O)=O)C)C2)=O)c(F)ccc(Cl)c1N Cc1ncn(C)c1C(N1CCCC(C2CCCN2C(C2CC3(CC3)C2)=O)C1)=O c1(C(=O)NC2CN(C(=O)CCn3cccn3)C2)cnc2cc(O)ccc2c1 C1(CNC(c2cc[nH]n2)=O)CCCCC1NC(c1cnc(O)o1)=O C(=O)(C(O)(C(F)(F)F)c1ccccc1)NC.C(C1CCOC1)=CC(N1CCC1)=O C1(C(=O)NCCC2(NC(C3N(C)CC3)=O)CCC2)CC1[N+](=O)[O-] C1(NC(CCOCCC)=O)CN(C(=O)C(F)CC)CC1(C)C CCC(CCC(=O)N1CCC(NC(=O)C(=O)NCCCOC)CC1)OC C1(NC(CCC#CC)=O)COC2(CCN(C(c3cn(C)cc3C)=O)C2)C1 c1(C=O)ccccc1O.C1(C(=O)NC2CC(C)C2)(OC)CS(=O)(=O)C1.N C1(NC(CCCN(C(C)C)C)=O)CCN(C(=O)C=CC2CCCC2)CCC1(F)F c1nc(=N)cc[nH]1.C=C1CC(C(=O)N)(CSC(C)C(C)C)C1.c1ccccc1 C(=O)(CC(C)(C)F)NCC(c1cccc(Cl)c1)NC(CSC(C)C)=O N1(C(C(C)(C)OC)=O)CC(C(=O)NC2CCC(=O)N(CC)C2)CC(C)(C)C1 C(=O)(C(C)CC(C)C)N1CCCC(NC(c2c(OCC)nccc2)=O)C1 CCC(CC)(CO)C(=O)N1CCN(C(=O)CC(C)c2cccnc2)C(CCO)C1 c1(CCC(=O)NCC(CC=C)NC(c2noc(C3CC3)c2C)=O)nccnc1C c1(NCC2(OC)CCSCC2)cc(=NC2CCC3CC3CC2)[nH]c(C(F)(F)F)n1 CCCC(C)C(=O)NCCc1cc(C(=O)NC(C)(CC)CCC)no1 N1(C(C=C(C)C2CC2)=O)CC=C(C(=O)NCC(N2CCCCC2)=O)CC1 CC1CCN(C(C23CC(F)(C2)C3)=O)CC1.C12(C=O)CC(c3ccccc3)C1C2.N C1(N(C)C(C2CCC23CCC3)=O)CCCN(C(=O)CCNC(N)=O)CC1 C1(CCNC(C2CCCO2)=O)CCCN(C(c2ccc(-c3cccs3)[nH]2)=O)C1 CC1C(NC(=O)C=CCN(C)C)CCCN1C(c1cnn[nH]1)=O c1(CC)[nH]c(C(N2CCC(C(C)NC(=O)CCN3CCCC3=O)C2)=O)nc1Cl N1(C(c2cnn(C(F)F)c2)=O)CCC2C(CCCN2C(=O)C2=CCOC2)C1 C1(NC(COCCCOC)=O)C2CC(O)C1N(C(c1cc3sccc3cn1)=O)C2 c1(C(N(C2CCCN(C(CC(C)O)=O)C2)C)=O)cc2ncccc2cc1Cl C1CC(O)(C2CCN(C(=O)C(C)=C(C)C)CC2)C1.c1(CC)ncc(C=O)s1.C c1(CNC(COC)=O)cn(C2CCN(C(=O)CCC=C(C)C)C2)nn1 Cc1cccc(Cl)c1S(=O)(=O)N1CC(NC(c2ccc(Br)c(F)c2)=O)CC(F)C1 C1(C(=O)NC(C2C(C(=O)NCCn3c(C)nnc3)C2)C)CCC2(CC2)C1 C(C(=O)NCC1(C)CCCN1C(=O)CCCF)(C(C)C)OC c1(C(=O)NC2CCCN(C(c3c(OC)ccs3)=O)C2)c(Cl)ccc2c1OCO2 c1(C(N(CC(CN(C(C(C(C)C)F)=O)C)O)C)=O)nccc2c(Br)cccc12 N#Cc1nc(Cl)ccc1CN(c1nccs1)C(=O)NCc1ncc(Br)s1 c1(C(=O)NCC(=C)CCNC(c2coc(Cl)c2)=O)csc2cncn12 C12(CNC(=O)NCC(N3CCCC(C)C3)=O)CCCC(C)(C1)OC2 c1(C(N2CCN(CC)CC2C)C(=O)NCC=C)cc2ccccc2o1 N1(C(CCCN=[N+]=[N-])=O)CCCC2(CCC(NC(=O)CSCc3ncc[nH]3)C2)C1 C1(C)(C(=O)NCC(c2ccc(C)cc2)NC(CSCCCC)=O)CC=CCC1 N1(C(c2ccccn2)=O)CCSCC1C(=O)NON1CCCCCC1.O=C1CN1 c1(C(=O)NC2CN(C(CCCOCC=C)=O)C(C)C2)ccc2c(c1)CCOC2 C1(C(=O)OC)CN(N2CCC(Cc3cccc(Cl)c3)CC2)C(C)CO1 C1(C(=O)NCCOC(C)C)CC2CCC1N2C(=O)CC12CCCC1C2 O=S(=O)(c1cnccc1N1CCC(c2nncs2)C1)N1CCC(SCCO)CC1 C(=O)(C(C(C)C)NC(=O)C(C)(C)C)NCC(CC)NC(c1ncn[nH]1)=O