SMILES c1(OC)cc(C(=O)NCC#CCNC(C2(OC)CC2)=O)cc(Br)c1OC CCCCC(C)(F)C(=O)N1CC(CC(C)(C)CNC(=O)CC(C)C2CCCCC2)C1 Cc1cc(NC(=O)COC2CN(C(C3C4CC(=O)CC34)=O)C2)cnc1C n1(C(C(=O)NC(C=C)C2CCC2)C)cc(CCS(C)(=O)=O)nn1 C1(NC(C2CC=CC(NC(c3c(C)n[nH]c3C)=O)C2)=O)CC(=O)NC(=O)C1 C1(COCC(=O)N(C2CCN(C(C3CCCO3)=O)C2)CC)CCOCC1 N1(C(C(C)C)=O)C(C)C2CC1C2NC(c1ccn(-c2cccnc2)n1)=O C1(NC(C2CSCC(=O)N2)=O)CC2CCC(C1)N2C(C1C2CCCCC12)=O C12(C=O)C3CC(CC13)C2(F)F.c1(C(=O)OC)ccoc1C(=O)NCCC C12(NC(c3nnc(C(F)(F)F)s3)=O)CC1CN(C(=O)CO)C2.C1CCCC1 N1(C(c2cnc(CSCC)s2)=O)CC(OC)C(c2cccc(F)c2)C1 N1(C(C)=O)CCCCC1CN(C(=O)CSCCNC=O)C.C(C)(C)C c1(OC)c(C)ccc(C(N2CCCC(NC(=O)CC(O)CC(C)C)C2)=O)c1F c1(C(N2CC(C(C)NC(=O)CC(O)c3ccccc3)C2)=O)ccnc(C2CC2)c1 C1(CNC(c2ccc(CC)nc2)=O)CN(C(=O)CCC(C)SC)C(C)(C)C1 c1(C(N2C(CNC(=O)C(O)C(F)F)CC(O)C2)=O)cn2cccnc2n1 C1(C2CCN(C(c3ncccc3O)=O)CC2)(NC(C(CC)COC)=O)CC1 N1(C(CSC(C)C)=O)C2CCC1C(NC(=O)C(C)Cc1ccnn1C)C2 C1(C(=O)NCC2C(NC(c3ccc(Cl)[nH]3)=O)CC2)CCc2nc[nH]c2C1 c1(SCC(=O)NC2CN(C(C=CCOC)=O)C3C2C3)nc2ccccc2n1C c1(CC)cccc2[nH]c(C(=O)NC3C4CC3N(C(=O)C(C3CCC3)O)C4)cc12 C#Cc1ccc(F)c(C(N2CCC(COC)(NC(c3ccc(F)cc3)=O)C2)=O)c1 N1(C(C(CC)(CC)c2ccccc2)=O)CCC2(NC(=O)C3=CCCC3)CCCC12 C1(C(N(C)CC2CCN(c3c(OC)cncn3)CC2)=O)CCCC2(C1)CC2(F)F c1(OC)c(C(=O)NC(C)CCCNC(c2cc(C#N)on2)=O)ccnc1F N1(C(Cc2cc(OC)no2)=O)CC(CNC(=O)C)CC(C)C1.CCN(C)C N1(C(C=CC)=O)CC(NC(=O)C(F)(F)c2nccn2CCC)C(C)C1 c1(C(N(C)CC2(NC(c3cnco3)=O)CC2)=O)cnn2ccn(C)c12 CC1C(C(=O)N2C(C(=O)NCc3cc(O)ncn3)CC3CCCC23)=NOC1C Cc1ccc(C(=O)NCC2(C)CCC(NC(c3cc(F)c[nH]3)=O)C2)nc1O C1(NC(C(C)N(C(=O)Cc2cccs2)CC)=O)CC2(C1)CC21CCC1 C(=O)(C(CNC(c1cc[nH]c2nccc1-2)=O)C(C)(C)C)NC(C)CC(C)(C)O CCCCC(O)C(C)C(=O)NC1(CCNC(=O)CC2OCCCC2(C)C)CCC1 C1(CNC(Cc2ccc(C)cc2)=O)CN(C(c2cc(Cl)no2)=O)CCC1CO C1(C)(C(=O)NCc2cnc(C)[nH]2)CCCN(C(=O)CCc2scnc2C)C1 C(=O)(CCC1=CCCCC1)N1C2C(C(N3CC(CN=[N+]=[N-])C3)=O)CC(C=C2)C1 CCCC(F)C(=O)NC1CCC(NC(C2(N(C)C)CCCSC2)=O)CC1 N1(C(C(C)CC(C)(C)C)=O)CCC2(NC(C3CC(N=[N+]=[N-])C3)=O)CCCCCC12 CC1CCOCC1C(=O)NCCN(C(c1coc(C2CCCCC2)n1)=O)C1CC1 Cc1cnc2n1CC(C(=O)NCC1(C)CCN(C(=O)CCC=CC(C)C)C1)CC2 C1(CC)CC(C(=O)NC2(C(=O)NCCSC)CCC2)CCC1=O NC(=O)CCCCC(=O)NCC1(C(=O)NC2CN3CCC2CC3)CCCC1 CC(F)(F)CC(=O)NCC1COC(CNC(C2CC2)=O)C1.C1CCC1.C Cn1nc(C(N2CC3CC3(NC(=O)C(C3CCOCC3)F)C2)=O)c(Cl)c1Cl Cc1cc(CC(=O)NC(C2CCCN2C(C2CCCS2)=O)C)ccc1CO C1(N(C)C(=O)C2CC2)CCCC2CN(C(=O)Cc3nccn3C)CC12 CC1(C#CC(=O)N2CCC(O)(CCNC(c3ccc(CO)cc3)=O)C2)CCCO1 CC1(C(=O)NC2CCN(C(c3snc4ccccc34)=O)C2)Cc2ccccc2C1 c1ccccc1C#N.CC(C)C(C(C)NC(=O)CC)NC(C12CC(F)(C1)C2)=O CC1CCN(C(c2sccc2F)=O)C(CNC(=O)CS(N)(=O)=O)C1 c1(C(C(=O)NCC#CCNC(C(COC)OC)=O)O)cc(Cl)cc(Cl)c1 C(=O)(N=c1[nH]nc2[nH]ccnc1-2)C1OCCN(C(C(=C)C(F)(F)F)=O)C1 C1(C(N2CC(CCO)(NC(c3ccc(COC)o3)=O)C2)=O)CCCC(=O)N1 CCC(C)C(C(=O)NC1CCN(C(c2c[nH]cc(Cl)c2=O)=O)C1)NC(=O)OC C(C)(c1cnn(C)c1)=CC(=O)NC(C(C)NC(CCCCC)=O)C(C)C C1(CNC(CC=C)=O)CCN(C(=O)CC(O)COCc2ccccc2)C12CC2 N1(C(C(C)P(C)(C)=O)=O)CCN(C(C2CN(C3CCC3)C2)=O)CC12CCC2 c1(C(=O)NC(C(=O)NC(c2cccs2)C)C(C)(C)C)n[nH]c2ccccc12 O=C(CCCC1CCC1)NC1CCC(NC(c2cc(C3CCOCC3)[nH]n2)=O)C1 C(C(C)(C)C#CC(=O)NCCOC1CC1(F)F)NC(CSSC)=O N1(C(CCC(C)=O)=O)CCC2(C(=O)NCC(=O)N(C)C)CC2C1 C1(C(N(C2CCCN(C(CNS(NC)(=O)=O)=O)C2)C)=O)CC2(CCO1)CC2 N1(C(CC(C(C)OC)NC(=O)C(O)CC(C)(C)C)=O)CCCC12CCCCC2 C1(C(N2CC(Cn3cc(-c4ncc(C)cn4)nn3)OCC2)=O)CC2COCC2C1 Cc1[nH]nc(Cl)c1C(=O)NC1CC(CO)N(C(=O)C(C)O)C1.c1ccncc1.C c1(C(=O)NCC2CCN(C(c3coc(C(F)F)n3)=O)C2)cccc2ccsc12 c1(CC)nc(C(=O)NCC2CCCC2)c(C)o1.n1(CC=O)ncc(Br)n1.N C1(C(N2CC(CC=C)(C(=O)N(C3CC3)C)C2)=O)COCCC1C.c1cccnc1 C1(C)(CC)C=C(C(=O)NCCCCOC)C1.C(c1cn(C)cn1)=CC=O.N CC(C)CCC(=O)NC(C1CCCN1C(c1sccc1C(F)F)=O)C Cc1nc(=N)[nH]cc1C(=O)NC1CCN(C(=O)C=C(Cl)Cl)C1 Cc1c(C(C)NC(=O)C(N2CC3(CCNC3=O)C2)=O)oc2ccccc12 n1(CCC)cccc1C(=O)NCCCC1CCCN1C(=O)CC1(O)CC1 N1(C(CSC(C)C)=O)CCC(NC(c2ncc(C(F)(F)F)cc2Cl)=O)C(C)C1 CC1(C)CN(C(C2OCCC2(C)C)=O)CC1CNC(c1cnc(N)c(Cl)c1)=O C1(C)(CNC(Cc2c(C)cco2)=O)CN(C(=O)C(F)(F)C(C)O)CC1C Cc1ncc(C(N2CCCCC2C(=O)NCC2CC3(CCC3)C2)=O)c(=N)[nH]1 c1(-n2cc(C3(O)CN(C(C)=O)C3)nn2)cccc(CNC(=O)C(C)(C)CO)c1 C#CC1(C)CCCN(C(C2CC(C)(C)CN2C(=O)CC2CCCSC2)=O)C1 c1(C(N2CCS(=O)C(C)(C)C2)C(=O)NCCCOC)ccc([Si](C)(C)C)cc1 C1(OC)CCCC(CC(=O)NCCCCCN(C(=O)CNC(=O)NC)C)C1 N=c1[nH]c2ccc(=NCCNc3ccc(C(F)(F)F)cn3)[nH]c2[nH]1 C(CCS(N)(=O)=O)c1cn(CCCC(=O)N2CC(CC)C2)nn1.c1cc(Cl)c(Cl)s1 C(=O)(CCC[N+](=O)[O-])NC(C(C)C)CCN(C(=O)CN1CCN(C)CC1)C C1(CNC(CCOCCC)=O)CC(NC(c2c[nH]nc2F)=O)C1(C)C c1(NC(CN(C(C2Cn3c(C)nnc3C2)=O)C)C)nc2c(cc1C#N)COCC2 N1(C(CCN(CCCCC)CC)=O)CC2CC(NC(c3ccnc(O)c3)=O)C2C1 Cc1cnc(C(=O)NC(C)(C(=O)N2CCC(OC(C)C)C2)C2CCC2)c[n+]1[O-] C1(CNC(CN(C(=O)OCC)C)=O)CCCN(C(C2CC(C)CCO2)=O)C1 c1(N2CCC(CCNC(CC(CC)C)=O)CC2)c(F)cc([N+](=O)[O-])cc1F N1(C(C(CC2CC2)NC(C2C(C)(C)CCO2)=O)=O)CCOCC2(CC2)C1 C#CC12CCC(C(=O)NC3CCC(NC(c4nccn4CC)=O)CC3)(CC1)CC2 c1(NC2(c3nnnn3C3CC3)C(CCCF)CCC2)ccc(OC(F)F)c(F)c1 c1(C(N2CC(C)(C)C(NC(=O)C(O)C(F)F)C2)=O)cccc2ccnn12 c1(C2(C(=O)NC3C(C(=O)Nc4ccccc4)C3)CC2)ccncc1Cl C12(C(=O)NC3CCN(C(Cc4cnc(C)s4)=O)CC3C)CCCC1CC(=O)CC2 c1(C(N2CCCC(N(C)Cc3c(C)cccc3C)C2)=O)cc(F)c(F)cc1Cl c1(SC)ccccc1CC(=O)NC(C)CN(C)C(C1CC2(CSC2)C1)=O Cc1nc2c([nH]1)C(C(=O)NC1CCCCC1NC(C13COCC(C1)C3)=O)CCC2 C(CC(=O)NC(CO)CCSC)(C(C)(C)C)NC(C(CCCOC)C)=O Cc1cc(-c2ccccc2)ccc1CNC(=O)C(C1CCCCO1)N C1(NC(C=CCCC(C)C)=O)CC(O)CN(C(=O)CCSCC(N)=O)C1 N1(C(C(CC(N)=O)O)=O)C2CCC1CN(C(=O)C(CC=CCl)c1ccccc1)C2 C(=O)(CC(C)C(C)(C)C)N1CCC(CC(=O)N(C2CCCC(C)C2C)C)C1(C)C C1(NC(C2CCN(C(C)=O)C2)=O)CCC(O)CN(C(=O)Cn2ncn(C)c2=O)C1 C(=O)(CCCCC=CC)N1CC(NC(C(CC#C)C2CC2)=O)C(OC)C1 c1(Oc2c(NC(N(C(C)C)CC)=O)cn(C)n2)cc(Br)ccc1F.C.O N1(C(CC(C(=C)C)OCC)=O)CC(NC(c2cnn(C)n2)=O)C2CCCC12 N1(C(C(C2CC2)SC)=O)CCN(C(c2ccc(C(C)C)cc2)=O)CC1CCO CCC1=NOC(CC(=O)NCC=CC(N2CCC(SC)C2)=O)C1 C(=O)(CC(C)C(C)C(C)C)NC1CCCC(NC(CSc2nc(C)[nH]n2)=O)C1 Cc1c(Cl)ccnc1C(=O)NCC1(NC(c2cc(C#N)c[nH]2)=O)CCCCC1C C1(CCC(=O)NCC=CC(C)(C)C)CCCCN(C(=O)CC2CCCOC2)C1 CP(C)(=O)c1cccc(C(N2CCCC(CNC(=O)CC3CCOC3)CC2)=O)n1 c1(C=O)cc(C2CC2)ccc1O.C(=O)(C1=NOC(C)C1)N1CC(COC)C1.C c1(C(=O)NCCC2CCN(C(CN(C(COC)=O)C)=O)C2)ccc(C)cc1.O c1(-c2n(-c3ccn(CCOC)n3)nc(CC(C)(C)CO)n2)ccc2n[nH]cc2n1 c1(N(C)C)ccc(C(N2CCC(C)(NC(c3csc(Cl)n3)=O)C2)=O)cc1F c1(NC(C2C(NS(CC(C)C)(=O)=O)C2)=O)cccc2nc(O)ccc12 C(=O)CC(C)C(C)C.C1(CSC)CCC(C(=O)NCCC2(C)CC2)O1.N CCC(CCCC(=O)N1CCC([N+](=O)[O-])CC1)NC(C1CC(=C2CCC2)C1)=O N1(C(CNC(C)=O)=O)CCCCCCC1C(=O)NC(C)CF c1(C2(C(=O)NCCN(C)CCC(N)=O)CC(N)C2)cccc(F)c1 c1(C(N2CC(CC=C(C)C)C(C)C2)c2cnccn2)c(C)cc(C)nc1Cl c1(-n2c(-c3cccn3C)nc(C)n2)cccc2c1CCCC2 C1(C(NC[Si](C)(C)C)=O)(COC)CN(C(=O)CC(O)C2CCCC2)C1 N1(C(CC2CC(C)C2)=O)CCC2C(NC(=O)CNC(N)=O)C2C1 C1(NC(C(C)SC(F)(F)F)=O)CCC(CNC(=O)C(C)S)C1.c1ncccn1 c1(C(N2CCC(CNC(CC(CC)(F)F)=O)C2)=O)ccnc2c1ccn2C C12(CNC(c3cc(OC)ns3)=O)COCCN1CCN(C(C1(O)COC1)=O)C2 C1(COC(=O)CC2CSCCS2)CCC2(CCCC2)O1 C1(C(=O)N)CC(O)CN1C(c1ccnn1C(C)C)=O.C(=O)(CCC)OCC C(=O)(C1CSc2ccccc21)N1CCN(C(c2ccc(CC)o2)=O)CC1COC CN1C(=O)CCC1C(c1ccccc1Br)NC1(c2nnnn2C2CCC2)CCC1 c1(C(N(CCCNC(C2COCCC2C)=O)CC)=O)cn2cc(C)sc2n1 CN(CCCC(=O)NC1CCN(C(=O)CN2CCCC2)CC1(C)C)N=O c1(CC=O)cccc(F)c1.Cc1ncc(C(C)N(C(=O)CC2CCC2)CC)s1 c1(C(=O)NC2CCCN(c3ncc(Br)cn3)C2)cccc(C(F)F)c1F CCCC(C(=O)NCC1(COC)CCN(C(=O)C=COCC)C1)OCC N1(C(C(CO)NC(C(C)C)=O)=O)CCN(C(=O)C=O)CC(C)(F)C1.CC(F)F.N CC1CN(C(=O)CC2CCC(C3CC3)O2)CC1NC(=O)C(=CC1CCCCC1)F C1(C=O)CC1[N+](=O)[O-].c1(C(=O)NCC2CC2)scnc1C(F)(F)F.C CC12CCC(C(=O)NC3CC3)(CO1)C2.C(c1ccc(C(F)F)cc1)=CC=O c1(OCC(=O)NC(C(C)NC(C2CCC(O)C2)=O)CO)ccc(Cl)cc1F N1(C(CC(CC)C(C)C)=O)CCCC2CN(C(=O)CC(=O)NC)CC12 Cc1ccc(C(C)C(=O)NC2CC(CNC(=O)Cc3ccc(Cl)cc3)C2)cc1 C1(CC(=O)N(CC(C)NC(C2CCC(C)CC2)=O)C)CCc2sccc2C1=O C=CCC(CC=C)C(=O)NCCOC1CN(C(=O)Cc2cc(C)cc(F)c2)C1 N1(C(C=Cc2ncc(C)[nH]2)=O)CC(NC(c2nccn2C)=O)CCC1C Cc1sc(O)nc1C(=O)NC1CC(O)C1.c1(C=O)c[nH]nc1C(F)(F)F.C c1(C(C=O)N(C2CC2)CC)ccc2nc(C)sc2c1.C(CC)SCCOC c1(C(=O)NC2C(CNC(c3n(C)nc(C)c3Cl)=O)CCC2)ccn2ccnc2c1 N1(C(C2(COC)CC2)=O)CCC(C2CC2)C1.c1(C=O)ccc(F)c(F)c1F.N CCCC(CNC(=O)CC1CCCOC1)C(=O)N(CC(F)(F)CC)C C(C1CCN(C(C2CC(C)(C)CCO2)=O)CC1)=CC(=O)N(C(C)C)CC c1(N2CC(CCOC)OCC2)nc2c(c(=NC(C)CC(F)(F)F)[nH]1)CCCC2 C1(N(C(CC(C)C)=O)C)CCCN(C(c2ccc(-c3ccc(F)cc3)s2)=O)CC1 C1(C(=O)NCC=CC(=O)NC2CCN(CCOC)C2)CCSC(C)C1 C1(C(N(CCF)CC)=O)COC2(C1)CN(C(=O)CC1CC(C)C1)C2 C1(CNC(CC(CC)O)=O)CC2CCC(C1)N2C(C1(C)C=CCCC1)=O C1(CNC(=O)C=CC=C(Cl)Cl)C(O)C(O)CN1C(=O)C=O.CC(F)F.N Cc1nc(Cl)ncc1NC(C12CC(CN(C(=O)CC3CC4C=CC3C4)C1)C2)=O C1(CN(C(C(=O)OC)(C)c2ccccn2)C)CC(C)(C)NC(=O)O1 c1(C(C)C)ccc(CC(=O)NC2CCN(Cc3ncoc3C3CC3)C2)cc1 c1(C(=O)NC2CCC(NC(c3cnc[nH]3)=O)CC2)cc2c([nH]1)CCOC2 c1(C(F)F)nc(C2CCN(CC(F)(F)F)CC2)n(CC2CC2)n1 C1(CC=O)COCC2(CCC2)O1.C1(C(C)C)(CC)CC1C(=O)N.C1CCC1 N(C(=NCCCc1cccs1)NCc1n[nH]cc1Br)C(C=C)C c1(C(C)NC(c2nnc(C)s2)=O)ccc(F)cc1OCC1CCOCC1 C1(C(N2C(CC(C)C)COCC2)=O)CC(F)CN(C(=O)C(c2ccccc2)O)C1 N1(C(c2ccc(C)nc2)=O)CCN(C(c2cc(O)cc(O)n2)=O)C2CCCCC12 C1(CC)CCN(C(C2CCC(NC(c3ccnc(SC)c3)=O)CC2)=O)C1C C(=O)(CCN=C(NCc1cn2c(n1)CCCC2)NCC1CN(CC)CCO1)NC CN1C2(CCN(c3ncccc3S(C)(=O)=O)CC2)C(NC(=O)C=CI)CS1(=O)=O C1(C)(CC)CCCN(C(C2CCCN(C(c3ccc(C#N)n3C)=O)CC2)=O)C1 C1(CC(C)C)CCCCN1C(=O)NCC(c1ccccc1Cl)O C1(C(N2CC(CC(C(=O)NCC(C(C)C)C)F)C2)=O)CCOC1(C)C C1(NC2CCCC(OC)C2)CN(C(=O)OC(C)(C)C)CC(F)(F)C1 CCCCC(C(=O)NC1(CNC(c2cc(F)c(C)cc2Cl)=O)CCOC1)C(C)C S(=O)(=O)(c1ccc(Br)cc1Cl)N1C(C(=O)Nc2cnn(C(F)F)c2)CC(F)C1 N1(C(C(CC)(C)OC)=O)CCC(NC(=O)CCOCCOC)C2(CCC2)C1 N1(C(=O)CCC2CCC2)CCOC2(CCC(NC(C3(F)CC=CCC3)=O)CC2)C1 c1(N2CCC(Oc3ccc(C)cn3)CC2)ncnc(NC(=O)C#CC2CC2)c1C N1(C(c2cncc(OCC)c2)C(=O)NC(C)C(=O)OC)CCCC(C)(CC)C1 C#CC(C(C)OC)NC(C1(N(C)C(c2csc(C)c2)=O)CC1)=O C1(OC)CCC(C)N(C(C2OCCC2CNC(c2cnc(C)s2)=O)=O)C1 C1(CNC(=O)C(F)C2CCC2)CC2(CO1)CN(C(=O)C=Cc1ncc[nH]1)C2 C1(CCC(=O)N(CCCC)C)CCCCCC1.C1(CC(=O)N)(C(F)(F)F)CCC1 c1(C(N(CCCCNC(Cc2cc(CC)no2)=O)C)=O)cc(F)ccc1Cl N1(C(c2cnc(C)s2)=O)CC2CC1CN(C(=O)CC1C=NN(C)C1=O)C2 c1(NC(C2CC23CCNC3)=O)cc(F)c(O)c(F)c1.c1cc(Cl)c(F)c(Cl)c1.C c1(C(=O)NCCn2ccc(C(=O)NC3C(C)CCCC3)c2)nnc(O)nc1O CC1(C(=O)NCC(C)(C)OCC(=O)NCCN2CCCCC2)CCCCCC1 c1(C(=O)NCC2N(C(C3CCC(=O)NC3)=O)CCOC2)cc2c(Cl)cccc2[nH]1 C1(C(N2CCN(C(C3N(C)CCC3)=O)C(CCO)C2)=O)CC2(C1)CS(=O)(=O)C2 CC(C(C)(C)C(=O)N1CC(OC(=O)CO)C1)NC(=O)C(F)C(C)(C)O Cc1nc(C)c(C(=O)NC(C)CC(C)NC(c2cccn2C(C)C)=O)s1 N1(C(C(C)NC(=O)NC2CC(C)(Cc3cc(Br)no3)C2)=O)CCCCC1 CC1(CCNC(C2(F)CCCCC2)=O)CCN(C(=O)Cc2ccns2)C1 N1(C(c2ncc(C)c(Cl)c2)=O)CCC2(C1)CN(C(=O)Cc1cn(C)cn1)C2 C1(C(=O)NC(CNC(C(C=C)C)=O)CCCC)CCC(F)(F)CC1 C#CCCCC(C)C(=O)NC(CNC(c1c(C)[nH][nH]c1=N)=O)CC(C)C C1(CC)CCOC1C(=O)NCC1CN(C(C2(COC)CC(=O)C2)=O)C1 Cc1ccc(C(=O)NC(C2CCCN2C(c2c[nH]c(=O)cn2)=O)C)c(Cl)c1 c1(CC(=O)NCC2CCN(C(C3C4CC5C(C4)C35)=O)C2)ccc(Cl)c(Cl)c1 N1(C(c2ccc(I)cc2)C(=O)NCCC)Cc2cnc(C(F)(F)F)nc2C1 CC(CNC(=O)C=CC(=O)NC1CC1)C(F)C=O.CC(O)CC(F)(F)F c1(C(=O)NCC(C)(C)NC(C2C(C)OCC2)=O)cc2sc(F)cc2[nH]1 c1(SCCC(N2CCC(C(N(CCC)C3CC3)=O)C2)=O)cc(OC)nn1C C1(C(CNC(C2(OC)CCSC2)=O)(C)O)CCN(C(c2ccc(O)nn2)=O)CC1 N1(C(C2N(C(CC(CC)O)=O)CCC2O)=O)CC(CN)C(F)(F)C1 C1(C(=O)NC2(C)CN(C(c3c(OC)cc(F)cc3)=O)C2)Cc2cc(C)ccc2S1 C#CCC(C)(C)C(=O)N1CCC(C(C)NC(=O)CCCCF)CC1 C1(CC(=O)NC2(CO)CC(C)C2)CCC1(C)C.C1(CC(=O)N)CC(=O)C1 c1(C(C)NCCNC(=O)OC(C)(C)C)nnc2ccccn12.c1nccs1.C N1(C(C(c2n(C)cnc2)O)=O)CCC2CCC(C1)N2C(=O)C(F)(F)CO c1(CC)cccc(C)c1.C1(C=O)CC2(CC2)CN1C(=O)CC1OCCC1(C)C.N O=C(C1CCCCc2ccccc21)NCC1COCCN1C(=O)CSC(F)(F)F C1(COC)CCN(C(=O)C=CC2CCCN2C)CC1.C(=O)(C(C)n1cccn1)N N1(C(C2(F)CCN(C(C(C(C)C)C#N)=O)C2)=O)CCCc2ccccc21 N1(C(C(C(C)(C)C)=O)=O)CC2(C=C(C(=O)NC3CC(CCO)C3)CO2)C1 c1(C(=O)NC2C3N(C(Cc4cn(CC)nc4)=O)C(CC3)C2)cccc2[nH]ncc12 C(=O)(C1CCOc2c(F)cccc21)NC1(COC)C(C)(C)C1(C)C Cc1cnc(C(N2CCC(C)C(NC(=O)CC3(CO)CCC3)C2)=O)c(C)c1 N1(C(C2N(C(c3ccc(C#N)o3)=O)CC(=O)C2)=O)C2CCCC1CC2 C12(NC(C(C)N(C)C)=O)CCCC1N(C(=O)CC1SC3=NCCN3C1=O)CC2 N1(C(N(c2ccnn2Cc2cc(Br)cs2)C)=O)CC2(C1)OC1(C)CC2(C#N)C1 N1(C(CC=CCC)=O)CC=C(CC(=O)NCC(C)(C)C(C)(C)C)CC1 C1(C(N2CCC(C(C)NC(c3ncccc3N)=O)C2)=O)CN(C)CCN(C)C1 O=C(CCc1ccco1)NCC(O)CNC(=O)COCC1CCCO1 C1(C)(CNC(C2C(CC)CCO2)=O)CCCN(C(c2cnc3sccn23)=O)C1 c1(C(N(CCCCN(C(CC=CCC)=O)C)C)=O)nc(Cl)c(Cl)s1 c1(C(=O)NCC2(C)CCCN2C(c2cc3n(n2)CCC3)=O)occ2c1CCOC2 CCCCCCC(F)C(=O)NC1CC(C)(NC(c2nccc(OC)c2O)=O)C1 c1(C(=O)NC2COCCN(C(=O)C=CC3CCCO3)C2)cc2nc(=O)ccn2[nH]1 Cc1nc(C)n(CC(=O)NC2CC(NC(C3(C(N)=O)CCC3)=O)CC2O)n1 C1(OC)CCCCCC1NC(=O)CCCCNC(=O)C(C1CCC1)OC N1(C(=O)CC2CCC(F)(F)C2)CCCCC1C1CCCN1c1nnc(C2CC2)o1 C(C(CC(=O)NC1COCCN(C(c2ccncn2)=O)C1)C(F)(F)F)N(C)C C(=O)(C(C)(F)C(=O)N(C)CCN(C(=O)C(F)C(C)(C)O)C(C)C)OC N1(C(Cc2c(C)cccc2)=O)CCC(F)(C(=O)Nn2ccnn2)CC1 N1(C(c2c(C)nccn2)=O)CCCN(C(C2CN(C(C)C)C2)=O)C(CO)C1 C(=O)(CC(C(F)F)c1ccccc1)NC(CNC(c1c(C(C)C)noc1)=O)(C)C c1(COC(=O)NCC(=O)Nc2ccccc2)cccc2cnncc12 Cc1nc(O)nc(C)c1CC(N1CC(NC(c2cn(C)cn2)=O)C(C)C1)=O C1(F)(C(N2C(CNC(c3cnn(C(F)F)c3)=O)CC2)=O)CCOCC1 CS(C)(=O)=NC(=O)C(=O)N1CCCC(CNC(=O)CCCc2cc[nH]n2)C1 C1(CC(F)F)(C(=O)NCC(C)NC(c2ncoc2C2CC2)=O)CCOCC1 C1(C(=O)NCC2CCN(C(CCC(=O)OCC)=O)CC2)CNC(=O)CC1C C1(NC(Cc2n(C(C)C)cnn2)=O)CC(O)CN(C(c2cn(C)nc2CO)=O)C1 C(=O)(C1=COCCC1)NCC(CN(C(c1c(C)snn1)=O)C)(C)C C(=O)(CC(C)CCC)N1C(C(N(CCCC)CCCC)=O)CC2CC21 c1(OC)ncc(Br)cc1CC(=O)NC(C)CC(=O)NC(C)(C)C c1(C(N2CCCCC(CNC(COCCCC#C)=O)C2)=O)cc(C)c(C)cc1C c1(C=O)ccc(C)nc1C.C1(CCC)CCCC1.C1(C)(CC)CC1C(=O)NC C1CC(C=O)=NO1.C1(C(N(C)C)=O)(C(=O)NC)CC1.C(CO)C1(O)CC1 CC1CN2CCN1CC2C(N1CCC1)=O.C1(C(=O)N)CSCN1C(=O)C(C)(C)C C12CC(CO1)N(c1nccc(C(F)(F)F)n1)C2.n1(CC)cc(C(=O)N)c(C)n1 c1(OC)nccnc1C(=O)NCC(O)C(=O)N(CC(C(C)C)OC)C C1(C(=O)NCC(CNC(COCCC=C)=O)C)CNC(=O)CC12CCOC2 c1cccc(Cl)c1C.Cc1[nH]nc(-c2cn(C3C4CCC(F)C34)nn2)c1C c1(C2C(C(=O)NC3CC(CNC(C=C(C)Cl)=O)C3)C2)ccc(F)cc1 C=CCC(C)(CC)C(=O)NCC1CC(C(C)C)CCN1C(=O)C1=CCSC1 C1(C(=O)NC(C(=O)OC)C2CCOC2)CC(F)CN1c1ncccn1 C(C1CCN(C(=O)CC2CCOC2(C)C)CC1)=CC(=O)NCC(CC)(F)CC C(C(C(C)(C)C)NC(=O)C(F)(F)c1ccccn1)NC(CC(C)OC)=O C1(C(N(CCNC(c2c(CC)c[nH]n2)=O)C)=O)Cc2nncn2C1.C1CC1 C=C1CC(C)(C(N2CC(O)(C(F)C(=O)NCc3nc(=O)o[nH]3)C2)=O)C1 c1(-c2nnc(N(C)C3CC3)n2CC2CCCCO2)cc2cc(C#N)ccc2o1 N1(C(C(CC#C)C2CC2)=O)CCCC2CN(C(=O)C3=CCCS3)CCC12 C1(NC(Cc2cc(COC)on2)=O)CN(C(=O)C(O)CC)CC1C(F)(F)F c1(OC)ncccc1S(=O)(=O)N1CCOC(C(N2CCC(c3ccccc3)C2)=O)C1 C12(C(N(CC)Cc3ccc(C)c(Cl)n3)=O)CCCN(Cc3ccccc3)CC1C2 N1(C(Cc2cc(C)sc2)=O)CC2CCC1C2NC(c1cn(C)ccc1=O)=O C1(CC(=O)NC2C(NC(C=C3CCN(C)C3)=O)CCC2)CCCS1(=O)=O c1(CNC(c2n(CCCOC)nnn2)c2conc2C)nnc2n1CCCCC2 C1(C)(C(=O)NCC(CNC(COCC(=C)C)=O)(C)O)CCC(=O)NC1 N1(C(CC2CC(=O)NC2=O)=O)CC2(C(=O)NCC(F)CO)CC1CO2 C(=O)(C1CCc2nccn21)NC(C(=O)NCCC(=O)N(C)C)c1ccco1 c1(CC(=O)OC)ccc(NC(=O)C#CCCc2ccccc2)c(OC)c1 C(CC(=O)N(C)C)(C(C)C)OCC.c1(C(N2CCOCC2)=O)cc2c(s1)CCC2 N1(C(=O)OC(C)(C)C)C(C=O)CCC12CC2.C1(C=O)OCCC1(C)C.CC.N C(=O)(CC(C)C=C)N1C(CC(=O)NC2(CC#C)CCC2)CCC1 C1(CNC(CC(=O)N(C)C)=O)CC(NC(=O)CCCCC2CC2)CCO1 Cc1csc(=O)n1CC(=O)NC(C1(C)CC1)C.C1(C=O)CCS1(=O)=O.N C(CC(O)CC(=O)NC(CNC(=O)CNC(C)=O)C1CC1)SC C1(NC(CC2CCC(C)C2)=O)CC2CCC1CC2NC(=O)C(C)(C)CO C1(C2CCC2)(C(N(C2CCN(C(C(CC)(C)C#N)=O)CC2)CCO)=O)CC1(F)F c1(NC(C(C(C)c2ccccc2F)O)=O)cc(Br)cc2c1NC(=O)CO2 c1(C(=O)OC)c(C(=O)NC2CN(C(c3coc(C)n3)=O)CC2C)cnn1C c1(SC)ncc(C(=O)N(C2CCN(C(C3CN(C(N)=O)C3)=O)CC2)C)c(O)n1 C(CNC(c1csc(C#N)c1)=O)(CC(=O)N1CCC(CSC)C1)OC Cc1nc(C)c(C(N2CCC(CO)C(NC(=O)CC(C)CN(C)C)C2)=O)nc1C c1(C(N(C2C(C)CC2)C(C2OCCC2CNC)=O)=O)cccnc1O.c1ccco1 Cc1cc(C(N2CCC(O)(CN(C(=O)CC3CC=CC3)C)C2)=O)n2nccc2n1 C1(C(=O)NC(C)C(CO)NC(=O)C(F)=C2CCCC2)CCC2(CC1)CC2 C1(NC(c2nc(C)sc2)=O)CN(C(=O)Cc2csc(C3CC3)n2)C2CCCCC12 CCC(C)C(O)C(=O)NC1CN(c2cc(Cl)nc(C(C)(C)C)n2)CC1(C)C O=C(C#CC1CC1)NCC=C1CCN(C(=O)C(c2cccc(F)c2)O)CC1 CCC(C(=O)N(CC)CC1CCCN1C(c1cnc(OC)nc1)=O)C(C)C C1(NC(CCC(C)OC)=O)CN(C(c2cc(C(N)=O)cs2)=O)C2(CCC2)C1 S(=O)(=O)(c1cn(C)nc1C1CCCC1)N1C(CC#C)COCC1 CS(=O)(=O)CCC(=O)NCC1(C)CCC1.C1(CC=O)NC(=O)NC1=O.N c1(CNC(C(C)c2cccs2)=O)cc2n(n1)CCN(C(=O)C(F)=C1CCCC1)C2 C=CCCN=C(NCC(N1CCOCC1)(C)C)N1CCC(Cc2ncccc2C)C1 C1(CC(=O)NC2CC23CCCCCC3)CCc2sccc2C1=O c1(C(=O)N)nc(C2CC2)cs1.C1(CCNC(=O)CC2(CO)CC2)CCOC1 C(=O)(C(CO)C(F)(F)F)N1CCC(C)C1C(N1CC(CO)(CF)C1)=O Cc1ccc(CC(=O)NC2CN(C(=O)C(C)(O)C3CC3)CC2(C)C)cc1[N+](=O)[O-] Cc1cc(NC2CCCC3CN(C(=O)CN(C)C(N)=O)CC23)n2ncc(C)c2n1 C1(NC(c2nc(CCC)sc2)=O)(CO)CCCN(C(C2CCC23CCC3)=O)C1 c1(OC)cc(C)c(Br)cc1C(N1CCC(CNC(=O)CC2CCOC2)C1)=O Cc1cc(C(=O)NC(C)(C)CCCNC(=O)CC2CCC3CC23)cc(N)c1O C1(O)(CNC(Cc2c(C)nn(C)c2Cl)=O)CCCN(C(=O)C(F)C(C)C)CC1 N1(C(c2c(C)n(C(C)C)nc2)=O)CCC(NC(c2cc3n(n2)CCC3)=O)C12CC2 c1(C(=O)NC2(NC(=O)OC(C)(C)C)CCCOC2)cccc2c1CCCC2 Cc1nn2ccccc2c1C(=O)NC(CNC(C1CCC1(C)C)=O)CC(C)C C1(CCNC(C(=O)Nc2scc(C)n2)=O)CN(C(=O)O)CC1C.C(C)(C)C c1(OC)cc(CC(=O)N(CC)C2CC2)ccc1C.C(c1ccccc1)=CC=O.N N1(C2CCC(N)C2)CCN(c2ccnc(NCC3CCC(O)CC3)n2)CC1 C1(NC(CCN(C(c2cc[nH]c2C)=O)CC)=O)CCCC1C C1(OC)CN(C(C2CNC(=O)N2)=O)CC1C(N1CC(F)(F)C1)=O c1(C(=O)NCCC(C(C)C)NC(c2c(Cl)nsc2Cl)=O)cc(F)cc(F)c1 c1(OC)nn(C)cc1C(N1CCC(C)(C(N2CCC2(C)C(C)C)=O)C1)=O C(=O)(C1=CCCOC1)NC(C1CCN(C(=O)C=CCn2cncn2)C1)C Cc1cc(NC(=O)CN(C(=O)C(=C2CCCCC2)F)C2CC2)c(O)c(C)c1 C1(C(N(CCNC(C(C)C2CC2)=O)C)=O)CCc2ccnn2C1 C12(CNC(c3cccc(CC)c3)=O)CCC1CN(C(c1scc(C)c1)=O)C2.O c1(C=O)ccc2c(c1)OCCN2.C1(NC(CN(CCC)C)=O)CCC(C)(C)C1.N C1(CNC(Cc2c(C)ccnc2)=O)CN(C(=O)CCCCNC(N)=O)CCCO1 c1(OCC)ccccc1C=O.C1(C)CC1NC(=O)CN(C)C(=O)O CCC(F)(C(=O)N1CC(n2cc(CNC(C3CC3C)=O)nn2)C1)C=O.OC c1(OC)nc(C(=O)N(CCC(C)NC(=O)C(C(C)C)SC)C)ncc1F Cc1cc(N2CCC(CCNC(C3CCN(CC4CC4)CC3)=O)CC2)nc(Cl)n1 C=C(Cl)C(C)(C)C(=O)NCCN(C(=O)C(O)CSC)C1CC1 C1(NC(c2cnc(C)[nH]c2=N)=O)CN(C(c2c(Cl)cnn2C)=O)CC12CCC2 c1(C(=O)NCC2N(c3ccnc(C(C)C)n3)CCCC2)cc2[nH]ccc2s1 c1(C(=O)OCC)cnc2c(N3CCc4ccccc4C3C)cccc2c1 c1(N2CCC(CCOC)(NC(=O)CCC3CC3)C2)c(C#N)cccc1[N+](=O)[O-] c1(C(N2CCC(CNC(c3ccn(C(C)(C)C)c3)=O)C2)=O)noc2ncccc12 N1(Cc2ccc(NC(=O)CN3C(=O)CCC3=O)cc2O)CC2CCC1CNC2 C(C(C(=O)NC(C)CC(C)NC(c1sccc1OC(F)F)=O)OC)OC C(=O)(C1CCCc2sccc21)NC(C(C)C)CNC(C1C2CC3C(C2)C13)=O C12(C=O)CC3CC(C1)CC(O)(C3)C2.C1(C(=O)N)CC1(F)F.C(C)C1CC1 c1(NC(C2CN(C(C3(C#N)CC3)=O)C2)=O)ncc2[nH]ccc2n1 c1(C(C(=O)NC2C(CNC(C3(SC)CC3)=O)CCC2)C)c(F)cccc1F C1(C(=O)NCC2C(C)(C)CCCC2)CCC2(CCCCN2)CC1 c1(C(N2CCCC(C(C)NC(c3ccccc3O)=O)C2)=O)ccn2ccnc2c1 C(=O)(CC(F)(F)CC)NC(C(=O)NC(C#C)C(C)C)Cc1cn[nH]c1 c1(C(=O)NC2CC(NC(c3c(C)n(C)cc3)=O)C23CCC3)ccccc1[N+](=O)[O-] CC(CC(F)(F)F)C(=O)NCC(O)CC(=O)NC1(C(O)CO)CCC1 Cc1cc(C(=O)NCC(C)NC(c2cncc(Cl)n2)=O)cnc1F C1(O)CN(C(C2CCCCO2)=O)C1.c1(C(N(C)C)=O)coc(-c2cnn(C)c2)n1 CC1(C(=O)NCC(F)(F)CC2CC2)CN(C(c2ccc(C(F)F)o2)=O)C1 CN1CCOCC1C(=O)NC1CN(C(=O)CNC(N)=O)C1 n1(CC(=C)C)nnnc1C(c1c[nH]nc1C)NCCC(C)SC N1(C(C(C)OCC(F)F)=O)CCCCC1C(=O)N(C)CCC1CC1 Cc1cc(C(=O)NCC2CCN2C(=O)C(c2ccc(Cl)nc2)(C)C)c(C)s1 Cc1ncc(Br)cc1C(N1CCC2(CC2C(N2CCCC(F)C2)=O)C1)=O C1(NC(=O)Nc2c(CC)n(C)nc2)CCOC12CCOCC2 CC(C)C(C(=O)N1CCOC(C(=O)NC(C)C(=O)NO)C1)NC=O C1(C)(NC(C(CSC)C)=O)CCN(C(c2cc(O)nn2-c2ccccc2F)=O)C1 c1(C=O)cc2c(cc1Cl)OCO2.c1(OC)ccc(C(=O)NCCC2CC2)nc1.N N1(C(C2(NC(c3cn(CC=C)nc3)=O)CCCC2C)=O)CCC(O)(C2CC2)CC1 C(CCCC(=O)NCC1CCCCN1C(c1ccccc1C(N)=O)=O)OCC C12(NC(CCOCC)=O)CCCC1N(C(=O)CCCCCOCC)CC2 C#CCC(CC(F)F)C(=O)NC(CCC)CC(=O)N1CCC1CN=[N+]=[N-] c1(NC(c2ccc(C)o2)C)ccc(S(=O)(=O)NC2CCCc3occc32)cc1Br C1(NC(C2N(CC)CC2)=O)CC2CCC1CN(C(c1ccc(S(C)=O)cc1)=O)C2 c1(C(C(N2CCC(NCCNC(=O)OCC)CC2)=O)C)cccc2ccccc12 NS(=O)(=O)c1ccnc(C(=O)NC)c1.C1(F)CCC1.C1(CC=O)C=CCC1 C1(NC(C(C=CCCC)O)=O)CN(C(=O)C)CC(C)(C)C1.N1(C=O)CCCC1 c1(C(=O)N)cnc(N2CCOCC2)nc1.C1(NC(CSCCC)=O)(C)CCOC1 CC1CCn2ncc(C(N3C4CCC3CN(C(=O)C#CC3CCOC3)C4)=O)c2C1 C1(NC(C(CC)NC(C)=O)=O)CC(OC)CN(C(=O)Cc2c(C)cccc2C)C1 N1(C(c2c(C)cc(O)cc2)=O)CCCC(O)(CNC(=O)CC23CCCC2C3)CC1 C(c1c[nH]nc1C)=CC(=O)NCCN(CCCCCC)C(c1nc(O)sc1C)=O Cc1cc2c(C(=O)N3CC(n4cc(CCN(C)C)nn4)CO3)cccc2o1 c1(C(=O)NCC2CCN(C(C(CC)n3cncn3)=O)C2)c(F)ccc(Cl)c1F C1(OCC)CC(N(C(C(=O)NC2(C)CC2)c2ccco2)C)C1COC C1(NC(CC=C)=O)CC2CC(NC(c3cnn(CCO)c3C)=O)CC2C1 C1(CC(N2CCN(C(CNC(C3CCCS3)=O)=O)CC2)=O)CCS(=O)(=O)CC1 CC1(C)C(C)(C)C1(F)C(=O)N.CC1=CCCN(C(C2CC(n3ccnn3)C2)=O)C1 C(=O)(C(C)CCCC(C)=O)NCC1N(C(C(OC)OC)=O)CC(C)CC1 C(=O)(C(=O)N=S(C)(C)=O)N1CC(C)C(C)C1.c1(SC)ccc(Cl)c(C(=O)N)c1 c1(Nc2cncc(C(=O)NCC(C)(C)C(N)=O)c2)ncc2ccc(Br)cc2n1 C1(CC(=O)N(C(C)CNC(=O)Cc2ccnn2C)C)(CC=C)CCCC1 C1(CCC(C)C)CCN(C(=O)C(=O)N(CCN2C(=O)CCC2=O)C(C)C)CC1 CC1CCN(C(c2sc(C(F)F)nc2Br)C(=O)NCSc2ccccc2)C2(CC2)C1 c1(SC(C(=O)NC(C2CN(C(CN(CC)CC)=O)C2)C)C)ccccn1 C1(CNC(CCCOCCC)=O)CN(C)CCN1C(c1csc(C(F)F)n1)=O C(=O)C(C)(F)C(C)(C)F.c1(NC)ccc(C(N2CCCC2C2CC2)=O)cc1Cl.N N1(C(c2c(C)cc(Br)o2)=O)CCCN(C(C2CC(=C3CC3)C2)=O)C(C)C1 CC(C)CC(C(=O)NCC(C(=O)N(CC(C)(CO)CO)C)N(C)C)C(N)=O Cc1cc(=NC(=O)c2cccc(C(N3CCOCC3)=O)c2)c(C)c[nH]1 c1(OC)ccc2c(c1)OCC(NC(=O)C(=O)N(C)Cc1csc(C)n1)C2 CC(C)CC(CO)NC(C1C(O)CCN1c1ncc(Br)cn1)=O C=CCCCCCC(=O)N1CCC1CNC(c1cc(N)c(F)cc1C)=O C(CCCC(=O)N1CCC(N(C)C(C2CCOC(=O)N2)=O)C1)OC N1(C(=O)NC2CCC(COC)C2)CCC(CO)(OCC)CC1 C1(CC(=O)N(CC(=O)NC)C)CCC(NC(c2cccnc2OC)=O)CC1 C#Cc1ccc(C(=O)N(C2CCCN(C(=O)CN3CC=CC3)C2)C)cc1F C(=O)(NN1CCCC1C(=O)NCC#CCC)C1(C=C)CCC1 c1(CCN(C(CCC2CCCOC2)C(=O)NC)CCC)ccc(Br)cc1F c1(C(=O)NCCCCCCN(C)C(c2cn[nH]c2)=O)nccc(Cl)c1O CC#CCCCC(=O)NCC1C(C)CCN1C(C1CN(C2COC2)C1)=O N1(C(CC=CC=C)=O)CC2C3CCC(C2C1)N(C(=O)C(C)OCCCC)C3 c1(C(=O)OC)ccc2c(c1)N(CC1(C)CC(=O)N(C)C1)CCC2=O c1(C(=O)NCC2CCC(NC(c3n(CC)ccn3)=O)C2)cccc(Cl)c1N c1(NC(C2C3(CN(C(c4nc(COC)oc4)=O)C3)C2)=O)ccc(Br)cc1F c1(C(=O)NC(CNC(CCN(C(CCC)C)C)=O)CC)cnn(C)c1CC N1(C(=O)NCCc2scc(C(=O)OC)n2)CCC(C2CCOC2)CC1 c1(OC)cc(N)cc(C(=O)NC2CCCN(C(C)(C)C)C2)c1OC C(CC(=O)N1CCCC1CC(=O)OC)(C(F)F)NC(C(C)NC(=O)OC)=O O=C(CC(F)(F)Cl)NC(CNC(C1CCO1)=O)CO C=CCN=C(NCCC(C)CC)N1CCCC1.N1(CCC)CCOC1=O c1(C(N2CCN(C(C(CC(C)(C)C)(C)C)=O)CC2)=O)cc2n(n1)CCCNC2=O c1(C(=O)NC(C(C)NC(c2cc(CO)n(C)n2)=O)(C)C)nnn2c1CCC2 C1(=CCNC(c2cc(Cl)no2)=O)CCN(C(=O)C=Cc2ccccc2)CC1 n1(C(C)C)ncc(Cl)c1C(N1CC(N(C(=O)C=Cc2cnccn2)C)C1)=O C(=O)(CC(C)CCC)N(CCC(=O)NC(C)CCn1cncn1)CC=C Cn1nc2c(c1NC(=O)NCCc1cccnc1F)CCCC2 CC(CCNC(C1CC(CNC(=O)CC#N)C1)=O)N(C)C C1(NC(Cc2c(C)non2)=O)CCN(C(=O)Cc2c(C)noc2Cl)CC1CO CC1CN(C(=O)C2CC2)C1C(N1CC(OC(F)F)C1)=O.N1(CCO)CC(C)C1 C12(NC(c3cnc(CC(C)C)[nH]3)=O)CCCC1N(C(c1csc(CO)n1)=O)CC2 C(CC(C(C)C)NC(c1cscc1C(N)=O)=O)NC(c1c(C)nco1)=O c1(C(N2CC(C)N(S(=O)(=O)CC3CCC3)CC2)=O)c(F)cc(Cl)cc1F C(=O)(C(CC)C(=O)OC)NCC(CC=C)NC(C1(CCC=C)CC1)=O C1(NC(c2cnncc2O)=O)(CO)CCCN(C(=O)C(F)(F)C(O)C2CC2)C1 C#CC1(C(=O)NCCCCC(C)(F)F)CCN(C(=O)Cc2cnc(C)s2)CC1 C#CC1CN(C(C2(F)CCCN(C(=O)CC(C)=C=C)C2)=O)CCN1C c1(OC)cc(C(N2CC3CC3(CNC)C2)=O)cc(O)c1.c1cc(Cl)cc(Cl)c1 c1(C(=O)NC2C(C(C)C)N(C(c3ccc(F)cn3)=O)CC2)n[nH]c2c1CCSC2 C1(NC(c2c(C(C)C)ocn2)=O)CCCCC1NC(c1ccn(C)n1)=O C1(CC)CN(C(c2cncc(OC)c2)=O)CCC1NC(c1nc(C)ncc1Cl)=O N1(C(CCc2ccc(CC)cc2)=O)CCCCC(NC(c2cscc2C)=O)CC1 N(C(=NCC1CC12CC2)NC1CC1C(F)F)C(CC)CC N1(C(C2ON=C(C)C2)=O)CCN(C(c2n[nH]c(C3CC3)n2)=O)CC2(CC2)C1 c1(C(=O)NCC2CC(O)(CNC(C(CC#C)O)=O)C2)ccnc2ccnn12 C1(C(N(CC)CC)=O)CC(c2ccccn2)=NO1.C(=O)C(F)=CC1CC1.CO c1(CN2C(C(=O)NC3CC(=O)OC3)COCC2)ccc(Br)c(F)c1F n1(CC)ncc(NC(c2ccccc2)=O)c1C(F)(F)F.C12CCCC1(C)N2 N1(CCNC(c2ncc(OC)cn2)=O)CCCN(C(=O)CC2(O)CCOC2)CC1 n1(CC(C)C2CC2)ncc(Cl)c1C(N1CCOC(c2cn(C)cn2)C1)=O N1(C(C(C)OC)=O)CC2(CC(NC(c3ccc4ccnn4c3)=O)CO2)C1 C1(NC(=O)CCc2ccco2)CN(C(c2nc(C3CC3)ncc2Cl)=O)CC12CC2 C1(CC=O)CCCC2(CCC2)O1.c1(C(=O)NCCC(C)C)ccc(N)c(F)n1.N N1(C(c2c(CC)scc2)=O)CC2(CCC(CNC(c3ccno3)=O)O2)C1.C C(=O)(C1CCc2nccn21)NC(C(=O)NCC(c1ccsc1)C)CC(F)F N1(C(CN(c2ccc(C)cc2)CC)=O)CCCN(Cc2cccc(F)c2)CC1 CC(C)CCCCCC(=O)N1CCC2CN(C(c3cccc4cnsc34)=O)CC12 C1(NC(C(COC)OC)=O)CC2CCC1CN2C(=O)CC1OCCCO1 C1(C=O)CC2(C1)NC(=O)NC2=O.Cc1cc(C(N2CCC(C)C2C)=O)[nH]c1C.N C1(O)(CC(=O)NC(CCC2CCC2)C(=O)NCc2cnns2)CCCOC1 c1(C(=O)NC(COCC)C(=O)N(C2CCC2C)C)cnc(C)c(C#N)c1 CCC(CC(=O)N)c1ccc(C)cc1.C(=O)(C(C)(F)F)N(CCCN(C)C)CC c1(C(=O)NC(C(C2CCCCC2)NC(c2c(CC)scc2)=O)C)nn(C)cc1Cl C1(CN(C)C(C2CC(C)(F)C2)=O)CN(C(c2ccccc2CC#N)=O)CCO1 C(C1CCCCC1)=C(C(=O)NCC(CC)N(C(CCOCC#C)=O)C)F C1(NC(C=CCCC(C)C)=O)CCC(C)N(C(=O)C=C(Cl)Cl)C1 C1(O)(CNC(C)=O)CCN(C(=O)CCc2ccc(C#N)cc2)CC1 N1(C(CN(C2CCC2)C)=O)CCC(C(F)C)CC1.c1(C=O)ccc(C2CC2)o1.N C1(CNC(=O)Cc2cc[nH]n2)CCCC(NC(c2scnc2C2CC2)=O)C1 c1(NC2CC(c3n(C)cnn3)CC2O)ncc2[nH]c(=N)sc2n1 C(C1=NOC2(CCC2)C1)NC(C1(CNC(C(C)C#N)=O)CCCCC1)=O c1cccc([N+](=O)[O-])c1.CC(C)CCC(=O)NCC1CC(NC(=O)C)C(O)C1 N(C(=NCC(C)CSC)NCc1c(C(F)(F)F)cnn1C)C(COC)C c1(C(=O)NCC(CNC(C2C(=C)C2)=O)C)ccc2nc(C3CC3)[nH]c2c1 CCC(CN(C)C)C(=O)N1CCCC1C1CC1.C1(CC(=O)N)COC(C)(C)C1 Cc1ccc(C(=O)NCC2CC2NC(=O)C(N2CCOCC2)C)c(F)c1Cl C1(C(=O)NCC2CC(O)CN2C(=O)CCOCC(F)F)CC12CCSCC2 C(CC(=O)N1CC(C)(C)C1Cn1cc(CCCC#N)nn1)(C(F)(F)F)OC c1(C(N2CC(OC)CC2)=O)ccc(Cl)c(Cl)c1OC.C(=O)C(C)(C)CC(F)F.N c1(CC(N2CC(F)(CNC(C(CCOC)C)=O)C2)=O)coc2cc(F)ccc12 c1(C(=O)OC)[nH]c(COc2ccccc2NC(=O)OC(C)(C)C)cc1C C1(C(=O)NC(CNC(CCC(=O)NC)=O)CO)COc2cc(O)ccc2C1 N1(C(C2N(C(c3cnc(CC)s3)=O)CCOC2)=O)Cc2cccnc2C1 c1(CCC)ccccc1C(=O)NC(CNC(c1nc(Cl)sc1C)=O)CC C1(NC(C=C(C)C)=O)CC2(CCN(C(=O)Cc3cc(F)cc(F)c3)CC2)C1 c1(OC)c(C(N2CC(CNC(C3(C)CSC3)=O)CCC2C)=O)ccnc1Cl CN1CSCC1C(N1CCCC1CNC(C1(C)CC1C(F)(F)F)=O)=O C(=O)(CC(C)C(=O)OCC)NCC(CC=C)NC(c1ccc(CC)cc1F)=O c1(CCC(=O)NC2CCCC23CN(C(=O)CCC2CC2)C3)cccc([N+](=O)[O-])c1 Cc1cccc(NC(=O)C(=O)NC2C3CC2N(C(=O)CN2CSCCSC2)C3)c1 c1(NC(Cc2ccn(C)n2)=O)ccc(NC(=O)C=Cc2ccccc2)cc1F c1(OC)ccc(CCC(N2CCN(C(C3CC3(C)C)=O)CC2C(C)C)=O)cc1O N1(C(=O)CSC(F)F)CCN(C(=O)C2=CSCCO2)C(C2CC2)C1 C12(C(N3C(CCC(=O)N)CCCC3)=O)CCCC1C2(F)F.C(C)(C)OCC#C CON1CCC(C(=O)NCC2COCC2NC(=O)CCn2nc(C)nc2C)CC1 C1CCCC(C)(C)O1.C(C)(C)(C(=O)N1CC(F)(C(=O)N)C1)NC(=O)OC C1(C(N2CC=C(CNC(c3coc(O)n3)=O)CC2)=O)CCOC2(CCCC2)C1 CCC(CCOC)C(=O)N1CC(C)(C)CC1CC(=O)N(C1CCOC1)CC CC1C(NC(c2cnn(-c3ccncc3)c2)=O)CCCN1C(c1c[nH]c(Br)c1)=O c1ccc(Cl)c(F)c1.CCCC(O)C(=O)N1CC(CNC(=O)C(F)F)C(C)C1.O CC1=C(C(=O)NC(C)C2CC2)SCCO1.C1(C=O)CC(O)(c2ccccc2)C1.N N1(C(C(=O)NCCCC(=O)OCC)C2COC2)CC(C)NC(=O)C1(C)C c1(C(=O)NCC(C)CNC(C2CC2C)=O)ccc2ccc(Cl)cc2n1 C1(C(=O)NCCCCCc2nc(-c3cccs3)no2)COc2ccccc2O1 C1(n2cccn2)CCN(C=O)CC1.CC(CC1CCC1)NC(=O)N.C(C)(C)C c1(C(N2C(C)CCC(NC(C3CC(N(C)C)C3)=O)C2)=O)cc(F)cc(F)c1N C1(O)CCCN(C(c2nccn2C(C)C)=O)C1.c1(CCC)cc(C(=O)N)no1.C CC1CN(C(=O)CCCc2ccccn2)CC1NC(=O)CCc1nncs1 CN=c1[nH]c(=NCc2coc(C)c2)[nH]c(=NCC2(c3ccccc3)CCC2)[nH]1 N1(C(c2cc(CCNC(CN(CC)CC)=O)on2)=O)CCOC(C2CC2)CC1 C12(C=O)CC3CC(C1)CC(O)(C3)C2.N#Cc1ccc(C(=O)N)o1.C1CCC1.C CCCCCC(F)C(=O)N1CC(C(=O)NC(c2ccco2)CO)C(F)(F)C1 c1(C(=O)OC)cc(=NCCC2CCN(C(=O)CCCC(C)(C)C)CC2)[nH]c(C)n1 C(CN=c1cc(C(F)F)nc[nH]1)N(C(c1cc(C)n(C)n1)=O)C Cc1nc(-c2cccc(OC(C)(C)C)c2)n(C(C2CCOCC2)C)n1 N1(C(CC(=O)NCC)=O)CC(F)(F)CC1C.c1(C=O)[nH]c(C2CC2)nc1C.C C1(C(N(CCCCCNC(=O)C=Cc2cnc[nH]2)C)=O)C2CC3C(C2)C13 c1(CN2C(C(=O)Nc3cc(C)cc(C)n3)CC(F)C2)ccc2ccccc2c1O Cc1ncc(CC(=O)NC(Cn2ccnn2)C(=O)NCc2nc(CO)n[nH]2)s1 c1(N2CCC(CCCCCNC(CCC)=O)CC2)ncc2c(n1)COC2 CC1(C)CCCC1NC(c1ccc(CNC(=O)CC2CCSC2)o1)=O CC(CC(C)(F)F)C(=O)N1CCN(CC(C)NC(c2scnc2Cl)=O)CC1 C#Cc1c[nH]nc1C(=O)N(C)CCNC(C1CCC(OC(F)(F)F)CC1)=O CCP(=O)(CC)c1cccc(NC(=O)N(C(C)C)C2CC2)c1 c1(C(=O)NC2CN(C(=O)Cc3cnc[nH]3)C3CC23)c(F)cccc1F C1(NC(CC(=C)C)=O)CCN(C(=O)C(CCCC)N2CCCS2(=O)=O)C1(C)C c1(C(=O)NCCC2CCN(C(C(C3CCC3)OC)=O)C2)cccc(C)c1 N1(C(C(C2CC2)OCC)=O)CC(C)C2(CC2)C1.c1(CC(=O)N)ccoc1 N1(C(C(C)=CC)=O)CC2(CCCC2NC(=O)C=C2CCC(C)CC2)C1 c1(C(=O)NCCCCC2CN(C(C=CC)=O)C2)cc2c(s1)C(C)(C)CCC2 N1(C(c2cnc(CC)s2)=O)CCC(C(N2CCC(n3ccnc3)C2)=O)C1CC C1(C)(CC)CCN(C(=O)CCC2CC(NC(=O)CCCOC(C)C)C2)CC1 C12(NC(C(C)OCC)=O)CCCC1(F)CN(C(=O)C(C(C)C)C(C)C)C2 C1(CNC(CCNC(COC)=O)=O)CCN(C(c2ccncc2Cl)=O)C12CC2 N1(C(C(CN(CC)CC)F)=O)CCC2(CCN(C(C3(CF)CC3)=O)C2)C1 c1(-n2cc(CNC(CC3CCC(=O)N3)=O)nn2)cccnc1C(=O)O c1(C(N2CC=CC(NC(C=C(C)C(C)C)=O)C2)=O)cc2c(O)cccc2n1C c1(C(=O)NC(C(CC)C)C)c(CNC(c2cnsc2)=O)nnn1C C1CCCC2(CC2)C1.C1(C(=O)NC2CC(CC(=O)N)C2)CC2OC1C1CC21.C C1(NC(c2cc(CC)[nH]n2)=O)(COC)CCN(C(C2CCN(C)C2=O)=O)C1 c1(NC(C2(C)CCCN(C(CC)=O)C2)=O)cccc(F)c1C#N Cc1nc(N2CCCC(C)(NC(=O)C3=NOC(C(C)(C)C)C3)C2)cc(Cl)n1 C1(CNC(c2c(C)ccn2C)=O)C(C)CCCN1C(=O)C.C1(C)CCCC1.O c1(OC)ccc(C)c(C(N2CC(CNC(c3ccncc3)=O)(OC)C2)=O)n1 CC(C)S(=O)(=O)CC(=O)N1CCC(C)(CCNC(=O)Cc2cc[nH]c2)C1 C1(NC(=O)COCC2CCCO2)CC(NC(c2csc(S)n2)=O)CC1O C(=O)(C(C)C(C)NC(=O)Cc1cscn1)NCc1cc(COC)no1 N1(C(CC(COC)C)=O)CCC(N=[N+]=[N-])(C(N2C3CCC2COC3)=O)C1 C(C)(CC)(CC)NC(C1(CCOCC)CCC1)=O.c1(C(=O)N)ccno1 C(C(C(=O)N1CC(NC(c2cncn2C)=O)CCC(O)C1)C(C)(C)C)OCC=C N1(C(Cc2c(C)non2)=O)CCC2CC(NC(=O)C(F)(F)C3CC3)CCC2C1 C(=O)(C(F)CC(C)C)NCC(CC)NC(CCCCOCC)=O N1(C(=O)C=CCF)CCC2(CCN(C(=O)Cc3csc4nccn34)CC2)C1 CC(C)C1=NOC(C(=O)NCCC2CCCN(C(C3(C#N)CCC3)=O)CC2)C1 c1(C(N(C2CCCN(C(C3C(CCC)C3)=O)C2)C)=O)cc(N=S(C)(C)=O)ccn1 c1(C(=O)NC(C(=O)NCCC(CCC)C)(C)CSC)cccc(C)c1N N1(C(C=CC(C)(C)NC(C2N(C(C)C)CCC2)=O)=O)C2CCCC1CC2 N1(C(c2cncc(NC(CCc3ccc(OC)nc3)=O)c2)=O)CCC(C)C(O)C1 N1(C(c2cc(COC)[nH]n2)=O)CC(NC(c2nccc(C)n2)=O)CCC1C c1(C(=O)NCC2(NC(CCn3c(C)csc3=O)=O)CC2)nnc2n1CCCCC2 C(=O)(C(C)(C)C(F)(F)F)N1CCN(C(C2ON=C(C)C2)=O)C(c2ccncc2)C1 N1(C(CC(C)OC)=O)CCC(C(C)CNC(=O)C=Cc2cnn(C)c2)CC1 CC1CC=C(C(=O)N2CCC(C(C)C(=O)NCC(O)C(F)F)CC2)CC1 C1(NC(COCCC#C)=O)CS(=O)(=O)CC1NC(c1ccc[nH]1)=O N1(C(COCC(=O)NC)=O)CCOCC(F)(CNC(=O)CC)C1.C(C)C C1(C=O)CC(C)(C)CCO1.c1(OC)cc(C(=O)NCc2nccs2)ccn1.C C(=O)(C(C(C)NC(c1cnn(C)c1C#N)=O)C(C)C)N(CCCC(=O)NC)C C1(CC)CN(C(c2cnn(C)c2SC)=O)CCC1NC(C12CC(CO1)C2)=O N1(C(C(C=C)O)=O)CCCC(C2CN(C(=O)C=Cc3cccc(OC)c3)C2)C1 C(=O)(N1Cc2ccccc2CO1)C1C(C(N)=O)C1.C(=O)CCC1CC1CCO c1(OC)cc(C(N2CC(NC(=O)C(C)(C3CC3)OC)C(C)C2)=O)ccc1Cl C1(C)(CNC(C(C)CN(C)C(C2(CCCF)CC2)=O)=O)CC=CCC1 N1(C(c2cc(F)cc(N)c2N)=O)CC2CCCN(C(=O)Cc3csnn3)C2C1 N1(C(CC2N(C(CCC=C)=O)CCC2)=O)CCC(c2ccn(C)n2)CC1 CC(CCC(=O)NOCCO)NC(=O)CC1CCCNC1=O C(C(=O)Oc1ccc(N2CCCC2)cc1C)(C(C)(C)C)OC CC1CN(C(C2CCCC2(C)C)=O)CCN1C(c1ccncc1F)=O CCCCCC(C)CC(=O)NC1(CCC(=O)NCC2(C(C)(C)O)CC2)CCCC1 c1(OC)ccc(N)c(C(N2CCN(C(c3sc(Cl)cc3Br)=O)CC2)=O)c1 C1(C(NOCCCOCC)=O)CN(C(c2coc(N(C)C)n2)=O)CC1C(C)C c1(N2CCC(CC)(CO)C2)nc2c(F)cccc2c(=NCCOCCC(C)C)[nH]1 CC(C)(F)C(C)(F)CNC(C12CC(CN1C(C1(C)CC=CCC1)=O)C2)=O C12(C(N(C)Cc3c(C)noc3C)=O)CCCC1CN(C(C1C3CCC(F)C13)=O)C2 S(=O)(=O)(c1cccnc1C(=O)NCC)N(C)C.C(=O)CS(=O)(=O)C1CC1.N N1(C(=O)OC(C)(C)C)CC(C)C(C)(C)C1.c1(CC(=O)O)ccc(Br)cc1Cl CC(C)C(C(=O)NC1CC(O)CN(C(C2(O)CCCCCC2)=O)C1)C(C)C c1(OC)cc(CN2CCC(O)C(C(N3CCC(O)C3)=O)C2)cc(Cl)c1 C12(CNC(CC(C=C)C)=O)CCC1CN(C(=O)C(C)(C)CN1CCN(C)CC1)C2 N(C)(C1CCc2ccccc21)c1n(CC(C)Oc2cccc(Br)c2)nnn1 C(c1cnc(OC)nc1)=CC(=O)NC(CNC(c1ccc(C#C)o1)=O)CC(C)C c1(C(=O)NC(CC2CN(C(CNC(C)=O)=O)C2)C)cn(CCO)c(=O)nc1O c1(OC)cc(C(=O)N(C)C)cc(Cl)c1.C1CCCN(C(=O)Cc2cc(C)no2)C1 c1(N2CCC(NC(C3(C)ON=C(C)C3)=O)C(F)C2)ncnc2cc(C3CC3)nn12 Cc1cc(C(=O)NCC23CC(NC(=O)C=C(Cl)Cl)(C2)C3)cn(C)c1=O c1(OCC(N2CC(N(C(C(C)OC)=O)C)C2)=O)nn(C)cc1Br Cc1cc(C)c(CNC(C2CC(NC(=O)C(F)C(C)(C)O)C2)=O)cn1 C1(CC(=O)NCCC2CC(NC(C3(CC)CCCC3)=O)C2)CCN(C)CC1 C(CCCN=C(NCC1CCC1)N1CCC(C2CC2)C1)N(C)C N1(C(C2CCC(C)(C)C2)=O)CC2CC(C)C2C1.C1(CC=O)CCC(F)(F)CC1.N C1(NC(c2c(CC)c[nH]n2)=O)CCCC(N(C)C(C2CN(C(C)=O)C2)=O)C1 c1(SC)cccc(NC2CCCCN(C(=O)Cc3cnccc3C)C2)c1[N+](=O)[O-] C1(NC(C2(C(N)=O)CC2)=O)CCC(C(=O)NC2CCC2O)C1 c1(C(=O)NC(CN(C(c2cnn(-c3nccs3)c2)=O)CC)C)cccc(C)c1O C1(N(C(C(C)OCC#C)=O)C)CN(C(=O)CCc2ccc(C#C)cc2)CCC1C C=CCC(C(=O)NCC1(O)CC(C(=O)NCCOCCCC)C1)C(C)C c1(C(N2CCOC(C)C2(C)C)C(=O)NCC)ccc(OC)c([N+](=O)[O-])c1C N1(CCCC(=O)N(C2CN(C(C3(CF)COC3)=O)CC2F)C)C(=O)CCC1=O c1(CC)cnccc1C(=O)NC(CC(=O)NC(c1cnc(C)s1)C)C1CC1 C1(C(N)=O)CC2CCCCC2N1C(=O)C(c1ccccc1F)(F)F C1(CN(C)C)(NC(C2C(NCC)C2)=O)CCOCC1.c1cc(Br)c(Br)s1.S C#CC1CN(C(=O)CN2CCC(F)(F)C2)CCN1C(=O)CCC(=O)C1CC1 CC(C)CS(=O)(=O)CC(=O)NCC1CCCN1C(c1cn(C2CCOC2)nn1)=O C1(C(=O)N(C(C)C=O)C)(NC(COCCC#C)=O)CCC(C)(C)C1.CCF C1(CNC(c2ccncc2O)=O)CCCN(C(c2n[nH]cc2Cl)=O)C1 C1(C(=O)NC2CCC(OC(F)F)C2)(CSC)CCOCC1 C1(NC(c2cc3c(s2)CCC3)=O)CC2CCC1N2C(c1ccc(O)c(Br)c1)=O CN1CCC(C)(C(=O)NC2CC(C)(NC(C3CCO3)=O)C2)C1 C1(C(=O)OC)SCCN1C(=O)C(c1ccccc1)NC(N)=O c1(CC(=O)NCC(Cn2cc(C3CCC=CO3)nn2)OC)cc(Cl)ccc1Cl c1(NC2(CO)CCN(C(C=C(C)C(C)C)=O)CC2)ncc(C#N)c2ccsc12 Cc1ccc(CC(N2CC(CNC(=O)C=Cc3ccncc3)CC2C)=O)cc1Cl C12(C(=O)NC(C3CN(C(C4CCCC5CC45)=O)CCO3)C)CCC(CC1)C2 C12(NC(c3ccc4scnc4c3)=O)CCCC1CN(C(c1cnncc1O)=O)C2 C(=O)(NN=c1ccc2nccn2[nH]1)NCc1cncc(OC)c1 N1(C(C2N(C)CCCC2)=O)CC(NC(=O)CCCCc2cnn[nH]2)C2(CC2)C1 C1(CNC(c2n(C)c(S)nn2)=O)CCCC2(CN(C(=O)CSC(F)F)C2)O1 c1(C(=O)NC2C(NC(=O)Cc3cncc(F)c3)CCC2)c(F)cccc1Cl c1(C(N(C2CCCCC2N(C)C(C2CC3(CC3)CO2)=O)C)=O)cc(Cl)ccn1 c1(NC(C2CC(=C)CN2Cc2ncccc2C(=O)OC)=O)ncc(C)cc1Cl c1(C(=O)NCCC=CC=C)cc(CNC(=O)C)no1.C(C)(C)CC.O C1(CC)C(NC(C2CCC(O)CC2)=O)CCN1C(=O)CCc1ncccc1C Cn1ncc2ccc(C(=O)NC3C4CC3CN(C(c3ccsn3)=O)C4)cc12 CCCCC(C)CCC(=O)N1CC(C)C(C)(CNC(c2cnc(CC)nc2)=O)C1 c1(OC)cc(C(N2CCN(C(C3CCSCC3)=O)CC2CCO)=O)ccc1CO c1(C(=O)NCC23CC2CN(C(c2cnc(O)s2)=O)C3)ccc2nn[nH]c2c1 c1(OC)nc(C(N2CC(NC(=O)CCC3CCOC3)C(C)(C)C2)=O)ncc1F c1(OC)cc(OC)c(C(=O)N)cn1.C1C=CCC1.C(c1cn[nH]c1)=CC=O.C Cc1csc(NC(=O)NCCCCC=C)c1Br C(=O)(CCC(F)F)NCC(C(=O)NC)(C)C.C(=O)(C(O)CN1CCCC1)N Cc1ncnc(O)c1CCC(=O)NCC1CCCN(C(C)C(=O)NC(C)C)CC1 c1(C(=O)OC2C(CC)CC(C)CC2)cc(C)cc(Br)c1C O=C1COc2ccc(C(=O)NCC3CN(C(c4ccc(Br)c(Cl)n4)=O)C3)cc2N1 C12(NC(c3c(Cl)cn(C(C)(C)C)n3)=O)CCN(C(c3csc(O)n3)=O)CC1C2 c1(C(CCC(=O)NC(C2(c3c(Cl)cccc3Cl)CCC2)C)=O)ccc(O)c(F)c1 CON1CCC(C(N2CCCC(C(=O)NCCCOCC(F)F)CC2)=O)CC1 c1(C=O)cc2ccccc2o1.C1(CCNC(C2(C(C)(F)F)CC2)=O)CCCC1.N c1(C(N(CC(O)CN(C(=O)C(C)(C)O)C)C)=O)ccc(-n2cncn2)cn1 c1(C(=O)NC2CC(CCNC(CC3(C)CC3(F)F)=O)C2)cc(Cl)c(Cl)s1 C(=O)(CC(N)C(F)F)NC(C(CC)CC)c1cccs1 N#Cc1cccc(CN2CCC(C(=O)Nc3cccc(C(N)=O)c3)C(O)C2)n1 CCC(CNC(C1CCN(C(C2C3CCC(F)C23)=O)C12CC2)=O)(CC)CC c1(-c2cnc(C)nc2)cc(C(=O)Nc2c(C)cccc2[N+](=O)[O-])cc2[nH]ccc12 CC1=NOC(C)(C(=O)NCC(C)CN(C)C(C2(O)CCCCC2)=O)C1 c1(OC(C)C(=O)NCC(O)CCNC(c2cccc(=O)o2)=O)ccccc1F CC(C)CC(O)C(=O)NC(C(=O)NCC(=O)N(C)C1CC1)C1CC1 Cn1nc(CNC(=O)C=CCNC(=O)CC(O)C2CCCC2)n(C)c1=O Cc1nc(C(C)NC(C2(NC(c3cocn3)=O)CC(CO)C2)=O)no1 N1(C(C2C(C)OCCO2)=O)C(C(=O)NC(C)(C)C(O)C(F)F)CCC12CC2 Cc1cc(C(=O)NCC(CNC(=O)C(C)(C)c2cccnc2)CO)ccc1Cl C1(NC(c2[nH]cc(C(C)(C)C)c2)=O)CN(C(C2CCSC2)=O)CC12CCC2 CC1CCC=C1C(=O)NC1CCC1NC(c1cscc1C(N)=O)=O C(CCN(C(=O)CN1CCCC1=O)C)(C(C)C)NC(C1(CC)COC1)=O C1(CC(=O)NC2C(C)(C)CN(CC3CCOC3)C2)COc2ccccc2O1 Cc1cnncc1C(=O)NC(C(=O)NCCCCN=[N+]=[N-])C1CCCO1 C1(C=O)CN(C(C2OCCC2C(C)C)=O)C2(CCC2)C1.C(=O)(C(C)CC)OC C(=O)(C(F)(F)C(C)O)NC(C(C)C)CCN(C)C(c1ccnc(CO)c1)=O CC1(C)OCc2ccc(C(=O)N)cc2O1.C1(O)CN(C(=O)CC2(O)CCC2)C1.C c1(C(N2CC=CC(NC(c3nc[nH]c4ncnc3-4)=O)C2)=O)cc(O)cc(F)c1F c1(OCC)cc(C(=O)O)cc(Br)c1.N12CC(C1)CNC(=O)C2 N1(C(C(C2CC=CCC2)NC(CC=C=C)=O)=O)CC2(C1)NC(=O)NC2=O c1(C(C)NC(C(CSC)C)=O)ccc(C)cc1.c1(C=O)cc(C(N)=O)c[nH]1.N C1CCCC(C(=O)N(C2(C=O)CC2)C)CC1.c1(OCC)cc(C(=O)N)on1 N1(C(Cc2c(C)cc(O)cc2)=O)C2CCC1CC(NC(=O)CC(F)(F)C(C)C)C2 C(c1cncc(O)c1)=CC(N1CC(CNC(CCC=CCC=C)=O)OCC1)=O c1(C(=O)NCC2(O)CN(C(C(C)NC(CC)=O)=O)C2)ncc(Br)cc1O CC1CN(C(C2(CCN(C)C)CC2)=O)CCC1NC(C1(F)CCOC1C)=O C1(CC=C)(NC(=O)Cc2ccc(C)cc2)CCCN(C(C2NC(=O)OC2C)=O)C1 C1(CNC(C=C(CCC)CCC)=O)CN(C(=O)Cc2csnc2C)C(C)(C)C1 Cc1ncc(C(=O)NCCC2CCC2)cc1N.c1(C=O)ccc(C(C)(C)C)[nH]1.N Cc1cnc(C)c(C(N2CCC(N(C)C(c3ncncc3Cl)=O)C2)=O)c1 N1(C(=O)Cn2cnc([N+](=O)[O-])c2)CCC2(CC(NC(C3(C)CCC3)=O)CO2)C1 C=C(Cl)C(C)(C)C(=O)NCC(C)(C)CCNC(c1ccc(CO)nc1)=O C1(C(=O)NCCN(C)C)CCN(C(C2CC2C(F)(F)F)=O)C12CCC2 Cc1ncncc1C(=O)NCC1CCN1C(=O)CN(C1CCSC1)C C(CC(C(=O)NCC(C)(C)CN(C)C)NC(C1CCCSC1C)=O)OC CC(C)CCC(C(=O)NCC1CCC1)NC(C1CCCC(=O)C1)=O.C1CC1.C CC(C)CC(CNC(=O)C(C)(F)C(=O)NC)C(=O)NCCCSCCO Cc1cnc(C(=O)N(C(C)C(=O)NCc2ncccc2Cl)C)c(C)c1 C12(C(=O)NC3CC(COC)C3)CC(CN1C(=O)CC1CC=CC1)C2 Cc1nn(-c2ccccc2)c(C)c1CC(=O)OCc1ccc(C(N)=O)nc1 C1(N(C)C(C2CC3C=CC2C3)=O)CCCCN(C(=O)CN2C(=O)CNC2=O)C1 C(CC(C)C(=O)N(CC(C)C(=O)N1CC(N(C)CC)C1)C)=CC C#CC1CN(C(=O)C2=NNC(=O)CC2)CCN1C(=O)C(C)OCCN(C)C c1nc(-c2ccccc2)sc1CCO.C1(C)(CC(=O)NC(CC)C2CC2)CCCC1 C#Cc1cccc(C(=O)N(CCNC(=O)C(C)CC(C)CC)C(C)C)c1F CC(C)CCC(F)C(=O)N1CC(C(=O)N(C)Cc2cnco2)C(F)(F)C1 CC(C)C1=NOC(C(N2CCCC(C(C)C(=O)NC3C4CCCCCC34)C2)=O)C1 Cc1nc2cc(C(N3CCOCC3CNC(=O)COC3CCC3)=O)cnc2s1 c1(C(N(C(C)CCNC(=O)CC2COC3CC2C3)C)=O)cncc2ccccc12 N1(C(Cn2c(C(F)F)cc(C)n2)=O)CCC(NC(=O)CCC(C)N(C)C)CC1C c1(C(=O)NCCN(CCC)C(c2cnn(C)c2F)=O)ccc2snnc2c1 C1(C(N(CC(CN(C(CCN(C(C)=O)C)=O)C)O)C)=O)CN2CCN1CC2 c1(CC)nc(Cl)c(C)c(=NCc2ccccc2CNC(=O)C(C)(C)C)[nH]1 C1(CN(CC)Cc2cnc(Br)s2)CCN(C(=O)CC2(C)CNC2)CC1 C(CC(O)C(=O)N=c1ccn(CCF)[nH]1)NC(C(C(C)C)SC)=O C1(CNC(=O)C=CC(N2CCOCC2)=O)CCCCCN1C(c1cccnc1)=O N1(C(CCSc2nc(C)[nH]n2)=O)CCC(NC(=O)C(C)O)C(C)(C)C1 CCCC(CC)CCC(=O)NC(Cn1ccnn1)C(=O)N(C)CCc1cnc[nH]1 O=C(C1=CCCN(C(c2ccc3[nH]ccc3c2)=O)C1)Nc1cc(Cl)c(F)cc1Br c1(C(=O)Nc2ccc(Cl)nc2)cc2c(C3=CCNCC3)cccc2s1 C(=O)(C(C)(C)C(O)CC)NC(C=CC(N1CC(C=C)(CC)C1)=O)C c1(C(=O)NC(CC(C)NC(C2CC(SC)C2)=O)C)ccccc1CC#N c1(C(=O)N)ccc(F)c(O)c1.Cc1ncsc1C(N1CC(n2cc(C)nn2)C1)=O Cc1ccc(C(N2CC(NC(=O)CC3(C)CC3)CC(F)C2)=O)c(Br)c1 C(CCC(=O)NC(c1cn(C)cn1)C)NC(CNC(=O)OCC=C)=O C#CCCCC(C)C(=O)NCC(C)(C)C(N1CCC(O)(CO)CC1)=O c1(C(N2CC(CC)N(C(C3CCCCS3)=O)CC2)=O)cn2ncccc2n1 c1(N(CC(N2CC(CCNC(=O)CCn3cncn3)C2)=O)C)ccc(Cl)cc1 CC1=C(C(=O)N2CCC(NC(=O)C3=COCCO3)C(C(N)=O)C2)CCCO1 CC1CN(C(=O)C(C)(C)c2ccccc2)CCN1C(C1(CC(F)(F)F)CC1)=O C1(NC(COCC(=O)NC)=O)CN(C(c2cnncc2O)=O)CCC1C Cc1ccn(CC(=O)NC2CC(C(=O)NC3CC3C(C)(C)C)C2)c1 c1(N2CCC(N(C(=O)C(C)C3CCCO3)CC)CC2)c(C)c(C)nc2ncnn12 N1(C(CC(=C=C)C)=O)CC2CCC(NC(=O)CC3CCCCC3(C)C)(C2)C1 c1(C(N2CC(C)(C(=O)NOCC(N)=O)C2)=O)ccc(F)cc1F CCC(CC)(CC)C(=O)N1CCC(C)C(N(C)C(C2COC2)=O)C1 c1(NC(CN(C(C2CC(C)NC2)=O)C)=O)cc(F)ccc1O C(=O)(C1=NN(C)C(=O)CC1)NC1C(C(=O)Nc2cnc(C)c(Br)c2C)C1 C1(NC(c2ccc(COC)cc2)=O)CC(F)CN(C(=O)CC(C)(O)COC)C1 C12(NC(CC(CC)C)=O)CCCC1N(C(=O)COc1ccccc1C(F)F)CC2 N1(C(CCOCC(C)C)=O)CCCCC1C(=O)NCC1CC2CCC1O2 N1(C(CN(C(=O)OCC)C)=O)CCCC(CO)C1.C1(C=O)CC(=O)NC1.N C(=O)(C1=CC2CCC=CCCC12)NCCCNC(C12NC(=O)C3CC(C1)CC23)=O c1(N(C)CC)ccc(-c2nc(-c3cn(C)nn3)n(C(c3cnn(C)c3)C)n2)cc1 N1(C(C2N(C(C(C)Sc3cccs3)=O)C3C(C2)C3)=O)CCC(O)C(C)(CO)C1 c1(CC)ccc(C)cc1C(=O)N(CC(C)NC(C1CC(C)C(C=O)O1)=O)C CC1(CNC(c2nnnn2Cc2cccs2)c2ccoc2)CCC(=O)N1 N1(C(c2ccc(Cl)cn2)=O)CCN(C(=O)CCc2ccncc2)C(CCO)C1 c1(-c2ccc(CNC)c(C)c2)ccc2[nH]c(C(N3CC4CC3CN4C)=O)nc2c1 N1(C(CCSc2n(C)ccn2)=O)CC(NC(=O)C)CC(O)C1.C=O.C1CC1.N C1(C(=O)NCc2cn(CC(=C)CC)nn2)CCC(COCC(=O)OC)CC1 C1(CCCNC(CCC)=O)(CNC(=O)CCc2nccn2CC)CCCC1 CN1CC(C(=O)NCCC2CCCCN2CCSCC#N)CC1=O C1(COC(c2nn(C)c(C(F)F)c2)=O)CC12CCCCC2 c1(C(=O)NC2CCN(C(c3nccc(OC)c3F)=O)C2C)cccc2cnnn12 C1(OC)CCN(C(=NCCCNc2c(F)cccc2F)NC2CCCC2)C1 c1(C(N2C(C)CC(CNC(=O)Cn3cncn3)C2)=O)csc2c(Cl)cccc12 NC1CCCCC1CC(CC(N1CCC(SC(F)F)C1)=O)=O.c1ccccc1 CCC(C)C(C(=O)N(C)CC=CC(=O)NC1CC12CCC2)N(C)C C#CCCCCC(c1nnnn1-c1ccccc1Cl)NCC12CCC(CC1)OC2 C(CCC(=O)N1CCC(C)CC(C)C1)(C(C)C)NC(C(COC)(C)OC)=O c1(C(=O)NC2CC(NC(c3cccc(O)n3)=O)C2)ccc(-c2cnccn2)cc1 CCC1=C(C(=O)NC2CCC(NC(c3cnc(S(C)(=O)=O)s3)=O)C2)CCCO1 c1(OC)cc(C(=O)NC2CCC(C)C2)nnc1C1CC1.C(=O)CC.C(C)=O C1(C(=O)NCCOCC)Cc2ccccc2CN1C(=O)CN=Cc1ccco1 N1(C(c2[nH]c(=NC)sc2)=O)CC(NC(c2cc(F)c(F)c(F)c2)=O)C(C2CC2)C1 C=CC(CCC)CC(=O)NC1C2CC3C1C3C2C(=O)NCC1CC(CF)C1 C1(N(CCC=O)CCC)CC(C)(C)OC1=O.C1C=CCN(C(=O)C2CC2)C1.CO Cc1c(C(N2CC3(C2)CN(C(C2CC4C=CC2C4)=O)C3)=O)cc(C2CCC2)n1C Cc1c(CC(N2CC3CC2CN3C(=O)CC2COC(=O)C2)=O)cccc1Br C1(CC(=O)NC(CN(C(=O)CCc2cn[nH]c2)CC)C)COC(C)(C)CO1 Cc1cncc(-c2cn(C3CC4(C(N5CC(CS(C)=O)C5)=O)CC34)nn2)c1 C12(CNC(c3cn(C4CCOC4)nn3)=O)CC1CN(C(=O)C(F)F)C2 c1(C(NC2CCN(C(C3CC(=O)N(OC)C3)=O)C2)=O)nc2c(s1)COCC2.CC CCC(C)(C(=O)N1CC(CCNC(C2(C)CSC2)=O)C(C)C1)OC c1(OC)c(C(=O)NC(CCN(C(=O)CC(C)F)C)C(C)C)cc(F)cc1F C(CC(C)(C)C)(C(=O)N1CC(CC)C1)OC.N1(C2(C=O)CC2)CCCCC1=O.N C1(NC(COC(CC)C)=O)CCCC1(C)CNC(=O)CC1(O)CCOCC1 Cc1cc(C(=O)NC2(CN(C)C(c3cnc(CO)nc3C)=O)CC2)c(F)cc1F N1(CC)CC(C(=O)N(CCC(C)NC(C2(C(F)F)CCC2)=O)C)c2ccccc21 Cc1ccc(CNC(=O)C(C)NC(=O)CNC(C2CC2C)=O)s1 CN1CCOCC1C(=O)N(CCNC(C1(C)CC2CC2C1)=O)CC1CC1 C1(C(N2CCC(C(C)OC)CC2)=O)CC2CC1CN(C(C1CN(C(C)=O)C1)=O)C2 CC(C)CC(C)C(=O)N1CC2C(NC(c3cncc(N4CCOCC4)c3)=O)C2C1 C1(C(N(C(CNC(C(Br)=C(C)C)=O)Cc2ccccc2)C)=O)COC2COCC12 c1(C(=O)NC2CN(C(C3C(CC)OCC3)=O)C2)cc2c(cc1Cl)NC(=O)CO2 Cc1ccc(C(C)C(=O)NCC=CCC(=O)NCCC(C)O)o1 N1(C(c2c(C)coc2C)=O)CCC2(CO)CN(C(=O)CCOCC(C)C)CC2C1 C1(C(=O)NC(C)C(=O)NC2(CF)CC2)CCNC(=O)C1 Cc1nc2cc(C(N3CC(N(C(=O)C(C)N(C)C)C)C(O)C3)=O)ccc2o1 c1(CC(=O)NCC(CC=C)NC(C2CC2CC)=O)cnc(Cl)cc1C C1(C)(NC(CN(CCOC)C(c2cncc(CO)c2)=O)=O)CC(F)(F)C1 CN1CC(C(=O)NCC2(C)CCC(NC(=O)C=C(Cl)Cl)C2)NC1=O c1(C(=O)NC(CCCC)CO)cn2cc(-c3ccc4[nH]cc(C)c4c3)ccc2n1 C(=O)(CC(O)CCCC)NC(CCCCN(C(C1C(C=C)C1)=O)CC)C C(=O)(C1Cc2ccccc21)NC(CN(C(=O)CC1(C)CC1)C)(C)C C#CCC(C)(C(=O)N(C1CCN(C)C1)C)NC(=O)C(C)CCCC c1(CNC(C2(C)N(C)CC(O)C2)=O)nn(C)c2c1CN(C(c1ncc[nH]1)=O)CC2 N1(C(c2cc(CC)nnc2C)=O)CCC2CN(c3cc(CC)ncn3)CC2CC1 N1(C(C(COC(C)C)NC(C(CC)OC)=O)=O)CC2CCC(C1)C(=O)N2 c1(OC)cc2c(C(N3CC(NC(=O)CCCF)CC(C)(C)C3)=O)c[nH]c2cc1Cl Cn1cnc2ccc(NC(=O)CC3(C)CN(Cc4cccn5ccnc45)C3)cc12 c1(CC)ccc(CCC(C(=O)NC2CCOC2)N2CC3CCC3C2)cc1 C(=O)(C1SCCc2ccccc21)NC(C(CO)NC(C(CC(C)C)O)=O)C c1cc(F)ccc1F.c1(C(N(CC(C)(C)C)C)=O)cc(=O)n(C)o1.C(=O)C.N c1(CC(=O)NCCC(C)(C)C)cccc([N+](=O)[O-])c1.C(=O)(CC1=CCOCC1)N C12CCC(CN(C(=O)CC(O)C3CCCC3)C1)C2.NS(=O)(=O)C1(C(=O)N)CC1 C1(NC(CCC(=C)C)=O)CC2(NC(C3CCOCC3(C)C)=O)COC1C2 C1(C)(CNC(Cc2ccc(OC)cc2)=O)CC(OC)CN1C(c1csnc1Cl)=O C#Cc1ccc(C)c(NC(=O)C(CNC(=O)CSCCC#N)CC(C)C)c1 C(=O)(CCC(F)(F)F)N(CC(C)C(=O)N1CCC1C1CCCC1)C c1(N2C(CNC(C(CCC)OC)=O)C(C)CC2)nc(C(=O)OC)cc(C)n1 C12(C(=O)NCC3C(C)CCCC3)CC(C)(CN1C(C1COCC1(C)C)=O)C2 c1(N(CC=O)C)ccccc1[N+](=O)[O-].CCC(CC1CC1)C(=O)NC1CCC1.N C12(CC(=O)NC3CCCCN(C(C4CCC4)=O)C3)CC3CC(CC(C3)C1)C2 c1(NC(C=COCC)=O)sc2c(c1C(=O)N(c1ccc(C)cc1Br)C)CCCC2 C1(NC(=O)OC(C)(C)C)CCCOC1C1CCN(C(=O)NC2CCCC2)CC1 Cc1cn2c(n1)CC(C(=O)NC1CCN(C(c3cnn(C)c3C(F)F)=O)C1)CC2 C(CC(=O)NCC1CC(O)C12CCC2)(C(F)F)NC(c1cncc(CC)c1)=O Cc1c(C(=O)NCC(C)CC2(C)OCCO2)oc2c(C)cc(Br)cc12 C1(NC(C(C2CCCN(C(c3cnn[nH]3)=O)C2)C)=O)CN(C)CC1(C)C C1(C(=O)OC)CCN(Cc2ccn(C)c(=O)c2)CC1(C)C S(=O)(=O)(c1sccc1I)N1CCC(N)CC1CO N1(C(CC(C)(C)O)=O)CC2CCC1(CNC(c1coc(Cl)n1)=O)C2 C1(c2n(CCC=C)c(N3CCC4C(C3)C4(F)F)nn2)CCc2cnc(C)n2C1 Cc1cnc(C(=O)NCCC(C)NC(=O)C=C(C2CC2)C2CC2)cc1Br N1(C(C(CSC)O)=O)CC2CCCN(C(c3sc(C4CC4)nc3C)=O)C2C1 CC1(C)NC(=O)N(CCNCc2cc(Cl)c(F)cn2)C1=O C1(C(N(C)Cc2nc(C)on2)=O)C(C2CC2)CCN1C(=O)CCC1CCC(C)O1 c1(CNC(C(C)O)=O)ccc2c(c1)CCN(C(c1cncc3ncccc13)=O)C2 N1(C(Cc2n(C)ncc2)=O)CC(NC(C2CCC(C(C)(C)C)CC2)=O)CC(O)C1 c1(C(N(CC(O)CN(C)C(c2cn(C)cn2)=O)C)=O)ccccc1OC(F)F c1(CNC(C=CCOC)=O)c(C)nn2c1CN(C(=O)CC(COC)C)CC2 N1(C(c2c(CCC)n(C)nc2)=O)CC(NC(c2cccc(C#N)c2)=O)C(C)(C)C1 c1(C(C(=O)OCC)=O)ccc(NCCN(C(=O)CCC2CCCCO2)C)nc1 c1(NC(CC(C)C)CCO)cc(Br)ccc1S(=O)(=O)N1CCC(c2ccco2)C1 Cc1ccc(CNC(C2CC23CCN(C(=O)N(CCCCl)C(C)C)C3)=O)cc1F C1(N(C(c2ccn(CC)n2)=O)C)CN(C(=O)CCC2CCCN(C)C2)CC12CC2 c1(C(N2C3CN(C(c4cscc4F)=O)C(CC3)C2)=O)c[nH]c(=O)c2ccnn12 C1(C(N2CCC(N(C(C3N(C)CCCC3)=O)C)C2)=O)CCOC(C)(C)C1.C1CC1 c1(C(=O)NC(c2cn(CCC(C)C)nn2)CC(N)=O)cc(Br)cn(O)c1=O C1(NC(c2c(CCC)n(C)nn2)=O)CN(C(=O)C2=CCCS2)CC1S(C)(=O)=O CC1C(NC(=O)C(c2ccccc2)C2CC2)CCCN1C(C1CCC(F)CC1)=O c1(C(=O)NCC(=O)N(C)CC2(C)CCCO2)c(C)noc1N Cc1ccc(C(=O)Nc2cc(C(N3CCCC(C(N)=O)C3)=O)cc(Br)c2)c(O)n1 Cc1cccc(C2(CNC(=NCC3CCOC3)NC(C)CC(F)(F)F)CC2)c1 C1(CNC(C2(CC)CCC2)=O)CN(C(C2(OC)CCOC2)=O)CCC1(F)F c1(C(=O)NCC2C(C)CCN(C(C3CCCC3(C)C)=O)C2)cc([N+](=O)[O-])nn1C c1(C(=O)NCC#CCNC(CCc2cc(C)nc(C)c2)=O)c(O)cc(Cl)cc1F c1(C(N2C(CN(C(CCC3CCC(C)O3)=O)C)CCCC2)=O)cc(N)c(F)cn1 C1(NC(c2n[nH]c(CC)c2Cl)=O)CC2COC1C2.C1(C(=O)N)CCC2(CCC2)O1 Cn1cnc2c1CCCC2C(=O)NCC12CC(CO1)N(C(=O)C(C)(C)C#N)C2 CC1=C(C(=O)N2CC(F)(CNC(=O)C(C)(C)C(C)C)C2)C(C)(C)CCC1 C1(NC(c2c(C)c(Cl)c(Cl)s2)=O)CC2CCC1C(NC(C1CC1(F)F)=O)C2 C1(NC(CCCC)=O)CC2CC(NC(=O)C(Cc3ccccc3)C3CC3)C2C1 Cc1cccc2c(C(N3CC(CNC(=O)CC4CCCCC4O)C3)=O)n[nH]c12 CC(C)(C)CC(O)C(=O)N1CCOCC1CC(=O)NCCCn1cccn1 c1(C(N2CCCC(C)(NC(=O)Cc3csc(S)n3)C2)=O)cc2ccccc2o1 C(Cc1ccccc1)(CC(=O)N1CC(Cc2n(C)ccn2)C(O)C1)NN c1(CNC(NC2CN(C)C(=O)C2)=NCCF)c(F)c(F)c(F)c(F)c1F N1(C(CC2(OC)CN(C(c3ccn(C)n3)=O)C2)=O)CCn2c(C)cnc2C1 C(=O)(CS(=O)(=O)C1CCCC1)N1CCN(C(CCCN(C(C)C)C)=O)C(C)C1C CC(C)S(=O)(=O)C(C)C(=O)N1CCCC(O)(C)C1.C1(CC(=O)N)CN(C)C1 C=C(Br)CCC(=O)NC(C)(CNC(=O)CN1CCC(N(C)C)CC1)CC Cc1ccc(C(=O)N(CCCCNC(C2(C)CC2Br)=O)C)cc1F N1(C(C(CC=C)(C)C)=O)CCC(C2CCCN(C(c3nccs3)=O)C2)C1 CN1CC(NC(C2C=CCN(C(C3COCCN3C)=O)C2)=O)CC1(C)C N1(C(C=NOC)=O)CCOC(C2CN(C(=O)C(C)(C)c3csc(C)c3)C2)C1 C1(C(N(CC(C)NC(c2ncsc2C)=O)CC)=O)CCC(C)CC1 c1(C(=O)NC2CC(NC(c3ncc(OC)cc3F)=O)C2)ccc2nccnc2c1 N(C(=NCCCN1CCOCC1)NCc1ncccc1Cl)C1CC(OC)C1(C)C C1(C(=O)NC(c2cc(C(=O)O)on2)(C)C)CCc2ncsc2C1 C(=O)(C(CC(C)C)C(C)C)N(CCC)C(=O)Nc1ccc(-c2ccco2)nc1O C1(c2nc(CC)[nH]n2)CCN(C(C2(NC(=O)CN(C)C)CCC2)=O)CC1 C1(O)(C(C(=O)N)NC(C=C(COC)C)=O)CCCCC1.c1(CC)cn(C)cn1 C1(C(=O)NCC#CC(=O)N(C2CCCOC2)C)(OC)CCOC1 c1(C(C)C)cc(N(CCCCNC(=O)C(c2cccnc2)NC)C)nc(CO)n1 CCC(CC(=O)N1CCN(CCNC(C2CCS2(=O)=O)=O)CC1)C(C)(C)C C(C)(CO)(C(=O)N)NC(C)=O.C1(C)CCCN1C(C1CC2(CSC2)C1)=O.C N1(C(C(c2ccccc2)OC)=O)CCN(C(C2CC=CCC2)=O)C2COCC12 C#CC1C(C(=O)NC2CCN(C(=O)CC3CC=CCC3)C2)C1(C)C CC(C)C(F)(F)CNC(C1C2CN(C(C3CC(F)C(=O)N3)=O)CC12)=O C1(ONC(C2CCN(C(CN(C(COC)=O)C)=O)C2)=O)CCN(C)CC1 C12(NC(=O)Cc3ccc(F)c(F)c3)CCCCC1N(C(C1SCCS1)=O)CC2 CCC(C)(C)C(O)C(=O)NCCCC(C)NC(c1cc(C(F)F)ncn1)=O C=CC(O)(C(=O)N1C2CCCC1CN(C(=O)C(C)c1cccs1)C2)C(F)(F)F c1(C(=O)N)cn2ccnc2s1.C1(NC(=O)CCOC2CCOC2)CC(O)(C)C1 N1(C(C2(C)CSC2)=O)CCC2(CCN(C(=O)Cn3nnnc3C3CC3)C2)C1 CCCCC(CN=c1[nH]c2cccc(C)c2s1)NC(=O)CN(C)C(C)=O C(C)(C(=O)NCC1CC1(F)F)(C(C)C)OC.C(=O)C(C)CN(C)C.C C12(NC(C(CCC)OCC)=O)CCCC(NC(c3cc(OC)ccn3)=O)(C1)C2 C1(NC(C(C)(C)OCCC)=O)CN(C(C2CCCOC2)=O)CC1CC C1(CNC(C(CC)OCC)=O)CCN(C(=O)CCC(=O)c2ccc[nH]2)C1(C)C C1(CC(=O)N(C(C)CNC(c2nonc2N)=O)C)CCS(=O)(=O)CC1 C(=O)(C1CCCn2cnnc21)NCC(C)(C)CNC(=O)CCc1cncnc1 CC1CCC(CC(=O)NC(C(=O)NCCCCN2CCCC2)c2ccoc2)C1 c1(CCNC(CCC)(C)c2nnnn2C(C)(C)C)ccc(Br)cc1F c1(C(=O)NC(C2CN(C(c3cnc(O)nc3O)=O)C2)C)ncc(Cl)nc1Cl C1(CC(=O)N(C(C)C2CC2)C)CC(O)C12CCC2.C1(CC=O)CC1.CC.O N1(C(CSCC)=O)CCC2(CCN(C(c3ccc(N)cc3Cl)=O)CC2)C(C)C1 c1(-n2cc(CC3N(C(COC(CC)C)=O)CC=C3)nn2)ccc(Cl)cc1 C1(CNC(CC2(CNC(Cc3nc(C)oc3)=O)CC2)=O)CC(F)(F)CO1 N1(C(c2cn(CCCC)nn2)=O)CCC2(NC(=O)CSc3nncn3C)CC2C1 c1(-c2c(C)ccc(CO)c2)ccc2nnc(C(=O)Nc3onc(C)c3C)n2c1 c1(C(=O)NC(C2CCN(C(C3CC3C(N)=O)=O)CC2)C)cccc(N)c1O C#CCCC(O)C(=O)N1CCCC(NC(=O)CCNC(=O)NC)C1 C1CN(C(=O)COC(F)F)CCC12CCC2.c1(CC(C)C)c[nH]c(C(=O)NC)c1 c1(NC(CC)CNC(=O)C(CC)n2ccnc2)ncnc2c1CCO2 N1(C(C(C)C2CCCC2)=O)CCC(NC(c2cnn(CC(F)F)n2)=O)CC1 c1(-c2n(CCS(N)(=O)=O)nc(C(F)F)n2)cc(F)c(Cl)cc1Cl CCC(CC)C(C(=O)NC1CCC(F)(F)CC1)N(C)CCN1CCOC(C)(C)C1 C1(CC(N2CC(OCC(N)=O)C2)=O)C=CCC1.C(=O)(CC)N.C1CCCC1 C1(NC(CCN(C(c2cc(C)cc(F)c2)=O)C2CC2)=O)CCCC(C2CC2)C1 Cc1nn2c(c1C(N1CCC(CNC(=O)C(C)(Cl)Cl)CC1)=O)CCCC2 c1(N2CCC(C(C)NC(=O)C(F)CC3CC3)CC2)nc(Cl)ncc1C(F)(F)F C#Cc1cnn(C)c1C(=O)NC(C)CC(C)C.C1(CC(=O)N)CC(F)(F)C1 CC1CCCC1CC(=O)NC1(CN(C(=O)Cc2cnc(C3CC3)[nH]2)C)CC1 C(CCCCC(=O)NC1C2CCN(C(=O)CSC(C)C)CC12)=CC C1(COC)CN(C(c2cc(C)sc2N)=O)CCN1C(=O)CCC1CCCOC1 C(=O)(CCC(=O)C(C)(C)C)N1C(C)(C(=O)NC2CC(=O)N(C)C2=O)C=CC1 Cc1nn(C)c2c1CC(NC(=O)NCC(C)(C)Cn1cccn1)CC2 C(=O)(C(C)(C)C(C)C)N1CCN(c2ccc(OC)cc2)CC1 C1(NC(C2CCN(C)C2=O)=O)CC2CCC1N2C(c1ccc(C#N)cn1)=O C1(CC(=O)NCC(C)OC)CCCS1(=O)=O.c1(C=O)ccn(C(C)C)n1 c1(-c2cn(CCO)nn2)nc(C2COc3ccccc32)nn1-c1ccccc1 C1(C)(CC)CC(NC(C2COCC2NC(C2(C)CCC(=O)C2)=O)=O)CCO1 c1(C(N2CCC(O)(C(C)NC(c3csc(S)n3)=O)C2)=O)cc2ncccc2[nH]1 C(CC(=O)N(C1CCCN(C)C1)C)(C(C)CC)NC(c1ccc(C=C)cc1)=O N1(C(c2c(C)cc(C)o2)=O)CC(S(C)(=N)=O)C1.C(=O)(CCCn1ccnn1)N c1(C(=O)NC(C(C)C)C(C)NC(C23CCC(CC2)O3)=O)sc2nccnc2c1N c1(CN2CCN(C(C)CC(c3ccc(F)cc3)=O)CC2)ncc(Br)cc1Cl N1(C(C(N2C(c3cc(C)cc(Br)c3)CCC2)=O)=O)Cc2ccc(F)cc2C1 N1(C(c2ccc3c(c2)OCC3)C(=O)NCCCSCC)CCOc2ccccc21 CCCCS(=O)(=O)CC(=O)N1CCC(NC(C2CC(O)CN2C(N)=O)=O)C(F)C1 C12(COC)CC1CCN2C(=O)CCCNC(c1ccc(C)nn1)=O c1(OC)cc(Cl)c(Cl)cc1C(=O)NC1CCC(CN(C(=O)CC#N)C)CC1 c1(N2CC3(C(NC(c4ccc(OC)nn4)=O)CCC3)C2)nnc(C)c(C)c1C#N CC1CC(C(=O)N(C2CCCCN(C(=O)C(F)(F)C3CCCC3)C2)C)CC(=O)N1 O=C(CC(C(F)F)n1cccn1)NC1CCN(Cc2n[nH]c(O)n2)C1 CC1=C(C)CC(C)(NC(C2CC(N=[N+]=[N-])CN2C(C2CC=CC2)=O)=O)CC1 CC(CN(C)C)CCC(=O)NC1C2CC(NC(=O)Cc3cncs3)CC12 c1(NC(Cc2cc(CC)no2)=O)cc(C(=O)OC)nc(Cl)n1 C1(C)(NC(c2c(CC)onc2C)=O)CCN(Cc2nnc(C3CC3)s2)CC1 CC(C)CCC(O)C(=O)N1CCN(C(C2CCN(CC(C)C)CC2)=O)C(C)C1 c1(C(=O)NCC2(NC(CC(CC)C)=O)CCOC2)cnc(N)c(N)c1 c1(C=O)cc(C)n(C2CC2)c1C.Cc1oc(C(F)(F)F)nc1C=O.C1CC1.N C(=O)(C(C)C(O)CC(C)C)NC(C(CC(=O)N1C(COC)CCCC1)C)(C)C C1(CCOC)CCN(C(=O)C(O)C2CCC2)C1.C1(=CC(=O)N)CCC(C)C1 N1(C(C2(OCC)CC2)=O)CCC(C(C)(C)C)CC1.c1(C(=O)N)ccncc1C c1(C=O)ccc([N+](=O)[O-])[nH]1.C(c1ccc(C)s1)=CC(=O)N(CCC)CC.N C1(C(=O)NC2(C)CCN(C(c3c(NC)cccc3)=O)C2)CC(F)(F)C1(F)F Cc1sc(Cl)nc1C(N1CCCC(N2CCN(C(=O)CP(C)(C)=O)CC2)C1)=O C1(C)(NC(c2cc(C(C)=O)on2)=O)CCC(NC(=O)CN2CCCC2=O)CC1 CN1CCC(C(N2CC=CCC2)C(=O)NC(c2ccccc2)c2cccs2)CC1 C12(NC(C3CCC(=C)CC3)=O)CCCC1N(CC1CN(c3nnnn3C)C1)CC2 c1(OCC)nn(C)cc1NC(=O)CC(O)CNC(=O)C(O)C1CC1 Cc1ncc(N)cc1C(=O)Nc1cccc(NC(C2CCNCC2C)=O)c1 N1(C(C=CCN(C)CC)=O)CCC12CC(CNC(C1(CO)CCC1)=O)C2 Cc1nc(Cl)c(C)c(=NCC2CCCCN(C(=O)CN3CCNC(=O)C3)C2)[nH]1 c1(CC)cc(C(N2CC(CNC(=O)C(C)NC(N)=O)C2)=O)n[nH]1 c1(CC(=O)NC(c2cn(C)nc2)C(=O)NC2CCCC2(F)F)ccccc1O c1(NC(N2CCC(CC(=O)NCC(O)CO)C2)=O)ccc(-c2ncccn2)cc1 c1(OC)cc(O)ccc1CN1CCCC(C(=O)N(CC=O)C)CC1.C(C)(C)C.O C(C1C(C(=O)NC(C2CCN(C(c3ncccc3Cl)=O)C2)C)C1(C)C)=C(C)C c1(C(=O)NCC2N(C(CCCOCC=C)=O)CCC2)cc2ccccc2nc1O N1(C(CCC(=C)Br)=O)CCC2(CCCCN(C(=O)CC3CCC(=O)N3)C2)C1 N1(C(CC(=O)OC)=O)CC2CCCN(C(=O)CS(=O)(=O)C3CC3)C2C1 N1(C(COc2c(C)cccc2)=O)C(C)CC(C)CC1C C(C1=NOC2CN(C(c3cc(Br)c[nH]3)=O)CC12)NC(Cc1ccc(C)s1)=O N1(C2CC3CN(C(C(CCC)NC(C)=O)=O)C2C3)CCC(=C(F)F)CC1 C1(NC(C(CNC(CN(C(C)C)C)=O)CC2CCCC2)=O)CN(C)CCC1O C1(C(=O)NCC2CCCN(C)C2)CCN(C(=O)C(O)C(F)(F)F)O1 c1(C(=O)NC2C(C(N3C(CN)CCCC3)=O)C2)ccc(O)c2ncccc12 C1(C(N2C(C(C)NC(CC(C)N(C)C)=O)CCC2)=O)CC2(COC(=O)N2)C1 N1(C(C(C)N(C(=O)C(c2ccn(C)c2)C)CCC)=O)CCCCC1CCOC N1(Cc2c(OC)ccs2)CCCC2(CCN(C(c3cc(=O)ccn3C)=O)CC2)C1 CC1(C)CCC(F)(F)CC1C(=O)NCC1CCC1.C(=O)(CS(N)(=O)=O)N CCCCCCn1nnnc1C(c1coc(C)n1)NCCCNS(C)(=O)=O.C Cc1ccc(Br)cc1S(=O)(=O)NC1CCN(Cc2sccc2C(=O)O)CC1F Cc1n[nH]c(C)c1C(=O)NCCN(C(=O)CCc1cscn1)CC.CCO.O CCCC(CNC(=O)C(C(=O)OCC)OC)C(=O)NCCc1ncccc1F c1(SC)nc(N2CC(=C(F)CNC(=O)CC3(O)CCCOC3)C2)cc(Cl)n1 N1(C(CCCC(C)C)=O)CCC(C2CCN(C(c3cccc(N)c3F)=O)C2)C1 CC1CC2CC2CC1C(N1CCCC1CN(C)C(c1cscc1Cl)=O)=O C1(C(N2CC(NC(=O)C=Cc3cc(C)no3)CC2CO)=O)(OC)CCSCC1 c1(C(=O)NC(C(=O)NC2CN(CCC)C2)C2CCC2)ccc(O)c(C)c1 C(c1cccc(Cl)c1)=C(C)C(=O)N1CCC1C.C1(C(=O)N)CC(=O)NC(=O)C1 c1(C(=O)NC2C(NC(CCC)=O)CCCCC2)ccc2nc(=N)[nH]n2c1 c1(CC)cncc(C(N2CCCC2C(C)(C)CNC(=O)CC(O)CC)=O)c1 c1(C(N2CCCC(CCNC(C3CCS(=O)CC3)=O)C2)=O)ccc(O)nc1Cl S(=O)(=O)(c1cnc(NC2CC(Cl)(Cl)C2)c(Cl)c1)NCCCC(=O)N1CCCC1 c1(CC(c2nnn(CCC3COCC(C)O3)n2)OC)ccccc1Br N1(C(C(C(C(C)C)OC)O)=O)CCCC2(CCN(C(c3occc3C)=O)C2)C1 CC1(CC(N2CC(OC(F)F)C2)=O)CCCN1C(C1C2CC(=O)CC12)=O C1(C(N2C(C)CCC2)=O)CCC2(CN(C(c3[nH]ccc3-c3ccccc3)=O)C2)O1 N1(C(c2c(C)cc(F)s2)=O)CCCC2(CCN(C(C3CCC=CO3)=O)C2)C1 N1(C(CCCCOC)=O)CCC(c2cn(-c3cc(OC)nc(C)c3)nn2)CC1C c1(C(C)=O)ccc(C(=O)NCCCCCN(C(=O)C(C)N2CCC2)C)cc1F Cc1cc2c(C(=O)NC34CCC(C3)N(C(c3cnc(S)n3C)=O)C4)cccc2o1 N1(C(C(C)SCCCC)=O)CCC2(CNC(=O)CC3C=CCC3)CCCC12 C1(NC(c2ccc(-c3ccccn3)o2)=O)C2CCN(C(=O)CCn3cncn3)C12 N1(C(c2n(CCOC)ncc2)=O)CCCCC1CNC(C1CC=CCC1)=O CC1CN(C(c2cncnc2)=O)CCN1C(=O)CC1CC2C=CC1CC2 C(=O)(CCC(=O)N=c1ccc2nc(C)cn2[nH]1)c1cccc(OC)c1 c1(CC=O)ccc(S(N)(=O)=O)cc1.Cc1ccc(C)c(C(=O)NCCC)c1C.N N1(C(C2C(=O)NCCC2)=O)CC2CS(=O)(=O)CC2C1.C(=O)C(F)(F)C1CC1.C C1(C(=O)NCC(C)N(C(=O)CCc2nccs2)C)CCCCN1C1CCCC1 C1(C(N2CC3C(CNC(c4cncc(F)c4)=O)C3C2)=O)CCCCNC1=O c1(C(=O)NCC(CC)NC(=O)C(C)OCC2CCCCO2)ccncc1C Cc1cc(C=CC(=O)NC2C=CCN(c3nnc(C(C)C)o3)C2)ccc1F C#CC1(NC(C2CC(=O)CN2C(c2ccnn2COC)=O)=O)CCOC1 C1(N(C(C=C(COC)C)=O)C)CCCC(N(C(=O)Cc2ccnc(Cl)c2)C)C1 C1(CNC(CN=S(C)(C)=O)=O)CN(C(c2sccc2C#N)=O)C2CCN1C2 C=C(C)CCC(=O)NCCOC1CCN(C(=O)CCOc2ccccc2F)C1 c1(C(N2CC(SC)C(NC(C3CCC(O)CC3)=O)C2)=O)sc2ccsc2c1C N1(C(=O)C=Cc2ccc[nH]2)CCC(N(C(c2cnc(S)[nH]2)=O)CC2CC2)CC1 N1(C(C=CC=CC)=O)CCc2ccc(C(N3CC(C)(O)C3)=O)cc2C1 Cc1cc(NC(c2cccc(Br)c2)Cc2ccccn2)ncn1 C#CCCCC(=O)NC1CC(CO)N(C(C2CC2C(C)(F)F)=O)C1 c1(C=O)ccc(C)nc1C1CC1.C(Cc1ccccc1)(CC)NC(CSC)=O.N c1(N2CC3(OCC(C)C3)C2)cccc(S(=O)(=O)NCC2CCC=CCC2)n1 c1(N(C)CC2CCCN(C(C3(OCC)CCOCC3)=O)C2)nc(C#N)ncc1Cl C1(CNC(=O)NCCc2cccc(-c3nn[nH]n3)c2)CCOC2(CCCOC2)C1 c1(C(N2CC(C(C(=O)NC3CCC3(C)C)OC)C2)=O)cccc(C)c1C#N C1(NC(C2C(CNC(c3ccc(C#C)o3)=O)CCC2)=O)CCn2nnnc2C1 c1(C(N2CCC(C(F)F)C2)=O)ccc(C(C)C)nc1C.C(=O)(C(C)C=O)OC.N c1(NC(c2c(-c3cc(OC)cc(OC)c3)csc2)=O)cc(F)c(C#N)cc1OC C1(NC(CN(CCC)C)=O)COC2(CCN(C(c3cnc(C(=O)O)s3)=O)C2)C1 O=C(NNC(=O)c1cnsn1)N(c1ccccc1)CCSc1ccccc1 C1(CC)CC(C(N2CC(CO)(NC(=O)CS)C2)=O)CCO1.c1c(C)noc1C C12(NC(=O)NC3CC3)CCCC1(F)CN(C(=O)CC1CN3CCC1CC3)C2 c1(C(=O)NC2CCC(N(C(Cc3c(C)con3)=O)C)C2)cc(Cl)c(O)cc1C c1(CNC(COCC#C)=O)ccccc1CNC(=O)C(C)O.CCC=C c1ccccc1Cl.Cc1n[nH]cc1C(=O)NC1CC1NC(=O)CC.C(=O)C.N c1(C(CNC(C(=O)NC(C(C)C)C2CC2)=O)C)ccc(F)c(F)c1 c1(C(N2CC(OC)C(NC(=O)C(C)C(C)(C)O)C2)=O)ccc(F)cc1Br C1(C)(CC)CCC(C(=O)NCC(C2CC2)N(C)C(c2cc(C)cnn2)=O)O1 C1(NC(c2c(C)ccnn2)=O)CCC2(CC1)CC(NC(C1CNC(=O)C1)=O)C2 C(N=c1[nH]c(=NCCC2=CCCCC2)c2ncccc2[nH]1)c1ccc(C#N)o1 c1(C=O)cc2ccccc2[nH]1.C(C)(C(=O)NC1CC1NC(=O)C)OCC n1(CC=O)nc(C)c(C=NO)c1C.CCCCNC(=O)CC1CC1.C=O.O C12(CC=O)CCCCC1C2(F)F.CC1CCCN1CC(=O)NC12CC(C1)C2.C CC1(C)C=C(C(=O)NC(CCOCCO)C(=O)NC(C2CCCO2)CO)C1 N1(C(C2C(CC(C)C)C2)=O)CCCC1CCC.c1(CC=O)cnc(C2CC2)[nH]1 CC1(C)OCCC1C(N1CC(CNC(=O)CCc2nc(O)n[nH]2)C1)=O N1(C(=O)C(F)F)C2CN(C(=O)C(F)(F)c3ccccc3)CC12 C1(O)(C(N(CCCNC(COCCCC)=O)CC)=O)CC2(CCOCC2)C1 Cc1oc(C(C)C)cc1C(=O)NC1(C)CC(NC(C2CCC(=O)O2)=O)C1 C(=O)(C1CCCc2c[nH]nc21)NC1C2CN(C(CCCC)=O)C(C2)CC1 N1(C(Cc2ccc(C)o2)=O)CCC2CN(C(c3cc(S(N)(=O)=O)co3)=O)C2C1 N(C(=NCCOC(F)(F)C(F)(F)F)NC1CCCCC1C)CC(=C)CC Cc1cc(C(=O)Nc2ccccc2OCCC(N)=O)cc2[nH]ccc12 c1(C(=O)NC2CCN(C(CCC(=O)NC)=O)CC2F)ccn2c(O)nnc2c1 c1(C(N2CCCC(C)C2CNC(c2ccccc2Cl)=O)=O)ccc2nccn2n1 C(=O)(CCC(C)(F)F)N(CC(=O)NCC(C)S(C)(=O)=O)CCC C(=O)(C(C(C)CC)N(C)C(C1CCCC12CCC2)=O)NCCC=C=C n1(CC(N2C(CNC(c3cc[nH]n3)=O)CCC2)=O)cnc2ccc(F)cc2c1=O c1(N2C(c3cccc(OC)c3)CCC2)nc(NCC2CC2(F)F)c2ncsc2n1 c1(C(=O)NC(C)CCCNC(C2CCSC2)=O)ccccc1NS(C)(=O)=O c1(-c2cc(C(=O)NCC(CC)C)n[nH]2)cccc(Cl)c1.c1(CC(=O)N)cnsc1 c1(C(=O)NCC(CC=C)NC(=O)C(C(C)O)N(C)C)sc(C)c(C)c1Br N1(C(c2oc(C)cc2)=O)CCCC(O)(CC(=O)NC2CC(CN(C)C)C2)C1.C c1(CC(C)(C)C)ccc(C(=O)NCC(F)C)cc1.c1(C=O)c[nH]nc1C1CC1 CN1CC=C(CC(=O)N2CC(NC(C3CC(N=[N+]=[N-])C3)=O)C(C)(C)C2)CC1 N1(C(CSc2n(C)cnn2)=O)CC2(C1)SCCC2NC(C1CC12CCC2)=O N1(C(C(C)(C)F)=O)CCC2C(CCCN2C(=O)Cn2cnc3ccccc23)C1 CCCCCC(O)CC(=O)NCC1CC(F)(CNC(=O)C(CC)CC(C)C)C1 C1(NC(=O)COc2ccccc2)CCSC12CN(C(=O)CCn1cnnn1)C2 c1(CC(=O)NC2C(NC(C3N(C(C)=O)CCCC3)=O)C2)cccc(Cl)c1Cl C1(NC(c2nnc(C)s2)=O)CC(NC(c2noc(C3CC3)c2C)=O)C12CCC2 C1(NC(C(CC)O)=O)CCCN(C(c2cc(C)n(CC(F)(F)F)n2)=O)CC1 C1(OC)(CNC(C2CSCCS2)=O)CN(C(c2nn[nH]c2Cl)=O)C1 C1(C(=O)OC)CCC(F)CN1C(C1CCCCN1)=O c1(-n2c(C)cc(C=O)n2)ccc(F)c(Cl)c1.C1C(C)C1C.C(C)(C)C.C(=O)N C(=O)(C(C)CC(C)(C)C)N1CC(CNC(c2c(CC)cns2)=O)C(C)CC1 C(=O)(C1CCCn2ccnc21)NCC(CN(c1ncc(C(=O)OC)nc1)C)C c1(C(=O)NC(CCOC)CNC(=O)C(C)c2ccsc2)sc2nnc(S)n2c1C S(=O)(=O)(CC(=O)N1CCCC1CCC)NC.c1ccccc1.C1(C(=O)N)CCCC1 C1(CNC(N2CC(C)(C)C2C2CC2)=O)CCOCC1(C)C C1(NC(C(c2ccc(F)cc2)OC)=O)CC(O)CN(C(=O)C(C)(C)C2CC2)C1 C(CC(C)C(=O)NC(C)(C)CCNC(=O)C(F)CC1CCOC1)=CC C1(=CC(N2CCCCC(NC(CC3C(C)CCC3)=O)C2)=O)CC2CCC(C1)N2C C(=O)(C(O)CC(N)=O)NC(CC(C)C)CNC(=O)CCCc1cccc(Cl)c1 C1(C2CC2)(C(N2C(CCC=C)CCC2)=O)CN(C(=O)C(C)NC(=O)NC)C1 c1(OC)ccc(C(=O)NCCCCCCN(C)C(C23CCCCC2C3)=O)nn1 c1ccc2c(c1)CN(C(C1CC1(C)C(C)C)=O)C2.CC1=CC(C(=O)NC)SC1 C1(OCCC(CNCC(=O)Nc2nn[nH]n2)O)CCCCCC1.c1ccccc1Cl c1(C(N)=O)ccccc1NC(C1CCCCC1NCc1ccccc1CCBr)=O N1(C(c2ccc3[nH]nc(Cl)c3c2)=O)CC(C2CCCCN(C(C34CC(C3)C4)=O)C2)C1 C#Cc1cnc(C(N2CCC(O)(CNC(c3cn(CC)cn3)=O)C2)=O)c(C)c1 N1(C(=O)NCC2(c3ccc(F)cc3)CCCC2)CCc2cccc(O)c2CC1 c1(C(N2CCC(C(C)NC(C3CC(N(C)C)C3)=O)C2)=O)ccc(=O)oc1 c1(N2CCN(c3cccc(OC)c3)CC2)nccc(=NC(C)Cn2cncn2)[nH]1 C1(NC(CN(CCC#C)C)=O)CCC(CCC(=O)NCCC(Cl)Cl)C1 CCC(CC(C)C)C(=O)NCC(O)CC(=O)NCC1(CC(C)C)CCC1 Cc1c(F)c(F)c(COC(C2(Cc3ccc(F)cc3)CCNCC2)=O)c(F)c1F N1(C(Cc2n(C)ccc2)=O)CCCC2(NC(c3cc(C(N)=O)cs3)=O)CCCC12 C(CCN(C(=O)CO)C)(C(C)(C)C)NC(CC(=C=C)C)=O.C1CCCCO1.C CCC(CC(C)C)C(=O)NC1C=CC(CNC(C23CC4CC(CC2C4)C3)=O)C1 C1(C(=O)NC2(C)CN(C(C3(CC=C)CCC3)=O)C2)CCc2n[nH]cc2C1 c1(N(CC)CC2CCC2)cccc(CC(=O)NC(C2CCCN2NC)=O)c1 N1(C(c2cc(C(C)(C)C)no2)C(=O)NC)CCC(O)(CC(=O)OC)C(F)C1 C(=O)(C(C(C)(C)C)OC)NC1CC(N(C(C(C)OCC=C)=O)C)C1 N1(C(c2cc(C)c(C(F)(F)F)cc2)=O)C2CCCC1CN(C(C1CC=CC1)=O)C2 CP(C)(=O)c1ccc(C(N2CCC(C(C)(C)C)C2)=O)o1.C1(C=O)C=CCC1.C n1(CCC)cc(CN2CCCC2CN)c(C)n1 c1(C(N2CC(CC(C)NC(=O)CCC3CCOC3)C2)=O)c(F)ccnc1Cl c1(NCC2N(C(c3c(C)nc(OC)s3)=O)CCCC2)ncc(Br)c(C)n1 c1(C(N2CC3C(C3)C2)=O)coc2c(C)cccc12.C(C)(C(=O)N)OCCC#C.C N1(C(C2CN(CC)C(=O)C2)=O)CCN(C(=O)C(C)n2cccc2)C(C)C1 c1(C(=O)NCCN(C(=O)CCC2CC2(F)F)C)ccc2cncn2c1 c1(C(N2C(C)C(NC(C3(CO)CC3(F)F)=O)CC2)=O)cn2ccccc2n1 C1(CC)CCC(N(C(=O)C(O)C2CN(C(c3ccc(CO)s3)=O)C2)C)CC1 C=CCC(F)(F)C(=O)N1CC2C(CC(=O)NCCOC3CCOC3)C2C1 c1(C(C(=O)NC(C)CN(C)C(C2(CC3CCC3)CC2)=O)O)ccc(Cl)cc1 C1(NC(C2CC(C)OC2)=O)CCCC12CN(C(c1c(C(F)F)cnn1C)=O)C2 C1(C)CCCN(C(c2cn(C)nc2-c2cccs2)=O)C1.C(=O)(C(=O)N)NCC N1(C(CCC2CCC(=O)NC2)=O)CC(CNC(c2ccns2)=O)CC12CCC2 c1(C(N(CC(CC)NC(=O)C(CC(C)C)N(C)C)C)=O)ccc2ncnn2n1 CN1CCCCN(C(=O)C=CCNC(c2cn(C)c(=O)n2C)=O)CC1 C1CC(F)(F)CN1C(=O)C(C#N)CC1CC1.CC(C)CCC=CC(=O)NC C(=O)(CCCCC(F)(F)F)N1CC(C)(CNC(C2CCC(C)O2)=O)OCC1 C1(CC(=O)NCC(CC)(CC)NC(c2ccc(C)cc2Cl)=O)CCC(C)(C)CO1 N1(C(c2n(C=C)ncc2)=O)CCN(C(=O)C(C)CC(=O)OC)C(C(F)F)C1 C=CCCC(C)(C)C(=O)NCC(C)(C)CC1CN(C(=O)CN2C(C)CCC2C)C1 C1(NC(C(C)NC(C)(C)C)=O)CCC(N(C)C(c2cnnn2C)=O)CC1 N1(C(CC(C)CN(C)C)=O)CC2CC1CN2C(=O)Cc1nccn1C c1(C(=O)OC)c[nH]c(C(=O)NC2CCN(C(=O)C(Br)=C3CC3)C2)c1 c1(NCC2CCC(C)(C)CO2)ncccc1S(=O)(=O)NCC1CCC2(CC2)C1 N1(C(C(CC(=O)OCC)C)=O)CC2CCC1CC2NC(=O)CC1CCOC1.O C1CCCN1C(=O)C(N1CCOC1=O)C.c1(CCC(=O)NCC)nc(C)no1.C Cc1ccsc1CC(N1CCCC1CN(C(=O)C=C1CCC1)C)=O CC1=C(C(=O)C2CC2)C(c2cc(C(C)C)nn2C)NC(=S)N1c1cccc(F)c1F C1(N(C(C=C(CCC)C)=O)C)CCCCN(C(C2CC(C)N(C)C2)=O)C1 c1(OC)ccccc1-c1cccc(COC(C23CC(C)C2C3)=O)c1 C(=O)(C#CC1CCCOC1)N1CC(CC)C(Nc2nnc(C)c(C)c2C#N)CC1 c1(NC(c2nc(C)sc2)C)ncccc1S(=O)(=O)N(CC(O)C1CCC1)C C(=O)(CC(C)C(C)(C)C)NCC1C2CN(C(C(CCSC)OC)=O)C1C2 C#CCC(CC#C)C(=O)NC(C)CN(C(=O)C=Cc1ccc(SC)cc1)C N1(C(C(C)NC(CC)(C)C)=O)CCN(C(=O)CO)CC(C)C1.c1c(F)cccc1F N1(C(c2cncc(C#C)c2)=O)C2COCC1CC(NC(C1(Cl)CC1(F)F)=O)C2 C1(NC(c2cnn(C)n2)=O)CC2CC(C1)CN(C(c1ncn3c1CCC3)=O)C2 c1(N(C)C(C2C=CCN(C(c3ncccn3)=O)C2)=O)cccc(C#N)c1 C12(C(=O)NCCC(C)N(C(=O)Cc3ccco3)C)CCC(C)(C1)OC2 N1(C(c2cc[nH]n2)=O)CCCCC1C1CCCN(C(C2(n3ccnn3)CC2)=O)C1 c1(C(C(=O)N(CC(C)(C)CNC(C2CCCC2O)=O)C)(F)F)ccc(F)cc1 c1(NC(C2(C)CCN(Cc3ccc4cc[nH]c4n3)C2)=O)cccc2c1C(=O)NC2 N1(C(CN(CC)CC)=O)C(C(=O)NC2(CSC)CCOC2)CC1C c1(C(=O)OC)ccc(NC2CCCCC2NC(=O)C(c2ccc(Cl)cc2)C)nc1 N1(C(C(CC2CC2)NC(c2c(CC)nccc2)=O)=O)CC2C3CCC(C3)C12 N1(C(c2ccc(N)c(F)c2)=O)CCc2ccccc2C1CNC(=O)C(F)(F)CO n1(CCC(=O)O)cc(Cl)c([N+](=O)[O-])n1.c1(C(=O)OC)cc(C(=O)N)ccc1 C1(F)(CNC(CCc2n(C)c(S)nn2)=O)CCCN(C(=O)CC2CCOC2)C1 N1(Cc2ccc(C)cc2O)CCC2(CCCN2C(c2ccncc2Cl)=O)CC1 Cc1cc(F)ncc1C(N1CCC(NC(=O)CC2CCC(=O)C2)C(C)C1)=O C(=O)(C1Cc2ccc(Cl)cc21)N1CC(CCNC(CN(C2CCC2)C)=O)OCC1 N1(C(c2c(CC)[nH]cc2)=O)CC2CC(NC(C3CC=CCO3)=O)CC1C2 c1(C(N2C(C)CCC(CNC(c3c(OC)csc3)=O)C2)=O)cccc2ncsc12 c1(C=O)cc2sccc2n1C1CC1.C12(C=O)CCC(C(F)F)(CO1)C2.CC.N C1(CC=C)(NC(=O)C(F)C(C)C)CCN(C(=O)Cn2cnnc2O)C1 C1(C2CC2)(NC(CC2CCN(C(C(CCC)OC)=O)CC2)=O)CCOC1 c1(C(N2CCC(C(=O)OC)(CCF)C2)=O)sc2cccnc2c1N N1(C(CCOCCOC)=O)CCN(C(C2COCC2C(=O)OC)=O)C(CF)C1 C1(NC(C2CC(C)(F)C2)=O)CCN(C(c2ccnc(F)c2)=O)CC1F c1(C(=O)NC2(CO)CCN(C(C(F)=CCC)=O)CC2)cn2ccc(OC)cc2n1 C1(C)(CC(=O)NC2C(NC(c3n(C(CC)C)ncc3)=O)CC2)CCOCC1 c1(C(=O)NC(C)C(C)NC(C2(C)CS(=O)(=O)C2)=O)ccnc2c1CCC2 c1(C(N2CCC(CNC(=O)CC3CCOC3)C2)=O)cc2cc(F)cc(F)c2[nH]1 CC1(C)CCCCC1NC(C1CC12CCN(C(=O)C1=NNC(=O)C1)C2)=O C(C)(C)(CCCNC(C1(C=O)CCC1)=O)NC(c1c(CC)nc[nH]1)=O.N Cc1ccc(C(=O)N)c(=O)n1C.C1CN(C(=O)CC2(C(F)(F)F)CC2)CCC1F C1CCS(=O)(=O)C12CN(C(=O)CCN1C(=O)CCC1=O)C2.C(C=O)OC(C)C C(CCCCC(=O)NC(c1ccc(F)cc1)CNC(C12CCC(CC1)O2)=O)SC C1(NC(=O)CSCc2cccnc2)CCC(O)CN(C(C2CC=CCO2)=O)C1 c1(SC)ccccc1CC(=O)OCC(C1CCCC(C)C1)=O N1(C(CCN(C)CC)=O)CCC2CN(C(=O)C(C)S(C)(=O)=O)C2C1 N1(C(CCC)=O)CC2CCC(C1)N2C1CCN(C(=O)C(C)SCC)CC1 c1(NC(CC)C(=O)NC2CCN(C(=O)CCCn3ccnc3)C2)cccnc1Cl Cn1cc(C(F)(F)F)nc1C(N1CCOC(CC)C1)=O.C1(C=O)CCC(=O)N1.N c1(C(=O)NCC2CC(NC(C(C(=C)C)(C)C)=O)C2)cc([N+](=O)[O-])ccc1 N1(C(c2cn(C(C)C)nc2)=O)CC2(C)CC1(C(=O)NCCc1cnnn1C)C2 C1(OC)CCCC(CC(=O)NC2COCC2NC(=O)C(=O)N(C)C)C1 c1(C=O)cc(N)cc(O)c1.c1(CC)c[nH]nc1C(=O)NC(C1CCCCC1)C.N C(=O)(C1=CC2C=CC1C2)NCCCCC(=O)NCC(c1ccsc1)O N1(C(CN(C(=O)CC2COC(=O)C2)C(C)C)=O)CC(O)C(N=[N+]=[N-])C1 CC1CN(C)CCN1C(=O)CN(C(=O)Cn1ccnc1)C1CCC1 c1(C(c2nnnn2CCSC)NCC(CC)C)cc2ccsc2n1C c1(C(=O)NCC(CO)NC(CNS(N(C)C)(=O)=O)=O)ncc2[nH]ncc2n1 C#CC1(C(=O)NCC(C)S(C)(=O)=O)CCN(C(=O)CNc2cccnc2)CC1 C1(NC(CC=C)=O)CCOC2(CCN(C(c3cc4cccn4c(O)n3)=O)CC2)C1 C(C(=O)N=c1nc(Sc2ccccc2)[nH]s1)N(C(CC)C)CCO N1(C(CC2(C)CC2)=O)C2CC=C(C(=O)N3CC4CC3C4)C1CC2 c1(C(C(=O)NCCC2(O)CN(C(C3(C)CC=CC3)=O)C2)O)cc(F)cc(F)c1 N1(C(C(=O)N(C)C)=O)CCN(C(=O)CC23CCCC2C3)C2CS(=O)(=O)CC12 C1(NC(CCC(C)C)=O)C2CC(O)C1N(C(C1CCOC(C)(C)C1)=O)C2 C1(CCC)(C=O)CCNC1=O.c1(C(N(CC)C2CC2)=O)ccc(C(C)=O)o1 CCC(CC)C(C(=O)NC(C1CC(NC(C2CN(C(C)C)C2)=O)C1)C)OC c1(NC(C2C(NC(C#CC)=O)CCC2)=O)cccc(C(=O)OC)n1 CCC(C)C(CNC(=O)C(=O)NCCCOC1CCCCC1)OC C(=O)(CCS(=O)(=O)N1CCOCC1)NCC1N(C(C2C(C)CCC2)=O)CCOC1 N=c1ccc(C(=O)NCCC2CCC(NC(=O)CCOC3CCC3)C2)c[nH]1 CC1CCCCC1CN(CC(=O)NCc1ccc(C(C)(C)C)s1)C C1(O)(C(=O)NC2CC(CCNC(c3ccsc3Br)=O)C2)CCCCC1 C(C(O)CC(=O)N1CCOC(CCF)C1)NC(c1ccc(SC)o1)=O N1(C(c2c(OC)c(F)ccc2)C(=O)NC(C)(C)C)CCC2(CC1)CN(C)CCO2 c1(CC)cccnc1CNC(N1CCOC(C2CCOCC2)C1)=O C1(C(=O)NCCCNC(CCC(=O)OCC)=O)CCCCN1S(N)(=O)=O.O c1ccc(O)cc1.C1(CCNC(C2(SC)CCC2)=O)CCC(NC(=O)C)C1 c1(C(N2CCC2)=O)cn2ccncc2n1.c1(C(=O)OC)ccccc1C(=O)NC N1(C(C2(C)CC2)=O)CCCC(C(C)(O)CNC(c2ccoc2C2CC2)=O)C1 c1(NC(c2n(CCSC)nnn2)(C)CC2CCC2)cccc(-c2cncnc2)c1 C1CCN(C(C2CN(C)C(=O)N2)=O)CC1.C(=O)CN(C)C(=O)C1CC1.CC Cn1ncc(Cl)c1C(=O)NCC(C)(C)CC1CN(C(C2CC3C=CC2C3)=O)C1 c1(CC(=O)N)ccc(C#C)cc1.C1(C(N(C2C3CCCC23)C)=O)(C)CCCO1 c1(CN2CCC(O)(CC(=O)OCC)C2)ccc(F)cc1O n1(CC=C)nnnc1C(c1ccn(C(C)(C)C)c1)NCC1COC(=O)N1 C=CCC(C)(C)CC(=O)NCCC(O)C(=O)NCc1conc1C(C)C c1(C(C)C(=O)NCC2(C)CCCN2c2nncs2)ccc(C(F)(F)F)cc1 C#Cc1ccc(NC(c2cc(Br)cs2)c2nnnn2C(C)(C)C)c(C)c1 N1(C(c2c(C)nn[nH]2)=O)CC2CCC1CN2c1ncnc(C(F)(F)F)c1Br N1(C(C2(C(=O)NC)CCC2)=O)CCC(C)(C)C1.C1(C=O)CCCC(=O)O1.C N(C)(C1CCCc2ccccc21)CCOC.C1CN=C2C=CN=C(N2)N1 C1(NC(C(C)SC)=O)CCCC(NC(=O)CC2CCC=CCC2)C1 c1(C(=O)NCC2(NC(C(C)c3ccsc3)=O)CCC2)ccc(Br)o1 c1(CN(C(c2ncc(C)o2)C(=O)NC2CCOCC2)CC)noc2c1CCCC2 C1(CNC(CC2C(C)(C)CCCO2)=O)CCC2(CN(C(c3cscn3)=O)C2)O1 N1(C(C(CNC(c2ccsc2)=O)CC2CC2)=O)CCc2cccc(O)c21 c1(CC)[nH]c(=N)sc1C(=O)NC(C)C(C)NC(=O)CC1CCCC1 c1(CC)nc(C)cc(=NC(C)CC(C)NC(=O)CN2CCCCC2)[nH]1 n1(CC)cc(Cl)c(C(=O)NCC(C)CO)n1.c1(C=O)csc(-c2ccoc2)n1.N C1(C(=O)NC(CCNC(C2=C(C)CCC2)=O)C)CCc2ccc(F)cc2O1 c1(-c2ccc(COC)cc2)ccc2nc(CC(=O)NCC(O)C(F)(F)F)cn2c1 C1(NC(=O)CC(=O)OC)CC(NC(c2nc(OCC)sn2)=O)C1(C)C C1(C(=O)NC2(C)CC(O)C2)CCCCCC1NC(=O)C=Cc1cccnc1 C1(CC(=O)N(CCC(=O)OC)CC=C)CCCN1C(c1c[nH]cc1CC)=O C1(C(N2C(COC)CC2)=O)(CNC(=O)CCCC2CCCO2)CC=CC1 C1(CC=C)(NC(c2nocc2C)=O)CCN(C(c2nccnc2C(=O)OC)=O)C1 c1(SC(C(=O)NCC(C)N(C(CN(C)CC)=O)C)C)ccc(C)cc1 CCC(C)(C(=O)NC1CCCC1NC(c1ccncn1)=O)C(N)=O C1(CNC(CSCCOC)=O)CN(C(=O)Cc2cc[nH]n2)C2(CCC2)C1 C#Cc1cnc(N(C(C)CNC(=O)C(C)Cc2ccncc2)C)nc1 c1(C2C(C(N(C3CCCC3)C)=O)C2)cccnc1.C(=O)(C(C)(F)c1ccon1)N c1ccccc1[N+](=O)[O-].C1(CC(=O)OC)CCN(C(=O)NCC2CC2)CC1.C C1(C(N(CCCC)C2CC2)=O)CC2CC1CN(C(=O)C=CC(C)(C)SC)C2 c1(OC)cc(S(=O)(=O)Nc2cnn(Cc3ccncc3)c2)ccc1F N1(C(CC2(C(=C)F)CCC2)=O)CC2CC(C(N3CCC(C)C(F)(F)C3)=O)CC2C1 N1(C(=O)NC(C)Cn2cncn2)CCC(C(c2ccc(Cl)cc2)O)CC1 C1(C(=O)NCC(C)C)(NC(=O)CCC2CCC2)CCc2cc(Br)ccc2C1 c1(CN2C3C(C(=O)Nc4c(O)ncc(C)c4)C(C3)C2)cc(Br)c(F)cc1Cl C1(CC)CC(C(=O)NC(C)CNC(=O)CCC(=O)NC)CC(=O)N1 CC1(CNC(c2ccc(C(F)(F)F)o2)=O)CCN(C(=O)C(O)CC(F)F)CC1 Cc1ccoc1C(=O)NCCOCc1ncnn1C.CCCNC(=O)C.O C1(NC(CCc2cnc(C)s2)=O)CCOCC1NC(=O)CCOCC1CCCO1 C(=O)(C1=CNC2=NCCC2=C1)NC1(COC)CCN(C(c2ncc[nH]c2=O)=O)C1 c1(CC)ncccc1C(N1CCC(C)(C)C1)=O.c1(C(=O)N)cnc(C(C)C)[nH]1 N1(C(c2c(C)noc2C(C)C)=O)CCC(NC(=O)CCCF)C(C(C)C)C1 c1(C(N2CCN(C)CC2)=O)ccc(F)c(S(N)(=O)=O)c1.C#CC(C)(C)C(=O)N.C C1(C(=O)NCC2(O)CCN(C(=O)CO)C2)OCC2COCCC12.C1CCCCC1 N1(C(c2ncc(CC)cn2)=O)C2CCC(C2)C1C(=O)NCc1cc[n+]([O-])cc1 C1(NC(c2cnc(C(C)C)[nH]2)=O)CCN(C(=O)CC(F)(F)Cl)C(C)C1 C1(CCC)CCc2nc(NC(C3CS(=O)(=O)C3)=O)sc2C1 C1(C(=O)NCCC(C)N(C)C(c2cnn[nH]2)=O)CCCCC1c1nnc(S)n1C C1(C(=O)NC2CC(NC(c3nc(C(C)(F)F)sc3)=O)C2)C(F)(F)C12CC2 c1(C(=O)NCCC2CCN(C(Cc3ccn(CC)n3)=O)CC2)cc(O)nc(O)n1 C12(CNC(C(CC)(C)C#N)=O)CCCC1CN(C(=O)CC)C2.C(=O)C(C)(C)C C=CCC(C)(C)CC(=O)N1CC(NC(=O)CC2(CO)CCCC2)C(C)(C)C1 N1(C(c2nnc(C3N(C(C4CN(C(C)=O)C4)=O)CCC3)s2)=O)CC2(CCS2)C1 C1(O)(CCNC(C(CC#C)O)=O)CCCN(C(=O)C=Cc2cscn2)C1 CC(C#N)CCC(=O)NCC.C(=O)CC.C(C)(C)C.C(C)(C)C.C(N)=O.O Cc1ncc(CCC(=O)N2CCC2CNC(c2cc(Cl)ccc2F)=O)c(O)n1 C1(CC)CN(C(C2CCCC(F)C2)=O)CCC1CNC(c1cc(C)sc1N)=O N1(c2nc(C(C)C)cc(C)n2)CCC2(CCCN(C(=O)CCC(F)F)C2)C1 c1(N(CCN(C(Cc2scc(C)c2)=O)C)C)nnc(C#N)s1 C=CCCCC(=O)NCC(CO)NC(c1c[nH]nc1-c1ccc(OC)cc1)=O N1(C(C2(N(C(=O)OC(C)(C)C)C3CC3)CC2(F)F)=O)CC(=O)CCC1C Cc1ccc(N2CCOC(C)(c3cnn(C)c3)C2)c([N+](=O)[O-])c1 CN(CCCC(=O)NCCCCN(C(=O)CCC1CCCO1)C)N=O C1(C(=O)NCCCCCNC(c2csnn2)=O)C2CCC1(c1cccnc1)C2 N1(C(c2c(CC)noc2)=O)CCCC2(NC(=O)Cn3ncc(Br)c3C)CC2C1 N1(C(C(C)=CC(C)(C)C)=O)CC(F)CC1C(=O)N(C1CCOCC1C)C c1(C(=O)NCCCCc2cn(CC(=O)O)nn2)cccnc1N1CCCC1=O C1(C(N2C(C(=O)NC(CO)CCO)C3CC3C2)=O)CC2CC(=O)C1O2 c1(OCC)ccccc1C(C)N(c1nnc(Cn2cncn2)n1CCOC)C c1(NCC(c2nncn2C)C)ccc(S(=O)(=O)N2CCC(C#N)CC2)cc1Cl CCCC(CC(C)C)C(=O)NC1CCC(CNC(=O)CC2(C)CC2)C1 C(=O)(CCN=c1[nH]ccs1)N1C(CN(C(CS(=O)(=O)NC)=O)C)CCCC1 c1(OC(c2ccccc2)C)ccc(CN2CCCCC2CCS(N)(=O)=O)cc1 c1(C(N2CCC(NC(C(CC)CC(F)F)=O)C2)=O)ccc(S(C)(=O)=O)c(C)c1 Cc1sc(C(N2CCC(C)(NC(C3SCCCS3)=O)C2)=O)nc1O N1(C(C(CC#C)O)=O)CCC2(CCC(NC(C3CCc4ncnn4C3)=O)C2)C1 N1(C(C(=O)NCCC(COC)(C)C)=O)CCCC2(C1)NC(=O)NC2=O N1(C(COCCSC)=O)CCN(C(=O)CC2CCN(C)C2=O)CC1.C1CC1.C C1(C(N2CCC(CN=[N+]=[N-])C2)=O)(COC)CN(C(C23CSCC2C3)=O)C1 CC1CN(C(C2(CO)CC(C)(C)C2)=O)CC(C(=O)NC(CO)C(N)=O)O1 N1(C(CC2CN(C(C)=O)C2)=O)CC2CN(C(=O)CCC(=O)NN(C)C)CC(C1)O2 C(C(=O)NCC1CN(C(=O)Cn2cnc(Br)n2)CC1O)(C(C)C)SCC c1(C(N2CCCC2)=O)ccnc(N(C)C)c1.c1(C(N(CC)C)=O)csc(C)c1 C1(CC)CC2(CCO1)CCN(C(=O)NCC(c1cccc(C(F)(F)F)c1)(C)C)C2 C(=O)(C1Cc2ccc(Cl)cc21)N.CC(C)CCCNC(c1ccc(C(N)=O)[nH]1)=O c1(NC(C(Cc2cnc[nH]2)NC(CN(CC)CC)=O)=O)cccc(F)n1 C1(C)(NC(C2C3CN(C(C#CC(OCC)O)=O)C2C3)=O)CCC2CC2C1.C c1(C(C)NC(=O)C=CC2CCCC2)cccc(Cl)c1.C(=O)(CCn1ccnn1)N C(=O)(C#CC1CCC1)N(C1CN(C(C2CC23CCOCC3)=O)CCC1O)C c1(CC(C)C)ccc(C(C)C(=O)NCCOCC)cc1.C1(C=O)C=CCCC1 c1(C(C)NC(COC)=O)nc(-c2cc(C)oc2C)nn1-c1cccnc1C N1(C(C(CC)CC)=O)CC(NC(c2cc(OC)ccc2Cl)=O)CC(C)C1 N1(C(c2cnc(C(C)=O)s2)=O)CCC(NC(=O)C=C2CCCCC2)C(C)(C)C1 N1(C(C2CC(O)(CNC(c3c(C)cccn3)=O)C2)=O)CCc2c(O)noc2C1 CCCS(=O)(=O)CC(=O)NC1CN(C(C2(F)CCC(C)CC2)=O)CCC1F C1(CNC(CCCC)=O)CN(C(c2cc3n(n2)CCC3)=O)CC1(C)C C=C(C)CC(C(=O)N1CCC(C)(CC)C1)NC(c1ccnn1CCOC)=O c1(OC)cc(OC)c(S(=O)(=O)N2CC3C(Br)C3C2)c(OC)c1 c1(N2CCC(C)(NC(C(CN(CC)CC)F)=O)C2)nc(C=O)nc(C)c1C.O c1(CC(=O)NC2CCN(C(C(C(C)C)NC(C)=O)=O)CC2)ccc(Cl)cc1Cl c1(C=O)coc2ccccc12.c1(C(=O)NC2CC2C)cc(-c2ccco2)on1.N c1(CC(N2CCC(CN(C(CN(CCC#C)C)=O)C)C2)=O)ccc(C)cc1 C1(NC(c2c(CC)c[nH]c2)=O)CC12CC(NC(=O)C(C)c1ccco1)C2 c1(OC)cc(F)c(F)cc1C(=O)N(C1CCN(C(C2CCCC(C)(C)C2)=O)C1)C c1(C(=O)NC2C(C)CN(C(c3cccc(CO)c3)=O)CC2)nc(O)nc(O)c1F C1(NC(C2CC3(CC(=C)C3)C2)=O)CCOC2(CCN(C(C3CCCC3)=O)CC2)C1 N1(C(CCc2ncc(C)[nH]2)=O)CC(CNC(=O)C(C)(C)CN(C)C)C(O)C1 CC(C)(CC(=O)NC1CN(C(=O)C#CC2CC2)CCC12CCC2)CC(F)(F)F c1(C(C(=O)NCCNC(c2cc(C)cc(N)c2)=O)O)cc(F)c(F)cc1F N1(C(CN(C(c2ncccc2O)=O)CC)=O)CC(F)(C#N)C1 c1(CC(N2C(C)(CC)CC(NC(c3ccsn3)=O)C2)=O)ccc2nc(O)[nH]c2c1 C1(CNC(C2CC(=C(F)F)C2)=O)CC2CCCC2N1C(=O)Cc1ccoc1 C#CCCCC(=O)N(C)CC1CN(C(=O)CCCNC(=O)OCC)CCO1 C1(C)(CC(=O)N(CC(C)(C)C)C)CCS(=O)(=O)N1.c1(C=O)ccc(F)s1 O(NC(=O)C(c1ccco1)NC(c1nc(Cl)cs1)=O)CCOCCOC c1(C(=O)NCCCNC(CC=CCCCCC)=O)ccc(CCO)cc1 N1(C(=O)NCCC(C)N2CCCC2)CCC2(CCCC2N2CC(C(N)=O)C2)CC1 C1(C(N2C(CC(=O)O)COCC2)=O)CCC2CCCCN2C1 C1(C(N(CC(CNC(C2CN(C(C)C)C2)=O)O)C)=O)Cc2c[nH]cc2S1(=O)=O N1(C(C(=O)NCC)=O)CCC(C(F)(F)F)CC1.c1(C(=O)N)cnc(=N)[nH]c1 CC(C(=O)N=c1c(F)c[nH]cc1Br)N1CCS(=O)(=O)CC1 N1(C(c2ccc(C)s2)=O)CC(NC(=O)C(O)C(C)C)CCC(O)C1 CN1CCC(C(=O)NCCC2(C)CCOCC2)(NC(c2c[nH]c(=O)cn2)=O)C1 c1(NC(C(C(=O)OC)Cc2cc(F)cc(Br)c2)=O)c(OC)ccc(F)c1Br CN(C)S(=O)(=O)N1CCC(C(=O)NCC(O)CCNC(c2ncccn2)=O)C1 C1(C(C)C(=O)NC(C)CC2CCOC2)CCN(C(c2cc(O)nn2C)=O)CC1 N1(C(c2ccnc(N(C)C)c2)C(=O)NCCCSC)CC(OC)CCC1C c1(CN2CC(C(=O)NC(C3CCOCC3)C)C(O)CC2)cc(O)c(F)c(F)c1 c1(C(=O)NCC(C)CNC(=O)C(F)(F)c2cccnc2)cc(O)cc(O)n1 c1(CNC(COCCCC)=O)cnn2c1CN(C(C1CC(F)(F)C1)=O)CC2.C Cc1nn(C)cc1C(N1C(CNC(C2CCC(N(C)C)CC2)=O)CC2CC12)=O c1(CC(=O)NC2CN(C(C3(C)CC3(F)Cl)=O)C2)c(F)cccc1F c1(C(N(CC(C)NC(C(CC)(C)F)=O)C)=O)ccc(O)cc1[N+](=O)[O-] c1cc2ccccc2s1.C1(C(C)NC(C2(OCC)CC2)=O)CCOC1.C=O.N c1(C(=O)NC(c2ccccc2)C(=O)NC2(CC)CCOC2)cccc2nccn12 C=CC1(C(=O)NC2CCCN(C(=O)C=C(C)c3ccsc3)C2)CCCCC1 C(CC(CC)C(=O)N1CC(F)CC1CNC(=O)Cc1ccccc1)=CC Cc1cccn2nc(C(=O)OCC(c3ccc(F)c(F)c3F)=O)cc12 c1(CC)ccc(C(=O)NCC2CCCCN2C(=O)C(C)COC)c(C)n1 c1(C(=O)NCC(c2ccccc2F)NC(C=C(CCC)C)=O)c(C)cnn1C CC(C)(F)C(C)(F)C(=O)N.C1CN(C(C2C3(CC3)C23CC3)=O)CC1C(F)F C1(NC(c2cnc(N(C)C)s2)=O)CC2CCC1(Nc1ncccn1)C2 c1(OC)ccccc1N1CCC(NC(=O)NC(c2ncsn2)C)C1 c1(C(N2CCC(CC)C2C(N2CC3CC2CC3O)=O)=O)c[nH]c2ccncc12 c1(N(CCN(C(C(C(C)C)N)=O)C(C)C)C)nccc(C#N)n1.[SH](C)(=O)=O C12(C(=O)NCC3OCCN(C(CCC(=C)C)=O)C3)CCC(F)C1CC2 N1(C(CCN(CCC)C)=O)CC(O)(C(C)(C)CNC(=O)CCCC2CC2)C1 C(=O)(C(C)N(OC)C(=O)c1oc(C2CC2)nc1C)N1CCOCC(C(=O)OC)C1 Cc1cc(N2CCOC(c3cccnc3)C2)nc(N2CCC(C)(CN(C)C)C2)n1 C1(C(C2CCOCC2)NC(C2(F)CC2)=O)CCCCC1 c1cc(F)ccc1F.C12CCC(N1CC)NCC(=O)NC2.C(C)O.CC.O Cc1nc(C)c(C(N2CC(CCNC(=O)C3CC3)C(C)C2)=O)s1 C1(C(N2CC3(CN(C(C)=O)C3)C2)=O)CC2CCCC2N1.C12C(=O)C3CC1C2C3.C C(C)(C)(C(O)C(F)F)NC(CCC1CCC(NC(COCCOC)=O)C1)=O N1(C(C(c2cncnc2)C)=O)CC(CC(N2CC(C)(C)C2)=O)C2(CC2)C1 N1(C(Cc2n3c(nc2)C(C)CCC3)=O)CC(S)CC12CCOCC2 c1(C(N(CCC)C)=O)ccncc1.c1(C=O)cc[nH]c1C1CC1.C(C)(C)(C)O CCC(C)C(O)C(=O)NCCn1cc(CCN2CCCCC2)nn1.C1CN1 Cc1c(C(=O)NC2CN(C(c3cc(C)n(C)n3)=O)CC2(C)C)ccc2cncn12 N1(C(c2cn(C(C)C)nc2)=O)CC=C(C(=O)N2CCCC(C(C)(C)C)C2)C1 C1(N(C(Cc2cnc(C)s2)=O)C)CN(C(C2(CN(C)C)CCCCC2)=O)CC1O N1(CC(c2c(F)cc(C)c(F)c2)=O)CC=C(c2cccc(Cl)c2F)CC1 C1(NC(c2n(C(C)C)ccc2)=O)CC2CCC1CC2.C1(CC=O)CNC(=O)C1.N C1(C(=O)NCC2CCN(C(C3(CCCC)CCCC3)=O)CC2)COCC(C)(C)O1 c1(C(c2nnnn2CC(F)F)NC(CSCC)C)cn(CC2CC2)nn1 C1(OC)CC(CNC(=O)CCc2ccnn2C)N(C(=O)CCC2CCC2)C1 C=C=CC(C)C(=O)N(CCC(=O)N1CC(OCC(F)F)C1)C1CC1 c1(C(C)C)cc(NC2CCCN(C(c3cc(Br)co3)=O)CC2)n2ncnc2n1 N1(C(CCN(CC#C)C(c2ccnc(C)c2C)=O)=O)CCC(CO)CC1C N(C(=NCC(C)N1CCCCC1)NCc1cnc(C)s1)C(CC)C CS(=O)(=O)c1ccc(C(=O)NCC2(NC(c3ccoc3Cl)=O)CC2)[nH]1 c1(CC(N2CCC(CC)C2)=O)cnc2n1CCCC2C.C(=O)(C)N.