c1(C(N(C(C)C(N2CCOC(CCN(C)C)C2)=O)C)=O)ccc(F)c(F)c1 C1(NC(c2c(OC)cc(C)cn2)=O)C(C)CCN(C(c2cccnc2O)=O)C1C N1(C(Cc2c(SC)cccc2)=O)CC(C2(NC(=O)Cn3nc(C)nc3C)CC2)C1 C(=O)(C(C)CS(=O)(=O)Nc1ccc(-n2cccn2)c(OC)c1)OC C12(CNC(c3cc(C)sn3)=O)CC1CN(C(=O)COC(F)F)C2 N1(C(Cn2c(C)cc(C(F)F)n2)=O)CCC(C)CC1.S(S(C)(=O)=O)CC=O.C Cc1ccn2ncc(C(N3CCC(C)(CNC(C4(C)CC5CC5C4)=O)C3)=O)c2c1 C1(CC)CCCN(C(=O)C)C1.C1(CC=O)C=NN(C)C1=O.C1(O)(C)CCC1 C(c1ccc(S(C)(=O)=O)o1)=CC=O.CC(C)(C=O)C(N)=O.C1CCCCC1.N C1(NC(c2sc3c(c2)C(=O)CC3)=O)C2Cc3cc(Cl)ccc3C12 N1(C(C2(COC)CN(C(=O)CSC)C2)=O)CC(C)C1(C)C N1(C(CCCC=C)=O)Cc2ccnn2CC(CNC(=O)CC2CC3(CC3)C2)C1 C(=O)(CC(C)C(=O)NCc1cc(O)ncn1)OC.C(=O)C(C)(C)C1CC1.C c1(C(=O)NC2CC(C(C)C)OC2)ccc(N2CCOCC2)cc1F C=CCC(C)(C)C(=O)N1CCC(OCC(=O)N(CCC)CCC)C1 c1(CN2C(C(N3CCC(C#C)CC3)=O)CCC2C)c(C)ccc(C)c1O N1(C(C(C)n2cccc2)=O)CC2(C1)CN(C(=O)C(F)OC(F)(F)F)CCO2 C(C)(CCC(=O)NCC(=O)NCC(N1CCOCC1)C)SC C1(CC(=O)N)(OCCNC(C(CC)C)=O)CCCCC1.c1cc(C)nn1C c1(SCC(=O)NCC(C)NC(C2(C#C)CC2)=O)nccc(OC)n1 C1(C(=O)NCC(CN(C)C(C2(C(C)(C)O)CCC2)=O)O)CC2(C1)CC2F c1(-c2cn(CC(C)NC(C3C(CCC)C3)=O)nn2)nc(C)c(C)s1 C1(C(N(c2ccsc2)CC)=O)CC12CCN(C(=O)C(C)C)C2 C12(NC(=O)CC3CCC4CC34)CCC(CC1)N(C(=O)CC=Cc1ccccc1)C2 c1(NC)ncnc(NCCCc2ncc[nH]2)c1C CC(C(=O)NCCC1CCN(C(c2cc(F)ccc2Cl)=O)CC1)C1=CCCC1 c1(C(=O)NC(C2CCN(C(=O)C(C3CCCCC3)O)CC2)C)cn2ccnc2s1 CCC(=O)CCC(=O)N1CC(O)CC1(C)C(=O)NCCCc1ncn(C)n1 C(=O)(C1=C(C)CCC1)NCC1CN(C(CCOCCCOC)=O)CC1C C(=O)(CCC(C)C)N1CCC(C)(CNC(CCNC(C)=O)=O)C1.C(C)=O.N CC(C)(C(=O)NCCN(CC)C(C1C2COCC12)=O)C1CCCO1.CCO.O C=CCC(C)(C)CC(=O)NCCOC(C)(C)CNC(C1CCC(C)O1)=O N1(C(C(c2cc(C)sc2)(C)C)=O)CCC2(NC(c3ncncc3Cl)=O)CC2C1 c1(SC)ncc(CNC(C)C(C2CCCCC2)O)s1 Cc1ccc(C)c(CC(=O)NCC#CCNC(C2(C)CC2(Cl)Cl)=O)c1 CCCCCCC(CC)C(=O)N1CCN(C(=O)CSc2nncs2)CC2(CC2)C1 Cc1nocc1C(=O)NC(CNC(=O)C)C(C)C.C(=O)CCC1CCCC1 N1(C(C2(COC)CCN(C(=O)CCC3CC3(C)C)CC2)=O)CCCCCCC1C c1(OC)cc2ccc(Cl)nc2cc1S(=O)(=O)NCC1CCN(OC)CC1 N1(C(C2CCC(C)(F)CC2)=O)CC2CCN(C(=O)CCC3OCCO3)CC12 c1(OC)ccc2c(N3CCC(OC(=O)N(C)C)C3)nc(=NC(C)C(C)C)[nH]c2c1 Cc1cc(N)c(C)nc1C(=O)NC1CCCCC1NC(=O)CN1CCN(C)CC1 c1(C(N2CC(C(N)=O)C2)=O)ccc2sncc2c1.C1(C)(COC)CC1C=O C(=O)(CCCN=[N+]=[N-])N.n1(CC)nc(C2CC2)cc1C(=O)N(CCC)C(C)C CCC(CC)=CC(=O)NCC1CC1C c1(C(c2nnnn2C2CC(F)(F)C2)NC(c2cc(Br)cs2)C)cc(Cl)ccc1Cl c1(CC)ccccc1CCNC(=O)CCc1ccon1.C1(C)(C=O)CC(F)C1 C(=O)(C(CNC(c1cccc2cncn12)=O)CC(C)C)NCC(CC#C)(C)CO c1(C(=O)NC(C2CN(C(c3c(C)oc(C4CC4)n3)=O)C2)C)nccc2nn[nH]c12 C1(CC=O)CCCS(=O)(=O)C1.C1(OC)CC(C)N(C(c2coc(Cl)n2)=O)C1 c1(C(=O)NCC(C)(C)NC(CC(C)c2cnn(C)c2)=O)ccc(Cl)c(Cl)c1 C1(NC(C(=O)NC(CC(N)=O)c2cccs2)=O)CCCCC1O CC1(C)CCC(C(=O)NCC2(F)CCCN(C(c3cc4sccc4s3)=O)C2)CO1 C1(CC=C)(NC(=O)CSC(=N)N)CCCN(C(=O)C(C2CCC2)OC)C1 C1(Cn2cc(CC(=O)O)nn2)CCCCN1C(=O)COC1CCOC1 C#CC1(NC(C2CC(C(C)C)=NO2)=O)CCCCC1.C12(C)C=CCN1C2=O.O N1(C(C2C(C)OCC2)=O)CC2(CO)CC1(C(=O)NC(C)CO)C2 N1(C(CCC(Cn2cc(CNC(C)=O)nn2)(F)F)=O)CC2(CC1C)CC(F)(F)C2 N1(C(C(C)OC2CCCC2)=O)CC2CCN(C(=O)CCCS(N)(=O)=O)C2C1 N1(C(C2C(CCC)C2)=O)CCC(OCC(N2CC(C(=O)OC)C2)=O)CC1 N1(C(C(CC2CCCC2)NC(C2CCC=CCC2)=O)=O)CCc2nn[nH]c2C1 C(=O)(C(C)(C)CCCNC(c1nc(=N)cc[nH]1)=O)NC(CC)C1CC1 C1(CNC(CC(C)C2CC2)=O)CC(C(=O)Nc2cn(C)nc2O)=NO1 Cc1ccc(CCC(=O)NCCCNC(=O)CC2(O)CCCCC2)cn1 C1CC(C)(C)CN1C(=O)CC1CCC(C)O1.C1(OCC)C(C(=O)N)C1C C(=O)(CCCC(C)(C)C)N(CCOC)Cc1cc(Cl)c2c(Cl)[nH]nc2n1 C1(NC(C(C(C)C)OCC)=O)CCN(C(C2(C(F)F)CC2)=O)CC1C C1(NC(C2(C)CC(F)(F)C2)=O)CC2CCC1(NC(=O)CS)C2.c1cccs1 c1(C(C)C)ccc(CN2C(C(=O)NCCC3(C)OCCO3)CC3CC23)cc1 N1(C(CC2C(C)(C)C2)=O)CC2CCCC1C2CNC(=O)C1=C(Cl)CCOC1 C(CCCC(=O)NC1CN(C(c2occc2C(=O)OC)=O)CC1SC)OC N1(C(c2cc(C)c(C)s2)=O)CC2CCCC1CN(C(C1CCCC(C)(C)O1)=O)C2 C1(CCNC(CCCOCC)=O)CSCCN1C(C1CC1(C)C)=O c1(OC)cccnc1C(=O)NCc1cn(CC)nn1.C(=O)(CC)N.C1CC1 Cc1ccc(C(=O)NC2CCC(NC(=O)C(O)Cc3cnc[nH]3)C2)nc1C c1(C(N2C(CCNC(c3cn(C)nc3)=O)CCC2)=O)cccc2cccc(O)c12 N1(C(CCC(=O)NCC)=O)CC(C)C(NC(c2cnc(O)c(Cl)c2)=O)C(C)C1 C1(NC(c2n(CC=C)ccc2)=O)CC(F)(F)CC1.c1(C=O)cccc(Cl)c1O.N C=CC1(CC(=O)NCc2cc(OC)ns2)CN(C(=O)CN(C)CCOC)C1 c1(OC)ccc(C(N2CCCCC2CC)=O)cc1O.C1(C(=O)N)C(F)(F)C12CC2 c1(C(=O)NC(CC)CN(C)C(C2(N(C)C)CC2)=O)cn2c(Br)cnc2s1 N1(C(C(C)n2cccc2)=O)CCCN(C(=O)CCS(C)(=O)=O)CCC1 C(=O)(C1=COCCO1)N1CC(O)(CCNC(Cn2c(C)cnc2)=O)C1 C1(C(=O)NC2CCN(C(c3cc(OC)no3)=O)C2)(COC)CCCC1 N1(C(C2(C#C)CCC2)=O)CCN(C(C2CCC(F)(F)C2)=O)C(CO)C1 N1(C(C(CCC)O)=O)CCC(NC(c2sccc2C(C)C)=O)CC(C)(C)C1 c1(C(=O)OC)cc(C)nn1CC(=O)NC(C)CC.c1(CC(=O)N)cocn1 C1(NC(CCCC#C)=O)CCCC(C(=O)NCC(C2CC(C)(C)C2)O)CC1 N1(C(c2cc(C)c(C)o2)=O)CC2(CCN(C(=O)C(C)CC(N)=O)CC2)C1 c1(C(=O)NCC(C(=O)NC(C)CP(C)(C)=O)C)cc(=O)n(C)cn1 CC1(C)Cc2cccc(CNC3(c4nnnn4CCF)CC4CCC3CC4)c2O1 c1(C(=O)NCC2CCCN2C(C2COCCC2(F)F)=O)ccc2sncc2c1 C1(C(=O)NC2CCN(CC)CC2)CCN(C(=O)CCC2OCCO2)CC1(C)C