[SH](C)(=O)=O C=CC(C(F)(F)F)NC(=O)CC(C)CNC(=O)COCCCCC C12(OC)CCCC1(C(=O)OCCc1ccnc(C3CC3)c1)C2 C12(C(N3CC(=CC)C3)=O)CC(CO)(CN1C(C1CC(OC)(O)C1)=O)C2 c1(NC(C2(C)N(S(CCC)(=O)=O)CCC2)=O)c(Br)c(C(=O)OC)nn1C Cc1cc(C(=O)N(C(C)(C(=O)NC(CO)C2(O)CC2)C2CC2)C)n(C)n1 C#Cc1ccc(C(N2CCC(CC)C2CNC(=O)C2=C(C)CCC2)=O)c(C)c1 c1(C(=O)NC2C(C)CN(C(C3(C)CC=CC3)=O)C2)c(NC(N)=O)cccc1F N1(C(C2(NC(C)=O)CCC2)=O)CCOC(C)(C)C1.C(C1CCOC1)=CC=O C#CCC(CC#C)NC(=O)CC(COC)NC(=O)Cn1cccnc1=O c1(C(N2C3CN(c4c(F)cnc(C)n4)C(C3)C2)=O)ccc(O)c([N+](=O)[O-])c1 C1(C(=O)NC2C(OC)CN(C(=O)CCc3c[nH]c(=N)[nH]3)C2)CC(C)(C)CN1C C(=O)(C(O)C(C)C)N.C(COc1ccccc1)(C(=O)N1CC(CCCC)C1)OC C1CCCN(C(c2nocc2C(C)(C)C)=O)C1.c1(C(NCC)=O)cc(C)cs1 c1(C(NOCC(=O)NCc2sccc2C(=O)O)=O)cnn2ccccc12 C(=O)(C1=C(SC)CCCC1)N1C(C)CCC(NC(c2cc(COC)no2)=O)C1 N1(C(c2c(C)ncs2)=O)C(C(=O)NCc2cnns2)CCC1C1CC1 Cc1cc(C(N2CCCCC2CNC(=O)C(F)C2CCOC2)=O)ccc1[N+](=O)[O-] C(=O)(CCC(=O)NN(C)C)NC(C)CN(C)C(C1(CO)CCCO1)=O c1(C(=O)NCCCCCCNC(=O)C#CC2CCOC2)ccc2nnc(O)n2c1 N1(CC2CCN(c3ncnc4ccc(C)cc43)C2)CCc2c(O)nc(C)nc2C1 c1(C(=O)NC2CCN(C(C(C)S(C)(=O)=O)=O)C2)cc(N)c(Cl)c(O)n1 c1(C(=O)NC2C(NC(c3ccc(O)cc3)=O)C2)ccc(F)c(Br)c1 CC1(NC(=O)CSCCC#N)CCN(C(c2cc(-c3ccncc3)on2)=O)C1 c1(C(=O)NC(CCN(C(c2c(OCC)cccn2)=O)C)C)sc(C)c(C)c1C N1(C(C2(F)CCN(C(c3ccc(OC(F)F)cc3)=O)C2)=O)CCC2(CCOCC2)C1 N1(c2c(C)c(N(C)CC3CCCN3C)ncn2)CCC2(CC1)CCC21CCC1 C1(C(N(C2CC3(CCC3)C2)C)=O)CN(C(=O)CC2CCCO2)CC1(C)C C(=O)(C1=CCCC1(C)C)NCC1CN(C(c2occ(C)c2C)=O)CC1C CC1CN(C(C)C(=O)NC(=O)NCc2ccccc2)CCCO1 C1(N(C(=O)C(CO)NC(C2CCCOC2)=O)CC)CCC(NC(=O)C)CC1 c1(C(=O)NC2(c3cn(C4C(SC)CCC4)nn3)CCC2)c(F)ccc(C)c1F N1(C(Cc2cc(C)[nH]n2)=O)CCN(C(C2CC(CF)C2)=O)C(CCO)C1 C1(OCC(C)C)CN(C(=O)CCNC(=O)C=CC2CCC2)C1 C(C(C)CC(C)C)NC(c1ccc(COC)o1)=O.n1(C(C=O)C)nccc1C.N C(C(C)C(F)C(=O)N1CC(C)(O)CO1)NC(C(C1CC1)OC)=O C(C(N=[N+]=[N-])C(=O)NCCOCCCNC(C1CCCC1)=O)OCC.C C1(NC(C(CCC)O)=O)CCN(C(c2ccn(C)c2CC)=O)CCC1CO Cc1cncc(C(=O)N(C2CC3CNC2C3)Cc2ncc[nH]2)c1 C1(SCc2n(C3CC(F)(F)C3)nnn2)CCC2(CCNCC2)C1 CC1CCC(CNC(=O)CC(C)(C)C)N(C(=O)CCC2CCC(O)CC2)C1 N1(C(C2C(c3ccc(C)cc3)CCCC2)=O)CC2(CCC2)c2cc(Br)ccc21 CCC(C)CC(=O)C(=O)NCC(C(=O)N(CCCC(C)C)C)N(C)C CC(CCc1ccccc1)CC(=O)NC(C)CCN(C)C(C1(C)CSC1)=O C1(C(N2CCCC(N3CCCCC3)C2)=O)CCCN(C2CCS(=O)(=O)C2)C1 N1(C(C=CC=CCC)=O)CC2CC1CN2C(c1nc(C)ncc1Cl)=O N1(C(C(c2c(C)cccc2)(F)F)=O)C(CNC(=O)CC2CC2)CC2COCC12 c1(C(N2C(CNC(C3OCCN(C)C3)=O)CC3(CC3)C2)=O)cc2n(n1)CCCC2 N(C(=NCC1CC12CC2)NCc1ccco1)CC(C1(O)CCOCC1)O C(=O)(CCCC1CCC1)N.C(=O)CC.N(CC)(CC)CC.C(=O)C1CC1 C(C(F)(C(=O)NCCN(CCCF)C)C(C)C)NC(c1cnn(CC)c1C)=O N1(C(CCCC(C)C)=O)CC2COCCC2(NC(C2CC=CCC2)=O)C1 C1(C(=O)NCC2CC2NC(c2ncccc2N)=O)(CC)CCC(F)(F)CC1 c1(C(N(CC#C)C2CC2)=O)c(C)nnn1C.C1(CC=O)CC2C=CC1C2.N C1(Nc2c(OCC(=O)OC)cccc2)(C)CC2CCC1C2.c1csc(C)n1.N C(=O)(C(CC(N)=O)NC(c1cncnc1)=O)N1CC(C(=O)NC)OCC1 c1(C(N2CC3C(NC(c4nc(Cl)c(Cl)s4)=O)C3C2)=O)ccc2scnc2c1 c1(CC(=O)NCC(Cn2cc(-c3cncs3)nn2)OC)ccc(Cl)cc1Cl N1(C(CC(CC)C)=O)CCN(C(c2nn(C)c(C)c2Br)=O)C(CC)C1 CCCCCCC(C)C(=O)NC1(COC)CCN(C(c2c(C)cc[nH]c2=N)=O)C1 Cn1cc(C(=O)NC2CCCCC2NC(=O)C2=C(Cl)CCC2)n(C)c1=O C=CC(CC)CC(=O)N1CCOC(C(=O)NC(c2nc[nH]n2)C2CC2)C1 C1(C(=O)NC(C(C)C)CNC(=O)C=CC(N)=O)CCCOCC1 C1(CNC(C(C)S(C)(=O)=O)=O)CCC2(CN(C(c3ccnc(Cl)c3N)=O)C2)O1 O=C(CS(=O)(=O)NC1CC(c2ccccc2F)C1)OCCOCC1CCCO1 Cc1nc2[nH]c(C(=O)N(CCCCCNC(C3CSC3)=O)C)cc2s1 N1(C(c2nc(Cl)cs2)C(=O)NC2(C)CC2)CC(=O)N2CCCCC2C1 c1(C(N(CCNC(C=C(CC)C)=O)CC2CC2)=O)cnc2c(c1)CCCO2 CC1CSCC1N=c1cccc(S(=O)(=O)NC2(C3CCS(=O)(=O)CC3)CC2)[nH]1 N1(C(CSC)=O)CCC2(CCC(NC(=O)CCC3CCCCO3)C2)C1 N1(C(c2c(C)nc(C)[nH]2)=O)CCC(F)C(NC(C2C(C)C2C)=O)C1 C1(C)CCN(C(C2CCC(C)(C)O2)=O)C1.C1(CCC#C)(CC(=O)N)OCCO1.C O=C(CC1=CCCC1)NCC1CCC(C)CC1.c1(CC=O)cc(F)cc(F)c1.N C1CN(C(c2c[nH]nc2-c2cnn(C)c2)=O)CC1O.C(C(=O)N)(C1CC1)SC.C C#CC1(C(=O)N(CC(C)CC)C2CC2)CCN(C(C2CN(C(C)=O)C2)=O)C1 c1(C(N2C(C#C)C(C)(C)C2)=O)c[nH]c2nc(Cl)ccc12 C(=O)(CC(C(F)(F)F)NC(c1ncn2c1CCC2)=O)N(CC(C)O)CC(F)F C1C2CC3CN(C(=O)C=CCN4CCCC4)C1C3C2.C(c1cc[nH]n1)=CC=O.N c1(OCC(=O)NCC(CC=C)NC(=O)CC2CC2(Cl)Cl)ccc(Cl)cc1F Cc1cnc2c(C(=O)NC)cnn2c1.C1(CNC(C2CC2)=O)CC1.N(C)C N1(C(CCc2c(OC)cccc2)=O)CCC(CNC(=O)C(C)C(C)O)C(C)C1 N1(C(c2cc(C)c(=N)[nH]c2)=O)CC=C(C(=O)NCCc2ncccn2)CC1 c1(OC)ccc2nccc(C(=O)NC3CC(C)(NC(c4ccccc4)=O)C3)c2n1 C1(C(C)O)CC2(C1)CN(C(=O)Cc1cccnc1)C2.C1(C)(S)CCC1.C(=O)C c1(C(=O)NC2CN(C(c3c(O)cc(C)nn3)=O)CC2F)cn(C)c(C)cc1=O C#Cc1cccc(C(=O)N(C)CC2(NC(=O)C(C)n3cccc3)CC2)c1Cl N1(C(C2(OCC)CCC2)=O)CC2(C1)CN(C(=O)C1=CCSC1)C2 c1(C(=O)NC2C(N(C(CCCC#C)=O)C)CCCC2)ccn2c(C)cc(C)nc12 c1(N2CCN(C)CC2CNC(c2ccc(Cl)nc2Cl)=O)nc2cccc(F)c2s1 c1(CC)cc2c(c(=O)o1)C(c1nnsc1Br)N(C)C(=S)N2CCC#N c1(C=O)cc(F)c(F)c(O)c1F.C(c1cccc(Cl)c1)=CC(=O)NC1CCC1.N Cc1cccc(C(C)Nc2cc(NCCCS(C)=O)ncn2)c1C c1(CCC(N2CCC(OC3CCOC3)CC2)=O)ccc(O)c(O)c1 CCCC(F)C(=O)N(CCCNC(=O)COc1ccon1)C1CC1 N1(C(=O)NC2CC(C)SC2)CCN(C(=O)C(=O)N(C)C)CC1 C1(NC(C2(OC)CCSC2)=O)CCC(NC(=O)CC2CC2(C)C)CC1 C1(C(=O)NCC(CC)N(C(=O)Cn2nccc2C)C)CC2CC1CC2O CC1(C)CC(CC(N2CCCN(C3CC3)CC2)=O)N(C(C2CC3CCC(C2)C3)=O)C1 C(=O)(N1CCC(C(=O)NC(C)C(C)(C)CC)O1)c1c(C)cc(CC)o1 O=C(Nn1ccccc1=O)C1=NOC(CNC(=O)C(CO)C(F)(F)F)C1 c1(COC)nc(Cl)cc(=NCC(C(C)(C)C)NC(=O)C(C)(F)C(C)(C)F)[nH]1 CCC(C)(C(=O)N1CC(OCCNC(=O)COc2ccccn2)C1)OC CC(O)C(F)(F)C(=O)NCC(C)(C1CCC1)NC(C1COCCOC1)=O c1(C(N2CC3(CN(C(C(c4ccncc4)C)=O)C3)C2)=O)[nH]nc2c1COC2(C)C c1(CC)ccccc1.C1(CNC(CSCCN)=O)CCC1NC(=O)CS C(=O)(CCC(F)(F)CN=[N+]=[N-])NC1CN(C(C(CC)CO)=O)CC1C(F)(F)F c1cc(=NCc2ccc(C)c(Cl)c2)[nH]c(C(F)(F)F)n1.C(CCCNCCC)SC c1(CN2CC3C(C(=O)Nc4c(C(N)=O)ccs4)C3C2)c(Cl)c[nH]c2nccc1-2 c1(C(=O)NC(CCC)C(=O)NC(c2nccn2C)C)ccc(C)c(CO)c1 CCC(F)(F)CCNC(c1c(CNC(C2(C)CCSCC2)=O)nnn1C)=O O=S(=O)(c1cnc(N2CCC3C(C2)C3(F)F)c(Cl)c1)NCCCCn1cnnc1 Cc1ccc([N+](=O)[O-])c(C(=O)NC2CCCN(C(c3cccc(Br)c3)=O)C2)c1 N1(C(C(C)c2ccco2)=O)CC=CC(NC(c2[nH]nnc2-c2ccccc2)=O)C1 c1(CC(N2CC(CC(C)NC(c3ccc(CO)nc3)=O)C2)=O)nnc(O)nc1O Cc1nccc(Cl)c1C(=O)NC12CC(C1)C2.c1(C=O)cc(C(F)(F)F)cs1 Cc1cccc(COCC(=O)NC(C2CN(c3ncns3)CCO2)C)c1 C(=O)(CCC(C)(C)C)N(C1CCCN(C(=O)Cc2csc(S)n2)C1)CC N1(C(c2cncc(NC)c2)=O)CCCCC(CNC(C2(C#N)CC3CC3C2)=O)C1 c1(SC(C(=O)NCC(C)N(C(C(c2cnn(C)c2)C)=O)C)C)ccnn1C CC1CCCC(C(=O)NCC(C)NC(=O)Cc2ccco2)O1 N1(C(c2ncn(C)c2)=O)CC=C(C(=O)NC2(C3CCCO3)CCC2)C1 C(=O)(C#CC1CCCO1)N1C(CCN(C)C(C2CC3C=CC2CC3)=O)CCCC1 N1(C(=O)OCC)CCCC2CCN(C(c3nc(C(C)C)ncc3NC)=O)CC12 N1(C(CCc2n(C)ccc2)=O)C2CCC1CC(NC(c1ccnc(Cl)c1)=O)C2 C1(NC(CN(C)C)=O)CCOC12CCN(C(c1cc(C3CC3)ccn1)=O)CC2 N1(C(c2c(C)oc(C#N)c2)=O)CC(NC(=O)CC23CCCC2C3)C2CCCC12 c12cccc(c1)CNC2=O.c1(NC(C2CCN(CC)C2)=O)ccccc1C CCCCCCCCC(=O)NCC(C)CNC(C1(CC)CCOC1)=O c1(OC)c(C(N2CCC2(C)CCO)C(=O)Nc2ccccc2C)cccc1F Cc1ccc(CCC(=O)NCCCCC2CN(C(c3ccc(F)cc3)=O)C2)cn1 c1(C(N2C(Cn3cc(C(C)OC)nn3)C(C)(C)C2)=O)cc(Cl)c(F)cc1F C1(C(=O)OC)CC2OCCC2N1C(=O)C(C1(O)CCOCC1)(F)F N1(C(=O)Nc2c(SCCC)cccc2)CC2(CCCC2)C1COC c1(CC(=O)NC2(C)CC(NC(C(CC(C)C)O)=O)C2)ccc2nc[nH]c2c1 C12(CC(=O)N)CCC(CC1)OC2.C1(C=O)CCS(=O)(=O)C1.C1CC(F)C1.C N1(C(=O)OC(C)(C)C)CCOC(C2CC2)CC1.c12nc(=N)nc([nH]1)SCCC2 c1(C(=O)OC)nn(C(F)F)cc1NC(C1CCOCC1)C.C(C)(C)C.C=O N1(C(C2(CC=C)CC2)=O)CCCC1CCC(=O)C(N1CC(CCC)C1)=O N1(C(C(CC)C)=O)CCN(C(c2ccc(F)c(C(F)F)c2)=O)C2(CC2)C1 C(CCCC(C)(C)C(=O)NNC(=O)c1ccc(N)cc1Cl)NC(COC)=O CC1=C(C(=O)NC2CC2NC(=O)CCN(C)CCO)C(C)(C)CCC1 C1(C(=O)NCCCCOC)C2CC(O)C(C2)N1C(=O)C=C1CCOCC1.O c1(C(N2CCN(C(C(CC)N(C)C)=O)C(CF)C2)=O)cnc2[nH]c(C)nc2c1 c1(C(=O)NCC2N(C(c3c(CC)nco3)=O)CC(OC)C2)ccc(C#N)n1C c1(SC)cn(C)nc1C(=O)NC(C)CCN(C(=O)Cc1ccc(O)cc1)C N1(C(C(C(=O)OC)C)=O)CC2(CCCC2)C1C(N1CC(CC(F)F)C1)=O Cc1cnc(C(N2CCC(OCCNC(=O)C=CBr)C2)=O)cc1C C(C)(CCCCNC(C1CC1(C)C(C)C)=O)NC(C=C(C)C)=O C(CN=c1nc(C)[nH]s1)(N(C(c1cc(OCC)no1)=O)C)C1CC1 C1(OC)CCC2(C(N3CCC(CC(=O)NCCCOC4CCC4)C3)=O)CC12 CC(C)CC(CNC(=O)C(C)CSC(F)(F)F)NC(c1cc(O)ncn1)=O c1(C(N2CCOCC(NC(c3c(C)cnn3C)=O)C2)=O)cncc2sccc12 CCCCC(F)C(=O)N1CC(C(F)Cn2cc(-c3ccc(C(F)F)nc3)nn2)C1 c1(CC)ccc(C(=O)N)cc1N.C1(C)CCN(C(C23CC(C)(C2)C3)=O)CC1.C CCCC(C)(CCC)C(=O)N1CCC(N(C(C2CCCC(=O)N2C)=O)CC)CC1 CCC(C)(C)C(=O)NCC1CCCN1C(C1(n2cccn2)CC1)=O c1(CC)ccnc(C(=O)NC2CC(CNC(=O)CC(C)CN(C)C)C2)c1 C1(C)(CNC(CC2C(C(=O)OC)C2)=O)CCCN1C(=O)C.c1cn[nH]c1 c1(C(=O)NC(C)CCNC(C2C=CCC2)=O)ccc2c(n1)NC(=O)CO2 c1(C(C(=O)NCC=C)N(CC(C)OC)C)ccc(OC)c(SC)c1 N1(C(C(Cc2cc[nH]n2)NC(C(CCC)CC)=O)=O)CCOCC(F)(F)C1 c1(-c2nc(Cc3ccc(C)cc3)n(-c3cccnc3)n2)cccc(S(C)(=O)=O)c1 CC1CCOC(C(=O)NCC(C)(C)C(=O)N2CCSCC2C)C1 c1(C(=O)NCCCC2N(C(c3ncc(NC)nc3)=O)CCC2)c(C)ncnc1O c1(C(=O)NCCCCNC(c2ccc(C)c(CO)c2)=O)cc(O)c2ccsc2c1 N1(Cc2c(C(=O)OCC)c(OC)ns2)c2ccncc2CC1C.C(C)C CC(C)C(O)C(=O)NCC1(F)CN(C(C2OCCOC2c2ccccc2)=O)C1 c1(N2CCC(NC(C)=O)C2)ccncc1S(=O)(=O)N1CCN(C)C2(CC2)C1 c1(C(=O)NC(C)CCN(C(=O)Cc2cc[nH]n2)C)cc2ccccc2o1 n1(CC(=O)N(CC(C)(C)CNC(c2sccc2F)=O)CC)ncc(Cl)c1C c1(-c2c(C(N(CC(C)O)C)=O)nco2)ccc(C)cc1.C1CC1C=O.CCO C1(CC)CCN(C(=O)CC(CC)N(C(=O)CC2(C)OCCO2)C)CC1 N1(C(CC2CC(=C)C2)=O)CC2CCCC2(CNC(c2cnn(CCC)c2)=O)C1 C(=O)(C(C)(C)CN=c1[nH]c(=NCc2ncoc2CC)c2cc(Cl)ccc2[nH]1)NC c1(NC(C2CC(=C)CN2C(c2ccc(Cl)c(O)c2)=O)=O)cnc(Cl)nc1C N1(C(C2(CCCC)CC2)=O)CCC(O)(CCOC)C1.C123CC1CN(C2)C3=O Cc1cc2ccc(NC(C3CN(Cc4cnn(C)c4C)CCO3)=O)cc2[nH]1 Cc1ccc(C)c(C(=O)NCCCc2nn[nH]n2)c1N C=C=CC(C)C(=O)NCCCCC1CCCN(C(C2(COC)CC2)=O)C1 N1(CC(=O)N(C)CC)CCC(C(=O)NC(C2OCCO2)C)CC1 N1(C(C2(CC)COC2)=O)CCC2(C1)c1[nH]cnc1CCN2C(=O)C1=NOC(C)C1 C1(c2cn(C3CN(C(C4CC4C#N)=O)CC3O)nn2)(CC(=O)OC)CCOCC1 c1(C(N2CC(COC)(CNC(=O)C)C2)=O)ccnc(Cl)c1.C1CC1.O C1(C=O)Cc2c[nH]cc2S1(=O)=O.C1C=CCC1.C1(C(=O)N)(NC(N)=O)CC1 Cc1cc(C(=O)NC(C2CCN(C(=O)CN(C3CCC3)C)C2)C)c(C)cc1Cl c1(C(=O)NCCC2(O)CN(C(Cc3n[nH]c(=NC)s3)=O)C2)cnc(O)cc1C c1(CNC(C(C2CN(C(C3(C(C)=O)CC3)=O)C2)O)=O)cc(O)ns1 C1(NC(c2n(C(C)C)nc(C3CC3)c2)=O)C2CC1CN(C(=O)C(C)(C)C)C2 C1(CNC(Cc2cc(C)sc2C)=O)CC(C)CN(C(c2ccc(O)c(N)n2)=O)C1 C#Cc1cc(C(=O)NC(CC)CC(=O)NC(c2cccs2)CC)ccc1C C=CC(C)CC(=O)NC1CC(CCNC(c2cnccc2N2CCOCC2)=O)C1 C(=O)(CCCN=c1nccc[nH]1)NCC(=O)Nc1n2c(nc(C)c1C)ncn2 N(C(=NCCN1CCC1)NC1CCN(c2ccc(F)cc2F)C1)C(C#C)C CC(C)CC(C(=O)NC1CC(C)N(C(c2ccc(F)nc2)=O)C1)n1ccnc1 c1(CNC(=O)NC2(c3ccccc3)CCOC2)cccnc1Br c1(SC)cccnc1C(=O)NCC1CCCC(NC(c2cccc(=O)o2)=O)C1 c1(Cc2ncc(C(=O)NC3CC3NC(C3CCOC3=O)=O)s2)ccccc1F N#CC1(C(N2CCC(CCCNC(C3COCCO3)=O)CC2)=O)CCCCC1 C1(C)(CCC(=O)N(C(CC)C)C)CN(C(=O)C(C)SC)C1 C1(C(=O)NC(C)CCCNC(c2coc(O)n2)=O)CCc2ncc(Br)n2C1 N1(C(C2CCc3ncnn3C2)=O)CCC2C(CCN2C(c2ncccc2F)=O)C1 c1(COC)ncsc1C=O.c1(C(N(CCC)C)=O)sccc1-n1cnnn1.N c1(C(=O)NCC(C)CN(C(=O)C(O)c2ccsc2)C)cnnc(O)c1 N1(C(c2ccc(C)c(C)n2)=O)CCN(C(=O)Cc2ccon2)CC12CCC2 C1(NC(CCn2ncc(C)c2)=O)CCCC(C(=O)NCCCC2CCOCC2)C1 c1(OC)ccc2cc(Cl)nc(N3CCOC(c4c(OC)cccc4Cl)C3)c2c1 Cc1ccccc1NC(=O)C(C(C)C)N1CCC(CN2CCCC2=O)C1 C1(CSc2c(C)nc(C)s2)Cn2c(-c3ccccc3)nnc2S1 c1(CC(=O)NC2CCC3CC23)noc2ccc(O)cc12 Cc1oc(C(=O)NCC#CC)cc1S(N)(=O)=O.C1(C=O)CC(n2cccn2)C1.N C1(O)(CNC(c2scc(CNC(C3(CCC)CC3)=O)c2)=O)CCOCC1 Cc1c(C(=O)NCCOCCNC(C2(C)SCCCS2)=O)cccc1N O=C(CCC1CCCCO1)NOCc1cn(C2CCCCC2)nn1 C1(CNC(CCc2n(C)ncc2)=O)CCC2(CCC2)CN1C(=O)Cc1cccs1 N1(C(=O)C=C(C2CC2)C2CC2)CCC2(CCN(c3ncnc4c3CCC4)C2)C1 c1(C(N2CC(CNC(=O)CO)CC(C)(C)C2)=O)cc2ccc(Cl)cc2[nH]1.CCF c1(OCC)ccc(N)c(C(N2CC(NC(C3CC3(C)C)=O)CC(O)C2)=O)c1 N1(C(CNC(=O)CCCCO)=O)CCC2(CCCN2C(C2CCSC2)=O)CC1 C1(NC(c2ncc(C)nc2)=O)CN(C(=O)COC2CCCOC2)CC12CC2 C=CCC(CC(=O)N(CC(=C)C)CC(=C)C)NC(=O)CC(C)CC C(C)(C(C)C(=O)NCCCOC(C)C)NC(c1ccn(CCC)n1)=O N1(C(c2c(C)nsc2N)=O)CCC2(CCCN(C(C3(C)CC3C)=O)C2)CC1 c1(Cc2nc(-c3n(C(C)C)ncn3)n(CC3CCCCO3)n2)cccc(Cl)c1Cl C1CN(C(=O)C=C2CC2)CCC1(C)C.C(C(=O)NC)N(S(C)(=O)=O)C Cc1cc(=NCC2CC(C)CO2)[nH]c(Cl)n1.C1(C(=O)N)CCCN1S(C)(=O)=O C1(NC(C(C2CC(NC(CSCC#C)=O)C2)F)=O)COCCN(C)C1 c1(SC)cncc(C(N2CC(F)CC2CNC(=O)CCCC)=O)c1.C(N)=O.N C(=O)(C1=C(C)NC2=NCCCC2=C1)NCC(C)NC(Cn1ncc(C#C)c1)=O N1(C(C(C(CC)C)O)=O)CCC2CCC(C1)N2C(c1ccn(C(C)C)c(=O)c1)=O N1(C(C=CC(=O)N(C)C)=O)CC=CC(CC(N2CC(c3ccccc3)C2)=O)C1 Cc1nnc(-c2ccccc2)n1CC(=O)NCCOC1CCCCO1 N1(C(CCCOCC)=O)CCCC(CCNC(C2(C)CC=CCC2)=O)CC1 N1(C(c2c(N)cc(S(N)(=O)=O)cc2)=O)CCC2(CCc3ccccc3C2=O)CC1 N1(Cc2ccc(C)c(Cl)c2)CCC2(CCCC2C(N2CC(=O)NC(C)C2)=O)C1 c1(OC)cncc(C(=O)NC2CC2NC(=O)C(C)C)c1C.c1ccccc1F.S c1(C(=O)NC(C2CCN(C(c3ccoc3)=O)C2)C)snc2ccccc12 CCCCC(CC)CC(=O)N1CCCC(NC(=O)C(C)NC(=O)NC)C1 Cc1nn(C)c(Cl)c1C(N1CCCC(CCCO)C1)C(=O)NCCCOC1CC1 CCCC(CC)C(=O)NCC1CCC(C(=O)N(CCN(C)C)CC)CC1 Cc1cc(CCC(=O)NCC2(C(N)=O)CN(C(C3CC4CCC3C4)=O)C2)nn1C CCCC(CC(=O)NCCCC1(O)CC1)NC(C1(CC)CCCC1O)=O Cc1nc(-c2ccccc2)c(C(=O)NC(C(F)(F)F)c2ccccn2)s1 Cc1ncc2n1CC(C(=O)NC1CC3C1CCN3C(c1sccc1C#N)=O)CC2 CC1(C)C(C(=O)NC2CC(C(=O)NCC3C(CO)C3(F)F)C2)C1(C)C N1(CC(=O)NCCC2(C)N=N2)C(=O)OCC12CN(C=O)C2.C(C)(C)C.O N1(C(c2csc(C)c2C)=O)CCC2(COC(CNC(c3ccc(O)nn3)=O)C2)C1 c1(C(=O)NCc2n(C)cnc2)noc2cc(-c3ccc4scnc4c3)ccc12 c1(NCC)ccc(Cl)cc1C(=O)NCCCC(C)C.C(=O)C(O)C(F)(F)F.N C1(NC(c2ccc(F)c(F)c2)=O)CN(C(=O)CCOC2CCOC2)CC1C1CC1 C1(C)(C(N2CCN(C(C)=O)CC2)=O)CCCN(Cc2cccc(C(C)(C)C)c2)C1 C(=O)(C1=C(C)OCCC1)N1CCC(C(=O)NCC(C)(C2CC2)OC)C1 C1(F)(CNC(=O)CCNC(c2cc(F)c[nH]2)=O)CC(O)C1 C1(NC(C(N2CC(C=C)C2)=O)(C)C)CCCCC1OC(F)(F)F CC(C)(C)CN=c1[nH]c2ccc(S(=O)(=O)NC3CCCC3CO)cc2s1 N1(C(CCCCCN(C(c2cc(C)c(O)nc2)=O)C)=O)CCCC2COCC12 CC(C)C(CC(=O)N(c1cnn(C)c1)C)NC(=O)CN1CCOC1=O Cn1cc(C(=O)NCc2ccc(CNC(c3n[nH]cc3Br)=O)cc2F)ccc1=O C=CCCCCC(=O)NCC(O)CC(=O)N(C)CC1CC(F)(F)C1 N1(C(C(CCCC)C)=O)CCC2(CCC2NC(c2cc(COC)no2)=O)CC1 c12ccnc(c1)NC2C1CCC1.c1(CC(=O)OC)ccn(C)n1 N1(C(c2cncc(C)c2)=O)CC2CC(NC(c3cc(Cl)c(Cl)[nH]3)=O)CC2C1 CC1(C)C2CCC(C2)C1C(=O)NCCCCNC(c1ncc(Br)cn1)=O N1(C(c2cc(CN3C(CC)C(=O)N3)[nH]n2)=O)CCn2cc(C)nc2C1.CC c1(NS(C)(=O)=O)ccccc1C(=O)NC1CCC1.C12(C(=O)N)CCC1C2 C1(CNC(C2(CC=C)CCCC2)=O)(NC(C2C(C)CC2C)=O)CCOCC1 N1(C(CC=O)=O)CCCC(F)(CNC(=O)CCSC2CCCC2)C1.C1CC1.N c1(C(=O)NCCCCC(CO)NC(CC2CC(C)C2)=O)ccnc2ccsc12 N1(C(c2ccc(C)nc2O)=O)CC2CCCCN2CC1CNC(c1cnns1)=O C(=O)C(F)C(C)(F)F.c1(C(C)(C)C)c[nH]cc1C(=O)NC(C1CCOC1)C.N c1(CNC(CC)=O)cn(CC(N2CCC2CC(=O)NC)=O)nn1 CC1CCCN1C(=O)C=CC(=O)N(C)C.N(C)(S(N)(=O)=O)CC(=O)N Cc1cccc(C(=O)NCC(C2CCOC2)NC(=O)C2=CCOC2)c1Cl c1(CC(=O)NC2(CF)CCN(C(=O)CCc3cnn[nH]3)C2)ccccc1[N+](=O)[O-] C1(F)(C(=O)NC2CCN(C(=O)CCc3ccccc3)CC2F)CCCCC1(F)F C12(CNC(=O)Nc3nnc(C(C)(C)C)s3)CCC(CO)(CC1)CO2 C(CCCCNC(=O)C=C(C)Cl)NC(C=CCN(CC)CC)=O C1(NC(c2cnc(CC)s2)=O)CC(C2CCN(C(c3cccnc3N)=O)C2)C1 C(=O)(CC1=CCOCC1)NC1(CC=C)CCN(C(=O)CN2CCC(F)(F)C2)C1 c1(CCC(=O)N(CC(C(=O)NC)C)C)c(C)nc2nnnn2c1C CN1CCN(CC(=O)NC2(C(N3CCOC(C4CCC4)C3)=O)CC(CO)C2)CC1 c1(CN2C(C(F)(F)F)CC(C)C(C)C2)c(Br)ccc2c1OCO2 C(=O)(C1=CC2(CCN(C(c3ccnnc3)=O)C2)C1)NCCCc1n(C)nnn1 Cc1ncc(C=CC(N2CCOC(C)(CNC(c3cccnn3)=O)C2)=O)c(O)n1 Cc1cc(F)c(C(=O)NCC2CC(C)CO2)c(F)c1.C(=O)(C(F)(F)CO)N c1(N(CCCN(CC)CC)C)ccc(S(=O)(=O)N2CCC(C(F)F)C2)cc1C#N c1(N(CC(CCC)=O)C(=O)CCc2cc(O)ccc2C)ccc(Br)c(F)c1 C#CC1(O)CCN(C(c2ccc(CNC(C3C=CCCC3)=O)cc2)=O)C1 C1(NC(CCSCCCC)=O)CCCC1C.c1(C=O)c[nH]nc1C(F)(F)F.N c1(OC)ccc(C(=O)NCCCNC(C2CC23CCOC3)=O)c(C)c1 C1(NC(CCC(=C)C)=O)CCC12CN(C(=O)Cc1cc(C)nn1C)C2 N1(C(c2c(C)nns2)=O)CCN(C(c2ccc(OCC(F)F)cc2)=O)C(C)C1C Cc1cc(OC(F)F)c(C(=O)NC2CC2)s1.N1(CC=O)CC(=O)NC1=O.C C12(NC(c3cc(Cl)ncc3Cl)=O)CCCC1N(c1ncc(F)cn1)CC2 C=C(C)CN=C(NCC1(C)CCCC1C)N1CCn2c(nn(CC(F)F)c2=O)C1 CC(C)CCC(F)C(=O)N1CC2CCCC2(CNC(=O)Cc2cccn2C)C1 c1(-c2ccc(C)o2)nnc(N2CCC(c3ccc(F)cn3)C2)n1CC1CCCO1 C1(C(=O)NCC2CCN(C(CCCCOC)=O)CC2C)CCCC2C1C2(F)F c1cnn2c1CN(C(C1CCCC1C1CC1)=O)CC2.C(C)(C)(C(=O)NC)OCC c1(C(=O)NCC(C)(C)NC(c2ccc(CC)cc2)=O)c(Cl)ccc(O)c1F C1(C(C)C(N2C(CO)CC2CO)=O)CCN(C(c2ccc(C#N)s2)=O)CC1 N1(C(C2(C)CC(C#N)C2)=O)CCC(C2CCCN(C(c3ccnc(F)c3)=O)C2)C1 N1(C(Cc2c(CC)cc(F)cc2)=O)CCC(C)N(C(=O)CN)CC1.[SH](C)(=O)=O c1(NC(C=CCC(C)(C)NC(c2cc(C)cc(F)c2)=O)=O)cnn2c1CCCC2 c1(C(N(CCNC(C2CC2COC)=O)CC)=O)cc(Cl)c(F)cc1 CC(CC(C)NC(c1ccc(C2CC2)s1)=O)NC(=O)CCCn1cccn1 C1CC2(C1)CN(C(=O)C(C)C(C)(C)C)C2.c1(NCC)nc(C)c(C=O)s1.N CC1CCN(C(=O)CSCCC#N)CC1NC(=O)Cc1cccc(C(N)=O)c1 Cc1occc1CN(C(=O)C(C)(C1CCC1)NC(C)=O)C C(=O)(C(S(C)(=O)=O)C1CC1)N(C1CCCN(C(CCCC)=O)C1)C C1(C(N2CCC(N(CCO)CC3OCCCO3)C2)=O)CCc2cc(F)ccc2O1 O=S(=O)(c1cccc(=NCC2CCCCC2)[nH]1)NCC1CC(C2CC2)C1 c1(N(C)C)ccc(C(=O)OCc2cn(C3CCOCC3)nn2)cc1F N1(C(c2ccc(C)nc2C)=O)CCCC2(CCC(NC(C3CC(CF)C3)=O)C2)C1 Cc1c(Cl)ccc(C(N2CC3CC2CN3C(=O)Cc2cc(F)cc(Cl)c2)=O)c1F C1(N(CCO)Cc2cnc(C)o2)CCCN(C(=O)Cc2csc(C(C)(C)C)n2)C1 c1(C(=O)NCCCN2CCN(C(c3cc(C)oc3)=O)CC2)cnn2cnnc2c1 C1(NC(CCCC#N)=O)CCN(C(c2cncc(Cl)c2Cl)=O)CC1CO c1(C=O)cccc2ncnn12.C1(NC(CCNC(COC)=O)=O)CC(O)(C)C1 C1(CNC(=O)Cc2cscn2)CCCC1NC(=O)CCN1CCCCC1 c1(OC)c(F)ccc(C(=O)NC2CCCN(C(=O)C(C)C(C)O)C2C)c1F N1(C(C)=O)CC(O)CC1C(=O)NCC(Cc1cccnc1)CN c1(C(N2CCn3nncc3C2)C(=O)NCCCF)cc(F)c(Cl)cc1Cl C1(C(C(=O)NCCSCCOC)C)CCCN(C(C2(O)CC(C)C2)=O)C1 C1(CC)(NC(c2nc(C)oc2O)=O)CCCN(C(C2CC3(CCC3O)C2)=O)C1 n1(CC(=O)NCC(C)=CC(=O)NCC2CC2C)cccn1 c1(NC(C(CC#C)NC(=O)CCn2cnc(=N)[nH]2)=O)ccc(F)c(CO)c1 C1(CC(=O)Nc2c(C)noc2C)CCCN(C(=O)Cc2ccncc2)CC1 Cc1cncc(CNC(=O)C(c2cccnc2)NC(=O)Cc2cncs2)c1 C(=O)(C(C)(C)CC(F)(F)F)N1CCC(NC(CCCCNC(C)=O)=O)C(C)(C)C1 C1(CNC(C2(NC(=O)C=Cc3cc[nH]n3)CCCC2)=O)CC(O)C12CCC2 C1(NC(C(C)CC(N)=O)=O)CC2(CCN(c3nncs3)CC2)C1 Cc1ccc(C)n1Cc1cccc(C(=O)NCCC2CNCCCO2)c1 N1(C(c2c(C)ncnc2)=O)CC=C(C(=O)NCC2CCCNC2=O)C1 C1(CNC(c2cnns2)=O)CCCC2CN(C(=O)C(c3ccccc3F)F)CC12 c1(NCCCCCC(C)C)cc(Br)c(O)cc1F c1(C(N2C(C)CC(NC(=O)C(=O)NCCC(N)=O)C2)=O)cccc2oncc12 C(=O)(CCN(C(C1(CNC(=O)C(C)SC)CC1)=O)CC)OCC c1(OCCOC)ccc(C(N2CCC2)=O)cc1.C1(C)(C=O)CCC(=O)C1.C c1(C(=O)NC2CC(C)N(C(c3csc(S)n3)=O)CC2)cc(C#N)ccc1Cl c1(C(N2CCOCC2)=O)ccc(C#N)cc1F.C1(C(=O)NC)(OCC)CCCC1 C(=O)(CCP(C)(C)=O)N1CCC(NC(C(C)N(CC)CC)=O)CC1 C1(C(CC)CC)CCCN(C(C2C3CN(C(=O)OC(C)(C)C)CC23)=O)CC1 c1(OC)cc(C)cc(C(=O)N(C2CCN(C(=O)CC3CCCCCC3)C2)C)c1O Cc1cc(C(=O)NC2CCN(C(CN)C(C)C)CC2)ccc1F C(C)(C(C)(C)C(=O)NCCCCCc1cn(-c2cncc(Br)c2)nn1)OC C1(NC(C2CCC(C(=O)OC)C2)=O)CC(C)CN(C(=O)Cc2cccn2C)C1 C1(CNC(c2n(CC=C)ccc2)=O)CC(OC)CN1C(=O)C(C)c1cc[nH]n1 C1(C)(NC(c2cc(C)ns2)=O)CCCCC1C(=O)NCC(=O)NC1CCC1 S(=O)(=O)(c1cc(C)cnc1NC1CCC(C)C1)NCCc1ccc(C)cc1 C1(C(=O)NC2(C(=O)NC)CC2)CCC=CC1.C(C1CCOC1)=CC(=O)N c1(CC)ncc(C(=O)N(CCNC(=O)CC23CCCC2C3)C(C)C)[nH]1 c1(CC(C)(C)C)ncc(C(=O)NCC2CCC2)o1.c1nccs1.C(=O)C.N CCC(CCC(=O)N=c1cc(C(N)=O)n(C)[nH]1)NC(=O)C#CC1(C)CCCO1 CC1(C)C(C(=O)NCC2CN(C(N)=O)C2)CCN1C(C1CCO1)=O CC(=O)C(C)(C)CC(=O)N1CCC(CNC(C2CC23CCC3)=O)C1(C)C c1(CC(=O)NC(C2N(C(C(C)SC)=O)CCC2)(C)C)ccc2n[nH]cc2c1 O=C1CCCCC(C(=O)NCC2CC(C(=O)N(CCF)C3CC3)=NO2)N1 C(=O)(C(C)CC(C)C)N1CCC(NC(c2c(C)cccn2)=O)(CF)C1 Cc1cn2c(-c3nc(C(C)O)nn3-c3ccc(Cl)cn3)cnc2s1 C1(C(=O)NC2CCC(NC(CCNC(=O)NC)=O)C2)CCCCNC1=O C1(C(=O)NC2CCCC(NC(Cc3c(C)noc3C)=O)C2)CC2C(C1)C2(C)C Cc1nccc(CCC(N2CCC(C)(NC(C3CC3(F)F)=O)C2)=O)n1 N1(C(CCC(CC)C)=O)CC(CNC(C2(CF)CCOCC2)=O)OC2(CCC2)C1 c1(C(=O)NCC(C)N(C)C(c2ccncc2N)=O)ccc(-c2coc(O)n2)cc1 C(C)(CCC(=O)NC(C)CCCNC(=O)COc1ccccc1Cl)OCC c1(C(=O)NC2CC3(C(NC(=O)C4=C(Cl)CC4)C3)C2)ccc(OC(F)F)cc1.O N1(C(c2c(OC)ccc(C)c2)=O)C2CCC1CN(C(=O)C(F)C1CC1)C2 Cn1ncc(C(=O)NCC(O)C)c1C(F)(F)F.c1(CCC=O)ccc(=N)[nH]c1 N1(C(CSC(C)C)=O)CC2OC(=O)N(C3CCN(C4CCCC(C)C4)CC3)C2C1 S(=O)(=O)(CCCCCl)N1C2CN(c3ccnc(OC)n3)CC21 C1(C(N2CC3CC2CN3C(C2CC3CC3C2)=O)=O)(CC)CCC(O)CC1 C=CCC(C)(O)C(=O)N1CC(CC(F)C(=O)NC(c2noc(C)n2)C)C1 Cc1[nH]c(NC(C2CN(C(c3cn(C)cn3)=O)C2)=O)c(C#N)c1C c1(CCC(C(=O)OCC=Cc2ccccc2)C)ccc(F)c(F)c1 C1(CCC)CN(C(C2CC(=O)N(C)C2)=O)CC1C(=O)NC1(CO)CC1 C1(C)(C(=O)Nc2nc(C)sc2)CCN(Cc2ccc(C3CC3)cc2)C1 Cc1cc(C(C)NC(=O)C(Cc2cc[nH]n2)NC(=O)CCc2cnccn2)no1 O=C(C1=CS(=O)(=O)CCC1)NC.C1CN(C(=O)CN2CCOC2=O)CCC1(F)F c1(C(=O)NC2CN(C(C3C(C)(C)C3)=O)C2)cnc(Cl)c(F)c1N N1(C(c2nc(C)sc2C)=O)CC(C(=O)N=c2ccn(C(C)(C)C)[nH]2)C2(CCC2)C1 N1(C(C(C(C)C)O)=O)CC(C)OC2(CCN(C(c3cc4n(n3)CCCC4)=O)C2)C1 C1(NC(C2CCS(=O)(=O)C2)=O)CC2CCC1CN(C(=O)C1=CS(=O)CCC1)C2 c1(CC)nc(C)oc1C(=O)N(CC(O)CN(C)C(c1nonc1CC)=O)C C(=O)(CCC(N)=O)NCCN(CCOC)C(c1cc(-c2ccco2)c[nH]1)=O C1(C(=O)OC)Cc2c(Cl)cccc2CN1C(c1[nH]cnc1C)C(=O)NCCCF c1(OCC)ccc(OS(=O)(=O)N(C)C2CC(=O)NC2=O)c(Br)c1 c1(C(N2CCCC(CNCc3ccc(Br)[nH]3)C2)=O)ccccc1-c1cnco1 N#Cc1c(I)nc[nH]c1=NCc1nc2c(n1C1CCCC1)CCCC2 c1(CN2CC(C(C)(C)COC34CC(F)(C3)C4)C2)ncccc1O N1(C(C(C)OC)=O)CCCC1C1CCN(C(C2CCN2C(C)(C)C)=O)C1 Cc1cccc(C(=O)NCC2(C)CCCC2)c1N.c1(C=O)ncsc1C(C)C.N N1(C(CC2CC(SC)C2)=O)CCC2CCC(C1)N2C(=O)CCS(C)=O N1(C(C2(F)C(C)C2)=O)CC2OCCN(C(=O)CCNC(C3CCCO3)=O)C2C1 O=C(C1=CNC2=NCCC2=C1)NC1CC2CC(NC(=O)C(Cl)=CCl)CC12 c1(NC(CC2N(C(c3ccnc(OC)n3)=O)CCC2)=O)ccc2sc(Cl)nc2c1 N1(C(CCOCCCOC)=O)CC2CCN(C(c3cc(N)ccc3O)=O)CC2C1 C1(NC(c2c(F)ccc(C)n2)=O)CN(C(C2COCCN2C)=O)C2(CCC2)C1 C1(C(N(CC(C)(C)CNC(=O)C2=CCCC2)CC)=O)CCc2[nH]nc(O)c2C1 O=C1CNc2nc(C(=O)NC3CCCN(C(c4ncccn4)=O)C3)ccc2N1 N1(C(c2nc(Cl)ccc2Cl)=O)CC2CCCN(C(C3CC3F)=O)C2C1 c1(NC(c2ncccc2NCc2cnccc2Cl)=O)cccc(Br)c1CO S(=O)(=O)(c1cccnc1N)N1C(CF)CC(OCC)C1.C1CC(F)(F)CO1.C CC1(C)OCc2c1n[nH]c2C(N1CCCC1CNC(C1CCCC1)=O)=O c1(C(C)=O)ccc2oc(O)nc2n1.CC(O)C(C(=O)O)NC(C1CC(F)(F)C1)=O N1(C(c2ncn(C)n2)=O)CCC2(CCC2NC(c2ncoc2C2CC2)=O)CC1 c1(N(CCCS(C)(=O)=O)C)ccc(S(=O)(=O)NCCS(=O)(=O)C2CC2)cc1Br c1(C(C(N2CCN(CC(C)NC(=O)C(C)(F)F)CC2)=O)(F)F)cccc(F)c1F c1(C(=O)N)coc2cc(O)ccc12.C1(NC(c2cnc(O)s2)=O)CCC(CC)C1 CCS(=O)(=O)CC(=O)N1CCOC(C(=O)Nc2cncc(C3CC3)c2)CC1 C(=O)(C(O)CC(F)(F)F)N(CC)CC1CCCN1C(c1sc(F)cc1C)=O N1(C(=O)O)CCC2CN(CC)CC12.c1(C=O)ccc(S(C)(=O)=O)s1.CC(C)C c1(C(=O)NCC(CNC(C2C(C)(C)CCC2)=O)CO)cc([N+](=O)[O-])ccc1O Cc1nc(S)sc1CC(=O)N(C1CC1)CC1CCCN1C(c1cc(F)c[nH]1)=O C1(C(=O)NCC2CC(OC)C2)C2CC3C(C2)C13.C1(C(=O)N)CCOCC1 N1(C(CCc2n(C)ccn2)=O)CC2(CCOCC2)CC1CNC(=O)C(Cl)=CCl N1(C(CC(C)(C)C)=O)CCC(C)(NC(=O)Cn2ccsc2=N)CC1 c1(C(N2C(COC)COCC2)C(=O)NCCC2(C)CC2)ccc(Cl)c(C)c1 C(C(=O)N1OC2CCC1C2)(C1CN(C(=O)C#CC2CCOC2)C1)C(=O)O N1(CCC(=O)NC2COCC2n2cc(CC3CCCCO3)nn2)CCOCC1=O Cc1ncccc1CC(=O)NC(C)CC1CN(C(c2cnc(CC(C)C)s2)=O)C1 c1(OC)ccc(C(N2CCN(C(c3ccoc3C(F)(F)F)=O)CC2)=O)cc1C C1(C(C)NC(c2ccc(C(C)C)o2)=O)CCCN(C(=O)C=Cc2ccncn2)C1 C(CCCCNC(=O)CC1CC(=O)C1)N(C)C(c1cc(C2CCCC2)no1)=O C1CC(F)(F)CN1C(=O)C.c1(C(=O)N)cnc(C2CC2)nc1.c1cn[nH]c1.C c1(N2C(CNC(CC3CCN(C)C3=O)=O)CCC2)ncnc2c1CCO2 CC1CN(C(=O)CCc2ccoc2)CC1CNC(c1cccnc1)=O.N(C)C.C CC1CCN(C(C23CC(CCO2)C3)=O)CC1NC(=O)CC1CCCO1 C(=O)(C(C)CC(F)(F)F)NC1C(OC)CN(C(c2ccncc2O)=O)C1 C(C(C)(C)C#CC(=O)NC)NC(c1cc(C)c(O)cc1)=O.C1(O)CCC(C)(C)C1 C(=O)(C(C)(O)CC(F)(F)F)N(CCCN(C(C(CCCC)O)=O)C)C c1(OCCCCCC)cccc(CNC(CO)C(C)(C)C)c1 C=CCC(CC=C)C(=O)N1CCCC(C(=O)NC2(C)CCCC2(F)F)C1 N#Cc1ccc2c(c1)CN(C(=O)NCCN(C1CC1)Cc1ccc(Br)cc1)C2 C1CC2CN(C(=O)CC(C)C)CC2C1.c1(OCC)cc(C(=O)N)on1.C(C)=O CC(C)(C(=O)NC1CC(NC(c2nc(Cl)cs2)=O)C1)C(F)(F)F C1(C)(C=O)CCC(C)=C(C)C1.c1(COC)nc(C(=O)NC(C)CCO)cs1 Cc1cc(C)c2sc(N3CC4(C3)OCCCC4O)nc2n1 CC1CN(C(C2CNC(=O)CN2C(C2C(C#N)C2(C)C)=O)=O)CC2(CCC2)O1 O(N1CCC(NC(C2CCN2C(C2CCN(C)C2)=O)=O)CC1)CC C12(NC(C(=Cc3ccccn3)C)=O)CCCC1N(C(=O)CO)CC2 CCC(C(=O)N1CC(CNC(=O)CCC#N)C2(CCC2)C1)C(C)(F)F c1ccccc1C.c1(C=O)cncs1.C1(NC(C2(SC)CC2)=O)CC(C)C1.N CC1COCC(C(N2CC(CC(F)C(=O)N(C)Cc3nc[nH]n3)C2)=O)O1 c1(C(=O)NC(CNC(CC2(C#N)CC2)=O)C2CC2)ncsc1C(F)(F)F CC(C)(CNC(C1COCCN1C(=O)CC1CCOC1=O)=O)CCO Cc1ccncc1CC(N1C(C(=O)NC(C)(C)CNC(N)=O)CC1C)=O c1(-c2cn(C)nc2)ccc(F)cc1CN1CC(=O)NC(C(=O)O)C1 N1(C(c2c(C)n[nH]c2)=O)CCOC2CN(C(=O)CNC(c3cccs3)=O)CC12 C12(NC(c3cc(OC)ns3)=O)CCC(C1)N(C(c1ccccn1)=O)C2.CCF.O Cc1c[nH]ccc1=NNC(=O)CN1CCC(C)C1 C1(NC(c2cn(CCNC(C3N(C)CCOC3)=O)nc2)=O)CC2(CCOC2)C1 C1(C(N(CC=C)C)=O)CN(C(=O)Cn2ncnn2)CC1CCC.C1CC1 c1(CC(=O)NCC(C)NC(Cn2c(C)nnn2)=O)cccnc1C(F)(F)F c1(OCC)cc(C(=O)NCCN(C)C(c2ccoc2CC)=O)ccc1OC N1(C(C(C(C)NC(C(CC(=C)C)OC)=O)(C)C)=O)CCCC(C)(C#N)C1 C1(CC)CN(C(=O)C(Cc2ccccc2)C2CC2)CCN1C(=O)C1=CSCS1 c1(CC(C)C)nc(Cc2ccccc2Br)nn1C1CCOC1 c1(C2(C=O)CC2)cc(F)ccc1F.C1(CC(=O)N)CCS(=O)(=O)N1.C1CCC1 C1(C(=O)NCC2(C=C)CCOCC2)CC2CCCC2N1C(=O)CCC(C)N(C)C c1(CN(C(C(=O)NC(c2cccc(C(F)F)c2)C)=O)C)ccc(F)cc1 C1CC2(C1)CCC2.C(=O)C(F)(F)C1CCOCC1.C1(C(=O)N)CN(C2CC2)C1 CC1CC=C(C(=O)NCC(C)C)CC1.n1(CC=O)cc(S(C)(=O)=O)cn1.C Cc1nc2ccnn2cc1C(N1CC(c2cccc(F)c2)(F)C1)=O C(=O)(C(F)C(C)CNC(=O)Cc1cccnc1)N(C(c1nccs1)C)C N1(C(c2c(COC)scc2)=O)CC2CCCC(NC(=O)CC3CCC3)C2C1.O CS(=O)(=O)c1cc(C(=O)NCC2(CN)CCOCC2)cc(C(F)(F)F)c1 C1(C(=O)NC2C(C(C)(C)C)C2)CC2(C1)C(C(=O)O)C21CCC1 CC1CC(C(=O)N(C2CN(C(=O)CSCc3cccnc3)C2)C)CCS1(=O)=O C1(NC(COCc2onc(C)n2)=O)CC2(C1)CN(C(=O)CCO)C2.C(N)=O CCCCN=C(NCC1CCCSC1)NC(C)COC(F)F C1(C(=O)NC2CN(C(CCCC(=O)N(C)C)=O)CC3C2C3)CNC(=O)C(C)(C)C1 N1(C(c2cc(C)sc2)=O)CCOC(Cn2cc(CNC(N)=O)nn2)C1 C1(NC(c2c(C)ncs2)=O)CCCC12CCN(C(c1cnc3[nH]nnc3c1)=O)C2 C1(CNC(c2cn(C)nc2)=O)(CNC(C2(F)CCOC2)=O)CCCCC1 C1(O)(C(C)NC(c2cc(Cl)n[nH]2)=O)CCN(C(=O)CCc2nccn2C)CC1 c1(CC=O)ccc(S(=O)C2CC2)cc1.N1(CC(=O)NCCCC)CCCC1=O.N c1(C(=O)NCCCN(C(=O)C)C(C)C)csc(C2OCCO2)c1.CC(F)F.O c1(C(N(C)CC2(O)CN(C(C3C(C)SCCC3)=O)C2)=O)ccc2[nH]c(=N)sc2c1 C(=O)(C1=NOC2COCC12)NCC(CCNC(CNS(CC)(=O)=O)=O)OC c1(C(=O)NC(C2CCCN2C(C2CCCSC2)=O)C)cccc(C(C)(F)F)n1 c1(OC)cc(C(=O)NC2CC(F)(C)C2)ncn1.C1(C=O)CCS(=O)(=O)N1 CCC(C)C(O)CC(=O)NCCCN(C(=O)CCc1ncco1)C CCCC(CCC)CC(=O)NCCC1(CNC(C2CCCC2CC)=O)CC1 C1(NC(C2OCCN(CC)C2)=O)C2CC3CN(C(C4CC=CC4)=O)C1C3C2 c1(NC(=O)C(F)F)ccc(N2CCN(Cc3cccnc3Cl)CC2)cc1 C(=O)(CCC1=NNC(=O)CC1)NCCCN(C(C(C(C)O)C)=O)CCO C(=O)(CCCC(=O)N1CC(NC(=O)CN2CC3CC3C2)C(F)C1)OC C(CCC(=O)N1CCC(C(N2CCC2C(C)O)=O)C1)OCC c1(OC)ccccc1C(=O)NCCN(C(=O)CN1CCNC(=O)C1)C Cc1cccc(C(=O)NC2CC3(C2)CC(NS(=O)(=O)C2CC2)C3)c1I CC1(C)C(NC(=O)Cn2cncn2)CCN1C(=O)Cc1cncc(C#N)c1 CCC(CC(=O)NCC1CCN(C(c2ccsc2)=O)CC1C)C(C)(C)C c1(N(c2c(C)cccc2)CC(N2CCCC(O)C2)=O)sc2c(c1C#N)CCC2 Cc1ncc(C(N2CCCC2C(=O)Nc2cn(C)nc2O)=O)c(=N)[nH]1 C(CS(=O)(=O)NCC=O)OCC.C(C1CCCC1)=CC(=O)N(C(CC)C)C Cc1nnc2n1CC(C(=O)NC1CCCC1CNc1nccc(CC#N)n1)C2 CC(C)(C#N)C(=O)NCC1CCC(C(=O)NC2CCN(C3CC3)CC2)C1 CC(CO)C(=O)N1CC(N(C)C(C2CC3(CC3)C2)=O)C1 C(=O)C(C=O)C(C)(C)C.C1(=CC(=O)NCCCC)CCCCC1.C(C)(C)C CC(CC(C)(C)CO)NC(=O)C(C)(C)CN(C)C(c1cc2occc2[nH]1)=O C=CCC(C)(C)CCN=c1cc(C)[nH]c(=NCC(C)(C)C2CCCO2)[nH]1 c1(C(N(C(C)CNC(c2cnc(Cl)cc2Cl)=O)C)=O)c(F)ccc2occc12 c1(OCC)ccc(Cl)c(C(c2nnnn2CC)NC(C)(C)CSC)c1 C(=O)(NNc1cccc(OC)c1Br)Nc1ccc(OC)nc1OC c1(SCC)ccc(CNC(c2ccc(-c3ccsc3)cc2)=O)cc1F O([Si](C)(C)C(C)(C)C)CC1CC(C)SC1.N12CC(C1)C2 N1(C(CCC(=O)NCC)=O)CCC(C)C(NC(C2CCc3cncn3C2)=O)C1C N1(C(c2c(C)snc2)=O)CC=C(C(=O)Nc2cnn(C)c2C(N)=O)CC1 C1(C(C)NC(c2c(OC)ccs2)=O)CN(C(C)=O)CCO1.C(=O)CC(F)(F)F N1(C(Cc2c(C)noc2C)=O)CCC2C1CCN2C(C1CN(C)C1)=O N1(C(COCCCC#C)=O)CCC2(CC1)CC(NC(=O)CC1CCCCC1F)C2 CC(C)CS(=O)(=O)CC(=O)NCC1(F)CCCN(C(C2(C)CCCOC2)=O)C1 C1(CCNC(C2CC(N(C)C)C2)=O)CCCCN1C(=O)COCC(F)(F)F Cc1c(C(=O)NCC(O)CC)cnn1C(C)(C)C.C(C1CCCC1)=CC=O.N c1(NC(CCCCNC(C)=O)=O)ccc(NC(c2cncc(C)c2)=O)c(C)c1 c1(OCC)ccc(C(N2CCN(Cc3ccc(CC)cc3)CC2)C(=O)NC)cc1 c1(C(N(C2(C(N(c3ccc(F)cc3)C)=O)CC2)C)=O)ccc([N+](=O)[O-])o1 Cc1ccc(F)cc1C(=O)NC1CC2CC1CN2C(=O)CO.c1ccc([N+](=O)[O-])s1 C=C=C(C)CC(=O)NCC(C1CCCC1)NC(C1CCN(C)C1)=O Cc1ccc(N(C(=O)C(=O)NCCCc2nncs2)C(C)C)cc1F C1(NC(Cc2c(C)nsc2)=O)CCN(C(=O)COC2CCOCC2)CC1C CCC(N=c1cc(C)[nH]c(=NCCC(C(F)(F)F)OC)[nH]1)c1ncccn1 c1(C(N(C(c2ccccc2)CO)C)=O)c[nH]c(=O)c2ccncc12 N1(C(c2nc(COCC)sc2)=O)CC2CCCC2(CNC(=O)C=NOC)C1 Cc1cc(=NCCn2ccc(=O)cc2)[nH]c(N(C)CCN2CCOC2=O)n1 c1(OCC)ccc(Br)cc1CN1CCCC(F)(CNC(c2ccon2)=O)C1 C(=O)(CCCNC(N)=O)N(CCC(=O)N(CCCC)C)CCOC Cc1n[nH]cc1C=CC(N1CCN(C(C2CCCCC2n2cccn2)=O)CC1)=O N1(C(c2cc(CCC)ncc2)=O)CC2(C1)CN(C(c1cc[n+]([O-])cc1)=O)CCO2 C(=O)(CC(C)(C)C(F)F)N1CC(C)N(C(C2CCC2C(C)(C)C)=O)CC1 c1(CC)nn(C2CC2)cc1C(N1CCC1)=O.C1(CCC=O)C(=O)ON=C1C.C N1(C(C(=O)NC(C(=O)OC)C)C(C)C)CCc2cc(Cl)cc(C)c2C1 C1(C(=O)NC)CCCCN1C(c1ccc(SC)s1)C(=O)NCc1ccco1 C#CCCC(O)C(=O)N(C1CN(C(=O)CC(n2nc(C)cc2C)C)C1)C N1(C(c2nn(C)c(F)c2)=O)CCC(C2CCN(C(=O)CC3CC4CC4C3)C2)CC1 c1(C(=O)NC(COCCCNC(C(C)=C(CC)C)=O)(C)C)cnn(C)c1Cl c1(C(=O)OCC)cncc(S(=O)(=O)NCCCOc2ccc(F)cc2Br)c1 c1(C(=O)NCC2(C)CN(C(C3(F)CC3)=O)CCO2)cc2ccsc2c(O)n1 Cc1cc(=NC2C3CCC(F)(F)C23)[nH]c(NC(c2ccccc2Br)C)n1 CC(CN=c1ccc([N+](=O)[O-])c(O)[nH]1)NC(C1CC(C)(C)C1C(F)(F)F)=O N1(C(C2CC(C)=C(C)CC2)=O)CCC2(CCCN2C(c2cc(Cl)c(C)cn2)=O)C1 N1(C(C=CCOC)=O)C2CCC1CC(NC(C1CCC(=O)NC1)=O)C2 c1(OC)cc(C(N2CCN(c3ccnc(C4CC4)n3)C(C#N)C2)=O)cc2n[nH]cc12 c1(N2C(C)CCC2)nc2cc(F)cc(F)c2o1.CC(C)C(C=O)NS(C)(=O)=O.N C(=O)CCC=CC.c1(CN(C(=O)CC=CC(C)(C)C)CC)ncc[nH]1.N N1(C(=O)CCCc2ccsc2)CCC2(CCN(C(=O)C(O)c3ccco3)C2)C1 N1(Cc2nc(CCCC)on2)CCCC2(C1)CN(C)C(=O)O2 C1(C(=O)NCCCOCCCO)CCN(C(C2C3CCCC23)=O)C12CC2 C(C(O)CC(C)(C)C)NC(CONC(c1c(OC)cncc1)=O)=O c1(CC(CNC(C2(O)CCSCC2)=O)O)ccccc1F C1(C(N2CC(NC(c3cc(CO)[nH]n3)=O)C2)=O)CC2CCC1NC2=O N1(C(c2[nH]cc(C)c2)=O)CCC2(CCCN(C(C3CC(=O)N(C4CC4)C3)=O)C2)C1 c1(NC(c2n(CCC)nnn2)c2cncn2C2CC2)ccc(N(C)C)cc1 C1(C(CNC(CC(C)C2CC2)=O)(C)C)CCCCN1C(=O)COC1CCOCC1 N1(C(CCC(=O)NCC)=O)CC2(CCCCN2C(=O)C(C)C2CC2)C1 CC(C)CC(C(=O)NC1(C)CCOC1)ONC(=O)C(C)(Cl)Cl C1(NC(C(C)C#N)=O)CN(C(=O)CSCC(F)F)CC1(C)C C12(C(N(C(C)CCNC(=O)C(C)O)C)=O)CCC(F)(CC1)C2.CC(F)(F)F N1(C(c2cc(C(C)C)n(C)n2)=O)CC2CCN(C(=O)CC(C)n3ccnc3)CC12 C1(CC)(CC)CCCN1C(=O)CC1CCCN(C(=O)C(F)C(C)C)C1 Cc1ncnc(O)c1CCC(N1CC2(CCN2C(C2(C)CCOCC2)=O)C1)=O Cc1ncc(CNC(c2cnc(C3CC3)o2)c2nnnn2C(C)C)n1C Cc1nn(CC(=O)NC(C)CCCCNC(=O)C(F)C2CC2)c(C)c1Cl c1(C(=O)NCC2(O)CSC2)coc2c1CN(C(C1CC3CCC1O3)=O)C2 N1(C(C(CCCC#C)C)=O)CCC2(CC1)CC(NC(=O)C(CC)NC(C)=O)C2 CCCC(CC)CC(=O)NC(C1(O)CN(C(c2cn(C)nc2C2CCC2)=O)C1)C C1(CNC(C(Br)=C(C)C)=O)C2CN(C(=O)CP(C)(C)=O)CC12 c1(C(=O)NC(c2c(C)n(C)nc2)C(=O)O)ncnc2c1nnn2Cc1cccs1 N1(C(C2CCC(CC)O2)=O)CCC2(CC1)CC(NC(c1cnc(SC)s1)=O)C2 CCC(C)C(O)CC(=O)NC1CC(OCC(=O)NCC(C)(C)C(N)=O)C1 N1(C(C2CCC(F)(F)C2)C(=O)NC2(C)CC2)CCc2cccc(Br)c2C1 CC(C)CC(F)C(=O)NCC(C1CCN(C(C2CN(C(=O)N(C)C)C2)=O)CC1)C CCC(O)C(C)C(=O)NC(C1CCCCC1)CNC(c1csnn1)=O C(=O)(CCCCCCS(N)(=O)=O)N(C)CCNC(c1ccc(F)cc1Cl)=O C1(CNC(C2(C(F)F)CCOC2)=O)CC(c2cccc3ncccc23)=NO1 C1(C(=O)NC2CC(CNC(CSCC=C)=O)OCC2)NC(=O)OC1(C)C c1(C(N2CCC(CN(C)C(c3nccnc3N)=O)C2)=O)ncncc1F Cc1nn(C)c(C)c1C(C)C(N1CCN(C(c2c[nH]nc2C(F)F)=O)C(C)C1)=O C1(C(=O)NCCc2cccc(F)c2)CN(C(c2ccc(F)cc2Br)=O)CCC1O C1(NC(CCN(C)CC)=O)CCN(C(c2sc(CO)nc2C)=O)CC(C)(C)C1 c1(CC)nocc1C(=O)NC(C)(CNC(=O)CC)C1CC1.c1nnnn1C c1(C(N(CC(COC)C)C)=O)occc1C.c1(C(=O)N)cn(C(C)C)nn1 C(CC(C)C(=O)NCCCN(CCCNC(c1cc(O)ncn1)=O)C)=CC c1(C(=O)NC2(C)CCN(CCCC(=O)O)C2)cc2ccccn2n1 N1(C(CC(C(F)F)NC(CC(C)F)=O)=O)CC2(CCC(=O)O2)C1 Cc1ccc(N2CCC(NC(c3nnnn3CCC3CC3)c3cn[nH]c3)C2)cc1 N1(c2ccc(-n3nc(C)c(Cl)c3C)cn2)CCc2c(cc(C(=O)O)n2C)C1 Cc1c(F)ccc(CN2CC(C)(CC(N3CCn4cncc4C3)=O)C2)c1Cl c1(C(=O)N)cn(C)c2c(Cl)cccc12.C1(C(=O)NCCC)CCN1C1CCCC1 C1(NC(C(CC)C(C)O)=O)CC(N=c2nc(C3CCCCC3)[nH]s2)C1 C1(NC(c2ccn(CC)c2C)=O)CN(C(=O)Cn2ccnc2C)CC1(C)C C#Cc1cccc(CC(=O)NCC2(F)CCC(NC(=O)C(C)COC)C2)c1 C(C)(C(CC(=O)NC1CCCC1CN=[N+]=[N-])NC(C1CCCCCN1C)=O)OC CC(C)CC(CNC(C1(O)CCSCC1)=O)C(=O)N(CC1=CCSC1)C N1(C(CC(C)n2cccc2)=O)CC(C)C(C)(C(=O)N(C)CCc2cnn(C)c2)C1 c1(CN2CC3CN(C(c4cc(C)[nH]n4)=O)CC3C2)c(Br)ccc2c1OCO2 C(=O)(CCC(C)(C)C)N1CCN(CCN(C(=O)CC(O)c2ccccc2)C)CC1 C1(NC(C2CCC3(CC3)C2)=O)C2CCC1CN(C(c1cc(F)ccc1F)=O)C2 S(=O)(=O)(c1ccco1)OC(C1N(C(=O)OC(C)(C)C)CCS1)=O CC1(C)CC(NC(=O)CSC(F)F)CCN(C(=O)CC2CSCCO2)C1 C(C(CNC(C1(O)CCC1)=O)S(C)(=O)=O)NC(C1CCC(OC)C1)=O c1(NC(c2c(C)cc(OC)c(Br)c2)=O)c(Cl)cccc1[N+](=O)[O-] N1(C(CC(=C)C)=O)C2CCC1CN(C(c1ccc(F)cc1OCC=C)=O)C2 CCC(C)C(C)(O)CNC(=O)CCCCCn1cc(C(C)(C)C2CC2)nn1 N1(C(C2(C)CCCNC2=O)=O)CCC2(CC1)CN(C(=O)CC1COC3CC1C3)C2 c1(-c2nccc(N3CCN(C(C4(C)COC4)=O)CC3)c2)cc(F)cc([N+](=O)[O-])c1 Cc1cnc2n1CCCC2C(=O)N1C2CCC1CN(C(C1(C(C)C)CC1)=O)CC2 Cc1cc(C(N2C3CN(C(=O)C(C)(CO)CO)CC23)=O)ccc1[N+](=O)[O-] c1(C(N2C3CN(C(c4scc(C(=O)OC)c4)=O)C(C3)C2)=O)cccc2nc[nH]c12 C(C(CC#N)NC1CC(NC(=O)OC(C)(C)C)C1)(OC)OC CC1CSCCN1C(=O)C(Cc1ccco1)NC(c1csnc1Cl)=O C1(CCC(=O)N(CC(CN(CC(=O)NC)C)O)C)CCN(C)C1.c1ccccc1 c1(SC)cccnc1C(=O)NCC1CN(C(c2sccc2C)=O)C2CC12 c1(COC(c2ccc(Cn3ccccc3=O)cc2)=O)c(Cl)cccc1Br C(=O)(CCC(C)(C)C#N)N1CC(CC(N2CCC(SC)C2)=O)OCC1 c1(C(N2C3C(CNC(=O)CCc4nc[nH]n4)C(C3)C2)=O)c(F)ccc(O)c1F N1(C(C(C)=CC)=O)CCCC1CC(=O)NC(c1ccccc1)C1CCC1 O=S(=O)(c1ccc(NCCN2CCC2)c(Br)c1)NCCN1CC2CC2C1 Cc1ccc(CC(=O)NC(C2CCCC2)CNC(=O)CCO)c(C)c1.C1CC1 C#CCCC(O)C(=O)N=S(C)(=O)c1cccc(OC)c1 C1(CNC(C2CCCS2(=O)=O)=O)CC2CC2N1C(=O)Cc1ccccc1Cl N1(C(C2CCN(C)C2)=O)CCN(C)C(C(=O)NCC2(C)CCCC(=O)N2)C1 C1(C)(CNC(C2(C3(C)CC3)CC2)=O)CN(C(c2cncs2)=O)C(C)(C)C1 c1(CC)cc(F)c(C(=O)NCCC(F)Cn2cc(C3(SC)CCC3)nn2)c(F)c1 C(CC(CNC(C1(c2ccccc2)CC1)=O)NC(=O)CSC(F)F)OC N1(C(c2scc(C(=O)Nc3ccc(C(C)=O)cn3)n2)=O)CC2C(C1)C2(F)F N1(C(c2cccc(I)c2)C(=O)NC(C(=O)OC)C)CCCSCC1C Cc1c(C(N2CC(O)CC2C(=O)NCC(C)CC2CC2)=O)cncc1F c1(C(CNC(COCCCCC)=O)NC(c2snnc2C)=O)ccccc1F C(CO)(CCCCNC(=O)Cc1nnc(O)s1)NC(c1nc(C)sc1C)=O c1(OC)ccc2c(c1)CCCC2CC(=O)Nc1ccc(N2CCCC2)cn1 C1(C=O)CCCCN1C1CCCC1.C1(F)(CNC(C2(C#N)CC2)=O)CCC1.C C(=O)(C(CC)CC(F)(F)F)NC1C2N(C(c3cc(OCC)ncc3)=O)C(CC2)C1 C1(C(N2CC3CC(NC(C(C)(C)n4cccn4)=O)C3C2)=O)CCCC1S(C)(=O)=O Cc1[nH]nc(C(F)(F)F)c1C(=O)NC(C)CC.N1(C(C=O)C)CCCCC1=O.N N12CC(CC1(C)C)NC2=O.Cc1nc(COCCCN=[N+]=[N-])sc1C CN=c1[nH]c(C(N2CCC(N(C(=O)CC3CCCN(C)C3)C)C2)=O)cs1 C1(C(=O)NCC2C3CN(C(C4SCCS4)=O)CC23)C2CC3C(C2=O)C13 Cc1cc(C)c(C(N2CCC(CNC(c3c(Cl)nn(C)c3Cl)=O)C(C)C2)=O)cn1 N1(C(C(C)(C)OCC)=O)CC2(C1)CN(C(c1sc(-n3cccc3)nc1C)=O)C2 CC(C)(C#N)CCC(=O)NCC1CCCC1C(=O)Nc1cccc(C(F)F)c1 c1(N2CCC(CC=C)(NC(=O)Cc3[nH]cnc3C)C2)nc(Cl)nc(C2CC2)c1F C1(C(=O)N(CCc2cccc(Cl)c2)Cc2cccc(F)c2)(CN)CC12CCC2 C=CC(CC)CC(=O)N1CC2CC2(CNC(C2(COC)CC=CC2)=O)C1 C(c1c(F)cccc1F)=CC(N1CCC(N(C(C=CC(CC)C)=O)CC)C1)=O c1(C(=O)NCC(C)(CO)OC)cccnc1C.c1(CCC(=O)N)cccnc1 Cc1cc(CC(=O)N(C(C)CNC(c2ccnn2C(F)F)=O)C)ccc1O C1(NC(=O)Cn2nc(Cl)ccc2=O)CCCCN(C(=O)CCc2nccs2)CC1 Cc1ccccc1C(C)NC(=O)CCCN(C(=O)C(C)CN(C)C)C c1(OC)ccc(OC)c(CN(C(C)C(C(=O)OC)C(=O)OC(C)C)C)c1 Cc1cc(C)c(C(=O)N(C2CCCC2)CCCNC(C2COCC(C)O2)=O)o1 CCC(CC)CC(=O)N1CC(CNC(c2cc(CO)oc2C)=O)CC(C)C1 c1(C(N(CC)CC2CCCN(C=O)C2)=O)ccc2nccn2c1C.C(C)(C)C.O CCCCCC(=O)O.C(C)(C)(CCCNC(C1COCCN1C(C)=O)=O)NCC C1(NC(CCOCC)=O)CC(F)(F)CC1NC(c1ncoc1C1CCC1)=O C1(CC(=O)NCC2(C#N)CCC2)(OC)CN(C(=O)CCOC2CC2)C1 Cc1ccc(F)c(C(=O)NCC2(O)CN(Cc3ccc(Br)cc3Br)C2)c1Cl C1(C(N(C(C#C)C2CCC2)C)=O)CN(C(C2(C(N)=O)CCC2)=O)CC1C1CC1 CCC(C(=O)N1CC2(CCC2NC(=O)Cc2ccsc2)C1)C(C)C c1(C(=O)NC2C3CC(CN)(C3)OC2)coc2cccc(Br)c12 N1(C(C(CCOC)C)=O)CC(F)(F)CC1C(=O)NCc1cnns1 CCCCC(C(=O)N1CC2CC1CCN2C(c1ncc([N+](=O)[O-])n1C)=O)C(C)C C1(C(=O)NC(C)CCCNC(=O)C2=CCCCO2)CCn2cnnc2C1 c1(C(=O)NCC2C3CN(C(CC(=C=C)C)=O)CC32)c(Cl)ccc(Br)c1F C(=O)(CC(C)(C)CNC(C1(C)CCOC1)=O)N1C(C)(COC)CC1 N1(C(c2nnn(C)c2C(F)F)=O)CCN(C(c2ccc(=O)oc2)=O)C(C2CC2)C1 c1(CNC2CN(C(c3ncc(C)c(Br)c3)=O)CC2C)cc(O)c(O)cc1O N1(C(c2c(CC)nco2)=O)CCN(C(c2cn(C)c(O)n2)=O)CC2CCCCC12 C1(NC(c2c(C)cc(C)o2)=O)CCCC(N=c2[nH]nc(-c3ccccc3)s2)C1 N1(C(c2n(C)nc(C3CC3)c2)C(=O)NC2CCCC2)C2CCC1CC(=O)NC2 C1(CNC(C2C(CC)C2)=O)CCCCN1C(C1CCCC1OC)=O C(c1ccc(F)c(OC)c1)=CC(N1CCN(C(c2c(CCC)nns2)=O)CC1)=O C1(NC(=O)CCc2cc[nH]n2)CC2CCC(C1)N2C(C1CC2(CCC2O)C1)=O Cc1cc(Cl)ccc1OC(C)C(N1CC2CC(NC(=O)COC(F)F)C2C1)=O Cc1c(C(N2CC(C)(C)CC2CNC(c2cccnn2)=O)=O)[nH]c2ccccc12 c1(C=O)ccn2c1CS(=O)(=O)CC2.C12(NC(=O)CCC3CCCO3)CC(C1)C2 C1(CC(=O)N(C2CCN(C(C3(C#N)CCCCC3)=O)CC2)C)C(=O)N(C)N=C1C C1(C(N2CCC(C(C)C(N3CCC(C)(CO)C3)=O)CC2)=O)C(C)(C)C1(F)F CCCC(CCCNC(C1CC1(C)C)=O)NC(C1COCCO1)=O c1(C(N(CC(CN(C(C=C(CCC)CCC)=O)C)O)C)=O)c(C)cc(O)nc1C c1(N2CC(C)C(NC(=O)C(C)C(C)(F)F)CC2)ncc([N+](=O)[O-])cc1CO c1(C(N2C(C(=O)NCCCOCCCC)CC2)=O)c(C)nn(CC)c1C c1(C(N2CCCCC2)=O)cc2c(F)cc(F)cc2[nH]1.C1(C(=O)N)CCS1(=O)=O.C c1(C(=O)NCC2CN(C(C=Cc3n(C)cnc3)=O)C2)c(Cl)nc2cc(Cl)ccn12 Cc1nnc2n1CC(C(=O)N(C)CCN(C)C(c1cnccn1)C)CC2 CC1CC(NCC(O)COCc2ccccc2Cl)CC(C)S1 Cc1c(C(=O)OCC(=O)Nc2nccs2)cc(C)c2ncccc12 c1(OC)cc(NC(C2CN(Cc3ccc(O)nc3)CCO2)=O)cnc1Cl C1(NC(CC(=O)N(C)C)=O)CC2CCC1N(C(C1(C(N)=O)CCC1)=O)C2 c1(N2CC3C(C)(C)C3C2)cc(Br)ccc1S(=O)(=O)N1CCCC(C(F)F)C1 CC(C)CC(C)CC(=O)N1CCN(C(c2ccc(O)nc2)=O)C(C2CC2)C1 N1(C(C(C(=O)OCC)F)=O)CCN(C(=O)Cc2ccc(Cl)s2)C(CF)C1 C(C(CN=c1[nH]c(=NCCOC2CC2)[nH]c2c(F)cccc12)c1ccccc1)SC C1(CNC(C(C)NC(C(C=C)CC)=O)=O)CC12CCOCC2 CN1CCN(C)CC(NC2(C3CCCCO3)CC2)C1 CCC(CC)(CCNC(=O)C(C)=C1CCC1)NC(=O)C(=CC1CCCCC1)F CC(C)CC(CNC(c1cnc(C(C)O)s1)=O)NC(C12CCC(CC1)C2)=O c1cccn(C)c1=O.N1(C(CN(C(C2CC2)=O)CC)=O)CCN(C(C)=O)CC1 CS(=O)CCC(O)C(=O)NCCCCNC(=O)Cc1ccc(O)cn1 c1(OC)cc(C(N2CCN(S(=O)(=O)c3cccs3)C(CO)C2)=O)cc(Cl)n1 C1(NC(c2csc(Cl)c2)=O)CCN(C(=O)COc2cccnc2)CC1CO Cc1ncnc(O)c1CCC(N1CC2CC1CN2C(=O)Cc1c(C)noc1Cl)=O C(C(C)(C)C=O)NC(C)=O.C1(CCC(=O)N(C2CCOC2)C)CCN(C2CC2)CC1 CC12CCOC(C(=O)NCC(C)(F)CNC(c3csc(O)n3)=O)(C1)C2 C1(NC(C(CC)N(C)C)=O)CN(C(c2cc(Cl)n[nH]2)=O)CC12CCCC2 CCC(C)(O)C(=O)NCCn1cc(C(N2CCC(c3cnn[nH]3)C2)=O)nn1 N1(C(C2CC23CCOC3)C=O)CCCN(CC(N)=O)CC1.C(C)N(C)C(C)=O.N C1(O)CC1(C)C.C1(C=O)CCN(C(=O)C)C1.N1CCCC1.CC(C)C.C=O.O Cc1cc[nH]c1C(=O)NCC1CC(NC(=O)C(C)Cc2ccnn2C)C1 C(CCC(=O)N1C(C(=O)N(C)CC2CC(F)(F)C2)CC1C)NC(C)=O N1(C(CCc2c(C)ncs2)=O)CC2CC1CCC2NC(c1ccccc1CO)=O CCCCCCCCN(C)C(C1NCC(C)CC1C)=O N1(C(CC=CC)=O)CCC2(CCCN2C(=O)C(C)C(C)CC)CC1 Cc1cc(C(=O)N(C)CC2C3CN(C(=O)C4=CCOC4)CC23)nn1C Cc1ccc(C)c(C(=O)NCC(C)CC2CN(C(=O)CC3CCCOC3)C2)n1 C1(C(=O)NC2C(NC(Cc3c(C)occ3)=O)CCC2)CCN(C)C(C)C1 C1(C(=O)NCC(CCCC)NC(C2CSCC(=O)N2)=O)Cc2ccccc2O1 C1(NC(CCC(C)OC)=O)CCN(C(C2(CCF)CCOCC2)=O)CC1F N1(C(C(C)OCC=C)=O)CCOC(CC(=O)Nc2ccc(CCF)cc2)C1 c1(CC(N2C(CNC(C(C)OC)=O)COC(C)(C)C2)=O)nccc2ccccc12 c1(CC)ncsc1NC(=O)CC(C1CC1)NC(=O)C(C)(C)OC(C)C CC1(C)CC(C(=O)NC)C(C)(C)O1.c1(C=O)cc(C2CC2)ccn1.C1CC1 c1(CNC(Cc2ccn(C)n2)=O)cnn(C)c1C(N1CCC1C(C)(C)O)=O C(=O)(C1=CCCC1C)N1C(CC=C)(C(=O)NCCC(O)CCC)CCC1 Cc1cc(=NCC2CC=CCC2)[nH]c(N2CCC(c3ccncc3)C2)n1 n1(C)cc(Cl)ccc1=O.C1(C(=O)OC)CC=CC(NC(=O)CCn2ccnn2)C1 C1(NC(=O)Cc2ccsc2)CCC12CN(C(=O)CN1CCSCC1)C2 Cc1cc(C(=O)NC2CCC(NC(=O)C=C3CCC(C)C3)C2)c(O)nc1C C1(CC(=O)NC2CCCN(CCNC(=O)NC(C)C)C2)CCn2cncc2C1 C1(C(=O)NC(C)CC2CCC2)(CC)CN(C(C2CCN2C)=O)C1 c1(CCCNC(C2CCCNC2=O)=O)cc(O)cc(Br)c1 Cc1nc(O)nc(C)c1C(=O)NC1CCCN(C(=O)COC2CCC2)CC1F N1(C(C(CN(C)C)O)=O)CCC(NC(=O)COC2CCCCCC2)C(CO)CC1 Cc1ncnc(C)c1CC(=O)NC1CC1NC(=O)CCCO.c1cccc(F)c1 CC1(O)COCCN(C(=O)CC2CCCN(C(=O)C3=C(Cl)CCC3)CC2)C1 Cc1ccnc(NC(c2cccc(CN(C3CCN(S(C)(=O)=O)C3)C)c2)=O)c1 CCCCCCNC(c1occc1C)c1nnnn1Cc1ccccc1 N1(C(CCc2ncc(C)[nH]2)=O)CCC(NC(c2nocc2Br)=O)C1C(C)C N1(C(c2c(C)ncs2)=O)CC2CC1C2CNC(c1ccoc1C)=O N1(C(C(C(C)C)(C)C)=O)CCn2c(CNC(=O)C)nnc2C1.C1(C=O)CC1C C(CCO)C(F)(F)F.S(=O)(=O)(CC(=O)NC(COC(C)C)C=O)NC.N C1(NC(=O)CNC(=O)C2CC2)CCC(C)C1.N1(CC=O)CCOC1=O.N Cc1nc(C2CCC2)sc1CC(=O)NC1CC(NC(=O)C(O)C(C)C)C1 N1(C(CCC(=C)C)=O)CCC2CN(C(=O)C(O)C3CC3)CC12 CC1COCCC1N=c1ccnc(NCc2cccc3c2NC(=O)CO3)[nH]1 N1(C(c2c(C)ccc(C#N)c2)=O)CCC(C(=O)NCCC(=O)N(C)C)=C(F)C1 N1(C(C(Br)=C(C)C)=O)CC(NC(=O)CCc2ccccc2Cl)CC1C Cc1cc(C(=O)NC(C)CC2CN(C(=O)Cc3cn[nH]c3)C2)n(C2CCC2)n1 C1(C2CCC(=O)NC2)(C(N(CCCNC(=O)CCCCC(C)C)CC)=O)CCC1 N1(C(C2(C)CCN(C)CC2)=O)CCCCCC(NC(c2cccc(F)c2F)=O)C1 c1(CC(C(=O)N(CCCO)CC#C)NC(C2CSC2)=O)ccc(Cl)cc1Cl C(C(C(=O)N1CC(n2cnnn2)C1)NC(=O)C(C)NC(C)=O)OC N1(C(C(C)(C)OC)=O)CC2(C(=O)NCCN(C)C)CC1CO2 O(P(C)(=O)CNC(=O)C(C)(C)CNC(c1cnncc1O)=O)CC C1(C(=O)NCC2C3CN(C(C(=O)NC4CC4)=O)CC32)CCCC2(CC2)C1 n1(CC)c(C(N2CCC(NC(=O)COCc3ncc(C)o3)C2)=O)cnc1O C1(NC(c2c(C)noc2C)=O)COC2(C1)CN(C(c1ccc(N)cc1Br)=O)C2 C1(CNCc2c(C3OCCO3)ncs2)CCC2(CCC2)O1 S(=O)(=O)(c1cnc(N(C2CCCCC2)C)cc1C)N1CCC(OCC)CC1 CCC(C)CCCCC(=O)N1CC(O)(CN(C)C(c2nccc(Cl)c2F)=O)C1 c1(C(=O)NCCNC(=O)Nc2c(-c3cn(C)nc3)cccc2)ncc(Br)cc1Br N1(C(COCCC#C)=O)CC(NC(=O)C=C(C)C)C(n2ccnn2)C1 N1(CC)CCCCC1C(=O)N(C)CC1(C)CCCC1NC(c1cccnc1N)=O c1(C(N2CC(CNC(C(C3CCCO3)OC)=O)C2)=O)cnc2nccn2c1 C1(C(c2n(CCC)nnn2)NC(C)Cc2ccco2)CCCCCCC1 N1(C(c2c(C)nc(CNC(=O)C(C)O)o2)=O)CC2(CCOC2)C1 C1(C2CCCN(C(=O)C(C)C(C)C)C2)(NC(CCCn2c(C)ncc2)=O)CC1 C(=O)(C(=O)CC(C)CC)NC(C(=O)NC1CCN(CCC)CC1)CC1CCCC1 N1(C(CCC(CC)NC(C2OCCC2(C)C)=O)=O)Cc2ccc(C#N)cc2C1 C#Cc1cnc(C(N2CCC2CNC(C2CCOCC2(C)C)=O)=O)c(C)c1 c1(N2CCC(C(C)O)C2)nccc(=NCCNC(c2ccccn2)=O)[nH]1 C1(CC)CN(C(C23CC=CC(C2)OC3)=O)CCN1C(C1CC(C#N)C1)=O Cc1nccnc1C(=O)NC1CC(CC(=O)NCC2(C3CC3)CC2)C1(C)C C12(NC(C3(CC)CCOCC3)=O)CCCC1CN(C(c1cnn(CC(F)F)c1)=O)C2 N1(C(c2ccc(CC)cn2)=O)CC2CCCC(C2)C1.C(=O)(C(C)CS(C)(=O)=O)N N1(C(C2C(C)CCO2)=O)CC(CO)C2(C1)CN(C(=O)C1CCc3snnc31)C2 c1(C(=O)NC2CCN(C(=O)CSCc3ccncc3)C2)cc2ccccn2c1 C12CN(C(c3ncoc3C3CC3)=O)CC1CS(=O)(=O)C2.CC(C)(C)CCC(=O)N N1(C(CC(=C)C)=O)CCC2(COC(CNC(=O)CC=CCC)C2)C1 c1(C(=O)NCC2CCCN(C(=O)CCC3CCC3)C2)ccc2ccsc2c1 C1(NC(c2c(COC)cc[nH]2)=O)CCCN(C(=O)CC(C)C(F)F)CC1 c1(N(C2CCCC2C(=O)C2CC2)C(C)=O)nc(C=O)cs1.C1CCC(C)C1 c1(CC)cc(C(=O)NC2CCN(C(=O)CCc3ccc(Cl)nc3)C2CC)ccn1 N1(C(c2c(C)coc2C)=O)CC2(CCN(C(=O)C(C)C3CC3)C2)C1 C1(C2CN(C(c3ccc(Cl)cn3)=O)C2)(NC(C=Cc2cn(C)nn2)=O)CC1 Fc1cccc2c(CCNCCn3ncnc3Br)c[nH]c12 C(=O)(CC1=NNC(=O)C1)NCC(CC(C)C)(C)NC(C1CCCCCCC1)=O C(=O)(CC(C)C(F)(F)F)N1C(CNC(C(C)Cc2ccccc2F)=O)CC1 c1(CCC(=O)NC(c2ccco2)Cc2ccccc2)cn(C2CCC2)nn1 c1(C(C(=O)N(C)CC2CCN(C(c3c(CC)nco3)=O)C2)O)ccc(Cl)cc1Cl CC1CN(C(=O)C(C)(C)C(F)F)CCC1CNC(=O)CC1CCC2(CCC2)O1 CC(C)(CO)C(C)(C)NC(=O)C(CNC(N)=O)CO C1(N(C(c2cc(CC)[nH]n2)=O)C)C2CN(C(=O)C=CC3C(C)C3(Cl)Cl)CC12 Cc1nnc2c(C(=O)NCC(C)(C)NC(c3ccc4c(c3)COC4)=O)cccn12 C(=O)(C(C)CC(F)(F)F)NC(CCOC)CNC(C1(C(F)F)CCCO1)=O c1(CC(=O)NCCC(C)N(C(C(CCOC)C)=O)C)ccc2nc[nH]c2c1 N1(C(C(c2cccnc2)NC(COCCCN(C)C)=O)=O)CCC(C(F)(F)F)C1 C(CC(C)C)(C(=O)NC)NC(C(c1ccco1)NC(C(CC)C)=O)=O C1(CNC(C(CC)n2nccc2C)=O)CCCCN1C(=O)C(C)(C)SC c1(C(=O)NCC2CCN(C(C(CC)(C)C(N)=O)=O)C2)ccc(F)c2ccccc12 C1(NC(CCC(CC)CC)=O)CN(C(c2nncs2)=O)CCC12CCC2 c1(C(N2CCC(c3scc(C)n3)C2)C(=O)NCC(F)F)ccc(S(C)(=O)=O)s1 N#CC1(CNC(=O)CCN(C(=O)C(O)C2CC2)C2CC2)CC1 c1(-c2n(CCOC)nc(CCCN(C)C)n2)cc2cccnc2cn1 C(CN=C(NCc1nc(-c2ccccc2)n[nH]1)NC1CCC1)c1c(C)n(C)nc1 c1(CC)ccc(C(=O)C(C)OC(C2(c3ccccc3)CCOC2)=O)cc1 CCC(C)(C)CCCC(=O)NC1CCN(CCNC(=O)C2CC2)CC1 Cc1nn(C)cc1C(C)C(=O)NC1CC2(C1)CC2.c1(C(=O)N)sc(F)cc1Cl N1(C(C(=Cc2ccco2)C)=O)CCN(C(C2CCC(C)(C)CO2)=O)C2COCC12 Cc1nc2ccnn2c(C)c1C(=O)NC1CC2CC1N(C(=O)Cc1nc[nH]n1)C2 Cc1noc2ncc(C(=O)NC3CCC(NC(C4CCNC(=O)C4)=O)CC3)cc12 N1(C(CCN(CC)CC)=O)CCC2(CC1)CC2C.C(=O)C(C)(C)C(O)CC.N C1CC2CCC1CC2.c12cn(nn1)C1CN(C(=O)C2)C1.C(=O)(OC)NC(C)C C1(CNC(C(C)OCC=C)=O)CCCN(C(=O)C2=CCCOC2)CC1 c1(COc2cccc(C3C(C)(C)C3(C)C)c2)nc2cc(F)ccc2[nH]1 C(C1=CCN(C(C2(O)CCOC2)=O)CC1)NC(C1CCCS1(=O)=O)=O c1(C=O)c(C)cc(C)nc1S.CCCC(C(=O)NC1CC(F)C1)NC(N)=O.C N1(C(C(CC)N(C)C)=O)CC(C(=O)Nc2cc(OC)cc(F)c2)CC12CCC2 Cc1ccc(-n2cc(CSCCNC(C3Cc4nccn4C3)=O)nn2)cc1C Cc1cc(=N)[nH]cc1C(N1CCN(C(=O)CC(C)c2ccncc2)CC1)=O N1(C(C(CCCNC(CCCSC)=O)(C)C)=O)Cc2nncn2C(C)C1 C1(O)(CN(C)C(=O)C2CC2)CCCN(C(=O)CC2COCC(C)(C)O2)C1 C=CCCCCC(=O)NC1(C(=O)NC2COC(C3CC3)C2)CCCC1C C(C(C(=O)NC(C)(CC)C1CC1)n1cc(Cn2cncn2)nn1)OCC CC1C(NC(c2c(Cl)cncc2Cl)=O)CCCN1C(=O)CCC=CBr c1(NC(C2(CNC(=O)C#CC3CC3)CCCO2)=O)ccc2cnccc2c1 Cc1cc(C(N2CCC3CN(C(=O)Cc4ccn(C)n4)C3C2)=O)c(C)nc1C N1(C(CC(CCC)(C)C)=O)CCC2(CC1)CN(C(C1CCC1OC)=O)C2 CCC(F)(F)CC(=O)NC1CCN(C(=O)Cc2nc(Br)sc2C)CC1C C1(NC(CNC(C(CC)C)=O)=O)CCN(C(=O)Cc2cc(C)no2)CC1F c1(C(N2CC(C)C(C(=O)NC(C)CC(F)(F)F)CC2)=O)c[nH]c2cccnc12 C1(N(C(=O)Cc2cnco2)C)CN(C(c2cc(-c3ccco3)no2)=O)CC1O N1(C(c2cc(Cl)cnc2F)=O)CCC(F)(F)C(NCc2csc3ccccc23)C1 C1(N(C(=O)CC2CS(=O)(=O)C2)C)CCCN(C(c2c[nH]nc2F)=O)C1 C1(C#N)(C(N(C2CCN(C(=O)C=C3CCC3)C2)C)=O)CC12CCOCC2 c1(N2CC(C)N(C3CC3)CC2)nc(=NCCc2cn[nH]c2)[nH]c2c1ncn2C CC1(CN2CCC2CNC)CCCC1.c1(C2CC2)cnn(C2CC2)c1 Cc1nc(Cl)ccc1CC(=O)NC1CC2C1CCN2C(=O)Cn1cccc1 C1(O)(CNC(C(F)=CC)=O)CCN(C(=O)CCCn2ccnn2)CC1 O=C(CC1=CCCCC1)NC(CO)CCCCNC(c1ccnc2cc[nH]c12)=O C(=O)(CCC(C)(C)F)NCC(CC(C)C)NC(=O)CCC1CCCC(=O)N1 N1(C(Cc2c(C)ccnc2)=O)CCCC12CCN(C(C1CC1C1(C)COC1)=O)C2 c1(CNC(C(=O)NCCNC(C)=O)=O)ccc(C)[nH]1 C1(NC(c2cc(C)c(C)o2)=O)CCN(C(=O)C=Cc2ccnn2C)CC1O c1(C(=O)NCCC(C(C)C)NC(=O)CC(C)C2CCCC2)cccc2c[nH]nc12 c1(CCC(=O)NCC2CN(C(CC)=O)CC2O)ccnc2ccccc12 Cc1ccc(C(N2CCC(NC(=O)C(C)Oc3ccccc3F)C2)=O)c(F)c1F N1(C(C=CC(C)(C)C)=O)CC(NC(c2cc(F)c(F)cc2O)=O)CC(C)(C)C1 C1(F)(C(N2CCC(C3(C)N=N3)C2)=O)CCN(C(=O)Cc2cccc(F)c2)CC1 C1(C(=O)Nc2c(CC)nn(C)c2)CCCN(C(=O)C(C)NC=O)C1C C(C(F)C(=O)N1CCCC1CN(C)C)C1CN(C(C(C)NC(CC)=O)=O)C1 Cc1cc(C(=O)NC23CC2CN(C(=O)CCCC2CCCC2)C3)ncc1CO CC1(C)CCC=C1C(=O)N1CCCCC(NC(c2nc(Cl)c(Cl)s2)=O)C1 CC(C)CC(F)(F)C(=O)NC(C)CCNC(=O)CSC1CC1 C1(NC(C2(C(C)(C)O)CCC2)=O)CCC(CNC(=O)Cc2cnoc2)C1 C(=O)(C1=CCCSC1)N1CCCC(N(C(c2ccc(C(C)O)cc2)=O)C)C1 c1(C(N2CCCC2)=O)cn2cc(C)nc2s1.n1(CC)nnc(C)c1C(=O)N(C)C c1(C(=O)NCC2(NC(c3ncc(OC)nc3)=O)COC2)ccc(Br)c(F)c1 C12(C(=O)NC(COC)C)CC(CO1)N(C(C1(F)CCCC=C1F)=O)C2 CN1CC(CC(=O)NC2CCN(C(=O)CC3NC(=O)NC3=O)CC2)C(O)C1 N1(C(C(CO)NC(=O)COCc2ccccc2)=O)CCC(C2CCC2)C1 Cc1c(C(N2C3CCC2C(CNC(=O)C(=O)N(C)C)C3)=O)ccc2n[nH]cc12 CC1(C)CCc2[nH]c(C(=O)NC3CCN(C(=O)CC4(CO)CC4)CC3O)cc2C1 C=CCN=C(NCC1CCOC1)N1CCC(F)(c2ccccc2)CC1 C1(CNC(Cc2cc(C(C)C)no2)=O)CCC(N(C(=O)CC2CC2)C)CC1 CC1CCC2C(CCCN2C(c2ccccc2CC2(C)CC2)C(=O)NC)C1.C=O C12(C(=O)NCc3c(C(=O)NC4CCN(CC)C4)n[nH]c3)CCC(CC1)CC2 C(=O)(CCC(C)OC)NCC(CCOC)NC(c1ccc(SC2CC2)cc1)=O C1(CC(=O)N(CC#C)C(C)C)C2CCC(C2)N1C(=O)Cc1ccns1 C1(CCC(C)(C)OC)CCCCN1C(=O)C(F)CC1CCOC1.C(=O)CCF C(C(O)CC(F)(F)F)N1C(C2(NC(c3cccc(COC)n3)=O)CC2)CCC1 c1(CC(N2C(C)CC(CNC(CN(CC)CC)=O)C2)=O)c(F)cncc1Cl C1(C#N)(C(N2CCN(C(C(C)Br)=O)CC2)=O)CCN(C(=O)OC(C)(C)C)C1 C(=O)(C(C1=CCC2CC1C2(C)C)N1CC=CC(O)C1)NCC c1(C(=O)NCC2(C3(O)CN(C(C(CC)C)=O)C3)CC2)cc(F)c(F)c(F)c1F c1(NC)nc(C)ccc1C(=O)NC1(CO)CCCN(C(C2CCCN2N=O)=O)C1 C(=O)(CCCCC(C)C)NCC(CC(N1CC2(CC2)CC1C)=O)OC N1(CC(=O)N(C(C)CC)C)C(=O)NC(C)(C)C1=O.C1(C=O)CCC(C)(C)CC1 C1(NC(=O)Cc2ccccc2)CCC2CN(C(C3CC34CCC4)=O)CC2C1 CC1(C)CCCC(C(=O)NC2CCC2)O1.c1(CCC(=O)N)ccc(C(F)F)cc1 C1(C(N2CCCC(Cn3cc(C(CC)N(C)C)nn3)C2)=O)CCCC(=O)N1C CCC(C)CCC(=O)N1CCC(OCCNC(c2c(C)oc(C)c2C)=O)C1 c1(C(NC(C)C)=O)cc(N)c(O)c(F)c1.N1(C2(CC=O)CC2)CCCC1 CC1CN(C(C2(CNC(=O)C(F)CC(C)(C)C)CCCC2)=O)CC(C)C1O c1(C(N2C(CNC(C(n3cc(Cl)cn3)C)=O)CCC2)=O)nn(C)nc1Br CCC(CC(C)C)C(C(=O)NCCCF)N1CCCC1Cc1nccn1C c1(C(=O)NC2C3CN(C(C4CN(CC)C(=O)C4)=O)CC32)ccc2cncn2c1C C(=O)(C=CS(C)=O)N(C)CC1N(C(CCn2ncc(C)c2)=O)CCC1 C12(C(=O)NC3C(CC)CCCC3)CCC(C)(CC1)OC2.C(=O)CC.CCCO.N c1(C(=O)OC)ccc(C(=O)NCCN(C)C(C2CCNC2=O)=O)c(Cl)c1 C1(C(N(C)Cc2n(CC)cnn2)=O)CN(C)CCN1C(=O)CCC(C)OC CC(CC(F)(F)F)C(=O)Oc1ccc2c(c1)OCO2 Cc1cc(C(F)(F)F)nn1CCc1nc(-c2nnc(C(C)C)s2)no1 CC(C)(CC1CC1)C(=O)N1CC(OCCC(=O)NCC2(O)CCCC2)C1 c1(C(N2CC(N(C(=O)CC3CCCOC3)C)C(O)C2)=O)coc2c(Cl)cccc12 N1(C(=O)CN2CCS(=O)(=O)CC2)CCCC2(CCCN(c3nccc(Br)n3)C2)C1 c1(C(=O)NC2(CO)CCN(C(C34CCC(CC3)O4)=O)C2)cc2c(F)cccc2[nH]1 CC(=Cn1ccnn1)C(=O)NC1CCN(C(C2CC(S(C)(=O)=O)C2)=O)CC1O C(c1cccc2ccccc12)=CC(=O)NC1(C)CC(NC(C2C(C)CCO2)=O)C1 N1(C(C(CC)CC)=O)CCOC2(CCCN(C(C3CC4CCCN(C3)C4)=O)C2)C1 C(C(=O)NCC(C1CCCO1)O)(C(C)(C)C)NC(CCNC(C)=O)=O Cc1c(F)ccc(N)c1C(=O)NC(C)CCNC(C1CCn2nccc2C1)=O c1(CCC)cc(N2CCC(C(=O)NCC3CCCO3)(OC)CC2)n2ncnc2n1 Cc1nc2ncnn2cc1C(=O)NC1CCN(C(=O)C2=COCC2)CC1O N1(C(C(CC)OC)=O)CC2CN(CC)CC2C1.c1(OCC(CN(C)C)O)ccccc1 N1(C(C(CC)F)=O)CCN(C(=O)C=C(C)C2CC2)C(C(C)C)C1 C1(NC(c2c(C)ccc(C)c2N)=O)CN(C(c2ccoc2)=O)CC2(CCC2)C1 N1(C(CC2C(CC)C2)=O)CCC(NC(=O)Cc2nccc(OC)n2)C1C CC(C)C(CCN(C(=O)Cc1ccoc1)C)NC(c1c[nH]nc1C1CC1)=O c1(C(=O)NC(CNC(C(COC)O)=O)C2CCC2)c(C)ncn1C c1(C(=O)NCC2C(NC(C(CC)O)=O)CC2)cc2ncn(C)c2cn1 O=C(C1=Cc2cc(Cl)ccc2OC1)NCC1COCCN1C(C1(F)CCOC1)=O CC1(C)OCCc2cc(C(=O)NCC3COCCN(C(=O)CC4CC4)C3)ccc21 C1(NCc2ccc(C(F)F)cc2)C2Cc3ccc(Br)cc3C12 C(=O)(CCCCCF)N1CCC(CCC(=O)NCC(C)CC2CC2)C1 CC1CCC(NC(C23CCCC2(C(N)=O)C3)=O)CN1C(=O)CC(C)(C)C c1(C(=O)NC2(C)CN(C(C3CCC3C(C)(C)C)=O)C2)cc(O)cc(O)n1 Cc1ccc(C(=O)N(CC(C)NC(=O)CCc2cc(Br)cs2)C)c(F)c1 CCCCCCN(C1CN(C(=O)CN(C)C(c2cc(OCC)no2)=O)C1)CC c1(C(=O)NCCC(C)NC(C2(C)CCCN2C)=O)cnc(O)c2ccccc12 c1(COC(C(N2CC(C(c3ccnnc3)C)C2)=O)C)ccccn1 C(=O)(C1=C(C#N)CCC1)NC(C(=O)NC1C(C)CCCCC1)C1(C)CC1 c1(C(C)N(C)CCN(C)C(C2(c3ccccc3)CC(F)(F)C2)=O)ccc(F)cc1 N1(C(C(CC)SC)=O)CC2(C)CN(C(=O)C(C3CC3)C3CC3)CC2(C)C1 N1(C(CC2C(C)=NN(C)C2=O)=O)CC2CCN(C(=O)Cc3cnccn3)C2C1 c1(C(=O)OC)c(C(=O)N)n[nH]c1C.C(=O)(CCCCN1CCCC1)N(CCC)C C(=O)(CC(C)(C)C(=O)NCC1CCCC1NC(c1ccns1)=O)OCC CC1(CNC(=O)C(C)(C)C#N)CCC(NC(=O)CO)CC1.C1CCCCO1 Cc1cc(C)c(C(N2CC(NC(C3CCC(C)(C)O3)=O)C3(CCC3)C2)=O)cc1N N1(C(C2(CC)CCCC2O)=O)CC=C(C(=O)NC2CCNC2=O)CC1 C1CC2(C1)CN(C(C1CCCCN1S(C)(=O)=O)=O)C2.Cc1ncc(C(=O)N)[nH]1 C1CC2(CCC2)C1.N1(C(C(C)(C)OCC)=O)CC(C(=O)N)C(C(C)C)C1 C1(C)(CNC(CN(CC)C)=O)CCCN1C(=O)C.C1(OCC)CCOC1 C(CCCCC(=O)NC1CCC(C2CC2)C1)N(C)C(C1CCC=CCCC1)=O c12ccccc1CN=C(NC1CCC1)NC2.C1(NCc2cnsc2)CCCCS1 c1(C=O)cc2c([nH]1)CCOC2.C1(C)(CN(C(C2(C=C)CCC2)=O)C)CCCC1.N N1(C(C2C(C=C)OCC2)=O)CC2(C=C(C(=O)N3CC(=O)N(C)C(=O)C3)CO2)C1 S(=O)(=O)(c1ccc2c(c1)CCCC2)N1CC(CC(=O)NCCC2CCCC2)C1 C1(NC(CC(=C)C)=O)CN(C(C2CC(=O)OC2(C)C)=O)Cc2nccn2C1 C(=O)(C1=NN2CCCN=C2N1)NCC(CC=C)NC(=O)C(C)(C)C1CCCCO1 CCCCN=C(NCc1c(C)cccc1C)NCC1CCC2(CC2)C1 C1(CC#C)(C(N2CC(O)(C(F)C(=O)OC)C2)=O)CCCCC1 CCC(CC)CCNC(=O)C.C1(C=O)CS(=O)(=O)CN1C(C)=O.CCF.O N1(C(c2c(CC)nc(C)s2)=O)CCC(C2CCN(C(=O)CC3CCOC3)C2)CC1 c1(C(N2CCC(F)(F)C(NS(=O)(=O)C(Cl)(Cl)Cl)C2)=O)c[nH]c2cc(Cl)ccc12 C1(CC(=O)NC2CCCC(NC(C(Br)=C(C)C)=O)C2)CCC2(CCC2)O1 C1(C(=O)NC2CCN(C)CC2(C)C)CCc2ncccc2C1 c1(CC(N2C(CNC(c3cc(C)n(C)n3)=O)CC3CC32)=O)cncc(C#N)c1 C(CCCCCNC(=O)C=CC1CCCCC1)NC(C1C(CCOC)C1)=O n1(CC=O)nc(C)c([N+](=O)[O-])c1C.Cc1ccoc1C(=O)NCC1CC1.N c1(-n2cc(CC(C(=O)OC)SC3CCCCC3)nn2)cc(C#N)ccc1F N1(C(C(CSCC)NC(c2cc(O)cs2)=O)=O)CC2(COCC(=O)N2)C1 CC(C)CCC(=O)NCCC(C)NC(=O)COCc1ncnn1C c1(-c2nc(C)c(C(N3CCC(CO)CC3C)=O)s2)c(F)cccc1Cl c1(OC)cc(NC(=O)C(CN(C)C)NC(=O)C(C)CN(C)C)ccc1C CC(CC(F)F)C(=O)NCC(C)(C)CC(=O)NCC1CC(C(N)=O)=NO1 CCCC(C(O)C(=O)Nc1cnn(CC(N)=O)c1)NC(=O)CC1OCCC1(C)C C12(CNC(C=C(C)C)=O)CCC(CN(C(=O)CCc3cc(C)[nH]n3)C1)C2 C1(CNC(c2ccc(C)o2)=O)CCC(CNC(c2c(C)[nH][nH]c2=N)=O)CC1 Cc1cc(F)ccc1C(N1C(C(N2CCN(C)C(=O)C2)=O)CC1C)=O c1(C(=O)NC2(CF)CN(C(=O)CC3CC(F)(F)C3)C2)ncc(Cl)cc1O c1(C(=O)NC(C2CCCCC2)C(=O)NC(CC)CCOC)cn(C)cc1C c1(CC(=O)NCCCC(C)(C)NC(=O)CC2CCCC(O)C2)cc(O)nnc1O C1(CC)CN(C(c2nc[nH]c2C(C)(C)C)=O)CCN1C(=O)C(N1CCOCC1)C C(=O)(C(C)(C)C1=CCN(C(c2ccco2)=O)C1)N(C(C(=O)NC)C)C C(=O)(C1COc2ccccc21)NCCC(C(C)C)NC(=O)CSc1nncn1C N1(C(C2(CC)COC2)=O)CC2CCC1C1CN(C(C3CCCN3C=O)=O)CC21 N1(C(C(C2CCC(C)CC2)CC)=O)CC2(NC(c3ccc(C#N)[nH]3)=O)CC1C2 C1(CC=O)CCCCN1C.C1(C)(C=O)CC(C(N2CC(O)(CC)C2)=O)C1.CO CCC(CC)CCC(=O)N1CC(CC(=O)N(CC(N2CCCC2)C)C)CC1C C1(NC(C2CCCN(C(c3c(CC)nccn3)=O)C2)=O)CC2CCC(C1)S2 N1(C(c2cc(C(C)(C)C)on2)=O)CC2CC3CC2C1C3NC(c1csc(Cl)n1)=O CC(C(=O)NCC1CN(C(=O)CN(C)C(c2ccsc2)=O)C1)=CC1CC1 C1(CCN(C(CCOC(C)=O)=O)C)CCN(C(=O)Cc2ccoc2C)CC1 N1(C(C=CS(C)=O)=O)CCN(C(=O)C2=CCCOC2)CC1c1cccc(F)c1 C1(C=O)CCCCC12CC2.c1(CCC)nc(C)c(C(=O)NC23CC(C2)C3)o1.N C1(CNC(C2CC2C(F)F)=O)CCN(Cc2cnc(Cl)s2)C1 C(C)(CC(=O)N(C1CC1)CC1CCOC1)N(C(CC=CC)=O)C c1(C(=O)NC2(CO)CN(C(C3C(COC)C3)=O)C2)cnc(SC)n1C c1(OC)ccccc1CC(=O)NCCC(C)(C)NC(C1CC(C)(O)C1)=O c1(C(=O)NCC2CCCN(C(C(C=C)(C)CC)=O)C2)noc2c(F)cccc12 N1(C(CCCCC(C)=O)=O)CC2CC(C)N(C(c3cn(C(C)C)nc3C)=O)C2C1 CN=c1[nH]c(=NCC2CC(O)CN2C)[nH]c(=NCCC=CBr)[nH]1 C(=O)(C1CCc2c[nH]nc21)N1CCCC(NC(c2c(C)cc(C)nc2C)=O)C1 c1(C(N(CC(CO)CO)C)=O)ccc(F)c(Cl)c1.C1(C(=O)N)C(C)(C)C1(F)F C1(C(=O)NC2(c3ncco3)CCC2)CCN(C(c2ccc(O)nc2)=O)CC1 c1(C(C)OCCSC)ccc(S(=O)(=O)N(CCC(C)C)C)cc1Cl c1(C(=O)NC2C(NC(C(C)n3cncn3)=O)CCC2)cccc2c1CC(=O)N2 c1(C(=O)NC2(C)CCCN(C(=O)C3=NNC(=O)C3)C2)cc2c(nn1)CCOC2 c1(CCC)nnc(S)n1CC(=O)NCCC1CCCCN1C(=O)C1=CCSC1 n1(CC(=O)NC2(C3N(C(C=CC(CC)C)=O)CCC3)CC2)ncc(O)nc1=O CC1CN(C(c2cccnc2)CNC(=O)CC2CCCC2)CC(C)O1 Cc1ccc(C(=O)NC(C2(O)CCN(c3ncc(F)cn3)CC2)C)c(F)c1 c1(C(N)=O)c[nH]c(C(N2CC(CCCCNC(C3CC3Cl)=O)C2)=O)c1 C1(COC)(NC(=O)CCCCCc2ccccc2)CCOC1(C)C c1(NC)c(C(=O)NCC2(C)CCN(C(C3CC3(C)Br)=O)C2)cccc1N C1(C(N(C(CNC(Cc2cccc(OC)c2)=O)C)C)=O)CCc2c(ncn2C)C1 n1(CCCC(=O)N(CCCCNC(c2n(C(C)C)ccn2)=O)C)ccccc1=O C(=O)(C(CCC1CC1)N1CCCCC1Cc1ccccc1F)NCCC C1(OC)(CNC(C2CCOC2C)=O)CCN(C(c2sc(C)nc2C)=O)C1 C1(C(N2C(C)(C(=O)OC)CC2)=O)CC12CCN(C(=O)CN(C)C(N)=O)C2 CC1CN(C)CC1C(=O)Nc1ccccc1.C1(C=O)CC(O)(c2ccccc2)C1.N CCC(CC(F)(F)F)C(=O)N(C(C)Cc1ccc(C)cc1)C C(=O)(CC(O)CC(C)(C)C)N1C(C(=O)NC2CC(C)OC2=O)CC(O)CC1 c1(CCC)ccccc1C(=O)NCCOCCN(C)C(C1CCCNC1)=O.C C1(C(N2CCN(C(C=CC)=O)C(CC(F)(F)F)C2)=O)CC(c2ccccc2)=NO1 N1(C(C(CC=C)(C)C)=O)CC2(CCC(NC(C3CC4CCCCN4C3)=O)CC2)C1 c1(CC(C(=O)NC2CC(NC(C(C)OCC(C)C)=O)C2)C)ccccc1F CN1CCCC1C1COCCN1C(=O)C(C)(C)C1CCCCN1 C1(C(N(C2CCN(C(=O)C(C)C)C2)CC)=O)CC2CC1CO2.CC(F)(F)F.O c1(OC)cccc(F)c1CC(N1CCCC(CO)(CNC(=O)C(C)(F)F)C1)=O Cc1sc(Cl)nc1C(N1CCC(N(C)C(C2CCOC2C2CC2)=O)C1)=O C(=O)(C(O)C(C)(C)C)NCCC(C)NC(=O)CC(c1ccccc1)N(C)C N1(C(c2cc[nH]n2)=O)CCC(C2CN(C(=O)C(F)F)C2)CC1 c1(OC)ccccc1C(C(N1CCC(O)(C(=O)N)C1)=O)OC.N1(CC)CCOCC1 CC(F)(F)CCCC(C(=O)NC(C)(C)C)N1CCC1(C)C1CC1 C1(F)(CNC(=O)CC(O)c2ccccc2)CCC(NC(=O)C(F)(F)C2CC2)C1 CC1CN(C(C2CCCN2CC(F)(F)F)=O)CCN1C(C1CC(N(C)C)C1)=O C1(CNC(c2occ(C)c2)=O)CN(C(c2scnc2C(F)F)=O)CCCO1 c1(N2CC3CCN(C)C3CC2)nc2ccsc2c(=NC2CS(=O)(=O)C2)[nH]1 C1(C(=O)NC(C)C(C)NC(C2(C)CC2)=O)(COC)COC1 Cc1nn(C)c(F)c1C(N1CC(NC(=O)CS)C(F)C1)=O.c1ccc(F)cc1 c1(C(N2CCCCC2)=O)cc(=O)n2nccc2[nH]1.C(=O)(C(C)(F)C(=O)N)OC.C CC1CN(C(c2cccc(Cl)n2)C(=O)NCC2CCCO2)CCC1C(=O)OC C1CCCCCN1C(=O)CC1(C(F)F)CC1.c1(CCC)ccc(C(=O)N)cc1.C CC1CN(C(=O)CCc2ccncn2)CCCN1C(=O)CC1CC(C2CC2)C1 c1(C(=O)NCCC(=C)CNC(C2(O)CCC2)=O)nnc(O)nc1O.C(C)C C1(C)(NC(Cc2n(C)ccc2)=O)CCN(C(C2CN(C(N)=O)C2)=O)C1 c1(C(=O)NCC2(CNC(CC(C=C)C)=O)CCOCC2)nnc(O)nc1O C=C1Cn2c(C(N3CCN(C(C4CCCC4)=O)CC3CCC)=O)nnc2S1 c1(C(N(C)CC2CCN(C(C(CC)(C)CC)=O)C2)=O)nnn2cc(C)nc(O)c12 CN1CCCC(F)(C(=O)NCC2CC(NC(=O)Cc3n[nH]c(=N)s3)C2)C1 c1(NC(C)CCCO)cc(N2CCN(CC(C)(C)F)CC2)nc(C(F)(F)F)n1 c1(CC)cc[nH]c1C(=O)NC(CSC)C(=O)NC(C)(C)CCF c1(OC)cc(C(=O)NC(C)CC(C)NC(=O)CN2CC(C)(O)C2)ccc1Cl C1(C)(N(CC(C2CCCC2)OC)C)CCCN1C(=O)OC(C)(C)C c1(OC)ccc(OCC(N2CCC(O)C2)=O)cc1C.C(=O)(C(F)=C1CCCC1)N c1(C(=O)NCCCN(C(c2ccc(N)cc2OC)=O)CC)nccc2[nH]ccc12 c1(C(N2CCCC2CCC(C)C)C(=O)NC(CC)(C)C)ccc(F)cc1I N1(C(C(C(=O)OCC)OC)=O)CCn2c(CNC(=O)C=CSC)nnc2C1 c1(-c2nc(CCCCCC)nn2C2CC2)ccc2ncc(=O)[nH]c2c1 c1(C(=O)NCC2(CNC(CCSC)=O)CC2)cc2ncccn2n1 CCC(C)(C)C(O)C(=O)NC(C)CN(C(=O)C(C)(O)COC)C N1(C(c2c(C)cc(C)o2)=O)CCC(C)(C)C1C(=O)NCCc1cnnn1C Cc1cnc(C)c(C(C)NC(Cc2cnn(C)c2)C(=O)O)n1 C(=O)(C(C)C(C)C)NCC(CC(=O)NC)C.n1(CC(=O)N)cnc(=N)[nH]1 Cc1cc(C(N2CC3CC2(C(=O)NC2CCOC2=O)C3)=O)nnc1O C(CNC(C1CCC(C(F)(F)F)O1)=O)(CC)(CC)NC(COCCC)=O C(CC(F)F)(C(=O)N1CCC1(C)CCO)N(C(C(C)OCC)=O)C c1(NC2CC(NC(c3cn[nH]c3)=O)C2)ncc(Br)c(C(F)(F)F)n1 C1(NC(CCNC(C)=O)=O)CCC(C)(C)CC1CNC(c1cccs1)=O c1(C(C)C)nccc(=NC(C)C2CCCN(C(=O)CCC3CCCC3)C2)[nH]1 C1(C(C)C)CCN(C(=O)C=CC)C1.C(=O)C(O)c1cnc[nH]1.C(C)(C)C c1(SC)nc(C(=O)OCC2CCCSC2)c2ccccn12 C1(NC2CC(CS(C)(=O)=O)C2)CC2(CCC2)C1O c1(C(=O)OC)cnc(NC(C2CCCC2N)=O)c(Br)c1.c1ccc(C)cc1C.C Cn1nc(C2CC2)cc1CC(N1CCOC(CNC(=O)CCc2ncc[nH]2)C1)=O Cc1cc(C(=O)NCCSCC(N(C)C[Si](C)(C)C)=O)ccn1 C1(NC(c2cnc(OC)nc2)=O)CCN(C(=O)C2=CC(C)(C)C2)CC1F c1(CNC(C(CC#C)C)=O)nc(CNC(=O)CCCC(N)=O)cc(O)n1 C1(C(=O)NC2CCN(C(C3CN(CCOC)C(=O)C3)=O)CC2)CCCCC1(F)F C(CCN=C(NCc1cccc(SCC)c1)NC1CCCCC1)N(CCC)C c1(C(=O)NC(CC)CNC(=O)CC=C(C)C)cnc(C(C)(F)F)s1 C1(O)(CCNC(=O)CCc2csc(Br)c2)CCN(C(C2CCOC2)=O)C1 C(c1scnc1C)=CC(=O)NC(CNC(C(c1cccc(Cl)c1)CC)=O)C C(CCC(C)(C)C(=O)NCC(C)(C)CC(F)F)NC(C(CO)N(C)C)=O C1(C(=O)NC(CO)C2CCC2)(CC)CCCN1C(=O)CCc1ccncc1 c1(C=O)cn(C)c2c(Cl)cccc12.C1(CNC(C=CCC)=O)CC(F)C1.C Cc1nnn(C)c1C(=O)NCC1CCC(NC(=O)Cc2sc(O)nc2O)CC1 CCC(O)C(F)(F)C(=O)N(C)CCN(C(=O)CC(F)(F)Br)C C1(C(N2CC(O)(C3CCCN3C(C34CC(CO3)C4)=O)C2)=O)CC12CCOC2 C1(COCC)CCCN(C(C2(CNC(c3cccn3C)=O)CC2)=O)C1 C1(C(=O)OC)C2CC1N(C(C1CCCN(C)C1)C(=O)NC1CCOCC1)C2 N1(C(C2(OCC)CCC2)=O)CCN(C(C2CC(=O)N(C)C2)=O)CC12CCC2 c1(CCC(N2CCN(C(C3CCC(C)CC3)=O)CC2)=O)cc(F)ccc1F c1(C(=O)NCCNC(c2cn(C(C)C)nc2)=O)nc2cc(O)ccc2[nH]1 c1(C(N2CC(NC(CSCCC)=O)CC23CCC3)=O)cc2ccccc2n1C C(=O)(C1Cc2ccccc21)N1C(CNC(C2(CC)CCOCC2)=O)C2CCC1C2 c1(C(=O)NCC(=O)NCC(=O)NCCc2onc(C)n2)[nH]cc(C)c1C N1(C(c2nc(OC)c(C)s2)=O)CCC2(CC1)CC2C.n1(CC(=O)N)nccc1C c1(NCC(CNC(=O)CC2CC(F)C2)O)ccc([N+](=O)[O-])cc1Br Cn1ccc(OCC(=O)NC(C)(CNC(c2cnsn2)=O)CO)n1 c1(OC)ccc(-c2ccc(CN(C)C)cc2)c2ccccc12 C(=O)(CCOC1COC1)NC1(C(C)(C)OC)CC1 N1(C(C2CC(C)C2)=O)CC2(NC(=O)COCc3ccnn3C)CCCC2(F)C1 N1(C(C2CCN(C)C2)=O)CCC(NC(=O)COC2CCCC2)C12CCC2 C#CC1(C(=O)N(CC)Cc2cccs2)CCN(C(C2CC(C)CO2)=O)CC1 Cc1ccc2c(n1)CCCN2Cc1nnc(-c2cccc(F)c2)o1 c1(OCCOC)ncccc1C(=O)N.C1C2CN(C(C)C(=O)N(C)C)CC12 C1(NC(=O)CCn2ccnc2)CC(F)(F)CC1.c1(CC=O)ccc(Cl)c(F)c1.N c1(C(=O)NCC)cnc2c(c1)CCCC2.C1(C(F)(F)F)(C(=O)N)CC=CCO1 N1(C(C2CCCN(C(c3cnc(Cl)cn3)=O)C2)=O)Cc2cccc(Cl)c2C1 C1(NC(C(C)=C2CC2)=O)CCCC12CN(C(=O)C(O)C1CCCC1)C2 c1(C=O)cc([N+](=O)[O-])c(C)s1.N1(C(C2(COC)CC=CC2)=O)CCC(C)C1 c1(C(=O)NC2(CF)CCN(C(COCCCCC)=O)C2)cc2occc2n1C CC1(C)CN(C(c2ccncc2N)=O)CCC1C(=O)NCCc1cnccn1 C1(CNC(C(C)S(C)(=O)=O)=O)CCC2(CCC2)CN1C(c1nccn1C)=O N1(C(c2ccc(Cn3cc(CSC)nn3)o2)=O)CCOC(C2CCCO2)C1 c1(C(=O)NC2C(C(=O)NCCCOC)C2)c(F)cc(Br)c(F)c1F Cc1ccc(C(=O)NC2(C(=O)NC3(C)CCOC3C)CCCCC2)cc1C#N CCCCC(O)CC(=O)NCCC1CCN(C(=O)CSCc2cccnc2)C1 Cn1nccc1CC(=O)NC(CNC(=O)Cc1coc(C(F)F)n1)CO c1(-c2nc(C(CCCCC)C)on2)ccc([N+](=O)[O-])cc1C C1(CC(=O)NCC2(NC(c3coc4c3CSC4)=O)CC2)Cc2ccccc2O1 C1(C(=O)NC(c2ccccc2)CNC(C2(C)CCC2)=O)CC2C=CC1CCC2 c1(CNCc2ncn(C)c2Cl)ccn2ncnc2c1 C(=O)(C(CCC)CCC)N1CC(F)CC(NC(c2c(CCC)n(CC)nc2)=O)C1 C(CCC(=O)NCCOCCCNC(c1ccn(CC#N)n1)=O)C1C(C)C1 c1(C(N2CC(n3cc(-c4nccc(C)n4)nn3)C2)=O)nc(=NC)cc[nH]1 C(=O)(C1=CC2(CCN(C(=O)CC3CCCNC3=O)C2)C1)NC(CC)C1CC1 c1(C(=O)NC(C(C)C)CCN(C(=O)C(F)=CC2CC2)C)cc2n(n1)CCC2 C1(N(C(COC(CC)(C)C)=O)C)CC2CCC(C1)N2C(=O)CCCCC(N)=O CC1CC(N=c2[nH]c(=NC3CC(CSC)C3)[nH]c3c2CCCCC3)CC(C)(C)O1 c1(C=O)nn(C)c(C)c1Cl.C1CCCC1.C(=O)(C=O)NCCNC(C)=O.N c1(CC)ccc(CC(=O)NCCOCCN(C)C(C2(Cl)CC2)=O)cc1 c1(CC)ccc(C(=O)NCC(CC)(CC)NC(C2CC2(F)F)=O)cc1N CC1(C(=O)N2CCCCC(CNC(C3CC=CC3)=O)C2)CCc2ccccc21 c1(C(=O)NC2CC(NC(Cn3ncc(C)c3)=O)C2)cccc(S(C)(=O)=O)c1 C1(C(=O)NC(C)CCNC(=O)C(C)(C)c2cnsc2)(OC)CCCCC1 C=Cc1ccc(NC(N2CC=CC2(C)COC)=O)nc1F n1(CC(C)C)ccc(C(=O)NCC(C)CO)n1.C1(C=O)(C(F)F)CC(=O)C1 C1(C)(CC(=O)NCCC(C)NC(C=C(C)CN2CCCC2)=O)CC1(F)F c1(C(=O)NC(CNC)C)cn(C2COCC2n2cccn2)nn1 c1(OC)cc(OC)c(C(=O)NC2(C)CCN(C(C3CC3(C)C)=O)CC2)cc1.O C(=O)(CC(C(=O)N1CCCCC(NC(=O)C)C1)NC(C)=O)OC.c1cccs1 C=CCC(C)(C)CC(=O)N1C(C(=O)NCC2OCCC2(C)C)CCC1C1CC1 N1(C(c2c(C)cn(C)n2)=O)CCC(C)(C)C1CNC(=O)CO.C1CCOC1 c1(CNC(C=CC)=O)nnc2n1CCN(C(C1(CCO)CCCC1)=O)C2.C C1(OC)CCCC(C(=O)N(CCC(=O)N(CCCN=[N+]=[N-])C)CCO)C1 C1(C(=O)NC2(CC=C)CN(C(=O)C(C)CC3CCC3)C2)CCc2ccnn2C1 c1(OC)ccc(C(N2CC(NC(=O)C(C)O)CC(F)C2)=O)c(Cl)c1OC c1(NC(C(C)C)CNC(=O)C(F)(F)c2cnccn2)c([N+](=O)[O-])cnn1C C1(CNC(CCCC)=O)CCCN(C(c2nccnc2C(N)=O)=O)CC1 c1(C(=O)OCC)cccc(CCC(=O)OC(C)Cc2cccnc2)c1 c1(C(N2CCC2)=O)cc(C(C)(C)C)nn1C.C1(C(=O)N)(COC)CCOC1 N1(C(C2N(C(c3cc(C(N)=O)[nH]c3)=O)CSC2)=O)CCOC(C2CCC2)C1 CC1(C)CN(C(=O)CC2CCC2)CCC1C(=O)NCC1CC1C1CCC1 C(CC(CC)C(=O)N(CCCNC(=O)Cc1nnc(C)s1)CC)=CC c1(C(=O)NCCC2CCCCN2C(C2CCCSC2)=O)ccc2nccnc2n1 C1(C(=O)NCCCN2CCN(C(c3c(Cl)cn(C)n3)=O)CC2)CCCCC1(C)C c1(C(=O)NC2(C(C)C)CCNC2=O)cc(Br)cc2c1OCCO2 c1(CC(C(N)=O)NC(=O)Cn2cc(-c3csnn3)nn2)ccccc1Cl C(CN=C(NCc1nnc(C(C)C)s1)N1CCCC2(C=C2)C1)OCC CC1CN(C(=O)Nc2nc3ccccc3c(=O)n2C2CC2)Cc2cccc(Br)c21 C12(C(N3CC(NC(c4c(Cl)nsc4Cl)=O)C3)=O)OCCCC1C2(F)F c1(NC2CN(C(C3(COC)CC=CCC3)=O)CC2C(=O)O)nc(Cl)ncc1F c1(OC)cc(F)c(CNCC2CCC(n3cc(CO)nn3)C2)cc1Br c1(C(N(C)CC)=O)cnc2cccnn12.c1(C(=O)N)ccc(C(F)(F)F)c(F)c1 O=C1NC(CCC2CCCCC2)C(=O)N1Cc1ccc(Br)nc1 CCC(N=c1cc(NCCC2CC2(Cl)Cl)nc(COC)[nH]1)c1ncc[nH]1 c1(C2N(C(c3ccc(-n4c(C)cc(C)n4)nc3)=O)CCC2)nnc2n1CCCC2 N(C(=NCC1Cc2ccccc2C1)NC1CCCc2nc(C)sc21)C(C=C)C c1(C(N2CCOCC(NC(CC(C)(C)C3CC3)=O)C2)=O)ccc2n[nH]cc2c1 c1(C(=O)NCCCC2N(C(C=CS(C)=O)=O)CCC2)cc(F)c(Cl)cc1Cl c1(C(=O)NCCC2CCC(NC(c3c(C)snn3)=O)C2)cc(F)c2cn[nH]c2c1 C1(O)(CNC2C(O)CCN(C(=O)OC(C)(C)C)C2)CCC(F)(F)CC1 c1(OC)cc(C(=O)NC(C(=O)N2CC(CC(N)=O)C2)C2CCCO2)[nH]n1 CC(C)(CCCN)C(=O)ON.C1(C(C)(F)F)C(=O)N1 C#Cc1ccc(C(N2CCC(N(C(=O)C=Cc3cc[nH]n3)CC)C2)=O)cc1C C1(N(C(=O)CN2CC3CC3C2)C)CCN(C(C23CCCC2C3Br)=O)CC1 N1(C(C(C)(C)N(C)C)=O)CCC2CN(C(C3CCCS(=O)(=O)C3)=O)C2C1 Cc1cccc(CC(N2CCCC2c2nccn2C)=O)c1Cl c1cc(F)cc(F)c1.c1(C(N(CC(C)CNC(=O)C)C)=O)ccc(F)cn1.O C1(NC(C2(C)C=CCN2C(=O)CC2CC3CC3C2)=O)C(=O)OC2CCCC12 c1(C=O)cc(C(N)=O)c[nH]1.c1(C(N(CC(C)C)C)=O)cnc(-c2ccncc2)s1 c1(C(=O)NC(c2ccccc2)C(=O)NCC(=O)NCC)scnc1Cl CC#CCC(C(=O)N1CCC(CC2CC2)C1)NC(C1CCCN1C=O)=O c1(OC(CCC)C(=O)NCCN(C)C(C2CCCC(=O)O2)=O)ccc(Cl)cc1C C1(OC)(CNC(c2ccncn2)=O)CCN(C(=O)Cc2cnsc2)CC1 C#CCCCCCCC(=O)NC1C2CCC1CN(C(=O)Cc1sc(C)nc1C)C2 C(=O)(CC1=NNC(=O)C1)N1CC(C)(CNC(CCNC(C)=O)=O)OCC1 c1(CN2CC3C(C(=O)NC(C)CN(C)C)(C3)C2)cc(O)cc(F)c1 c1(C(=O)NCC2N(C(c3nc(C)c(Br)cc3)=O)CCC2)cc(Cl)c(O)c(Cl)c1 N1(C(C(=Cc2cccs2)C)=O)CCC2(CCCN(C(c3occc3Cl)=O)C2)C1 C(=O)(CCCNC(C1CCN1C)=O)NC1(CCC)CC1 CCCC(CC)CC(=O)NC1CC2CN(c3nccc(CC#N)n3)CC2C1 Cc1cc(C(=O)NCC2CC2C(N2CCC(C(F)(F)F)C2)=O)cc(C)n1 Cc1cc(CNC(C2CCCCS2)=O)oc1C(=O)Nc1csnc1C1CC1 N1(C(CC)=O)CCN(C(C2CCCC2S(C)(=O)=O)=O)C2(CCC2)C1.C(=O)(OC)N C1(C(=O)NC(CNC(C2C(=C)C2)=O)C)CCC(C(C)C)CC1 c1(-c2nccn2CCNCC2N(C(c3ccco3)=O)CCOC2)ccc(Cl)cc1Cl C(CS(=O)(=O)CC(=O)N1CCN(c2ccccc2C)CC1)OC.C(=O)(C1CC1)N c1(OC)ccc(O)c(C(N2CCCC(NC(C3CCCCC3O)=O)C2)=O)c1 c1(C(N(CC(C)NC(=O)C(C)C2CCC2)C)=O)cc(CCCO)on1 CCC(C)(COC)C(=O)NC.c1ccc(Cl)c(F)c1.C1CC(O)CN1C(=O)C S(=O)(=O)(CC(=O)NCC(C)CO)NCC.c1(C=O)cnn(C2CC2)c1C.N c1(C(=O)NC(CNC(C(c2c(C)cccc2)C)=O)C2CCC2)cccc(O)c1C c1(C=O)ccc(=NCC2CC2)[nH]c1.C(c1ccc(F)cc1)=CC(=O)NCCC.N c1(N(C)C)cnc(C(=O)N(c2ccnc(OC(F)F)c2)N2CC(O)C(F)C2)cn1 C1(CC(N2CC(O)(CC)C2)=O)OCCOC1(C)C.c1(CC=O)ccc(F)cn1.N C1(c2cn(CC)nc2)CS(=O)CCN1C(=O)CCCCCNC(=O)OC c1cc(F)ccc1F.C1(CN(C(C2(SC)CC2)=O)C)COCCN1C(=O)CS N1(C(Cn2nc(C)n(CC)c2=O)=O)CC2CN(C(=O)CCCN(C)C)CC2(C)C1 c1(-c2cn(C(CNC(C3C(=C)C3)=O)C)nn2)cnc(F)cc1C C1(NC(C2N(C(=O)NC(C)C)CC(=O)C2)=O)CCc2c(nnn2C)C1 C1(NC(C(CCC)CCC)C)CCOC2(CCNCC2)C1 C12(CC=O)CCC(CC1)OC2.C1(C(C)NC(=O)COC2CCC2)CCC1 c1(CCCC(N2C(CNC(C=CCCC)=O)C=CC2)=O)nc2ccccc2s1 Cn1nnc2c(C(=O)NCC3CCC(NC(c4cc(Br)c[nH]4)=O)C3)ccnc12 N1(C(C2(NC(C)=O)CCC2)=O)CC2(NC(c3ccc(F)cc3O)=O)CCC1CC2 CC1=C(C(=O)N2CCC(CCNC(C3(C)CC(C(F)(F)F)C3)=O)C2)CCCO1 C1(N=[N+]=[N-])(C(N(CC=C)CCOC)=O)CCN(C(=O)C(CO)OC)C1 c1(OCC)ccc(C(N2CC(O)CC2CNC(=O)CO)=O)cc1C.CCF C1(N(C(C(CC)C2CCOCC2)=O)C)CC2CCC(C1)N2C(=O)C(C)(CC)OC C1(NC(C(C#N)C2CC2)=O)CCC12CN(C(c1ccc(OC(F)F)cc1)=O)C2 c1(COC(C(N2CCN(C)CC2)(C)C)=O)ccc2c(c1)OCCCCO2 C12(CNC(C(=O)N(C)C)=O)CCC(CN(C(c3cccn(C)c3=O)=O)C1)C2 C=CC(F)(F)C(=O)N1CCN(C(CNC(=O)CC(=C)C)C(F)(F)F)CC1 C1(C(N2CC(F)C2)=O)CC2(C)CC1CO2.N1(C(C)C)CC(C(=O)NC)CC1=O c1(C=O)csc([N+](=O)[O-])c1.c1(COC)nc(C(=O)NC2(CC)CC2)co1 c1(OC)cc(N)c(Cl)cc1C(=O)NCC1CCC1.C1(CC=O)CC=CCC1 O=C(CC1OCc2ccccc21)N1CCC(CNC(C23CCCCC2C3)=O)CC1 N1(C(c2occ(C)c2)=O)CCC(C)C(NC(=O)Cn2ccc(=O)cc2C)C1 Cc1cncc(CC(=O)NCc2ocnc2C(N2CC(O)CC2C(C)C)=O)c1 c1(CC(=O)N(C(C)C(=O)O)CCOC)cccc(Cl)c1I N1(C(C(C=C)(C)O)=O)CCN(C(=O)CSc2ccccc2OC)C(C2CCC2)C1 C1(C)(C(=O)N)C2CC3CC(C2)CC1C3.C1(C)(CC)CC1C(=O)N(CCC)C C1(CC)CN(C(c2cc3c[nH]nc3s2)=O)CCC1NC(=O)CN1CCN(C)CC1 C1(NC(Cc2c(C)nc[nH]2)=O)CC2CC1N(C(=O)C(C)Cc1ccccc1Cl)C2 Cc1cc(F)ccc1C1(C(=O)NCCC2CC=CCC2)CC1 c1(CCC(N2CC(OC)(C)C2)=O)ccccc1O.c1(C=O)cscc1C(F)F.N c1(OC)ccc(C=CC(=O)NC2CC(C)CN(C(=O)C)C2)nc1.C(N)=O.N CC(N=c1nc2sccc2c(N(C)Cc2nc[nH]n2)[nH]1)c1ncn(C)n1 N1(C(C(C(C)(C)F)(C)F)=O)CC2CCCC(CNC(=O)CCc3nccs3)C2C1 CC1CC=CCC1C(=O)NC(Cc1cn[nH]c1)C(=O)NC(c1ncc[nH]1)CO Cc1cc([N+](=O)[O-])c(C)cc1C(=O)NC1(c2cnn(C)c2)CC1 c1(C(=O)NC2(C#N)CCN(C(C(C)OC)=O)C2)cc2nc(C)ccc2o1 N1(C(C(CC(C)C)NC(c2[nH]cc(C(C)=O)c2)=O)=O)CC2CCC(C1)C(=O)N2 N1(C(C(COC)O)=O)CCC2(CC1)CCN(C(=O)C(c1ccccc1O)OC)C2 c1(-c2n(C)nnc2)ccc(C(=O)NC(C)(C)CC)cc1.C(=O)(C(F)C1CCC1)N C12(C(N(CCNC(c3ccnnc3O)=O)CC)=O)CCCN1CC(O)C2 C1(C(=O)NCC(C)(C)CO)CC12CC(NC(c1ccc(C3CC3)o1)=O)C2 C1(CC(=O)NCCN(CCC)C(C2CC(N(C)C)C2)=O)COC2CC1C2 c1(NC(c2cnc3ccccc3n2)c2n(CC)nnn2)ccc2c(c1)CCOC2 C1CN(C(c2cc(C(N)=O)co2)=O)CC(F)(F)C1.C(=O)(C(=O)N)NC(C)C N1(C(C(=O)Nc2c(OC)cccc2)CC2(C)CC2)Cc2ccccc2CCC1C c1(OC)nccc(N2CC(NC(c3ccc(C(F)F)cc3)=O)C(C)C2)n1 c1cc(Cl)cc(F)c1F.c1(CN(C2CCCCC2)C(C)=O)cn(C(C)C=O)nn1.N N1(C(c2c(CC)cccc2C)=O)CCN(C(=O)CC(C)(C)O)CC(C)(F)C1 Cc1[nH]c(C)c(C(=O)NCCOC2CCN(C(C3(O)CC3)=O)CC2)c1C C1(NC(C(CC2CCC2)NC(C(C=C)C)=O)=O)CCCN(O)C1=O N1(C(C#CC(C)C)=O)CCOC(C)C1C(=O)NOCC1CC2C=CC1C2 C(c1cc(Br)ccc1F)=CC(=O)NCC1(O)CCCOC1 c1(C(N2C(CN(C)C)C=CC2)=O)cc2c(Br)ccc(F)c2[nH]1 C1(C(C(=O)NCC(CN(C)C(c2ccc(C(C)(C)C)[nH]2)=O)O)F)CCCCC1 N1(C(c2cccc(Cl)c2)=O)CCC2CC2(C(=O)NCC(C2CC2)C2CC2)CC1 c1(CC)cn2c(n1)CC(C(=O)NCCCCNC(=O)C)CC2.C(C)(C)C.O CCC(F)(F)C(C)(C)C(=O)N.c1(CCC(=O)N(C(C)C2CC2)C)cn(C)nn1 C1(CNC(c2cc(C(C)C)on2)=O)CN(C(C2CCO2)=O)CCC1(C)C CCC(Cc1cccc(C)c1)C(=O)NCC1CCN1C(=O)CCOC1CC1 C=C=CC(C)C(=O)NCCC1CCN(C(=O)Cc2cccnc2)C1 c1(C=O)cnn2cccc(Cl)c12.C(=O)(C(O)CC(C)(C)C)N(C(C)C1CC1)C.N c1(C(=O)N)ccn(C)c(=O)c1.Cn1nc(C)cc1C=O.C1(C)CC(F)(F)C1 C1(F)(CNC(=O)C2=CCOC2)CCCN(C(C2CC2C(F)F)=O)C1 C1(C2CCN(C(=O)C(CO)C(C)(C)C)CC2)(NC(C2(F)CCCN(C)C2)=O)CC1 CCCCC(C(=O)N(CCC(=O)NCc1ccc(C)o1)CC)C(C)C N1(C(c2cc(Cl)c(Br)s2)=O)CCC2CN(C(c3cnc(Cl)cc3Cl)=O)CC2C1 c1(C(C)C)cc(C(=O)NC2CCC(NC(=O)C(C)Cc3ccccn3)C2)n[nH]1 N1(C(C2(C#N)CC=CC2)=O)CCC(NC(=O)CCN2CCCC2=O)C(O)C1 Cc1nnnn1CC(=O)NC(C1CCCCC1)CNC(=O)CCc1cnc(O)[nH]1 N1(C(C2(C(=O)O)C(=C)CC2)=O)CCCC2(CCC2)C1.C(=O)C(C)=C1CCC1 C1(N(C(=O)CCC2CCN(C(c3csc(CO)n3)=O)C2)C)COCC1(C)C Cc1[nH]c2ccccc2c1C(=O)NCC12CC(NC(c3ccon3)=O)(C1)C2 C1(Cn2cc(C3(C)CN(C(c4n[nH]cc4Br)=O)C3)nn2)CC2(CCC2)CO1 c1(C(=O)NC(CC#C)C(=O)NC2(C)CCC(C)CC2)cc(C)cc(C)n1 c1(C(=O)NC(C)CCCNC(c2cncc(Cl)c2Cl)=O)n[nH]c2c1C(=O)CCC2 C1(C=O)CCCCS1(=O)=O.N1(CC(=O)N(C(C)CC)C)CCC(C(N)=O)CC1.N c1(C(C)C)ccc(C(=O)NCC(O)CNC(C2CCCO2)=O)c(O)n1 N1(C(CSCCC)=O)CCC(C)(C)C(C(=O)NCC2C(C)(C)C2(F)F)C1 c1(C(C)NC(=O)NC(CC=C)C)ccc(NC(C)=O)cc1 c1(OCCC(=O)NC2C3CN(C(c4c(C)cc[nH]4)=O)C2C3)cccc(Cl)c1Cl c1(CC(=O)NCC(CN(c2nccc(SC)n2)C)C)cn2c(n1)CCCC2 N1(C(C2(O)C(C)(C)C2)=O)CC(C2(NC(=O)CO)CC2)C1.C1CC(F)(F)C1 c1(C(C(=O)NCC2(NC(=O)C3=CCC3)CCOCC2)O)ccc(F)c(Cl)c1 C1(C=O)CCCCC(=O)N1.C(c1ccc(C)s1)=CC(=O)N(CCOC)CC Cc1cc(O)ncc1C(N1CCCCC1CNC(=O)CCSCC(C)C)=O c1(C(N(CC=C)C(C)C)=O)n[nH]c2c1CN(C(=O)CC=C)C2 c1(C(N2CC(NC(=O)CC3CC3)C(F)C2)=O)ccc2occc2c1O N1(C(C(=Cc2cccs2)C)=O)CCCC(NC(=O)CS)CC1.c1csc(=N)[nH]1.C CC1CN(C(=O)CC2CCCC2NC(=O)CCOCC(F)F)CC1CO C(=O)(C(F)(F)C(C)(C)O)N1CC(C)(C)C(NC(=O)CC(F)(F)F)C1 C1(NC(CN(C)CCO)=O)COC2(C1)CN(C(=O)C(C1CCCCCC1)O)C2 CCC(C)C(C(=O)NC)NC(=O)CC(C(F)F)NC(=O)COCCF c1c(F)cc(F)cc1F.C(=O)(C(Cl)(Cl)Cl)NC=O.C123CC(C1)(C2)C3=O.N C12(NC(CCCN(C)C)=O)CC1CN(C(=O)CSCc1ncc[nH]1)C2 C(=O)(C#CC(C)(C)O)NC1CC(C(=O)NC(c2ccccc2)C#C)CC1O N1(C(c2ncn(C)c2)=O)CCN(C(c2n[nH]cc2[N+](=O)[O-])=O)CC1CC#N c1(C(N2CC(C)C(NC(=O)Cc3ccc(F)cc3F)C2)=O)n[nH]c2c1CCCC2 N#Cc1ccc(SCC(N2CCCN(C(c3cccc(O)n3)=O)CC2)=O)cc1 c1(N(CCN(C(CCOc2c(C)cccc2)=O)C)C)[nH]c(=O)n(C)c(=O)c1C#N O=C(CCN1C(=O)COc2ccccc21)NC1CCC1CNC(c1cnc[nH]1)=O c1(CCC(N2CCC(NC(C(C)C)=O)C2C(C)C)=O)ccc(C#N)cc1 c1(N2CCCC(C(=O)NCC3(CO)CCOC3)CC2)nc(Cl)nc2c1COCC2 CC1CCN(C(=O)C(=O)NCCN(C(c2occc2F)=O)C)C1.C1CCCCC1 N1(C(CC(C)C)=O)CCCC(O)(CN(C)C(c2ncncc2Cl)=O)C1 CC1(C)CN(C(C2CC=CCC2NC(c2coc(CO)c2)=O)=O)CCC1O c1(C(N2CC(CCNC(C(CC#C)O)=O)OCC2)=O)cc(Br)c(O)nc1C C(=O)(CC(C(=O)OC)NC(=O)Cc1ccc(OC)c(C)c1)OC C(=O)(CC(C(C)C)C(C)C)N1CCC(C)(CCNC(C(COC)(C)C)=O)C1 C(C1CCCN1C(=O)CCc1nccs1)=CC(=O)N(C)Cc1ncccn1 c1(C(=O)OCCOCC(=O)OCC)cccc(N2CC=CC2)c1 C(CC(C(=O)N1CCC(C)(O)C1)NC(=O)C(C)N1CC(C)C1)=CC c1(C(=O)NC2CCC(NC(CCOCC)=O)C2)cc(C)c(C)c2ncccc12 c1(CNCc2c(C)cccn2)ccc2c(c1O)C=CC(C)(C)O2 C(=O)(C(CCOCCO)NC(=O)CN1CCNC1=O)N(CCCC)CC c1(C(=O)NCC2CC(OC)CN2C(=O)CC(C)C)ccc2c(c1)CCCC2 C(C(C)C(=O)NCCC1(C(N2CCC2C(C)O)=O)CCC1)OC(C)=O C(=O)(CC(CCC)NC(=O)CC1CCOC1(C)C)NCCOCCCC C(CC)(C(=O)NCC1CCC(C(N2CC(c3ccccn3)C2)=O)O1)OCC c1(C(C(=O)NC(c2cccc(O)c2)C)N)ccccc1F c1(OCC(=O)NCC2N(C(C#CC)=O)CCOC2)ccc(C#N)cc1Cl c1(C(N2C(CNC(C(C)OC)=O)COC(C)(C)C2)=O)cnc2nc(O)ccc2c1 N1(C(CCOCC)=O)CCCC2(C)CCCC12.c1(CC=O)nnc(C2CC2)o1.N C=CCCC(F)(F)C(=O)NCC1(O)CN(C(c2ccc(N)c(SC)c2)=O)C1 N1(C(CC2(C)N(C(CNC(=O)OCC)=O)CC2)=O)CCCN(C2CC2)CC1 N1(C(=O)NC(c2ccnn2C)C)CC2(C=Cc3ccccc3O2)C1 O=C1Cc2ccc(NC(C3CCCN3C(C3CC4(CCC4)C3)=O)=O)cc2N1 c1(C(N2CCC(NC(C(C)(C)OC)=O)C(C)C2)=O)ccc2n[nH]cc2c1F N1(C(CCN(C(C)=O)C)=O)CCOC(C(C)NC(c2cccnn2)=O)C1 N1(C(c2nnc(C)s2)=O)C2CCC1C(CNC(c1cc(C(C)C)no1)=O)C2 C1(C(N2CCC(F)(F)C2)=O)Cc2n[nH]cc2C(=O)N1.CC(CC(N)=O)C(=O)NC N1(C(CC(COC)(C)C)=O)Cc2n[nH]cc2C1C(=O)Nn1nnc2c1CCCC2 c1(OC)cc(F)c(C(=O)NC(C)C(CO)NC(=O)C(C(C)C)SC)c(F)c1F C(C(C)C(C)C(=O)NCC=CCNC(=O)Cc1nc(C)sc1C)OC N1(c2nccc(OCC)n2)CC2CN(C(c3ccccc3OC)=O)CC2C1 N1(C(C(c2cn(C)nc2)O)=O)CC2(C1)CN(C(=O)Cc1cnn(C)c1)C2 C=Cc1cc(C(=O)N(CC(O)CNC(=O)CCS(C)(=O)=O)C)cc(F)c1 C#CCC(C)(C)C(=O)NCC1CCCCC1NC(=O)C(C)(CC)CC C=CC(C)CC(=O)NCC(C1CCC1)NC(=O)C(C)(C)n1cc(Cl)cn1 C1(CN(C)C(C2(Cl)CC2(F)F)=O)CCN(C(=O)CSC)C1.c1cscn1 c1(Cc2nnnn2CCC2(C)CC2)c(F)cc(F)cc1Br.C=CCOCC.N C1(NC(c2cc(C)ns2)=O)CC=C(C(=O)N2CCCC(C(C)C)CC2)C1 Cc1cc(C(N2CC(NC(C3CCC(C)(C)CC3)=O)CC2C)=O)cc(C)c1C c1(C(N2CC(C)C(NC(c3cncc(O)c3)=O)C2)=O)cnnc2ccccc12 Cc1c(OCC(=O)NC2CCC23CN(C(C2CCOC2(C)C)=O)C3)cccc1Cl C1(C(C)NC(c2cn(CCOC)nn2)=O)CCCN(C(c2nocc2C)=O)C1 N1(C(c2n[nH]c(C)c2C)=O)CCC2(CC1)CC(NC(C1CCCC1O)=O)CO2 C12(C(=O)NCC3C(C(N(C4CC(C)OCC4)C)=O)CCC3)CCC(CC1)C2.C c1(OC)ccc(Cl)c(NNC(=O)NCC(C2CCCO2)N(C)C)c1 C1(CNC(=O)CO)CCCCC1.C1CCCC(O)C1.n1(C)cc(CC2CC2)nn1 N1(C(C=Cc2ccc(CC)o2)=O)CCCC2CCC(C)CC12 C1(F)(CNC(c2cncc(C(N)=O)c2)=O)COCCN(C(=O)CC2CCOC2)C1 C1(NC(=O)NC(c2ccc(OC)nc2)CC(N)=O)CC(C)(C)OC1(C)C C(CNC(c1[nH]c(C)nc1C)=O)(CC(F)(F)F)NC(c1c(C#C)c[nH]n1)=O c1(NC(C)CC2CCCNC2)ncnc2sc3ccccc3c12 n1(CC(=O)NCC(C)NC(=O)C(C)(C)F)ccc2ccccc12 C1(NC(CCOC)=O)COC2(CCN(C(=O)CC3(C)CCC3)C2)C1 c1(OCC)ncc(C(N2CC(NC(C3CCNC3=O)=O)C(CO)C2)=O)cn1 C1(CC(N2CC(CC)C2)=O)CCN(C(=O)CSCCOC)C1(C)C C=CCCCC(=O)N1CCOC(CCCNC(c2cnn(CC(C)C)c2)=O)C1 N1(C(C2CC3CCCCC23)=O)CCC2(CC1)CCN(C(=O)C(F)(F)CO)C2 C1(C(N(C(CCNC(CC=CCC)=O)C)C)=O)COC(=O)N1C N1(C(C(=O)NCC)=O)CCCCC(F)C1.c1(CCC=CC(=O)N)ccccc1 c1(CC)cncc(C(C(=O)NC2CCOC2)N(C(C)C(C)CC)CC2CC2)c1 C1(CC=C)(C(N2CCC(CN(C(=O)C(C)(C)F)C)C2)=O)CC=CC1 N(C(=NCCc1ccc(F)cc1)NC1CC(S(C)(=O)=O)C1)C(C)CC(F)(F)F c1(C(=O)NC2C(C)CN(C(=O)CC(C)(F)F)CC2)cccc2nncn12 C1(CC)CN(c2ncc(C(=O)O)o2)CCC1NC(=O)OC(C)(C)C N1(C(C(C)SC)=O)CCC2CN(C(c3ccc(F)cc3OC(F)(F)F)=O)CCC12 CCC(C)C(C(=O)NC(C)(C)C)N1CC2C(CN=[N+]=[N-])C2C1 C(=O)(C1=CCCN(C(=O)CCc2ccn(C)c2)C1)N1CCC(C)C(C)C1 n1(C(C(N2CC(O)(CC)C2)=O)C)cnc2c(N)ncnc12.C=C1CCC1C(=O)N Cc1ncn(C)c(=O)c1C(=O)NC1COCCN(C(C2CC23CC3)=O)C1 C1(NC(C(CC)N(C)C)=O)C2CC3C1C3C2C(N1CCCC1CC(C)(C)C)=O C1(C(N2CCC(C(C)C)(C(=O)N(C)C)C2)=O)CC2(CC(=O)C2)C1.C1CCCS1 CN1CCC(C)(C(=O)NCC(N2CCN(C(C3CNC(=O)C3)=O)CC2)=O)C1=O Cn1cnc(C(N2CCC(C)(CCNC(=O)CC3CCSC3)C2)=O)cc1=O C1(CN=C(NCc2n(CC)ncn2)NCc2ccnn2C)CC(C)(C)OC1(C)C N1(C(c2c[nH]c(=N)o2)=O)CCCC12CCN(C(c1cncs1)=O)CC2 c1(COC(CC(Cc2c(OC)cccc2)C)=O)ccc2nccnc2n1 c1(N(C)C)ccc(C2CCN(C(=O)C(=O)Cc3cccc(Cl)c3)C2)cc1 c1(C(N(CC(C)NC(C2CCCNS2(=O)=O)=O)C)=O)cn2cnnc2cn1 c1(CCC(=O)NC2CC23CC(NC(c2cccs2)=O)C3)cnc2ccccc2c1 c1(CC)sc(C(=O)N(C)CC2CCCN(C(C3CC(=O)C3(C)C)=O)C2)cc1C C1(NC(C(C)OCC#C)=O)CCN(C(=O)C(c2cnccn2)C)C(C)C1 N1(C(c2c(NC)scn2)=O)CCCC(C(=O)Nc2csc(C)c2)CC1 C1(CC(=O)NC(C)CCCNC(c2cccc(=O)o2)=O)CC(=O)NC(=O)C1 c1(C(=O)NCC(C)NC(c2c[nH]nc2C(F)F)=O)cc(C(C)(C)C)ccn1 C1(CNC(C=CC)=O)(OC)CCCN(C(c2cc(C)on2)=O)C1 c1(C(N(C2CN(C(COCC=C)=O)CC2(C)C)C)=O)cc2cc(F)ccc2o1 C1(C)(CNC(c2n(C)c(Cl)cn2)=O)CCN(C(=O)C(CO)c2ccccc2)CC1 c1(CC)nncn1NC(=O)C(C)(C)NC(C1CC2CC2C1)=O c1(NC(c2nn(C)c(Br)c2Br)=O)nc2cccnc2[nH]1 O=C(C(CC1CCCO1)C(F)(F)F)NCC1(O)CCN(C(c2cnn[nH]2)=O)CC1 N1(C(C2C3(CN(Cc4n(C)ncc4Br)C3)CCC2)=O)CCc2cc(O)ccc2C1 c1(C(=O)NCC2(C)CCN(C(C(CC(C)C)F)=O)C2)c2c(nn1C)CCOC2 N1(Cc2ccc(C(=O)OC)cc2)CC(C(=O)NC(CO)C2CC2)CC(F)C1 Cc1cnc(C(=O)NCCCN(CCO)C(c2cc(C)nc(O)c2)=O)c(F)c1 c1(SC)ccccc1C(N1CCCCC1CCCNC(c1cnnc(O)c1)=O)=O C12CCC(CC1)CO2.c1(NCC)cccnc1C(=O)N.C(=O)C(C)=C1CC1 N1(C(c2ccc(CC)s2)=O)CCCCC(NC(c2cc(C(C)=O)on2)=O)C1 C1(NC(c2c(OC)noc2C)=O)CCCCN(C(c2c[nH]c(=O)cn2)=O)CC1 C1(C(C(=O)O)NC(=O)Cc2ccon2)CC2CCC1C2 c1(C(N2CCC(NC(CCCNC(N)=O)=O)C2)=O)cc(N)cc(F)c1 C1(CC)C(C(=O)N(CCCN(C(=O)Cc2ccnn2C)C)C)CCN1C S(=O)(=O)(c1cnc(-c2ccc(Br)cc2)s1)N(C1C(C)(C)CC1)CC1CCCO1 C(=O)(CCC=O)OCC(c1ccc(Br)cc1)=O.C=C1CC(C(F)(F)F)(C=O)C1 c1ccc(C2CC2)nc1.C(C(=O)NCC=CCC(=O)N)(C1CCC1)OCC Cc1ccnc(C(N2CC(N(C)C(C3CCC3C)=O)C2)=O)c1Br Cc1c(CC(=O)NCC2CCN2C(C2(C)CCCC2C)=O)oc2ccccc12 O=S(=O)(c1ccc(NCCc2ccncc2Cl)c(Br)c1)NCC1CCOCC1 N1(C(C2C(NC(=O)Nc3ccc(Cl)c(Cl)c3)C2)=O)CCc2c(O)cccc2C1 CCC(C(=O)N1CC(C(C)NC(c2c(OC)noc2C)=O)C1)C(C)O N1(C(C2(N(C(=O)C(c3ccnn3C)O)C)CC2)=O)CCCC(O)CC1 N1(C(C(C2(C)CC2)NC(Cc2ccn(C)n2)=O)=O)CC(=O)NC2(CC2)C1 Cn1cc2c(n1)CC(C(=O)NC1CC(F)(F)CC1O)NC2=O N1(C(CC2(OCC)CC2)=O)CC=C(C(=O)N(C2CCN(CC)C2)CC)CC1 C(=O)(C1CCCc2ncnn21)NC1C2(CN(C(C(C)(C)CF)=O)C2)CCC1 C1(CNC(CC(C=C)C)=O)CC(F)(F)CN1C(c1ccc(C(C)=O)o1)=O c1(C(N2CCC(NC(C(C)C3CCOC3)=O)CC2)=O)cccc2nc(O)ccc12 N1(C(C(C)C#N)=O)CC(NC(=O)CCc2cscc2Br)CCC(O)C1 CC1C(NC(c2csc(Cl)c2)=O)CCCN1C(c1ccc(O)c(Cl)n1)=O C1(CC=O)COC(C)(C)CO1.c1(CC)nnsc1C(=O)N.C(C)(C)C1CC1 c1(N(C2CCOCC2)C)cnc2c(F)c(F)ccc2c1Cl c1(C(=O)OC)cc(CNCCCCN)n2c1COCC2 C1(C(N)=O)CCCC(NCc2ccc(C(F)(F)F)nc2)C1 CC(C)(C(=O)N1CCC2(CC2)C1)C1=CCN(C(C2CCCS2)=O)C1 c1(C(=O)NC2(CC)CCN(C(=O)CCC(C)OC)CC2)ccc2ocnc2n1 S(=O)(=O)(CCC(=O)NC1(CO)CCCN(C(=O)CCCCCSC)C1)NC CN1CCCCC1CC(=O)NC12CC(NC(C3CC3C(F)F)=O)(C1)C2 N1(C(C2(CC(C)C)CC2)=O)CC2(C(=O)N)CCC1CC2.c1(CC)cccc(O)n1 C1(CC=C)(C(=O)NCC(F)(F)COC)CN(C(c2csnc2Cl)=O)C1 c1(CC)ccc(F)c(C(=O)NC2CC2CNC(C2CCC(C)CC2)=O)c1 C(=O)(C#CC(C)(C)C)NCC1CCCN(C(C(CC#C)SC)=O)C1 C(=O)(CCN=c1[nH]ccs1)NCC(CC)NC(c1csc(C(F)F)c1)=O N1(C(c2nn(C)c(=O)cc2)=O)CCN(C(=O)CN2CCCC2CO)CC12CCC2 C1(C(NOCC=C(C)C)=O)CC(C)CCN1C(c1ccc(C(N)=O)cc1)=O C1(CNC(C2(CC)CCC2)=O)CCN(C(C2(C(F)F)C=CCC2)=O)C1.C C1(C(C)NC(C(C)c2ccco2)=O)CN(C(c2nnn(C(C)(C)C)n2)=O)CCO1 c1(C(=O)NC2CC(CNC(C(F)OC)=O)C2)cc2c(cn1)CCCC2 CC(C)(O)C(F)C(=O)Nc1cnn(Cc2ccccc2NC(=O)C2CC2)c1 N1(C(CCN(C(C2CC2(Cl)Cl)=O)CC)=O)C2CCC1CC(F)C2 c1(OC)nc(OC)nc(N2CCN(C)CC2CNC(=O)CC(C)(C)O)n1 C(=O)(CC(C)C(=O)N1CC(F)CC1CC(=O)NC1CCC1)OC.C(N)(=O)N C#CCN(OC)C(=O)C1CC1CNC(=O)CC1CCCC12CC2 c1(OC)ccc(OCCCC(=O)NCC(CO)NC(=O)C=CCO)cc1 C1(CNC(c2[nH]cc(C)c2C)=O)CCC2CN(C(C3CCC3)=O)CC12 C1(NC(c2cc(OC)nn2C)=O)CCN(Cc2ccc(C)c(C)c2)CC1(C)C c1(OC)ncccc1S(=O)(=O)NCC1CN(Cc2cccc(C)c2)C1 c1(C(=O)Nc2nc(-c3ccccc3)ns2)ccc2cc(Br)ccc2c1 CCC(CC(C)C)C(=O)NCC1CC1NC(c1c(C)ncn(C)c1=O)=O NS(=O)(=O)CCN=c1cc[nH]cc1S(=O)(=O)NCCC(=O)Nc1ccccn1 N1(c2nc(N3CCC(N(C)C)CC3)cc(C)n2)CCC(C2CNC(=O)C2)C1 N1(c2c(CC)ccs2)CCC(NCc2cccnc2C(=O)NC2CC2)C1=O Cn1nc(CC(N2CC(CC)C2)=O)cc1C(F)(F)F.n1(CC=O)cnc(=N)[nH]1 C1CC2(CCC2)C1.n1(CCC=O)nc(C)cc1C.C1(OC)CC1C(=O)NC C(=O)(CC(CC)C(F)F)NCC1N(C(CCC(=C)Cl)=O)CC(O)C1 C(=O)(CCC(=O)N(CC(C)CNC(c1cc(Br)co1)=O)C)OCC C1(C(=O)NCCCC(CO)NC(C2CC3C(C2)C3(F)F)=O)CCc2nn[nH]c2C1 Cc1ccc2c(CN3CCC(CNC(C4COCCO4)=O)CC3)cc(=O)oc2c1 C12CCCC1(F)CN(C(=O)CC1CC(F)(F)C1)C2.C1(C(=O)N)CC2C=CC1O2 C1(COC)CN(C(c2ccn(CC(F)F)n2)=O)CCN1C(c1ccc(O)nc1)=O Nc1cnc(Cl)cc1C(=O)NCC1(O)CCN(C(=O)C(O)C2CCC2)CC1 CC(C)(CNC(C1(C#N)CCOC1)=O)CC(=O)N1CCCC(C(N)=O)C1 c1(C(N2CCN(C(C=C(C)C)=O)CC2C)=O)cc(S(N)(=O)=O)c(C)s1 c1(C(N2CC(C(=O)NC)OCC2)=O)csc2c1CCC(C)(C)C2 C1(NC(CC(=C)C)=O)C2CCC1CN(C(c1ccc(OCCF)cc1)=O)C2 c1(C=O)ccc(SC(F)(F)F)s1.C1(C(N(CCC)CC)=O)CC(F)(F)C1.N C1(NC(c2ccc(CC)nc2C)=O)CN(C(c2[nH]cnc2C#N)=O)CC12CCC2 N1(C(CCn2cc(CCN(CCOC)C)nn2)=O)CCC12CCC(C)CC2 c1(C2(C(c3nnnn3CCCF)NCCc3cc(C)no3)CC2)ccc(F)cc1 c1(NC(c2n(CCSC)nnn2)CCOCC(F)(F)F)ccc2c(c1)OCCC2 C1(NC(C2N(CCC)CCC2)=O)CC2(C1)CCC2.c1(C=O)cnc(C(F)F)s1 C1(NC(c2nnn(C)c2N)=O)CCC12CCN(C(=O)C=CC1CCCCC1)CC2 n1(CCCC(=O)NCC(CN(C(C2(OCC)CCC2)=O)C)O)ccccc1=O c1(C(N(CC(F)(F)F)CCCN)=O)cccc(OCC(F)F)n1 C12(C(N3CCCC(CNC(CCC#C)=O)C3)=O)CCC(CC1)OC2 c1(C(N2CCCC2)=O)c(F)cc(F)cc1F.c1(C(=O)NC)ccnn1CC(F)F C1(NCc2c(C(F)(F)F)cn(C)n2)CCC2(CCO2)CC1 Cc1c(C(=O)NCCCCCCNC(=O)CC23CCCC2C3)ccn1C C1(CN(C(CN(C(C)C)C)=O)C)CCCCN1C(=O)C(F)CC1CCCCC1 N1(C(C(c2ccc(C)s2)C)=O)CC(NC(C2(C)CCCC2)=O)C(C)C1 O=C1CCc2c(C(N3CCCCC(CNC(C4CC=CCC4)=O)C3)=O)cccc21 C1(CNC(c2scc(C)c2Cl)=O)CCN(C(=O)CC2(O)CCOC2)C1(C)C N#Cc1cc(CNC(C2(CCNC(=O)CCc3ccsc3)CCC2)=O)ccn1 C(CC1=CCN(C(C2CCCCN2C)=O)CC1)NC(C(C)NC(C1CCC1)=O)=O c1(C(=O)NCC#CCNC(C(c2cccc(OC)c2)C)=O)cccc2scnc12 C(c1ccc(Br)cc1)=CC(N1CCOCC1)=O.c1(C(=O)N)ccc(O)c(Br)c1.C N#CC1(C(=O)NCC2CCC(NC(C3CCOC3)=O)C2)CC2CCC1CC2 C1(N(C(=O)Cc2cn[nH]c2)C)CCN(C(C2CC(O)C2)=O)CC1 C12(CNC(c3c(C(C)C)occ3)=O)CCC1CN(C(=O)C(C)CO)C2 C1(CC=C)(C(N2CC3C(N(C)C(C4CC(CC(F)F)C4)=O)C3C2)=O)CCOCC1 CC(CCC(=O)NCCN1CCOC(C)C1)NC(=O)CC1(C)OCCO1 c1(C(=O)NCC2N(c3ccnc(C(C)(C)C)n3)CC3(CC3)C2)cnc2ccccn12 Cc1nn(C)c(Br)c1C(N1CCCC(C)(NC(=O)CC2CN(C)C2)C1)=O c1(C(N(CCCCNC(c2ccns2)=O)C)=O)c[nH]c(C(N)=O)c1 N1(C(C(C(=O)OCC)C)=O)CCC(NS(=O)(=O)CCC(=O)OC)C(F)C1 C(CC(=O)NCC(O)CF)(C(F)(F)F)NC(c1cccc(CC=C)c1)=O CC(C)CC(=O)NCC(C1CCC1)NC(c1cn(C2CC2)cn1)=O Cc1ccsc1CNC1CCC1CN=[N+]=[N-] C1(CC=C)(NC(=O)CC(C)F)CCN(C(c2cc(C)cs2)=O)C1 c1(CC(=O)NCC=O)cccc(F)c1.C12(C=O)CC(O)C1C2.CC(O)C.N C1(CN(CCNC(C(C)OCC2CC2)=O)C2CC2)CC2CCC1CC2 n1(CS(C)(=O)=O)cc(CC(C=O)C2CC2)nn1.C1CCCN1C(=O)CCCC c1(C(C)C)noc(C2=NOC3(CCN(c4ccccn4)CC3)C2)n1 C1(C(N2CC(CCO)(CC)C2)=O)CC(NC(=O)CC2CCOC2=O)CCO1 C=CCCCC(=O)N1CCC(C(=O)NCC(n2ccnn2)C)(CF)C1 N#Cc1ccc(NC(C2CC2CNC(=O)CC=C(Cl)Cl)=O)c(O)c1 Cc1scc(C(N2CCC(N(C(=O)CCOCCOCCCO)C)C2)=O)c1N C(=O)(CCC(F)(F)Cn1cc(CC(C)(C)C)nn1)NC1C(C)CCC1C CCC(CC)CC(=O)N1CCC(O)C(N(C(=O)C=CCCC(C)C)C)C1 c1(C(N(CCC(=O)NCc2nc(C)c(C)s2)CC#C)=O)cc(C#N)ccc1C C1(C(=O)N)CCc2nncn2C1.Cc1cc(C(N2CC(C(C)(C)O)(C)C2)=O)on1 CCCCC(F)(F)C(=O)N1CCC(O)(CCNC(C2CC3(CCC3)CO2)=O)C1 CC(CNC(=O)Cc1cnn(C)c1)C(F)C(=O)Nc1ccc(CCO)cc1 C(=O)(C1CCc2cc(Cl)ccc21)N1CC(N(C)C(c2csnn2)=O)C(C)(C)C1 N1(C(C(=Cc2ccco2)C)=O)CCC(F)(C(=O)NC2CNC(=O)OC2)C1 C1(CC)CC(C)CN1C(=O)C=CCNC(c1nccnc1OC)=O c1(CC(=O)N(CCC(=O)N(CC(C)CC)C)CC#C)c[nH]nc1C c1(C(N2CCC(C(C)NC(c3c(C)snn3)=O)C2)=O)cn(C)c(=O)nc1O C12(NC(=O)CC3(O)CCCCC3)CCC(CC1)N(C(=O)CC1C=CCC1)C2 c1(CNC(CN(C(CC=CCCCCC)=O)C2CC2)=O)cc(OC)ncn1 N1(C(=O)CCCC2CCCC2)CC2(C(N3C4COCC3C4)=O)CCC1CC2 C1(C(N(CC#C)CC2CCCO2)=O)CCN(C(=O)CC(O)CC)C1C N1(C(C2C3CN(C(C4C5C=CSC45)=O)CC23)=O)Cc2ccccc2C(O)C1 N1(C(C2C(c3c(C)n(C)nc3)OCC2)=O)CC(=O)N2CCCCC2C1 CC1(C)CC(NC(c2ccc(F)cc2N)=O)CN1C(C1CCCO1)=O C1(NC(C(C(CC)C)OC)=O)CC2CCC(C1)N2C(=O)CC1COC(C)(C)C1 c1(C(=O)NCC(CO)NC(CCN(C)CC)=O)ccc2nnn(C)c2c1 C1(N(C(Cc2cn(CC)nn2)=O)C)CCCCN(C(C2(n3cccn3)CC2)=O)C1 c1(C(=O)NCCOCCCNC(=O)CC2CCC3CC23)ccncc1F C(=O)(CCC(=O)NN(C)C)N1CC(C2C(C(=O)N)C2)C1.C1(COC)CC(C)C1 CC1(C)C(CNC(c2c(O)cccc2Cl)=O)CCN1C(=O)CCS(N)(=O)=O N1(C(C(C)O)=O)CC(n2cc(-c3ncccc3C(F)(F)F)nn2)C(O)C1 C1(CNC(C(F)=CC)=O)CC2(CC2)CN1C(c1c(C)nn(CC)c1C)=O c1(NC(C2C3(CC(NC(c4n(CC)nnc4)=O)C3)C2)=O)cc(Cl)cnc1O C(=O)(CCCCC(N)=O)N(CC(C)CNC(C1(C)CC1(F)F)=O)C C1(CNC(CN(C(=O)OC)C)=O)CCN(C(c2nc(C)n(C)c2C)=O)CC1C Cn1ncc(C(N2CCC(CC(=O)O)C2(C)C)=O)c1C#N C1(NC(CCC2C(C)C2)=O)CCCCC1NC(=O)C(c1cccc(Cl)c1)O Cc1nn2cc(C(=O)NC(C3CCN(Cc4cc(F)ccc4F)CC3)C)nc2s1 N1(C(c2c(CC)scn2)=O)CC2CC1CCN2C(c1cnc(Cl)cc1N)=O N1(C(C2C(C=C)OCC2)=O)CCC2(CC1)CC2C(N1CC(CC)(CC)C1)=O c1(OC)cc(C)c2[nH]c(C(=O)NCC(CS(C)(=O)=O)OC)cc2c1Br C(C(CC(C)C)C(=O)NC1(CCNC(c2sncc2C)=O)CCCC1)OC N(C(=NCc1ccc(N2CCCC2)nc1)NCC1CC1)C1CCC(C(=O)OC)C1 c1(C(=O)NC(CNC(CC(C=C)c2ccccc2)=O)C)ccc(Cl)c(F)c1O N1(C(c2cc(N)nc(Cl)c2)=O)CCCC1C1CCCN1C(=O)CCn1cccn1 C1(C(N2C(C(N3CCCC(OC)C3)=O)CC3CC32)=O)CNCC(F)(F)C1 c1(NC(c2cncc(-c3ccc(C)o3)n2)=O)cc(Cl)c(Br)cn1 c1ccc([N+](=O)[O-])cc1.C(=O)(C(C)(F)C(=O)NCCNC(=O)C)OC.O CCS(=O)(=O)C1(CNC(=O)NCc2noc(CC(F)(F)F)n2)CC1 Cc1c(Br)ccc(F)c1C(=O)Nc1c[nH]nc1C(=O)NCC=O.C(C)(C)C CCC(CC(=O)NCC1CC(C(=O)N(CC(C)C)CC(C)C)C1)SC c1(NC(C2C=CCN2C(c2csc(-c3ccccc3)n2)=O)=O)cc(Br)ccc1I c1cc(C(F)(F)F)cc([N+](=O)[O-])c1.N1(C=O)CC(F)(F)C(F)(F)C1.C1CCN1 N1(C(CSC)=O)CCN(C(C2CCC(OCc3ccc(CO)cc3)C2)=O)CC1 n1(C2CN(C(CC)=O)C2)ccnn1.C(=O)C=CC=O.C(C)(C)C.CCS C1(NC(C2CCC(C(N(C)C)=O)CC2)=O)(C)CCCN(C(=O)C2=C(Cl)CC2)C1 c1(C(=O)NC(c2ccc(C(C)C)cc2)CNC(=O)C(C)O)csc2nnsc12 C1(CNC(C(C2CCC(C)CC2)N)=O)Cc2ccc(C(=O)O)cc2O1 CCCCCCC(C(=O)NC)NC(=O)Nc1ccc2[nH]ccc2n1 S(=O)(=O)(c1ccccc1F)NC1CC(C(=O)OC)(CC)N(Cc2ccccc2)C1 C(=O)(CCCC(C)(C)C)N1CCC(C(=O)Nc2nccc(C(=O)OCC)n2)C1 c1(CC(=O)NC(CCCNC(Cc2cc(C)no2)=O)C)oc2ccccc2c1C N1(C(C(C)OCC2CC2)=O)CCCC(NC(=O)CCC(=O)N2CCC(O)CC2)C1 S(=O)(=O)(c1ccccc1Br)NC1C(C(=O)Nc2cccc(Cl)c2CO)C1 N1(C(c2c(C)occ2)=O)CC2(CC2)CC1CC(=O)NC1CCC(C2CC2)C1 c1(C(=O)NC2CCN(C(CCSC)=O)CCC2CO)c(Cl)ccc2ccncc12 N1(C(CCCC2(NC(CC(C)SC)=O)CCC2)=O)Cc2ccc([N+](=O)[O-])cc2C1 c1(C(=O)N)ccc(F)c(F)c1N.c1(NC)cnccc1C(=O)NCCC(C)(C)C c1(C(N(CCN(C)C(c2cc(-c3ccoc3)on2)=O)C)=O)c[nH]c(=N)s1 c1(C(N(C2CCN(CC(C)O)CC2)CC2CC2)=O)cccc2ncn(C)c12 Cc1cc(C)c(C(=O)NCC2(C)CCN(C(c3cc(N)ccc3F)=O)C2)cn1 c1(OC)ccc(CC(=O)NC2CCN(C(c3sccc3SC)=O)C2C)c(Cl)c1 C1(C(N2CC(NC(C(C)=C(CC)C)=O)C(CO)CC2)=O)CN2CCN1C(C)C2 Cc1[nH]cc(C(N2CCC(F)C(NC(=O)COC)C2)=O)c(=O)c1Cl.C1CCC1 C1(NC(N2Cc3ccc(CO)cc3C2)=O)CCCC12CCCCO2 c1nc(C(N2CC(O)C2)=O)c(N)s1.c1(C(NC)=O)cc(C2CC2)n(C)n1.C C1(NC(C=CC(C)C)=O)CN(C(c2ccnc(O)c2Br)=O)CC12CCC2 C1(NC(Cc2cn(CC)nc2)=O)CCCC(NC(=O)C(C)(C)c2sccc2Cl)C1 C(=O)(C1CCCc2cncn21)N1CCC(C(F)(F)F)C1.C(=O)(CC(=O)NC)OC Cc1cc(C(=O)NC2(C(=O)NC(c3nncn3C)C)CC2)n[nH]1 CCCCCC(C(=O)NC(C1CCN(C(c2cc(Br)n[nH]2)=O)CC1)C)C(C)C C12(CNC(C3CCCN(C)C3)=O)CN(C(c3cccc(F)c3N)=O)CC1CCO2 c1(C(=O)NCC(C2CC2)NC(c2cncc(SC)c2)=O)ccc2nccnc2n1 Cn1c(C(=O)NCCC2(O)CCN(C(=O)Cn3cnnc3O)C2)ccc1[N+](=O)[O-] CC(C)(O)C(C(=O)NCCc1ncccc1F)NC(=O)CC1CC2CCC1O2 c1(CC)cccc(F)c1C(=O)NC(CO)C(C)NC(=O)Cn1nnc(C)n1 Cc1nc2cc(-c3ccc(NC(c4cccc(O)n4)=O)s3)ccc2o1 N1(C(C2CN(OC)C(=O)C2)=O)CC2CN(C(c3csc(C)n3)=O)CCC12 C(=O)(C1CCCc2c[nH]nc21)NC1CCCC(NC(CCNS(CC)(=O)=O)=O)C1 C1(C(=O)NC2CCN(C(c3cncc(F)c3)=O)CC2)CC2CCCCN2C1 c1(C(=O)NCC2(C(=O)NC(C(=O)N(C)C)CO)CC2)cccc(F)c1O c1(CC(=O)NCC(CCC)NC(=O)C(C)OC2CCOC2)cccc(C)c1F N1(C(c2cc(CSC)c(C)s2)=O)CCC(NC(=O)Cc2cccs2)C(F)C1 N1(C(C=CC=CCC)=O)CC(C(=O)N(C2(CC)CC2)C)C(F)C1 N1(C(C2(C)CC(=C)C2)=O)CCC(F)(C=O)C1.c1(CC(=O)N)csc(C)n1 c1(C(N(C2CCC(NC(CCCC(=O)OC)=O)C2)C)=O)cn2cc[nH]c(=O)c2n1 CC(C)(C#N)CCC(=O)N1C2CCC1CN(C(C1CCCN1C1CCCC1)=O)C2 N1(C(C2C(=C)C2)=O)CCC2(CCC(C)O2)CC1.c1(C(=O)N)c(C)ccc(C)c1C C1(CC(=O)OC)NC(=O)CCN(CC(c2ccc(Cl)cn2)(C)C)C1=O N1(C(C2(CC)CC(C)(C)C2)=O)CCC(C=O)CC1(C)C.C1CC2CC(O)C1C2.N c1(C(N(CCN(C(=O)CN2CCOCC2)CC)CC)=O)cccc(C)c1N C(C(O)C(=O)NC(C)CC(C)NC(c1cnc(C)s1)=O)SC c1(-n2ccc(CNC(c3ncnn3C)C)n2)ccc(Br)cc1 c1(CC(C)C)ccc(C(=O)N(C2CN(C(C3CCOC3(C)C)=O)CC2O)C)cn1 C#CC(C)(C)C(=O)NC1CC(C)N(C(c2ccc(C3CC3)cn2)=O)C1 C1(C)(C(=O)NC2CC(C(C(=O)NC)F)C2)CCN(C)CC1 CC1CN(C(=O)C(=O)N(C)C)CCC1NC(c1cccc(N2CCC2)c1)=O C1CCCC2(CN(C(C3(O)CCC3)=O)C2)O1.c1(OC)ccc(C(=O)NC)cc1C c1(N(C)C)cnc(NCC(c2cccc(F)c2)O)cc1Br c1(CC(=O)NCC2(C(N(C3CCCC3O)CC)=O)CC2)cc(F)ccc1C N1(C(=O)C2=CCOC2)CCC2CC(C1)CN(C(=O)Cc1cc(Cl)sc1Cl)C2 N1(CCC)CCCC1C(=O)NCCC1CCN(CCCOC)C1 c1(C(N2C(C(=O)Nc3cccc(F)n3)CC(O)C2)=O)cccc(Br)c1O Cc1cccc(C(=O)NC(C(=O)NCCN2CCCCC2)C2CC2)c1O C1(CC(=O)NCC2(C#N)CCC2)CCCN(C(=O)CCCC2CC2)C1 C1(CCC)CCCN(C(c2nc(CNC(C3(C)CCCO3)=O)oc2C)=O)C1 c1(C(N(C)CC2N(C(C3(OC)CCOCC3)=O)CCC2)=O)c(Cl)sc(C)c1C C1(CNC(C2C(=C)CC2)=O)CCCC1.c1(C=O)c[nH]nc1-c1cnn(C)c1.N C1(CCC)CCC(N=c2[nH]c(N(CCCCO)C)nc3c2CSC3)CC1 C1(NC(c2ccccn2)=O)CC2(C1)CC2C(N1CCC(n2ccnc2)C1)=O CN1CCC(CC(=O)NCC(O)CCNC(c2cncc(O)c2)=O)C1=O C(=O)(C(C(C)(C)C)NC(C1CC12CCCC2)=O)NC1(C=C)CCCC1 c1(C(=O)NCC)cc(-c2ccnc(C(=O)NC(c3nccs3)C)c2)ccc1F N1(C(c2cc(C)nnc2)=O)CCC2(CCC(NC(=O)CC(C)P(C)(C)=O)C2)CC1 c1(C(=O)NC(C(C)NC(c2c[nH]nn2)=O)C)ccc(O)cc1C(F)F C1(OC)(OC)CCC1C(=O)NCCCO.c1(C(=O)N)cc(-c2ccccc2)[nH]n1 C1(NC(CSCCOC)=O)CCCCC1NC(=O)Cn1cc(Br)cn1 CC(C)CC(CNC(C1CCCCNC1=O)=O)C(=O)NCC1CC(C2CC2)=NO1 C(=O)(C(F)C(F)(F)F)NCC1N(C(c2cnn(C(C)C)c2F)=O)CC(O)C1 N1(C(C(CC)OCC)=O)CCC(NC(c2ccc(N3CCOCC3)cc2)=O)CC1 Cc1ccc(C)c(CC(N2CC3C(C2)N3c2ncc(Br)c(C)n2)=O)c1 c1(C(N2C(CNC(c3cccnc3S)=O)CCC2)=O)csc([N+](=O)[O-])c1 C=Cn1nncc1C(N1CCC(C(C)CNC(=O)C(=O)NC2CC2)CC1)=O C=CC1(C(=O)NCC2CC2C)CCN(C(=O)C2=C(C#N)CCC2)CC1 C1(C(=O)NCCN(CCC)C(c2nc[nH]c2C(C)(C)C)=O)CCC(C)CC1 C1(CC(N2CC(C(C(N3CCCC3C)=O)OC)C2)=O)CCCC(=O)C1 C1(C(N2CC=CC2)=O)CCCCN1C(C)C.C1(OCC)CCC1C(=O)N.C C(=O)C(C)(C)C(O)C(C)C.n1(CC)cnnc1CN(C)C(c1occc1)=O.C Cc1nc(C(=O)NCC(F)CNC(c2nccnc2C(F)(F)F)=O)n(C)n1 N1(C(c2c(C)n(C)cc2)=O)CC(CC(=O)NC(C)CCCO)C2(CC2)C1 c1(C(=O)NC2CC(NC(=O)CCC(F)(F)F)C2)cc2c(cc1[N+](=O)[O-])OCCCO2 C1(NC(=O)C(F)C2CCC2)COC2(C1)CN(C(=O)CN1Cc3ccccc3C1)C2 C(=O)(C(CC(C)C)C(C)C)NCCCN(C(c1cc2cnccc2[nH]1)=O)CC c1(CNC(c2ccc(Br)cn2)CCO)cc(F)c(F)cc1F Cc1nc2cc(C(=O)N)c(F)cc2[nH]1.C1CC(C)(C)CN1C(=O)C(F)C1CC1.C Cc1ccc(CN=C(NCC2(C)CCCO2)NC2CCOCC2)c(Cl)c1 S(=O)(=O)(c1cc(C)cnc1NCc1ccc(C2CC2)cc1)N(CCO)CC c1(OC)ccc2cccc(CCNC(=O)C(N)CC(N)=O)c2c1 c1(NC(C(N2C(c3cc(C(=O)OC)no3)CCCC2)=O)=O)c(C)cccc1O c1(C(=O)N)cc(O)n(C)n1.Cc1nccn1CCCNC(=O)CCn1cccn1 c1(CNC(COCCOCC)=O)ccccc1.c1(C=O)ccnc(F)c1.N O=C(C(C(F)(F)F)C(F)(F)F)N1CCN(C(=O)Cc2ncn3c2CCC3)C2CC12 c1(C(N2CC(CC(C(=O)NCCN3CC=CC3)F)C2)=O)c(F)cncc1F C=C1CC2(C1)CC(C(=O)NCC(C)CNC(C1CC1)=O)C2.c1ccccc1 C1(C(=O)NC(CC=C)CC=C)COC2(C1)CN(C(=O)CN1CSCC1=O)C2 c1(CN(C(=O)CCC(F)F)C(C)C)cc(Cl)nc2ccccc12 N1(CCNC)C(=O)CC(=O)N(C2C=CC(=O)NC2=O)C1=O.c1ccc(Cl)c(F)c1 c1(C(=O)NCC2(O)CCN(C(C(C#C)(C)C)=O)C2)cccc(F)c1CC Cc1nn2cc[nH]c(=O)c2c1C(=O)NCCCN(CCC)C.C1(C(=O)N)CCC1 C(N=c1[nH]cncc1C)C1(CCNC(c2c(C)n[nH]c2)=O)CC1 Cc1ccc(C(=O)N(C(C(=O)Nc2cccn3ccnc23)C2CC2)C)cc1C#N CCCC(C)(CCC)C(=O)NC(C)C=CC(=O)NC1CC2CC2C1 c1(CC)ccc(C=CC(=O)N(CC(C)(C)CNC(c2[nH]ncc2Cl)=O)C)o1 C1(C)(C(=O)NC(CCC)C2CCC2)CCN(C(c2cc(C)on2)=O)C1 C(C1=CCCN(C(C2CN(C)C2)=O)C1)NC(c1c(C)scc1)=O CCCCCC(C)CC(=O)NCC1C(C)CCN1c1cncc(C#N)n1 CCCCCC(C)(CC)C(=O)NC(C)CNC(=O)C(CC)C(C)C C1(C(=O)NC2CC(CC)(CC)C2)COCCN(c2nc(CCOC)ns2)C1 c1(C(=O)NCC(C)CC(N2CC(=O)NCC2C(N)=O)=O)ccc2occc2c1 c1(C(=O)NCC2CCCN(C(CCC3CNC(=O)N3)=O)C2)c(F)cc(F)cc1F c1(CC(N2CC(Cc3cn(CCCO)nn3)C2)=O)ccncc1Cl c1(OC)cc2[nH]ncc2cc1C(N1CC(C2CCN(C(=O)C(C)SC)C2)C1)=O c1(C(C(=O)NCC(CCOC)NC(c2ncc[nH]c2=O)=O)C)ccc(F)cc1 N1(C(c2cccnc2OC(F)F)=O)CCN(C(c2cnsc2)=O)C(CO)C1 CC(C)CC(F)C(=O)N1CCC(C)(NC(=O)Cc2nccn2C)C1 c1(C(=O)NCC(CO)NC(c2c(CC)noc2)=O)ccc(C(C)(F)F)cc1 c1(C(=O)NCC(CNC(C2CN(OC)C(=O)C2)=O)O)nccc2ccncc12 N1(C(c2cc(CC)[nH]n2)=O)CCC(CO)(NC(=O)CCn2c(C)csc2=O)C1 c1(NC(C)CC2CC2)ncccc1S(=O)(=O)N(C)Cc1cnccn1 c1(CC)nnsc1C(=O)N(C1CN(C(=O)C(C)=CC2CC2)C1)C C1(C(=O)NCC(C#C)CC2CC2)CCC2(CC2)N1C(=O)C(C1CC1)O C1(C(N(CCN(C(CC)=O)C)C)=O)(NC=O)CC2CCC1C2.C(C)(C)C.O C12(CC(N3CC(C)C3)=O)COC(C)(C1)C2.N1(CC(C)C)CCC(C=O)C1.N N1(C(C(C)=CC=C)=O)CCC2CC2(C(=O)NCC(C)(C)C2CCCC2)CC1 c1(C(=O)NC(CNC(CC(c2ccccc2F)C)=O)(C)C)csc2ccncc12 N1(C(C2CC(C(=O)OC)C2)=O)CCCC(C)CC1.C(c1cn[nH]c1)=CC=O.N N#Cc1ncc(Cl)c(N2C3CCC2C(CNC(=O)CC2CCCCC2O)C3)n1 N1(C(CC(C(=O)O)NC)=O)CCC12CCCN(C(=O)C(C)CSC)C2 C1(NC(C(CC)OC)=O)CC2CC1CN(C(c1sccc1F)=O)C2 C1(NC(=O)CSc2nc[nH]n2)CCOCC1C(=O)NCCOCCF CC(C)C(C(=O)NC(CCC1CCC1)C(=O)NCCC1CC1)C(C)C N1(C(c2c(C)coc2)=O)CCN(C)CC1C(=O)NCc1cccc(C)c1C c1(C(=O)NC(CNC(C(C=CCCC)O)=O)CC)cc(C)c(C)cc1C c1(CC)cc([N+](=O)[O-])ccc1NC(CNC(c1cnn[nH]1)=O)C1CCC1 N1(C(CCCCCCC)=O)CCCC12CCN(C(=O)CNC(=O)C(C)(C)C)CC2 N1(C(C2CCC(C(=O)OC)O2)=O)CC=C(CNC(c2nc(O)sc2C)=O)CC1 N1(C(C2CC3N(C)C(CC3)C2)=O)CCC2(CCC2)C(NC(c2cscc2Cl)=O)C1 CC1CCN(C(=O)COc2cccnc2)CC1NC(C1CCCN1C)=O Cc1c[nH]c(C(N2CCC(N(CCO)C(c3csc(C4CCCO4)n3)=O)C2)=O)c1 CC(C)CCCCCC(=O)N1CC(CNC(=O)COCP(C)(C)=O)C(O)C1 c1(C(N2CC(C)C(NC(C3(CCN(C)C)CC3)=O)CC2)=O)n[nH]c2c1CCCC2 C#CCCCC(=O)NCc1ncccc1CNC(=O)CCC1CC1 c1(OCC(=O)OC)cc(Cl)c(Cl)cc1NC(=O)C(N1CC(C)NCC1C)=O CN1CCN(C(C2CN(C(C3CC3c3ccco3)=O)C(C)(C)C2)=O)CC1CO CC1Cc2cc(C(C)NC3CC4CC3CC4(O)c3ccccc3)ccc2O1 c1(C(=O)NC2CC(C)N(C(c3cnco3)=O)C2)ccnc2ncccc12 C(=O)(C(O)CC(N)=O)NCc1c(C2CN(C(c3c(C)cncc3)=O)C2)ocn1 Cc1[nH]nc(C(N2CCN(CCCc3ccccc3C(F)(F)F)CC2)=O)c1O c1(C(=O)NC2C(NC(CC3(C)CCCO3)=O)CCC2)cc2ncccc2s1 N1(C(C)C)CCOC(C(=O)NCCCN(C)C(c2sccc2-n2ccnn2)=O)C1 Cc1cccc(OCCC(=O)NC2CCOCC2NC(=O)CC(C)CF)c1 c1(-n2cc(C(C)NC(c3c(CC(=O)OC)scc3)=O)nn2)ccccc1CCO CC1Cc2ccccc2N(C2CCN(c3ccc(Cl)cc3)C2)C1C O(NC(=O)CCC1CCN(C(c2n[nH]cc2Cl)=O)C1)CCC(C)O Nc1ccc(F)c(F)c1C(=O)N(CCNC(=O)C1=CCC1)C1CC1 C1(NC(c2cn(C)nc2)=O)C(C)CCC12CCC2.C(c1ccccc1)=CC(=O)N Cc1cc(C(N2CC=CC(NC(=O)C(C)C(F)(F)F)C2)=O)cc(N)c1O C1(C(=O)NCC(=C)CCNC(c2cn(C)nc2Cl)=O)CC(C)CC(C)C1 c1(-c2nnc(N3C(C4CCC(=O)NC4=O)CCCC3)n2O)cc2c(s1)CCOC2 c1(NCC2(N(C)C)COC2)ncnc2c1ccn2CC(=O)OC C(=O)(C1=CCCCC1)N1CCC(NC(=O)C(Cl)=CCl)(CO)C1 Cc1cc(C)n2ncc(C(N3CCOC(C(=O)N(CCCO)C(C)C)C3)=O)c2n1 C(C(C)(C)CC(=O)NCCC1CC1C)NC(c1cc(CC)ncn1)=O c1(OCC=C)ccc([N+](=O)[O-])c(C(=O)NCC(n2cc(C(C)O)nn2)C)c1 C1(C=O)CC2(C1)CC1(CC1)C2.c1(C(=O)N)cc(C2CCOC2)[nH]n1.C1CCC1 c1(CC(N2CC(CC(C)NC(CCC)=O)C2)=O)nc(C)sc1Br C1(C(N2C(CC)CN(C(c3scnc3COC)=O)CC2)=O)CCOC2(CCC2)C1 Cc1cc(C)c(C(=O)NCCC(C)N(C(=O)CC(C)O)C)c(C)c1Br S(=O)(=O)(c1ccccc1)N1CCC(C(N2CC3OC(=O)OC3C2)=O)CC1 c1(C(=O)NC2CCN(C(C(C)OCC)=O)CC2CC)[nH]c2c(c1C)CCCC2 c1cccc(C2CC2)c1F.Cc1oncc1C(=O)NC1CCCC1NC(=O)C.O C#CCC(O)C(=O)NC1C=CC(CC(N2CCN(CC3CC3)CC2)=O)C1 c1(C(N2C(COC)CCCC2)=O)coc2cc(N)c(-c3cc(C)ccc3O)cc12 N1(C(=O)OC(C)(C)C)CCC1C#CC(=O)N(c1ccc([N+](=O)[O-])cc1)CC(F)F c1(COC)ccoc1C(=O)N.C1(C2CC2)CCCC1.C(C)(C)C.C=O.C CN1CCN(C)CC(C(=O)NCCNC(c2ccn(C)n2)=O)C1 C1(F)CCCN(C(c2cnc(CC(C)C)s2)=O)C1.C(C)(C(=O)N)OCCOC C1(C(N(CCO)CC)=O)CCN(C(C)=O)CC1 c1(C=O)n[nH]c(C(C)C)c1[N+](=O)[O-].c1(SC)cn(C)nc1C(=O)N.CC(O)C CC1OCCCC1C(N1CCC(CCC(=O)N(CCn2cccn2)CC)CC1)=O C(=O)(CC(C)(C)C(F)F)N(CCOCCN(CC(F)(F)C(F)F)C)C C(=O)(C1CCCc2scnc21)NC(CC=C)CNC(c1cncc(C)n1)=O C1(NC(CC(C)(F)F)=O)CC2CC1CC2C(=O)O C1(C)(C(c2nnnn2CC2CC2)NC(COC)C2CC2)CCOCC1 c1(C(N2CC(=O)N(C)C(=O)C2)=O)oc2ccccc2c1CSc1nccs1 c1(SCCNC(c2n(C(CC)C)nnn2)COC(C)(C)C)cccc(Cl)c1 N1(C(c2c(CC)nc(C)s2)=O)CCN(C(=O)C(=O)NCC2CC2)CC(O)C1 C1(C(=O)N)CCC2(CCC2)CC1.c1(CC(N2CCC3C2C3)=O)ccc(Cl)c(F)c1 CC(C)(CC(F)F)C(=O)NCC1COCCN1C(c1cc2[nH]ccc2s1)=O c1(COC)nsc(NC(=O)CCC2(NC(C)=O)CCC2)n1 c1(OC)ccc(S(=O)(=O)CN2CCNCC2CC(N2CCN(C)CC2C)=O)cc1 C1(CC(C)C)CN(C(=O)C#CCNC(=O)C(C)(C)c2ccno2)CCO1 N1(C(=O)NC(=O)CN2CC3COCC23)CCSCC1C1CCOCC1.CCO C=CCC(C)(C)CC(=O)N1CC(OCC(=O)NCC2=NOC3CCCC23)C1 C=CCC(F)(F)C(=O)NC1COCC1CNC(c1ocnc1C)=O N1(C(c2cn(C)c(=O)cn2)=O)CC2CCN(C(c3cc4c[nH]cnc-4n3)=O)CC12 N1(C(C2CC(OC)C2)=O)CC2CCC(C1)N2C(C1CC(CCO)C1)=O c1(C(N2CCCCC(CNC(C(C(CC)C)OC)=O)C2)=O)cncc2nc[nH]c12 C1(NC(C(CO)N(C)C)=O)CN(C(=O)C(C)(C)C(N)=O)CC(F)(F)C1 c1(C(=O)NC2C(CNC(c3ccccc3)=O)C2)nnc(O)nc1O.CCO.S C#Cc1cc(C(N2CCC(C(=O)NC3C(O)CC3O)C2)=O)ccc1C O=C(C#CC1CCCC1)NC(CCOCCO)C(=O)N1CC(NC(N)=O)C1 CC1OC2(C)CC1(C(=O)NCCN1CCCOCC1)C2 Cc1c[nH][nH]c1=NC(=O)C1CSCCN1C(c1ccncc1F)=O c1(C(N2CCN(C(C=C(C)c3ccco3)=O)CC2)=O)ccc2c(c1)C(C)C(C)O2 CC1(C(=O)NCC(c2ccccc2)NC(=O)CC(F)F)CC=CC1 N1(C(C(OC)OC)=O)CCC2(CC1)CC(NC(c1cnc(Cl)cn1)=O)CO2 C(=O)(CC(C(F)F)n1ccnc1)NCCC1N(C(c2n(C)c(S)nn2)=O)CCC1 c1(NCc2c(OCC)cc(C)cc2)nc2ccccc2[nH]c1=NC1CC1C(N)=O c1(CCC(c2noc(-c3ccnc(-n4cccn4)c3)n2)N)cccc(F)c1F n1(CC(N2CCCCC2c2ncc(Br)cn2)=O)ncc2nc(Br)ccc12 CCCCC(C)CCC(=O)NC(CCN(C)C(C1(CC(C)C)CCC1)=O)C(C)C N1(C(c2c(CC)n(C)nc2)=O)CCCCC(CNC(=O)C)C1.CCC(F)(F)F.S N1(C(CCS(=O)(=O)N(C)C)=O)CC(NC(c2n[nH]cc2[N+](=O)[O-])=O)CC12CCC2 c1(C(=O)NCC2C(C)CN(C(=O)CC3CC=CC3)C2)cnc(Br)c(N)n1 N1(C(C2C(CC)C2)=O)CC(NC(=O)C(C)Oc2ccc(Cl)cc2C)C2CC2C1 CCCCCCC(=O)N(C)CC1CCN(C(C2CC(=C(F)F)C2)=O)C1 C1(c2cn(C)nc2)NC(=O)N(CCCN2CCCC2C(N)=O)C1=O c1(N(C)C)nc(C(N2CCC(CCS(C)(=N)=O)CC2)=O)[nH]c(=N)n1 Cc1ccc(O)c(CN2CCC(O)(C(=O)NCc3cnn(C(C)C)c3)C2)c1 NC(=O)CCCCC(=O)N1CCN(C(c2ccc(C(F)F)o2)=O)CC(CO)C1 c1(C(N2CC(C)(C)C(NC(C3CC(=O)C34CCC4)=O)C2)=O)c[nH]c2ccccc12 N1(C(C(CC)(C)C)=O)CCCC(NC(=O)CC2(O)CC2)C1C N1(C(COC2CN(C(c3oc(CC)c(C)c3)=O)C2)=O)CC(S(C)(=N)=O)C1 Cc1nn(C)cc1C(=O)NC12CC(NC(C3CC(CCO)C3)=O)(C1)C2 N1(C(c2ccc(OC)c(Cl)c2)C(=O)NCCSC)CCC(C2CCCOC2)CC1 c1(C(N(CCCCNC(C23CC(O)C2C3)=O)C)=O)ccc(C2CC2(F)F)cc1 C1COCCN(C(=O)C(F)=CC2CC2)C1.C1(C(=O)NC)(COC)C=CCC1 CCC(N=c1cc(NCC2=CCCCC2)nc(COC)[nH]1)c1ccn(C)n1 C1(NC(CC=C=C)=O)CCC(C)N(C(c2ccc(CN(C)C)cc2)=O)C1 C1(CC)(CC)CC(NC(c2ccc(F)c(S)c2)=O)CN1C(=O)CCC(C)(F)F c1(NC(=O)NC2(OC(C)C)CCC2)cccnc1-c1ccc(Cl)cc1 C1(C(N(CCSC)C)=O)C=CCCN1C(C1COCC1C(N)=O)=O C1(C(=O)NCCCN(C(CCCSC)=O)CC2CCCC2)CCOC1(C)C N1(C(C(C)N(CC)CC)=O)CC2CCN(C(c3cc(CC)n(CCO)n3)=O)C2C1 Cc1ncn2ccc(C(=O)NC3COCC3NC(=O)CCC3CCCN3C)cc12 c1(C(N2CCC(Cn3cc(-c4ccccc4)nn3)C2)=O)ocnc1C1CC1 C1(C(=O)NCc2c(C(C)C)n[nH]c2)CC12CCC2.C1(C=O)CC2(CC2)C1.C c1(NC(C)=O)ccc(C(=O)NCC(O)CNC(=O)C(F)=CCCF)cc1 C(=O)(C(C)CC(C)(F)F)NCCC1N(C(Cc2nc(C)oc2)=O)CCC1 C12(C(N3C(CNC(CCc4n(C)ccc4)=O)CCC3)=O)CCC(CC1)CC2 C1(CC)CCN(C(c2ccnn2COC)=O)C(C(=O)NOCCC(C)O)C1 CC1CC(NC(=O)O)CN(C(=O)Cn2c(-c3ccc(Cl)cc3)nnc2S)C1 N1(C(Cc2c(C)nc(CCCC)s2)=O)CCN(C(c2occc2F)=O)CC1CC Cc1ccsc1C(=O)NCC1COC(CNC(=O)C=Cc2cc[nH]n2)C1 C1(OCC)COCCC1(c1nnnn1C1CCOCC1)NC1CCN(CC)C1=O C12(C(=O)NC3C(OC)CN(C(c4c[nH]ccc4=O)=O)C3)COCC1C2(F)F C=Cn1nccc1C(=O)NCCC(C(C)C)NC(c1ncccc1C(C)(C)C)=O c1(C(C)(C)C)cnnc(NC(C2CNOC2)=O)n1 c1(OC)cc(C)cc(C(N2CCN(C(c3cc(F)n[nH]3)=O)CC2C(C)C)=O)c1C Cc1cc(F)ccc1C(N1CC2C(CC(N3CC(F)(F)CC3CO)=O)C2C1)=O C(CCCCCO)(C(=O)Nc1ccc2c(c1)OCO2)N1CC(C)OC(C)(C)C1 c1(C(N2CCC(n3cc(C(C)OC)nn3)C2)=O)ccc(C(C)O)cc1 N1(C(C(C)(N(C(c2[nH]cc(C)c2)=O)C)C2CC2)=O)CC2CCCC12 C(CC(=O)N1CC(C)C1)(c1cccs1)NC(C)=O.C1CCOC1.C(=O)(C)N.C C(C(CC1CC1)C(=O)N1CC(Cc2ccco2)C1)NC(c1c(C)[nH]cc1)=O C1(C(=O)NC(C(=O)Nc2ccc(OC)cc2)(C)C)CC2(C1)CC2(F)F C1(Cc2onc(C)n2)CCN(C(C2(c3cccs3)CCOCC2)=O)CC1 C1(COC)CN(C(=O)C2=CSCS2)CCN1C(=O)CC1(C)CCC1 c1(C(N2CC3CC(NC(C4(CF)CC4)=O)C2C3)=O)cccc2c1OCCC2 C1(CNC(C=NOC)=O)CN(C(=O)CCC2CCCN(C)C2)CC1O C(C(C)(C)CCNC(=O)CCOCCN(C)C)NC(c1n(C)cnc1)=O c1(C(=O)NCC2(C)CN(C(C(CC(=C)C)C)=O)C2)cn2c(n1)CCC(C)C2 C1(CNC(C2CCN(C(C)=O)CC2)=O)CN(C(=O)C(O)CC(C)C)CCN1C c1(C(=O)NC2(CC(N3CC4(C=CCO4)C3)=O)CC2)occ2c1CCC2 C1(C(N2CCC(C)(CNC(C#CC(C)(C)O)=O)C2)=O)CC(c2cccnc2)=NO1 N1(C(c2c(C(C)C)con2)=O)CCN(C(C2CCCCCS2(=O)=O)=O)C2(CC2)C1 c1(C(N2C(C)C(NC(=O)C(O)C3CCC3)CC2)=O)cc(=O)c2ccccc2n1C Fc1cc(CC2CC3CN(c4nnnn4Cc4ccccc4)CC23)c(F)cn1 N(C1CCc2ccccc21)C1(c2nnnn2C2CCC2)CCC(C#N)CC1 c1(NC2CC(CNC(C3CCC3)=O)C2)ncc2ccc(Br)cc2n1 c1(CNC(C2(NC(CCC3C(C)C3)=O)CC2)=O)csc(C)n1 c1c(Br)cnc(Cl)c1[N+](=O)[O-].Cc1ccc(F)c(CNC2C=CC(C(=O)N)C2)c1 C=CC1(O)CCN(C(=O)C(CNC(c2ccccc2Cl)=O)C(C)C)C1 N1(C(C(C)(Cl)CCl)=O)CCC2(CCC(C(=O)NCC3CC3)O2)CC1 C1(O)(C(N(CCC(c2cccs2)NC(=O)CCC2CC2(C)C)C)=O)CCSC1 C1(CC(=O)NCCC(=O)NCC)CC(C)N(C(c2nonc2CC)=O)C1 Cc1cc(C(N2CCCC(C(=O)NCc3cscn3)C2)=O)cc(Br)c1 c1(NCC2CCC(SCC)CC2)ncc(C(=O)O)n2cncc12 C1(C)(C(=O)NCCSC)CCN(C(=O)Cn2ccnc2)C1 c1(C(=O)NCCCC(C)NC(CCC#CC)=O)cc(=O)c2ccccc2[nH]1 Cc1cnn(C)c1CC(N1CC(OCC(N2CCC(C(N)=O)C2)=O)C1)=O C(C)(CC(=O)NCc1csc(C(=O)NC2(c3cccnc3)CC2)c1)SC C1(C(NOC)=O)C(C2CC2)CCN1C(=O)C=CC(C)(C)C N1(C(c2cnn(CC)c2C)=O)CC(C)N(C(c2cnc(SC)s2)=O)CC1C CCCCC(O)C(=O)NCCNC(C1CCCN(C(=O)Cc2csc(S)n2)C1)=O C(CC(O)C(F)(F)F)NC(C=CCN(C(c1ncn(C(C)C)n1)=O)C)=O c1(CNC(c2c(Cl)cn(CCC)n2)=O)cc(O)ncn1.C(=O)C(C)C(C)C.C c1(C(=O)NCCC(C)(C)NC(C(CCC#C)O)=O)cc(Cl)nc(Br)c1N c1(C(N2C(CO)CC(NC(=O)CC3CC3(Cl)Cl)C2)=O)cccc2nccnc12 C(=O)(C1=CC2(CCOCC2)C1)N(C)CC1CC1.c1(C(=O)N)cc2ccccc2s1 c1(OC)ncnc(N2CCNCC2C(=O)NCCCCN(C)C)c1C n1(CC(=O)NC)ccc(=O)n(C)c1=O.N1(C(C(C)OCC#C)=O)CCCCC1 C1(NC(C(C)SC(F)(F)F)=O)CCCCC12CCN(C(C1CC(N=[N+]=[N-])C1)=O)C2 Cn1cc(C(C(=O)NCCC2CC2)NC2CC2)c(I)n1.C1COC(C)(C)O1 c1(C(N2C(C(=O)NCC=C)CCC2)C(=O)NC2CC2)cnn(C)c1F C1(CNC(c2ccncc2)=O)CN(C(=O)CCc2cncs2)C2CC12 c1(C(N2CCC(O)(CC)C2)=O)ccc2c(O)nncc2c1.C1(C(=O)N)CC(=O)N1 Cn1cc(C(=O)NC2CC3CCCC(C2)N3C(c2cncs2)=O)c2cccnc12 c1(OC)nccc(S(=O)(=O)NC(c2cccc(C(F)(F)F)c2)CC2CC2)c1Cl n1(CC(=O)NC2CCN(C(CN3CC(CC)C3)=O)C2)cc([N+](=O)[O-])nc1C Cc1nn(C2CC2)cc1C(=O)NCCOCC.C(=O)(CCc1cc[nH]n1)N c1(CC)cc(N(CCCNC(=O)C(C2CCCCC2)O)CC)ncn1 c1(C=O)cn(C)c(=O)cn1.C1(C(=O)OCC)(NCC)CC(=O)C1.CC CCCCC(CNC(C1CSCC(=O)N1)=O)NC(=O)CCOCC(F)(F)F C1(CCC(=O)N(CCOC)CCNC(c2ccc(F)s2)=O)CCCC(O)C1 CC1CC2(CCN(C(=O)C(C)(C)O)CC2)CN1C(=O)CCC=CBr c1(C(N2CC(OCCNC(C(COC)OC)=O)C2)=O)ncc(N)nc1C N1(C(C(C(CC)O)C)=O)C2CCC1CC(N(C)C(C1CN(CC(C)C)C1)=O)C2 c1(-c2nnc(N3CCOCC(C)(O)C3)n2CC2CC2)cc2ccccc2nc1O CC(CC1CC1)C(=O)NCC1(F)CC(CNC(c2c[nH]nc2Cl)=O)C1 c1(C(N2CC(NC(C(C)C)=O)C(C(F)F)C2)=O)ccc(F)cc1.[SH](C)(=O)=O C1(C=O)CCCN1C1CCCC1.C1(CC(=O)N(CC)CC)CC2(CC2)C1.N c1(CCC)ccc(N)c(C(N2CC(NC(c3ccc[nH]3)=O)C(C)(C)C2)=O)c1 Cc1ccc(=O)n(CC(N2CCC(NC(c3nc(C)oc3C)=O)C2C)=O)n1 c1(CN(C(=O)CC)CC)cnc2cc[nH]c2c1.N12CCC1C(=O)N1CC2C1.S N1(C(C(C)CF)=O)CCC(F)(CNC(=O)Cn2cc(CO)nn2)C1 N1(C(C23CC(CC)(C2)C3)=O)CCC(O)(CNC(=O)CC(C)C(C)C)CC1 N1(C(c2csc(Cl)c2)=O)CCC(NC(N)=O)CC1.C1(=O)CC2(CC2)N1C CC1=C(C(=O)N2CC(C(N)=O)(CNC(C3(C)CC3(F)Cl)=O)C2)CCCC1 c1(C(=O)NCC(C)CNC(c2cc(N)cc(O)n2)=O)ccnc2ccsc12 N1(C(C2C(OCC)C2)=O)CCCC(NC(c2ccnn2CC(F)F)=O)C1C Cc1cc(C(=O)NCCc2ccc(C3CC3)cc2)c(Cl)cc1N c1(CN(C(=O)C=CC(C)NC(=O)CCc2ccnn2C)CC)occc1C C1(OCCN(C)C)CCN(CC2C3CN(CCCS(=O)(=O)N(C)C)CC23)CC1 C1(OCC)CN(C(C2(F)CC2C)=O)CC1CNC(=O)CCCn1cccn1 C12(NC(=O)CC3(NC(c4cncnc4)=O)CCC3)CCC(CC1)C2 C1(N(CCCC#C)C(c2cnc(C(F)(F)F)s2)=O)CCCCC1 C12(C(N(CCN(C(c3ccccc3)=O)C(C)C)C)=O)CC=CC(C1)OC2.C C1(O)(C(C)NC(CCOCCC)=O)CN(C(=O)C(C)CS)C1.c1ccccc1 C12(NC(COC(CC)C)=O)CC1CN(C(c1[nH]ccc1C1CC1)=O)C2 CC(C)(C)CC(O)C(=O)N1CC(C(=O)NC(C2CCOC2)(C)C)C2(CCC2)C1 N1(C(c2c(C)nc(C)o2)=O)CCCN(C(c2ccccc2F)=O)C(C)C1 N1(C(CN(CC)CC)=O)CCC(F)C(NC(C2CCC(C)(C)C2)=O)C1 CC(C)CC(C(=O)NCCCCN1CCCC1)ONC(=O)C(C)NC=O C(=O)(CC(=O)NC1CCN(C(=O)C(C)OCc2ccccc2)C1)NCC c1(C(=O)NCCN(CCOC)C(C2CCCOC2)=O)cnc(O)c2cnccc12 c1(OC)ccc(F)c(CNC(C2CCC2)=O)c1.c1(CC(=O)N)ncccc1F N1(C(c2cncs2)=O)CCN(C(=O)C(F)(F)Cc2ccccc2)C2(CCC2)C1 C1(C(=O)NC2CC(CC(=O)Nc3ccc(F)cc3CO)C2)CCCCC1(F)F C1(C)(OCC)CCN(C(C2CCN(C(C3COCOC3)=O)C2C(C)C)=O)CC1 C(=O)(CN=c1cc[nH]cc1)NCCOC(c1cc(C)c(=N)[nH]c1)C C1(N(C(c2c(C)ccnn2)=O)C)CCCCN(C(=O)CN(C2CCSC2)C)C1 C=C(C)CC(C(=O)N(CCN(C)C)CC)NC(c1ccnn1CC)=O N1(C(C2CC2F)=O)CC2C3CCC(C2C1)N(C(C1(F)CCOCC1)=O)C3 C(=O)(CCC(C)c1ccccc1)NC1(C)CN(C(Cc2cc(C)ns2)=O)C1 c1(C(N(CCCCCNC(c2ncoc2Br)=O)C)=O)ccccc1CO C1(C(=O)N(CC(C2CCCC2)O)C)(OC)CCN(C(C2CC2C2CCC2)=O)C1 c1(CC)c(C(=O)NCCCC(C)C)nnn1C.c1(C2C(C=O)C2)ccc(Cl)s1.N CC1CCCCN1CCNC(=O)CC1CCN1C(=O)Cn1cnc(=N)[nH]1 Cc1cc(=NC(=O)C(=O)NC2(CO)CN(C(=O)C=Cc3cscn3)C2)[nH]o1 C(=O)(C(CCC1CC1)NC(C1CCOCC1)=O)NC1CCN(C)C1 N1(C(CCN(C(COCC#C)=O)CC=C)=O)CCC(F)(F)CC1 Cc1cc(O)c(Cl)cc1C(=O)NC1CCCC12CN(C(C1CC1(C)C)=O)C2 CC1CN(C(C2CC3C(C2)C3(F)F)=O)CCN1C(C1CCC(=O)N1C1CC1)=O C1(NC(CN(C(C)=O)C)=O)(C)CCOCC1.n1(CC(=O)NCC)cnnn1 C1CN(C(=O)CCc2ccn(C)n2)C(C)(C)C1.C(=O)(CCC=O)N(CC)CC C12(C(N3CCCC(C(C(=O)NCCOCC=C)C)C3)=O)CC(C)(CCO1)C2 C1CN2CCC1C2.C(Cn1cncn1)(C(=O)N)NC(c1cc(C2CC2)[nH]n1)=O Cc1nnc2n1CCC(COC(=O)COc1ccc(Cl)c([N+](=O)[O-])c1)C2 C1(NC(c2cc(CC)on2)=O)CCN(C(C23CC(OC)C2C3)=O)CC1CO C#Cc1cccc(C(=O)NC(COCC)C(N2CCCC(O)(CO)C2)=O)c1 C1(NC(Cc2c(C#C)cccc2)=O)CCN(C(=O)C=CCOC)CC(C)(C)C1 c1(C(N2CCC(NC(C3CC(C(C)(C)C)C3)=O)C2)=O)c(O)nnc2c1CCC2 CCCC(CC(=O)N1CCCC(OC)C1)NC(C1CC2(CCCO2)C1)=O C1(CC)COC(C)(C)CN1C(=O)C1=CC(O)C(NC(=O)CC2=CCCC2)C1 C(C(CC(C)C)C(=O)NCC1C2CCCC12)NC(CCCC(=O)OCC)=O N1(c2c(F)cnc(C)n2)C2CCC1CN(C(c1cc(F)cc(F)c1)=O)C2 c1(OC)cc2c(cc1F)N(C(c1ccc(C#N)s1)C(=O)NC(C)C)CCC2 Cc1ccc2nccn2c1CN1CCC(C(N)=S)CC1 CC(O)C(C)(C)C(=O)NCCC1(O)CCN(C(c2c[nH]c(Br)c2)=O)C1 C=C(C)CC(C(=O)NC(c1cn(C)nn1)C(=O)N(C)CCN1CCOCC1)OC C1(CC(=O)OCC)CCN(C(=O)Cc2cc(Cl)cc3c2OCC3)CCC1(F)F N1(C(CCCN(C(=O)OC)C)=O)CCC(NC(c2ccc(CO)cn2)=O)C(F)C1 CC1CC(NC(C2CCS(=O)(=O)N2)=O)CCN1C(C1(c2cccs2)CC1)=O N1(C(CCNC(C)=O)=O)CCCC(Cn2cc(Cn3cc(Cl)cn3)nn2)C1 c1(N(C)C)ccc2c(n1)CCC(=Cc1cncc(O)c1C)C2=O C1(CNC(CNC=O)=O)CCCN(C(=O)CC2CCCC(F)(F)C2)CC1 N1(CC(C)C)CCCC(C(=O)N(CC(O)CNC(=O)Cc2ccccc2)C)C1 N1(CC)CCC(CCN)CC1.Cc1nc(SCC(N2CCOCC2)=O)n[nH]1 C1(C(=O)NC2(CN(C(C(COCC)C)=O)C)CC2)CC2C=CC1CC2 CCCC(CC)CCC(=O)NC(C(=O)Nc1cc(O)c(C)cc1C)C(C)(C)C C1(C)(CNC(C2OCCN(C)C2)=O)CN(C(=O)COCCF)CCO1 c1(CCCC(N2CC(CNC(CCC(C)OC)=O)OCC2)=O)ccc(C)c(C)c1 Cc1cccc(C(C)C(=O)NC2CCC2NC(c2ncccn2)=O)c1 N1(C(=O)C#CC2CCC2)CCCC1C1CCCN1C(=O)CCc1cscn1 C(C(C(=O)OCc1nc(CS)no1)c1ccccc1)OCC=C.c1ccccc1 C(=O)(CCCC(F)(F)CO)NC1CCN(C(CC=C(C)C)=O)C(C)C1 c1(CC(=O)NCC(CC)NC(=O)C(C)(C)N2CCOCC2)ccncc1Cl C1(NC(C=CSC)=O)CC2(C1)CN(C(c1ccc(-n3ccnn3)cc1)=O)C2 c1(C=O)cc2cc(Cl)ccc2[nH]1.C1(OC)CN(C(=O)C=C2CCN(C)C2)CC1.N CC1CCC(CNC(C2(NC(=O)CSC(F)F)CCCC2)=O)C1 Cn1ncc2c1CC(C(=O)NCC(CNC(=O)CC)C(F)(F)F)CC2.C(N)=O C1(NC(C(C)(C2CC2)OC)=O)CCC(O)C1.c1(CC=O)ccc(Cl)cn1.C C1(NC(CCC)=O)CCC(C)(C)CC1CNC(=O)COC C1CC(O)C12CCC2.C=C(F)C1(CC(=O)NCC2CC2CC(=O)N)CCC1 c1(CCCNC(c2n(CC)nnn2)C2CCCOC2)cccc(F)c1 C(=O)(CS(=O)(=O)CCC)NCC1(n2cccn2)CCN(C(C(CCC)O)=O)CC1 CCC(C(=O)N(C)CCN(C)C(c1nc(C)sc1Br)=O)C(C)(F)F N1(C(c2[nH]cc(C)c2C)=O)CCC2CN(C(C3(O)CC3)=O)CC12 Cc1ccc(C(N2CC(NC(C3(c4ccccc4)CC3)=O)C(C)C2)=O)c(Cl)c1 N1(Cc2c(OC)nccc2)CCC(NC(c2n[nH]c3c2COCC3)=O)CC(C)(C)C1 N1(C(C2C3CN(C(=O)C4CC4)CC23)=O)CCc2ccccc2C1c1cccnc1 N1(C(C2C(C)C2)=O)C2CCC1C(F)C(NC(c1cccc3c1OCCC3)=O)C2 CCCC(C(=O)N(C(CNC(=O)CC=Cc1ccc(C)cc1)C1CC1)C)C(C)C C1(NC(=O)C2=CCOCC2)CC2CCC1CN2C(c1cnn(C(F)F)c1)=O CC1(C)C(C(N2CCCC(c3ccc(NC(C4(O)CC4)=O)cc3)C2)=O)C1(C)C N1(C(C(C(C)C)(C)C)=O)CCN(C(C2C(C3CC3)C2(F)F)=O)CC(O)C1 c1(C(N2CC(CNC(CNC(C)=O)=O)C(F)(F)C2)=O)cnc2ccnn2c1N C(N=c1ncc2cc(F)ccc2[nH]1)C1CCC(NC(=O)Cc2ccccc2F)CC1 N1(C(c2ccc(C)n2C)=O)CCC2CCN(C(=O)CCC3CC(F)(F)C3)CC12 c1(CC(=O)N(CCCNC(=O)CCc2cc(Cl)no2)CC)cccnc1.O c1ccc(F)cc1.C1(C2(NC(C(C)NC(CC)=O)=O)CC2)CCCN1CC.C CCCCCC(O)CC(=O)NC12CCC(NC(=O)Cc3cccnc3O)(CC1)C2 S(=O)(=O)(c1ccc(Br)cc1Cl)N1CCC(COCC)C(C)CC1 C(C)(N=c1[nH]c(=NCCCC(=O)N(C)C)[nH]c2c1CCC2)c1ncc(CC)s1 CC1(C)CC1(C(=O)NC)NC(C12CCCC1C2)=O.c1cc(C2CC2)no1 C1(NC(=O)Cc2ccc(C3CC3)cc2)CC2CC1CC2SC Cc1ccc(Cl)c(OCC2CCCC(C)(C)O2)c1 CC1(C)CNC12CCN(Cc1cccc3c1nnn3C)C2 CCCCCCC(C(=O)NCCCNC(C12COCC(C1)OC2)=O)NC(C)=O C(=O)(C#CC1CCOCC1)NCCCN(C(C=C(C)c1ccccc1)=O)C(C)C N1(C(c2c(CC)cc(C)cc2)=O)CCC2CCN(C(=O)C=CSc3nc[nH]n3)CC12 CC1(C)CCC(C(=O)NC2(C(F)F)CC2)CN1C(=O)C(C1CCCCC1)=O c1(C(=O)NC2(CNC(C(CC)NC(N)=O)=O)CCOC2)cc2ncccc2o1 c1(CNCC2CN(C(c3cc(C(C)(C)C)on3)=O)C2)coc2ccccc12 c1(C(C(=O)NC2CCCCC2)N(C)CCC2CCC(C)(C)O2)cc(F)cc(Cl)c1 Cc1nc(=NCC2CC(NC(=O)CC(C)(C)CC(F)F)C2)[nH]cc1[N+](=O)[O-] C1CN(C(=O)C(F)(F)c2cnccn2)CC1C.C(C)(C)C=O.C(=O)(NCC)N C(C1CCCC1)=CC(=O)N(CC(CC)NC(C(C)OCCC=C)=O)C N1(C(CSSC)=O)CC(NC(=O)COc2ccccc2F)CC1C Cc1nn(C)cc1S(=O)(=O)N1CCCC(C)(C(=O)NCc2ccc(F)c(Cl)c2)C1 c1(OCCN(C)C)cc(C(=O)NCCCNC(=O)C=C2CCC2)ccn1 CCCCC(CC)CC(=O)N1CCN(C(c2cnc3ncccn23)=O)CC(O)C1 CCC(C)CC(=O)NC(C(=O)N(C(C)CC(F)(F)F)C)c1cccs1 N1(C(CCCCCC#C)=O)CC(C)OC2(CCN(C(=O)C(F)(F)CC3CC3)C2)C1 Cc1cc(C(=O)NCC2CC3CCC2N3C(c2cnco2)=O)nc(C)n1 CC1(CNC(c2ccc(C)c(Cl)c2)=O)CC(F)(F)CN1C(=O)C.C1CC1 c1(C(=O)NCCN(C(C(CC)C(=O)OC)=O)C2CC2)cc2c([nH]1)CCCC2 C1(C(=O)NC(CNC(CCCCC)=O)CCCC)CCc2ncnn2C1 c1(CC)cc(F)ccc1C(N1CC(NC(c2cc(OC)n[nH]2)=O)C1)=O N1(c2ccnc(NC(c3ccc(OC)cc3)CCC)n2)CC2CCCC2C1 c1(C2C(NC(=O)NCCN(C3CCCCC3)C)C2)ccc(Cl)cc1 CCC(CC(=O)NC(CCF)C(N1CCCC2C(O)CC12)=O)CC(C)C C(=O)(C1=CCOCC1)NCC1CCC(C(N2C(CC(=O)OC)CCC2)=O)O1 C(C1=C(C)CCC1)NC(C1C(CNC(c2c(CC)cco2)=O)CCC1)=O C1(NC(C(C)(C)N(C)C)=O)CC2CC1N(C(=O)CCc1cscn1)C2 C1(C)CS(=O)(=O)CC(=O)N1.c1(C(C=CC(=O)NCC)=O)cccnc1 c1(C(=O)NC(CNC(CCCCCOC)=O)(C)CO)cc2c(C)ccc(Cl)c2[nH]1 N1(C(C2CCC(NC(c3cnc(C(C)C)o3)=O)C2)=O)CC(=O)NC2(CC2)C1 c1(C(=O)NC(CC)(C)CNC(C2CC(F)C2)=O)sc(C(C)OC)nc1C N1(C(C)=O)CCC(N=c2[nH]c(=NCc3c(Cl)cnn3C)[nH]c3cccnc23)CC1 Cc1cc(C(N2CCCC(C(C)C(=O)Nc3cn(C)nc3Cl)C2)=O)c(C)cn1 C1(CC(=O)N(CCC#C)CCO)COCCN1C(=O)CN(C)C(=O)OC C1(C(=O)NCC2CC(C)C2)(NC(=O)C(O)C2CC2)CCCC1 c1(C(N2CCCN(C(C3CCSCC3)=O)CCC2)=O)cccc2c1CCO2 c1(OC)cc(CC(=O)NC2(C)CC(NC(c3cncc(Cl)c3C)=O)C2)ccc1C C1(OCC)CCCCC1NC(C1CN(C(=O)CC2(C)CC2(F)Cl)C1)=O C1(CNC(C2(C)CCOC2)=O)CCCCN(C(c2cnncc2C(F)(F)F)=O)C1 N1(C(c2c(CC(C)C)cccc2)=O)CCC(NC(=O)C(F)(F)C(C)O)C(O)C1 C1(C(=O)Nc2cc(C)no2)CCCN(C(=O)C(O)Cc2ccc(O)cc2)C1 N1(C(C(CCCC)NC(c2nccn2C)=O)=O)CCCN(CC)C(=O)C1 C(C(C)C(=O)N1CC(C(=O)NCc2ccc(C)o2)(CC)C1)OCC N1(CC#C)CCc2ccccc2C1CNC(c1cc(C#N)c[nH]1)=O c1(N2CCC(C(N3CCCC(COC)C3)=O)CC2)ccc([N+](=O)[O-])cc1Br C(=O)(CC(F)(F)CC)NC1(C(=O)NCC(=C)Cl)CC1(C)C N1(C(C(CSC)(C)C)=O)CC(NC(=O)CC2CC3(CCC3)CO2)C(N=[N+]=[N-])C1 N1(C(C(=O)NCCC)C(C2CCOCC2)OC)CC(C)CCC1C N1(C(Cc2n(C)ccn2)=O)CCCC2CCN(C(=O)CC(C3CC3)C3CC3)CC12 C(CC(=C)Cl)(C(=O)NC(c1scnc1C)C)NC(COCC(=C)C)=O C12CC(=NO1)C(=O)NC2.C1(NC(CC=C(C)C)=O)CC2CCC1C2 C(C(COC)N=c1[nH]c(N2CCCC(C)(F)C2)nc2cc(OC)ccc12)OC Cc1nocc1C(=O)NCc1ccoc1C(=O)N(C1CCSC1)C c1(NCCOC(CC)(C)C)cc(N(CCCC(C)O)C)nc(C)n1 N1(C(c2c(C)ncs2)=O)CC(NC(c2cnc3n2CCC3)=O)C(C2CC2)C1 C(=O)(CC(O)(CCC)CCC)N1C(C#C)CN(C(=O)C2=CCCSC2)CC1 c1(NC(C)=O)cccc(F)c1C(=O)N.C1(C=O)C(C)(C)C1(F)F.C1CC1 CCCCC(O)CC(=O)NC1CCCCC1CNC(c1coc(C#N)c1)=O N1(c2ncc(F)cn2)CCC2C(CCN2Cc2cc3ncccc3o2)C1 N1(C(CN(CCC)C)=O)CCC(CC(=O)N(C(CC)CO)C)CC1 C1(NC(CC2(C)CCCCC2)=O)CCN(C(C23CCCC(C2)OC3)=O)CC1O C(=O)(C1COc2ccccc21)NCCC1CN(C(CC(n2ccc(C)n2)C)=O)C1 N1(C(COCCCCC)=O)CCC2CN(C(=O)C(C(C)C)C(C)C)C2C1 C1(C(N2CC3C(NC(c4ccc(OC)cn4)=O)(C3)C2)=O)CC12CCCCCC2 C1(c2ccccc2)(CN2CC(CCC=C)(NC(C)=O)C2)CCNCC1 C1(CCNC(Cc2c(C)cc(C)s2)=O)CCN(C(=O)Cn2cc(Cl)cn2)C(C)C1 C(=O)(CCC(=O)NN(C)C)N1CC(C#C)(C(=O)N(CC)Cc2ncc[nH]2)C1 C1(C(=O)N(CC(C)NC(=O)CCc2csc(=N)[nH]2)C)(COC)CCOC1 CCCC(F)(F)C(=O)NC1CCCCC1NC(C1CCCO1)=O C1(NC(C2C3(CC(NC(c4c(C)csc4)=O)C3)C2)=O)CC2OCCCC12 CCCC(CC)C(=O)NC(CC(C)C)C(=O)NC1COCC1CN(C)C c1(C(=O)NC2CN(C(C3CCC3)=O)CC2O)ccc(F)c(O)c1 CC(C)(O)C(=O)N(C)CCN(C(=O)C=CCn1cncn1)C(C)C.CO C(C)(C(C(=O)NC(C)C(C)F)NC(C1CC(C)CCO1)=O)OC C(=O)C(C)(C)C(=O)N(C)C.n1(CC)c(C(=O)N)cnc1O.C1CCC(CC)C1 N1(C(Cc2c(C)cco2)=O)CCC2CCN(C(=O)COCC(F)F)CC12 CCC(CC(=O)NC1(C)CC(NC(C2(c3ccc(Cl)cc3Cl)CC2)=O)C1)C(F)F c1(N2c3ccccc3CC2)nc2c(c(=NC3CCC4CC34)[nH]1)SCC2 C(COCC1CC1)N=C(NC1CCCC1)N1CCC2OCCC2C1 Cc1cc(=O)n(C)cc1C(=O)NC1CN(C(=O)C)CC12CCC2.C1CC=CC1.O c1(NC)cccc(C(=O)NCCCCCCNC(=O)CNC(C)=O)n1 c1(CN(C(C)CCO)Cc2ccccc2)nc2cnccc2s1 N1(Cc2c(O)ncc(Cl)c2)CC=C(c2ccc3c(c2)OCCO3)CC1 c1(CC2(C(=O)OCC(=O)OCCC)CC2)ccc(Cl)cc1 c1(C(=O)NC(COCC)C(=O)N(C2CCOC2)C)ccncc1Cl CC(C)CC(C)CC(=O)N1CCC2CCCC12C(=O)NC(c1ncc[nH]1)CO C1CC2(C1)CN(C(C1CC1C1CCCO1)=O)C2.C1(CCC=C)(C=O)CCCC1.N Cc1ccc(Br)c(F)c1C(=O)NC1CCCC1NC(c1ccncn1)=O c1(C(N2C(CCN(C)C(C3CC=CCO3)=O)CCCC2)=O)nnc(O)cc1O C(c1ccc(C#N)cc1)=CC(=O)NCC1CC(NC(C)=O)C1(C)C C(=O)(CC(F)(F)C(F)(F)F)N.c1(C(C)(F)F)cccc(C(N2CCC2C)=O)n1 Cc1nnc(CC(=O)NCC2CC2CNC(=O)COC2CCC2)s1 C1(C=O)OC(C)(C)OC1(C)C.C12(C(N(C)CC)=O)CC=CCN1CCC2.CC.O CON(C(=O)C1CCN(C(c2csnc2Cl)=O)CC1(C)C)C1CCCC1 c1(C(N2CCC(CNCc3ccc(C(=O)O)cn3)C2)=O)ccc(Cl)c(Cl)c1 C1(NC(CCN(CCCCOC)C)=O)C2CC1N(C(c1cc(C(C)C)[nH]n1)=O)C2 Cc1[nH]nc(C(=O)NC2CCN(CCCNC(=O)CS(N)(=O)=O)C2)c1C N1(C(C2(C)N(C)CCC2)=O)CC2=C(C1)CN(C(=O)C=Cc1c(F)cccc1F)C2 C1(CNC(c2nc(CCC)oc2)=O)CCC(C)N(C(c2cn(C)nc2Cl)=O)C1 c1(NC(=O)NCC)ccc(CC)nc1.C(=O)C(C)CNCC.CCO.N C1(CC)CC(c2nnnn2C2CCOCC2)(NCc2ccno2)CCO1 Cc1cc(=O)c(C(N2CCOCC(F)(CNC(=O)Cn3cccn3)C2)=O)cn1C CC1(C)C(NC(C2C3CCCCC23)=O)CCN1C(=O)CNC=O C1(C(=O)NC(CC=C)C)(CNC(=O)C=CC2CCCN2C)CCCCC1 c1(CNC(C(CC)NC(C)=O)=O)cnn2c1CN(C(c1cc(C)ns1)=O)CC2 c1(NC(C2(NC(c3ccc(C)nn3)=O)CSC2)=O)c(C)ccn(C)c1=O c1(C(N(CC(C)CNC(c2ccc([N+](=O)[O-])s2)=O)C)=O)scc2c1OCCO2 C(=O)CS(=O)(=O)C1CC1.c1(C(=O)N)cccc(C(F)(F)F)c1F.C=C(C)CC C1(C(=O)NCCC(C)N(C(C=C(C)Cl)=O)C)CCCSC1 C1(CNC(c2c(CCC)n[nH]c2)=O)CC2CCC1N2C(=O)CC.C1CCCC1.O C(=O)(CS(=O)(=O)C1CC1)NC1CN(C(c2cn(C(C)C)nc2)=O)CC1CO C1(NC(c2c(C)nncc2)=O)CCN(C(=O)COCCN(C)C)CC1F c1(CN(C(=O)CC2CCCCO2)CC)cccc(OC)c1.C(=O)(C(O)CF)O C1(C(=O)OC)CCOCC1C(=O)Nc1oc(C)nc1C C(=O)(C1=NN(C)C(=O)CC1)N(C(CC(F)F)C(=O)NCc1cnc[nH]1)C C1(NC(C(n2cc(C(N3CCOC3=O)(C)C)nn2)C)=O)CCC(C)(CO)CC1 N1(CC(=O)N)CCNC(=O)C1.c1(OC)cc(CNC(C2CCC2)=O)on1 C(=O)(CCCC(=O)OCC)N(C(C)C(=O)NCCC1(CO)CCC1)CCC c1(C(N(C2CCN(C(C(CC)C)=O)C2)C)=O)cccc(C(F)F)c1F N1(C(c2nnc(C(C)(C)C)s2)=O)CCC(CNC(c2ccoc2)=O)C(F)(F)C1 C1(C)(CNC(C(CC#C)O)=O)CCN(C(=O)COc2ccc(F)cn2)CC1 C1(NC(c2ccc(C(C)C)s2)=O)CCC(F)(CNC(=O)C(C)CF)C1 C1(C(N2C(C(=O)NCC3CC=CC3)C=CCC2)=O)CC2OC1C1CC21 N1(C(c2cnc(COC)s2)=O)CCC2CN(C(c3cc(F)n(C)n3)=O)CC2CC1 c1(C(=O)NC2CCN(C(C(C#N)C3CC3)=O)CC2O)c[nH]c2nccc(Cl)c12 c1(CC(=O)NC2C3CN(C(C4C(C)CCC4)=O)C2C3)ccc2c(cnn2C)c1 C(=O)(C(CC(C)C)N(C)C)N(C1CCCC1)CCNC(CCC=C=C)=O C1(CC)(CC)CC(NC(C2CCS(=O)(=O)C2)=O)CN1C(c1ccnnc1)=O Cc1cnc(C(=O)NC2(C3CN(C(C4CCOC4)=O)C3)CC2)c(F)c1 c1(C(=O)OCC)cccc(S(=O)(=O)N2CCC(O)CC(C)C2)c1 N1(C(Cc2c(C)occ2)=O)CCN(C(C2(CC3CC3)CCC2)=O)CC(O)C1 C1(CNC(CCC2(C)CC2)=O)N(C(C2CCCC2C(F)F)=O)CCCC1(C)C C(=O)(CC(O)CN(C)C)N(CCCNC(=O)C=Cc1cncs1)C(C)C c1(C(C)(C)C)ncsc1C(=O)NCCC1CC1.c1(CCC=O)ccccc1.C c1(CCC(N2C(CO)CC(NC(C3CCCSC3)=O)C2)=O)ccc(Cl)c(Cl)c1 N1(C(c2nc(=N)[nH]cc2)=O)C2CC=C(C(=O)C(=O)NOC#N)C1CC2 CC1(Cn2cc(CSCCNc3cccc4ccnn34)nn2)CCCCC1(F)F C1(NC(C2(CC)CCCO2)=O)CN(C(c2ccc[n+]([O-])c2)=O)CC1CO c1(C(N(CCN(C(c2cncc(C)n2)=O)C(C)C)C)=O)cnnc(C)c1C C1(C(N2CC3(CCOC3)C2)=O)CC2(CCN(C(C3(O)CCOCC3)=O)CC2)C1 C1(NC(C2(CSC)CC2)=O)CC(C)CN(C(C2(C)CCNC2=O)=O)C1 C(C)(C(C)C(=O)NOC(C)(C)CO)NC(C(C=C)(C)C)=O N1(C(c2c(OC)n[nH]c2)=O)CCC2C(CCCN2C(=O)CC2CS(=O)(=O)C2)C1 N1(C(COCCOC)=O)CCC(O)C(N(C(=O)CC(C)C)C)C1 C1(NC(c2c(C)nc(CC)s2)=O)CCN(C(=O)C(F)C(C)C)CCC1(F)F N1(CC)CC(C)N(C(C2(NC(c3cnccc3C#N)=O)CCC2)=O)CC1C c1(CCN2CCC(c3nc(C(C)C)cc(C)n3)CC2)ccccc1S(C)(=O)=O C1(O)(CC)CCCN(C(c2ccc(F)c(C)c2)C(=O)NC(C)C(=O)OC)C1 C1(NC(c2c(CC)non2)=O)CCC2(CCN(C(c3cc(C)c[nH]3)=O)C2)C1 N1(C(C(C=CC)O)=O)CCCC(NC(c2cnn(CCCC)c2C2CC2)=O)C1C Cc1nsc(C(=O)NC2CCCC(NC(=O)C(C)Cc3ccccc3)C2)c1N C(C(C)(C)CC(=O)N(C)CC1(CO)CCC1)NC(C(C(C)C)SC)=O C1(O)(CNC(CCCc2scc(C)n2)=O)CCCN(C(=O)C=Cc2ccco2)C1 N1(C(Cc2c(C)ncs2)=O)CCCC(N(C(=O)C(C)(C)N(S(C)(=O)=O)C)C)CC1 Cc1cc(Br)cc(C(=O)NC2CN(C(c3cnco3)=O)CC(F)(F)C2)c1O C1(N(C(CCCc2onc(C)n2)=O)C)CN(C(C2CC2C(C)(C)C)=O)CC1(C)C c1(OC)ncc(C(N2CC(OCC(=O)NCC(C)(C)COC)C2)=O)s1 C(=O)(CCC(C(C)C)NC(=O)CNC(N)=O)N1CCCCC(COC)C1 C1(NC(c2n(C)ncc2Cl)=O)CC(N=c2ccnc(C(F)(F)F)[nH]2)C12CCC2 C(=O)(C(C)(CO)NC(=O)CN(C1CCC1)C)NCc1c(C)nsc1 CC(CS(C)(=O)=O)C(=O)NC1CCN(C(c2ccc(N)c(Cl)n2)=O)CC1O C=C1CC(C(=O)NC2CC(CN(C)C(C3(SC)CCC3)=O)C2)C1 C(c1cccc(Cl)c1Cl)=C(C)C(=O)NCC1CN(C(=O)CC2(O)CCCOC2)C1 C1(NC(=O)COC2CC=CC2)CCCCC1.c1(CC=O)nc(C2CC2)cs1.N CC12CC(C(=O)OCC(N3CCOCC3)=O)(CCO1)C2 N1(C(C(=O)N(C(C)C)CCN(C(=O)Cc2ccon2)C)C)CCOC1=O C12(C(N3CC(CNC(COC)=O)OCC3)=O)CCCN1S(=O)(=O)CC2 N1(C(C2CN(C(CNC(C)=O)=O)CC2F)=O)CCc2c(cnn2C)C1 C1(CNC(C(C)n2cccn2)=O)CCN(C(C2CCCC2O)=O)C1(C)C Cc1ncc2ccc(NC(=O)CC3CC4(CCC4)CO3)cn12 N1(C(C2CC2c2ccsc2)=O)CC(NC(C2CC2)=O)C(c2ccccc2)C1.C N1(C(N2CCC(c3ccccc3)(C(C)=O)C2)=O)CC(=O)Nc2c(C)cc(C)nc21 Cc1cc(C(=O)NCC(CNC(C2CCNC2=O)=O)C(F)(F)F)cc(C)c1O CCCC(C)C(=O)NCC1(C)CCCCC1.C1(C=O)CCCN1C(=O)C1CC1 c1(SCC)nc(C)c(CC(=O)NC2CCCCC2)s1.N1(CC=O)CCCC1.C c1(OC)cccc(C)c1C(N1CC(NC(c2ccc(Cl)nc2O)=O)CC(C)C1)=O N1(c2nc(C)nc3c2scc3)CCC2(CN(C(c3cc(=O)cco3)=O)CCO2)C1 C(=O)(CC(F)(F)C(F)F)N1CCCC(C(C)NC(COCC(=O)OC)=O)C1 Cc1nn(C)c(C(N2CC(NC(C3CCOC3C(F)(F)F)=O)C(F)C2)=O)c1Cl CCC(CC(=O)N1CCCC1C)C(C)(C)C.C12(C(=O)N)CC(C(C)C)(CO1)C2 CC1(C#CC(=O)NC2CCCCC2NC(=O)C2=CCCCC2)CCCO1 C1(C(=O)NNC(=O)c2c[nH]nc2COC)CC(CO)N(Cc2ccccc2)C1 C1(C2CCOCC2)(C(N(C(CNC(CNC(=O)OC)=O)C)C)=O)CC1 c1(C(N2CCC(O)(CCNC(C3CC(CC)C3)=O)C2)=O)ccc(OC)cc1N CCC(C)C(C)C(=O)NCCOCCNC(=O)CCC.c1ccc(F)cc1F.O C1(F)(C(=O)NCC2CN(C(C)C)C2)CN(C(C2CC=CCO2)=O)C1 C(C(COC)CC(=O)N1CCC(F)C(NC(C2CC2F)=O)C1)OC c1(C(=O)NCC(C)CNC(=O)C)cccc(=S)n1O.c1ccccc1.CC.O C(=O)(C(C(C)C)c1cnn(C)c1)NC(CCNC(c1nc(C(C)C)oc1)=O)C c1(SC)nc(C(=O)NC2CCN(C(=O)CC(=O)O)C(C)C2)c2ccccn12 C1(CNC(c2n(C)cnc2)=O)CN(C(C23CCCC2OCC3)=O)CCC12CCC2 C1(NC(CNC(CNC(CCOC(CC(C)C)C)=O)=O)=O)CC1C1CC1C C(C(C)(C)CC(=O)NCC1CC(F)(F)CN1C(=O)CCO)OC.CC(F)F c1(CCC(=O)NC2CCC(C)C2)cncc(F)c1.c1(C=O)c[nH]c(C(F)F)c1.N C(=O)C(CC)C(C)(F)F.C1CCOC1.CCCCOC(=O)C=CC(=O)N.C C1(NC(c2cc(C)oc2C(F)(F)F)=O)CCC(C)(NC(=O)C(C)(F)F)CC1 Cc1cnn(C)c1C(C)NC(c1ccc(Br)s1)C C(=O)(CCN(OC)C(=O)C(C)O)N(CCCOC)C N1(C(c2nc(C)n(C)n2)=O)CCN(C(c2cnc(C(C)(C)C)[nH]2)=O)C(C2CC2)C1 C1(CNC(COC)=O)CCN(C(=O)CN2CCN(C)C(=O)C2=O)CCC1(F)F N1(S(C)(=O)=O)CCCC1C=O.C1(F)CN(C(=O)C=CC)C1.C(C)(C)C CC(C)(C)C(CNC(c1cnn[nH]1)=O)C(=O)NCC1CC2CCC(C1)C2 c1(CC(N2CCC2)=O)coc2ccccc12.c1(CS(C)(=O)=O)nc(C=O)cs1.N C1(NC(c2ccc(C(C)=O)[nH]2)=O)COC2(CCN(C(=O)CC)CC2)C1.C(C)C.O N1(C(C(COC)(C)C)=O)CCC(C(=O)N(C)CC2CCCS2)C(C)(C)C1 C1(C(C)NC(c2ccc(COC)o2)=O)CCCCN1C(c1cc(Cl)ccn1)=O N1(C(C(C)CC2CCCCC2)=O)CC2CCN(C(C3CCCO3)=O)CC2C1 n1(CC(=O)NC(C(C)NC(C)=O)C)ncc2ccccc2c1=O c1(CN2C(C)CC(C)CC2C)ccccc1S(=O)(=O)c1ccccc1 c1(-c2cn(CC(CNC(=O)Cn3cccnc3=O)OC)nn2)cccc(Cl)c1Cl C1(C(=O)NCC(C)N(C)C)CCC(c2cc[nH]n2)O1 c1(C(=O)NC(C)CN(C)C(C2(N(C)C)CCC2)=O)ncc(N)cc1Cl CC(O)(CC(=O)NC1CCOCC1NC(C1CCC2CC1CO2)=O)C(F)(F)F N1(C(C(C)NC(C)=O)=O)CCCCC2(CCN(C(C3CC3C)=O)C2)C1.C(C)C.O C1(C(=O)NCCC(C)(F)F)CN(C(=O)C(F)(F)C2CC2)CC1C1CC1 Cc1noc(C)c1CN(C)C(c1ccccc1-c1nncn1C)=O Cc1cccc2oc(C(N3CC(O)CC3CNC(c3ccncc3F)=O)=O)cc12 c1(C(N2CCCC(C(=O)Nc3c(C)nc[nH]3)C2)=O)c(C)nc2ccc(F)cn12 c1(NC(CN(C(=O)C(C)c2ccco2)CC#C)=O)ncoc1C1CC1 CC1(C)CCC(CNC(C2CCSC2)=O)CC1.C1(C(=O)N)CCC2(CCCC2)C1 O=C(C1=CC2(CCOC2)C1)NC1CC2(CCN(C(=O)CC3CCCCC3O)C2)C1 C1(C(=O)NCC2(CO)CCN(C(C(COC)OC)=O)CC2)CCOC2(CCC2)C1 Cc1cc(F)c(C(=O)NCC(C2CCN(C(c3csc(C)n3)=O)CC2)C)c(F)c1 c1(-c2n(CC)c(N(C)CC3(C)CCCO3)nn2)ccc(C)c([N+](=O)[O-])c1 c1(N2CC3C(N(C)C)C3C2)nccc(=NCC2CCC=CO2)[nH]1 CCCC(C#N)C(=O)NC1C=CC(CC(=O)NC(CO)CCF)C1 C1(CC)CCN(C(=O)CCC(C)CC)C(C(=O)NCc2cncc(Cl)c2)C1 Cc1cccc(F)c1CC(=O)NCC(CC(C)C)NC(C1OCCC1C)=O C1(O)(C(C)NC(CC=CCNC(C=NOC)=O)=O)CCCCC1 C1(CNC(C(C)CN(C)C)=O)CCN(C(C2CCC3(CC2)N=N3)=O)CC1C [SH](=O)(=O)c1cn(C)cn1.Cc1conc1CC(=O)NC1CCCC1.C(=O)(C)N N1(C(C2(CC)CCCC2O)=O)CCN(C(c2ccc(C)c(N)c2)=O)CC12CCC2 C1(CC(=O)N(CCNC(=O)CCC2CCOC2)CC)OCCOC1(C)C Cc1nc(N(C2CC(N)C2)C(c2ccc(C(C)(C)C)nc2)=O)c2c(n1)CCC2 c1(SC)ccc(C(=O)NC2CCN(C(=O)Cn3ccnc3C)CC2)c(Cl)c1 N1(C(C(c2ccc(C)cc2)C)=O)CCC(O)C(C(=O)NCCF)C1 CC(C(=O)N1CCC(CCO)CC1)C(C)NC(=O)CC1CC2C=CC1C2 c1(C(N2CCC(N(CCC)C(C3CC=CCC3)=O)C2)=O)cc2ccncc2o1 c1(CC(=O)NCC(C2CC2)NC(c2ccc(Br)o2)=O)noc2ccc(F)cc12 CC1CCN(C(c2cn(C)nc2C2CC2)=O)C1c1cn(-c2ccnc(F)c2)nn1 C12(C(N(CC(C)C)CC)=O)CC(C)(CN1C(=O)C(O)CSC)C2 C1(CC(=O)NCCC2COCC2O)CCCCC1NC(C1CNC(=O)C1)=O Cc1ncc(C(=O)NCC2(C=O)CC(C)(C)C2)c(=N)[nH]1.C1CCCCCC1C.N c1(C(N2CCN(C(C(CC=C)C)=O)CC2CC(F)F)=O)ccnc2c1ccn2C C1(C(=O)NC(C)(C)C(N)=O)CC(F)CN1Cc1cnc(Br)s1 O=C(CC(O)C1CCCC1)NC(CNC(C12CC(F)(C1)C2)=O)C1CC1 c1(C(=O)NC2CCN(C(c3c(C)ccc(OC)c3)=O)CC2)ccc(Cl)c(Cl)c1N S(=O)(=O)(c1ccccc1F)N1C(C(N(CC(=O)NC)CCC)=O)CC(O)C1 C1(CC)CN(C(C2(C(=O)N(C)C)CC2)=O)CCN1C(=O)CC(C)(C)CC C1(OC)CCC(C)(C(=O)NCCC(C)N(C)C(c2ncccn2)=O)CC1 N1(C(C(C)(C)n2cnnn2)=O)CC2C(CC(=O)NC)C2C1.C1C(C)(C)C1(F)F c1(CC(=O)N(C)CCN(C)C(c2ccn(CC#N)n2)=O)nc(C2CC2)nn1C C1(C2(NC(C3CC3(C)C)=O)CC2)(OC)CCC1.c1(C=O)ccc(F)cc1F.N C#Cc1cccc(C(=O)NCC(C)(C)NC(=O)CCCCC=O)c1Cl.C(C)(C)C.O C1(C(=O)NCC(C(N2CC(CC#C)OCC2)=O)O)CCC(=O)C(C)C1 C1(C(=O)NCC2CC(NC(C(C)NC(c3cccs3)=O)=O)C2)CCSCC1 C1(NC(N(C2CCN(C)C2)C)=O)CCc2c[nH]nc2C1 c1(C(=O)NCC2COCCN(C(CCCCCC)=O)C2)cc2sccc2cn1 C1(OCc2n(C)ncc2)CCN(N2CCC(CC#N)C2)CC1 c1(OC)ccc2[nH]c(-c3nccn3Cc3ccoc3)cc2c1 C(=O)(C1=C(Cl)CCOC1)NC1CCCC(CNC(C2C(C)C2)=O)C1 c1(CNC(C2C(NC(C3C(C=C)CC3)=O)C2)=O)ccccc1SC c1(C(C)OCC)nc(CC(=O)NC(c2ccccn2)Cc2ccccc2)cs1 c1(C(=O)NCCN(C(C2C(=C)CC2)=O)Cc2ccccc2)cccc(Cl)n1 C12(NC(C3C(C)C3)=O)CC(CNC(c3sccc3F)=O)(C1)OC2C C1(NC(c2c(C)c[nH]n2)=O)CCCCC1.c1(C(=O)N)cccc(CS(C)(=O)=O)c1 Cc1c(C(N2CCN(C(=O)CCC(C)CN(C)C)CC2)=O)cccc1Cl Cc1ccc(C(=O)NCCC2COCCN2C(C2COC(=O)O2)=O)cc1C C(=O)(C1=C(Cl)CCCC1)N1CCC(C)(NC(c2ncc(NC)nc2)=O)C1 Cc1cc(C(C)C)ccc1C(=O)NCC1(C)CCN(C(=O)CCC(C)(F)F)C1 N1(C(C2CN(C(C)=O)C2)=O)CCC(O)C1.N1(CCC(=O)N(C)C)CCC(F)C1 C1(F)(CNC(=O)CC(O)c2cccnc2)CCCN(c2ncc(Br)cn2)C1 c1(OC)ccccc1Oc1ccccc1C(=O)NCC(C)NC(=O)CSC N1(C(c2nc(C(C)C)oc2)=O)CCC2(CC1)CC2NC(=O)CCn1cnnn1 C1(NC(CC2(OC)CCC2)=O)C2CC(O)C1N(C(=O)C(C)S)C2.c1nncn1C Cc1ccc(C(=O)NCCC23CCC2CN(C(=O)CC2(C)CCC2)C3)c(N)c1 c1(C(N2CCC(c3cn(Cc4c(C)c[nH]n4)nn3)C2)=O)cc(F)c(F)c(F)c1 C(=O)C#CC1CCOCC1.C1(NC(C2C(C(=O)OC)C=C2)=O)CC2CCC1C2.N C(CC(CC)(CC)NC(=O)CCc1ccn(C)n1)NC(Cc1c(CC)con1)=O c1(CC)cc(=NCC2CN(C(c3cc(Cl)on3)=O)CCO2)[nH]cn1 N1(C(C2(C#N)CC23CCC3)=O)CC2(C1)CN(C(=O)COC1CCOC1)CCO2 CC(C)C(F)(CNC(=O)C(O)c1ccsc1)C(=O)N1CC(C)(CO)C1 c1(C2CC(C(N(CCCN(C(C=CCCC(C)C)=O)C)C)=O)C2)ccc(Cl)cc1 NC(=O)CCCC(=O)N1CCCC(NC(C2CCN(c3nncs3)CC2)=O)C1 N1(C(CN2CCN(C)CC2)=O)CCCC2CCN(C(=O)C3=CSCS3)CC12 N1(C(CN(CCC#C)C)=O)CC(CNC(=O)C)C(F)(F)C1.c1ccccn1.S N1(C(C2(OC)CCSC2)=O)CCC(C(CO)NC(=O)C(F)CC2CCC2)CC1 N1(C(C2C(C)OCC2)=O)CCCN(C(N(c2cc(O)cc(O)n2)C)=O)CC1 Cc1c(C(=O)NC(CCNC(=O)C(C)(C)CF)C(C)C)c2ccccc2n1C c1(OC)ccc(CCC(=O)NC2CC(F)CN(C(C3CC(C)=NO3)=O)C2)cc1F c1(C(=O)NC2C(NC(c3c(C)cc(=N)[nH]c3)=O)C2)cc2c(F)cccc2[nH]1 C(=O)(C#CC1CCOCC1)N1CC(F)(CNC(=O)CC2CCSCC2)C1 C1(NC(c2nc(C#C)sc2)=O)CC2CCC1N(C(c1ccncn1)=O)C2 C1(NC(c2ccc(SCCC)cc2)=O)CC2CC(NC(=O)C)C1C2.C(C)C C(=O)(C(O)CC(C)(C)C)N1CCCCC1.C1(CC(=O)NCC)CCC(C)(C)O1 C1CN(C(=O)CCS(C)(=O)=O)CCC1C(F)(F)F.c1(OC)n[nH]cc1C(=O)N Cc1nc(C(N2CCC(N(C(=O)C(O)Cc3cnn(C)c3)C)CC2)=O)c(C)n1C c1(C(N2C(C)CN(C(C3CC(OC)C3)=O)C(C)C2)=O)cc2nc[nH]c2cc1F CCC(C(=O)N1CCCC(CN(C(=O)C=C2CCOCC2)CC)C1)C(F)(F)F C(CN=C(NCCF)N1CCN(c2ccc3c(c2)CCC3)CC1)c1c(C)nn(C)c1 c1(C(N2CC(CC(=O)Nc3cnccc3C(=O)O)C2)=O)c(Br)ccnc1Cl N1(C(C(C)N(C(=O)Cc2ccsn2)C2CC2)=O)CC(F)(CO)C1 C1(CNC(C(C)=C2CCC2)=O)CCCN(C(c2cnc(N)c(CO)c2)=O)CC1 C1(C(N2C3C(NC(CCC4CC(C)C4)=O)CC(C3)C2)=O)CCN(S(N)(=O)=O)CC1 c1(C(N(CCN(C(c2cnco2)=O)C)C(C)C)=O)ccc(C)cc1C.CC=O C1(C(N(CC(CN(C(c2c(CC)cccn2)=O)C)O)C)=O)CCC(C)(C)C1.S c1(CC)ccc([N+](=O)[O-])cc1N1CCN(C(=O)C(C)CN(C)C)CC1 C1(C(=O)NCC(C(C)C)NC(C2(C)CCCC2C)=O)Cc2ccccc2N1C c1(SC)cc(Br)ccc1C(=O)NC1(C)CC(NC(=O)CCc2cnc[nH]2)C1 c1(SC)nc(N2CCCC(C)C2C)cc(C(F)F)n1.c1(CC=O)cnc(C)o1.N Cn1cnc([N+](=O)[O-])c1C(=O)NC1CN(Cc2ncccc2Cl)CC1(F)F C1(CC)CN(C(C2CCCN(C(=O)O)C2)=O)CCN1C(=O)C.C(=O)C1CC1 c1(N(CC(C)NC(c2cn(CC3(C)COC3)nn2)=O)C)nc(Cl)ncc1Cl c1(C(=O)NC(CC=C)CNC(=O)CC2CCC2OC)cc(OC)c(Cl)s1 C(N=c1[nH]c2c(C)cc(C)cc2s1)C1C(C)CCN(C(c2n(C=C)ncc2)=O)C1 Cc1cc(C(=O)NCC2CN(C(C3CCC(C)NC3=O)=O)C2)nnc1O C1(C(=O)NCCC2(NC(C(COC)OC)=O)CCCC2)CCC(C)=C(C)C1 N1(C(C(=O)Nc2c(C)cccc2)CC2CCOC2)CCC2(CCCCO2)C1 N1(C(CCCOC)=O)CCN(C(=O)C(C)(F)CC2CCCC2)CC1C1CC1 C1(NC(c2c(CC)oc(C)c2)=O)CCN(C(C2CCN(CC)CC2)=O)CC1CO C1(NC(C(C)NC(=O)NC)=O)CC2CN(C(c3cc(SC)ccc3C)=O)CC12 C(=O)(CC(CC(C)C)NC(c1ccn(C)c1-c1ccccc1)=O)OC C(=O)(N1CC(C)(O)CO1)C1(CC)CCN(C(=O)Cc2ccon2)C1 C1(C)(NC(=O)NC2C(C(=O)NCC)CCCC2)C2CC3CC(C2)CC1C3 c1(C(=O)NC(C=CC(=O)NC(CCC)C)(C)C)cnc(O)cc1C C(=O)(CCC(=O)NCC1(O)CCN(C(c2cc(-c3ccccn3)ns2)=O)C1)NC Nc1c(C(N2C3CCC2C(CNC(=O)C(F)OC(F)(F)F)C3)=O)cccc1Cl C=CC(C)(O)CC(=O)NC(CNC(=O)CCc1cc(C)[nH]n1)C1CCC1 c1(CC)nnc(C)cc1C(N1CCC(C)CC1)=O.C(=O)C(F)(F)C1(O)CCC1.N C(=O)(CCC(C)NC(C1CC12CC2)=O)N(C(C)C(F)F)C N(C1CCc2cc(CNC(c3ncn(C)n3)=O)ccc21)C(c1nc(C)n(C)n1)=O Cc1cc(C(=O)N(CCNC(=O)CC(C)(C)C)Cc2ccccc2)cn1C C1(NC(c2c(C)nn(CC)c2C)=O)CC2CC(C1)N(C(C1CCC(O)C1)=O)C2 CC1(C)CC(NC(=O)CCc2ccc(F)cc2)CN(c2cnc(F)cn2)C1 c1(C=O)cc2n(n1)CC1(CC1)C2.N1(C(C2(COC)CC2)=O)CCCCC1.O N1(C(=O)CCc2ccco2)CCC2CN(C(C34CC5CC(CC3C5)C4)=O)CC2C1 CC1CN(C(C2(n3nccn3)CC2)=O)C1.c1(C=O)cc(-c2csc(=N)[nH]2)c[nH]1.N N1(C(c2ccc(C)nn2)=O)CCCCCCC1C(=O)NOCC(O)C(C)(C)C c1(C(=O)NCC(CCOC)N)c(F)cc(C(=O)OC)cc1F C(c1c(Cl)cccc1Cl)=CC(=O)NC1CC(NC(c2ncc(C)cc2F)=O)C1 c1(CC)ccc([N+](=O)[O-])cc1C(=O)N(CCCC)C.C(=O)CC(C)P(C)(C)=O.N C(=O)(N1OC2CCC1CC2)N1C(C)CCC(C(=O)NC2CN(C)CC(C)O2)C1 c1(OC)cncnc1C(=O)N(C1CCN(C(=O)CCN2CCNC(=O)C2)C1)C c1(C(N2C(C(C)C)CN(C(C3(O)CC3)=O)CC2)=O)coc2cc(O)ccc12 C(CO)(CCCCNC(=O)C(c1ccc(Cl)cc1)=O)NC(C1(CC)CCOC1)=O C(=O)(C(O)CC(F)(F)F)NC1CC(NC(c2cc(Br)no2)=O)C(O)C1 Cc1c(C(=O)NCC2CC2NC(c2n[nH]cc2F)=O)nnn1-c1ccccc1 C(=O)(CCCC(C)NC(=O)CN=[N+]=[N-])NCC(C)CCCO N1(C(Cn2ccc(C)n2)=O)CCSCC1CCNC(c1cnn(C(C)C)c1Cl)=O C1(CNC(C(C)SCCCC)=O)(CO)CCN(C(C2(OC)CCCOC2)=O)C1 C(C(C(=O)NCCCc1ccccc1)C(C)(C)C)NC(CCC=C=C)=O C1(CC)CN(C(C2CC23CC(NC(=O)C#CC2CCC2)C3)=O)CCCO1 c1(CCC(=O)N(C(CCNC(C(C)CC2CC2)=O)C)C)ccc(Br)cn1 Cc1ccc(C(CNC(C2CCCCC2O)=O)NC(C2CC(=O)N(C)C2)=O)cc1 C1(CC)CC(C(=O)NC2(CNC(C3CCCN3C)=O)CC2)CCC1=O c1ccc(C(F)(F)F)cc1.N1(CCN(C(=O)C(=O)NC)CC)CCCCC1 O=C1CCC(CC(=O)N2CCOC(Cn3cc(CO)nn3)C2)c2ccccc21 CCC(CC)CC(=O)N(C(C)CNC(=O)COc1ccc(Br)cc1Cl)C c1(C(N2CCC(CC)C2)=O)cc(F)cc([N+](=O)[O-])c1.C1(C=O)CCS1(=O)=O.N C1(OC)CN(C(c2ccccc2)=O)CCC1NC(c1c[nH]c(C)c1)=O n1(CC)cnc2c(NC(c3cncs3)C)[nH]c(=NC3CCC4(CCCC4)C3)nc12 CC1CC(CNC(=O)CCCCN2CCCC2)CN1C(=O)Cn1cnccc1=O C1(N(C)C(=O)NCc2ccn(CC(F)(F)F)n2)CC(CC(N)=O)C12CCC2 c1(C(N2CCCC(CCNC(CC3(C=C)CCC3)=O)C2)=O)cc(C)nc(O)n1 CCCCC(O)CC(=O)NC1CCN(C(=O)CCC(=O)N2CCOCC2)C(C)C1 N1(C(CC)=O)CCCC2(NC(c3nc(Cl)ccc3F)=O)CCCC12 CCC(N=c1cc(NC(c2cn(C)cn2)C)nc(C(C)C)[nH]1)c1ccccc1F c1(OC)cc(OC)c2c(=O)c(C(=O)Nc3ccc(OC(F)F)nc3)c[nH]c2c1 c1(OC)ccc(F)c(C(N2CC(NC(=O)C(c3ccc(F)c(F)c3)O)C2)=O)n1 N1(C(C(c2cccnc2)NC(C(CC)C#N)=O)=O)CC(C)=CC(C)C1 C1(C)(C(N(CC(CN(C(c2cn(C)cc2)=O)C)O)C)=O)CCC(C)(C)CC1.CC c1(C(N2CC(O)(CNC(c3ccon3)=O)C2)=O)cccc(O)c1.[nH]1cccn1 c1(C(=O)NC2CN(C(C3CC4C=CC3CC4)=O)CCC2O)ccn2cnnc2c1 N1(C(C2(NC(CC(CC)CN(C)C)=O)CCSC2)=O)CCC(O)C(C)(O)C1 Cc1nc(CN2CCC(C(=O)N(CCO)Cc3ccccc3)CC2)sc1C c1(C(=O)NCC2CC(OC)CN2C(c2csc(Cl)n2)=O)ccc2c(n1)CCC2 c1(C(N2C3C(NC(=O)CSCC(F)(F)F)CC(C3)C2)=O)[nH]nc2ncnc(O)c12 C12(NC(C3N(C)CCOC3)=O)CCCC1(F)CN(C(=O)Cc1sc(O)nc1O)C2 C(=O)(C1=CCCSC1)NCCCCN(C(c1nc(OCC)oc1)=O)C N1(C(CC2N(CC)CCC2)=O)CCC2(CCC2)C(C)C1.n1(CC(=O)N)nccn1 CCC(CC)(CCNC(c1ccn(C)c(=O)c1)=O)NC(C1COCCO1)=O CCC(C(=O)NC(C)CC1CN(C(=O)CC2CC(=O)NC2=O)C1)C(C)(C)CC CC(CO)C(=O)NCCC1(NC(c2coc(N(C)C)n2)=O)CC1 CCCCCC(=O)N1CCC(NC(=O)CNC(=O)OC(C)(C)C)C(CO)C1 c1(C2N(C(c3cncnc3C)C(=O)NC)CCC2)ccc(OC)nc1 C(CC(C)(C)CNC(=O)C(=Cc1cccs1)C)NC(CN(CC)CC)=O C1(NC(C(COC)NC(=O)C=C(C)c2ccco2)=O)CC(C)N(C)CC1C C#Cc1cccc(CNC(=O)CC(CC2CC2)NC(C2CCC(CC)O2)=O)c1 c1(C(=O)N)nc(Cl)c(Cl)c(N)c1Cl.C1(C(N2CCCC2)=O)(CC)CC(C)(C)C1 c1(C(N2CC(CC(C)NC(C=CCCC)=O)C2)=O)ccc(C2CCOCC2)cc1 c1(C(N2CC(O)CC(NC(c3n(C)c(C#N)cc3)=O)C2)=O)ccc2ccsc2c1 N1(C(CC(=O)OC(C)(C)C)=O)CCC(C2CCCN(C(=O)C=C(Cl)Cl)C2)C1 C1(C(CNC(C=CCC)=O)F)CCN(C(c2cc(F)n[nH]2)=O)CC1 Cc1nc2c(s1)CC(C(=O)NCC(C)(C)NC(=O)Cc1nnc(O)s1)CC2 N1(C(Cc2ccc(C)nc2)=O)CCC(C)C(NC(=O)OC(C)(C)C)C1C NC1CCOC1COCc1nn[nH]c1C1CC1.C1CN1 C(=O)(CC(C)(C)C)NCc1nnc(CC)s1.C12(C(=O)N)CCC(CC1F)C2 Cc1noc(C(F)(F)F)c1C(=O)NCCCC.c1(C=O)ccn(CC(F)F)n1.N CC1CN(C(=O)OC(C)(C)C)CCC1N(C)C(c1cccc(C2COC2)c1)=O C=C=CC(C)C(=O)NC(COCC)C(=O)NC(C12CCC(CO1)C2)C C1(C(=O)NCc2c(C)n[nH]c2)Cc2nnc(C)n2C1 C1(CC(=O)N(C2CN(C(C)C)C2)C)CC(F)CN1C(C1CC12CCCC2)=O CN1C(=O)COc2cccc(NC(=O)C(=O)NC3CCc4cnn(C)c4C3)c21 C(=O)(C1=NN(CCO)C(=O)CC1)N(CCN(C(c1c(C)oc(C)c1C)=O)C)C C1(C(N2CCCC(C)(NC(CC3C(C)CCC3)=O)C2)=O)CCC(C2CC2)CC1 N1(C(C(C2CCCCC2)C)=O)C(C(N2Cc3c[nH]nc3C2)=O)C2CC(O)C1C2 c1(C(C)=O)cc(C(N2CCC2C)=O)oc1C.c1(C=O)ccc(C(=O)CF)cc1.N C1(C(=O)NCCc2onc(CC)n2)CC2(CCC2)C1.C1(CC=O)CCCC1O CC1(C2CC2C(=O)NCc2cncc(C(N3CCOC(C#N)C3)=O)c2)COC1 Cc1oc(C#N)cc1C(N1CC=CC1(C)C(=O)NCC1(N(C)C)CC1)=O n1(C(C)C)nccc1C(N1CC(C)(NC(=O)C(F)CC2CCCC2)C1)=O c1(C(=O)NC(C(C)NC(c2c(C)cc(N)cc2)=O)C)cc(Cl)c2[nH]c(O)nc2c1 C(=O)(C(F)(F)C(O)C1CC1)NC(C1CCN(C(=O)CC=O)CC1)(C)C.C1CC1 c1(OC)cc(N2CC(NC(c3ncsc3C)=O)C2)nc(OC)n1 Cc1oc(C(=O)NCC2COC(CNC(C3(C)CCC3)=O)C2)cc1Br c1(C(=O)N)cccc2ccc(C)nc12.C(=O)(CC1(C)CC1)N(C(C)C)CC C(C)(CO)(C=O)NC(CCNC(=O)OCC)=O.C(CC1CC1)CC(C)C C1(NC(c2cnc(CCC)s2)=O)CN(C(c2ccncc2Cl)=O)CC1(C)C Cc1cc(C(N2CCCCC2)=O)nc(N(C)C)n1.C(=O)(C=CCN(C)C)NC N1(C(c2ncn(C)n2)=O)CCC(C)(NC(=O)CC2CCCCCO2)C1 n1(CC)nnc2c1C(C(=O)N1CCCC(C)(F)C1)CN(C(c1cccs1)=O)C2 C(c1cc(F)c(F)c(F)c1)=CC(N1CC(NC(c2cc(Cl)cs2)=O)C1)=O c1(CC(C)NC(N2CCS(=O)(=O)CC2)=O)ccc2ccccc2c1 N1(C(CCCOC)=O)CCC(C2(O)CCN(C(c3cccc(C)c3O)=O)C2)CC1 c1(OC)ccc(N2CCN(Cc3ccc(OC(C)C)nc3)CC2)c(OC)c1 C(=O)(C1CCCn2cnnc21)NCC(C)(C1CC1)NC(c1cc(Cl)on1)=O CC(C)C(C(=O)N(C)CC1CC(F)C1)NC(c1cnn[nH]1)=O C1(C(=O)O)CC(=O)N(CC)C1.C(CCCCOC)NC(c1ccccc1)C1CCC1 Cc1ccccc1SCC(=O)N(C)C.C1CCN(C(C2CC2C(F)(F)F)=O)C1 c1(C(=O)OC)nc[nH]c(=NCC(CNC(C2CCC(C)O2)=O)C(F)(F)F)c1O Cc1cn2c(n1)CCC(C(=O)OCc1cccc(C#N)n1)C2 C(=O)(C1CCCc2sccc21)NC1CC2(CC(NC(c3cscn3)=O)C2)C1 C1(COC)CN(C(=O)CC)C1.C1(CC=O)CCC(=O)N1.C1(C=O)CCC1 C1(C(=O)NCC2(OC)CN(C(=O)C(C(C)C)SC)C2)CCOC2(CCC2)C1 C1(C(N2CCCC(NC(CN=S(C)(C)=O)=O)C(F)C2)=O)CCC2(CC1)OCCO2 C1(CNC(c2cncc(CC)c2)=O)CCCC12CCN(C(=O)C(O)CSC)CC2 C=CCC(C(=O)N)NC(=O)OC(C)(C)C.C1CCCN(C(=O)C(C)CC)C1 CCC(C)CC(C(=O)O)OC(=O)CNc1cccc(C(F)(F)F)c1 C1(F)(C(=O)NC2CC(CNC(c3ncc(OC)nc3)=O)C2)CCCN(C)C1 c1(C(=O)NCC(O)CCNC(=O)C(F)C2CCC2)n[nH]c(C2CC2)c1Br c1(OC)ccc(F)c(CC(=O)NCCCNC(c2ncoc2-c2ccco2)=O)c1 N1(C(C(CC2CCOCC2)NC(CC2(C)CC2)=O)=O)CCC2(CCC(O)C2)C1 CCC(CC(=O)NC1CCC1NC(=O)C(C)(C)OC)CC(F)(F)F C1(O)(CC(N2CC(CNC(CCC=CC)=O)C(C)C2)=O)COC(C)(C)C1 N1(C(c2c(C)nsc2)=O)CC2CCCC2(NC(c2ccc(F)c(C(F)F)n2)=O)C1 CCC(CC(=O)NCc1ccc(C(N2C3CCC2CC(OC)C3)=O)cn1)C(C)C C=CCC(C)(O)C(=O)NCc1cc(C(N2CCCCCC2C)=O)cs1 N1(C(C(=Cc2cccnc2)C)=O)CCC(C)C(NC(=O)COC)C1.c1nccs1 c1(C(C(=O)NCC2(O)CC(C(N3CCCCC3)=O)C2)=O)cc(F)c(F)cc1F S(=O)(=O)(c1cccnc1NCCCCO)N1C(C)CC(C)C1 C(=O)(CCCCCN=[N+]=[N-])NC1C(C)(C)C1C(N1CCC(O)(C(N)=O)C1)=O c1(C(=O)NCCCNC(c2coc(-c3ccccc3)c2)=O)ccc(F)c(O)c1 c1(OC)ccc(S(=O)(=O)NC2CCN(C(c3cc(Cl)cc(Cl)n3)=O)CC2)cc1Br C1(N(C(CCN(CCCCOC)C)=O)C)CCCC(N(C(=O)CCC(N)=O)C)C1 N1(C(C2CCN(C)C2=O)=O)CCCC2C1CCN2C(c1ccc2occc2c1)=O N1(C(CSCCOC)=O)CCCC12CCCN(C(c1cc(C3CC3)ncn1)=O)C2 c1(C(=O)NCCC2CN(C(c3ccncc3)=O)C2)cc2cccnn2c1 N1(C(C2C(C)N(C)CC2)=O)CC23CCCCC2(C1)CN(C(=O)C#CC1CCC1)C3 N1(C(C2CCC(C)O2)=O)CCCCC12CN(C(c1cn3c(n1)SCC3)=O)C2 C(=O)(C(C)(C)CC(=O)N1CCCC1CCNC(C1CCC(C)(C)CC1)=O)OC Cc1sc(-c2nc[nH]n2)nc1C(=O)NCC1COCC1NC(=O)C(C)C C(c1cc(Br)ccc1OC)=CC(=O)NC(CNC(C(C(=O)OC)C)=O)CO Cn1nnc(C(N2CCC(F)(CNC(C3CCCS3)=O)C2)=O)c1N n1(CC)c(C(=O)NC(C2(O)CCN(C(=O)CN(C)C)C2)C)cnc1O C1(C(N2CCCC2)=O)C2C3CC4C1C1C2CC3C41.C1(CC)CC1C(=O)NC N1(C(c2c(OC)cncc2)=O)CCN(C(=O)CN2CCC2)CC(C)C1.C(C)=O.O N1(C(CNc2ccc(C)cc2)=O)CCCC(O)(C)C1.C(c1cc[nH]n1)=CC(=O)N C1(CCNC(=O)Cc2csnn2)CCCN(C(=O)Cc2ccnn2C2CCC2)C1 CC(C)CCC(=O)N(CCCNC(=O)C(C)(C)C1(O)CCOC1)C.C1CCCC1 c1(C(N2CCN(C(C)=O)CC2)=O)ccc(Cl)c([N+](=O)[O-])c1.C=C1CC1C(=O)N C1(C(=O)NC(C)C(CO)NC(=O)C(C)(C)C2CCCCC2)CCC(N(C)C)CC1 C(=O)(CC1CCCc2ccccc21)N1C(CNC(=O)C=CBr)CC1 Cc1nc(=N)[nH]cc1C(=O)NC1CC(F)(C)C1.c1(C2C(C=O)C2)ccsc1 C(=O)(C(C)(C)CC(F)F)N1CCC(CCNC(C(C2CCOC2)OC)=O)CC1 c1(C23CC(C2)C3)cccc(F)c1F.Cc1cc(CCC(=O)N2CCC2)n[nH]1 C(=O)(C(CC)(CC)CC)NC(CCCC)CNC(c1c(O)cccc1O)=O C1(CC=C)(NC(c2cc(F)n[nH]2)=O)CCCN(C(c2ccnc(C)c2C)=O)C1 c1(NC(=O)N=c2cc[nH][nH]2)cc(Cl)nc2ncccc12 C(=O)(CC(c1ccccc1)c1ncc[nH]1)NC(C)CNC(=O)Cc1ccno1 c1(CC(N2CCC(NC(C(CC)SC)=O)C2)=O)ccc(OC)cc1OC C#Cc1cn(C)nc1C(=O)NC1CCCC1C(=O)NCC(C)(Cl)CC C1COC2(C1)CN(C(=O)C=CC(=O)NC)C2.CCC=O.C1(C=O)CCCC1 N1(C(C(C(C)C)SC)=O)CC2OCC(NC(c3ccc(C(F)F)cc3)=O)C2C1 C1(CNC(C2C(C(C)C)C2)=O)CCCCN1C(=O)CCOc1ccccc1Cl c1(C(N2CC(OCCNC(C3C(C=C)CC3)=O)C2)=O)ccnc2ccc(O)cc12 CC1CN(C(c2ccc(F)c(Br)n2)C(=O)NCCN2CCOCC2)CC(=O)N1 N1(C(Cc2c(C)non2)=O)CCN(C(=O)Cc2csc(S)n2)C(C)C1C CC1CCN(C(c2cc(CO)n(C)n2)=O)CCN1C(C1CC(=O)N(C)C1)=O n1(CC)c(CN2CC(C)N(C(C)=O)CC2C)nc2c(F)cccc12 N1(C(C(CCN(C)C)NC(C(CC)C)=O)=O)CCN2CCC1CC2 C1(C2CN(C(C3(C)CC=CC3)=O)C2)CN(C(=O)CCN2CCOC2=O)CCO1 c1(CC(=O)N(C2CN(C(C3CC34CC4(F)F)=O)C2)C)cc2ccccc2cc1O N1(C(CCOCC)=O)CCC(COC)(NC(C2CCCC(C)(C)C2)=O)CC1 c1(C(C(=O)O)NC(=O)C(n2cc(Br)cn2)F)ccc(O)nc1 C1(OCC)(OCC)CC(C)(C(=O)NCCCC)C1.c1(C=O)ccn(C)c1 C(N=c1[nH]c2c(c(=NCCCn3cnnc3)[nH]1)CCC2)c1cnc(O)[nH]1 N1(C(CCC(CC)=O)=O)CC2CCN(C(C3(COC)CC3)=O)CCC2C1 c1(OC)ccc2c(c1)CC(NC(C1CC3OC(C)CC3N1)=O)CCC2 C1(NC(C(C)Cc2ccccn2)=O)CCC(C(N2CC3CC3C2)=O)CC1 Cc1ccc(C(=O)NC(C)C(C)NC(=O)Cc2cc(C)[nH]n2)c(O)c1 N1(C(CCn2c(C)cc(C)n2)=O)CCC2(C1)CN(c1cc(Cl)c(O)nn1)C2 Cc1nc(CNC(=O)CN2CCCC2)oc1C(N1CCCC1CCCO)=O C(=O)(C1=CC2(CN(C(C3CCCC(CF)C3)=O)C2)OC1)N(C)CC1CCCOC1 Cc1ccc(CC(=O)NC(C)CCN(C(=O)C(C)(Cl)Cl)C)c(C)c1 c1(C(N(CCN(C(CCCCCOC)=O)C)C)=O)cccc(NC)c1[N+](=O)[O-] c1(OC)ccc(C(=O)NC2CCOCC2NC(C2CCCCO2)=O)cc1C1CC1 C1(CNC(=O)NCC2(COC)CCC2)CCC2CCCCC2C1 C1CCN(C(=O)CN(C(=O)C(C)C)C)CC1C(C)C.Cc1ncccc1C=O.N Nc1nc(Cl)cc(Cl)c1C(N1CC2=C(C1)CN(C(c1ccc([N+](=O)[O-])[nH]1)=O)C2)=O C12(CNC(C(C)N3CCC3)=O)CC(CN1C(C1CCCN1C1CC1)=O)C2 c1(OCC)ccc(C(=O)NC2CC(COC)C2)cc1.c1(C2CC2)cccs1 C1(C)(NC(c2ccc(CC)[nH]2)=O)CCN(C(c2cn(C)nc2C2CC2)=O)CC1 c1(CC(=O)N)nc([N+](=O)[O-])n[nH]1.CC(C)CCCNC(C1(Cl)CC1(F)F)=O C1(NC(N2CCCC(C)(C(=O)OCC)C2)=O)CN2CCC1(C)CC2 C1(C(N2CCN(C(C(C)N(C(C)=O)C)=O)CC2)=O)CCCC2(CCOCC2)O1 Cc1ccnn1CC(=O)NCc1occc1C(=O)NC(C)(C)CC1CCC1 c1(C(N(C)CC2CCCN2C(c2cscn2)=O)=O)cc(F)c(O)c(Cl)c1 CC1CC(C(=O)NC(C(=O)N(C(C)C(C)(C)O)C)C2(O)CCC2)CC(=O)N1 Cc1cnc(N)c(C(=O)NC2CCCCC2N(C(=O)C(c2cncnc2)C)C)c1 N1(C(c2[nH]cc(C)c2)=O)CCC2CC2(NC(=O)CCCS(N)(=O)=O)CC1 c1(C(N2C3(CN(C(c4ccon4)=O)C3)CC2)=O)cn2ccccc2n1.CCSC CC(=O)CCCC(=O)N1CC(N(C)C(C2C3CN(CC(F)(F)F)CC23)=O)C(F)C1 C1(F)(CNC(CN(C)C)=O)CCCN(C(c2cccc(Br)c2F)=O)C1 Cc1nc(C)c(C(=O)NC(C2CN(C(=O)C=Cc3cc[nH]n3)C2)C)c(C)n1 c1(C(=O)NCC2(F)CCN(C(CCC3C(C)C3)=O)C2)cc2c(F)cccc2[nH]1 N1(CCNC(C2(OCC)CCC2)=O)CCCCC1.c1(C(=O)N)coc(Cl)c1 c1(CC(=O)NC(CNC(c2ncoc2Br)=O)CO)cc(F)ccc1F C(C)(CO)(C(=O)N(CC(F)F)Cc1nccc(C2CC2)n1)OC c1(C(=O)NCC2N(C(c3cccc(SC)n3)=O)CC2)c(O)ccc(Cl)c1O N1(C(C(CC(N)=O)O)=O)CCCCCC(NC(c2ncccc2Cl)=O)C1 N1(C(CC(=O)NC)=O)CC(C)OC2(CCN(C(c3ccnc(C)c3)=O)C2)C1 c1nc2c(s1)CCCC2=O.c1(OC)ncc(Cl)cc1C(N1CC(C)(C(=O)N)C1)=O Cc1cnc(C(N2CC3(CCN3C(=O)CC(C)C3CC3)C2)=O)c(Br)c1 CC(CNC(=O)CCc1nncn1C)CC(=O)N1CCSCC1CO C1(CNC(C=CCC)=O)C(C2CC2)CCN1C(=O)Cc1sc(C)nc1C N1(C(C=CC(C)=O)=O)CC2CCC1C(NC(=O)C(O)C(C)c1ccccc1F)C2 N1(C(=O)C(F)Cc2ccccc2)CCN(C(=O)Cc2sccc2Cl)C(C2CC2)C1 C(CCCCC(=O)N1CCC(C)C1CNC(c1ccsc1C(F)F)=O)OCC c1(OC)cc(N=[N+]=[N-])ccc1NC(N1CCCC(N(C)C)C1)=O C1(C)(CNC(C2(F)C(C)C2)=O)CCC(NC(c2coc(CO)c2)=O)CC1 CCC(CNC(C1CC=CCC1)=O)(CC)C(=O)NC(C)(C)CCCO Cc1c(C(N2CCN(C(C3CCC3)=O)CC2CC#N)=O)cccc1F c1(C(N(CCNC(c2ccc(CN3CCCC3)o2)=O)CC)=O)ccoc1C C1(C(=O)NCc2c[nH]nc2C(=O)NOCC2CCCO2)CCCOCC1 C#CC1CCCN1C(=O)C(=O)N(CC1CCC1)CC1CC1 c1(C(N(CCCOCCNC(C)=O)C)=O)ccc(-n2cnnn2)c(C)c1 C1(NC(c2c(C)cccc2)=O)CC2(C1)CC(NC(=O)CCS)C2.c1nccn1C C1(CNC(c2cccc(-c3nc(NC)c(N)s3)c2)=O)NC(=O)OC1(C)C c1(NC(Cc2ccc(OC)cc2)=O)ccc(C2=CCCCC2C)nc1 C1(C(N(C)Cc2ncc(C)o2)=O)CCC(C)CN1C(=O)CSC(F)F Cc1cc(O)c(C(N2CCC(n3ccnn3)C2)=O)cc1F CC1=C(C(=O)NCC(F)C)S(=O)(=O)CCO1.c1(C(C=O)=O)ccc(C)cc1.N CCCC(C)(O)CC(=O)NCC(C)(C)CN(C)C(c1coc(CO)c1)=O CCC(C)CCCC(=O)NCC1(OC)CCN(C(C2CCN(OC)CC2)=O)CC1 N1(C(C2(C3N(C(c4c(C)con4)=O)CCC3)CC2)=O)CCCN(C2CC2)CC1 C(CCNC(=O)N(C)C)(C(F)(F)F)OC.C1CCC(=O)N1 N1(C(=O)CCC2CCN(C(=O)CCCC3CCCC3)C2)CCc2ccncc2C1 C(C(C)(C(=O)NC1C(C)CCC1C)NC(=O)CCC1CCC(=O)C1)SC c1(C(=O)NC(C(C)NC(c2ccnc(C)n2)=O)CO)ccc(S(=O)C(C)C)cc1 CC1(C)CC(C(=O)NC2CN(C(=O)Cn3cc(CO)nn3)C2)CC(C)(C)O1 CC(c1ccccc1)=CC(N1CC(O)CC1CNC(c1nc(O)sc1C)=O)=O N1(C(c2cc(OC)nn2C)=O)CCC2(CC2C(=O)NCC)C1.CC(F)F.O N1(C(Cc2c(C)nsc2)=O)CCOC(C(=O)NCC2(C(N)=O)CC2)C1 Cc1ncc(C(=O)NCc2ccccc2)c(=N)[nH]1.C1(C=O)CC(=O)N(O)C1.C N(C(=NCCN1CCCOC1=O)NC1CS(=O)(=O)c2ccccc21)C(C=C)C N1(C(CCCOCC=C)=O)CCC(C)(C(N2CC(C(C)(C)C#N)C2)=O)C1 C(c1ccc(F)c(F)c1)=CC=O.N1(C(C2CN(C(C)C)C2)=O)CCCC(F)C1.N CN1CCOc2ccc(C(N3CC(OCCNC(=O)C(C)(C)F)C3)=O)cc21 N1(C(CSCCC#N)=O)CC2CC(NC(C34CCCC3OCC4)=O)CC2C1 Cc1cc(Cl)c(C(=O)NC2CCN(C(C3(O)CCC(C)CC3)=O)C2)cc1[N+](=O)[O-] C1(C(=O)NC2CCC(C#C)C2)CCN(C(c2ccc(CO)o2)=O)C(C)C1 c1(OC)ccc(NC(=O)CCCC(C)NC(c2ncsc2C)=O)c(C)c1 c1(C(=O)NCCC(C)NC(=O)CC2CCCO2)cc2cnccc2cc1F N1(C(Cc2c(C)ccc(F)c2)=O)CC2=C(C1)CN(C(C1CN3CCC1CC3)=O)C2 C(=O)(CCCCNC=O)OC(C)(C)C.C12CC1CN(C(c1nc[nH]n1)=O)C2.N CC1(CNC(=O)Cn2cnnn2)CN(C(=O)CCCCc2cnc[nH]2)CCO1 N1(C(C(CC)(C)CNC(C2CCOC2(C)C)=O)=O)CCC2(CC1)CSC2 c1(C(=O)NC(CC(C)NC(=O)CC2COCCOC2)C)cnc(C(F)(F)F)nc1 Cc1cc(C(=O)NC2CN(C(=O)C(C)CF)C2)nc(C(F)F)n1 C1(NC(c2cc(N(C)C)ncc2)=O)CC(NC(c2cscn2)=O)C12CCC2 c1(C(C)C)nc2cccc(C(=O)NC3(C)CCC3)c2[nH]1.C1(C(=O)N)CCC1(C)C C1(C(C)C)CN(C(=O)CSCCC#N)CCCN1C(=O)C(=O)N(C)C C1(C(=O)NC2CCOCC2NC(C2COC(=O)O2)=O)(OC)CCCCCCC1 c1(CCC(N2C(C)CC2C(=O)NCCC(O)C(C)C)=O)cc(F)ccc1Br c1(C(=O)NC(CCNC(CC(C)c2cnn(C)c2)=O)(C)C)cc(CO)ccc1Cl C1(C(=O)NC(C(=O)OC)c2cccs2)CC(=O)N(c2ccc(SC)cc2)C1 N1(C(C(CC)Oc2cccc(C)c2)=O)C2CCC1CN(C(C1OCCOC1C)=O)C2 CC(C)C(CNC(C1(C)CCCC1C)=O)N=c1[nH]cnc2cnn(C)c12 N1(C(C2(N(C)C)CC2)=O)CCCC(NC(C2=NC=C2c2ccccc2F)=O)C1 c1(C2C(NC(=O)NCC3CC=CCC3)C2)c(Cl)cccc1Cl CCC(F)(F)C(=O)NCC(C1CC1)N(C)C(c1ccc(N2CCOCC2)cc1)=O N1(C(C2(NC(c3cn(C)nc3)=O)CC2)=O)CCCC(CC2CCC(C)(C)C2)C1 N1(C(C2CC(C)OCC2)C(=O)NC2CCCC2)CCCCC1C#N.C1CC1 N1(C(C(C=C)O)=O)CCC(CN2CCN(C(=O)CCN(C)CCC)CC2)CC1 n1(CC(=O)N(C2CCCC2)C)ccc(=O)c2ccccc12.C(=O)(C(C)(C)C#N)N c1(N(C(CNC(C(C(C)C)F)=O)C)C)nc(C(F)(F)F)c2ncnc-2[nH]1 c1(C(C=Cc2nnc(CC)o2)=O)cc(OC)c(OC)c(C(N2CCCCC2)=O)c1 C(CCC(C)C)(C(=O)N1CC(C)=CC(C)C1)NC(c1c(CC)nn[nH]1)=O C=CCC(C(=O)NCc1ccc(C(=O)NC(C)(C)C2CC2)cc1)C(C)C.O C1(C(=O)NC2CN(C(C3(C(F)F)CC3)=O)C2)OCCCC1c1ccccc1 C12CCCC1(F)CN(C(C1(C(C)C)CC1)=O)C2.C(CC(C)(C)C)(C(=O)N)OC C1(NC(c2c(C)nn(C)c2)=O)CCCCN(C(c2cccc(Cl)c2F)=O)C1 N1(C(CN(C)CC)=O)CC2OCCN(C(=O)CN3CCS(=O)(=O)CC3)C2C1 c1(C(N2CCC(NC(=O)CC(F)(F)C(F)F)C23CC3)=O)cc(Cl)c2c(c1)OCCO2 c1(COC)ccnc(C(=O)N(CC(O)C)C)c1.c1(CCC=O)ccc(N)cn1.N c1(NC(=O)CC2CN(C(c3ccncn3)=O)C2)c(Cl)cc(Br)c(Cl)c1Br S(=O)(=O)(c1ccc(Cl)c([N+](=O)[O-])c1)NC1CC(NC(c2ccc(C)cn2)=O)C1 Cc1nn(C)c(Cl)c1CC(=O)NC1CCCN(C(c2cc(N)cc(N)c2)=O)CC1 c1(C(=O)NC2C(CNC(C3(C=C)CCCCC3)=O)C2)[nH]c2ccccc2c1C C#Cc1ccnc(C(=O)NCC(F)CNC(C2CCN(CC(C)C)CC2)=O)c1 Cc1ncc(F)c(=NCC2(NC(=O)C(C)CSc3ccccc3)CCOCC2)[nH]1 c1(NC(C2(C)CC2)C)ccc(S(=O)(=O)N2CCC(O)C2)cc1C#N C1(C=O)CC(=O)N(C(C)(C)C)C1.CC1=NOC(C(=O)N)C1.C12CC(C1)C2 C(=O)(CC(C)(C)C(F)(F)F)N1CC(C)C(CNC(=O)CO)CC1.c1nc[nH]n1 c1(C(NCCNC(C2CC3CC(=O)C2C3)=O)=O)cnn2c1N(C)CC2.CC C1(C(=O)NCCn2c(CC)ncc2)CCN(C(=O)CC2CC3CCC2C3)CC1 c1(CCC(=O)OCCN(C(C2CC2CC(C)C)=O)CC)cccc(F)c1 c1(OCC)ncc(C(N2CC3(CC3)CC2)=O)cc1Cl.N(S(N)(=O)=O)CC=O C#CCCCC(C)C(=O)NCC(C(=O)NC(C)Cc1nncn1C)N(C)C N1(C(C(C)n2cccn2)=O)CCC(S(=O)(=O)Cc2ccccc2)C1 N1(C(C2C(C(=O)OC)C=C2)=O)CCC1(C)CC(=O)NCCc1cc(C)no1 N#CCC(C(=O)N1CCN(C(C2CC2c2ccccc2)=O)CC1)c1ccccn1 c1(C(=O)NC2C(CNC(=O)CN3CCCS3(=O)=O)C2)cc2ccccc2s1 C1(NC(C2(NC(Cn3c(C)ncc3)=O)CCCC2C)=O)CC12CCCCCC2 Cc1ccc(N)c(C(=O)NCCC(O)C)c1.c1(C(=O)N)cc(C(F)(F)F)ncn1 Cc1cc(C(N2CC(F)(C)C2)=O)ccn1.C1(C=O)CCS(=O)(=O)N1.C1CC1 Cc1nn(C)c(C)c1C(=O)NCC1CN(C(=O)C(C)C(C)C)CC1C c1(OC)cccc(COC(C)C(=O)OC(c2ccccc2O)C)c1 Cc1cc(C(=O)NCC2(C)CCCN(C(c3c(Cl)csc3Cl)=O)C2)ncc1N Cn1cnc2[nH]c(=NC3C4CC3CN(C(=O)CC3CC5CCC3C5)C4)nc(O)c12 C1(OC)CCCC(CC(=O)NCC2CC(F)(F)C2)C1.C(=O)CCC1CC1.N N1(C(CCN(C)CC)=O)CC2CCCC2(NC(c2cc(F)ccc2N)=O)C1 Cc1ncsc1CCC(N1CC=CC1Cn1cc(-c2cnn(C)c2)nn1)=O Cc1ncc(S(N)(=O)=O)cc1C(=O)N.C(=O)(C(C)(O)CC(F)F)N1CCC1.C C1(C(F)(F)F)(C(=O)NCCC(Cn2cc(CC(C)O)nn2)F)OC2CCC1C2 Cc1ncc(C(=O)NC(C)C(C)(C)C)c(C)n1.c1(C(=O)N)ccc(O)c(Cl)n1 N1(C(CCCN(C)N=O)=O)CC2CCC(C1)N(C(=O)CN1CCN(C)C(=O)C1)C2 CC(c1ccccc1C)=CC(=O)NCC1=CCN(c2ncc(F)cn2)CC1 Cc1c[nH]c(NC(C2CCCC2NCc2ccc([N+](=O)[O-])o2)=O)c1C#N C1(NC(C2C(C#N)C2)=O)CCC2CCN(C(=O)CCc3cscn3)C12 C1(CNC(COCCC=C)=O)CN(C(=O)Cc2c(O)ncnc2O)CC1(F)C c1(OC)ccccc1CC(=O)NCC1(F)CCC1.C1(CC=O)COCCO1.C c1(C(=O)NCC2CC(NC(=O)CCN3CCC(F)C3)C2)cnc(O)c(Br)c1 C(N=c1c(C#N)c[nH]c2c(C)cccc12)C1OCC(CC)C1 C1(CCNC(C2CC2(Cl)Cl)=O)CCN(C(=O)CCc2cnc(C3CCC3)o2)C1 C1(OC)CCC(C(=O)NC2COCC2CNC(C2(CF)CC2)=O)C1 C(=O)(C(C)(C)CCCNC(=O)CN(CC(C)(C)C)C)NCCCCS(C)=O c1(C(N2CCC(N(C)C(C3CC34CC4)=O)CC2)=O)cc2n(c1)CCSC2 N1(C(C(CO)NC(C)=O)=O)CCC(S(C)(=O)=O)C1.c1(CC(=O)N)ccsc1 N1(CCc2ccc(F)c(Br)c2)CCNCC12CCCC2 Cc1cnc(C(C)CNC(=O)C(=O)NCc2ccnn2C2CC2(F)F)s1 c1(C=O)cc2c(F)c(F)ccc2[nH]1.CCC(C)(C)OCC(=O)NCC1CCC1 N1(c2ccc(C(=O)OC)cn2)CC(F)(F)CC1CNC(=O)C(C)C1CCOC1 c1(C=O)cccc(C)c1.C(CC(C)C)NC(C1CC(CCC)C1)=O.C(C)=O.N N1(C(CC2(OC)CCOCC2)=O)CCC(C)C(CNC(c2ccns2)=O)C1 N1(C(C(NOC)=O)=O)CC(NC(=O)C(N2CCOC2=O)C)CC12CCCC2 Cc1ccccc1CC(=O)NCC1(C)CCC(NC(=O)Cc2ccn(C)n2)C1 CC(C)C(C(=O)OCCC1CCCCCC1)c1ccccc1 c1(C(=O)NCC2C(NC(CCC=C(C)C)=O)C2)cnn2c(N)ccnc12 C1(NCc2c(C(=O)O)cccn2)CC12CCOCC2.C12CN(C1)C(=O)O2 C(=O)C1=NNC(=O)C1.Cc1cc(C)n(-c2ccc(C(=O)NC3CCC3)cc2)n1.N c1(C(=O)NC23CC(C)(C2)C3)cc(CNC(=O)CCc2ccccc2)ccn1 CCCCC(=O)N1CSCC1C(=O)NCCC(C)(C)NC(C1CCCC1)=O n1(CC(C)C)c(N(C2CCCSC2)CCF)nnc1-c1cccs1 n1(C(C)C)nnnc1C(c1ccc(Br)s1)NCC(C)(C)Oc1ccccc1 NS(=O)(=O)CCC(=O)N1CC2CC2(CNC(C2(CC#N)COC2)=O)C1 N1(C(C(C)CCC(C)(C)C)=O)CC2(C=C(C(=O)NC(c3ccnn3C)C)CO2)C1 N1(C(CC2CC(N(C)C)C2)=O)CC2COCC2(C(N2CCC(OC3CC3)C2)=O)C1 Cc1ccc(C(N2CCN(C(=O)CCc3ccn(C)n3)CC2C(F)F)=O)c(C)c1 C1(NC(CCc2onc(C)n2)=O)COCCN(C(c2cccnc2N(C)C)=O)C1 C(C(C)CC(=O)N1CCC(=CCNC(C2(CCN(C)C)CC2)=O)CC1)OC CC(C(=O)NC12CC1CN(C(c1cccc(N)c1F)=O)C2)C(C)(F)F c1(N(CCCC(F)(F)F)C)nc(=N)nc(N2CCN(Cc3cccn3C)CC2)[nH]1 C1(C(C#C)C)CCN(C(=O)C(C2CCN(C(C3(C)CCC3)=O)CC2)C)CC1 c1(CC(N2CC(CNC(CCSCCC)=O)OCCC2)=O)ccc(S(C)=O)cc1 C=CC(C)(O)CC(=O)N(C1CCC(NC(=O)CO)CC1)C.c1ccnc(O)c1.C Cc1ccnc(C(N2CCC(N(C(c3cc(C)c(Cl)s3)=O)CC3CC3)C2)=O)n1 c1(C(N(C)CCN(C)C(C2(C)CC(=O)C2)=O)=O)ccc(-c2ncc[nH]2)nc1 c1(C(=O)NCC2OCCN(C(CC)=O)C2)ccc(C)c(-c2ccccc2)c1 C=CCCCCC(O)CN1CCOCC1Cc1ccccc1 C=C=CC(C)C(=O)N(CCC(C)NC(=O)Cc1ccon1)C c1(CCC(=O)NCCN(C2CCCC2)C(=O)CN2CC3CC3C2)cnc(O)[nH]1 C1(CNC(CSCC)=O)CC2(CCC2)CN1C(C1CCN(CC)C1)=O c1ccccc1F.C(CC(=O)NCC(C1CCOC1)NC(=O)CO)OC(C)=O C(C(C)(O)C(C)(C)O)NC(=O)Nc1cn(C)nc1C1CCCCC1 Cc1cc(S(=O)(=O)O)ccc1NC(C1CCN(Cc2ccncc2Br)C1)=O c1(N2C(C(=O)NC3(CC)CCCCC3)CC(F)C2)cc(C(=O)OC)nc(Cl)n1 c1(CNC(C(=O)N(C)CC2CC=CCC2)=O)cccc(Cn2cccn2)c1 Cc1scc(C(=O)NC2CCN(C(=O)C(C3CCCCC3)C)C2C(C)(C)C)c1C N1(C(CC(=C=C)C)=O)CCCCC(C2CN(C(=O)COCC3CCOC3)C2)C1 N=c1[nH]c2ccc(C(N3CC4C(CNC(=O)CN5CCOCC5)C4C3)=O)cc2[nH]1 c1(C(N2C(CCNC(C(CCCC)O)=O)CCCC2)=O)ccc2nccnc2c1 c1(C(=O)NC(CCNC(c2c(C(C)C)con2)=O)C)cccc2c1C(=O)NC2=O C1(OC)(CNC(=O)C)CCCN(C=O)C1.C(C)(C)CC.C1(C=O)CC1C CC1CCCC1N(C)C(c1cn(CCNC(=O)CCOC2CC2)nn1)=O N1(C(COCc2onc(C)n2)=O)CCN(C(=O)C(=O)NCCO)CC12CCC2 C1(CC(N2CC(CN=[N+]=[N-])C2)=O)CC2(CC2)CN1C(C1CC12CCCCC2)=O CC1CC(C(=O)NCC=CC(=O)N(C)CC2CN(C)C2)CCC1=O n1(CC(C)C)c(NC(c2cncc(C#N)c2)=O)nc2ccccc12 Cc1n[nH]cc1C(=O)NC(Cc1cnc[nH]1)C(=O)N(C)Cc1nccs1 c1(C(=O)NC2CC(NC(C(C)C3CC3)=O)C2)cc(-c2ccccc2)nn1C c1(OCC#C)c(OC)cccc1CNC(C12CCC(CC1)C2)C1CC1 N1(C(C)=O)CC2CC(C)N(C(=O)Cc3c(C(F)(F)F)n[nH]c3C)C2C1 c1(NC(N(C)C)=O)ccc(C(=O)Nc2n[nH]c(-c3ccccc3)c2Br)cc1 CP(C)(=O)c1ccc(C(=O)NC2CCN(C(C3(C#N)CC3)=O)CC2CO)s1 N(C1CCc2cc(CNC(=O)C(C)CSC)ccc21)C(c1ccc(C=C)cc1)=O N1(C(COC(CC)(C)C)=O)CC2CCCC(C1)N(C(c1ccnc(C)c1C)=O)C2 N#CC1(C(N2CCC(NC(=O)C(F)CC3CCCCC3)CC2)=O)CC=CC1 c1(C(=O)NC2CC(N(C(=O)C(F)C3CC3)C)C2)ccnc(OC(F)F)c1 C1(C(N2CCCC(CO)C2)=O)CN(Cc2ccc(Cl)cc2)CC12CC2 N1(C(c2c(C)nc[nH]2)=O)CC2(CC2C(N2CC(O)CC2C(N)=O)=O)C1 CCCCCC(CC)C(=O)NCC1(NC(=O)CC(C(C)C)c2ccon2)CCC1 CC(C)C(O)C(=O)N1CCC(NC(C2CCC2c2nc[nH]n2)=O)C1 c1(CC)ncccc1C(=O)NCC1CCOC1C(=O)NCc1nccs1 C(=O)(C1=NOC2(CCOC2)C1)NC(C)CN(C)C(c1cccc([N+](=O)[O-])c1Cl)=O C1(C(=O)N)CCC(=O)C(C)C1(C)C.CC1CCCN(C(=O)CCCC2CC2)C1C c1(C=O)ncnc(C)c1C.CC1=NNC(=O)C1CC(=O)NCC1CC(F)C1.C Cc1cc(O)nc(C)c1C(N1CCC(N2CCN(C(C3(C)CC3Br)=O)CC2)C1)=O C(c1sc(Cl)nc1Cl)=CC=O.CC(C)(C)C(=O)N1CC(C(C)(C)O)(C)C1.N c1(C(CNC(=O)CC(C)SC)NC(c2cc(CCC)on2)=O)cccc(Cl)c1 CCCCC(C)CCC(=O)NC(CCF)C(=O)NCC(n1cccn1)C CCC(CC(=O)NC1(C(=O)NCCc2ncc(C)cn2)CCSC1)C(F)F c1(C(=O)NCC(C)NC(c2cccc(F)c2)=O)ccc(C(F)(F)F)c(O)n1 CC1(C#CC(=O)N2CCN(C(c3cccc(CF)c3)=O)CC2C(F)F)CC1 C(=O)(C1=C(Cl)CCOC1)NC(C(C(C)C)NC(Cn1c(C)cc(C)n1)=O)C C1(C(N(CCC(=O)N(C)Cc2cccs2)CCCO)=O)CC2(CC2)C1 n1(CC)cc(NCCN(CCC#N)C(C)=O)cn1.C1(=O)C(O)CN1 O=C(CCC[N+](=O)[O-])N1CCC(O)(CNC(=O)COc2ccccc2)C1 C(=O)(C#CC1CCCOC1)NC1C(C)(C)N(C(C2CN(C(N)=O)C2)=O)CC1 C1CN(C(=O)C(n2ccc(C)n2)C)CC1C(=O)N(C1COCC1O)C1CC1.CO Cc1n[nH]c(C)c1S(=O)(=O)N1CC2CC1CN2C(=O)Cc1ccccc1I C1(CC)C(C(=O)NCC2(C3CC3)CCC2)CCCN1C(=O)C(F)C(=O)O N1(C(=O)NC(c2cc3[nH]ccc3s2)CC)CC(N(C)C)C(C)(C)C1 C(=O)(C1=C(Cl)CCCC1)NC(C(C(C)C)NC(=O)CN(S(C)(=O)=O)C)C C12(NC(CC(C(=O)OC)C)=O)CCC(CC1)N(C(=O)CCC(N)=O)C2 Cc1cc(C(=O)NCCC(C)NC(=O)C(C)NC(C)(C)C)c(C)cc1Br Cc1ccc(C)c(NC(=O)NC2CN(C(c3ccc(CO)cc3)=O)CC2(F)F)c1 Cc1cc(N2CC(CCCCNC(c3[nH]nnc3C)=O)C2)ncn1 C1(C)(C(N2CCC(=CCNC(c3nnc(C)s3)=O)CC2)=O)CCCS1(=O)=O C#CC1CN(C(=O)C(CNC(C2C=CC=CC=C2)=O)C(C)C)CCN1C N1(C(C2CC(C)(C)C2)=O)CCC2C1CCCN2C(c1csc(S(N)(=O)=O)c1)=O c1(OC)ccc(OCC(O)CNC(C)C(=O)Nc2cc(Cl)ccc2Cl)c(C)c1 c1(C(=O)NCC(CCNC(C2OCC(C)(C)C2)=O)O)ccc(=O)n2c1CCCC2 C1(NC(C(COC)N(C)C)=O)CN(C(C2(n3nccn3)CC2)=O)CC1(C)C C1CCC12CN(C(c1ccc(C(F)(F)F)o1)=O)C2.c1(C=O)cc(O)nc(Cl)c1.N Cc1ccc(CNC(=O)CCSCCCC=O)cc1C.N12CCCOC(C1)NCC2 O=C1CCCCC(C(=O)NC2CC(OCC(=O)NCc3cncnc3)C2)C1 Cc1[nH]nc(C(=O)NCC(C)(C)OCC(=O)N(C(CCO)C(F)F)C)c1C N1(C(c2n(C(C)C)ncc2)=O)CCC(CCCCNC(C2CC(CF)C2)=O)CC1 Cc1ccc(CC(=O)NCC2(NC(c3cc(C#N)on3)=O)CCOC2)c(F)c1F C1(CO)CN(CC2(c3ncco3)CCC2)CCO1 C1(CNC(C(C)Oc2cccc(F)c2)=O)CC2CCC1N2C(C1(F)CCC1)=O Cc1oc(Br)cc1C(=O)NC1CCC(NC(C23CC(C2)C(C)O3)=O)C1 C1(CSCC(N2CC(CC(C)NC(c3cnc(S)[nH]3)=O)C2)=O)CCCCO1 c1(C(CC)NCc2cn(Cc3cccs3)nn2)cnc(C)cc1Cl CC(CC(F)F)C(=O)N1CCCC(N(C(=O)CCc2ccccc2Cl)CCO)C1 C(=O)(C1=C(C(C)C)N(C)C(=O)NC1c1ccc(C(F)(F)F)cc1C)OCC.O C1(OC(C)C(=O)NC2C3CC2N(C(C2CS(=O)(=O)C2)=O)C3)CCCCCC1 c1(CNC(CCNC(=O)OC)=O)cc(C(=O)NCCc2cnco2)no1 N1(C(c2cnc(CNS(C)(=O)=O)s2)=O)CCN(C(=O)CN2CCOCC2)CC1 C1(C(C)C)C(NC(C2CC3CCC2O3)=O)CCN1C(C12CC(CO)(C1)C2)=O c1(C(=O)NC2C3(CCN(C(C4CN(C)C4)=O)CC3)C2)ccnc2ccncc12 N1(CCCC(=O)NCCC(C)NC(C(C)Cc2ccccc2)=O)C(=O)CCC1=O c1(NCc2c3n(nc2)CC(C)CO3)cccc2c1OC(C)(C)CC2 C1(CNC(CC(C)=C(C)C)=O)CCN(C(C2(C(N)=O)CCC2)=O)CC1O N1(C(C(CC)OCC)=O)CC2C3CCC(C2C1)N(C(=O)CCOCC1CC1)C3 C(=O)(C#CC(C)C)N1C(C(N(CCC(=O)NC)C(C)C)=O)CC1C CCCCCCC(C)C(=O)NCC=CC(=O)N(C1CCOC1C)C1CC1 c1(C(=O)NCC(=O)NCC2CCC3(CCC3)O2)ccc2cncn2c1 c1(NCCN2CC(C3CN(C(C)=O)C3)C2)cc(=O)n(C)c(=O)n1C c1(N2CCOCC(CNC(C3(C)CC3)=O)C2)nc(C(F)F)nc2ccc(F)cc12 C1(C(=O)NC(C(=O)OCCC)C)CC12CCN(C(C1CN(C)CCO1)=O)CC2 Cc1nc2ccc(C(N3CCCC(CO)(NC(C4CCC4)=O)C3)=O)cc2s1 O=[N+]([O-])c1c(CNCC2Cc3ccccc3CO2)ccc2ccccc12 C(CN=c1[nH]c(OC)ncc1Cl)(CC(C)C)NC(C1(CC#C)CC1)=O C1(OC)CN(C(=O)CC2CCCN2C(c2n[nH]cc2Cl)=O)CC12CC2 CC(C)C(C)CCNC(=O)CCCOC(C)C.c1(CCC=O)ccc(=N)[nH]c1 Cc1c(F)ccc(N)c1C(=O)NCC(O)CN(C)C(c1cc(O)ncn1)=O Cc1nonc1CC(N1CC=CC1CNC(=O)C(C)NS(C)(=O)=O)=O N1(C(CN(CC#C)C(C2CNC(=O)C2)=O)=O)CCCCC1CF c1(C(=O)NCC(C)(O)CNC(=O)COC(F)F)cccc(CC#N)c1 C12(C(N3CC4C(C=O)C4C3)=O)CC(CN(C(=O)CN3CC4CC4C3)C1)C2.C Cc1nc(CC2CC2)oc1C(N1CC(C)CC1C)=O.C(c1ccc[nH]1)=CC=O C(=O)(CC1OCCc2ccsc21)NCC1(NC(c2nccc(N)c2)=O)CC1 c1(C(N2CCC(=CCNC(C3C(CC)C3)=O)CC2)=O)nn(C)c2c1COCC2 c1(CC(=O)N)ccnc(Cl)c1.c1(CC(=O)NC2CCC2)ccn(C2CCCC2)n1 N1(C(C=CC(=O)N(C)C)=O)CC2CC2(C(N2CC(CC3CC3)C2)=O)C1 c1(NC(COC(COC(CC)C)=O)=O)sccc1C(N)=O Cc1ccn(CC(=O)NC2CC(C)N(C(c3nnc(Cl)cc3N)=O)C2)c(=O)c1 CC1(C(=O)NCC2CCN2C2CCOCC2)CCS(=O)(=O)CC1 C1(NC(c2ccc(CO)o2)=O)CC2(C1)CN(C(C1(c3cc[nH]n3)CCC1)=O)C2 N1(C(C(C)OC)=O)CCCC(C)(NC(=O)CC2CC3CC3C2)C1 c1(CC)nsc(N(C)CCOCCNC(=O)CC(C)c2ccco2)n1 CC(CC1CC1)N=c1[nH]c(N(C)CC2CC2(C)C)nc(=N)[nH]1 N(C(=S)N1CCCc2c(Cl)cc(Cl)cc21)S(c1cccc(OC)c1)(=O)=O c1(C(=O)NCCCc2cn(-c3ccncc3F)nn2)cc2c(nc1Cl)CCSC2 Cc1cc(C(=O)NCC2CCN(C(=O)C(C)CC3CCC3)C2)ccc1Br C(=O)(C1c2ccccc2-c2ncccc21)N(CCNC(C1C2CCCC12)=O)CC Cc1cc(C(N2CC(O)(CC)C2)=O)ccc1S(C)(=O)=O.c1(C=O)cnc(Cl)[nH]1.N c1(CCC(N2CCC(O)(CC)C2)=O)ccc(F)c(F)c1.c1(C=O)coc(Cl)c1.N C1(C(N(C)CCc2ccccc2)=O)CC(C)(C)CCN1C(=O)CC1CCOC1=O c1(NC(C(CC2CCCC2)NC(CCC)=O)=O)cnc(OC)nc1 C(C(C)(C)CC(=O)NC1C=CC(CC(=O)NCC(O)C(=O)NC)C1)OC C(=O)(C1=CCC(F)(F)CC1)N1CCCC2(NC(CSC(C)(C)C)=O)C(C1)C2 c1(NC(CN(S(=O)(=O)c2ccccc2)C)=O)ccc(C#N)c(Cl)c1F C1(NC(CCN(C(C=CC=CC)=O)CCO)=O)CCCCC1.C1CCC1.C c1(C(=O)NCC(C(=O)NCCCc2nnnn2C)N(C)C)ccc(O)c(F)c1 C1(C(=O)NCC(C)NC(=O)C(C)C2CCCO2)(CC)COC1 CCCC(C(=O)N1CCOCC1CNC(c1scc(Br)c1C)=O)N(C)C c1(C(N2CC(C)C2)=O)cccc(S(=O)(=O)C2CC2)c1.c1(CC)ncoc1C=O C1(NC(C)=O)CCC(CC(N2CCC(NC(=O)Cn3cc(Cl)cn3)C2)=O)CC1 C1(C#N)(C(=O)NC2C(N(C(COc3cc(C)on3)=O)C)CCCC2)CCCOC1 c1(CN(C=O)Cc2cnc3n2CCC3)ccc(Cl)cc1F C1(NC(=O)NC(C)CCC(=O)OC(C)(C)C)CC[Si](C)(C)CC1 n1(CCc2nc(-c3cnccc3)nn2C2CC2)ncc2ccccc12 N1(C(c2nc(C)[nH]n2)C)CC(NC(c2cncs2)=O)CCC1C C1(C(C)C#N)CCN(C(C2(C)CCCN2C(c2ccc(Cl)cn2)=O)=O)CC1 C(c1nc2ccccc2o1)=CC(=O)NC(CNC(c1c(C)c[nH]n1)=O)CO CC1C(NC(=O)CC2C=CCCC2)CC2CCC1N2C(c1cc(F)ccc1O)=O C(=O)(C(CNC(c1sncc1C)=O)C(C)(C)C)N(C)Cc1ncc(C)nc1 C1(CC)C(NC(c2csc(NC(C)=O)n2)=O)CCN1C(=O)C(C)CF C1(NC(C(CN(CC)CC)F)=O)CC2CCCC(C1)N2C(=O)C=CBr N1(C(c2c[nH]c(=NC)o2)=O)CCC(N=[N+]=[N-])(C(=O)N(C)Cc2cc(=O)cc[nH]2)C1 C1(O)(CC(=O)NC23CC2CN(C(C2CCS(=O)(=O)CC2)=O)C3)CCCCCC1 C1(NC(C2(NC(c3c(C)cco3)=O)CCCC2C)=O)CC2CC3C(C2)C13 C(=O)(C1=NNC(=O)C1)N.n1(CCC)cncc1CNC(=O)CC1CCCC1 C(=O)(CCS(N)(=O)=O)NC(CCNC(CCSC)=O)C Cc1[nH]nc(C(=O)NC2CCC2NC(=O)CCC(C)N(C)C)c1C C1(C(=O)NC(CNC(C(C)(C)C2CC2)=O)(C)CO)CCC2(CCCC2)CC1 C(CC(C)(C)CC(=O)N1CCC(O)(CNC(C2(C#N)CC2(C)C)=O)C1)OC CC1=CC(C)CN(C(=O)CC2(NC(C3CCOCC3(C)C)=O)CC2)C1 c1(C(=O)NC(C(=O)NCc2nnn(CC)n2)CC2CCC2)ccccn1.C Cc1ncc(CC(=O)NC2CCCCC2NC(C23CCC(CC2)CC3)=O)c(O)n1 c1(NC(c2nncs2)C)cc(Br)ccc1S(=O)(=O)NCC1(C)CC=CCC1 c1(C(=O)NCC(C2CC2)NC(C(c2ccc(F)cc2F)C)=O)ccc(C#N)cn1 N=c1[nH]cnc2cc(C(=O)N)ccc12.C12CC(C1)C2.c1(C2C(C=O)C2)cn[nH]c1 Cc1nc(CC(C)C)oc1C(=O)NCC1(NC(C2CC2[N+](=O)[O-])=O)CC1 C(=O)(C1CSc2ccccc21)N1CCC2(CN(C(C(C(CC)O)(F)F)=O)C2)CC1 C(=O)(CCC(=O)NC1CCCCC1CNC(c1c(Br)n[nH]c1C)=O)NC C1(C)(C(N(CC(C)C)CC(=O)NC2C3CCCOC23)=O)CCOCC1 CC(C)CC(CC(C)C)NC(c1c(F)ccc(I)c1F)=O C=C1CCN(C(c2ncc(C)cc2F)=O)C(C(N2CCC(CC)CC2)=O)C1 N1(C(COC(CC)(C)C)=O)CCCC(C2CCN(C(=O)Cn3nnc(C)n3)C2)C1 CCC(CC(=O)N1CCCC(NC(=O)C(=O)Nc2ccccc2)C1)C1CCC1 CC1CCN(C(=O)CC2CN(C(c3cnc4cc[nH]c4c3)=O)C2)CC1(F)F N1(C(C(C)O)=O)CC2(C1)OC1(C)CC2(C(N)=O)C1.C1CCCC1.C(=O)(C)N c1(NCC)cccc(C(=O)NC2CC(C)N(C(C34CC5CC3C4C5)=O)C2)c1 Nc1c(C(N2CCC(NC(C3CCS3(=O)=O)=O)C23CCC3)=O)cc(Cl)cc1F c1(C(N2CCC(CNC(CCC(=C)Cl)=O)C2)=O)cc(C)nc2c(C)cccc12 C1(C(N(C2CCN(C(=O)C(C)CSC)C2)CC#C)=O)CCNC(=O)C1 C1(C(N2CC(NC(COCCC=C)=O)C3(C2)CC3)=O)CCc2nnc(O)cc2C1 N1(CC(=O)NCCC(C)(C)NC(=O)Cc2cccnc2N)CCCNC1=O c1(C(N(CCCN(C(CN(C)C(N)=O)=O)C)C)=O)cccc2ccn(C)c12 CCC(CNC(C1CC(C#N)C1)=O)(CC)NC(c1csc(C(F)F)n1)=O CC(C)CCC(=O)NCCN(C(c1nn(C(F)F)cc1Cl)=O)C(C)C C1(C(=O)NC(C)(C)CCNC(c2cnc(S)[nH]2)=O)CCCOCC1 C1(C(=O)NCCCCCN2CCN(C(C3C(C)CC3)=O)CC2)CCCC12CCC2 CC1=NOC(C(=O)NC(C)CC(C)NC(c2ncoc2-c2cnn(C)c2)=O)C1 C1(CC(=O)NC(CCOC)CO)CCN(C(=O)CCSC)C1(C)C C1(CC)C(C)CCCN1C(c1cc(C)cc(F)c1)=O.n1(CC)nncc1C(=O)N c1(C(=O)NC2CC(CNC(CCC#N)=O)C2)cc(F)c(Cl)cc1Cl C(c1c(C)noc1C)=CC(=O)NCCC1CCN(C(C2C(=C)CC2)=O)CC1 c1(-c2ccc(OCC(N3CCC(C)(C#N)C3)=O)cc2)cncc2cc[nH]c12 C1(CCNC(C(Cc2ncn(C)c2)O)=O)CCN(CC(F)(F)F)CC1 c1(C=O)c[nH]c2cccc(C)c12.n1(CCOC)cc(C(=O)NC2CCC2)nn1.N C1(C)(COC)CCN1C(=O)C=CCN(C(=O)CCc1cccn1C)C C(CCC(=O)NCCn1cnc(C(=O)N(C)Cc2cccnc2)c1)N(C(C)C)C c1(SC)cc(C(=O)N(C(c2ccccc2)C)C)ccn1.C1(C=O)CC(C)(F)C1.N C1(CNC(C(CC=CC)NC(c2cc(CCC)on2)=O)=O)CC12CCCCC2 n1(CC(=O)N)ccc(=O)n(C)c1=O.C=CC(F)(F)C(=O)N(CCC)C1CC1 C1(C(=O)NCCN(C)CC)CN(Cc2cc(C)sc2C)CCC1O c1(C(=O)NCCC(C)N(C(=O)CCOC2CCOCC2)C)c[nH]ccc1=N CC1CCCCN1C(=O)N(C1(CC(=O)NCC2(CC(N)=O)CC2)CC1)C C(=O)(C1=NOC(C)C1)N(C)CC1CCOC1.c1(C=O)ccc(C(N)=O)o1.N N1(C(CC#N)=O)CCC2C1CCCN2C(c1ccc(C#N)cc1Br)=O C1(NC(c2c(OC)c[nH]n2)=O)CCC12CN(C(=O)C(C(C)C)c1ccccc1)C2 C1(C=O)CCCCC1.C(C)(CC(=O)NCC=CC)OCC.c1ccccc1.N c1(C(=O)NCC2NCC3CCCC23)cccc2cc(O)ncc12 CC1CNc2c(C(N3CC(F)(CNC(=O)C(O)CC(C)(C)C)C3)=O)cnn2C1 N1(C(C(CC(C)C)OC)=O)CCC2(CCC2)C(C)C1.C(=O)(C(F)(F)C1CC1)N CC(=O)CCCCC(=O)NCC12CN(C(=O)C(F)CC3CCOC3)CC1CCO2 c1(C=O)cnccc1C(C)(C)C.CC(F)(F)F.C(CC)N(C(=O)C)CC.N C1(NC(C2(CC)CCN(C(=O)CC3CCOC3)C2)=O)CC2(C1)CC21CCC1 N1(C(C(C(C)C)SC)=O)CC2(CC(C(=O)NOCC(F)(F)F)CO2)C1 C=CC1OCCC1NC(=O)CN(C(=O)CCc1ncccn1)C1CC1 CC1(C(N2CCC(CCNC(c3c(F)cccc3F)=O)C2)=O)CC(C2CC2)=NO1 C1(C(=O)NCCNC(c2c(CC)ncnc2)=O)CC12CCC1(CC1)CC2 C1(NCc2cccc(CC=O)c2)CC2CN(c3cc(C)nc(CSC)n3)CC12.O c1(C(=O)NCCCCC(C)NC(C23CCC(CC2F)C3)=O)ccc2nccn2c1 c1(NC(CC)CNC(=O)Cn2nnc(-c3ccsc3)n2)ncccc1C(C)=O CC(CC(=O)N1CCC(NC(c2cccc3c2NCC3)=O)C1)C(F)(F)C(F)(F)F CS(C)(=O)=NC(=O)C(=O)N.c1(CC=O)cc(-c2ccccc2)on1.C1CC1.C c1(CC(=O)N)ccc(S(=O)(=O)CCO)cc1.N1(C(C2C(C)C2)=O)CCC(F)CC1 C1(C(=O)N)CS(=O)(=O)CC(=O)N1.c1(CC(=O)NCCCCC)ccc(O)cc1Cl C1(F)(CNC(c2cnc(CCC)s2)=O)CCN(C(c2nnn(C)n2)=O)C1 C1(C(=O)N)(COC)CCCCO1.C1CCN(C(=O)CN(C)S(N)(=O)=O)CC1 C1CN2CCCCC2CN1C(=O)C=CC.C1(C(=O)N)(COC)C=CCC1.C C1(CC(N2CC(NC(c3c(C)nn(C)c3)=O)C(C)(C)C2)=O)COC2(CCC2)CO1 C1(CNC(C(CC)(C)CC)=O)(CNC(c2c[nH]cn2)=O)CC2CCCC2C1.C Cc1cc(Br)sc1C(N1CCCC(C(N)=O)C1)C(=O)NCc1ccco1 c1(C(=O)NC(C)CCNC(c2cnn3ccn(C)c23)=O)ncnc2c1cnn2C C1(SC)CCN(C(C2CC(NC(c3ccnc(CO)c3)=O)C(O)C2)=O)C1(C)C Cc1nn(C)c(C(=O)N(CC(C)NC(C2CC23CCOC3)=O)C)c1Cl CCCC(C(=O)N1CC(C)(CCC(=O)NCCC2CC3CCC2O3)C1)NC(N)=O C(=O)(C(CO)C(F)(F)F)N1CC(CNC(c2c(C#N)scc2)=O)C(F)(CO)C1 c1(C(N2CC(CC)N(C(C3CC3(C)C)=O)CC2)=O)ccc2ccnn2c1 C#CCC(C)C(=O)N1CCC(O)(CCNC(c2cc(-c3ccc(Cl)s3)on2)=O)C1 N1(C(c2ccnc(OCC)c2F)=O)CCCc2cc(OC)ccc21 C12(NC(C(CSC)C)=O)CC3CCC(C1C2)N3C(c1ccn(C(C)C)n1)=O CC1CCN(C(C2(C)CCC(F)(F)C2)=O)CCN1C(=O)CC1(C(F)(F)F)CC1 n1(CC)cnc2[nH]c(=NCC3CCC(=O)N3)nc(N3CC(C)=C(C)C3)c12 c1(C(N(CCN(C(C2CN(C)C(=O)CC2)=O)C)C)=O)cnc2cccnn12 c1(C(=O)NCCCN(C(=O)C(C2CCOC2)OC)CC)ncnc2c1ccn2C n1(CCCC)nc(C)c(CNC(=O)CCc2cc(C)sc2C)c1Cl C1(CC=O)CCCC2(CC2)C1.N1(C(C2(CC#C)CCCC2)=O)CC2CC1C2C N1(C(c2c(C)nncc2)=O)CCCC(C)C1CNC(c1cnc(O)s1)=O c1(C(N(CCCC(C)C)C)=O)cn2c(n1)SCC2.C1(C=O)(C=O)CC1.CC N1(C(c2cc(C)c(C)o2)=O)CCC(NC(=O)CNC(c2ccncc2)=O)C(F)C1 c1(C(N2CC(F)C2)=O)cc(C(F)(F)F)cc(O)n1.C(=O)(C(=O)N)N(C)C.C CC1CN(C(c2ccc(C3CC3)nc2O)=O)CCC1N(C)C(c1cscc1F)=O c1(CC)nc(C(=O)NCC2CN(C(C3CCC3C(N)=O)=O)C2)co1.C c1(C(N(CCN(C(C2CC(C(C)C)C2)=O)C)C)=O)ccc2c(c1)CC(=O)N2 c1(N2CCC(S(C)(=O)=O)C2)nc(N2CC3CC3C2)c2[nH]ccc2n1 C1(CC(=O)NCC2C(NC(C(SC)SC)=O)CCC2)CCC(F)(F)CC1 Cn1cc2cc(C(=O)NCC3CC4CCC3N4C(C3CC(F)(F)C3)=O)ccc2n1 c1(CNC(C2(C)CCN(C(CCCCCCC)=O)C2)=O)ccc(C)c([N+](=O)[O-])c1 C(=O)(C(CNC(C1(CC)COC1)=O)CC1CC1)NC1(CC=C)CCCC1 c1(-c2n(C)ncc2)nc(-c2ccoc2)n(C2CCS(=O)(=O)C2)n1 N1(C(C)=O)CCCCC1C(=O)NC1CCC(NC(C23C=CC(CC2)C3)=O)CC1 C=CCN=C(NCc1ccc(Cl)o1)NCc1ccc(-n2ccnc2)c(F)c1 C(=O)(CCCC(C)CCC)NCCCOCCNC(C1CCC(C#C)CC1)=O c1(C(N(CCNC(C2N(CCC)CCC2)=O)CCO)=O)cc2cn[nH]c2cn1 C1(C(=O)NCC(c2ccc(F)cc2)OC)(CC)CCN(C(C)=O)C1 C1(N(C(CC(C)F)=O)CC2CC2)CCN(C(=O)CCC2CCOCC2)CC1 C1(C(=O)OC)CCCN(C(C2(NC(c3nccs3)=O)CCC2)=O)CC1 C1(CNC(C(c2n(C)cnc2)O)=O)CCCCC1.c1(C(=O)N)nc(=O)n(C)[nH]1 N1(Cc2cn(C3CN(C(c4c(C)nn[nH]4)=O)C3)nn2)CCCN(C)CC1 C(CN=c1[nH]c(=NC2CC3(CCCO3)C2)c2sccc2[nH]1)OCCCO c1(CN2C(C(=O)Nc3c(C)ncc(C)n3)CC(F)C2)ccc2ccc(Cl)cc2n1 C(CS(=O)(=O)NCCCN(C(C)C)Cc1ccco1)(c1ccccc1)OC N1(C(c2c[nH]c(=NC)o2)=O)CC2(CC2)CC1C(=O)NCCC(C)N1CCC1 c1(N(C(C(N2CCN(CC)CC2)CC)=O)Cc2ccccc2)cncnc1C c1(NC2CCN(C(c3c(C)cnc(F)c3)=O)C(C)C2)ncnc2c1cnn2C C1(NC(C2(NC(C(CC(=C)C)OC)=O)CCCCC2)=O)CCc2n[nH]cc2C1 c1(CNC(c2nnnn2CC2CCOC2)CCC)ccnc(OCCOC)c1F CCC(C)C(O)C(=O)N1CC(CNC(C2(C(C)C)CCC2)=O)(COC)C1 CC1(C)OCC2CC12C(=O)N.C1COCCN(C(c2cc(C(N)=O)cs2)=O)C1.C c1(C(N2CC(CCNC(CC(=C)C)=O)OC(C)C2)=O)ccc2n[nH]c(C)c2c1Cl c1(C(N2CCC(N(C(CSCCOC)=O)CCO)C2)=O)ccc(OC)c(F)c1 n1(CC(=O)NCC2N(C(CC(C)OC)=O)CCN(C)C2)c(C)cc(O)cc1=O C1(CC)CN(C(=O)C(C(C)C)OC)CCC1NC(c1cc(C2CC2)on1)=O C(=O)(C1=CCCOC1)NC(C(C)C)CCN(C)C(C1(F)CCCC1)=O c1(C(N2CC(COC)N(C(c3ccno3)=O)CC2)=O)cccc2nc(O)[nH]c12 N1(C(c2c(C#C)cnn2C)=O)CCC2(CCC2NC(=O)C(C)=CC2CC2)CC1 C(C(CNC(=O)C(F)C(C)C)S(C)(=O)=O)NC(c1ccc(OC)o1)=O N1(C(C(CC(C)C)N(C(C(CO)OC)=O)C)=O)CCC2CCCC2CC1 CC1CCC(NC(=O)CC2CCOC2)CN1C(=O)CCC1(N(C)C)CCCCC1 CCC(C)CCCC(=O)NCC(CC(F)(F)F)NC(=O)CCc1ncc[nH]1 c1(C(=O)NC(CC(C)NC(c2cc(C)cc(O)n2)=O)C)n[nH]c2c1CCCCC2 c1(CC)cc(F)ccc1C(N1CCCC(CNC(c2oc(C)cc2C)=O)C1)=O c1(CC)c(C(N2CCC2C(=O)NCCCc2ccsc2)=O)ccn1C C1(C(N(C)CCc2ncon2)=O)(CNC(=O)CCc2cncs2)CCCC1 C1(NC(CCOCCCOC)=O)CCN(C(=O)C=COCC)CC1(C)C C1(C(=O)NCCC(C)N(C(CCOCCOC)=O)C)CCCC2CCCCC12 c1(NCC(C)Cn2cccn2)nc(N2CC3CC2C2CC32)nc2scnc12 C1(OCCCNC(c2ncccc2F)=O)CCN(C(c2cnc(CO)[nH]2)=O)CC1 C1(OC)CCN(C(C23CC(CO)(CN2C(C2CC2C)=O)C3)=O)CC1C c1(C(=O)NCC(CC=C)NC(=O)C(C)(C)C2CCCC2)ccc2nc(S)oc2c1 N1(C(c2cccc(C)n2)C(=O)NC2CCCCC2)CCOC(C2COC(C)(C)O2)C1 c1(N2CC(C=C)OCC2)nc(N2CCOC(c3cc[nH]n3)C2)c2c(n1)CSC2 c1(C(N(CC(C)NC(C2CC3CC3C2)=O)C)=O)ccc(C(F)(F)F)cc1Br CC1CN(C(c2cscn2)=O)CC1(C)CNC(=O)C(F)C1CC1 C1CCC2CN(C(C3C4C5CCC(C5)C34)=O)CC12.c1(C(=O)NC)nc(Cl)cs1 CCCCC(C)C(=O)N(C1CN(C(c2c(C)nsc2Br)=O)CC12CC2)C N1(C(CONC(C2(CC)CCCO2)=O)=O)CCN2CC(C)CC2C1 C(=O)(C1=CN=C2N=CNN2C1)N(CC(C)NC(C(c1ccccc1)C)=O)C CC1(C)CCCC(C)C1.C1(C)(CCC(=O)N)CCCN1C(C1CC(C2CC2)C1)=O c1(C(=O)NC(CN(C(C2(CCCC)CC2)=O)C)C)cc2c(C)nn(C)c2s1 c1(CCC(=O)N(C)CCNC(c2cccnc2C(F)F)=O)c(F)cccc1F n1(CC(=O)NCCC2CN(C(C3N(S(C)(=O)=O)CC3)=O)C2)cc(Cl)cn1 c1(C(=O)NCC2C(C(N(C)Cc3cccnc3O)=O)OCC2)nnc(O)nc1O CC(CC(=O)NCCN(C(=O)CC1CN2CCC1CC2)C)P(C)(C)=O c1(OC)ccc(CC2CC(NC(=O)C(C)SC3CC3)C2)cc1 c1(C(C(=O)N(C(C)C(=O)OC)CCC)N(C)C2CC2)cncn1C C#Cc1ccc(C(=O)NC2C=CCN(C(=O)C(C)(C)N3CCOCC3)C2)nc1 C1(CNC(C(C)=C(C)C)=O)CCC1(C)C.C(=O)C=CCN1CCC1.N CCCCC(CC)C(=O)NC(CCCC)C(=O)NC1(C)C(C)(C)C1(C)C N1(C(c2c(C)nco2)=O)CC(CNC(=O)Cc2nc(Br)sc2C)C(C)C1 C1(CNC(CN(CCOC)C(c2coc(N(C)C)n2)=O)=O)CCCCC1C C1(COC)(NC(c2cccnc2Cl)=O)CCN(C(C2CCC(C)C(C)C2)=O)CC1 C(=O)(C(CC)(CC)CO)NCC(CC)NC(c1ccc(Br)cc1O)=O N1(C(C2C(C)C2C)=O)CC2CC2C1C(=O)NCC(C)CC1CCCC1 C(CCCC(=O)NC(C)C(c1ccccc1)NC(=O)CC1CC1)NC(C)=O N1(C(CC=CCNC(CCCOCCC)=O)=O)CC2C(C1)C2(F)F Cc1cccc(C#N)c1.C12(CC(=O)N)CCC1CN(C(C1CN(C)C(=O)N1)=O)C2 C1(C(=O)NC2(CN(C)C(c3cn(C4CC4)cn3)=O)CC2)C2CCCCC12 N1(C(C(COC)O)=O)CCN(C(=O)Cn2cnccc2=O)C(CF)C1 C1(CNC(c2n(CC)nnc2)=O)CC2COCC2N1c1cc(O)nc(O)n1 c1(NC(C2CN(C(c3n(CC)ncc3)=O)C2)=O)cc(Cl)nc(C)n1 N1(C(c2c(CCNC(C(C)OC(C)=O)=O)n[nH]c2)=O)CC2CCC2(CO)C1 c1(C(=O)NC(CCCNC(C2CCN(CC(C)C)C2)=O)(C)C)csc2nccn12 CC1(C)CCOC(CC(=O)NCC2CCCN2C(=O)Cn2cnccc2=O)C1 N1(C(C)C)CCCC(NC(=O)C(CO)NC(=O)CCN(C)C)C1 c1(C(N(C2CCN(C(=O)CSC(F)F)C2)CC)=O)cc(OC)n[nH]1 C(=O)(CCCCC(F)F)N(CC(O)CN(C)C(C1CCCCC1)=O)C C(=O)(C(CNC(=O)CC1(O)CCC1)CC1CC1)NC(CC(=O)NC)C C(CC(O)C(=O)NCC1(O)CCC1)SC.c1(CC=O)nc(C2CC2)cs1.C CC#CCC(C(=O)NCC(CO)N(C)C)NC(c1cnc(S)nc1)=O C(c1cccc(Cl)c1)=CC(=O)NC(C1CCCCN1C(=O)Cc1nc[nH]n1)C N1(C(COCC=C)=O)CCC(NC(c2ccccc2C(C)C)=O)CC1C c1(CNC(CC2C(C)(C)C2)=O)n[nH]cc1C(N1CCC(CO)C1)=O C1(NC(C2C=C(C)CS2)=O)CN(C(=O)CCN)C2(CCOC2)C1.