C(=O)(C1=C(C)OCCS1)NC1(COC)CCN(C(CC(C=C)(C)O)=O)CC1 CCCCC(C)(F)C(=O)N(C)CCN(C(c1n[nH]c2c1CCC2)=O)C(C)C C1(NC(c2ccc(COC)o2)=O)CCN(C(=O)C(C)C(=O)OC)C1(C)C O=C(C(O)C(F)(F)F)N1CCCC1c1cn(CCCN2CCC(O)CC2)nn1 N1(C(N(CCO)Cc2ccc(OC)cc2)=O)CC2(CCOC(=O)N2)C1 c1(OC)cc(N)c(C(=O)NC(C)(C)CC)cc1F.C1(=CC(=O)N)CCCC1 C1(CN(C(Cc2c(CC)con2)=O)CC)CCCCN1C(=O)CCC(C)C C(CCCCCC(=O)NCCCn1cnnc1)NC(CC1N(C)CC=CC1)=O C1(C)(CCC)CCN(C(=O)C(CCF)NC(=O)COc2cccnc2)C1 C1(N)(CC(=O)OC)CCN(CCc2cc(F)ccc2Cl)CC1 C(=O)(C(CCN(C)C)NC(c1ccsc1Cl)=O)NC(C(=O)OC)CO N1(C(c2c(COC)cco2)=O)CCC2CCN(C(=O)CCn3cncn3)CC2C1 C1(NC(C2CCN(C)C2)=O)CCCN(C(=O)Cc2ccc(Cl)c(F)c2)CC1 C1(NC(=O)CSc2nc[nH]n2)CCN(C(c2cccnn2)=O)C12CC2 C(=O)(C(CC(C)C)NC(C1CC2CC2N1C(C1(OC)CCSC1)=O)=O)NC Cc1ccc(O)cc1C(=O)NCC1(C(=O)NCc2cnns2)CC12CCC2 C1(NC(C2C(C)CC(C)O2)=O)CN(c2nnco2)CC1S(C)(=O)=O CCC(CC(=O)N(C(C)CN(C(=O)CCN1CCN(C)CC1)C)C)SC N1(CCCCNC(CNC(N)=O)=O)CCCN(C(C2CCC3CCC23)=O)CC1 N1(C(c2c(C)c[nH]n2)=O)CCN2CCN(C(c3cc4cc[nH]c4cn3)=O)CC2C1 C1(C(=O)NCCC(C)CO)CCCN(CCN(CCO)CCO)CC1 n1(CC)nc(C)c(C(=O)NC2CN(C(=O)C(CC(C)C)OC)CCC2C)c1C c1(NCc2nccc(C(=O)Nc3onc(C)c3C)c2)ncc2[nH]ccc2n1 c1(C(=O)NC2CC(NC(C3CC(=O)NC(=O)N3)=O)C2)nc2ncc(Br)cc2[nH]1 N1(C(CCOC)=O)CC2CC1CCC2NC(c1cc(Cl)c(C)c(Br)c1)=O Cc1cc(C(N2CC(N(C(=O)CC3OCCC3C)C)C2)=O)c2[nH]cnc2c1 C1(Cn2c(C3CCCN(C(C)C)C3)nc(C)n2)COc2ccccc2O1 c1(Cc2n(-c3cn(CC)nc3)nc(C3CC3)n2)c[nH]c2ncccc12 c1(C(N(CC(=O)NC(c2ccon2)(C)C)CCC)=O)cc(O)ccc1C c1(C(N2C(C(=O)Nc3ccnn3C)CC(C)C2)=O)ccnc(Br)c1F N1(C(C2C(OCC)C2)=O)CC2CC(C1)C2.c1ccc(F)cc1.C(=O)(CC)N C12(NC(CN(C(=O)CN3CC(C)(C)C3)CC)=O)CC1CN(C)C2 CCC(CCOC)C(=O)NCC1CN(C)CCN1C(c1ccc(C)s1)=O CCC(F)(CNC(C1CCCCC1NC(=O)CCn1cnnn1)=O)CC CN(CC1CCc2ccccc21)N1CCc2c(C(F)(F)F)cccc2C1 CCC(C)C(C(=O)N(C)CCNC(=O)C(C)C)Nc1cc(C)ncc1C C12(C(N3CC(C(N)=O)C3)=O)CC(CO)(CN1C(C1CN(C(N)=O)C1)=O)C2 CN=c1[nH]c(C(=O)NC2CCN(C(=O)CC(C)C3CCCO3)CC2)cs1 c1(C(N2CC(CC)N(C(=O)C(C)Cn3ccnc3)CC2)=O)cnc2cc[nH]c2c1 n1(CCOCC)nnnc1C(C)(CCSC)NCC(N1CCOCC1)=O N1(C(C(C2CCCC2)OC)=O)CC=CC1(C(=O)NC)COC.c1ccoc1C.C c1(C(=O)NC2(CF)CN(C(C=Cc3ccn(C)c3)=O)C2)ccc(Cl)nc1N CC1CN(C(C2CCC(=O)CC2(C)C)=O)c2ccccc2N1CCO Cc1cc2ncnc(N3CC(C)CN(C(c4cc5n(n4)CCO5)=O)CC3C)c2[nH]1 c1(CC(=O)NC2CCOCC2N(C(=O)CC(F)(F)F)C2CC2)cccc(F)c1F N1(C(C(CC)(C)COC)=O)CC2(C1)CN(C(c1ccnnc1)=O)CCO2 N1(C(Cc2cc(C)[nH]n2)=O)CCCC(C)(C(N2CCC(CC(=O)O)C2)=O)C1 