[SH](C)(=O)=O c1(OCCC)ccc(CC(=O)NCC2CCN(CC(C)O)CC2)cc1OC C(C)(CSC)(C(=O)N)NC(c1cc(COC)no1)=O.n1(CCC)nccn1 C(CNC(C1(Cl)CC1)=O)(CC(F)(F)F)NC(=O)CC(O)C1CCCC1 c1(C(=O)NC2(C3N(C(Cn4c(C)ncc4)=O)CCCC3)CC2)cc(Cl)nnc1Cl C1(C)(C(=O)NCCN(C(CCCCC)=O)CCO)CC2(C1)CC2(F)F.CCO Cc1ccc(CN2CC3CN(C(c4ncc(Br)cc4F)=O)CC23)c2ccccc12 O=C1C2CCC3C1C3(C(=O)Nc1cncc(-n3cccn3)n1)C2 c1(CC)cc(CC(N2CC(C(C(=O)NC(C)(C)C(C)O)OC)C2)=O)on1 CC1CN(C(=O)CCCN(C)C)C(C)CN1C(=O)C(c1ccc(Cl)cc1)=O c1(NCC2(F)CCN(C(c3ccc(C)nc3)=O)CC2)c(F)cccc1[N+](=O)[O-] CCC(CC)C(C(=O)NCCC(C)NC(=O)CSc1cccs1)N1CCOCC1 c1(OC)ccc(CCOC(=O)Cc2ccc(Cl)c(I)c2)cc1Cl c1(C(=O)NCCOC2CCN(C(c3c(C)n[nH]c3)=O)C2)ccc(N)c(Cl)n1 N1(C(c2c(C)cc(C)[nH]2)=O)C2CCC1CC(NC(=O)C(O)Cc1ccccc1)C2 c1(CNC(=O)NC2(c3ccccc3)CC(F)C2)nc(Cc2ccccc2)no1 C=CC(C)(C)CCCNC(c1ccncc1Cl)c1nnnn1CC(F)F CC1CC(C(=O)NOC)CN(C(C2OC3CCC2C3)=O)C1 C1(CC#C)(C(=O)NCCCC)CCCCO1.c1(CC(=O)N)coc(COC)n1 C(N=c1cc(C)[nH]c(=NCCN(C)C)[nH]1)c1cc(C)cc2c1CCC2 O=C(CCOCC1CCCO1)NCCC1CCCC1.C(=O)(CC1CCC1)N Cc1coc2ccc(C(=O)NCC3(C)CCCN3C(c3c[nH]c(=N)s3)=O)cc12 c1(OC)cc(C(=O)NCC2CCC2)c(N)c(C)c1.c1(C=O)ncc(Cl)cc1F C1(C2(O)CCOC2)(C(N(CCCNC(c2coc(C3CC3)n2)=O)C)=O)CC1 C(=O)(C1=C(Cl)CCOC1)NC(C(C)NC(c1csc(-c2ncc[nH]2)n1)=O)(C)C Cc1ncc(C(=O)NC2(C(N3CCC3CC(C)C)=O)CCN(C)C2)n1C C#CC1CCC(NC(=NCCOC)NCC(c2c(OC)cccc2Cl)(C)C)CC1 Cc1oc(C)c(S(N)(=O)=O)c1C(=O)NCC(O)Cc1ccccc1F CC(C)C(C)(CNC(=O)Cc1ncncc1Cl)NC(=O)C1=CCC1 c1(OC)cc([N+](=O)[O-])ccc1C(=O)N.C1(C=O)CC2CCC1O2.CCC1CC1 C1(CNC(C2C3CCCCCCC23)=O)CCCC2(CN(C(C3SCCS3)=O)C2)O1 c1(C(=O)NC2CCN(C(c3c(C)ccs3)=O)C2C2CC2)ccc(=O)n(C)c1 C1(C(=O)NCCSCC(NOCC(=O)OC)=O)C2CCC(C2)C1C C=CC(C)(CC)C(=O)NCCCCC(=O)NCC(CSC)OC C1(C2CC2)(SCC(=O)NCCNC(=O)COC2CC2)CC1 CC1C(C)N(C)CCN1C(=O)NCCCN(C)Cc1ccncc1 CC(CCCCCO)NC(c1cc(CCNC(=O)Cn2cccn2)on1)=O C1(C(=O)NCCC(=C)C)CCC2C(C1)C2(F)F.c1cnn(C)c1.C(=O)(C)N N1(C(C2(F)CCN(C(c3c(CC)nccc3)=O)C2)=O)CC(N(C)C)C(C)(C)C1 N1(C(CCCN(C)C)=O)CC2CCCC(C)(C2)C1.C1(C(=O)N)CC(=C2CCC2)C1 CC1(C)COC(CCC(N2CCC(CCNC(c3n[nH]cc3F)=O)C2)=O)C1 N1(C(c2n(C)ncc2)C(=O)NCCC2(C)CC2)CCCC(C2(C)CC2)C1 c1(NC(C2N(C(C)=O)CCC2)=O)ccccc1N(C)C O=C1CCC(NC(=O)CCCCCNC(C2CC(O)C(F)C2)=O)CCN1 c1(-n2c(C(CCC=C)NC3CSC(C)C3)nnn2)cccc([N+](=O)[O-])c1 C(=O)(CCCCC(C)(C)C)NC12C(CN(C(CP(C)(C)=O)=O)C1)CCC2 c1(C(N2CC(N(C(CC(=C)C)=O)C)C(F)C2)=O)ccc(C#N)cc1C Cc1nccc(C(N2CC3CC2(C(=O)N(CC(=O)NC2CC2)C)C3)=O)c1C c1(C(=O)NC(CNC(CCCOCC=C)=O)CC=C)c(F)cc(F)c(F)c1F N1(C(c2cc(COC)[nH]n2)=O)CCC(CO)(NC(C2CCCCO2)=O)C1 c1(C(C(C)OC(C2(COC)CCNC2)=O)=O)ccc(OC)c(OC)c1C CCC(C(=O)N1CC(CNC(=O)Cc2cnco2)(OC)C1)C(C)O C1(NC(CC2(C(=O)OC)CC2)=O)CCCCCC1.C1(C=O)CN(C2CCC2)C1 CCC(F)(F)CCNC(c1cccc(F)n1)c1nnnn1CCC1CC1 C1CS(=O)(=O)CC1.c1(C=O)ccc(F)s1.c1(N(CC=O)CC)ccccc1.N C1(NC(C(C(C)C)SC)=O)CN(C(=O)C2=NOCC2)CC2CC12 C1(C(N(C2CCN(C(c3csc(CCC)n3)=O)C2)CCC)=O)CCN(C)C(C)C1 c1(CNC(C)CCC(=O)O)ccn2cncc2c1 C1C(C)CCCN1C(=O)CC.C(CC)(C(=O)N)OCC.c1(C=O)cccs1.C c1(C(=O)NCCN(C(Cn2c(C)nnn2)=O)C)cccc(I)c1 Cc1nc(C(C)C)sc1C(N1CC(NC(c2cocn2)=O)C(n2ccnn2)C1)=O N1(C(CCCNC(C)=O)=O)CCC(C2CC(NC(c3oncc3C)=O)C2)C1 n1(CC)nc(C)c(C(=O)NCC2CCCCN(C(=O)C(C)O)C2)c1Cl C1(C(=O)NCC(CC=C)NC(c2c[nH]nc2[N+](=O)[O-])=O)CCCN2CCCC12 c1(N2C3CCN(C(CC#C)=O)CC3CC2)ncc2c(Br)cccc2n1 N1(C(C2CN(C)C2)=O)CC=CC(C(=O)NCCNS(C)(=O)=O)C1 c1cccc(Br)c1F.C(=O)(C(C)COCC)NCCN(CC(=O)N)CCC C1CC2C(C1)C2(F)F.c1(OCC(=O)OCC)ccc(OCC(=O)N)cc1 CCC(CCC(=O)NCC1(OCC)CN(C(=O)CC(C)n2ccnc2)C1)OC c1(C(=O)NCC(CC(C)C)NC(c2cnn(CC)c2C)=O)cc(N)cnc1Cl C1(C(N(CC(C)N(C(=O)CC2COC2)C)C)=O)CN(S(=O)(=O)N(C)C)C1 Cc1cc(Cl)ccc1CC(=O)NC1CCCC(NC(=O)Cc2csc(S)n2)C1 C=C=CC(C)C(=O)NCCN(CCCN(C)C)C(c1ccncc1Br)=O N1(C(c2c(CNC(c3ccccc3)=O)noc2)=O)CCC2(CC1)N=N2 N1(C(CC=C)=O)CC(OC)CC1(C)CNC(c1c(C)ncn1O)=O c1(NCCCC(C)NC(c2c(C)nncc2)=O)snc(C)c1C#N C1(CC(=O)N(CCCCOC)CCO)CCOCC1OC n1(CC(=O)NCC(CC)NC(=O)CCCOc2ccccc2)nnc(=O)[nH]1 C(=O)(CC(C)(C)C(F)S(=O)(=O)N1CCC(O)(c2cccc(Br)c2)C1)OCC N1(C(c2cc(C)nc(C)c2)=O)CCCC2C1CCN2C(=O)CCS(C)(=O)=O C1(CNC(C2CC(OC)C2)=O)CCC(C)(C)CN1C(c1cncs1)=O CCCCCCC(=O)NC1CCC(NC(=O)C(C)(F)c2ccon2)CC1 C1(CC)CC(C(N2CCC2CC2CC2)=O)CCN1C(=O)C(CSC)OC C1(NC(c2n(C)nc(C(F)F)c2)=O)CCC12CCC2.c1(C(=O)N)cc(Cl)ccn1 c1(C(=O)NC2CC(C)N(C(=O)CCCF)C2)cc(O)c2ccccc2c1 c1(OC)ccc2oc(C(C=O)N(CCC#N)C3CC3)c(C)c2c1.CCC1CC1.N c1(CN2C(C(=O)NCCOCC(F)(F)F)CCC2)nnc(O)nc1O CN1CC(C(N2CCC(C(C)(C)NC(C3CNC(=O)N3)=O)CC2)=O)CCC1=O c1(COC)ccc(CC(N2CCC(NC(=O)CCOC3CCCC3)C2)=O)cc1 N1(C(C(CCCC#C)C)=O)CC2CC(C1)C(CO)C2NC(=O)CC1(C)OCCO1 N1(C(C)=O)CCC2(CC1)CC(NC(c1cccnc1C)=O)c1ccccc1O2 c1(CC=O)c(Cl)ccc(O)c1Cl.c1(CC)nc(C)[nH]c1C(=O)NC1CCC1.C C1(C)(NC(C2(C#C)CN(C(=O)CC3COCCO3)C2)=O)CC(C)(C)OC1=O Cc1cc(-n2cc(CONC(c3ccc(F)c(C(F)F)c3)=O)nn2)cnc1Cl C(=O)(CC1=NNC(=O)C1)N1CC(Cn2c(C)cc(C)n2)OCC1 c1(C(C)NC(C)C(C)O)c(F)cc(F)cc1F c1(N2CC(NC(c3cccc(C)c3)=O)C(F)C2)ncncc1C#N c1(NC(C2N(C(c3c(C)cncn3)=O)CCC2)=O)ccc2c[nH]nc2c1 c1(C(=O)NC2CC(C(C(=O)N(CC(=C)C)C)F)C2)ncc(C)cc1C Cc1nc(C)c(C(=O)NCC2CC(C)N(C(=O)CCc3ncc[nH]3)C2)c(C)n1 N1(C(C2(NC(c3c(CCC)n[nH]c3)=O)CCOCC2)=O)CC2(CCC(C)OC2)C1 C(=O)(CCCCCC(C)O)NCC1CC2(CN(C(c3c(C)nc(C)[nH]3)=O)C2)C1 CC1(CNC(C23CC(F)(C2)C3)=O)CCCN1C(=O)CNS(N)(=O)=O Cc1oncc1C(=O)NCC1N(C(C(C)OC)=O)CCC1.C1(C=O)CCCC1 C(=O)(CCCC(F)F)NC(CCN(C(c1nnc(C)s1)=O)C)C(C)C c1(C(C)C)ccccc1-c1cn(CCCC(=O)N(C(C)C)Cc2cccs2)nn1 c1(C(=O)NCC(C)(CO)NC(CN2CC(CC)C2)=O)ccc(Cl)cn1 c1(OC)ccc(C(N2CC=C(CNC(=O)C(C)Cc3ccco3)CC2)=O)cc1O c1(C(C)(C)CNC(=O)CN2CCOCC2)ccc2ccccc2c1 c1(C(N2CCCC3(NC(CCOC(C)C)=O)C(C2)C3)=O)ccnc2c1ncn2C c1(C(CO)NC(c2cc(C)[nH]c2C)=O)ccc(Br)c(Cl)c1 C1(C(N(C2CCC(NC(c3c(CC)ncs3)=O)C2)C)=O)CCc2nnc(O)n2C1 c1(C(N2CCC(C(C)NC(C34CC5CC3C4C5)=O)C2)=O)ccc2nc(O)sc2c1 c1(CCC(=O)NC2C(NC(COC(C)=O)=O)CC2)ccc2ccccc2c1 c1(C(=O)NC2CCC(NC(=O)CCc3cc[nH]n3)CC2)cnc2ccnn2c1 c1(C(N2CCC(C)(CNC(=O)C(F)(F)C(F)F)C2)=O)ccn2ccccc12 c1(CC2C(C(C)NC(=O)Nc3ccccn3)C2)cc(Br)cc(F)c1C#N C(=O)(C#CC1(C)CCCO1)N1CCCC(C)(CO)C1 c1(C(N2C(CNC(CCCCN(C(C)C)C)=O)CCC2)=O)cn(C)c(=O)nc1O CCCC(CC)C(=O)NCc1cc(C(N2CC(C)(O)C2)=O)on1 C1(NC(c2c(OC)scc2)=O)CC2CN(C(=O)C(C)c3cccs3)CC2C1 CC1N(C(=O)CC2(C)CCN2C(=O)Cn2nccn2)CCCC1(C)C c1(C(N2CCC(C(N3CC(SC)C3)=O)C2C(C)C)=O)ccc(=O)n(C)c1 C1(OC)CCC(C)(C(=O)NCCC2CC2)CC1.n1(CC=O)nc(C)oc1=O C#CC1(C(N2CCCCC2CC(C)C)=O)CN(C(=O)C(C)C(C)C)C1 CC1C(NC(c2snnc2C2CCC2)=O)CCCN1C(C1CCC2(CC1)CC2)=O CC(C)CC(O)C(=O)NC(CC(=O)NC(C)(C)C(C)(C)C)C(F)F C(CNC(=O)C(O)CC1CCCC1)(CCNC(=O)Cn1cnnc1O)OC Cc1ccc(CC(N2CCCC(NC(c3c(C)ccnc3O)=O)C2C)=O)c(Cl)c1 c1(N(CC#CC)C)nc(NCC2(S(C)(=O)=O)CCC2)c2ncsc2n1 c1(C(N(C2CN(C(C3CNC(=O)CC3(C)C)=O)C2)C)=O)cc2ccc(F)cc2[nH]1 C1(O)(CCNC(c2nocc2Cl)=O)CCN(C(C2CC2c2ccccc2)=O)CC1 c1(CCC(=O)NC2(c3ccccc3)CCN(C(=O)COCCF)C2)cccc(O)n1 c1(C(=O)NC2CC(C)(NC(C(Br)=C(C)C)=O)C2)ccc(Cl)c(C#N)c1 C1(C=O)CC12CC(C)(C)C2.N(C)(S(N)(=O)=O)CC(N1CC(CCC)C1)=O C1(c2cn(CCNC(CN(C3CCCC3)C)=O)nn2)CCC(=O)CC1 c1(C(N2CCn3cncc3C2)=O)ccc2[nH]cc(-c3ccc4scnc4c3)c2c1 c1(SCC)ccccc1CC(=O)NC1CCC1NC(=O)Cc1ncc[nH]1.C c1(C(N(C2CCN(C(C(N3CCNC3=O)C)=O)CC2)C)=O)ccc2n[nH]cc2c1 CCC(C)C(O)C(=O)NCC1(F)CC(NC(c2cn3ccnc3s2)=O)C1 CCCC(CCNC(=O)C(CN(C)C)NC(c1cccc(C)c1)=O)C1CC1 C1(N(C(c2cnc(CC)[nH]2)=O)C)CCC2CN(C(c3coc(C(F)F)n3)=O)CC12 C1(C(=O)NC2(COC)CC=CC2)CCCN(C(=O)CC(C)n2ccnc2)CC1 CN1CCOC(C(=O)NC2CC2CNC(c2ccccc2-n2cncn2)=O)C1 CCC(CC)C(C(=O)NC(c1ccccc1)C)N1CC2CCCC2(CO)C1 c1(C(N(CCCCN(C(c2c(C)nc(C(C)C)o2)=O)C)C)=O)cc(F)cnc1O c1(N2CCCC(CCCC)C2)nc(=NCCC2CC2)[nH]c2ccccc12 O=C(CNC(C1CCOC1)CO)N=c1ccn(CC2CCNCC2)[nH]1 c1(C(N2C(C)C3CC2C3)=O)cn(C)c(=O)nc1O.C1(CC(=O)N)CCC=CCC1 N1(C(Cc2ccc(OC)nc2)=O)CCC(C)C(N(C(=O)C=CC(C)(C)S)C)C1 C(=O)(CCCC(C)(F)F)NCCc1ccc(C)cc1.c1(C=O)cnc(C2CC2)o1.N N1(C(C2(OCC)CC2)=O)CC2CN(C(=O)C=CC3CCOC3)CC(C1)O2 N1(c2ccc(C(=O)OCC)cn2)CC(F)(F)CC1(C)C.C1(CC=O)CCOC1 c1(Nc2ccc(C)cc2)ccc(N=c2ccnc(OCCF)[nH]2)nc1 C1(CCC)CN(C(c2coc(Cn3cccn3)c2)=O)CCN1C(=O)CC(C)CF CCCCC(CC)CC(=O)NCC1(NC(C2CCCN(C(N)=O)C2)=O)CC1 C=CCC(C)C(=O)NC1(CCNC(c2ccnn2CCCC)=O)CCC1 Cn1cc2ccc(C(=O)NC3CCOCC3NC(c3ccc(O)nn3)=O)cc2n1 CC1SCCCC1C(=O)NCC(O)C(=O)N(C)CC1(F)CCC1 S(=O)(=O)(c1c(F)cccc1F)NC1C(C(=O)Nc2c[nH]c3ncccc23)CCC1 c1(CC)nc(C(N2CC3C(CNC(C4(C)CCCN4C)=O)C3C2)=O)c(N)s1 Cc1cc(NC(C2CCCC(NC(=O)CCc3ncccn3)C2)=O)cnc1O N1(C(C(n2ncc(C)c2)C)=O)CCC(C(N2CC(N(C)C)C2)=O)(CO)C1 c1(NC(=O)C(O)Cc2ccc(Cl)cc2)ccc2cnn(C(F)F)c2c1 N1(C(CC(CC#C)NC(c2cnn(C)c2Cl)=O)=O)CCN2C(=O)NCC2C1 c1(CNC(=O)CC2COCCN2C(c2cnn(C3CC3)c2)=O)cnc2n1CCC2 N1(C(C2=NOC(C)(C)C2)=O)CCOC2(CCN(C(=O)C(O)Cn3cncn3)C2)C1 C1(NC(CC2N(C(COC(C)=O)=O)CCC2)=O)CCCC(O)CC1 Cc1nn2c(c1CNC(c1ccnc(C)c1C)=O)CN(C(=O)C(O)C1CC1)CC2 C(CCCCC(=O)NCC1CC2(CC2)C1)N(C)C(c1cncnc1)=O CC(C)(CCCF)C(=O)NC1CN(C(c2cc(F)cc(F)c2N)=O)CCC1O Cc1cccc2cc(C(=O)NC3CCC(NC(=O)OC(C)(C)C)C3)nnc12 C=CC(CCC)CC(=O)NC(C1CCCCC1)C(N1CCN(CC)CC1)=O C1(C(=O)NCC(C(C)C)NC(c2snc(C)c2N)=O)OCC2COCCC12 CC#CCCC(=O)NCC1(C(=O)NCC2CC(C)C2)CC12CCC2 c1(C(=O)NCC2C(NC(CCC(=C)C)=O)CCCC2)ccc(C#N)c(F)c1 c1(C(=O)NCC2C(C)CCN2c2ccnc(CO)n2)cnc2[nH]ccc2n1 N1(C(C2=CCN(C(CC(CC)(F)F)=O)CC2)=O)CC2CCN(C)CC2C1 C1(CN(c2ncc(C(C)(C)O)cn2)C)CCCN(C(C2(O)COC2)=O)C1 Cc1oc2ccccc2c1CC(=O)NC12COC(C1)C(NC(=O)CC(F)(F)Cl)C2 N1(C(c2nn(C)c(Br)c2C)C(=O)NCCSC)CCn2cc(C)nc2C1C c1(CC(=O)Nc2c[nH]nc2C(=O)NCC2CCC(F)C2)cc(Br)ccc1Br Cc1nc(NCC2CCC(NC(=O)C(C)c3cccs3)C2)c(Cl)cc1C#N N1(C(c2ccc(OC)cc2O)=O)CCC2(NC(=O)C(F)OC)CCCC12 c1(C(=O)OC(C)(C)C)cc(C(=O)O)cc(F)c1.c1cnc(-c2ccccc2)o1.C c1(C(c2cn(C)nc2)NC(=O)NCCC2(O)CCCC2)ccc(Cl)cc1 C#CC1(C(=O)NC2CCC(C)(CNC(=O)C3=NOCC3)C2)CCCC1 C1(C(=O)NCC2CCN(c3cccc(Br)c3)C2)CCC(N=c2cncc[nH]2)CC1 c1(C(=O)NCC(C)NC(c2ccnc(C3CC3)c2)=O)ncc(Cl)n1C c1ccc(Cl)c(Cl)c1.C=Cn1nccc1C(=O)NCC1CN(C(=O)C)C2CC12 C1(C(N(CCCNC(c2c(C)csc2)=O)C(C)C)=O)CC(C)(C)OC1(C)C CONS(=O)(=O)c1ccc(C(=O)NC2CC2NC(c2ccnn2C)=O)cc1 c1(CNS(c2nccc(C)c2)(=O)=O)nc(O)c2cc(Br)cc(Br)c2n1 C1(C(C(=O)N(CCC)C)O)CCS(=O)(=O)CC1.Cc1c(C=O)ccn1CCC N1(C(C(C2CCCC2)NC(C)=O)=O)CC2CCCCC2(NC(c2csnn2)=O)C1 c1(CCC(=O)NC(=C2CCN(C(C3CC3CF)=O)CC2)C)cccc(Cl)c1 N1(C(c2nc(C)n(C)n2)=O)CCC2(CCCN2C(C2CC=CCO2)=O)C1 C1(C(N(CC(CNC(c2c(SC)n(C)nc2)=O)C)C)=O)CCCCC1(F)F N1(C(c2cc(C)on2)C(=O)NCC=C)CCN(S(=O)(=O)C(C)C)CC1C.O c1(OC)cccc(C=CC(N2CC(CNC(=O)C(C)(Cl)Cl)CC2C)=O)c1 C1(C(=O)NC2CCN(C(CCCOC)=O)CC2O)(OC)CCCC(C)(C)C1 C(N=c1[nH]c(N2CCCC3(CCCCO3)C2)nc2c1CCCC2)c1c(Br)scc1 C1(CC)CCCN(CC(=O)NCC(CNC(c2nc(OC)c(C)s2)=O)OC)C1 N1(c2nnc(C(CC)C)n2CCC(=O)N(C)C)CC=C(c2ccccc2)C1 n1(CC(=O)NCCOc2c(C)nccc2)cc(C#N)c(O)nc1=O N1(C(c2ccc(SC)s2)=O)CCC(O)C(NC(=O)C(C)=C2CCC2)C1 N1(C(CCC2CC(OC)C2)=O)CC(CN(C)C(c2ccnnc2O)=O)C2(CC2)C1 N1(CC(C)(C)NC(c2cc(Cl)c[nH]2)=O)CCN(C(=O)Cc2cccnc2O)CC1 C12(NC(C3CC(SC)C3)=O)CCC(CC1)N(C(c1ccc(F)c(C)c1)=O)C2 c1(CCC(=O)NCCN(C(=O)CC(C)C(C)C)CCC)nnc(S)nc1O Cc1occ(C(F)(F)F)c1C=O.C1(F)CCN(C(C2CC(F)C(=O)N2)=O)C1.N c1(C(C(=O)NCCCn2cc(C(N3CCOC3=O)C)nn2)(C)C)ccccc1Cl N1(C(c2cc(CCC)c(C)s2)=O)CCC(O)(C(C)NC(c2sncc2C)=O)CC1 C(=O)(C1=CCC(NC(=O)C(=O)C(C)CC)C1)N(c1ccc(Br)cc1)CC#C C1(NC(CCCCC=C)=O)CCN(C(c2cc3c(ccn3C)s2)=O)CCC1CO CC1=C(C)CC(C(=O)NC2C=CC(CNC(=O)CN3CCOCC3)C2)CC1 N1(C(C2Cc3nccnc3C2)=O)CCC2OCCN(C(c3ccc[nH]3)=O)C2C1 c1(C(N2CCCC(O)(CN(C(CSC)=O)C)C2)=O)cc2c(=O)[nH]ccn2c1 c1(C(N2CCC(CC)(NC(C3CCCCN3C)=O)CC2)=O)c(C)cc(C)cc1N C12(C=O)CCC(CC1)C(C)(C)O2.Cc1nn[nH]c1C(=O)NCCC1CCC1.N C1(OC)CC2(CCN(C(c3cn(CC4CC4)nn3)C(=O)NCC(F)F)CC2)C1 Cc1ccc(SCC(=O)N(C2CCN(C(c3nc(C)n(C)n3)=O)C2)C)c(C)c1 Cc1csc2nc(CC(=O)N(C)CC3CCCN(C(C4CCC4(F)F)=O)C3)cn12 c1(C(C(=O)NC(C)C)N(C(C)C(=O)OC)CCC)cc(Cl)c(F)cc1F CC1CN(C(=O)CC2COC(=O)N2)CC1CNC(=O)CC(C)(C)C1CC1 c1(OCCCC(N2CCCC(CNC(C3(F)CC3(F)F)=O)C2)=O)ccccc1F c1(C(C)C)nccc(C(=O)NCCC(C)NC(=O)CN(C)C2CC2)n1 c1(-c2nc(N(CCCC(=O)NO)CC=C)sc2)c(C)cc(C)cc1C c1(OC)ccc(C(=O)N(CC(CO)(CO)NC(c2occ(C)c2C)=O)C)c(C)n1 C1(COC)CCN(C(C2CCC3CC3C2)=O)C1.C1(C(=O)N)CN(C(C)=O)C1 CN1CC(O)CC1(C)C(N1CCN(C(=O)C=Cc2cncc(O)c2)CC1)=O Cc1nnc2n1CC(C(=O)NCC(C)(O)CNC(=O)Cc1ccc(Cl)nc1)C2 c1(CC(C)NC(=O)NCc2nc(C(CC)(C)C)on2)ccc(C)cc1C c1(CC(=O)NC2CC(NC(=O)COCC(F)F)C2)c(Cl)ccc(O)c1Cl Cc1nccc(Cl)n1.c1(C(N2C(C(=O)N)C=CC2)=O)ccc(C(F)(F)F)c(Br)c1 N1(c2c(C)cc(C#N)cn2)CCC2(CC1)CN(C(=O)CC=C(Cl)Cl)CCO2 C1(C(=O)NCC(CNC(c2ccn(COC)n2)=O)(C)F)CCn2nncc2C1 c1(C(N(C)C)=O)ccc([N+](=O)[O-])cc1.C1CN(C(C2(F)CCOC2)=O)CC12CC2 C1(CC(=O)NCC(=O)OC)CCN(C(=O)CN2CCCNC2=O)CC1 c1(CCC)ccc(C(=O)NC2CCCC2NC(=O)C(C)Cc2cccnc2)[nH]1 c1(OC(C)C)ccccc1C(=O)NC1CCOCC1.c1(C(=O)N)cnc(C#N)s1 c1(OC)cc(Cl)ncc1CN1CCOC(C(=O)Nc2cc(Br)ccc2Cl)C1 N1(C(C=CCN(C)CC)=O)CC=CC(C(=O)Nc2ccc(Cl)cc2)C1 C(=O)(C1CCc2nnc(C)n21)N1CCCC(CNC(c2ncc(C)c(Cl)c2)=O)C1 C1(n2c(C(c3cn(CCC(C)(C)C)nn3)C3CC3)nnn2)CCCCCC1 c1(C(=O)NCC(C)(CO)NC(C=Cc2ccc(C)nc2)=O)csc2ccccc12 C1(C)(C(=O)NC(CC)CNC(=O)C(=Cc2ccncc2)C)CCC(OC)CC1 C12(C(N3CCCC(NC(C(C)n4cnnn4)=O)C3)=O)CCC(CC1)C2(C)C c1(OC)cc2c(cc1F)N(C(C1(O)CN3CCC1CC3)=O)CC2 Cc1nccnc1C(=O)NCCN1CCN(C(=O)C(C)Cc2cnn(C)c2)CC1 C1(C(=O)NOCCCCC2CC2)COCCN(C(C2(CF)CC2)=O)C1 C1CCC2(CO1)CCC2.C(=O)C(O)C(F)(F)F.C1(CC=O)(C(=O)OC)CC1.N C(=O)(C(C)C(C)(C)C)NCCC(C)(C)OC.c1(C(=O)N)ccnc2cc[nH]c12 c1(OC)ccnc(C2(CN3CCCC3c3cc(I)nn3C)CC2)c1 C1(CC)CCOCC1NCC1COC(C)C1 N(C(=NCCCF)NCc1ccc(OC)cc1OC)C1CC(C#C)C1 CC1C(C)N(C(c2ccc(N)cc2O)=O)CCN1C(c1ccc(C(N)=O)cc1)=O CCC(CCCC(=O)NCCCC1CC(C)C1)NC(=O)CC1CC2CC2C1 S(=O)(=O)(c1ccc(NC2CCCSC2)cc1Br)NCC(n1cccn1)C N1(C(c2sc(C(F)F)nc2Br)C(=O)NCCCOC)CCOC(C(F)F)CC1 Cc1c(C(=O)NC2CCC(N(C)C(c3cc(Br)n[nH]3)=O)C2)ccn1C c1(C(=O)NC2(CC)CCC2)occ2c1CCC2.c1(C(=O)N)cscc1C(F)F C(=O)(C(C#N)C1CC1)N.C(C(=O)NC1(C)CC1)OCCOCC#C CC(C)CC(O)CC(=O)NCC1(C)CC(F)(F)CN1C(C1CCCO1)=O C1(NC(C(C(C)(C)C)O)=O)CC2(CCN(C(c3ccc(C4CC4)nc3)=O)CC2)C1 N1(C(=O)NCCc2c(CC)cccc2)CCCCCC1CCN(C)C C1(CNC(COCC(=C)C)=O)CCCN(C(C2CC(n3ccnn3)C2)=O)C1 C12(NC(CCOC)=O)CC(C1)N(C(c1csnn1)=O)C2 C#CC1CN(C(=O)C=CC)CCN1C(=O)C(F)CCCC c1(N(CC(C)(O)c2ccco2)C)nnc(CC(F)(F)F)n1CCCS(C)(=O)=O Cc1ncnc(NC2(CO)CCCN(C(C3(C)CS(=O)(=O)C3)=O)C2)c1F C1(N(C(C(CC)CC)=O)C)CCCN(C(c2c(C(F)(F)F)ncn2O)=O)CC1 C1(n2cc(C(C)(C)O)nn2)CC2CCC1(NC(C1CCCO1)=O)C2 c1(SC)cscc1C(=O)N(C)CCN(C(=O)CC1CC2(CC2)C1)C C(=O)(CCC(C)CC)N1CCC(CNC(c2cc(CC)[nH]n2)=O)(OC)C1 C=CCC(C(=O)NC(CCF)C(=O)N1CCC(F)(CF)C1)C(C)C CCC(CC(=O)N1CC(CNC(c2cn3cc(C)sc3n2)=O)CC1C)C(C)(C)C c1(C(=O)NCC2CCCC(CNC(c3c(C)scn3)=O)C2)ccc2nnnn2c1 Cc1cc(C)c(C(N2CC(NC(=O)CC3(O)CCCC3)CC(C)C2)=O)cn1 CCC(CC(=O)N1CCC2(CCCN2C(c2cnc[nH]2)=O)CC1)CC(F)(F)F Cc1csc2ccc(C(N3CCC(NC(=O)CCOCC(F)F)C(C)C3)=O)cc12 CC1(C)CC(CN2C(=O)NC(CCC(F)(F)F)C2=O)CCO1 C#CC(CNC(=O)CC1(C)CCN1C(c1ccnc(OC)n1)=O)CC(C)(C)C Cc1c(C(=O)NC2(CC)CCC2)nnn1C.c1(C=O)ncccc1C(C)(C)C.N c1(C(N2CCCC(c3n(CC)c(S)nn3)C2)=O)c(F)ccc2n[nH]cc12 N1(C(C(C)CF)=O)CC2(CCC(CNC(c3c[nH]cc(Cl)c3=O)=O)O2)C1 C1(CNC(CC2C(C)C2)=O)CCN(C(c2c[nH]c3ncccc23)=O)CCC1(F)F Cc1ccc2[nH]c(C(=O)NC3CC(C)C3)cc2c1.C(=O)C(C)(C)CC1CC1.C Cc1cc(C(=O)NCC2CN(C(c3ccccc3CO)=O)C2)c(C)cc1F c1(C(=O)NCC2(F)CN(C(C(CC)(C)F)=O)C2)cc2ccccc2n1C C1(CC=C)(NC(c2cncc(COC)c2)=O)CCN(C(C2C=CCCC2)=O)C1 C(C)(C(C)(C)C)NC(C1(C)CC(C)C1)=O.n1(CC=O)cnc(C(N)=O)n1 Cc1cc(C(=O)N(C(C)CCNC(C2CC2OC(C)(C)C)=O)C)[nH]c1C N1(C(C2N(C(c3c(C)non3)=O)CC(F)C2)=O)CCCN(C)CC1 CCC(C)(CC(=O)NN1CCCC1C(=O)NCc1nncs1)C(=O)OC C1(CNC(CCN(CCCO)C(c2c(C)nc(C)s2)=O)=O)CC(O)C12CCC2 C1(C2CCN(C(=O)C#CC(=O)N(C)C)CC2)(NC(C2CC(C)OCC2)=O)CC1 C1(CC=O)CCCCC1.CCS(=O)(=O)N1CC(C(=O)NCC=CC)C1.N CC(C)C(C(=O)N1CCN(C(=O)CNS(=O)(=O)C(F)(F)F)CC1)n1cnnn1 C1(CC)C(C(=O)NCCc2ccccc2C)CCN1C(C1CC1)=O.C1CC1.O N1(C(C(CCC)O)=O)CC2(CCN(C(=O)C(c3c(C)nn(C)c3C)=O)C2)C1 C(=O)(C(C)CC(=O)N1CCCCC1CC(=O)NCCC1=CCOCC1)OC N1(C(COc2cc(C)c(F)cc2)=O)CC(C2CCCN(C(c3cncs3)=O)C2)C1 Cn1nnnc1C(CC1(C)CC1)NC(=O)CCc1ncccn1 Cc1cnc(NC(=O)CC2CCC(NC(c3cccc(Br)c3Br)=O)CC2)cc1Br c1(SC)ncc(Br)c(N2CCN(C(=O)Cc3ccc(F)c(F)c3)C3CC23)n1 c1(C(=O)NC2CC(O)C23CCC3)nc2sccn2c1I CN1CCC(C(=O)NC2(C(=O)NC3CC(N4CCCC4)C3)CCOCC2)CC1=O N1(C(C2(C)CCNC2=O)=O)CC2CCC2(CNC(=O)C(F)(F)c2ccccc2)C1 CCC(C)CCC(O)Cc1nc(-c2cc(F)ccc2OC)no1 C(=O)(CCCC)N.C(C(F)(F)Cl)N(C(=O)C=CCC1CCC1)C.C(N)=O C(C(=O)N1CC(CC(C)NC(c2cc(C(C)=O)cs2)=O)C1)(C(C)C)OC Cc1ccc(F)c(NC(C2(F)CN(C(c3cc(C)cc(Cl)n3)=O)C2)=O)c1 C1(NC(C(COC)N(C)C)=O)CCC(N(C)C(c2cc(C)c[nH]2)=O)CC1 CN1CCN(CCNC(c2cc(O)n(C)n2)=O)CC1=O c1(C(N(CCNC(C2(C)C(C)(C)C2)=O)C2CC2)=O)ncc(Br)cc1N c1(C(=O)NC(C2CCN(C(C(F)=C(C)C)=O)C2)C)ccc(S(C)(=O)=O)o1 c1(NCC(CC)C(C)(F)F)cc(=NCC(CN(C)C)OC)[nH]cn1 C1(N(C(=O)Cn2cnnn2)C)CCCN(C(=O)CC(C)c2ccccc2)C1 N1(C(C(c2cncnc2)C)=O)CCN(C(=O)CCCCNC(N)=O)CC1C1CC1 Cn1cnc2cc(C(N3CCCC3C3CCN(C(C4(C)CCC4)=O)C3)=O)cnc12 CC1COc2c(C(=O)N(CC(C)CNC(=O)Cc3sc(O)nc3O)C)cccc21 N1(C(c2cc(C)sn2)=O)CCOCCC1C(=O)NC1CNC(=O)C1 N1(C(C(COC)NC(C)=O)=O)CCC2(CC2)CC1C(=O)NOC CC(c1cccc(F)c1)=CC(=O)NCC(C)NC(c1cnc(C2CCC2)s1)=O N1(C(c2cncc(OC(C)C)c2)=O)CCCC(N(C)C(C2CCCCS2)=O)CC1 CCC#CCCN=c1[nH]c(N2CCC(CC(C)C)C2)nc2c1CCCCCC2 C(=O)(N1CCC(C(=O)NCc2ccsc2C)O1)c1cc(C)ns1 CCCC(CCCNC(=O)C(C)CO)NC(c1cc(O)nc(Cl)c1)=O C(CCCC(=O)NCCC1CC=CCC1)N(C(C(C1CCC1)OC)=O)C Cc1oc(C(C)C)nc1C(N1CCC(O)C1)=O.C1(CNC)CC1C(F)(F)F c1(C(N2CC(C3N(C(CSC)=O)CCC3)(O)C2)=O)cc(C)nc(C)c1 c1(CC)cc(C(=O)NC2CC=CCC2)c(C)cc1F CCC(C)(C)C(O)C(=O)NCC1CC2(CC2)CN1C(=O)CC1(C)CCCC1 Cc1c(C(=O)NCC(C2CC2)NC(=O)C)sc2ccc(C#N)cc12.C(C)C N1(C(c2cnc(C)o2)=O)CCN(C(C)CNC(c2scc(C)c2C)=O)CC1 Cc1nc(C2CCCC2)sc1C(N1CC(CC(C)NC(=O)C=CS(C)=O)C1)=O C1(CC(=O)N)CCCC2(CCC2)O1.C#Cc1ccc(C(=O)NC(C)C(C)C)nc1 CCCCCC(C(=O)NCC1(OC)CN(C(C2Cc3nccn3C2)=O)C1)C(C)C C(CC(C)C)(C(=O)NCC(C)(C)OCC(=O)NC)OC.C1(C#N)CCCC1 Cc1ncccc1CCNC(=O)NC(c1ccccc1)(C)C N1(C(Cc2c(C)cccc2)=O)CCc2sc(-c3ccccc3)cc2C1.C1(=O)CO1 C(=O)(C(O)CCSC)NCC(COC)NC(c1nccc(C)n1)=O C(=O)(CCCCCc1cccs1)NC1CCN(C(C(c2cnn(C)c2)C)=O)CC1 C1CC2(C1)CN(C(c1ccc(C)cc1OC(F)(F)F)=O)C2.C(C(C)C=O)OC.N CCC(CC(F)(F)F)C(=O)N1CC(N(C)C)C(CNC(=O)CCCCOC)C1 CC1CN(C(=O)COc2ccsc2)CC(C)CN1C(=O)CC12CC(C1)C2 N1(C(C(C=C=C)C)=O)CCC2CCC(C1)N2C(c1ncccc1C1CC1)=O n1(CCCC)nc(-c2ccc(CC)cc2)nc1C1CN(C(C)=O)C1 N1(C(c2c(C(C)(C)C)c[nH]c2)=O)CC2(CC(C)C2)C1.c1(C=O)sccc1C#N.N c1(OC)cc(C)c(C(=O)NC(C2CN(C(=O)C3=NOC(C)C3)C2)C)cc1Br Cn1ncc(-c2cncc(C(F)(F)F)n2)c1NC(=O)NC1CC1.c1ccccc1 N1(C(c2c(SC)ccs2)=O)CCCC2(NC(c3cnc(C(C)O)s3)=O)CCCC12 c1(C(N(CC(F)F)C)=O)cnc2n1CCN(C(c1ccc3nc(O)[nH]c3c1)=O)C2 C#CCC(C)(C(=O)N1CC2CC1C2C(=O)OC)NC(c1ccccc1C)=O CC(C)CCC(=O)NC1(C)CC(NC(=O)C(C)Cc2ccncc2)C1 N1(C(c2c(C)nn(CC)c2C(F)(F)Cl)=O)CCOC2(CCC2)C1 CC(N=c1nc2c(ncn2C)c(NCc2nc[nH]n2)[nH]1)c1csc2ccccc12 C1(C(=O)NCCN(C(c2n(C)nnc2)=O)C2CC2)CC2(C1)CC2(F)F c1(NC(c2ccc(Cl)c(Cl)n2)=O)ccc(-c2ccc(Cl)cc2)nc1O N1(C(COC(C)=O)=O)CCC(C)(NC(c2nsnc2O)=O)C1 C(=O)(C1=CCC2(COC2)OC1)N1CCC(N(C(C(F)=C(C)C)=O)C)C(C)C1 C1(N(C(C(C)N(C(c2c(C)n(C)cc2)=O)C2CC2)=O)C)CCN(C)C(C)C1 c1(C(N(CC(CC)NC(C2(COC)C=CCC2)=O)C)=O)ccc2cccnc2n1 c1(C(=O)NC2(CC=C)CCN(C(c3occc3C)=O)C2)ccnc2[nH]ncc12 Cc1nc(C)c(C(N2CCOCC(NC(C34CC(O)C3C4)=O)C2)=O)nc1C C1(NC(C2CC3(CC3)CO2)=O)CN(C(=O)C2=CCCS2)CCC12CCC2 C(=O)(C1c2c[nH]nc2CCC1C)NCCCCCNC(C(C)=CC1CC1)=O C=C=CCCC(=O)N1CCC(c2nnc(CNC(C3CNC(=O)C3)=O)s2)CC1 C(CN=c1cc(C)[nH]c(=NCC2CCN(CC(F)F)C2)[nH]1)N1C(=O)CC(CC)C1 N1(C(c2c(C)n(CCO)cc2)=O)CC2CC1CC2NC(=O)CN1CCC(C)CC1 n1(CC=O)nc(C)c(C)c1C.c1(OC)oc(C)nc1C(=O)NCC1CC1 C1(N(CC(CNC(=O)NCCOCC=C)(C)C)C)CC(OC)C1(C)C C(CCCCCC(=O)N(CC(C)C(C)C)C)NC(c1cnn(CC)c1C)=O C12(CNC(c3cccc(C(C)C)n3)=O)CC(CO1)N(C(=O)CC(O)C(C)C)C2 N1(CC)C(=O)CCC1C(=O)NC(C)(C)C1CC1.C1(C(=O)N)CCCCC1O c1(C(=O)NC(CC)CNC(c2c[nH]cc2-c2ccccc2)=O)oc(C)nc1SC c1(C2C(C(=O)OC)C2)cn(C2CCCC2NC(=O)CCC2CC2(F)F)nn1 c1(CNC(C)=O)ccc(C(=O)N)cc1F.C1C2CN(C(=O)C(C)CF)CC12.C N1(C(c2cc(C)cc(Cl)c2)=O)CCc2c(CNC(=O)CC(C)F)cccc2C1 Cn1c(=O)nc(O)c2nc(CCC(=O)Nc3nc4c(s3)CNC4)[nH]c12 C=CC1(CC(=O)NCC2(CC)CCOCC2)CN(C(C2CCC(=O)C2)=O)C1 C1(C(N2CC(C#N)(CC)C2)=O)CC2(CCN1C(=O)CCOCCOC)CC2 c1(CNC2C(C(=O)Nc3c(F)cccc3Br)C2)cc(F)cc(Br)c1Cl C1(NC(C=C(CC)CC)=O)CCSC12CN(C(C1CC1c1ccco1)=O)C2 CCCCCC(CC)C(=O)NCC1(O)CC(C(=O)NCC(C2CC2)SC)C1 c1(OCC#C)ncccc1C(N1CCC(NC(C2C=CCCC2)=O)C1)=O N1(C(C=Cc2ccc(C(C)C)cc2)=O)CCCN(C(C2CCCOC2)=O)C(C)C1 C1(C(=O)NCCNC(=O)OC)CN(C(=O)C=Cc2cocn2)CC1(C)C c1(CNC(N2CCC(F)(CC3CC3)C2)=O)cc(Cl)c(Cl)s1 CC(c1ccccc1F)=CC(=O)NC1CC(C)(C(N)=O)C1 C1(NC(CC(=O)N(C)C)=O)CCCC1O.c1(CCC=O)cnc(C2(C)CC2)o1.N CCC(CC)C(C(=O)N1CC(CO)(CNC(C23CCCCC2CCC3)=O)C1)OC c1(CNC(=O)NCCS(=O)(=O)N(CC)CC)ccc2c(n1)NCCC2 c1(OC)cc(OC2CC(O)(CO)C2)ccc1[N+](=O)[O-].c1nn[nH]c1C(C)(C)C c1(C(N2CC(NC(C=CC(=O)OCC)=O)CC2)=O)ccc(N=[N+]=[N-])cc1 Cc1ccc(C)c(C(=O)NCC(C(C)C(C)C)NC(=O)Cc2n[nH]c(C)n2)n1 c1(C(=O)Nc2cnn(-c3c(C)cccc3)c2C)ccc(P(C)(C)=O)cc1 CCC(C(=O)N1CCCC1C1CCN(C(=O)C(N)=O)CC1)C(F)(F)F C1(C)(NC(C(C)O)=O)CCN(C(c2ccccc2N2CCCC2=O)=O)CC1 N1(C(C)C)CC(NC(c2ccc(CN3CCC(F)C3)nc2)=O)C(C)C1 C1(C(N2CCN(C(CNC(C(F)=CC)=O)=O)CC2)=O)CC(C=O)C12CCC2 Cc1nc2cc(C(=O)NCC34CCC(CN3C(c3nccn3C)=O)C4)ccc2o1 C1(C(N2CC(OCC#C)C2)=O)(CC=C)CCN(C(C2CC=CCC2)=O)C1 C1(CCNC(C2C(C=C)C2)=O)CCCN(C(=O)CCC(=C)Br)C1 c1(CC(=O)NC2CN(C(C3C(C)C3)=O)CC2F)c(F)cccc1Cl c1(CCC(=O)NCCNC(c2c(C)noc2C(F)F)=O)cccc2c1OCCO2 c1(C(=O)NC(C2(O)CN(C(=O)C=CBr)C2)C)cc(C#N)c2n1CCCC2 CC1CCC(NC(=O)C(C)(F)F)CN1C(c1ccc(CO)cn1)=O C1(C=O)CCn2ncnc2C1.c1(OC)nsc(OC)c1C(=O)NC1CC1C.N c1(C(=O)NCC2CC(C(=O)Nc3ccc(C)nc3)C2)cccc(F)c1F N1(C(C2N(C(c3ccc(OCC)cc3)=O)CSC2)=O)CC2CCCC2C1 C=CCC(CC(C)C)C(=O)N1CC(C(=O)NC2C3CCCC2CC3)CC12CCC2 CCCCCCC(=O)NCC(c1cccc(C)c1)NC(C1CCCSC1)=O C=CCCCCC(=O)N1CC(O)CCC1C(=O)NCC(O)CC1CCCC1 CCC(C)(CC)C(=O)NC(C1CCN(C(=O)Cn2ccnn2)CC1)C.N(C)(C)C CC1CCC(C(=O)NCCc2csnn2)N(C(=O)CN2CC3CC3C2)C1 c1(C(=O)NC2CC3(C(NC(C(C)OCC#C)=O)C3)C2)ccc(N)cc1O Cc1nc(C(=O)NCC2(O)CCCN(C(=O)C(C)CF)C2)ccc1C#N C1(C(=O)N)CCc2nnnn2C1.Cc1n[nH]c(C)c1C(=O)NC(C)(C)C1CCC1 c1(NC(C(CC=C)CNC(C2(C)COC(=O)N2)=O)=O)ccc2ccncc2c1 N1(C(C2(SC)CCC2)=O)CCC(NC(=O)C(=Cc2cn(C)nn2)F)C(F)C1 c1(CC(=O)NC2(CC=C)CCN(C(=O)C(C#N)C(C)C)C2)ccc(OC)cc1F N1(C(C(CCSC)O)=O)CCCn2nc(C(=O)NC34CCC(CC3)CC4)cc2C1 C1(NC(C2CC23CN(C(c2cccc(Cl)c2)=O)C3)=O)CCc2ccccc2C1 c1(C(N2C(C(C)NC(=O)CCCN(C)C)CCC2)=O)ccc2c(c1)CC(=O)N2 N1(c2cc(NCC3(C)NC(=O)NC3=O)nc(C)n2)CCS(=O)(=O)C(C)C1 c1(C(C)=O)ccc(S(=O)(=O)N2CCC3CN(C(c4csnc4C)=O)CCC23)cc1 c1(OC)ccc(C(=O)NCC2(C)CCCN(C(=O)CCSC)C2)cc1O C12(C(N3CCCC3)=O)CC3CC(C(=O)N1)C2C3.C=CC1(C(=O)N)CCOCC1.C C(=O)(C1=CCCC1)NC(C)C(C)(C)CN(C)C.N1(CC(=O)N)CC2CC2C1 Cc1nc2ncc(C(=O)OC3CCCC(n4ccc([N+](=O)[O-])n4)C3)cc2o1 C1(SCC(c2ccc(N(C)C=O)cc2)=O)CCc2ccccc2C1 N1(CC#CC)CCC2(CCN(C(C3(C4CCCC4)CCNC3=O)=O)CC2)CC1 C1(CNC(CNC(=O)NC)=O)CN(C(C2(C)CC(C)=NO2)=O)CC1C Cc1cc(F)ccc1CC(=O)NC(C1CN(C(c2ccc(O)nc2)=O)CCO1)C N1(C(C2CCC(NC(C(C3CC3)OC)=O)CC2)=O)CCC2CCN(C)CC12 C1(OC)CC(O)CN(C(=O)NC(c2cc(C(F)(F)F)ncn2)c2ccccc2)C1 c1(OC)cc(Cl)cc2[nH]c(C(=O)NCCCCNC(c3c[nH]c(C#N)c3)=O)cc12 c1(C(N2C(CNC(C3(OC)CCSC3)=O)C=CC2)=O)cnn2c1C(=O)NCC2 c1c[nH]nn1.c1(C(N2CCC2)=O)cc(C2CC2)on1.C(=O)(C(=O)N)NCC N1(C(=O)NC)CCC(C(N2CCC(CC(=O)Nc3cnccc3CO)C2)=O)CC1 N1(C(CSC)=O)CCN2CCN(C(C3CN(C)C3)=O)CC2C1 c1(N(C)CC2CCCCN2C(C2CCN(C3CC3)CC2)=O)ncc2c(n1)COC2 C1(CNC(=O)CN2CSCC2=O)CC(F)CN1C(C1CNC(=O)O1)=O CC(C)(C)CC(=O)NCC(N1CCCC(c2nnc(C3CC3)n2CCO)C1)=O C=C(C)CC(C(=O)NC1CC(C)N(C(c2ccc[n+]([O-])c2)=O)C1)NC(C)=O Cc1cc(Cl)cnc1C(=O)NCC1CN(C(=O)Cc2ccc(C#N)cc2)C1 Cc1c(C(=O)NCC2(C)CCN(C(=O)C(c3ccc(F)cc3)C)C2)cccc1F Cc1sc(C(=O)NC(C)C2CC2)cc1[N+](=O)[O-].C(=O)CCCN(C)C(C)C.N CC(=Cn1ccnn1)C(=O)NC1COCC1CNC(=O)C1CCc2c[nH]nc21 C1(C2CCC2)(NC(c2ccc(C(F)(F)F)cc2)=O)CCC1 c1(C(N2CC(C)(NC(c3n(CC#C)ccc3)=O)C2)=O)cnc(C2CC2)nc1O C(=O)C1=CCC(F)(F)CC1.c1(C(=O)NCC(C)OC)ccc2c(c1)CCN2.N CC(CNC(=O)CNC(=O)C)C(C)(C)C.C1(C(C(=O)N)O)CCOCC1 CC1CCN(C(=O)C=Cc2ccc(O)cc2)CC1N(C(=O)CC12CCCC1C2)C Cc1nn(C)c(C)c1C(C)C(N1CCOC(C)C1)=O.C1(C#N)(C=O)CC=CC1.N N1(C(CC(C)CF)=O)CC23CCCCC2(C1)CN(C(=O)C(CO)N(C)C)C3 c1(C(=O)NC(C2N(C(c3c(OC)nn(C)c3)=O)CCCC2)C)c(C)ncnc1O Cc1cc(NC(=O)CC2CCCCC2F)ccc1NC(=O)CCC1CCCCC1 C(CCNC(=O)C(C)(CSC)NC(C12CCCC1C2)=O)(C(C)C)OC.O N1(C(C2CC(=C)C2)=O)CCCCC2(C1)CN(C(C1CC=CCC1)=O)C2 Cc1ccnc(C(C)(C)C(=O)N2CCC(CCNC(=O)C#CC3CC3)C2)c1 CCCCCC(O)C(=O)N1CC(NC(=O)CCc2cnn(C)c2C)C(O)C1 C1(NC(c2scnc2Cl)=O)CCSC12CN(C(c1cn3ccncc3n1)=O)C2 n1(CC(C)C)nc(-c2ccoc2)nc1-c1cnc(N2CCOCC2)s1 C(=O)(CC(C)CC(=O)NCC(C)CO)OC.N1(C(C2(C=O)CC2)=O)CCCC1 CN1CCCC1C=CC(N1CCN(C(c2ccc(-c3ccccc3F)[nH]2)=O)CC1)=O C1(C#N)(C(N(CC(=O)NC(C)C(=O)N(C)C)C2CCC2)=O)CCCC1 c1(C(N(C2CCC(NC(C(C#C)(C)C)=O)C2)C)=O)cccn2cncc12 c1(C(N2CC(N(C)C(C3C4CCC3(c3ncco3)C4)=O)C2)=O)cc2scnc2[nH]1 CC1(C)C(C(N2CCCC2)=O)C1(F)F.C1(C=O)CCN(C(=O)C(N)=O)CC1.C C(C)(C)(CC(C)C)NC(C1C(CCOC)C1)=O.C12(C(=O)N)CSCC1C2 C1(C(N2CC=C(CNC(C(=Cc3cccs3)C)=O)CC2)=O)CCn2nccc2C1 C(=O)(C1=CC2CCC(C1)C2)NC(C(=O)NCC(C#C)OC)CCOC N1(C(C2CCC(C(=O)OC)CC2)=O)CCOC2(CCN(C(=O)CC(C)(C)C)CC2)C1 Cc1ccc(Cl)c(F)c1NC(N1CCNC(c2cn[nH]c2)C1)=O CC(C)(CC(F)C(=O)NC(CO)C(N)=O)NC(=O)CCc1nccs1 Cc1cc(C)n2nc(C(=O)NC(C)C(C)(C)NC(=O)Cc3ccoc3)cc2n1 CC1CN(C(C2CC3CC3CC2C)=O)CCC1CNC(=O)C(=O)N(C)C C(=O)(N=S(C)(=O)C1CC(O)C1)c1nc(C(C)C)n2c1CCCC2 c1(C(N2CC3CCN(Cc4c(C)nn(C)c4Cl)C3C2)=O)n[nH]c2c(C)cccc12 CC1CCCN(C(c2ncc(C(F)F)s2)=O)C1C.C1(O)(CC(=O)N)CCCCC1 CCC(CC)(CC)C(=O)NC(CNC(=O)CCC1CCOC1)C1CC1 c1(CC(C)C(=O)NC2(C)CCN(c3nc(C4CC4)ns3)C2)ccccc1Cl C=C1CCN(C(c2cc(C)cc(O)c2)=O)C(C(=O)NCCCC(F)F)C1 c1(OC)cc(N)ccc1C(=O)NC(CNC(c1sccc1Br)=O)C1CC1 C1(C(N2C(CN=[N+]=[N-])CC2)=O)CC(O)(CNC(c2sccc2CO)=O)C1 N1(C(CNC(=O)NC)=O)CC(CNC(C2(C)CC(C#N)C2)=O)C(C)C1 c1(-c2cc(C(N3C(CC)CCCC3)=O)n[nH]2)ccc(=O)n(C(C)C)c1 C1(C(=O)NCC(C)(OC)OC)CCC(n2cc(C3(O)CSC3)nn2)C1 CCCCC(CC)CC(=O)NC(CC1CCOCC1)C(=O)NC1(COC)CCC1 C12(C(N(CCC(=O)NCCNC(C)=O)CC#C)=O)CC1CNC2=O n1(CC)nc(C)c2cc(C(N3CC4(CCC4)C3)=O)sc12.c1(C=O)cc(C)c[nH]1.N C(=O)(CCCC(=O)NC(C)CC)NCC.c1(C(=O)N)ccco1.N(C)CCO CC(C)(C(C)C)C(C)C.Cc1cc(C(=O)NCC2(C(=O)N)CC=CC2)ccn1 C(CC(CC)C(=O)NC1CCCCC1)=CC.C12(CC=O)CNC(=O)C(C1)C2.C C1(C(N2CC(C(C)OC)C2)=O)CN(C)CCN1C(=O)CCc1csnn1 C1(C(=O)NC(C(=O)NCC(C)C(F)(F)F)C2(C)CC2)CCC(O)CN1C C(=O)(N=c1cc[nH]cc1C)C1CCN(C(c2cc(CC)nn2C)=O)CC1O c1(C(C(=O)NC(CNC(Cc2nc(C)sc2)=O)C)(C)C)cccc(Cl)c1F CCC(CC(=O)N(C(C(=O)N(Cc1ccccc1)OC)C1CC1)C)C(C)C N1(C(c2ccc(C)c(O)c2)=O)CCN(C(=O)C(n2cc(Cl)cn2)C)C2(CC2)C1 N1(C(C2C(C)CC2)=O)CC(C(=O)N(C2CCOCC2)C)CC12CCC2 C12CCC(CN(C(C3(n4cncn4)CC3)=O)C1)C2.Cn1ccc(CC(=O)NC)n1 c1(CSCC(=O)NCC2CC23CCOC3)nc2ccccc2[nH]1 c1(NC(CSc2ccc(C)cc2)=O)ccc(Cl)c(NCCN2CCCCC2C)c1 Cc1cc(=NCCOCCS(C)(=O)=O)[nH]c(NC2CN(C)C2c2ccccc2)n1 C(=O)(C1=CCCOC1)N1CCCC(NC(=O)CCSc2ccccc2)C1 CON1CCC(C(=O)NCC2CC(NC(C3(C(F)F)CCCO3)=O)C2)CC1 C1(C(=O)NCC(CN(C(=O)CC2(O)CC2)CC)(C)C)COCCN1C N1(C(CC(C)c2ccco2)=O)CCC(O)C1C(=O)NCCCCCCO c1(CNC(c2cc(C)oc2)=O)nc2c(s1)CN(C(=O)CN1CCC(C)C1)CC2 C(=O)(C(CCCOC)NC(c1ncc(C)cc1C)=O)NC1CC(C=C)C1 CON=CC(=O)NCC(F)CNC(=O)CCn1ccnc1C N1(C(CCc2nc(=N)[nH][nH]2)=O)CCC(NC(c2cn3c(n2)SCC3)=O)CC(O)C1 C(=O)(C1=COc2ccccc2O1)NC1CCN(C(c2nc(CCC)sc2)=O)C1 C(=O)(CCC(=O)N1CC(C(N)=O)C1)N.C1(C=O)CCC(C(F)(F)F)O1.CC N1(C(C2(F)CN(C(C3OCC(C)C3)=O)C2)=O)CCC(F)(CO)CC1 N1(C(C(c2c(C)noc2C)C)=O)CC2CCC1C(NC(c1cnn[nH]1)=O)C2 c1(C(N(CCN(C(c2ccc(Cl)cn2)=O)CC)CC)=O)nc(C)oc1.N C=CCCCC(C(=O)NCC(=O)NOC)NC(c1ncncc1OC)=O CC(=O)CCCCC(=O)NC1(C(=O)NC2COCC2CO)CCC1 Cc1cccc(NC(c2c(Cl)ncn2C)c2nnnn2CCN2CCOCC2)c1 N#Cc1ccc(C(=O)NC(CCC2CC2)C=O)s1.C(CC1CC1)CC1CC1 C(CCC(C)(C)C(=O)NCc1cncc(F)c1)NC(CN1C(C)CCCC1)=O C#CC1(C)CCN(C(c2cc(CNC(c3ccncc3OC)=O)ccn2)=O)CC1 C(=O)(C1=C(C#N)CCC1)N1CCC(C(=O)NC(c2ncc[nH]2)C)OCC1 Cc1nccc(C(=O)NCC(C2CCN(C(C3CCCSC3)=O)CC2)F)c1C N1(C(CC(C)N(C)C)=O)CCOCC(C)(CNC(=O)C=Cc2cnn(C)c2)C1 N1(C(COC)=O)CCC2CN(C(c3[nH]ccc(=O)c3C)=O)CC12 c1(C(=O)NC2CC(O)CN(C(c3cc(CF)on3)=O)C2)cc2cccc(Cl)c2s1 c1(C(=O)NC(C)CNC(C2CCCC2(C)C)=O)cc(N)c(Br)c(F)c1 c1(-c2cn(CCC=C=C)nn2)ccc2c(c1)N(C(c1nnsc1C)=O)CC2 Cc1ccc2[nH]c(C(=O)NCC(C)(F)CNC(C3CC(C)(C)C3)=O)cc2c1 c1(NCc2cccc(C)c2)n[nH]c2ccc(C(=O)N=c3[nH]onc3C3CC3)cc12 C1(C(N2C3CC(NC(C(C)C4CCOC4)=O)(C3)C2)=O)CCc2ccccc2O1 c1(C(=O)NC2C(OC)CN(C(=O)CNC=O)C2)nn2c(c1C)CCCC2 CCCCC(C)C(=O)N(C)CC1(CNC(=O)C(F)C(C)(C)O)CC1 C(CN=C(NCCc1nnc(CO)s1)NCc1ccc(Cl)cc1Cl)OCC c1(C(=O)NCC2N(C(Cc3cn(C)nn3)=O)CC=C2)noc2c1CC(F)(F)CC2 c1(N2CCC(NC(C(C)NS(CCC)(=O)=O)=O)C2)nc(C)ncc1C(=O)OC C1(NC(=O)NCc2c(C(C)(C)C)[nH]nn2)CC2CS(=O)(=O)CC2C1 C1(NC(c2ccc(CCC)cc2)=O)CC2(CCCN(C(=O)C(C)(Cl)Cl)C2)C1 N1(C(c2scc(C)c2Cl)=O)CC(C(F)(F)F)OC(CNC(c2cccnn2)=O)C1 c1(CC(NNC(c2c(Cl)ccc(C)c2O)=O)=O)ccc2c(c1F)CCC2 c1(C(=O)NC2C(NC(C(C)(C)N3CCCC3)=O)C2)n[nH]c2ccc(F)cc12 CCCC(CNC(=O)C(F)(F)CCC)C(=O)NCCn1cnnc1CC CCCCCCCCC(=O)NCC1(CNC(=O)CCC(F)F)CC1 N1(C(c2c(C)[nH]nc2C(F)(F)F)=O)CCCC2(CCN(C(=O)CS(N)(=O)=O)C2)C1 N1(C(CC(=O)OCC)=O)CC(NC(c2cncc3c[nH]nc23)=O)CC(C)(C)C1 N1(C(C23CC(NC(C(C(=O)OC)C)=O)(C2)C3)=O)CCCC(C)(O)C1 c1(OC)ccc(C(N2CCCC(CNC(=O)CCC(C)C)CC2)=O)cc1Cl c1(C(=O)NCC(CNC(Cc2c(C)nc(S)s2)=O)O)c(Cl)ccc(F)c1N c1(C(=O)NCC(C)N(C)C(c2cc(C(F)F)n(C)n2)=O)csc2cncn12 O=C1Nc2ncc(Br)cc2CC1NC(=O)C(c1ccc(F)cc1)CN1CCCC1 C1(C(=O)N)C2CCN(C(C)=O)C12.C(C)(C)C.N(CCOC)(C=O)CC c1(C(=O)NC2C(C(=O)Nc3n(C)nc(O)c3)CCCC2)cc(F)c(F)c(Cl)c1 CC#CCCCC(=O)N1CCC12CN(C(=O)CCNS(=O)(=O)CC)C2 Cc1cc(C)nc(SCC(=O)NCCC2CCCN2C(c2sc(=N)[nH]c2C)=O)n1 Cc1ncc(Br)cc1C(=O)NC1CC(O)CN(C(c2cccn2C)=O)C1 C(=O)(CC1=CCN(C)CC1)N.C1(C(=O)NCc2ccc(CC)o2)CCC1(C)C C.c1(C(N(C(C(=O)N(C2CCOC2)CC#C)C)CCC)=O)cc(O)ncn1.C C=C(Cl)CC(C(=O)NCC(C)CN(C)C)NC(=O)C=Cc1cnccn1 C1(C(N(C(C)CN(C)C(C2(C)CCCS2)=O)C)=O)CN2CCCN1CC2 C1(C(N2CC(CC(C)NC(C3(OC)CCC3)=O)C2)=O)CC(C)OC(C)C1 C#CCC(C)(CC)C(=O)NCCCCN(C(=O)COCCN(C)C)C Cc1cccc2ccc(C(=O)OCC3CCCN(C(=O)C4CC4)C3)nc12 CCCC(C(=O)N1CCCC1C1CCN(C(=O)CCn2c(C)csc2=O)C1)OC Cc1nc2cc(C(=O)NC3CC(C)(NC(=O)C(CO)N(C)C)C3)c(F)cc2[nH]1 N1(C(C2CC(=O)OC2)=O)CCC2CN(C(c3sccc3-n3ccnn3)=O)CC2C1 Cc1nc(S)sc1CC(=O)NCC1(O)CCN(C(=O)C(CCO)N(C)C)C1 Cc1c(NC2CC(=O)N(C)C2)ncnc1N1CCC(CC(F)F)C1 N1(C(c2cc(CNC(CCC)=O)no2)=O)CCCCC1C(=O)OC c1(NC(C2CC(O)CN2Cc2cccc(I)c2F)=O)cccc2c[nH]nc12 c1(CC)sc(=N)[nH]c1C(N1CC(O)CC1C)=O.C(=O)C(F)(F)c1ccncc1 Cc1sc2ncnc(NC3CN(C(c4cccnc4F)=O)CC3C)c2c1C CC1CCN(c2cc(NC(c3n[nH]c(=N)s3)C)ncn2)CC12CCC2 c1(C(=O)NC(C(=O)NC2CC(CNC(C)=O)C2)CO)cc(Cl)cc(Br)c1 C12(C(=O)NC3CC(C(=O)OC(C)(C)C)C3)CCCC1C2(F)F c1(C(=O)NC(CC(C)(C)OC)C)cc2cccc(C)c2o1 c1(C(=O)NC(C2CN(C(c3cnc[nH]3)=O)C2)C)onc2ccccc12 C1(NC(CCCOC)=O)COC2(C1)CN(C(c1cccc3c1COC3)=O)C2 O=C(CCCOC1CCOCC1)NCC1(NC(=O)C(F)=CC2CC2)CC1 c1(C(N2CC3CCC(NC(CSC)=O)(C2)C3)=O)cccc2[nH]cc(Cl)c12 CS(=O)(=O)c1ccsc1C(=O)NC1CCCC1CNC(c1ncccc1N)=O Cc1cc(C(=O)NCCc2ocnc2)nn1C(F)F.C1(C=O)CC1[N+](=O)[O-].C c1(OC2CCN(c3nc(C4C(C)C4)on3)C2)ccc(F)c(Cl)c1 C1(NC(c2[nH]cnc2-c2ccccc2)=O)CN(C(=O)C2=NOCC2)CC1C1CC1 C1(C(=O)NC2C3(CC(NC(c4cnnc(O)c4)=O)C3)C2)CCCC12CCC2 c1(OC)cc(F)ccc1C(=O)NC(C1CCN(C(=O)CC2CC2(Cl)Cl)CC1)C C(=O)(CC(C)CC(C)C)N1CCC(C(C)NC(c2cn(CCC)nc2C)=O)CC1 C1(C(CNC(C2(C(=O)NC)CCC2)=O)O)CCN(C(c2cnns2)=O)CC1 N1(C(c2cn(CC3CCC3)nn2)=O)CCCC(c2cn(-c3ccccn3)nn2)C1 Cc1cc(Cl)c(Cl)cc1C(N1CCC(Cc2cn(-c3ccc(Cl)cc3)nn2)C1)=O Cc1nc(CO)sc1C(=O)NC1CCN(C(=O)C(C)(F)F)C1C(C)(C)C C1(C(N2CC(C)C(CNc3snc(Cl)c3C#N)C2)=O)C2CC3CC(C2)CC1C3 C(=O)(CC(CC)NC(=O)C(C)(C)C#N)NCCN(CCC)C(C)C N1(C(c2c(CC)noc2)=O)CCC(F)C(NC(C2CCN(C3CC3)CC2)=O)C1 c1(C(C)(C)C)nnn(CC(=O)NC2CCCC2NC(=O)C(Cl)=CCl)n1 CCCCC(CC)CC(=O)NC1CC12CCN(C(=O)Cc1ccnn1C1CC1)C2 C(=O)(C(C(C)C)C1CCC1)N1CC(CNC(C2(CC)C=CCC2)=O)C1.C C1(CNC(C2(C)CC2(F)F)=O)CC2CN(C(C3(C4CC4)CC=CC3)=O)CC12 c1(OC)cccc(F)c1C(=O)NC1(C)CN(C(C23CC(OC)C2C3)=O)C1 C1(N(CC)CC)CCN(C(C2CCN(C(C3(OC)CCCC3)=O)C2)=O)C1 CN1C(=O)Cc2c(C(N3CC(NC(=O)Cc4cc[nH]c4)CC(O)C3)=O)cccc21 C1(CNC(CC2CCCC(C)C2)=O)CN(C(=O)CCc2ccon2)CC(C)(C)O1 C1(NC(Cc2ccc(C)cc2Cl)=O)CC2CC1CN(C(=O)CCF)C2 C(=O)(C(=O)N=S(C)(C)=O)N1CCN(C(CN(CCC)C)=O)C2C1C2 N1(C(c2cn(CCNC(C3CCCC(C)C3)=O)nc2)=O)CCC2(CC=CCO2)C1 Cc1ncccc1CCC(=O)NC(C)C(C(C)C)NC(=O)C=C1CCN(C)CC1 c1(C(=O)NC(C(C2CCCCC2)NC(CCCOCC=C)=O)C)cnccc1C C#CCC(C(=O)N1CCC(CC=C)C1)NC(c1cc(CCC)on1)=O C1(NC(C(C)=CC)=O)CCC(C)(C)CC1CNC(=O)Cc1ccnn1C CCS(=O)CC(=O)NC(C1CCCC1)CNC(c1cn(-c2cnn(C)c2)cn1)=O C(=O)(CC(C(=O)OC)OC(C1CCN1CCN1CCCS1(=O)=O)=O)OC C(=O)(CC(C)(O)c1ccccc1)NCC(C)NC(C1CC(=O)C1)=O c1(-c2nc(-c3c(C)ccnn3)on2)c(Cl)nc2sccn12 C1(COC)CCC(NC(C)(C)C(=O)NCc2cn(C)cn2)CC1 Cc1cncc(CCC(N2CCOC(CNC(C3CC3c3ccsc3)=O)C2)=O)c1 N1(C(C2CC2NCc2cccc(F)c2)=O)CCC(F)(c2ccccc2)C1 C1(O)(CN(C(=O)COC2CCCCC2)C)CN(C(C2(N=[N+]=[N-])CC2)=O)C1 N1(C(Cc2n(C(C)C)ncc2)=O)CCN(C(C2CCCCC2)=O)C(C)C1C Cc1csc2c(C(=O)NCc3ccc(C)cc3)ncnc12.C1(C=O)CC(F)C1.N C1(C(=O)NCC2OCCN(C(C=CC(C)C)=O)C2)CC2(CC(=O)N2)C1 Cc1ccncc1C(=O)NCCOCCCNC(=O)C(C)(C)c1sccc1Cl Cc1ncc(Cl)cc1CC(=O)NC(C)CC(C)NC(c1cncc(O)c1)=O N1(c2n(CCCCCN(C)C3CC3)nnn2)CC2C(C1)C2(C)C CC(F)(F)CCCCS(=O)(=O)Nc1csc2nc(-c3ccc(F)cc3)cn12 C1(C(N2CC(CNC(c3c(C)snn3)=O)N(C)CC2)=O)CN2CCN1CC2C CC1=NOC(=O)C1CCC(=O)NC1CC(C)(NC(=O)CC2CSCCS2)C1 c1(CC)nn(C)cc1C(=O)NCC1COCC1NC(C1CC1(F)F)=O CCCC(CCC)C(=O)N1CCC(C(N2CCC(OCCF)C2)=O)O1 c1(C(N2C(C(C)(C)NC(=O)CCO)CCC2)=O)cc(F)cc2c1CCC2.C1CC1 N1(C(C2C(C)C2)=O)CCN(C(=O)CNC(=O)CCC(=O)c2ccccc2N)CC1 N1(C(CS(=O)(=O)NC)=O)CCC(C)N(C(C2CCc3nn[nH]c3C2)=O)CC1 N1(CC2CCN(C(=O)OCC(C)C)C2)CCC(NC(C)(C)C)CC1 Cc1nc(C=CC(=O)NCC2CCS(=O)(=O)CC2)[nH]c1C N1(C(c2c(C)coc2)=O)CCC2C(C1)CN2C(=O)C(=O)Nc1ncc[nH]1 C1(C(=O)OC)CCCN(N2CCC(Cc3ccc(C)c(C)c3)CC2)C1C N1(C(CC)=O)CCC2(CCN(C(C3(F)CC=CCC3)=O)CC2)C1.C(C)OCC.O CCC1=NOC(CC(N2CCC(C(=O)NCCCC3CCCCC3)C2C)=O)C1 Cc1ccc(Cl)c(C(N2CCC(C)N(C(=O)C#CC3CCOC3)CC2)=O)c1O CN1CCCC(CNC(=O)CCc2cncnc2)C1=O.C12(CCCCC1)C(=O)N2 C(=O)(CCC(C)(C)C#N)N1CC(Cn2cc(CN3C(C)COCC3)nn2)OCC1 C1(C(N2CCC(C(C)NC(c3cnc(CC)s3)=O)C2)=O)(CO)CCOCC1 N12C3CCC1CC(C3)CNc1nccc2n1.C1(COC)(OC)CCOCC1 N1(C(CCC)=O)CCCSC1C(=O)Nc1cnc(N2CCOCC2)nc1 c1(C(N2C3C(NC(C=CC(C)C)=O)CC(CC3)C2)=O)cccc2oc(=N)[nH]c12 N1(C(C(C=CC)O)=O)CCC(C)C(NC(c2cc(C(C)(C)C)n[nH]2)=O)C1C c1(NC(C2N(C(Cc3nnc(C)o3)=O)CC(F)C2)=O)cccc(Br)c1CO C(C1CCc2nccn21)NC(CCC1CCCN(C(C(CC(C)C)C)=O)C1)=O C1(CN(C(C=CC(CC)C)=O)C)COCCN1C(=O)CN(C)CC C1(C(=O)NCC2=CCN(C(C3N(C)CSC3)=O)CC2)CC(=O)NC2CCCCC12 C#CC1(C(=O)NC(C2CC2)C2CC2)CN(C(=O)Cc2cccnc2)C1 C1(C)(OC)CC(NC(C2CCCC2C)=O)C1(C)C.C(=O)C=O.C(C)C.N C1(C(=O)NC2C(C)(C)CN(C(c3nccc(Cl)c3O)=O)C2)CCC(=C(F)F)CC1 CCC(C)(C)CC(=O)NC1(CNC(=O)CCCn2cc(C)cn2)CCOC1 c1(C(N2CCC=C(CNC(CCCOCC)=O)C2)=O)cn2cccnc2n1 C=CCCCC(C(=O)N(C)CCc1cnc[nH]1)NC(c1ccn(C(C)C)n1)=O C(CC(C)N=c1nc(NCC(F)(F)C(C)C)c2c([nH]1)c(C)nn2C)OCC c1(C(=O)NC23CC(NC(CN4CCC(C)C4)=O)(C2)C3)cc2ccccc2cc1O n1(C(C)C)ccc(C(c2nnnn2C(C)(C)C)NC2(C(C)C)CC2)n1 N1(C(C2N(N=O)CCC2)=O)CC2(COC(CNC(c3ccccc3Cl)=O)C2)C1 C(C(C)CC(=O)NCC1(F)CC(NC(C2CC(C)(F)C2)=O)C1)OC c1(NC(C2CCCN2C(=O)COCC2CCOC2)=O)ncc(Br)c(O)n1 N1(C(C)=O)CC(C(=O)NC(C(F)(F)F)c2nc(C)cs2)Oc2ccccc21 C1CC2CCC(C1F)N2C(C1CC1)=O.S(=O)(=O)(CC(=O)N)NC.N1CCCC1 CC(CCNC(=O)Cn1cnnc1O)CCNC(c1ccc(Br)cc1)=O C(=O)(CCC(C)(C)C)NC1(CNC(c2cn(CC=C)nc2)=O)CCOCC1 N1(C(C(C(C)O)(F)F)=O)CC2CN(C(c3ccc(Cl)c(F)c3)=O)CC(C1)O2 C1(C(N2CCC(COC)C2)=O)CC2CC(=O)C1O2.C1(CC=O)CSCCO1.C CC1CC(NC(C2CC(O)C2)=O)CN(C(=O)CCc2ccccc2F)C1 c1(CC)cccc(CNC2CC(C)(C)C2c2ccccc2)c1 C1(CNC(=O)CCc2nncs2)CCCN(C(c2ccc(Cl)cc2)=O)CC1 N1(C(c2nc(C#N)c(Cl)cc2)=O)CCC(NC(C2CC23CC3)=O)C2(CCC2)C1 C1(CNC(c2cn(C)nc2Cl)=O)CCCN(C(=O)CCC2CNC(=O)N2)CC1 c1(C(=O)N)csc(S(C)(=O)=O)c1.CC(C)CCCNC(=O)CN1CCCC1C C1(CC)(CC)CC(NC(=O)C(N2CCOCC2)C)CN1C(=O)C#CC1(C)CC1 Cc1cc(N2CCCC(C)(NC(C3CCNC3=O)=O)C2)ncc1C#N Cc1cc(Br)cnc1OC(C1CCC2(CC2)N1C(=O)OC(C)(C)C)=O C1(NC(C2(CCN(C)C)CC2)=O)CC2CC(NC(c3ccc[nH]3)=O)C1C2 CCS(=O)CC(=O)N1CC(NC(c2ccnn2CC)=O)C(CC2CC2)C1 c1(C(=O)OCC)cc2cc(C(N3CC(C)C3)=O)ccc2[nH]1.C(=O)C1=CCCC1 c1(C(N2CC(C(C(=O)N(C)CC)(C)C)(O)C2)=O)nccnc1N.C(C)(C)C.O C1(NC(c2ccc(F)s2)=O)CC2C1CCN2C(c1cc(O)ncn1)=O CCCC(O)CC(=O)N(C1CCN(C(c2ccc(OC)cn2)=O)CC1)CC N1(C(C2(C)CC2F)=O)CC(O)(CCNC(c2ccnn2C2CCCCC2)=O)C1 N1(C(C(C2CCOCC2)OCC)=O)CCCCC(NC(C2(SCC)CC2)=O)C1 C(=O)(CCN(OC)C(=O)C(CCC1CC1)NC(=O)CC1CCCOC1)OC Cc1ccc(CSCC(=O)NC(CNC(c2cc(C)sc2C)=O)CO)cc1 c1sc(=N)[nH]c1C=O.C(CN(C(=O)CC1CCCC1)C)CC.C(C)=O.CC c1(C(=O)NCC(CN(C(C2CC=C(C)CC2)=O)C)C)nccc2cnn(C)c12 O=S(=O)(c1ccc2cc(Br)ccc2c1)N(C1CCCc2ccccc21)CCO N1(c2nc(C)nc(C(C)C)c2)CC2CC1CN(C(=O)Cc1sccc1C)C2 CCC(C)CC(C)C(=O)NCC1CCCCC1NC(c1cccc2nccn12)=O O=C(C1=Cc2ccccc2C1O)NCC#CCNC(C1CCn2nnnc2C1)=O N1(C(CNC(c2c(OC)scc2)=O)C(F)F)CCN(C(=O)C(C)(C)CO)CC1 C(=O)(C(F)(F)C(F)(F)C(F)(F)F)NCC(N1CCCCC2CCCC12)=O C1(NC(C(CSC)(C)C)=O)CN(C(=O)C(=O)N)CC2(CCOCC2)C1.CC(F)F N1(C(C(CC)OCC)=O)C2CCCC1CN(C(=O)Cc1cccs1)C2.C(C)=O.N c1(COC)ccccc1CC(=O)NC(C1CCN(C(C2CCCO2)=O)CC1)C C(=O)(C(CCS(C)(=O)=O)NC)NCCCN(C(=O)C#CC(C)(C)O)CC C1(NC(C(C2CC2)NC(C(CC2CCC2)OC)=O)=O)CCn2cnnc2C1 C1(NC(c2cc(C3CCC3)no2)=O)CN(C(c2ccc(Cl)c(O)c2)=O)CCC1O N1(C(c2c(C)nc(O)cc2)=O)CC2CCN(C(=O)CC3(C)CC3(Cl)Cl)C2C1 c1(C(=O)N)ccccc1N1CCCC1=O.C=C(C)CCNC(c1ccc(F)o1)=O C1(CC)CN(C(c2c(Cl)nn(C)c2Cl)=O)CCN1C(C1CCCO1)=O C1(N(C)Cc2ncoc2C(C)(C)C)CCCN(C(=O)OC(C)(C)C)C1 N1(C(C2CCCCCC2)C(=O)NCC2CCOC2)CCC(C2CCOC2)CC1 CC(C)C(C(=O)N1CC(NC(=O)C(C)N2CCC2)C1)C1CCC1 C=C1CCC(C(N2CCC(C)C2CNC(c2ccc(OC(F)F)nc2)=O)=O)CC1 c1(C(C)NC(=O)CN2CCNC(=O)CC2)ccc(S(=O)(=O)NCCO)cc1 CC(C)CCCCCC(=O)NCC1CN(C(c2ccccc2C(C)O)=O)CCO1 C1CC2(CO1)CN(C(C1CN(c3nnnn3C)C1)=O)C2.CC(C(=O)NC)C1CC1 CC1(NC(=O)Cn2ncnn2)CCN(C(C2(C3CC3)CC2)=O)C1 CC1C(C)N(C(c2cnc(C#N)s2)=O)CCN1C(=O)COC(F)F C=C(Cl)CCC(=O)N1CCC(N(CCC)C(C2CCCCO2)=O)C1 c1(C(=O)NCc2c(C(=O)NC(CCC)(C)CO)con2)cc([N+](=O)[O-])n[nH]1 CC1CN(C(c2cnoc2)C)CCN1Oc1ccccc1.C1CC2C=CC1C2 CC(C)C(CCO)NC(c1ccc(CCC(=O)NC(c2cncnc2)C)[nH]1)=O N1(C(C2C(C)CN(C)C2)=O)C2CCC1CN(C(=O)COc1ccc(Cl)cc1)C2 C1(NC(=O)CC2CCCCCC2)COC2CN(C(=O)C=CBr)CC12 S(=O)(=O)(CCCCCl)NCC1N(C(CNS(C)(=O)=O)=O)CC1 C1(c2nc(-c3ccc(OCCOC)cc3)nn2CC(C)(C)C)CC(O)C12CCC2 C1(NC(C2(CC#C)CC2)=O)CCN(C(c2c(OC)cccc2O)=O)CC1CO C(CC(C)(C)C(=O)N1CC(O)(C(F)C(=O)N(CC(=O)N(C)C)C)C1)SC C1CN(C(c2ccncn2)=O)CC1C(F)(F)F.C(=O)(CC(=O)N)OCC.C C1(NC(CCCc2cn(CCCCOC)nn2)=O)CCCCC1CCO c1(C(=O)NC(CC)CNC(c2n[nH]c(C)c2C=O)=O)cnc2n1CCCCC2.O c1(C(=O)OC2CCCC(C(C)(C)C)C2)cnc2c(c1)CCCO2 C12(NC(CN(C(C(C)SC(C)C)=O)C)=O)CCCC1OCC2 C1(CNC(NNC(c2cccc(C)n2)=O)=O)CCC2(C1)NC(=O)NC2=O c1(N2CCCC(c3nc(C)on3)C2)ccc(F)c(-c2cccs2)n1 Cc1nnc(CNC(=O)CCC2(NC(C3CC=CC3)=O)CCC2)o1 C1(C(=O)NC(C#C)CC)C(O)CCN1C(c1ccsc1Cl)=O S(=O)(=O)(c1cc(F)ccc1OC)N(CCOCC)CCOC c1(C=O)cnn2cc(C)cnc12.S(=O)(=O)(CCC(=O)N1CCC(C)C1C)NC.N CCC(O)C(C)C(=O)NCCCCCNC(c1ccc(N)cc1C)=O CC1(F)CN(C(c2cnn3ccncc23)=O)CCN(c2ncnc(Cl)c2CO)C1 c1(NCCC(CCC)O)ncccc1S(=O)(=O)NCCc1ccc(Br)cc1 c1(CC(=O)NCCCCN(C(C(C)SC(F)(F)F)=O)C)csc(Cl)c1 c1(CCNC)cn(C)nc1C(F)F.C1CCCN(C(=O)C(C)(C)C)C1.C=O.C N1(C(C(C2CCCN(C(C3(COCC)CCC3)=O)C2)C)=O)CCCN(C)CCC1 c1(-c2n(CCCC)nc(C3CN(C)CCO3)n2)[nH]c2cc(C)cc(C)c2c1C c1(C(=O)NCCCN(C(C2(F)C(C)C2)=O)C)ccnc(N2CCN(C)CC2)c1 c1(C(=O)NCC2CN(C(C(C)C3(O)CCC3)=O)CC2O)cccn2nnnc12 N1(C(C(=O)NCC23CCC(C)(C2)CO3)=O)CCc2c(O)n[nH]c2C1 C1(CCOC)(C(=O)NCCC(O)CNC(=O)C(C)SC)SCCCS1 C1(CNC(C(C)OC)=O)(OC)CCN(C(=O)C(c2ccccc2F)O)C1 c1(C(N2CCCC(N(C(=O)C(O)Cn3cncn3)C)C2)=O)ccc(Cl)c(Cl)c1O N1(C(C2CCC(OC)CC2)=O)CCC2(NC(C3CCC4(CC4)C3)=O)CCCC12 c1(CC)ccc(C(N2CCCC(O)C2)=O)c(C)n1.C1(CC=O)CC(F)(F)C1.C c1(C(=O)NCC(C2CCN(C(c3cc(CO)[nH]n3)=O)CC2)O)ccc([N+](=O)[O-])[nH]1 N1(C(Cc2c(C)nc(C3CC3)s2)=O)CC2CCOCC2C1 Cc1ccc(C(=O)NCC2CC3CC3N2C(=O)CC2(C)CCCC2)c(F)c1F CS(C)(=O)=NCC(=O)NC1CC(CNC(C2CCCC2(F)F)=O)C1 c1(N2CC=CC(NC(C3(CO)CC3)=O)C2)cc2c(cn1)C(=O)CCC2 c1(CCC=O)cc(C)n(C)n1.c1(COC)ncsc1C(N1CCC(CC)C1)=O C(=O)(C(C#N)C(C)(C)C)N1CC(CC=C)(C(=O)OC)C1 c1(C(N)=O)ncc(C(=O)NC2CCN(C(=O)CCCC3CCCC3)C2)s1 CC(C)(CC(=O)N1CC2(CCCC2NC(c2cc(Cl)cnn2)=O)C1)CC(F)(F)F Cc1nnc(NC(=O)N)n1CCCN(C(C)CN1CCCC1)C.C1CCCO1.C C1(C(N2CC3(CNC(=O)O3)C2)=O)(OC)CCS(=O)(=O)CC1 c1(CNC(C2CC(=C)CN2Cc2nc3ccccc3s2)=O)cc(C)c(F)c(F)c1 c1(NC(CC2CCN(C(C(CCOC)C)=O)C2)=O)cccc(C#N)c1 Cc1nc(Br)sc1C(=O)NCC(C1CC1)NC(=O)C=Cc1cn(C)nn1 N1(C(C(Cc2ccoc2)NC(COC(C)C)=O)=O)CCCC(C2CC2)CC1 C(=O)(CC(O)C1CCCC1)NCC1CN(C(C(C)NC(C2CCCC2)=O)=O)C1 Cc1cn2c(n1)CCC(C(=O)NCC(C1CCCC1)NC(C13CC1C3)=O)C2 c1(NC(c2n(CCC)nnn2)c2csnc2OC)ccc(-c2ccccn2)cc1 C(COC)(CC(=O)NCC1CCN(CC)C1)NC(CSCC=C)=O c1(C(=O)Nc2cc(OC)ncc2)cc(-c2cccc(C)c2)cn2ccnc12 n1(C(C)C)ccc(C(=O)NC2CCCCC2)cc1=O.C1(C=O)CCCSS1.N(C)C.N C=CC(C)(O)CC(=O)NC1(CNC(C2(F)CCOC2)=O)CCCCC1 N1(C(C(CC)CC2CCCCC2)=O)CCC(O)C(NC(C2(Cl)CC2)=O)C1 CCCC(CC(C)C)C(=O)NC(CNC(=O)Cc1cccn1C)C1CCC1 C(CC(C)(C)C(=O)NC1COCCC1NC(=O)CC12CCCC1C2)OC c1(C(=O)NC2CCN(C(CCCc3scc(C)n3)=O)CC2)cnn2c1CCC2 Cc1cc(C(=O)N(C2CC(C(=O)NCc3c(C)cnn3C)C2)C)c(C)o1 CN1CC(C(=O)OCCC2CCCCC2)CCC1C(F)(F)F c1(CC(=O)N(C(CN(CC(c2cccs2)O)C(C)C)=O)C)ccc(F)c(Cl)c1 C1(C)(CC)CCN(C(=O)Cc2csc(NS(C)(=O)=O)n2)C1 C(=O)(C1=CNC2=NCCC2=C1)NC1CCN(C(CC23C(C)(C)C(CC2)CC3)=O)C1 CC(CC(=O)N(C)CCN(C)C(C1CCC(=O)N1)=O)N(C)C C(=O)(C#CCNC(=O)CC1CC=CC1)NC(c1ccncn1)C Cc1nc(C(=O)N(C)CC2(O)CCN(C(=O)Cc3ccsn3)C2)cn(C)c1=O c1(C(N2CC(CNC(C(C=C)(C)CC)=O)OCC2)=O)cc(Cl)cc(C)c1C C1(C(N2C(C)(CC(=O)NCC(c3ccccc3)C)CC2)=O)CCN(C)CC1 c1(C(N2CCC(C(=O)N)(COC)C2)=O)cc(C)c(C)nn1.c1ccc(O)nc1 N1(C(C(C)c2cc[nH]n2)=O)CCC(C(N2CC(C)(O)C2)=O)C(O)C1 Cc1cc(C)c(C(N2CC(CNC(c3cn(C)nc3O)=O)C(O)C2)=O)c(S)n1 C1(NC(CCSC)=O)CCCN(C(=O)CC2CCC3CC3C2)CC1 C(C(F)(C(=O)NC1COC(C(C)C)C1)C(C)C)NC(CCCCNC(C)=O)=O Cc1ccc([N+](=O)[O-])cc1C(N1CCC(NC(=O)CCc2ncc[nH]2)C(O)C1)=O c1(C(=O)NCC(COC)NC(c2cnc(O)o2)=O)coc2ccc(C)cc12 n1(CCSC)nnnc1C(c1cccnc1)NC(C)(C)CCc1ccco1 C1(NC(CN(CCC)C)=O)CCC(C(=O)NCCc2cccs2)CC1 C1(CCNC(=O)NCCC2CCC3CC23)CCCCC12CCC2 N=c1ncc(C(=O)NC2CCCCC2CNC(c2ncc[nH]c2=O)=O)c[nH]1 c1(OC)cc(C(=O)NC2(C)CCC2)ccc1C#N.C(C)(c1ccsc1)=CC=O c1(N2CCCC(C)(CNC(C(C=C)O)=O)C2)ccn2c(Br)cnc2n1 N#Cc1ccc(C(N2CC3CC2CN3C(=O)Cn2ccc(Br)n2)=O)c(F)c1 C1(CNC(C2CCCOC2)=O)C2CCC1CN(C(c1ccc(O)nc1Cl)=O)C2 C1(C(C)(C)NC(C(C)SCC)=O)CCN(C(=O)CCCC2CCOCC2)CC1 c1(C(N2CC(CC)C(N3CCOCC3)C2)=O)cc2[nH]ccc2s1 c1(C(=O)NCC(CNC(C(CC)C(C)C)=O)O)cccc2oc(O)nc12 C=CC1CN(C(=O)Cc2csc(C(F)(F)F)n2)CC1NC(=O)C=C(C)Cl CC1(C)CN(C(c2ccsn2)=O)CC1NC(c1ccc(C2OCCO2)cc1)=O N1(C(C(c2cccc(F)c2)(C)C)=O)CC(C)C(F)(F)C1.C(=O)(C)N.C1CCC1 c1(OC)cc(C=CC(=O)NCC=CC)ccc1.C(=O)C=CSC.CC#N.N CC12CCN(CC1)CC2NC(=O)C(Cc1cc[nH]n1)NC(C1CCCCC1O)=O CC(C)CC(O)C(=O)NCC1CN(C)CCN1C(=O)Cn1nnc(C2CC2)n1 C12(C(N3CCC(NC(=O)Cc4ccccc4)CC3)=O)COCC(C1)C2.C(CO)N c1(C(=O)N)cccc([N+](=O)[O-])c1Cl.CC(CC(=O)NC1CC(F)(C)C1)N(C)C C1(C(=O)NCC2CCC(C#C)C2)CN(C(=O)C(C)C)CC12CC2.C(C)(=O)O N1(c2nc(NCC3=CCN(C)CC3)cc(C)n2)CCc2c(C(N)=O)cccc2C1 C123CCC(CC1)(OC2)C(=O)NC3=O.N1(CC)CC(C)C(F)C1 CC1=C(C(=O)NCC(C)(C(C)C)NC(C2CCC3(CCC3)C2)=O)CCCO1 c1(C(N2C3CC(NC(C4(CC)CC4)=O)C(C3)C2)=O)c([N+](=O)[O-])c(C)nn1C c1(C(N2CC(CCCNC(C(CC)C(C)C)=O)OCC2)=O)cccc2cncn12 CCC(C(=O)N(c1nc(-c2cccc(F)c2)cs1)C(c1ccc[nH]1)=O)C(F)(F)F C12(CNC(C3C(CNC(C4CC(=O)C4)=O)CC3)=O)CC(CCO1)C2 N1(C(C2(OC)CC(C)(C)C2)=O)CCOCC(C(=O)NCC2(C)CCCOC2)C1 CCC(C)C(O)C(=O)NCC1CC1CNC(=O)C(c1ccc(F)cc1F)=O Cc1cc(N2CCSCC2)ccc1NC(N1CCN(CC)CC1CC(C)(C)C)=O CC(O)(CC(=O)NCC1CCC(NC(C2CC23CCCC3)=O)CC1)c1ccccc1 C1(C(F)(F)F)(C=O)CCCCO1.C1(NC(C2CC(OCC)C2)=O)CCCC1 N1(C(C2(C)COC2)=O)CCCC2(C1)CN(Cc1ccc3ccccc3c1)CCO2 C(=O)C1CCc2ccccc21.N1(C(=O)COCC2CCCC2)CCCC(C(=O)O)C1 c1(CC(=O)NCC=CCC(=O)NC(CCC)C2CCC2)cnccc1C CC1CC2CCC(C1)N2C(c1cc(C2CC2)nn1C)C(=O)NC(C)(C)C Cc1ccc2c(c1)CCC(C(=O)OCc1cc3c(cc1Br)OCCO3)O2 C(C1(C)COC1)=CC(=O)NCCN(C(=O)CSc1ccccc1)CC c1(CC(=O)N(C2CCC(NC(C3(C(=O)NC)CC3)=O)C2)C)cccnc1Br C12(C=O)CC3CC(C(=O)N1)C2C3.C1(C=O)CCS(=O)(=O)C1.C1CCCC1.N C1(NC(Cc2cncc(C)c2)=O)C2CCN(C(=O)CCc3cnoc3)CCC12 CC1(C2CC2)CN(C(C2CCCN(CCOC3CCC3)CC2)=O)CCO1 c1ccc([N+](=O)[O-])cc1.c1(OC)nsc(OC)c1C(=O)NC(C)C=O.CCO.O C(C(=O)NC(C)CCc1cn[nH]c1)(C(C)C)NC(C(COC)N(C)C)=O c1(C(=O)NCC(C)N(C(=O)CC#N)C)ccc(OC2CCOC2)cn1 Cc1cc(CNC(=O)CC(C)(C)NC(=O)CC2CCCN(C)C2)oc1C N1(C(c2c(C)nsc2)=O)CCN(C(=O)CCN(c2ccccc2)C)CC(O)C1 C(=O)(C(C(C)(C)C)C1CCC1)N1CCC(N(C(C(F)=CC)=O)CCC)C1 N1(C(CC=CC=C)=O)CC2CCN(C(c3csc(C)c3C)=O)CCC2C1 c1(NC(c2nc(NC(c3ccc(C)nc3Br)=O)sc2)=O)c[nH]c2ncccc12 C1(C)(CC(=O)NCCNC(C(C)C)=O)CCN(C(c2cnc(S)nc2)=O)C1 C1(CNC(=O)C2=COCC2)CC2CCC1N(C(=O)CC(F)(F)C(F)F)C2 Cc1ccc2c(c1)CCC2C(=O)NCCCCC(C)NC(=O)C=CCF NC(=O)CC(O)C(=O)NCC(CNC(c1ccccc1Oc1nccs1)=O)CO C1(C)(CC#C)CCCN(C(c2cccc(C(=O)OC)c2)C(=O)NCC(=C)C)C1 C(=O)(C1=CCCOCC1)N(C(CCNC(c1c(OCC#C)nccc1)=O)C)C c1(C(=O)NCC2CC(OC)CN2C(c2sccc2SC)=O)ccc2nnnn2c1 C(CN=c1cc(C)nc(CC)[nH]1)C1CCCN(C(CCCOCC=C)=O)C1 C1(C(=O)NC2(CO)CN(C(c3c(C)ccnn3)=O)C2)CS(=O)(=O)CC(=O)N1 Cc1cccc(F)c1C(=O)N(CCCOCC)C.C(=O)C=O.CC(F)(F)F.N c1(CN2CC(CC(=O)Nc3ccc(C)cc3Br)OCC2)ccc2occc2c1 CCC(C)C(C(=O)NC(CO)CCO)N(C(=O)C=Cc1cc[nH]n1)C C(CCC(F)(F)F)NC(C(CC=C)NC(C)=O)=O.c1(C=O)ncoc1C1CC1 N1(C(CCOCCC)=O)CCC(CCC(=O)NCCOCC(=O)OC)CC1 C1(C(N(C(C)CNC(=O)COC(F)F)C)=O)CCN(c2ncccn2)CC1 C1(C(=O)NC(CCNC(c2cc(C)[nH]c2)=O)C(C)C)CCc2ccccc2O1 C(=O)(CCC(=O)OC)N(CCNC(CCCOCCC)=O)CC.C(C)=O.N C1(CC=O)CCc2nncn2C1.N12CCCCC1C1(CC2=O)CC1.NC(=O)CS C1(C(N(CC)CC2CC2)=O)CC2(CCC2)C1.C1(CC=O)CC(C)C1.N N1(C(CCc2cc(C)n(C)n2)=O)CC(CNC(=O)CCC(F)(F)F)CC12CCC2 C1(F)CC2C=CC1C2.C1(N(C)C(=O)OC(C)(C)C)CC1CNC=O C1(NC(C2CC23CCCC3)=O)CCCC12CN(C(=O)C(O)C1CCCC1)C2 C(=O)(C1=Cc2cc(F)ccc2OC1)N1CCC2OCCN(C(C(C)OC)=O)C2C1 c1(N(C2CCC3(CC2)CNC3)C(C(C)(C)O)=O)nc2ccc(F)cn2n1 C(COC(C1C(COC)(COC)C1)=O)C=O.C1(CO)CC(F)(F)C1 C1(C(N(C)Cc2ccccn2)=O)CCC(C2CC2)N1C(=O)Cc1cnns1 N1(C(Cc2cc(C)on2)=O)CC2(CC2C(=O)NCCC2CCCCCC2)C1 c1(C(C)O)nc(C2CC3CCC2C3)n(Cc2ccccc2Cl)n1 C(CF)(C(F)(F)F)NC(C1C(CNC(=O)CC2OCCO2)CC1)=O C1(=O)C(F)(F)S(=O)(=O)N2CCCC2CN1.N1(CC(=O)OC)CCOCC1 CN1CC(C(=O)NC(CO)C(=O)NCCC(C)(C)C2CC2)NC1=O N1(C(c2c(C)n(C3CC3)cc2)=O)CC2CCC(CNC(=O)C3=CCSC3)C2C1 c1(C(C)C)nnnn1CC(=O)NCC(C)(C)CNC(=O)Cc1cnoc1 C1(CNC(=O)CC2C=CCCC2)CN(C(c2cncc(F)c2)=O)CCC1(F)F c1(OC)cc(OC)cc(CN2CCN(C(C3(C#N)CCC3)=O)CC2C(C)C)c1 N1(C(=O)NC(CC)C(C)NC=O)CCOCC12CCS(=O)(=O)C2.C(C)(C)C.O C=CCC(C)(C)CC(=O)N1CC(F)CC1CNC(c1ccc(C(=O)CF)cc1)=O C12(C(=O)NC(CNC(CCc3c(C)noc3C)=O)(C)CO)CCC(C)(C1)OC2 C(CN=c1nc(N2CC3C4C=CC(C4)C3C2)c2c([nH]1)CCC(C)C2)OCC(=C)C S(=O)(=O)(C1CC2CC1C2)Nc1cc(-c2onc(CC(=O)NC)n2)[nH]n1 Cc1cc(C(=O)NC(COC(C)C)C(=O)N)c(C)cn1.c1(CC)n[nH]cn1 C1(C(=O)NCCOCCCNC(CCc2cnc(C)s2)=O)CCOC1(C)C c1(NC(CC(C)CNC(C2(CO)CCCCO2)=O)=O)cccc(F)c1O C(=O)(CCCCCCNC(c1c[nH]nc1C)=O)N1CCC(O)(CC)CC1 c1(C(=O)NCC(C(C(C)C)C)Nc2ccnc(F)n2)ccc2c(n1)NCC2 C1(NC(C=C(CC)C)=O)CN(C(=O)C(C)(C)F)CC1OCC N1(C(C=C(C)C2CC2)=O)CCCC2CN(C(c3nocc3C(C)C)=O)CCC12 Cc1c(CN2CCCC(NS(=O)(=O)c3ccc(Cl)cn3)C2)nc2ccccn12 C(=O)C(CC(C)C)n1ccc(C2CC2)n1.C(C)(C(=O)NC1CC1)=C(C)C.C c1(C(=O)NC2C(NC(c3ccn(C(CC)CC)n3)=O)C2)cscc1S(C)(=O)=O N1(C(C2C(=C)C2)=O)CCCC(CNC(c2cc(C(C)C)ccc2C)=O)CC1 CC1(C#CC(=O)NC(CNC(=O)C#CC(C)(C)O)C(C)(C)C)CC1 Cc1nc(Cl)ncc1NC(C1(C)CCCN1C(c1cc(Br)cs1)=O)=O C1(NC(CNC(=O)OC)=O)CCC(NC(c2c(C(C)C)cnn2C)=O)CC1 N1(C(COc2c(C#N)cccc2)=O)CCC2C1CCCN2C(c1cc(F)c[nH]1)=O N#CC1CN(Cc2ccsc2Br)CCN1C(c1ccc(O)nc1)=O n1(CC)nc(C(N2CC(NC(=O)Cc3cccc(F)c3)C(O)C2)=O)ccc1=O C(=O)(CCCCCCCN)Nc1c(C(N)=O)cc(I)c(F)c1 O=C(CC1OCc2ccccc21)NCC(CO)NC(=O)Cc1cnns1 C(=O)(C(N)CP(C)(C)=O)NC(CCc1ncno1)CCO.CS n1(CC(=O)NCCCC(C)NC(c2ncc(C(F)F)s2)=O)ncc2ncccc12 CC1(NC(C2(CO)CCN(C(C3CC4(CC4)C3)=O)C2)=O)CCCC1(F)F C1(OC)CN(C(=O)C(C)(C)C2CCOC2)CC1C(=O)NC(C)C(O)C(F)F c1(C(=O)NCC(C)NC(CC2(CSC)CC2)=O)cccc2cc(F)ccc12 C(=O)(CC(C)(C)C(F)F)NC(CCCNC(COCC#C)=O)C C(=O)(C1=NOC(C)(C)C1)N(C1CCN(C(c2cccc3ccnn23)=O)C1)CCC C1(C2C(C(=O)NC3(C)CC3)C2)COCCN1C(=O)COCC(F)F C12(CC(=O)NC3CC(CCNC(=O)Cc4ccns4)C3)CCCN1CCC2 Cc1cn[nH]c(=NC(=O)c2ccc(C3(NCc4cc(Cl)cnc4F)CC3)cc2)c1 C(=O)(C(C#N)C(C)(C)C)N1CCC(CC)C1.c1(OCC)ccc(Cl)nc1C=O C1(CN(C)C(C2CCOCC2)=O)CCCCN1C(=O)CC1CCCOC1 c1(C(=O)NC2(CC)CN(C(=O)C(F)n3ccnc3)C2)cc(C)ncc1C C(=O)C1=CC2CCC(C1)C2.c1(C(N2CC(COC)C2)=O)cc(C)c(Cl)s1.C Cc1cc(N)cnc1C(=O)NC1(C(=O)Nc2ccc(Cl)nc2C)CCC(C)(C)C1 c1(C(=O)NCC2N(C)CCN(C(c3cnn(C)c3Cl)=O)C2)coc2ccccc12 Nc1cc2c(cc1C(N1CCOC(CNC(c3cnsn3)=O)C1)=O)OCO2 N#Cc1ccsc1C(=O)N(c1ccc[nH]1)Cc1cn(C2(C(=O)O)CC2)nn1 C1CC2(CCN(C(c3nc(Cl)c(Cl)s3)=O)C2)CO1.C1(C(=O)N)CCCC(O)C1.C c1(CC(N2CC(C)C(CNC(C3SCCS3)=O)C2)=O)ccc2occc2c1 c1(NC(C)=O)cncc(C(N2CCC(NC(=O)C=CC3CC3)CC2)=O)c1 C1(C(=O)NC(c2onc(C)n2)C)CCC(C)CN1C(=O)C(C)NC=O C(=O)(C#CC1CCC(=O)CC1)N1CC2CC(NC(C(C(C)C)O)=O)CC2C1 C1(COC)CN(C(=O)COc2ccccc2)CCN1C(c1cc(O)ccc1O)=O c1(OC)cc(NC(=O)CC2CCN(C(C)=O)CC2)ccc1Cl c1(C(N(CCC(C)NC(C(C)=CC)=O)C)=O)ncc(C(F)F)s1 C(C(C)(COC)C(=O)NC1CC(C(C)NC(c2cc(O)nn2C)=O)C1)OC c1(C(=O)N)cnc(S(C)(=O)=O)s1.C12(C=O)COC(CCO1)C2.CC(C)(C)C N#Cc1cc(C(N2CC3CC(NC(c4cc(Cl)on4)=O)CC3C2)=O)cc(O)c1 C(CC(C)C)(C(=O)NC)N(C(c1nccc(OC)c1)=O)C.c1cc(C)cc(F)c1 N1(Cc2c(C)nccc2)C(=O)CCN(CCC2CNC(=O)C2)C1=O Cc1ccc(C(=O)NC2CC3CCC2CN3C(C23C=CC(CC2)C3)=O)c(F)c1F CC1CCC(O)(C(=O)NC2C=CCC(C(=O)NCc3cccc(O)n3)C2)CC1 C1(c2n(CCOC)nnn2)(Nc2ccc[n+]([O-])c2)CCCN(C2CC2)C1 c1(CC(=O)N(CCNC(C2CCCC(C(N)=O)C2)=O)C)cnc2ncccn12 c1(Cn2cc(-c3scc(C)n3)nn2)cc(C)ccc1F C1(CNC(c2cnc(CC)o2)=O)CC(F)CN1C(=O)CC1CCCNC1=O C1(C(=O)NCC(C2CC2)NC(c2cccc(C)n2)=O)CC(=O)NC(C)C1 Cc1c(Cl)cnn1CC(N1CCCC(C(C)N)C1)=O N#CCCCC(=O)NCc1cncc(C(=O)NCC2CC23CC3(F)F)c1 C(=O)(C1COc2ccc(Br)cc21)N1C2(CNC(C3(C)CC3)=O)CC(C1)C2 C#CC1(O)CC(C(N2CC(NC(=O)C(C)=CC)CC2CO)=O)C1 Nc1c(C(N2CC3CC(NC(=O)Cc4cnns4)C(C3)C2)=O)ccc(F)c1F C1(CNC(C(CCC)F)=O)CN(C(C2CC23CCC3)=O)CC12CC2 CC1(C)CCC(=CC(=O)NC2CN(C(C3CN(C4CCOCC4)C3)=O)CC2F)CC1 C1(C(=O)N(C)Cc2c[nH]nc2CC)CC=C(C)CC1.C1(C(C)=O)CCC1C=O CCC(CC(=O)NCCOCCN(C)C)N(C(=O)C(C)C1CCC1)C N1(C(C(C)Cc2cccc(Br)c2)=O)CC2CCC(C1)C2C(=O)Nc1cnc[nH]1 c1(N(CCCC(=O)N2CCOCC2)CCO)c([N+](=O)[O-])cccc1[N+](=O)[O-] c1(OCC(=O)NC(CC)CNC(=O)C(CC)N(C)C)c(F)cccc1F Cc1cc(C)c(C(N2CC(O)CC2CNC(C2(C)CC=CC2)=O)=O)cc1C n1(CC)ncc(C=O)c1Cl.C1(CC)CCN(C(c2nn[nH]c2C(F)(F)F)=O)C1.N N1(C(CC)=O)CSCC1C(=O)N(CCCNC(c1ccc(-c2cccs2)[nH]1)=O)C C=CCC(CC(=O)NC1(C)CC2CCC1C2)NC(=O)C(C)C(O)CC c1(C(N2C(CCNC(c3ccc(OC)cc3)=O)CCC2)=O)cc2occc2[nH]1 n1(CC(=O)NCC2CC(NC(c3cccc(F)c3O)=O)C2)ncc(O)nc1=O c1(C(N2CCN(C(c3[nH]c(=N)sc3)=O)C(CC(F)F)C2)=O)ccc2c(c1)CCO2 c1(CN2CC3CCN(c4cc(SC)nc(C)n4)C3C2)ccc2ccn(C)c2c1 c1(OC)c(C(=O)N(CC(O)CN(C(=O)C(O)C2CCCC2)C)C)cnn1C N1(C(Cn2c(C)csc2=O)=O)CCN(C)CC1C.C1(CC=O)CCC(=O)NC1.N c1(N2CC3C(NC(C4CC5CCCC45)=O)C3C2)ncc2c(n1)COC2 CN1CCCCCC1C(=O)NCC1COCCN(C(=O)Cn2cnc(=N)[nH]2)C1 N1(C(C2C(=C)CC2)=O)CCN(C(CNC(=O)C(C)CCO)C(F)(F)F)CC1 CCC(COC)(CC)C(=O)N(CCNC(C1CC1F)=O)C1CC1 c1(N(C)Cc2scc(C)n2)nc(=N)nc(N2CCC(NS(C)(=O)=O)C2)[nH]1 C1(CNC(C2CNC(=O)N2)=O)CC(F)CN1C(=O)C.c1(C(C)=O)ccccc1 C1(CNC(=O)C#CC2CC2)CN2CCCCC2CN1C(=O)C=Cc1ccccn1 C1(n2cc(CC(C)O)nn2)CCC(C(=O)NCc2cccc(I)n2)CC1 CC1Oc2c(C(N3CC(NC(c4ncccc4Cl)=O)C3)=O)cccc2C1C CC1CN(C(c2cc(C3CC3)cs2)=O)CCC1NC(=O)C1=NNC(=O)C1 n1(CCCC)ccc(C(N2CCCC2C(C)NC(C2CCCC2C(C)C)=O)=O)n1 c1(OCCNC(=O)OC2CCCC2c2nc[nH]n2)ccc2c(c1)CCCC2 C(C)(CC)C(F)(F)F.C(C(C(=O)N)NC(=O)COC1CCOC1)OCC c1(NC(C2N(Cc3c(C)ccs3)CC(O)C2)=O)ccc2ccnc(O)c2c1 N1(C(CCC=CCC=C)=O)CC=C(CCNC(=O)CC2CCCCC2O)CC1 C#CCCC(C(=O)NCc1ccc(C)s1)NC(c1scc(C)c1C)=O c1(C(N2C(CNC(c3ccc(C)cc3)=O)C(C)CC2)=O)cc(F)c(Br)cc1N Cc1cc(C(=O)NC2COCCN(C(=O)Cn3ccnc3)C2)ccc1OC(C)C C1(CC(=O)NC(c2c[nH]nn2)(C)C)(COCC)CCOCC1.c1ccccn1.C C1(C(=O)NCC2C(NC(c3nc(CCC)oc3)=O)C2)CC2CCC1O2 C1(C(C)C)C(C=O)CCN1C(=O)CC(C)O.C1CC(=O)N1C.C1CC1 C1(CNC(CNC(CCC)=O)=O)CCC(C)N(C(c2cn(C)ccc2=O)=O)C1 C1(NC(C2CCC(C(F)(F)F)CC2)=O)CN(C(=O)CC2CCOCC2)C2CC12 C(=O)(C1OC(=O)c2ccccc21)N1CC=CC(NC(c2cnc(C3CC3)o2)=O)C1 N(C1CCCc2cc(OC)ccc21)C(CONC(c1cc(CCC)on1)=O)=O C=CC(CCC)CC(=O)NCC1CN(C(c2occc2COC)=O)CCN1C C1(CNC(C(c2ccc(CC)s2)=O)=O)CN(C(c2ncc(Cl)n2C)=O)CC1C c1(OC)ncc2c(n1)CN(C(c1nc(-n3nc(C)cc3C)ccc1Cl)=O)C2 N1(C(c2n[nH]c(C)c2C(F)(F)F)=O)CCN(C(=O)C(C)CN(C)C)C(C)C1 c1(C(=O)NCCN(C(C(CC(CC)C)C)=O)CC2CC2)cnc2ccnn2c1C c1(NC(c2ncc(OC)nc2)=O)sc2c(c1C=O)CCC2.CCS(C)(=O)=O.N c1(NC(C2C(c3nc(C)[nH]n3)C2(C)C)=O)ccnc2c(Cl)c(C)ccc12 c1(CNc2cn(C)c(C(=O)NCc3cccc(CO)n3)c2)cccc2[nH]ccc12 Cc1cc(Br)c(F)cc1C(=O)NC1CCCN(C(C2(C)CCC2)=O)CC1 C1(c2ccc(C)cc2)C(C)CCCN1C(=O)Nc1cn(CCCCCC(C)C)nn1 C1(CNC(C(C)C(F)(F)F)=O)CCC2(CCC2)CN1C(=O)CC1CCCOCC1 N1(C(C(CNC(=O)CC2CC3CC3C2)OC)=O)CCCC(C2(C)CC2)C1 CC1(C)CCCC1C(=O)NCC1CCCN(C(=O)CCCSC(C)(C)C)C1 N1(C(CCS(N)(=O)=O)=O)C(CNC(=O)Cc2ccc(F)cc2)CC2CCCCC12 C1(NC(=O)CC2CCNC2=O)CC(F)CN(C(c2cccc(Br)c2)=O)C1 C1(F)(C(N2CC3C(CC(=O)N(CC=C)C)C3C2)=O)CCC(C)CC1 C1(N(C(c2scc(C(C)=O)c2)=O)CCO)CCN(CC23CC(C2)C(C)O3)CC1 N1(C(C(C)CC2CC2)=O)CCOC2(CCN(C(C3CC(C)(C)C3)=O)C2)C1 c1(C(C)OC)nc(C(=O)N(C(C)CNC(=O)CS)C)co1.c1ccccn1 C1(NC(C(C(C)C)C)=O)CCSC12CN(C(=O)C(F)(F)c1cnnn1C)C2 N1(C(CN(C(=O)OCC)C)=O)CCCC(CC)C1.C1(C)(C(=O)N)CCCOC1 N1(C(C2CC(C)SCC2)=O)CCC2(C1)CN(C(c1cccc3cc[nH]c13)=O)C2 c1(C(N2CC3(CN(C(CC4CC(C(=O)OC)C4)=O)C3)C2)=O)ccc2cccnc2n1 N1(C(C2CCC(C#C)CC2)=O)CCCN(C(=O)COCc2ncnn2C)CC1C N1(C(CNC(C)=O)=O)CCC(NC(c2cnc(O)s2)=O)C12CCC2 C1(c2cn(CC3C(CNC(=O)CCCn4cccn4)C3)nn2)CC2CCC1CC2 N1(C(C(C)(C)C)=O)CCC(CO)(NC(=O)CNC(C2CCC(=O)N2)=O)C1 C1(CNC(CC2(NC(C=CC)=O)CC2)=O)CCCSC1 N1(C(C2N(N=O)CCCC2)=O)CCC2CN(C(C34CCC3CC4)=O)CCC12 C1(NCC2Cc3n(C)ncc3CC2)CCc2ccc(F)cc2C1 C1(CNC(CCOCC(C)(C)C)=O)CCN(C(=O)C(F)(F)c2cccnc2)C1 N1(CCCC)CCC(C(=O)O)(CNC(=O)Cc2c[nH]nc2C(F)(F)F)CC1 O=C(CC(C(F)(F)F)c1c[nH]c2ccccc12)N1CCC12CCCOC2 n1(CC)cc(CC(=O)NC(CO)C(C)NC(c2ccn(C3CC3)n2)=O)nn1 c1(C(=O)NC2(C)CCN(C(c3c(C)[nH]c(C)c3C)=O)C2)csc2c(F)cccc12 CC(C)CC(O)C(=O)N1CCC1CNC(C1(CN2CCCC2)CCCC1)=O CC1CCN(CCNC(C2CCCC2NC(=O)Cc2ccccc2Br)=O)CC1 C1(CC(=O)NCC(CC)(C)NC(=O)CC(C)(C)N(C)C)OCCOC1(C)C c1(C(N2CCCC(NC(C3(C)CC=CCO3)=O)C2)=O)cc(N)c(Cl)cn1 c1(C=O)nnc(O)nc1O.CC1CCCN(C(=O)C(=O)NC2CC(F)(C)C2)C1.N C1(CNC(c2cnc(C(N)=O)s2)=O)CCC(F)C1.C1(C=O)CC2CCC2C1.C CC(C)CC(CNC(=O)CC(C)CC(C)C)C(=O)NCc1ccc(F)c(O)c1 N1(C(c2c3cc(C)nn3ccn2)=O)CCCC12CCCN(C(=O)C1=CCCC1)C2 N1(C(C2C(C(C)NC(c3cccc(C)c3C)=O)C2)=O)CCOC2C(O)CC12 N1(C(c2nnn(CC)c2C)=O)CCC(N(C(=O)CCCc2nccs2)C)C(C)C1 C1(C)(C(=O)NCC2(OC)CN(C(C3CCCN3C=O)=O)C2)CCOCC1 c1(N(CC(N2CCC(F)(C(N3CCC(Br)C3)=O)C2)=O)CC)ccc(F)c(F)c1 N1(C(c2nc(COC)oc2)=O)CCOC2CN(C(=O)CCC3CCCOC3)CC12 Cc1cc(Cl)nc(Cl)c1C(=O)NC1CC(C)CN(c2ncncc2Br)C1 c1(C(N2CC(F)(CC)C2)=O)cncc(CNC(=O)CC2CC2(C)C)c1 Cc1nc(Br)ccc1C(N1CCC(CNC(=O)Cc2ccc(Br)cc2)C1)=O CC(C)C(C)C(=O)N1CC(NC(c2cccc(-c3nnco3)c2)=O)CC1C c1(CNC(C)Cc2c[nH]c3ncccc23)ccc2c(c1)CCCO2 C1(C(N(CC(C)O)CCNC(c2coc(Cl)n2)=O)=O)COCCN1C Cc1occc1CC(=O)N(C1CCC(NC(c2coc(Cl)c2)=O)C1)C C1(NC(C(c2ccc(C)cc2)C)=O)CC2CC1N(C(C13CC(C1)C(C)O3)=O)C2 c1(OC)cc(-c2cccc(CN3CCN(C(C4(C#N)CCC4)=O)CC3)c2)ccn1 n1(CCOC)cc(C(=O)NCCC)c(C)n1.C1(CC=O)CC(C(F)F)C1 S(=O)(=O)(c1cc(Br)c(F)cc1F)N1CC2C(C(=O)Nc3n(C)cnc3)(C2)C1 Cc1nn(C)c(-n2cncn2)c1C(=O)N.C(=O)(CN=S(C)(C)=O)N1CC2C(C2)C1 N1(C(c2c(CC)[nH]c(=N)s2)=O)CCN(C(=O)C(C)N(C)C(C)=O)CC1CF Cc1cnncc1C(=O)NCC1(C)CC12CCC2.C(=O)(C)N.C(C)(C)C Cc1ccc(N)c(C(N2CC3CC3(NC(C3(F)CCOC3)=O)C2)=O)c1F C1(NC(CN(C)C2CC2)=O)CN(C(=O)CCC(C)(C)C)CC12CCC2 Cc1cccc2oc(N3CCC(C(C)NC(=O)CCc4cn(C)nn4)CC3)nc12 C12(CNC(CS(CC)=O)=O)CCCC1CN(C(c1c(C)cc(O)nc1C)=O)C2 CC(C)(C#N)C(=O)NCCN1CCC(C)(F)C1 C1(CNC(C2CC(C(C)C)C2)=O)C2CN(C(=O)C(F)(F)C3CCCC3)CC12 Cc1cnc(C(=O)NCC2(NC(=O)C3CC3)CCOCC2)cc1Cl C1(C(=O)NCC#CC(=O)NC(C)CCN2CCCC2)(OC)CCOCC1 C#CCCCC(C)C(=O)N1CCCC(CC=C)(C(N2CC(N=[N+]=[N-])C2)=O)C1 CC12CC(C=O)(CCO1)C2.C1(CCC)CCN(C(=O)CC2(C)CC2(F)Cl)CC1.N C1(C(=O)OC)CCC2(CCCC2)N(Cc2c(F)ccc(F)c2Cl)C1 N1(C(C2(OCC)CC2)=O)CCCC(C)C1.c1(C=O)cnn(CCN(C)C)c1 c1(-n2c(NC(C(=O)NCCC3(O)CCOC3)=O)ccn2)ccc(Cl)cc1 N1(C(C=CC(CC)C)=O)CC(CC(N2CCC(NC=O)CC2)=O)C2(CC2)C1.O c1(C(NOCC2OC(C)(C)C(F)(F)CC2)=O)cc(Br)c(O)c([N+](=O)[O-])c1 CCC(C)C(C(=O)N1CCC(O)(C(C)NC(=O)COc2ccn(C)n2)C1)OC C(C(C)(C)C(=O)N(C)CC1CCCN1C(c1ncccc1F)=O)OC N1(C(C(C)Sc2ccccc2)=O)CCC2(CC1)CC2(C#N)CO C1(C2CCC2)(C(=O)NCC2(CNC(C(C)(C)F)=O)CC2)CCC1 c1(C(=O)NCCCNC(CN2CCCC(CC)C2)=O)ccc2c(O)nccc2n1 CC1=C(CC(=O)NCc2ccc(C(C)=O)cc2)c2ccccc2C1 c1(C(=O)NCC=CCNC(=O)CC2CCOCC2)ncnc2c1OCCO2 CC(C)CCC(=O)NC(Cc1ccccc1)CCNC(C1(C)CCSCC1)=O c1(C(N(C)CC2CN(c3ncnc4n[nH]cc34)C2)=O)ccc2c(cnn2C)c1 C(=O)(C(C)(C)C(C)NC(c1cnco1)=O)NCC1CCN(CCC)C1 C(=O)(C1=CCOCC1)NCC(CCOC)NC(=O)Cc1sccc1Br C1(C(=O)NC2CC(C)N(C)CC2)CC2(C1)CC(C#N)C2 c1(OC)ccc(F)c(C(N2CCC2C)=O)c1.c1(C(=O)N)cn(C)c(=O)cn1 c1(C(=O)NCC(CNC(c2onc(CC)c2C)=O)C)cc2ccccc2[nH]c1=N Cc1nn2cc(C(N3CCN(C(c4cccc(Cl)c4O)=O)CCC3C)=O)nc2s1 n1(CC(=O)NC2(C)CC(NC(=O)CCc3cccs3)C2)ncc(O)nc1=O C1(CNC(Cc2c(OC)nccc2)=O)CCCCCN1C(=O)CC(C)C CCCC.C(=O)C=CC1CC1.C(=O)C=CC=O.C(C)(C)C.C(N)=O.N Cc1ccc(F)c(S(=O)(=O)N2CCN(C(c3cc(Br)c4cn[nH]c4c3)=O)CC2)c1 C(=O)(C(CNC(c1cc(Cl)n[nH]1)=O)CC1CC1)N(C)Cc1cncn1C c1(C(=O)NCC23CN(C(CC(C)OC)=O)C(CC2)CC3)coc2c1C(O)CCC2 c1(NC(C(=O)NC)=O)ccc(C(C)=O)cc1C(C)C.C1(C)CCC(=O)O1 c1(NC(=O)C2=CCN(C(=O)C#CC3CC3)C2)ccn2nccc2c1 C(CCN=C(NCc1nc(C(F)(F)F)cs1)NC1CCCC(C(C)C)C1)OC c1(CNC(C2N(C(C(CC)O)=O)CC=C2)=O)ccc(F)cn1 C1(CNC(=O)Nc2cccc(-n3c(C)cnc3O)c2)CCCN(C(=O)CO)CC1 C(=O)(C(CCOC)NC(=O)CC1CC2CCC1O2)N(CC(=O)NCC)C CCC(C)(CNC(C1CC(Cl)(Cl)C1)=O)NC(=O)C(COC)OC N1(C(c2cn(CC=C)nc2)=O)CCC2C(NC(=O)Cc3ccc(F)cc3)C12 c1(C=O)cc2n(n1)CC(F)C2.N1(CC(=O)N)C(=O)CNC1=O.C(CCC)OC N1(C(C2(F)CC(C=O)C2)=O)CC(C)CN(C(c2cc(F)c[nH]2)=O)C(C)C1.CC C1(C(C)C)CCN(C(=O)Cn2nnc(=N)[nH]2)C1.c1(C=O)nc[nH]c1C(F)(F)F C1(C=O)CCC(C)(O)CC1.C(C(=O)NCC(=O)N)NC(C)=O.C1CC1.C C1(C(N2CCNC3(CC3)C2)=O)CC2(CC2)CN1S(=O)(=O)Cc1ccc(Br)cc1 CC1(NC(=O)CSC2CC2)CN(C(C2(c3ccccc3)CC2(C)C)=O)C1 c1(C(=O)NCC(C)NC(C(CC)(C)CC)=O)cn(C)c(C)c(Br)c1=O c1(CC)cc(C(=O)NC(COC)C(=O)NCCCC2CCCCC2)ns1 c1(C(=O)NCC(C)NC(Cc2n(C)nc(CC)c2Br)=O)cnc2[nH]ncc2c1 c1(CC)nn[nH]c1C(=O)NC(Cc1cn[nH]c1)C(=O)NCc1[nH]cnc1C C1(CNC(C(C)N(C(C2CC(=O)CCO2)=O)C2CC2)=O)C2CCCCCC12 CC(=O)C(C)CCOC(C12COCC(C1)C2)=O C1(C)(CNC(CC(C)n2cccc2)=O)CCN(C(c2nscc2Br)=O)C1 CCC(CC(C)C)C(=O)N1C(C)CN(C(C2(CSC)CC2)=O)CC1C N1(C(C2CC(SC)C2)=O)CCN(CC(=O)NC(C)CN2CCCC2=O)CC1 C(=O)(C1=CC2(CCOC2)C1)N1CCN(C(c2cc(C(C)C)c(F)cc2)=O)CC1C c1(C(N2CCCC3(CCCO3)C2)=O)ccc2[nH]nc(I)c2c1 C1CCCCC1.c1(C=O)snc(O)c1Cl.C12(C(=O)OC)CC(CC(=O)N)(C1)C2 c1(C(=O)NC2C(CNC(COCCOC)=O)CCC2)sc2sccc2c1Cl C=C(C)C(CC(=O)NC1(CC(=O)NC2CC3CC(OC)C3C2)CCC1)OCC Cc1cccc(C(=O)NC(CC(C)C)C(=O)NCC2CC2(Cl)Cl)c1N c1(OC)cc(NC(C23CCCCC2C3)=O)ncn1.C1CC12CC(NC=O)C2.O C(C(C(=O)N1CC(NC(=O)CCCc2nncn2C)C1)NCC(F)(F)F)N(C)C Cn1nc(Br)c2c(NCC(C3CCCC3)NC(=O)CCC3CCCO3)ncnc12 Cc1cnc(Cl)c(CN(c2ccc(C)c(Br)n2)C)c1.C12CCC(CC1)CC(=O)N2 c1(C(=O)NCC2N(C(c3c(CCC)[nH]cc3)=O)CC2)cc(Br)c(C)cc1F CC(C)CCCCC(=O)NCC1CCCN(C(=O)C(C)Sc2ccccn2)C1 C1(C(N2CC(c3ccc(OC)cc3)C2)=O)CC2CCC1N(C(c1cncs1)=O)C2 c1ccc(O)cc1.C1(CC)CCCC1C(=O)NC.C1(C=O)(C=O)CC1.N c1(CC)c(I)c(C(N2CC3(C2)CN(c2ncc(Br)c(C)n2)C3)=O)nn1C N1(C(CC(=O)NCC)=O)CC2(CCCC2NC(C2C3CCCCC23)=O)C1 C1CCC(C)(C)CN1C(=O)CC1CC1C(F)(F)F.CC(C)(C)C#CC(=O)N N1(C(Cc2cc(C)on2)=O)CC2CC1CN(C(c1cc3ccsc3s1)=O)C2 C1(C(N2CCCC(CC=C)C2)=O)CC2C=CC1N(C(=O)CC(COC)COC)C2 C1(C(=O)NCC2C3N(C(CSC(C)(C)C)=O)C(CC3)C2)CCc2nccn2C1 C1(C(N2CCC(NC(c3cc(C)on3)=O)C2(C)C)=O)CC2(CCCCC2)C1 c1(C(=O)NC2CCN(C(=O)CC3CC4(CC4)C3)C23CC3)onc2c1CCCC2 C1(CC(N2C(C)(CNC(=O)CC3CC34CC4)CCC2)=O)CCCCCCC1 N1(C(C(OC)OC)=O)CCC(C)(C)C1.c1(C=O)ccc(CS(N)(=O)=O)cc1.C CC(C)(C)C(C(=O)NCC1CC2CCC(C1)C2)NC(c1ncccc1O)=O C1(C(=O)NCCN(C(=O)CS)C)CC(c2ccccc2)=NO1.C1CCCO1.C c1(OC)cc(C(=O)NCC2(OC)CCN(C(=O)C(N)=O)CC2)cc(OC)n1 C1(NC(C)=O)CC(NC(=O)CCC2(C#N)CCC2)C12CCC2 C1(O)(C(=O)NC2C(C)CN(C(c3cnc(Cl)[nH]3)=O)C2)CCCC(C)(C)C1 c1(NCC(N2CC(c3ccccc3O)C2)=O)cccc(Cl)c1 N1(C(CC2N(C(C3=NNC(=O)C3)=O)C3C2CCC3)=O)CCc2ccncc2C1 N1(CC(=C)C)CCC2(CC1)COC(CNC(C1C3CC4CC(C3)CC1C4)=O)C2 c1(C(=O)NCCNC(C(CC#C)(C)CC)=O)cc(S(=O)(=O)NC)cn1C N1(C(C(C)OCC)=O)CCCCC1C1CCN(C(c2nc(C3CC3)cs2)=O)CC1 CCCC(CC)CC(=O)N1CC2(CC2)CC1CNC(c1ccnc(S)c1)=O C1(CNC(Cc2cn(CC)nc2)=O)(C)CCN(C(=O)C=CC2CC2)CC1 S(=O)(=O)(c1ccccc1)CCCNC(=O)C(N1CCC(C2CCCCO2)CC1)=O c1(N2C(C(NOCC3(C)CCC3)=O)CCC2)nccc(S(C)(=O)=O)n1 N1(C(c2c(C)n(CC3CC3)cc2)=O)CCN(C(c2cc(O)cc(O)c2)=O)C(C)C1 C1(NC(=O)CCc2ccco2)CN(C(=O)CC2CCC(F)(F)CO2)C2(CCC2)C1 C1(NC(C(CCOCC)NC(c2cc(=N)[nH][nH]2)=O)=O)CCCC(C2CC2)C1 C(=O)(C#CC1CCOC1)NCC1CCCN(C(Cc2c(C)cc(C)s2)=O)C1 N1(C(c2nc(C(=O)OC)sc2)=O)CCN(C(=O)Nc2cnccn2)C2CC12 C(C(C)(C)C(C)(C)C)NC(C(COCC)n1cc(CCN(C)C)nn1)=O Cc1coc(C(=O)NC2CCC(NC(=O)C(C)OCc3ccccc3)CC2)c1C N1(C(C(C)OC)=O)CC(C2CCN(c3nc(C)nc4n[nH]cc34)CC2)C1 CCCCCCCC(=O)N(C1CCC(NC(=O)C2=NOC(C)C2C)CC1)C c1(CCC(=O)NC2C(NC(C3CC(CCC)C3)=O)CCC2)nnc(C)n1C.C C=CC(O)C(=O)N(C1CCN(C(=O)Cn2cnc(-c3ccccc3)n2)C1)C1CC1 N1(C(c2cnc(COC)s2)=O)CC(CNC(C2CCC(=O)N2)=O)C(C)C1 Cc1nnc(N2CCCC(CO)(NC(=O)C(F)CC3CCCC3)C2)nc1C c1(C(N2C(CCNC(=O)C(C)(C)S)CC(OC)C2)=O)[nH]nc2c1COC2(C)C c1(CCNC(c2n(CC)nnn2)c2ccsc2)cn(C)nc1C c1(C(=O)NCC(c2c(CC)cccc2)NC(c2cnco2)=O)cccc(F)c1F c12ccc(S(=O)(=O)N3CCCCC3)cc1N2.c1(COCC)ccn2nccc2n1 Cc1c(F)ccc(F)c1CN1CC(NC(=O)C=Cc2cnc[nH]2)C(F)C1 C1(N(C(C2CC2(C)CO)=O)CC)CCN(C(=O)C(=Cc2cnc[nH]2)C)CC1 C1(CC)(CC)CC(C(=O)N)C1.C(C)CC=O.C1OCCC1C=O.C(C)C.C c1(C=O)ccc2c(c1)N(C)C(=O)CC2.C(=O)(C(F)(F)C(O)C1CC1)N.CCC Cc1ccc2cc(C(N3CCC4CN(C(=O)C5=CCN(C)C5)C4C3)=O)cn2c1 N1(Cc2n(C)nc(Cl)c2)CCC2C(O)C(C)(C)C12 C1(C(N2CC(NC(C3CC3C)=O)C2)=O)(CC)CCC1 Cc1cccc(C(CNC(N2CC(c3ccccc3)CC2C)=O)N(C)C)c1C Cc1ccc(C(=O)NCC(O)COc2cc(F)ccc2F)c2[nH]cc(C#N)c12 C1(C(=O)NC2CCC(C(F)(F)F)O2)CCN(C(=O)C2CC2)CC1 C1(C(N2C(COC)(C)CCC2)=O)CCOCC1(C)C.C(=O)C(C)c1ccsc1.N C1(C2CN(C(C=CC(C)(C)NC(C3CCC3(C)C)=O)=O)C2)CCCCO1 C1(C(N(C(C2CCCC2)C)C)=O)CC12CCN(C(=O)CCC(C)CN(C)C)C2 CC1CC(C)CN(C(=O)NC2CCCN(c3ccnc(N4CCCCC4)n3)C2)C1 c1(NC(C2N(C(c3cc(OCC)n[nH]3)=O)CCCC2)C)cc(O)nc(O)n1 N1(C(Cc2cnc(C)[nH]2)=O)CCC(NC(c2cncc(F)c2C)=O)CC1C n1(CC(=O)NCC2CCN(C(C3(C)CC=CCO3)=O)C2)ccc2ccc(Cl)cc12 CC1COCCCN1C(c1ncccc1Cl)C(=O)NC1CCCCC1 Cc1c(NC(=O)NC2CN(C(=O)C=Cc3ccco3)CC2C)cccc1F C1(C(N2C(C(C(=O)NC3C(C)(C)CC3)(C)C)CCC2)=O)CCS(=O)CC1 C1(C)CN(C(c2ccnc(N(C)C)c2)=O)C(C)(C)C1.C=C=C(C)CC(=O)NC c1(-n2c(C(c3c(C)nn(C)c3)NCC3CCC(=O)O3)nnn2)ccc(Cl)cc1F c1(C(N2CC(C)OCC2C)C(=O)NCC(=C)C)csc2ccc(C)cc12 C1(NC(=O)C(O)C2CC2)CCN(c2nnc(C3CC3)o2)CCC1CO C(c1ccccc1)=CC(N1C(C(=O)NCCc2cc(C)no2)C(C)C1)=O N1(C(CC2(CSC)CC2)=O)CCOC(Cn2cc(-c3sccc3C)nn2)C1 N1(C(C2(CCN(C)C)CCCC2)=O)CCC(O)(C)C1.c1(CC(=O)N)ccon1 Cc1cc(C(=O)NC2CCC23CCC3)cc(=O)n1C.C(C1CCCC1)=CC(=O)N c1(C(C2CCC2)NCC(N(C)C)C2CC2)ccc(F)cc1OC(F)F CC1CCC(CNC(=O)CCC2(NC(=O)Cc3ccoc3)CCC2)C1 Cc1nc(C(=O)NC(CC2CCCC2)C(=O)NCCc2cc[nH]n2)ccc1C#N C1(NC(C(C)S)=O)CCCCC12CN(C(c1n[nH]c3ccccc13)=O)CCO2 O=S(=O)(c1cccnc1N1CC2CCC(C1)O2)NCCN1CC=CCC1 N1(C(C)C)C(=O)CN(C(=O)CCc2cnccc2Sc2ccccc2)CC1(C)C c1(C(N2CCC(C)(CCNC(C=CC)=O)C2)=O)ccc(OC)nc1OC C(=O)(CC(O)C(C)C)NCCN(CCC)C(c1cc2sccc2[nH]1)=O c1(CC)nn(C)cc1C(=O)NCCCC1CCCCN1C(C1CNC(=O)C1)=O Cc1ccc(CC(=O)N(CCCN(C)C)CCNC(=O)CC(F)F)cc1C CCCCCC=CCC(=O)NCC#CCNCC1CC1CC(=O)NC C(=O)(CCC1CCc2ccccc21)NC1CC(NC(C(C)OCC(C)C)=O)C1 C1(CNC(COCCC(C)C)=O)CN(C(=O)CCC2CC2)C(C)(C)C1 CCCCCCC(=O)N1CCCC1C(C)NC(=O)Cc1csc(C2CC2)n1 C1(NC(C2C(CCC)CCC2)=O)CN(C(=O)CCC(F)(F)F)C2CCCC12 c1(C(=O)NCC2CC23CC3)cccc(Cc2ccccc2)n1 C(=O)(C(O)CCc1ccccc1)NC1C(CNC(c2cnc(OC)s2)=O)C1 C1(NC(CC(CCC)CC)=O)CC2CCC(C1C)N2C(C1CCC1(C)C)=O C1(NC(C(C)C2CCOC2)=O)C(C)CCN(C(=O)CC2CCCCCC2)C1C C(=O)(C(CCC(C)C)NC(C)=O)Nc1ccc(C(=O)OCC)cn1 c1(CN2C(C(N3CC(O)C3)=O)CC(O)CC2)ccc(Br)cc1[N+](=O)[O-] C1(CNC(c2nc(OC)nc(O)c2)=O)CC12CCN(C(c1nccn1C)=O)CC2 c1(C(=O)NC(CNC(c2cc(CCOC)on2)=O)CCOC)cnccc1.O C1(C(=O)NC)SC2C=CC1CC2.C1CCCCC1.C1(C=O)CC(O)(C(F)F)C1 c1(C(=O)NC(C)CNC(=O)C(C2CCCO2)C2CC2)csc(C2CC2)n1 CC(C)(O)C(=O)NC1CC(OCC(=O)NC2(CCCF)CC2)C1 c1(C(=O)NC(CNC(C(n2ncc(C)c2)C)=O)(C)CO)cnc(Br)c(N)n1 C1(N(C(=O)C(F)(F)c2ccccn2)C)CCS(=N)(=O)C1 C1(C(=O)NC23CC(NC(C(C)OC4CCOC4)=O)(C2)C3)CCCS1(=O)=O c1(C(N2CCC(CCC(=O)OCC)C2)C(=O)NCCCSC)ccc(Br)cc1F c1(OC(C)(C)C)ccc(F)c(CNS(=O)(=O)N2CCC2)c1 CC(CN=c1cccc(S(=O)(=O)NCCc2cncc(Br)c2)[nH]1)S(C)(=O)=O c1(C(N2C(C)CC(NC(c3cc(C#N)n(C)n3)=O)C2)=O)cncc([N+](=O)[O-])c1 C1(NC(CCSCCC)=O)CCCCC1NC(c1ccsc1NCC)=O c1(CNCC2(NC(c3ccon3)=O)COC2)c(Br)ccc(Cl)c1Cl C1(C(N(CC(CNC(CC=C=C)=O)(C)C)C)=O)CC2(CCOC2)C1 C(=O)(CCCC(C)CC)NC(C(=O)NCC1(OCC)CCC1)CC(F)F N1(CC)CC(C(=O)NC2CCC(NC(c3sc(=N)[nH]c3C)=O)C2)CC1=O Cc1cccc2[nH]cc(C(=O)NCC3CN(C(=O)CCc4ccoc4)C4CC34)c12 c1(C(=O)NC2CN(C(C(C)OCC3CCCO3)=O)C2)cc(CO)n(C)n1 c1(C(N2CCC(C)C2)C(=O)NC2CC(CNC3CC3)C2)ccccc1Br c1(NCCCCC(=O)NC)nccc(=NCCn2cc(Cl)cn2)[nH]1 S(=O)(=O)(c1c[nH]c(C(=O)NC(C)CC)c1)NC.C1(C=O)CCC2(CCC2)C1 C1(CCC(=O)NCc2cnco2)CCCCN1C(=O)COCCF N1(C(C(C2CCC2)OC)=O)CC(C)(C(=O)NC2CCC3(CC3)C2)CC1(C)C C1(CCNC(C(C)SCCCC)=O)COCCN1C(=O)C.c1(C=O)nccs1 c1(C(N2C(CNC(C3C(C)OCC3)=O)CCCC2)=O)ccc(C#CC2CC2)cc1 CC1CC(C)(C(=O)NCCC2CCN(C(c3cc(O)ncn3)=O)CC2)CCO1 c1(C2C(C(=O)N)C2)cc(Br)ccn1.C1(NC(C=CC=CC)=O)CCCC1 c1(C(N(CC(C)(C)C)C)=O)ccc(C)c(Cl)c1.N1(C(C)=O)CC2CC2(C=O)C1 c1(CNC(N2CCC(NC(CCC)=O)(CO)CC2)=O)ccc2c(c1)CCO2 c1(C(C(C)N(C(=O)C(C)(C)C)CC(F)(F)F)OC)ccc(Br)cc1 C1(C=O)CCC(C)(C)N(C(c2cc(C(N)=O)c[nH]2)=O)C1.C#CCCC(C)(C)C.N C1(OC)CN(C(=O)NC2(CO)CC(C)C2)CC1(C)C c1(C(N2CC(C(C)NC(C3CCCCO3)=O)C2)=O)ccc(C#N)c(F)c1 c1(C(N2CCCC(C(C)NC(CC(C(=O)OC)C)=O)C2)=O)cccn2nccc12 c1(C(=O)NC(C)CNC(c2cnn(C)n2)=O)ccc(OC)cc1.C1CCC1 C1(NC(C2N(CC(C)C)CCC2)=O)C2CC1CN(C(C1CC3CCC1O3)=O)C2 c1(C(N2CCC(CCNC(c3cocn3)=O)C2)=O)nnn2c1CCCC2 N1(C(CC2CC(SC)C2)=O)CC2CCCC2(NC(c2sccc2C)=O)C1 C12(C(=O)NC3C(C)CN(C(C4CC(=O)NC(C)C4)=O)CC3)CCC(C)(CC1)OC2 c1(C(=O)NCCC(C)NC(C2CC23CCCC3)=O)cc(F)cc2ccoc12 Cc1cc(C(=O)NOCC(=O)NCC(c2ccccn2)C)nnc1C CC1(C)C(CNC(=O)Cc2ccccc2F)CCN1c1ccnc(CO)n1 C1(N(C(C2C=CCC2)=O)CCO)CCN(C(C2(N3CCCC3)CC2)=O)C1 c1(OC)ccnc(C(N2CCC(NC(=O)C(c3ccccc3)C)C2C)=O)c1N C1(CCC(=O)N(CCC)CC)CCS1(=O)=O.c1(C2C(C=O)CC2)nncn1C c1(NCCC)ccc(S(=O)(=O)NCCN)cc1Cl.C(C)(C(C)C)SC N1(C(C2CC(C#C)(O)C2)=O)CCC2(CC1)CC(NC(=O)C(C1CCOCC1)F)C2 CC(C(=O)N1CCCC(CN(C(=O)C)CO)C1)S(C)(=O)=O.c1nncn1C.S C(C(C)N=c1[nH]c(N2CCC(C)C2)nc2c1SCC2)C1CC(C)C1 c1(C(=O)NC2CC(CCNC(C(C=CC)O)=O)C2)ccc(N)c(F)c1F C(=O)(CCC(=O)N(C)CCn1cc(-c2ccn(CC(F)(F)F)n2)nn1)NCC C=CCCCC(=O)NC(c1ccccc1)C(=O)NC(C)CC(N)=O N1(C(C=CCC)=O)CC(C)OC2(CCN(C(c3nccc(C)n3)=O)C2)C1 N1(C(CC)=O)CC(N(C)C(c2cc([N+](=O)[O-])c[nH]2)=O)C(C)(C)C1.C(C)(C)C.O c1(CC(=O)N)ccc2c(c1)CCCO2.CC(C(=O)N(CC)C1CC1)n1ccnc1 C1(CNC(COCC)=O)CCCN(c2nnc(C(c3ccccc3)C)o2)CC1 CC1(C)CC(C)(C(N2CC3C(CNC(=O)CCN4CCOCC4)C3C2)=O)C1 N1(C(CN(C)C(N)=O)=O)CCC(NC(c2cnc3ccsc3c2)=O)C12CCCC2 N1(C(C(C)C)=O)CC(NC(=O)C(C)Cc2ccnn2C)CC2(CCC2)C1 N1(C(C(C)C#N)=O)CC2(CCC2)CC1CNC(C1(CO)CC(F)(F)C1)=O c1(OC)cccc(C(N2CC3C(CN=[N+]=[N-])C3C2)C(=O)NC2CCOC2)c1C CC(F)(F)C(F)F.CC1(C)CC(CC(=O)Nc2ncoc2C)C1.C(=O)CC.N CC1CN(C)CC(C(=O)NCC2CC2C(=O)NCCCCCF)O1 c1ccc(CC#N)cc1.CC1CCC1C(=O)NCCNC(=O)C.C1CC1.O N1(C(C(CC)CC)=O)CC(NC(=O)C=Cc2nnn(C)n2)CC1(C)CC N1(C(CC2CCCC(NC(C(CC)COC)=O)C2)=O)CCC2(CCCO2)C1 n1(CC)cnc(C(N2CCCC2C(=O)NCC2(CO)CCCO2)=O)c1 C#CCCCC(=O)NCC(C(=O)NCC(O)C(C)CC)N(C)C CN1C2CCC1CN(C(C1CCN1Cc1cc(Cl)cc(Cl)c1)=O)C2 O=C(C(O)C1=CCCCC1)NC(C(=O)NCCc1ncccn1)C1CC1 Cc1ncccc1C=CC(=O)NCCCCC(C)NC(C1SCCCS1)=O c1(C(CCN(CCC(C)C)CC(=O)NC(=O)NCC(C)C)C)ccccc1 C(CCCCCNC(C1CC2CCC2C1)=O)N(C(=O)CCn1cncn1)C N1(C(C2CC(F)CN(S(=O)(=O)c3ccccn3)C2)=O)CCc2ccc(Br)cc2C1 Cc1cc(C(=O)N(C2CN(C(C3(O)CC(CF)C3)=O)CC23CC3)C)c(C)c(C)c1 C1(C(=O)NC2CCN(CC)C2)CC(NC(=O)CSC(F)(F)F)C12CCC2 Cc1nncc(C(=O)NC2CCN(C(=O)CN3C(=O)CNC3=O)CC2F)c1C Cc1ncn2ccc(C(N3CCCC(CNC(C4(N(C)C)CCC4)=O)C3)=O)cc12 c1(C(=O)NCC(CNC(C(COC)(C)O)=O)OC)ccc(OC)nc1C C1(C(=O)NCC2C(NC(CCn3cc(C)nc3)=O)COC2)CCCC12CCC2 c1(C(=O)NCC(CC=C)NC(=O)C(CO)N(C)C)cc(F)c(Br)cc1C n1(CC(=O)OC)c(C)cc(C=O)c1C.C(C)(C)CC.C1(C=O)C(C)C1C.N Cc1cc(CNC(C2CCCC(CF)C2)=O)oc1C(=O)N.C(C)C(O)C(F)F c1(C(N(C(C)CCNC(=O)Cc2cncn2C)C)=O)cccc(Cl)c1 n1(CC(=O)NCC2(C(C)C)CC2)cccn1.c1ccccc1.C(=O)(CC=C)N C1(NC(c2c(C)[nH]nc2Cl)=O)CCN(C(=O)CSc2ccncc2)CC1F C(=O)(CC(O)C(C)C)N1C2C(CNC(C3CC(SC)C3)=O)C(C2)C1 c1(CCC(N2CCC(OC(c3ncc(Cl)cc3C)=O)C2)C)ccc2c(c1)OCO2 c1(C=O)cccc(C=C(F)F)c1.O=C(COCC1CCC1)NCC=CC c1(CCO)ccc(C=O)cc1.C1(N(CCCN)CC(N)=O)CCOCC1 Cc1ccc(-n2ncc(C(=O)NCC3(F)CCC3)c2C)cc1.C1(C=O)CC1F.N C(=O)(C(CC)C(F)(F)F)NCCC1(NC(C(CCCC)C)=O)CC1 C1(N(C(=O)CC2CC3(CC3)C2)C)CCN(C(=O)C(C)(C)c2cncnc2)CC1 CC1OCCCC1C(=O)NCCN(C(=O)CP(C)(C)=O)CCCN(C)C C1COC(C(F)(F)F)CN1C(C1CCC2(CC1)CC2)=O.O=C(C#CC1CC1)NC C12(NC(CCC(=O)NC)=O)CCC(CN(C(c3ccc(C#N)[nH]3)=O)C1)C2 Cc1cc(N2CC(NC(c3cn(C)nn3)=O)CCC2C)nc(S(C)(=O)=O)n1 CCC(C(=O)NC12CCC(n3cc(COC4CCOCC4)nn3)(CC1)C2)C(C)O c1(C(=O)NCC2C(C)CN(C(=O)C=Cc3ccc(Cl)s3)C2)cc(F)cnc1Cl Cc1cnc2n1CCC(C(N1C3CCC1(CO)CC3)=O)C2 CCCC(C)CC(=O)N1CCCC1C(=O)NCCCc1ncccc1C C=CC1CCCN(C(=O)C=CCC2(NC(C3C=C(C)CS3)=O)CCC2)C1 N1(C(C2CCCC(C)C2)=O)CCC(C2(NC(c3c[nH]c4cccnc34)=O)CC2)C1 C(=O)(C1CCCc2nc[nH]c21)N1CCC(NC(c2nn(C)c(C(F)F)c2)=O)C1 c1(N2CCCC(c3nc(C)[nH]n3)C2)ncnc(NC2CCS(=O)C2)c1C c1(C(=O)NCCCNC(C(C)NC(COC)=O)=O)ccc2ncsc2c1 c1(CC)ncc(C(=O)N(C(C)CC(=O)NCCOC2CC2)C)cn1 c1(NC(CC(C)(C)CBr)c2nnnn2CCCC2CC2)ncc(Cl)c(I)c1F C1(COC)(NC(C2(c3ccccc3)CC2(Cl)Cl)=O)CN(C(=O)C(C)SC)C1 C1(NC(CC(COC)(C)C)=O)CN(C(C2CCC(C)(C)C2)=O)C2(CCC2)C1 N1(C(CC2N(CC)CCC2)=O)CC2C(N(C)C(C3C4CC5C(C4)C35)=O)C2C1 N1(C(C(OC)OC)=O)CC(C)(C)CC1CNC(=O)CCCC(F)F c1(C(=O)NCC2CC(C)(C)N(C(c3occc3Cl)=O)C2)c(F)ccc2nc[nH]c12 C1C(C2CC2)CCN1C(=O)C=Cc1cncc(O)c1.CC(C)(C)C=CC=O.N c1(OCCC(=O)NC(CC(C)NC(=O)CCCC#N)C)ccc(Cl)c(Cl)c1 C1(CC(N2CCc3sccc3C2C)C(=O)NCC)CC(C)(C)OC(C)(C)C1 c1(C=O)cccc2nccn12.C1(CCNC(C2C(C)(CC)C2)=O)CCOCC1.N CC(O)(CC(=O)NC(C1CCCC1)C)C(F)(F)F.C1(C=O)CCCCS1(=O)=O.N C(=O)(C1=C(C)CCC1)N(C1CC(C(N(CC#C)C)=O)C1)C C1(CC(=O)NCC2N(C(C3N(C)CCCC3)=O)CCOC2)CCC2(CCC2)CO1 Cc1oc(Br)cc1C(=O)NC1CN(C(=O)COc2cnn(C)c2)CC1O CC1C(NC(C2(CO)CC2)=O)CC2CCC1N2C(=O)C(F)(F)C12CC(C1)C2 c1(-c2cn(C3CN(C(CC(C)C)=O)CC3C)nn2)ccc(C#N)c(F)c1.CC(=O)N S(=O)(=O)(c1cnc(NCc2ccc(C)o2)c(Cl)c1)NC(c1ccccc1F)CC C1(CC(=O)NCC2CN(C(c3cnc(CC)[nH]3)=O)C2)CCC(C#N)C1 CC(CS(C)(=O)=O)C(=O)NC1CCCN(C(=O)COc2ccccc2O)C1 c1(N2CCCC(c3cc(C)[nH]n3)C2)nccc(=NCCCCC(F)(F)F)[nH]1 N1(C(C2C(C)C2)=O)CC2CCC1CN2C(c1cc(F)ccc1I)=O CCCC(C(=O)NC)NC(C1CC12CC(NC(C1(C)CCCN1C)=O)C2)=O c1(C(C)C(=O)NC2CCC2NC(c2cn(C)cn2)=O)cccc(Br)c1F C1(NC(=O)CC2C=CCC2)CC2CCC1N2C(=O)C=Cc1ccncc1 C(C(O)C(=O)NC1CC(O)(CNC(=O)CC=O)C1)=CC.CC(F)(F)F c1(CN)cccc(S(=O)(=O)NC(C23CCC(C(N)=O)(CC2)C3)=O)c1 C=CCCC(C(=O)NC(C)C(C)SC)NC(=O)Cn1c(C)ccc1C N1(C(C2CCN(C(CCCSC)=O)CC2C)=O)CCOCC(C)(O)C1 c1(C(=O)N)cnc2n(c1=O)CCS2.CC(CNC(C1(C(N)=O)CC1)=O)CO CCCC(C(=O)N1CC2CC1(c1cn(C)nn1)C2)S(N)(=O)=O.[nH]1nc(C)n(C)c1=O C(C(C)(C)C(=O)NCC1CCCCC1NC(c1cc(C)ncn1)=O)OCC CN1CC(C(=O)NC2(C)CCN(C(C3CCN3Cc3ccccc3)=O)C2)CC1=O Cc1ccc(CNC(=O)NCc2ccc(Cl)c(Cl)c2)nc1F N1(C(c2c(C)nccc2Cl)=O)CCC2(CCN(C(=O)C3=COCCO3)C2)C1 O=C(N=c1nc[nH]n2cc(Br)cc12)C1CC(NCc2cccc3[nH]ncc23)C1 CCCC(O)C(CO)NC(=O)CCC(C)NC(C1CC(=O)NC(=O)N1)=O Cc1cc(C(=O)N(CCCCN(C(=O)COCC2CCCO2)C)C)cc(O)n1 C1(C)(CCC(=O)N(C(C2(C)CC2)C)C)CN(C(=O)CCc2cncnc2)C1 c1(C=O)c(C)nn(C)c1C.C(=O)(CCC(=O)N1CC(C)C1)Nc1nnc(C)s1.N C1(C(=O)Nc2ccns2)CC2CC2N1c1nccc(-c2cccnc2)n1 C1(C(N2CC3(CC(F)C3)C2)=O)CCN(C(=O)C(O)C2CCC2)CCO1 c1(C(N2C(C)C(NC(C3CCCC(C)(C)C3)=O)CC2)=O)cc(F)c(F)c(C#N)c1 c1(OC)cc(F)c(C=O)cc1N.C1CCN(C(=O)C=CCN(C)C)C(C)C1.N N1(C(C(CC=C)CC)=O)C2CCC(C(N3CC(C)=C(C)C3)=O)C1CC2 N1(C(c2c(C)nsc2)=O)CCC2(CCC(C(=O)NC(C3CCOCC3)C)C2)CC1 C(=O)(CC(C)C(C)(C)C)NCC(C)N(C(c1c(CC)nc(=N)[nH]c1)=O)C C1(CNC(c2n(C)c(O)nc2)=O)CN(C(c2ccsc2)=O)CC12CC2 C1(O)(CNC(CCCC(N)=O)=O)CCCN(C(c2cc(O)ccc2F)=O)CC1 N1(C(c2c(Cl)cc(C)s2)=O)CCN(C(=O)CCCCCN(C)C)C2(CCC2)C1 C1(NC(C(CC#C)C2CC2)=O)(COC)CCCN(C(c2ccc(F)cc2)=O)C1.C c1(C(C=O)(C)O)ccc(F)cc1.CC(C)(C)CC1CN(C(=O)C=O)C1.CCC C(=O)(C1=CC2CCCCCC12)N1CCC(CNC(CCCCC(=O)OC)=O)CC1 CCC(C)C(O)C(C)C(=O)NCc1cccc(CNC(=O)C(C(C)C)OC)c1 Cc1c(C(N2CCCC(NC(C3(C)COCCO3)=O)C2)=O)cncc1F Cc1nn(C)cc1CCC(=O)NC1CC(NC(C2CCN(C)C2C)=O)C1 Cc1nsc2cc(C(=O)NCC3CN(C(=O)C(=O)N(C)C)CCC3C)cnc12 C(=O)(C1=CCOCC1)N1CCC(C)(C(=O)NCC2CC2Cl)C1 c1(C(CC(C)C)OC)nc(SC(C)C)n(-c2ccn(CCOC)n2)n1 C1(O)(CC(=O)N(CC(C)N(C(CNc2ccccc2)=O)C)C)CCOCC1.C c1(NCc2c(OC)cc(OC(F)(F)F)cc2)ncc(C2=COCC2)s1 Cn1cc(C(=O)NC(c2ncoc2C(F)(F)F)c2ccccc2)cn1 N1(C(c2ccnc(Cl)c2Br)C(=O)NC(C)(C)C)CC2CCCC2(CO)C1 N1(C(CC2(C(=O)OC)CCC2)=O)CCCC(C)C1.C(c1csc(C)n1)=CC=O c1(C(=O)NC(CCNC(Cc2c(C)ccc(Cl)c2)=O)C)cc(C)c2[nH]nnc2c1 c1(C(=O)OC)cc(Br)cc(S(=O)(=O)NC(=O)C(C)(F)C2CCCCC2)c1 c1(C(=O)NCC(C)(O)CNC(=O)CC=C(Cl)Cl)ccc(CO)c(Cl)c1 N#CC1(F)CCN(C(=O)C(CCF)NC(=O)CC2CCOC2)C1 C1(C(=O)NC2CCCC23CC3)(CC)CCCN(C(c2ccc(C)nc2O)=O)C1 c1(OCCCC(=O)NC(C(C)NC(CN(C(C)C)C)=O)(C)C)ccccc1F c1(C(=O)NC(CCOC)C(=O)NC2CCCCNC2=O)cc([N+](=O)[O-])n[nH]1 Cc1cc(C)c(C(=O)NCC(C)NC(=O)C(C)(C)C2CCOC2)c(C)c1Br C1(C(N(CC(CC)NC(=O)Cn2cnnc2)C)=O)(CC)CCOCC1 c12nc(c3c(n1)CCC3)N(C)CCCN2C.c1(C(C(C)OC)C)ccc(Cl)cc1 N1(c2n(CC)c(Cc3ncccc3C)nn2)CCOC(C)(CC)C1 c1(C(N(C(C)C)CCN(C)C(C2(C)CCCO2)=O)=O)c(C(F)F)cnn1C CCCCCCC(F)C(=O)NCC1(O)CCCN(C(=O)C(C)(C)CCC)C1 Fc1cc(-n2nc(CCCCN(C)C)nc2-c2c(F)ccnc2F)ccc1Cl c1(C(NC)=O)ccc2cn(C)nc2c1.C(=O)(C(C)C(=O)NCC1CC1)OC N1(C(C(CC#C)C2CC2)=O)CC(F)(F)CC1CCNC(=O)C(=O)N.C(C)C C(=O)(CC(C)(C)C(F)F)NC1(C(=O)NC2C(C)C2)CCCC1.N1CCCC1=O c1(OC)cc(OC)c(CN2CC3CC2CN3C(c2cccc(Cl)c2O)=O)c(O)c1 CC1(CNC(=O)CCn2ccnn2)CC(F)(F)CN1c1cncc(C#N)n1 c1(NCC(c2ccc(C)cn2)(C)C)ccc([SH](=O)=O)cn1.C1(C2CC2)CCCC1.N Cc1ccc(CNC(C2CC(O)CCN2C(=O)CC2CC3CC3C2)=O)cc1C c1(C(=O)OC)cccc2c1CCOC2C(=O)NC1CCC(C(C)O)CC1 c1(N2CCC(Cc3cc(OC)n(C)n3)CC2)ncc2ccc(Br)cc2n1 N1(C(c2c(C)nn[nH]2)=O)CCC2(CC1)OCCCC2NC(=O)CC1CCN(C)C1 O=C(CC(F)(F)F)NC(Cn1cccn1)C(=O)NC1(CCF)CCC1 n1(C(C)C)cc2c(n1)CC(NC(=O)NCC1CC(=O)NC(=O)C1)CC2 c1(C(N(C2CCN(C(=O)C(c3cncnc3)C)C2)CCC)=O)ncn2c1CCC2 C1(COC)(C)CCN(C(C2CCC3CCC23)=O)CC1.c1(C=O)ccc(O)nn1.N C1(CC)CCC(C(N2CCN(CC(C)NC(=O)Cn3ccc(=N)[nH]3)CC2)=O)CC1 Cc1sccc1C(=O)NCc1ccsc1C(=O)NC.n1(C2CC2)nccn1 CCCC(C)(O)C(=O)NCCSCC(=O)NCc1ccoc1 C(CN(CC(C)C)N1CCC(=O)N2CCCC12)c1cccc(C)c1 C(=O)(CCCCCC(C)O)NC1C2C(C)N(C(C=Cc3cncc(C)c3)=O)C1C2 c1(C(C)C)c(NC(N2CCN(C3CN(C=O)C3)CC2)=O)cnn1C.C(C)(C)C.O Cc1c(C(=O)NC(C)C=CC(N2CCC2C(N)=O)=O)ccn1C N1(C(c2cncc(SC)c2)=O)CCCC(C)C1CNC(=O)Cn1ccnn1 Cc1nc[nH]c1C(=O)NCC=CC.c1(CC(=O)N)c[nH]nc1C(F)(F)F C1(C(=O)NCC2N(C(C3N=C(C)SC3)=O)CCCC2C)CC(C)CC(C)(C)C1 C1(C(=O)NC2CCCN(C(C3(O)CC(F)(F)C3)=O)CC2)CCc2ccccc2O1 C#Cc1ccc(C(=O)NC2(CNC(C3C4CC(F)(F)CC34)=O)CCC2)cc1 c1(OC)c(Cl)ccc(C(=O)N(C)CC2CCN(C(=O)CCc3ccoc3)C2)c1F CCS(=O)(=O)c1ccccc1C(N1CCC(NC(=O)C=C2CC2)C(F)C1)=O N(C(=NCC1CCCOC1)NCC(C1(OC)CCOCC1)(F)F)CCSCC=C Cc1nsc(C(=O)NC(C)(C)CC)c1N.c1(C(=O)N)cccc(C2CC2(F)F)c1 C1(CC(N)=O)(NC(c2c(Cl)cn(C)n2)=O)CCN(C(=O)C2=NNC(=O)C2)CC1 c1(C(=O)NCCCN(C(=O)C=CSC)CC)ccc(N)cc1OC N1(C(CC2CCN(C)CC2)=O)CCC2CN(C(c3c(F)cc(Cl)cc3Br)=O)CC12 C1(CNC(c2cnn(CCC)c2C2CC2)=O)CCN(C(=O)COC)CC1C CC1(C(=O)NCCNC(=O)CCC2CC2)CC2CC2C1 CCC(C)CCCCC(=O)N1CCC(NC(c2cn(C)nc2C)=O)CC(C)(C)C1 C(CN=c1[nH]nc(C(C)(C)C)s1)C1C(C)CCCN1C(=O)CC1CC(C)(C)CO1 C(=O)(C=CS(C)=O)N(C)CCN(C1CCCCCC1)C(=O)Cc1cnoc1 N1(C(C(C)CO)=O)CCN(C(c2cc(-c3ccc(C(F)(F)F)cc3)[nH]n2)=O)CC1 N1(C(CCC)=O)CCCC(C(N2CCC(NC(C3(C)CC3)=O)C2C(C)C)=O)C1 N1(C(C(=C(C)C2CC2)F)=O)CCOCC(NC(=O)CC2COCCO2)C1 C1(C)(CNC(C2(COC)CC2)=O)CCCN1C(C1CCCCC1C)=O c1(C(C)=O)ccc(C(=O)NCC2(O)CCN(C(c3cncnc3)=O)C2)nn1 N1(C(c2cnc(C)nc2C)=O)CCC2(CC1)CC2NC(c1cn(C2CC2)nn1)=O c1(C(=O)NC2(n3cc(CCS(C)(=O)=O)nn3)CC2)ccccn1.C1CCCC1.N C1(CNC(COC)=O)CN(C(c2cc(Cl)ncc2OC)=O)CCN1C N1(C(C(CC2CCOCC2)NC(CCC2(C)CC2)=O)=O)CCOC2C(O)CC12 C1(NC(Cc2scc(C)n2)=O)CC1C1CCCN(C(c2ccccc2O)=O)C1 c1(C(=O)NCC2CCN(C(CC(C)(F)F)=O)C2(C)C)cccc2sncc12 C=C1CCN(C(C2CCN(C(C3CCC(C)O3)=O)C2CC)=O)CC1 C(=O)(C#CC1CCCO1)N(CCCCNC(C(C)Cc1cnc[nH]1)=O)C c1(CC(N2CC(C3(NC(C(C(C)(C)O)F)=O)CC3)C2)=O)coc2cc(F)ccc12 c1(CC)cccc(C(=O)NC2(CO)CCN(C(c3n[nH]c(C)c3Br)=O)C2)n1 C1(Cn2cc(C(C)(C)C)nn2)COCCN1C(c1cc(Cl)ccn1)=O N1(C(CN(C(C(CC#C)O)=O)C2CCC2)=O)CCc2nn[nH]c2C1 CCCS(=O)(=O)CC(=O)NC1CC(CNC(c2cnoc2C)=O)C12CCC2 C1(NC(C2C(CNC(C(=O)N(C)C)=O)C2)=O)CCCC1C1CC1 S(=O)(=O)(c1n[nH]c(=NC(=O)OC(C)(C)C)s1)Nc1nn(C)c2c1CCNC2 N1(C(c2nc(CC)sc2)=O)CC(CC(N2CC3CC(C)C3C2)=O)CC1(C)C Cc1ncc2c(n1)CCC(C(=O)NCC(C)CN(C)C(c1cncnc1)=O)C2 CC(C)(CCCO)C(=O)N1CCC(C(C)(C)CNC(c2cnc[nH]2)=O)CC1 c1(C(=O)NCC(C)CNC(C2(c3cccs3)CC2)=O)nn(C)cc1Cl C12(C(N3CCC(C)(CC)C3)=O)CCC(CN(C(C3CC(SC)C3)=O)C1)C2 O=C(CCCCCCc1ccccc1)NCC1CCCN1C(=O)CSC(F)(F)F N1(C(c2ccc(OC)s2)=O)CC2(C=C(C(=O)N3CCC(C)C3)CO2)C1 CC1C(NC(=O)CC2CCOCC2)CCCN1C(c1ccn(C)n1)=O C1(C(=O)OCC)CCC(NC(=O)NCC(C2CCCN(C=O)C2)O)CC1.O C(=O)(C(CNC(=O)CCCF)CC1CC1)NCC1N(CC)CCC1 Cc1c(C(=O)NCC2CCCN(C(=O)C(O)C3CCC3)C2)sc2cccc(F)c12 Cc1ccc(CNC(c2cc(-c3cnn(CCF)c3)cnc2N(C)C)=O)c(O)n1 C(=O)(CCCCCC#N)NCCCOCCCNC(c1ccc(NC)cc1F)=O CC(C)S(=O)(=O)CC(=O)NC(C)(CNC(=O)OC(C)(C)C)C(C)C n1(CC(C)NC(=O)C(C)C2CCOC2)cc(-c2cnccn2)nn1 N1(C(C2C(C)(C)NC(=O)C2)=O)CCC(NC(c2cnc(F)c(Cl)c2)=O)C12CCC2 N1(C(C(C)NC(CC)=O)=O)CCC(CNC(=O)COc2ccccc2)CC1 N1(C(c2n(C(C)C)ncc2)=O)CC(C2CN(C(C3CCn4cnnc4C3)=O)C2)C1 N1(C(C(C)NC(=O)NC)=O)CC(O)(CNC(=O)CC2CSCCS2)C1 Cc1ncc(Br)cc1C(=O)NCC1(NC(c2ccncn2)=O)CCOC1 C=CC(C)CC(=O)NCC1CCN(C(c2cccc(-c3csc(C)n3)c2)=O)C1 c1(C(C)N(C(CC2(C#N)CCC2)C(=O)NC2CC2)C)ccccc1F c1(C(C(=O)NCC(CC)(C)NC(=O)Cc2cncn2C)O)ccccc1Br C(CC(=O)NC=O)(C(F)(F)F)NC(C)(C(F)(F)F)C1CC1.c1ccccc1.N C1(NC(CC2(OCC)CC2)=O)COC2CCOC12.C1(C=O)CCC(F)(F)C1O N1(C(C(CN(CC)CC)F)=O)CCC2(CCC2)C1.c1(C2CC2)ccc(F)cc1.N CC1CCC(NC(c2cnsn2)=O)CN1C(c1ccc(OCC(F)(F)F)nn1)=O c1(CCC)occc1C(=O)NC(C1CC(NC(=O)CSCC(C)C)C1)C C1(CNC(c2ncn(C(C)C)n2)=O)CN(C(c2ncc(Br)cn2)=O)C2CC12 c1(C(=O)NC(CNC(CC2C(C)C2)=O)(C)C)cc(Cl)ccn1 Cc1nn(C(C)(C)C)c(C(N2CCCC(OCc3ccccc3)C2)=O)c1Br CC1CCN(C(=O)CCCc2cnn[nH]2)C1C(N1CCNC(=O)C1)=O c1(-n2cc(CN(C(=O)CCC(=O)C3CCCC3)C)nn2)ccc(Cl)cc1C(=O)O C=CC1(C(N2C3CCC2C(NC(=O)C(C)(C)OCCCC)C3)=O)CCCCC1 C1(C(=O)NCC2=CCCC2)C(C2CC2)CCN1C(=O)C(O)C1CCC1 N1(C(C2C(OC(C)(C)C)C2)=O)CCCC1(C)CNC(c1cc(C)[nH]n1)=O c1(CCC(N2CC(N(C(=O)C(c3ccc(Cl)cc3)CO)C)C2)=O)cccc(Cl)c1 c1(C(=O)NCCN(C(C(C(C)C)c2ccccc2)=O)C)cccc(F)c1Cl N1(C(Cn2ncc(C)c2)=O)CC(NC(c2csc(C(C)C)n2)=O)CC(C)C1 CC(N=c1ccnc(N2CCC3(CCC3)C2)[nH]1)c1ccoc1 C1(CNC(c2c(C)c[nH]n2)=O)CN(C(=O)CCNC(=O)C=CCl)CC12CCC2 CC1=CCC(C(=O)N(C)CC=CC(N2CCC(CO)C2C)=O)CC1 c1(C(=O)NC23CC(NC(CC(C)N(C)C)=O)(C2)C3)cn2cc(Cl)cnc2n1 C1(CC(=O)NC(CNC(C(C)OCC)=O)(C)C2CCC2)CCC=CCC1 C#CCC(C(=O)N1CC=CC(NC(=O)C(C)C(C)C)C1)C1CC1 N1(C(C(CC)C(C)O)=O)CCCC(C2CCCN(C(C3CC(=O)N(C)C3)=O)C2)C1 C1(OC)CC(NC(=O)Cc2c[nH]nc2C)CN(C(C2COC2)=O)C1 c1(C(=O)NC2CN(C(c3n(CC)cnn3)=O)C(C)(C)C2)cc2c([nH]1)CCCC2 Cn1cc(Br)c(C(=O)NC2CCN(C(c3ccc(C#N)[nH]3)=O)CC2)n1 c1(NC(C(C)OCC)=O)ccncc1-c1ccccc1 Cc1cncc(C=CC(=O)NCC(c2ccccc2F)O)c1 c1(C(N(C)CC2CCCN(C(C(CC)C)=O)C2)=O)cccc2ccoc12 C1(C)(NC(C(=Cc2cn[nH]c2)C)=O)CCCN(C(c2ccc(O)cc2Cl)=O)C1 C(=O)(C1=CC2CCCCCC12)N(C1CCCCC1)C.C(=O)(COCC(=O)N)OC C(=O)(C1=CC2(CN(C(C3CC4(CC4)CO3)=O)C2)OC1)N(C(C(C)C)C)CCC N1(CCCC)C(=S)NC(c2[nH]cc(C(=O)O)c2C2CC2)C(C(=O)OC)=C1CC c1(N2CCN(C(CCCC(=O)NC)=O)CC(O)C2)c(F)cccc1[N+](=O)[O-] C(C(O)(CNC(C1CCCCO1)=O)CO)OC.n1(C2(CC=O)CC2)cccn1 N1(C(Cc2c(C)non2)=O)CCN(C(=O)CNC(C2CCCCC2)=O)C(C)C1C N1(C(c2c(C)ocn2)=O)CCC(C)(C)C(CNC(=O)C(C)(F)C(F)(F)F)C1 C1(CNC(=O)COc2ccccc2F)CC2CCCC2N1C(=O)C=CBr C1(C(N(C(C)CCO)C)=O)CCC(C)(C)N(C(c2ccc(Cl)s2)=O)C1 C1(CCC(=O)OC)CN(CCNCc2nn[nH]c2CO)CC2(CCOCC2)O1 C1(C(N2CC(N(C(C(C)=C(CC)C)=O)C)C3(C2)CC3)=O)Cc2ccccc2O1 c1(C(N2CC(CC)N(C)CC2)C(=O)NCCOC)cncc2ccccc12 CC1CN(C(c2ncccc2Cl)=O)CCN1C(c1cc(O)ccc1F)=O C1(C)(C(=O)N)COc2ccccc2O1.C(C(O)C(=O)NCC1(CC)CC1)OC CC(C)(C)C(CNC(c1cncc(Cl)c1)=O)NC(=O)CCC(F)F c1(C(C(F)(F)F)NC(C2CC(CCN)C2)=O)c(F)cccc1F C1(C(C)(C)NC(C(CC)C)=O)CCN(C(=O)C(CCSC)NC(N)=O)CC1 Cc1cc(C(=O)NC23CC(Nc4ccncn4)(C2)C3)sc1Br N1(C(c2c(CC)n(C)nc2)=O)CC(NC(=O)CC2(O)CCCCCC2)C(C)(C)C1 N1(C(C(CCC)(C)O)=O)CCC(NC(C2(c3cccs3)CC2)=O)C(CO)CC1 CC(C)S(=O)(=O)c1ccccc1C(=O)Nc1nccc2c1OCO2 N1(C(C=C(CC)C)=O)CCC2CC2(NC(c2ccc(O)cc2)=O)CC1.C1CC1.C CC1CCC(NC(C2CCCC2C)=O)CN1C(=O)CSc1ccccc1 O=S(=O)(c1ccc2c(c1)CCCO2)NC1(Cc2cccc(Br)c2)CCOC1 CC1CC2(CO1)CN(C(C1CCCN(C(=O)CCC3CC3)C1)=O)C2 c1(C=O)cccnc1S.C1(COC)(C)CN(C(=O)CC2CC(C)(C)C2)C1.N C=CC(C)(C)CC(=O)NC1CCOC(CNC(=O)C)C1.c1cc(F)cc(Cl)c1 C1(C(N2CCC(SC)C2)=O)CN(C(=O)COC2CCC2)CC12CCC2 c1(NC(=O)NCC(CC2CCOCC2)OC)ccn(C2CC2)c1C CC(C)C(C(=O)NCC1(C(=O)N(C2CC2(C)C)C)CC=CC1)C1CCC1 c1(-c2cc(C(N(CCCNC(C(C(C)C)F)=O)C)=O)no2)c(F)cccc1F c1(C(N(C(CCNC(CSCCCC)=O)C)CC)=O)cncc(OC)c1 Cc1cc(C(N)=O)cc(C(=O)NCC)c1.C1CCN(C(C2CNC(=O)C2)=O)C1 C1CCN(C(C2CC23CC(O)C3)=O)C12CC2.N1(C(C)=O)CCCC1(C)C(=O)N.C C1(NC(c2n(CC)ncc2Cl)=O)CN(C(C2(CC(C)C)COC2)=O)CCC1C C1(N(C)C(C2CCS2(=O)=O)=O)CCCC2CN(C(=O)CC3CC=CCC3)CC12 c1(NCC)ccc(Cl)cc1C(=O)NC1CCC1.c1(C=O)cncc(O)c1Cl.C c1(C(=O)NCC(CC)NC(c2nc3cnccc3s2)=O)cc(C)c(F)c(C)c1 Cc1ccc(C)c(C2CCCN2C(=O)Cc2nncn2C(C)C)c1 c1(CNC(=O)CC2C=CCC2)cc(C(=O)O)ccc1F Cc1ccc(OCC(=O)NCC2C=CCN2C(=O)CC2CCOCC2)c(Br)c1 Cc1[nH]nc2cc(C(=O)N(CCCCC)CCO)ccc12.N(S(N)(=O)=O)CC=O.N C1(CNC(c2c(CCC)n(C)nc2)=O)C(C2CC2)CCN1C(=O)C(C)O Cc1nc(N2CC(NC(c3cnn(CCN(C)C)c3C)=O)CC2C)[nH]c(=N)n1 N1(C(c2cnc(C)[nH]2)=O)CC(NC(c2ccnnc2)=O)C(F)C1 C=C1CCN(C(=O)Cc2cnn(CC)c2)C(C(=O)NC(c2nnc(C)o2)C)C1 C12CN(CC1(F)F)C2=O.C(=O)(CNC)N(CCOCCO)CC.C1CC1 C12(CNC(C(c3c(C)cccc3)C)=O)CCC(C1)N(C(c1ncncc1Cl)=O)C2 CN1CCCN(C(=O)CC(C)(C)CNC(=O)CCc2cn[nH]c2)CCC1 c1(C(=O)OCCC2(CC)OCCO2)cnc2c(c1)N(C)CCO2 C1CC(C)(C)CCO1.C(C(COC)C(=O)NC(CN(C)C)C(=O)N)OC.C c1(C(c2nnnn2CCCSC)NCC(CC)(F)F)nn(C)nc1Br.C1CC1 N1(C(c2c(C)cc(O)nn2)=O)CCC(C2(O)CC(N)C2)CC1 c1(C(N(CC(C)C)C)=O)cccc2nn(C)nc12.c1(CC)[nH]c(=N)sc1C=O C1(CNC(C(C)Oc2ccc(Cl)cc2)=O)CC2CCCC2N1C(=O)C1=CCC1 N(C(=NCCN(CC(F)F)C)NC1CC1)C(C)C1CC1.c1(CO)c(C)noc1C CC1CN(C(C2CCCN(C)C2)=O)CC1(C)C(=O)NCC1C(C)C1C C(=O)(C(C)CC(=O)NC1CC(CNC(C2(OC)CC2)=O)C(O)C1)OC N(C1CCCc2cccnc21)(CC(C)C)C(=O)NC1CC2C=CC1O2 C(C1=CCN(C)CC1)NC(C(C)N(C(c1c(CC)nn(C)c1)=O)C)=O c1(OCC=C)ccc(C(=O)NC2CCC2NC(C2CCCC2)=O)cc1OC C(=O)(CCCCCNC(=O)C(C#N)C(C)C)NCCC(C(C)C)O C(C#Cc1cccnc1)NC(C1(CNC(CC(C)OC)=O)CC12CCC2)=O CN1CC2CC1CN(C(=O)C(CCC1CCC1)NC(=O)CC1CCCCO1)C2 CCC(CC(=O)NCC(C(=O)NC(C)(CO)C(C)C)C(C)(C)C)CC(C)C c1(C(=O)OC)ccc2c(c1)CC(NC(=O)C(F)Oc1ccc(Cl)c(F)c1)C2 Cc1ocnc1C(=O)N(CC(C)N(C(=O)Cn1nnc(=O)[nH]1)C)C CCC(CC)C(C1CC1)NC(Cc1ccccc1)C(=O)NCCc1ccccc1 C(=O)(C(F)(F)C(O)CCCCCCC)NCc1cn(CC=C)nn1.C1(CO)CC1 C1(CNC(C2C(=C)CC2)=O)CC2(CO1)CN(C(c1ccc(C3CC3)o1)=O)C2 c1(C(=O)NC(C)CNC(=O)C=CC2CCC2)cccn1Cc1ccncc1 n1(CC)ccnc1C(C)NC(=O)CONC(C1CNC(=O)O1)=O N1(CC(=O)NC2CCCN(Cc3nc(C)sc3)C2)C(=O)NC(C)(C)C1=O N1(C(C2C(CCOC)C2)=O)CC(O)CC1.C(CCC=C(C)C)=CC=O C1(NC(C=CCOC)=O)CCCCN(C(=O)Cc2ccn3cncc3c2)CC1 Cc1cc(Cl)c(C(N2CCOC(CN(C)C(c3cc(CO)on3)=O)C2)=O)s1 c1(C=O)ccc(C(F)C(F)(F)F)cc1.C(=O)(C(C)(C)NC(=O)CC)OC.N C1(CCC)CN(C(c2ccnn2C2CCOCC2)=O)CCN1C(=O)C(O)C1CC1 N1(C(c2cc(OC)c(Cl)s2)=O)CCC(C2CC2)(CNC(C2(O)CCC2)=O)C1 Cc1ncoc1C(=O)NCC1CCN(C(=O)C(c2ccccc2)n2cccc2)C1 CCCC(C(=O)N(C1CCN(C(=O)C(C)C2CCC2)CC1)C)OCC CCC(CO)C(=O)N1CCC(C(C)NC(=O)CC#N)C1 C1(OC)(CNC(=O)CCCc2ncc(C)o2)CN(C(=O)C(C)N2CCC2)C1 C(C)(c1ccc(F)cc1F)=CC(=O)N.c1(C(N(CCC)CC)=O)ccnnc1O C(=O)(CS(=O)(=O)CCC(F)(F)F)N1CCOCC1.C1(C)(C(N(C)C)=O)CCOC1 c1(C(=O)NCCCC)cnc(C2CC2)nc1O.C1(F)(C=O)C(C)(C)C1(C)C.N O=C1CN(C(C2CN(c3cc(CO)ccn3)C2)=O)CCO1.C12CCCCN1C2=O C12(NC(C(CC)=CC)=O)CCCCCC1N(C(=O)Cc1ccccc1OC)CC2 N1(C(C2CCC(CC)O2)=O)CC(N=c2cc(COC)nc(C(C)(C)C)[nH]2)CC1C N1(C(CCc2c(C)nn(C)c2)=O)CCC(CNC(c2cccc(Cl)c2)=O)CC1C CCCC(C(=O)N1CCCC(NCC(=O)N(CC(F)(F)F)C)C1)S(N)(=O)=O C1(CNC(CSCC(=O)OC)=O)CCCCC1.c1(CC=O)cc[nH]c1.C c1(OC)nccc(Br)c1C(=O)NCCN(C(=O)CN1CCOCC1)C c1(NC)ccccc1NC(c1ccc(CN(C)Cc2ccno2)nc1)=O N1(C(c2ccc(CC)o2)C(=O)NCC2CCOCC2)CC(=O)NCC12CC2 CCCC(C)(CC)C(=O)N1CCN(CCNC(C2CC3CC3C2)=O)CC1 n1(CCOCC)nnnc1C(CCC=C(C)C)NCC1COC(=O)C1 O=C(CC1=CCCC1)NC1CC1NC(C1(CSc2ccccc2)CCOC1)=O c1(C(=O)NCc2occ(C(=O)NCC(CCCC)CC)c2)cccc2occc12 N1(C(C2C(C)OCCN2C(C2C=CCS2)=O)=O)CC2(CCCN2C)C1 C1(F)(CNC(C(C)C2CC2)=O)CCCC1.C(=O)(CCCCc1cccc(O)c1)N C1(NC(c2c(C)nc(C)[nH]2)=O)CC(C)CN(C(=O)C(C2CC2)C2CC2)C1 N1(C(c2cc(C)c(Cl)cc2)=O)CCc2ccccc2C1CNC(=O)C1=CCOC1 c1(C(N2CCCC2Cc2ccccc2)C(=O)NC)cnc2c(C(N)=O)cnn2c1 Cc1cc(C)c2cc(C(=O)NCC(O)CNC(c3c(C)cc[nH]c3=N)=O)[nH]c2c1 Cc1nc(Cl)[nH]c(=NCC2CN(C(c3ccnn3CCF)=O)CC2C)c1[N+](=O)[O-] N1(C(c2cccc(OC)c2)=O)CCN(C(C2CSCC(=O)N2)=O)CC1C1CCC1 C1(C(N2CC(NC(C3CC(n4cnnc4)C3)=O)C2)=O)CC2CC2C1 N1(C(C2(CC)CC2)=O)CCC2C(C1)NC(=O)CCN2C(=O)C1=C(C)OCCC1 C(=O)(C(CCC(N)=O)n1cc(-c2cn[nH]c2)nn1)Nc1ccc(OCC)c(C)c1 CC(C)(CC(F)F)C(=O)N1CCN(C(C2CCCN2C2CCOCC2)=O)CC1 N1(C(C=CC=CC=CCC)=O)CCCN(C(c2ccc(F)c(F)c2N)=O)CC1C C1CN(C(=O)CC(C)(F)F)CCC1C(F)(F)F.C1(SC)CC(CC(=O)N)C1.C C(=O)(C(C)P(C)(C)=O)NCC1(COC)N(C(CCCOC)=O)CCC1 CCC(C)(O)C(=O)N1CCCC1CN(C(=O)CSCc1ncc[nH]1)C C(=O)CCC(F)(F)F.c1(CC)cccc(Cl)c1.C(C(=O)N)NC(=O)OCC N1(c2nnc(C(C)(F)F)n2CC2CCCCO2)CCOCC12CCSC2 C1(CC=O)C(=O)N(C)N=C1C.n1(C2CC(C=O)C2)ccnn1.C=O.CC.O C(C(C(=O)N1CC(CC(C)NC(c2csnc2C)=O)C1)C(C)(C)C)OCC=C C1(C(=O)NC(C(=O)NC2(CC)CCCC2)CO)CC(=O)CCO1 c1(C(N(C2CN(C(=O)C(C)(C)C#N)CC2F)C)=O)cc[n+]([O-])cc1 C1(NC(C(COC)O)=O)CCN(C(=O)CCN(c2ccncc2)C)C1C(C)C c1(NC(CC2CN(C(c3cccc(C)c3C)=O)C2)=O)ccc(I)c2cccnc12 N1(C(c2ccncc2Cl)=O)CCN(C(c2cnc(O)o2)=O)C(c2ccccn2)C1 c1(CC(=O)NC(CC2CC2)C(=O)NC(c2cscn2)CO)cccc(F)c1 C(=O)(C(CCN(C)C)NC(=O)C(C)Sc1ccccc1)NCC=C N1(C(C(C)C2CC2)=O)CCC12CN(C(=O)CN(C)C(c1ccsc1)=O)C2.CO S(=O)(=O)(c1ccc(O)cc1)N1CC2(N(C(c3cccc(C(=O)OC)c3)=O)CC2)C1 C1(NC(C2CCC(CNC(c3nocc3Cl)=O)O2)=O)CCCC(O)CC1 C=CC(C)(C)CC(=O)NCC1CCC1NC(=O)CCc1nnc(S)n1C N1(C(c2ccc(CCC(N)=O)cc2)=O)CC(O)(C2CC2)C1 CCCCCC(O)C(=O)N1CCCN(C(c2ccc(N)c(SC)c2)=O)C(CO)C1 C(=O)(C(F)C(C)(C)O)NC(c1cn(-c2ccc(SC(F)(F)F)cc2)nn1)(C)C Cc1ccc(SCC(=O)N)cc1.C1C2CN(C(c3cnn(C(F)(F)F)c3)=O)CC12 N1(C(C)C)C(=O)COCC1C(=O)NC1(C)CC(NC(C2COCCN2C)=O)C1 CC(N=c1nnn(C)[nH]1)c1ccc(CNC(c2scnc2C(C)(C)C)=O)cc1 N1(c2ccnc(NCc3c(C)c4c(o3)cccc4)n2)CCCC2(C1)CC2(F)F c1(C(=O)NC2CC(C)(C(=O)NC(C=C)C3CCC3)C2)sc(O)nc1C c1(-c2cn(CCN(C(=O)C(O)C3CCCC3)C)nn2)cccc(C(=O)O)c1 c1(OC)ccc2cc(C(=O)NCC(C)NC(=O)C(C)(O)C(C)(C)C)[nH]c2n1 C1(NC(C2CCC(=O)N2)=O)COC2CN(C(C3CC4(C3)CC(F)(F)C4)=O)CC12 C1(C=O)CC2CCC(C1)N2C(=O)CC1CC(C)(C)CO1.Cc1ncsc1CC.N C1(C)(C(=O)NCc2scc(C)c2)CCCN(C(=O)C(O)C2CC2)C1 C1(C(=O)NCCCCOC)CC(C)(C)CCO1.c1(C(=O)N)ccc(C(C)C)o1 c1(C(=O)NCC2(NC(C(CC)CC(F)F)=O)CCOC2)nc2nc(C)ccn2n1 c1(NC(C(=O)NC2(C#C)CCOC2)=O)cc(Cl)c(Cl)nc1C N1(C(C2C(C)(C)CCN(C(C(CC=C)CC)=O)C2)=O)CCC2(CC1)CC2C#N C1(CC(=O)N)CCCS(=O)(=O)C1.N1(C(C2CC(C)(F)C2)=O)CCSCC1CC C#CCCCCCCCNC(c1ccoc1CNC(C1(O)CCCCCC1)=O)=O CC(C)(C)CC(O)CC(=O)NC1(C(=O)NC2CCC(N=[N+]=[N-])CC2)CSC1 C12(C(=O)NCCC(C)N(C)C(c3csc(O)n3)=O)CC1COC2(C)C C1(CC(N2CCCC(C(F)F)C2)C(=O)NCC=C)CCOC(C)(C)C1 c1(CSc2ccc(OC)cc2OC)nnc2n(C)c(=O)c3ccccc3n12 c1(C(=O)NCC(CCOC)NC(C2CC(=O)CCO2)=O)c[nH]cc(C)c1=O N1(C(c2c(CCC)[nH]cc2)=O)CCC(CC(N2CC(C)C2(C)C)=O)C1(C)C c1(SC)cccc(F)c1C(=O)NC1CCN(CCNC(C2CCCN2C)=O)CC1 CCCC(C)(CC)C(=O)NC1CC2(CCN(C(C3CCC3)=O)C2)C1 c1(CC)ncc(C(N2CCCCC2C(C)NC(=O)CC2(C)CC2)=O)c(C)n1 c1(C(N2C(CNC(C3CC(=O)OC3)=O)CC2)=O)ccccc1C#CC1CC1 Cc1cc(-n2cc(C3(C)CCCN3C(c3ncc(Br)cn3)=O)nn2)cc(F)c1 CC(O)C(C=O)NC(=O)C(C)(C)C.CCC(C)N(C(=O)CCn1cncn1)C.N CC1Oc2ccc(C(=O)N(CC(C)(F)F)C)cc2C1C N#Cc1cc(Cl)c(C(=O)NCC(C2CC2)NC(c2cc3c(s2)CCC3)=O)s1 c1(C(N2CC(OC(C3C(=C)C3)=O)C(F)C2)=O)cccc(OC(F)(F)F)c1C CCCC#CCCNC(C1CC(O)CN1C(c1[nH]cc(C)c1C)=O)=O C1(F)(CNC(C(CC=C)(C)C)=O)COCCN(C(C2CCC(C(N)=O)C2)=O)C1 N1(C(=O)NCCc2ccc(I)s2)CCc2sccc2C1c1cccs1 C(CCCC(F)(F)F)N1CCN(CCC(=O)Nc2nccs2)CC1 N1(C(C2C(C)C2)=O)CC2(CCCC2NC(=O)Cn2cnnn2)C1 C1(C(N2CCN(Cc3cnc(O)nc3O)C3CC23)=O)CCc2nc[nH]c2C1 C1(O)(CNC(C2(CC)CCOC2)=O)CCCN(C(=O)CN2CCCCC2=O)CC1 C(c1cscn1)=CC(=O)N(CCC(=O)NCCCc1ccccc1)CC c1(CC(=O)NC2CCN(C(CC3CC(OC)C3)=O)C2)sc(C)cc1Br C(C(=O)N1CCOCC1)(C(C)C)NC(=O)OC.n1(CC(=O)NC)nccn1.C c1(C(C(F)(F)F)NC(c2cn(-c3cccc(C)c3)nc2)=O)c(F)cc(F)cc1F c1(C(=O)NCC2N(C(CC3CC(C)(C)OC3)=O)CC2)cc2cc(F)ccc2[nH]1 c1(CC)nnc(O)c(C(N2CCCN(C(c3cccs3)=O)C(CO)C2)=O)c1CC c1(C(=O)NC2(CC=C)CN(C(C3(C)CCC(C)C3)=O)C2)cnn(C)c1C Cc1ncc(CCC(=O)N(CC(C)NC(C2C(c3ccccc3)C2(F)F)=O)C)o1 CC(C)CCCC(=O)NCC1CC1CNC(c1cnn(C(C)C)c1Br)=O N1(C(c2ccc(Br)c(C)c2)C(=O)NCCCSC)CCc2nc(C)ncc2C1 C(=O)(C1CCc2cc(F)ccc21)N1CCC(N(C(Cc2c(C)noc2)=O)C)C1 c1(N(CCCNC(CCOCCCOC)=O)C(C)C)cncc(C#N)n1 c1(CCNC(C(C)NC(C)CC(N)=O)=O)ccc(C(F)(F)F)cc1 C1(CCNC(Cc2cnc(C)[nH]2)=O)CN(C(=O)C#CC(=O)N(C)C)CC(C)O1 c1(C(C(=O)OCCCC#N)N)cc(Br)ccc1C(=O)NC1CCOC1 Cc1ccc(C(n2cc(-c3ccc(NC4CCCC4)cc3)nn2)C2CC2)cc1 CC(CC(=O)N1CCCC(Nc2nccc(C(F)(F)F)n2)CC1)CC(F)(F)F c1(C(=O)NC2(C(=O)O)CC(F)C2)cc2c(nn1)CCCO2 CC1CCCC1(C(=O)N(C1CCOC(C)C1)C)NC(=O)C1=NOCC1 N1(Cc2c(C)ccc(N)c2)CCC2CC(C(=O)NCC(C)(C)CN(C)C)C2C1 CC1(C)Cc2[nH]nc(C(=O)NCc3cccnc3)c2C1.C(=O)CS(N)(=O)=O.C Cc1ccc(F)c(C(N2CCSCC2C(=O)NCCCC(=O)NO)=O)n1 C1(C(=O)NC(C2CCOC2)CNC(C2(OC)CC2)=O)CCN(C)C1=O N1(C(c2n[nH]c(C)c2[N+](=O)[O-])=O)CC2CCOCC2(NC(=O)C2=NNC(=O)C2)C1 C12(NC(CC=CCC)=O)CC(C)(C1)OC21CCN(C(=O)CCCCC(F)F)CC1 C1(NC(C(C)(C)C2CCCCC2)=O)CC2CCC(C1)N2C(=O)C1=CCCC1 C=CC1CN(C(c2cn3ccsc3n2)=O)CC1NC(=O)CC(C)C(C)C N1(C(CSCCC(C)C)=O)CCC(C(N2CC(C)C(F)C2)=O)(CO)C1 C12(O)CN(C1)C(=O)C2F.C(=O)(C(C)(C)C1CCN(C(C2CCC2)=O)C1)OC c1(OC)cnc(C(=O)NCC(C)(CO)NC(=O)Cc2cccc(C)c2)cn1.O c1(C(N2CCC(CN(C(C(C)N(CC(F)(F)F)C)=O)C)C2)=O)ncc(F)cn1 c1(C(=O)NC(CC)CN(C)C(c2coc(CO)c2)=O)snc2ccccc12 c1(C(=O)NC)ccc(OC)c(-c2ncn(C)n2)c1.c1(CC)nc(C(C)C)sc1C N1(C(C(CC#C)O)=O)CCN(C(c2cnn(CC3CCCO3)c2)=O)C2(CC2)C1 CCCCCC=CCN(CCC)C(=O)Cc1cc(CC)no1.C(=O)C1CC1 CC1(C)CN(CC(=O)NCCCC2(NC(=O)C=Cc3ccsc3)CC2)C1 CCCCCC(O)C(=O)NCC(C)(C)CNC(=O)C(O)CN1CCOCC1 c1(C(=O)NCC2(CNC(CC(CC)C)=O)CC2)cccc2c1NC(=O)CC2 C1CC12CCCCCC2.C1(NC(c2c[nH]c(=NC)s2)=O)C2CC3C(C2)C13C(=O)N C(=O)(C(C(C)NC(=O)CCCC(=O)C1CC1)C(C)C)N(CCCC)CC c1(SCC(=O)NC)ncnc2[nH]cnc12.C1CC(O)CN1C(C1C2COCC12)=O C1(NC(=O)CCCOCc2ccccc2)CCN(C(C23COCC2C3)=O)CC1O N1(C(c2cc(CC)oc2C)=O)CCC(C)C(C)C1.c1(C=O)n[nH]c(C2CC2)n1 CCC(CC)(CO)C(=O)N1C(CNC(C2CC2C(=O)OC)=O)CC2COCC12 Nc1ncc(C(=O)NCCC2CCCN(C(=O)CC34COCC(C3)C4)C2)cc1Cl C1(C(N(c2cccc(C#C)c2)C(C)C)=O)CC1C1CCCNC1 C1(NC(C(CC)N(CC)CC)=O)CN(C(c2ccc(C(C)C)cn2)=O)CC1(C)C N1(C(Cc2c(C)noc2)=O)CC(NC(=O)Cc2cc[nH]n2)C2(CC2)C1 c1(C(=O)NCCCC2N(C(c3ccc(CC)o3)=O)CCC2)cnc(OC)c(C)n1 S(=O)(=O)(c1cc(Br)ccc1Br)N1CC(N(C)C(C2CCC3CCC(=O)N3C2)=O)C1 c1(OC(C)C)cccc(CC(=O)NC2C=CCN(C(=O)C(F)=C3CCCC3)C2)c1 CC1(NC(=O)Cc2csnn2)CCN(C(C2(c3cc[nH]n3)CCOCC2)=O)C1 N1(C(CNC(CC)=O)=O)CC(CNC(c2ccnnc2S)=O)OC(C)(C)C1 C(CCC(=O)N(CC(C)N(C(=O)Cn1cc(C2CC2)nn1)C)C)=C(C)C CCCCS(=O)(=O)CC(=O)NC(C)CN=[N+]=[N-] C(=O)(C(CCCC)C(C)C)NCCC1(CNC(CC=CC=C)=O)CC1 n1(CCNC(CC2(NC(C(C)C3CCOC3)=O)CC2)=O)cnccc1=O C1(F)(CNC(=O)C=Cc2ccncc2)COCCN(C(C2CCO2)=O)C1 Cc1cnc(C(C(=O)NC(c2ccccc2)c2ccccc2)N(CC(F)F)C)s1 C1(C(=O)NCC2(NC(=O)CCc3cc[nH]n3)CCC2)(OC)CCC(C)C1 N1(C(C(c2ccccc2)C)=O)CC=CC1C(=O)NOCCCCC1CC1 c1(OC)cc(OC)c(N)c(C(N2CC(O)C(NC(C3CC(C)C3)=O)C2)=O)c1 C1(NC(C2CC23CCN(Cc2ccccc2Br)CC3)=O)CCc2n[nH]cc2C1 C1(C(N2CC(CC(C)NC(C34CCC(C3)OC4)=O)C2)=O)CCOC2(CCC2)C1 c1(C(=O)NCC(C)C2CCC2)cccc(Cn2cc(C3CCC3)nn2)c1 N1(C(COCC)=O)CCC2CN(C(C3(c4cncnc4)CCCC3)=O)CC12 c1(C(=O)NCC(C(C)C)NC(C(C2(O)CCCCC2)CC)=O)cc(Cl)nnc1O C1(NC(CC2C(C)CCN(C(c3ccncc3F)=O)C2)=O)CCCC(C2CC2)C1 C(C)(CCCC(=O)NCC(=C1CCCCC1)F)NC(CC1COCC(C)O1)=O Cc1cc(C(N2CCC3CN(C(=O)C(O)C4CCC4)CCC23)=O)cc(C)c1C#N c1(NC(=O)Cc2cccc(-c3cnc(F)nc3)c2)c(Cl)ncc2ccccc12 c1(C(C(C)C)NC(=O)NC2CCOCC2F)nnc2n1CCC2 c1(C(=O)NC2CC3CN(C(CC(C=C)C)=O)C2C3)cc(F)cc2cc[nH]c12 c1(C(N2CC(C(=O)NC(C)(C)CCO)CC(C)C2)=O)ccc2cc[nH]c2c1 CC(C)(CC#N)C(=O)NCc1cn(C2CCCN(C(c3ccc(Cl)o3)=O)C2)nn1 C(N=c1cc[nH]cc1C(=O)OC)C1CCC(NC(CC(CC)OC)=O)C1 N1(C=O)CCC(C)C1.C1(NC(C(C)SC(F)(F)F)=O)CCOCC1.C(=O)CC.N n1(CC)ccnc1C(=O)NCC(=C1CN(C(C2CC2C(C)O)=O)C1)F C1(CNC(CC#N)=O)CCCN(C(C2CC2c2ccc(Cl)cc2)=O)C1 N1(C(C2C(C)=C2)=O)CCC(CCNC(c2cc(C(N)=O)cn2C)=O)CC1 c1(CC(C(=O)O)NCc2c(F)ccc(F)c2O)cn2cc(Cl)ccc2n1 N1(C(c2cn(C)nc2O)=O)CCC2(CCN(C(=O)C=CSc3ccccc3)C2)C1 N1(C(CSC)=O)CC2(CCN(C(C3(NC(N)=O)CC3)=O)C2)C1 C(C)(C(C(=O)N1CCC(C)(CC(=O)NCC2(C)CCCO2)C1)N(C)C)OC Cc1cc(C(=O)NC2CC(C)(CNC(=O)C(C)CN(C)C)C2)cc(Cl)c1 C1(C)(CC)CC(NC(c2cnc[nH]c2=N)=O)CN1C(c1cc(C)c(CO)cn1)=O c1(C(=O)NCC(=C)CCNC(=O)C=CCOC)cnc2nc(C)oc2c1 c1(C(=O)NCCN(C(=O)Cc2cnco2)CCOC)nnc(C)s1 C12CCC(CN(C(=O)CC)C1)C2.c1(CN(C)C)ccc(C=O)o1.[SH](C)(=O)=O C1(CNC(CS(CC)=O)=O)CC(C)(C)CN1C(=O)Cc1cc(C)on1 CC(C)(O)C(F)C(=O)NCC(CC(=O)NC12CC(C1)C2)C1CCC1 Cc1cc(O)cc(C)c1C(=O)NC1CN(C(=O)CC(C)F)CC1C(F)F C1(CC=O)(CNC(C)=O)CCCCC1.c1(C=O)csc(C(N)=O)n1.CCC.N Cc1cccc(N)c1C(=O)NCC(C)(C)CC1CN(C(C2(C)CCCO2)=O)C1 N1(C(c2cccc(OC(C)C)c2)=O)CC2CC(C1)N(C(c1ccn(C)c1)=O)C2 C1(CC)C(NC(=O)Cc2cnc(O)nc2O)CCCN1C(=O)C(C)CCCOC C1(C(=O)N(C2CCN(C(C3CC(O)C3)=O)C2)CCO)CC2C(C1)C2(F)F.C c1(C(=O)NCC2C(NC(=O)CCc3nncs3)CC2)ccc2nc[nH]c2c1 c1(OC)ccc(C(N2CC(NC(c3cc(C)nn3C)=O)CCC2C)=O)c(F)c1 c1(CN2CCN(C(c3cscc3Br)=O)CC2)cc(F)c(F)cc1O C1(CNC(c2ncncc2F)=O)COCCN(C(=O)Cn2cc(Cl)cn2)C1 N1(C(CC(CC)C)=O)CC(C)(C)CC1CNC(=O)CCn1cccn1 C(N=c1[nH]c(N(C)Cc2ccncc2)nc2ccc(Cl)cc12)c1cnc(CC)[nH]1 CCCC(C(=O)N1CC(C(C)NC(=O)CC)C1)OCC.C1(C=O)CCOCC1.N N1(C(CCCSC)=O)CC2CN(C(=O)Cc3noc(C)c3C#N)CCC2(CO)C1 c1(CN(C(CSC)=O)C)cnn2c1CN(C(c1cnc3c(F)cccn13)=O)CC2 c1(N(CCn2c(C)ncc2)C)nc(NCCC(=O)N(C)C(C)C)c2ncsc2n1 Cc1cnc(C(N2CC(NC(=O)C(c3ccccc3)F)C3(CC3)C2)=O)c(C)c1 C1(C)(CNC(c2cn(CCC)nc2)=O)CCCN(C(C2CC2(C)C)=O)C1 c1(C(N(C(C)C)C)=O)cn(C)c2ccccc12.C1(CC=O)CCS(=O)(=O)CC1.N c1(CC)cc(C(N2CCCC2c2ccco2)=O)c(Br)s1 N1(C(CCOc2ccc(C)cc2)=O)CC2(CCCCN2C(=O)COCCCF)C1 N1(C(C2(COCC)CC2)=O)CCC(F)(CNC(=O)CC(O)CC)CC1 c1(OC(C(=O)OCC(C)=CBr)(C)C)cc(F)cc(F)c1 CC1CN(C(c2ncc(F)cc2N)=O)C(C)CN1C(c1occ2c1CCC2)=O c1(C(N2CC3C(N(C)C(c4cccc(=O)o4)=O)C3C2)=O)cc(=O)c(Br)c[nH]1 Cc1cc(=NC(=O)C(=O)NC(C)CC)[nH]o1.c1(C2(C=O)CCC2)cc(C)on1.N C(C(C)(C)C1=CCCC1)NC(C1N(C(c2c(CC)ocn2)=O)CCC1C)=O CC1(CN=c2nnc(C(F)F)c(CO)[nH]2)Cc2ccccc2C1 c1(NCCCC(C)NC(=O)OC(C)(C)C)ncc(CO)cc1Cl.C1CCOCC1 c1(NC(CCC(=C)C)C)ccc(S(=O)(=O)N2CCCC(CF)C2)cc1C#N CC(C)C(O)C(=O)N.c12ccc(n1C)C1COCCN1C2=O.C(C)(C)C.C1CC1Cl C(CC)(C(=O)N1CCC1(C)CC(=O)N(C1CC1)CC1CCOC1)=CC C1(CCC)CN(C(C2CSCC(=O)N2)=O)CC1C(=O)N(CCC(N)=O)CC C=CC(C)(CCOC)C(=O)NCC1(O)CCCN(C(=O)CCCc2ccsc2)C1 C1(NC(C(CC=C)C)=O)CCC2CN(C(C3C4CCCCCCC34)=O)CC2C1 C(=O)(C(C)(C)C(F)F)NCc1ccc(C(N2C(CO)CC(OC)C2)=O)s1 c1(N2CC(CNC(C(CCC)(C)C)=O)OCCC2)ccccc1[N+](=O)[O-] N1(C(C(C)C2CCC2)=O)CCCN(C(c2cc(F)cnc2O)=O)CC1CO S(=O)(=O)(CC(=O)N(CCCN(C(=O)C(CC)n1ccnc1)C)C)NCC c1(NC(C2CC(F)CN2Cc2c(O)cccc2Br)=O)c(F)c(F)nc(F)c1F CC1C(c2ccccc2)CCN1C(=O)C(=O)NC1COCC1CC1CC1 N1(C(CC(C)C)=O)C(CNC(=O)CC2(C)CCCO2)CC2COCC12 C(=O)(C1CCCc2sccc21)N1C(C(C)(C)NC(C2CC2F)=O)CCC1 Cc1ncc(CCC(=O)N(C)CCN(C(=O)CC2CCC(C)O2)CC)c(O)n1 CC1(C)CC(C)(C(=O)NC2CCCC2)C1.C1(O)(C(C=O)(F)F)CCOCC1.C C1(OC)CC(NC(=O)Cc2cnccn2)CN(C(=O)C=CC2CCCCCC2)C1 C12(CC(=O)NC3CN(C(c4cncc(SC)c4)=O)CC3C)CCC(CC1)CC2 Cn1cc(C=CC(=O)N(CC(=O)NCC(c2cccs2)O)C2CCC2)cn1 C1(NC(c2cc(C)oc2)=O)(CNC(C2CCOC(C)C2)=O)CC2CCC1CC2 C(=O)(C(C)(C)CN(C)C(c1ccn(C)n1)=O)N(CC(C1CC1)OC)C Cc1cccc(-n2nc(C3CC34CC4)nc2C2CC(n3cncn3)C2)c1 N1(c2[nH]c(=NCc3c(C)nc[nH]3)[nH]c(=N)n2)CCC(C)C2(CCCCC2)C1 c1(C(N)=O)cccc(C(N2CC(NC(=O)COCCF)CC(F)C2)=O)c1F C1(NC(c2c(OCC)scc2)=O)CC2CC(NC(c3cnncc3C)=O)CC12 N1(C(C(C)c2ccco2)=O)CCCC2(CNC(c3n[nH]c(O)n3)=O)CCCC12 CCC1=NOC(C(=O)NC2CCN(C(=O)CNC=O)C2)C1.C(C)(C)C.O C=C=CC(C)C(=O)N1CC2CC1C2NC(=O)CC(N1CCCCC1=O)C Nc1c(C(N2CCC(CCNC(C3CCCS3)=O)C2)=O)cccc1Br C1(CCC)CN(C(c2cnccc2C)=O)CCN1C(C1COC(=O)N1)=O C12(C(N3CC(O)(CC=C)C3)=O)CCC(CN(C(=O)CN(C)C(C)=O)C1)C2 CCC1=NOC(C(N2CC(O)CC2C(N2CC(F)CC2C)=O)=O)C1 C(=O)(CCC(CC)CC)N1CCN(C(c2ccc(CC)c(O)c2)=O)C2C1C2 C1(C(=O)NCCc2cccc(C)n2)CC2(CCN(C(=O)Cc3cnns3)C2)C1 CC(C)C(CCC(=O)N1CCOCCC1C)NC(c1coc(C(N)=O)c1)=O C1(C(NOCC(=O)OCC)=O)CCN(C(C2CCC=CCC2)=O)CCO1 C(=O)(C1=C(C)CN(C(c2ccccc2-n2cc(CC(C)C)nn2)=O)C1)OC c1(C(N2C3C(C(=O)NC4CCCC(C)C4)C(C3)C2)=O)c(F)ccc([N+](=O)[O-])c1F c1(-c2cn(CCCN(C(C(n3ccc(C)n3)(C)C)=O)C3CC3)nn2)cccc(N)n1 C1(NC(=O)C=CC2CCOC2)CC2CC(C1)N(C(=O)Cc1ccc(F)cc1F)C2 c1(C(=O)N(Cc2ccccc2)CC2(C3(O)CCOC3)CC2)ccc2nccn2c1 C1(C(N2C(NC(=O)OC(C)(C)C)C(C)CC2)=O)(NC)CC2(CCC2)C1 c1(CN(CCCCCC)C(C)C)cccc(-c2nc(-c3ccncn3)nn2C)c1 N1(C(C2CCN(C(C)=O)C2)=O)CC2(CC(NC(c3cc4sccc4[nH]3)=O)CO2)C1 c1(SCC)cnccc1C(=O)N(C)C.C1COCCN1C(=O)C(O)CN(C)C C1(C(N(CCC(C)C)C)=O)CC2(CCC2)CO1.c1(C(C(=O)N)OC)ccccc1 CC(C)(C)C(O)CC(CO)NC(c1cc(F)c(F)cc1Cl)=O N1(C(=O)Nc2cccc(C)c2)CCOCC(C(=O)NCc2ccc(Cl)nc2)C1 C12(C(N3CCC3)=O)CC1COC2(C)C.C1(C(=O)OC)CCCC1C(=O)NC c1(C(=O)NC2CC(CNC(C3(CC#C)CC3)=O)C2)ccc(C#N)cc1F c1(N2CC(C=O)C2)ccccc1C#N.C1(C(=O)OC)CC1CC(=O)N.C1CC1 C(=O)(C#CC(C)(C)C)NCc1c(F)ncc(C)c1.C(c1nccs1)=CC=O.N Cc1ccc(F)cc1-c1nc(C2CSC2)nn1C1CCC(F)(F)CC1 CCCC(CC(=O)Nc1conc1CC)NC(C1CC(O)C1)=O c1(NC)ccc(CC(=O)NCC(C)(C(C)C)NC(c2c[nH]nc2)=O)c(F)c1.O N1(C(CCOC)=O)CC(NC(=O)Cn2cnc(Br)n2)CCC1C C1(N(C(CCC(=O)NCCC)=O)C)CCCN(C(=O)C(O)C2CC2)CC1 Cc1ccc(C(N2CCCC2c2ccc(C)nc2)C(=O)NC2CCCC2)c(Cl)c1 C1(C(=O)NCc2nnn(CC)n2)C(C)CCN1C(=O)CCCc1ncco1 C(C)(CCCC(C)C)(c1nnnn1C1(C)CC1)NCc1cnc(C)n1C c1(OC)ccc(Cc2scc(NC(C3CC34CCOC4)=O)n2)c(OC)c1 N1(C(C2(CCC)CCC2)=O)CCCCC2(CCN(C(=O)C=C(C)Cl)C2)C1 N1(C2CCCN(C(CC(COC)C)=O)C2)CCN(C(c2cc(Br)co2)=O)CC1=O C(=O)(C(CCCC1CC1)N1CC(C)OCC1C)NCCCC(=O)OCC C1(COCC(=O)NCC(C)N(C)C(c2csnc2Br)=O)CCCCC1 c1(OCC(=O)N(C)CCN(C)C(c2ccc(Cl)s2)=O)ccc2c(c1)CCCC2 C12CC(C1)C(C)O2.C(=O)CCCn1ccnc1.C(C(=O)N)OCCOC.C c1(C(N(CC(C)N(C(c2nc(CC)oc2)=O)C)C)=O)ccc(CO)cc1 CC(C)C(O)CC(=O)N1CCCCCC1C(=O)NC(c1ccc(O)cc1)C Cc1cc2ccc(C(=O)NC3C4CN(C(=O)Cc5cscn5)CC34)cc2[nH]1 C(=O)(C1=CCC2CCC1N2C(c1nn(C)cc1Cl)=O)NCCC(=O)NC n1(CC)cc(C=O)c(C(C)C)n1.C1CCC1.C1(C=O)CN(S(C)(=O)=O)C1 CS(=O)CCC(O)C(=O)N1CC(O)(CNC(C2(Br)CC2)=O)C1 c1(C(N(C(CCNC(CCC)=O)C)C)=O)cc(S(C)(=O)=O)ccc1CC Cc1ccc(C=CC(=O)NCCC2COCCN2C(=O)C(N2CCCCC2)C)o1 c1(C(N2CCCC(CN(C)C(c3ccc(Cl)o3)=O)C2)=O)ccccc1C#N CCC(C(=O)N1CCC2CCN(C(=O)COC(C)(C)CC)CC12)C(C)(C)CC c1(C(=O)NC(CNC(C2CCCC(=O)N2)=O)CO)[nH]cc2c1CCCC2 c1(CN2CCCC(C(N3C(C)CCCC3)=O)C2)cc2c(cc1Cl)OCCO2 C#CC1CCC(C(=O)NCCC2CCN(C(=O)CC3CCC(=O)N3C)C2)CC1 c1(C(=O)NCCC(C)N(C)C)cnn(CC)c1.c1(CC)cccs1.C(=O)C.N c1(NC)cnccc1C(N1CCCC1C(C)NC(=O)CCc1cccs1)=O NC1C(C(=O)NCc2cnn(-c3ccccc3)c2)CC1C(F)(F)F c1(N2CC(Br)=C(C)CC2)nc(=N)[nH]c(=NCCn2ccc(O)nc2=O)[nH]1 c1(NCCC2N(C(CC3CCC(C)CC3)=O)CCCC2)cc(O)nc(O)n1 C=CC(CCC)CC(=O)N1CCCC(NC(c2coc(COC)n2)=O)CC1 Cc1ncnc(C)c1C(N1CC(CNC(C2CC2F)=O)C(c2cncn2C)C1)=O C1(NC(C2CN(C)C(=O)N2)=O)CC1C1CCCN(C(=O)CCCCCNC(N)=O)C1 Nc1ccc(C(=O)NCC(C2CC2)NC(C2CC2C=O)=O)cc1O.CCO N1(C(C(CC)CC(C)C)=O)CC2(CCN(C(=O)Cc3cncnc3)CC2)CC1C c1(C(=O)NCCCC2N(C(CC(=O)NC)=O)CCC2)nn(C)cc1C C1(C(=O)NC2C(C(C)C)CCC2)CCC(c2nc(-c3cccnc3)no2)CC1 C1(C(=O)NC(C2CCN(C(=O)CCCCCF)CC2)C)CSC2(C)CCC(=O)N12 C(=O)(CC(CC)C(C)C)NC(CC=C)C(N1CCC(C2CC2)C1)=O CCC(C(=O)N1CCC(C(C)(C)C)C1)NC(=O)OC(C)(C)C C1(C(N(C2CCCN(C(C(=Cc3cn[nH]c3)C)=O)C2)C)=O)C2CCC(F)(F)C12 c1c(C)occc1=O.C1CCC(F)C1.C(C(=O)NC)=CC=CC.C(=O)C C1(NC(=O)Cc2c[nH]nc2O)CCCCCC1NC(c1cc(O)cc(=O)o1)=O Cn1c(=O)n(C)c2cc(N3CCCC3CCCO)c([N+](=O)[O-])cc12 c1(OC)ccc(N)c(C(N2CC3CC2CN3C(C2CC2c2ccnn2C)=O)=O)c1 C1(NC(C(CC#C)(C)NC(C2CCC2(F)F)=O)=O)CC(C)(C)C12CCC2 c1(C(N2CCC(N(C(=O)C3CC3)CC)C2)=O)cccc(NS(N)(=O)=O)n1 C=C(C)C(C)(O)C(=O)N1CCC(O)(CNC(c2cc(O)ncc2Br)=O)C1 C1(C=O)CCCN(c2ccc(Cl)nn2)C1.c1(C(=O)NCC)coc(C(F)F)n1.N Nc1c(C(=O)NCC=CCNC(c2cccc(=O)o2)=O)cc(Cl)cc1Br C12(NC(C(CC)O)=O)CC3CC(C1)CC(NC(=O)Cc1cnco1)(C3)C2 N1(C(CC(C=C)(C)O)=O)CC(NC(=O)C(C)=CCC)CC2(CCC2)C1 O=C(C1=CC2CCOCCC12)NCCNC(c1cnc(Cl)cc1Cl)=O N1(C(C(CCC)N(C)C)=O)CC(C)OC(C)(C)C1.c1(C(=O)N)cn(C(C)C)nn1 CC1CCN(C(C2CCC(NC(=O)CP(C)(C)=O)CC2)=O)C(C(N)=O)C1 c1(CC(=O)NC2CN(C(=O)C(F)F)CCC2O)cn2cc(F)ccc2n1 c1(C(N2C3C(NC(C4C(C)CCC4)=O)C(C3)C2)=O)ccc([N+](=O)[O-])nc1 c1(CC)nc(C)c(C(=O)NCCC(O)CNC(C2(OC)CCSC2)=O)o1 C1(NC(C2CC2[N+](=O)[O-])=O)CCC(NC(C2CC2C2CC2)=O)CC1 C(=O)(C(C(C)(C)C)n1ccnn1)N1CCC(O)(CN(C(c2cc(C)ns2)=O)C)C1 Cc1ccccc1-n1nnnc1C(c1cn[nH]c1)NC1(C(=O)N(C)C)CC1 C(C)(C(C)(C)C(=O)NCc1cccc(O)c1F)NC(c1cnc(CC)nc1)=O c1(CC(=O)NC(CN(C(c2cn[nH]c2)=O)CC)C)cccc(C)c1 C1(C(N(C2CN(C(C3CCSCC3)=O)C2)C)=O)CC2C=CC1C21CC1 c1(NCCCN(C(C2(CC#C)CCCC2)=O)C)ncnc2sc(C(F)(F)F)nc12 CCC(C)CC(=O)NCC(C)CNC(c1oc(Br)nc1C(F)(F)F)=O CC(C)C(CO)CN=c1nc2c(ncn2C)c(NC(C2CSC2)C)[nH]1 N1(C(C(CC)n2cncn2)=O)CC2CCC(C1)N2C(C1(C)CC1(F)F)=O C1(CN(C(=O)COCC2CC2)C(C)COCC)CCOC1 Cc1ccc(C(=O)NC23CC(NC(c4nn(C)c(Cl)c4Cl)=O)(C2)C3)c(C)n1 C(CC(O)CC(=O)N1CCC(CNC(C2CCCCC2(C)C)=O)CC1)SC C(C(CC(C)C)C(=O)NCCCCCCNC(=O)C(=O)NC1CC1)OC c1(C(=O)NCCCCCNC(CCOCCC)=O)cccc(S(C)(=O)=NC)c1 c1(CCOC)c(C)[nH]c(C=O)c1C.C1CCC(N(C(=O)C)C)CC1.C(C)=O.N C1(C(N2CC(NC(C(CSC)C)=O)C2)=O)Cc2nccnc2C1 CCC1=NOC(CC(N2CCC(C(O)CNC(=O)C(F)C3CCCC3)CC2)=O)C1 C12(NC(CC=C=C)=O)CCC(F)(F)CC1CN(C(=O)CC1CC=CCN1C)C2 c1(C(N(C)CC2CCN(C(=O)CCC3CCCCO3)C2)=O)ccc2nc[nH]c2c1 C1(C(=O)NC(C(CCC)C)CO)CCN(C(=O)C2=CCC(C)(C)CC2)O1 C(=O)(CC1C(=O)Nc2ccc(Cl)cc21)N(CCNC(c1cc(CC)c(C)s1)=O)C C12(NC(C3C4COCC34)=O)CC(NCc3n[nH]cc3Cl)(C1)C2 c1(C(N2CCCC(F)(C(N3CCCCC3C3(O)CC3)=O)C2)=O)occ2c1CCC2 CCC(CC)C(c1nnnn1C)NCc1csc(Cl)c1 C(C)(C(=O)NC1CC(NC(C2CC(OC(F)F)C2)=O)C1)NC(C)=O C(=O)CCCCCN(C)C.C1(C(=O)NC(c2cn(C)cn2)C)(C)CCCCC1.N CCCC(C)(CC)C(=O)NC1CCCCC1NC(c1cc(C(F)F)cc(C)c1)=O c1(N2CCC(OC)(CO)CC2)nc2ccccc2c(=NCCC#CCO)[nH]1 N1(C(C2N(C(C(c3ccccc3)C)=O)CC2)=O)CCC(N(C)C)C1 c1(CC(C)OC(c2c(C)n(C)cn2)=O)ccc([N+](=O)[O-])cc1F C1(NC(c2c(C)ccs2)=O)CCN(C(=O)C(c2ccccc2)F)C(C)C1 N1(C(C(C2(OC)CCCC2)(F)F)=O)CC2(CCN(C(C3CCCC3O)=O)CC2)C1 c1(C(=O)NC(C)(CNC(C2CCC3CC23)=O)C2CCC2)ccc2[nH]ccc2c1F c1(C(=O)NC2C(C)(C)CN(C(=O)CCCN=[N+]=[N-])C2)ccc(C#N)c(Cl)c1 C1(C)(OCC)CCN(C(=O)C(C)C)CC1.C(C(C)C)=CC=O.C(C)=O Cc1ccc(F)c(N2CCCC(NC(=O)CC3CNCC(C)(C)O3)C2=O)c1 N(C1c2ccccc2CC1NC(=O)CCCF)C(C(C(C)(C)C)SC)=O C=CCC(C)(CC)C(=O)NC1CCN(C(=O)CCOCC(C)C)C1C1CC1 CC1(NC(C2CC3CC3N2C(=O)CC2CCCOCC2)=O)CC(F)(F)C1 c1(C(=O)NCC(C)CNC(=O)CC2CC=CCC2)n[nH]c2c1CC(C)(C)C2 C1(OC)CC(CNC(=O)C(C)c2ccco2)N(C(c2ncccc2Br)=O)C1 C1CC1C1CCCN(C(=O)CC2CC(C)(C)CO2)C1.C(C=CC=O)(CC)=CC C1(C(=O)NC2CC(n3cncn3)C2)C(O)CCN1C(C1CC=CC(O)C1)=O N1(C(=O)CCOC2CN(C(C3(O)CCCCC3)=O)C2)CCC2(CC1)CC2CO c1(C(N2CC(F)(C(=O)NCCC3CCC3)C2)=O)cc(F)cc(Br)c1Cl c1(OC)cc(C(=O)NC(C(=O)N(C2CCNC2=O)C)C(C)C)n(C)n1 c1(CC)ccc(C=CC(=O)N(CC(C)NC(c2cc(F)n[nH]2)=O)C)cc1 C(C1OCCc2sc(F)cc21)NCc1c(F)c(Br)ccc1Br C1(C)(C(N(C)CC2(CO)CC2)=O)CCN(C(C2CC2(C)C(F)F)=O)CC1 C=CCC(CC=C)C(=O)N1CCC(CN(C(=O)C2=C(C#N)CCC2)C)C1 Cc1cc(C(=O)NC2CC3(C2)CC3NC(=O)C(C)C2CC2)oc1Br c1(C=O)ccc(F)c(C)c1.CCC(C)(C(=O)NCC1(C)CC1(F)F)OC.N c1(N2CCC(CS(N)(=O)=O)CC2)ncnc2c1ncn2C1COCC1O N1(C(CCCCN(C(CC2C(C)OCC2)=O)C)=O)CCC(O)C12CCC2 C1(CC(=O)NC(c2onc(C)n2)CO)CC(C)N(C(c2cn(C)nc2C)=O)C1 c1(C(N2CCC(CCC)CC2)=O)ccc2c(n1)CN(C(c1cc[nH]c1C)=O)CC2 Cc1occc1.c1(C(C(=O)N)N(C)C(C2(C)CC2)C)ncc(-c2ccccc2)s1 c1(C(N(CCNC(C2N(CCC)C(=O)CC2)=O)CC)=O)cccc2c[nH]nc12 c1(C(N(CC(C)NC(c2cc3occc3s2)=O)C)=O)cnc2c(c1)CCC(=O)N2 N1(C(CC=CC=C)=O)CCc2[nH]nc(CNC(c3cnn4c3CCCC4)=O)c2C1 c1(OC)ccc(C(=O)NCC2COCCN2C(C2CCC(C)CC2)=O)cc1 C=C(C)CC(C(=O)N1CC(CC(=O)NCc2cnc(C)c(C)c2)CC1(C)C)OC Cc1ccc(NC(c2ccc(F)c(C(C)O)c2)=O)cc1C(=O)NC(C)C C1(C)(CCC(=O)NCC(CC)OC)CN(C(=O)C(c2ccnn2C)C)C1 Cc1ccc(C(=O)N(C2CCCC(NC(=O)C=CC3CCC3)C2)C)cc1[N+](=O)[O-] c1(CNC(CC)C(C)C(F)F)cc([N+](=O)[O-])c(C)cc1C CCC(CC)C(=O)N(CCNC(c1ccc(F)s1)=O)Cc1ccc(Cl)nc1 C(=O)(CCC(C)(C)F)NC(C)CN(C)C(c1ccc(C(C)(C)C)cc1)C C1(CC#N)CCN(C(=O)CCC2CCCN2C(=O)CCCCBr)CC1 c1(C(N2CCC(NC(c3csnn3)=O)CC2)=O)n[nH]c2c(Cl)cccc12 C1(C(N2CCN(C(CC)=O)CC2)=O)CC12CCN(C(=O)CN1CCCC1=O)CC2 C(=O)(CCCCCCCS(C)(=O)=O)N1C(C(C)NC(C(F)OC)=O)CCC1 C1(NC(c2c(C)nc(C3CC3)s2)=O)CN(C(c2ccoc2)=O)CC12CCC2 c1(C(=O)NCCC2(CNC(C(CCCC)N(C)C)=O)CC2)cc2ccccc2[nH]1 C(=O)(C(C)(C)CC(=O)N1CC2C(CNC)C2C1)OC.C1CC2CCC(C1)C2O.C N1(C(COCCC)=O)CC(NC(c2nccs2)=O)C(C)C1 C1(NC(C2C(CC)OCC2)=O)C2CC3C1C3C2C(=O)NC1CCN2CCC1C2 C#Cc1ccc(C(=O)NC(CNC(=O)C(=Cc2ccccn2)C)CO)c(F)c1Cl C1(C)(CNC(c2cc(C(C)(C)C)ncc2)=O)COCCN(C(C2(O)CC2)=O)C1 C1(C#N)(C(=O)NCC(CNC(c2cn(C)c(=O)n2C)=O)CO)CCCC(=O)C1 Cc1cc(C(=O)NC2CCC(CNC(=O)Cn3nccc3C)C2)cnc1O Cc1cc(C(=O)NC2CC(C)CN(C(=O)C=CCN3CCOCC3)C2)nnc1O C(=O)(CC1OCCc2sccc21)NC(CC1CN(C(Cn2ccc(C)n2)=O)C1)C c1(NCCC(=O)NCC2(C(=O)OC3(C)CCCC3)CC2)ccc(Cl)cc1Cl Cc1cc(C(=O)NCC2CN(C(=O)C(N)=O)CC23CCC3)c2n[nH]cc2c1 CC1C(C(=O)Oc2ccc(C(=O)OCCSc3ccccc3)cc2)=NOC1C Cc1cc2c(ncn2C)c(NCC2CN(S(=O)(=O)C(C)C)CC2C)n1 C(=O)(C1OCCc2ccccc21)N1C(C2CCN(C(C3CCOC3)=O)C2)CCC1 c1(C(N2C(CC(C)(C)C)CN(C(C3(C)CC3)=O)CC2)=O)ccc2c(n1)CCC2 CC1(C)CCC(C=O)(NC(=O)CC2CC(C3CC3)C2)C1.C1COCC1N=[N+]=[N-].N c1(C(=O)NCC(CNC(C(C)Cn2ccnc2)=O)O)cnc(=N)[nH]c1 c1(C(=O)N)cn2cnnc2cn1.C1(CC(N2CCCC2)=O)CCCS(=O)(=O)C1.C C1(C(N2CC(CNC(C3CC(=O)NC3)=O)C2)=O)CCc2nnc(O)n2C1 c1(C(=O)NCC(CNC(c2c(C(C)C)c[nH]n2)=O)F)cccc([N+](=O)[O-])c1N C1(NC(CC(C)N(C)C(c2ncccc2O)=O)=O)CCC=CCCC1 C1(NC(CCN(C(C)C)C(c2cnco2)=O)=O)CCC(C)(O)CC1 C(C)(CC1=CCCCC1)NC(CC1CC(NC(COC(C)=O)=O)C1)=O c1(C(=O)OC)cc(Br)ccc1S(=O)(=O)NC1CCc2cc(C#N)ccc2C1 C1(CC(=O)NCCCNC(C(CSC)O)=O)OCCOC1(C)C.C1CCCC1.C C1(C(N2CCC2CNC(c2cc(-c3ccccc3)ns2)=O)=O)(CC)CCCC1 N1(C(COCC(=O)NC)=O)CCCC(F)C1.c1(C(C(=O)N)=O)cnn(C)c1 c1(CNC(c2cc(-c3cccc(F)n3)cnc2F)=O)ccnc(F)c1F C(=O)(C1=NN2CCCN=C2N1)N1CCC(N2CCN(C(CC(C)CF)=O)CC2)C1 c1(N(C(C)CNC(=O)CC2OCCC2(C)C)C)nc2cccc(Br)c2o1 N1(c2cc(COC)ncn2)CCCC(NC(C2C=CCCC2)=O)C1C c1(C(=O)NC(c2ccc(F)cc2)(C)C(=O)O)cc(F)cc(I)c1N Cc1nccc(C(=O)NC2C3CN(C(c4cc(CC5CC5)on4)=O)CC23)c1O C1(OC)CC(CNC(C2CNC(=O)N2C)=O)N(C(C2CNC(=O)N2)=O)C1 N1(C(C=C(CCC)C)=O)CCC2CCCN(C(C3(C(=O)OC)CC3)=O)C2C1 S(=O)(=O)(c1cccnc1NCCCCCCF)NCC(C)(C)N(C)C c1(CNCCC2CCN(C)C2)cccc2c(O)cccc12 Cc1cnccc1C=CC(=O)N(C1CN(C(C2CC(F)C2)=O)CC12CC2)C C1(CC(=O)N(CC(C)(C)C)C)C2CCC(C2)N1C(C1CC=C(C)CC1)=O.C c1(-c2cn(C3CCN(C(c4ccc(C(F)F)o4)=O)C3)nn2)ncc(F)cn1 C1(NC(CC2(OC)CCOCC2)=O)CC(O)CN(C(=O)Cc2ncoc2C)C1 c1(C(C)NCC(=O)NCCCCC)c(F)cccc1Cl N1(C(C=Cc2ccc(C)o2)=O)CCC2(CCC(NC(c3ccnnc3)=O)C2)CC1 Nc1cc(Cl)nnc1C(=O)NC1(CNC(c2c[nH]cc(Br)c2=O)=O)CC1 c1(C(N2CC(NC(CC3N(C(C)C)CCC3)=O)C(C)C2)=O)cccc2sncc12 N1(C(C#CC2(C)COC2)=O)CC2(CCC(NC(C3CC4(CCO3)CC4)=O)CC2)C1 C=C=CCCC(=O)N(CCC(=O)NCc1csnc1C)CC c1(C(=O)NCCC(=C)C)cc(Br)n2c1CCC2.c1(C(=O)N)ccc([N+](=O)[O-])o1 CCCC(C)CCCC(=O)NCC1CN(C(c2oc(CC)cc2C)=O)CCO1 CC1CN(C(C2(C3(O)CCC3)CC2)=O)CCC1NC(c1cc([N+](=O)[O-])c[nH]1)=O C(=O)(C1=CC(O)C(NC(=O)COC2CCNCC2)C1)OC c1(C(=O)N)cnc2ccc(C)cn12.N1(C(C2(C(F)F)CC(=C)C2)=O)CCC(C)C1 C1(CCNC(C(CC)OC)=O)CCN(C(c2cc(OC)no2)=O)CC1(F)F C(=O)(C1=CC2(CCOC2)C1)N(C)CC1CCN(C(=O)C=CC2CCOCC2)CC1 c1(OCC)cccc(CC(=O)NCCN(C(=O)C(F)OC)CCOC)c1 c1(CC)nc(C(N2CC(F)(C(=O)C3CC3)C2)=O)co1.c1(C=O)ccccc1.N C(=O)(C(F)C(F)(F)F)N1CC(CNC(C2OCCN(C)C2)=O)OCC1 c1ccccc1C#N.C1(C=O)(CNC(C(C)OCCN(C)C)=O)CCCCC1.N C(=O)(C(CCC1CC1)NC(=O)C(C)CCN(C)C)NC(c1nc(C)on1)C C(CC(O)C(=O)N1CCCCC1CCNC(c1[nH]nnc1C)=O)SC CC1=C(C(=O)N(C2CCCCN(C(=O)CCC(C)N(C)C)C2)C)CCC1 C(=O)(C1=C2CCCN=C2NN1)NC(CCCNC(CSC)=O)C c1(CC)cc(C(=O)NC2CC(C)(NC(C3CCCCC3O)=O)C2)ccc1Br C(=O)(C(C)CC(=O)c1ccccc1F)NC1CCN(C(Cc2nc(C)[nH]n2)=O)C1 CC1c2cc(C(=O)O)ccc2OC1CNC(C1CC(=O)C1C(C)(C)C)=O Cc1ccc2c(C(N3CCC(C4(NC(=O)Cc5cnsc5)CC4)C3)=O)coc2c1 c1(C(=O)OC)cccc(NC(c2ccc(SC)c(SC)c2)=O)c1O CC1CCC(NCc2ccc(F)c(F)c2)C(OCc2ccccc2)C1 CC1CC(NC(C2(c3cc[nH]n3)CCC2)=O)CN(C(c2ccc(C#N)cn2)=O)C1 C1(NC(c2ccc(C)cn2)=O)CC1C1CCCN(C(c2cc(F)ccc2F)=O)C1 C#CC(C)(C)C(=O)NC1CCC(N(C)C(c2cc(N(C)C)ccn2)=O)C1 C12(NC(C3C(CC)CCCC3)=O)CCC(C1)N(C(c1cnc(SC)n1C)=O)C2 c1(C(N2CC(CC(=O)C(F)(F)F)C2)=O)ccc2ccnc(O)c2c1 N1(C(=O)CCCCF)CCN(C(=O)Cc2ccccc2CO)C(CO)C1 C1(NC(C2C(C(=O)OCC)C2)=O)CCC(NC(c2cscc2Cl)=O)C1 Cc1oc2ccccc2c1CC(=O)NC1CN(C(C2CCC=CCC2)=O)C2CC12 Cc1cccc2c1CC(C(=O)N(C)CCOCC)N2.C1(C(=O)N)NC(=O)CC1C c1(CC(=O)NC2CC(NC(CCC(=C)Cl)=O)CC2O)cccc2sccc12 C1(C(C(=O)N(CCC)C(C)C)C)CCCN(C(=O)CC2(O)CCCC2)C1 N1(c2ccnc(N(C)Cc3nc(C)sc3)n2)CC2CC1C1CC21 CC(C)C(O)C(F)(F)C(=O)NCC1CN(C(=O)Cc2cccs2)C1 c1(NC(CCC)CCO)[nH]c(=NCCN(C)C(C)C)nc2c1ncn2C C(=O)(CCC(C)N(C)C)N1CCC(CCC(=O)NCC(COCC)(C)C)C1 C(C1=CCN(C(C2(F)CCN(C(=O)C(C)S(C)(=O)=O)CC2)=O)CC1)OC N1(C(C(CC)OCC)=O)CCC2(CCCC(C)O2)CC1.c1(CC(=O)N)ccsn1 CCCCCCCC(=O)N(C1CCN(C(=O)Cc2cc(F)ccc2Cl)C1)CCO C1(C(N2CC(N(C)C)OCC2)=O)CCN(C(C2C3CCC(F)C23)=O)C1(C)C C1(C(=O)NC2(C(N(OC)C)=O)CC2)CN(C)CCN1C(C1COCCC1C)=O C(CCCCCC)(C(=O)NC)N(c1ccc(CN(CC=C)C)cc1)CC.C1CC1 C(=O)(C1=CCC(F)(F)CC1)N1CC(N(C)C(c2ccc3ccn(C)c3c2)=O)C1 C1(NC)(CO)CN(C(=O)CCc2ccccc2)C1 Cc1ccc(OCCC(=O)N(CC(C)NC(=O)C(c2ccnn2C)C)C)cc1C c1(N2CCCC(CCOC)C2)ccc(S(=O)(=O)NCc2ccc(C)cc2)c(Br)c1 C1(CC=C)(NC(c2cncc(SC)c2)=O)CC2CCC(C1)N2C(C1CC1C)=O CC(C)CCNC(c1nccn1C(C)C)=O.C1(C(=O)N)CN(C2CCOC2)C1 C1(NC(C(c2ccc(F)cc2)C)=O)COC2(C1)CN(C(C1CCCC(=O)N1)=O)C2 N1(C(Cc2nc(C)on2)=O)CCC2CN(C(C3COCCN3CC(F)F)=O)CC12 c1(CC)ccc(C(N2CCC(C)(C(=O)Nc3cccc(C)c3)C2)=O)nc1 c1(CC(N2CC(CC)N(C(=O)CC)CC2)=O)ccc2c(c1)OCO2.C(=O)(CO)N N1(C(CC(C)NC(C2CC2OC(C)(C)C)=O)=O)CCC2(CC(F)C2)C1 C(=O)(CC(C)C(C)(C)C)NC(C(=O)NCC(CC#C)(C)CO)Cn1cncn1 C1(NC(c2cc(CC)n(C)n2)=O)C(C)CCC12CCC2.c1(C=O)ccn(C)c1.N C1(C=C)(C(=O)NCC(CC=C)(C)C)CCN(C(c2ccc(C(C)C)o2)=O)C1 N1(C(C(=O)NC2N(C)CCCC2)=O)CC(c2ccccc2)C2(CCC2)C1 Cc1cc(OC(C)C(=O)NCC(C)N(C(=O)CC2CCC(=O)N2)C)ccc1Cl C1(CC(=O)NCC(C)CNC(=O)C(C2CCOCC2)=O)CC2CCC1O2 c1(C(=O)NC(CO)C(c2ccc(Cl)cc2)O)cc(N)ccc1C(F)(F)F c1(C=O)cccn2nnnc12.C1(F)(CNC(C(N2CC(C)C2)C)=O)CC(C)C1 C1(CNC(c2cc(C)c(O)nn2)=O)CC2(CO1)CN(C(c1cc(Cl)cn1C)=O)C2 N1(C(c2nc(CC)sc2)=O)CC(=O)NCC1C(N1CC2CCOC2C1)=O CC1CCc2[nH]c(NC(N3CC(CNC(=O)C(F)(F)F)C3)=O)cc2C1 C1(C(=O)N)CCN(S(=O)(=O)N(C)C)CC1.CC1CN(C(c2cc(F)c[nH]2)=O)CC1 C1(NC(C2C(CNC(c3cn(CC)nn3)=O)C2)=O)CC2(CCOC2)C1 CCCC(C)(O)C(=O)NC1CCCC(NC(=O)CCCN=[N+]=[N-])C1 C(=O)(C1=NN(C)C(=O)CC1)N1CC(C)N(C(C2CCCC2)=O)CC1C Cc1nnc2n1CC(C(=O)NCC(C)(C)CNC(C1(C)CCN(C)C1)=O)C2 N1(C(C2CCCNS2(=O)=O)=O)CCC2OCCN(C(=O)C=Cc3ncc[nH]3)C2C1 c1(OC)cccc2c1C(C(=O)NCCC1CCCN1C(C1CC1C)=O)CC2 C(C(=O)N=c1cc(CC)n(C)[nH]1)N1CCN(C(C(CCCC)F)=O)CC1 C(=O)(C1CCCc2c[nH]nc21)NCCN(C(c1ccc(C)n(C)c1=O)=O)C1CC1 C(=O)(CC(C)(C)C(F)F)N1CCC(CNC(c2nc(C)n(C)n2)=O)(CO)CC1 O=C(CCNC(=O)C(C1(O)CN(C(=O)CC2OCCO2)C1)F)NO C1(C(=O)N)CCCC1S(C)(=O)=O.N1(C(CCOCC#C)=O)C2CCC1C(C)C2 Cn1cnn(CCC(=O)NC2CC(O)(CNC(=O)CCCn3cccn3)C2)c1=O Cc1ccc2sc(C(N3CCCC3CCNC(C3CCSC3)=O)=O)cc2c1 C1CC(=O)N(C)C1=O.C1(C(=O)N)(CNC(C2N(CC)CC2)=O)CCCC1 N1(C(C(C#N)C2CC2)=O)CCN(CC2CN(C(C3CCCCS3)=O)C2)CC1 c1(SC)cc(C(=O)NCC2CCCC2)c(C)o1.C12(C=O)CC(C1)C(C)O2 C1(CC(N2CCN(C)C(=O)C2)=O)C2CCC1CN(C(c1ncccn1)=O)C2 C(CN=c1cccc(S(=O)(=O)NCCC2CC2)[nH]1)c1c(C)[nH]c2c(C)cccc21 c1(C(N2CC(C)(NC(=O)Cc3cnc[nH]3)C2)=O)cnccc1Cl C1(CC(=O)NC(COC)COC)CCC1O.C(C1(C)COC1)=CC(=O)N c1ccc(P(C)(C)=O)o1.c1(OCC)ccccc1C(N1CCC(C(=O)N)C1)=O C1(=CC(=O)N(CCC)C)CCOc2ccccc21.C1(C#N)(C(=O)N)CC2CC2C1 c1(OC)ccc(C)c(C(=O)NC2CC2C(=O)Nc2cc(F)ccc2OC)c1 C1(C(=O)NCC2CC(C)N(C(c3ncccc3N)=O)C2)CCC(=C(F)F)CC1 C#Cc1cc(C(=O)NC)cc(F)c1.C1(C)CCN(C(=O)C(O)Cn2cncn2)C1 C#CCC(C)(C(=O)N1CCCC1CCC)NC(C1CNC(=O)N1)=O C1(SCCC2C(C(F)(F)F)C2)C(F)(F)C12CCC2 C1(NC(C(=O)NCCNC(C)(C)C)=O)CCNC2(CCC2)C1 c1(C(N(CC(CC)NC(=O)Cc2ccc(Cl)cc2)CC)=O)cc(C)[nH]c1C O(C1CC(C)(C)Oc2ccccc21)C(C(C)N(C)C(=O)OC(C)(C)C)=O N1(C(C(=O)NC(CC)C)C(C)=Cc2ccc(Br)s2)CC2(CCOC(=O)N2)C1 Cc1cccnc1C(=O)NC(CCC1CC1)C(=O)NCCN1CCC(C)(C)C1 C(=O)(C1=CCC(F)(F)CC1)N1CC(N(C(=O)Cc2ccn(C3CCCC3)n2)C)C1 C1(NC(C)=O)CCC(C(=O)NC(C)C)CC1.c1(C(C=O)=O)ccc(Cl)s1.N c1(NC(CNC(CC)=O)(C)C)ncnc2[nH]c(C)cc12 C1CC2(CCC2)CN1C(=O)Cc1cn2ccccc2n1.Cc1cocc1C(=O)NC c1(OC)ccc(C(N2CC3CC(NC(c4nc(Cl)cs4)=O)C3C2)=O)cc1C c1(C(N(CCN(C(C(F)=C(C)C)=O)C)CC)=O)coc(-c2ccccc2)c1 N1(C(C(C)CO)=O)CCCC(C)(NC(c2ccnc(OCCO)c2)=O)C1 N1(C(COC(CC)C)=O)CC2CCC(NC(=O)C(CO)c3ccccc3)CC2C1 c1(C(c2nnnn2CCOC)NC(CC)(C)CC)cn(CCO)nc1C.C1CC1 c1(C(=O)NC2CN(C(CNC(=O)NC)=O)CC2SC)ccc(F)c(C)c1C C1(CNC(=O)NC(CNC)C)CCN(CCOC)C1 C(=O)(C(CC(C)C)NC(c1cnc(C(C)C)o1)=O)N(C(C#C)C1CCC1)C C(C(CNC(=O)C(C)NC=O)CO)NC(C(C)=CC)=O.c1ccccc1 C#CCC(O)C(=O)NCC1C=CCN1C(=O)Cc1ccccc1C Cc1ccc(C(=O)NC2CC2CNC(=O)CC2COCCO2)cc1 N1(C(CN2C(C)CC2)=O)CCC(NC(C2CC2Br)=O)CC1 CC(C)C(CC(=O)NC1CCN(C(c2sccc2C2CC2)=O)CC1(C)C)C(C)C C(=O)(CC(C)C(=O)N1CCN(C(c2cc(CO)[nH]n2)=O)CC1CCO)OCC c1(OC)cc(F)c(C(N2CCC2C)=O)cc1N.c1(CC(=O)N)cc(F)ccc1C N1(C(c2cc(C)sc2)=O)CC2CCC2(NC(c2ncc(Cl)cc2F)=O)C1 C1(C(=O)NC(C)CC(C)NC(c2coc(Br)c2)=O)(COC)CCCCC1 CCC(CNC(=O)C)OC.c1cc(C)cs1.C1(C=O)CCCC1.C(=O)(C)N CCC(C)C(C)C(=O)N(CCCNC(c1n[nH]c(C)n1)=O)C1CC1 N1(C(Cc2nc(NC=O)sc2)=O)CC2CC1CCC2NC(c1cnoc1)=O N1(C(C2COCCN(C(CCC)C)C2)=O)CC2COCC(C1)N(C)C2=O c1(C(N2C3CC(NC(C(C)CN4CCCCC4)=O)(C3)C2)=O)cc(Cl)ccc1N N1(C(C(CN(CC)CC)F)=O)CCCN(C(c2onc(Br)c2C)=O)CC1 CC(C)CC(C)C(=O)NC(C)CC1CN(C(c2cnn(C)c(=O)c2)=O)C1 C1(NC(c2cc(Cl)nnc2Cl)=O)CC2CC(C1)N(C(c1cc(C(F)F)cs1)=O)C2 c1(NC(CN(C(C(C)N(C)C)=O)C)=O)cn(C)nc1C#N C1(C(=O)NCCC2(OC)CN(C(c3coc(C)n3)=O)C2)CCOC(C)(C)C1 N1(C(C2(N(C)C)CCCCC2)=O)CCCC(CO)C1.C1(C=O)CC1C(F)(F)F.N CC1COCC(CNC(=O)CC(C)NC(C2COCC(C)O2)=O)O1 N1(C(C2OCCN(C(C)C)C2)=O)CC2CCN(C(=O)C(C)(Cl)Cl)CCC2C1 CC1CC(C(N2CCOC(C(N3CC[Si](C)(C)C3)=O)CC2)=O)CC(=O)N1 CCC(C)C(O)C(=O)NCCNC(C1CN(C(=O)CS)C1)=O.c1cscn1 CC1(C)CCCC(C(=O)NCC2CCC(NC(c3cc4c[nH]nc4s3)=O)CC2)O1 C1(CC(=O)NCC(CC=C)NC(=O)CC(C)C)(CN(C)C)CCCCC1.O C1(C(N)=O)C2CCN(C(CCc3ccc(Br)cc3)C(=O)NCC3CC3)CC12 c1(C(=O)NCC2(C)CCN(C(c3ccc(CCC)[nH]3)=O)C2)cnn(C)c1C#N c1(C(=O)Nc2c(C)cc(OC(F)F)cc2C)cc2ccnc(N(C)C)c2[nH]1 Cc1ccc(C(N2CCC(CC(=O)N(C)C)C2)=O)cc1.N12CCC(C1)CC2 C1(c2cn(Cc3nc(C)sc3)nn2)CN(C(=O)CCSc2ccccn2)CC1O N1(C(=O)CSc2ccccc2)CC2CC2(C(=O)NCC2(CO)CCCC2)C1 C1(NC(C2CCCS2(=O)=O)=O)CCN(C(c2cnc(C(F)(F)F)s2)=O)C1.C c1(C(=O)NC2C(C)N(C(=O)Cc3cncs3)CCC2)cncc2c[nH]nc12 N1(C(c2cnc(OC)s2)=O)CC2CCN(C(=O)C(C)(C)C#N)CC(C2)C1 C1(CNC(C2CCOC2)=O)CN(C(=O)CCc2cscn2)CC1O c1(C(C(=O)NCCOC)NC)ccccc1.c1ccc(C)s1.CC(F)(F)F.O N1(C(C(=O)Nc2cccc(OC)c2)C=Cc2ccco2)CCOC2CCCC12 c1(C(N2CCC(N(C(CC3ON=C(C)C3)=O)CCO)CC2)=O)ccc(C)c(O)n1 N1(C(COCCC#C)=O)CCc2ccccc2C1CNC(C1CC(OC)C1)=O C1(CNC(=O)CC2COCCOC2)CCCCCN1C(c1ccc(CO)cn1)=O c1(C(=O)OCC)nn(C)c(Oc2ccc(C(C)(F)F)cn2)c1Br C1(O)(c2nnc(N(C)Cc3nnc4n3CCCCC4)n2C)Cc2ccccc2C1 C1(CCNC(C(C)=C(CC)C)=O)CCN(C(=O)CC2C=CCC2)C1 C12(NC(c3ccc(CNC(c4cncs4)=O)o3)=O)CCCCC1OCC2 O(NC(=O)C1=NOC(CNC(=O)C2=C(C#N)CCC2)C1)CCCOC c1(SCC(=O)NC2CCN(C(CN3C(C)CCC3)=O)C2)ncnc2[nH]cnc12 c1(COC)cc[nH]c1C(=O)NCC1CCC1NC(c1cc(Br)no1)=O C(=O)(C1=COCCC1)N1C(C)CC(CC(=O)NCCN2CCCC(C)C2)C1 c1(C(=O)OC)cc(C(=O)NC2CCCCC2)ccc1C.C(=O)(CSC(C)=O)N c1(OC)ccc(CC(=O)NCCC(O)CNC(=O)C=Cc2cccnc2)cc1Cl c1(C(CC)C)ccc(C(=O)N(CCCOCCNC(=O)C2=NOCC2)C)cc1 C(=O)(CCC(=O)NN(C)C)NC1(C(N(CCC#C)C)=O)CSC1 CC(C)C(O)C(C)C(=O)NCC(CC(C)C)C(=O)NCc1ccccc1Cl N1(C(=O)OC)CCN2CC1Cn1c2nnn1.C1(C(F)(F)F)(OC)CCC(O)CC1 CC(C)(C(=O)N1CC(NC(c2cn(C3CC3)nn2)=O)C2(CC2)C1)C1=CCSCC1 C1(NC(CCN(C(=O)C(O)CC2CCCC2)CC=C)=O)CCCC1CC c1(CN2CCC(NC(C3CC(=O)NC3)=O)C2)ccc2cc(F)ccc2n1 c1(C=O)c(C)nn2ccccc12.C(=O)(C(C)S(=O)(=O)CCC)N(CCC)CC.N N1(C(Cc2c(C)nccc2)=O)CCC2(CCN(C(=O)Cn3cnccc3=O)C2)C1 C1(C=O)C2CCCCCC12.c1(CC)ccc(C(C)C(=O)N(CC)C(C)C)cc1.N Cn1nc(C(=O)NCC2(Nc3ncccn3)CCCCC2)cc1F Cn1ccc(C(=O)NCCOCCC)c1C(F)(F)F.C1(C=O)CCCO1.N C(=O)(C1=CC2C=CC1C2)NC(C1(O)CCN(C(=O)CC2CCCSC2)C1)C c1(C(C(=O)Nc2ccc(C3(C(=O)O)CCC3)cc2)O)cccc(Cl)c1Cl C1(N(C)C(C2CC2C(F)(F)F)=O)CCN(C(c2cnc(O)o2)=O)CC1 N1(C(C(CC)=CC)=O)CCC(C)(NC(c2ccnc(C3CC3)n2)=O)C1 C1(CNC(CC2(C)CC2)=O)(CO)CCN(C(c2cnc(O)o2)=O)C1 C=C1CCN(C(=O)C=CCCC)C(C(N2CCN(CCOC)CC2)=O)C1 Cc1cc(C(=O)NCCOCCn2cc(C(C)(C)O)nn2)c(-n2cccc2)s1 c1(CC(=O)NC(CCC)C(=O)NC(Cc2cnc[nH]2)CO)ccc2c(c1)CCC2 C1(C(=O)NCC23C(CN(C(C(CCCC)O)=O)C2)C3)(CC)CC2CCC1CC2 C1(C)(CC(N2C3CN(C(C)=O)C(C3)CC2)=O)Oc2ccccc2O1 c1(C(N2CC(C(C)NC(=O)C(C)(C)C3CCCC3)C2)=O)[nH]nc2ncccc12 Cc1cccc(COC(=O)CCc2cccc(N)n2)c1Cl N1(C(C(C)=CC)=O)CCN(C(c2ccc(C#N)cn2)=O)C(c2ccccn2)C1 c1(C(N2CCC(O)(CN(C(CC(C)OC)=O)C)CC2)=O)cc(C)nc(C)c1O C1(NC(CCN(C(=O)CC2COCC2O)C(C)C)=O)CCc2n[nH]cc2C1 Cc1nc2ccc(C(=O)NCCC3CCC(NC(c4ccncc4)=O)C3)cc2s1 C1(NC(CC2(COC)CCCC2)=O)CCC(C)C1.C1(C)(C=O)CCCCC1.C N1(C(C(CC)F)=O)CCN(C(=O)Cc2ccccc2CC#N)C(C2CC2)C1 c1(C(CN2CCN(CC(O)COc3ccccc3Cl)CC2)=O)ccc(Br)c(Cl)c1 Cc1onc(CC(N2CCC(NC(c3ccsc3C)=O)CC2C)=O)c1C#N c1(OC)cccc(C(C)(C)C(=O)N2CCC(SCCCC(C)(F)F)C2)c1 Cc1nc(CCC(N2CCCC(CNC(=O)CC3CCCC3(F)F)C2)=O)oc1C C(=O)(C(O)(C(F)(F)F)c1cn[nH]c1)NC1CC(NC(=O)CCc2ncc[nH]2)C1 N1(C(c2c(OCC)cccc2)=O)CCC(NC(C2CC3CCC2O3)=O)CC(O)C1 N1(C(C2(C)CC2)=O)CCC(C)(C)C1C(=O)NCc1cc(O)ns1 c1(CC)ccc(Br)cc1C(N1CCC(C)(NC(C2CC(F)C2)=O)C1)=O c1(C(CC)C)nnc(N2CCC(CN3CCCCC3C)CC2)n1C C(C1CN(C(=O)C(C(=O)OC)OC)Cc2ccccc21)NC(COCCOC)=O Cc1[nH]c2ccccc2c1C(=O)N.C(=O)(C(C)S(N)(=O)=O)N1CCCC1C1CC1 c1(CN2C(C(=O)Nc3ncccc3F)CC(C)C2)ccc2[nH]ccc2c1 c1(C(C)NC2C(CCC(C)C)CCC2)cccc2cnccc12 C(CC(=O)N(C)Cc1nc[nH]n1)N(C(=O)Cc1csnn1)C c1(C(=O)NC2CN(C(Cn3nc(C)c(Cl)c3)=O)C(C)C2)cccc2cnccc12 c1(CCC(C)NC(c2csc(Br)n2)c2nnnn2C2CC2)ccccc1 c1(C=O)cccc(S(=O)(=O)N2CCC2)c1.O=C(CSC(F)F)NC1CC1.C c1(C(C)NC(C2N(C(C3C(CCOC)C3)=O)C(C)C2)=O)nn(C)cc1O c1(N2CCN(C(c3cc(CSC)c(C)s3)=O)CC2)ccc(C#N)cn1 N1(C(C(C)OCCOC)=O)CC(C)CCC1C(=O)NCC(C1CCCCC1)O N1(C(c2nccc(C)c2)=O)CCCC(CCNC(c2ccc(Cl)c(Cl)c2)=O)CC1 c1(CC)ccc(-c2cn(C3COCC3NC(=O)COc3cnn(C)c3)nn2)nc1 c1(C(N2CCN(C(C(C)C3CCOC3)=O)C(CCO)C2)=O)nccc2[nH]ccc12 CCCC(CNC(=O)C(C)CC(N)=O)C(=O)N1CC(CC(F)(F)F)C1 c1(CNC(c2cc(C(=O)C(F)(F)F)c[nH]2)=O)ccc(C(F)(F)F)o1 c1(C(=O)NCCN(C(c2noc(CC)c2C)=O)CC)cn2cnnc2cn1 Cc1coc2ccc(NC(c3cc(Cl)cs3)c3nnnn3C(C)C)cc12 N1(C(CNC(c2ccccc2)=O)=O)CC2CN(C(c3ccno3)=O)CC(C1)O2 c1(C(=O)NCC2C(NC(C(CCC)C#N)=O)C2)cc(C)nc2onc(C)c12 c1(C(=O)OC)cc(NC(C2CCCN2C(c2cccs2)=O)=O)on1 C12(NC(C(C(CC)C)OC)=O)CCCC1N(c1nc(C)cc(C)n1)CC2 C(=O)(CC(C)CC(=O)OC)N1CC(NC(C2CN(CCC)C2)=O)C(C)C1 C1(C(=O)NCCNC(C(C)n2ccnc2)=O)CCCN(C(=O)C2=CCSC2)C1 N1(C(C2C(C(=O)OC)CCC2)=O)CCC(C)(NC(C2CC2OC)=O)C1 CC1(CNC(=O)NCCNc2ccccc2)CCNC1 C(C)(CCCC(=O)N(C)Cc1n[nH]c(C)n1)NC(c1n(COC)ncc1)=O c1(OC)ccccc1CC.C(=O)C(O)CN(C)C.C(=O)C(C)N1CC(C)C1.N N1(C(c2nc(CC)oc2)=O)CCC(NC(c2snnc2C)=O)CC(C)(C)C1 C1(NC(CN(CCC)C)=O)CCC(C)CC1.c1(C(=O)N)ccc(-c2cccs2)s1 C1(NC(=O)CCCCC2CC2)C2CC1CN(C(=O)COCC1CCCCO1)C2 C12(CC(=O)N(C)Cc3ccco3)CCC1CN(C(=O)Cc1cc[nH]n1)C2 N1(C(c2cc(OCC)n[nH]2)=O)CC(O)CCC1C(=O)NCCN1CCCOCC1 N1(C(C(C)N(C)C)=O)CCC(C(=O)NCc2cccs2)C(C)(C)C1 c1(C(N2CCCC(C#N)C2)C(=O)NCCCSC)cccc(Br)c1Cl c1(CN2C(C(=O)NC(C(=O)OCC)C(C)O)CNCC2)ccc(C#N)cc1Cl N1(C(C(N2CC(N)C(F)(F)CC2)=O)=O)CCN(S(=O)(=O)N2CCOCC2)CC1 S(=O)(=O)(c1cccc(Br)c1)NCC(C(F)(F)F)OC.c1c(C)nn(C)c1C.N C1(NC(c2cnn(CC)c2Cl)=O)CN(C(C2(C)CC3CC3C2)=O)CC1(C)C N1(C(c2ccc(CSCCC)o2)=O)CC(CC)OC(C)C1.C(=O)C.C1CC1 c1(NC(C2C(OC)CCCC2)=O)ccc(OCCC(C)C)c(N)c1 C(=O)(C1=C(C)OCC1)N1C(C=CC(N2CC(O)(CC)C2)=O)CCC1 CCCCC(O)C(C)C(=O)NCCCCC(C)NC(=O)C(N1CCCCC1)C N1(C(CN(CCC)C(C2(CC)CCC2)=O)=O)CCC(OC2CC2)CC1 C1(NC(C2C(CC)C2)=O)CCN(C(=O)CCCN=[N+]=[N-])CC12CCC2 c1(C(=O)NCC(C)NC(=O)C(O)Cc2ccccc2)cnn(C)c1C#N C(C(CC(=O)NC(CC(N)=O)C1CC1)NC(=O)CCC1(C)N=N1)OC CCCCC(C(=O)NCC1CC1NC(=O)CCOc1ccccc1)C(C)C Oc1ncccc1C(c1nnnn1CSc1ccccc1)Nc1ccc(I)cc1 N1(C(c2onc(CC)c2C)=O)CC(NC(C2CCOC2C)=O)C2(CC2)C1 c1(CC)cc[nH]c1C=O.C1(C(N(CCC)C(C)C)=O)CCCN1C(N)=O.N c1(CCC)ccc(C(=O)CCC(=O)ON(C)Cc2cn(CC)nc2C)cc1 N1(C(c2ccn(C)n2)=O)CC2CCOC2(CNC(=O)C(c2ccccc2)O)C1 C12(C=O)CCCCC1C2.c1(C(=O)NC2(CC)CC2)ocnc1-c1ccccc1.N c1(COC(C2C(CC(=O)OC)CC2)=O)cc(C)ncn1 c1(C(c2n(CCOC)nnn2)NCc2cccc(O)c2C)cc(C)c(F)cc1Br CCC(CC(=O)NCC(=O)NC)N(C(C1CCCCC1)=O)C c1(OC)c(C)cnc(CN(C(=O)Cn2cc(CCC3CCCCC3)nn2)C)c1C C(C(COC)CC(=O)N1CCCC(N(CCO)C(C2CCC3(CC3)C2)=O)C1)OC c1(OCC)ccc2c(c1)CN(C(=NCCOC)NCc1ccccc1)CC2 C(c1cnc(C)nc1O)=CC=O.C(C)(CO)(C(=O)N1CCC(C)(CC)C1)OC.N O(NC(=O)CCCN(C)C(C1(C#N)CCCOC1)=O)CC(C(C)C)O c1(CC(=O)NC2C(C(=O)Nc3n(CC)ncc3)C2)ccccc1C.C(C)C c1(CC(=O)NCC2(C)CC(NC(c3nn[nH]c3Cl)=O)C2)cc(F)cc(Cl)c1 C1(NC(COC)=O)CC2CCC(C1)N2C(C1CC1C(N)=O)=O C(=O)(C1CCOc2ccccc21)N(C(C)C)CCN(c1cnc(F)cn1)C c1(COC)ccccc1C(=O)NC1COCC1.c1(C=O)ncoc1-c1ccon1 Cc1nsc(C(N2CCOCC2CC(=O)NC2C=CCCC2)=O)c1N c1(C(=O)NCCCC)ccc(P(C)(C)=O)nc1.c1(C=O)cnc(C(C)=O)s1.N c1(N(C(CCNC(c2c(C)cno2)=O)C)C)nc2cccc(C)c2s1 c1(N2CC(C)CC(OC)C2)nc(N(C)Cc2cnccn2)c2ccsc2n1 C1(C(N(C(C(N)=O)C2CC2)C)=O)C=CCN(C(=O)CCCn2cccn2)C1 Cc1nn(C)cc1C(N1CC(NC(c2ccnc(OC(C)C)c2)=O)C(C)C1)=O C(=O)(C(F)(F)C(O)C(C)C)N.C12(C=O)CCC(C1)OC2.C(C)(C)(C)OC CC1CCC=C1C(=O)NCCCC1CCN(C(=O)CC2C=NN(C)C2=O)CC1 CC(C)C(C)C(CNC(=O)CCc1cc(Cl)no1)NC(c1ccnc(F)c1N)=O C1(OCC)COCCC1N(C(=O)NC1CC(C)OC1C)Cc1ccc(F)cc1 CC1CCCCC1(C)C(=O)NCCNC(c1cccc(Oc2ccccc2)n1)=O c1(-c2cccc(CC(=O)Nc3cc(C)on3)n2)ccc(CO)cc1F c1(NCC2CN(C(=O)C=CI)CC2C(F)(F)F)ccc(Br)cc1[N+](=O)[O-] S(=O)(=O)(c1cccnc1)NCC(N1CCC(CNC(CC)=O)C1(C)C)=O N1C(=NCCC2CCCO2)NCC1=O.c1(C(N2CCCC2=O)C)ccc(F)cc1 N1(C(c2cn(CCN(C)C)nn2)=O)CCN(C)C(C)C1.C(=O)(CCC(C)(F)F)N N1(C(c2ccc(C(C)(C)C)[nH]2)=O)CCCC2(CC(NC(=O)C=CCO)CO2)C1 c1(CNC)cc(C)[nH]c(=NCC(C)NC(c2cnc(F)c(Cl)c2)=O)n1.C1CC1 CCCCC(=O)C(=O)NC(CNC(c1cc(C)sc1C)=O)CO C(CCS(=O)(=O)c1ccc(F)cc1)Sc1nnc(CC)n1C C(=O)C(C)C1CCC1.C(=O)C(C)C1CC1.C1(C(=O)OCC)(CC)CC1 C1(CC)CN(C(C2(n3cccn3)CC2)=O)CCC1NC(=O)C.CC.CCO.O C1(COC)CCN(C(N2CCC(NC(=O)NCC(C)C)C2)=O)CC1 Cc1ccc(Br)c(C(=O)NCC23CC(C2)C3)n1.C1(C(=O)N)CCN(C)CC1 CN1C(=O)COC(C(N2CCC2)=O)C1c1cccs1.C1(C(F)(F)F)(C=O)CC1 c1(C(N2C(CNC(c3snnc3C3CC3)=O)CCCC2)=O)ccn2cnnc2c1 N1(C(CN(CC)CC)=O)CCOC2CCN(C(=O)C(COC)OC)CC12 C1(CC(=O)NCc2c(C(=O)NCC(COC)C)c[nH]n2)CCCC(=O)C1 c1(NC(C2N(C(C3CCC(CC)O3)=O)CCC2)=O)ccc(C)c(F)c1F c1(CC(=O)N(C(CCNC(C2CCN(CC)C2)=O)C)C)ccccc1OC C1(C)(C(N2CCN(C(COCC)=O)C(CC)C2)=O)CC2(C1)CC(F)(F)C2 c1(C(N(CC(C)NC(C(C)=C(CC)C)=O)CC)=O)cnc2sc(C)cn12 N1(C(c2c(CC)[nH]cc2)=O)CCCN(C(=O)Cc2c[nH]c3ccccc23)CC1C N1(C(C2(OC)CCSC2)=O)CC=CC(C(=O)NC(C)C(C)SC)C1 N1(C(C(CC)SC)=O)CCC(C)C(N(C(=O)CCCNC(=O)OC(C)C)C)C1 C(C(C(=O)NCC(C1CCCCC1)NC(c1ccoc1Br)=O)OC)OC Cc1cc2occ(C(N3CC(CNC(c4ccc(F)o4)=O)CC3C)=O)c2cc1C c1(C(=O)NCC(CC2CCCO2)OC)ccc2c(c1)nc(S)n2C c1(C(=O)N)cc(C)c(Cl)cc1C.c1(OCC)cccc(CC(=O)NC2CC2)c1 C(CCCCCCC(=O)N1CCOCC1)NC(C1C(NC(=O)OC(C)(C)C)C1)=O C1(C(N2CCC2)=O)CC(=O)N(CC(F)(F)F)C1.O=C(CC(O)C1CCCC1)N.C C1(CN(C)CCn2cccn2)CCCN(C(=O)CC2CCOC2)C1 C1(CC)CCCC(CNC(c2ccn(CCNC(=O)C3=CCCC3)c2)=O)C1 C12(C(=O)NC(c3cccnc3O)C)CCCC1CCN2C(=O)C=CC1CC1 O=C(C1=CC2CCC1C2)NC1CCC(NC(c2c[nH]cc(Br)c2=O)=O)C1 N1(C(C2N(C(c3cncc(OC)c3)=O)C3C(C2)C3)=O)CCCC2(CCO2)C1 CCCCCC(O)C(=O)OCc1cc2ccsc2n1C C1(C(N2CCN(C(C(C)OCCC(C)C)=O)CC2)=O)CC2(C1)CC(C)(C)C2.C N1(C(c2c(OC)n[nH]c2)=O)CCC(C)C(CC(=O)N(C2CCC2C)C)C1 C(=O)(C1CCCc2n[nH]cc21)NCCC(C)NC(=O)CNC(=O)C1CC1 C(=O)(C(CCCO)c1ccccc1)N(C)CNC1(O)CN(C=O)C1.C(C)(C)C CCC(C)C(O)C(C)C(=O)NC(C)(C)CC(=O)NCC1CCCCO1 CN1C(=O)CSC1=CC(=O)N1CC(NC(=O)Cc2csc(Cl)c2)C2(CCC2)C1 C12(CNC(C3CCC4CC4CC3)=O)CCCCC1N(C(=O)Cc1cnsc1)CC2 N1(S(CCN(C)C)(=O)=O)CCC2CN(C(=O)OC(C)(C)C)CCC2C1 C1(C(=O)NC2CCC(C(N3CC(COC)C3(C)C)=O)C2)CCCCCN1C C(=O)(N=c1ccn(C2CCC2)[nH]1)C1OCCN(C(C(C(=O)OC)OC)=O)C1 CCCC(CC)CCC(=O)N1CCC(CCC(=O)NCC(O)CNC(=O)OC)C1 c1(CC)cnn(C)c1C(C(=O)NC1CCCC1)N(C)CC1C(C)(C)C1(C)C C1(CC)CCCCCCN1C(=O)C(c1ccccc1)NC(C1CCCN1C=O)=O C1CC2CCCC2N1C(C1CCS1(=O)=O)=O.c1(COC)nn(C)cc1C=O.N c1(NC(CC)CNC(c2cc(Cl)c[nH]2)=O)ncc2scc(Br)c2n1 N1(C(c2cn(CCC)nn2)=O)CCCC(C2(NC(c3coc(CC)n3)=O)CC2)C1 C1(C(=O)NC(C(=O)NC(c2nccs2)CC)CO)CC2(CCO1)CC2 CC(C)C1=NOC(C)(C(=O)N(C)CC2CCCCN2C(=O)CCC=CBr)C1 C1(C(=O)NCc2c(C(N(C)CC3(C)CC3)=O)[nH]cc2)CCCC(=O)N1C CCCCCCCCS(=O)(=O)N1CCOC(CC(=O)Nc2c(C)cccc2O)C1 c1(NC(C2CC(F)CN(C(C3(F)CCCCC3(F)F)=O)C2)=O)ccc2[nH]nnc2c1 N1(C(c2ncn(C(C)C)n2)=O)CCC(CF)(NC(=O)CCCn2ccnn2)C1 N1(C(C2C(C)CCO2)=O)CC2CCC1CN(C(c1cccc3ncnn13)=O)C2 Cc1ccnc(NC2CC2CNC(c2cnn(Cc3ccccc3)c2)=O)n1 CCC(CC)CCCC(=O)N1CCC(O)(CNC(c2ccnc3[nH]ncc23)=O)C1 C(=O)(C(C)(C)C(=O)N(CC)C1CC1)NC.c1(C=O)ccccn1.CC(F)F N1(C(c2c(C)nco2)=O)CCC2(CC1)CC(NC(=O)CCC#N)CCO2 CC(C)CC(C(=O)NCCC1CCCCC1)NC(C1CC(C)(C)C1)=O C(=O)(CC(C)(C)C(C)(F)F)N.N1(C(Cc2scc(C)n2)=O)CCCC(C)(C)C1C c1(C(N(CCOCCN(C(C(CCC)C)=O)C)C)=O)cccn2[nH]c(=N)nc12 CC1CN(C(c2coc(C(F)F)n2)=O)CC1NC(c1cnc(C(=O)O)[nH]1)=O C1CC(C=O)CCO1.CCCN(C(=O)C=CC)CCN(C)C.CCO.CC C12(C(=O)NCc3cc(C)cc(C)n3)CCCC1CCN2C(=O)Cc1ccnn1C C(=O)(CC(C(F)(F)F)NC(C1(C)CCC1)=O)N1CC(CC(C)C)OCC1 C12(OC)CCCC1(C(=O)NCC(C)N(C)C(c1cc(F)ccc1C)=O)CCO2 C1(C)(NC(C=CCN(C(c2c(CC)occ2)=O)C)=O)CCCC1(C)C CC1(CNC(=O)CCCC2CCC2)CCC(=O)N1.C(=O)(CCC1CCCC1)N C12(NC(CN(C(COC)=O)C)=O)COC(CNC(=O)CCO)(C1)C2 N1(C(C(CC)(C)O)=O)CCC2CCN(C(=O)C3=NN(C4CC4)C(=O)CC3)C2C1 CC(CCCCNC(C1CCCN1C1CCOCC1)=O)NC(c1ccon1)=O c1(N(C)C)ncc(C(=O)NC2CC(CO)N(C(=O)CC3(O)CCCOC3)C2)cn1 c1(C(C)OC(CC(c2cnccn2)=O)=O)cccc(C(F)(F)F)c1 N1(C(C(C)SC)=O)CCC(C)(C)C(C(=O)NCCC(O)CO)C1 Cc1c(C(=O)NCC2CC2CNC(=O)CCC(F)(F)F)nn(C)c1Br Cc1cc(C#N)ccc1C(=O)NCC(C)C(=O)NCC1CCCCS1 CC1CC(NC(C2(C)COC(=O)N2)=O)CN(C(=O)CCCNC(N)=O)C1 c1(C(=O)NCC(CO)NC(Cc2c(C)n[nH]c2C)=O)cc2n(c(=O)c1)CCS2 C(=O)(C1=CC2CCCCC12)N1CCN(C(C=C(COC)C)=O)C(c2cccnc2)C1 C1(C(=O)NC2C(CNC(CCN(CCCCC)C)=O)COC2)C2CCC1CC2 N1(C(c2nc(C#C)sc2)=O)CCOCC(NC(C2CCCN2C)=O)C1 c1(-c2c(C(=O)Nc3c(OCC)nccc3)csc2)c(F)ccc(OC)c1F CC1C(NC(c2cnc[nH]2)=O)CCCN1C(=O)CCc1cnn(C)n1 c1(C(=O)NCCN2CCN(C(CCC3CC(OC)C3)=O)CC2)ccc(C)nc1C C1(C(CNC(c2ccc(Cl)s2)=O)F)CCN(C(c2cnc[nH]2)=O)CC1 N1(C(c2ccc3c(c2)CCCC3)C(=O)NC)CCC2(CC1)COC(=O)N2C Cc1ccc(C(=O)NC(C2CCCN(C(c3nnc(O)nc3O)=O)C2)C)c(C)n1 N#Cc1ccc(CC(=O)NC2CCCCN(C(=O)Cc3ccnc(Br)c3)C2)cn1 c1(OC)cc(C(=O)NC2CC2)c(N)c(C)c1.c1(C(CC(=O)N)C)ccccc1C C1(C(=O)NC2CC(C)(NC(c3ccc(OC)cn3)=O)C2)CCC(C)NC1=O Cc1nc(C(C)(C)C)sc1C(=O)N.C1CCCN(C(c2ccnn2C(C)C)=O)C1 C=CCC(CC(C)C)C(=O)NCCCC(C)NC(=O)CN1CC2C=CC1C2 c1(NC(=O)NCc2c(CC)nn(C)c2)c(C#N)cnn1-c1ccccn1 N1(c2n(CC)c(-c3cc(-c4ccncc4)[nH]n3)nn2)CCC(OC)C(C)C1 C1(N(C)C(c2coc(Cl)n2)=O)CCCC(NC(c2coc(C(F)(F)F)c2)=O)C1 CC(C)(CC(=O)N1CC(NC(C2CC(C)(F)C2)=O)C2CCCCC12)CC(F)(F)F C1(c2ccccc2)(NC(=O)C2CC2)CCN(C(C2CC(N3CCOCC3)C2)=O)C1 N1(C(c2c(C)csn2)=O)CC2(CCN(C(=O)CC(C)O)CC2)CC1C Cc1ccc(C(N2CCC(NC(c3cncc4n[nH]cc34)=O)CC2)=O)c(F)c1F CC1CCN(C(=O)C=Cc2cnccn2)CC1NC(=O)CC1CC2C=CC1CC2 N1(C(C(CC)C(C)C)=O)CCC2OCCN(C(c3ccc(CC4CC4)s3)=O)C2C1 c1(OCC)cccc(C(N2CC(C)C(O)C2)=O)c1N.c1(C=O)sc(F)cc1C.N c1(C(=O)NCCC2(O)CCN(C(C(CC(=C)C)C)=O)C2)c(OC)ccc(Cl)c1Cl c1(CN(CCC)C(C2CC23CCCCC3)=O)cc(C)cc(Br)c1OCC c1(C(=O)NC2(CCNC(C(CC)COC)=O)CCC2)ccccc1C#N C1(CC)CN(C(C2CCCCC2)C(=O)NC(C)C(=O)OC)CC(C)S1=O c1(C(N(CC(C)N(C(C2CCCN(CC)C2)=O)C)C)=O)cnn2cccc2c1 O=CN1CCCC1C(=O)NCCCNC(C1(C2CCCCO2)CCC1)=O Cc1cc(NC(C2CC(C)CN(C(=O)CC(C)(F)F)C2)=O)cc(C#N)c1 CC1SCCCC1C(N1CCN(C2CCCOC2)CC1)=O C1(C(N(CC(CO)CO)C)=O)CCCC1P(C)(C)=O.C(=O)(CC(C)C=O)OC.N CC1CCC(O)(C(=O)N)CC1.C1(C)CN(C(C2CC(=O)NC(=O)N2)=O)CC1C.C CC1(C(=O)NC(CNC(c2c[nH]c3ncccc23)=O)CO)CC2CCC(C1)S2 C=C(C)C(C)(C)C(=O)NC1CCCCN1CC(=O)NC(=O)NCC Cc1cnc2ccccc2c1C(=O)NCC1(C)CCCN1C(C1CC(Cl)(Cl)C1)=O C1(C(=O)NCC2CCN2C(c2ccc(O)nc2)=O)CCS(=O)(=O)C12CCC2 Cc1cc2c(cc1C(N1CCC3(CC1)CN(C(=O)C(C)CF)C3)=O)OCO2 C1(CNC(C(C)N(C)C)=O)CCC12CCN(C(=O)CC(C)(C)C(F)F)CC2 N1(C(C2CCC2)=O)CCN(C(c2ccc(I)c(Br)c2)=O)C(Cc2ccccc2)C1 N1(C(C2CN(C(c3c(OC)nccc3)=O)CC2C)=O)CCCCC(C)C1 C1(CC(=O)NC2(C(N)=O)CC=CC2)CCCN(C(c2ccccc2)=O)CC1 C1(NC(C2(CC)CC2)=O)CC2CCC(C1)N2C(=O)CC1CCC(O)C1 c1(C(N2C(C)CCC(NC(C3(c4ccno4)CC3)=O)C2)=O)cc2ccncc2s1 Cc1n[nH]cc1C(N1CC(c2nc(C(F)F)no2)C1)=O c1(C(=O)NC2CN(C(C(OC)OC)=O)CC2c2nccn2C)ccnn(C)c1=O C#CCC(C)(C)C(=O)NC1COCC1NC(=O)CC1(O)CCOCC1 c1(C(N2CCCC(N(C(=O)C(C)=C3CCCC3)CC)C2)=O)ccc(O)cc1F C(C)(C(C(=O)NC(c1cnn[nH]1)C)NC(C1C2CC3C(C2)C13)=O)OC c1(N2CCC(CCC)C2)ccn2ncc(S(=O)(=O)N3CCC(C(N)=O)CC3)c2n1 C12(C=O)CC(C)(CN1C(C1COCC1C(N)=O)=O)C2.CCCCC(=O)OC.N C1(NC(c2c(C)ocn2)=O)CN(C(=O)C)Cc2ccnn2C1.C(=O)(C(C)(C)C)N N1(C(C(C)n2cnnn2)=O)CC2(C)CC1(C(=O)NC(C1CSC1)C)C2 c1(C(C)NC(=O)NC(C)C(=O)N2CC(F)C2)ccccc1O C1(CC)CN(C(c2cc(C)on2)=O)CCC1NC(=O)COC1(C)CCC1 C(=O)(N1OC2C=CC1CC2)C1C2C(NC(=O)CCC3CCCO3)C3C(C2)C31 c1(C(C(=O)NC)N(C2CCN(CC)C2)CC)ccc(Cl)c(Cl)c1Cl C1(C(=O)Nc2ccco2)CCCN(c2cnccn2)C1 N1(C(C(C2CC2)SC)=O)CCOCC1(C)c1cn(-c2nc(C)c(C)s2)nn1 CC(C)(CCCO)C(=O)NC(C1CCCC1)CNC(c1cccc(N)n1)=O N1(C(CC(COC)(C)O)=O)CCC(NC(=O)Cc2nonc2C)C(CO)CC1 c1(C(N(CCCN(C(C(CC)COC)=O)C)C)=O)cccc2c1OC(C)C(=O)N2 O=C(C1=NOC(CNC(C2CC=CCC2)=O)C1)NCCC12CCCC1C2 N1(C(Cc2nc(C)sc2)=O)CC2CC(O)C1C2NC(C1CC2(CCCCO2)C1)=O Cc1cc(C(=O)NCC2C(C)CCN2C(=O)CCc2cc[nH]n2)c2n[nH]cc2c1 C(CC(C(=O)NCC(c1ccc(F)cc1)NC(=O)CC1CC=CC1)OC)OC C(=O)(C1=CCCOCC1)N(C1CCCC(NC(=O)CC2(C)OCCO2)C1)C c1(C(=O)NCc2c(CCNC(Cc3c(C)ccs3)=O)ocn2)cc(Cl)ccn1 C1(CNC(c2csc(-c3nc[nH]n3)n2)=O)CCCCN(C(c2ccc(Cl)o2)=O)C1 CCC(C#N)(CC)C(=O)NCCC1CCCN(C(=O)CCCCCSC)C1 CCC(C)(C(=O)NC(c1ccc(C)cc1)C)OC.c1cnn(C)c1.C(=O)(C)N Cc1ccc(C(N2CCN(C(=O)CCOC)C(C(C)C)C2)=O)c(N)n1.C1CCC1 C1(CC(=O)NCC2CN(c3nc(C4CCOCC4)ns3)CCO2)CCC(F)(F)C1 C1(NC(c2ccc(CO)nc2)=O)CCN(C(c2ccnc(O)c2F)=O)C12CC2 C1CN(C(c2ccsc2Cl)=O)CC2CC12.c1(NC(=O)NC)ccc(C(=O)N)cc1 C1(NC(CC(CC)C)=O)CCC(C)(NC(c2ccc(F)c(F)c2)=O)CC1 C=CC(C)(CCOC)C(=O)NCC(c1ccccc1)CNC(=O)CC(C)(C)C Cc1cccc(C(N2CCCC(NC(=O)CC3(O)CCOCC3)C2)=O)c1[N+](=O)[O-] c1(CCC(=O)N(CC(CC)NC(=O)C(C)(C)COC(C)C)C)ccccc1C N1(C(C(C)OCCCC)=O)CC(CO)C2(C1)CN(C(=O)C)C2.C(=O)C1CC1 C12(NC(c3nc(Cl)sc3Cl)=O)CCC(CC1NC(C1CCCOCC1)=O)C2 Cc1cnc(O)c(NC(=O)NCCC(N(C)C)C2CC2)c1 CCC(N=c1nc(N2CCn3c(O)nnc3C2)c2ncn(CC)c2[nH]1)C1CCC1 C1(NC(=O)CC2CC2)CN(C(c2n[nH]c(O)n2)=O)CCC1F Cc1nc(C)c(C(N2CCC(C(=O)NCc3csc(C)c3C)C2)=O)s1 c1(CN(C2C3CCC2CNC3)CC(C)NC(=O)CN)c(F)cncc1Br c1(CC)ccc(-c2noc(COC(C3(CC(C)=O)CCC3)=O)n2)cc1 N1(C(C(C(C)C)O)=O)CCCC(NC(C2CC(=O)N(C3CCCC3)C2)=O)CCC1 N1(C(C2(CCCC)CC2)=O)CCCCC1CNC(=O)CC1CCOC1=O C(C(O)CCO)N(C)C(C1CC(N(C(=O)C=CC2CCOC2)C)C1)=O Cc1cc(N2CCCC2C2CCN(C(=O)C(C)(C)NS(C)(=O)=O)C2)ncn1 N1(C(c2ccc(SC)s2)C(=O)Nc2c(CC)cccc2)CCC2CCC(C1)N2C C(=O)(C(C(C)(C)C)NC(N)=O)NCC(=C)CCNC(=O)CC(=O)NC Cc1nn(C)c2ccc(C(=O)NC3CCCCN(C(C4C5COCC45)=O)C3)cc12 Cc1ccc(CCC(=O)NC(C)(C)CNC(=O)CSCC2CCCO2)cn1 c1(OC)cccc(C(C(=O)NC2CCCCC2C)OC)c1.C(=O)C(O)C(C)C.N C1(NC2(C(=O)NCc3occ(C(N)=O)c3)CCCCC2)CC2CCCC2C1 C#CCC1C(=O)NCCCC(=O)NCC(NC(=O)OCC)CC(=O)N1 N1(C(CC2CN(C(=O)NC)C2)=O)CCCC1CNC(C1CCOC1C)=O.C C=C(C)CCCC(=O)NC1CCC(NC(C2CC2[N+](=O)[O-])=O)C1 Cn1ncc(CNC(=O)C(F)CC2CN(C(=O)C3=COCC3)C2)c1O C1(C)(CNC(C(CC)CC)=O)COCCN(C(c2ccc(C)c(O)c2)=O)C1 C1(C(=O)Nc2cncc(Br)c2Cl)CN(Cc2ncccc2Br)CC(F)(F)C1 c1(CN)nnc2n1CCN(C(=O)NC1CCCC(O)C1)C2 C(=O)(C1CCc2ccccc21)NCCC(C(=O)NCC1CN(C)C(=O)C1)O C12(Nc3ncnc(C)c3Br)CCCC1CN(C(=O)C=CC(N)=O)C2 N1(C(C2(c3ccc(Cl)cc3)CCC2)=O)CCOC(C)C1.C1(F)(C(=O)N)CCOC1 C12(CSC)CC(C(=O)N)(CO1)C2.C1CCCC1.C1CCCCO1.C(=O)C.C c1(C(=O)NCC2N(C(CC(CC)C3CC3)=O)CC=C2)cn(C)ccc1=O C1(NC(C)=O)(CF)CCN(C(=O)CN(C)C)C1.C1CCCCC1O Cc1cn2cc(C(N3CC4CC(NC(=O)Cc5ccn(C)n5)CC3C4)=O)sc2n1 C1(NC(N2C(CC(C)C)(CC)CCC2)=O)CCN(C)C(=O)C1 C1(OC)CC(C(N2CCC2C2CCC2)=O)N(C(=O)Cn2ncccc2=O)C1 c1(CN(C(C2C(C)C2)=O)C)ccc(I)cc1 N1(C(c2ccc(C)nn2)=O)CCCC(CNC(=O)Cc2ccc(O)cc2)CC1 Cc1noc(C2CC2CNC(C23CSCC2C3)=O)n1.C1(=O)CCN1C c1(N(C)C)cccc(C(=O)NC2CCC(F)(C)C2)n1.C(=O)CCN1CCCC1.N CCC(C)CC(=O)NCC(C)NC(c1csc(-c2ccccc2Cl)n1)=O C(=O)(C1=C(C)OCCS1(=O)=O)NCC1CN(C(C(CC)NC(N)=O)=O)C1 c1(C(=O)NC(c2ccccc2)CNC(C2C(C)C2C)=O)c[nH]cc(Cl)c1=O C1(NC(Cn2c(C)nnn2)=O)CN(C(C2(CCO)CC2)=O)CC2(CC2)C1 CC1CCCC(C(=O)NCCC2CC(NC(c3cnn(CC(F)F)n3)=O)C2)C1 c1(C(C)NC(=O)C(C)(c2ccccc2)N2CCCC2)cn(C2CC2)nn1 c1(C(=O)NCC)ccco1.C1C(=O)OCCN1C(=O)N(C)C CN1CCN(C(C2C=CCS2)=O)CC1C(N1CC(C(C)(C)O)C1)=O C1(NC(c2c(CNC(C(c3cn(C)nc3)=O)=O)occ2)=O)CC12CCOCC2 C1(NC(=O)CN2C(=O)CNC2=O)CCN(C(=O)CSc2nncs2)CC12CCC2 c1(C(=O)O)ncc(C2CN(C(=O)Nc3ccnn3C3CCC3)C2)s1 C=CC1(c2cn(CC3CCOC3)nn2)COCCN1C(=O)Cc1nc[nH]n1 C(N=c1[nH]cc2ccnc-2[nH]1)C1CCN(C(C2(C(N)=O)CC2)=O)C1 C1(CC)OCCC1C(=O)NCc1cc(C(N2CC(C)(C(N)=O)C2)=O)no1 c1(C(C(=O)NCC(c2ccccc2)NC(N)=O)CO)ccc(F)cc1 C1(C(N2CCC3(CN(C(C4C(CCC)C4)=O)C3)C2)=O)Cn2c(C)nnc2CN1C C#Cc1ccccc1CC(=O)NC12CC(C1)N(C(=O)C(N1CCCCC1=O)C)C2 C1(C(N(C2(CCO)CC2)C)=O)CCCCC1NC(=O)Cc1cncnc1 Cc1csc(C(=O)NCC#CCNC(C2CC3CCC2O3)=O)c1C C(CN=c1nc(C(F)F)[nH]s1)OCCNC(C1CCCC1c1ccccc1)=O c1(C(N(CCC(C(C)C)NC(C(CCC)N(C)C)=O)C)=O)cc(O)nc(O)n1 C=CCCCC(C(=O)NCc1cn(C2CC2)nn1)NC(=O)CN1CCC(C)C1 Cc1cc(C(=O)NCC(C)CNC(=O)C(C)N(C)C)sc1Br N1(C(C(CC(C)C)O)=O)CC(C2CN(C(=O)C(C)NC(c3cnoc3C)=O)C2)C1 C1(NC(c2ccn(C(C)C)n2)=O)CC(CC(=O)NC(CCO)C2CCC2)C1(C)C CCCC(C)(CC)C(=O)N(CCC(C(C)(C)C)NC(=O)CN(C1CCCC1)C)C C1(NC(C(C2CCCC2)OCC)=O)CC2CN(c3ncc(C)cn3)CC2C1 N1(C(=O)NCC)CCC(C=O)CC1.C1(CC=O)CC12CC2.C(C)C1CC1 c1(C(N(C(c2ccc(OC)nn2)C(=O)NCCOC)C)C)ccccc1Br N1(C(CC(c2ccccc2)NC(C)=O)=O)CC2=C(C1)CN(C(C1C(C)C1C)=O)C2 n1(CC=O)ccc([N+](=O)[O-])n1.C(CCC(C)C)NC(C=CC=CCC)=O.N C1(O)(CC(N2CC(COC)C2)=O)CCCCCC1.C(=O)C.CCN(C)C.C C12CCCN(C(c3nccc(C(F)(F)F)n3)=O)C1C2.c1(C(=O)NC)ncccn1 c1(NC(C(N2C(C)CC(NC)C2)=O)=O)ccnc(F)c1Cl C(C(O)C(=O)N1CC(O)(C(C)NC(=O)C(C)Cc2ccncc2)C1)OC N1(C(CC)=O)CC=C(CNC(c2nn(CC(F)(F)F)cc2Cl)=O)CC1 CC(C(=O)NCC1(CNC(=O)CC(C)(C)C)CCC1)C(=O)N1CCOCC1 c1(C(N(C2CCN(C(=O)CNC(C3CCC3)=O)C2)C)=O)ccn2c1CCC2 CC(CCC(C)(C)C)C(=O)NC1CCCCC1Nc1c([N+](=O)[O-])cnn1C c1(C(CC)C)ccc(C(=O)NCC(CO)NC(=O)CC(F)F)c(O)n1 C1(C2CCC(=O)CC2)(NC(N2CC3C(C(N)=O)C3C2)=O)CC1 O=C1CC(C(=O)N2C3CCC2C2CC2(NC(=O)CCC(F)F)C3)c2ccccc21 C1(C(=O)N)CC(C)(C)CCN1C(c1cc(=O)n(C)cn1)=O.n1(CCC)cnnc1 C(=O)(C1=C2CCCN=C2NN1)NCC1C(C)CCN(C(=O)Cc2csc(S)n2)C1 c1(CC)nn(C)c(CC)c1CNC(=O)NC(c1nc(C)no1)(C)CC c1(C(=O)NCCCCN(C)C(C2CC(O)C(F)C2)=O)nccc2[nH]ccc12 c1(C(N2CCN(C(CC(CCCC)O)=O)CC(O)C2)=O)nncc2c1CCCC2 c1(OC)ncc(C(=O)NCc2cn(CC(=O)N)nn2)s1.C1(CCO)CCOCC1 C1(C(C)C)CN(C(=O)C(C)(C)CF)CCC1NC(c1cn(C(C)C)nn1)=O Cc1nc(C(C)C)nc(O)c1C(=O)N.c1(C=O)cn(C)nc1Cl.CCC1CCC1 c1(C(=O)OC(C(C)SC)C)cccc(C2=CCOCC2)c1 CC1(C)C(NC(=O)CCOC2CCOCC2)CCN1C(=O)C(F)CC1CCCC1 Cc1ccccc1C=CCNC(C1CC(O)CN(C(C2(CO)CC2)=O)C1)=O N1(C(C2(CC#C)CCOC2)=O)CCOCC(NC(c2cn(CCCC)nn2)=O)C1 C(=O)(C1=CCCCCC1)NC(C(C(=O)NC(C(=O)NC)CC1CC1)(C)C)C CC1(CNC(C2CC(n3cnnc3)C2)=O)CCCC1.C1(O)(C=O)CCOCC1.N c1(NCCCN(C(c2ccsc2OC)C(=O)NC)CC)ccc(OC)cc1C C(=O)(CCCCCCC)NC1(CCCC(N2CCCC(C#C)C2)=O)CCC1 CC1CCN(c2ncc(O)cn2)C1CNC(=O)CCN1CCCCCC1 c1(C(N2C(C=C)CCC2)C(=O)NCCC2CC2)cccc2c1CC(C)(C)O2 c1(C(=O)NC(c2nc(=O)o[nH]2)C)coc(CNC(=O)Cn2ccnc2)c1 C=CC(C)(C)CCNC(C1CC(C)(NC(C2CC2C(F)(F)F)=O)C1)=O N1(Cc2ccc(OC)c(C)c2)CCC2(NC(c3cnco3)=O)CCCC12 c1(OCCC(=O)N(CC(C)N(C)C(C2CC2C2CCC2)=O)C)ccc(Cl)cc1 CCC(CNC(=O)CN1CCC(C)CC1)(CC)C(=O)N1CC(C)(CCO)C1 CCCC(C)CC(=O)N1CC(OCC(=O)NC(C)C(C)C(=O)OC)C1 CN1N=CC(CC(N2CCCCC2C(=O)NC(CC2CC2)C2CC2)=O)C1=O Cc1c(C(=O)NCCC2(O)CN(C(c3coc(Cl)n3)=O)C2)cnn1C1CC1 N1(C(c2cc(C)sc2)=O)CC2CCC1C1CN(CCCc3ccccc3C)CC21 c1(C(N2CCC(CNC(CC3CC(=C)C3)=O)C2(C)C)=O)cc2ccc(C)cn2c1 n1(C(C)C)cncc1CNC(C1(N(C)C(c2ccon2)=O)CC1)=O CC(C)(C)CCC(=O)NC(C1CCCC1)CNC(=O)Cc1ccc(Cl)cc1F N1(C(CC2(C)CC2(F)Cl)=O)CCOC2(CCN(C(C3SCCS3)=O)C2)C1 c1(CN2CC(CC(=O)NCCc3ccc(O)cc3)OCC2)cccc(Cl)c1Cl CCC(CCC(=O)N1CCNC(=O)C1CCO)NC(=O)Cc1csnn1 Cc1ccc(-c2nnn(CC(=O)NC3CC(NC(=O)Cc4cocn4)C3)n2)cc1 c1(C(=O)NC(c2cccc(O)c2)C(N2CCC(CC(F)(F)F)C2)=O)ccccc1O Cc1ccc(C(N2C3CN(Cc4cc5cnccc5[nH]4)CC23)=O)c(F)c1F c1(Nc2cccc(OCC(=O)N(C)C)c2)ncnc2ccccc12 C1(C(N(CCC(C(C)C)NC(=O)CN2CCCC2=O)C)=O)CCC2CC1CO2 c1(OC)cc(NC(C2CCCN(C(c3cc(O)cc(Cl)c3)=O)C2)=O)cc(Br)c1Cl O=C1OC(C(N2CCCC2c2cccs2)=O)Cc2ccccc21 CCC(C(=O)OC)C(=O)NCC(C)CNC(c1ccccc1-c1ccccc1)=O C1(C)(NC(Cc2ccc(C)o2)=O)CCCCC1C(=O)NCCCc1cccs1 c1(C(N(CC(CC)NC(C2CCCOCC2)=O)C)=O)cccc(C)n1 N1(C(c2nnc(C)s2)=O)CCCC(N(C(=O)CCc2cnc(C3CCC3)o2)C)C1 CC(=O)CCC(C)(C)C(=O)N1CCC(c2nn[nH]n2)C(F)(F)C1 C#Cc1ccc(C(=O)N(CCC(C)NC(=O)C=Cc2cc[nH]n2)C)nc1 c1(C(C)(C)C(=O)N)ccc(F)cc1F.C1(CC)CCCN1C(C1CC1C(F)F)=O c1(C(=O)NCC(C2CCCCC2)NC(C2CCCSC2)=O)cc2ccc(F)cc2s1 C(=O)(CCCC(C)C)NC(CNC(C(c1c(C)noc1C)C)=O)C(C)C Cc1cccc2c(CN=c3cc(NCCCC(=O)NC(C)(C)C)nc[nH]3)c[nH]c12 c1(OC)cc(CNC(c2ccccc2F)c2nccn2C)ncn1 C(=O)(CC1=CCCC1)N(C1CCN(C(C2CCCN2C(=O)OC)=O)C1)CC N1(CC(c2nccs2)C)C(=O)CCN(CCC2CC3(CCC3)C2)C1=O c1(C(N2CCCC(Cc3ccc(Cl)cc3)C2)C(=O)NCCSC)ccc(Cl)cn1 N1(C(C(C)SCC)=O)CCC(N2CCC(NC(=O)C(C(=O)O)OC)CC2)CC1 C=CCC(F)(F)C(=O)NC1CC2C(NC(=O)CC(C)n3cccc3)C2C1 N1(CC(=O)OC)C(=O)OCC12CN(S(=O)(=O)c1csc(C(=O)O)c1)C2 Cc1cc(C(N2CCN(C(c3cc(C(N)=O)[nH]n3)=O)CC2CO)=O)cc(C)c1 c1(CC)cc(C(N2CCC(C3CCCN3C(=O)C3CC3)CC2)=O)ncn1 CC1(CNC(=O)CN2CCSCC2)CCC(NC(=O)C2=COCCC2)CC1 C(CC(=O)N(C)CCOCC)(C(C)C)OC1CC(C)(C=O)N(C)C1.CC.N N#Cc1cc(C(=O)Nc2ccc(C(N3CCCCC3)=O)cc2)n2c1CCCC2 CN1CC(O)CCC1C(N1CCCCC1C(N1CC2CCC1C2)=O)=O c1(CC(C(=O)NC2CC(NC(C(C)(C3CC3)OC)=O)C2)O)ccccc1Cl Cc1noc(C)c1C(C)C(=O)NC(C)CC(C)NC(c1csc(Br)c1)=O C(=O)(C(C)(C)CC(F)F)N1CC(CNC(c2c(C)c(Cl)sc2Cl)=O)C1 C12(Cn3cc(C4N(C(CC5C(C)C(=O)CC5)=O)CCC4)nn3)COC(C1)C(O)C2 C1(C(=O)NCCCCCCC2CC2)(CC)CCCN(C(=O)C(C)c2cc[nH]n2)C1 C(=O)(CC(C)CC(F)(F)F)N.N1(C(CCNC(=O)OC)=O)CCOC(C)(C)C1 c1(C(N(C(c2ccccc2)C)C)=O)cc(F)cc([N+](=O)[O-])c1 c1(C(=O)NC(C)CNC(c2cc(Cl)cnn2)=O)c(Cl)ccc(F)c1F C1(C(N(CCC2CCC2)C)=O)CC(C)(C)CN1C(c1cnn(C(C)C)n1)=O O=C1CCC2(C(=O)NC3CCCC4CC34)CCCC2C1 C1(CNC(CCC2CC(OC)C2)=O)CCCCN1C(=O)C=C1CCN(C)C1 N1(C(c2ccc(OC)nc2)=O)CCCCCC(NC(C2CC2[N+](=O)[O-])=O)C1 c1(C(N2CC3CN(C(=O)C(F)Cl)CC3C2)=O)ccc(I)c([N+](=O)[O-])c1 c1(C(=O)NCCN(C(C(CC#C)(C)C)=O)CCC)nccc2nn[nH]c12 C(CCCCC(=O)NCC(=O)NCC(c1ccsc1)O)OCC N1(CC)CCC(=O)N(Cc2ccc(OCC(F)(F)F)o2)C1=O C1(N2C(=O)NC(C3CC3)C2=O)CCCOC12CCOCC2 N1(C(c2c(OC)ncnc2C)=O)CCCC2(NC(c3ccccc3Cl)=O)CC2C1 Cc1cc(C(=O)NCCCNC(=O)C(=O)NCC(F)(F)F)cc2ccoc12 N1(C(C2CC2c2ccc(Cl)cc2)=O)CCN(C(=O)C(O)C(F)F)C2(CC2)C1 C1CN(C=O)C1(C)C.CC(C)N(C(=O)C=CC=O)C.C(C)(C)C.CCC C(CCCC)(CC(=O)N1CCCC(O)C1)NC(C(CC=C)CC)=O C1(NC(C(C(C)(C)O)F)=O)CN(C(=O)C(c2csc(=N)[nH]2)=O)CCC12CCC2 N1(C(C=Cc2n(C)cnc2)=O)CCC2(CCC(NC(C3CSCCS3)=O)C2)C1 c1(C(C)C)nn(C)c(NC(C2CC2C(N2CCC(C)(C)C2C)=O)=O)c1Cl c1(CN2CCN(CC(=O)N(CC(F)(F)F)CC)C(=O)C2)c(O)cc(O)cc1Br c1(C(=O)N)ccc2c(c1)NC(=O)C1CCCN21.C(C(O)C)NC(c1ccoc1)=O C1(CNC(C(CC)(C)CO)=O)CC12CCN(C(c1ccoc1Cl)=O)CC2 c1(C(C(=O)NCC2CC3(CC3)CO2)F)ccccc1Br c1(C(=O)NC)ccc(C(=O)NC2CC(C)N(C(=O)C(C)C)C2)cn1 C=C(C)C(O)CC(=O)NCCC1CCN(C(c2ccccc2CC#N)=O)CC1 C1(CN(C)C(c2c(Cl)ncn2C)=O)CCN(CC(F)(F)F)CC1 Cc1nc(C2CCCCC2)sc1C(=O)NC1CC1NC(=O)C(C)C C1(CNC(c2n(CC)ncc2)=O)C2CCC1CN(C(c1nn(C)cc1Cl)=O)C2 C1(CC=O)CCCC(C(F)(F)F)O1.N1(CC=O)CCC(C)C1.CC=O.CC.N c1(-c2ccc(C(=O)NCCC(C)NC(C=CCOC)=O)[nH]2)ccccc1F N1(C(C)=O)CCC(C)(C(N2CC3CC2CN3C(=O)CNc2ncccn2)=O)CC1 N1(c2c(C)nccn2)CCC2(CC1)CC2C(=O)NC1CN(S(C)(=O)=O)CC1C C(=O)(CCC)NCCN(CCOC)C(C12CC(C)(C1)C2)=O.C(C)=O CC1CC(C(=O)N2CC=CC(NC(c3csc(-c4cnn(C)c4)n3)=O)C2)=NO1 C1(C(=O)N)CC2C(C1)C2(F)F.C(=O)(C1=CCCC1)N1CC(COC)(C)C1 N1(C(CCCC(N)=O)=O)CCCC12CCN(C(c1cc3cccn3c(O)n1)=O)C2 c1(OC)ccccc1C(C)N(C)C(C1CC12CN(Cc1cccs1)C2)=O C1(C(N(C(C)C)CC)=O)CCC([N+](=O)[O-])CC1.C(=O)(C(F)(F)C1CCCC1)N C(C1CCOc2ccccc21)OC(c1cc(F)c(F)c(Cl)c1F)=O N1(C(=O)CC2CCN(C(C3CC34CCCC4)=O)CC2)CCN2CC(O)CC2C1 Cc1cc(C(N2CC(NC(=O)C(N3C(=O)CCC3=O)C)C(C)C2)=O)c(C)n1C Cc1nc(C(=O)NC2CCCCN(C(=O)CC3CCCC4(CC4)C3)C2)c(C)n1C c1(OC)cccc(C2(C(=O)NCC(C)(C)C)CC2)n1.C(=O)(CC(C)(C)C)N Cc1noc(C)c1CC(N1CCCCC1CCCNC(c1csnn1)=O)=O CC(CC(C)(C)C)C(=O)NC1C2CC(NC(=O)Cn3ncc4ccccc34)CC12 c1(CN2C(C)CN(c3cc(C(F)(F)F)ncn3)CC2)ccc(Cl)c(Cl)c1O C1(NC(C(CCC)N(C)C)=O)CN(C(=O)COC2(C)CCCC2)CCC12CCC2 c1(N2CCCCC(COC)C2)nc(NCC(C)N(C)C2CC2)c2ncsc2n1 C1CCN(C(c2ccc(C(C)C)c(F)c2)=O)CC1C.C1(C(=O)N)(OCC)CC1 c1(C(N(CCNC(CCCCN(C)C)=O)C)=O)cc2scc(Cl)c2[nH]1 Cc1ncc(Br)cc1CNC(=O)C(=O)NC1CC1C1CC1 CC(C(=O)NO)NC(C1(CNC(C2CNC(=O)N2)=O)CCCC1)=O N1(C(CC(N2CCCCC2=O)C)=O)CC=CC(NC(=O)CCN2CCOC2=O)C1 CC1(C)COc2c(C(=O)NC3CCCC3NC(C3CC3F)=O)cccc21 N1(C(C(F)=CCC)=O)CCN(C(=O)CC2OCCC2(C)C)C(CCO)C1 C1(C(N(CC(C)CO)C)=O)CC(NC(=O)Cn2ccnc2)C12CCC2 N1(C(C2=C(C)Oc3c(cccc3)C2)=O)CC(N=c2[nH]c3ccccc3cc2C#N)CC1C c1(C(=O)N)nc2ncccn2n1.C1(O)(CC(=O)NCC2CC2C)CCCCC1 N1(C(C2CN(C(C(C)CC#N)=O)CC(C)(C)C2)=O)CC2(CCC2)C12CCC2 CS(=O)(=O)c1cccc(-c2ccc(C(=O)NCc3cccc(F)c3F)nn2)c1 c1(C(N(C(CCNC(C(c2ccc(C)cc2)O)=O)C)C)=O)c(C)nc2sccn12 c1ccc(C#N)cc1.C1(CNC(C(C)CO)=O)CCC(CNC(=O)C)CC1.S c1(C(N2CC(F)C2)=O)cn(C(C)C)cc1C.c1(CCC)nc(C(=O)NC)co1 N(C1CCCc2cnn(C(C)C)c21)C(C1C(C(=O)OC)CCCN1)=O CCC(O)CN(C(=O)CCOCCNC(=O)C=CC1CCC1)C1CC1 C1(NC(CN2C(C)CC2)=O)CN(C(=O)Cc2csc(NC=O)n2)CC(C)(C)C1 Cc1cccc2[nH]c(=NC3CCN(C(c4c[nH]c5cccnc45)=O)CC3C)oc12 c1(C(=O)O)cnc[nH]c1=NCC1CCCCN1C(=O)Cc1cc(F)ccc1Cl Cc1c(C(=O)NCC(O)CNC(C2CCCCS2)=O)cccc1F C1(CC=C)(NC(c2cc(C)cs2)=O)CCCN(C(C2(C)CC2(F)Cl)=O)C1 c1(NCC(C2CC2)OC)cc(=NC(C)c2cn(C)nn2)[nH]c(C)n1 C(C)(C)(CCCN=c1[nH]nc(C2CC2)o1)NC(c1ccc2cc(C)cn2c1)=O C(CC(C)CC)(C(=O)NCc1ccnc(Cl)c1)NC(CCN(CCC)C)=O C1(CNC(C(C)=CC2CC2)=O)CCCN(C(C2CC3CCC(C2)O3)=O)CC1 CCCC(C)(O)C(=O)N(C)CC1CCN(C(=O)Cc2ccc(OC)cc2F)C1 CC(C)CCC(O)C(=O)NCC1(F)CC(NC(C2CCN(C)C2)=O)C1 c1(C(=O)NC2C3N(C(c4cn(CC)nc4C)=O)C(CC3)C2)n[nH]c2c1COCC2 CC1CCN(C(=O)C(c2cnn(C)c2)NC(=O)C(C)CC#N)CC1 CCCC(O)(CCC)CC(=O)NC1(CNC(c2ccc(F)c(SC)c2)=O)CC1 c1(NC(C2(C)CCCN2Cc2cnc(-c3ccccc3)s2)=O)cc(Cl)cnc1Cl C1(NC(CC(CN(C)C)O)=O)COC2(C1)CN(C(=O)CCCC#N)C2 Cc1ccc(C(N2CCCC2C(=O)N(CCC(=O)NC2CC2)C)=O)cc1C c1(C(=O)NC2CCN(CCNC(c3nc(C)oc3)=O)CC2)cn2ccccc2n1 c1(C(C(=O)N)C)cccc(N(C)C)c1.CC(C(C)(C)C)=CC(=O)NC1CC1 c1(C(N2CCC(NC(c3cc(OC)ncc3F)=O)C2)=O)ccc2cncn2c1 Cc1ccc(NC(=O)CO)cc1.N1(C=O)CC(O)CC1C1CC1.C(C)(C)C N1(C(c2cc(C(C)=O)c(C)[nH]2)=O)CCC(C)N(C(=O)Cc2cnoc2)CC1.CC c1(N(CCC)C(=O)NC(C)(COC)CO)cccc(C#N)c1 O=C(CC1NC(=O)c2ccccc21)N1CCN(C(C23CC(C2)C3)=O)C(CCO)C1 CCC(C(=O)Nc1sccc1CN1CCOC1=O)NC(=O)OC(C)(C)C C1(NC(c2c(C)scn2)=O)COC2(CCN(C(c3nc4ccccc4[nH]3)=O)C2)C1 N1(C(C2(C#C)CCN(C(c3nscc3C)=O)C2)=O)CCC(=C(F)F)CC1 Cc1nc(C(=O)NCCCCCNC(=O)C(C2CCOCC2)C)c2ccnc-2[nH]1 c1(C(=O)OCC)cc(CNC(=O)NC2(C(=O)O)CC(F)C2)cn1C N#CC1(CC(=O)NC2CC2CNC(=O)CCC2CCC(=O)N2)CCCCC1 c1(C(N(CCCC)C)=O)cc2c(s1)CN(C)CC2.c1(C(=O)N)occc1C1CC1 c1(C(N2C(CC)CN(CC)CC2)=O)noc2cc(-c3ccc(CO)s3)ccc12 C1(NC(C2OCCN(C(C(C(C)C)CN(C)C)=O)CC2)=O)CCc2ncnn2C1 c1(C(=O)NCC2C3CC2N(C(=O)CC2CCOC2)C3)ccc(F)c2ccncc12 Cc1onc(Cl)c1C(=O)NCC1CC(NC(C2CC(C)C2)=O)CCO1 N1(C(C2NC(=O)OCC2)=O)CCN(C(C2(c3ncco3)CC2)=O)CC(O)C1 N1(C(C(C)(C)C)=O)CCC(F)C(NC(c2cc(CC3CCCC3)ccn2)=O)C1 Cc1ccc(C2CC2)c(C(=O)NCC(F)CNC(=O)CCc2nncn2C)c1 C(N=c1[nH]cnc2ccc(O)cc12)C1(CNC(C(C(CC)O)C)=O)CCC1 C#CC1CN(C(C2CCCN(C(C3OCCC3C(C)C)=O)CC2)=O)CC1O c1(NCc2nnc(SCC(=O)NC)n2C)nnc2n1CCN(C)C2=O c1(C2(C(C)NCCOC(=O)C(C)Cc3cccnc3)CC2)ccccc1F Cc1csc2nc(CC(=O)NC3(c4ccccc4)CCN(C(=O)C(N)=O)C3)cn12 N1(C(c2ccc(CC)[nH]2)=O)CC(NC(c2[nH]nc(OC)c2Cl)=O)CC2(CCC2)C1 C1(NC(=O)Cc2cscn2)CC2(CCN(C(=O)CCN(CCO)CCO)C2)C1 n1(CC(=O)NCCCC)nc(C)cc1C=O.c1(C=O)cc(C(C)C)sn1.O N1(C(C(C)CSc2ccc(F)cc2)=O)CCN(C(=O)CC(C)(C)C)C2CCC12 c1(C(N2C(CO)CC(NC(COC3(C)CCC3)=O)C2)=O)cccc(F)c1F c1(COC)nc(C(=O)NCC(F)CNC(=O)C(C2CCOCC2)O)cs1 C(=O)(CP(=O)(C(C)C)C(C)C)NC1CN(C(C=C(CC)CC)=O)CC1O C1(N(C(C(CCC)C#N)=O)C)CC2CCC(C1)N2C(C1(OC)CCSCC1)=O N1(C(C2C(C)C2)=O)CCN(C(C2CCC3(C2)CC3(F)F)=O)CC(C)(F)C1 C1(NC(N2CCN(c3ccccc3)CC2)=O)CC2(CCCC2)C1.C12(CC1)NC2 C(=O)(CCCN(C(=O)COC1CCOC1)C)NC1(CCC)CCC1 C1(CN(C(=O)Cc2sccc2Br)C)CCCN(C(=O)C=CC(C)(C)C)C1 Cc1cc(CNC(=O)NC2CCCNCC2F)cc(C)c1O CC1OC2CCC1(C(=O)NCC(CNC(=O)CC1CCCNC1=O)CO)C2 N1(C(C2N(C)CSC2)=O)CC=C(CNC(=O)CCN2CCCCC2)CC1 c1(OC)c[nH]c(C(=O)NCCC2CC2)cc1=O.C1(C)(C=O)CCN(C)CC1.N c1(OC)cc(NCC(N2CCC(Nc3cnn(C)c3)CC2)=O)ccc1F c1(SCC)cccc(C(=O)N(C(C)CNC(c2ccnnc2C)=O)CC)c1 C1(C)(CNC(C(CC#C)C)=O)CN(C(=O)CN2CCC(CO)CC2)C(C)(C)C1 N1(C(c2nc(CC)oc2)=O)CC(CO)C2(C1)CN(C(=O)C(C)N=[N+]=[N-])C2 c1(C(=O)NC2(CC=C)CN(C(C3CCOC(C)C3)=O)C2)cccc2nc(C)nn12 c12ccc(Cl)c(c1F)CN=C1C=CC(=CN1)CN2.N1(CC)Cc2ccccc2C1 c1(CC(=O)N(C(C)(C)CC(=O)NC2COC(C)(C)C2)C)cccc(C#N)c1 CCCCCCCCCCC(C)(C)C(=O)NCCOCCN(C)C(C)=O c1(-c2cc(C)c(Nc3ncccn3)nc2)cccc2c1CCC2 c1(OC)n[nH]c(C(=O)NC2CCCC2NC(C2CCC(=O)N2)=O)c1Cl CCCC(O)CC(=O)N1CCOC(C(C)NC(=O)CCC[N+](=O)[O-])C1 N1(C(CC=CC=C)=O)CC2(CCOCC2)CC1CNC(=O)C(C)C(F)F N(C1COc2ccc(F)cc21)C(C(=O)NCc1n(C)nc2c1CCCC2)=O C(=O)(CCC(=O)NN(C)C)N(CC(=O)NC1CNC(=O)OC1)C(C)C c1(N(C)C)cnc(C(=O)NCC2CC2)nc1.c1(C=O)cc(C(C)(C)C)no1 N1(C(CC(C)C)=O)CCC2(CC2NC(=O)CCOC(C)C)C1 c1(C(=O)NC(C2CN(C(=O)CC3CCCC3)CCO2)C)cc(F)c(F)cc1N c1(C(C2(C(=O)NCC(C)=CC(=O)O)CC2C)=O)ccc(F)cc1 C1(CC(=O)N(CC(C)C)CC(=O)NCCC(F)F)CCCC12CC2 N#CC1CCCCC1NC(=O)CCOCCCNC(C1(CCF)CCC1)=O c1(N(C)C)ncc(C(=O)NC2CC(NC(C3CCCN(C4COC4)C3)=O)C2)cn1 C(=O)(C(CNC(=O)C(C)CCCOC)C(C)C)NC(CCC)C(=O)N(C)C C1(NC(C2CCCS2)=O)CN(C(C23CCCCN2CCC3)=O)CC12CCOCC2 C1(C#N)(c2ccc(C)cc2)CCN(C(C2CC3CCCC2N3)=O)CC1 Cc1nnc2c(C(=O)NCCC34CCC(C)(C3)OC4)nccn12 C1(C)(C(=O)NCC(C)CNC(=O)COCCCF)CCC(O)CC1 CC(=O)CCCC(=O)NCC1CC(NC(=O)C(F)CC2CC2)CC1O C(C1CCCN1C)=CC(=O)N(C(C)CNC(=O)CN1CCCCC1)C N1(C(c2c(CC)[nH]nc2Cl)=O)CCC2(CCC2)C1.C12(C=O)CCCC(C1)OC2.N C1(CN(C(=O)C(O)C(F)F)CC)CCN(C(=O)CCOC2CCOCC2)CC1 C1(C2CC=CCC2)(C(N2CCN(CC(C)NC(=O)C(N)=O)CC2)=O)CC1 C#Cc1ccc(CC(=O)N)cc1.C1CCN(C(=O)CC2C(C)(C)C2(C)C)C(C)C1 N1(C(C(COC)O)=O)CC2CC1CN2C(C1(CO)CCCCO1)=O C1(C(=O)NC(C(C)C)CNC(=O)CC(=O)NC2CC2)Cc2ccccc2O1 Cc1nscc1C(=O)NC(C)(CNC(C1(C)CCCS1)=O)Cn1cccn1 Cc1cc(N)cnc1C(=O)NCC1CCN1C(c1cc(Br)oc1C)=O c1(CCC=O)ccccc1C(N)=O.C12(CCC)CC(C(=O)N)(C1)C2.CCCC c1(CC(=O)NCCOCCCNC(=O)CC2CCCCCO2)cccc(O)c1 C1(NC(C(=O)N(C)CC2CCC(C)CC2)=O)CNCC2(CCOCC2)C1 N1(C(C=Cc2ccc(OC)cn2)=O)C2CCCC1CN(C(=O)C(C)CC(F)F)C2 c1(NC(c2ccsc2-c2cnn(C3CCCC3)c2)=O)nccc2[nH]ccc12 C=CCCC(C(=O)OC)NC(C1CCCN(C(C2(COC)COC2)=O)CC1)=O N1(C(CC(C)SC)C(=O)NCCC#N)CCc2cc(Cl)ccc2C1C S(=O)(=O)(c1ccc(Br)cc1N1CCN(C)C(CC)C1)NC(COCC)C(C)C CC1CCCC(C(=O)NC2CC23CC(NC(c2cnn(C)c2)=O)C3)O1.C1CC1 CC1(C)CN(c2nnc(CS(C)(=O)=O)s2)C1CO N1(C(c2n(CC)ncc2)=O)CCCC(C)C1C.c1(C=O)cc(C(F)F)n(C)n1 C1(NC(C(CCOC)(C)C)=O)CC2CCC(C1)N2C(C1CC(=O)CO1)=O CC1C(C=CC(=O)NCCNC(=O)C(C)(C)n2cccn2)C1(Cl)Cl O(N1CCC(NC(c2nn(CC)c(Br)c2Cl)=O)CC1)CC C(=O)(CC(C)(C(F)F)NC)N1C(CC)CN(C(=O)CCc2ccc(O)nn2)CC1 N1(C(c2cnc(C)nc2)=O)CC2=C(C1)CN(C(C1CC3CCC(C1)S3)=O)C2 C(=O)(C(C)C(C)(F)F)N.C1(CCNC(CCOCCCOC)=O)CCCCC1 Cc1cccc(C(N2C3CCC2C(C(=O)NC2CC(O)C2)C3)=O)c1I c1(CN2CCC(NC(COc3c(C#N)cccc3)=O)C2)cc(F)c(Cl)cc1Cl N1(C(CC2N(C)CCC2)=O)CC(F)(F)CC1(C)C.C(=O)(C)N.C1(C=O)CCC1 CN1CCOC(C(N2CCC(CCC(=O)NCc3ccc(C#N)o3)CC2)=O)C1 CCCC(CCC)=CC(=O)OCc1nc(C#N)cs1 C(=O)(C1=CC2(CCOC2)C1)NCC1CC(NC(c2c(CC)[nH]nc2)=O)C1 c1(C(N2CC(C)(CNC(c3c(C)cns3)=O)C(C)C2)=O)n[nH]c2ccc(Cl)cc12 Cc1cccc(C(=O)N(C2CC2)CC2CCCN2C(C2CC(O)C2)=O)c1 C1(N(C(C(=O)NCc2cccs2)C2C(C)C2)C)CCNC1=O c1(N2CC(CN(C)C(c3ccc(C(F)(F)F)o3)=O)C2)nc2ccc(Cl)cc2s1 CC1(C)Cc2cc(NC(C3(O)CCN(Cc4ccccc4)CC3)=O)ccc2O1 C1(OC(C2(C(=O)OCC)CCOCC2)=O)CCCC(C)C1C C1(NC(c2n(C)ccc2)=O)CCCC(NC(=O)CCCN2CCCCC2)C1 N12CCCC(CC1)N(C)C(=O)C2C.c1(C=O)cncnc1.C(CNC=O)OC.N c1(C(=O)NCCOCCNC(CC=CCC)=O)cc(OCC)ccc1Cl C1(C2(NC(c3nc(C4CC4)no3)=O)CC2)CCCN1C(=O)CCF C1(=C(C(=O)NC2C(NC(C3C(C(C)(C)C)C3)=O)C2)F)CCCCC1 N1(C(Cc2scc(C)c2)=O)CCCC(C2CN(C(c3cnc(Cl)cn3)=O)C2)C1 C(C1CCCN1C)=CC(=O)NCC(CNC(C(C)Cc1ccnn1C)=O)(C)C c1(OC)cc2c(cc1C(N1CCC(CNC(=O)C)C1)=O)CCC2.c1ccsn1 c1(NC2(c3nccc(OC)c3)CCC2)nc(C)cc(=NCCC2SCCS2)[nH]1 c1ccccc1.C(=O)CC.C(C(=O)NCCCC1CC1)SCC#C.C(=O)CO N1(C(C2(OCC)CCC2)=O)CCN(CC)CC1.c1(CC(=O)N)ncn(C)c1C C1(OC)CC(C(=O)NCCC2CCCN2C)N(C(=O)CCc2ncc[nH]2)C1 c1(CNC(C2CC(NC(CCC(=C)Cl)=O)C2(C)C)=O)cc(F)ccc1F c1(C(=O)NCC(C)NC(c2c(C)cc(Cl)cc2)=O)ccc2c(c1)COC2(C)C c1(C(CNC(C(CC)CC)=O)NC(c2nnsc2C)=O)ccc(F)cc1F CCCC(C)C(C(=O)Nc1ccccc1OC)N1CCC(C)C1 C1(C(=O)NC2C(NC(CCCOCC)=O)COC2)CC12CC(O)C2 N1(C(CC(C)c2ccco2)=O)CCC2(C1)CN(C(C1CC13CCCC3)=O)C2 c1(C2C(C(=O)OC)C2)ccc(C(=O)NCC2(CCCCl)CC2)cc1 C1(CNC(C(C)OCC=C)=O)COCCN(C(=O)Cc2ccc(F)cc2Cl)C1 N1(c2ncc(C(=O)OC)cn2)CCN(Cc2ccc(O)c(OC)c2)C(C(C)C)C1 c1(C(C)C)cccc(NC2CC(C(=O)NC(=O)C(C(C)C)C3CC3)C2)c1 C1CC2(C1)OCCO2.c1(-n2cc(CN(C(C)=O)C)nn2)ccccc1C(=O)N.C c1(C(=O)NC2CCC(NC(CCCN(C(C)=O)C)=O)C2)ncccc1OC(F)F Cc1ncccc1CC(=O)N(C)CCC1CCCCN1C(C1CC1(F)F)=O Cc1sc(=O)n(CC(=O)NC23CC2CN(C(C2CCCC2)=O)C3)c1C C#CC1CCCN(C(=O)CCN(C(C2CCCN2C(C)C)=O)C(C)C)CC1 c1(OCC)cccc(C(=O)NCCC2CC(NC(C3CC3F)=O)C2)c1 c1(C(=O)NC2C(NC(C(CC)O)=O)CCC2)c(C)nc2ccc(Br)cn12 c1(-n2cc(C3N(C4CCN(C(=O)CCn5ccnn5)C4)C3)nn2)ccc(F)c(Cl)c1 Cc1ncc(Br)c(C(=O)NCC(C)(C2CC2)NC(C2CC2(F)F)=O)n1 C1(CC(N2CCC(F)C2)=O)CCCC(F)(F)C1.CC1(C)CCN(CC(=O)N)C1.C N1(C(CCSC)=O)C(CNC(=O)C(C)OCc2ccccc2)CC2CC12 c1(CC(N2CC(N(C(=O)CC3(C)CC3)C)C2)=O)csc(C(F)(F)F)n1 C1(C(C)NC(CCc2c(C)ncs2)=O)CCCN(C(c2c(C)ncn2C)C)C1 C(=O)(C(F)(F)C(C)O)N1CC(F)(CNC(c2ccc(CCCC)cc2)=O)C1 c1(-c2n(-c3cnc(OC)nc3)nc(-c3cc[nH]n3)n2)nccc2ncccc12 c1(C(N(CCCN(C(=O)CC2CCCCN2C)C)C)=O)cc(O)cc(Cl)c1 C(=O)(C1=NOC(C)(C)C1)NC(C(=O)NC(C1CCCC1)C)CC1CCCC1 CCCC(CC)C(=O)N(C1CN(C(C2CCCC(C)CC2)=O)C1)C Cc1c[nH]c(C(=O)NC2CCC(CC(=O)N(C)CCc3cccs3)CC2)c1C c1(NC(C2CC3CC3N2C(c2ncc(Cl)cn2)=O)=O)ccc(-c2ccccn2)nc1 c1(OC)cccc(C(=O)NC(C(=O)NCC2(C)CCC(=O)N2)C(C)O)n1 c1(CC(=O)NCC2(O)CN(C(C3(CO)CCCO3)=O)C2)csc(Br)n1 Cc1ncncc1C(=O)NC1CC(CNC(c2ccc(-n3cccc3)cc2)=O)C1 N1(C(C2CCC(C(F)(F)F)CC2)C(=O)NCC(=C)C)CCC(C(N)=O)CC1C C1CC2(CO1)CN(C(c1oncc1)=O)C2.C(C(=O)N)NC(=O)OCC=C CC1(C)CCCCC(C(=O)NC(C(=O)OC(C)(C)C)c2cncs2)C1 c1(NC(=O)NCC(=O)NC(c2ccccc2)CC)cc(C)ccc1C#N N1(C(C(C2CC(NC(C3CNC(=O)N3)=O)C2)F)=O)CCNC(=O)C1 CC(C)CCC(=O)NC1CCOCC1NC(c1coc(C(F)(F)F)n1)=O N1(C(C2CC(C(=O)OC)C2)=O)CC(C)C(F)(F)C1.C(=O)CCc1cnoc1 c1(C(C)N(C)C)cn(CC(N2CCCC2c2nncn2C)=O)nn1 Cc1nn2ncccc2c1C(=O)NC1CCN(C(c2cc[n+]([O-])cc2)=O)CC1 C1(O)(c2cn(CC)nn2)CCCN(C)C1.N1(C(C2(C(C)=O)CC2)=O)CCCCC1.O C1(NC(C=CC=CC)=O)CC2(CCC(NC(=O)CCCN(C)N=O)CC2)C1 c1(COC)ccc(NC(=O)NC(C)Cc2cncn2C)cc1O c1(C(CC)C)nnc(N2CCOC(c3ccc(Cl)cc3)C2)n1CC CC(C)CS(=O)(=O)CCC(=O)NC1CN(C(=O)C(C)C(C)C)C1 N1(CCCNC(C(CC)OC)=O)CCN(Cc2cccc(N(C)C)c2)CC1 Cc1cccc(C)c1NC(=O)C(CNC(C1CC12CCCCC2)=O)C(C)C c1(C=O)ccc(=O)n(C)n1.Cc1nc(CO)sc1C(=O)NC(C1CC1)C.C N1(C(C2(CC#C)CCCCO2)=O)CCCC(N=c2[nH]nc(C(F)F)s2)(CO)C1 c1(C(=O)NCCCOCCN(C(CC2CC(C)C2)=O)C)nnn2ccccc12 CC1CCN(C(=O)CCC2CCOC2)C(C(=O)NCC2CSCCO2)C1 c1(CN2CCC(NC(C(C)COc3ccccc3)=O)C2)ccc(Cl)cc1.C(C)N c1(C(=O)NC2CCC(NC(Cc3nc(C)sc3)=O)C2)nnn(C2CCOC2)c1C N1(CC23CC(C#N)C(C2)C3)CC(NS(=O)(=O)C2CC2)C2(CCC2)C1 c1(C(=O)NC(C)(CO)C(N2CC3CCC(CC3)C2)=O)cc2cnccc2[nH]1 N1(C(C(C)OC)=O)CCOCC(C)C1.c1(C(=O)N)c(C)nn(C)c1-n1cccn1 c1(CCC(=O)N(C(c2ccncc2)C)CC)ccc(-c2sccc2C)s1 N1(C(C2(COC)CCCCC2)=O)CCOCC(F)(CNC(=O)C(C)SC)C1 CC1(C)CC(NC(C2(F)CCCN(C(=O)CC3CCSC3)C2)=O)C(=O)O1 N1(C(C=CC(=O)O)=O)CCOC(C)(C)C1.C(=O)C(O)P(C)(C)=O.CCCC C(=O)(CCCn1ccnc1C)NCCN(C(=O)CC1CCOC1=O)CC C1(C(=O)NCC(CN(C)C(C2(F)CC2)=O)O)CCCC(c2ccccc2)O1 CC(C)(C)CCC(=O)N1CCOCC(CNC(c2ccncc2Br)=O)C1 Cn1c(N2CCCC(CCNC(c3cccc(C4CC4)c3)=O)C2)cc(O)nc1=O N1(C(C(CSC)O)=O)CC2C3CCC(C2C1)N(C(=O)CCc1cc(C)no1)C3 C(=O)(C1=CNC2=NCCC2=C1)NC1CCN(C(C2CCCN(C(C)C)C2)=O)C1C N1(CCN(c2ccccc2)CC(N)=O)CCCC2(CCCc3ccccc32)C1 c1(NC)ncccc1C(=O)NC(C(=O)N1CCC(C)CC1)C(C)OC C1(C(=O)NCCNC(c2cnn(C)c2Br)=O)CCC2(CC1)CC2 n1(CC)cnc(C(=O)NCCCCCN(C(=O)COC(F)(F)F)C)c1 CC1CNCC(c2nc(Cc3ccc(N(C)C)cc3)no2)O1 c1(NC(c2c(C)nn(CCO)c2C(F)F)=O)ncnc2ccnn12 c1(CC)nc(C#N)cc(=NC(C)C(C2CC2)NC(=O)C(CC)CC(F)(F)F)[nH]1 C1(CCOC)(NC(C2CC=CCC2)=O)CCN(C(C2(C)CC3CCC2O3)=O)CC1 N1(CCNC(CC2(OC)CN(C(=O)Cn3cccc3)C2)=O)C(=O)CCC1=O N1(C=O)CCC2C(CC(=O)NCC(F)F)CC12.C1CCS(=O)(=O)C1.CC(C)C C12(C(=O)NC(c3cn(C)nn3)C=O)CCC(CC1=O)C2.C1(O)(CC)CCCC1.N c1(CC(=O)NCC2CC3COCC3N2C(c2cocn2)=O)c[nH]c2cnccc12 N1(C(C(CC(C)C)F)=O)CCCN(C(c2ccc(C(F)F)cc2)=O)C(CO)C1 C(=O)(C1=CCC2CCC1N2C(c1n[nH]cc1[N+](=O)[O-])=O)NCc1ncc(C#N)o1 c1(C(=O)NC2CCC(NC(Cc3cccc(OC)c3)=O)CC2)cccc(N)c1C C1(NC(C(c2cn(C)nn2)NC(CCCC2C(C)C2)=O)=O)CCC2(CC2)C1 C12(CCNC(c3n(CCCOC)nnn3)c3scnc3Cl)CC(CCO1)C2 N1(C(C2(C)C(C)OCC2)=O)CC2CCC(C1)N2C(=O)CCCC1CC1 C#CCC(O)C(=O)NC1(CN(C(=O)CCc2ccc(OC(F)F)cc2)C)CC1 CC1C2CCC(C2)C1C(=O)N(CCCC(=O)NCC1NC(=O)OC1(C)C)C C(CC1CC1)(C(=O)N(C(C)CCO)C)NC(C(C1CCOCC1)C)=O CC1(C)COC(C(=O)NC2(CC(=O)NC3CCOC(C(N)=O)C3)CC2)C1 C1CN(C(=O)C2CC2)C2(CCC2)C1.O=CCCCNC(C1CC1C(F)F)=O C12(C(=O)NCC3(NC(=O)Cc4c(F)cccc4Cl)CC3)CCCCCC1OCC2 C#Cc1ccc(Br)c(C(=O)NCC(CC=C)NC(=O)CCC#CC)c1 CC(C)CC(O)CC(=O)NCC1(O)CN(C(=O)C(C)C(C)(C)C)C1 CCCCC(CC)CC(=O)N1CCOC(C(=O)NCCCC(=O)NO)CC1 C1(C=O)CC2CC1C1C2C1(F)F.c1(C(C)(C)C)ncc(C(=O)N)s1.C1CC1.C N1(C(C2C(NC(C3(C)C=CCCC3)=O)CCC2)=O)CCc2nc(O)[nH]c2C1 c1(CNC(C(=O)NC(C)C)C2C(C(=O)OC)C2)ccc(O)cc1OC C1(CN(C(CO)C2CC2)C)(NC(=O)OC(C)(C)C)CCCC2CC12 c1(C(N(Cc2cn(CC(=O)O)nn2)CC2CC2)=O)ccn2nccc2c1 CC1CCCC=C1C(=O)N1CC2(C(=O)NC3CC4CC5C(C4)C35)CC1CCO2 Cc1c(F)ccc(C(N2CC(C3CN(C(=O)C(O)C(F)F)C3)C2)=O)c1Cl c1(C(=O)OC(C(=O)OC)C(C)(C)OC)csc(S(N)(=O)=O)c1 Cc1ccccc1C(C)C(=O)NCC1CCCC1.c1(C=O)csc(C(F)F)n1.N c1(CC(C(=O)NC(CCO)C2CCC2)NC(COCCC)=O)ccc(Cl)cc1Cl CC1CN(C(C2(C)CC2C)=O)C(C)CN1C(C1CN(C)C1)=O C(=O)(C(CC(C)C)C(N)=O)NCC1(O)CN(C(C=C(C)C)=O)C1 C12(C(N3CCN(C(C4CC=C(C)CC4)=O)CC3)=O)CCC(CC1)C(C)(C)O2 CCC1=NOC(C(=O)NCCNC(C2CCCCC2C(N2CCCC2)=O)=O)C1 C(=O)(C1c2ccccc2C(=O)N1C)N1C(C)CC(N2CCOCC2)C1 C1(C(=O)NCc2cn(C)nn2)CN(C(=O)CC2(C)CCOC2)CCO1 CN=c1cc(C(=O)NC2CC(C)(CNC(=O)Cc3cnns3)C2)cc[nH]1 c1(C=O)nc[nH]c2nccc1-2.C1(CC(=O)N)(C(F)(F)F)CNC(=O)C1.C1CC1 C1(CNC(C(NOC)=O)=O)CN(C(C2CCC(C#N)CC2)=O)C2(CCC2)C1 N1(Cc2cncc(OC)c2)CCN(C(=O)Cn2cc(-c3nn[nH]n3)cn2)CC1C C=CCC(CC)C(=O)NCC1(C)CCN(C(=O)CCc2c(C)nn(C)c2C)C1 c1(C(N2C(C)C(O)CC2)C(=O)NC(C)(C)C)ccc(F)c(Cl)c1 N1(C(c2ccc(OCCC#C)cc2)=O)CC(NC(=O)CCC#CC)CC1(C)CC c1(C(=O)NC(c2ccccc2)CNC(C(C)N(C)C)=O)cc(Cl)cc(F)c1F CC1(C)COCCC1C(=O)NCCC1CN(C(=O)CCn2ccnc2)CCCO1 CC#CC(C)(C)NC(=O)CNC(=O)CCNC(C1CCCCC1)=O c1(N(C)C)ccccc1C(=O)NCC(CO)NC(=O)CNc1ccccc1Cl C1(CNC(c2cnn[nH]2)=O)C2CN(C(c3occc3Br)=O)CC12 Cc1oc([N+](=O)[O-])cc1C(=O)NC(C)C1CC1.C1(O)(C(=O)N)CC1(C)C c1(C(=O)NC(CC2CCN(C(c3cnc(CC)o3)=O)CC2)C)cc[nH]c(=N)c1Cl C1(C(N2CCC(N(C(CCC)=O)C)C2)=O)CC2CCCCCC12 Cc1nc2c(NC(C)CCNC(c3ccc4nc(Cl)nn4c3)=O)ncnc2s1 C(CCCC(=O)NC(CCF)C(=O)NCCN1C(=O)CCC1=O)OC C1(NC(C(=O)Nc2cccc(N3CCOCC3=O)c2)=O)CC2CNC(C1)C2 c1(C(N(CCC(C)NC(C(CCCC)N(C)C)=O)C)=O)c(O)nnc2c1CCC2 c1(C(=O)NC2(CCCC(=O)NCCCCN(C)C)CCC2)cc2n(n1)CCO2 C(C)(CO)(C(=O)N1CCOC(CCNC(=O)Cc2ccccc2O)C1)NC(C)=O C(CC(C(C)C)NC(C1CN(C)CC1C)=O)NC(c1nc(CC)sc1)=O.O C(=O)(NN=c1[nH]ccnc1F)c1ccc(-c2cccc(C(C)(C)C)c2)o1 C1(O)(CNC(c2sncc2Br)=O)CC(NC(C2CCNC2=O)=O)C1 C(=O)(C(CCc1ccccn1)N1CCC(N(C)C(=O)NC2CC2)CC1)NC c1(C(N2CC(CNC(c3n(CC)cnn3)=O)C(C)CC2)=O)cc(C#N)ccc1Cl C=CCCC(CC(C)C)C(=O)NCC1CC(O)CN1C(c1cc(Cl)c(C)cn1)=O N1(c2cc(N3C4CCC3CC4)nc(COC)n2)CCC2(CCCCO2)C1 c1(NC(C(N2CC(C)C(O)C(C)C2)=O)=O)ccc(I)cc1[N+](=O)[O-] CN1CCC(C2(C(N3CC(O)(C(C)(C)C)C3)=O)CC2)CC1.c1(C=O)cc[nH]c1.N N1(C(CCOC(C)=O)=O)CC(C)OC2(CCC2)C1.c1(CC=O)ccc(Cl)nc1.N N1(C(CCCSC(C)(C)C)=O)CC(CC(N2CCN(CCO)C(=O)C2)=O)CC1(C)C CC1CN(C(C2(C3CCCO3)CC2)=O)CCC1NC(=O)CCn1cnnn1 C12(n3c(-c4cc(CC)c(Cl)cc4)nc(C(C)O)n3)CC(C3CCCC3)(C1)C2 CC1CN(C(C2(C#N)CCC2)=O)CC1C(=O)NCCC1CC2C=CC1C2 O(NC(=O)C(C1CCC1)NC(c1cc(CC)oc1C)=O)CCC#C CC(CC(=O)NCC(C)(C)OCCNC(=O)CCC1CC1)C1CCCCC1 C1(C(=O)NCCN2CC(C)OC(C)C2)CC2(CCO1)CC(F)(F)C2 N1(CC)CCCCC1C(N1CCCC(NC(c2c[nH]nc2Br)=O)C1)=O CCC(C)C(O)CC(=O)N1CCN(C2CN(C(c3ccc(O)nc3Cl)=O)C2)CC1 Cc1ccc(SCCC(=O)OCC(=O)N(c2ccccc2)C)cc1 C(=O)(CC(C)OC)N1CC(C(C(N2CC(OC)C2)=O)O)C1 C1(NC(c2c(C(C)C)scn2)=O)CCCCN(C(C2(C)CCC(F)(F)C2)=O)C1 C1(CNC(COCC=C)=O)CCN(C(=O)CC2CCCCN2C)C12CCC2 C1(OCC)CN(C(=O)CCCNC(N)=O)CC1.c1(CC=O)cccnc1Cl.C C1(NC(C(C(C)C)C)=O)CCN(C(C2CCC(N(C)C)CC2)=O)CC1C C1(CNC(C(C=C)CC)=O)CC2(CC2)CN1C(=O)C(C)=CC1CC1 