N1(C(c2c(CC)ocn2)=O)CCOC(C(=O)NC2(CC(C)(C)C)CC2)C1 C1(C=O)CCCC(C)(C)C1.C1(CN(C)C(C2CCC(=O)N2C)=O)CCCCC1.N N1(C(C(CC)(C)C)=O)CC2CCN(C(=O)C(C(=O)OC)c3ccccc3)C2C1 C1(CC(N2CCC(CCO)CC2)=O)CC2(C1)CN(C(c1cnc(OC)cn1)=O)C2 C#CCC(C)(C(=O)NCC1CCN(C)C1)NC(c1ccn(C)c1CC)=O C(CCCCC(=O)NCC(C(C)C)NC(=O)C=C=C(C)C)=CC Cc1c(C(=O)NCC(C)CNC(C2CCC(C)(C)C2)=O)oc2c1C(=O)CCC2 c1(C(=O)NCCC(C)NC(=O)CC2(C)CC2)ccc2c(c1)CCCS2(=O)=O N1(C(COCC(C)C)=O)CCOCC(NC(C2(C)CC=CCO2)=O)C1 c1(NCC)ccc(CNS(=O)(=O)CCCOC(C)=O)c(F)c1 C1(CNC(=O)CCC2CCOCC2)C(O)C(O)CN1C(=O)CC1CC2CC2C1 N1(C(C2(CC#C)CCCO2)=O)CC2C(C(=O)NCCc3cccc(O)n3)C2C1 C#Cc1ccc(C(=O)N(C2CCN(C(c3sccc3Cl)=O)CC2)CCCC)o1 N1(C(C2C(C)CC(=O)CC2)=O)C2CCC1CC(NC(=O)C(C)N(C)C)C2 C=CCC(F)(F)C(=O)NC1CN(C(=O)CCC(=O)OC(C)(C)C)CC1O CCCC(CCC)CC(=O)Nc1ccc(C(C)C(F)(F)F)cc1 c1cccc(C)n1.N1(C(CC2(COCC)CC2)=O)CC(CC)C1.C(=O)N N1(C(c2cc(C(C)C)on2)C(=O)NC(CC)(C)C)CCOCC(C)(O)C1 Cc1ccncc1C=CC(=O)NCC(n1cc(CN2CC3CC3C2)nn1)C Cc1c(C(N2CCCC(N(C(=O)CCC#N)C)C2)=O)oc2c(Cl)cccc12 c1(OCC=C)ccc(F)c(CN(C)Cc2ccc(F)cc2F)c1 C#CCC(C)(C(=O)Nc1cc(CO)cc(F)c1)NC(C1C=C(C)CS1)=O N1(C(C(CCN(C)C)O)=O)CC(NC(c2cccc(=O)o2)=O)CC12CCC2 N1(C(C=C(C)c2ccsc2)=O)CC2CC(NC(c3c(Cl)cnn3C(C)C)=O)C1C2 CC(C)CS(=O)(=O)CC(=O)N1CC(NC(=O)C(C)C)C(C(F)F)C1 C12(CNC(C3CSCCN3C(=O)CCc3cnn[nH]3)=O)CCCC(CO1)C2 C1(C(N(CC(=O)NC2CCOC2C2CC2)C(C)C)=O)CCC(=O)N(C)C1 O=C(NNc1cnc(Cl)cn1)C1CC2CCC(C1)S2 C1(NC(c2ccccc2OC2CC2)=O)CC2CC1N(C(=O)C#CC1CCC1)C2 C(C)(CNC(=O)C(C)SC)(CNC(c1snnc1C)=O)OC C1(C(=O)NCC(CCCC)NC(=O)CC(C)(C)C2CC2)CC(=O)NC1(C)C C1(C(N(CCCCN(C)C(c2ccnn2CCF)=O)C)=O)CCc2ccnn2C1 c1(C=O)cc(C)nn1CCO.C(C)(C(=O)NCC1CC1)N(C(C)=O)C.C CS(=O)c1cccc(C(N2CC3CC2C3NC(C2CC3(CC3)CN2C=O)=O)=O)c1 C(=O)(C(C)(CC#C)NC(c1cnc(S)nc1)=O)NC(C1CCOC1)C#C C1(N(C(=O)C(O)Cc2ccccn2)C)CCCN(C(=O)Cc2ccccc2)CC1 N1(C(CC(CC)SC)=O)CC2CC(C1)N(C(c1ncc(C)cc1C)=O)C2 C1(C(N(C2CCN(C(=O)CO)C2)CCC)=O)CCOC(C)(C)C1 N1(C(c2sc(C)c(C)c2C)=O)CC(NC(C2(F)CCOC2)=O)C2(CCOCC2)C1 C1(CS(=O)(=O)N(C)CC2CCOCC2)CCC2(CCCCCC2)O1 C(=O)(CCCC(=O)N1CCOCC1)NCC.C1(CC(=O)N(C)C)CCC(=O)NC1 N1(C(C)=O)CCCC2(C1)CN(S(=O)(=O)c1cccc(Br)c1Cl)CCO2 C1(NC(C(=C)C(F)(F)F)=O)CC2CCCC(C1)N2C(c1ccc2nn[nH]c2c1)=O C1(CNC(CCc2cc(C)no2)=O)CCN(C(c2c(C)cncc2C)=O)CC1C c1(O)ccccc1.C1(C(=O)OC)(CF)CCN(C(C2COC(=O)N2C)=O)C1 c1(C(=O)NC23CN(C(C=Cc4ccn(C)c4)=O)C(C2)C3)cccc2nc(O)[nH]c12 C(=O)(C(C)CNC(=O)CCc1cn(C)nn1)NC1CC(C(=O)OC)C1 