CCCC(O)(CCC)CC(=O)NC(C)CC1CN(C(=O)Cn2cc(C#N)cn2)C1 C1(C(N2CC(CCNC(c3c(C)coc3)=O)OCCC2)=O)Cc2cccnc2C1 c1(C(N(CC)CC)=O)ccc2c(c1)CCCC2=O.C12(C=O)CC(C)C1C2.CO Cn1cccc1-c1cc(C(CNC(C)=O)NC(=O)COC2CCOC2)n[nH]1 N1(C(=O)NC2CCCN2Cc2ncccc2Br)CCC(C2=NOCC2)CC1 c1(C(=O)NC2C(NC(CCC(C)(C)OC)=O)CCOC2)ccc2oncc2c1 c1(C(N2CC=C(C(N3CCC(CC)OCC3)=O)C2)=O)cc2cc[nH]c2cn1 C1(NC(CCc2n(C)c(S)nn2)=O)CCN(C(=O)OC(C)(C)C)CCO1 c1(C(N(C)CCN2CCN(C(=O)C(C)(Cl)Cl)CC2)=O)nccc2nn[nH]c12 CC1CC(C2CC2)CC(C)N1C(c1c(OC(C)(C)C)sc2cccc(F)c12)=O C1(NC(C(C)n2ccnn2)=O)CC12CCN(C(=O)CC1CC(=O)NC1=O)C2 c1(C=O)csc(Cl)c1Cl.C(C(=O)NCC1CC1)OCCOCCOC N1(C(C2CCN(C(CC(C)(C)O)=O)C2)=O)CCCC(C)(O)CC1 Cn1c(C(=O)OC(C)(C)C)cnc1C=O.c1(C2C3C2CN3)ccccc1 C1(NC(C2CCCN(C(C)C)C2)=O)CCN(C(C2CC2(C)Br)=O)CC1(C)C N1(C(CCC=C=C)=O)CC2CCC2(CNC(c2cncc(CO)c2)=O)C1 Cn1cc(S(C)(=N)=O)c(CNC(C)(C#N)COc2ccc(F)cc2F)n1 Cc1csc(=O)n1CC(=O)NCC=CCNC(=O)CCC1CCCN1C c1(CNc2nc(C(=O)NC(C)CCO)n(C)c2)ccc2c(cnn2CCF)c1 c1(NC(COC(C(C)CC(N)=O)=O)=O)cc(I)cc([N+](=O)[O-])c1 N1(C(c2n[nH]c(C)c2F)=O)CCn2c(nc(C(=O)NCC3CN(C)C3)c2Cl)C1 C(=O)(CCC(=O)NCCNC(C1(c2ccc(O)cc2)CCCCC1)=O)NCC CC(CCO)C(=O)N1CCCC1CCCNC(=O)C(F)CC1CCCC1 C1(C(=O)NCCCCNC(c2ccc(SC)cc2)=O)CC2(CCCCC2)CO1 C(C(C)(C)C(=O)NC1CCCCC1CNC(=O)C(C)(O)c1ccccn1)OC N1(C(CCc2c(C)ncs2)=O)CC2(C1)CN(C(=O)C=CCO)CC2CO c1(C(C(=O)NC(C)C)N(CC(C2CCC2)OC)C)ccnc(Cl)c1Br Cc1cc(S(=O)(=O)O)c(NC(C2CC2C(=O)N)=O)cc1Cl.c1csc(Br)n1 N1(C(C(c2ccccc2)NC(=O)CC2CCOCC2)=O)CCOCC1 n1(CC)ncnc1C(=O)NCC1CCC1NC(=O)C(C)CC1CCC1 c1(C(N2CCC(C(=O)NCCc3onc(C)n3)C2)=O)c(F)cc(F)cc1F CN1C(=O)NCC1C(=O)N.C1(F)CN(C(c2ccc(CS(C)(=O)=O)o2)=O)C1 CCC(C(=O)NCCOCCNC(C1CCC1)=O)n1cnc(-c2nccs2)n1 C(=O)(C#CC1CCCO1)N(CCCOCCNC(CN(C(COC)=O)C)=O)C C12(C(N3CC(C)(OCC(=O)NCCCCCC4CC4)C3)=O)CCCCC1C2 CCCC(C(=O)OC)C(=O)N(C(C)C(=O)N(C)Cc1cncn1C)CC N1(CC(=N)NOCCC2CCCCN2)CCCC(CC(c2ccccc2)=O)C1 c1(SC)nccnc1C(N1CCC(O)(CN(C(=O)CCC2CC2(Cl)Cl)C)C1)=O C1(CC=O)CC2(C1)CN(C(=O)CP(C)(C)=O)C2.C1(C=O)CC12CCC2.CO C12CN1CCC2O.c1(C(=O)NC(CC)C(=O)O)cncc(N2CCCC2)n1 c1(CN(C(=O)CCN2CCC2)Cc2ccccc2)ccc(Cl)cc1 c1ccc(S(=O)(=O)N2CCC(CS(C)(=O)=O)C2)cc1Br.Cc1nc(CN)c(C)o1 C(C(C)CC(=O)N1CC(=C(F)CNC(c2[nH]nnc2C2CC2)=O)C1)OC Cn1ncc2c(C(N3CC(NCc4ccc(I)o4)C4(CC4)C3)=O)cccc12 c1(N(C)CC2C(C)C2)ccc(S(=O)(=O)N2CCC(C)(F)CC2)c(Br)c1 Cc1ccc(I)c(C(N2CCCCC2CNC(c2sc(Cl)nc2C)=O)=O)c1 C12CCCN(C1)c1ccc(cn1)C(=O)N2.Cc1cc(C(C)NC2CCCC2)on1 N1(C(C(=O)NCC2CC2)C2C(CC)C2)CCCC1C.C(C)(C)C.C=O.C c1(C(N2C(CNC(c3c(CC)occ3)=O)CCCC2)=O)cc(C)c(N)cc1Cl CC1CCN(C(C2CC(C)(C)CO2)=O)C(CNC(c2c(Br)nnn2C)=O)C1 c1(C(=O)Nc2ccccc2C(=O)O)cc2[nH]c(=O)ccn2n1.CCSCC.O c1(OC)ccc(-c2ncc(-n3c(-c4cc(C=C)[nH]n4)ncc3)s2)c(C)c1.C(F)(F)F Cc1cc(C(=O)NCC(C2CC2)NC(=O)CC(C)c2ccccc2)c(Cl)cc1N c1(OC)cccc(C(C(=O)N(CC(C)CNC(c2c[nH]c(Br)c2)=O)C)OC)c1 N1(C(C2CC(C)OCC2)=O)CC(C2CN(C(=O)C3=CCCC3(C)C)C2)C1 N1(C(C)=O)CCC2(CCN(C(=O)CC3CNC(=O)C3)CC2)C1.C(=O)OCC.N c1(C2C(C(N3C(CCNC(CC(C)(C)C)=O)CCC3)=O)C2)ccc(C#N)cc1 N=c1ccc(C=CC(=O)NCC(O)CNC(=O)CCn2cncn2)c[nH]1 C(C(=O)N1CCC(N(CCOc2ccccc2OC)C)CC1)(C(C)C)OC C1(NC(Cc2c(C)cc(Cl)nc2)=O)CCC2CCN(C(=O)CC3CCCO3)C12 c1(CCC(=O)N(CCC)CC)ccccc1C.C(=O)(C(C)Cc1cnn(C)c1)N C1(CC(=O)NCCN(C(C2C(CC)C2)=O)C)CC2CCC1O2 c1(CN(C(=O)C=Cc2ccnn2C)C)ccccc1.C(=O)C(C#N)C1CC1.C C=CC(CCC)CC(=O)N1CC(C(=O)NC(C)Cc2nncn2C)CC(C)(C)C1 Cc1ccncc1C(=O)NCC(CC(C)C)NC(=O)CN1C(C)CCC1C c1(N2CC(OCCNC(C(CC)c3ccccc3)=O)C2)nc(O)c2c[nH]nc2n1 C=C1Cn2c(C(N3CC(NC(=O)C(C)(CC)C(F)F)C4(CC4)C3)=O)nnc2S1 N1(C(C2CCCN(C(C)=O)C2)=O)CCC(NC(=O)C=CCN(C)C)C(F)C1 C1(CC)(CC)CC(NC(=O)CCc2ccon2)CN1C(=O)COC(C)C N1(C(Cc2ccc(C)c(O)c2)=O)CCC2(C1)CN(C(=O)CC1CCOC1)C2 C=CCC(CC(C)C)C(=O)NCC1CC(C)(C)CN1C(=O)C(O)CN(C)C c1(OC)cc(Br)cn2ncc(C(=O)NC3COCCC3=O)c12 CC1(CO)CCCN(C(C2CCN(C(=O)CN3CCCCC3)CC2O)=O)C1 C1(NC(C(C)(C)OC)=O)CC2CC(C1)CN(C(C1CC(C)N(C)C1)=O)C2 N1(C(C(CCSC)N(C)C)=O)CC2OCC(NC(=O)Cc3ccsc3)C2C1 N1(C(C2(SC)CC2)=O)CCn2nccc2C1.c1(C(NC)=O)ocnc1C1CC1.C c1(OC)cscc1C(=O)Nc1nc(C)no1 C1(O)(C(=O)NC(C)C=CC(=O)NCCN(C)C)CCSCC1 CCCCCC(F)C(=O)NCC1CCC1NC(C1(C(=O)N(C)C)CC1)=O C1(CNC(C(C)SC(F)(F)F)=O)CN(C(=O)C(c2ccccc2)F)CCN1C C(=O)(C1=CCCC1)N(CC=CC(=O)N(C(C)CS(C)=O)C)C C1(C(N(C)CC2N(C(C(CCSC)OC)=O)CC(F)C2)=O)CCn2nnnc2C1 C#CCC(CC#C)C(=O)NC1CC2CC(C1)N(C(=O)CCc1ccncc1)C2 O=C1CC(CC(=O)N2CCC(NC(=O)C(C3(O)CCCCC3)(F)F)C(F)C2)=NN1 c1(N2CC(N)C2)n[nH]cc1-c1nc(C2CC=CCC2)no1 C12(NC(C3CCCN(C)C3)=O)CC(C)(C1)OC21CN(C(=O)CCn2ccnn2)C1 N1(C(CCc2cnc(C)s2)=O)C2CCC1(CNC(=O)CC1CCC(=O)N1C)CC2 N1(C(C2(CC)CC2)=O)CCC(CCCNC(C2CCC(OC)C2)=O)CC1 C(=O)(C(CO)C(F)(F)F)NCC1CC(C)N(C(=O)C(C)C2(O)CCC2)CC1 CC1CC2CCC(C(=O)NCC3(CO)CCCOC3)CN2C1 C(C)(C)(CC(=O)N(CCNC(C1CCCN(C(C)C)C1)=O)C1CC1)SC C1(C(=O)NCCCN(C(C(C=C)(C)C)=O)C)CCc2nnc(C(C)(C)C)n2C1 CCC(CC)C(F)C(=O)NC(COC(C)C)C(=O)NCCOCCN=[N+]=[N-] CCC(CC(=O)NC1(C(=O)NCC(C)CN(C)C)CC(CO)C1)C(F)F C#Cc1ccc(C(=O)NC2(CN(C)C(c3ccc4scnc4c3)=O)CC2)cc1Cl C1(NC(C2N(CC)CCC2)=O)CN(C(c2ccccc2C(N)=O)=O)CC1OC Cc1cc([N+](=O)[O-])cc(C(=O)NC(C)CCCCNC(C2(C#N)CCCO2)=O)n1 c1(-c2c(OC)ncc(C)c2)nc2c(s1)CC(C(=O)NCC(C)(C)C(N)=O)CC2 c1(OC)cc2c(cc1NC(=O)C(=O)Nc1cnc3c(c1)COCC3)OC(C)C2 C1(C(=O)NCCNC(c2c[nH]cc2C(F)(F)F)=O)(CC)CCOCC1 S(=O)(=O)(c1cc(-c2cccc([N+](=O)[O-])c2)c(C)cc1C)N(C(CC)C)C c1(C(N2CC(O)(CNC(C(CCC)C)=O)C2)=O)cc2scc(C)c2[nH]1 C1(NC(c2ccc(Cl)c(C(F)F)c2)=O)CCCCCC1.c1(C(=O)N)cnc(O)o1 c1(CC=O)ccc(S(N)(=O)=O)cc1.CC(C)CCCNC(C1CCC2CC12)=O C#CCC(CCOC)NC(C1(COC)CCCN1C(=O)CC)=O.C(N)(=O)N CC(C)(C)C(C(=O)NC1CN(C(C2COC2)=O)C(C)(C)C1)N1CCCC1=O C#CCC(CC(F)F)C(=O)NCCCN(C)C(C1CCCN(C(=O)N(C)C)C1)=O C1(NC(CC(=C)C)=O)CN(C(c2cccnc2NC(C)C)=O)CCC1(C)C C1(N(c2cccc(C#C)c2)C(=O)CC)CCC2(CC1)CNCCO2 CC(C)CC(C(=O)NC1COCC1CN(C)C)N(C(=O)CC(C)(C)C)C C(=O)(C(CCC(C)C)NC(=O)CCn1ccnc1)N(CCOC)CCO C(=O)(C(CC1CCCC1)NC(C12CCN(C1)C2)=O)N1CC(N(CC=C)C)C1 C1(C(=O)OC)Cc2ccccc2CN1N1CCN(C)C(=O)C12CC2 CC1CN(C(=O)Cn2cncn2)CC1CNC(=O)Cc1ccon1 C=CCCCCCC(=O)N1CCN(C(c2cc3cccnc3[nH]2)=O)C(CCC)C1 c1(CC)ccc(C(C)C=O)cc1.N1(CC(=O)N(CCC)C)CCCS1(=O)=O.N c1(CC)ccc(CNC(c2nnnn2CC)C2CC(CC(C)(C)C)C2)o1 c1(C(N2CCCC(c3n[nH]cc3C(N)=O)C2)C(=O)N)cncc(F)c1.C(C)SC N1(C(c2c(C)cc[nH]2)=O)CC(C2CN(C(C3CC3C)=O)C2)C1 N1(C(c2nc(CCC)sc2)=O)CC(NC(C2(OC)CCSCC2)=O)C(C)C1 N1(C(C(C)OCCC=C)=O)CCN(C(=O)CCCOC2CC2)C(CC(C)C)C1 c1(Cc2nc(-c3cc(C)c(C)o3)on2)ccnc(Cl)c1C C(CC(C)CC)(C(=O)N1CCC=C(Cl)C1)NC(CC=CCCCCC)=O c1(OC)cnc[nH]c1=NCCC1C(C)CCCN1C(=O)CCC(C)OC Cc1nc2ccccn2c1C(N1CCCN(C(C2(C)CCCC2C)=O)CCC1)=O c1(C(N2CC(CNC(c3c(C)cc(F)cn3)=O)C2)=O)cc2ccc(Cl)c(F)c2[nH]1 c1(CC)c(C(=O)NCCCN2CCN(CCC3CC3(Cl)Cl)CC2)cnn1C C1(CNC(c2c(Cl)cn(C)n2)=O)CN(C(C2CCS2(=O)=O)=O)CC12CC2 c1(CCC(=O)OCC#CCOC)ccccc1-n1cc(CCO)nn1 Cc1oc(C#N)cc1C(=O)NCC1(O)CN(C(C2CC2C(F)F)=O)C1 c1(NC(CC(C2CC2)NC(C(C=C)C)=O)=O)ccc(C)nc1OC C1(N(C)C(=O)NC2CCN(CC(F)(F)F)C2=O)CCN2CCC1C2 C1(NC(c2c(C)scc2)=O)CC2CC(C1)N(c1snc(Cl)c1C#N)C2 C1(CNC(C(C)O)=O)COCC2(CCN(C(c3ccnc(S)c3)=O)CC2)O1 c1(OC)cc(NC(=O)NCC(F)C(C)(C)O)ccc1Cl C(CCCCCN=[N+]=[N-])NC(C1C2(CCN(C(C3C(OC)(OC)CC3)=O)C2)C1)=O C1(C(=O)NCCN(CCCC)C)CCCN(C(C2CCC(C(=O)O)CC2)=O)CC1 CC1CCN(C(=O)CNc2ccccc2Cl)CCN1C(=O)Cc1ccc(F)cc1 N1(C(C(C)SC(F)(F)F)=O)CCN(CCNC(C2CN(CCF)C2)=O)CC1 N1(C(C(c2ccccc2)=O)=O)C2CCC(C2)C1CNC(c1cscn1)=O c1(C(=O)NC(C(C)NC(C23CC=CC(C2)OC3)=O)(C)C)ccc2ncnn2c1 C1(NC(c2cc(C(N)=O)oc2)=O)CCC2(CCN(C(N)=O)C2)C1 C1(NC(C2C(C(C)C)N(C(c3ccoc3)=O)CC2)=O)CCCCCCC1 C12(CCNC(c3nccc(F)c3Cl)=O)CCC1CN(C(c1ccoc1)=O)C2 C1(CCC)CN(C(c2nn(C)cc2Cl)=O)CC1NC(C1(C)CCCOC1)=O C(=O)(CC(O)CNC(=O)CC(=O)N(C)C)NCc1cn(CCC)nn1 c1(C(=O)NCC2N(C(C(C=C=C)C)=O)C3C(C2)C3)ccc(C(C)C)cc1F C1(NC(=O)CO)CC(NC(c2c(Br)noc2C2CC2)=O)C12CCC2 c1(C(N2CCN(C3C(NC(CSC)=O)COC3)CC2)=O)cc2cnccc2[nH]1 c1(C(N(C2CCN(C(CSC(C)=O)=O)CC2)C)=O)ccc(Br)c(F)c1C Cc1cnc(C#N)c(NC(C2CC2C(N2CC3CC(C2)O3)=O)=O)c1 O=C(C1CNCc2n[nH]cc21)N1CC2C(C1)C2(F)F C1(C(N(C)Cc2scc(C)n2)=O)CCCCN1C(=O)Cc1cc[nH]c1 C1(C2CCCN(C(=O)CCCCCO)C2)(NC(c2ccc(C)cn2)=O)CC1 N1(C(C(CCC)C#N)=O)CC(NC(=O)COc2ccsn2)CC12CCC2 CC(C)C(F)(F)CCn1cc(C2CCCN2C(=O)C(F)(F)c2ccccn2)nn1 N1(C(CC2CCC(=O)C2)=O)CCC2CCN(C(c3cn(C(F)F)cn3)=O)CC2C1 c1(NC(c2cc[n+]([O-])cc2)=O)ccc2c(c1)CN(Cc1c(Cl)ccc(F)c1F)C2 Cc1ccc(C(=O)N(CC(N2CC(C)CCC2C)=O)CC2CC2)c(C)c1 C1(NC(c2nnc(C)s2)=O)CN(C(=O)CCNS(C)(=O)=O)CCC1(C)C c1(C(=O)NC(CC(C)NC(CCn2ncc(C)c2)=O)C)c(C(C)C)n[nH]c1C C1(C(=O)N(C2CC3CNC2C3)CCO)CCC2CCC(=O)N2C1 C1(NC(CC(=O)NC)=O)CCN(CCNC(=O)CCCOCCOC)CC1 CCC1c2ccccc2CCN1C(C(=O)NCCOC)c1ncco1 C(C)(CO)(C(=O)NCc1cn(CC(N2CCCC(O)C2)=O)nn1)OC C#Cc1ccc(C2CCCCN2C(=O)Cc2ccc(C3CC3)cc2)cc1 c1(CC)cc(C(=O)NC(C)CC2CN(C(c3c[nH]nc3C)=O)C2)ccc1Br c1(OCC)c(C(N2CCCC(NC(=O)C=CC=C(Cl)Cl)CC2)=O)cccc1F CCC(C(C)Cc1ccccc1)NC(=O)N(C1CCCCC1)CCC#N C=CC(CC)CC(=O)NCCC(C)N(C)C(c1ccc(Cl)c(N)c1)=O CC1(CO)CCN(C(c2cc(F)n[nH]2)=O)CC1.c12cncc(c1)NC2=O.C1CCC1 N1(C(c2cccn3nccc23)=O)CC2CCCC(C1)N2C(=O)CC(F)(F)Cl C1(N2CC(NC(c3cccc4ccoc34)=O)C(O)CC2)CC2CCCC(C1)N2 N1(CCNC(C2C(C)CC2C)=O)CCCN(C(=O)CC2OCCCO2)CC1 c1(NC(C2(NC(CCC(C)C)=O)CCN(C)C2)=O)ccc(OCF)c(F)c1 Cc1cc(S(C)(=N)=O)cnc1N1CCCC(C(F)(F)F)C1C C1(CCCC(=O)NCCCNC(C(C)CC2CCCO2)=O)SCC2NC(=O)NC12 Cc1nc(CC(=O)NC2CCCC2NC(=O)CSc2ccncc2)cs1 N1(CC(=O)Nc2ccc(NC(C)=O)cn2)CCC2(CCN(C)CC2)C(CO)C1 C(C(O)CC(F)(F)F)NC(c1c(CNC(C(CSC)O)=O)ccs1)=O C1(C(=O)NC(C=C)(C)C)CCC(O)CN1C(=O)Cn1cnnn1 C(CC(CNC(=O)CNC(C)=O)NC(=O)Cc1cncnc1)OC c1(-c2cn(CCCCNC(c3ccc(C)cn3)=O)nn2)cc(Cl)c(C#N)c(Cl)c1 c1(C(=O)NC2C(NC(C=C(CC)C)=O)CCCC2)ccc(F)c(CC)c1 c1(OCC)ccc(C)nc1C(=O)NCCC(C)C(C)C.c1(C=O)n[nH]cc1F.N N1(C(C2(C=C)CCCC2)=O)CCCCCC(NC(=O)C(C)c2cc[nH]n2)C1 c1(N(C(C)=O)CC)ccc(C(=O)NCCCC(C)(C)OC)cc1 c1(CC(=O)N(CCCNC(C2CCC(C)S2)=O)C)c[nH]c2cc(F)ccc12 CN(CC1CCOCC1)N1CCC12CCC(C)(C)CC2 CC1CC(C)(C(=O)NCc2ccnc(C(=O)NC3CCCC3C#N)c2)CCO1 C1(C(=O)NC(c2nc(CC)[nH]n2)C)C=CCCN1C(=O)CP(C)(C)=O C1(F)(CNC(c2sccc2-n2cccc2)=O)CCC1.C1(C(=O)N)CCCOC1 N1(C(c2c(C)oc(CNC(=O)C)n2)=O)CCN(C)CC1C(C)C.CCC(C)C CC1CCCN(C(C2C(C)OC(C)C2C)=O)C1CNC(c1cccc(Cl)c1F)=O c1(NC(C(N2CCS(=O)CCC2C)C(CC)C)=O)cccc([N+](=O)[O-])c1 C1(C=O)CCC2(CC1)CC2(F)F.c1(COC)ccsc1C(=O)NCCC(O)C CC1C2CC(C2NC(C2CCCCN2C)=O)N1C(c1ccc(N)cc1O)=O C1(CNC(COCCCOC)=O)CCC(NC(=O)COC2CC2)CC1 C1(NC(c2c(C)cc(C)[nH]2)=O)COC2C(NC(c3oncc3C)=O)COC12 N1(C(C2N(C(C(C=C)O)=O)C3CCC2C3)=O)CC2OCC(F)(F)C2C1 Cc1nc(CNC(c2occc2CNC(=O)CC2OCCCO2)=O)sc1C c1(OC)ccc(Cl)c(-c2cn(Cc3cccc(OCC(C)(C)C)c3)nn2)c1N c1ccn2c(C)cnc2c1.C1(N(CCNC(C(CNCC)C)=O)C)CCCCCC1 N1(C(C2CC(C)(CC)OCC2)=O)CC2(CCC(NC(=O)C3=NOCC3)CC2)C1 N1(C(=O)OC(C)(C)C)CCN(C)C(C(=O)NC(C(CO)C2CC2)C2CC2)C1 CC1(CCN(C2CC2)CC2CC2c2cccs2)CCN1 c1(NC(C2=CCCN(Cc3c(O)ccc(C)c3)C2)=O)ccnc2c1CCO2 CCC(C)(C(=O)NCC1(C)CCN(C(C2(O)COC2)=O)CC1)C(F)F Cc1cc(=N)[nH]cc1C(=O)NCC1CN(C(=O)CCCCC)CCO1.C(N)(=O)N c1(OC)ccc(CC(N2CC(NC(=O)C(Cl)=CCl)C(F)C2)=O)c(Cl)c1OC C1(n2cc(C(C)(C)NC(C)C)nn2)CCCN(C(=O)CC(C)c2ccco2)CC1 CC1(C)CC(C(N2CCC(O)C(C)(O)C2)=O)CN(C(C2(C#N)CC2)=O)C1 c1(N)ncc(Cl)c(C)c1C#N.c1(SCC)ccccc1C(=O)NCC1CCC1 N1(C(c2ccc(OCC#C)cc2)C(=O)NCCCOC)CCC(O)C(F)C1 C1(NC(CC)=O)CCCN(N2CCCC(c3cc(OC)n(C)n3)C2)C1 c1(CC(=O)NCC2C3CN(C(c4c(C#N)ccs4)=O)CC32)cc(F)ccc1F C=C(C)CC(C)C(=O)N1CCC(CN(C(=O)C(C)(C)CC2CCOCC2)C)CC1 CC1(C(N2CCC(O)(CCNC(=O)CCc3ncccn3)C2)=O)CCNC1=O C#CC1(NCc2c(C)cccc2C)CCCOC1 c1(C(=O)NCC(CNC(=O)CC(=O)NC2CC2)F)cccnc1.C1CC1.N N1(C(C2(CC)COC2)=O)CC(CC(=O)NCc2ncc(C)o2)C2(CC2)C1 c1(C(N(CC(CC)NC(c2ccc(OC)c(C)c2)=O)C)=O)ccc(OC)nc1F N1(C(C2OCCN(S(C)(=O)=O)C2)=O)CCC2(CC1)C(=O)Nc1ccccc12 N1(C(C(CC)(C)O)=O)CCC(NC(c2cccc3nccn23)=O)CC(C)(C)C1 C=C(C)c1cccc(NC(=O)C(C)C(C)NC(=O)CCNC(=O)OC)c1 c1(CNC(=O)C=O)ccc(C)cc1.c1(C(=O)OC)sc(C(=O)OC)nc1C c1(NC(C)=O)cccc(F)c1C(=O)NC1CCCCN(Cc2c(C)nsc2N)C1 CCC(C(=O)NCC1(CC(=O)NC(C2CCOCC2)C)CC1)SC Cc1cc(C(N2CC(CCNC(c3scnc3Cl)=O)OC(C)C2)=O)cc(C)c1O Cc1ccc(C=CCC(=O)NC23CCN(C(=O)Cn4cccc4)CC2C3)cc1 c1(C(=O)NC(C)(CNC(C2CC(CF)C2)=O)C2CCC2)cc2cccnc2s1 N1(c2ccnc3ccc(C)cc32)CCC2(CNc3ccccc32)C1 C1CC(C)(C)CCO1.CCC(C)(C)OCC(N1CC(C(C(=O)NC)OC)C1)=O c1(CN(C)C(C2C=CCN2C(c2nonc2N)=O)=O)ccnc(O)c1 Cc1cc(Cl)cc(C(=O)NCC(CNC(=O)CS)CO)c1C.c1ccccc1.C N1(C(C2CN(C)C2)=O)CCC(NC(C2CC(C(C)(C)C)=NO2)=O)C2(CCC2)C1 N1(c2nc(C)cc(SC)n2)CCC2C1CCCN2C(c1cc2sccc2[nH]1)=O C1(C(N(CC(CNC(C2N(S(CC)(=O)=O)CCC2)=O)O)C)=O)CCCCCCC1 c1(N2CCC(N(C(=O)C(C)SC)CCCC)CC2)ncnc2c1CCC2 C(CCO)(C(F)F)N(C)C(C1C(C)CN1C(=O)CCCCC1CC1)=O C(=O)(CC=C(Cl)Cl)N1CC(CCNC(=O)CC(=O)NC2CC2)(OC)C1 Cc1ccc(F)c(N)c1C(N1CC2C(NC(C3CCC(C)(C)CC3)=O)C2C1)=O C1(NC(C(=O)NCCOC)=O)COCCC1.c1(C=O)ccc(CC#N)cc1.N C1(CC)CCN(C(=O)CC2(C)CC(F)(F)C2)C1C.C1(CC=O)CSCCO1 CC1(NC(=O)C(C)(C)c2ccccn2)CC(NC(=O)CC2CCCOC2)C1 c1(C(=O)NC(C)CC(C)NC(=O)CC2COCCOC2)ccc2nc[nH]c2c1 S(=O)(=O)(c1cc(C(F)(F)F)ccc1N)NCC1CC(C)C1.C1(C)CC1.C C1(CNC(=O)Nc2c(OC)ccc(C(C)(C)C)c2)COc2cscc2O1 c1(NC(CC)C2CCC2)nc(N2CCCC(CSCC)C2)nc2c1ncn2CC CC(CCC(C)(C)C)C(=O)NC1CC(CNC(=O)CC(O)C2CCCC2)C1 C(=O)(CCCN=c1nccc[nH]1)NCCC(C)NC(C(CC=C)(C)CC)=O C1(CN(C)C(C2(c3ccccc3)CC2)=O)CCN(C(=O)CCc2ccc[nH]2)C1 c1(OC)cc(C(N2CCOCC(NC(c3coc(Cl)n3)=O)C2)=O)ccc1[N+](=O)[O-] C#CCCCCC(=O)NCC1(NC(=O)C(c2c(F)cccc2F)C)CCOCC1 C1(C(N(C)C(c2cccs2)=O)=O)CC2CCC(C1)N2C(C1CCCO1)=O C(C(C(=O)NC1COC(C(C)C)C1)C(C)C)NC(C1CC(OC)(OC)C1)=O C1(N(C)C(C2CCOCC2)=O)CN(C(C2(S(N)(=O)=O)CC2)=O)CC1O c1(C(N2CCC(CNC(C(C=C)CC)=O)C2)=O)cc(F)cc(C)c1N c1(OC)ncccc1C(=O)NC1CCCN(C(C2(C3CC3)CC2)=O)C1 CC1OC2CCC1(NC(C1COCC1NC(=O)COC(N)=O)=O)C2 N1(C(C(CCOC)C)=O)CCN(C(=O)CCn2cnccc2=O)C(CCOC)C1 c1(C(=O)NCCCN(CC(CC)CC)C)cc(C(C)=O)cn1C Cc1ccc(O)c(C(=O)N(C(C)CNC(=O)C(c2nc(F)ccc2Cl)C)C)c1 C12(C(=O)NCC(CCC)C)CC(CN(C(=O)CCNC(=O)OC)C1)C2 C#CCC(C)(C(=O)N1CCC(C)(C#N)C1)NC(=O)COCC(F)F Cc1ncc(Cl)c(C(=O)N(CC(C)NC(=O)CCCc2ccc(F)cc2)C)n1 N1(C(C(C(=O)O)(C)C)=O)CCC(N=[N+]=[N-])C1.N1(CC=O)CCCC1.CC(C)C c1(CC)cccc(C(=O)NCC(O)CCNC(=O)C(=O)N(C)C)c1C N1(C(C(C)c2cc[nH]n2)=O)CCCC(O)(CCNC(c2cc(C#N)n(C)n2)=O)C1 CCCCC(CNC(=O)CCOC1CC1)NC(=O)C(c1ccccn1)(F)F.O C1(Sc2ccc(SC(C)(C)C)cn2)CCCN(c2ccc(Cl)c(Cl)c2)C1=O N1(Cc2cccc(C(=O)NCCO)c2)CCS(=O)(=O)CC1.C(=O)C1CC1.N C1(OC)CN(C(=O)Cc2ccccc2Br)CC1NC(=O)C(C)C(C)O CC12CC(C1)C(C(=O)NCCC1COCCN1C(c1cccnc1)=O)CO2 c1(C(=O)NCCCCCNC(C(C(=C)C)(C)O)=O)cc(C)cc(Br)c1F CCCC(C)(C)C(=O)NC1CN(C(C2(c3ccc(Cl)c(Cl)c3)CCC2)=O)C1 O=[N+]([O-])c1cccc(C(C2CCOC2)NC2CCC2)c1 c1(C(=O)NC(CCCNC(C2CCN(CC#C)CC2)=O)C)cccc(C#N)c1C N1(C(c2ccc(-n3cc(CCCCC)nn3)cc2)=O)CCS(=O)(=O)C(CO)C1 N1(C(CCC=C)=O)CC(CNC(=O)C2=CCN=[SH]2)C(C2CC2)C1.c1ccncc1.C c1(N2CCN(C(=O)NCC)CC2)nc(=NCCOC2CCC2)[nH]c2c1SCC2 CC1(C)CC(CC(=O)NC2CCC(NC(c3ccc(C#N)[nH]3)=O)CC2)CO1 CC1ON=C(C(=O)N2CCC(C3CC3)(CNC(=O)CCN3CCCCC3)C2)C1C c1(C(C)C)ccccc1C(=O)N.C1CC(C(F)(F)F)CN1C(=O)CCS(C)=O.C C(=O)(CCC(C)(C)NC(C1CCC(F)CC1)=O)NC(CCC)C1CCC1 c1(NS(CC)(=O)=O)ccc(COc2c(C)cccc2C)cc1F C1COCCN(C(=O)C=CC(=O)N(C)C)C1.Cc1cc(C(F)F)n(CC=O)n1.N Cc1scc(C(=O)Nc2c[nH]nc2C(=O)Nc2ccc(-c3nn[nH]n3)cc2)c1C C(=O)(CCC1=CCCCC1)N(CC(C)CNC(c1nnc(S)n1C)=O)C c1(CN(C2CN(C(c3ccc(C)c(O)c3)=O)C2)C)ccc(Br)c(Cl)c1Cl N1(C(C(CCC)C)=O)CCCC(NC(c2cnn(CCOC)c2)=O)CC1 CC(C)C(C(=O)NCCN(C)C(C1CCC(C(C)C)CC1)=O)c1ccn(C)n1 c1(CC(=O)NCC2(NC(C3CCCCO3)=O)CCOCC2)ccc2[nH]ccc2c1 C1(NC(c2cc(C(C)=O)sc2)=O)C2CC1N(C(C1C3CCOCC13)=O)C2 C(=O)(CC(C)C(C)(C)C)N1CCN(C(c2cc(C(=O)OC)sn2)=O)CC1C C1(C(=O)NCC(C)O)(CC)CCCCN1 C12(CNC(=NCC)NCC3CCSC(C)C3)CCC(CC1)OC2 c1(CC)nnc2n1CCCC2C(=O)NC1(C)CCCN(C(c2csc(O)n2)=O)C1 C(=O)(C(C)(O)C1CC1)NCCC(C)N(C(CSC)=O)C CC1(O)CN(C(=O)CONC(c2ccc3c(c2)CCC3)=O)CCC1O C1(CNC(C(CC2CCCC2)OC)=O)CCN(C(c2sc(F)cc2Cl)=O)CC1 Cc1cc(N(C)CCc2ccccc2F)ncc1S(=O)(=O)N(CC(C)(C)CO)C n1(CC)cnc(C(=O)NCC2CC2NC(c2cnnn2CC)=O)c1 c1(C=O)cc(C)c(Br)o1.C1(C(N(C(C)C)CC)=O)CCN(C(=O)NC)C1 CC1CC(NC(=O)CCC(C)c2ccccc2)CCN1C(=O)CC1CC(O)C1(C)C CC1(c2noc(C3CCC3)n2)CS(=O)(=O)C1 CC1(C)CN(C(=O)CC2(C)CCC2)CC1C(=O)NCCO.C1CCOC1.C C(CN=c1ccnc(N2CCc3nc(O)[nH]c3C2)[nH]1)OCCC(C)C N1(C(=O)OC)CCCC(C(=O)NCC2CCCC2)C1.c1(C=O)oc(C)cc1C c1(NC(=O)CC2CC(NCc3cc(Br)ncc3Br)C2)ccc2ccnc(O)c2c1 c1(C(=O)NCc2cn(CCCC(=O)NC)nn2)ccc(CC)cc1.C(=O)CC C1(C(N2C(C(N3CCC3)=O)CCC2)=O)C2CC1N(C(=O)C=Cc1ccco1)C2 N1(C(C(C)C)=O)CC2CCCC(CNC(c3cc(Cl)n(C)n3)=O)C2C1 Cc1cc(-c2ccc(C(=O)NC3CCCN(C)C3)cc2)c(F)c(C)c1 C(CNC(C1(CO)CCCCO1)=O)(CC(=O)N1CCCC(CF)C1)OC Cc1scc(C(=O)N(C2CCN(C(=O)C(Cc3ccccc3)N(C)C)C2)C)c1N c1(C(C)C)c(C(N2CCCCC2CNC(c2cncs2)=O)=O)cnn1C CN=c1[nH]cc(C(N2CCC(C(C)C(=O)N(CC(C)C)CCN(C)C)CC2)=O)o1 Cc1cc(C(=O)NC2CCN(C(=O)C(C)(O)C(C)C)C2)c2sc(=N)[nH]c2n1 C(C)(C)(CCC)NC(CCNC(=O)NC)=O.c1(C(C=O)O)ccc(Cl)cc1.N C=CC1OCCCC1C(=O)NCC(C)(C)CNC(C1(C2CC2)CC=CC1)=O c1(C(CC)O)nc(-c2ccc(N3CCCCC3=O)cc2)n(CC2CCOC2)n1 c1(C(N2CC(F)CC(NC(c3ccc(OC)cn3)=O)C2)=O)ccc(Cl)c(F)c1O c1(CN2C(C(=O)NCCC3CCCC3)CC(F)C2)ccc(Br)c(F)c1 C(=O)(CC(O)C(C)C)NC1CCCC(NC(c2c(C)[nH]nc2Cl)=O)C1 c1(-n2c(N(CCC(=O)NO)C(c3cccc(C)c3)=O)nnn2)ccc(F)cc1Br c1(C=O)cc(=O)cc(Cl)[nH]1.c1(C(NC(C)C)=O)cccc(CS(C)=O)c1.C C1(CC)C(NC(c2nn(C)cc2Cl)=O)CCCN1C(=O)CC1CCCC(O)C1 c1(OC)ccc(C)cc1-n1ccc(CNc2cccc(Oc3ccccn3)c2)n1 c1(C=O)cnc(O)c(F)c1.c1(CN(C)C)ccc(C(N2CCC2)=O)o1.C(C)O n1(-c2cc(C)on2)c(C)cc(C(=O)NOCc2nnnn2CCC2CC2)c1C N1(C(COCC#C)=O)CCN(C(=O)CCOc2cccc(C)c2C)CC1CO C1(C(N(CC(C)N(C(=O)Cc2cccc(Cl)c2F)C)C)=O)CC12CC(F)(F)C2 C1(CNC(c2c(COC)cc[nH]2)=O)CCC(C)N(C(=O)C2=CCOCC2)C1 C(=O)C(O)C(C)(C)C.C=C(C)CCNC(C1(C)CC(C(F)(F)F)C1)=O.N c1(C(C(=O)NCC2CC2)N(C(C(C)C)C)C)coc(-c2cc[nH]n2)c1 c1(C(=O)NC(CNC(CCCOCCOCC)=O)C2CC2)cnccc1Cl c1(C(=O)NCCN(C(C2(COC)CC=CC2)=O)C)nnc(O)cc1C c1(C(=O)NCCC2CCCN(C(C(CC#C)C)=O)C2)n[nH]c2c1CS(=O)(=O)CC2 C1(NC(COCC)=O)CC2(CCCN(C(=O)CN(c3ccccc3)C)C2)C1 C1(CNC(c2c(OC)ccs2)=O)CCN(C(=O)CC2CC(C3CC3)C2)CC1C C1(CC(=O)NC(C)CC2CCN(C(=O)Cc3cn[nH]c3)CC2)CCCCNC1=O N1(c2nccc(=NCc3nnc(C)s3)[nH]2)CCN2C(CCS2(=O)=O)C1 C(=O)(N(CCO)OC)C1(CC=C)CN(C(=O)C2=COCCC2)C1 Cc1nc(C(N2CC(N(C(=O)CC3CC(N(C)C)C3)C)C(O)C2)=O)cc(O)n1 CC(C)(C)C(O)c1cn(CC2CC(NC(=O)CCn3cc(Cl)cn3)C2)nn1 Cc1ccc(S(=O)(=O)N2CCC3(CCN(C(=O)C(C)(CO)CO)C3)C2)cn1 C1(C(=O)NC2C3(CN(C(C4(C)CCC4)=O)C3)SCC2)CC2CCC(C1)S2(=O)=O C(=O)(CN=c1[nH]c2c(c(=NCCSC(C)C)[nH]1)SCC2)NCCC C1(C(N(CCC)C2CC2)=O)CN2CCCN1CC2.C(C)C=O.C(C)OCC.O c1(N2CCC(CC)C2)nc(N(C)Cc2cccc(Cl)c2Cl)c2ncn(CC)c2n1 c1(C(N2CC3C(NC(CCCN(C)C)=O)(C3)C2)=O)c(Cl)c2ccccc2n1C C(CCC(=O)N1CC(O)(CCNC(c2ccnn2CC#N)=O)C1)=CC c1(C(N2CC(C)C(NC(=O)Cc3nc(=N)[nH][nH]3)CC2)=O)[nH]nc2ncnc(O)c12 N1(C(c2c(C)cc[nH]2)=O)CCC(C2CCN(C(c3ccc(CC4CC4)s3)=O)C2)C1 C1(C)(CNC(C2N(C(CCC)=O)CSC2)=O)CCN(C(C2CN(C)C2)=O)CC1 c1(OCCOC)cc2[nH]c(=NCc3cnn(C)c3OC)cc(I)c2cc1OC Cc1ccc(S(=O)(=O)NCC(=O)N(CCC(O)CO)C)cc1 CN1CC(C)(C)CC1C(N1CCCC(N(C)C(c2ccc(F)cc2N)=O)CC1)=O C(C)(C(=O)N1CC(CNC(=O)CCC2CC2(C)C)C1)SCCCC c1ccc(Cl)cc1.CC(C)(CNC(C1(CC2CC2)CCC1)=O)C.C(=O)C Cc1[nH]nc(C(C)C)c1C(=O)NC1CCCCC1N(C)C(C1CC1(C)C)=O c1(OC)cc(C)nc(N2CCC(NC(=O)Cc3noc(C4CC4)n3)C(F)C2)n1 N1(C(c2ccc(CC)nc2C)=O)CCCC12CCN(C(c1ccncc1N)=O)C2 N1(C(c2ncn(CC)n2)=O)CCCC1C=CC(=O)NC(C(F)(F)F)C1CC1 C1(CC(=O)NCCC2(C)CCOC2)CN(C(C2(F)CCOCC2)=O)CCO1 c1(OCC)cc(F)ccc1CN1CCC(CNC=O)CC1.C(C)(C)C.O CC1(C)C(NC(=O)C=C2CCCC2)C2CCCN(c3cc(Cl)ncn3)C12 C1(NC(CCOCCN(C)C)=O)CCSC12CN(C(c1cccc(F)n1)=O)C2 c1(NC(C2CCCN(C(c3ccc(CCC)cc3)C)C2)=O)c(C)cc(Cl)cc1Cl C=C1CC(C(=O)NCCCCN(C)CC)N(C(c2cnc(C3CC3)s2)=O)C1.O N1(c2c(C)c(NCc3nn(C)cc3C(F)F)ncn2)CC2CCCCCC2C1 N1(C(c2cc(C)no2)=O)CCC(CC(C)NC(c2coc(C(F)(F)F)c2)=O)CC1 c1(-c2cn(CC(C)C)nc2)nc(Cc2ccccc2)nn1CC1CCCO1 N1(C(C(C)NC(=O)NC)=O)CCC(C(=O)NOC2CCC2)C12CCC2 Nc1ccc(C(=O)NC2CCCN(C(=O)C=Cc3ccco3)C2)nc1Cl c1(NC(=O)NCC(CCCC=C)(C)C)sc2c(c1C(N)=O)CCCC2 C1(NC(c2c(CC)c[nH]n2)=O)CCC2(CC1)CN(C(c1coc(C)n1)=O)C2 c1(-c2ccc(C=O)[nH]2)nc(-c2ccccn2)nn1CC1CCC1 c1(OC)cccc2c1C(C(=O)N(C)CCNC(=O)CCC1CCCN1C)CC2=O CCC(CNC(=O)C(C)(CC)CC)N=c1nc[nH]c2[nH]c(Cl)cc12 c1nc(C)cc(C)n1.C(=O)(C(C)C(=O)NC1CCCC1NC(=O)C)OC.S c1(C(CC)=O)ccc(N2CC(CNC(c3ccccn3)C)CC2=O)cc1.C(C)(C)O C(C1C(C(=O)NCCC2CCCN2C(C2CNC(=O)N2)=O)C1(C)C)=C(C)C C1(CC(=O)NCC2CCCCC2NC(=O)Cn2ncnn2)CCC(F)(F)CC1 N1(C(CNC(CNC(C)=O)=O)=O)C2CCCC1CCC2.C(=O)C#CC(C)(C)O.N c1(CC)cc(C(N2CCC(C(N3CCC(CCCO)C3)=O)(CC)C2)=O)c(C)o1 C1(CNC(C(C)O)=O)CN(C(c2nc(Br)c[nH]2)=O)CC1(F)F c1(OCC(=O)NCC(CNC(CCNC(C)=O)=O)C)cccc(F)c1F c1(C=O)ccc(S(C)(=O)=O)cc1.CC1(C)CCCN1C(C1CCCC2(CC2)C1)=O C1(C(=O)NCCC=CCCC)(CC)CCCN1C(=O)CC1CCOC1 N1(C(C(CC)(C)C)=O)CC2CCCC2(NC(=O)CN2CC=CC2)C1 C1CN(C(C2(F)CCCC2)=O)C2(CCOCC2)C1.C1(C(=O)N)CC2C(C1)C2(F)F c1(NCCN2CC(=O)NCC2)nc2cccnc2c(=NCC2CC23CC3(F)F)[nH]1 CCCCC(O)C(=O)N1CCN(C(=O)Cc2cn(C)nc2C)CC1CCC C(C)(C(C(=O)N(CC(C)C(=O)N(CCCCN(C)C)C)C)N(C)C)OC C=CC1CN(C(=O)C(S(C)(=O)=O)C2CC2)CC1NC(c1ncccn1)=O CCS(=O)CC(=O)N1CC(CC(F)C(=O)NC2CCC3CCC23)C1 c1(C(N(C(C)C)CCNC(=O)CC2CCCCC2F)=O)ccc2nc(O)[nH]c2c1 Cc1ccc2cc(C(N3CC(NC(C4(F)C5CCCC45)=O)C3)=O)[nH]c2c1 C=C1CC(C)(C(=O)NC2CC(CNC(=O)C(N3CCNC3=O)C)C2)C1 CN=c1nc(N2CCc3nc(N4CCOCC4)ncc3C2)[nH]c(=NCC(F)F)[nH]1 c1(CC)cc(C(=O)NCc2ccccc2)nn1C.C1(C(NC)=O)CNC(=O)N1 c1(C=O)cccc(F)c1.C1(C(=O)OC(C)(C)C)CCC1C(=O)N.C1CCC1 Cn1cnn(CC(N2CCC(C3CCCN3C(c3cncc(Cl)c3)=O)C2)=O)c1=O Cc1nn(C2CC2)c(Cl)c1C(=O)NCCN(C)C(c1cc(C#N)c[nH]1)=O C1(C(N2CC(C(N)=O)C2)=O)CCC(C)CC1.N1(CCC)CCCC1C(=O)N.C C1(C(=O)NCC2(OC)CN(C(=O)CC3CCCCN3C)C2)CC2C=CC1C2 c1(CC)cc(O)ccc1NC(C1CCN(C(C2CC=CC2)=O)CCO1)=O N1(C(CC2(OC)CCC2)=O)CCCC(C(=O)NCCCN(C)C)C1 c1(C(N2CCCC(NC(C3C4CCCC34)=O)CC2)=O)n[nH]c2c1CCSC2 N1(C(=O)C=CC#N)CC(C2CCCN(C(c3cc[n+]([O-])cc3)=O)C2)C1 C(C(N=c1cc(Cl)nc(C2CC2)[nH]1)C1CC1)NC(Cc1ccn(C)n1)=O C1CC(F)CN1C(=O)CCc1ccc(C)cn1.C(CC=O)NC(=O)OCC.N C(=O)(CS(=O)(=O)C(C)C)N.N1(CC(N2CCCC2)=O)C(=O)CCC1=O.CC c1(C(=O)NCCSCc2cn(CCSc3cnn[nH]3)nn2)csc(Br)c1Cl c1(C(N2C(C)CCN(C(=O)Cn3cccn3)CC2)=O)cc(N)c2ccccc2n1 CC1(C)C(CNC(c2ccc(N)c(F)c2)=O)CCN1C(C1CC1C1CCC1)=O C1(NC(Cc2ccn(C)n2)=O)CCc2onc(C(=O)N=c3cc[nH]cc3)c2C1 C1(C(C)C)C(C(=O)NCc2ncc(Cl)cn2)CCN1C(=O)C(N)=O C1(C(=O)NC(C(=O)OC)CCF)CN(C(C2CC(NC)C2)=O)C(C)(C)C1.C CC1c2cc(F)cc(F)c2CCN1N1CCN(Cc2ccsc2)CC1 C1(NC(C(Cn2ccnn2)NC(CCC)=O)=O)COCC(C)(C)C1 c1(C(C)C)ccc(OCC(=O)NC2CC2)cc1.C(=O)CS(=O)(=O)N(C)C.C c1(CCC(N2CCC(NC(CCNC(C)=O)=O)C2(C)C)=O)cccc([N+](=O)[O-])c1 Cn1ccc(NC(=O)C(=O)NCc2ccccc2OC2CCCC2)cc1=O c1(C(=O)NC2C3CC2CN(C(C2CC24CC4(F)F)=O)C3)ccc2ncsc2c1 N1(C(c2c(C(C)C)ccs2)=O)CCN(C(=O)CC2CCCC(O)C2)C2(CCC2)C1 Cn1cc(C(=O)C(=O)NC(Cc2ccco2)C(=O)NCCC(F)(F)Cl)cn1 C(=O)(CCCCC(=O)NC(C(=O)N(C1CCSC1)C)C(C)O)OC c1(NC(C2CCN(C(c3cn[nH]c3)=O)C2)C)ncnc2c(Cl)cc(Cl)cc12 C1(C(N2CCC(CC3CC3)CC2)C(=O)NC(CC)(C)C)CCc2ccccc2C1 C1(NC(=O)CCCCC(F)F)CCCC12CCN(C(=O)CN1CCCC1)CC2 C1(CCC)CN(C(=O)C2=CCOC2)CCN1C(c1cn(-c2ncccn2)cn1)=O N1(C(C=CC)=O)CC2CCN(C(=O)CCNC(=O)OCC)C(C2)C1 c1(CC(C(=O)NCC(CO)NC(CC(=O)OC)=O)C)ccccc1C CCC(C)(C)C(O)C(=O)N(CCCOCCNC(C1CCC(O)CN1C)=O)C c1(OC)cccc(C(=O)NC2CC2NC(C2(C)CC=CCC2)=O)c1C C1(C(N2CCC(c3ncc[nH]3)C2)=O)(CC)CCN(c2nncs2)C1 c1(N2CCN(C(c3c(C)c(Cl)ccn3)=O)CC2)nsc2ccccc12 CC1CN2CCN1CC2C(=O)NC1(CF)CCN(C(c2cccnc2Cl)=O)C1 C(=O)(C1=CC2(CCOC2)C1)NC1CCN(C(c2cncc(C=C)c2)=O)C1 N1(C(C2CC(C(C)C)C2)=O)CCC(NC(=O)C(c2cccnc2)N(C)C)C1 C1(CC(N2CCC(NC(C(C=C)(C)CC)=O)C2)=O)CCC2(CC1)COC2 Cc1cc(=NCCC2=CCC3CC2C3(C)C)[nH]c(N2CC=C(Br)CC2)n1 c1(C(N2CC(NC(CC(C)C)=O)C(O)C2)=O)cccc2ncccc12 C1(C2(O)CCN(C(C3(Cl)CC3)=O)CC2)(NC(CCc2n(C)ncc2)=O)CC1 C1(NC(C(C)CSCc2ccccc2)=O)CCC(F)(C)C1.C1(C=O)CCC1 CCC(N=c1[nH]c(=NC)[nH]c(=NC(C)c2ncc(C)cn2)[nH]1)C1CCC1 C1(NC(c2c(C(N)=O)nccn2)=O)CC2CC1CN2C(=O)Cc1cccs1 C12(NC(Cn3ncc(C)c3)=O)CCC(CC1NC(=O)CCc1cccnc1C)C2 CC(CCCCNC(=O)C=Cc1ccccn1)NC(c1nn[nH]c1Cl)=O C1(C(=O)Nc2ccc(C)c(C#N)c2)Cc2nccnc2CN1C(=O)C(O)C(C)C C(=O)(C(c1ccccc1)=CC(C)(C)C)NC.C1CCN(C(=O)C=CS(C)=O)CC1.C CC1CC(N(C)C)CN(N2CCC(C(N3CCCCCC3)=O)C(O)CC2)C1 c1(CN=C(NCC(NOCC)=O)NC(C)C2CC2)ncc(F)cc1F C1(C)(CC)C=C(C(=O)N2CC(F)(C(=O)NCC(F)(F)C(=O)OC)C2)C1 N1(Cc2c(C)nc(C)s2)CCCCCC(N)C1 CCC(C)(C(=O)NCC1C=CCN1C(=O)CCCSc1ccc(Cl)cc1)OC C1(C(N2C(CNC(C(CC)n3cccn3)=O)CC(O)C2)=O)CC2(C1)CC(O)C2 CC1CC2CN(C(C3CCN(C)CC3)=O)CC2N1C(=O)CC1CC2CC2C1 c1(NC(C(C)C2CCC2)=O)c(F)cc(C(F)(F)F)cc1F c1(C(N(CCCCN(C(C(C(C=C)C)C)=O)C)C)=O)cc(C#N)ccc1F CC1CN(C(C2(C)CN(C=O)C2)=O)C(C)(C)C1.c1ccc(F)cc1.C(C)(C)C c1(CNC(c2cc(Br)c3nccn3c2)=O)cc2n(n1)CCN(C(=O)C1CC1)C2 CC(C)CC(C(=O)NCc1ncc(CO)[nH]1)ONC(=O)CCC1CC(C)C1 C1(NC(C(CC)=CC)=O)CC2CCC1N(C(=O)CC)C2.c1cc(Cl)cc(Cl)c1.O C1(NC(C=CCC)=O)CN(C(C2CCCOC2)=O)CCC1(C)C C1(NC(CN(C(COC)=O)C)=O)CCCC1C.C1(C)(C(=O)N)CC(C)C1 c1(C(=O)N)cnc(N(C)C)nc1.N1(C(C2C(CCOC)C2)=O)CCCC1C N1(C(Cc2ccc(CC)cc2)=O)CCC(CNC(c2ccoc2Br)=O)C12CC2 Cn1ccc(CCC(=O)NC2CC2CNC(C2(n3cncn3)CC2)=O)n1 CC(C)(CF)C(=O)NC1CC1NC(c1ccccc1-c1cn[nH]c1)=O C(C)(CCC(=O)NC1CCN(C(=O)Cc2csc(C(C)C)n2)CC1)OCC.C c1(N2C3CC(NC(c4cc(CC)[nH]n4)=O)CC2CC3)[nH]cnc2nc(Cl)cc1-2 c1(NC(c2n(CC)nnn2)(C)CC2CCOCC2)ccc2c(Cl)n[nH]c2c1 Cc1ccc(N)c(C(=O)NC2CN(C(=O)C(c3ccccc3)O)CCC2CO)c1 C1(C)(C(=O)NC(COC)C)CCCN(C(c2sc(Br)cc2Br)=O)C1 C1(CN=[N+]=[N-])(N(C2C3(CC(C)(C)C3)C2)C2CC2)CCC(F)(F)CC1 C1(CN(C(c2oncc2C)=O)CC)CCCN1C(c1ccn(COC)n1)=O C1(CCN(C(=O)CN2CCNC(=O)C2)C)CCN(C(=O)C)CC1.c1cn[nH]c1.S N1(C(CCCCCCSC)=O)CCCC2CN(C(C3CC(=O)N(C)C3)=O)CCC12 Cc1cncn1CC(=O)NC(C1CCCCC1)CNC(=O)C.C1(C)CCCC1.O C#CC1(C(=O)NCCc2cocn2)CCN(C(c2csc(Cl)n2)=O)C1 C=CC(C)CC(=O)N(C)CCNC(c1c[nH]c(C(N2CCCC2)=O)c1)=O N1(Cc2cc(C)n(C)n2)CC2(CC(C(=O)Nc3cc(Cl)cc(Cl)n3)C2)C1 C(=O)(C(CC#C)NC(=O)C(C)Cn1cccn1)N1CCC(OCC#C)C1 CCCCCCC(=O)N1CCCC(CCCCNC(=O)Cc2ncc(C)[nH]2)C1 C1(N=c2ccc(C#N)c(C)[nH]2)(CCNC(C(C(C)C)SC)=O)CCC1 C1(NC(CC(C)O)=O)CCN(C(c2cc[nH]c2)=O)C12CCC2 Cc1cnc(C(=O)NC2CCC23CN(C(c2cc(C(C)C)on2)=O)C3)c(Br)c1 c1(C(C)C(N2CC=CC(NC(C34CCC(C3)C4)=O)C2)=O)ccc(C#N)cc1 Cc1nn2c(c1C(=O)N)CCCC2.C1(CC)CN(C(=O)C(=O)N(C)C)CC(C)O1 c1(-c2scc(C=O)c2)ccc(Cl)cc1.C(=O)(CC(=O)NC1CC(O)C1)OC.C C1(NC(C2(CC)COC2)=O)C2CCC(C2)C1C(=O)N.C(C(C)C)C1CC1 C1(NC(C(CCC)c2ccccc2)=O)CCN(C(=O)CN(C)C)CCC1(F)F C1(C=O)CSCCS1.C1(CC(=O)N2CC(=C(F)C)C2)CC(F)(F)C1.CCO Cc1c(Br)cnc(O)c1C(N1CC2(CNC(=O)C(N)=O)CCC1CC2)=O S(=O)(=O)(c1ccc2sccc2c1)NC(C(=O)O)(C(F)(F)F)c1cccc(Cl)c1 c1(OCC(c2ccc(C)cc2)n2nnnc2C2C3COCC23)ccc(Cl)c(C#N)c1 C1(NC2CC(OC)CN(C(=O)OC(C)(C)C)C2)COc2ccccc2C1 CC1CN(C(=O)NC2CCN(C3CCCCC3)CC2)CC(C)S1(=O)=O c1(C(=O)NC2CC(CNC(C(CC#C)C3CC3)=O)C(O)C2)ccc(C)nc1C C(=O)(C1CCc2snnc21)N1CC2(CCOC2)C1.C1(C(=O)N)(CSC)CC1.C N1(C(CCc2nc(=N)[nH][nH]2)=O)CC(NC(=O)C=Cc2ccoc2)C(O)C1 c1(COC)nc(C)cc(=NCC2CN(C(c3ccc(CSC)cc3)=O)C2)[nH]1 C1(C(N2C(CNC(c3ccc(C)cc3F)=O)CC(O)C2)=O)CCOCC12CCC2 Cc1ocnc1CC(=O)NCCCC1(C)CCCC1.C(=O)CN(C)C1CC1.N C1(NC(c2c(C)nn(-c3ccccc3)c2)=O)CCN(C(C2COC2)=O)CC1C Cc1nc(C)c(CNN2CCN(C(=O)CSc3ccccc3)C3CC23)nc1C c1(C(N(CC(C)C)C)=O)cc(F)n(C)n1.c1(C(=O)N)cnnn1-c1ccccc1 C(C1(C)CCOCC1)=CC(N1CC(CC)OCC1)=O.c1(CC)ncc(C(=O)N)[nH]1 C#CC1(C(=O)NCC(C)(C)C(=O)NC2(C3CCCCO3)CC2)CCCCC1 Cn1ccc(C(N2CC(NC(c3cnc(O)[nH]3)=O)C2)=O)c1 C1(CC)(CCl)CCN(C=O)CC1.C1(CC#C)CCCC1NC(C)(C)C c1(N2CC(OC)(CNC(=O)CC3CC3C)C2)nc2ncc(Cl)cc2o1 C1(F)(C(=O)NCCc2cccs2)CCN(Cc2ccc(O)c(Cl)c2)CC1 C=CCC(CNC(C1C2CC3C(C2)C13)=O)C(=O)NC(C)(C)CC(N)=O c1(C(N2CCN(C(C(C)(C)O)=O)CC2C#N)=O)cnc2ccc(C(F)(F)F)cn12 C(C)(C(=O)N)(C(C)C)NC(C)=O.c1(C2C(C=O)C2)ccsc1.C1CC1.C Cc1cc(N)c(C(N2CCN(C(C3CCC(C)CC3)=O)C(C(C)C)C2)=O)cc1C c1(C(=O)NC(CNC(COC(CC)C)=O)C2CC2)cn(C)nc1SC C=CC(C)(C)CC(=O)NCC1CC1CNC(=O)Cc1ccc(O)cn1 Cc1cc(=NCc2ccc3c(c2)OCO3)[nH]c(N(CCC(C)O)C)n1 C1(C(=O)NC(CC)CN(C)C)CC=CCN1C(=O)CC1CCC=CCC1 c1(C(=O)NCC2OCCN(C(c3cc(N)c(Cl)nc3)=O)C2)cccc2c[nH]nc12 c1(C(NCCNC(C(CC)F)=O)=O)coc(S(=O)(=O)N(C)C)c1.C1CC1 Cc1cccc(CC(=O)NC2CCCC(NC(=O)C(C3CCCCC3)O)C2)c1O C1(c2nnnn2C2(C)CC2)(NCCOCC=C)CCCCC1F C1(C(N2C(CC=C)(C(=O)NC3CCN(C)CC3C)CCC2)=O)CCC=CCCC1 C#CCC(CC#C)NC(=O)C(C1CC1)N(C)C(C1CCC(O)C1)=O c1(C(=O)NCC2CCC(F)(CNC(C)=O)C2)ccc(C(F)F)cc1Cl C(=O)(C1Cc2ccc(C)cc21)N1CC(N(C(c2cccc(CCC)c2)=O)C)C1 C1(N(C(C(C)Cc2ccc(F)cc2)=O)c2nn[nH]n2)CCn2cnnc2C1 Cc1cc(Br)cc(CN=C(NCC2CNC(=O)C2)NCC(F)F)c1F N1(C(C2(CC=C)CC2)=O)CC2(CCC(NC(=O)C)CC2)C1.c1ccccc1Cl.O N1(C(c2c(C)cc(C(F)F)o2)=O)CCC2(CCN(Cc3nnc(C(C)C)o3)C2)C1 S(=O)(=O)(c1ccc(C#N)cc1C(F)(F)F)N1CCCC(n2ccc(C)n2)C1 CCCCC(O)CC(=O)N1CC(CNC(=O)CCCCNC(N)=O)C(O)C1 Nc1c(C(N2CCC(CCNC(=O)Cc3nccs3)CC2)=O)cccc1F Cc1cnc2c(C(N3CC(CNC(C4CCC(=O)N4C)=O)C(C)C3)=O)cnn2c1 C1(NC(CCCC#C)=O)CCN(C(c2ccc(F)c(CC)c2)=O)CCC1CO C12(NC(C3CCSCC3)=O)CCCC1N(C(c1ccc(Cl)c(Cl)c1O)=O)CC2 N1(C(=O)Nc2ncccc2Br)CC2CCCC1(NC(=O)C(F)(F)F)C2 N1(C(CC=CC=C)=O)CCC2(CC1)CCN(C(=O)CCc1ccncc1)CC2 Cc1cc(C(=O)NCC(C)C(=O)NCC2CN3CCC2C3)cc(O)c1 C1(c2nnnn2CCOC)(Nc2ccc(C#C)c(OC)c2)CCN2CCCCC2C1 C1(N(C(Cn2c(C)cnc2)=O)C)CCN(C(=O)CCc2ccsc2Cl)CC1C N1(C(C(n2c(C)cc(C)n2)C)=O)CCN(C(=O)CS(=O)(=O)CCO)CC2(CC2)C1 c1(C(=O)NC2CCC(N(C(C=CC=CC)=O)C)C2)ccc(C(N)=O)cc1 C(C(C)CC(C)C)NC(CCN(C(C)=O)C)=O.C1(C(=O)N)CC1C(C)(C)C Cc1ccc(Cl)cc1C(=O)NCC(O)CNC(=O)C(O)c1ccsc1 N1(C(C2C(C=C)CC2)=O)CCN(C(=O)CCOC)C(c2ccccc2OC)C1 CCC(C(=O)NCC1CCN1C(c1ccnn1C1CC1)=O)c1ccccc1 N1(C(C2C(C)(C=O)C2)=O)CC(O)(CC)C1.C1(CC=O)CCCO1.CC.O C12(C=O)CCC(C(F)F)(CO1)C2.n1(CCC)cc(C(=O)NCCC(O)C)nn1 C1(CC#C)CC2(CCN(C(=O)C(=O)NCCc3cccc4nc(C)sc34)C2)CO1 Cc1ncc(Br)cc1C(=O)NC1CC(NC(=O)Cc2cc(Br)ccc2Cl)C1 CCCCCCCCC(C)C(=O)N1CCC2CN(C(=O)CC3OCCO3)CC2C1 N1(C(C)=O)CCC(O)(C(C)C)C1.C(=O)(CC)N.C(C)(C)C.C=O.CC(F)F c1(C(N2CCC3C2C3)=O)cnc(O)c2ccccc12.C1(C(=O)N)(COC)CC1 N1(C(C2CC(C)OC2)=O)CCC(n2cnnc2O)CC1 c1(-n2c(C(COC)(C3CC3)NC3CCC(F)CC3)nnn2)cccc(Cl)c1C c1(OC)c(C)csc1C=O.c1(C(C(=O)NCC)C)ccc(C)s1.C1CC1.N C1(NC(c2cn(CCCC)nn2)=O)CCCN(C(C23CCCC2(C(N)=O)C3)=O)C1 c1(C(N(C2CN(C(Cc3cc(C)[nH]n3)=O)CC2O)C)=O)cn2c(n1)CCC2 N1(C(C(C)c2ccsc2)=O)CC2CCN(C(=O)Cn3cccnc3=O)CC2C1 C(=O)(C(F)CC1CN(C(=O)C(C)OCOC)C1)N1CC(C(C)OC)C1 C1(CNC(C(CC)(F)F)=O)CN2CCCCC2CN1C(c1coc(C)c1)=O C(C)(CNC(C12CC(C1)OC2C)=O)(CC(C)C)NC(c1c(C)nc[nH]1)=O.C c1(C(N2CCN(C(C34CCC(C)(CC3)OC4)=O)CC2)=O)cc2c(O)ccc(F)c2[nH]1 C1(N(C(C=CSC)=O)C)CCCN(C(=O)Cc2ccn(-c3ccccc3)n2)C1 n1(C(C(=O)OC)C)ccc(CC2(c3ncco3)CC2)n1 c1(C(N2CCC(N(C(=O)CC(C)n3ccnc3)CC)C2)=O)cnc2scc(C)n12 Cc1cc2nc(C(=O)NC(C)CNC(=O)C(N3CCC(C)CC3)=O)cn2cc1C N1(C(C2(N(C(C3=C(C)OCC3)=O)C)CC2)=O)CCc2nncn2CC1 C1(NC(c2cc(F)c[nH]2)=O)CC2CC(C1)N(C(C1(CO)CC1)=O)C2 C#Cc1cc(C(=O)NC(CCN(C(=O)C(C)CF)C)C(C)C)cc(Br)c1 CC1(C)CC(C(=O)NCC(F)CNC(c2ccc(O)c(Cl)n2)=O)CNC1=O Cc1cncc(C(=O)NCC2(O)CCN(C(c3csc(C#N)c3)=O)C2)c1Cl Cc1c(C(c2nnnn2Cc2cccs2)NCc2cnc(C3CC3)o2)cnn1C C1(CC(=O)Nc2c(C)ccnc2Br)C2CCC1CN(C(=O)CCc1cccs1)C2 C(=O)(C1CCc2cccnc21)NCC1C(NC(c2nc(C)oc2C)=O)CC1 CC(C)C#CC(=O)NCCC(C)NC(C1CC(N2CC(O)C2)C1)=O c1(CCC(N2CC(CC)C2)=O)nnc(S)n1C.C1(=CC=O)CCC(C)C1.CO C1(C(N2CCC(C(=O)NC(C)C(=O)OC)C2)=O)(COC)CCCO1 C(=O)(C(C(=O)NCC(O)CNC(c1nn[nH]c1Cl)=O)c1ccccc1)OCC N1(C(=O)OCC)CCCC1C(=O)NC1CN(C(=O)Cc2ccn[nH]2)C1.C N1(C(c2n(COC)ncc2)=O)CCC(C)(C)C(C(=O)N(C(CCO)C(F)F)C)C1 Cc1ncc(CC(=O)NCCC2CC(C(=O)NCCc3ccnn3C)C2)o1 CCC(C(=O)NCCC(C)N(C)C(c1n[nH]c(C)c1Cl)=O)C(C)(C)CC C1(CC(=O)N)COCC(C)O1.C12(C)CC(C1)C(=O)N2.C1(CCOC)CC1 CCCCCCC(=O)NC1CC2(C1)CC2NC(c1ccn(C2CC2(F)F)n1)=O C1(C(N(C2CCCN(C(C(C)(F)F)=O)C2)CCO)=O)CCc2n[nH]cc2C1 S(=O)(=O)(c1ccc([N+](=O)[O-])c(F)c1)N1CCC(C(N2CCS(=O)CC2)=O)C1 n1(CCCC)nc(C(=O)N)ccc1=O.C1(C=O)C(F)(F)C12CC2.CCC1CC1 CC(C)C(O)C(C)C(=O)N1CCC2(CC1)CC2NC(c1csnn1)=O CC1=CC(C)CN(C(=O)C(CC(F)F)NC(=O)COC2CCCCC2)C1 O=C(C1=NOCC1)NCC(N1CCN(C(c2c[nH]nc2C2CCCO2)=O)CC1)=O N1(C(c2cccc(-c3nc(C)[nH]n3)c2)=O)CCC(O)C(C)(C)C1 C12(CNC(CC)CN(C)C)CCCCC1C2 C1(C(=O)NC(C#C)C)CC12CC(NC(C1(COC)CCCC1)=O)C2 Cc1[nH]nc2ncc(C(=O)NC3CCCC3NC(C34CCCN(CC3)C4)=O)cc12 C12(C(N3C(CCNC(=O)C4=CCOCC4)CCCC3)=O)C3C4C1C1C2C3C41C C(=O)(C(C)(O)C(F)(F)F)N1CCC(NC(c2c(CC=C)cccc2)=O)C1 N1(C(c2cn(C)c(O)n2)=O)CCC(C(=O)OC(C)(C)C)C(O)C1 O(NC(=O)C(CNC(=O)C(C)n1cccc1)CC1CCCC1)C(C)C c1ccc(Cl)c([N+](=O)[O-])c1.C(=O)(CCCNC(C1CCCN1)=O)OC(C)(C)C CC1(C)CN(C(=O)C(F)CC2CN(C(=O)CC3NC(=O)NC3=O)C2)CCCO1 c1(C(=O)NC2CCC(N(C(=O)CSC(F)(F)F)C)C2)ccc(CO)s1 Cc1ccc(N(C2CC3CC2CN3)C(=O)C(C)Cc2ccco2)cn1 C1(CC(=O)OC)CN(N2CCCC2c2cccc(C)n2)CC1CSC c1(C(=O)NCC(C=C)O)cc(CNC(C2SCC=C2C)=O)[nH]n1 N(C(=NCCCCl)N1CCC2(CNC(=O)C2)C1)CC1(C)CCCCCC1 N1(C(C=C(CCC)C)=O)CCC(CNC(c2cc(C3CC3)on2)=O)(OC)C1 c1(NC(C2C(C=CC)CNC2)=O)cc(F)c(C(=O)OCC)c(Cl)c1 c1(C(=O)CCOC(=O)C(c2ccc(Br)cc2)(F)F)ccc2c(c1)OCCO2 C(=O)(CCCN=[N+]=[N-])N1C(CNC(c2ccn(CCCC)n2)=O)CCC1 CCCC(CCC)C(=O)NCc1csc(C(=O)N(C(c2cccnc2)CC)C)c1 c1(C(=O)NC(C(C)NC(C(C)Oc2ccccc2Cl)=O)(C)C)cncc(C#N)c1 N1(C(=O)CC2CC2)CC(C2CCN(C(c3ccc(CO)c(F)c3)=O)CC2)C1 C1(C(=O)OCC)CCN(C(c2cccnc2Br)=O)C(C2CC2)C1 c1(C(N(C2CCN(C(c3c(CC)nn[nH]3)=O)CC2C)C)=O)ccc(C)c(C)c1F N#Cc1cc(C(N2CCC(C(F)CNC(C3CCC4(CC4)C3)=O)CC2)=O)co1 C(=O)(C(CNC(C1CCCSC1C)=O)CCC)NC(C=C)COC Cc1ccc(C(N2CCC(NC(c3ccnnc3O)=O)C(O)C2)=O)cc1O c1(OC)cc(Br)ccc1CCC(=O)NC1CCC(C)(C(=O)O)CC1 C=CC(O)C(=O)NCC(C1CCCC1)NC(=O)C(CC)n1cncn1 N1(C(C(C=C)OC)=O)CCC(NC(c2occc2CC)=O)C1C(C)C c1(OC)ccccc1CC(=O)NCC(C)CNC(C1(C(C)(C)O)CCC1)=O CC1(C(=O)NCc2nc(-c3ccccc3)no2)CC(N)CCO1 c1(C(N2CCN(CC3(NC(C(CC)C)=O)CC3)CC2)=O)cc([N+](=O)[O-])c[nH]1 N1(C(COCCNC(C(C=C)(C)O)=O)=O)CCC(C#CC)C1 N1(C(CC2(C)CC2(Cl)Cl)=O)CC(NC(c2ccc(C3COC3)cc2)=O)C2(CC2)C1 c1(CC(N2CC(OCC(N)=O)C2)=O)cccc(C(F)(F)F)c1Cl C1CN(C(=O)C=CC2CC2)CC2CCCC12.c1(OC)cccc(OC)c1C(=O)N c1(C(=O)NCC2(O)CC(NC(CC(C(C)C)C)=O)C2)cc(Cl)cc2ccncc12 Cc1cccc(C=O)c1.C1(N(C(CC)=O)C)C2CN(C(C34CC(C3)C4)=O)CC12 CC(C)(C(=O)NCC(C1CCOC1)NC(=O)Cc1cnoc1)C1CCCC1 C(=O)(C(C)(C)CC1CC1)NC(C1CCCN(C(=O)CCCc2nncn2C)C1)C C1(NC(=O)CCN2CCCC2)COC2(CCN(C(c3cnc(CBr)s3)=O)CC2)C1 Cc1ccc(Cl)cc1C(N1CCC(C)(CN2CCCC2)CC1)C(=O)NCC(F)F Cc1cc(F)cnc1C(N1CC(NC(c2ccccc2CC(C)C)=O)C2CC12)=O N1(C(CNC(=O)OCC)=O)CC(NC(C2C3CCCC23)=O)CC(F)(F)C1 N1(C(C#C)=O)CC(C2CCN(C(c3ccccc3N3CCCCC3)=O)CC2)C1 S(=O)(=O)(c1ccc(F)c(Cl)c1)N1C(C(=O)O)CCCC1.C12CN(CCC1O)C2=O C=CC(C)(C)CC(=O)N1CCCCC1C(C)(C)CNC(=O)CCS.C1CCCC1 c1(C(=O)NCC2N(C(CC(C=C)CC)=O)CCCC2)cnn2c1NCC(C)C2 C1(CCC)CN(C(C2(C(=O)OC)CC2)=O)CCN1C(=O)CCC1CC1C c1(C(C)NC(C(C)N(C(=O)CCC2CC2C)CC)=O)cccc(F)c1 Cc1cc(=NCc2csc(C3CC3)n2)[nH]c(=NCC2(F)CC2)[nH]1 CC1CCC(=CC(=O)NCCC(C)(C)NC(=O)CNS(C)(=O)=O)C1 N1(C(C(C)c2cc[nH]n2)=O)CCCC(n2cc(CNS(C)(=O)=O)nn2)C1 C1(NC(CCSC)=O)CC2(C1)CC(CNC(=O)C(C1CCCCC1)C)C2 C(N=c1nc(O)c2c(ncn2C)[nH]1)C1CN(C(c2c(C)cco2)=O)C1 c1(OC)cc2c(cc1C(=O)NC1CN(C(=O)CCSC)C(C)(C)C1)CCC2 C(=O)(C1=CCC2(COC2)OC1)N.c1(SC(C(=O)NCCCC)C)ccc(F)cc1 Cc1ccccc1C=CC(=O)NC12CC(NC(c3cnc(S)nc3)=O)(C1)C2 C(C)(CC(=O)N1CC(CCNC(=O)CC(C)n2ccnc2)C1)SC CC1C(NC(c2ccc(=O)n(C)n2)=O)CCCN1C(=O)Cn1cccnc1=O C1(C(=O)NCC2CCC(C)(C)O2)CC12CCN(C(=O)CCS(C)(=O)=O)CC2 N1(C(c2c(C(C)C)nco2)=O)CC(C)CC(C)C1.C(=O)(C(C)CC1CCCC1)N N1(C(c2n(CC)c(O)nc2)=O)CCCC2(CCN(C(C3(CO)CC3(F)F)=O)C2)C1 c1(C(=O)NC2C(NC(C=Cc3c(C)ccs3)=O)CCOC2)ncc(N)cc1Cl C1(NCc2c(C)nc(C(C)C)cc2)CCC(O)C(C)(C)C1 CC1CCN(C(=O)C#CC2CC2)CC1N(C)C(c1cnc(C(F)F)s1)=O N1(C(CCNC(COC)=O)=O)CCN(C(=O)C(F)=C2CCC2)C(C(C)C)C1 Cc1ccc(CC(CC2CCC2)CO)cc1.C1(=O)CC(C)Cc2ccccc2N1 C1(NC(=O)Cc2ccc(O)cc2)CCC12CCN(C(=O)Cc1cc[nH]n1)CC2 c1(C(N2CC(CCOC)N(C(C3CC3C)=O)CC2)=O)cn2c(C)cccc2n1 CC(O)CC(=O)NC(C)C(C)(C)NC(=O)CC1CC=CCC1 c1(SC)nccc(=NC2CC(C)N(C(=O)C(C(C)C)C3CCC3)C2)[nH]1 N1(C(C2N(CC)CCOC2)=O)CCN(C(=O)CC(=O)N(C)C)CC1CF N1(C(C2(CC(C)C)CC2)=O)C(C(=O)N(CCCc2ccco2)C)CC1C C=CCC(CNC(=O)C(C)(C)N=[N+]=[N-])C(=O)NC(C)COCCOC C12(NC(=O)C=Cc3ccccn3)CCOCC1CN(C(C1(C3CC3)CCC1)=O)C2 c1(C=O)cnc(C(F)(F)F)c(Cl)c1.Cc1cc[nH]c1C(=O)NC1CC1C.N N1(C(=O)Cc2cccc(F)c2)CCc2[nH]nc(-c3ccc([N+](=O)[O-])cc3)c2C1 N1(C(Cc2c(C)cccc2F)=O)CCC2(NC(=O)C=Cc3ccco3)CCCC12 C(=O)(N1CC(O)C(O)CO1)C1(C(C)C)CCCN1C(C1CC1(F)F)=O c1(OC)cccc(CCC(=O)NCC(O)CNC(c2cnn[nH]2)=O)n1 C1(CC(=O)NCC2(C(N3CC(c4nc(=O)o[nH]4)C3)=O)CCC2)CCCCO1 N1(C(c2c(C(C)C)cco2)=O)CCC(NC(=O)CCc2ccc(N)cn2)CC1 N1(C(C2CC3(CC(C)C3)C2)=O)CC(N=[N+]=[N-])CC1C(N1CCCCC1)=O CC1(C)CCCN(C(C2OC(C)(C)OC2(C)C)=O)C1.C1(C2CCC2)(C(=O)N)CC1 C1(NC(C(C2CC2)OCC)=O)(C)CCCCCC1.C1(C=O)CCCC(C)C1.N c1(OC)cc(C(=O)NC2CCN(C(=O)C(O)CC(N)=O)C(C)C2)cc(OC)c1C C1(NC(C2N(S(C)(=O)=O)CCC2)=O)CC2CC1N(C(c1cc(Cl)ccc1O)=O)C2 CCN=C(NCC1(OC)CCOC1)NC1CCc2sc(Cl)cc21 c1(C(N2CCC(C(C)(C)NC(c3c(C)scc3)=O)C2)=O)ncncc1F O=C(C1=CCCC1)NCc1nc(C2CCCN(C(C3(CO)CCCC3)=O)C2)n[nH]1 C1(NC(C2CC(C#C)(O)C2)=O)CN(C(=O)CC2CCC2)CCC12CCOCC2 C1(C)(C(=O)Nc2ccc(CNC(=O)OC(C)C)cc2)CCCCC1C c1(NC(C2(CNC(CCCC3C(C)C3)=O)CC=CC2)=O)cc(O)c(C)cc1C C1(O)(CCNC(C2N(CC)CC2)=O)CN(C(C2(C(F)(F)F)CC2)=O)C1 C1(CNC(COCCCCCC)=O)CN(C(c2cn(C)nc2C(F)F)=O)CC1C Cc1ncc(NC(C2CN(Cc3c[nH]ccc3=N)CCC2O)=O)c(Cl)n1 C(=O)(CC(C)CC(C)C)NC(CC)(C)CCNC(=O)C(C)C1CCCC1 c1(CC(=O)NCC2C(NC(c3c(OC)cccn3)=O)C2)c(F)cccc1F C1(NC(=O)C(F)=CC2CC2)CCN(C2CCN(C(=O)CC3(O)CCC3)C2)CC1 O=C(CNS(=O)(=O)CCBr)N=c1cc(NCCc2nc3ccccc3[nH]2)[nH][nH]1 C(=O)(CCCCCn1cc(C(C)(CC)C(=O)OC)nn1)N(C(C)(C)C)CCC S(=O)(=O)(c1ccc(CCn2nccn2)cc1)NCCF C(C(=O)NC1CCCCC1N(C)C(c1ccc(Br)o1)=O)(C(C)C)NC(C)=O CC1N(CC(=O)NCCC2CC(C)(C)NC2=O)CCC1(C)C C1(C(N2CCN(C(C(C)(C)OC(C)C)=O)CC2C)=O)CN(C)C(=O)CCO1 Cn1cccc1C(=O)NCC1CCCN1C(=O)C(C)(C)c1ccno1 c1(C(=O)NC(CNC(C(C=CCCC)O)=O)C(C)C)cncc(Cl)c1.C(C)C n1(CC)cnnc1C(=O)NCC1CC(O)(C)C1.C(=O)C(C)CC1CC1 C(CS(=O)(=O)CC)NC(c1ccc(CN(C2CC2)CC)cc1)=O Cc1cc(C(N2CC=C(CCNC(=O)CSC(F)F)CC2)=O)c2cnn(C)c2n1 c1(CCC)cc(C(=O)NCC#CCNC(=O)C(CCC)N(C)C)cc(O)n1 C(=O)(C1CCCn2nccc21)N(CCNC(c1nccc2c1NCCC2)=O)CC CCC(O)C(=O)NC(COC)CNC(=O)CCc1cnc[nH]1 CC1(F)CN(C(c2nc(O)[nH]c(=O)n2)=O)CCN(C(c2c(O)cccc2Cl)=O)C1 CC(C)C(CCN(C)C(C1(C)CC1(F)Cl)=O)NC(C1CC1(F)F)=O C(=O)(C1c2c[nH]nc2CN1C(c1ccncn1)=O)N1C(C(N)=O)CCC1 N1(C(C2NCCN(C(c3cc(F)c(Br)cc3Cl)=O)C2)=O)CCN2CCOCC2C1 c1(NS(CC2(OC)CCC2)(=O)=O)c(C(C)C)cccc1C Cc1[nH]ccc(=NC(=O)C2(C)CN(c3ncnc4cc[nH]c34)C2)c1C C1(C(=O)NCC(CCOC)NC(C2(OC)CC2)=O)CCc2n[nH]cc2C1 CC1CN(C)CC(C(=O)NC(C)(C)CNC(C2CC(CF)C2)=O)O1 C1(C(C)C)(C(=O)O)CCCN1C(C1(CCF)CCOCC1)=O c1(C(=O)OC)cc(C(F)F)n(C)n1.C1(CC2CCC2)C(=O)NCCO1 c1(C(=O)NCC(C)(C)NC(=O)CCC2CCOC2)cccc(C(C)(C)C)n1 C1(NC(c2cn(CCC=C)nn2)=O)COC2C(NC(=O)C(C)C=C)COC12 Cc1c(Cl)c(C(=O)NC(CNC(c2ncn(C)n2)=O)CO)nn1C N1(C(c2c(CC)ncnc2)=O)CCN(C(=O)CCP(C)(C)=O)C(CC)C1 CC(C)C(Cc1ccccc1)C(=O)NC(c1cn(C2CC2)nn1)(C)C N1(C(=O)CCCF)CCCC(N(C(c2cccs2)=O)Cc2ccccc2)C1 N1(C(c2c(NCC)cccn2)=O)CCC(CO)C(NC(=O)CCc2nccs2)C1 c1(OC)ccc(F)c(C(=O)N)n1.c1(C(N2CCCC2)=O)cn(C2CC2)nc1C.C C(=O)(C(C)(C)C1CCCN1C(=O)C=Cc1cc[nH]c1)N(C)CCN(C)CC CC(N=[N+]=[N-])C(=O)NCc1cccc(C(N2CC(O)CC2C)=O)n1 N1(C(CC2(CCC#C)OCCO2)=O)CCOC(C(C)NC(c2ccoc2)=O)C1 c1(C(=O)NC2C(C(=O)NCC(COC)(F)F)CCOC2)cccc2cc[nH]c12 C(=O)(CC(C)(O)C(F)(F)F)NC1C(CC)CN(C(C2C=CCC2)=O)CC1 N1(C(c2c(C)cc(F)s2)=O)CC2(CCN(C(C3CCCC34CC4)=O)CC2)C1 N1(C(C2NC(=O)OCC2)=O)CC2CC(C1)C2NC(c1cc2sccc2s1)=O N1(C(C(=O)NCC(CN(C(c2c(CC)nns2)=O)C)C)C)C(=O)CCC1=O O=C(CS(=O)(=O)C1CC1)N.c1(C(N2CC(O)C2)=O)ccc(-n2ccnc2)cn1.C c1(OC)ccc(C(=O)NCC2CCCC2NC(C2CCCO2)=O)nc1Cl Cc1cccnc1C(C)NC(=O)CCC1CCN(C)C1=O.C(C)(C)C.C(=O)N C(C(=O)NCCC1CC1)(C(C)C1CCOCC1)N1CCC(C)C1 CC(C)CC(C(=O)O)NC(=O)CSCCCn1cc(C2(O)CCOC2)nn1 c1(C(N2CCN(C(C3CC3(Cl)Cl)=O)C(C3CC3)C2)=O)ccn2ncnc2c1 c1(C(=O)NCCCCNC(CCC#CC)=O)ccc(OCC)c(C)c1 Cc1c(C(N2CCCC2CNC(c2ccc(CO)cn2)=O)=O)cccc1C#N n1(CC)nc(C(=O)NCC23CC2CN(C(C2CC2)=O)C3)cc1C.C(C)=O CN=c1nc(C(=O)NCC(C)CNC(C2CC=CCC2)=O)cc(C)[nH]1 C#CCC(CC(=O)Nc1cccc(C#C)c1)NC(=O)C=C(C)C1CC1 c1(CC)nc(C)c(CN2CCC(CC(=O)NC(c3nc(O)n[nH]3)C)C2)[nH]1 C(=O)C(C)(C)CC(C)(C)C.N1(C(Cn2c(C)csc2=O)=O)CC(C)C(C)(C)C1 C(=O)(C(C(C)C)N(C)C)NCC1(CNC(C(F)=CCC)=O)CC1 Cc1ccccc1SCC(=O)NC1CCC(C(=O)NC2CC2(C)C)CC1 C1(C(=O)NC(C)C(CO)NC(=O)COc2ccsn2)CCCN(c2nccs2)C1 N1(C(c2c(CC)ocn2)=O)CC2CN(C(=O)C(F)(F)c3csc(=N)[nH]3)CCC12 c1(C(N(CC(C)(C)NC(COC(CC)(C)C)=O)C)=O)nccc(OC)c1F C(=O)CC(F)(F)CS(C)(=O)=O.C1(C(N(CCC)C)=O)CCC1.C(C)(C)C.C C1(C)(CNC(C2CN(C(N(C)C)=O)C2)=O)CN(Cc2cc(Cl)no2)CCO1 CC(C)(CO)C(=O)N1CCC(CNC(C2(Br)CC2(F)F)=O)C1 Cc1nc(C(C)C)ccc1C(=O)NCC1CCC(NC(c2cccnc2S)=O)C1 C(C(=O)N(CC(C)CO)C)(C1CN(C(=O)CN(C2CCC2)C)C1)OC c1(CNC(C2CC3CC3N2C(c2sc(Br)cc2Br)=O)=O)ccc(F)nc1F C1(C)(OC)CCCN(C(=O)C(O)C2CN(C(c3cncc(F)c3C)=O)C2)CC1 CCC(CC(=O)NCC1(N(C)C)CCC1)N(C)C(c1[nH]ccc1COC)=O C(=O)C1SCCc2ccccc21.C12(NC(C=CC=CC)=O)COC(C)(C1)C2 c1(OCC(=O)C2(CC(=O)C3CC3)CC2)ccccc1[N+](=O)[O-] c1(OC)ccnc(NC2(CNC(=O)CC(C)C)CCCC2)n1 O=C(CCC(=O)c1ccc(Cl)cc1)NCC(O)CNC(=O)Cn1cccn1 c1(CC(=O)NCCCCCNC(CC(C)C2CC2)=O)noc2ccc(F)cc12 N1(C(c2cc(C)c(C)s2)=O)C2CCC(C2)C1CNC(C12CCCC1C2)=O CCCC(CNC(=O)COc1ccn(C)n1)NC(C1(Br)CC1)=O C1(C(=O)NCCC(C)C(F)F)C2CC3C(C2)C13.c1(C=O)cc(C(F)F)[nH]n1 c1(C(=O)NC2CN(c3nnc(CCC)s3)CC2(C)C)ccc(F)c2ccccc12 C1(NC(c2c(CC)n[nH]c2)=O)CCN(C(C2C=CCS2)=O)CC1C c1(C(=O)NC(CNC(c2c(C(C)C)nns2)=O)C2CC2)cc2ccccc2s1 C#CC1(NC(=O)CCOCCC)CC(F)(F)C1.C1(C(=O)N)CC1C=O Cc1nc(S)sc1CC(=O)NC1CCCN(C(c2ccc(C(F)(F)F)cn2)=O)C1 C(=O)(CC(CC1CC1)NC(=O)COCCCC)NC(CC=C)C1CC1 C1(CC=C)(C(=O)NC2CC(=O)N(C)C2)CCN(C(=O)C(F)(F)COC)C1 c1(C(N2CCC(NC(C(=C)F)=O)CC2)=O)cc(Br)c(F)cc1C c1(C(=O)NC2COCCN(C(C(CC)(C)C)=O)C2)sc2nccnc2c1N C1(C(=O)NC2C(C)NC(=O)CC2)CC2(CCN1C(=O)Cc1ccn(C)c1)CC2 c1(SC)ccc(C(N2CC3C(C2)N3C(=O)Cc2cccc(Cl)c2)=O)cc1 C1(C(=O)NC(C(=O)NCCCSCC)CCOC)C2CCC(C2)C1C C1(NC(CCC(C)C)=O)CC2(CCC(CNC(=O)CN(C)C3CC3)OC2)C1 c1(C(=O)NC23CN(C(Cc4ccn(CC)n4)=O)C(CC2)C3)cc(C#N)ccc1O C1(C(N2CCC(C)(CNC(C3(Br)CC3)=O)C2)=O)CSc2ccccc2O1 C1(C(=O)NCC(CNC(CSCCC(C)C)=O)(C)C)CCOC(=O)CC1 CC1CC(NC(=O)CCc2ccccn2)CCN1C(=O)Cn1ccc(O)nc1=O c1(OCC)cc(N2CCC(CNC(c3cccc(C(C)(C)C)n3)=O)C2)ncn1 Cc1cc(=O)n(C)c2ccc(NC(N3CC4C5CCC(NC5)C4C3)=O)cc12 c1(OC)cccnc1C(N1CC(N2CCN(C(c3sc(C)cc3C)=O)CC2)C1)=O c1(CC=O)ccc(S(N)(=O)=O)s1.CC1OCCCC1C(=O)N.C1(CCC)CC1 C1(CN(C(c2ccc(CSC)o2)=O)C)CN(C(c2ccncc2)=O)CC12CC2 C(C(CO)C(C)CC)NC(CCC1CC(NC(C2C(=C)C2C(=O)O)=O)C1)=O C1(CC(=O)NCCCn2cc(CCN3CCOCC3)nn2)CCCCC12CC2 c1(SC)ncc(NC(C2CCC(C)CC2)=O)cn1.C1(C=O)CC(=O)C1(C)C.N CCCCCC(C)CC(=O)N1CCC2(CCCN2C(=O)CCc2ccccc2)C1 C1(C(N2CC(CCNC(CC(C)c3ccncc3)=O)C2)=O)(CO)CC(C)(C)C1 C(=O)(C(CCC1CC1)NC(=O)C(C)(C)F)N1CC(C)(C(F)(F)F)C1 c1(Oc2c(C=CC(=O)NNC(=O)C3CC3)cc(Br)cc2)cccc2c1CNCC2 c1(C(N2CCC(N(C(CC3C(CC)C3)=O)CC)C2)=O)cnccc1C c1(C(=O)OCCS(=O)(=O)Cc2cccc(NCC)c2)cncc2[nH]ccc12 C1(NC(CN(C(c2n(CC)ccc2)=O)C2CC2)=O)CC(CO)C12CCC2 c1(C(N2CCC(CO)C(F)(F)C2)C(=O)NCCCF)csc2cccc(F)c12 N1(C(C(=O)N(C2CCSC2)C)=O)CCC(c2cncn2C)CC1 c1(C=O)ccc(Cl)cc1F.c1(CCNC(c2occc2C)=O)ccc(F)cc1.N c1(CC)ccoc1C(=O)NCC1CCN1C(=O)CC1CCCN1C(C)C Cn1cnc(CC(=O)NCc2cn(C3CN(C(c4coc(CO)c4)=O)C3)nn2)n1 C1(C(=O)NC(CC(C)(C)OC)C)CCCCCCN1C(c1cnc(C)s1)=O CCC(CC)(C(=O)NCC1CC1CC(=O)NC1CCN(C)C1=O)OC c1(CN(C(c2n(CCC)ncn2)C(=O)NC(C)C)C)cn(C)nc1C(C)C c1(C2(CNC(NC(C=C)C)=NCc3noc(C4CC4)n3)CC2)cccc(F)c1F CCC(C)C(C)C(=O)N1CCN(CC(C)(C)NC(c2ccc(C3CC3)s2)=O)CC1 C1(COCC)CCCN(c2ccnc(NCC3CCN(S(C)(=O)=O)C3)n2)C1 c1(C=O)c[nH]c(=N)cc1C.Cc1cc(C)c(C(N2CCC(C(F)F)(C)C2)=O)o1.N c1(OC)ccc(CN2C(C(N3CCCCC3CO)=O)CC3CC23)c(O)c1N C(=O)(C1=CCN(C(C2CC(F)CN2C)=O)CC1)NC(c1ccc(O)cc1)C c1(SC)n[nH]c(=NC(=O)Nc2ccc(SCC(O)C3CCC3)cc2)s1 Cc1nn2ccccc2c1C(N1CCCC(CNC(=O)CCCC(F)(F)F)C1)=O CC1CC(C(=O)NCC2(C)CCOC2)CCN1C(=O)CC1(O)CCC1 CC1CC2(CCN(CC(=O)NC3CC3)CC2)CN1C(=O)CCSc1ccccn1 CC#CC1CCN(C(C2CCC(NC(C3SCC=C3C)=O)CC2)=O)C1 C1(C)(C(=O)NCC23C(CN(C(C(C)(C)C(N)=O)=O)C2)CC3)CCCCC1(F)F N1(C(Cn2c(=O)sc(C)c2C)=O)CC2C3CCC(C2C1)N(CCOCCO)C3 N1(CC2C(C)CCC2)CC(=O)N(Cc2cscn2)C1=O CC1(F)CCN(C(=O)C(Cn2cccn2)NC(c2csc(Cl)n2)=O)C1 c1(C(N(C(C)C)CCF)=O)ncccc1NC(=O)OC(C)(C)C c1(C(=O)NC2(CC=C)CCCN(C(CCC=C)=O)C2)nc2nc(C)cc(C)n2n1 c1(C(CC)=O)ccc(NCC2(O)CCN(C(=O)CC(=O)NC)CC2)c([N+](=O)[O-])c1 c1(C(C)=O)ccc(C(=O)NC(C2CCN(C(=O)COCCCF)C2)C)cc1O N1(C(C2(NC(c3ccc(C(C)C)o3)=O)CC2(C)C)=O)CC(=O)NC(=O)C1 N1(C(c2cnc(C(C)C)[nH]2)=O)CC(C)C(C)(C)C1.c1(C(=O)N)cc(F)ccc1Cl CC1COCC(C(=O)NCC2(F)CN(C(=O)CCCc3cc[nH]n3)C2)O1 CC(C)C(C(=O)N1CC(N2CCN(C(=O)C=CI)CC2)C1)c1ccccc1 N1(C(C(CC)(CC)CC)=O)CCC(C(=O)N2CCC(CO)C(O)C2)=C(F)C1 C=CCCC(F)(F)C(=O)N1CCCC(CNC(C2(OCC)CCCC2)=O)CC1 c1(C(N2CCC(NC(C(CCC)O)=O)C(F)C2)=O)cccc2ccoc12 Cc1nc(C)c(C(=O)NC(C)CCN(C)C(C2CCC2)=O)o1.c1ccccc1.C c1(N2C(C(=O)Nc3c(Cl)ncc(OC)n3)CSCC2)ncnc2sc(Br)cc12 Cc1cc(C(=O)NCC(=O)NCC2(C)CCCS2)cc(F)c1 O=C(CCCC(=O)NCC1(C(N2CCCC(F)(F)C2)=O)CC=CC1)C1CC1 C1(C2CN(C(COCC=C)=O)C2)CN(C(=O)C(=Cc2ccco2)C)CCO1 C1(C(=O)NC(C#C)(C)C2CCCC2)CN(C(=O)C=CC(C)C)CC1(C)C c1(NC(C(CC)F)=O)cccc(NC(=O)C(F)OC(F)(F)F)c1 C1(O)(CC(=O)NC2C(C)CN(C(c3sccc3Br)=O)C2)COC(C)(C)C1 c1(C(N2CCC(N(C(C(CC)O)=O)CCO)C2)=O)c[nH]cc(C)c1=O N1(C(CC(CC)OC)=O)CC(F)(F)CC1CNC(=O)CCC(C)OC CC1(C)CCN(C(C2(C(N)=O)CC2)=O)CC1NC(c1ccncc1)=O c1(OC)cncc(NC(C2CCCCN2Cc2c[nH]ccc2=N)=O)n1 C1(C(N2CC(c3cn(CC(C)(C)O)nn3)(N(C)C)C2)=O)CC1C1CCC1 N1(C(C(C)C2CC2)=O)CCOC2(CCN(C(c3cccc(O)c3F)=O)C2)C1 N1(C(c2c(CC)n(C)nn2)=O)CCC2CCN(C(=O)Cc3cn(CC)nn3)CC12 C1(C(N2CCC(COC)CC2)=O)CCN(C(c2cc(C(C)C)on2)=O)C12CCC2 C(=O)CCCC=O.C(C(C)O)N(C(=O)CC1(C)CC1)CC.C(C)(C)C.N CC1CCN(C(=O)CN=S(C)(C)=O)CC1NC(=O)CC1CCC(=O)NC1 c1(NC(c2c(C)nc(CNC(CCOCC)=O)o2)=O)cc(C)cc(F)c1 Cc1cncc(C(=O)NC2CC3CC(NC(=O)C(F)(F)C(F)F)CC23)c1C c1(C(=O)NC2C(F)CCN(C(c3c(C)cc[nH]3)=O)C2)cccc2c1CCO2 N1(C(CCCC(=O)OC)=O)CC(C)(C(=O)Nc2ccc3c(c2)CCC3)CC1(C)C C#CC1CCCN1C(c1ncc(C(C)(C)C)s1)C(=O)NCCOCCOC CC1(O)CC2(CN(C(=O)CCOCCCNC(c3c[nH]nc3[N+](=O)[O-])=O)C2)C1 C(=O)(C1=C(F)CN(C(=O)CC2(C)CC2)CC1)NC1C(CC=C)CCCC1.O C(=O)(C1=C(C)OCCS1)NC1(CO)CCCN(C(CC2ON=C(CC)C2)=O)C1 C1C(O)C(O)CN1C(c1cc(Cl)ccn1)=O.c1(C(=O)N)c[nH]nc1C(F)F.C C1(COC(C(C)Cn2cccn2)=O)CCCNC1=O C(=O)(C(C)C(C)(C)C)NCC1(O)CC(NC(CC=CC)=O)C1 C1(NC(C2(SCC)CC2)=O)CCCN(C(c2ccccc2F)=O)C1C.C(CF)O N1(C(Cc2c(C)ccnc2)=O)CC(O)CCC1C(=O)NCC1(O)CCC1 c1(C(N2CCN(C(=O)CC3CC3)C(CC(F)(F)F)C2)=O)c(Cl)nc2ccccn12 C1(C(C)C)CCC(CC(=O)NCCOCC)CC1.C(=O)(CCCC1CCCC1)N C1(CNC(=O)C=CCF)CN(C(c2cncc([N+](=O)[O-])c2)=O)C2(CCC2)C1 C1(NC(=O)CCc2cccc(Cl)c2)C(CO)(CO)CC1(CO)CO c1(C(N2CC3C(NC(COC(CC)C)=O)(CC3)C2)=O)cc(C)nc2[nH]c(=N)sc12 c1(NC(C)Cc2c(F)cccc2F)[nH]c(=NC2CC3CC3C2)nc2c1cnn2C C=C(Cl)CC(C(=O)NCc1n[nH]cc1C1CC1)NC(=O)C(C)=C(C)C c1(C(=O)NCC(CN(C)C(C2CCCC2F)=O)O)c[nH]c2cccnc12 CCC(CC(=O)N1CCC(OCCNC(c2cnn(C)c2C#N)=O)C1)C(C)(C)C Cc1nccc(C(=O)NCC2CN(C(C3CC(OC(F)F)C3)=O)CCN2C)c1C c1(C(=O)NCCC(CNC(CCS(=O)(=O)N(C)C)=O)O)cccc2[nH]ccc12 C(=O)(CC(O)CC(C)(C)C)N1C(C(=O)NCc2n(CC)ccn2)C(O)CC1 C1(COC)(NC(c2cnco2)=O)CCN(C(=O)CC(C)(C)C2CC2)CC1 c1(OC(C(=O)N(C2CCCN(C(CCOC(C)=O)=O)C2)C)C)cccc(Cl)c1Cl c1(C2CCC2)ccc(Cl)cc1.C(C)(C(=O)N(CC(=O)N)C(C)C)OC(C)=O C12(NC(CC3(C)CC3)=O)CCCC1N(C(=O)C(C)(C)CCCO)CC2 c1(CC)ccc(Cl)cc1C(=O)NCCC.C1(C=O)CCCN1C1CC1.CC.O c1(C(N2C(CC#N)CCC2)=O)cc(Cl)ccc1OC1CCCC1 C(C1=CCCN(C(=O)CCCCCF)C1)NC(C(C1CCOCC1)C)=O O=C1CC2(C(N3CCN(C4CCCOC4)CC3)=O)CCCCC2N1 c1(C(=O)NC2CC(OC)CN(C(C3(F)CCCOC3)=O)C2)ccn2ncnc2c1 Cc1cc(C(=O)NCC(C2CC2)NC(C2(CF)CC2)=O)c(Br)c(C)c1 N1(C(C(C)N=[N+]=[N-])=O)CCCC(CC(=O)NOCC2CCCCN(C)C2)CC1 c1(C(=O)NC2CC(CNC(C=CC)=O)C2)ccc(O)c(Br)c1 C1(NC(c2cc(C)oc2)=O)CCN(C(=O)CCCn2ccnc2C)C(C)C1 N1(C(C2CC(CC(C)(C)C)C2)=O)CCCCC1CNC(C1COCC1(C)C)=O N12C(CCC1C)C(=O)NCC(O)C2=O.c1(C(CSC)O)ccncc1 C=CC(C)(C)CC(=O)NC1CCCN(C(=O)CC2C=CS(=O)(=O)C2)C1 C12(C(=O)NCC(CC)(CC)NC(C3CC=CCC3)=O)CCCCN1CCC2 N1(C(C(CC=CCC)C)=O)CCN(C)C(C(N2CC(C)=CC(C)C2)=O)C1 C1(C(=O)NCC2CCN(C(c3ncc(CC)cn3)=O)CC2)CCC(C)(C)OC1 C#CCC(O)C(=O)NCC1CC(F)CN1C(C1CCCN1C(C)=O)=O c1(C(=O)NCC2CC(NC(C(C)C(C)(C)O)=O)C2)ccc2ncncc2c1 C1(O)(CCNC(=O)COCCCF)CCN(C(=O)CSC2CCOC2=O)C1 C1(C)(NC(c2ccn(CCOC)n2)=O)CCN(C(C23CCC2C3)=O)CC1 c1(C(=O)NC(CN(C(=O)Cc2coc(C3CC3)n2)CC)C)cncc(Br)c1 c1(CC(=O)NC(CC)CNC(=O)CNC(c2ccco2)=O)ccccc1F CON(CCC(=O)N(C)CC1CCCOC1)C(=O)C1(O)CCOCC1 C1(C(=O)NCCN(C(=O)Cc2ccccc2)C)CC2(CCC2)C1 Cc1noc(C(N2CC(CNC(c3ccc(CC(C)C)nc3)=O)C(C)C2)=O)c1C C1(F)(C=O)C(C)(C)C1(C)C.c1(C(CC(=O)NCC(C)C)=O)ccc(O)cc1 Cc1ccc(CC(=O)N(O)Cc2cn(C(c3ccc(Cl)cc3)C)nn2)cc1 c1(OCCn2c(C)ncc2)cccc(COCC2(C(C)(F)F)CC2)c1 C1(F)(C(=O)NCCN(CCOC)C(c2cn(C)c(C)n2)=O)CC=CCC1 CN1C(=O)CCC1CC(=O)NC(c1ccccc1)CN1CCOCC1 CC(C)CCCCCC(=O)NC1CC(C)(CNC(=O)C=C2CCCCC2(C)C)C1 c1(NC(C2(C(C)C)CCCN2C(=O)CCC2CCCO2)=O)ccc2ncnn2c1 c1(NC(=O)OC)cccc(C(=O)NC(CO)C(C)NC(c2ccoc2)=O)c1 C1(NC(c2nc(C)n(C)n2)=O)CN(C(=O)CC2CCCC2(F)F)CC1(C)C C1(CNC(C(C)C)=O)CCC(NC(c2cn(C)nc2O)=O)CC1 CC(C)CC(C(=O)NCC(C)C(=O)N1CCC(CCN(C)C)C1)N(C)C Cc1ccc(C(=O)NC2CCC(C)N(C(=O)C(c3ccccc3)=O)C2)c(C)c1 C1(C(=O)NCCC2N(C(C(CC)CC(F)F)=O)CCC2)CCc2ccccc2C1 N1(c2nc(CC)nc(=N)[nH]2)CC(C)(C)CCC1CNC(=O)CC1CCCOC1 c1(CC)ccc(C(N2CCN(C(c3ccc(CO)o3)=O)CC2C(F)F)=O)c(Cl)c1 N1(C(COCc2n(C)c(S)nn2)=O)CC2CN(C(C3(C)COC3)=O)CC2(C)C1 Cc1nc(C(N2CCC(NC(c3cnccn3)=O)CC2C2CC2)=O)cn(C)c1=O N1(C(c2cc(C)nc(C)n2)=O)CC2ON=C(CNC(=O)C=C(Cl)Cl)C2C1 C1(C(=O)NCC2C(C)=NNC2=O)CCC2(CCN(C(=O)C)CC2)O1.C1CC1 C(=O)(C(CCC(C)C)NC(=O)COCC)N(CCC(=O)OC)CC=C c1(C(=O)NCC2(C)N(C(c3c(C#C)c[nH]n3)=O)CCC2)cc2ccc(F)cc2s1 C(=O)(CCCC(=O)NC(C)C)N(C(C)C)CC.N1(CCC=O)CCC(F)C1 c1(NC(c2c(Nc3cc(COC)ncn3)c[nH]n2)=O)nc2cc(Br)cnc2[nH]1 N1(C(C(C)OCCOCC)=O)CCC(CO)C(O)C1.C(=O)CC.C=O.N C(C(C)(C)CNC(=O)CC1(N(C)C)CC1)NC(C(N1CCCCC1)C)=O c1(C(=O)OC)sc2nccnc2c1NC(=O)C(C1CC2COCC2C1)C C1(C(=O)N(C2CCN(Cc3ccccc3)C2)C)(COC)CNCCO1 N1(C(CC(C)(C)OC)=O)CC=C(C(C)(C)C(=O)N2CCC23CCC(C)CC3)C1 C12(C(=O)NCC3(NC(COC(C)=O)=O)CCOC3)CC=CC(C1)OC2 C(CO)(CCCNC(c1cnc(C2CC2)nc1)=O)NC(c1n(CC)ccc1)=O c1(NS(=O)(=O)CCCC2CCCCC2)ncnc2c1ccn2C1CC1 CCC(CO)(C(=O)N(CCCCCNC(=O)C(C)Cc1ccccc1)C)OC C(=O)(CN=c1[nH]c(C)cs1)N1CCN(C(c2n(CC)ncc2)=O)CC1C(C)C c1(C(=O)NCCC2N(C(C(CC#C)O)=O)CCC2)c(F)cc(Br)cc1F C#CC1(C(=O)N(C)CC2CCN(C(=O)C(C3CCCN(C)C3)(C)C)C2)CCCC1 Cc1oc(CNC(C2(F)CC=CC2)=O)nc1C(=O)NC.C1CC2CCC1C2 Cc1cc(NC(=O)CC2CN(C(=O)CCCN=[N+]=[N-])CCC2C)cc(CO)c1 c1(C(C)(C)C)noc(CCCC(=O)NC2CCC2NC(C2CC(F)C2)=O)n1.C N1(C(C2C(c3n(C)nnc3)C2)=O)CCN(C(=O)CCN2CCOCC2=O)CC1 C(=O)(C1=C(Cl)CCOC1)N1C(CNC(Cc2nc(C)oc2)=O)CC(O)C1 Cc1cc(Cl)cc(C(=O)NCC2(CNC(=O)C)CC2)c1C.c1ccccc1 c1(C(N2CCC3(C(NC(C4CCCN4C4CC4)=O)C3)C2)=O)ccc2n[nH]cc2c1 Cc1cc(C(=O)NC23CCC(C(=O)N)(CC2)C3)cc(Br)c1.c1cc(C)on1.C C1(C(=O)NC(C2(O)CN(C(C(COC)OC)=O)C2)C)CC2CC2CC1C C1(CNC(CCOC)=O)CCC2(CN(C(c3cncc(C)n3)=O)C2)O1 c1(C(=O)NCCC(C)C)cccnc1-n1cccn1.C(c1ccoc1)=CC(=O)N CC(CC(=O)NC(C)C(C)(C)C(=O)N1CC(CO)C1(C)C)CC(C)(C)C c1(C(=O)NCCN(C2CCCC2)C(C23CC(OC)C2C3)=O)nc(Cl)sc1C c1(-c2nn(C(C=C)C)c(-c3cccc(Cl)n3)n2)cc(F)cc(F)c1 c1(CC)ccc(C(=O)NC2CCOC2C(=O)NC2CCCOC2)cc1 N1(C(C(C2CC2)OCC)=O)CCC2(C1)CN(C(C1CCCCN1C)=O)CCO2 C(=O)(C1COc2ccc(Cl)cc21)NC1C(C)N(C(C2CCCCN2C)=O)CCC1 C(CN=C(NCC(F)F)N1CCc2c(Br)cccc2C1)N1C(=O)CCC1 C1(N(c2ncnc(OC)c2C)Cc2c(C)noc2C)CC2CCCC(C1)N2 c1(NC(C(CC)(C)O)=O)ccc(NC(c2cc(F)cs2)=O)cc1C C1(CCCCNC(c2ccc(Cl)o2)=O)CCCN(C(=O)CCc2ncc[nH]2)C1 C1(NC(C2CC3C=CC2CC3)=O)CC2CC1N(C(=O)Cc1c[nH]nc1O)C2 C(CCC(F)F)NC(C1C(C(C)NC(CN(C(C)C)C)=O)C1)=O c1(CC)ccc(F)cc1C(=O)NC1CC(O)CN(C(c2c(C)[nH]c(C)c2C)=O)C1 C=CC(CC)C(=O)NC(C)CC(=O)NC(C)(C)C(=O)NO Cc1c(Cl)ccc(C(=O)NC2CCN(C(=O)C(F)C(C)C)C2)c1Cl CCC(CC)CC(=O)NC1COCCC1NC(c1ncc(OC)cc1F)=O CC1CC(C)CCN1C(=O)CN1CCC(C)(O)C1.c1(C=O)ccc(F)c(Cl)c1.N CC1CCOC(C(N2CC(O)CC2CNC(=O)COc2cncc(Br)c2)=O)C1 CC(C)CC(CNC(=O)C(F)CC1CCCC1)NC(c1ccccc1)=O C1(C(=O)NC2(CC(N3C(C=C)CC3)=O)CC2)CCOC(C)(C)C1 c1(C(=O)N)cccc(F)c1C.C(=O)(C(C(C)C)n1ccnc1)N1CC(OC)(C)C1 C1(NC(c2cc(C)c(Cl)s2)=O)CCN(C(=O)COc2ccc(O)cc2)CC(O)C1 C1(NC(c2cn(C)nn2)=O)CN(C(C2CCCC(O)C2)=O)C2CCCC12.C1CC1 Cc1ccc(C(=O)NCC2(C)CCCN2C(c2cc[nH]c(=N)c2Cl)=O)c(=O)n1C N1(C(C(C(=O)OC)C)=O)CC2(NC(=O)Cn3c(C)csc3=O)CCCC2(F)C1 C1CC2(CCCN(C(=O)Cn3cccc3)C2)C1.c1(CC)ccc(C=CC=O)o1.N N1(C(C(C(C)C)OC)=O)CCCN(C(C2(c3cccs3)CCCC2)=O)CCC1 C=CC(C)(O)CC(=O)NC(C1CCCCC1)C(=O)NC1CC(CC)(CC)C1 C1(C(N2CCC(C(C)(C)C)C2)=O)(CNC(COCCCC)=O)CC12CCC2 C#CCC(C)(C(=O)N(CC)OCC)NC(c1ccc(C#N)cn1)=O Cc1nc(O)nc(C)c1CC(N1CCC(NC(=O)CNC=O)C1)=O c1(CC(C)C)ccc(C(=O)N(CCCCN(C)C(C2(C#N)CC2(C)C)=O)C)cc1 O=C(C(C(F)(F)F)C(F)(F)F)NCCC1=CCN(C(c2ccc(O)nn2)=O)CC1 N1(C(C2C(CC)(CC)C2)=O)CC(CNC(c2cccnc2C)=O)C2CC12 N1(C(C(C2CC2)OCC)=O)CCC(F)C(NC(=O)CCC2CCCCC2)C1 C(CC(=O)NC1CC(OCC)C1)(C(C)CC)NC(COCC(=C)C)=O c1(OC)cc(OC)cc(C2(CNC(=O)Nc3ccc(F)nc3O)CC2)c1 C(CCCCCNC(C1CCCC(F)C1)=O)N(C(=O)Cc1ccc(CO)cc1)C CC(CN=c1[nH]c(N2CC3CCC(O)C3C2)nc2cccnc12)c1ncc[nH]1 C1(CNC(c2n[nH]c(CC)c2C)=O)CC(C)CN(C(c2c[nH]nc2OC)=O)C1 c1(CNC(C2CCN2Cc2nccs2)=O)cc(C(F)(F)F)ccc1F C(=O)(C(CNC(c1cnns1)=O)C(C)(C)C)NC(c1c(C)nn(C)c1)C N1(C(c2cccc(SCCC)c2)=O)CCC(NC(=O)C(C)(CO)CC)C1(C)C CC1C(NC(=O)C(F)=CC2CC2)C(C)CCN1C(c1cc(CF)on1)=O C1(NC(c2cnc(CC)[nH]2)=O)CC12CCN(C(C1COCC1C(F)F)=O)CC2 C1(O)(C(=O)NCC2CCCC(NC(Cc3scc(CC)n3)=O)C2)CCCCCC1 C1(CNC(CCCOC(C)C)=O)CCCCC1.C1(C(F)(F)F)(C=O)CCC1.N C1(CNC(c2c(CC)occ2)=O)CC12CCN(C(=O)CS)CC2.c1cccs1 C1(C(C)(C)C)CN(C(C2CC(=O)NC(=O)N2)=O)CCN1C(c1cnc(N)cn1)=O C1(CCC(=O)Nc2ccccc2Cl)CCCN(C(c2cc[n+]([O-])cc2)=O)C1 C(c1nc2ccccc2o1)=CC(=O)N.C(C)(C)(C(=O)N(CC(C)(C)C)C)OC C1(NC(c2ncc(Cl)cc2Cl)=O)CN(C(=O)CC2(O)CCC2)CC12CCC2 C(C1CCN(C(C2CCC3(CCC3)C2)=O)CC1)=CC(=O)NC1CC1O C1(CCNC(c2cnc(C)s2)=O)COCCN(Cc2nc(C)c(C)s2)C1 c1(C(=O)NC2CC(NC(CCSC)=O)C23CCC3)cnc2nc(C)[nH]n2c1=O C1(C(=O)NC2CCN(C(C(C)OCCC(C)C)=O)CC2C)CCc2c[nH]nc2C1 CC(C)CCCNC(C1CCN(c2nccn2C)C1)=O.C1(=CC(=O)N)CCCC1 c1(C=O)cc(C2CC2)nc(O)c1.C(=O)(C(C)NC(C)C1CC1)OCC.N CC(C)(C)C(CNC(=O)CCCN1CCCC1)NC(C1(C)CCCO1)=O Cn1ccc(C(N2CCCC2(C)C(=O)NCCc2cc[nH]n2)=O)c1CC(=O)O CC1(C)COC(C(=O)NC2C3CC2N(C(=O)C=CCF)C3)C1 CCC(Cc1cccc(C)c1)C(=O)NCC1C=CC(NC(c2cncs2)=O)C1 C1(CNC(CN(C)S(N)(=O)=O)=O)CN(C(c2cscc2Cl)=O)CC12CCC2 C(CCN=c1nc(N2CCc3c(CO)n[nH]c3C2)cc[nH]1)OCC=C C1(C(=O)NC)(CC)CCCC1O.C1C2CN(C(=O)C)CC12.C(=O)CCC(C)C CC(CCNC(=O)C(=O)NCCCc1ncnn1C)CC(C)(C)C C1(N(C(CN(C(=O)COCCOC)CC)=O)C)CCCC1C#N C(CC(C)(C)C(=O)NC1COCC1C(=O)NCC(C)CN(C)C)OC c1(C(C)O)cc(NC(C2CCN(C(=O)OC(C)(C)C)CC2C)=O)ccc1F C1(NC(C(C)(C)CCNC(=O)C(O)C2CC2)=O)CC(O)CC(C)(C)C1 N1(C(C)=O)CCCNC(=O)CC1.c1(N2C(=O)C2)ccoc1 C(CC(=O)NNC=O)c1c(C)nc(-c2ccc(-c3c(C(=O)OC)noc3C)cc2)s1 Cc1ccc(C)c(S(=O)(=O)NCCNc2cc(-c3ccco3)nc(C)n2)c1 Fc1cc(-n2nc(CC3CC3)nc2C(F)C(F)(F)F)cc(F)c1F c1(C(=O)N)ccc2ncn(C)c(=O)c2c1.CCC(C)(COC)C(=O)NC1CCC1 C1(CC(=O)NC(C)C)CCCCN1C.C12(C=O)CC(C(C)C)(CO1)C2.CC c1(NCC2C(C)CCO2)cc(N2CCC(c3ncccc3Cl)CC2)ncn1 N1(C(c2nc(C3CC3)cs2)C(=O)NC(CC)C)CCC(C#N)CC12CC2 C1(NC(c2cccc(CNC(c3ccsc3)=O)n2)=O)CN2CCCC1C2 Cc1cc(C(N2CCC(O)(C(=O)NC)C2)=O)cn1C.c1c(-c2ccccc2)noc1Cl c1(C(=O)OC)cc(Br)ccc1CN1CC=CC1C(=O)Nc1ccnc(F)c1F c1(CCC(=O)NCC(CNC(C(C)(CO)OC)=O)(C)O)cc(Cl)cc(Cl)c1 O(NC(=O)CC(C(F)F)NC(=O)C(C)C(=O)OC)C(C(=O)OC)(C)C C(=O)(CCC(=O)NN(C)C)NC(C)C(C)C(=O)NOC1CCN(C)CC1 C(=O)(CCC(C)(C)C#N)N1CCCC(CC(=O)N(CC(O)CO)C(C)C)C1 N1(C(C(CC)c2cccnc2)=O)CCN(C(C2CCCN(CC)C2)=O)CC1CO CN1C(=O)OCC1C(=O)NC(C)(C)CCNC(c1cnn(CCO)c1)=O C(=O)(C(C)C(=O)N(C1(CC(=O)N(C)CC2COC(=O)N2)CC1)C)OC CC(C)C(CCN(C)C(c1ccn(C(C)C)n1)=O)NC(C1(O)CCOCC1)=O C1(CNC(Cc2c(C)con2)=O)CC2CCC(C1)N2C(C1(F)CCOC1C)=O Cc1ccc(Br)c(CC(=O)NCc2nc(-c3ccc(F)cc3)n[nH]2)n1 C1(CCN(C)C(c2ccc(CO)nc2)=O)CCCCN1C(C1CCCN1C=O)=O c1(C(N2C(C)(C(N(C)Cc3ccccc3)=O)CCC2)=O)cnc(Cl)c(I)c1 C=C(Cl)CCC(=O)NC(CCC1CCC1)C(=O)NCc1ncnn1CC C1(C(N(CC(C)(C)NC(C=CCC)=O)C)=O)CCC(=O)N(C(C)C)C1 N1(C(C2(CC)CCCCC2)=O)CC2CCN(C(c3sc(F)cc3C)=O)CC(C2)C1 C1(C(=O)NC(C(=O)OC)Cc2cccs2)CC2(C)CC1CO2 C1(NC(C23CC(CN(C(C4CC(C)(C)C4)=O)C2)C3)=O)CCCN2CCCC12 CCC1=NOC(C(=O)N(C2CCCN(C(c3ccc(Cl)o3)=O)C2)CC)C1 Nc1cc(C(=O)NCC2(C)CC2)cc(F)c1.C12(C=O)CC(F)(C1)C2.N c1(CC=O)cnn2ccccc12.n1(CC)cc(Cl)cc1C(=O)NCC1CCC1 c1(C(N2C(C)CC(NC(c3ccc(=N)[nH]c3)=O)C2)=O)cccc(S(C)=O)c1 c1(CNC(CC=CC)=O)occc1C(=O)NC(c1cncn1C)CO N1(C(Cc2nnn(C)n2)=O)CC(NC(=O)CCn2ccccc2=O)C2(CCC2)C1 c1(C(=O)NC2CCC2NC(C2CC(F)(CO)C2)=O)cc(F)cc(Cl)c1O c1(CC(=O)N(CCNC(c2ncc(F)cc2N)=O)CC)ccccc1[N+](=O)[O-] c1(C(N2C(CC(=O)N(C)CC34CCC(CC3)C4)CCCC2)=O)cc(O)ncc1F c1(C(=O)NCC#CCNC(C(CCC=C)(F)F)=O)ccccc1S(=O)(=O)C(F)F CC(C)(F)C(C)(F)C(=O)NCCC1CN(C(=O)C=CC)C1.C1CCOCC1 c1(C(N2CCN(C(C(CC)C3CCOCC3)=O)CC2)=O)cnn(C)c1C#N N1(C(CCSCCC)=O)CC(OC)CC1CNC(c1coc(OCC)n1)=O C1(CNC(C2NC(=O)OC2)=O)CCC2CN(C(c3ccc(Cl)s3)=O)CC12 C1(C(=O)NC2C(C)(C)CN(C(C3CSC3)=O)CC2)Cc2cc(Br)ccc2O1 C=CCC(C)(CC)C(=O)N1CC2CCOC2(CNC(c2cc(C)nc(C)n2)=O)C1 C1(NC(c2ccc(C(=O)OC)o2)=O)CC2COC1C2.C(=O)CC.CC(C)C.N c1(SC)c(-n2cc(C3OCCO3)nn2)ccc2c(C)cc(=O)oc12 C1(C(=O)NC(CNC(C(CC)(C)OC)=O)C)Cc2cccnc2C1 c1(C(=O)NCCN(CCC)C(c2ccnc(OC)c2F)=O)cccc(Cl)c1C CC1CN(C(C2CCCSC2)=O)C1C(=O)NCc1nc(N(C)C)no1 C1(NC(C2CCN(C3CC3)C2=O)=O)CCCN(C(=O)C=CC2CCCC2)CC1 C(=O)(C1=NN2CCCN=C2N1)N.N1(C(C(C)NS(CC)(=O)=O)=O)CCC(C)C1 c1(CCC=O)ccc(Cl)c(F)c1.c1(CNC(C)=O)cc(C=O)no1.C1CC1 Cc1ncc(C(N2CCC(=CCNC(=O)C(C)Cn3cccn3)CC2)=O)cc1N CCCCC(O)CC(=O)N(C1CN(C(=O)CCNC(c2cnccn2)=O)C1)C Cc1c(C(=O)NCC2CCN(c3ccc(Br)cc3)C2)ccc2ccccc12 CCCCCCC(=O)NOCC(N1CC23CCC2(COC3)C1)=O c1(OC)ccc(-c2nc(-c3[nH]c(C)cc3C)n(CCCN(C)C)n2)cc1Cl C(=O)(C1CCc2c[nH]nc21)N1C(C(C)(C)NC(C2CCC(CC)O2)=O)CCC1 C1(C(N2C(CNC(Cc3n(C)ncc3)=O)CCCC2)=O)CCc2nnc(O)n2C1 C12(CNC(CN(C3CCCC3)C)=O)CCCC(CN1C(=O)CCC(F)(F)F)C2 C1(C(=O)NCC2(COC)CCC2)CC12CCN(c1nc(C)ncc1F)C2 C1(C)(NC(C(CC)N2CCCC2=O)=O)CCCC1NC(=O)C=CC(C)C c1(CC)cccnc1C(N1CCOC(CCNC(C2(F)CC2C)=O)C1)=O CC12CC1CCN2C(C1CCC(CNC(C2CC2F)=O)CC1)=O C1(C(N2CC(OCc3ncc(C)o3)C2)=O)CCCCC12CCC2 CC(CC(F)F)C(=O)N(CC(C)(C)CNC(=O)Cc1ccc(O)cc1)C c1(OC)c(C(=O)N)c(C)nn1C.C1C2CN(C(=O)CC3(C)CCCO3)CC12.C C1(C(CNC(C2(OC)CCSC2)=O)(C)C)CCN(C(c2cnc(C)nc2)=O)CC1 N1(CCC)CCCCC1C=O.C(C)CC(C)C.[SH](=O)(=O)CC.C(=O)CC1CC1 Cc1cccc2c(CC(N3CCC(NC(=O)CC4=CCCC4)C(O)C3)=O)c[nH]c12 CS(=O)(=O)C1CCCN(C(C2C(O)CCN2Cc2cc(CO)ccc2O)=O)C1 C(=O)(CCC(CF)CF)NC1C(CNC(CCCOC)=O)CCCC1 C(=O)(CCCCC1CC1)N(CC(CC)NC(=O)CNC=O)C c1(CCC(=O)NCCC2(CNC(Cc3ccn(C)c3)=O)CC2)ccccc1F c1(-n2ncc(C(=O)NC)c2C2CC2)ccc(Cl)cc1Cl.c1cccc(OC(F)F)c1 N1(C(c2cnc(N(C)C)nc2)=O)CCc2sc(-c3cnn4cccnc34)cc2C1 Cc1cn2cc(C(=O)NC3CCCCC3NC(=O)C=C3CCCC3)cc(C)c2n1 c1(C(=O)NC(C)(CO)CO)cc(CNC(=O)CC2CCCCC2)ccn1 c1(CC(=O)N(CC(CNC(c2ccn(C(C)C)n2)=O)C)C)cccc2cn[nH]c12 c1ccc(F)c(F)c1.C(=O)(CCCO)N1CC(CNC(=O)CC2CC=CC2)C1 C1(NC(C(=O)NCCCCNCC(F)(F)F)=O)C2C=CC(C2)C1CO N1(C(c2c(CC)nco2)=O)C2CCCC1CN(C(C1(C)CC1)=O)CC2 c1(C(=O)NC(C(C)NC(=O)CN2CC3CC3C2)CO)coc2c1NC(=O)CCC2 C1(NC(=O)Cn2cc(Cl)cn2)CC2(C(N3CC(OCCF)C3)=O)COC1C2 N1(C(CN(C(COC)=O)C)=O)CC2CCCC2C1C(=O)NCc1cocn1 c1(OC)ccc(C(C(=O)O)NC(=O)C2=C(Cl)CCC2)c(C(F)(F)F)c1 c1(C(=O)NCC(CC=C)NC(c2cnsn2)=O)ccc([N+](=O)[O-])s1 C1(F)(C(=O)OC)CN(C(=O)C(=O)NC(C)C(C2CCCOC2)OC)C1 Cc1cc(C(=O)NC(C)C(C)NC(=O)Cc2cnns2)n(CC(F)F)n1 C(=O)(CC(F)(F)C(F)(F)Br)N1CC2C(CNC(C(F)=C(C)C)=O)(C2)C1 CCC(C)(C)CCCC(=O)N1CC2CCC1CC2NC(C1CC2(CCCO2)C1)=O C12(C(N(C3CCN(C(CCC=CC)=O)C3)CCO)=O)CCCC(OC)(CC1)C2 c1(OCCOCC)cc(CNCC(C2CC(F)(F)C2)O)cc(O)c1 C1(C=O)CCC([N+](=O)[O-])CC1.O=C1CC(C(=O)N)NC(=O)N1.C1(O)CCC1.C Cc1nccc(C(=O)NC2(C)CN(C(C3(C)CC(C(F)(F)F)C3)=O)C2)c1N Cc1cc(C)c(CC(=O)N(CCC(C(C)C)NC(C2CSC2)=O)C)c(O)n1 N1(C(c2ccc3ccnn3c2)=O)CC(C2CCN(C(C3CCC3)=O)CC2)C1 O=C(C1=CC2C=CC1C2)NC1CN(C(c2ccc(O)nc2)=O)C2CCCC12 C1(NC(C(CC#C)(C)C)=O)CC2CCC(C1F)N2C(=O)C(CC)C(C)(F)F C(C(C(=O)N1CC(NC(C2C3CCCC23)=O)C(SC)C1)C(F)(F)F)OC Cc1cc(C2(C(=O)NCC(C3CCCCC3)NC(c3nn[nH]c3Cl)=O)CC2)on1 C1CC2(C1)CCC2.c1(CCC=O)ccc(F)cc1.C1(OCC)CC1C(=O)N C1(CN(C(=O)C=CC(F)F)CC)CCCN1C(c1csnn1)=O CC1CN(C(=O)C(C)Cc2ccc(C#N)cc2)CCN1C(=O)CC1CCC(C)C1 CCCCS(=O)(=O)CC(=O)NCC1CCCC1NC(c1cccc2ccnn12)=O c1(C(=O)NC2COCCN(C(C3N(C)C(=O)NC3)=O)C2)ccc2c(n1)OCCO2 N1(C(C2(CNC(CCCSC)=O)CCCC2)=O)CC2CCC1C(O)C2O C#CCC(C)(CC)C(=O)NCc1csc(C)n1.C12(C=O)CCC(N=[N+]=[N-])C1C2 C1(CC)(NC(=O)C=Cc2ccncc2C)CCCN(C(c2cc(Cl)n(C)n2)=O)C1 Nc1cc(F)c(F)cc1-c1cn(CCNC(c2cnc(Br)s2)=O)nn1 N1(C(C(C)n2cncn2)=O)CCC(C2(NC(=O)CC3SC(=N)NC3=O)CC2)CC1 c1(NC(=O)OC(C)(C)C)ncc(Br)cc1NC(C1C2CC3C(C2)C13)=O C1(NC(C(COC)O)=O)CCC2CN(c3ccc([N+](=O)[O-])c(C)c3)CC2C1 c1(C(=O)NC2CC(C)N(C(c3cc4c[nH]nc4s3)=O)C2)ccc(F)c(Cl)c1 N1(C(=O)C=Cc2cncnc2O)CC2CCN(C(=O)CCCC(F)(F)F)C(C2)C1 c1(CC)nc(Cl)nc(NC2(CNC(=O)CCC3CCC3)COC2)c1C#N N1(C(c2c(CC)n(CC)nc2)=O)CC(NC(C2(CCO)CC2)=O)CCC1C C1(CNC(=O)C(=O)Nc2ccc3cc[nH]c3c2)CCCCC12CCC2 c1(OC)ccc(OC)c(CC(C)N(C)CCN(C)C)c1 c1(C=O)ccc(C(C)C)nn1.c1(N(CCOCC)CC)nnc(C(F)F)s1 c1(OC)ccc(Cl)cc1-c1cscn1.N1(C(C(=O)N)=O)CCC(O)(C(N)=O)CC1 Cn1c(O)ncc(C(=O)NCC2(C)COCCN(C(=O)Cc3cnsc3)C2)c1=O C(=O)(CC(C(F)(F)F)NC(=O)COCCF)N1CC(NC(C)=O)C1 C1(C(N2C(CC(N)=O)COCC2)=O)CCCN1NC(=O)c1ccccc1F c1(C(=O)NC2C(C)CCN(C(C(C(C)C)F)=O)C2C)nnc(O)c2ccccc12 c1(CNC(CS(CC)=O)=O)nc2c(s1)CN(C(c1csc(O)n1)=O)CC2 CCC(O)C(F)(F)C(=O)N1CCOC(CNC(c2ccoc2C)=O)C1 N1(C(C2CC(C)OC2)=O)CC2CC(NC(C3(C)CCC(=O)NC3)=O)CC2C1 c1(C(N2CC(C)(C(=O)NC(c3ccncc3)C)C2)=O)cc2ccncc2[nH]1 N1(C(C(C)OC)=O)CC(CO)C2(CCN(C(c3cc4cnccc4o3)=O)CC2)C1 C(=O)(C(C)CC1CCCCC1)N(CCCNC(COC(CC)(C)C)=O)C C(=O)(C#CC(C)(C)O)NCC1CC(NC(CC(C)CN(C)C)=O)C1 CC(C)(C)C(O)C(=O)N1CCC(NCc2ccccn2)CC1 C(=O)(C1=CCC2CCC1N2C(C1(CF)CC1)=O)N1CCCC(C)(CO)C1 C1CCN(C(=O)C(C)Cn2ccnc2)CC1(F)F.C(C(=O)N)NC(=O)NC.C c1(C(N2CC(CC(C)NC(=O)C(C)(Cl)Cl)C2)=O)cocc1Br CCC(CC)CCC(=O)NCCC(C)N(C)C(c1cccn2cnnc12)=O Cc1n[nH]cc1C=CC(=O)NCCC(C)NC(c1cnn(C(C)(C)C)c1)=O C1(C(N2CCC2)=O)CCCN(C(=O)N)C1.Cc1nc(CC(=O)NCC(C)C)cs1 c1(CN2CC(C(C)NC(C3CC34CCOC4)=O)C2)ccc(OCCO)cc1 C1(C)(CC)NC(=O)N(CC(=O)NC2CCCCC2)C1=O.C(=O)(C)N.C1CC1 N1(C(CCc2cc(C)on2)=O)CC(C2CN(C(C3(C#N)C(C#N)C3(C)C)=O)C2)C1 CCC(CCOC)C(=O)NCC(F)CNC(c1cn(C2CC2)cn1)=O O=S(=O)(CCCN=c1[nH]c2c(c(=NC3CCN(c4ncc[nH]4)C3)[nH]1)CCCC2)C(F)(F)F C1(CC(NOCC=CC)=O)CCCN(C(C2CC(OC)C2)=O)C1 C1(F)CCCN(C(c2cc[nH]c(=NC)c2)=O)C1.C(=O)(CC(=O)NC)NCC#C c1c(Cl)c(F)nc(F)c1Cl.C=CCC(C)(C)C(=O)NC1CC2(C1)CC(C=O)C2.N c1(N2CCC(NC(=O)NC(N(C(C)C)C)=O)C2)ccc(F)c(F)c1 N1(C(C2C(C)(C)C2(C)C)C(=O)NC2CCCC2)CCC2(CC(C(F)F)=NO2)C1 CC1(C)CC(CO)N(C(C2COCCN(C(C3OCCC3(C)C)=O)C2)=O)C1 N1(C(C(CC)=CCCC)=O)CC2CC(C)N(C(c3cc(C)co3)=O)C2C1 c1(C(N2CC(CNC(c3c(C)nn[nH]3)=O)C2)=O)sc(C#N)cc1Cl C1(C(N2CC(C(CC)CC)C2)=O)CCN(C(C2CCCN2C=O)=O)C12CCC2 CC1CCC(C)CN1C(c1ncn(-c2ccccc2)n1)=O.C(=O)(C1=NNC(=O)C1)N C1(C(=O)NCC2COCCN(C(C3CCN(C)C3=O)=O)C2)Cc2nccnc2C1 N1(C(CN(C(=O)OC)C)=O)CC2CC(C1)N(C(=O)CSC(C)(C)C)C2 N1(C(C(C)OCC)=O)CCCC(CNC(C2CCCC3CC23)=O)C1 Cc1ccc(F)c(CC(=O)NC(C2(O)CN(C(c3cc(Cl)n(C)n3)=O)C2)C)c1 C1(NC(c2ccc[nH]2)=O)(CO)CCCN(C(=O)COc2cnn(CCO)c2)C1 c1(C(=O)NCC=CCNC(C(CC)C)=O)cc(C)n(C)c1C.c1ccncc1 c1(C(=O)NC2CN(C(c3ccn(CC)n3)=O)CC23CC3)ccc(Br)c(O)c1Br C1(C(=O)NC2(C)CC(NC(CN(C(COC)=O)C)=O)C2)CCCCN1C c1(SC)cncc(C(=O)NCCCCCCNC(c2c(C)coc2C)=O)c1 N1(C(CCOCC#C)=O)CC2CC1CCC2NC(C1CC12CCOCC2)=O C1(CN(C(=O)C(C)C)CC)CCN(C(c2ccc(O)nn2)=O)CC1.C(C)=O Cc1nc(C(=O)N(C)CCNC(=O)CC2CCCCO2)nn1-c1nc[nH]n1 Cc1ncc(C(=O)NC2(C(=O)NCC3CC(C)CO3)CC2)cc1C#N c1(CCNC(C(=O)Nc2cc(C)nn2C(C)C)=O)c(F)cc(Br)cc1F C(=O)CC(C)(CN(C)C)C(F)(F)F.c1(OC)cnc(C(=O)NC2CC2)nc1 Cc1[nH]nc(C(C)C)c1C(N1CCC(NC(=O)CCn2cccnc2=O)CC1)=O c1(C(C)C)cc(C=O)cc(O)n1.C1CN(C(=O)C(F)OC(F)(F)F)C(C)(C)C1.N Cc1nc(NCC2CC23CCC(O)CC3)cc(=NC(C)c2cccc(Cl)c2)[nH]1 C(=O)(CCCC(=O)N1CCCC(CCC(=O)NC2CC3CC3C2)C1)OCC c1(C(=O)NCCCC(C)NC(C(C)SCCCC)=O)cn(C2CCC2)nc1C N#Cc1ccnnc1N1CC2CC1(CNC(=O)CC=C(Cl)Cl)C2 c1(C(N2CC(COC)(NC(=O)CC3(C)OCCO3)C2)=O)cnccc1C C1(C(N2C3CC(CNC(C(C)(C)CF)=O)(OC3)C2)=O)OCC2CCCCC12 NC1CCCc2c(C(=O)NC(C3CCOC3)CO)n[nH]c21 c1(N2CCC(C(C)C)(CO)C2)nc2ccc(Cl)cc2c(=NCC=CBr)[nH]1 c1(SC)ccc(C(N2CC(CNC(C3(CCF)CC3)=O)CC2C)=O)cc1 N1(C(C(C)(C)OCC)=O)CCCC(O)(CN(C)C(C2CCCS2)=O)C1 N(C(=NCCN1CCC(C)CC1)NC1(C)CCCOC1)C(COC)C c1(C(NCC(C)C)=O)ccc(CC(C)C)cc1.CC=O.C(CO)OCC C(=O)(C(CC(C)C)CC(C)C)N.c1(CCC)cc(C(=O)NCCC2CC2)nn1C c1(C(=O)OC)c(Br)ccc(NC(C23CC(C2)C3)=O)c1C.c1cccc(F)n1.N Cc1nc2cc(C(N3CCCC3(C)C(=O)N(C)CC3CCNC3)=O)ccc2s1 c1(C(=O)NCCN(C(C)=O)CC2CC2)cnc(-c2ccccc2)s1 c1(C(N2CCN(C(=O)NC)CC2)=O)cc(Cl)cc(Cl)c1OC c1(C(N2CC3CC3C2)=O)cnc(N)c([N+](=O)[O-])c1.Cc1cccc(C(=O)NC)n1 c1(C(=O)NCC(CNC(CCSCCC)=O)C)c[nH]c2c(F)c(F)ccc2c1=O C(CCN(C(=O)CC1CC=CCC1)C)(C(C)(C)C)NC(c1nc(C)n(C)n1)=O C1(CNC(c2ncc(OC)cn2)=O)CN(C(C2C(C)C2(F)F)=O)CC1(C)C C(=O)(C(F)(F)C(F)F)CCN(C(c1cnc(C#N)s1)=O)CC.C(=O)O O(C=CC(=O)N1CCCC1CN(C)C(c1cn(CC(F)(F)F)cn1)=O)CC C1(CN(C(=O)C(F)C2CCC2)C)CCCCN1C(=O)CCCCC1CC1 CN1N=C(C(=O)NC2CCCCC2C)CCC1=O.n1(C2(C(=O)N)CC2)cncn1 N1(C(C2(C=C)CCC2)=O)CC2(CCCC(CNC(C3CC(C)CO3)=O)O2)C1 Cn1ncc(C(=O)NCC(C)(C)NC(=O)C=CC2CCCO2)c1S(C)(=O)=O c1(C=O)cc(C)nc(Cl)c1N.c1(OCC)cncc(C(=O)NC2(C)CC2)c1 c1(C(=O)NC2C(C)CCN(C(C=CCCC)=O)C2)cc(F)c(CC(=O)O)cc1N C12(C(NOCCCC(=O)OC)=O)CCCC1CCN2C(=O)C=CC1CC1 N1(CC2CCN(C(C(CC(=O)OC(C)(C)C)O)=O)CC2)Cc2ccccc2C1=O c1(C(=O)NC2CCC(C)N(C(=O)CCc3ccsc3)C2)cc2n(n1)CCCC2=O C1(CC)CCN(C(=O)Cn2cccnc2=O)C1C.C(=O)CN(C)C(N)=O.N c1(CC(N2CCCC(NC(C(C)(CO)OC)=O)C2C)=O)cccc2sccc12 c1(OC)c(O)cc(C(N2CCCC2(C)C(N2CC(C)C2)=O)=O)cc1O N1(C(CN(CC)CC)=O)CC=CC1(C)C(=O)N(CCC(C)C)CCO C(CCCC(=O)NCCCCCN(C)C(C)C)N(C(C(CSC)O)=O)C C1(C)(NC(C2C(C)=CCS2)=O)CCCN(C(C2COCCC2(F)F)=O)C1 c1(CCCC=O)c(F)cccc1F.CCCC(C)=CC(=O)NCCC1(C)CC1.N C1(C)(COC(C(c2ccc(Cl)nc2)(C)C)=O)CC(=O)C12CCC2 c1(C(N2CCN(C(C(C)OCCC#C)=O)CC2C)=O)cc(F)c(O)c(F)c1 Cc1cnn2cc(NC(COCc3ccccc3)C(C)C)cnc12 c1(CC(=O)NC2CCCC2NC(c2ccc(-c3cc[nH]n3)s2)=O)sc(O)nc1O C1(C)(NC(c2c(SC)cn(C)n2)=O)CCCCC1(F)F N1(C(CC=CC=C)=O)CCC(C2CCN(C(c3cc(SC)ccc3O)=O)C2)CC1 c1(COC)n[nH]c(=NC2CCC(NC(=O)CC3CCNC3=O)c3ccccc32)s1 N=c1ccc(C(=O)NCC(C2CC2)NC(C2CC2c2ccncc2)=O)n[nH]1 c1(C(N2CCC(O)(C(C)NC(CSCCCC)=O)C2)=O)cc(F)ccc1O CCCC(CC(=O)NCC(C)N=[N+]=[N-])NC(c1cnc(O)cc1C)=O CC1=CCC(C)(C(=O)NCCC2CCCN(C(=O)CCc3ccc(Cl)s3)C2)CC1 C(=O)(C1=CS(=O)(=O)CCC1)NCC1CCCN(C(CC=O)=O)C1.CC(F)(F)F C1(NC(C(CC)n2ccnc2)=O)CC2CC1CN(C(c1cc(OC)ncn1)=O)C2 C1(CNC(CC2(OCC)CC2)=O)CCCCN1C(=O)C(N1CCNC1=O)C c1(C(=O)NC(C(=O)N2C(COC)CCC2)CCC2CC2)cnc(O)cc1C C(CC(F)F)(C(=O)NCCCS(C)=O)NC(c1c(C)cncn1)=O c1(C(N2CCC(NC(C(C)CO)=O)C2(C)C)=O)ccc2c(c1)OC(C)(C)C(=O)N2 c1(C(=O)NC2(C(=O)NC(C(=O)OCCC)C)CC2C)ccc(C#N)cc1C N1(C(CC(C)(F)F)=O)CCC2C(CCCN2C(=O)Cc2ccc3[nH]ccc3c2)C1 c1nn(C)c2c1CN(C(C13CCCC(C)(C1)OC3)=O)CC2.C(C)(C(=O)N)SC.C N1(C(C(CC#CC)NC(c2cncc(C)n2)=O)=O)CCC2(CCCCO2)C1 CC1CCCc2ncc(C(=O)NC3CCCCCC3NC(c3cscn3)=O)n21 C1(CN(C)C(C2CC=CC2)=O)C2CN(C(c3n[nH]cc3Cl)=O)CC12 CC1CCc2ncc(C(=O)NCCC3COCCN3C(=O)C(=O)N(C)C)n2C1 c1(C(N2CC3CC3C2)=O)cc(Cl)nc(Cl)c1.c1(CC)cc(C(=O)N)n(C)n1.C C(C1=CCCOC1)NC(CC1C(CNC(C(C2CCOCC2)C)=O)C1)=O N1(C(CSC(C)C)=O)CCC(C2CCN(C(=O)CC3CCC(C)C(C)C3)C2)CC1 c1(C(C)C)ccc(C(N2CC(CNC(C3CCCC4CC34)=O)C2)=O)cn1 CCC(C(=O)NCCCN(C(=O)Cn1ccc(C(F)(F)F)n1)C)N(C)C c1(C(=O)NC2(CC=C)CCN(C(C3CCSC3)=O)C2)cccc2c1OCCCO2 C1(O)(CC(=O)OCC)CCN(Cc2cnn(C3CCOCC3)c2)C1 c1(C(C)C)nc2ccccn2c1NCC(C1CCN1C(C)(C)C)n1ccnc1 c1(C(=O)NCC2N(C(C3CCC(CC)O3)=O)CC(O)C2)nnn2ccccc12 C(=O)C(C(C)(C)C)C1CCC1.Cc1noc(Cl)c1CC(=O)NC.C1(F)CCC1 C1(N(C=O)C)CCN(C(=O)CC(=O)N(C)C)CC1.c1(OCC)cc(CC)on1 N1(C(CC(C)(C)O)=O)CCC2C(CCCN2C(c2cccc3c2CCC3=O)=O)C1 N1(C(c2ccc(=NC)[nH]c2)=O)CCC2CN(C(c3ccc(F)c(C)c3)=O)C2C1 S(=O)(=O)(c1cccc(Cl)c1)NC(C)C(N1CC2(OC(F)F)CC1C2)=O C1(NC2C(=O)N2)CCC=CCCC1.c1(C2(N)CC2)nccc(O)n1.c1ccc(N)cc1 N#CCCCCC(=O)N1CC2CCC2(CCNC(c2n[nH]cc2Br)=O)C1 c1(C(N(CCCCCNC(CNC(CC)=O)=O)C)=O)ccc(-c2nc[nH]n2)cc1 c1(NC(C(C2C3CC=CCC23)N(C)CC)=O)ccccc1CO c1(OC)cc(Cl)ccc1CN1CCCC(NC(c2n[nH]c(C)c2C)=O)C1 CN1CC2(CC2)CC1C(=O)NC(CCF)C(=O)NC1(CCCF)CC1 c1(NC(=O)CCC2CCCO2)cnc2sccn12 N1(C(=O)NCCc2nnc(CC)n2C)CCCC(N2CCCS2(=O)=O)CC1 c1(CC)cc(CNC(C)(C)CCO)ccc1C CC(C)C(C(=O)NCC1CC2CC2N1C(=O)CN(C1CCCC1)C)NC=O N1(C(C(CO)N(C)C)=O)CCC2CN(C(=O)CCSc3nnnn3C)CC12 O=C1CC(C(N2CCN(Cc3cccnc3)CC2)=O)CN1Cc1ccc(F)cc1 N1(CC)CC(C(=O)NCCC2CCCC2)CC1=O.C(=O)CN(C(=O)C)C C(CC(=O)NCCC(=O)NCC(C)CC)NC(=O)NC C(=O)(C(O)CCC(C)C)N(C)CC1CCN(C(Cn2c(C)cc(C(F)F)n2)=O)C1 C1(C)(NC(Cn2nc(C)c(Cl)c2)=O)CCN(C(=O)CCCCCF)CC1 C(=O)(C(F)(F)CO)NCC(C)CN(C(=O)CC(C)(C)c1ccccc1)C c1(OCC(=O)OC(c2ccccn2)C)cccc(N2CCCC2=O)c1 c1(CCC(=O)NC(C2N(C(C(COC)OC)=O)CCC2)C)cc(C)sc1C Cc1cn(C(C)(C)C(=O)N2CCC2CON)cn1 Cc1ccc2[nH]nc(CN3CC4CN(C(c5ccc(O)cc5Cl)=O)CC34)c2c1 Cc1ccccc1NC(=O)C(N1CCCC(c2ccc(O)cc2)C1)C1CC=CC1 C1(C)(C(NOCCN(C)C)=O)CN(C(=O)CC23CCCC2C3)C1 N1(C(C2CCCC(C(=O)OC)C2)=O)CCCc2cc(N(C)C)ccc21 C=C=CCCC(=O)NC(CNC(c1cn(CC(=O)N(C)C)nn1)=O)CC=C C1(CNC(CC(=C)C)=O)CCC2(CN(c3nnc(CC)s3)C2)O1 c1(CC)c(C(=O)NCC2CCCC2NC(=O)C(C)SC(C)C)csc1C C=CCC(CC)NC(=O)CC1CC1CNC(C1CC(F)(CF)C1)=O C1(C(=O)NC(CCN(C)C)C(N2C3CCC2COC3)=O)CC2CCC(C1)O2 c1(CC(=O)NC(C(=O)N(CCCOCC)C)CC2CCCC2)cccnc1C C(=O)(CCCCCN=[N+]=[N-])N1CCC(C(C)C)(C(=O)NCc2cnsc2)C1 N#Cc1cccc(CNC(C2C3CN(C(C4CC=CCC4)=O)CC23)=O)n1 N1(C(CCS(N)(=O)=O)=O)CCC2(CCCC2NC(c2nn[nH]c2Cl)=O)CC1 CCC(C)(CNC(C12CSCC1C2)=O)NC(=O)CC(=O)OC c1(N(C(C(OC)OC)C)C)ccc(S(=O)(=O)NCCC2=CCOCC2)cc1Cl N1(C(CS(N)(=O)=O)=O)CCN(C(c2cnc(C3CCC3)s2)=O)CC1C1CC1 C1(Cn2cc(C(C)OCC)nn2)CN(C(=O)CSc2cccs2)CCO1 N1(C(C2C(CC)CN(C(=O)C(F)C3CCCC3)C2)=O)CC=C(CO)CC1 CC(C)(C#N)CC(=O)NCC1COCC1NC(C1CCS(=O)(=O)C1)=O C1(CNC(=O)CCOc2ccccc2Cl)CC2CCC1N2C(=O)CC1CCCO1 Cc1cc(Br)cc(C(c2nnnn2C2CC2)NC(C)COC(C)C)c1F c1(NC(C2(C(C)(C)F)COC2)=O)ncc(C(=O)C2CC2)s1 N1(C(c2ccc[n+]([O-])c2)=O)CC2(CCCN2C(C2CC2c2ccccc2)=O)C1 C1(NC(Cc2c(C)nc(C)s2)=O)CCC2(CCN(C(C3CC3F)=O)CC2)C1 C=C(Cl)CC(C(=O)N1CCCC(C)(N(C)C)C1)NC(c1cc(C)c(F)cn1)=O CCC(C)CC(C)CC(C)C(=O)N1CC(CN)CCC1C C1(CN(C(Cc2ccc(C)o2)=O)C)CCN(C(=O)CCC2CCCCN2C)CC1 Cc1cc(C(=O)NCc2nnn(C)c2C(=O)N)ncn1.C(CC1CCC1)CO Cc1ccncc1C=CC(=O)NC1COCC1.C(=O)(CN(S(C)(=O)=O)C)N CC(C(=O)NCC=CCC(=O)NC1CC(n2cccn2)C1)OCC1CC1 S(=O)(=O)(c1ccc(N(C)Cc2cn(C)nn2)nc1)N1C(CCC)COCC1 N1(C(CC2(OC)CCC2)=O)CC(CO)C2(C1)CN(C(C1C=CCCC1)=O)C2 C1(C(=O)N(C)CC2CCCCN2C(c2cncc(C)n2)=O)(OC)CCSCC1 c1(OC)cccc(Cl)c1CC(=O)N(CC(C)CNC(C1CC12CCOCC2)=O)C CCCC(CCCNC(=O)CCC1CCCO1)NC(=O)CC(C)(C)SC N1(C(C(C)(F)F)=O)CCCN(C(=O)CSc2nnc3ccccn23)CCC1 Cc1cc(C)nc(N2CCC(OCCNC(c3cc(-c4ccco4)on3)=O)C2)n1 CCCC(C(=O)NCc1csc(CNC(C2(Cl)CC2(F)F)=O)n1)N(C)C CS(=O)CCC(=O)N1CCCC(CCNC(=O)CCc2cncs2)C1 C(CCC(=O)N1CCCC1CCCNC(=O)CC1CC(F)C1)=C(C)C CCCCCCC(=O)N(C1CCCCC1)CCNC(=O)C(CC)OC CC(C)C(C)C(C)CC(=O)N1CCC(NC(=O)C(C)C2CCCO2)C(CO)CC1 c1(N2CCN(C(c3cc(C)nc(NC(C)C)n3)=O)CC2)cc(F)c(F)cc1F CC1C(C)N(C)CCN1C(c1c(Cl)nc(Cl)n1C)C(=O)NCc1cccc(Cl)c1 c1(C(=O)NCC2(COC)CCN(C(c3cnco3)=O)C2)cnc2[nH]ccnc1-2 c1(C(=O)NC(CC=C)CNC(=O)C(C)(C)C2CC2)ccc(Cl)cc1 C(=O)(CS(=O)CCC(F)(F)F)NC(CC)CNC(=O)C=C1CCCCC1(C)C C1(C(N(CC(=O)N(C)C2CC2)C2CC2)=O)C(C)(C)C1(F)F c1(CC(=O)NCC2(C)CCN(CC3CC3)CC2)ccc(C#N)cc1F N1(C(c2cc(C)sn2)=O)CCCCC(CCC(=O)N(C2CCCOC2)C)C1 C(=O)(C1(C)CCn2c(C)nnc21)NCCCC(CCC)NC(c1csc(C)c1)=O C1(NC(c2cncc(COC)c2)=O)CCN(C(=O)C)CC1F.C1CC(F)(F)C1 CC1C(NC(C2(NC(=O)C(C)n3ccnc3)CCN(C)C2)=O)CCN1C c1(OC)cc(NC(=O)C(=O)NCCc2nc(C(C)C)cs2)cc(OC)c1O CCCCC(CC)C(=O)N1CC(CNC(c2cncc(OC)n2)=O)(OC)C1 c1(NCc2cc(CC)[nH]n2)cc(NCCn2ccc(Br)n2)nc(C)n1 c1(-n2c(C)nnc2)ccc(C(=O)NC2CCC(NC(=O)C(C)C3CC3)CC2)cc1 C1(C(=O)OCC)CN(CC(=O)N)CC1.c1ocnc1C(C)C.[nH]1cccn1.C C1(O)(CC#C)CC(C(=O)NC(CNC(=O)CC(C)n2cccn2)CO)C1 CC1CN(C(c2csc(S)n2)=O)CCC1CNC(=O)C(C)N(C)C C#CCC(O)C(=O)NC1CCCCC1C(=O)N(C)CC1COC(=O)N1 C1(CNC(C=C(CC)C)=O)CC(C)(C)CN1C(c1ccc(O)c(Br)c1)=O c1(COCC)nc(N2CC(C)(C)CC2CNC(=O)CO)cc(Cl)n1 Cc1[nH]c2ncccc2c1C(=O)NCCOC1CN(C(C2CC23CC3)=O)C1 C1(C(CNC(C2(C=C)CC2)=O)NC(=O)COC)CCCCC1 N1(C(C(C)CO)=O)CCC(C)(NC(=O)CC(c2ccc(F)cc2)C)C1 C1(CC)CCN(C(=O)CN(CC(C)(C)C)C)C(C(=O)NCC(O)CCO)C1 N1(C(C(COC)O)=O)CC2CCC(NC(=O)C=Cc3ccccc3OC)(C2)C1 CC(C)CC(CNc1ccc(C(=O)O)cn1)NC(=O)OC(C)(C)C Cn1cnc2sc(C(=O)NCCC3CCN(C(=O)C(C)(C)C4CCC4)C3)cc12 CCC(C(=O)N(CC)C1CC1)C(C)(C)CC.C1(CC=O)CCCC2(CCC2)O1.N C12(NC(C(CC)NC(N)=O)=O)CC1CN(C(=O)CCC13CCC(CC1)C3)C2 C12(CNC(=O)CN3CCCS3(=O)=O)CCC(CC1)N(C(c1ccccc1Cl)=O)C2 Cc1ccc(C(=O)NC2(CCO)CN(C(C3CC4(CCC4O)C3)=O)C2)cc1F C12(C(N3CCCN(C(CCN4C(C)CCCC4)=O)CC3)=O)CCCC1CC(=O)C2 C(=O)(NNC(=O)c1ccccc1)C1CCN(C(=O)OC(C)(C)C)C1 N1(C(c2cnc(CC)[nH]2)=O)CC2CC(NC(c3cncc(OC)c3)=O)CC(C2)C1 C1(S(=O)(=O)N2CCCCC2CSc2ncccc2C(=O)O)(CC=C)CC1 c1(OC)cc(NC(C2CCC23CCOCC3)=O)c(C(N)=O)cc1OC O=C(C1CCCc2nncn21)NC1(CO)CN(C(c2cccc3cc[nH]c23)=O)C1 C(N=c1[nH]c(=NCC2CCCCC2)c2[nH]ccc2[nH]1)C1CC(=O)N(C2CC2)C1 Cc1nn(CCC(=O)NCC2COCC2)c(C)c1C.C(=O)(C(C)S(C)(=O)=O)N Cc1ccc(F)c(C(=O)NCC(CNC(c2cc(Br)c(C)o2)=O)CO)c1 c1(C(=O)NCCC2CN(C(CCc3nnc(C)o3)=O)C2)c[nH]ccc1=O C1(C(=O)NCC(C)CN(C)C(c2nc[nH]c2C(C)(C)C)=O)CCCCN1N=O C#CC1CC2(CC(C(=O)NC3CN(C(=O)C(C)S(C)(=O)=O)CC3(C)C)C2)C1 c1(OC)c(-c2ccc(CN3CCCC(N(C)C)C3)c(F)c2)cccc1F CC1(C)COC(CC(=O)NC2CC(NC(=O)CCC(=O)c3cccnc3)C2)C1 c1ccc2ccccc2c1.C(=O)(CC)NC(CNC(C1C(C(=O)OC)C1)=O)C c1(C(=O)NCC2N(C(CSCCC)=O)CCCC2C)cc(F)c(F)cc1O C1(C(=O)NCC(CC)NC(=O)CNS(=O)(=O)C2CC2)CCC12CCC2 CCCC(C)C(=O)NCCCCCNC(=O)C(c1cccn1C)=O C1CCN(C(C2(c3ccsc3Cl)CC2)=O)CC1.N1(C(C2C(OC)C2)=O)CCC1.O C1(NC(CN(C)CCO)=O)CN(C(c2ccncc2Cl)=O)C2(CCCC2)C1 Cc1ccncc1CN(C(=O)C)C.C1CCN(C(C2CCN2C(C)(C)C)=O)C1 Cc1n[nH]c(C)c1C(=O)NC1CCC(C)(CNC(=O)CC)C1.C1COC1.O c1(CCC)ccc(CCCC(=O)NCC2CCCCN2Cc2nccn2C)cc1 CCS(=O)(=O)CCN=c1cc[nH]c(-c2ccc(SC)cc2)n1 C1(NC(C(C)(C)SC)=O)CN(C(C2(O)CCCC(C)(C)C2)=O)Cc2nccn2C1 C1(CCC)(C(=O)NC2CC(CNC(C3OCC3(C)C)=O)C2)CCNC1=O c1(C(N2CCCC2)=O)cnc(O)c(Br)c1.C1(CC)CCCC1C(=O)N(CC)C CCCC(CNC(=O)CC1CCN(C)C1=O)C(=O)N1CC2(CC2)CC1C N1(C(c2nc(C)[nH]c2Br)C(=O)NC(CC)C)CCC2(CC1)CC(O)(C(F)(F)F)C2 C1(CC(=O)NC2CN(C(C3(CC(F)F)CCC3)=O)C2)CC2COCC12 N1(C(Cn2ncc(C#C)c2)=O)CCC(C2CC2)C1.N(C)(S(N)(=O)=O)CC(=O)N CC1CC(NC(=O)C2CC2)CN(c2nccc(N3CCCCC3)n2)C1 c1(C(N2C(CC(NOC(C(=O)OC)(C)C)=O)CC(F)C2)=O)ccnc(C)c1C C1(=CCNC(CC=CC)=O)CCN(C(=O)COC2CCN(C)CC2)CC1 Cc1cc(C(F)F)n(CC(=O)NC2CC23CC(NC(=O)C=CS(C)=O)C3)n1 c1(CC)cnc(C(=O)NC2CN(C(c3nc(O)sc3C)=O)C3CC23)cn1 C(=O)(Nn1cnnc1C)C1CCN(C(c2c(C)cn(C)n2)=O)C(C)C1 C=CC1(CC(=O)NCC2(CC)CCCC2)CN(C(=O)CC(C)O)C1 c1(-c2nc(C(N3CCC(F)(Cc4cn(CCO)nn4)C3)=O)[nH]n2)ccccc1Br N1(C=O)CC(F)CC1C.Cc1cnn(CCC(=O)N2CC(C(O)C=O)C2)c1 C1(CC(C)NC(C2C(C)CN2C(c2csc(F)c2)=O)=O)CCCCO1 C1(Cc2nc(-c3c(C)cco3)nn2-c2ccc(C)cc2C)CC12CCC1(CC1)CC2 N1(C(CC2(N(C)C(C3CC3(F)F)=O)CC2)=O)CC(CO)CC1CO C1(C(F)(F)F)(C(=O)NC(=O)CNc2nccs2)CC2(CCC2)C1 Cc1ccc2nc(C(=O)NCCNC(c3ccc(F)cc3)=O)cn2c1 C=CCC(C(=O)NCC1CC(F)(F)C1)NC(C)=O.C(=O)CCS(C)=O.C C1(C(=O)NC(C2CCN(C(C3CC4(CSC4)C3)=O)C2)C)CCC(N=[N+]=[N-])C1 Cc1nn(C)cc1CC(N1CC(C(C)(C)O)(CNC(=O)CCF)C1)=O c1(OC)cc(C(c2nnnn2C2(C)CC2)NCc2n[nH]c(C)n2)ccc1Br c1(C(N)=O)ccc(CC(N2CCC2CNC(=O)C(C2CCOCC2)O)=O)cn1 C1(C(=O)NCCC2(C)CCN(C(c3cccs3)=O)C2)(OC)CCC(C)(C)C1 N1(C(C(C=C=C)C)=O)CCC(C(=O)NC(CC2CC2)C2CC2)C(C)(C)C1 C(=O)(C(CC)C(C)(C)CC)NC(C(=O)NCc1c(C#C)cccc1)(C)CO C1(CCOC)(NC(C2CC(C)CO2)=O)CCN(c2ncncc2C)C1 C(=O)(C=C1SCC(=O)N1C)N(C(C)CNC(c1ccncc1N(C)C)=O)C C1(NC(=O)Cc2n[nH]c(C3CC3)n2)CC2(C1)CC2NC(=O)C1=C(Cl)CC1 C1(C(N2CC(CCNC(COCCCC)=O)OCC2)=O)COC2(C)CC1C2 c1(SCC)cnc(O)c(C(=O)N(C2CN(C(C3CCN3CC)=O)CCC2C)C)c1 C(C)(CCCCN=c1nc(C(C)C)[nH]s1)NC(c1cc(C)nc(O)c1)=O Cc1cnccc1CC1(C(=O)NCC)CC1.C1(C=O)CCCNC1.C1CC1.N CCCCCCCC(=O)N1C2CCC1C(NC(c1ccc(CC(C)C)cc1)=O)C2 C1(n2cc(CN(C)C)nn2)CCCN(c2ncccc2Cl)C1 c1(C(=O)OCC)sc2[nH]c(N(C3CCN(CCO)C3)C)nc(=O)c2c1C Cc1cccnc1C(N1CCC(NC(c2cncc(Cl)c2)=O)C1)=O c1(CC(C)C(=O)NCC(CNC(=O)CCC(F)F)CO)cccc(F)c1 N(C(=NCCN1CCOCC1)NCC(C)C)CC(c1ccccc1C)OC C1(NC(c2cnc(C(C)C)[nH]2)=O)CC2CN(C(=O)Cc3cn(C)nn3)CC2C1 c1(C(N(CCCCNC(C2C3COCC23)=O)C)=O)c(Cl)cnn1C Cc1nc2c([nH]1)CC(C(=O)N(CCNC(=O)CCC#N)Cc1ccccc1)CC2 CN1CC(CC(=O)NCC2CCC2)C(O)C1.C1(C=O)CC(=C2CCC2)C1.N c1(C(=O)NCCCNC(CCC(C)OCC)=O)c(N)cc(Cl)nc1Cl Cc1ccc(CC(N2CCOCC2CNC(=O)CCCn2ccnn2)=O)cc1C CC1C(NC(=O)C(C)(C)CNC(=O)CC2CCCCC2C)CCCC1C C1(C(N(CCC(=O)O)CC=C)=O)CN(C(=O)Cc2cncnc2O)C(C)(C)C1 C1(NC(C(F)=C(C)C)=O)CN(C(=O)CC2(O)CCCCCC2)CCC12CCC2 c1(C(N2CCCC(C(C)(C)O)C2)C(=O)N)ccc(C(F)(F)F)c(Cl)c1Cl.CCC c12ccc(N(C3CCNCCC3C)CC)cc1N2.C1(NS(C)(=O)=O)CCCC1 CC(C)(C)CC(F)C(=O)NC1CCCC1C(=O)NCC(C)(C)C1CCC1 C(CCS(=O)(=O)c1cc(Cl)ccc1Cl)N(C1CCCC1(C)C)C CC(C)(CC#N)C(=O)NC1CCC1NC(=O)CCCc1cccnc1 CC1(C)CC(C(=O)NC2CC(NC(c3c(Br)ccc(N)c3F)=O)C2)=NO1 CCCCC(CO)NC(N1CCCC(C(N2CCCCCC2)=O)C1)=O c1(OC)ccc(-c2cn(CC(F)(F)CCNC3CCCN3C=O)nn2)cc1F N1(C(C2(NC(CSCC)=O)CSC2)=O)CCCC(C(C)(C)C)C1 CC1CC(NC(C2CCCCN2C)=O)CN1C(c1cnn(C2CCCC2)c1)=O CC1CC(NC(c2cccnc2S)=O)CN(C(c2ccnc(C3CC3)c2)=O)C1 C1(CNC(CC(C)C)=O)CCN(C(C2CCC2c2nncn2C)=O)CC1 n1(CC(=O)N(CC(=O)NC)C)ccc2ccc(Cl)cc12 C#CCC(C(=O)N(C1CN(C(=O)CCC)C1)C)C1CC1 c1(C(=O)NCCN(C(=O)CCc2cn[nH]c2)CC(C)O)nccn2nccc12 CCC(CC(=O)NCC1CCCC1NC(C1(C(C)C)CC1)=O)OC O=C(C1c2c[nH]nc2CN1C(c1ccnn1CCF)=O)NCC1(CO)CCC1 N1(C(c2n[nH]c(CC)c2C)=O)CCOCC(NC(=O)C=CC2CC2)C1 C1(CNC(c2c(SC)n(C)nc2)=O)CCC(C)N(C(C2CCC(C)CC2)=O)C1 Cc1ccc(C(C)CC(=O)NC(C2CN(C(c3ncnn3C(C)C)=O)C2)C)cc1 Cc1cc(C(N2CC(O)(CNC(c3cc[nH]c3C)=O)C2)=O)cc(C)n1.C1CC1 c1(C(=O)NC23CCC(C2)N(C(=O)Cn2cnnc2)C3)n[nH]c2c1CCCC2 c1(N2CC(NC(=O)Nc3ccccc3Br)C3(C2)CC3)ncnc2cc(F)ccc12 N1(C(C2ON=C(C)C2)=O)CCN(C(=O)C(Cl)=CCl)C(c2cn[nH]c2)C1 CC1(CNC(=O)Cc2ccco2)CCC(NC(=O)C=Cc2ccco2)CC1 C1(C(=O)NC2CC(NC(=O)CCOC3CC3)C2)CC2CC(O)CC(C1)C2 C(N=c1cc(C(F)(F)F)c(Cl)c[nH]1)c1c(NC)nccc1 c1(C(N2CC(CNC(c3cc(C)oc3)=O)N(C)CC2)=O)cnc2ccccc2n1 c1(C(=O)NC2CN(C(C3C(CCC)CCC3)=O)C(C)C2)cccc2nn[nH]c12 C(c1ccc(C)c(C)c1)=CC(=O)NCCCC.c1(C=O)cccc(C(C)=O)c1 CCCCC(O)C(=O)NCC1(O)CCN(C(c2cccc(CS(C)=O)c2)=O)CC1 c1(NC(C2N(c3ncc(CC)cn3)CCC2)=O)cc(OC)c(OC)cc1I C#Cc1ccc(F)c(C(c2nnnn2CCC2CC2)NCCc2ccsc2)c1F C(=O)(CCCC(F)(F)F)NC1CCC(C)(NC(CNS(CC)(=O)=O)=O)CC1 C1(C=O)CCCCCS1(=O)=O.N1(C(c2ccn(CC#N)n2)=O)CC2CC1C2C.N C(CCCCCC(=O)N1CC=CC(NC(=O)Cc2c[nH]c3ncccc23)C1)SC O=C(CS(=O)(=O)Cc1cccs1)NCCOCC.C1(C=O)CCC(O)C1.N CC(c1cccc(Br)c1)=CC(=O)NCC(C)(C)NC(C1CC(CF)C1)=O N1(C(C2CCN(C=O)C2)C(=O)N)CCC(O)C(F)(F)CC1.C(C)(C)C.CCC C12(C(=O)Nc3cn(CCC)nc3)CCC(CC1)N(C(=O)C(=O)NC(C)C)C2 C=CCCCN=C(NCC(=C)C)NCC1(c2ccccc2)CCC1 C(c1ccc(Cl)nc1)=CC=O.N1(C(C2(CC)CCC2)=O)CC(O)(CC)C1.C N1(C(C(C)CC2CC2)=O)C2CCC1CC(NC(c1nc(O)nc(O)c1F)=O)C2 C1(F)(C(=O)NCC(C(C)C)(C)F)CCN(C(C2CC(O)CN2C)=O)CC1 c1(C(N2CCC(C(N3CC4C(C(N)=O)C4C3)=O)C2)=O)cccc2ccoc12 CC(C)(C)CC(F)C(=O)NCCC1CCCN(C(c2ccc(Cl)c(O)c2)=O)CC1 C1(CNC(C2C(=C)C2)=O)CN(C(=O)CO)CCO1 C1(CNC(C2C(=O)NCC2)=O)CCN(C(C2(CC(F)F)CCC2)=O)CCC1(F)F N1(CC)CCCC(C(=O)NC2C=CC(C=O)C2)C1.c1cc(C(C)(C)C)no1.N c1(C(C)=O)cc(CCC(N2CC(O)CC2c2nc[nH]n2)=O)oc1C Nc1cnc(Cl)cc1C(N1CC(CO)(NC(=O)Cc2ccoc2)C1)=O c1(C(=O)NCC2(C)CC2)cccc(C(F)(F)F)c1Cl.c1cc(CCBr)ccn1 C12CCN(C(c3cccc(-n4ccnn4)c3)=O)CC1C2.C1(C=O)CC(=C2CC2)C1 c1(NCCn2c(CC)ncc2)nc2c(c(=NC3CCCCC3SC)[nH]1)COCC2 c1(CO)nc2ccccc2c(=NCCc2cccc(F)c2)[nH]1 C1(C#N)(C=O)CCOCC1.CC(Cn1cccn1)C(=O)NCC1CC1(F)F.C C1(NC(C2CCS2(=O)=O)=O)CCCCC1Sc1ccccc1Cl CC(=NOCC#N)C(=O)N1CCC(C(=O)NC2CCN(C(C)(C)C)C2)O1 N1(C(C(c2ccccc2)OC)=O)CCCC(N(C(=O)Cc2cnn(C)n2)C)CC1 Cn1cc(C(=O)NCC(C2CCOC2)NC(=O)CCc2cscn2)nn1 Cn1[nH]c(=NC(=O)C2CC2NC(c2sccc2F)=O)c2cc(Cl)ccc12 C(=O)(C1CCCc2nc[nH]c21)NC1CC(NC(c2n(C)nc(C3CC3)c2)=O)C1 CC1CN(C(=O)CN(c2ccncc2)C)CCC1N(C(=O)C(C)(F)F)C C1(OC)CCN(C(c2coc(C(C)(C)C)n2)=O)CC1.C1(C=O)CCC(=O)N1.C c1(CC(=O)NCC(C)(C)NC(Cc2cc(C)sc2)=O)cc(O)ccc1Br C1(CC)CN(C(=O)COc2ccccc2C)CCN1C(=O)CN(C)C1CC1 CC(CNC(C1CCCC(NC(c2cccn2C)=O)C1)=O)S(N)(=O)=O N1(C(c2ncc(-c3cn(CC)c(=O)cc3)nc2)=O)CCCCC(C)(F)C1 C1(C(N2CCC(N(C(=O)C=Cc3ccsc3)C)C2)=O)CC2CCC(C1)C2 C1(C(=O)NC2(C)CC(NC(CCCN(C(C)=O)C)=O)C2)CCC2(CCOCC2)O1 C1(CCC)(NC(C(CC=C)C)=O)CCCN(C(=O)C(c2cnn(CC)c2)=O)C1 c1(OCc2cn(C)nn2)cccc(NC(c2n[nH]c(C(C)(C)C)n2)=O)c1 C1(CNC(C2CC(=C)C2)=O)CC(C(=O)NCC(CO)C(C)CC)=NO1 c1(C(=O)N)cc(S(C)(=O)=O)ccc1Cl.C(CSC)(C(=O)NCC(C)C)OC N1(C(Cc2c(C)n[nH]c2C)=O)CC2CCOCC2(NC(=O)CCc2cnn[nH]2)C1 Cn1cc2c(C(N3CCC4CN(C(C5C=CCN5)=O)CCC34)=O)cccc2n1 C1(CC(=O)NCC2CCCC2)(CC)CCOCC1.n1(CC(=O)N)cccnc1=O c1(CC(=O)N(C(C)CCNC(c2cnn(CC(F)F)c2)=O)C)cccc(F)c1 c1(NC(CC2(C)CN(Cc3c(F)ccc(F)c3F)C2)=O)nc2cc(Br)ccc2s1 C1(C)(NC(C2C(OCC)CC2)=O)CCN(C(c2ncncc2Cl)=O)CC1 C1(NC(CCC(C)O)=O)CN(C(=O)CN2CCS(=O)(=O)CC2)CCC1C Cc1nc(CC2CCNC2)sc1C(=O)NC(C1CCN(C)CC1)C N1(CC)CCOCC1C(=O)NCC1CCCC1NC(c1cccnc1O)=O N1(C(c2cncc(C(C)(C)C)c2)=O)CCCC(CO)(C)C1.C1(C(=O)N)CC=CC1 c1(NC(C2(C)N(C(C3C(C)C3)=O)CC2)=O)nccc2scc(Br)c12 Cc1nc2[nH][nH]cc-2c(=NC2CCN(C(=O)CN3CCCNC3=O)C(C)C2)n1 C(C(C(=O)NC(C)Cc1cc(C)[nH]n1)NC(=O)CCC1CCCC1)OC c1(NC(C(C)SCCCC)=O)ccc(NC(=O)CC2CCSC2)c(C)c1 S(=O)(=O)(c1cnn(C(F)F)c1)NC(c1ccc(C)cc1)c1cccc(Cl)c1 N1(C(CCC2CCCN(C)C2)=O)CCCCCC(NC(c2ccnnc2S)=O)C1 C=CCCC(C)(C)C(=O)NC(CCC)CC(=O)NC(c1cccnc1)CO C1(C=O)OC(C)(C)OC1(C)C.c1(CC)cc(C(=O)NC2CCC2)cc(O)n1.C c1(NCC2(NC(=O)C=CI)COC2)ncnc2sc(C(F)(F)F)nc12 N1(C(C2(NC(C(C(CC)C)=O)=O)CCC2)=O)Cc2nncn2C(C)C1 C1(CNC(c2ccncc2O)=O)CCCCC1NC(C12CC(F)(C1)C2)=O N1(C(CC=C=C)=O)CC2(CCC2)CC1C(=O)NC(CO)C(N)=O N1(C(C(C)(N(C(C2ON=C(CC)C2)=O)C)C2CC2)=O)CC2CCCCC12C Cc1c(C(N2CCN(C(=O)CC3(O)CC3)CC2C2CC2)=O)[nH]c2c(Cl)cccc12 C1(NC(C=COCC)=O)COCCN(C(C2CCCN2C(C)=O)=O)C1 c1ccc(C(N)=O)cn1.N1(CC)CCCC1C(=O)NC(C)CC.C(=O)(C)N N1(C(c2nc(C(=O)OC)sc2)=O)CC=CC(NC(=O)Cc2ccnc(O)c2)C1 C1(OC)CC(CC(N2CCC(C)CC2)=O)C1(C)C.C1(C)(CC=O)CC1(F)Cl.N N1(C(=O)CCSc2ccccn2)CCN(C(=O)C2=CCCOC2)C2CCCCC12 C1(C(N2CCC(C)(C)C2)=O)(CC)CNC(=O)C1.c1(C=O)ocnc1C1CC1 N1(C(c2cc(SC)c(C)o2)=O)CCC(NC(=O)CC2CCCOC2)C1(C)C CC(C(=O)N1CCCC(F)(CNC(c2n[nH]cc2C2CC2)=O)C1)P(C)(C)=O Cc1cc(CC(=O)NC2CN(C(=O)CC3CC(=O)C3)CCC2C)ccc1F C(=O)(C1=CC2CCCCC12)N1CCC(CN(C(c2nc(C(C)C)sc2)=O)C)CC1 c1(NC(COCCOCC)=O)cccc(NC(=O)C(CC)c2cccnc2)c1 N1(C(C2(OC)CCC23CCC3)=O)CC2CC(NC(=O)C#CC3CC3)CC1C2 C12(C(N(CCn3ncc(C)c3)C)=O)CCN(C(=O)C(C)(C)C(C)C)CCC1C2 N1(CCC)CCCCC1C(=O)NCCCN(C(=O)C(F)CC1CC1)C(C)C C1(C(=O)NC(CNC(C(CC2CCC2)OC)=O)(C)C)C(C)(C)C1(F)F c1(C(=O)NCC(CC(=O)N2CCC(OC(C)=O)C2)O)c(C)ccnc1C c1(OCC#N)ccccc1C(=O)NCC(CNC(=O)CCC1CC1)CO C1(C(C)OCCC(C)C)CCN(C(=O)NC2(C)CC2(C)C)CC1 Cc1cccc2[nH]cc(C(N3CC(C)CN(C(=O)CNC=O)CC3C)=O)c12 C(=O)(C(F)(F)c1csc(C)c1)NCCN(C(=O)Cc1ccns1)CC C1(C(=O)N)CC2COCC2N1C=O.c1(C(=O)OC)cccc(N)c1.C(C)(C)C C1(CC)CCN(C(=NCC(=O)OC(C)(C)C)NC(C)CC)C1 c1(C(N2CCNC(=O)CC2(C)C)C(=O)NCC(C)C)n[nH]c2cc(Br)ccc12 c1(C(N2CC(C(C)(C)O)C2)=O)c(C)ccnc1O.Cc1ccnnc1C(=O)NC C1(N(C(C(=O)NC(C)C)=O)C)CCCN(C(C2CN(C3COC3)C2)=O)CC1 C=CC1(C(=O)OCCc2ccc(CC(=O)OC)cc2)CCCCC1 Cc1csc(CNC2CCCC2C(=O)NC2CC2)n1 C(C1CN(C(c2nn(C)cc2C)=O)Cc2ccccc21)NC(C(CC)C(C)O)=O C(=O)(C#CC1(C)CCCO1)N1CCC(C2CC2)C1.c1(OCC)sccc1C(=O)N N1(C(c2c(CC)c(F)ccc2)=O)CCCC(C2CCCN(C(=O)CO)C2)C1 c1(C(C=O)N(c2ccc(Br)c(C)c2)CC(C)C)c(C)nn(C)c1C.C=C(C)C CC(C)(C(=O)NCCC1CCN(C(=O)CO)C1)n1cc(Cl)cn1.C1CCOCC1 CC(CS(C)(=O)=O)N(C(=O)C(=O)Nc1ccccc1N1CCCCCC1)C N1(C(CNC(C2(CCC)CCC2)=O)C)CCN(C(=O)CCc2ccc[nH]2)CC1 C1(CC=C)(C(=O)NC2CC(F)(C)C2)CCCCC1.c1(C=O)ccc(O)nc1.N CC1CSCCCN1C(=O)C(Cn1cncn1)NC(C1CCOCC1)=O Cc1cc(C)n2ncc(C(N3CC4CC(NC(C5(F)CC5C)=O)C3C4)=O)c2n1 Cn1cnc(NCC2CCC(NC(c3occc3Br)=O)C2)cc1=O CC(C)C#CC(=O)NCC1(NC(=O)Cn2nnc(C3CC3)n2)CCC1 c1(N2CCC(Cn3ncc(C)c3)C2)cc(NCC(=O)NC2CCOC2)ncn1 CC(C)(O)C(F)(F)CNC(c1ncoc1CNC(c1cscc1Cl)=O)=O N1(C(C(Cn2ccc(C)n2)C)=O)CCN(C(=O)CCCc2ncco2)CCC1C C(=O)(CC1=CCOCC1)N1CCCC(NC(CC=CCC)=O)(COC)C1 C1(C(=O)N)CC(=O)c2ccccc2C1.Cc1coc(C=CC(N2CCC2C)=O)n1 N1(C(C2C(CC)C2)=O)CCN(C(=O)CC2CC3CC3C2)CC1CCO C1(CNC(=O)CSCc2ncc[nH]2)CN(C(c2ccnnc2)=O)CCCO1 CCCCCC(C)CC(=O)NC1CC2CC(NC(C3CS(=O)(=O)C3)=O)C1C2 N1(C(c2c(CC)nco2)=O)CCC2CCCC12C(=O)NCc1ncc(CO)o1 CC(C)(F)C(C)(F)CS(=O)(=O)N.N1(C2(CN)CC2)CCOCC1 C(=O)(CN=c1[nH]c(C)cc(=NCCc2ccc(Cl)c(F)c2)[nH]1)NCC C(=O)(C(C)C(C)(F)F)NCC1CN(C(C(c2cccc(OC)c2)OC)=O)C1 N1(C(CC(C)C)=O)CCC(F)(CNC(C2CC2(C)C=O)=O)CC1.C(C)(C)C c1(C(=O)NC(C(=O)NC2(CCCF)CC2)C2CCC2)c[nH]c(=S)cn1 CCS(=O)(=O)c1ccc(C(=O)NC)cc1.C1CCCN1C(C1CC(C)(C)O1)=O.C c1(C(N2CCN(C(C(C)OCC)=O)CC2)=O)cc(NC(=O)OC)ccc1F c1(C(N2CCC(N(C(CSS(C)(=O)=O)=O)CCO)C2)=O)ccc2n[nH]cc2n1 c1(C(N2C(C3(C(=O)NC(c4cnsc4)C)CC3)CCC2)=O)cnn(C)c1C#N c1(C(=O)NCC(C)CN(C)C(C2(O)CCSCC2)=O)cnc(C2CC2)nc1O CCC(O)C(F)(F)C(=O)NCC(Cc1ccccc1)N(C(=O)Cn1cccn1)C N1(C(c2cnn(C)c2N)=O)CCC(NC(=O)C(C2CCCCCCC2)O)C(O)C1 C1(O)(C(C)NC(CSCCOC)=O)CCN(C(=O)CCSCC(C)C)C1 c1(C(C)OC(C2(OC)CC(C[Si](C)(C)C)C2)=O)ccc2nc(C3CC3)[nH]c2c1 C1(CNC(CNC=O)=O)CCCC2(CN(C(=O)C(C3CCCCCCC3)O)C2)O1 N1(C(C2CNC(=O)O2)=O)CCCCC1CCC.c1(C(=O)N)ccc(SC(F)(F)F)o1 C(=O)(CC(C)(C)C)NC1(CC=C)CN(C(=O)CNC(=O)C(F)(F)F)C1 C(C)(C(C(=O)NC1(C(O)CO)CC1)C(C)C)NC(C(=O)NCC)=O c1(C(=O)N)ccc(Br)c(Cl)c1Cl.C12(NC(C3(C(C)C)CCC3)=O)CC(C1)C2 CC1(CO)CCN(C(C2CC23CC(NC(C2C4CC(=O)CC24)=O)C3)=O)CC1 C1(N(C)C(c2cccnc2CNC(=O)Cc2cnoc2)=O)CCOC(C)(C)C1 N1(C(C(n2nc(C)c(OCCOC)c2C)C)=O)CC2CC(C2)c2ccc(Br)cc21 C1(NC(c2n(CC)nc(C)c2)=O)CCC2(CCN(C(c3cc(O)ncn3)=O)C2)C1 c1(C(CC)COC)nc(CC2CCCC2)nn1-c1nc(Br)nn1C Cc1cc(C(=O)N(C2CCN(C(C3CC3CC(C)C)=O)C2)CCO)nnc1C Cc1ccc2c(c1)C(c1nc(CCN(C)C)nn1-c1cc(F)ccc1C)C2 C(=O)(CCC(CC)NC)N(C1CCN(C(CN(CCCCCC)CC2CC2)=O)C1)C N1(C(=O)CCc2ccncc2)CCN(c2cccc(F)c2)C(=O)C1 c1(C(=O)OC)cc(S(=O)(=O)NC2CN(Cc3cnc(Cl)c(C)c3)C2)ccc1F c1(OCC)ccc(CNC(COC)C(=O)O)c(F)c1F N1(C(c2cn(CC)nn2)C(=O)NCCc2cccnc2)CC(C)C(O)C(C)C1 C1(NC(C(=O)NCC)=O)CCC2CCN(C(=O)Cc3cc(OC)ccc3F)C1C2 c1(C(N(C2CCCN(C(C3CC3C(F)F)=O)C2)C)=O)ccc([N+](=O)[O-])cc1.C C(=O)(C1CCCc2nn[nH]c21)NC(C1CCN1C(c1ccc2c(c1)OCC2)=O)C C(=O)(C1=NN(C2CC2)C(=O)CC1)N1CCC(NC(C(C)C(F)F)=O)C1 N1(C(=O)Oc2ncc(OC)nc2)CC2CC1CN(C(=O)OC(C)(C)C)C2 c1(C(N2CC(NC(C3(C4CC4)CC3)=O)CC(C)C2)=O)ccc2c(c1)COCO2 C1(C(=O)NOC2CC3CCC2C3)CCCCCN1C(c1ccc(CO)cc1)=O CC1(CNC(=O)CCOCC(F)F)CC(F)(F)CN1C(c1cccnc1S)=O Cc1cccc(CNC(=O)CC2(NC(=O)Nc3cccc(C)n3)CC2)c1 C(=O)(C1=CCCN(C(C2CCCCN2C(C)=O)=O)C1)N1CC2C(CC)(C2)C1 C12(NC(c3c(CC)nns3)=O)CCCC1(F)CN(C(C1CCN(C)C1C)=O)C2 c1(OC)c(C(=O)NCC(C2CCCC2)NC(C2(OC)CC2)=O)ncnc1C c1(C(N2CC(C(C)NC(c3cc(OC)ns3)=O)C2)=O)cccc2oc(C)cc12 CC1C(NC(C2(O)COC2)=O)CCCN1C(c1ncc(Br)cn1)=O C(=O)(C(C)CC(F)(F)F)NC1CC(F)(CNC(C(CC(C)C)OC)=O)C1 CC1CCCCC1(C)NC(=O)CC(F)(F)c1cccnc1Br N1(C(c2cc(C(N)=O)[nH]n2)=O)CC2(CCC2)CC1CNC(c1occc1F)=O c1(C(N2C(CN(c3nccc(CO)n3)C)CCCC2)=O)cncc2ccsc12 N1(C(C(C=C)C)=O)CCCC1(C(N1CCCCC1CC)=O)C(C)C CCC(CCC(=O)N(C)Cc1cncs1)NC(c1ccc(C#N)o1)=O c1(CCNC(CC2(C)N(C(c3cc(C(C)C)on3)=O)CC2)=O)cccc(O)n1 c1(NC(C2CCN(C(=O)OC(C)(C)C)CC2)C)ccc(C#N)cc1[N+](=O)[O-] C1(CC(=O)NCC(c2ccccc2)C)CCCN(C(c2ccon2)=O)C1 Cc1nn(C)c(C)c1C(C)C(N1CCN(C(C2C3COCC23)=O)C(C)C1)=O C(C(O)CS(=O)(=O)c1cccs1)NC(=O)N=c1[nH]ncn1-c1ccccc1 c1(-c2c(C(N3CCCCC3c3nccs3)=O)n[nH]c2)cccc(OC(F)(F)F)c1 C1(C(=O)NCCC2CCOC2)(CC)CCN(C(C2CCC2(F)F)=O)C1 C1(C(N2CCC(c3ccccc3C)C2)=O)(OCC)CC(F)(F)C1 c1(NCCN2CCN(C)C(=O)C2)[nH]c(=NCC2(C)CCOC2)nc2sccc12 C1(CCOCC2(CC)CC2)(COC)CCN(C(C2CC=CC2)=O)CC1 c1(C(=O)NC2(CNC(C=C(COC)C)=O)CCOCC2)ncc(OC)nc1 c1(NC2C(CC)CN(C(=O)C(F)OC(F)(F)F)CC2)ncnc2c1CCC2 C12(NC(c3cc(Cl)c[nH]3)=O)CC(C(=O)NCC3(O)CCSC3)(C1)C2 C1(NC(c2cccc(CC)c2)=O)CCC12CCOCC2.C1(C(=O)N)CC(F)(F)C1 C=CC1(C(=O)NC2CC(N(C)C(c3cnc(CC)[nH]3)=O)C2)CCCCC1 CC(C(CO)NC(=O)C=CC(C)(C)C)NC(=O)CSCC(F)(F)F C(C)(C)(CC(F)C(=O)N1CCN(C)C(C)(C)C1)NC(c1c(C)cc(F)s1)=O N1(C(c2cccc(C#C)c2)C(=O)NCC(C)C)CCC2(CCCC2)CC1 Cn1cc(C(N2CC(CCO)(NC(=O)CCc3ccco3)C2)=O)cn1 C(=O)(C(C)(C)CC(C)(C)C)NCC(C(=O)NC(CC#C)CC)CC1CC1 C1(C(N2C(C(N3CC(C(N)=O)(OC)C3)=O)CCC2)=O)CC2C=CC1C2 S(=O)(=O)(c1cccnc1NC(CC)C1CC1)NC(CCCCC)C CN=c1cc(C(=O)NC2(C(=O)NCC3CCCN(C)C3=O)CC2C)cc[nH]1 C=CC(CC)CC(=O)N1CC(NC(C2SCC=C2C)=O)C(C)C1 C1(OC)CCC(NC(=O)C(N2CCN(c3cncc(F)c3)CC2)=O)CC1 c1(C(N(CCCCS(N)(=O)=O)C)=O)cnn2cc(C#N)cnc12 N1(C(CNC(=O)OCC=C)=O)C2CCC1CC2.c1(C=O)ccc(Cl)nc1O.C C(N=c1ccn2ncc(S(=O)(=O)N3CCC(CF)C3)c2[nH]1)c1c(C)c(Br)ccc1 CC1CN(C(=O)CC2CCC(C)C2)CC(C)N(C(C2CCC(=O)N2C)=O)C1 C1(CNC(Cc2ccc(OCC)cc2)=O)CCN(c2nnc(C(N)=O)s2)CC1C c1(C(C(=O)NCCC#N)N(CC(C)C(=O)OC(C)(C)C)CC)ccccn1 C#CCCCC(C)C(=O)N(CC(=O)NOC(CO)C(C)C)CC1CC1 N1(C(COCC(=O)NC)=O)CCOCC(NC(=O)C(c2nc(F)ccc2Cl)C)C1 N1(C(C(CC(C)C)N(C)C)=O)CCC2CN(C(C3CC(=C4CCC4)C3)=O)CC2C1 C=CCC(CC)C(=O)NC1(CNC(=O)C(=C2CCCCC2)F)CCOCC1 c1(NC(C23CC2CN(Cc2c(F)cc(Cl)cc2Cl)C3)=O)nnc2ccc(Cl)nn12 N1(C(c2c(C)nc(CO)o2)=O)CCC2(CO)CN(C(=O)CC3CC3)CC2C1 C1(CC(=O)NCCCCCNC(C(=Cc2cccs2)C)=O)CCC(=O)NC1 c1(C(N(CCCNC(c2cccnn2)=O)CC)=O)cccc(C#N)c1C C(=O)(C(C)CC(F)(F)F)NCC1C(C)CCN1C(=O)COCCCF N1(C(c2onc(C)n2)=O)CCC2(NC(C3CCSC3)=O)CCCC12 C1(c2ccc(C)c(OC)c2C)NC(=O)N(C(C)C)C(C)=C1C(=O)NC(C)C c1(C(c2nc(C(C(C)C)SC)on2)(C)C)cccc(C(F)(F)F)c1 CN=c1nc(N2CCCC(NC(=O)C3CC3)C2)[nH]c(=NC2CCN(C(C)(C)C)C2)[nH]1 N1(C(C(C(C)NC(C23CC(F)(C2)C3)=O)C)=O)CCCC(O)(C(N)=O)C1 C1(CC)CN(C(C2(OC(C)=O)CCOC2)=O)CC1C(=O)NCC(C)OC CCC(C(=O)NC(c1ccnn1C)C(=O)NCC1CCSC1)N(C)C CC1C(NC(C2CC3CCC2N3C(=O)CCCC(F)(F)F)=O)CC2CC1C2(C)C C(CN=c1ccnc(NC2CCCN3CCCCC23)[nH]1)c1c(C)ncs1 C=CCC(C)C(=O)N(C(C)CC(=O)NC1(CO)CC(C)C1)C Cc1cccc2c1OCC2C(=O)NCCOCCN(C(=O)C1=CCCS1)C C1(CNC(CCc2onc(C)n2)=O)CC(C(=O)NC2COCC(C)(C)C2)=NO1 C1(CN(CC(F)(F)F)C(C2(NCCO)CCNCC2)=O)CCCC(F)(F)CC1 c1(-c2c(C(=O)NC(c3ccccc3)C3CC3)n[nH]c2)ccc(C(=O)O)cc1.C N1(CCC)C(=S)NC(c2c(Cl)ccnc2F)C2=C1C(C)CN(C)C2=O N1(C(c2cc(C)oc2)=O)CCCC2(CCC(NC(c3cnn(C)c3)=O)C2)C1 C12(C=O)CCC(CC1)CC2.CC1CN(CCNC(=O)CCOCCC)CCO1.N C1(CNC(C(CSC)C)=O)CC(NC(c2cccc(C)c2)=O)CCO1 CCCC(C(=O)NCC1CCC1NC(C1(COC)CCOCC1)=O)OCC N1(C(C(c2cccc(C)c2)=O)=O)CCC(C)C(F)(F)C1.C1(C(=O)N)CC2CC1C2 c1(CC)ccc2cc(C(N3CC4CC(NC(=O)CS)CC4C3)=O)[nH]c2c1.C(C)C CN1CCOc2c(C(N3CC4CC4(CNC(=O)CCC#N)C3)=O)cccc21 Cc1ccc(NC(=O)COC(F)(F)F)cc1N(S(C)(=O)=O)C C1(C(N2CCCCC2)=O)(CC)CCN(C(=O)C=CC2(C)COC2)C1 CC1CC2(CC(C(=O)NCC(CC(C)C)NC(=O)C#CC(=O)N(C)C)C2)C1 c1(OC)csc(C(=O)NCC2CCCN(C(=O)Cc3c(C)noc3C)C2)c1.O CC1=C(C(=O)NC(C)(CNC(=O)Cc2cncs2)CO)Cn2nnnc2N1C C#Cc1ccc(CC(=O)NC(C)(C)C=CC=O)cc1.c1cn(C)nc1C1CC1 N1(C(C2CC(C)OC2)=O)CC2CCC1C1CN(C(=O)CC3(C)CC3(Cl)Cl)CC21 N1(C(C2CN(Cc3csc(Br)c3)C2)=O)CCC2(CC1)COc1ccccc12 C1(CN(C)C)COCCN1C(=O)C(C1CCN(C(=O)Cn2ncn(C)c2=O)C1)F Cc1nc(C)c(C(=O)NC(CNC(C2(CF)CC2(F)F)=O)C(C)(C)C)s1 N1(C(C(C(CC)O)(C)C)=O)CC2OCCN(C(=O)CC(C)(F)F)C2C1 N1(C(CCc2nnc(C)o2)=O)CC(CNC(=O)C(c2ccc(Cl)s2)=O)C(C)C1 Cc1cnccc1C(=O)NCC1C=CC(NC(C23COCC2C3)=O)C1 Cn1cc(CNC(c2[nH]ccc2C)=O)ccc1=O.C1(C(C(=O)N)F)CCOCC1 c1(NC(N2CC(C)(C(=O)OC)OCC2)=O)cc(C)c(Cl)nc1Cl c1(C(N2CCCC2)=O)cc(N)ccc1F.CC1=NNC(=O)C1CC(=O)NCCO N1(C(C=CC=CCC)=O)CCOCC2(COCCN2C(=O)CC2CC2C)C1 c1(C(C)NC(=O)CCN(C(C2CC2)=O)C2CC2)ccccc1F C1(NC(C2C(C=C)C2)=O)(CNC(=O)CCCCC(=O)OC)CC2CCC1CC2 C(=O)(C1=CCOCC1)NC(CCOCC)C(=O)N(C)Cc1cc(C)cs1 N1(C(C=CCCC)=O)CCN(C(C)CNC(C2CNC(=O)O2)=O)CC1 CC(O)CCCCCC(=O)N1CCCCC1CNC(C1(C#N)CCCOC1)=O C1(CNC(c2ccc(O)nc2Cl)=O)CCN(C(=O)C(O)C2CCCC2)CC1(F)F c1(CN(C)C)ccc(O)c(Cl)c1.c1(C2C(C(N3CCC3)=O)C2)ccc(F)cc1 C1(CC)CN(C(c2sccc2F)=O)CCN1Cc1cc(O)ccc1OC C(C)(CC(=O)NC1CC(F)(CNC(=O)C(F)(F)c2ccccn2)C1)OC Cc1nc2c(C(=O)NC3CCCN(C(c4ccn(C)c(=O)c4)=O)C3)cccc2o1 N1(C(C(C(CC)C)C)=O)CC(O)(C2(CNC(c3cc(C)nc(O)n3)=O)CC2)C1 c1(CC=O)ccc(Cl)cn1.C1(OC)CC(CNC(c2cn(C)cn2)=O)C1.N c1(CCOC)cccc(NC(c2cn(C)nc2-c2ccco2)=O)c1 N1(C(C(CO)OC)=O)CCOC(CC(=O)NCCC2CCCOC2)C1 N1(C(CC)=O)CSCC1C(=O)NCC(C)(C)NC(=O)C.N1(C=O)CCCC1 c1(CC)ncc(C(=O)NC2CC3CN(C(=O)C=Cc4cc[nH]n4)CC23)c(O)n1 O=C1NCc2ccc(C(N3CC(C(c4cnn(C5CCC5)c4)=O)C3)=O)cc2N1 CCC(CC(=O)NCCC1CCCN(C(c2cnc3c(c2)NCC3)=O)C1)C(C)C C(C(CO)(CO)NC(=O)Cc1ccn(C)n1)N(C(=O)C(F)CC1CCCCC1)C c1(NC(=O)NCc2ncc(C(C)C)[nH]2)c(I)cc(Br)c(F)c1F c1(C(=O)NC(CNC(=O)Cc2cc[nH]n2)C2CCC2)cncc(-n2cccn2)n1 Cc1oc([N+](=O)[O-])cc1C(N1CCCC(C)(C)C1)=O.C(c1nccs1)=CC=O.N c1(C(N2CCCC2CC#N)C(=O)NC(C(=O)OC)C)ccn(C)c(=O)c1 Cn1cncc1C(=O)NC1CCN(C(=O)Cc2cc[nH]c2)C1 N1(CC(=O)N(CCN(C(c2[nH]c(=NC)sc2)=O)C)CC)CCCCC(O)C1=O c1(CC)ccccc1C(N1CCOC(CC(N2CCN(CC(C)C)CC2)=O)C1)=O c1(SCC)cccnc1C(=O)N(CCCCNC(c1cc(CC)oc1C)=O)C N1(c2ccc(Br)cn2)CCc2cc(Cl)c(Cl)cc2C1 c1(C(=O)NC(C)CN(C)C(C2(O)CCOC2)=O)c(C(F)(F)F)cccc1Br C(=O)(C(O)CCS(C)=O)N.c1(C(N2CC(COC)C2)=O)nc(C)c(C)[nH]c1=O C1(NC(c2c(C)ccc(C(C)(F)F)c2)=O)COC2C(NC(=O)C(N)=O)COC12 Cc1ccc(F)cc1C(=O)NC(Cc1ccoc1)C(=O)NCCn1cncn1 Cc1nn(-c2ccccc2)c(Cl)c1CNCCCCCC(=O)N(C)C c1(C(C)NC(=O)C(=O)N(C)CCc2nc[nH]n2)c(N(C)C)cccc1F N1(C(CCOCCC)=O)CCC(C2CCN(C(=O)C#CC3CCCC3)CC2)CC1 C(C(CC(F)(F)F)NC(c1csc(-c2ncccn2)n1)=O)NC(C(C(C)C)F)=O C12(C(NCCC)=O)CCCC1(C(N)=O)C2.C1(C=O)CCN(CC(C)C)C1.C c1(C(N2CCC(CN(C(c3oc(CC)c(C)c3)=O)C)C2)=O)csc([N+](=O)[O-])c1 C1C2CN(C=O)CC12.c1(C=O)[nH]cnc1.C1(CC=O)(OC)CC1.C(C)(C)C N1(C(c2c(NCC)scn2)=O)CCCC2(NC(c3ccccn3)=O)CCCC12 c1(C(=O)N)cc(F)c(C(F)F)cc1F.Cc1csc(C(C)C(=O)NCC(C)C)n1 CC1CN(C)CCN1C(c1c[nH]cc1-c1ccc(Cl)s1)=O Cc1cnc(C(N2C(C(=O)Nc3nnc(Br)s3)CC3CC23)=O)cc1Br C1(C)(CNC(CC=C)=O)COCCN(C(C2(C(F)F)CC(F)(F)C2)=O)C1 c1(C2C(=O)N2)c(C)cccc1Br.O(NC(=O)COC)CC.C1(=O)C(C)N1.O c1(CN(C)C(C2CC2C(N)=O)=O)ccccc1.c1(C=O)cnn(C)c1F.C c1(C(=O)NC2C(NC(CCCCC=C)=O)COC2)n[nH]c2c1CC1CC21 C(=O)(CCCCCCC)N1CCC(C#C)(C(=O)NC(C2CCC2)C2CC2)C1 C1CCC(C)N(C(=O)CCC(C)(C)N(C)C)C1.Cc1ccc(C=CC(=O)N)o1.C C1(C(=O)NC2CCC(N(C(C3CC4(CC(C)C4)C3)=O)C)C2)CN2CCN1CC2C Cc1ccc(NC(=O)C(CCC2CCC2)NC(c2ncccc2N)=O)cc1C C1(NC(c2c(C)cc(C)o2)=O)CCCCN(C(=O)C(C(C)C)n2ccnc2)C1 C(CC(C)(C)C(=O)N1CCC(C(=O)N(CCCC(O)CO)C)(CF)C1)SC C=CCN=c1[nH]cc(C(=O)NC2CC23CCC(NC(=O)C2=CCCCC2)CC3)s1 N1(C(C=CC(C)NC(C(CCC)C)=O)=O)CCOC2(CC2)C1 Cc1cc(O)c(C(=O)N(C)C(c2cn(CCCCC(=O)O)nn2)C)nn1 Cc1cn2cc(C(N3CC4CCCC(C3)N4C(=O)C(F)C(F)(F)F)=O)ccc2n1 c1(C(CO)NCC(O)Cc2ccc(Cl)cc2)cccc(F)c1F N1(C(C2CN(C(=O)CC3COCC3O)CC2(F)F)=O)CCCc2occc2C1 N1(C(c2c(CC)ocn2)=O)CC2(CCN(C(C3CC3C)=O)CC2)C1C(C)C N1(C(CC2N(C(C3N(C)CCC3)=O)C3C2CCC3)=O)CCC(C2(C)CC2)C1 C1CC(F)CN(C(C2(c3ccccc3)CC(O)C2)=O)C1.c1(C(=O)N)cccc(F)c1 C=C(C)CC(C(=O)NCC(O)(C1CC1)C1CC1)NC(c1ccc(C)o1)=O c1ccc(C(=O)C=CC2CC2)cc1.CCCC.C(=O)C.C(=O)CN(C)C.N Cc1ccc(C2=NOC(C(=O)NC3C=CCN(C(=O)CN(C)C(C)C)C3)C2)cc1 S(=O)(=O)(c1cnc(C(C)C)n1C)N(C)CC1(OC(C)C)CCOC1 N1(c2n(CCSc3c(C)cccc3)c(C)nn2)CCN(C)C(=O)C1.C(C)(C)C.O Cc1cc(Cl)cc(C)c1C(N1CC2CC(F)(C1)C2)=O.C(C(C)(C)C)=CC=O C(=O)(C(C)Cc1ccco1)N(C(C)CNC(=O)CC1(C)CCC1)CC C1(C(=O)NC2CCN(C(c3ncc(F)cc3F)=O)CC2)CC2CCC1NC2=O c1(C(N(CC)C)=O)cnn(C)c1S(N)(=O)=O.C(C)(C(O)C(=O)N)SC.CC c1(C(=O)NCC(CCNC(=O)CCCn2cccn2)OC)sc(F)cc1C C#CCCCC(=O)NCC=C1CCN(C(=O)C=C(C2CC2)C2CC2)CC1 C1(C(N(C(C)C(F)F)C)=O)CN(C(=O)CN2CC3CC3C2)CC(C)(C)C1 CC1COCCCN1C(c1coc(CNC(=O)C(O)C(C)(C)C)n1)=O C#CC12CC(NC(=O)NC(c3ccccc3)Cc3ccc(F)cc3)(CO1)C2 c1(OC)ncc(C)cc1C(=O)NCC(C)(CO)NC(C1(F)CCOC1)=O N1(C(C(C)OCC#C)=O)CCC2(CCCN(C(=O)C(C)CC#C)C2)CC1 CC1(C)CCCC(CC(=O)NCC23CC2CN(C(C2CCC2)=O)C3)C1 C1(SCC)CCC(C(=O)NC2C3CC2N(C(C2(C#N)CCCC2)=O)C3)CC1 c1(C(=O)NC(C(=O)NCCC(C)(C)F)CC2CCOCC2)cc2occc2[nH]1 N1(Cc2cn(CCCN(S(C)(=O)=O)C)nn2)CCCc2ccc(N)cc21 C1(C)(C(=O)NCC2N(CC)CCC2)C=CCN1C(=O)C(C1CC1)SC C(CC1CCOCC1)(C(=O)NC(C)CCF)NC(CNC(C)=O)=O C1(CC(N2C(C)C(NC(=O)CCc3cnn(C)c3)CC2)=O)CCCCC12CC2 c1(C(N2CC(C)(CCNC(=O)CCCN=[N+]=[N-])C2)=O)sc2cc(Cl)ccc2c1Cl N1(C(CCN(C)CC)=O)CCCC(C)(NC(C2CC2C(F)F)=O)C1 C(=O)(C1CCc2nccn21)NCCC(C(=O)Nc1ccc(OC)nc1C)OC N1(C(CC2(NC(CC(C(CC)C)O)=O)CC2)=O)CC2CCCN2CC1C C1(CCNC(C2(CNC(CCCN(C)C)=O)CCC2)=O)CCN(C)C1=O N1(CC(=O)OCC)CCN2CCOCC2C1.C1(=O)C(C)(c2ccccc2F)CN1 O=C(C1=NOC2(CCN(Cc3cc(F)c(Cl)cc3Cl)C2)C1)NCC1CCCO1 c1(C(N2CCN(C(C#C)(C)C)CC2)C(=O)NCCCF)cc(OC)c(Cl)cc1F O=C1CN(C(C2CCCCO2)=O)C(C(=O)NC2CC(O)C2O)CN1 N1(C(C(C)Cc2cnc[nH]2)=O)CCN(C(c2sccc2OC(F)F)=O)C2CCC12 c1(CC)cc(C(N2CC3CC2C3NC(c2ccsc2C)=O)=O)ccc1F N1(C(CN(C(=O)CC(C)n2ccnc2)CC(C)C)=O)Cc2ccnn2CC1C N#Cc1cccc(C(N2CCOCC(NC(=O)Cc3cn4ccsc4n3)C2)=O)c1 C1CCN(C(=O)Cc2ccc(C(F)(F)F)cc2)C1.C1(F)(C(=O)N)CCC1.C C1(C2CC2)(CNC(CC)=O)CCN(C(C2CCCN(C(=O)C(C)C)C2)=O)C1 C1(CC)(CC)CC(NC(c2ccco2)=O)CN1C(c1ccoc1Cl)=O n1(CC(=O)NCC2(C)CCN(C(=O)CCCCC3CC3)C2)ncc2ccccc12 C1(C=O)(COC)C=CCN1C(c1cc(C)c(C)[nH]1)=O.C(C)CC1CC1.N C12(C(N3CCCC(=C)C3)=O)CCC(CN(C(c3coc(CCC)n3)=O)C1)C2 N1(C(CSCCC)=O)CCC(CCOC)(NC(C2CC(=C3CC3)C2)=O)C1 c1(C(N2CC=CC(NC(c3c(N(C)C)nccc3)=O)C2)=O)ccn2c1CCCC2 C1(CNC(C=C(C)C(C)C)=O)CCN(C(=O)CCCc2csc(=N)[nH]2)CC1C C1(C(=O)Nc2cnc(CC)nc2)CCN(C(=O)CC2CCSC2)C12CCC2 C=CC(C(F)(F)F)NC(C1CN(C(c2cn(C3CC3)cn2)=O)CC1CCC)=O c1(-c2cn(C)nc2)nn(C)cc1C(N1CC(NC(C2(C(N)=O)CC2)=O)C1)=O c1(C(=O)NC(C(=O)NC(C#CCC)(C)C)C(C)C)cnn2c1OCC2 C1(CNC(c2nn(C)c(Cl)c2Cl)=O)CN(c2nc(Cl)ncc2F)CCC1(F)F C1(CC)CCCN1C(=O)Cc1ccccc1.C(=O)CC1(C)CC1.C(C)=O.N c1(C(COC)N(C2CCC3(CC2)COC3)C=O)ccc2c(c1)OCCO2 C1(CCC)(NC(C(C=C)CC)=O)CCCN(C(=O)CC2(CSC)CC2)C1 CC(CC(=O)NCC1(F)CCN(C(c2cc(CO)[nH]n2)=O)C1)CC(F)(F)F N1(C(C2(CCOC)CCC2)=O)CCCC2CN(C(c3ncccc3O)=O)CCC12 C(=O)(C1CCc2c(Cl)cccc21)N1C(CCNC(=O)CC2=CCOCC2)CCC1 N1(C(c2cc(C)on2)=O)CC(NC(=O)C(C)n2cncn2)C(C)C1 C1(CNC(COC)=O)CN(C(c2ccnc(N3CCN(C)CC3)c2)=O)CC12CC2 c1(OC(C)C(=O)NCC(c2ccccc2)NC(=O)C(F)F)cccnc1 N#Cc1ccc(F)cc1-c1cnc(C(=O)O)c(Br)c1 c1(Cn2cc(-c3c(F)ccs3)nn2)ccc(Cl)nc1 c1(C(=O)OC)cncc(C(=O)NC(C)C2CCC2)c1.C(=O)CC.C1CC1.N C1(CNC(=NCC=C)NCC(c2cc(C)cc(C)c2)O)Cc2cccnc2C1 C1(CNC(CCNC(CC2(C#N)CC2)=O)=O)CC2(CC2)C(=O)O1 C12(C(=O)NCC3CN(C(C4C(C)C4)=O)CC3(C)C)CCC(F)(CC1)CC2 C1(C=O)CCN(C(=O)C(=O)NCC)C(c2ccccc2)C1.CC(C)CCF c1(C(=O)OC)cc(C(N2CCCC2C)=O)cs1.C1(C2(C=O)CC2)CCCCO1 C1(Nc2c(C)c(Cl)ncn2)CCC2CN(C(=O)CN3CCN(C)C(=O)C3)CC12 N1(C(C(C2CCN(C(=O)C(C)CC(F)F)CC2)C)=O)CCC2(CCOC2=O)C1 Cc1ccc(C(N2CC(C)(NC(C34CC(CO3)C4)=O)C2)=O)cc1N c1(CC)ccc(CC(N2CCC(C(F)F)(CNC(C3CC3)=O)C2)=O)cc1.C C1(CCC(N2C(CC(=O)NCCOc3ccccn3)CC2)=O)CCCOC1 c1(CN2CC3C(NC(c4c(C)csc4)=O)C3C2)ccc([N+](=O)[O-])cc1F C(=O)(C(C#N)CCC)N1CC(CC=C)(C(N2CCC(C)(CN(C)C)C2)=O)C1 C1(C(=O)OC)CC12CCC(NCc1cc(Cl)c(C)cc1Br)CC2 C1CCC2(CCC2)C1.N=c1[nH]cc(C(=O)NC)o1.C1(C=O)CN(CC(F)F)C1 C1(C(C)(C)O)CCN(C(=O)C(C)(C)C2CC2)CC1.c1(C(C)C)ncc(C(=O)N)s1 C=C(C)C1OCCC1C(=O)N(C(C)(C)CC(=O)NC(CC(=O)OC)C1CC1)C N1(Cc2ncc(C)nc2)CCC2(CC1)CC2C(=O)NCc1cc2c(s1)CCC2 N1(c2ccnc(NC(Cn3c(CC)ncc3)C)n2)CCc2ccncc2C1 Cc1oc2c(F)c(F)c(F)c(F)c2c1C(N1C2CCC1(C)CC2)=O C#CCC(C)(CC)C(=O)NCCOCC.c1ccc(F)c(F)c1.C(=O)(CC)N N1(C(c2ccn(COC)n2)=O)CC(OC)C(OC)C1C.C(=O)(C1=CCCC1C)N C1(F)(CNC(c2c[nH]nc2Br)=O)CC(NC(=O)C(F)(F)C2(O)CCC2)C1 S(=O)(=O)(c1cc(C#N)ccc1C)NC1C(CC)CN(C(C)=O)CC1 C1(C(=O)NCCC(C)NC(C(C)O)=O)CC2CCC1O2 C1(NC(C=CCC)=O)CC(=O)N(C2CN(C(=O)CC3CCCN3C)C2)C1 C(=O)(C(O)CCC(F)(F)F)N1CCC(NC(C2=C(C)OCC2)=O)(CC)CC1 N1(C(C(c2cccc(F)c2)(C)O)=O)CCC(CCCNC(C2(CF)CC2)=O)CC1 N1(C(c2c(OC)cccn2)=O)CC2(CCC2NC(c2ncoc2C2CC2)=O)C1 N1(C(COCCSC)=O)CC(C2CC2)(C(=O)NC2(CO)CC(F)C2)C1 C1(C)(CNC(c2ccc(C)nc2)=O)CCN(c2cc(C)nc(C)n2)CC1 c1(C(=O)NCCC(C)Nc2ncc(C#C)cn2)ncnc2c(C)csc12 c1(NC)cnncc1C(=O)NC1CCOC(C(=O)NC2CN(C(N)=O)C2)C1 C1(CC(=O)N(C(CNC(C=C(CC)CC)=O)C)C)CCCC(C)(C)C1 c1(C2N(C(=O)CCn3cccn3)CCCC2)nc2ccccc2o1 C(=O)(CCC1CCOCC1)NC1(C(C)O)CC1.C(=O)CC1(N(C)C)CC1.N CC1CCN(C(=O)CCC(F)(F)F)CC1NC(c1csc(C(C)(F)F)n1)=O C1(NC(C2(NC(c3ccn(C)n3)=O)CCOCC2)=O)CC(=O)NC(=O)C1 C(=O)(CC(C)(C)CNC(=O)C(O)C(F)(F)F)N1CCC(CC(C)(C)C)C1 N1(C(c2cc(C)[nH]n2)=O)Cc2nccn2CC(NC(=O)C=Cc2nnn(C)n2)C1 Cc1nc(C(F)(F)F)sc1C(N1CCC(=CC)CC1)=O.C1(C=O)CCNC1=O.N c1(C(=O)NC2CC(N(C(Cc3cncc(C)c3)=O)C)C2)ncc(C)cc1C Cc1nc(C(=O)NCCN(C(=O)CSc2n[nH]c(O)n2)C2CC2)cn1C c1(OC)cccc(NC(=O)CC2CCCN(C(C3CC(=O)CCO3)=O)CC2)c1C N1(C(C(CCSC)O)=O)CCC2CN(C(C3(N(C)C)CC3)=O)CC12 c1(CNC(CSCC=C)=O)nc2c(s1)CCN(C(C1CCCC(OC)C1)=O)C2 Cc1ncc(C(=O)NC(C)(C)CN(C(=O)CCOC2CCCOC2)C)[nH]1 c1(C(N(C(C)CNC(=O)C(O)C2CC2)C)=O)cccc(C(F)(F)F)c1Cl c1(C(N2CCC(C(C)NC(c3nc(C)sc3)=O)CC2)=O)ccc(Br)c2cc[nH]c12 C1(NC(=O)CCc2cnoc2)CN(C(=O)Cn2cc(C(F)(F)F)cn2)CC1O C1(C=O)CCS(=O)CC1.C12(CNC(C3C(C)(C(C)C)C3)=O)CC(C1)C2 C(=O)(C=CS(F)(F)(F)(F)F)N.Cc1nn(CC(=O)NC2(C)CCC2)c(=O)o1 C1(C(=O)OC)C(C(=O)NCC(C)NC(c2ccc(Cl)s2)=O)C1(F)F N1(C(C2=CCN(C(C(C)N=[N+]=[N-])=O)CC2)=O)CCc2ccccc2C1 C(=O)(C(O)P(C)(C)=O)N(CCCNC(CC(c1c(C)cccc1)C)=O)C Cc1c(NC(C)C)cccc1C(=O)N.C12CC1CN(C(=O)C=CC1CC1)C2 CC1CN(C(c2occc2F)=O)CCN1C(c1cnc(O)c(F)c1)=O C1(CNC(CSCC#C)=O)CC(C)N(C(=O)Cn2cnnn2)C1 C1(C(=O)NCCC2CCCN2C(=O)Cc2cn[nH]c2)CCCOC1c1cc[nH]n1 C1(OC)CC(NC(=O)C)CN(C(c2ccncc2)=O)C1.[SH](=O)(=O)C1CC1.N C1(CNC(CSC)=O)(CO)CCN(C(=O)CSc2cccc(F)c2)CC1 c1(C(N2CC(C)(C)NCC2)=O)cccnc1C1=CCC(F)(F)CC1 c1(-c2scc(C(=O)NC(c3cccs3)CC)n2)cccc(C(C)O)c1 N1(C(C(C)=C2CCC2)=O)CCN(C)CC1CNC(=O)CO.C1CCCO1.C N1(C(c2c(CC)oc(C)c2)=O)CCC2(C1)CN(C(=O)CCc1cscn1)CCO2 C(=O)(C(O)CC(C)(C)C)N1C(C)C(NC(c2cc(Br)no2)=O)CCC1 c1(C(=O)NCC(C)(O)CNC(c2ccc(Br)o2)=O)cc(=O)cc[nH]1 CCC(CC(C)C)C(=O)N(C(C)CNC(c1ccc2n[nH]cc2n1)=O)C Cc1c[nH]c(C(N2CCC(C(C)C(=O)NCCc3ccccc3)CC2)=O)c1C C(=O)(C(O)CC)NCC(CC)NC(c1ccsc1Br)=O CC(=O)CCCC(=O)NCC1CN(C(=O)CCc2csnn2)CC1(F)F C1(C(N2CCC(CC(=O)N(C)Cc3cn(C)nn3)C2)=O)CCS(=O)CC1 CC(C(=O)NCC(C)Cc1cccs1)C(C)(C)C Nc1ccc(S(N)(=O)=O)cc1C(=O)NCC1CC(NC(=O)C2=CCC2)C1 Cc1nn(CC(=O)NC(C)C(CO)NC(C2CC(C#N)C2)=O)c(C)c1Cl c1(OCCO)ccc(Br)cc1NC(c1nnnn1CCCF)CC1CC1(Cl)Cl CC12CC(C1)C1(CN(C(=O)CCc3csc(=N)[nH]3)C1)O2.C(=O)C=CCO.N C(=O)(C1CCCn2ccnc21)N1CC(C(C)C)N(C(=O)CCOC2CC2)CCC1 Cc1nn(CC(=O)NCC(C)CN(C(=O)C(F)=CCCF)C)cc1Cl c1(CNC(C(C2CN(C(CSCC=C)=O)C2)O)=O)cnn(C)c1 C1(NC(c2c(C)scc2)=O)CC12CCN(C(=O)CNC(=O)CC(C)(C)C)CC2 N1(C(C2C3CN(C(CCC(C)C)=O)C2C3)=O)C2CCC1CC(CO)C2 c1(C(N2CC(NC(=O)C(=O)N(C)C)CC(C)C2)=O)cc2cn[nH]c2cn1 C1(CNC(C2C(c3n(C)ccn3)C2)=O)COCCN1C(=O)C=C1CCSCC1 C1(CNC(C(COC)O)=O)CN(C(c2cccnc2O)=O)C2CCCC2O1 C(C(=O)NCC(c1cccs1)C)(C(C)(C)O)NC(C1CC(=C)C1)=O C1(NC(C(CC#C)C)=O)(CNC(=O)CO)CCC(C)(C)CC1.C1CCCOC1 C(=O)(CCCCC(C)(C)C)N1CCC(F)(C(N2CCN(C)C(C)(C)C2)=O)C1 CCC(C(=O)NC(C)(C)CN(C)C(c1cn(C)cn1)=O)n1ccc(C2CC2)n1 c1(OC)ccc(C(c2ccc(Cl)cc2)NC(C2CCC(F)CC2)=O)cc1 CC1(C#CC(=O)NCC2CC2CNC(C2CCCC23CC3)=O)CCCO1 c1(C(=O)NC(CC)(C)CNC(=O)CCCOC(C)C)ccn2c1CCCC2 C(=O)(C(F)(F)CO)NCc1c(C(=O)NCC2C(N(C)C)CCC2)c[nH]n1 c1(N2CCC(C(CC)C)CC2)cc(C)c(S(=O)(=O)NC2CC2(C)C)cn1 C(=O)(C1=CCCC1(C)C)NCC(CNC(C#CC1(C)CC1)=O)O n1(CC)cc(S(=O)(=O)N2CCC(C)C2)c(C)n1.c1(C=O)ccc(C=O)s1.N n1(CC(N2CC(C3CC3)C2)=O)cc(S(N)(=O)=O)cn1.N#Cc1nc[nH]c1C=O c1(C(=O)NC(C2CN(C(c3c(CC)c[nH]c3)=O)C2)C)cccc(F)c1Cl Cc1cc(CNC(=O)CCCc2ccccc2Cl)ccc1S(N)(=O)=O C1CCCC(C)C1.C(=O)C(O)CCN(C)C.c12cc(no1)CNC2=O.CC c1(OC)ccc(C(=O)NC(C2CN(C(=O)CC3CCOC3)C2)C)cc1F CC1CN(C(C2(Cc3ccccc3)CN(C3CCOCC3)C2)=O)CCS(=O)C1 N1(C(CC(C)O)=O)CCC2CN(C(=O)CCc3ccc4c(c3)CCO4)CC12 O=C1CCC(CC(=O)NCC(O)C(=O)NC23CC(C2)C3)CN1 N1(C(c2cnc(C)[nH]2)=O)CC2CC(NC(=O)Cn3cc(Br)c(C)n3)CC1C2 CC(C)(C)C#CC(=O)N1CCC(C)(NC(c2ccc(F)o2)=O)C1 N1(C(C)CC2(C)CC2)CCc2nc(C(=O)NC(C3(O)CC3)C)cn2CC1 CC(C)C1=NOC(C(N2CCC2C(=O)NCC2CC23CCOC3)=O)C1 c1(OC)c[nH]c(C(=O)NC(C)(CNC(=O)C#CC(=O)N(C)C)CO)cc1=O C1CN(C(c2ccc(N)c(O)c2)=O)CCC1C.C(C)(C(=O)N)OCCOCC c1(C(c2nnnn2CC2CCCO2)Nc2cn(CC#C)nc2)c(Br)c(C)nn1C Cc1ccc2c(c1)CC(C(=O)NCCCC(C)NC(c1ncccn1)=O)S2(=O)=O c1(CCC(=O)NCC(CNC(=O)Cn2cncn2)OC)ccccc1 N1(CC(N(CCCC)CCC)=O)CCN(c2ccccc2O)CC1 c1(OC)cc(OC)c(F)c(NC(C2COCCN2C(c2ccnn2C)=O)=O)c1 C1(N(C(CCC2CC(OC)C2)=O)C)CCN(C(=O)CN2CCOCC2)C1 N1(C(C(c2noc3ccccc23)C)=O)CCC2(CCN(C(=O)CC3CC3)C2)C1 c1(C(N(C2CCN(C(CCCOCCC)=O)C2)CC)=O)cnn2c1CCC2 N1(C(CCCC#C)=O)CC2(CCCCN2C(C2CCSC2)=O)C1 CC(C)(C)CCCCC(=O)NCCCC1CCN(C(C2(O)CC2(C)C)=O)CC1 C12(NC(CCC(=O)NC)=O)CCCC1N(C(=O)C(F)CC1CCCC1)CC2 C(=O)(C(C)(C)C(=O)NC(C)CC(F)(F)F)N(C)C.c1(CC(=O)N)cncs1 n1(CC(N2C(CN(C)C(c3ncccc3Br)=O)CCC2)=O)ncn(C)c1=O C1(NC(CC2CCC(C)C2)=O)CCC(NC(c2cc(F)n[nH]2)=O)CC1 C(=O)(CC(C)(C)CNC(c1sccc1C#N)=O)N1CC(C#C)(N(C)C)C1 N1(C(C(=O)NC(C2COCCO2)CC)=O)CC(C)Oc2ccccc21 C1(CNC(c2cccc(SC)n2)=O)CC2COCC2N1C(C1CCCS1)=O C(=O)(CC1=CCCC1)N1C(C)(CNC(C2(C(C)C)CCCO2)=O)CCC1 CCC(CC)(CO)C(=O)NCCC(C)(C)NC(=O)Cc1ccc(C)c(OC)c1 c1(OC2CCN(C(c3nc(CO)cs3)C(=O)NC)C2)cccc(F)c1 C1(NC(CC2(CSC)CC2)=O)CCCCCC1.c1(C(=O)N)cc(C)nc(C)n1 N1(C(C2C3CC4C(C3)C42)=O)CC2(CC(C)CO2)C1.C(=O)(CC=O)OCC.O C1(NC(Cc2cnc(C)[nH]2)=O)CC(C)N(C(=O)C#CC(C)C)C1 C(CC(C)C(=O)NCc1ccc(CCNC(C2CC(C)C2)=O)cc1)=CC Cc1cccn2cc(C(N3C4CCC3CC(NC(=O)C(C)S(N)(=O)=O)C4)=O)cc12 N1(C(COCC=C)=O)CCC(C2(NC(C3CN(C4CCOC4)C3)=O)CC2)CC1 N1(C(C2N(C=O)CCC2)=O)CCC2(CCN(C(C3Cc4nccnc4C3)=O)C2)C1 S(=O)(=O)(c1ccccc1F)N1CC(NC(c2c(OC)cc(Br)cc2)=O)C(F)(F)C1 N1(C(c2ccnc(C)n2)=O)CCN(C(=O)CC(C)P(C)(C)=O)CC(C)(F)C1 S(=O)(=O)(c1ccc(NC(=O)NC2CCC2(C)C)c(C)c1)NC c1(C(=O)NC(CC)CNC(C2(C3CC3)CCC2)=O)cnc(O)c(C)c1 CC(CCCc1cccnc1)OC(c1cn(CCN(C)C)nn1)=O CC1(C)CN(C(C2CC2F)=O)CCN(C(C2(C#N)CC3CC3C2)=O)C1 CCN=C(NCC1(COCc2ccccc2)CCCCC1)N1CCC(OC)CC1 c1(C(=O)NCC2CN(C(C3C4COCC34)=O)CC23CC3)cc2cccc(Cl)c2o1 C1(NC(CCC(=O)NCc2nnc(C)s2)=O)CCCN(C(=O)C(C)(C)F)C1.C CC1CCN(C(c2cncn2C)=O)CCN1C(=O)C(c1ccc(F)cc1)=O N1(CC)CCOCC1C(=O)NCC1CCC(C(=O)NC2COCC2N=[N+]=[N-])C1 C(=O)(C(C)(C)CCNC(=O)CC1CNC(=O)O1)N1CCC(CC)C1 c1(CNC2C(F)(F)CCN(c3cc(C#N)ncn3)C2)ccc2ccccc2c1 N1(C(c2c(Cl)ncc(C)c2)=O)CCC(C2CN(C(=O)CC(C)(C)O)C2)CC1 C1(NC(=O)CNC(C2CCCCC2)=O)CN(C(=O)C2=COCCO2)C2(CCC2)C1 CCC(CCO)CN=c1[nH]c(N2CCC(CC)(CC)CC2)nc(=NC)[nH]1 C1(CC)CN(C(C2CCCC2F)=O)CCC1CNC(C1CNC(=O)O1)=O CC(CCC(=O)N1CCCCC1CN(C)C(C12CC(CO)(C1)C2)=O)N(C)C CN(CP(C)(C)=O)C(=O)CCN(CCCO)C(=O)C=CC1CCOC1 C1(C)(CNC(C2OCC(C)C2)=O)CCCN1C(=O)C(F)=C1CCCC1 c1(C(=O)NC(C(CC)C)C(=O)Nc2cc(C)ccc2C)cccc2c1OCC2(C)C N1(C(C(C(=O)OC)OC)=O)CC2=C(C1)CN(C(c1snnc1C)=O)C2 N1(C(C=NOC)=O)CCN(C(=O)C(C)SC(F)(F)F)CC1C1CCCC1 N1(C(CC2CC(=C)C2)=O)CC(NC(c2nc(C)ccc2OC)=O)CC12CCC2 c1(COC)cc(C(F)(F)F)ccc1NC(=O)NCCCCOC(C)C C(=O)CC(C)C.C1(CCO)CN(C)C1.C(C(=O)NC)N(C(=O)CO)C(C)C c1(C(=O)NCC(N(C(CCC(CC)C)=O)C)C2CC2)cnc2cc(C)nn2c1C N1(C(c2cncc(OC)n2)=O)CCC(C)(NC(=O)COCCCF)CC1 C#Cc1nc(C(N2CCC(OCC)C2)=O)cs1.c1(C(=O)N)ncccc1N(C)C c1(C(=O)NCC2(O)CN(C(C(C=C)(C)C)=O)C2)cccc(S(C)(=O)=NC)c1 c1(OC)ccccc1CN1CC2CC2(C(N2CCC2CO)=O)C1 c1(C(=O)NCC(CNC(C(C(=C)C)(C)O)=O)CO)c(Cl)ccc(Cl)c1Cl C=CC1(O)CCN(C(c2sc(Br)nc2Cl)C(=O)NCCCCCC)C1 C1(C(C(=O)OCC(CC=C)O)C)CCN(CCNC(=O)O)CC1.C(C)(C)C C1(C)CCN(C(=O)CC2(N3CCCC3)CC2)C1.C1(C=O)CCOC1.C1CC1.N C1(C(C)(C)C)(CNC(C)=O)CCN(C(=O)C(C)CF)C1 c1(OCC(=O)N(C)CC=CC(=O)NC2(c3cncs3)CC2)cccnc1 CCC(C(=O)N1CC(=C(F)C)C1)Nc1nc(C)cs1.C(=O)(CSC(F)F)N c1(C(=O)NCC(CC=C)NC(C2(C)CCC(=O)N2)=O)ccncc1OC C1(CNC(C(C)N(C(=O)CCCCSC)CCC)=O)CCCC(F)(F)C1 c1(C(N(C)Cc2cc(Br)cc(Br)c2)=O)cnn2cc(C3=CCCCO3)ccc12 C1(NC(c2cccnc2)C)C2CCN(C(=O)OCC(C)(C)C)CCC12 C1(C(C)C)OCCC1C(=O)NCCN(C(=O)CC(C)c1cccnc1)C(C)C CCCC(C)C(=O)N(C1(C(N2CC(C)(C(N)=O)C2)=O)CC1)C Cc1cn2nc(C(=O)NCC3CCC3c3ccccc3)ccc2n1 c1(OC)cc(CC(N2CCC(C)(NC(=O)CCSC(F)(F)F)C2)=O)ccc1F C12(C(=O)NCCN(C(C3CCOC3)=O)CC)COCC(COC1)O2 c1(N(C)C)cc(C(=O)NC2CCC(N(C)C(C3CC3F)=O)CC2)ccc1[N+](=O)[O-] c1(C(=O)NC(CNC(C(CCC)(C)O)=O)C(C)C)cc(C(C)C)n2ncnc2n1 CC1CN(C(C2C=CCC2)=O)CCCN1C(=O)CCc1cnc[nH]1 c1(OCC=CC(=O)NC2CCCC(c3ccc(Cl)cc3)C2)cccc(Cl)c1 C1(NC(CCOCC#C)=O)CCN(C)C12CCCN(C(C1(F)CCCC1)=O)C2 C12(NC(C(C)C3CCC3)=O)CCC(C)(C1)OC2.C(=O)(CCC)N.C(C)(C)C N1(C(Cn2c(C)cc(C)n2)=O)CC(CNC(=O)C(O)C(C)(C)C)CCC1C S(=O)(=O)(c1ccc(CBr)cc1)N1C(C#N)CN(C(c2cc(F)cnc2Cl)=O)CC1 c1(C(C)NC(C(C)N(C(CCSCCC)=O)C)=O)cn(C)nn1 c1(OC(C)C(=O)N(CC(O)CN(C)C(C2(Cl)CC2)=O)C)cccnc1 c1(CNC2C(C(=O)NCCC(C)CO)C2)cc(Br)ccc1I c1(NC(C(C(C)C)CNC(C2C=CCC2)=O)=O)ccc2c[nH]nc2c1 c1(C(NOC)=O)ccccc1NC(C1CN(C(=O)CC=CC(C)(C)C)C1)=O C1(C(=O)NCC2(CO)CC3CCC2C3)CCc2nn[nH]c2C1 C1(C(NOCC(=O)NCCCCC=C)=O)(CO)CCCCO1 Cc1nc(C(=O)NCC2CC2CNC(C2CCCC(=O)O2)=O)sc1C C1(C(=O)NCC2(C)CCCN2C(C2SCCS2)=O)CCc2cncn2C1 C(=O)(C1COc2c(C)cccc21)NCC(CCCC)NC(c1ccc(Cl)cc1)=O c1(CC(=O)N)nc(C)sc1C.C(F)(F)(C(=O)NCC(F)C)C1(OC)CCC1 N1(C(=O)CN2CCCCC2)CCc2c(cccc2C2=CCCCO2)C1 C1(CNC(=O)CCC2CCCC2)CCN(C(c2cc(Cl)on2)=O)CCC1(F)F C(=O)(C1=CCN(C(=O)CS(C)(=O)=O)CC1)N1CCC(OC)CC1C N1(C(CCN(C)CC)=O)CCN(C(c2ccc(C3CC3)nc2O)=O)C2(CCC2)C1 C1(C(=O)NC(c2cccc(I)c2)CC(=O)OC)CCC2(C1)N=N2 C12(NC(C3CCN(c4cc(Cl)ccc4Cl)C3=O)=O)CCCC1N(C(=O)CO)CC2 c1(SC)ncc(C#N)c(NC23CC(NC(=O)Cc4ccc(Br)cc4)(C2)C3)n1 C#CCC(C)(C(=O)N1CCC(O)(CC(C)C)C1)NC(c1cc[nH]c1CC)=O N1(CC(C)C)N=C(C(=O)N2CCOCC(NC(=O)CC3CCOC3)C2)CCC1=O Cc1cc(C(=O)NCC(C(=O)NC2(C3CCCO3)CCC2)N(C)C)cc(C)c1 CN1C(=O)NC2(CCCN(C(c3nc4cccc(Br)n4c3N)=O)C2)C1=O CC1CN(C(C2(C3CC3)CCCO2)=O)CCN1C(=O)C1CC1 C1(CNC(COC)=O)CN(C(=O)CCCS(N)(=O)=O)CCC12CCOCC2 c1(C(N2CCC(O)(CN(C(C=C(C)C)=O)C)C2)=O)cc(Cl)c(F)cc1C C=CC(C)CC(=O)NCC=CCC(=O)NC(C)CCSC C1(C(N2C(C(=O)OC)CCCC2CC(F)(F)F)=O)CCc2ncc(C)n2C1 c1(C(N2C(CCC(=O)NCc3c(C)non3)CCC2)=O)cnn(C)c(=O)c1 C(=O)(CCCS(=O)(=O)N1CCCC1)NCCCN(C)C(C1CCN(C)C1=O)=O c1(C(N)=O)cc(=NCCSCc2ccccn2)[nH]c(C(F)(F)F)n1 c1(C(N2CC(NC(c3c(C)ccs3)=O)C(C)CC2)=O)nn(C)c2c1CCCC2 c1(C(=O)NC2CCN(C(=O)CC(F)(F)F)CC2O)cc2ccc(Br)cn2c1 C1(C(N(CCC(c2cccs2)NC(CCCC)=O)C)=O)CC2OC(C)(C)OC2C1 N1(C(Cc2cccc(SCC)c2)=O)CC(NC(=O)C(CO)C(C)C)C(C)(C)C1 N1(C(C(CCCC)C)=O)CC2=C(C1)CN(C(C1(NC(C)=O)CC1)=O)C2 C(=O)(C(C)(CC)C(=O)OCC)NCC1(SC)CN(C(CC(C=C)C)=O)C1 CC1(C)CC(N=c2nc[nH]s2)CN(C(=O)CCN2CCC(F)C2)C1 c1(NC(C2(F)CN(C(c3[nH]cc(C(C)=O)c3)=O)C2)=O)ccc(F)c(O)c1 c1(CC)c(C(=O)NCCCN2CCC(N)C2)cnn1-c1ccc(Br)cc1 Cc1noc(C)c1NC(c1cc(CCNC(c2ccc(CO)cn2)=O)on1)=O c1(NC(CN(CC=C)C(C2CNC(=O)CC2C)=O)=O)ccc(CN)c(OC)c1 c1(C(=O)NCC(=O)NC(C)C2CC2)ccccc1F.C(=O)CSC(F)F.N N1(C(C2(CNC(C3CCCCC3)=O)CC(=C)C2)=O)CC2CCC(C1)N2C C1(C(=O)NCCC(C(C)C)CO)CC2C=CC1N(C(=O)CCCCC(N)=O)C2 c1(C(=O)NC(C(=O)NCC2CC(C#N)C2)C2CCOC2)ccccc1Cl c1(COC)c(C=O)oc2ccccc12.CC(C)CN(C(=O)C=C1CCCC1)C c1(OC)nc(N(Cc2cc(Cl)ccc2Cl)CC2CCCNC2)ncc1Br N1(C(c2nnc(C)s2)=O)CCC2CN(C(c3ccc4c(c3)NCC4)=O)CC12 n1(CC(=O)NC2CCCC(C)C2)nc(O)ccc1=O c1(C(N2CC3C(CCNC(CCC(C)(C)F)=O)(CC3)C2)=O)ccc(Cl)c(F)c1O N1(C(C=Cc2cc(OCC)c(O)cc2)=O)CCC2(CCC(C(=O)OC)C2)C1 N1(C(c2nc(C(C)(C)C)sc2)=O)CCC2CCC12CNC(c1c[nH]ccc1=N)=O C1(CC(=O)NCc2cc(C)c(C)s2)CC(C)(C)CN1C(=O)CC.CC(C)C.O c1(C(N2CCC(C)(NC(c3cc(C)oc3)=O)C2)=O)ccnc(C)c1N N#Cc1csc(NC(C2(F)CCN(C(c3snc(Cl)c3Cl)=O)C2)=O)n1 C(=O)(CC(CN(C)C)CC)N1CCC(N(CCC)C(C2CCN(OC)CC2)=O)C1 Cc1nc2ncc(N3CCC(O)(c4ccccc4F)CC3)nc2s1 N1(C(c2ccc(CCC)s2)=O)CC(C)(C)CC1CNC(=O)CC(C)(O)C.O c1(OCC)cc(C(=O)NC)ccn1.c1ccccc1Cl.C1(O)CN(C(=O)C)C1 c1(CCSC2CCN(C)C2)nc(C(C)(C)C)nn1-c1ccccc1C(=O)O c1(C=O)[nH]c(C)c(C=O)c1C.n1(CC)ccc(C(=O)NC(C)C(C)C)n1.N c1(OCC)oc(C)nc1C(N1CC(CNC(=O)CC2CCCOCC2)C1)=O C=CC(C)(CC)C(=O)NCC1=CCCN(C(c2cn(C(C)C)nc2C)=O)C1 N1(C(C2ON=C(C)C2)=O)CCC2(CCC2)C(NC(=O)CCC(C)(C)F)C1 C1(C2CCC2)(C(=O)OCCc2c(C)ccs2)CC1 c1(OC)cc(CN2CCSC(C(=O)Nc3sccc3C(N)=O)C2)c(OC)cc1C C(=O)(CC(C(F)(F)F)c1ccon1)NCCOCCCNC(C(CC)(C)C)=O CC(C)(O)C(C)CC.C1(C(=O)NCc2cc(C=O)no2)(COC)CCCO1 C#CCCCC(C)C(=O)NC1CCC(NC(c2ccc3ccoc3c2)=O)CC1 c1(CC(N2CCC(O)C2)=O)csc2ccccc12.C1(C(=O)N)C2CC3C(C2)C13 C1(NC(C2CC(C)(F)C2)=O)CN(C(c2cc(Br)no2)=O)C2(CCCCC2)C1 C(=O)(C=C(Cl)Cl)N(C(CNC(c1ncoc1)=O)C1CC1)C.c1ccccc1.C c1(-c2occ(COC(c3ccc(C)[nH]3)=O)n2)cccc(Br)c1 c1(C(N2CCC2)=O)ccccn1.c1(CC)conc1C(=O)N.CCN(C)C.C c1(CC)c(C(=O)NC(C)CCNC(=O)Cc2ccccc2SC)cnn1C c1(NCC(CC)(C)C)ccc(S(=O)(=O)N2CCOCC2CC(F)(F)F)cc1F CC(C(=O)N1CCN(CCNC(=O)CCCc2cnccn2)CC1)S(N)(=O)=O C1(CC(N2CCC(C)C2)=O)C(=O)N(C)N=C1C.C(=O)(COCC=O)NC.N c1(C=O)cnn(C)c1C#N.C1CCCCC1.C(=O)(C=CC(=O)N)OCC.C N1(C(CC(n2ccc(C)n2)C)=O)CCC(CO)(NC(=O)C=Cc2cnn(C)c2)C1 C1(C(=O)NC(CC)C(F)(F)F)C2CCN(C(=O)C=Cc3cncn3C)CC12 C1(C)(C(=O)N)CCC(=O)N(C)C1.C(CC(=O)N(C(C)C1CC1)C)N(C)CC CC(CC(=O)N1CCSCC(C)C1)C(C)(C)NC(=O)CC1(O)CCC1 C1(C(=O)NCC(CC=C)NC(c2ccc(F)o2)=O)CC(C(C)(C)C)=NO1 C1(NC(CCCCOCCC=C)=O)CCCN(C(C2CCCN2C)=O)C1C CC1CCC(NC(c2c(Cl)n[nH]c2C2CC2)=O)CN1C(c1csc(O)n1)=O n1(CC(C)C)ncc(C(=O)N(CC)C2CC2)c1C.C1(C=O)CC2CC1C2 C1(NC(c2ccc(N(C)C)cc2F)=O)CC2(CCCCC2)C1.C1(C(=O)N)CC1F C(=O)(C1=CC2(CN(C(=O)C3=CCCC3)C2)OC1)NCC1(C)CCCOC1 C1(C(N(CC(=C)C)C)=O)CCN(C(c2ncc(C)cc2F)=O)CC1C CCC(C)(C(=O)NC1CC(NC(=O)C(F)CC2CCC2)C1)C(F)F C1(NC(C2C(CC)=NC=C2)=O)CC12CCN(C(=O)Cc1ccc(C)s1)CC2 N1(C(CCC(=C)Cl)=O)CCCC(C2CCCN(C(=O)Cc3ccns3)C2)C1 C1(C(N(C(C#C)C)C)=O)CC(O)CN1C(=O)C=Cc1ccc(C)o1 C1(c2ccccc2)(N(C(C(OC)OC)=O)C)CCCCC1=O c1(OC)ccc2oc(C(N3CC(C)C(C)C3)C(=O)NCCSC)cc2c1 c1(C(=O)NC2CN(C(C(CC)C#N)=O)CC23CCC3)nccc2c(C)cccc12 CC1CC(CNC(=O)COC2CCOC2)CN1C(=O)CCC1CC1(C)C C(=O)(C(C)(C)CCNC(=O)CCN1CCOC1=O)N(C)CC1CC1(F)F C1(C(=O)NCCC2COCCN2C(C2CS(=O)(=O)C2)=O)CCn2ncnc2C1 N1(C(c2cc(C)c(-c3nn[nH]n3)nc2)=O)CCC2(C1)OCC1CC21 N1(C(C2N(C(=O)OC(C)(C)C)CCCC2)=O)CCCN(C(=O)CCC(F)F)CC1 C1(C(N2CC(CC(C)NC(c3c(C)nc(CC)o3)=O)C2)=O)OCCOC1(C)C C(=O)(C1CCc2c[nH]nc21)N(CCNC(c1cc(CCC)c(C)s1)=O)C1CC1 N1(C(C(C)OC)=O)CCC(C(C)(C)C(=O)NC2CC(c3ncc[nH]3)C2)C1 CCCCCCC(C)(CC)C(=O)NCC1CCCN1C(=O)Cc1ccc(N)cc1 C1(OCC)CC2CN(C(C3(NC(=O)CC(C)C(C)C)CC3(C)C)=O)CC12 Cc1nsc(C)c1C(N1CCN(C2CN(C(c3scnc3C(C)C)=O)C2)CC1)=O c1(CC(=O)NCC(CC)NC(C(C2CC2)OCC)=O)cc(C)cs1 C1(NC(c2cnn(C3CCOC3)n2)=O)CCC(CNC(c2ccnnc2)=O)CC1 C1(CC(N2CC(OCCC(N3CC(=C)C3)=O)C2)=O)CCC(C)(C)O1 C(C(O)CC(=O)N1CCCC1CNC(C1CCCN1c1ncccn1)=O)N(C)C Cc1[nH]nc(C(C)C)c1C(N1CCOC(CC)C1)=O.C(=O)CC.[SH](C)(=O)=O.N c1(C(=O)NCc2ccc(NC)cc2)cnc(C(C)(C)C)nc1C C1(OC)CCCCC1n1cc(C(=O)NC2(C3(OC)CCOCC3)CC2)nn1 N#Cc1ccc(C(=O)Nc2cncc(-n3cccn3)n2)cc1F C(=O)(C(C)C(C)NC(=O)C(CNC(c1cc(C)no1)=O)OC)OC C1(NC(C(CCOCC)NC(=O)CC2CC2)=O)CCCC2(CCC2)C1 NS(=O)(=O)c1cc(Br)cnc1NC1C2CCCC1CCC2 c1(CCC)nc(C)c(C(=O)N)o1.C(C(C)CC)=CC(=O)N(CC)C(C)C c1(C(C(N)=O)NC(C2(CNC3OCCO3)CC2)=O)ccc(Cl)cc1 N1(C=O)CCN(C(=O)N(C2(C)CCCOC2)CCN2CCOCC2)CC1.CC(C)C C1(n2cc(C3(F)CCOCC3)nn2)(C(=O)O)CCc2cc(Br)ccc2C1 N1(C(c2c(C)nsc2C)=O)CC(C2CCCCN(C(=O)CC3CCC(O)C3)C2)C1 N1(C(C(C)SC(C)C)=O)CC2CCOC2(CNC(c2cccc(F)c2F)=O)C1 c1(C(=O)NC2(C3CN(C(COCP(C)(C)=O)=O)C3)CC2)ccc2cnnn2c1 c1(OC)c(C(=O)NC2CC2)oc2ccccc12.C(=O)(C(F)(F)c1ccccc1)N O=C(C1=CCC(F)(F)CC1)NCC(F)CNC(=O)C(O)Cc1ccccn1 CC12CC(C(=O)N)(C1)C(C)(C)O2.C1(C)CCCN(C(C2CC(C)(O)C2)=O)C1 Cc1ccc(C(C)C(=O)NC(CNC(=O)CCCc2ccccn2)C2CC2)o1 CC(C)C(CCC(=O)NC1CC(=C2CC2)C1)NC(=O)C(C)Cn1ccnc1 N1(CC)CC(C(=O)NCC(CC(C)C)NC(=O)CCOC)NC1=O C(=O)(C1CSc2ccccc21)NC1CC(NC(c2cc3n(n2)CCC3)=O)C1 C12(C(=O)NC(CC)CN(C(=O)C(C)C3CC3)CC)CC(C=O)(CO1)C2 N1(C(C(c2cnn(C)c2)C)=O)CC2OCC(NC(c3cc(C4CC4)no3)=O)C2C1 CCCC(CC)C(=O)NC(CNC(c1cc(CC)ccc1O)=O)CO N1(c2c(C)cncn2)CCc2cc(NC(c3nccnc3Cl)=O)ccc2C1 N1(CC=O)C(=O)C(=O)N(C)C1=O.N1(CC)C(=O)CCC1C=O.C1CCC1 CN1CC(NCC(C)(C)CNC(c2cc(N3CCCC3)ncn2)=O)NC1=O N1(C(c2cc(C)n(C)c2)=O)CCC(NC(C2CCCCCCC2)=O)C(C)C1 CCCCCC(O)C(=O)N1C2CCC1CN(C(=O)C(=O)NCC)C2 Cc1ccc(CN2CCCC(NC(c3cnc(O)cc3O)=O)CC2)c(Br)c1 C1(C(N(C(CC)CC)CC)=O)CCCN(C(C2CCCN2C)=O)C1 Cc1ccc(CCCC(N2CCC(CCNC(C34CCC3C4)=O)CC2)=O)cc1 N1(C(=O)CCOCC2CC2)CC(NC(C2(Cl)CC2(F)F)=O)C(C2CC2)C1 c1(C(=O)OCC)c(NC(=O)C)cccc1F.c1(CCC=O)ccc(Br)cc1.O C1(NC(CC2CN(C)C2)=O)CCCC2CN(c3ncc(Cl)cn3)CC12 c1(C=O)cccc(C)c1Cl.C12COC(C(=O)NCC)(C1)C2.Cc1csc(S)n1 Cc1cc(NC(N2CC(=O)NC(C(C)C)C2)=O)nc(Cl)n1 Cc1ccc(C=CC(=O)NCCCCC(CO)NC(c2cncs2)=O)cc1Cl c1(CCOC)nc(=NCCC2CCN(C(c3cc(C)nc(O)n3)=O)CC2)s[nH]1 C1(C(N2C(C)CCC(NC(=O)CCc3cnoc3)C2)=O)COc2ccccc2O1 N1(C(C(C)C#N)=O)CCOCC(F)(CNC(c2ccc(F)cc2C(F)F)=O)C1 c1(N(CC(N2CC(NC(=O)CCF)C(F)C2)=O)C)nc(N2CCCC2)ncc1Cl c1(C(N2CC(NC(c3csc(O)n3)=O)C(F)C2)=O)cc(Cl)cc2c1NCCC2 C1(NC(c2cncs2)=O)CN(c2ncnc(Cl)c2[N+](=O)[O-])CCC12CCOCC2 c1(C(=O)N)nc(O)[nH]c(=O)n1.C(Cc1ccccc1)(C(=O)NCC(C)C)OC c1(OC)cccc(CNC(N2CCOC(C(C)(C)O)C2)=O)c1O.c1ccccc1 C1(COC)(COC)CC1C(=O)N(CCCNC(=O)C=O)C(C)C N1(CC)CC(NC(c2ccc(NC(c3nccnc3Br)=O)cc2)=O)C(C#N)C1 N1(C(C23CC4CC2C3C4)=O)CCn2c(C3CC3)nnc2C1.CC(C)C.C(=O)N Cc1ccc(C(N2CCC(F)C2)=O)c([N+](=O)[O-])c1.c1(C(=O)N)nccn1C(C)C C(=O)(CC(C)C(=O)N1CCN(C(=O)CCC2CCOC2)CC1CO)OC C1CC2CC2N1C(c1ccccc1)=O.Cc1csc(C(=O)N)c1.[SH](C)(=O)=O.C N1(C(c2c(CCC)nco2)=O)CC2C(C)C2C1.c1(C=O)nnn(C(C)(C)C)n1 CCCC(CCC)CC(=O)NC1CCN(C(=O)CCc2ccc(Br)s2)C1 C(=O)(CC(C)(C)N(C)C)N(C1CCN(CC(O)Cc2ccccc2)C1)CC C1(C(C)CNC(c2c[nH]c(=O)cn2)=O)CCN(C(=O)C(c2cncnc2)C)CC1 C1(CC(=O)N(C(CC)C)CCO)CC(C)N(C(=O)Cc2cc[nH]n2)C1 Cc1ccncc1C1CC1C(=O)NC1CC(NC(=O)CO)C1.c1ccnn1C C1(C)CCCC1.c1nc(C(C)C)c(C)s1.C1(CC(=O)NC)(OCC)CCC1 C(CN=c1[nH]c(=NCC2CSCCS2)c2[nH]ccc2[nH]1)N1CCC(C)C1 C(CCCCCC(=O)N1CCSCC1)n1cc(-c2cc(C)c(Br)nc2)nn1 CCC(O)C(C)C(=O)N1CCC(C)(c2cn(-c3cc(C)cnc3F)nn2)CC1 c1ccc(C)cc1.C1(C(=O)NC)(C(=O)N(CC(C)N(C(=O)C)C)C)CC1.O C12(C(=O)NCCCNC(=O)CC=CC(F)(F)F)CCC(CC1(F)F)C2 N1(C(C(C)C(C)O)=O)CCC2(CC1)COC(C)C2.C1(CC(=O)N)SC(=N)NC1=O C1(C(=O)NCC2(O)CCN(C(COC(C)(C)C)=O)C2)COc2ccccc2O1 CC(CN1CCOCC1)C(=O)NC1CCCC1NC(C1CC(F)(CO)C1)=O C1(=CC(=O)NCc2cc(CN(C)C)no2)CCN(C(=O)C=CI)CC1 c1(C(C)C)nnsc1C(=O)NCC(C)Cn1cccn1.c1(CC=O)ccsc1.N c1(C(N2C3(CNC(Cc4c(C)con4)=O)CCC2CC3)=O)n[nH]c2ccccc12 c1(C(=O)NCC2CC(C)N(C(=O)CN3CC(=O)NC3=O)C2)cccn2cncc12 C(=O)(CCCC(C)=O)NC(Cc1ccc(CNC(C(C)(C)SC)=O)cc1)C c1(C(=O)NC(C2CCN(C(c3c(C)cn(C)n3)=O)C2)(C)C)cc2c(s1)CCCC2 c1(C(=O)Nc2cn(C)c(C(N3CCC(O)C3)=O)n2)cc2cnccc2[nH]1 C#CC1(O)CCN(C(c2coc(CNC(=O)C(F)(F)C(C)O)n2)=O)CC1 N1(C(C2(CCC=C)CC2)=O)CCCC2(CC(NC(=O)CC3CCCCCC3)C2)C1 C1COC2(C1)CN(C(=O)C)C2.n1(CCC)ccnc1C(F)(F)C=O.C(N)=O.N c1(C(=O)NCc2c(CC)c[nH]n2)snc2ccc(Br)cc12 C#CCCCC(C)C(=O)NCC(CCCC)NC(c1scc(OC)c1OC)=O N1(C(c2ccc(N(C)C)nn2)=O)CCC2(CCCN2C(C2CC2Cl)=O)CC1 c1(C(=O)NC2CN(C(C34CC(OC)C3C4)=O)CC2C)cc(C)cc(Cl)c1 C12(C(=O)NCC(c3nccs3)C)CCC(CC1)C2(C)C C1(NC(CCOC)=O)CC2CN(C(=O)CCOc3cccc(C(N)=O)c3)CC2C1 C1(C(=O)NC(C2Oc3ccccc3C2C)C)CC(c2cccc(Br)c2)=NO1 CC(C)(O)C(F)C(=O)NCCCCCCNC(c1ccccc1C(F)(F)F)=O C(=O)(C#CC1(CN)CC1)NC1C(OC)CCCC1 C1(OC)CN(C(c2cc(C)cc(O)n2)=O)C(C)(C)C1.C(=O)CC.C(C)=O.N C1(F)(CNC(=O)C=C(Cl)Cl)COCCN(C(C2CCn3nncc3C2)=O)C1 N1(C(C(C2(C)CC2)NC(CC=C(C)C)=O)=O)CC(F)(F)C(F)(F)C1 c1(CCC(=O)NCC#CCNC(c2cc(Cl)no2)=O)ccc(F)cc1 C1(CC(N2CC(O)(CC)C2)=O)CC(O)C12CCC2.c1(OC)n[nH]cc1C=O.N C(=O)(CC(CC)CCCC)NC(CC=C)CNC(C1(C(C)(F)F)CCOCC1)=O c1(NCc2nn(C)c(C(F)F)c2)ncc([SH](=O)=O)cc1Cl.C1(CC#N)CC1.N c1(OCC)ccc(C(=O)NC2C=CCN(C(=O)C(C)N=[N+]=[N-])C2)cc1 C12(C(=O)NCCCCCC(C)(C)C)CCC(=O)N1c1ccccc1S2 c1(OCC)ccc(NC(c2cc(-c3ccc(CO)nc3)[nH]n2)=O)c(OC)n1 N1(C(C(C)n2cncn2)=O)CC2(CCN(C(=O)C(F)(F)C(F)F)C2)C1 Cc1nc(C(C)NC2(c3nnnn3C3CCC3)CC(c3ncc[nH]3)C2)no1 C1C2CC3C1C3C2C(N1CCN(C(=O)C2CC2)CC1)=O.O=CCCC1CCC1.N c1(CC)cc(C(=O)NCC2CCOCC2)nn1C.C1(C=O)CC1C(C)(C)C c1(CC)cc(C(=O)NC(C2(O)CN(C(c3n[nH]cc3F)=O)C2)C)nn1C C1(CNC(C(N)=O)=O)Cc2ccccc2CN1C(=O)C1=CCCCO1 CCC(C(=O)N1CC(CN(C(=O)Cc2cnc(C)o2)C)C1)n1ccc(C)n1.S CC1CN(C(=O)CC(C)(C)CN(C)C)CC(C(=O)N(C)CCN(C)C)O1 C1(N(C(c2csc(CC)n2)C(=O)NCC=C)C)CN2CCC1CC2 c1(C(N(CCN(C(c2nnc(C)o2)C)C)C)=O)sc2ccccc2c1Br N1(C(C2(C)COC2)=O)CCN(c2ccncn2)C2CC12 N1(C(c2c(O)cc(C)nn2)=O)C2CCC1CC(C)C2.C1(C(=O)N)CC(C(C)C)C1 CC1(n2nc(-c3cc[nH]n3)nc2Cn2ncnn2)CCS(=O)(=O)C1 c1(C(N2CCC3(NC(c4occc4Cl)=O)C(CC2)C3)=O)cccc2ncccc12 N1(C(CC=CC)=O)CCCC1C1CCN(C(C2(COC)CC=CC2)=O)C1 c1(-n2cc(C(CCC)NC(c3cccc(OC)c3)=O)nn2)ccccc1CCO c1(C(N(C2CCCC2)CC)=O)cc(F)cs1.c1(C(=O)N)cnn(C2CCC2)c1 Cc1ccc(C(N2CC3C(CC(=O)NCCC#CC(C)(C)C)C3C2)=O)cc1O c1(C(N(C)CC2OCCN(C(C(C(C)C)F)=O)C2)=O)cc2c(s1)CCCCC2 CC(Cc1cccnc1)C(=O)N1CCCC1CNC(=O)C.C(=O)N.C1CC1 C1(NC(C(C)NC(=O)NC2CCCC2)=O)CCN(c2nnnn2C)C1 C#CCC(CC(=O)NCC(F)(F)CO)NC(=O)Cn1cc(C)cn1 C1(C(=O)NC(C)CNC(=O)OC)(CC)CCCN1C(C1CN(C)C1)=O N1(C(C(C)CC(N)=O)=O)CCN(C(c2ccc(C(C)(C)C)cc2)=O)CC(CO)C1 c1(C(=O)NC2CCC(NC(c3ncccn3)=O)C2)ccnc2[nH]nnc12 n1(CC(=O)NC(CNC(C(CCC)O)=O)COC)nc(O)ccc1=O N1(C(c2c(OC)ccnc2)=O)CC2CN(C(C3CCCCNC3=O)=O)CC(C1)O2 Cc1cccc2n[nH]c(=NC(C)C(=O)Nc3ccc(OC(F)F)cc3)n12 c1(C(N2CCC(C)(CCNC(=O)C3=CCCS3)C2)=O)csc(=NC2CC2)[nH]1 C1(C(N2CC(N(C(c3c(C)nns3)=O)C)C3(C2)CC3)=O)COC2(CCC2)CO1 CCCCC(O)C(C)C(=O)N(CC(C)NC(c1cc(C)nn1CCC)=O)C CC1CCn2cc(C(=O)NCCCC3CCCN3CCc3cnn(C)c3)nc2C1 N1(C(c2cnn(C(C)C)n2)=O)CCC2CN(C(C3CCC=CCCC3)=O)CC2C1 CC(C)(C)S(=O)(=O)CC(=O)NC12CCC1CN(C(c1csnn1)=O)C2 C(=O)(C1=CC2(CCN(C(c3ccc(C(C)C)o3)=O)C2)C1)N1C(CC=O)CC1 c1(C=O)c([N+](=O)[O-])cnn1C.Cc1[nH]cc(C(N2CCC(C)C2C)=O)c(=O)c1.N Cn1nnc2cc(C(=O)NCC(O)CNC(c3cscc3Cl)=O)sc12 C(=O)(N=c1ccn(CC(N)=O)[nH]1)C1CC1CC=CC(=O)NOC(C(CC#C)O)=O CC1CN(C(C2(c3ccsc3)CC2)=O)CCC1NC(c1ccc(CCO)cc1)=O C(=O)(C1(C)CCOc2ccccc21)NCC(CN(C(=O)C)C)O.CC(C)(C)C.O C(c1cccnc1)=CC(N1CC(O)(C(F)C(=O)N2CC(C(F)(F)F)C2)C1)=O C(=O)(C(C)(C)C(C)(C)O)N1CCC(C(=O)NCC(C(CC)C)CO)OCC1 Cc1ccc(NC(=O)C(C)N(C)CCN2CCN(C)CC2)c(C)c1 c1(CNC(=O)CC(O)C2CCCC2)cccc2c1CCNC2 c1(C(N2CC(CC(C)NC(c3ccc(C)cc3C)=O)C2)=O)cc(F)c(F)cc1O C1(C(N(CCNC(CN2CC(C)(OC)C2)=O)C2CC2)=O)CCOCC1(C)C c1(C(N2C(CCC)CN(C(=O)C(C)C(O)CC)CC2)=O)cc(F)cc(F)c1OC C1(COC)CC(C)N(C(=O)Cc2c[nH]nc2C)C1.C(=O)(CCC1CCC1)N c1(C(=O)NC(C(CO)NC(COc2cccc(OC)c2)=O)C)ccc(Cl)cc1C C(C1CN(C(C2CC(C(C)C)C2)=O)CC1C(=O)N(C1CC1C)C)=CC C(=O)(C(C)(CO)NC(=O)CC#N)NC(CC=C)C O=C(CS(=O)(=O)CCO)N(C1CC1)CC1CCCN1C(=O)Cc1cnoc1 c1(C(N2CC(O)(CNC(C3CC(SC)C3)=O)C2)=O)sc(F)cc1C N1(C(C(C(C)OCC)n2cc(-c3cnn(C)c3)nn2)=O)CC2CCC=CC12 N1(C(C(C2CCOCC2)OCC)=O)CCC(C)CC1.c1(CC=O)c(C)noc1C.N c1(C(=O)NC(C)C(C)(C)NC(C2CCC(C(N)=O)CC2)=O)cc2cn[nH]c2cn1 C12CC(C1)N(C(c1cc(C(C)C)[nH]n1)=O)C2.C(=O)CN(CC=O)C.CCC N1(C(C2CCC(C)N2Cc2ccc(O)cc2Br)=O)CC(C(N)=O)C2(CC2)C1 C(=O)(CCC(C)(C)C#N)N1CCCCC(CNC(c2c(SCC)cccc2)=O)C1 CCC(CC)CCC(=O)N1CCC(O)CC1C(N1CCCOC(CC)C1)=O N1(C(CSCCOC)=O)CC2CCCC2(C(=O)NCC2CN3CCC2C3)C1 c1(N2CCC(NC(c3cc(C)c(F)nc3)=O)CC2C)cc(C#N)nc(C2CC2)n1 C1(CCC)(NC(=O)CC(C)CN(C)C)CCCN(C(c2cnn(CC)c2F)=O)C1 CN1C2CCC1CN(C(c1c(CNC(=O)CCNC(N)=O)nnn1C)=O)C2 c1(OC)cc(C(F)(F)F)nc(N2CCCC2C(C)(C)NC(=O)C(O)C(C)C)n1 N1(C(C(C)SC)=O)CCCC2(C1)CN(C(c1ccc(C(N)=O)nc1)=O)CCO2 C1CCC2CC(c3nnnn3C3COC3)(NC34CCC(CC3)C4)C2C1 N1(CC(=O)NCC(CC)N(C(=O)COCC(C)(C)C)C)CCCCC1=O C(C(=O)NCCNC(=O)CCc1ccoc1)(C(C)C)n1ccc(C)c1 c1(OCCNC(c2cc(C)c(C(F)F)cn2)=O)ccc([N+](=O)[O-])c(C)c1 CCCCC(C(=O)N1CC(CO)(NC(=O)CCC(C)(C)OC)C1)NC(N)=O c1(OC)cccc(-n2nc(-c3cnn(C)c3)nc2C2CCS2(=O)=O)c1 C(CN=c1ccnc(C(C)C)[nH]1)C1(O)CCN(C(c2n(CC)ccc2)=O)CC1 N1(C(c2nc(CCC)oc2)=O)CCCC(C)(C)C1.N1(CC=O)CCNC(=O)C1.N Cc1noc(N)c1C(=O)NC1CCCC1NC(c1n[nH]cc1-c1ccccc1)=O c1(CC)cc(F)ccc1C(=O)N(CC(C)N(C)C(c1ocnc1C(F)F)=O)C c1(C(C2CC2)NC(N2CCCC(C#C)(C)C2)=O)ccc2nc(C)oc2c1 c1(C(N2CC(C(=O)Nc3cccc(Br)n3)C2)=O)cc(OC(F)(F)F)ccc1O c1(C(N2CC(C#C)(C(N3CCC3C(C)O)=O)C2)=O)cc2cccn2cn1 C1(CNC(=O)Cn2cncn2)C2CC1N(C(c1cn(C3CCOCC3)nn1)=O)C2 c1(C(C)=O)cccc(-c2cn(CC3CCC(NC(=O)CO)C3)nn2)c1.C1CC1 CC(C)=C=CC(=O)NC1COCC1NC(=O)C(c1ccn(C)n1)C C1(CCCC)CCC(C(=O)NC(CN(C(=O)Cn2ncccc2=O)C)CC)CC1 c1(CNC)ccc(CC(N2CCC2CC2(CC(=O)OC)CC2)=O)cc1 C(=O)(C(O)CC(C)C)NCC1CCN(C(CCCc2ccc(OC)cc2)=O)C1 C(=O)(C(C)(C)CS(C)(=O)=O)N1CC(O)(CC)C1.C(=O)CN(C)C=O.C N1(C(Cc2c(C)cco2)=O)CC2CCC2(CNC(c2ccncc2Cl)=O)C1 c1(NC(C2(C)CCN(C(C(c3ccccc3)C)=O)C2)=O)ncnc2[nH]c(Br)nc12 C(=O)C(=O)N=c1cc(C)o[nH]1.C1(COC)CCN(C(C2CC(C)CO2)=O)CC1.N c1(CC)noc(COCC(=O)NCC2C=CCN2C(C2C=CCC2)=O)n1 C(=O)(C(C)N(C)N1CCN(C)C2(CCOCC2)CC1)OC C1CN(C(c2cc(C)cc(O)c2)=O)CC(C)(C)O1.C(CCC(=O)N)OCC=C.C C1(OC)CCN(CCNC(=O)CN(C(=O)C(O)CN(C)C)CC)C1.O c1(COC23CCCN(C(=O)OC(C)(C)C)C2C3)cc(O)c(O)c(O)c1 Cc1ccc(C)c(CC(N2CCC(CF)(NC(c3cnncc3O)=O)C2)=O)c1 C(=O)(C1CCCc2scnc21)N1CCC(NC(CNS(N)(=O)=O)=O)C12CC2 C1(NC(C2(OC)CCC2)=O)CC2CC1CN(C(=O)CC1CC(OC)C1)C2 N1(C(C)C(=O)NCC2CCCC2)C(=O)c2ccccc2C1=O.C(=O)(C)N.CCF N1(C(CC2C(C)(C)COC2)=O)CCOC2CN(C(c3cn(C4CC4)nn3)=O)CC12 c1(CC(N2CCC(C)(CNC(CCC(=C)Cl)=O)C2)=O)cc(Cl)cc(Cl)c1 C(=O)(C(C(C)CC)N(C(=O)Cn1cc(C)cn1)C)N(CC(CCC)C)C N1(C(COCCC=C)=O)CC2CC1(CNC(=O)CSc1nncs1)C2 C1(C2CCN(C(=O)CCc3ccccc3)C2)CCCCN1C(=O)C(O)C1CCC1 C(CCCCC(=O)N1CC(CNC(C23CC(CO)(C2)C3)=O)CC1C)=CC Cc1nc(Cl)ccc1S(=O)(=O)N1CCSC(C(=O)Nc2c(O)cccc2Br)C1 c1(OC)cnccc1C(=O)NCCCOCCC.C1(C=O)CCC2(CC2)C1.N C1(CNC(C2CCN(C)CC2)=O)CCN(Cc2scc3c2OCCO3)CC1(F)F c1(-c2cc(OCC)ncc2)c(C(=O)NC(C2CCOCC2)C)nn2c1CCCC2 Cc1cc(C(N2CCC(C)CC2C(=O)NC2COC(C(F)F)C2)=O)cnc1O c1(C(=O)NCCC(C(C)C)NC(C2CCO2)=O)c(S(N)(=O)=O)cnn1C N1(C(COC)=O)CCC2OCCN(C(c3ccn4c(O)nnc4c3)=O)C2C1 c1(NC(C2(F)CN(Cc3cccc(OC(F)F)c3)C2)=O)ccc2ncccc2c1 c1(C(N2CCCCC(NC(C(CC)(C)O)=O)C2)=O)cc(=O)c2cc(O)ccc2o1 C1(C(=O)Nc2ccc(C)c(O)c2)CN(C(C2CCC3CC23)=O)C2(CCC2)C1 N1(C(CCC(C)SC)=O)CC2(CCC2NC(=O)COC2(C)CCCC2)C1 c1(NC(C2OCCN(C(CN(C(C)C)C)=O)C2)=O)cc(N(C)C)ccc1Br CC1CC2(CO1)CN(C(C1CCCCCN1C(=O)CCCc1ncco1)=O)C2 c1(C(=O)N)n[nH]c2cc(C=O)ccc12.Cc1cccc(F)n1.C(C1CC1)C1CC1 C=CCCC(C)(C)CNC(=O)C(CCC=C)NC(C1C=C(C)CS1)=O C(C(C(=O)NCC(F)Br)NC(=O)C(C)OCC1CC1)OC C12(C(=O)NC3(C(N4CCC(CC5CCC5)C4)=O)CCC3)CC1CNC2=O c1(OC)ccccc1-c1ncc(C(=O)OCc2cc(C(=O)O)on2)s1 C#CCC(O)C(=O)NC1CCCC1NC(=O)Cc1csc(C)c1 c1(OCC=C)c(C(N2CC(CNC(=O)CC(C)(C)C)C2)=O)cccc1C C1(C(N(CCCNC(C(CC)C#N)=O)CCO)=O)CCc2ccccc2C1 c1(C(=O)N)cc(Cl)c(Cl)cc1.C1(C(=O)OC)CCC1C(=O)NC1CCC1 N1(c2nnc(Cc3c(OC)cccn3)n2CCC#N)CC(C)C(F)(F)C(C)C1 c1(NC(C2CCCN(C(c3nc(Br)cs3)=O)C2)=O)cc(Cl)c(F)c(Cl)c1 CCC(C)C(C(=O)NC1CC(C)CCC1O)N(C(=O)CCc1cncs1)C N1(C(=O)C(C23CCC(CC2)C3)F)CCC2CCN(C(c3cc(=O)cc[nH]3)=O)C2C1 N1(C(C2C(=C)C2)=O)CCCC(C)(CNC(c2c(C)cccc2F)=O)C1 Cc1ccc(NC(=O)C(=O)N)cc1C.C(=O)(CC(C)(C)C#N)N1CC2CC2C1.C Cc1c(C(N2CCC(C)CC2CNC(=O)C=Cc2ccsc2)=O)[nH]ccc1=O CCCC(C)(C)C(=O)N1CCC(CNC(C2(C)CC=CCO2)=O)(COC)C1 c1(N2CCCC(NC(C3CN(CCC)C(=O)C3)=O)(CO)C2)nc2ccccc2o1 Cc1cc(S(=O)(=O)Nc2nc(C3CC3(F)F)cs2)cc(C(=O)O)c1F C1(C(N2CC(F)CC(NC(=O)C=Cc3cocn3)C2)=O)Cc2ccccc2CO1 N1(C(C2(O)C(C)(C)C2)=O)CCC(NC(C2CCCOCC2)=O)C2(CCC2)C1 CCC(C)(O)C(=O)NC.C1CC(F)CN1C(c1ccccc1)=O.C(=O)C1CC1 c1(OC)ncc(C(=O)NCc2cc(F)ccc2Cl)cc1-c1cc(F)ccc1CO N1(C(COC)=O)CCC(NC(c2ccnn2CC(C)C)=O)C1(C)C N1(C(Cc2cc(C)ns2)=O)CCC2(CC1)CCN(C(C1CCC(C)C1)=O)C2 C1(C)(CNCc2c(OCC)cccc2)CCC(F)(F)C1 C(=O)(C#CC1CCCCO1)N1CCC(CCOC)(NC(=O)CCC(=O)NC)CC1 c1(CC(=O)NC(=O)CC(=O)NC2CCCN(c3ncccn3)C2)ncc(Cl)cc1F C#CC1(NC(=O)C(C)C(=O)OC)CN2CCC1CC2 Cc1cc(C(C)(C)C)ccc1NC(=O)NC(C(=O)O)C1CC(C(=O)O)C1 C1(C(N(CCCOC)CCO)=O)CC12CC(NC(c1occc1C)=O)C2 c1(C(=O)NCC(C)NC(=O)CC2CCN(C)C2)cccn2nnnc12 C(=O)(C(=O)C(C)(C)C)N1CCCC(CCNC(c2nc(CCC)oc2)=O)C1 c1(SCC(=O)NC(CN(C(c2ccc(O)s2)=O)CC)C)cccc(Cl)c1 c1(C(N2CCC3(NC(=O)C(F)=C4CCCC4)C(C2)C3)=O)ccc2cc[nH]c2n1 c1(CCN(C(=O)C(C2CCN(C(=O)C=Cc3cc[nH]n3)C2)F)C)ccccn1 C1(C(C(=O)NCCC(=O)OCC)N(CCC)CCC)CCCOC1 C(CCOCC)(C(=O)N1CC(O)(C(F)(F)F)C1)NC(CC=C=C)=O c1(C(=O)N)c(OC(F)F)cccc1F.C1(CNC(=O)COCCF)CCCCC1 CC1=C(C(=O)NCCC2CCN(C(C3(C(C)C)COC3)=O)C2)SCCO1 C(=O)(C1=CC2CCC(C1)C2)NC(c1occ(C(NOCCOC(C)C)=O)n1)C Cc1ccc(F)c(NC(C23CC2CN(C(=O)CN2CCOC2=O)C3)=O)c1 N1(C(CC(C)(C)O)=O)CC(CNC(C2CC2Br)=O)CC1(C)C C12(CNC(c3c(CNC(=O)CCC4CCCOC4)cc[nH]3)=O)CCCC1CCO2 N1(C(C2CC(C)(O)C2)=O)CC2CC(C(=O)NCCN3CCOCC3=O)C(C2)C1 c1(OC)cc(NC(=O)C(=O)NC2CC2)ccc1NC(=O)C(C)(C)C#N CC12CCN(CC1)CC2NC(=O)CC1CCCN(C(c2cnnc(O)c2)=O)C1 Cn1nccc1C(C(=O)NC1CN(C(N)=O)C1)NC(C1CC1[N+](=O)[O-])=O C1(CCC)C(=O)NCCN1C(=O)C(CCC1CC1)NC(=O)C(C1CCOCC1)=O c1(C(=O)NCC(CO)NC(C2ON=C(C)C2)=O)cc(S(N)(=O)=O)cs1 C1(NC(c2ccc(C3CC3)o2)=O)CC2(C1)CC2C=O.C1(CC)CCOC1.N N1(C(c2c(C)ncn2C)=O)CCC(C)N(C(c2ccnn2CCF)=O)CC1 Cc1nn[nH]c1CNC(C1C=CC(NC(c2ccc(C3CC3)o2)=O)C1)=O C12(C(=O)NCc3c(C(N4CCC(C(C)O)C4)=O)n[nH]c3)CCC(CC1)CO2 c1(C(N(C2CN(C(C(CC=C)OC)=O)CC2(C)C)C)=O)cn2c(C)cccc2n1 C1(C)(C(N2CC(C)(NC(c3ccsc3I)=O)C2)=O)CC=CCC1 c1(C(=O)NC2(CO)CCCN(C(COCCC#C)=O)C2)cc2c(cn1)CCCC2 c1(OCC)nc(C)ccc1C(=O)NC(C)CC(C)NC(C1CCC(C)C1)=O c1(CC)ncncc1NC(=O)C(F)=CC1CC1 c1(OC)ccc(OC)c(C(=O)NCC(O)C)c1N.N1(CC(=O)N)CC2CC2C1 C1(NC(C(C)NC(=O)NC)=O)CC(c2ccccc2)C1.C(=O)N.C(C)C C#Cc1ccc(CCC(N2CCN(C(=O)C(O)P(C)(C)=O)C(CO)C2)=O)cc1 c1(C(N2CC(NC(C3CC3(F)Cl)=O)(CO)C2)=O)ccc(F)cc1 Cc1oc(C#N)cc1C(=O)NC(CC(C)C)C(=O)N(C)C[Si](C)(C)C C(c1cccc(F)c1)=C(C(N1CCC(CCCCNC(C(N)=O)=O)CC1)=O)F CC1OCCNC1C(=O)NC1CC(Cc2nn[nH]n2)C1 C1(NC(CC(CN(C)C)O)=O)CC2CC1N(C(=O)Cn1ccc(C3CC3)n1)C2 Cc1ccc(S(C)(=O)=O)cc1C(=O)NC1CCCC1.C1(C=O)CCC(C)CC1.N C1(C(=O)N)CCS1(=O)=O.CC(CNC(C1(CC)CC1)=O)Cc1cn[nH]c1 N1(Cc2ncn(C)n2)CCCCC(C)(C)C1.C1(C=O)CC(=O)N(C(C)(C)C)C1.N Cc1nn2ncccc2c1C(=O)NCC(C)NC(C1CC(=O)N(C(C)C)C1)=O c1(C(=O)NC(CNC(c2cc(OC)c(C)cc2)=O)(C)C)cccc2nc(Cl)cn12 Cc1nccn1CCC(=O)NCC(CO)NC(C1(C(F)(F)F)CCCC1)=O C1(NC(c2c(C)sc(Cl)n2)=O)CC2CC(NC(C3(F)CCC(C)CC3)=O)C1C2 C(=O)(C1=CCCCC1P(C)(C)=O)NCCCNC(CCC1COC(C)(C)O1)=O Cc1cc(CCC(=O)N(C2CCN(C(C3COCCO3)=O)CC2)CCO)c(C)s1 c1(NC(C(=O)NCCCOC)=O)cc(Br)c(F)cc1C(=O)OC C1(NC(C2(SCC)CC2)=O)CCCN(C(=O)Cc2ccnc(Cl)c2F)CC1 Cc1cc(C#N)ccc1C(=O)N(C1(C(=O)NC2CCN(C)CC2C#N)CC1)C N1(C(=O)CC2(O)CCCC2)CCCN(C(=O)Cn2cnnc2)CC1 Cc1cc(CN(C(C(=O)NC2CCOCC2)c2nccs2)C)cc(C#N)c1 N1(C(c2cc(C(C)=O)oc2)=O)CCCC(CCNC(=O)Cc2cc[nH]n2)C1 C1(CCC(=O)N(C2CCC2)C)NC(=O)NC1=O.c1(C=O)csc(C(F)F)n1.N N#Cc1ccc(C(N2CC(NC(=O)C=CCN3CCOCC3)CC(F)C2)=O)nc1 O=C(O)C#CC(=O)N1CCSC(C(=O)Nc2ccc(N3C(=O)C=CC3=O)cc2)C1 N1(C(C23C(CN(C(C4C(C=C)OCC4)=O)C2)C3)=O)Cc2ccc([N+](=O)[O-])cc2C1 c1(CN2C(C(N3CCN(C(=O)OC)CC3)=O)CSCC2)c(F)c(F)cc(F)c1F N1(C(C2CCC(=C)CC2)=O)CC2CC(NC(=O)CN(C)C3CC3)CC(C2)C1 c1(SC(C)(C)C)nccc(=NCc2csnn2)[nH]1 N1(C(C2C(CC)N(C(=O)COC(C)C)CC2)=O)CCC12CCN(C)C2 C(CCCCCC(=O)Nc1cncnc1C)NC(C(C=C)O)=O CCCCC(C(=O)NOC1CCN(C)CC1)NC(C1CCS1(=O)=O)=O C=CCC(C)(CC)C(=O)NC(CC(N1CCOC(C2(C)CC2)C1)=O)C1CC1 C1(NC(c2cccs2)=O)CCN(C(c2ccnc(O)c2F)=O)CC1F c1(CCC(=O)NCCN(C(=O)CC2OCCC2C)CC)ccc(O)c(C)c1 c1(C(=O)OCCCC)ccc(SCCC)cc1 c1ccc(Cl)cc1F.C(C(C)C(C)C)NC(C=CC(CC)=CC)=O.C(=O)C c1(NC(C(C)C)=O)ccc(NC(=O)CC(N)c2cccnc2)cc1 Cc1nc(CNC(=O)C(c2cncn2C)O)oc1C(=O)NCC(O)CCO CCCCCCCCCC(O)C(=O)OC1CCC1C(F)(F)F C1(NC(CC(C)OC)=O)CN(C(C2CCCC2S(C)(=O)=O)=O)Cc2nccn2C1 N1(C(c2c(C)ncs2)=O)CCOC(C)C1C(=O)NCC(C)C(C)C c1(OCCOC)cccc(C(=O)NCC2CCC3CC23)c1Cl C(=O)(CC(C)(C)CCOC)NC(CC)(CC)CCNC(C1(O)CC1(C)C)=O CC(C)C(C)(C)C(=O)N1CC(C(=O)NCC)C1.C1(C=O)CCCC(C#N)C1.N c1(C(N2C(CC(=O)Nc3c[nH]c4ncccc34)CCC2)=O)cc2cc(Cl)ccc2[nH]1 C12(C(N3CCN(CC)CC3)=O)CC(C)(CN1C(C1CCCCO1)=O)C2 c1(C(=O)NCC2N(C(C3OCCN(C)C3)=O)CC=C2)cnc2[nH]cncc1-2 N1(C(C2CCCC2)CNCC(c2n(C)ccc2)=O)CSCCSC1 N1(C(C(C)SCCCC)=O)C2CCC1C(NC(c1cccnn1)=O)C2 CC1(C)CC(n2nnc(C3CC3)n2)(C(=O)Nc2ccc(OC3CC3)cc2)CCO1 C1(C(=O)NCC2CN(C(C3C4CCC34)=O)C2)CC2CC(O)CC(C1)C2 c1(C(N2CCC2)=O)ccc(-c2cnn[nH]2)cc1.c1(C(N)=O)ccc(C(=O)NC)[nH]1 C(CN(C(=O)CC(C)n1cccc1)C)(CO)(CO)NC(C(C)CC1CC1)=O CC1CN(C(=O)C(C)(F)F)CC(CCNC(c2cnnn2C)=O)O1 n1(CCOc2c(N)c(Br)ccc2Cl)c(=O)c(C2CC2)nc2ccccc12 C1(N(C)C(c2cnc(C(C)(C)C)[nH]2)=O)CCCN(C(c2ccncc2Cl)=O)CC1 c1(C(N2CCOC(c3cnn[nH]3)C2)C(=O)NCCC)nccc(OC)c1OC c1(C(N2CCN(C3CCCN(C(C=CC)=O)C3)CC2)=O)cc(C(F)F)cc(F)c1 CC(C(F)C(=O)N1C2CCC1(CNC(=O)CCCc1cccs1)CC2)C(F)(F)F c1(C=O)coc(C(N)=O)c1.C1(O)(CC)CN(C)C1.c1cnc(C(F)(F)F)s1 N1(C(COCCCC(C)C)=O)CC2CC1(C(=O)N(C)CC1(F)CCC1)C2 C1(NC(C2N(CCC)CCC2)=O)CCOCCC1(F)F CC(C)(O)CC(=O)NC(CNC(=O)C(C1CCCCC1)=O)C(C)(C)C C1(CC(=O)N(CCOC)CCO)CCCC(NC(C2(Cl)CC2)=O)C1 O=C(CCCC(F)(F)F)N(CC(=O)O)Cc1cn(-c2ccccc2Cl)nn1 c1(C=O)cnn2ccsc12.C(C)(C)C(C)C.C1(C(C(=O)N)OC)CC(F)(F)C1 Cc1nc(=N)[nH]cc1C(N1CCCC(C(C)(O)CNC(c2ncoc2C)=O)C1)=O CCCC(C)(O)C(=O)N(C(C)CNC(c1ocnc1CC)=O)C C1(O)(CNC(C(Cn2cccn2)NC(C(C)C2CCC2)=O)=O)CCCOC1 C1(C(=O)NCC2(O)CCN(C(c3ccsc3)=O)C2)CCC2(CCOCC2)O1 C(=O)(C(C1=NOCC1)N1CCC(OCCOC)CC1)OCC C=Cc1ccc(C(N2CCC(NC(C3CCCN(C)C3)=O)C(O)C2)=O)cc1 N1(CC)CCCC(CCO)C1.n1(CC)ccc(C(N2CCC(C(F)C=O)C2)=O)n1 CC(=O)CC(C)(C)CC(=O)N(CC(O)CN(c1nc(Cl)nc2c1CCC2)C)C S(=O)(=O)(c1ccc(Br)cc1N1CCCC2(CCOC2)C1)NC(c1ncn(C)n1)C N1(CCC)CC(C(N2CC(CNC(=O)C(C#N)CC)C2)=O)CC1=O C1(C=O)CC(C)(C)OC(C)(C)C1.C(C)(C(=O)NC1CC1)OCCC=C.C C1(CCC)CN(C(=O)C(C)OCCOC)CCN1C(=O)C.C(=O)(CCCCO)N Cc1cc(NC(=O)Cc2ccoc2)cc(-c2cccc(C(F)(F)F)n2)c1 N1(C(C(C(CC)C)OC)=O)CC2(CCN(C(=O)CCN3CCCC3)CC2)CC1C O=C(CCCCO)NCCCCn1cc(C2CCCCO2)nn1 N1(C(C2OCCN(CC)C2)=O)C2CCC(C2)C1C.C1(C(=O)N)CCS(=O)CC1 CCC(C)(C(=O)NCC(CCOC)NC(c1ccc(-n2ccnc2)cc1)=O)OC C1(NC(C2(CC)CC(=O)C2)=O)CCCC(CN(C)C)C1 c1(C(N(CC(C)NC(=O)C2=C(Cl)CC2)CC)=O)cnn2c(OC)cccc12 CCC(CCCC(=O)NC1COCCN(C)C1)NC(C1(C)CC=CCC1)=O CCCC(C)(CCC)C(=O)NC1CN(C(c2n[nH]cc2CC)=O)C(C)(COC)C1 CC1(C)OCCC1CCNC(=O)C(Cc1ccoc1)NC(c1cnn[nH]1)=O N1(C(C2(C)C(C)CCC2)=O)CCC(O)(CCNC(=O)CCc2cn(C)nn2)CC1 c1(OC)nccc(C(=O)NCC2CC2NC(=O)CNS(N)(=O)=O)c1F Cc1cnc(CNc2cnc(C(=O)O)c(F)c2)cc1Br Cc1cc(C(=O)NC(C)CNC(C2CCCC2C2CC2)=O)cc(N)c1Cl c1(C(=O)OC)ccc(C(=O)NC(C)(C)CO)cc1C.C(=O)C1=C(C)CCC1.N N#Cc1ncccc1-c1ccnc(NC(c2cc(=O)cco2)=O)c1 C1(NC(C(C(CC)C)O)=O)CCC2(CC1)CCN(C(=O)CCCOC(C)(C)C)C2 N1(C(C2N(C(C)=O)CC(O)C2)=O)CCC2(CCN(C(=O)C=CC=C(Cl)Cl)C2)C1 C1(CNC(C2(OC)CC2)=O)CCC2CN(C(c3cc(CO)oc3C)=O)CCC2C1 N1(C(c2ncc(C)s2)=O)CC2C(C(=O)NCc3cc(Br)cs3)C2C1 Cn1c(Cl)c(CN2CCC(c3ccc(Br)s3)C2)sc1=O NC1CN(C(=O)C(=O)NCc2ccccc2N)CCC1C(F)(F)F c1(CC)ccc(C=CC(=O)NCC(N2CCN(C(C3CCCC3O)=O)CC2)=O)o1 Cc1ccc(C(N2CCC(C(C)NC(C3CCCS3)=O)C2)=O)c2c1CCCN2 Cc1n[nH]c(C)c1SCC(=O)NCCC(C)CC.c1(C=O)scnc1C1CC1.N C1(NC(Cc2c(C)n[nH]c2)=O)C2CC3C1C3C2C(=O)NC.c1cc(F)ccc1F C=CCCCNC(C1(n2cc(Br)cn2)CC1)=O.C(=O)(CC)N.CCN(C)C C(CN=C(NCC(c1ccc(F)cc1)(F)F)N1CCC(OC)C(C)(C)C1)OCC CC(C)C1=CCC(C(N2CCC3(CC3NC(c3csnn3)=O)C2)=O)CC1 CC1CCCN(C(c2ncncc2Cl)=O)C1CNC(=O)C(C)(C)C1CCC1 C1(C2CCCC2)(C(=O)NC2CCN(C(Cc3nc(C)oc3)=O)CC2)CCNC1=O c1(C(c2nnnn2CC(F)F)NCCCOCC=C)csc(C#N)c1 c1(C(=O)NC2CCC(CNC(C3=C(C)OCC3)=O)C2)cc2n(n1)CC(F)C2 C1(=CC(=O)N(CCCNC(=O)CCCN2CCCCC2)C)CCCCCC1(F)F N1(C(CSCC)=O)CCN(C(c2cc(C(C)C)[nH]n2)=O)CC1CC C1(O)(CC)CCN(C(C2(C)CCN(C(=O)COCC3CCCO3)C2)=O)CC1 C1(C(N2CCCC(NC(C3CN(CC(C)C)C3)=O)C2)=O)(OC)CCCCCC1 C1(NC(=O)C=CC2CCC2)CC(C(=O)NC2COCCC2(F)F)=CC1O CC1(C)CCN(C(=O)C2=CCCOC2)CC1C(=O)Nc1cc(O)cc(F)c1 c1(C2(C(=O)NC(c3cn(C(C)C)nc3)C)CC2)ccccc1Br C1(C(=O)NCCCN(C(C)C)C(c2ccc(CCO)cc2)=O)CCCC(F)C1 Cc1cc(C(=O)NCC2CN(Cc3cccn3C)C2)cc(Cl)c1.c1ccccc1 c1(N2CCC(CCO)C2)nc2c(c(=NCC3(CO)CC3)[nH]1)CCCC2 c1(NC2C(C#N)CN(Cc3cncc(Br)c3)C2)ncc2sccc2n1 C1(NC(c2cc(C)c(F)nc2)=O)CN(C(=O)CSC(C)(C)C)CCC12CCC2 C(=O)(C1=CCC(NC(=O)CSc2nc[nH]n2)C1)N(C(C)C)CC1CC1 CCC(CCCC(=O)OC(C)=O)NCC(C)CC(=O)OC(C)(C)C N1(C(c2c(O)ccc(C)c2)=O)CCN(C(=O)CCc2ccccc2Cl)C2(CC2)C1 c1(C(N(C(C)CCNC(=O)COC2(C)CCCC2)C)=O)ccnc(Cl)c1O N1(C(COC)=O)CCCCC(CCC(=O)NC2CC(O)C2OC)C1 C1(NC(c2n[nH]c(C)c2F)=O)CCCCN(C(C2(C)C=CCCC2)=O)C1 CCCCC(CC(=O)NCCN1CC2CC2C1)NC(=O)CC1CN(C(C)=O)C1 c1(OC)cc(C)c(C)cc1S(=O)(=O)N1CC2CC1C2C(=O)Nc1ncccc1I c1(C(=O)NC2CC(F)(CNC(c3c(C)c[nH]c3)=O)C2)cc2cc(Cl)ccc2s1 c1(C(N2CC(NC(C3=NOC(C)C3C)=O)C2)=O)cnn2ccnc(N)c12 N1(C(CCc2n(C)cnn2)=O)CC2CC1CCC2NC(c1ccc(CO)o1)=O N=c1cc[nH]cc1C(=O)NC1CCC1NC(=O)Cn1cnc(Br)c1 N1(C(c2cn(CC)nn2)=O)CCCC(NC(=O)NC2(C3CCCCO3)CCC2)C1 C12CCCC1CN(C(=O)C)C2.C12(C(=O)OC)CC(C=O)(C1)C2.CC(F)F.N Cc1oc(C(C)C)cc1C(N1CCC(C(C)NC(=O)CC2COCCO2)C1)=O c1(N2CCCC(C(=O)NC3CC4CCC3C4)CC2)nc2cc(Br)ccc2s1 N1(C(c2ncc(F)cn2)=O)CC2CC(C(N3CC4(CC(CO)CO4)C3)=O)CC2C1 C1(C(=O)NCC(CCO)OC)CCC(NC(C2(C)CC(C)=NO2)=O)CC1 N1(C(c2c(C)coc2)=O)CCN(C(=O)CC2CC(n3cnnc3)C2)CC1C(C)C N1(C(c2c(COC)ccs2)=O)CCN(C(=O)CC2CC2)CC1C1CCCC1 CC(C)CC(CNC(=O)C(F)CC1CCCCC1)NC(=O)Cn1nnc(=O)[nH]1 N1(C(=O)Cc2ccccc2)CCC2CCC(C1)N2C(=O)CC1CCCO1 C(=O)(C(Cc1ccccc1)NC(=O)OC)NC(COC)CC1CCCO1 N1(C(CCc2ccc(C)o2)=O)CCC2C(C1)CN2C(c1cc[nH]c2nccc1-2)=O c1(CC)cc(C(=O)NCC2CC(C)N(C(=O)C=Cc3cn[nH]c3)C2)sc1C CC1COC2(CCC2)CN1C(C1(CNC(C2CC3(CC3)C2)=O)CCCO1)=O c1(C(=O)NCCC(=C)CNC(C2(c3cccs3)CCCC2)=O)cncc(N)c1 c1(C(=O)NCC(C)N(C(=O)C#CC(C)C)CC)nc(C)c(C)nc1O CC1OCCNC1C(=O)NC1(C)CCNC1=O C(=O)(CC(C)(C)NC(C1CCC(=O)N1C)=O)NCCC(=O)NCC#C c1(NC(=O)NCCc2ncn(C)c2)ccc(C2(C#N)CCCC2)cc1 c1(C(=O)NCC2(O)CN(C(c3cc[nH]c3)=O)C2)n[nH]c2c(F)cccc12 c1(C(=O)N)cccc(C(F)(F)C(F)(F)F)c1.C=CC1(C(=O)N(C)CC)CCC1 Cc1c(NC(=O)C(Cl)=CCl)ccc(Br)c1F n1(COC)nccc1C(=O)NC(C(=O)NCc1csc(O)n1)C1CCOC1 Cc1ccc2nc(C(=O)NCC(C)N(C)C(c3cc4n(c3)CCCC4)=O)cn2c1 C(=O)(CCCC(c1nnnn1CC1CC1)Nc1cc(Cl)cnc1OC)OCC Cc1ccc(C)c(C(=O)NCC2CCC(C)CC2)c1C.C1(C)(CC=O)CC1F CCC(C(=O)N(C)CCNC(=O)Cc1cn[nH]c1)N(C)C=O.C(C)(C)C.O O=C1CCC(C(N2CCCCC2CNC(C2(C3CCC3)CC2)=O)=O)CN1 Cc1ccc(C(=O)NC2CC3(C2)CC(NC(C2(O)COC2)=O)C3)cc1Br Cc1ccc(C(=O)C(=O)NC2CCCC2NC(=O)C(n2cc(Br)cn2)C)cc1 c1(OC)c(F)cc(F)c(C(N2CCC(N3CCCc4ccccc43)C2)=O)c1Br c1(C(N(C(C)CN(C)C(c2cncc(C3CC3)c2)=O)C)=O)cc2cnccc2[nH]1 C1(OC)CC(O)CN(C(C23CCC(NC(=O)CCCCCN(C)C)(CC2)C3)=O)C1 c1(C(N2CC(NC(C3(C(F)F)CC(=C)C3)=O)C(C)CC2)=O)cc2sccc2n1C c1(CCCC)nc(C(=O)N(C)CCN(C)C(C2(CCOC)CCCC2)=O)cs1 N1(C(C=C(COC)C)=O)CCCN(C(C2CC3(CCC3)CO2)=O)CC1C c1(OC(C)C)cc(C(=O)NC2CN(CC(=O)N(C)C3CC3)CCC2C)ccc1F C1(CC(=O)N(C)C(c2ccc(Cl)cc2)c2cccs2)CC2(CCNCC2)CO1 N1(CC(=O)NC(CC(=O)N(C(CCSC)C)C)(C)C)C(=O)CCCC1=O c1ccccc1-c1ccc(F)cc1.CC(C)(O)C(=O)NC1(CC(=O)NC)CCC1 N1(C(C2N(C)CSC2)=O)CCC2(CC(NC(=O)CC3CCCCO3)C2)C1 N1(C(c2cc(=O)cco2)=O)CC2CCN(Cc3ccc(O)c(Cl)c3)CC2C1 N1(C(C(CNC(C(C=CC)O)=O)O)=O)CCOC2COCC12 c1(C(C(=O)N)(F)F)ccc([N+](=O)[O-])cc1.CC(C(=O)N(C(C)C)C)c1cncs1 c1(NC(=O)CCF)cccc(NC(=O)C=CC=Cc2ccccc2)c1 C1(CNC(c2ncn(C)c2)=O)CCCC(NC(c2cncc(Br)c2)=O)C1 C=C(C)CC(C(=O)NCCCCN1CCC1)NC(=O)C(C)CCCOC C1(OC(c2nn(CC)c(C)c2I)=O)CCC2COCCC2C1 CC(C)(CCC(=O)NCC(F)CNC(C1CC2CC2C1)=O)[N+](=O)[O-] N1(C(C(C)=C(CC)C)=O)CC2OCC(NC(c3ncc(F)cc3F)=O)C2C1 c1(C(N2CCCC(C(=O)NCC(C(C)C)(C)O)C2)=O)c[nH]c2ccncc12 C1(CN(C)C(c2cnccn2)=O)CCCCN1C(C1CC(c2ccccc2)C1)=O N1(C(C2(C)CC(C(F)(F)F)C2)=O)CCCC(C2CN(C(C3CCC3)=O)C2)C1 c1(OC)cnnc(C(N2CCN(CC(=O)N(CC(N)=O)C)CC2)=O)c1 N1(C(c2ccc(CNC(C)=O)o2)=O)CCN(C(=O)CCCCC(=O)O)C(C#N)C1 c1(C2CC2)ccccc1.C=CC1(C=O)CC1.C(=O)(CC)N(CC(C)O)CC.N C1(C(=O)NCC(C)OC)C2CC2CN1C(=O)CN1CC2CC2C1 C#Cc1ccc(Cl)c(C(=O)NCC2(COC)CCCCCC2)n1 c1cn(C)c(C(=O)N(CC(O)CN(C(=O)C(C)CC2CCC2)C)C)cc1=O.C c1(CC(=O)NCC2CC(OC)CN2C(=O)C=CCO)ncnc2sccc12 NC1CC2CCC(C1)N2CC(=O)N(CCCO)Cc1ccccc1 c1(CC)cc(C(=O)NC2CCCC(CNC(c3nc(C)oc3C)=O)C2)sc1C N1(C(c2ccc(C#N)o2)=O)CCC=C(CNC(=O)C(C2CCOCC2)O)C1 N1(C(C2ON=C(C)C2)=O)CC2CCCC1(CNC(c1cccc(C)c1N)=O)C2 CCCCC(F)C(=O)N(CCC(C(C)C)NC(=O)CCCC1CCC1)C c1(C(=O)NC(CC(C)NC(CCOCC)=O)C)ccc(C(F)F)c(Cl)c1 c1(CC)nnc2cc(NCC3(F)CCC3)ncn12.C1(C=O)CC(=O)NC(=O)C1 N1(C(CC(n2c(C)cc(C)n2)C)=O)CCN(C(=O)C(O)C(C)C)CC(C)(F)C1 C1(C(N2CCC3(CC3)C2)=O)C(O)C(=O)N(C)C1C.Cc1cnn(C)c1C(=O)N Cc1ccnc(C(=O)NCC(C)CN(C)C(c2cncnc2)=O)n1 C#Cc1cc(C(=O)NC2COC3(C2)CN(C(=O)CCP(C)(C)=O)C3)cc(F)c1 C1(CCNC(c2n[nH]c(C)c2Cl)=O)CN(C(=O)C=Cc2ccoc2)CC(C)O1 Cc1c(CC(N2CCC(N(C(=O)CCNC(N)=O)C)C2)=O)ncn1C C1(C(=O)NCCC(=C)C)CC12CCN(C(=O)CCCCCSC)CC2 c1(N(C2CCN(C(C(CC)SC)=O)C2)C)ncnc2c(F)c(F)ccc12 NS(=O)(=O)c1cc(C(=O)NC2CCCN(C(=O)CCn3cccn3)C2)c(Cl)s1 C=CCC(C(=O)NCCCN(C(=O)C(C1CCCCC1)F)C)C(C)C c1(C(F)(F)F)cc(C(F)(F)F)ccc1-c1nc(C(c2ccc(Br)nc2Br)(F)F)no1 N1(C(c2ccc(CC)[nH]2)=O)CCN(C(c2[nH]ncc2C#N)=O)C(C(C)C)C1 c1(C(=O)OC(C)(C)C)ncccc1NC(=O)NCCc1ccnc(Br)c1 c1(N2C(CC(=O)Nc3nc(Cl)ccc3C(=O)O)COCC2)ncc2[nH]ccc2n1 Cc1cc(C(=O)NC2CCOC2C(=O)NC2CCCC2C#N)c(C)[nH]1 N1(C(c2c(C)c(C#N)[nH]c2)=O)Cc2[nH]nc(C(=O)N3OC4CCC3C4)c2C1 C1(NC(C(c2cccc(F)c2)(C)C)=O)CCN(C(=O)C=CI)CCC1CO CCC(C)(C)C(O)C(=O)N1CCCC(C(=O)NCc2cc(C)c(C)s2)CC1 C1(NC(c2nc(CCCC)sc2)=O)CN(C(c2ncc(Cl)s2)=O)CC2(CC2)C1 C1(C2CCC2)(C(N(CC(CNC)O)C)=O)CC1(F)F.C1(F)CCS(=O)(=O)C1 Cc1cc(C(C)N(C(=O)CC2CCCOC2)C)no1.C1(CC)CC(F)(F)C1 c1(C(C(=O)NC)NC(c2cc(C)ccc2C)CC)cnc(C)cc1OC C1(CC#N)CN(C(c2cn[nH]c2)=O)CCN1C(=O)Nc1ccc(Cl)cc1Cl C1(C(N2C(CN(C(=O)CCn3ccccc3=O)C)CCC2)=O)CCCC(=O)N1C Nc1cc(F)c(C(=O)NC2CCCCC2NC(C2CC=CCO2)=O)cc1F C1(CC(N2CCCC2C)=O)CCC2(CCC2)O1.c1(OCC)ccc(C(=O)N)cc1 c1(C(N2CCC3(CC(NC(CCC(N)=O)=O)C3)C2)=O)ccnc2ccc(F)nc12 C(N=c1[nH]c(N2CCCC(F)(F)C2)nc2c1CSC2)c1c(C)nn(C)c1 C#CCCCCCC(=O)NC(C)(C)CCN(C(=O)C=CC1CCC1)C Cc1cc(C(F)F)nn1CC(=O)NCC1CN(C(=O)C(C)C#N)CCO1 N1(C(C(COC)O)=O)CCN(C(C2C3CCC(F)(F)C23)=O)CC(C)(C)C1 c1(OCCOC)ccc(C(N2CC(N(C(=O)CCC3CCCO3)C)C2)=O)cn1 N1(C(c2scc(C)c2C)=O)CC2CCC(C1)N2C(=O)C(C)C1CC1 C(=O)(C(O)CCCNC(C1CCCOCC1)=O)N(CCCC(C)O)C Cc1cc(F)cc2[nH]c(C(=O)NCCC)cc12.C1(S(N)(=O)=O)(C(=O)N)CCC1 C#Cc1ccc(CC(N2CC(=O)NCC2C(=O)NCC#CC#CCO)=O)cc1 CC1CN(C(c2csc(C#N)c2)=O)CCC1CNC(=O)C.c1ccc(Cl)cc1.O C1(NC(CCC=C(C)C)=O)COCCN(C(=O)CC(C)N(C)C)C1 Fc1ccc(C(c2nnnn2C)NCc2ncc(-c3ccccc3)o2)c(Br)c1F c1(C(N2CCC(c3ncc[nH]3)C2)=O)cnc(CNC(C2(F)CC=CCC2)=O)nc1 c1(C(c2nnnn2-c2ccccc2)NC2(CC)COC2)sc(C)c(C)c1Br C1(CC)(CO)CCCN(C(C(=O)NCC2CCOC2)C2CC(OC)C2)C1 N1(C(CN2CCCC(NC(=O)OC(C)(C)C)C2)=O)CCn2ncc(Cl)c2C1.C=O c1(OC)ccc(CN2CC(C)(CC(=O)NCC(C)OC)C2)c(OC)n1 N1(C(COC)C)CC(NC(=O)C(c2ccccc2Cl)C)CC2(CCOCC2)C1 c1(C(=O)NC2(C(N3CC(CSC)C3)=O)CCC2)ccc(CO)s1 c1(C(=O)NCC2CCCN(C(c3cc(OC)ncc3)=O)C2)ccc2c(c1)CCO2 C1(C)(CNC(C(COCC)C)=O)CCCN(C(=O)CC2(OC)CC2)C1 CC1CCC(C(=O)NC2(CCCNC(c3ncccc3C3CC3)=O)CC2)CC1 C(=O)(C(C)CC(=O)NC(CCF)C(=O)Nc1ccc(O)c(F)c1)OC N(C(=NCCCF)NCc1ccc(C)c(C2CC2)c1)CC1N(CC)CCC1 CCC(CC(F)(F)F)C(=O)NCC(CNC(c1cccc(C(F)(F)F)c1)=O)CO C1(C(=O)NCC(CN(C(C(C)c2ccsn2)=O)C)C)CC(F)(CO)C1 c12ccccc1CNC(=O)C(O)Cc1nc-2no1.C1(SC)CC(C)(C(N)=O)C1 c1(NC(CC)=O)ccc(O)c(C(N2Cc3cncn3C2)=O)c1 C1(OC)CC2CC1CN(C(=O)C1=CCC(NC(C34CCCN3CCC4)=O)C1)C2 CC1CCN(C(=O)CCNC(=O)CC2CCCC(O)C2)CC1 Cc1c(C(=O)NC2C(C)CCN(C(c3cscc3Cl)=O)C2C)cccc1[N+](=O)[O-] c1(OC)cc(OC)n2[nH]c(=NC(=O)NCCC(C)N(C)C)nc2n1 C1(NC(=O)CCC2CC(NC(=O)CCC3CC3(F)F)C2)CN2CCC1CC2 N1(C(C(C)OC)=O)CC2CN(C(c3ccccc3N3CCCC3=O)=O)CC12 c1(C(N2C(C(CNC(C(CC(C)C)O)=O)(C)C)CCC2)=O)cc2cccnc2[nH]1 CCCC(O)C(=O)N1CCN(C2CCC(NC(c3ccc(=N)[nH]n3)=O)C2)CC1 C(CC(F)(F)C(F)(F)F)NC(N1CCN(Cc2nnc(C)s2)CC1)=O Nc1ccnc2c(C(N3CCC3CNC(=O)COC3CCCC3)=O)cnn12 C=C=CC(C)C(=O)N(CCCCCCNC(=O)C(O)c1ccsc1)C S(=O)(=O)(c1ccc(Br)c(Cl)c1F)NCCC(N1CCC(C)CC1)=O CCC(C)(O)C(=O)N=c1ccn(C2CN(C(c3nn(C)c(C)c3Br)=O)C2)[nH]1 c1(N(C(CCNC(C2C(C)C2)=O)=O)CC2CC2)cncnc1 c1(OC2CN(C(C(CC)NC(N)=O)=O)C2)ccc(F)cc1.C(=O)CC.CC.N C(CCC(C)NC(c1sccc1F)=O)NC(C(C)OC1COC1)=O N1(CCNC(=O)CC2CCC2)CCCN(C(C2CCOC2C(F)(F)F)=O)CC1 C1(CNC(=O)CN2CCCNC2=O)CN(C(=O)CC2OCCO2)C2CCN1C2 N1(C(C2CC(=O)NCC2)=O)CC2(CC(NC(c3ccc(CO)c(F)c3)=O)C2)C1 c1(OC)cc(C)ccc1C(=O)NC(CNc1cc(Cl)ncn1)CC(C)C c1(OC(C)C(=O)NC(C2CCCN2C(c2cnsc2)=O)C)ccc(O)cc1 CCCCC(CCCC)C(=O)NCCn1cc(CNC(=O)C(O)CCSC)nn1 CCC(C)(C(=O)O)N(C(=O)C(=O)NC1CN(C(=O)OC(C)(C)C)C1)C CC1(C)CC(C(=O)N(C2CC2)Cc2cnsn2)c2ccccc2O1 Cc1cc2scc(CC(=O)NC3CCCN(C(C4(C)CCC(=O)C4)=O)C3)c2s1 N1(C(CNC(N)=O)=O)CCC(O)C(NC(=O)CCOCC(F)F)C1 N1(C(CC(C)OC)=O)CCC(CCCCNC(c2ccns2)=O)CC1 N1(C(C(OC)OC)=O)CC=C(C(=O)NC(C)CC2CCOC2)C1 C12(C(N(CC)CC3CCOC3)=O)CC(CN1C(c1nc(Cl)oc1C)=O)C2 c1(CCC(=O)N(CC)CC)cccc2c1OCO2.C(=O)(C(C)Cc1ccco1)N Cc1nc(C(=O)NCC2C(C)CCN2C(c2ccc(Cl)s2)=O)cc(O)n1 C1(C)(CC(=O)N(C2CCNC2=O)C)CCN1C(=O)CCCOC(C)(C)C Cc1ccc2c(N3CCN(C(c4nc(Cl)sc4C)=O)CC3C)ncnc2c1 c1(C(N2CCC(CC)C2)=O)cc(Br)c2c(c1)OCO2.C12(C(=O)N)CC(F)C1C2 c1(C=O)ccc2c(c1)OCC2.C(=O)(CCC1CC1(F)F)N(CCC)C1CC1.N c1(N2CC(C(=O)OC)CC(C)(O)C2)ncnc2c1ncn2C(C)(CO)C1CCC1 c1(C=O)c(Cl)cnn1C.n1(CCOCC)cc(C(=O)NC2CCC2)cn1.C O=S1(=O)CCC(CN2CCCC2c2cn(-c3cnccc3Cl)nn2)C1 C1(NC(CC(CC)C(F)F)=O)CC1C1CCN(C(=O)CSC(C)(C)C)CC1 C1(CNC(COCC=C)=O)C(C)CCN1C(c1cc(C(=O)O)nn1C)=O N1(C(C2(N(C)C)CC2)=O)CCCCC(NC(c2ccc(-n3cncn3)nc2)=O)C1 c1(C(=O)NC(CC(C)NC(c2cncnc2C2CC2)=O)C)cnn2ccccc12 c1(C(=O)NCC(C)(F)F)ccc2c(c1)CN(C(c1cccc(=O)n1O)=O)CC2 C1(C(=O)NC(CC)Cn2cncn2)COC2(C1)CN(C(=O)C(C)(C)CF)C2 c1(OC)ccc(SC2(C(=O)Nc3cccc(COC)c3)CCC2)cc1 NS(=O)(=O)C1CCC(C(=O)NCC2CC(NC(=O)CC3CCC3)C2)CC1 C12(C=O)CCCC1(C(N)=O)C2.CCCCCN(CCC(=O)NC1CC(C)C1)C CCCCC(CC)NC(c1cc(CNC(C2(C#N)CCCO2)=O)ccn1)=O c1(C(=O)NC2CC(F)CN(C(C3CC=CCO3)=O)C2)cc2sc(Cl)cc2s1 c1(OC)cc2c(cc1NNC(=O)Sc1ccc(Br)cc1)CCC2 N1(C(=O)CCCC2CCC2)CCN(C(c2cnc3[nH]cnc3c2)=O)C2COCC12 C1(C(N(CC(C)CNC(=O)Cc2ccnn2C)C)=O)CCn2ncnc2C1 C1(NC(C(N2C(c3cccc(C)n3)CCC2)=O)=O)CC12CCC(F)(F)CC2 O=C1CCC(CNCC(c2nccn2C2CC2)N2CCCC2)CN1 C#CC1CCCCN1C(C1(C2CCCN2C(C2CCN(C)CC2)=O)CC1)=O c1(C(=O)NC(CN(C(C2ON=C(CC)C2)=O)C)C)cc(CO)ccc1Cl C(C1c2ccsc2CCN1C(=O)COC1CC1)NC(CNC(CC)(C)C)=O N1(C(CSc2nc(C)[nH]n2)=O)CCOC(C(N2CCOC3CC23)=O)C1 C1C2CN(C(c3c[nH]nc3C3CC3)=O)CC12.C1(OCC)CC1C(=O)N.C N#Cc1cccc(C(=O)OCCn2cc(CNCCN)nn2)c1.c1c[nH]nc1F c1(C(N2CCC23CN(C(=O)COC2CCCCC2)C3)=O)cc2ccncc2[nH]1 N1(C(C(C)NC(=O)C(C)(C)C)=O)C(C)CC2CC12.C(=O)CCCc1nccs1 c1(C(=O)NC2CC(CCNC(C3CCC(=O)O3)=O)C2)cnc2c(F)cccc2c1 C1(CCCC)CCCN(Cc2ccc(C(F)F)cn2)C1 Cc1nc(CC(C)C)sc1C(=O)NC1CC1NC(=O)CCc1nc(O)n[nH]1 c1(CNC(c2cc(OC)no2)=O)ccccc1.n1(CC=O)c(C)csc1=O.N Cc1cc(C(N2CC3CC3(CNC(c3n[nH]c(C)c3Cl)=O)C2)=O)c(C)cc1Cl CCCC(CNC(C1CC1(F)Cl)=O)C(=O)NCC1C(CO)C1(F)F C1(O)(CNC(CCCOCC)=O)CCCN(C(c2ccnc(O)c2Br)=O)C1 N1(C(c2cccc(C(C)C)n2)=O)CC2CCN(C(c3cnc[nH]3)=O)CC2C1 c1(OC)ccc(C#N)cc1NC(=O)NCCCC(N)=O CC(C)CC(F)(F)C(=O)Nc1cccc(CNC(C2CC2CF)=O)c1 C1(C(C)C)CCN(C(C2CN(C(C)=O)C2)=O)C1.CCCCCN(CCC(=O)N)C Cc1ccc(C=CC(N2CCCC(NC(=O)C=CS(C)=O)C2C)=O)nc1 c1(C(=O)NC2CCCCN(c3snc(C)n3)C2)ccc(F)c2occc12 N1(C(c2c(C)nc(CO)s2)=O)CCCCC(CNC(=O)C(C)(C)CN(C)C)C1 CC1CN(C(C2(F)CC2)=O)CCCN1C(c1csc(C(C)(F)F)n1)=O C(=O)(C(CN=[N+]=[N-])NC(=O)Cn1nnc(C)n1)NCC1CC(CC)C1 c1(C(=O)NC(CCN(C(c2c(OC)nsc2)=O)C)C)c(C)cc(C)nc1C C1(COC)CCN(C(=O)Cn2nc(C)nc2C)C1.n1(CC=O)cccnc1=O.N c1(C(=O)NCC(C2CC2)NC(C(C)CF)=O)cccc(Cl)c1O C1(C(=O)NCC2C3CC2N(C(=O)CO)C3)(OC)CCOCC1.C1CCCOC1 CCC(CC)C(=O)N1CC(O)CC1CNC(C12CCC(C1)C2)=O c1(C(N(CCCOCCN(C(C(C)SCC)=O)C)C)=O)ncncc1C#N CN=c1[nH]cc(C(=O)N(CCCCNC(c2ccc(-c3cnn(C)c3)o2)=O)C)o1 Cc1n[nH]c(C)c1NC(=O)CN1CCC(C2(C)OCCO2)CC1 CS(=O)(=O)CCC(=O)NCC1CN(C(c2cc(C3CC3)ccc2Cl)=O)CCO1 c1(C(=O)OCC(c2ccc(C)cc2)=O)onc(C)c1C#N c1(C(=O)NCC(CNC(c2n(CC#C)ccc2)=O)O)c(CCC)nsc1N C1(C(=O)NCC(CNC(c2ccn(CCCC)n2)=O)O)CC2C=CC1CC2 c1(C(N(C(C)C(=O)NC2CC3CCCC3C2)CCC)=O)cnn(C)c(=O)c1 C1(C(=O)NC(C(=O)OC2CC2)c2ccsc2)CC12CCNCC2 C(CCCC(=O)NCC1(C(=O)N(C2CCOCC2)CCO)CCCO1)SC c1(C(N2CC(NC(CCC=C(C)C)=O)(CO)C2)=O)ccc(C2(C)CCO2)cc1 c1(OC)ncc(C2CC2)cc1CN1CCC(O)C(C(N2CCC(N(C)C)C2)=O)C1 O=C(C1=CCCN(C(=O)Cn2ccnn2)C1)NC1CC(CF)C1 c1(C2N(C(c3cc(CC)c(CC)o3)=O)CCC2)cc(F)cc(F)c1 c1(OCCC(=O)N(CC(C)NC(=O)Cc2ccccc2F)C)ccc(Cl)cc1Cl N1(Cc2cnc(OC)c(Br)c2)CCc2sc(C(=O)Nc3cnccc3C)cc2C1 c1(C(N2CC(C)C(NC(=O)CNC=O)CC2)=O)cc(F)c(Br)cc1N c1(C(=O)NCC2(n3cccn3)CCOCC2)cc2c(F)cccc2[nH]1 C12(C(=O)N)CC(C)(CCO1)C2.C1(C(N(C2CCC2)C)=O)C(C)(C)C1(F)F c1(OC)cccc(C(N2CC(NC(c3ccccc3F)=O)CCC2C)=O)c1OC CCC(C)C(C(=O)N1CC(O)(CNC(=O)CCC2CCOC2)C1)NC(N)=O C1(C(=O)NC2(C)CCSC2)CCOCCN1C(C1CC1OC(C)=O)=O c1(C(=O)NC(CNC(COc2ccc(OC)cc2)=O)(C)CC)ccc(Cl)cc1N C(=O)(CCCCNC(=O)CCC(C)=O)N1CCC(CSC)C1 C=CC(CCC)CC(=O)NC(CC(=O)NC(c1cccnc1)C)C1CC1 CC1OCCC1CN(C)C(C1CCN1C(C12CSCC1C2)=O)=O c1(C(=O)NC(CC)CN(C(=O)Cc2cn[nH]c2)CC)cc(-c2ccccn2)ns1 N1(C(CC2CC(C)C2)=O)CC(O)CCC1C(=O)NCCCC1CCCC1 N1(Cc2nc(C)oc2)CCCC(C(=O)NCCN(C)C)C1 C1(C)(CC)CCCC(NCCc2ccc(C)c(OC)c2)C1 CC1(C)C2CCC(C2)C1C(=O)NC1C=CCN(C(c2cnc3ccccn23)=O)C1 c1(OC)cc(CN2CC3(CC(C(=O)Nc4ncc(F)cc4Cl)C3)C2)ccc1C#N N1(C(COc2ccc(OC)c(C)c2)=O)CC(CO)C2(C1)CN(C(=O)CCSC)C2 C1(NC(=O)C=Cc2ccc[nH]2)CN(C(=O)CS)CCC1C(F)(F)F.C1CC1 c1(C(N2C(CN(C)C(C3CC4C=CC3C4)=O)COCC2)=O)cc(O)cc(O)n1 CCC(C)CCCC(=O)N1CC2CCC(C(=O)N(C)CC3(O)CCC3)(C2)C1 c1(CN(C)C(c2occc2Cl)=O)cccc(CNC(C2CC2(Cl)Cl)=O)c1 CCC(CC(=O)N1CC(C)(c2cn(CC(F)(F)CO)nn2)C1)c1ccc(C)cc1 N1(C(C2(O)C(C)(C)C2)=O)CC2(CCN(C(c3cnc4c(c3)CCOC4)=O)CC2)C1 C12(NC(COCP(C)(C)=O)=O)CCC1CN(C(=O)CCS(N)(=O)=O)C2 C1(C(N(C2CC(C)OCC2)C)=O)CC2CCC1N2C(=O)CC1CCC(C)CO1 c1(CCC(=O)NCCCCNC(C2C(=C)C2)=O)ccccc1Br C1(CNC(c2cc(Cl)ns2)=O)(NC(c2n[nH]c(C3CC3)n2)=O)CCOC1 N1(C(C2N(N=O)CCC2)=O)CCC2(C1)CN(C(C1CCC(=O)O1)=O)C2 c1(CC(N2CC(CC(C)(C)C)C2)=O)ccc(C(N)=O)nc1.CC=O.C#CC.S N1(N(C(N2CCC(C)C2c2ccccc2)=O)C)CCCS(=O)(=O)CC1 C1(C(=O)NC(C(=O)NCCC(CC)CO)C(C)C)CC2CCCC2C1 c1(CC)ccc2c(c1)CCCN2C(c1cc(C(C)(C)C)ccc1C)=O c1(CNC(c2ccc3c(c2)NCCO3)=O)cccc2cc(C(=O)N=c3cco[nH]3)[nH]c12 C1(NC(CCSCCC)=O)CN(C(=O)COc2cc(C)ccc2Cl)C2CCCC12 N1(C(C(C)CNC(=O)Cc2cncn2C)=O)CC2(CCC2O)C1 Cc1c(C(=O)C(N2CC3CCC2C(NC(=O)C2CC2)C3)=O)sc2ccccc12 N1(C(C(C)NC(=O)NC)=O)CCN(C(=O)CC2C=CCCC2)CC1C(C)C Cc1cc(C(=O)N(CC(=O)NC2CCCC2)C2CC2)cc(C(F)F)c1 C1(C(N2CCCC(CNC(C3(C)C=CCCC3)=O)CC2)=O)CCn2ncnc2C1 C(C)(C(=O)N1CC(OCC(=O)NC2(CC(=O)OC)CC2)C1)SCC O=S(=O)(c1ccc(=NCc2ccncc2F)[nH]c1)NCC12CCCCC1C2 C1(CN=C(NCc2nc(COC)[nH]n2)NCc2cccs2)CCCCC1C1CC1 C(CC(=O)N1CCC2(NC(c3ccc(=O)n(C)n3)=O)CCCC12)(C(F)(F)F)OC N1(C(C2N(CC)CCC2)=O)CCN(C(c2cccc(C3CC3)n2)=O)CC(C)(F)C1 C1(C(=O)NCC2(CC)CCCO2)CC=CCC1.C(c1cocn1)=CC(=O)N Fc1cc(C2CCN(C3C=CCCCC3)C2)cc(Cl)c1 N1(C(c2c(OC)noc2C)=O)CCCN(C(C2CSCCS2)=O)CC1 Cc1ccc(F)c(C(C)(C)CNc2cc(NCC3C(C)C3(F)F)ncn2)c1 c1(C(=O)NC(COC)(C)C)c(F)ccc2c1CN(C(=O)OC(C)(C)C)CC2 C1(OC)(Cn2nnnc2N2CCOC(C)(C3CC3)C2)CCCC(C)(C)CC1 c1(C(=O)O)ncccc1-c1cn(CCC2CN(C(C3CCC(F)(F)C3)=O)C2)nn1 c1(OC)ccccc1NC(=O)C(CCN(C)C)NC(=O)CCNC(N)=O N1(C(C(C)=C2CC2)=O)CCN(C(c2ccc(-n3cnnn3)cc2Cl)=O)CC1CO C(CCC(=O)NC1(CC(=O)NCC2C3CCCC23)CCC1)=C(C)C CC1=C(C)CC(C(=O)NC2CCCC2CNC(=O)C2=C(Cl)CC2)CC1 Cc1onc(O)c1C(=O)NCC1CCC(O)C1.c1(C=O)ccccc1C1CC1 c1(C(=O)N)c(F)ccc(Cl)c1F.Cc1c(C(=O)NC2CCC(C)(C)C2)cnn1C N1(C(c2c(C)cn(C)c2)=O)Cc2[nH]nc(C(=O)NCC3CC(O)C3(C)C)c2C1 CCC(C)CCCCC(=O)N1CCCCC1CNC(c1ccc(F)c(CS)n1)=O c1(C(C(=O)NC(C)(C)CC)N(CCCN(CC)CC)C)cc(OC)ccc1F c1(NC(=O)OC)ccc(O)c(C=O)c1.C1(C(N2CCC2)=O)CCN(C)C1C.N C1(C(N2C(C=O)CC(F)C2)=O)CC2(C1)CC2(F)F.C(=O)CCC1CC1.CN c1(C(=O)NCC(C2CCOC2)NC(C(C)(C)n2cnnn2)=O)snc(O)c1Cl C(CCCCO)N(C(=O)CCC1CCCN1C(c1cccnc1)=O)C C1(CNC(c2cc(C(F)F)no2)=O)CCCC1NC(c1scnc1Cl)=O c1(C(N2C(C)(C(=O)Nc3c(O)ncc(C)c3)CC2)=O)cc2ccccc2cn1 C1(=O)C(CCC2CC2)NC(=O)OC2(C)CN1C2.C(C)(C)C.C(C)OC c1(C(N2CC(Cn3cc(C4CCCC(F)(F)C4)nn3)C2)=O)cncc2c1CCCC2 C1(NC(C=C(COC)C)=O)CN(C(c2c(F)cc(C)cc2F)=O)CCC12CCC2 C1(C(N2C(C(=O)NC(C)C(C)n3cccn3)CSC2)=O)CCCC(O)C1 C1(CNC(=O)C=CC=C(Cl)Cl)CC2(CC2)CN1C(C1CCCSC1)=O C1(CNC(c2ccc[n+]([O-])c2)=O)CCN(C(=O)CCc2cccc(O)c2)C12CC2 CC1(C(=O)NCC2(O)CC(C)C2)CCCCC1.c1(C(=O)N)cc(C#N)no1 C(=O)(C1CCCc2cncn21)N1C(C(C)NC(c2ccccc2)=O)CCCC1 c1(C(=O)NC(C2CCCN(C(C(c3ccccc3)C)=O)C2)C)cc(O)nc(O)c1 N1(C(c2ccnc(CO)c2)=O)CCN(C(c2ns[nH]c2=O)=O)C2(CCC2)C1 C1(C(=O)NC(C(C)(C)OCC)c2c[nH]nn2)C2CCC1(c1cncs1)C2.C Cc1ccc(CCC(=O)NC2CC2C(=O)N(C)C)cc1.C(C)(C)C.C(=O)N c1(C(=O)NCC(CO)NC(CCCCCCC)=O)ccc2c(c1)CCCC(=O)N2 N1(C(CCC(=O)c2cn(C)nc2)=O)CCCC(NC(=O)COc2ccon2)CC1 N1(C(C2N(CCCC)CCCC2)=O)CCC(CO)C(NC(=O)CCC(C)(F)F)C1 c1(C(=O)NC2CCC(NC(C(C)Cc3cnc[nH]3)=O)CC2)cc2n(n1)CCO2 N1(S(=O)(=O)c2cccc(OC(F)F)c2)CCC2(CC3CCC2C3)C1 c1(C(N2CC(C)C(CNC(=O)CCCC(C)(C)C)C2)=O)ccc(F)c2[nH]ccc12 c1(C(C(=O)NCC(C)C)N(C)CC2CC2C)cccc(I)c1 c1(C(N2CC(Nc3ccnc(C)n3)C(C)C2)=O)cc(F)c(Cl)cc1F N1(CCC(N)=O)CC(N=c2cc[nH]cc2S(=O)(=O)NCC(=O)NC2CCCC2)C1 c1(CNC(c2cc(C)[nH]n2)=O)cccc(CNC(c2snc(O)c2Cl)=O)c1 N(C1CCCNc2ccccc21)C(C1(c2cccc(F)c2Br)CC1)=O C1(CCOC)CC1N=c1[nH]c(N2CCn3ncc(C)c3C2)nc2c1CCCC2 CN1CCC2CN(C(C3(CNC(c4cc(C#N)n(C)n4)=O)CC3)=O)CCC12 c1(C(N(CC(O)CN(C)C(C2(C#N)CC3CC3C2)=O)C)=O)cccc2sncc12 c1(OC)cn(C)c(C(=O)NCC(C)(C(C)C)NC(=O)CC(C)CF)cc1=O c1(C(=O)NCCCN(C)CCO)cc(C(F)(F)F)nc(C(F)(F)F)c1 Cc1nc(C(=O)NC2CN(C(=O)C=Cc3cccs3)CC2O)sc1C c1(C(=O)NCC2(C)CC(NC(=O)CC3(C)CCCO3)C2)cccc2nc[nH]c12 N1(C(c2scc(-c3ccc(NC(C)=O)cc3)n2)=O)CCC2(COC2)C1.C1C(=O)N1 O(NC(=O)C(F)(CNC(C12CC(C)(CCO1)C2)=O)C(C)C)CCCOC c1(CC(=O)NCC(C2CCOC2)NC(CN(C(C)C)C)=O)ccc(O)cc1 CC1CN(C(=O)CC2=CCCC2)CC1(C)CNC(=O)C(C)(C)CN(C)C c1(COC)csc(NC(c2cnn(C3CC3(F)F)c2)=O)c1 c1(C(=O)NCCCC(C)NC(C2COC3(CO)CC2C3)=O)cc[nH]c2nccc1-2 Brc1cc2c(N3CCC4(C3)CN(c3ncnc5c(Br)c[nH]c35)C4)[nH]cnc-2n1 c1(C(=O)NCCC(C)N(C(c2cc(C)[nH]n2)=O)C)cc(C#N)c[nH]1 N1(C(CCCC(=C)C)=O)CC2(CCN(C(c3n[nH]c(C4CC4)c3Br)=O)CC2)C1 N1(C(C2N(C(C(C)NC(=O)NC)=O)CC(=O)NC2)=O)CCC2(CC=CCO2)C1 C(CCC(=O)N1CCC1(C)CC(=O)N(C)CC1CCCN1C)OCC Cc1nn(C)cc1C(=O)NCC(CO)NC(=O)C(N1CCSCC1)C n1(CC=O)cccc(C)c1=O.C(CCCNC(=O)CC1CC(OC)C1)OC.N C(=O)(C(C)NC(=O)C(C1CCCC1)NC(=O)C(C)NC(=O)O)NC C(=O)(C#CC1CCCCC1)NC1CCC(NC(c2c(Br)ccc(N)c2)=O)CC1 C1(C(=O)NOCCF)(CC)CN(C(c2cc(C)cs2)=O)C1 C(C1SCCc2ccccc21)N(CC1(C#N)CCCC1)CCOCc1ccccc1 N1(C(CCOC)=O)CCC2CCC(NC(=O)C(F)(F)c3csc(C)c3)C1C2 CC(C#N)CCC(=O)N1CCC(C)(NC(=O)CCCCN2CCOCC2)C1 N1(C(C2CCC(n3cc(CCN(C)C)nn3)CC2)=O)CCC2CC2(O)C1 CCCCCC(O)CC(=O)NC1CN(C(=O)Cc2ccc(Cl)s2)C2CCCCC12 C12(CNC(CCOCC(C)C)=O)CCCC1N(C(C1CC1C(C)C)=O)CC2 N1(C(C23C(CN(C(c4c(C)n(C)nc4)=O)C2)COC3)=O)CCc2c(nnn2C)C1 CN1CCN(C(c2ccc(CN3CCOCC3)o2)=O)C2CCC12 C(CC)(CCCCC)(c1n(CC(=C)C)nnn1)NCc1cnc(Cl)c(C)c1 C1(NC(c2c(C)cncc2)=O)CN(Cc2ccc(F)c(Br)c2)CCC1C C(C(C)CC(F)(F)F)NC(C(CC=CC)NC(=O)CCc1nncs1)=O C(=O)(CC1=CCCCC1)NCCC(CNC(CC(C(=C)C)OCC)=O)O c1(NC2CCCN(C(C)C(N3CCN(C)CC3)=O)C2)ncccc1Cl C#CCCCCCCC(=O)NC(CCSC)C(N1CCN(C2CC2)C(C)C1)=O C1(CNCC=CCC(=O)OC)CCC2(CCC2)O1 Cc1cnc(N(CCCC(C)(F)F)C)c(S(=O)(=O)N(CC(C)N(C)C)CCO)c1 N1(C(CCc2cc(C(C)=O)c(C)o2)=O)CCC2C(CCN2C(C2CC2(F)F)=O)C1 c1(NC(N2CCCC3(C(=O)OC)C(C2)C3)=O)cc2c(cn1)CCCC2 CCC(CC(=O)NC1CCC1NC(c1cc(OC)n(C)n1)=O)C(C)(C)C CCC(CC(C)C)C(=O)N1CC2CN(C(=O)CN3CCCCC3=O)CCC12 C12(NC(C3C(c4cccc(C)c4)C3)=O)CCOC(C)(C1)C2.C(=O)(CCC#N)N CCCCCC(C)(CC)C(=O)N1CCCOC(CNC(c2ccc(OC)s2)=O)C1 c1(C(=O)NC(CNC(C2C(OCC)C2C)=O)(C)C2CC2)nc(C)nn1C N1(C(C2CC(C)(O)C2)=O)CCN(C(c2c[nH]c(-c3ccccc3)c2)=O)C2CC12 c1(OC)cccc(CC(=O)NC2CC(CCNC(c3cc(F)c[nH]3)=O)C2)c1 c1(NC(c2ccc(F)c(F)c2Cl)c2n(C)nnn2)cc(Cl)c(F)c(Cl)c1 c1(CNC(CCC=C)(c2nnnn2C2(C)CC2)C2CC2)cnn2c1CCCC2 n1(CC)cnc2c(NCc3ccc(C)cc3F)[nH]c(=NCc3sccc3Br)nc12 c1(N(C)C(=O)N(Cc2ccccn2)Cc2cscn2)ccc(Br)cn1 C1(CC=C)(NC(=O)CCc2nccs2)CCCN(C(=O)C2=CCCCO2)C1 N1(C(=O)Nc2ccc(OCCC(N)=O)cc2)CC2(CCCC2)c2ccc(Br)cc21 c1(C(=O)NC2(C(=O)NCCCC#C)CCN(C)C2)cccc(C)c1C N1(C(CC2CCCC(=O)N2)=O)CC2(C1)C(NC(c1ccc(Cl)[nH]1)=O)CCS2(=O)=O CN1C2CCC1CC(=CC(N1CC3C(NC(C4CC4(F)F)=O)C3C1)=O)C2 c1(C(=O)NCC2CN(C(CNC(CCC)=O)=O)C(C)C2)cc(C)c(O)c(N)c1 C1CCCN(C(c2cnn3c2OCC3)=O)C1C.C(COC(C)C)(C=O)NC(C)=O C1(O)(CCNC(=O)CCc2cccnc2)CCN(C(c2n[nH]cc2Br)=O)C1 c1(C(=O)NC2CC(NC(=O)C=Cc3ccoc3)C23CCC3)c(F)cc(F)cc1F CC(C)C(C(=O)OCc1ccccc1)NCc1ccn(C2CCCCC2)n1 Cc1cc(C(=O)NCC2CN(CCCc3ccccc3C)CCO2)nn1C c12ccc(cc1)NC(=O)C2(C)C.N1(C(CCC)=O)CCCC1C(=O)NCC.O C=CCC(CC(C)C)C(=O)NCCCN1CCN(C(C2CSCCS2)=O)CC1 N1(C(C(c2ccn(C)c2)C)=O)CC(C)(C)CC1CNC(C1CCSC1)=O Cc1nc(C)c(F)c(=NCC2CN(C(c3cn(C)c(=O)n3C)=O)CCC2C)[nH]1 C(=O)(C(O)C(C)(C)CC)NC1CN(C(c2cc(CC)cc(F)c2)=O)CC1C c1(OC)ccc(C)c(C(=O)NC23CCN(C(C4(F)CCC4)=O)CC2C3)n1 CC1CN(C(c2ccc(CNC(c3cc(C#N)cs3)=O)cc2)=O)C(C)CO1 C1(CC)CCC(C)CN1C(=O)CC1CC(C)N(C(c2c[nH]nc2C)=O)C1 C1(C)(CNC(C(CC)N(C)C)=O)CCCN(C(C2(O)CCCCCC2)=O)C1 c1(-n2cc(C(N(CC(C)N(C)C(c3ccon3)=O)C)=O)nn2)ccc(F)cc1 C1(C2(O)CCOC2)(CNC(CCCC=C)c2ccccc2)CCC1 C1(CNC(c2c(C)cno2)=O)CC(C)CCN1C(c1cccc(CO)c1C)=O C1(CC)(NC(=O)Cn2ncnn2)CCCN(C(=O)Cc2cn[nH]c2)C1 