c1(NCc2c(C)cco2)nc(N2Cc3ccc(Cl)c(Cl)c3C2)nc2c1ncn2C C1(C(=O)NCC2C3CN(C(CCC(C)OC)=O)CC32)CC(S(C)(=O)=O)C1 C(CC(C(=O)NCc1ccccn1)NC(=O)Cn1cnc(=N)[nH]1)=CC C12(C(N(CC(=O)OC)C)=O)CC(CN(C(c3cnn(C)n3)=O)C1)C2 c1(C(=O)OC)nn(CN2CCOCC2Cc2ccccc2)cc1[N+](=O)[O-] C1(NC(c2nc(C)nn2C)=O)COC2(C1)CN(C(=O)COC1CCCC1)C2 C(c1ccc(C)c(C)c1)=CC(=O)NCC(CC)(CC)NC(=O)CC.C(C)C N1(C(C(COC)N(C)C)=O)CC=C(C(=O)NCC(C(C)C)C(C)C)C1 c1(C(N2CCCC(CNC(C(F)=CCC)=O)C2)=O)cc(Cl)ccc1.CC(C)C CCCCC(O)C(=O)NC1CCCC1(C)CNC(c1c[nH]nc1[N+](=O)[O-])=O c1(C(=O)NCCCC)cc2c(Cl)cc(Cl)cc2[nH]1.C1(C(=O)N)COCC1C(F)F CCCCCCCCCCC(=O)NCC(CNC(c1c(F)cccc1Cl)=O)CO c1(C(N2CCCC(NC(C(N3C(=O)CCC3=O)C)=O)C2)=O)cnn2cccnc12 C1(NC(c2c(C)sc(Cl)n2)=O)CN(C(c2ccnc3c2CCC3)=O)CCC1(C)C N1(C(C(=O)NC(C)C)=O)CCN(C)C(CNC(C2CCCO2)=O)C1 C1(C#N)(C(=O)NC2CCN(CCNC(COCC)=O)CC2)CC12CCCC2 C1(CNC(C2CCN(C)C2)=O)CN(C(c2[nH]nc([N+](=O)[O-])c2Cl)=O)CC12CCC2 Cn1ncc2c1CC(CN1C(=O)CCN(CC3(CF)CCOCC3)C1=O)CC2 C(=O)(N=c1ccn(C2CCCCO2)[nH]1)Nc1cccc(OC)c1OC C(=O)(C1=CCc2ccccc21)N1CC(CNC(CC(=C=C)C)=O)C(OCC)C1 Cc1cccc2oc(NC3CCCN(C(=O)CCC4(C)CC4)CC3)nc12 Cc1cccc(OCC(=O)NC2CN(C(=O)CCS(C)=O)CCC2O)c1C C1(C(=O)NC2(C)CN(C(Cn3ccc(C(C)=O)n3)=O)C2)C2C3CCC(C3)C12 O(C=CC(=O)NC(C1CCN(C(C2(n3cccn3)CCC2)=O)C1)C)CC N1(C(C(c2ccc(OC)cc2)OC)=O)CC(NC(c2nncs2)=O)CCC1C CC1CN(C(C2CCCO2)=O)CCCN1C(C1CC1c1ccsc1)=O Cc1cc(F)c(OC(=O)C2=CCOC2)cc1F N1(C(c2ccc(C)cn2)=O)CCN(C(C2CCC(C)(C)OC2)=O)C(C(C)(C)C)C1 c1(C(N2CCC(N(C(=O)C(C(C)(C)C)OC)CCC)C2)=O)cc2cccnn2c1 C1(CC(=O)NC2CC(NC(C3N(C(CCCC)=O)CSC3)=O)C2)CCC(C)CO1 C1(CC)CN(C(=O)CCCC2CC2)CCC1NC(C1CCN(CC(C)C)C1)=O c1(CCN=C(NCC(c2cccc(C)c2)O)NCC(F)F)cn2ccccc2n1 C(=O)(CCCCCCN(C)C)NC1CN(C(C23CCC(C)(OC2)C3)=O)CC(F)C1 Cc1ncc(C(=O)NC2CSC(C(C)(C)C)C2)cn1 c1(C(c2n(CCOC)nnn2)NCCC(=O)NC(C)CC)ncc(C)nc1.O N1(C(C2CCN(C(C(CC)CC)=O)C2C(C)C)=O)CCC12CCSCC2 c1(NC(C(CC2CN(C(COCC(=C)C)=O)C2)F)=O)cc(C)c(O)cc1C c1(CS(=O)(=O)N(CC(=O)NC(CC#C)C(=O)O)CCO)ccc(Cl)cc1Cl c1(C(=O)NCC2(F)CN(C(CCN(C(C)=O)C)=O)C2)ccc(Cl)c(C)c1Cl CC1(NC(=O)CC2CN(C(=O)C(O)C3CCCC3)CCO2)CCCC1O c1(C(N(CC(C)N(C(=O)CC2CC(F)C2)C)C)=O)cc(N)c2ccccc2n1 CN1CC(O)CC1(C)C(=O)NCC1(CCNC(c2csc(S)n2)=O)CC1 N1(C(C2CCCC(C)CC2)=O)CCN(C(c2cccc3scnc23)=O)C2(CC2)C1 c1(OC)cccc(C)c1N(C1CC2CC1CN2)C(c1cnc(O)[nH]1)=O C12(C(N3C4C(NC(c5nn[nH]c5Cl)=O)CC(C4)C3)=O)C3CCC(CC13)C2(F)F C(=O)(C(CNC(=O)CNC1CC1)C(C)(C)C)N1C(CC)(CO)CCC1 N1(C(c2csc(Cc3ccccc3)n2)=O)CCC2(CC1)COCC(CO)O2 N1(C(C2(F)CN(Cc3n(C(C)C)ncc3)C2)=O)CCC2(CC1)CC(=O)NC2=O CCCCCC(O)C(=O)N1CC(CNC(=O)C(C)NC(=O)CC)C(F)(CO)C1 C1(NC(c2c(CC)csc2)=O)CCN(C(=O)C=CCOC)CC12CCC2 c1(C(N2CC=CC(C(=O)NC(c3cn(CC)nc3)C)C2)=O)cc(C)cc(C)n1 CC(C)C(CCO)NC(=O)CC1CN(Cc2c[nH]ccc2=N)C1 O=C(CCCN1CCCC1)NC(c1ccccc1)C(=O)NC1CNC1 CCC(C)C(=O)C(=O)N1CCC=CC1C(=O)NC1C2CCC1CC2 c1(CC)cc(NC(C2CC3CC3N2S(=O)(=O)CCCl)=O)n(C)n1 N1(C(C=C(CC)CC)=O)CCCCC1C(C)NC(=O)CCCc1ccncc1 CC(C)(C)CC(F)C(=O)NCC1CCCC(NC(=O)CCC(C)(C)C#N)C1 C1(C2CCN(C(=O)Cc3ccccn3)CC2)(NC(c2n(CC)ccn2)=O)CC1 c1(N2C(C)CC(CNC(=O)C(F)F)C2)ncc(C#N)cc1F c1(N2CCC(OC)(CO)C2)nc2c(c(=NCc3nccs3)[nH]1)CCCCCC2 NS(=O)(=O)c1ccc(C(N2CCC(C3CC3)C2C)=O)o1.C(=O)CCC1CCC1 N1(C(c2c(C)ncnc2O)=O)CCCC2(CCN(C(C3CCC(F)C3)=O)C2)C1 C(c1nc2ccccc2o1)=CC(=O)NCCC1CC(NC(C2C(C)C2C)=O)C1 c1(-c2n(CC)ccn2)cnc(OC)cc1NC(c1ccc(O)cc1)c1nccs1 C1(NC(C(CN(C(CCC(C)OCC)=O)C)C)=O)C2CCC3C(C2)CC13 C1(C(N(CCNC(c2ccc(F)s2)=O)CC)=O)COCC(C)O1 N1(C(COc2ccc(OC)cc2)=O)CC(NC(=O)C(C)O)C(N=[N+]=[N-])C1 c1(C(=O)OC)ccc(SC(C)CCNN(C2(CO)CCCC2)C)cc1 C1CCCCN(C(=O)CC2(O)CCOC2)C1.n1(CC)nc(C2CC2)cc1C(=O)N c1(OCC=C)nc(OC)nc(-n2cc(-c3nccn3C)nn2)n1 C1(C#N)(CC)CCN(C(=O)C(CC(F)F)N(C)C(c2cnn(C)n2)=O)CC1 CC(C)(C)C(C)(C)C(=O)NCC.C1CC(F)(F)C1.C1CN(C(=O)CC)C1.O C#CCC(O)C(=O)N1CCC(CNC(C2CC2c2ccccc2OC)=O)CC1 c1(C(c2cn(C)nc2)NC(=O)CCn2cc(-c3ccncc3)nn2)ccc(F)cc1 C#CC1(C(=O)N)CN(C(C2CC(=C3CC3)C2)=O)C1.C1(CC)CC2C=CC1C2 c1(CC(=O)NC2CN(C(c3nnc(C(C)C)s3)=O)C2)ccc2nn[nH]c2c1 C1(C)(NC(c2ccn(C(C)C)n2)=O)CCN(C(=O)C(C#N)C2CC2)C1 CC1CCN(N2CCC(CCc3cccc(C(F)(F)F)c3)CC2)C(C)C1 C12(CNC(c3cocc3)=O)CC(CO1)N(C(=O)CN1CC3CCC1C3)C2.C n1(CC(=O)N)cc(C)nn1.C1(C(=O)OC)CCN1C(=O)CC.c1ccsc1 C(=O)(C1=NOCC1)NCCN(C(C(C=C)OC)=O)C1CCCC1 C1(NC(C#CCNC(C2(CC#C)CC2)=O)=O)CCCN(C)C1C C1(NC(C(C)C)=O)CC(NC(=O)COC2(C)CCOCC2)CC1O C(=O)(CCCC(=C)C)NC1C(NC(CCCC#C)=O)CCC1 C1(NC(Cc2[nH]c(=N)sc2)=O)CN(C(=O)CC2(O)CCC2)CC2CCCC12 N1(C(C=CC)=O)CCC(CCCN2CCN(C(=O)Cn3cnnc3O)CC2)CC1 Cc1nn(C)c(Br)c1C(=O)NCC1CC1.c1(C=O)cc(C(F)F)[nH]n1.C N1(C(c2c(C)noc2C(F)(F)F)=O)CCC2C(CCN2C(c2cnco2)=O)C1 C(C1(O)CCc2cc(F)ccc21)NC(c1ncc(F)cc1C(F)(F)F)=O N1(C(C(CC)OC)=O)CC(F)(F)CC1(C)CNC(c1ccc2ncsc2c1)=O Cc1scc(C(=O)NC2CC2NC(=O)C(C(C)C)N2CCCS2(=O)=O)c1N c1(OC)cc(O)ccc1C(C)NC1CCCN(c2nccs2)C1 S(=O)(=O)(c1ccc(C(N2CC(NC(=O)CC(C)F)C(O)C2)=O)cn1)NC N1(C(C(C)C#N)=O)CC2CCC1CN2C(c1ccc(C(C)(C)C)c(Cl)c1)=O c1(OC)ccc(C(=O)N)c(C)n1.C1(C)CN(C(C2CC2c2ccccc2)=O)C1 c1(C(N2CCC(C(=O)NCC3(CCC)CC3)C2C)=O)cccn2ccnc12 N1(C(Cc2nc(=N)[nH][nH]2)=O)C2CCC1CC(NC(=O)CC1CC3CC3C1)C2 N1(C(C2CCC2c2ccccc2Cl)=O)CCCCC(OCC(F)(F)F)C1 C(=O)(C1=CS(=O)(=O)CCC1)N1C2CC(N(C(CC(C)OC)=O)C)CC1CC2 C(CCC(=O)NCC(N1CCC1C)=O)N(C(C)=O)C C1(OC)CCCN(C(=O)CC2CC(F)C2)C1.C1(CC(=O)N)CC(C(F)F)C1 CCC(C)(CO)C(=O)N1CCCC(N(C)C(c2ccnc(C(C)(C)C)n2)=O)CC1 C(CCCC(=O)NCC(O)C(N1CC(OC)CC1CO)=O)OCC C(=O)(CC(O)CC(C)C)N1CCN(CCNC(c2cc[nH]c(=NC)c2N)=O)CC1 C(=O)(C1=CC(C)C1)NCCC1CN(C(C(C)NS(CCC)(=O)=O)=O)C1 C#CC1(C(=O)NCCc2ccc(C)cc2)CCN(C(=O)C(c2ccccc2)C)C1 CC(C)C(C)(C)CNC(=O)C(C1CCCC1)NC(=O)CC1CSC1 N1(C(C(C)N2CCC2)=O)CCCCC1CNC(=O)CCc1cncc(Br)c1 c1(C(=O)NC(C(C(C)C)NC(CSC)=O)C)cnc(C)cc1Cl C=CCCCC(=O)N(C1CCN(C)CC1)CC(N1CCCC1)=O c1(CNC2(c3nnnn3-c3ccc(F)cc3)C(CNC)CCC2)c(C)cccc1C N1(C(C=CCOC)=O)CCCCC1C.c1(C(C(=O)N)C)ccc(C(F)(F)F)cc1 C(=O)(CC1CS(=O)(=O)c2ccccc21)N1CC(O)C1.C(C)(C(=O)NC)=CC.C C(CNC(c1nocc1Br)=O)(CC)(CC)NC(C(CC)NC(C)=O)=O CCC(C)CCC(=O)N1CCN(C)CC1C(=O)NCC1CCC1C CC(C)(C(=O)N1CCC1Cn1cc(CCC2CCOC2)nn1)c1cscc1Cl C=C1CC2CC1CN2C(C1CCCN(C(=O)C(O)CC)C1CC)=O N1(C(c2c(CC)scc2)=O)CC2CC(NC(=O)CC(C)C)C2C1.c1ccccc1.O S(=O)(=O)(c1cnc(NC2CCCn3ccnc32)c(Cl)c1)N1CCOCC(C)C1 C1(C2CN(C(=O)CC3CC(CF)C3)C2)(NC(c2cnn(C)c2S)=O)CC1 c1(CCC(=O)NCC=CCNC(CN(C)CC)=O)nc2ccccc2[nH]1 C1(NC(c2cc(C)cc(Cl)c2)=O)CCN(C(C2CCC(F)CC2)=O)CC1(C)C Cc1cc(C(N2CCCC(N(CCO)C(c3cc(O)ncn3)=O)C2)=O)cc(O)n1 O=C(CC1=CCCCC1)NC1(CO)CCCN(C(c2coc3c2COC3)=O)C1 c1(CC(=O)N)cn2cc(F)ccc2n1.C1(C(N)=O)(C)CN(C(C2CC2)=O)C1 C1(NC(COCCCC)=O)CN(C(=O)Cc2cn(CC)nn2)CCC1CO Cc1ccccc1-n1cc(COC2CCCC(C(F)(F)F)O2)cn1.c1nc(CC)no1 O=C(C(C)CC1CCCC1)NCc1cccc(CO)n1.C1(C=O)CCS1(=O)=O C(=O)(C1=Cc2ccccc2C1C)NC1CCC(NC(c2c(C)occ2)=O)CC1 N1(C(C=O)=O)CC(N(C(=O)C=Cc2ncco2)C)C(O)C1.CCCCO.CC N1(CCN(C(=O)CS(N)(=O)=O)C)CCN(C(=O)CCc2cncnc2O)CC1 c1(C(=O)NC2CCC(NC(C(C3CCCCC3)C)=O)CC2)ccn2cncc2c1 c1(C(C)C)ccc(F)c(C(=O)NCC2CC2)c1.c1(C=O)ccsc1C1CC1 N1(C(C(CC)NC(C)=O)=O)CC2CC2(NC(=O)C(C)(C)c2csc(C)c2)C1 C(=O)(CC(C)(F)F)NCCC(C)NC(c1cc(Cl)nn1C)=O CC1(C)CCCC(CC(=O)NCCCCCCNC(=O)Cc2cnns2)CC1 C12(CC(=O)NCC(c3scc(C)n3)C)CCC1CN(C(=O)CC1CCCCC1)C2 C1(CN(C(C2N(CC)CC2)=O)C)CCCN1C(=O)CCc1ccon1 C(=O)(CC(C(C)C)c1ccccc1)NCC1N(C(Cc2c(C)n(C)nc2)=O)CC1