c1(C(=O)NCC(C)NC(c2cnc(SC)n2C)=O)ccc([N+](=O)[O-])cc1Cl C(=O)(C1=NOC2(CCN(S(=O)(=O)CC#N)C2)C1)Nc1c(C(=O)OC)c(C)sc1 c1(COC)nc(NCC(C)C(F)(F)F)cc(N(C)CC2CCCOC2)n1 O=C1CC(CC(=O)NCC#CCNC(c2cnc(C(F)F)s2)=O)CCCN1 C1(NC(c2cn(CCC)nc2)=O)CN(C(c2coc(C)n2)=O)CC1n1ccnn1 C1(NC(C=C(C)C(C)(C)C)=O)CC(F)(F)CC1.C(=O)C(C)S(N)(=O)=O.N CCCCCCCCCC(=O)N1CC2(NC(C3CC(C)=NO3)=O)CCCC2(F)C1 c1(C(N2C(C)(CC(=O)N(C3C(C)CCC3)C)CC2)=O)coc2c1COC2 C1(C(N(CCCCNC(C=Cc2ccc(C)nc2)=O)C)=O)CCC2CCCCN12 N1(C(C2(NC(=O)OC(C)(C)C)CCOCC2)=O)CCC(C2CCCCC2)C1 c1(C(N)=O)ccc(NC(c2cccc(C)c2)=O)cc1F.C12(C(=O)N)CSCC1C2 C1(NC(C2(F)CCN(C(COCCCCCC)=O)C2)=O)Cc2cscc2C1 N(C1CCCn2nccc21)C(C(C)CNC(=O)CNC(=O)C1CC1)=O c1(C(=O)NCCC2(NC(CN(C(C)C)C)=O)CCC2)cncc(C#N)c1 c1(CC(=O)NCC2(F)CCN(C(C3(CO)COC3)=O)C2)cccc(Cl)c1 Cc1ccc(C(=O)NCCC(C)NC(c2cnc(Br)s2)=O)n1C O=C(C(F)C(F)(F)F)NC1CCC(NC(c2cccc(OC(F)F)n2)=O)CC1 C1(CNC(C(C)O)=O)CCC2(CCN(C(c3ccc(C#N)cc3F)=O)CC2)CO1 C1(C(=O)NC(c2nccc(C(F)(F)F)n2)C)C2CN(CCc3ccccc3)CC12 C1(C(=O)N)CN(S(=O)(=O)N(C)C)C1.Cc1cccc(C(N2CCC(C)C2)=O)c1N Cc1cc(=NCCN2CCC2)[nH]c(=NCCC2CCN(c3ccccc3)CC2)[nH]1 C(N=c1[nH]c2c(c(=NC3CC(O)C3)[nH]1)COCC2)c1ccc(S(C)(=O)=O)cn1 N1(C(=O)Cc2cccs2)CCCC2(CCCN2C(=O)C(O)CN2CCOCC2)C1 C1CN(C)CCN1C(=O)CC.n1(CCOC)cc(C(=O)NC)cn1.C(C)=O C1(NC(CC=C)=O)CCCCC12CCN(C(c1scnc1C)=O)C2 c1(OC)cccnc1C(=O)NC1(CO)CCN(C(=O)C=C(C)c2cccs2)C1 c1(C(=O)NC23CC(NC(C4C(C)(CC)C4)=O)(C2)C3)ccn2nccc2c1 C=CC(CCC)CC(=O)NCC1(CNC(c2ncoc2C2CC2)=O)CCCC1 Cc1nc(NC2CCN(C(=O)CCCC3CCCCC3)CC2)c2c(C)csc2n1 N1(C(CCCOC(C)=O)=O)CCCC(NC(c2cc(-n3ccnc3)ccn2)=O)C1 N1(C(C2C(C(C)O)C2)=O)CCCCC1CCNC(=O)C=C(Cl)Cl C(CC(C(=O)NCCN(CC(F)F)C)NC(C1C=CCC1)=O)OCC c1(COC(C)C(=O)NC2CCC(NC(=O)C=CBr)CC2)ccc(F)cc1 c1(C(=O)NCCCN(C(=O)Cc2cccc(O)n2)CC)cc(C)n(C)c1C N#Cc1ccc(=NNC(=O)C(Cc2ccccc2)C2CCCC2)[nH]c1 C1(C2CC2)(OC(=O)CNS(=O)(=O)c2cccs2)CCOC1 CCC(C#N)C(=O)NCC1CCN(C(c2cn(C)nc2-c2ccc(Cl)cc2)=O)C1 c1ccnn1C(C)C.C(C)(C(=O)NCC1CCC1C(=O)N)OCC=C c1(C(=O)NC2CCCN(C(c3scc(C)c3C)=O)C2C)ccc2c(n1)CCCC2 CCC(C(O)C(C)C)NC(N1CCN(c2ncccn2)CC1)=O C1(CC)CCN(C(c2cccc(O)c2)=O)C1C(=O)N(C)Cc1nncs1 C1(C(C)(C)C)CCN(C(C2(N(C)C)CC2)=O)C1.C(=O)CC.CC(F)(F)F.C Cc1ccc2c(c1)C(C(=O)N(C)CC1CCN(C(=O)C=Cc3cccn3C)C1)C2 C(CCCCC(=O)NC1CC(=O)N(O)C1)N(C(C(C)(C)OC(C)=O)=O)C C(=O)(C1CCCc2ncccc21)N1CCCN(C(=O)CN2CC3CCC2C3)CC1 CCC(CC(=O)NC1CCC(NC(C2C3CCC4C(C3)CC24)=O)CC1)C(F)F CC1(CCNC(=O)CCc2cccnc2Cl)CCN(C(C2CCC(F)(F)C2)=O)C1 Cc1nc(CC(=O)N(C)CC2CN(C(C3OCCOC3C)=O)CCO2)c(C)s1 C1(OC)CCC2(C(=O)N(C)CC3CC3)CC12.C12(C=O)CC(F)(C1)C2.C c1(C(N2CC(F)(CNC(C3C(C=C)OCC3)=O)C2)=O)n[nH]c(C)c1[N+](=O)[O-] c1(C(=O)NC2CCC(NC(c3ccnc(C)c3O)=O)CC2)c2c(nn1C)CCC2 c1(SC)cc(C)ccc1C(=O)NCC(C)(C)CC.C1(C(=O)N)CC=C(C)CC1 c1(NC(c2nnnn2CCCSC)(COCC)C)cnc2ccc(Br)cn12 n1(CC(=O)NC2CC(C)N(C(=O)CS(C)(=O)=O)C2)c(O)nc2ccccc2c1=O n1(CC)nc(C)c(C(=O)N(CCC)C)c1Cl.C(=O)(CC)N(CC)C.C(C)C.O N1(C(c2c(C(C)=O)cccc2)=O)CC2(CC(NC(c3sccc3Cl)=O)CO2)C1 Cc1[nH]nc2c(-c3nc4c(s3)CCN(C(c3cc(CO)ccn3)=O)C4)cccc12 Cc1ccc(C=CC(N2CC(OCC)C2)=O)o1.c1(C=O)ccn(CCO)c1C.N C1(C(=O)NC(C2CN(c3ccnc(C)n3)C2)C)CCc2cncn2C1 C1(CC)(NC(=O)C(CC(F)F)C2CCC2)CCCN(C(=O)Cc2ccn(C)n2)C1 C1(CC(=O)N(C(CCNC(C2(CC(C)C)CC2)=O)C)C)C(C)C1(F)F c1(C(=O)Nc2ccc(OC)nc2OC)cnc2occc2c1 c1(-c2cc(C(=O)Nc3ncc(F)cc3Br)n[nH]2)ccn2cnnc2c1 c1(C(=O)NC(CC(C)NC(C(C#C)(C)C)=O)C)ccc(C)c(Cl)c1 N1(C(C(N2CC(C)OC(C)C2)=O)C)CCOC2CC(N(C)C)CCC12 C1(C(N2CC(CC=C)(C(=O)NC(C)CC(C)C)C2)=O)CC(=O)NC1(C)C N1(C(C(C)OCC=C)=O)CC(NC(=O)CCCCCC)CC(F)C1 C1(NC(C2C(CN(C)C)C2)=O)CC2C1CCN2C(=O)CN1CCOCC1 C1(NC(c2n(CC=C)nnn2)COCc2ccccc2)CC(C)(C)OC1=O C1(=O)C(CO)N1C.C1(C(C)OCC)CCOC1.C(=O)C.CC(C)C.C(N)=O C(=O)(C1=C2CCCN=C2NN1)N(CCN(C(CCOC(CC(C)C)C)=O)C)C N1(C(CNC(C)=O)=O)CCN(C(=O)CCc2cncn2C)C2CCC12 Cn1ncc2c(NCCC3CCCCC3O)[nH]c(=NCCNC(=O)N(C)C)nc12 CCC(CC(=O)N1CCC(C)(C)C(CNC(c2ccsn2)=O)C1)CC(F)(F)F C1(O)(CCNC(CN(C(C)=O)C)=O)CCN(C(=O)CC2CCCC2O)C1 c1(CNC(CSC(C)C)=O)cc(C(=O)NCC(C)O)on1 CCC(CC)CC(=O)NC1CCN(C(=O)Cn2ccc(Br)cc2=O)CC1 C(=O)(C(O)C(F)(F)F)NCCCN(C(=O)COCc1cccnc1)C C1(NC(c2cccc(N(C)C)c2)=O)CCN(C(=O)CC2CC2(C)C)C1(C)C C12(C(N(CCC)CCO)=O)CC(CO1)N(C(=O)Cc1nonc1C)C2 c1(C(=O)NCC2C3CN(C(CCOCC)=O)CC32)c(C)cc[nH]c1=N c1(CCC(N2CC(NC(c3c(C)cc(CC)o3)=O)C3C2C3)=O)ccccc1C#N N1(C(C2CCCN(C)C2)=O)CCCCC12CCCN(C(=O)C1CC1)C2 CC1(C)CCCCC1CC(=O)NCC1(C)CC12CCC2.c1(C=O)cnc(O)o1 c1(C(=O)NC(CC)(C)CCNC(=O)C(=CC2CCCC2)C)cc[nH]c2nccc1-2 Cc1cc(=O)c(C(=O)NCCC(C)N(C(=O)CCc2nnc(S)n2C)C)cn1C c1(C=O)cccc(C(N)=O)n1.C1(NC(C2(COC)COC2)=O)CCCC1.N C(=O)(C1=CCCC1C)N1CCC(CC)C1C(=O)NCCOCC(C)(C)O Cc1scc(C(=O)NC2CCOC(C(=O)N(C)CCN3CCCC3)C2)c1C C(=O)(C1CCc2nnc(C)n21)N1CC(CC(=O)OC(CCCCC(=O)NC)=O)C1 C=CC(F)(F)C(=O)N(C)CCOCCCN(C)C(C1(C)CC2CC2C1)=O c1(NC(c2c(OC)cc(C(F)(F)F)cc2)=O)cc(-c2ccoc2)c2[nH]ccc2c1 N1(C(CCC2CCC(=O)N2)=O)CCc2nc(SCC(F)(F)F)sc2C1 CCCC(C(=O)NC(C)C(F)(F)F)NC(=O)CN(CC(C)(C)C)C N1(C(C2(N3CCCC3C)CC2)=O)CCCCC1.C1(NC(C)=O)CCCN1C(=O)N C1(NC(N2CCC2C2CCC2)=O)CCCCC1O O=C1Cc2cc(C(N3CCCC3C(N3CC(O)CC3CO)=O)=O)ccc2N1 c1(NCc2c(C)nccn2)ccc(S(=O)(=O)N(C)Cc2ccns2)cc1Br N1(C(CC(C)F)=O)CCC(C2CCN(C(=O)CSCc3ccncc3)C2)CC1 N1(C(c2c(C)n(CCO)nc2)=O)CCN(C)C(C)C1.C1(C=O)CC(=C2CC2)C1 Cc1ccc(SCCNC(=O)NCc2cncc(Cl)c2)cc1 N1(C(C(CC(F)F)N(C(Cc2cc(C)[nH]n2)=O)C)=O)CCn2c(O)nnc2C1 c1(C(N2CCC2)=O)cc(F)cc(Cl)c1.S(=O)(=O)(C(F)F)N1CCC1.O=C.N c1(NC(C2CCN(C(c3cc(C)c(Br)cc3F)=O)C2)=O)ccc2nc(Cl)sc2c1 c1(NC(CCN(CC#C)C(c2cnc(OC)s2)=O)=O)cccnc1 CC1CCC(C)N(C(=O)C=CC2CCC2)C1.c1(C(=O)N)cc(C2CC2)nnc1O C1(NC(CC(CNC(C(C)OCCCC)=O)OC)=O)CCCCC12CC2 c1(C(=O)NCC(n2cccn2)C)ccc(=O)n(C2CC2)c1.C1(C=O)CCC1.C c1(C(=O)NC(CC(C)NC(c2c(COC)nn[nH]2)=O)C)ccc(O)cc1Cl C(=O)(C(C(C)NC(c1cc(Cl)cn1C)=O)C(C)C)NC(C(CC)C)CN(C)C N1(C(=O)CCOC2CCC2)CC2CCC1CN2C(=O)CC1(c2ccon2)CCC1 CCCCC(=O)NCC12CC(NC(C3CCC(C)C3)=O)(C1)C2 N1CCCN(C(=O)CC)CC1.C1(COCC)(C)CC1C(=O)N.C1COC1 c1(CNC(CCOCCCNC(C(C2CCC2)OC)=O)=O)ccccc1 Cc1c(C(=O)NCC(C)CNC(c2n[nH]cc2[N+](=O)[O-])=O)[nH]ccc1=O c1(C(=O)OC)ccc(CN2CCC(O)(C(F)F)C2)cc1Cl N1(C(CCOCCOC)=O)CCN(C(=O)CCSC)C(c2ccncc2)C1 Cc1nc[nH]c1CC(O)C(=O)NCCCOCCCNC(=O)C(C)(Cl)Cl c1(-c2c(NCc3cc(OC)nc(OC)n3)ccnc2)c(F)cc(F)cc1F C1(CCNC(CC2(C)CC2)=O)CCCN(C(=O)Cc2cnccc2Cl)CC1 CCCC(C=O)OCC.C1(=CC)CCN(C(C2(c3cc(C)on3)CC2)=O)CC1.N S(=O)(=O)(c1cccc(Cl)c1F)NCC1CCN(Cc2cc(C)c(Br)cc2C)CC1 C(=O)(C(C(C)C)n1cncn1)NCC=CCNC(C1(SC)CCC1)=O O=C(C1=CCCCCC1)NC1CCN(C(=O)CC2CCCC(F)(F)C2)C12CCC2 C1(C(N(CCCCCNC(c2c(C)onc2)=O)C)=O)CCCC(N(C)C)C1 N1(C(C2CC(O)(CC#C)C2)=O)CCC(COC)C1.c1(C=O)cc[nH]c1CCC C1(NC(C2CC(CC)C2)=O)CCCCC1NC(=O)CN1CCCC1 C1(CNC(C(C#C)(C)C)=O)CC(C)CCN1C(c1ccc(C2CC2)cc1)=O c1cc(O)ccc1Br.c1(OCCCC)ccc(C(C)NC(=O)NC2CC2)cc1.C N1(C(Cn2ccc(C)n2)=O)CCOCC12CCN(C(c1ccc(CO)o1)=O)C2 N1(C(c2cnc(CN)s2)=O)CCC(CO)CC1.C(=O)(C=CC)N(C)NC CC1CN2CCN1C(C(N1CCCC1Cn1cc(C3(S(N)(=O)=O)CC3)nn1)=O)C2 c1(CC(=O)NC2CCN(CCNC(C(C)=CC)=O)CC2)cc(C)ccc1F C1(CC)CCN(C)C1=O.C1(CC(=O)N(CCC(=O)N)C(C)C)NC(=O)NC1=O N1(C(CSCCOC)=O)CCC(CN(C(=O)C(CC2CCCC2)OC)C)C1 C1(C(N2CCC(CNC(=O)Cc3cn[nH]c3)CC2)=O)CCN(CCO)C(=O)C1 CN1CC(CC(=O)NC2CCOCC2NC=O)CCC1C(=O)O.C(C)(C)C.O C1(NC(CNC(=O)CC(F)(F)F)=O)CCN(C(C23CCC(CC2)OC3)=O)CC1F C(=O)(C(F)(C)C(C)C)NCc1cc(C)c(C)s1.c1(CC(=O)N)ccc(F)cc1 N1(C(C(C(C)C)NC(C)=O)=O)CCN(C(=O)C(O)C2CCCC2)CC(C)C1 Cc1cc(C2(C(N3CC(F)(CNC(=O)C(C)N(C)C)C3)=O)CC2)on1 C(=O)(CCCCN(C)C(C1CCOC1(C)C)=O)N(C(c1nccs1)C)C N1(C(CCC(C)=O)=O)CC2(CCC(NCc3cc(C)ccc3Br)C2)C1 Cc1cc(Cl)cc(N)c1C(N1CCOCC(NC(C2(C)CCC(F)(F)C2)=O)C1)=O C1(NC(C2CC(C(C)C)C2)=O)CCC2CN(C(C3CN(C)C(=O)N3)=O)CCC2C1 C(=O)(C1=NOC2(CCN(C(=O)C(N3CCCC(CC(N)=O)C3)=O)C2)C1)OC N1(C(C2CCCCS2)=O)CCCCC1CNC(C1(n2cccc2)CCCC1)=O CCCCC(F)C(=O)N1CC=CC1(C)C(N1CCC(C(F)(F)F)C1)=O N1(C(C2(CC)COC2)=O)CCC2(CC1)CN(C(=O)CC1(C)CC1(F)F)C2 Cc1oc(C(C)C)nc1C(N1CCC(CC(C)NC(=O)C(C)O)CC1)=O C(CN=c1[nH]nc2ccccn12)OCCNC(N1CCC2(CSC2)C1)=O C1(NC(C2CC(C(C)C)C2)=O)CCCC1CNC(c1ccn(CC#N)n1)=O C=CC1(C)COCCN1C(c1ccc(N2CCOCC2)nc1)C(=O)NC c1(C(C(=O)N(c2cccc(O)c2)C2CCCC2)O)ccc(F)c(F)c1.C1C(=O)N1 CCC(C)C(C)C(=O)NCC(CC)NC(=O)CCN1CCC(O)CC1 c1(-c2onc(C(c3cccc(F)c3)(C)C)n2)cc(OC(C)(C)C)c(C2CC2)nn1 C12(NC(c3c(CSC)cccn3)=O)CCCC1N(C(=O)CC1CSC1)CCC2 N1(C(=O)Cc2ccon2)CCN(C(c2cccc3occc23)=O)CC2(CC2)C1 Cc1cc(Cl)c(C(N2CCN(C3CCCNC3=O)CC2)=O)c(Br)c1 c1(C(=O)NC2CC(F)(CNC(C(CC)CC)=O)C2)cnc(C(C)C)nc1C c1(CN2C(C(=O)N(CCO)Cc3ccccc3)CNCC2)ccc2nonc2c1 Cc1cc(CN2CC3C(NS(=O)(=O)CCCN(C)C)C3C2)cc(C)c1Cl C12(C=O)CC(CN1C(=O)CC1CCC(C#N)C1)C2.C(C)(C(F)(F)F)OC C1(NC(CC(C)(C)NC(C=Cc2cn(C)nn2)=O)=O)CC2(C1)CC21CCC1 c1(OC)noc(C)c1C(=O)NCCN(C(=O)C(C(C)C)SC)CC(C)O C1(C(=O)NCCC2(C(=O)OC)CCC2)CC(c2ccncc2)=NO1 C1(C(N2CCN(C(C=C(CC)CC)=O)C(CF)C2)=O)CC(c2cnn(C)c2)=NO1 c1(CNC(Cc2n(C)ncc2)=O)ccccc1CNC(=O)CCC1OCCO1 N1(C(C(C)C2CC2)=O)CCC2(CCCC2Nc2ncncc2I)CC1 C=C=C(C)CC(=O)NC(C)(C)C=CC(=O)NCC(=O)N(C)C1CC1 C(=O)(C1SCc2cccnc21)N(CC(C)(C)NC(c1cc(SC)oc1C)=O)C c1(CN(C)C(C2(C)CC2F)=O)ccc(CNC(=O)CC2CCCC2)cc1 c1(C(=O)OC)oc(CSCC2CC(N)C2)cc1C N1(C(CCC2(NC(CCCC(C)C)=O)CCCC2)=O)CC2CCCC1C2CO C(=O)(C1=NOC(CNC(c2nc(C)c(C)s2)=O)C1)Nc1c(C)noc1 S(=O)(=O)(c1cccs1)N1CCCC1.C1(CC=O)CC(NC(=O)C)C1.C1CC1 n1(CCC)cncc1C(c1nnnn1C1(C)CC1)NCC(C)Oc1ccccc1 C1(N(C(c2c(CC)nns2)=O)C)CN(C(c2ccccc2COC)=O)CC12CC2 N1(C(C(C(C)C)C2CCC2)=O)CCN(C(=O)C=Cc2ccncc2)CC1C(F)F N1(CCN)CCCC(C(N2CCCCC2C(F)F)=O)C1=O N1(C(c2c(C)nc(C)o2)=O)CCC(C)CC1CNC(=O)C(C)C(C)(C)O N1(C(CN2CC(C)C2)=O)CC2CCC1CN(C(c1c[nH]c(=O)cn1)=O)C2 O=C1CCc2c(C(N3CC(CCNC(=O)C(F)C4CCC4)C3)=O)cccc2N1 CC1CN(C(c2ncc[nH]c2=O)=O)CC(CCNC(c2cc(CO)n(C)n2)=O)O1 c1(C(=O)NCC(C2CCC2)NC(CCc2scc(C)n2)=O)c[nH]nc1[N+](=O)[O-] C1(NC(=O)COc2cccnc2)CC(=O)N(c2ccccc2F)C1 C1(C(CNC(C2CCC(CC)O2)=O)C)CCN(C(C2CC(Cl)(Cl)C2)=O)CC1 C1(C(=O)Oc2ccccc2)(NC(NNC(=O)c2c[nH]c(=N)s2)=O)CC2CCC1C2 [SH](=O)(=O)c1cc(F)c(Br)c(F)c1.c1(C(=O)NC2CCCC2)cc(O)cc(F)c1 C=CCCC(N)C(=O)NC12CC(CN)(C1)C2 CP(C)(=O)C(O)C(=O)NC1CCN(C2CCN(C(=O)C3=CCSC3)C2)CC1 CC(C)CC(CC(C)C)C(=O)N(CC(C)O)CCNC(c1cnn(C)c1N)=O S(=O)(=O)(c1cccc(N2CCCC(CC)CC2)n1)NCC(CC)NS(C)(=O)=O O=C(C1=CCOCC1)NC1CCOC(C(=O)NC2CCSCC2)C1 c1(C=O)ccccc1F.C(CC(C)(C)C)NC(C1(COC)CC1)=O.CCF.N Cc1cc(C)n(CC(N2C3CN(C(C4(C#N)CC4)=O)CC23)=O)n1 CCC(CC(=O)NCC(C)N(C(=O)Cn1nc(C)cc1N)C)C(C)C C1(NC(=O)CSC(F)F)CCCC12CN(c1ccn3nccc3n1)C2 c1(C(=O)NC(C)CN(C(=O)Cc2ccsn2)C)cc(N2CCCC2)ccn1 c1(-c2c(C)c(F)ccc2F)cccc2ccc(C(N3CC4C(C3)C4(C)C)=O)nc12 Cc1c[nH]nc1C(=O)NC1CCOC1C(=O)NC(C1CCOC1)CO c1(CN)cc([N+](=O)[O-])c(C(=O)Nc2c(Br)cc(Cl)cc2Br)cc1F N1(C(CC2CC(SC)C2)=O)CCC(C)C1C(N1CCCC1C)=O c1(C(N(CC(C)NC(c2cnn[nH]2)=O)CC)=O)cnc2ncc(Cl)cn12 N1(C(c2c(C)nc(C(C)OC)s2)=O)CCCC(C)(C)C1.C1(O)(C=O)CC1.N N1(C(CCC=C)=O)CCC2(CCCCC2NC(C2CC=C(C(C)C)CC2)=O)C1 c1(C(N(C(C(=O)NC(CC)CCO)C)CC)=O)ccccc1OC c1(OC)nscc1C(=O)NC1CC(c2ccccc2)(CNC(=O)CCF)C1 c1(C=O)c(Cl)nsc1Cl.N1(C(CN(C)C(=O)C2CC2)=O)CCCC1C1CC1.N c1(C(C(=O)N(CC(C)(C)NC(C(COC)N(C)C)=O)C)(C)C)cccnc1F C(C(C)C)(C(O)C(=O)N1CCCC(C)(CNC(=O)CCc2nc[nH]n2)C1)OC CC1(C)COC(CCNC(=O)C(C)(C)NC(C2CN(C(C)C)C2)=O)C1 C(C(C)(C)CCCN=c1nc(N2CCOC(C)(C)CC2)c2ccccc2[nH]1)OC Cc1ncc(CCC(=O)NC(CNC(=O)C2=NNC(=O)C2)CO)c(O)n1 C(=O)(C1=COCCO1)NC1C(NC(Cc2cn(C(C)(C)C)nc2)=O)C1 N#Cc1ccccc1CN1CC(NC(=O)C(=O)N)C(F)(F)C1.c1ccc(Cl)cc1 c1(C(c2nc(-c3ccc(Br)cn3)nn2Cc2ccccc2F)C)cccc(Cl)c1 C(=O)(C1CCCc2ncc(C)n21)N1C(CC)CN(C(=O)Cc2cc(C)cs2)CC1 c1(CNC2CCN(CCCOC(C)C)C2)cnn2ccc(N)cc12 c1(CC(N2CCC(C(C)NC(c3c(C)cco3)=O)C2)=O)ccccc1O C1(C)(OCC(=O)NCC(CC)NC(C23CC(C2)C(C)O3)=O)CCOCC1 C(CC(=O)N1CCCCC12CC2)(C(F)(F)F)NC(CC)=O c1(CC(=O)N(CC)C)ccc(OCC)c(C)c1.C=CC(C(=O)NCC)OC N1(C(C(C)C2CCCC2)=O)CC(C)CN(C(c2cnn[nH]2)=O)C(C)C1 C1(C)(C(=O)OC)CCN(C(C2(OC)CCN(C(=O)Cc3cscn3)C2)=O)C1 c1(C(N2CC(C(=O)Nc3c(O)cccc3F)SCC2)=O)ccc2c(c1)OCCO2 c1(C(N2CCC(N3CCN(C(CC)C)CC3)C2=O)=O)cc(C)cc(C)c1 c1(C(=O)OC)cc(C(N2CCN(Cc3ccc(Br)cc3)CC2)=O)oc1C N1(CC)CC(C(N2CCN(C(c3cc(CO)[nH]n3)=O)CC2C2CC2)=O)CCC1=O c1(C(N2CC3C(NC(C(CCC)C)=O)(CCC3)C2)=O)cc(C)nc2c1cnn2C c1(C(=O)NC2C(CNC(C3(C)CCOC3)=O)COC2)ccc2c(c1)CCOC2 c1(C(N2CCN(C(CNC(=O)Cn3ccnc3)=O)CC2)=O)cc2ccccc2s1 C#CCC(C(=O)NC1CC(NC(=O)C=CCN2CCNCC2)C1)C1CC1.C N1(C(C(C(C)C)OC(C)=O)=O)CCC2(CCCN(C(=O)CCS(C)(=O)=O)C2)C1 C(C(=O)NNC(=O)C(C)(C)CCCCNC(C1(Cl)CC1(C)C)=O)C1C(C)C1 C1(OC)CC(NC(=O)CC2CCCS2(=O)=O)CN(C(c2cc(C#N)on2)=O)C1 CC(C)C(C(=O)NC1CCCC1)N1CCC(CS(C)(=O)=O)C1 c1(CCCC(=O)OC(C)(C)C)ccc(C(=O)NCCC(O)CO)cc1 C1(C(=O)N(C(=O)C(N2CCS(=O)CC2)c2ccccc2)CC)CNCC2(CCC2)C1 C(=O)C1=NOC2(CCN(C(C34CC(F)(C3)C4)=O)C2)C1.c1(CCC)ccncc1.N C1(C(=O)NCC(C)CC(F)(F)F)CCCN1NC(=O)C(C)(C)CC(C)(C)C c1(C(N2CC3C(C(=O)NC(c4ccc(Cl)cn4)C)(C3)C2)=O)c(Cl)cccc1Cl C=C=CC(C)C(=O)NCC(c1ccc(OCCC)cc1)NC(=O)C(C)(O)C C=CCC(F)(F)C(=O)N1CCC(=CCNC(=O)Cc2ncc(C)s2)CC1 Cc1nc(C)c(C(=O)NC2(CF)CCN(C(c3ccc(-c4cccs4)s3)=O)C2)[nH]1 C(=O)(C(F)CC(C)(C)NC(c1ccn(C2CC2)n1)=O)NCCCCCC(C)C c1(CCCC(=O)NC2CCCC(NC(=O)CCn3cncn3)C2)ccccc1Cl c1(CC(N2CCC(CNC(CSCC#C)=O)C2)=O)ccc(C#C)cc1 c1(CNC(=O)NCCCn2ncc(C)c2)ccc(N(C)C)cc1C c1(C(=O)N)ccc(C#N)c(O)c1.c1(N(CC(=O)NCCCC)CC)ccccc1 C1(OC)CCC12CC(C(=O)NCC1COCC1)C2.C1(CC(=O)N)CC=CC1 Cc1nc(C(=O)NCC(C)NC(C2COCC(C)(C)O2)=O)ccc1Br C1(CNC(=O)Cn2cncn2)COCCN(C(=O)Cc2c[nH]nc2O)C1 CCCC(C(=O)N1CC2C(NC(=O)CCc3nc(C4CCCC4)no3)C2C1)OC CC1CN(C(=O)CCCn2cnc(C#N)n2)CC1NC(C1(C)CC1)=O.C1CC1 C=CCC(C(=O)NC(C1CC1C(=O)OC)C)NC(C1CCOC1C=C)=O CCC(CC(=O)NC1CN(C(c2cc(C)c[nH]2)=O)CC(C)(C)C1)CC(F)(F)F C1(NC(C2(C=C)CCC2)=O)CC(C)CN(C(=O)C=Cc2nc(C)cs2)C1 C1(C(=O)NC(C#C)CC2CCC2)CN(C(c2ncc[nH]2)=O)CC1CCC(C)C c1(OC)ccc(I)c(NC(c2c(-c3ccc(F)c(F)c3)cncc2F)=O)c1 c1(OC)cc(C(=O)NC(C)C(C)NC(c2ccccn2)=O)cc2ccoc12 C(=O)(C(CNC(C1(C)CC=CC1)=O)CCC)N(CC=C)CC=C c1(C(=O)N)n[nH]cc1[N+](=O)[O-].C(C)(C(=O)N(CCCN(C)C)CC)=C(C)C CCC(CC)C(F)C(=O)N(C)CC1C2CN(C(c3cnc4ccnn4c3)=O)CC12 CC1=C(C(=O)NCCC(C)NC(C2CCC(F)(F)CC2)=O)CCCO1 Cc1c(NCC2CC2(F)F)nc[nH]c1=NCC(C)(C)CN1CCN(C)CC1 Cc1cc(NNC(=O)C2OCCC2CN)nc(-c2ccccn2)n1 CCCCC(C(=O)NCC1CN(C(=O)Cn2ccccc2=O)CCCO1)C(C)C CC1CCCCC1(CNC(=O)COC(F)F)NC(=O)Cn1ccccc1=O C12(CNC(C(CCC)(C)O)=O)CCCCC1N(C(c1oc(C)nc1C)=O)CC2 C1(C(=O)NCCC(=O)N(CC)CC)CCC(n2cc(C(O)C(C)C)nn2)C1 C(=O)(CCC[N+](=O)[O-])NC1C(CNC(c2nccc(N)c2)=O)CCCC1 C=CCC(CNC(C1CCCN1C)=O)NC(c1cnn(C(F)(F)F)c1)=O CC1CCN(C(C2CC(C)(O)C2)=O)C1C(=O)N(CC(C)(C)O)C C1(C(=O)NCCN(C(=O)Cc2cc[nH]n2)C(C)C)CCCCN1C(C)C c1(C(=O)NC2(CF)CCN(C(C(C=C=C)C)=O)C2)cc2c(F)ccc(F)c2[nH]1 C(=O)(C(CCC)CCC)NCC1N(C(C(C)OCCCCCC)=O)CC1 CCC(C)CC(C)N(C)C(c1cn(CC2CNC(=O)O2)nn1)=O C1(C(=O)NCC(C)N(C)C(c2ccc(C(C)(C)C)[nH]2)=O)CCCN(C)C1 c1(C=O)cc(C=O)ncc1F.C1(NC(C=C(COCC)C)=O)CCCC1.C CCC(CC(=O)NC1COCC1NC(=O)COc1cccc(C)c1F)C(C)C CC(C)CCC(C(=O)N1CC=CC1CF)NC(c1n[nH]cc1Cl)=O CC(C)CC(CNC(c1csc(O)n1)=O)NC(=O)Cn1cnc(Br)n1 C(=O)(C(O)C(C)(C)C)N1CCC(N(C(=O)CCc2ccsc2)CCC)C1 c1(C(=O)NC2CCCN(C(Cc3ccc(C)cc3)=O)CC2)ccc2c(n1)CCC2 C1(NC(c2c(N)cccn2)=O)CN(C(C2CC2(Cl)Cl)=O)CC12CCOCC2 C1(C(=O)NCC(CC)(C)Cl)CCN(C(=O)CCc2ncccn2)CC1(C)C CC(CC(=O)NCCN(C)C(=O)C1CC1)C(C)C.C1(C)(C=O)CCOCC1.N N#CC1(C(=O)NCC#CCNC(=O)Cn2ccc(O)nc2=O)CC2(CC2)C1 Cc1cnc2nc(C(=O)NCCCNC(c3c(C(F)F)cccc3F)=O)nn2c1 Cc1cc(F)cc([N+](=O)[O-])c1NC(C1CC1NC(c1snc(Cl)c1Cl)=O)=O CC(C)C(O)CC(=O)NCC(N1CCN(C(c2ccn(C3CCC3)n2)=O)CC1)=O C=CCCCC(C(=O)N(CC)Cc1ccncc1)NC(C1CCCC(C#N)C1)=O CCCCCCC(C)C(=O)N1CCCC(CNC(=O)C(F)(F)c2cncs2)C1.C(C)C c1(C(CNC(C2C(C)CC2)=O)N(C)C(C2CCCC2)=O)ccccc1 C(CC(C)C)(C(=O)NC1COCC1CO)ONC(CCN(C(=O)OC)C)=O c1(C(C)=O)cccc(C(=O)NCCC2CN(C(=O)C(C)CC3CC3)CC2C)c1 CC1c2ccccc2CC1NC(=O)N(C1CC1)Cc1cc(N(C)C)cc(F)c1 c1(C(=O)NCC2CCCN(C(=O)C=Cc3cnc[nH]3)C2)ncnc2c1OCCO2 C1(C(=O)NC(C(=O)N(CC)CC)C)CCCN1NC(=O)c1ccccc1O N1(C(C(C)=C2CC2)=O)CC(CNC(C23CSCC2C3)=O)CC(C)C1 CC(C)CS(=O)(=O)CC(=O)N(C)CC1CCCN1C(=O)CCc1cnc(O)[nH]1 CCCCCCC(=O)NCC(CC1CCCC1)C(=O)NCCc1ncc[nH]1 C1(C(C)NC(CC(=C)C)=O)CCCN(C(c2cnc(N(C)C)nc2)=O)C1 c1(C(N2CC(CC)CCC2)=O)cc(S(N)(=O)=O)c[nH]1.C(=O)(C(CC)(CC)CC)N Nc1ccc(F)cc1C(=O)NC.C12CCC1CN(C(c1ccoc1C1CC1)=O)C2 C(=O)(C(C(C)NC(=O)C(N=[N+]=[N-])C(C)C)C(C)C)NCc1cn(CC)nc1 c1(CCCC)nc(C(=O)NCC2CCCC2NC(=O)Cn2cccc2)cs1 C1(O)(CCNC(C2N(CC)CCOC2)=O)CCN(C(=O)C)CC1.C(N)(=O)N O=C1NCC(C(N2CCC(OCCNC(c3cncn3C3CC3)=O)C2)=O)N1 CCCC(C(=O)OC)C(=O)NCC1CC(NC(C2CCC(C)(C)CO2)=O)C1 N1(C(c2cc(C)nc(C)c2)=O)CCCC2CN(C(=O)Cn3c(C)ccc3C)CC12 CCCCC(C)C(=O)NC1CC1NC(c1ccn(Cc2ccccc2)n1)=O c1(-n2cc(C3N(C(CNC4C(OC)(OC)CC4)=O)CCC3)nn2)cccc(F)c1 Cc1noc2ncnc(NCC(C)(C3CC3)NC(=O)COCC(F)(F)F)c12 N1(C(CCC(C)C)=O)CCCC(C2CC2)C1.C(=O)C(Br)=C(C)C.C(=O)OC.N C(C(C)N=c1[nH]c2c(c(=NCC3CC(C(F)(F)F)CO3)[nH]1)CCC2)OCC N1(C(C2CCN(C(=O)NC)CC2)=O)CC2CN(C(=O)C(C(C)(C)C)OC)CC2C1 C1(NC(C2=C(C)OCCS2)=O)COC2(CCN(C(c3cn(C)cc3C)=O)CC2)C1 C#Cc1cc2nccc(N3CCN(Cc4ccc(C)cc4)C(=O)C3)c2s1 N1(C(C(=O)Nc2ccc(C)cc2)=O)CCN(C(=O)CCCS(N)(=O)=O)CC(O)C1 c1(CC(N2CC(C)C(NC(=O)CSC)C2)=O)nnc2n1CCOC2.c1cccs1 O=S(=O)(c1cn[nH]c1)N1C2CN(Cc3ncc(-c4ccccc4)[nH]3)CC12 C1(NC(C2(C)CC(=C)C2)=O)CC(NC(=O)CCc2cncnc2)CC1O C=CCCN=C(NCC(CC)N1CCCC1)NC1CN(CC(C)(C)O)C1 CCC(C)CCC(=O)NCC(C)CNC(=O)CCN1CCC(O)CC1 C1(C(N2CC(NC(c3c(C)scn3)=O)C(O)C2)=O)CCC2(CCC2)CO1 c1(C(=O)NC(C)C=O)cc(CNC(=O)CCc2ccco2)cs1.C1CC1.N c1(CC(=O)N(C2CN(C(=O)Cn3ncccc3=O)CC2O)C)cc(O)nc(O)n1 N1(Cc2cn(CC(=O)N(C)Cc3c(C)nsc3)nn2)CCS(=O)CC1 C1(CC=C)(NC(c2cnc(C)s2)=O)CCN(C(=O)CC2CCC(=O)NC2)CC1 C(=O)(C1=CCCCC1)C1CC(C)(C)C1.N12CCCC1(C)C2.C1Cc2nnsc2S1.NC Cc1cc(C=CC(=O)NCC(C)(CO)NC(C2CC3CCC3C2)=O)ccc1F c1(CS(=O)(=O)NC2CCCN(C(c3ccc(F)cc3)=O)C2)c(F)cccc1F CC(=O)CCCCC(=O)N1CCCCC(CNC(C2C=CCS2)=O)C1 c1(C(c2nnnn2C)NC2C(c3cn(C)nc3)C2)cc(C2CC2)nn1C c1(C(=O)NC2(CF)CCN(C(c3n(CC)ncn3)=O)C2)cnc(O)cc1C C1(C(=O)NC2(CC=C)CN(C(=O)CCn3cncn3)C2)CC2(CC(=C)C2)C1 CC1(C)CCN(C(=O)CCC2CCC2)C1CC(=O)NCCn1cccn1 c1(-n2c(C)ncc2)cc(C(N2CCC(CN(C)C(C)C)C2C)=O)ccc1F Cc1nc2c(C(N3CCC(C)C3CNC(=O)Cc3ccc(Cl)s3)=O)ccnc2[nH]1 CC1CN(C(=O)CNC(c2ccccc2)=O)CC(C)C1C.C(=O)CC(C)(C)O Cc1nc(NC2CC(F)(CNC(c3ccc(F)cc3Cl)=O)C2)c2cnn(C)c2n1 Cc1ccccc1S(=O)(=O)CC(=O)N1CC(NC(c2nonc2N)=O)CCC1C Cc1nc(N2CCOCC2)sc1-c1nc(Cc2csc(CCC(C)C)n2)nn1C Cc1c(Cl)cc(C(N2C3CC2CN(C(=O)C(C)Cc2ccccn2)C3)=O)cc1Cl N1(C(=O)OC(C)(C)C)CC2CCC(CNC(c3ccc(F)nc3O)=O)(C2)C1 c1(CNC(COC(CC)(C)C)=O)ccc(C(=O)NCCC2CCCO2)o1 c1(CNC(CCCN(C(c2cc(C(C)=O)on2)=O)C)=O)ccc(C)cc1F N1(C(C(CC)(C)F)=O)CCOC2(CCCN(C(c3cccc4ncnn34)=O)C2)C1 C12(C(=O)NCC(C)CNC(=O)CCCCN(C)C)CCCC1CC(=O)C2 C1(NC(C2(c3cc(C)no3)CC2)=O)CCC(C)C1.C(=O)C(C)CN(C)C.C Cc1c(NCC2=CCCC2)ncnc1N1CCCC(C(N2CCCCC2)=O)C1 c1(C=O)cccc(C(F)(F)F)c1C.C1(NC(CC)=O)CCC1NC(=O)CC.O C1(NC(C(CC)NC(N)=O)=O)C(C)(C)CC1(C)C.c1(C(=O)N)c[nH]nc1C C1(NC(C=CSC)=O)CCCN(C(c2cccnc2OCC2CCCC2)=O)C1 CCC(CC)(CC)C(=O)NC(C)CNC(=O)C(C)Cn1ccc(C)n1 c1(OCC)ccc(Cl)c(C(N2CCCC2)=O)n1.C(c1nc(C)cs1)=CC=O.C N1(C(C(CC=C)(C)O)=O)CCN(C(=O)C(C)c2cccs2)C2(CCC2)C1 CC(C)CS(=O)(=O)CCC(=O)NC1CC2CN(C(=O)CCC3CC(F)(F)C3)CC12 C1(NC(CC2(OC)CCC2)=O)CC(C)N(C(=O)CCSCC(N)=O)C1 c1(-c2nc(CO)nn2CCOCC(F)(F)F)cccc2cc(F)ccc12 c1(OC)ccc(CC=O)c(Cl)c1.CC(O)CN(C)C(C1CC(C(C)(C)C)C1)=O CC1(C)C(C(=O)NC2CC(C(=O)NC)CC2O)C1(F)F.C1CC12CC2(F)F C1(NC(c2scc(COC)c2)=O)CCCN(C(=O)C(C)NC(C)(C)C)C1C C1(C(N2CC(n3c(-c4ccc(F)cc4)nc(OC)n3)C2)=O)CCC([N+](=O)[O-])CC1 CP(C)(=O)CCC(=O)NCc1ccccc1CNC(=O)C1=CSCCO1 C1(C)(NC(C(C)(N(C(=O)CCC2CCCC2)C)C2CC2)=O)CCCCC1(C)C c1(NC)cccc(CCC(N2CCCC(NC(C3CCC3)=O)C2)=O)c1 CC1CN(C(c2cn(C3CC3)cn2)=O)CC1CC(=O)NCC(C)(C)C1CC1 c1(OC)c(C)csc1C(N1CCOC(C(C)NC(=O)Cn2ncnn2)C1)=O c1(CC)ccc(C(N2CCC(CC)C2)=O)cn1.c1(CCC(=O)N)nc(C)c(C)o1 C(=O)(CCC(C)(C)C#N)N.c1(CC)ccc(CNC(=O)CCCC2CCC2)o1 C(CCCC(=O)N(CCNC)C(C)C)N(C(C)=O)C.C1(C(=O)N)C2COCC12 N1(C(c2cnc(OC)nc2C)=O)C(C)CC2CN(C(=O)C(C)C3=CCCC3)CC12 C(=O)(CC(C)(C)CC(=O)N1CC2CC2(CNC(=O)C(C)N2CCC2)C1)OC n1(C(C)C)nc(I)c2c(NC(C3CCN3Cc3cc(F)cc(F)c3O)=O)ncnc12 N1(C(=O)CC2CCOCC2)CCN(C(=O)Cc2cncs2)C(c2cccnc2)C1 Cc1cc(CNC(=O)CNC(=O)C=Cc2ccc[nH]2)ccc1F N1(CC(=O)NC2CCCC(NC(c3c(CC)scc3)=O)C2)CCn2ccnc2C1 N1(C(C2C(C(=O)OC)C=C2)=O)CCC2CCC(C1)N2C(=O)COC(F)(F)F N1(C(C=CC(C)(C)NC(CC2CCN(C)CC2)=O)=O)CCC(C)(F)CC1 N1(CCC=O)CCN(C(C)C)CC1.CC1C(C(=O)NCCOCC)C1(F)F C1(C)(C(N2C(C(=O)NC(C)C(C)(C)C#N)CC2)=O)CC(=O)N(C)C1 N1(C(C(CC)F)=O)CCC(CNC(C2(n3cc(Br)nn3)CC2)=O)CC1 c1(C(=O)OC)ccc(CNC(=O)Nc2c[nH]nc2C(F)(F)F)cc1C#N c1(OC)ccc(-n2cc(C(C)(C)NC(=O)C(C)OCC3CC3)nn2)cc1Cl Cc1ccc(Br)cc1CNC(=O)C(=O)NC1CCNC2(CC2)C1 C1(NC(c2cnc(CC)s2)=O)C2CCN(C(c3ccn(CCO)c3C)=O)CCC12 CCCC(C)CC(=O)N1CCCC(N(C(=O)CCCC#N)Cc2ccccc2)C1 Cn1cc(C=CC(=O)NC)cn1.C1(C)CCCC1.c1(CCC=O)cnn(C)n1 C1(C)(C(N(C)C)=O)CC(C2CC2)=NO1.Cc1ccsc1C=CC(N1CCCC1)=O C=CCC(C)(C(=O)NCC1CCCN(C(C2CCC=CO2)=O)C1)N(C)C CCC(C)(C)CCCC(=O)N1CCCC(C(=O)NCCN2CC(CF)C2)C1 Cc1ccc2c(c1)CC(C(=O)NC(C)CO)S2.C1(C#N)(C=O)CC2(CC2)C1.N c1(C(=O)NC2C(NC(=O)CC34CCCC3C4)CCCC2)cnc2c(c1)COCC2 C1(C(C(=O)OCC)(C)C)CCN(C(=O)C(n2ccc(Br)n2)C)CC1 c1(C(C(=O)OC)NCc2ncc(CC)[nH]2)ccc(C(F)(F)F)cn1 C(c1cnc(OC)nc1)=CC(=O)NC(CNC(c1cnc(OC)nc1)=O)C c1(C(=O)NCC2N(C(CC(COC)(C)C)=O)CCCC2C)ccccc1N=[N+]=[N-] CC1(C)CN(C2CCN(C(c3cccs3)C)C2=O)CCC1NC(=O)C.C(N)=O.N O=C(C(CNC(C12CC(F)(C1)C2)=O)CC1CCCC1)NCC=CCl C1(NC(c2nc[nH]n2)=O)CC2(C1)CC(C(=O)Nc1cc(F)cc(F)c1)C2 C(=O)(C1=CCC(NC(=O)CCC(=O)CC)C1)N1CC(O)(CC=C)C1 c1(C(N2CCCC(n3ccnc3)C2)=O)c[nH]c2nc(Cl)ccc12 N1(C(C=CC=CCC)=O)CCCC(NC(c2c[nH]nc2CCC)=O)CC1 c1(CNC(CNC(CNC(C(C)SC)=O)=O)=O)nnn(C)c1C C1(C(=O)NCCCN(C(C(c2scc(C)n2)C)=O)C)COC2CCCCC12 C(C)(C(=O)N1CC(N(C(=O)COCC2CCOC2)C)C1)OCC Cc1cc(N)c(C(=O)OCCSCC2CC(C)OC(C)C2)cc1F N(C1CCCc2c1[nH]c1ccc(F)cc21)C1C(C)CN(C(=O)OC(C)(C)C)CC1 C(C(C)C(C)C(=O)N(CC(=O)NCCCc1n[nH]c(C)n1)CCO)OC c1(CCC(=O)NCCC(C)NC(C2(CF)CCOCC2)=O)ccc(N(C)C)cc1 CC(C)CC(C)(O)CNC(N1CCC(Cc2ccccc2Br)C1)=O N1(C(C2=C(C)OCC2)=O)CC2(C)CN(C(c3cc(F)c(Cl)cc3Cl)=O)CC2(C)C1 CC(C)CCC(F)C(=O)OCC(C(CCO)c1ccco1)=O.C1C(=O)N1 c1(CC(=O)NCCN(C)C(C2CCC3CCC(=O)N23)=O)c[nH]c2cccnc12 Cn1nnc(CNC(=O)CCC2CC(NC(=O)CCc3nc(O)n[nH]3)C2)n1 CC(CN(C)C)CC(=O)N(CCC(=O)NC(C)C(C)(C)CO)C(C)C c1(C(=O)NCC(CN(C(CN(C)CCO)=O)C)O)c(Cl)cc([N+](=O)[O-])cc1Cl C1(CC)CCN(C(=O)Cc2ccc[nH]2)C(C(=O)NCCNc2cccnc2)C1 c1(C(=O)NC(CC)CNC(c2c[nH]nc2C)=O)cccnc1N1CCCC1 C(CNC(c1conc1-c1ccccc1)=O)(C(C)(C)C)NC(C(C=C)O)=O N1(Cc2nc(-c3ccc(Cl)cc3)oc2)CCOc2ccccc2C1 C1(C(=O)NCC(C(C)C)NC(=O)C=Cc2cnccn2)COC2(CCC2)C1 C(CC(O)CO)NC(CC1N(C(CN(C(C)=O)C)=O)CC1)=O N1(C(C2C(C=C(C)C)C2(C)C)=O)CCC(C)C(NC(c2cnn(C)c2Cl)=O)C1 n1(CCC)cncc1C(C(=O)NCSC1CCOCC1)N(C1COCC1OC)C c1(C(N2CCC(NC(C3C4CCCCC34)=O)C23CC3)=O)cccc2cccnc12 N1(C(C2CN(CC)C(=O)C2)=O)CCOCC(CNC(=O)CCCCSC)C1 C1(CN(C)C(C2CNC(=O)C2)=O)CCN(C(C2CC(N3CCOCC3)C2)=O)C1 c1(C(=O)NCC2(C)CCN(C(CC3C(C)CCCC3)=O)C2)c(Cl)ccc(F)c1N Cc1nn(CC(N2CC(NC(=O)C(C)(C)C#N)CC23CCC3)=O)cc1[N+](=O)[O-] C(=O)C(C)P(C)(C)=O.Cc1n[nH]c(C)c1CC(C)C(=O)NCCC1CCC1.N CC1CN(C(=O)C(CC2CC2)NC(=O)CCCCC(N)=O)CC(C)N1C c1(C(=O)NCC2CN(C(C3(CCCC)CC3)=O)CC2O)cnc(OC)cc1C C12(C(=O)NCCC(=C)CNC(C3(C)CCCN3C)=O)CCC(C)(C1)OC2 c1(SC)nc(Cl)c(C)c(=NC2CC3(CCC(NC(=O)CCCC(N)=O)CC3)C2)[nH]1 C1(OC)CC(CNC(c2ccncc2C)=O)N(C(c2ccc(=O)oc2)=O)C1 N1(C(c2c(C)oc(Cl)n2)=O)CCC(C)(C)C(CNC(C2CC3CCC2C3)=O)C1 N1(C(C(C)OCCC(C)C)=O)CCCCC1CN(C(=O)C#CC1CC1)C CC1OC(C)CC1CC(=O)NCCC1CCCN(C(=O)CCCc2nccs2)C1 CCC(O)C(C)C(=O)NCCC1COCCN1C(=O)Cn1ccc(C)n1 C1(C(=O)NC2(CC(=O)N(CC)CC3CCOCC3)CC2)CC2C=CC1O2 c1(C(c2nnnn2CCC2CC2)NC(C)CCO)cccc(F)c1C(F)(F)F N1(C(Cc2nnc(C)s2)=O)Cc2ccccc2C(NC(=O)CCCNC(N)=O)C1 C1(NC(CC=C)=O)C2CN(C(=O)C(=O)Nc3ccc(N4CCCCC4)cc3)CC12 c1(C(N2CC(CNC(c3occ(C)c3)=O)C3(C2)CC3)=O)c(F)ccc2c1OCC2 C1(NC(c2cc(CC)n(C)n2)=O)CCC(C)N(CCOc2ccc(C)c(C)c2)C1 C1(NC(=O)NCCCN2CCCCC2)CC2(C1)CC(NC1CCC=CO1)C2 C12(CCC(N3C(CNC(C(C)OCC)=O)C=CC3)=O)CCC(CC1)C2 C(=O)(C(O)C1=CCCCC1)N(CC(C)NC(c1cc(C#C)cc(N)c1)=O)CC CC(=O)CCCC(=O)NCC1CCN(C(C2CCCC(OC(F)(F)F)C2)=O)CC1 c1(C(CCC)OC(C2OCCC2CC)=O)nc2ccccc2[nH]1.C(C)(C)C.C=O.N N1(C(CNS(NC)(=O)=O)=O)CCN(C(c2c[nH]cc2C)=O)C(C)C1 C1(NC(CCNC(=O)CO)=O)CCN(C(=O)C(O)Cc2cnc[nH]2)CC1O c1(OC)ccccc1CC(C)(C)C(=O)N.c1(C(N(CCC)C)=O)nn(C)cc1Cl CC1=C(C(=O)NCC2(C)CC(NC(C3CC3C3CC3)=O)C2)CCCC1 c1(C(=O)NC2CCN(Cc3cn(CC(C)C)nn3)C2)coc2c1COC2 C(=O)(C(C)CS(C)(=O)=O)N1CC(C)CC(CNC(C2=C(C)OCC2)=O)C1 N1(C(=O)Nc2n(C)cnc2[N+](=O)[O-])CCc2c(F)cc(F)cc21 N1(C(c2ccnn2C)=O)CCN(C(=O)C)CC(C)(C)C1.C(=O)CN(C)C.C CC1CCC2(CN1C(C1(S(C)(=O)=O)COC(=O)C1)=O)OCc1ccccc12 C1(C2CCCCC2)(C(=O)NC2COCCN(C(C3CCC(C)(C)CC3)=O)C2)CC1 c1(OC)cncc(Br)c1C(N1CCC(C)C(NC(=O)C(C2CC2)OC)C1)=O C#CCC(CC(=O)OC)NC(C1CC(N(C)C(C2CC2C(C)C)=O)C1)=O C1(N(C(C(CO)N(C)C)=O)C)CC2CCC(C1)N2C(=O)C(C)(O)C1CCC1 c1(C(N2CC(C=C)(CC(=O)NC3(C=C)CCCC3)C2)=O)ccc(C#N)cc1C c1(C(N2CCC(NC(C3CCCN3C3CC3)=O)C23CC3)=O)cncc2nc[nH]c12 CC(C)(F)C(C)(F)C(=O)NCC1CC2CCC1N2C(c1coc2c1CCCC2)=O c1(C(=O)NC2CN(C(CC3N(C)CCCC3)=O)C2)cc2c(s1)CCSC2 c1(OC)ccc(NC(C2CCN(C(=O)C(CO)N(C)C)C2(C)C)=O)c(C)c1 C1(NC(c2nc(CNC(C=CC(C)C)=O)oc2)=O)C2CCC3C(C2)CC13 N1(C(CC2C(OC)C2)=O)CCC2(CC1)COC(C)C2.C(=O)COCC=O.N c1(C(=O)NCCNC(CSc2n(C)ccn2)=O)cccc(Br)c1N N1(C(C(COC)C)=O)CC2CCC1C(CNC(C13CCCCC1C3(F)F)=O)C2 C(=O)(C(COC)CC(C)C)NCCCC(C)(C)NC(CCCCC)=O C1(CC(N2C(CC(C)O)COCC2)C(=O)NC2CC2)CCCCC12CC2 c1(C(=O)NC(C2CCCN2C(=O)C(F)C2CCCC2)C)cccc(CCO)c1 N1(C(CCC2N(C(Cc3nc(C)sc3)=O)CCCC2)=O)CC(C)OCC(C)(C)C1 C12(C(N(CC(C)C)C)=O)CC(C)(CN1C(c1cn(C)ccc1=O)=O)C2 CC1(C)CCN(C(c2ccccc2Br)=O)CC1CNC(C1C2CCCCC12)=O CC1(C)C2CCC1(NC1COC3CC1C3)CC2 c1(CC)ncc(C(=O)NC(C2CCN(C(=O)CC)C2)(C)C)s1.c1nccn1C.S N1(C(CCc2onc(C)n2)=O)CC(NC(c2cnoc2C)=O)CC(C)C1 c1(N2CCCC(CN(C(CC(C)c3cnn(C)c3)=O)C)C2)ncc(Cl)c(O)n1 C(c1cc(Cl)nc2ccccc12)=C(C)c1ccc(Br)cc1 C1(NC(c2c(CC)n(C)cc2)=O)CC2(CCC(NC(=O)CCC(C)SC)CC2)C1 c1(C(=O)N)ccc(S(=O)(=O)N(C2CCOC2)C)cc1.c1(CC)ccccc1OCF C1(CC(=O)NC2C(NC(Cc3c(C)ccs3)=O)CCC2)(CO)CCOCC1 Cc1cc(COC(=O)Cc2cc(C)c(Br)c(C)c2)c(C)c(C)c1 C1(C(N2C(CCC=C)CCC2)=O)C2CC(O)C(C2)N1C(=O)Cn1ccnn1 c1(C(C)C)ccc(C(N2CC(C)CCC2CNC(=O)CCC(C)(C)C)=O)cc1F c1(CC)ccc(C(=O)NC2C=CC(CNC(=O)CCCC3CC3)C2)nc1 C1(C(=O)NC2CCCN(C(=O)CSc3nncs3)CC2)CCc2ncncc2C1 C(=O)(C(C)C(O)C(C)C)N1CC(C(C)C)N(C(c2cn(C3CC3)nn2)=O)CC1 Cc1nc(N2CC3CC(NC(=O)CN4CC5CC5C4)C3C2)ccc1C#N c1(CCC(=O)NCCC(C)NC(C2(n3ccnn3)CC2)=O)ccccc1[N+](=O)[O-] c1(C(N2C(CNC(c3cnc(CC)[nH]3)=O)CC2)=O)cc([N+](=O)[O-])cnc1O O=C(C1=NOCC1)NCc1n[nH]cc1C(=O)NCCN1CCCCC1 C1(C(N(C(C(=O)N)(C)C2CC2)C)=O)CCC(F)(F)C1.O(C(F)(F)F)CCC C1(C(=O)NC2C(NC(CN(CC)CC)=O)CC2)(O)CCCCC1.C(C)C N1(C(CC2(OC)CN(C(C3(CO)CCCC3)=O)C2)=O)CCCCCCCC1 C1(C(CO)NC(C2C(CC)CCC2)=O)CCN(C(c2[nH]ccc2C2CC2)=O)CC1 c1(CNC(CSCC)=O)ccoc1C(=O)N(CC(C)C)CCOC CC1(C)CC(C)N(C(=O)CCC2CC2)C1.c1(C(C=O)(F)F)cccc(F)c1F.N c1(C(=O)NC2CCC(CCNC(CSCC)=O)C2)cc2n(n1)CCCO2 N1(C(CCC(=C)Cl)=O)CC(NC(c2ccc(O)cn2)=O)CC12CCOCC2 C(=O)(CC(C)(C)C#N)NCCC(CNC(c1c(OC)c(C)cs1)=O)O c1(NC(=O)C2=CCOCC2)nc2ccc(Cl)nc2s1 c1(C(N(CC=CC(=O)N(CCCC)C)C)=O)ccc2cc[nH]c2c1 CCCCC(F)C(=O)NCC(C1CCC1)NC(c1nccnc1C)=O C(CCNC(=O)C(CO)OC)(C(=O)NCc1cc(C)ns1)OC c1(CC)cccc(CC(=O)NC2CCCCC2NC(=O)C=Cc2cccn2C)c1 Cc1c2c(-c3cscc3C(N3CCCCC3CO)=O)cccc2nn1C C#Cc1ccc(C(=O)N(C2CCN(C(=O)CCc3ccnc(Cl)c3)C2)C)cc1Cl c1(OC)cccc(CC(=O)N(C(C)CNC(=O)CC2CC(F)(F)C2)C)n1 c1(C(N2C(CNC(=O)C#CC3CCCO3)CC2)=O)ccc2c(c1)SCC(=O)N2 c1(C(N2CC3CC(NC(C4CC(OC)C4)=O)CC3C2)=O)ccc2cccnc2n1 Cc1ocnc1C(=O)NCCc1cc(C(=O)NCCc2ncnn2C)no1 c1(NC(c2n(CCOC)nnn2)c2csc(-c3ccc(Cl)cc3)n2)cncnc1S Cc1nn(CC(=O)N(C)CCOCCNC(C2CCSC(C)C2)=O)c(C)c1C C(C(F)C(=O)NC(C1CCCN1C(=O)CC(=O)OC)C)N(CC)CC c1(C(=O)NCC(CNC(C(CSC)O)=O)(C)F)cnc(N(C)C)nc1 Cc1c(C(N2CCC(N(S(C)(=O)=O)CCO)C2)=O)c(Br)nn1C C1(C(N(CCCCCNC(c2c(OC)cccn2)=O)C)=O)CC2(C1)CC(O)C2 c1(OC)ccc(C(N2CCCCC2C(=O)NCCc2cnc[nH]2)=O)cc1Cl C1(CNC(c2n[nH]c(C)c2Cl)=O)CCC12CCN(C(c1nc(O)sc1C)=O)CC2 N1(C(C2C(CNC(C3CCC(=O)O3)=O)CCC2)=O)CC2CCCC(C2)C1 Cc1nnc2n1CCC2(C)C(=O)N1CCC1CNC(c1nocc1C(C)C)=O c1(C=O)ccc(O)c(C(C)(C)C)c1.n1(CC=O)ccc(C)n1.C(C)(C)OC CC1CCCN(C(=O)COCCN(C)C)C1C.c1ccccc1O.C(=O)(C)N Cc1cc(C(=O)NCC=CCC(=O)NCC(c2cccs2)O)on1 C1(C(=O)NC2(CF)CCN(C(C(CC)CC3CCCC3)=O)C2)CC2CCC(C1)C2 CC1(CNC(C2CCC(=O)NC2)=O)CCN(c2cc(Cl)c(O)nn2)CC1 Cc1ccc(C(F)(F)F)cc1NC(=O)C(=O)NCC(=O)NCCO CCCC(CCC)CC(=O)NCC(C1CCOC1)NC(c1ncc[nH]c1=O)=O Cc1ccc(F)c(C(N2CCC(CNC(c3sccc3CC#N)=O)C2(C)C)=O)c1 c1(CC(=O)NCCC(CNC(c2nnc(C)s2)=O)O)ccc(F)c(F)c1 N1(C(C=Cc2c(C)cncc2)=O)CCC(C)N(C(c2cccc(C)c2O)=O)CC1 Cc1ccc2oc(C(=O)NC3(CNC(=O)C(C)C#N)CC3)c(C)c2c1 c1(C(N(CCNC(C(C)Nc2ccccc2)=O)C)=O)ccc(-n2ccnc2)cn1 CC1CN2CCN1C(C(=O)NCC1(C)CCN(C(=O)C=Cc3ccsc3)CC1)C2 c1(C(N(C)CC2OCCN(C(C=CSC)=O)C2)=O)cc(S(N)(=O)=O)cc(C)c1C C1(C(N(C)Cc2nnn[nH]2)=O)CC2(C1)CC2(F)F C(C(CC(F)(F)F)NC(=O)C(N)=O)NC(C1CCC(CC)CC1)=O Cc1cc2cccc(NCCc3c[nH]c4c(F)cccc34)c2o1 CC1(NC(C2CC3CC2CN(C(c2nc(=N)cc[nH]2)=O)C3)=O)CCC(=O)NC1=O c1(C(=O)NCC(C2CCN(C(C3C(C)C3)=O)CC2)(C)O)ccc(CO)c(F)c1 C12(NC(CC=CCC)=O)CCN(C(=O)Cn3ncn(C)c3=O)CCC1C2 c1(-n2ncc(C)c2)ccc(C(=O)NCC2C3CN(C(=O)C=CCO)CC23)cc1 c1(C(=O)NCCN(C(=O)CCOCC(F)(F)C(F)F)C)cnc(Cl)cc1N N1(C(C(CCSC)(C)C)=O)CC2CC(C1)CN(C(c1cc(Cl)cn1C)=O)C2 CC(F)(F)C(C)(C)C(=O)NCC1CN(C(=O)CC2CCCC(O)C2)C1 C1(C(=O)NCCC(C)(C)NC(c2cccc(SC)c2)=O)CN2CCC1(C)C2 C12(C(=O)NC34CC(NC(COCC(=C)C)=O)(C3)C4)CCCCC1C2 c1(C(=O)NC2C(NC(Cc3cc(C)ns3)=O)CCOC2)cc2cccn2cn1 C(=O)(C(C)(C)CN(C)C(=O)NCC1CC1CF)NCC c1(C(N(C2CCN(C(C(N3CCC(C)C3)=O)=O)C2)C)=O)c[nH]c2cccc(F)c12 Cn1cccc1C(=O)NCc1nc(C(=O)NCC(c2cnc[nH]2)O)co1 C1(C(C)NC(c2ccncn2)=O)CCN(C(=O)CC2CC(C(C)(C)C)C2)CC1 c1(C(N(C(C)C)CC)=O)cc(C2CCC2)no1.c1(C=O)cnn(C(C)C)c1 CC1CN(C(C2CCCNC2=O)=O)CC1NC(c1ccncn1)=O N1(C(C(C=C=C)C)=O)CC(C(=O)NCC2(CC(=O)OC)CC2)C2(CC2)C1 c1(CC)ncc(C(N2CCC(C(C)C)C2)=O)cn1.C(c1cnc[nH]1)=C(C(=O)N)C C1(CC=C)(NC(=O)CC(C)C(C)C)CCN(C(C2CC(C(C)C)=NO2)=O)CC1 c1(N2C(C(=O)Nc3ccnc(C)n3)CC(F)(F)C2)ncc2c(n1)CCC2 C1(CNC(C2C(C)OC(=O)N2)=O)CN(C(c2csc3nnsc23)=O)C(C)(C)C1 C1(C(N2CCC(CNC(C3C(C)CC3)=O)(CO)C2)=O)CCc2cnnn2C1 CC1CC(C(=O)NC2CC(NC(=O)CCCSC(C)(C)C)C(O)C2)CCN1C c1(C(=O)NCC(CCOCC)NC(=O)CSCC)ncnc(C)c1C.O C(C(C)C(=O)NOCC1CCNC1=O)NC(c1c(OCC)ccs1)=O C#Cc1ccc(CC(=O)NCC(CNC(=O)C(C2CCC2)C2CCC2)CO)cc1 c1(CC)nn(C)c(CC)c1C(=O)NC1CC(Nc2cncc(Cl)n2)C12CCC2 CC1C(NC(=O)C(c2cccc(F)c2F)F)CCCN1C CC1CN(C(C2(CO)CC2(F)F)=O)CC1C.c1(C=O)ccncc1C(F)(F)F N1(C(C2=NOC(c3ccc(C)cc3)C2)=O)CCC12CCOCC2 CC(=O)CCCC(=O)NCC12CCC1CN(C(=O)Cc1cc(C)nn1C)C2 CC1C(NC(c2csc(Cl)n2)=O)CCCN1C(=O)CC(F)(F)F c1(C(=O)NCC2CN(C(COC)=O)CC2O)ccc(C#N)cc1 C(c1ccc(O)cc1)=CC(=O)NCCCC.C1(C(C=O)O)CCS(=O)(=O)CC1 c1(C(=O)NCC2(CO)CCN(C(C(COC)O)=O)CC2)c2c(nn1C)CCSC2 C1(CC=C)(NC(=O)COCC=O)CCN(C(C2CC23CC(O)C3)=O)C1.N c1(C(=O)NC(C(C)(C)NC(C(=O)NCC)=O)C)cc(Br)c(C)cn1 C(=O)(C(F)CCC(C)C)N1C2CN(C(c3c(OC)cccn3)=O)C(C2)C1 N1(C(CCC=CCC=C)=O)CCCN(C(=O)C(=O)C(C)C)C(C)C1 CC(C)CC(C(=O)N1CC2(CC(NC(=O)COC3CCOC3)C2)C1)C(N)=O c1(C(=O)NCc2ccc(C(=O)NCC3(O)C(C)CCC3)s2)cc2ccccn2c1 C(C(C)(C)CCCO)NC(CC(CC)N(C)C(c1cnc(Cl)n1C)=O)=O c1(C(=O)NC2CN(C(=O)C(O)c3ccco3)CC2O)cccc2[nH]ncc12 N1(C(CC(CNC(=O)C(C(C)OC)N(C)C)OC)=O)C2CCC1CN(C)C2 n1(CCC(N2CC(COC)C2)=O)cccnc1=O.C1(=CC=O)CCSCC1.C C1(C(N2CCN(C(CC)C)CC2)C(=O)NC)CC12CCOCC2 N1(C(CC(CC#C)NC(=O)C(C)(F)CCCC)=O)CCCC(C#C)CC1 C(c1ccc(F)cc1F)=CC(=O)NCc1cccc(F)c1Cl C(CN=c1ncc(Cl)c[nH]1)N1CCN(C(c2scnc2C(F)F)=O)CC1 c1(C(=O)NC2C(OC)CN(C(=O)CCC(N)=O)C2)cc2cc(Cl)ccc2s1 C1(C(=O)NC(c2nc[nH]n2)CC)CCN(C(=O)CCN(CC)CC)CCO1 C(C(C)(C)C(=O)N1CCOC(O)C1)N(S(=O)(=O)CCCl)C c1(NCC2CC(NC(c3cn(C)cc3C(F)(F)F)=O)C2)ncnc(Cl)c1C#N CCC(C)C(O)CC(=O)NCC(C(=O)Nc1cnn2cccnc12)N(C)C Cc1cc(C(=O)N(CCCNC(=O)C(C)CC2CC2)CCO)cc(O)n1 N1(C(c2ccc(CC)[nH]2)=O)CCOC(C2CN(C(=O)C(C)OC)C2)C1 C(=O)(C(O)CC(C)C)N(CCCCCC)CCNC(C1COCC1(C)C)=O CC1CN(C(=O)CC(c2ccc(F)cc2)C)Cc2[nH]ccc21 C1(C(N2C(CC)CC2)=O)CN(C(=O)CCCCC(C)C)CCC1(C)C C1(CN(CCCN(C(C2C(CCC)CCC2)=O)C)C)CCN(CCOC)CC1 C(=O)(C1=C(Cl)CC1)NC(C(=O)NCC(COCC)C)C1CC1 N1(C(COC(C(OC)OC)=O)=O)CCCC(C(=O)Nc2ccccc2F)C1 c1nc2c(s1)CN(C(=O)C1=CSCCO1)CC2.c1(C(=O)NC)ncoc1C1CC1 N1(C(CCNC(CC(CC)C)=O)=O)CC(C)(C)C2CCCC12 N1(C(C=CS(CC)(=O)=O)=O)CCC2(CC1)CN(C(C1(C)CC1(F)F)=O)CC2CO c1(SC)cncc(NC2(c3nnnn3C(C)C)CCC(C)C2)c1 N1(C(c2scc(C)n2)=O)CCN(C(c2ccc(N(C)C)nc2)=O)CC1C(F)(F)F c1(NC)ccc(C(=O)OCCNc2ccccc2C)nc1 CC1CN(C)CC(C(N2CCC(C(N3CCCSCC3C)=O)(CF)C2)=O)O1 N1(C(C2CCCN(C)C2)=O)CCC(CNC(c2coc3c2COC3)=O)C(O)C1 N1(C(c2n(C(CC)C)ncc2)=O)CC2(CCN2C(=O)C(F)C2CCOC2)C1 C1(CC(=O)N)COCCN1C(c1ccc(O)cn1)=O.C1(C(=O)OC)(C)CC1 c1(CC(=O)Nc2ccccc2CO)ccccc1C(N1CCCCC1CCO)=O c1(C(=O)NC(C2CCCCC2)CNC(=O)CC2CSC2)cc2ccnn2cn1 c1(C(=O)NC(C(=O)NC(C=C)(C)C)CCOC)cnn2c1OCC2.C(C)=O c1(CC)oc(C)cc1C(N1CCC(CCNC(C2(C)CC2(C)C)=O)C1)=O N1(C(C(CN(C)C)O)=O)CCOCC1CCNC(c1ccnc(C(F)(F)F)n1)=O CCCCC(O)C(=O)NC1CCN(C(=O)CCOc2cccc(C)c2)C(C)C1 C1(NC(CC(C)c2cnn(C)c2)=O)CCN(C(c2cnc(Cl)cc2N)=O)CC1O c1(C(N(C2CCN(C(C(CC)N(CC)CC)=O)C2)C)=O)cnc2ccccc2n1 C1(C2CCN(C(=O)Cc3ccoc3)CC2)(CNC(CC(CC)O)=O)CCOCC1 c1(N(C)Cc2cnc(C)s2)nc(N2CCC(F)(F)C(F)C2)c2c(n1)CCC2 O=C(CCCCC(F)F)NC(c1ccccc1)CNC(c1cnc(O)c(F)c1)=O C1(CCNC(c2c(C)n(C)nc2)=O)C(C)CCCN1C(C1CC2(C1)CC(F)C2)=O C12(C(N3CCCC(NC(C4C(COC)C4)=O)C3)=O)C3C4C1C1C2C3C41 N1(CCCCNCC#C)CCN(C(c2nc(Br)sc2C)C(=O)NCCOC=C)CC1 C1(NC(C2CCN(C(C)=O)C2)=O)CCN(C(c2cc(C)nc(O)c2)=O)CC1(C)C c1(CSCC(=O)NC(C(C)NC(CCN(C)CC)=O)C)ccccc1 CC1CC(C(=O)NCC2(NC(=O)C=Cc3cn(C)cn3)CC2)CCC1C c1(C(N2C(CCNC(=O)CCc3cnn[nH]3)CCC2)=O)nc(C2CC2)ncc1Cl Cc1ccnc2c(C(N3CC(N(C)C(C4CC5CC4C4CC54)=O)C3)=O)cnn12 c1(C(=O)NCC(CC)NC(=O)CCc2cn(CC)nn2)ccc2ocnc2c1 CC(=O)CCC(=O)N1CC(=O)CC1C(=O)NC(C)C(C)n1cccn1 CC1(C)CC(C(N2CC(Cc3ccoc3)C2)=O)CCN1C(=O)CN1CC2CC2C1 S(=O)(=O)(c1ccc(NCC2(F)CCOCC2)c(Cl)c1)N(C1CCSC1)C Cc1ccc(-c2cc(C(=O)NCCC(C)N(C)C(c3cncnc3)=O)n[nH]2)s1 N1(C(CNC(CC(C)C)=O)=O)CC(CNC(C2CCO2)=O)C2(CC2)C1 c1(C(=O)NC(CNC(C2(C)CCN(C)C2)=O)C2CC2)ccc(O)c(CO)c1 C(C(CCNC(=O)Cc1cc(C)ns1)OC)OC c1(SCC(=O)NC2CC(N(C(C(C=C)O)=O)C)C2)ccc(F)cc1F N1(C(CN(CC)CC)=O)C2CC=C(C(=O)NC3CN(C)CC3C)C1CC2 N1(C(c2ccc(C(N)=S)cc2)=O)CCC2(CC1)CC(NC(C13CC(C1)C3)=O)C2 CC(C)(C(O)C(F)F)NC1CCCC(CNC(=O)OC(C)(C)C)C1 c1(C(=O)NCC(C)CC(=O)N2CCCCC2C)nccc2cc[nH]c12 N1(C(C(CCC)OC)C(=O)NCCCOC)CCC2(CC1)CC(O)CO2 N1(C(c2ccc(COC)[nH]2)=O)CC(COC)CC1.C(=O)C(O)CCN(C)C C(=O)(C1=CCC(C)(C)CC1)NC(CC)CCCC(=O)NC(CO)CCOC C(C1CN(C(=O)C2=C(C)CC2)CC1C(=O)NCC1CCCN1C)=CC N1(C(c2cccc(CO)c2)=O)CC2CCN(C(c3nc(Cl)sc3Cl)=O)C2C1 CCCC(C)(CCC)C(=O)NC1CCN(C(c2cc3oc(C)cc3[nH]2)=O)CC1C c1(OC)cc(OC)cc(C(=O)Nc2c[nH]nc2C(=O)Nc2nc(C)ccc2Br)c1 N1(C(C2CCC(COC)C2)=O)CCCC1(C)C.C1(CC=O)CC2(CC2)C1.C CCCCC(C(=O)NC1(C)CN(C(=O)CC2CCCCN2C(C)=O)C1)C(C)C C1(C(N(CCNC(CNC(C(CC)C)=O)=O)CC)=O)CCCC(N(C)C)C1 N1(C(c2c(C)nco2)=O)CC2C=CC1C(C(=O)Nc1csnc1C(C)C)C2 C1(C2CCCN(C(c3cc(C(N)=O)nn3C)=O)C2)(NC(c2cc(C)sc2)=O)CC1 N1(C(CC=C=C)=O)CCC(C)(C(=O)N(C)Cc2cccc(C)c2)C1 C1(C(=O)NC(CC)CO)CC2(CC2)CN1C(=O)CCOc1ccc(F)cc1 Cc1nnc2n1CCC(C(N1CCOC(C3CCC3)C1)=O)C2 C1(NC(c2c(CC)ccc(O)c2)=O)CCCC12CCN(C(c1cocc1C)=O)C2 C(=O)(C(C(C)O)N(C)C)N(C1CCN(C(=O)Cc2sc(O)nc2O)C1)CC C#Cc1cccc(CNC(C2CN(C)CCN2C(=O)CCOC(C)C)=O)c1 c1(CNC2CC(C(=O)NCCCCC#C)C2)ccc(F)cc1Cl CC1CCN(C(c2ncc(F)cn2)=O)CCN1C(C1CC(C2CC2)=NO1)=O N1(C(C2CN(C(C)=O)C2)=O)CCN(C)CC1CNC(=O)C(O)CN(C)C CC(C)CC(C(=O)NC1CCC2(CC1)N=N2)NC(=O)C(O)CC(N)=O C1(CNC(CN2C(C)CCC2)=O)CC(F)(F)CN1C(C1CS(=O)C1)=O C1(CN(C(=O)C(C)c2ccsn2)CC)CCOC1 N1(C(=O)OC(C)(C)C)CCC(C(=O)O)(C)CC1.C1(C(=O)O)OC2CCC1C2 CC(CC(=O)NCCCC1CCN(C(C2Cc3nncn3C2)=O)CC1)C(F)(F)F N1(C(C(C)Oc2cccc(Cl)c2)=O)CCN(C(=O)C2=CC(C)(C)C2)CCC1C c1(C(=O)NCCCNC(c2nc(C)[nH]n2)=O)cnc2n1CC(C)CC2 CCC(CCC(=O)NCC(C1CCCCC1)NC(=O)CC(C)(C)COC)OC c1(N2CCN(CCC(C)C)C(=O)C2)nc(=N)[nH]c(=Nc2ccccc2)[nH]1 n1(CCC)cc(C(=O)NCCCNC(C2(C)CCC(=O)N2)=O)c(C)n1.O Cc1c(NC2C=CCCC2)ncnc1N1CCCC(COC(F)F)C1 N1(C(c2c(OC)c(C)sc2)=O)CC2CCC(C2)C1.c1(C(=O)N)c[nH]cc1C1CC1 C1(C(N2CCC(C(C)C)C2)=O)CCCCC1CNC(=O)CC(=O)N(C)C C(=O)(CC(C)(C)C(F)(F)F)N1C(CNC(c2ccc(C(C)C)o2)=O)CC1 N1(C(C2C(C)CN2C(=O)CC2CC3(CC3)CO2)=O)CCCC(C#N)C1 Cc1c(C(=O)N(C2CN(C(=O)C(C)c3cccs3)C2)C)ccc2c1NC(=O)C2=O CC1CCN(C(=O)CN2CCNC(=O)C2)CC1N(C)C(c1nc(Cl)ccc1N)=O C(=O)(NN(Cc1ccccc1)C=O)OCC(CC(C)O)(C)C.C(=O)C(F)(F)F.N S(=O)(=O)(c1cc(C)cnc1NC)NCC(CC)(CC)N.C1CCC(=O)NC1C C1(C=O)CS(=O)(=O)CC12CC2.Cc1noc(N)c1C(N1CCCC1)=O.C(C)O c1(CNC(c2c(NCc3n(C)ncc3)cccn2)=O)cccc(F)c1Br c1(-c2nc(CCN(C)C)nn2C2CCSC2)cc(Cl)nc(Cl)c1F CC(C)C(C(=O)NC1CCCC2(CCC2)C1)C(C)NC(C12CC(F)(C1)C2)=O c1(C(=O)N)cc(F)cc([N+](=O)[O-])c1N.C(CC(C)C(C)C)NC(C(C=C)(F)F)=O Cc1cc(C)c(C)c(S(=O)(=O)N2Cc3ccc(NC(=O)C(N)CN)cc3C2)c1C C=Cc1cncc(C(=O)NC23CC2CN(C(=O)Cc2cnc[nH]2)C3)c1 c1(C(=O)NC2(c3ccccc3)CN(C(C(C)SC)=O)C2)cc2sccc2n1C Cc1ccc(C(=O)NC2CCCC2NC(=O)CS)cc1.c1nncn1C(C)C c1(CCC)nccn1CC(=O)N(CC(C)NC(c1csc(Cl)c1)=O)CC c12ccc(cc1)CNC(=O)NCCCN2.C(CC(C)(C)C)C(C)(C)OC N#CC1Cc2cccc(C(=O)NCC3CCCN3C(=O)CCC(N)=O)c21 c1(C(=O)NC2(CCC)CCCN(C(C3CC3C)=O)C2)ccc2cc(C)oc2c1 CN1C2CCC1CC(C(=O)OCCCC(=O)NC(C1CCC1)=O)C2 Fc1cc(Cl)cc2c1CN(N1CCCC(c3ccc(Cl)cc3)C1)CC2 Cc1ccc([N+](=O)[O-])c(N2CCOC(CNC(c3onc4ccccc34)=O)C2)c1 C1(CNC(C(C)(C)F)=O)COCCN1C(c1ccc(SCCCO)cc1)=O CCCCC(=O)C(=O)NCC12CC1CN(C(=O)Cc1cccc(F)c1F)C2 N1(CCNC(C2(SC)CN(C(C(CC)OC)=O)C2)=O)CCC(O)CC1 CCC(C(=O)NCC(CCNC(=O)CCc1ccncc1)OC)n1ccnc1 N1(C(c2cncn2C)C(=O)NCCCSC)C2CCC1CN(c1ccccc1)C2 N1(CC=C)CCN(C(C2CN(C(C3CCC=CCC3)=O)C2)=O)CC1 CCC(C)C(O)CC(=O)OCC(N1CCN(c2cccc(Cl)c2)CC1)=O C=CC1OCCCC1C(=O)NCCOC1CN(C(C2(C(N)=O)CCC2)=O)C1 C1(NC(c2cnc(CC(C)C)[nH]2)=O)Cc2ccccc2N(C(C2CSC2)=O)C1 C#CCC(CC#C)C(=O)NC(c1ccccc1Cl)C.Cc1cccc(C)c1N=O C1(NC(c2c(C(C)C)nco2)=O)CCC(C)N(C(=O)C#CC(=O)N(C)C)C1 c1(C(=O)NCC2(C)N(C(C(C=C)O)=O)CCC2)c(O)nnc2c1CCCC2 C1(C(=O)NC2(C#C)CCCCC2)CCN(C(c2cnn3c2CCC3)=O)C(C)(C)C1 c1(C(=O)OC2C(NC(C)=O)CCCC2)cc(Cl)cc(OCc2ccccc2)c1O Cc1ncc(C)c(=NC(C)C2CCN(C(C3(F)CCCC3)=O)CC2)[nH]1 C1(NC(CCn2ncc(C)c2)=O)Cc2ccccc2C1NC(c1coc(Cl)c1)=O C=CC(O)(C(=O)NC1CCN(C(c2cc(C)c(O)nn2)=O)C(C)C1)C(F)(F)F c1(CC)cc2c(NCC(O)CNC(c3cccc(OC(F)F)n3)=O)ncnc2s1 C1(CC(=O)CCCC2(NC(=O)CN3C(=O)CNC3=O)CCC2)CCCC(O)C1 C1(CN(C)C(C2CC2c2ccoc2)=O)COCCN1C(=O)C=Cc1cnc[nH]1 c1(C(N2CC(OCCNC(C(C)=C3CC3)=O)C2)=O)cc(C)cc2c1CCC2 C1(C)(C(=O)NCCn2c(C)nnc2)CC(O)CN1C(=O)Cn1nccc1C N1(C(C(CC=C)OC)=O)CCC2(CC1)CC2C(=O)N(CC(=C)C)C1CC1 c1(C(=O)NC(CC(C)NC(C=NOC)=O)C)c(F)ccc(OC)c1OC C1(COC)CCOCCN1C(=O)NCCc1c(F)cccc1Cl c1(C(=O)NCCN(C(CS(C)(=O)=O)=O)C2CCCCC2)cnn2c1NCCC2 C(N=c1cc(Cl)c(O)n[nH]1)C12CCC(NC(C3C(OC)CCC3)=O)(CC1)CO2 C=CCCC(CC(C)C)C(=O)N1CCN(C(=O)CC(N2CCCCC2=O)C)CC1 C(N=c1[nH]c(=NCC2(C)CCOCC2)c2cccc(F)c2[nH]1)C1CC(C)SCC1 N1(C(c2nc(CC)sc2N)=O)CCC(NC(=O)C(C)N(C)C)C(C)(C)C1 Cc1ccc(CC(N2CC(O)CC2C(=O)NCC(=O)OC(C)(C)C)=O)cc1C C(=O)(CCC(=O)C(C)(C)C)N1CCC(N(C)C(C2CCC(CO)CC2)=O)CC1 C(=O)(C1=C(C)CCCC1)NCC1C2CN(C(c3nccc(C#C)c3)=O)CC21 c1(C(=O)NC2CC(CNC(c3nc(CC)sc3)=O)C2)cc(Cl)ncc1Cl N1(C(CN(S(C)(=O)=O)C)=O)CCOCC(NC(=O)CCCC(F)F)C1 CCCCC(C)CCC(=O)NC(C)CN(C(c1[nH]nc(OC)c1Cl)=O)CC Cc1ccc(CNC(=O)CC2CCN2C(=O)C2CC2)s1 C(=O)(C#CC(=O)NC1CCC(N(C(=O)CCc2cnc(O)[nH]2)C)C1)N(C)C CC1CC(C(=O)NC(C)(C)CCCNC(=O)C(C)(C)c2cccs2)CCO1 C1(OC)CN(C(C2CCCN2C)=O)CC1NC(c1c(C)c[nH]c1CC(N)=O)=O c1(C(=O)NC2CCN(C(c3ccc(C)cc3I)=O)CC2)cn2ncccc2n1 c1(CC)nn(C)cc1CNC(=O)C=CCNC(=O)CC1CCOC1 c1(C(=O)NCCN(C(C(N2CCC(O)CC2)C)=O)C)nn(C)cc1N.C1CC1 N1(CCNC(c2ccccc2F)=O)CCNC2CS(=O)(=O)CC12 N1(C(C(C)C)=O)CCC2CN(C(c3ccnc(C(N)=O)c3)=O)CC12 CCC(CC)(CCNC(c1cncn(C)c1=O)=O)NC(=O)CC1CC2C=CC1C2 C1(NC(C2(C)CC2)=O)CN(C(c2cnn(CC3CCCCO3)c2)=O)CCC1(C)C C(=O)(CC(C)CC(=O)N1CCCC(F)(CNC(=O)CC)CC1)OC.C(C)=O.N CC1CCCC=C1C(=O)NCC(C)(C)CNC(=O)CCN1CCC(F)C1 N1(C(C2=C(C)CCC2)=O)CC2CCCC(NC(C3CC34CCOC4)=O)C2C1 C(=O)(C(C(C(C)CC)OC)N1CCC(C)(OC)CC1)NCC1CCCN(CC)C1 N1(C(CCOCCOC)=O)CC2(CCC2NC(c2cncn(C)c2=O)=O)C1 Cc1cc(NC(=O)NCCCOC2CCOCC2)cc(CN)c1.C1CC1 C1(OCCC)CCCCC1C(N1CCC(CCNC(=O)C2=CCC2)CC1)=O C(CN=[N+]=[N-])(C(=O)NCc1ccccc1)NC(C(C)C1(O)CCC1)=O c1(NC(C2C(CNC(c3cc(C(C)C)on3)=O)CCC2)=O)cccc2[nH]ncc12 C1(NC(C2CCC(CC)O2)=O)C2CN(C(=O)CCN3CCN(CC)CC3)CC12 C1(C(C)C)(CO)CCN(C(=O)CONC(=O)C(C)C2CCOC2)C1 c1(-c2cn(C(C)C(=O)N(C)CC3CCCC3)nn2)ccc(S(C)=O)cc1 Cn1cc([N+](=O)[O-])cc1C(N1CC=CCC1)=O.c1(C=O)cc(C(C)(C)C)n[nH]1.N C(=O)(C(CO)NC(=O)CNC(=O)C(C)(C)C)N(CCCC)C c1(C=O)cc2c(Cl)cccn2n1.N1(CC)CC(C(=O)NC(C)(C)CC)NC1=O.N c1(C(N2CC(CC)C(C(N3CCC3C(N)=O)=O)C2)=O)cc(C)nnc1C c1(Cn2cc(CC(C(=O)O)C(=O)CCC3CC3)nn2)cc(Cl)c(F)cc1Cl C1(C(=O)NC(C)CN2CCCC2)(CO)CCN(C(C2CC3(CCC3)C2)=O)C1 c1(CNC(=NCc2ccccn2)NCC2CCCO2)nnc2n1CCOC2 N#Cc1n[nH]c(=NC2CC3CN(C(=O)Cc4cccc(C(F)F)c4)CC23)s1 c1(OC)c(CN2CCC(CO)(NC(c3ccc(Br)cc3Cl)=O)CC2)cccc1Cl CC1C2C(CCN2C(C2CCC3(CCCC3)C2)=O)CN1C(=O)CCCNC(N)=O c1(CN(C(C2(c3cccs3)C(C)C2)=O)C)ccc(Cl)nc1 Cc1ncc(N)cc1C(=O)NC1CN(C(=O)C(=O)NCCC(N)=O)CC1C c1(C(N2CCC(N(CCO)C(c3cccnc3)=O)C2)=O)cccc(I)c1 c1(C(=O)NCCCOCCNC(C2CC(C)C2)=O)ccc2occc2n1 N1(C(C(C)(C)C2CCC2)=O)CCC2(CC1)COC(CNC(C1CCCOC1)=O)C2 c1(COCC)ccc(Cn2nccc2)cc1.C1(C)(C)C(=O)N1.c1ccccc1 c1(CCC)cc(C(=O)NC(C)C(C)(C)NC(=O)CCCc2csc(C)n2)no1 N1(C(c2cc(C)no2)=O)CCN(C(c2ccc(OC(F)(F)F)cc2Br)=O)C(C)C1 c1(C(N(C)C)=O)ccc(F)c(-c2cncc(F)c2C(=O)NCCCS(C)(=O)=O)c1 c1(OCC(=O)NCCC2(O)CN(C(C(C)c3cccs3)=O)C2)ccc(Cl)nc1 c1(C(=O)NC(c2occ(C(NOC(C=C)C)=O)n2)C)ccc(=O)n(C)c1 Cc1onc(O)c1C(=O)NCCCC(C)(C)NC(c1cc(=O)cc[nH]1)=O c1(C(N(CC)C2CC2)=O)cc(C)[nH]n1.C1(C(C(=O)N)OCC)CCCOC1 Cn1cc(Cl)c(C(=O)NC2COCC2NC(=O)CC(O)c2ccccc2)n1 CCCS(=O)(=O)CC(=O)N1CCC(NC(c2ncn(C)n2)=O)CC(O)C1 Cc1cc(C(=O)N(C2CCN(C(c3cnc(S)n3C3CC3)=O)C2)C)cc(C)c1C C=CCC(C)C(=O)N1CCC(CNC(=O)C(C(C)C)C2CCC2)(OC)C1 S(=O)(=O)(c1cc(C=CC(=O)OC)ccc1OC)N(CCc1cccs1)CC C(C1CCCCCC1)=CC(N1CCC(N(C(=O)C(C)Cn2cccn2)CC)C1)=O CC1N(C(=O)C(CC(F)F)NC(=O)CN2CCCCC2)CCOC1(C)C S(=O)(=O)(c1cc(Cl)c(Br)cc1F)N1CCCC(F)(F)C1.C(=O)(CC(=O)NC)OC C1(C)(CC)CC(NC(C2(C#N)CCCCC2)=O)CN1C(=O)Cc1cc(C)cs1 C(C(CC(=O)NCC1(C)CCCC1O)NC(=O)C(C1CC1)SC)OC O=C1CCC(C(=O)N2CC(NC(=O)C)C3(CC3)C2)=NN1.c1(C=O)cscn1.N N1(CC(N2CC(CC(C)NC(=O)C(F)CC3CCCC3)C2)=O)CCN(C)CC1 C1(COC)CN(C(c2ccc(C(F)(F)F)o2)=O)CCN1C(=O)C(O)CCSC c1(CC(=O)NCCOCCCNC)cccc(O)c1.c1(C2CC2)cncn1C C1(C(NOCCCC#C)=O)CC(NC(C2CC(=O)C2)=O)C1(C)C Cc1cnn2ccc(C(=O)NC3CC(CO)N(C(=O)CC4(C)CC4)C3)nc12 C12(C(=O)NCC(C)CNC(=O)C(O)C3CCCC3)CCCCC1C2 n1(CC)c(C(=O)NC2(CO)CN(C(c3ccccc3OC)=O)C2)cnc1O N1(C(=O)NCC2CC(C(C)(C)C)C2)CCN2C(=O)C(N)CC2C1 C1(NC(=O)COC2CC2)CCC(CC(N2CCCC2COCCO)=O)C1 C1(C)(C(=O)NCC2(O)CC(NC(c3c(CC)ccs3)=O)C2)CCCN1C Cc1cc(C(=O)NCCOC2CN(C(=O)CC=C(Cl)Cl)C2)sc1Cl C1(NC(=O)Cc2ccno2)COC2(CCCN(C(=O)CCc3ccccc3)C2)C1 C1(C(N2CCC(C(C)(C)NC(C3OCCN(C)C3)=O)C2)=O)C2CCC3C(C2)CC13 C12CC1CN(C(=O)C=Cc1ncc[nH]1)C2.C1(OCC)CC(CC(=O)N)C1.C c1(C(N(CCCNC(=O)CCF)C)=O)cscc1C(F)F c1(C(N2CCC(F)CC2)C(=O)NCCC2(C)CC2)ccc2c(c1)CCO2 c1(C(N(CCC)C)=O)cnc2c(c1)CCCC2.C(=O)(C(C=O)C(C)C)OCC.N N1(C(CNC(N)=O)=O)CC2CC1CN2C(c1ccc(F)c(I)c1)=O C1(N(C(C(Cc2ccccc2)NC)=O)C)CCCN(C2CC2)C1=O C1(CNC(C2(F)CCN(C(C3OCCC(=O)C3)=O)C2)=O)C2CCCCCC12 C(=O)(C1CCCn2c(C)nnc21)N1CCC(NC(c2c(C)ncn2O)=O)C1C N1(C(CC2C(=O)NC(=N)S2)=O)CCC(NC(c2ccnc(C(F)F)n2)=O)C(O)C1 c1(CC(=O)NC2CCN(C(c3cnc(SC)nc3)=O)C2)c(F)cc(F)cc1F c1(C(N(C(C(=O)NC2CCN(CCOC)C2)(C)C2CC2)C)=O)ncncc1N C1(CNC(C(Cn2ccc(C)n2)C)=O)COCCN1C(=O)CCc1ncc(C)[nH]1 C1(N(C(CS(CC)=O)=O)C)CCN(C(c2nsc3ccccc23)=O)CC12CC2 C1(NC(=O)CCOC2CCNC2)CCOC2(CCNCC2)C1 c1(N2CCN(CCOC)CC2=O)cc(Cl)nc2c(C)c(C)nn12 NS(=O)(=O)c1ccc(C(=O)NC2CCCC2NC(c2ncc[nH]c2=O)=O)o1 C1CCCOC1C1CCN(C(c2ccc[nH]2)=O)CC1.C(C(=O)N)NC(=O)C1CC1 C(=O)C1=CNS(=O)(=O)N=C1C.C1(C(=O)N)(CC)CCNC1=O.C1CCOC1.C C1(C(=O)NCc2cc(C)sc2)CC2CCC1N2C(=O)CC1(O)CCCCC1 CC1CCN(C(=O)CSCC2CCCO2)CCN1C(c1cccc(N)c1F)=O C=CCC(CC)C(=O)N(CC(Cc1ccccc1)NC(C1(CO)CCCC1)=O)C c1(C(=O)NC2C(NC(C(CC)C)=O)CC2)c(C)cc(OC)cc1C Cc1cc(NC(C2(CCNC(=O)C=CC(C)C)CC2)=O)cc(C)c1F Cc1cccc(O)c1NC(=O)CC1CC(NC(C2CCCN(C)C2)=O)C1 CC1=C(C(=O)NCC(C)(C)OCC(=O)NCC(O)CN(C)C)CCC1 c1(OC(C)C(=O)NCCc2cn(CCCF)nn2)ccc(F)cc1F C1(NC(c2c(C)ncn2O)=O)CCCN(C(C2CCCN2C(C)C)=O)C1C C(=O)(CCC(CC)CC)N1CCCC(F)(CNC(CC=CC=C)=O)C1 N1(C(c2cn(C)nc2)=O)CC2(CCC(NCc3ccsc3Br)C2)C1 n1(CC)ncc(C(=O)NC2C3CC2N(C(c2cc(OC)nn2C)=O)C3)c1Cl c1(CC)[nH]ccc1C(=O)NCC1(F)CCC1.c1(C=O)cn[nH]c1.C1CCC1 N1(C(C2(NC(C)=O)CC2)=O)CC2(CCN(C(C3CCC(C)(C)O3)=O)C2)C1 C1(NC(c2cc(OC)n(C)n2)=O)CCOC2(CCN(C(=O)CC(C)(C)O)CC2)C1 Cc1nn(C2CC2)c(Cl)c1C(=O)NCc1ccccc1.C(=O)C(=O)N(C)C c1(CNC(C(c2ccn(C)n2)C)=O)nnnn1CC1CCCO1 C(=O)(C(C)(C)S(C)(=O)=O)NCC(CCCC)NC(=O)CC1(C)CCCO1 C1(C(=O)NCC2CCC(NC(COCCC=C)=O)CC2)CCc2ccccc2C1 CC(CC(N)=O)C(=O)N1CC2CC2C1.C1(C=O)CC(=O)N(C(C)C2CC2)C1.C CC(O)C(C)(C)C(=O)N1CC(N(C(=O)CCC(F)(F)F)C)C(C)(C)C1 C=CCC(C)(CC=C)NC(C12CC(CO1)N(C(c1cc[nH]c1C)=O)C2)=O C1(CCNC(c2c(C)nn(C)n2)=O)CCCN(C(C2CCC(C)(C)C2)=O)CC1 C1(C(N2CCC(CC=C)(NC(c3ccsc3)=O)C2)=O)CC12CC(F)(F)C2 Cc1cc(C(N2C3CCC2CC(N(C(=O)C#CC(C)C)C)C3)=O)cc(N)c1O N1(C(c2ccc(C)c(C)n2)=O)CCC2(CC(C(=O)N3CCOCC3)=NO2)C1 c1(C(N2C(CNC(C(C)N(C)C)=O)C(C)CCC2)=O)cnc2[nH]cncc1-2 c1(C(c2n(CC)nnn2)NCC2(COC)CCC2)ccccc1.N(C)C.C Cc1cccnc1C(=O)NCC1CC2CC2N1C(C1CCC1(F)F)=O c1(CC(=O)NCC2CC2NC(C2CC23CC(O)C3)=O)cn2ccsc2n1 C1(C(=O)NC(C)C(F)F)C2CC2CN1C(=O)C1=COCC1 c1(NC(C2(C#C)CN(C(=O)C(C=C)OC)C2)=O)ccc(F)c(O)c1 C1(C(N(C(Cc2c(C)ccc(C)c2)=O)C(C2CCC2)C)=O)CCCCC(F)(F)C1 C(CC(C)C(=O)NC(Cn1cccn1)C(=O)NC1CCCOC1)=CC c1(C(=O)N)cc(O)ncn1.c1(CC(CNC(C2CC2)=O)N(C)C)ccccc1 Cc1cc(CC(=O)NCC(O)CNC(c2csc(C(C)C)n2)=O)ccn1 c1(COC)cnc2[nH]cnc(NCC34CC(C3)C(C)(C)O4)c1-2.C(=O)CC C1(CNC(CC2N(C(CCCn3c(C)ncc3)=O)CCC2)=O)(CO)CC2CC2C1 C=CCCC(CC(C)C)C(=O)NC(C)C(C)n1cccn1 CC1(C#CC(=O)NC2COCC2C)CC1.c1(C=O)c[nH]cc1-c1ccc(Cl)s1.N N1(C(C(C)(CSC)NC(C=C(CC)CC)=O)=O)C2CCC1CN(C)C2 c1(N(C(C23CCC(C#C)(CC2)CC3)=O)C2CC2)cc(OC)c2ccccc2n1 c1(C(=O)NCc2cc(C(=O)NC3CCC(CCCC)C3)no2)ccc(F)cn1 Cc1ccc(CC(N2CCCC(CNC(=O)CN3CCOCC3=O)C2)=O)cc1O CCC(CC(C)C)C(=O)NCC1C(CC)CCN1C(=O)CCC1CC1C c1(CC(=O)NCCCn2cc(CCN(C)CCO)nn2)ccccc1CC(N)=O c1(CNC(=O)C(N2CCC(F)C(F)C2)=O)cc2c(s1)CCCC2 C1CN(C(=O)C(Cc2ccsc2)NC=O)CC1(C)C.CC=O.C(=O)(OCC)N c1(C(N(C2CCN(C(=O)CC3CC4CCC3O4)CC2)CCC)=O)c[nH]ccc1=N C1(CN(C(C2(CC#C)CC2)=O)CC)CCN(C(C2CC2(F)Cl)=O)CC1 C1(C(=O)NCCn2ccc(C(N(CC(C)SC)C)=O)c2)CC(C)CC(C)C1 N1(C(c2[nH]cc(CC)n2)=O)CCCC(NC(c2ncncc2N)=O)C1CC N1(C(C2C(CC)CCN2C(=O)Cn2cnnc2)=O)CC2CC3CC2C1C3 CC1=C(F)CN(C(=O)CC2CC2CNC(c2ccc(C)c(O)c2)=O)CC1 C1CC(C=O)C12CCC2.C(=O)(C=O)NCCOCCOCCOC.N C(N=c1ccnc(NCCc2cn[nH]c2)[nH]1)C1(C)CC(C)(C)C1 C1(CC(=O)NCC(O)COc2ccccc2)CCCC(C(F)(F)F)O1 N1(C(C(COC)Oc2ccccc2)=O)CC2CN(C(C34CCCC3C4)=O)CC2C1 C(C(O)C(=O)NCCC(O)C1CCC1)NC(=O)Cn1nccn1 C1(C(N2CC(NC(=O)Cc3ccccn3)(CO)C2)=O)CCCCC1O CC(C)CCCC(C)C(=O)NCC(C(C)C)NC(=O)CCSCC(N)=O Cc1ccc(C(=O)NCCCN2CCN(C(=O)CCCCCBr)CC2)c(F)c1 N1(C(C2N(C(c3c(C)cccc3O)=O)CCCC2)=O)CCCC2(CCNC2=O)C1 c1(CC(=O)NCCCN(C(=O)C(N2CCSCC2)C)CC)cn(C)nc1Cl C(C(CC(C)C)C(=O)N1CCC(n2cnnn2)C1)NC(c1c(CC)noc1)=O Cc1sc(C(N2CC(F)CC2CN(C)C(C2COC2)=O)=O)cc1[N+](=O)[O-] c1(CCC)ncoc1C(=O)NC(C)C1CC1.C(=O)C(C)C1CC1.C=O.N N1(C(C2(C)CCCO2)=O)CCC(F)(c2cn(CC3CCOCC3)nn2)C1 C1(CNC(C(=O)NCC)=O)CCC(F)C1.C(=O)CC(O)c1ccccc1.C C1(C(=O)NC(CCCC)CNC(c2ccc(Cl)cn2)=O)Cc2cncn2C(=O)N1 c1(OC)ccc(Cl)cc1C(F)(F)C=O.c1(C=O)ccn(C2CC2)n1.C1CC1.N c1(CCC(=O)N)cc(Cl)cc(Cl)c1.c1(NC(C2CC(C)OC2)=O)cccc(C)c1 N1(C(=O)NC(CC(CC)C)C)CCOC(CC)(CC)C1 N1(C(C2CN(C(C3(C=O)CC3)=O)CC2(C)C)=O)CCC(F)(F)C(C)C1.CN CN1CCC(O)(CNC(=O)CC2CC(NC(C3SCCS3)=O)C2(C)C)CC1 c1(CC(N2C(CCNC(c3cc(C)nnc3)=O)CCC2)=O)cc(Br)ccc1F CC(C)CCN=C(NCc1ccc(C(C)(C)C)cc1)NCC1CCCCO1 C(=O)(CCCC(C)(F)F)NC1C(C)N(C(=O)CCCN(C)C)CCC1 c1ccc(C#N)cc1.c1(CC)ncncc1C(=O)NCC(C)N(C(=O)C)CC CC1CCN(C(C2CCNC2=O)=O)CCN1C(c1cc(NS(C)=O)ccc1F)=O c1(C(N2CCC(CC(C)NC(=O)C(F)(F)CO)CC2)=O)cc(C2CC2)nc(Cl)c1 c1(CC(=O)NC(CNC(CC=C)=O)CC)cc(F)ccc1O C#CC1(O)CCN(C(=NCC(C)(C)Cc2ccccc2)NC2CCS(=O)(=O)C2)C1 Cc1conc1CC(=O)NCCN(C(C1CC1F)=O)Cc1ccccc1 c1(CC)[nH]c(=N)sc1C(N1CC(C(C)C(=O)O)C1)=O CC1(O)CC2(CN(C(C3CCN(C(=O)CCc4nc[nH]n4)C3)=O)C2)C1 C1(C2CC2)(C(=O)N)CCC1.C1(CC)CCN(C(C2CN(C(C)C)CCO2)=O)CC1 C1(C)(CC(=O)NC(CCNC(C2C(C)CCC2)=O)(C)C)CCCCCC1 C1(C(C)NC(C2ON=C(C)C2)=O)CCN(C(c2csc(-c3cn[nH]c3)n2)=O)CC1 c1(C(N(C(C)CCNC(C2CCC(C(N)=O)C2)=O)C)=O)ccc2ncnn2c1 Cc1cnc(O)c(NC(c2ncccc2NC(c2cn[nH]c2)=O)=O)c1 C#CCC(C)(C(=O)N1CCC1C(C)O)NC(c1ccc(C2CC2)cc1)=O c1(CC)c(C(=O)NCC(O)C)nnn1C.c1(C(=O)N)cncc(C(F)(F)F)n1 S(=O)(=O)(c1ccc(-c2cccc3scnc23)cc1)NCC(c1ccc(Br)cc1)C CC(C)(C)CCCC(=O)N1CC2(CCN(C(=O)Cn3cnnn3)C2)C1 c1(CC)nnc2cc(N3Cc4ccccc4C3)ncn12.C12CCN(CC1)N2 O=C1CC(NC(c2ccc(C)o2)=O)C(=O)N1.c1(CC(=O)N)ccc(O)cc1 N1(C(C=CS(C)(=O)=O)=O)CC2CCC1CN2C(=O)C(=O)C=Cc1cccs1 c1(CCC)ccc(C(N2CC(CC(C)NC(c3ccncn3)=O)C2)=O)s1 Cc1cc(-c2ccnc(C(=O)NC(CO)CC(C)C)c2)ccc1NC(C)=O c1(COC)nc(NC2CC(CC)C2)cc(O)n1.c1(C2(C=O)CC2)ccccc1 C1(NC(c2ccc(C)n2C)=O)CC2CCC(C1)N2C(=O)Cn1cccc(N)c1=O C=CC(C)CC(=O)NC1(C)CCN(C(=O)COc2cn[nH]c2)C1 O=C1CCCCN1C1CCN(c2nsc(N3CCOCC3)n2)C1 c1(CC(=O)N(CCC)C)cccc([N+](=O)[O-])c1.C1(CC=O)CCCS1(=O)=O.N C12(C=O)CCCC(C)(C1)OC2.N1(C(C2C(C(C)C)(CC)C2)=O)CC(C)C1 C(=O)(C1=NOC(CNC(=O)C(C)C2CCC2)C1)NC(c1cncnc1)C CCC(C)C(O)CC(=O)N(CC(CO)(CO)NC(=O)C(=O)N(C)C)C N1(C(c2ncc(N)cc2Cl)=O)CC=C(CCNC(=O)CC23CCCC2C3)CC1 C1(C(=O)NC23COCC(CO)(C2)C3)CC2CCC1(N=c1[nH]nc(C3CC3)s1)C2 c1(OC)cc(C(N2CC(CN(C)C)C2)=O)c([N+](=O)[O-])cc1O.c1cncc(Cl)c1 C(CN=c1ccc([N+](=O)[O-])c[nH]1)N1CCN(c2nc(SC)nc(O)c2)CC1 O=C1C=CC(C=O)N=N1.C1(N(C(=O)CC23CC(C2)C3)CC)CCCCC1.N Cc1nc(CNC(C2CSCN2C(c2cc(O)cs2)=O)=O)sc1C c1(C(=O)NC(C2(O)CN(C(=O)C(c3cncn3C)O)C2)C)ccc(CO)s1 N1(C(C2C(=C)C2)=O)CC(CNC(=O)Cc2ccc(F)cc2)C(C)C1 C1(c2ccc(OC)cc2)CN(C(=O)C(C)CF)CCN1C(c1cnn(C)c1F)=O Cc1cc(C(=O)N(CC(C)CNC(=O)C(C)Cc2cnn(C)c2)C)nnc1O C1(NC(C(C)OCCOCC)=O)CCN(C(c2[nH]cnc2C)=O)CC1(C)C C1(CNC(C(C=CC)O)=O)CC2CCC1N(C(C1(OC)CCSCC1)=O)C2 C(=O)(N=c1[nH]n(C)cc1C(N)=O)c1nc(NC(c2ccc(OC)c(O)c2)=O)sc1 c1(C(=O)NCC#CC(=O)NCC(=O)OC(C)C)ncccc1Cl N1(C(C=CC)=O)CC=CC1(C)C(N1CC2C(C(N)=O)C2C1)=O.C(C)OC.O C1(NC(C)Cc2cccs2)CCCNC1 C1(CNC(C(c2ccccc2)OC)=O)CCCN(C(c2occc2C(C)C)=O)C1 C(=O)(C1=CC2CCCCCC12)NC1(CNC(Cc2n[nH]c(=N)s2)=O)CCCCC1 c1(C(=O)NC2(CC(=O)NCc3cnc(C)s3)CCC2)sc(Br)nc1C N1(C(CSC)=O)CCC2CC(CNC(=O)COc3cn[nH]c3)CCC2C1 c1(C(=O)NCC(C)NC(C2CCc3cncn3C2)=O)ccn2c1CCCC2 CCCCCC(O)C(=O)NC1CCC2CC1CN2C(c1cc(Cl)ccc1OC)=O c1(C(=O)NCC(C)NC(CCOCCOC)=O)ccc(OC)cn1 N1(C(c2cc(C(C)C)on2)C(=O)NC)CC(N=[N+]=[N-])CCC1(C)C CC1CCC(N(C)Cc2nnc(-c3ccccc3)o2)(CO)C1 CC1CN(C(C2COCCN2C)=O)CC1NC(=O)CC1CC2(CCC2)C1 Cc1cc(C(=O)NCCN2CCCN(C(=O)C=CBr)CC2)nnc1C N1(C(C(=O)NCC2CCCC(C3CC3)O2)=O)CCOc2c(Cl)cc(Cl)cc2C1 CC(C)(C)C(CO)C(=O)NC1CC(CCNC(=O)C(O)C2CCCC2)C1 S(=O)(=O)(c1cccnc1N(C)CCN1CCOCC1)N1C(C)CCCC1C Cc1ccc(CN2C(C(=O)NCc3cnn(C(C)C)c3)CC3CC23)cc1C#N C1(CNC(CC2(C)CC2)=O)CCN(C(=O)CCc2cnn(-c3ccccc3)c2)C1 CC1C(NC(c2ncncc2Br)=O)CCN1C(=O)Cn1ncccc1=O c1(Nc2ccc(C(=O)NC(CNC(COC)=O)C)cc2)cnc(C#N)cn1 c1(C(=O)NC(CNC(C(C(C)(C)C)SC)=O)C)cc(C)c(C)nc1C C1(c2nnnn2CCCC2CC2)(NCc2cccc(C)c2C)CC2CCC(C1)S2 c1(N2CCC(C)(CNC(C3(CC#C)CCCO3)=O)C2)nc(OC)c2nc[nH]c2n1 CC1CN(C(C2CN(CC3CCCC3)C2)=O)CC1(C)CNC(=O)CC(C)(C)C c1(C)ccc(N2CCN(CC(C(=O)OC)CC3CC3)CC2)cc1Br.C(C)=O C(C(=O)NCC1CCCO1)(C(C)C1CCC1)N(c1ccccc1C)CC C(=O)(C1=CC2C=CC(C1)C2)N1CCC(C(N2CC(S(C)=O)C2)=O)C(C)(C)C1 C1CN(C(=O)CCc2ccncc2)CC(C(F)(F)F)O1.C1(C(=O)N)(CC)CC1 c1(C(=O)NC(CNC(CC(COC)(C)C)=O)(C)C)ccc2c(c1)COC2=O CC(O)CCCN(C)C(C1(NC(C2SCCS2)=O)CCCC1)=O c1(C(N2C(COC)CN(C(=O)CC(C)(C)CC)CC2)=O)cccc2c1CCCC2 c1(C(C)=O)ccccc1C(N1CCN(C(=O)CC23COC(C2)C3)CC1)=O Cc1cnc(C(C)NC(=O)C(C2CCN(C(=O)CN(C)C)C2)C)s1 C(N=c1cc(C)nc(N2CCc3cnccc3C2)[nH]1)c1ccc(OC)nc1 C1(C(N(CCCNC(c2n[nH]cc2F)=O)CCO)=O)CCc2nccn2C1 C(=O)(CCC(C)(C)NC(=O)CCC1CCOCC1)NCCOCC(C)C c1(OC)ccccc1OC(C)C(=O)NCCN.C1(n2ccnn2)CCCC1(C)O N1(C(c2cc(CCC)ncc2)=O)CCC(C)C(NC(C2(OC)CCSCC2)=O)C1 c1(C(=O)NC(C)CO)ccc(NCCCC2CCCC2)cc1 C1(CNC(C=CC(N)=O)=O)CCN(C(=O)C2=CCOC2)CC1(F)F C1(C(C)NC(C2OCCCO2)=O)CN(C(c2c[nH]nc2-c2cccs2)=O)CCO1 C1CC2(CO1)CN(C(c1ccnn1C1CC1)=O)C2.CC(C(=O)NC)C(F)(F)F C(=O)(CCCC(C)(C)C)N1C(CC)C(C(=O)NCC(c2ccccn2)O)CCC1 C1(C(=O)NCCCOC)CC12CCN(C(=O)C=CC(F)(F)F)CC2 C(=O)(CCC(C(=O)NCC(F)CNC(=O)CCc1cnoc1)N(C)C)OC c1(C(=O)NC2CCN(C(c3cc(Cl)c(Br)[nH]3)=O)C2)nc2ccccc2[nH]1 C1(C(C(=O)NCCN(C(C2(O)CCSC2)=O)CC)C)CCCCC1 c1(OC)c(C(N2CCC(C)C(NC(=O)Cc3csnn3)C2)=O)cccc1F C1CN(C(C2CCCCC2C(C)(C)C)=O)CC1O.C1(OCC)CC(CC=O)C1.N C(=O)(C(C)(C)CC(=O)N1C(C(=O)NCC2(C)CCC(O)CC2)CC1C)OC Cc1ccc(C)c(NC(=O)C(C)OC(=O)CSc2ccc(F)c(F)c2)c1 CCCCS(=O)(=O)CC(=O)NCC(C(C)C)NC(=O)CCCCC(F)(F)F C1(C(N(C(C)C)CC)=O)CCN(C(N)=O)CC1.C1(C(=O)N)CC1.C1CC1 c1(CN2CCC(C(=O)NCCCc3ccncc3)C2)cccc(Cl)c1 CC1(C)CCCc2c1nc(Cl)[nH]c2=NCCNC(c1ccccc1SCC#N)=O N1(C(c2n[nH]c(C)c2C(F)(F)F)=O)CC2CC(NC(C3(F)CC3)=O)CC2C1 C(CCCC(C)(C)C)NC(CC(C)(C)N(C(C(CC)NC(C)=O)=O)C)=O C(CN=C(NCc1nc(C(C)(C)C)n[nH]1)NC1CCC(=O)N(C)C1)OCC=C c1(C(=O)NC2C(NC(=O)Cc3ccncc3)CC2)cccc(C(F)(F)F)c1 N1(C(C(N2CC(C)C2CO)=O)=O)CCN(Cc2ccco2)CC1 N1(C(C2(CCC)CC2)=O)CCCN(C(C2(OC)CC2)=O)CC1 C1(O)(C(C)C)CCN(C(=O)CCCn2cc(CC3CC(F)(F)C3)nn2)CC1 N1(C(=O)CC2CCCCO2)CC2CCC1CN2C(C1(C(F)F)CCCO1)=O S(=O)(=O)(c1ccc(NCC(C)Cc2cccs2)c(Br)c1)N(CCO)CC Cc1nn2cccnc2c1C(N1CCC(NC(c2csnc2Cl)=O)C(F)C1)=O N1(C(C(=O)Nc2cccc(OC)c2)C(C)C2CCOCC2)CCC2(CCCO2)C1 c1(NC(CCCCCCSC)=O)nc2c(s1)CCN(c1ncccn1)C2 CC(CC(=O)N1CC2(CCCC2NC(c2cc(O)ccc2Cl)=O)C1)CC(F)(F)F C#Cc1ccc(C(=O)NC2(C(=O)N)CCC(C)(C)C2)cn1.C1CCOC1(C)C.C N1(CC(=O)NCCCC=C)C(=O)CNC1=O.c1(C=O)cc(C(N)=O)nn1C.N N1(C(C2CC2)=O)CCCC(N(C(=O)C(N2CCN(C)CC2)C)C)CC1.CCO.C c1(C(=O)NCC2CC(C(N3CCC(C(F)F)C3)=O)CO2)cc(F)ccc1O C(C(=O)N1CCC1Cc1cnn(C)c1)(C(C)(C)C)n1cc(C(C)(C)OC)nn1 C1(NC(C(CN=[N+]=[N-])NC(C(C(C)C)=O)=O)=O)CC2CCC(C1)C2O N1(C(CC(C)(C)C)=O)CC2CCN(C(c3nnn(C(C)(C)C)n3)=O)C(C2)C1.CS O=C(CC1CC(F)(F)C1)N=c1sccn1Cc1ccccc1F c1(N2CCC(CCNC(C3CN(CC)C(=O)C3)=O)C2)nc(Cl)nc(C)c1[N+](=O)[O-] N1(C(c2cnc(NC(C)=O)o2)=O)CC2COCCC2C1.C1(=CC=O)CCCC1.N c1(CC)ccc(C(=O)NC(C)(C)C2CCC2)c(F)c1.C(=O)CP(C)(C)=O.N CCC(CCC(=O)NCC12CCCN1CCC2)NC(C1CN(C)CCO1)=O c1(CC(C(=O)N)OC)ccc(F)cc1.C1(CC)CCCN1C(c1coc(Cl)n1)=O c1(C(N2CCCC(CNC(c3c(C)onc3)=O)CC2)=O)ccn2cnc(C)c2c1 CC1(O)CCOC2(CCN(C(C3C4CN(C(=O)CO)CC34)=O)CC2)C1 C(C(C)(O)CC(=O)N1CC(C)CC1C(=O)NCCCCCN(C)C)OC CCC(C)C(O)CC(=O)NC(CNC(=O)COC(C)=O)(CC)CC c1(CC)cnccc1C(C)NC(=O)NC1CC1c1cccs1 N1(C(CCCCC#C)=O)C2CCC1CN(C(C1(C(F)F)CCOCC1)=O)C2 N1(C(c2ccc(CS(N)(=O)=O)cc2)=O)C2CCC1CN(C(=O)Cc1cnc[nH]1)C2 N1(C(CC=C)=O)C(CNC(C2CC2(F)F)=O)CC2COCC12 C1(NC(CSc2ccc(C)cc2)=O)(CO)CCCN(C(c2nc(=O)n(C)[nH]2)=O)C1 C(=O)(C(C)(C)CC(=O)N1CCC(C)C(NC(C2CCCN(C)C2)=O)C1)OCC c1(CN(C(C)(C(N)=O)c2ccccc2)C)ccc(S(=O)(=O)N(C)C)cc1 N(C1CCCc2ccc(Cl)cc21)c1nnc(CC(C(C)(C)C)CCO)n1CCN C(=O)(C(C1=CCC2CC2C1)N)OC.[SH](=O)(=O)c1ccccc1.C(C)(C)C.C=O C(=O)(CCC(C(C)C)NC(C1(C#N)CCCC1)=O)N1CCC(NC(CC)=O)C1 N1(C(CC=C=C)=O)CCC2(C(=O)NC(C)CC=C)CCCC12 N1(C(CSCCCC(C)C)=O)C2CCC(C(=O)NC(C)C)C1CC2 c1(C(N2CCC(N(C(C(C)C3CCOC3)=O)C)CC2)=O)ccc(N)c(N)n1 N1(C(c2ncnc(OC)c2F)=O)CC(C2CN(C(=O)Cc3csc(C)c3)C2)C1 C(=O)(CCCCC(C)CC)N1CCC(C=C)(C(=O)N(CC(C)CO)C)C1 c1(C(=O)NC(C(=O)N(C2CCCOC2)CC)c2cccs2)ccc(C#N)s1 C1(C(N(CC(=O)N(C(C)C(=O)NC)C)CC)=O)COCC1C(N)=O C1(CNC(Cc2ccc(OCC)cn2)=O)CCN(C(=O)C(CC)CO)CC1C C1(NC(C)=O)CCN(C(c2cc(F)ccc2NS(C)(=O)=O)=O)CC1C C12(CNC(NC(C)CC(F)(F)F)=NCC3CCC3)CCC(C)(C1)OC2 N1(C(C2=NOC(C)C2)=O)CCOC2(CCN(C(C3(C(F)F)CCCO3)=O)CC2)C1 N1(C(CSCC)=O)CCC2(NC(C3CCCC34CC4)=O)CCCC12 C(CC(N)C(=O)NC(c1ccc(F)cc1)CCO)OCC N1(C(c2c(C(C)NC(=O)C(N3CCOC3=O)C)noc2)=O)CCCC(C)(C)C1C C1(CNC(C(N2CCOCC2)C)=O)(NC(C2CC2c2cccs2)=O)CCCC1 C(CCCN=C(NCC(F)F)N1CCC(C2(O)CC2)CC1)SCC C1(NC(CNC(CCC)=O)=O)CCCCN(C(=O)CC=Cc2ccccc2F)C1 Cc1ccc(C2CCC2NC(=O)NCc2cnc(F)cc2C)c(C)c1 N1(C(C(CCC)NC(C)=O)=O)CCCC2CN(C(c3ccc(C)o3)=O)CCC12 C1(CNC(C(N2CCOCC2)C)=O)(CNC(=O)C=O)CCCCC1.CC(F)F c1(C(=O)NC(C(C)C)C(C)NC(c2cc(F)cs2)=O)n[nH]cc1[N+](=O)[O-] c1(NC(C2CC(=C)CN2C(C2CC2(F)F)=O)=O)cccc(F)c1C(N)=O CCC(C(=O)OC)C(=O)NC1CC=CCC1C(=O)NCCCCCN(C)C c1(C(=O)NCC(C)CNC(=O)C(c2ccncc2)C)cccc[n+]1[O-] N1(C(C2=CC(C)(C)C2)=O)CCCCCC(NC(=O)C)C1.C(=O)(CCC(C)(C)C)N C1(C(=O)NCC(CN(C(C(=O)NCC)=O)C)(C)C)CCCS1(=O)=O Cc1cc(N(CCCNC(=O)C(F)(F)CO)C(C)C)c(F)cc1[N+](=O)[O-] n1(CC(=O)NC2CC(N(C(=O)Cc3c[nH]nc3O)C)C2)cnc2ccccc12 C1(NC(c2c(CC)[nH]cc2)=O)(CNC(c2cnn(C)c2C)=O)CCCCC1 c1(C(N2CCN(C(C(COC)(C)O)=O)CC2)=O)cnc2c(C#N)cnn2c1 C1(COC)CCCN(C(=O)CCN(C)CCO)C1.c1(C(=O)N)cc(O)n(C)n1 N1(C(C2CCC2)=O)CC(C(=O)N(C)CCC2CCCCC2)C(F)(F)C1.COC N1(C(c2c(C)ncc(N)c2)=O)CCC2(COCC(CNC(C3CC(O)C3)=O)O2)C1 C1(N(C)C)CCCC(C(=O)NC2CN(C(c3cncc(Cl)c3)=O)C2)C1 C1(CNC(c2c(Cl)nc(N(C)C)s2)=O)COC(C)(C)CN1C(=O)C1CC1 N1(C(c2nc(COCC)sc2)=O)CCCC12CCN(C(=O)CC(C)(C)C)C2 C1(C=O)CC2(C1)CC(O)C2.Cc1[nH]nc(C(=O)NCC2(C)CCCC2)c1O.N C1(CNC(CN2CCC(C)(C)C2)=O)CN(C(c2ccsc2)=O)CCC12CCOC2 Cn1c(C2CC2)nn(CC(=O)NC2CC(NC(=O)Cc3ccns3)C2)c1=O O=C(NNC(=O)c1csc(Cl)n1)NCc1csc(C(F)(F)F)c1 C1(C(N2CC(NC(Cc3c(C)con3)=O)C2)=O)CCCCC12CC2(F)F O(C=CC(=O)NCC1(O)CN(C(C2CC(O)(c3ccncc3)C2)=O)C1)CC N1(C(CNC(C(C)CC2CC2)=O)=O)CCC(C)C(F)(F)C1 C1(NC(C2C(C(=O)OC)CC2)=O)CCOC1C(=O)NC(COC)CO C1(NC(CCCc2nc(C)sc2)=O)CC1C1CCCN(C(C2CCC(=O)N2)=O)C1 Cc1ccc(CCCNC(c2nnnn2C(C)C)C2(C)CCCO2)c(C)c1 c1(C(N2CCC(CNC(Cc3ccc(C)s3)=O)C2)=O)ccc2sc(C)nc2c1 C(=O)(CCN=c1ccc(C)c[nH]1)N(CCN(C(=O)Cc1cccs1)CC)CC C(=O)(C#CC(C)(C)C)NCCC1(CNC(C2(C)C(C)CCC2)=O)CC1 Cc1c(Cl)ccc(C(=O)NC(C2CCN(C(C34CCC3CC4)=O)C2)(C)C)c1O Cc1ccnc(O)c1C(=O)N(C)CCC1CCN(C(=O)Cn2ccnc2C)CC1 c1(CC(CC)NC2(C)CCOC2)ccc(OC)c(OC)c1 N1(C(c2c(OC)noc2C)=O)CC2CCC2(CCNC(=O)C=CBr)C1 Cc1noc(C)c1CC(C)C(=O)OCc1cncc(C(=O)OC(C)(C)C)c1 Cc1nn(C)nc1C(N1CCCC(CN(C(=O)CCC2CC(C)(C)CO2)C)C1)=O N1(C(C2CCC(=O)N2)=O)CCC2(C1)c1[nH]cnc1CCN2C(=O)Cn1ncnn1 C#Cc1cc(C(=O)NC(C)(C)C)ccc1C.N12CCN(CC1)CCOCC2=O CCCC(CC(C)C)C(=O)N1CC(C(=O)NCC=C(C)C)C(C)(C)C1 c1(N(C)C)ncc(NC(=O)C(C2CCN(C(C3CC(C)(O)C3)=O)C2)F)cn1 S(=O)(=O)(c1cnccc1[N+](=O)[O-])NC(C)C(c1c(F)cccc1F)O C(=O)(N=c1ccn(C)[nH]1)C1N(C(CC(=O)OCC)=O)C(CO)CC1 CC(C(=O)N1CC(F)(F)CC1C(=O)N(C)Cc1cn[nH]c1)C(C)(C)C N1(C(C2N(C(=O)O)C3C(C2)CCC3)=O)CCC2(CCCC2)C1.CC(C)C.C(N)=O C1(CC=C)(NC(c2nnc(C)cc2O)=O)CCCN(C(=O)Cc2cncn2C)C1 c1(C(=O)NC(C(C)(C)C)CNC(C23CC(F)C2C3)=O)cc2sc(Cl)cc2[nH]1 C1(C(=O)NCC(CCC)NC(=O)CC(C)OC)CN(C)CCN1C CC1(C)CN(C(=O)C(C)(C)c2cccs2)CC(CNC(=O)C(O)C2CCC2)O1 CCCC(C(O)C(=O)N(C)Cc1ccccn1)NC(=O)C=C(C)c1ccco1 Cc1sc2ncc(C(=O)NC(C)CNC(C3CSCCS3)=O)c(=O)n2c1C C(=O)(C(CC(C)C)CC(C)C)NC1CCCN(C(c2n(CC=C)ccc2)=O)CC1 C1(C(=O)NC2(C)CCN(C(c3cnc(C(F)(F)F)s3)=O)C2)CCc2ncnn2C1 N1(C(c2ccc(C)n2C)=O)CCC(CNC(c2coc(O)n2)=O)C(C)C1 N1(C(c2c(C)sc(O)n2)=O)CC2(C1)CN(C(C1CC(OC3CC3)C1)=O)C2 CS(=O)CCC(O)C(=O)NC1(CNC(=O)Cc2cccc(O)c2F)CC1 C=CCCCC(C(=O)NC1CCC(O)C(O)C1)NC(=O)C(C)OCC(C)C N1(C(c2nc(CC)sc2)=O)CCC(C(=O)NOCCc2ccccc2)C1C(C)C C12(NC(CC=C)=O)CCOCC1CN(C(=O)CCN(C)CC)C2 Cc1ccc([N+](=O)[O-])c(NC(c2csc(C(N3CCC(F)(F)C(O)C3)=O)n2)=O)n1 CC1(C2CC2C(=O)NCCOC2CCCCCC2)COC1 N1(C(C(C(C)O)(C)C)=O)CC2CC(C1)CN(C(=O)C=Cc1cnc[nH]1)C2 Cc1cocc1C(=O)NCC(C)(C1CCC1)NC(=O)C=C1CCC(C)C1 C12(C(=O)NC(c3ccsc3)C)CC3CC1C2C3.n1(CC(=O)N)cccnc1=O c1(C(N(CCOC)CC)=O)c[nH]c2cc(C)ccc12.C1(C=O)CC2(C1)CC2F C(=O)(C1=NOC2(CCOC2)C1)NC(C1CCCN1C(=O)CCNC(N)=O)C C1(NC(=O)CC2NC(=O)NC2=O)CC2CCC(C1F)N2C(c1ncccn1)=O c1(CN(C)C(c2c[nH]nc2C(F)F)=O)cc(O)nc(=N)[nH]1 CCC(C)CC(=O)C(=O)NC(C(=O)NCc1cnccc1C)c1ccoc1 C1(C(=O)NC2COCCN(C(=O)CC(F)F)C2)CC12CCCc1ccccc12 N1(C(C2(OC)CCCC(C)C2)=O)CC2CCC(C1)N2C(c1cccc(C)c1)=O N1(C(c2cccc(OC)n2)=O)CC(CO)C2(C1)CN(C(C1(C)COCCO1)=O)C2 CC1CCCc2ncc(C(=O)NC(C)CN(C(=O)C(F)(F)c3nccn3C)C)n21 Cc1cc(O)cc(O)c1C(=O)NC1CC(C(=O)NCc2cnccc2Cl)C1 N1(C(N(CC(N2CCCC2)C)CC)=O)CCC(C(=O)OC)C1 c1(NC(C2CC(F)CN2Cc2ncc(-c3ccccc3)[nH]2)=O)cnnc(Cl)c1 c1(C(=O)NCC2N(C(C(COC)N(C)C)=O)CCCCC2)cccc2nc[nH]c12 O=C(CC(O)C(Cl)(Cl)Cl)NC1CC(CCNC(c2cnc(S)nc2)=O)C1 N1(C(c2c(C)nc(CCC)o2)=O)CCC(C2CCN(C(=O)CC3CC3)C2)CC1 N1(C(C(F)=C(C)C)=O)CCC(O)(CNC(c2c(C)nn(CCO)c2C)=O)CC1 CCCCCCC(CC)C(=O)N1CCN(C(=O)C(C)=O)C(C)C1 c1(NC(CNC(C=C(C)C(F)F)=O)C2CCC2)cc(Cl)nc(C2CCCO2)n1 C#CCCCCCC(=O)NC1C=CCN(C(=O)COc2ccccc2C(C)C)C1 C12(NC(c3cc4ccccc4s3)=O)CCCN(C(c3cc(Cl)c(Cl)[nH]3)=O)CC1C2 Cn1cnc(S(=O)(=O)NCC(=O)N)c1.C12CCC1CN(C(C1CCNC1=O)=O)C2 c1(C(N(C(C#C)C)C)=O)sccc1CNC(=O)C(CC1CC1)OC N1(C(CN2CCN(CC)CC2)=O)CC(CNC(=O)C(O)c2ccsc2)CC(C)C1 C1(C)(C(c2n(CCCOC)nnn2)Nc2cn(CCOC)cn2)CCCCO1 C1(F)(CNC(c2ccn(CC)n2)=O)CCCN(C(c2cc(C)cs2)=O)C1 Cc1cccc(CCNC(c2cn(CCNC(c3cnc(Cl)n3C)=O)nn2)=O)n1 c1(C(=O)NC2CC(OC)CN(C(C3CC3F)=O)C2)cc2ccncc2c(O)n1 C1(CC(=O)NCCc2cc(C)no2)CN(C(C2CN(C)C2)=O)CCC1C C1(NC(C2N=C(C)SC2)=O)CCN(C(c2ccc3nsnc3c2)=O)C12CCCC2 CC1CC(NC(C2CCC(O)C2)=O)CCN1C(c1cc(O)ncc1Br)=O C1(CNC(CC(CC)NC(=O)C2=CCCC2C)=O)COCC(=O)N1C c1(CC)cc(C)ccc1C(=O)N(C)C.C1CCCN(C(c2nc(Cl)c(Cl)s2)=O)C1 CC1CN(C(=O)C=CC2CCOC2)CCC1CNC(=O)CCC1CCCOC1 CC1CC(N2CCOCC2)CN1C(C1CC2CCC2C1)C(=O)Nc1ccccc1 c1(CC)cc(C(N2CCC(C(=O)Nc3cccc(-n4cccc4)c3)C2)=O)ccn1 c1(C(N2CCN(C(c3c(C#C)c[nH]n3)=O)CC2)=O)cc(Cl)nnc1O N1(C(Cc2c(C)nsc2)=O)CC2COCC(C1)C2NC(=O)C(F)C(F)(F)F N1(C(C)C)CCCC(CNC(=O)CCN(C)C(C)C)C1 C=CCCCCC(=O)NCC(C)(C)CN(C)C(C1CCC12CCCO2)=O Cc1noc(CCC(=O)NCCOC2CCN(C(C34CC(C)C3C4)=O)C2)n1 C1(CC)CCC(C(N2CC(C)C(C(F)(F)F)C2)=O)CC1.C(=O)CC.C(C)=O C(CCC)(C(=O)NC1CN(C(C2CCCSC2)=O)CC1C)=CCC C=CCC(C)(C)C(=O)NCC1CC2(CC2)CN1c1ncc(C(C)(C)O)cn1 c1(C(=O)NC2C(NC(COc3cn(C(C)C)nc3)=O)C2)cc(C#N)cn1C CC1CN(C(=O)Cc2csc(=N)[nH]2)CCC1NC(c1cncnc1C1CC1)=O N1(C(Cc2scc(C)c2)=O)CC2(CC2)CC1CNC(C1C(C)C1C)=O C1(NC(c2ccc(OC)s2)=O)CCCCC1NC(c1cccc(Br)c1)=O c1(C(=O)NCC(CC=C)NC(C2(OCC)CCOCC2)=O)nc(Cl)ccc1Cl CCCCCC(=O)NC1CC(NC(C2C=CCCC2)=O)C1 C1(CNC(C(C)SCCCC)=O)CN(C(=O)CN(C)C(C)C)CC1(F)F C1(C)(C(=O)NCc2nccc(C)n2)CCN(C(C2OCCC2C)=O)CC1 c1(C(=O)NCC(CC2CN(C(C=C(C)Cl)=O)C2)(C)C)onc(Br)c1C c1(C(=O)Oc2cccc(N(C)C(C3CCCCC3)=O)c2)cc2c(Cl)cccc2s1 c1(NC)ccc(F)cc1C(=O)NC1CCOCC1.c1(C=O)cc(C2CC2)[nH]n1.N C(CCCCCC(=O)NC(C1CCCN1C(=O)C(c1cccc(C)c1)=O)C)SC CCCCC(C)CCC(=O)N1CC(NC(c2cscc2F)=O)C2(CC2)C1 c1(C(N2CCCC(CNC(c3ccc[nH]3)=O)CC2)=O)ccc([N+](=O)[O-])cn1 c1(C(N(C2(C(=O)N)CC2)C)=O)ccc(CC#N)cc1.C1(CC)CCCC1.CO C1(NC(c2cccc(N)c2O)=O)CN(C(C2CC(=O)NC(=O)N2)=O)C2(CCC2)C1 C1(C)(CNC(CC(CC)OC)=O)CCN(C(c2ccsc2-n2cnnn2)=O)CC1 CC1C(NC(=O)CN2CCC(O)CC2)CCCN1C(C1CC(=O)N(C)C1)=O C1(C)(C=O)Cc2ccccc2C1.c1(COC)ccc(C(=O)NC(C)C)cc1F.N c1(C(=O)NC2CC3CC(C2)N(C(c2ccc[nH]2)=O)C3)noc2c1CC(F)(F)CC2 C1(C(C#C)C)CCN(C(=O)NC2CCN(c3cccnc3)C2)C1 N#CC12CC(C(N3CC(NC(c4ccccc4Cl)=O)C3)=O)(C1)C2 N1(Cc2cc(C)[nH]n2)CC(F)CC1C(=O)Nc1ncc(C#N)s1 c1(C=O)ccc(C(F)F)cc1Cl.C(C)(C)CO.CC(C(=O)N)NS(C)(=O)=O c1(C(=O)NCC(CC2CC2)C(=O)NC2CCC(CCO)CC2)cccc(F)c1F C=CCCCCCN=C1NC2=NCCS(=O)CCC(=CC(OC)=CC=C1)N2 c1(OC)ccc(C(=O)NC2CC(N(C)C(C34CC(C)C3C4)=O)C2)c(N)c1 C1(CCC)CN(C(=O)CC(C)C(C)C)CCN1C(=O)CSCC(F)(F)F C1(C(C(=O)NCCCOCC=C)F)CCN(C(C2CC2(C)C(F)F)=O)C1 N1(C(C(C(CC)(C)C)O)=O)CCOC2(CCCN(C(c3c(C)n[nH]c3C)=O)C2)C1 C=CCC(CNC(c1ccc(C)n1C)=O)C(=O)NC(c1ncc[nH]1)CO Cc1cnc(NC(C)CCNC(c2ccc(Oc3ccc(Cl)cc3)cn2)=O)nc1 c1(CC=O)ccc(C(F)(F)F)cc1.CC1OCCC1CNC(C1CC1)=O.C N1(c2snc(SC)n2)CCC2(CC1)C(NC(C1CCC3CC3CC1)=O)CS2(=O)=O C=CC(C)C(=O)NC(C)C(CO)NC(=O)CCCOC(C)C N1(C(C2CCC(CC)O2)=O)CCC(NC(c2cnn(C)c2N)=O)C2(CCC2)C1 CC1c2ccccc2OC1CC(=O)NC1(CO)CN(C(=O)C(O)CC(N)=O)C1 CC1CCCC(C)N1C(=O)C(C)NC1C=CCN(C(C23CC(C2)C3)=O)C1 N(C(=NCCCOC)N1CCC(C2CC2)C1)C(CC)CC c1(NC(C2C(Nc3nc(C)nc(-c4ccco4)c3)C2)=O)ccc2[nH]ncc2c1 Cc1ccc(SCC(=O)NC(CNC(C23CC(CO2)C3)=O)CC(C)C)cc1C Cc1ncc(CNC(C(=O)O)c2ccoc2)c2c1OC(C)(C)OC2 CC1(C=O)CCC(=O)N1.N1(CC(=O)N(C2CCCC2)CC)CC2C=CC1C2.N c1(C(=O)NC2C(C)CCN(C(=O)Cc3c[nH]nc3O)C2)cc(=O)n2nccc2[nH]1 C1(C=O)CCCC2(C1)CC2(F)F.C(CS(=O)(=O)CC(=O)NC1CCC1)OC.C S(=O)(=O)(c1ccc2c(c1)OCCO2)N1CC(NC(c2cnc(Cl)cn2)=O)C(F)C1 c1(C(=O)N)ccc(C)c(C)c1O.c1(OC)cc(C(=O)NC2CCCC2)cc(Cl)n1 n1(CC)ncn(NC(=O)CC2(NC(C34CCCC3C4)=O)CCC2)c1=O CCC(C)C(C(=O)N(CC(=O)Nc1cc(O)ccc1C)C)N(C)C c1(C(=O)NCC(CN(C(COC(CC)CC)=O)C)C)cccc2oc(C)nc12 N1(c2ncc(OC)c(C)n2)Cc2ccccc2C1C(=O)NC1(c2ncc[nH]2)CC1 CC1CN(C(c2ccnn2C)=O)CC1NC(c1cccnc1C(F)(F)F)=O c1(C(=O)NCC(C)NC(C2CCOC(C)C2)=O)cnc2c(C#N)cnn2c1 N#Cc1ccn2ncc(C(=O)NC3CCCC3NC(=O)CC3COCCO3)c2c1 c1(C(=O)NCCC(Cn2cc(C(C3CCCC3)C)nn2)F)cnc2ncccc2c1 C=C(C)C1CN(C(=O)CCCCNC(c2ccc(F)c(O)c2)=O)CCO1 C(=O)(C(F)C(F)(F)F)N1C2(C(=O)NCCn3c(C)cc(C)n3)CC2CC1 C1(CC=C)CCCCN1C(c1oc(CNC(=O)CC2CCC(=O)C2)cc1C)=O Cc1noc(CCC(=O)NCC2CC(NC(=O)C=Cc3cc[nH]n3)C2)n1 c1(C(N(CCNC(=O)CCSCC(N)=O)CC)=O)ncc2[nH]ncc2n1 c1(C(N2CCC(CNC(C(C)SCC)=O)C2)=O)cnc(C2CCOCC2)nc1C N1(C(C(C2CCC2)OC)=O)CC(C)OC(C)(C)C1.N1(CC=O)CCCNC1=O.N CCC1=NOC(CNC(C2C=CCN2C(C2CCC2C(C)(C)C)=O)=O)C1 CCC(C)CC(C)C(=O)N1CCC(NC(=O)C(C)=NOCC#N)CC1 C12(C(=O)NCC3N(C(c4c(OC(F)F)cc(C)s4)=O)CC3)CCC(CC1)OC2 C1(NC(c2c(C)nc(CC)o2)=O)CCN(C(=O)C2=NNC(=O)CC2)CC1(C)C Cc1cc(C)n(C(C)C(=O)NC2CN(C(=O)CCc3cn[nH]c3)CC2F)n1 C(=O)(C1=NNC(=O)CC1)NC(C)CCNC(=O)CC(c1cccc(F)c1)C c1(C(=O)NCC2CN(C(=O)Cn3cc(Br)cn3)C2)nc2ncccn2n1 C12(C=O)CCC(CC1)C(C)O2.C(C)(C)(CC(=O)NCCc1ocnc1)OC.C Cc1[nH]c(=N)oc1C(=O)NCC1(C(=O)NC)CC1.C1(C)CNC(=O)C1 c1(CNC(N2CCCC(C(=O)NC)C2)=O)cc2c(OC)cc(OC)cc2o1 C(=O)(C(N=[N+]=[N-])C(C)C)NC(CCC#C)C(=O)NC(CO)CCSC N1(C(C2(NC(=O)CC3CCCOC3)C(C)(C)C2)=O)CCC2(CC1)CSC2 c1(C(N(CCNC(=O)CS(=O)CC)CC)=O)cc(C)c2nc(C)nn2c1 CC1CN(C(=O)Cc2coc(-c3ccccc3)n2)CCN1C(c1coc(Cl)c1)=O c1(NC(=O)NCC(C)CS(N)(=O)=O)ccc(OC(F)F)c2ncccc12 C1(C(=O)NC)CCCN(C(CC2CCOC2)C(=O)Nc2ccc(OC)cc2)C1 C1(CC(=O)NCCS(=O)(=O)NC)CCCN(C(=O)CN2CCCCC2)C1 C#CCC(CC(=O)NC(C)C(O)C(F)F)NC(=O)C(n1nccc1C)C C1(NC(CC2(C=C)CCCCC2)=O)CCC2(CC1)CC2NC(=O)CC=C(Cl)Cl Cc1ccnc(C(=O)N(CCCNC(=O)C2=CCCS2)C(C)C)n1 c1(NC(C2C(COC)C2)=O)nc(=NCC2CCCO2)[nH]cc1Br C(c1ccncc1)=CC(=O)NC(C1CCCC1)CNC(C(N=C)=O)=O Cc1c(C(N2CCC(NC(C34COCC(C3)C4)=O)C2)=O)cccc1C#N C1(NC(C2Cc3cscc3C2)=O)CN(C(C2CC23CC3)=O)Cc2ccnn2C1 C1(N(C(=O)CC2CCOC2)C)CCCN(C(=O)CCNC(C2CCCC2)=O)C1 c1(OC)cc(CC(=O)NC(C)C(C)NC(c2nscc2Br)=O)ccc1C C12(CNC(COCC(=O)OC)=O)CCCC1CN(C(=O)C=CI)C2 C12OCCC1C(=O)N2.C(CC(=O)NC(C1CCCC1)C)NC(COC)=O N#CC1CN(C(c2ccccc2O)=O)CC1NC(c1cncc(F)c1)=O N1(C(C(C2CC2)SC)=O)CC(C(=O)N(C2(c3cc[nH]n3)CC2)C)C(C)C1 Cc1nn(C)c(=O)c(C(=O)OC(C)C(=O)NCC(C)C)c1C CCC(CC)CCNC(C1CCCN(C(C)=O)C1)=O.C1(C(=O)N)CCC2CC2CC1 N1(C(C(CC=C)CC)=O)CCOC2CN(C(c3ccc4nc(=N)[nH]n4c3)=O)CC12 CC(C)(C)C(COc1ccccc1)NC(=O)NCCc1c[nH]nc1O c1(C(=O)NC(CN(C(=O)CCCF)CC)C)occc1C(=O)OC c1(C(NC2CCN(C(c3ccccc3C3(C)CC3)=O)C2)=O)cc(C#N)c[nH]1.C c1(NC(=O)CCN(F)CCO)cc(C(F)(F)F)on1.C1(=O)COCCN1 c1(NC(C2CC(C)CN2Cc2cc(Br)c(F)cc2Cl)=O)ccc2ncccc2c1 C1(C(N(CCCCN(C(C(N2CCOCC2)C)=O)C)C)=O)CN(C)CCN(C)C1 c1(C(=O)NC2CCC(NC(=O)CCc3cscn3)CC2)nnc2n1CCCCC2 CCC(C)(C)C(C)CC(=O)NC1CCCC(NC(=O)C(C)=C2CCCC2)C1 Cc1cccc(C(C(=O)NCC2CC2)N(C)CCC2CCCN2C)n1 c1(C(N2CC(C)CC(NC(c3c(C)scc3)=O)C2)=O)ccc2c(c1)N(C)C(=O)C2 Cc1cc(CC(=O)N(CCCCN(C(=O)CC2CCC3CC23)C)C)on1 c1(CC(C(=O)N(CC(F)F)CCOC)N(C)C(C)=O)ccc(C)cc1 C1(CC)CCC(C(=O)NC(CNC(=O)C2=C(Cl)CC2)C2CC2)CC1 C1(C(=O)NCc2nc(COC)on2)CCCCC1(C)NC(c1cnccn1)=O N1(C(C2CCN(CC)C2)=O)CCC2CC12C(=O)NOCc1ccc(C)cc1 C(CCCC(=O)NC(c1ccc(C)cc1)CNC(c1csc(C)c1)=O)OCC CC1(NC(=O)COC2CCOC2)CCN(C(c2cnc(S)[nH]2)=O)C1 c1(NC(C2(CC#C)CCOC2)=O)cc(C(=O)OC)cc(F)c1C#N CCCCC(CC(=O)N1CCC(OC)C(F)C1)NC(c1n[nH]c(CC)c1C)=O C(C1=CCN(C(=O)CC2CC=CCC2)CC1)NC(=O)C(O)Cn1cncn1 c1(C=O)ccc(C)cc1.c1(CCC)nc(C(=O)NC2CC2C)cs1.C1CC1 C1(C(=O)NCCNCCOC)CC(=O)N(C)C1.c1ccn(C(C)C)n1.C C1(OC)CC(CNC(=O)C(C2CCCCC2)O)N(C(c2[nH]cnc2C#N)=O)C1 O=C(NNc1ccc(OC(F)(F)F)cc1)c1c(Cl)cccc1Br C1(NC(c2c(Cl)cc(C)s2)=O)CCC2(CC1)CN(C(=O)CC1CCCC1C)C2 CON(C(=O)C1CC2CN(C(C3CC34CCCCC4)=O)CC2C1)C1CCC1 c1(CN2CC(CNC(c3cc(F)cc(I)c3)=O)OCC2)cnc2ncccn12 C(CC)(C(=O)NCC(C)CNC(=O)C(n1cc(Cl)cn1)C)OCC C1(NC(CCC=C)=O)CC12CCN(C(=O)C(C)OCOC)CC2 N1(C(C(CCSC)OC)=O)CCC2CCN(C(=O)COc3c(C)cccc3Cl)C2C1 CC(CC(=O)NCC(CO)NC(c1nonc1N)=O)C(F)(F)F N1(C(C2(C#C)CN(C(c3ccsn3)=O)C2)=O)CCC(OC)CC1C C=CC(C)C(C)C(=O)N1CCC(N(C(=O)COCCc2cccs2)C)CC1 N1(CC(C)(C)CN2CCOCC2)CC2CCC1CN2C(=O)OC(C)(C)C C1(CC)CCC(C)N1C(=O)OC(C)(C)C.C12(F)CCN(C1)C2 C(=O)CC(C)(C(F)(F)F)N(C)C.C(=O)(CCC(=O)N(C)CC)OC.C(C)=O N1(C(c2ccc(OC)cn2)=O)CCCC(C)(NC(=O)CC2(C)CCCC2)C1 C1(CNC(Cc2c(C(C)C)con2)=O)(CO)CCN(C(=O)C(O)c2ccsc2)C1 N1(C(c2c(Cl)cnc(CC)n2)=O)CCCCCC(NC(C2CC23CCC3)=O)C1 CC1(C)CCC(C(=O)NC2CCC(C#N)CC2)CN1C(=O)Cc1csnn1 C1(C(=O)NCCOCC(=O)N(C(C)C(C)(C)O)C)CC(O)C(F)C1 Cc1nccn1Cc1cn(CC(C)NC(=O)CC2C=CCC2)nn1 c1(C(=O)NC(C2CN(C(C3(O)CC(F)(F)C3)=O)CCO2)C)cc(F)n(C)n1 c1(SC)cc(C)c(C(=O)NC2CN(C(=O)C(C)c3cncs3)CC2SC)o1 N1(C(C(c2c(C)nn(C)c2C)C)=O)CC(NC(c2cnnn2C)=O)CC2(CC2)C1 c1(C(c2nnc(C)n2C)NC(=O)CCSc2nnnn2C)ccc(Cl)c(F)c1 C1(CN(C)C)(CNC(=O)CC2CC23CC3)CCC1 c1(-n2cc(C(C)NC(c3cnc(C)n3C(F)F)=O)nn2)ccc(Cl)cc1Br N1(C(C2N(C(c3c(Cl)cnc(SC)n3)=O)CC(F)C2)=O)CCc2ncccc2C1 C(C(=O)NOCC1CCC1)(C1(C)CC1)NC(c1cnn(C(C)C)n1)=O Cc1cc(C(N2CC(NC(c3ccncc3Cl)=O)CC(O)C2)=O)c(O)nc1C N1(C(CC2(C)CCCCC2)=O)CCN(C(=O)CCCn2cccn2)CC1CF Cc1cnc2n1CCC(C(=O)NC1CCCC1NC(C13CC(F)(C1)C3)=O)C2 Cc1n[nH]c(C)c1-c1ccc(C(=O)N(C)Cc2ncc[nH]2)cc1 C1(C(=O)NCC(C)CN(C)C(C2(F)CCOCC2)=O)C(F)(F)C12CC2 C1(C(=O)NC2CCN(C(C3(SC)CC3)=O)C2)Cc2c(C)cccc2O1 n1(CC)ccnc1C1OCCC1C(=O)N(C(C)CNC(=O)C)C.C(N)=O N1(CC=O)C(=O)CN(C)C1=O.C=CCC(C)C(=O)NC(c1ccc(C)cc1)C C1(CNC(C(CC)=CC)=O)CCC2(CCC2)C1NC(=O)CCCC c1(C(N2CCC(C#N)CC2)C(=O)NC2CCC(F)(F)CC2)ccc(Cl)c(F)c1F CN(Cc1ccnn1C)N1CCN(C(C)(C)C)CC1 N1(CC=C)CCC(NC(=O)C(C)(C)CN(C)C(C2C=C(C)CS2)=O)CC1 N1(C(COCCOC)=O)CCC(N2CCOC(C)C2)C(C)CC1 N1(C(CCCOC)=O)CCC(NC(c2ccccc2COC)=O)C(CO)C1 c1(CC)nc(C(=O)NCCC(C)N(C)C(C2COC(=O)N2C)=O)c(C)o1 c1(C(N(CC(CNC(C(C(C)C)SC)=O)C)C)=O)cccn2c(C)nnc12 C(=O)(C#CC1CCC(=O)CC1)N(C(C)CNC(=O)CC1CCCOC1)C C1(CC)COCCN1C(=O)C(C)c1ccsn1.C(C=O)OCCOCCOC CC1CCC(N(C(=O)CCCNC(=O)COC(=O)CO)C)C1 N1(C(C2(COC)CC2)=O)CCCC(C2CN(C(C3CNC(=O)CC3C)=O)C2)C1 c1(C(=O)N)cc2c(s1)CCC2.CC1CCOC(C(=O)NCCNC(=O)C)C1 c1(C(=O)NCCCCN(C(CSCC)=O)C)ccc2cccc(Cl)c2n1 Cc1[nH]c2ccc(Cl)cc2c1CCNC(=O)NCc1nccn1C1CC1 CC1(C)CN(C(=O)CC(=O)NCC2CC2)CCC1.C12(C=O)CC(F)(C1)C2 N1(C(C)C)CCOC(C(=O)NCCCN(C(=O)Cc2cnnn2C)C2CC2)C1 N1(C(c2ccc(C#C)cn2)=O)CC2(CCC2)CC1C.C(=O)C(C)(C)C(C)(C)C.N Cc1nc(=NC(C)CNC(c2cc(CC(C)C)[nH]n2)=O)s[nH]1 c1(C(N2CCN(C(c3nc(Cl)sc3Cl)=O)CC2)=O)ccc2cncn2c1 CC1CCC(C(=O)NC2(CNC(=O)COC3CCCCCC3)CCC2)CC1C Cc1ccccc1CC(CO)NC(c1csc(C2CCCCC2)n1)=O C1(C)(COC)CC(c2nnnn2C2CC2)(Nc2ccccc2)C1 CC(CC1CCC1)N=c1[nH]c(=NCC2CC(C)(C)CCO2)c2c(F)cccc2[nH]1 c1(NC(C23N(C(c4n(C)c(S)nn4)=O)CC(C2)C3)=O)cccc(F)c1O C1CCCC2(CN(C(c3cc[nH]c3C(C)C)=O)C2)O1.C(CC(O)C(=O)NC)SC c1(C(=O)OC)cc(F)c(NC2CCCC2N2CCC(O)C2)c(F)c1 N1(C(c2cnc(CC(C)C)[nH]2)=O)CC2CCCC2(NC(=O)C(C)C2CCCC2)C1 c1(NC(C(=O)N(CC(O)CNC(=O)CSC2CC2)C)=O)ccncc1 N(C1C(=O)Nc2ccc(Cl)cc21)C(=O)NCCn1nnc(C)n1 c1(CC)c(C(=O)N(C)CCNC(=O)COCC2CC2)nnn1C CC1CN(C(c2cnc(N)cn2)=O)CCC1CNC(c1cncc(CO)c1)=O C(=O)(C(C)CC(C)(F)F)N.Cc1cc(C(=O)NCC2(CC)CC2)nc(C)n1 Cc1cc(C(=O)NC(C)CO)c2c(c1)C(C)CCN2.C(=O)(CCCS(N)(=O)=O)N c1(C(=O)NCC2CCN(Cc3ccc(C)cn3)C2)cc(Cl)nc2n[nH]cc12 N1(C(C2(CN(C)C)CC2)=O)CC(C2CCCN(C(c3cnc(O)cc3O)=O)C2)C1 Cc1cc(NC(=O)C2CC2)sc1C(=O)N.C1(C=O)COCCN1C.C1CCCC1 Cc1nsc(NC(c2ccccc2)CNC(C2COCCN2C)=O)c1C#N O=S(=O)(CC(F)(F)F)Nc1ncc(-c2cnc(O)nc2O)cc1O N1(C(C=C(C)C(C)(C)C)=O)CCC2CN(C(=O)C(=O)NCC3CC3)CC2CC1 c1(CC)[nH]c(C(=O)NC2CC(NC(=O)CCc3ccc(C)s3)C2)nc1Cl CC(CCC(C)(C)C)C(=O)NCC1(C)CC1(F)F.C1(C(=O)N)CCC1(F)F N1(c2nc(C)[nH]n2)CCN(N2CCCCC2C2(C(F)(F)F)CCC2)CC1 C1CN(C(=O)CO)CC12CCOCC2.c1(C(C)(C)C)ncc(C=CCNCN)s1 c1(C(=O)NCCC(=C)CNC(=O)CSC)ccc(S(C)(=O)=NC)cc1 c1(NC(C2(C)N(Cc3c(C)nn(C)c3)CC2)=O)cccc2c1cnn2C C1(O)(CNC(C2C(C)OCCC2)=O)CC(N=c2[nH]ccc(C#N)c2[N+](=O)[O-])C1 C1(NCc2cn(CC)nc2)CCCC2CN(C)CC12 c1(C(=O)NCC2C3CN(C(c4nc(CCC)oc4)=O)CC32)cc(C)cc(Cl)c1 C1(CN2C(c3ccccn3)CC2)OCC2CCOC12 CCCCC(O)CC(=O)NC1CCCCC1C(=O)NC1CCS(=O)(=O)C1 C1(C(=O)NC(CNC(CCC2(C)CC2)=O)C(C)(C)C)OC(C)(C)OC1(C)C c1(NC2C(C(=O)NCC3CC(OC)C3)C2)ccc(-c2cccs2)s1 Cc1cccc2c1CN(C(C1CC(NC(=O)CC3CCC3)C13CCC3)=O)C2 c1(NC(C2N(C(CN(CCC)C)=O)CCCC2)C)ncc(Cl)c(O)n1 n1(C(C)C(F)(F)F)cn[nH]c1=NCc1cc(C(F)(F)F)cc(F)c1 N1(C(C23CC(CCC)(C2)C3)=O)CCC(C)CC1.N1(CC=O)CC2CCC1C2.C Cn1nc(C(F)(F)F)c(CNC2CCCOC2)c1O.c1nn[nH]n1 N1(C(C2CCC(C)(C)C2)=O)CC2=C(C1)CN(C(=O)Cn1ncc(O)nc1=O)C2 c1(C(=O)NC2CC(NC(C3(CC#C)CCCCC3)=O)C2)cc2cscc2s1 C1(CNC(CC(=C)Br)=O)CCC(C)CN1C(c1cnn(CCN(C)C)c1)=O N#Cc1cc(Cl)c(C(N2CCC(OCCNC(=O)CO)C2)=O)c(Cl)c1 C(=O)C(C)CC1CCCC1.C(=O)(C(C)Cc1cnn(C)c1)N(CC)CC.C C12(C(N(C)CCNC(C3CCS(=O)CC3)=O)=O)CCCCCC1OCC2 N1(C(CC=C)=O)CC(NC(C2(N3CCOCC3)CCC2)=O)CC(C)(C)C1 c1(C(=O)NC2C(C)CN(C(C3CCCC(=O)N3C)=O)C2)cccc2ccsc12 C#Cc1ccc(C(=O)NC2CCCC(CNC(=O)C(C)(C)C3CCCC3)C2)cc1 C1(C(=O)NC2CC(CNC(C3(C)CCCS3)=O)C2)CSc2ccccc2O1 Cc1cc([N+](=O)[O-])cc(C(=O)N(C2CN(C(C3CC4C=CC3C4)=O)CC2O)C)n1 c1(C(C)CN(C)C(=O)C2CC2)nnnn1C1CCCCC1.c1(CS)nncs1 N(C1CCCc2c[nH]nc21)C(C(CC=CC)NC(=O)Cc1cc(C)on1)=O C#Cc1cc(C(=O)NC2CC(NC(=O)C(CCC)OCC)C(O)C2)ccc1Cl N1(C(C(C)SC(C)C)=O)CCC(C(N2CCCC(F)(CO)C2)=O)C(C)(C)C1 c1(SC)ccc2cc(C(=O)NCC3CC3NC(=O)C#CC(C)(C)O)[nH]c2c1 C1(C(N2CC(n3c(C(=O)OC)ccn3)C2)=O)CCCOC1c1ccc(C)cc1 CC1(NC(=O)CN)CCN(C(C23CC(CS)(C2)OC3c2ccccc2)=O)CC1 N(C1CCc2c(Br)cccc21)C(=O)CCCNC(C12CC(CC(F)F)(C1)C2)=O N1(C(C2CCC(=O)C2)=O)CC2(CCN2C(=O)CCn2cnccc2=O)C1 CCC(C)C(O)C(=O)NC(c1ccc(C)cc1)C.c1(C(=O)N)c[nH]cc1C1CC1 Cc1c(CCC(=O)NC)cnn1C.C1(F)CN(C(=O)C(F)(F)c2csc(=N)[nH]2)C1 C1(NC(C2(C(N)=O)CC2)=O)CCCN(C(=O)C(c2cccc(Br)c2)O)CC1 c1(C=O)cnn(-c2cccc(C)c2)c1C.C(C(=O)NC1CC1)N(CC)CC.N c1(C(=O)NCC2(NC(C3C(C#C)C3)=O)CCCC2)cc(=O)cc[nH]1 n1(CC=O)cc([N+](=O)[O-])cn1.Cc1c[nH]c(C(=O)NC(C2CCCCC2)C)c1.N CC(=NO)c1cc(C(N2CCN(C(=O)C(C)C3CC3)CC(O)C2)=O)cnc1O N1(C(C2(C)CC(=C)C2)=O)CCN(C)CC1C1CC1.C1(C(=O)N)C=C(C)CS1 c1(OC)cc(C)ccc1C(N1CCC(C)C1)=O.c1(C=O)cncc(C2CC2)c1.N C1(C(N(C(c2cccc(Cl)c2Cl)C(=O)OC)C)=O)CCc2c(C)nnn2C1 C(Cl)(c1ccccc1F)=C(C(C(=O)NCC=C)N(C1CCN(C)C(=O)C1)C)C N1(C(C2C(C(=O)OC)CC2)=O)CC2CCCC(C1)N2C(C1CCC(=O)NC1)=O c1(CC(=O)N(CC(CNC(C(C)(C)OCC)=O)C)C)cc(Cl)ccc1Br N1(C(Cc2cc(C)sc2)=O)CC2CC2(CNC(=O)CC(C)c2ccncc2)C1 N1(C(C2OCC(C)(C)C2)=O)CCCN(C(c2ccc(C3CC3)s2)=O)C(CO)C1 c1(C(N2CC(=C(C)F)C2)=O)cc([N+](=O)[O-])n[nH]1.C(CC1CCCC1)(C=O)OC c1(SCC)cnc(O)c(C(=O)NCCCCCCN(C(=O)C(O)CSC)C)c1 C(=O)(CCC(=O)N(C)C(C)C)NCC1OCC(CNC(CCC#C)=O)C1 Cc1nc2c(C(=O)NCC3CCCC(NC(=O)CP(C)(C)=O)C3)cccc2o1 C1(O)(C(=O)NCC(C2CCCCC2)NC(CC(C)=C(C)C)=O)CCSCC1 c1(C(C(N2C(CN(C(C(CC)OC)=O)C3CC3)CCC2)=O)C)c(F)cccc1F C1(F)(C(=O)NCC2(NC(C3COCCC3(F)F)=O)CC2)CC2(CCC2)C1 C(C(C)C(F)C(=O)NCc1c(C)nnn1CC)NC(c1ncn(CC)c1)=O c1(CC(=O)NCC(C2CCC2)NC(=O)Cc2csc(S)n2)ccccc1F c1(CC(C(=O)OCC)N2CCCC2C2CCCCC2)cc(Cl)sc1Cl C=CC1(CC(=O)NCc2coc(CC)n2)CN(C(C2CCC2C=O)=O)C1.O n1(CCN)ncc(C(=O)NC(Cc2ccccc2)CCc2nn[nH]n2)n1 CCC(CC)C(=O)N1CCC(C)C1C(=O)NCC=CCOC C(=O)(CCC[N+](=O)[O-])NC(C1CCN(C(=O)CNC(N2CCCC2)=O)C1)C Cc1cc(C(=O)NC2CC2C)c(N)c(Cl)c1.C1(C(=O)N)CS(=O)(=O)C1 CCCC(C)(C)C(=O)N(CC(C)(C)NC(c1ccn(-c2ccccc2C)n1)=O)C C1(NC(C(C=C=C)C)=O)CCC12CN(C(c1cc(C(C)(C)C)oc1C)=O)C2 c1(C=O)ccccc1.C(=O)(C(N)C(C)O)N(CC(N1CC(C=O)C1)=O)C.C c1(C(N2CC(CNC(C(CC)F)=O)C(O)C2)=O)cc(C(=O)OC)cc(O)c1 Cc1c(NCC2(CC3CCN(c4ccncn4)CC3)CC2)ncnc1NC(C)C CC1CC(C(=O)NC2CCCC2CC(N2CC3(CCC3O)C2)=O)=NO1 C12(C(N3C(C)(C(=O)NCc4cn(C)nn4)C=CC3)=O)CCCC1C2(F)F c1(NC(c2c(CCCC)ocn2)=O)ccc(Cl)c(S(=O)(=O)N(C)C)c1 C1(C=O)CC2CCC(C1)C2O.c1(CC)ccc(C(=O)N(CCC)CC)c(F)c1.N c1(CC=O)cc(C)cc(C)c1.C1(C=O)(OCC)CCCCC1.CC(C)(O)C.N C1(c2n(CC)nnn2)(NC(C)CSC)CCC2(CCCCC2)C1 C12(C(N3CC(CNC(C(C)NC(C)=O)=O)C3)=O)CCC(F)(CC1)C2 C(=O)(C#CC(C)(C)CNC(c1nccc2[nH]ccc12)=O)N1C(C)CN(C)CC1 CC1CN(C(c2n[nH]c(C(C)(C)C)n2)=O)CCC1CNC(C1CSCN1C)=O c1(CC)ccoc1C(=O)NCC(C)N(C(=O)CCc1cnco1)C Cc1ccc(OC(F)F)c(CNC(=NCC2CC2)NC(C)C)c1.OC(F)(F)F c1(C(=O)NC2C(C)N(C(c3cc[n+]([O-])cc3)=O)CCC2)cnc2c(c1)CCCC2 N1(C(C(CC)(C)OC)=O)CC(CNC(c2ccc(C)c(O)n2)=O)C2(CCC2)C1 c1ccc(Cl)cc1Cl.C1(C2(N(C(=O)C3=CCC3)C)CC2)CCCCN1C(=O)CO C(=O)(C(O)C1CCc2ccccc21)N(CC(=O)NC)CC=C CC(C(=O)NCC12CC(F)(C1)C2)(C1CCC1)NC(c1ccsc1)=O c1ccc2c(c1)CCN(C(C1CC1C)=O)C2.c1(OCC)cc(C(=O)N)ccn1.C C1(CCCNC(C2(CC)CC2)=O)CN(C(C2CCNC(=O)C2)=O)CCO1 c1(C(C(=O)NCc2cccs2)N(C)CCOC(C)(C)C)ccc(F)cc1I C1(NC(=O)C2CC2)COC2(CCN(C(=O)Cc3ccc(Cl)cn3)CC2)C1 c1(C(=O)NC(CC(C)NC(c2ccoc2)=O)C)cc(P(C)(C)=O)ccn1 C1(CN(C(C(C)CN2CCOCC2)=O)C)CCN(C(C2(C)CC3(CC3)C2)=O)CC1 C(C1CCCCCC1)=CC(=O)NC1CN(C(c2c(C)[nH]c(=N)s2)=O)C(C)C1 O=C(CC(C1CC1)C1CC1)NCC1(C(=O)NC)CCCC1.C1C=CCC1 C1(C2CCN(C(c3cc(OC)n[nH]3)=O)CC2)(NC(c2nc(C(C)=O)sc2)=O)CC1 N1(C(C2(C)CCOC2)=O)CC(NC(=O)Cc2noc3ccccc23)C2(CCC2)C1 C(=O)(N=c1[nH]n(C)c2ncccc12)c1c2ccc(C)cc2[nH]c1 C12(NC(c3ncc[nH]c3=O)=O)CCN(C(c3cccc(F)c3C(F)F)=O)CC1C2 N1(C(CCSCC)=O)CCC2(CC2)CC1C(=O)NCC(C)CC1CCC1 S(=O)(=O)(CC(=O)N(C)CC1COCCN1C(=O)CCNC(N)=O)NC CC1(C)CN(Cc2ncc[nH]2)CCC1NC(c1cc(Br)ncc1Br)=O c1(NCC(CC)C2CCC2)cc(=NCCNC(C)=O)[nH]cn1 N1(C(c2c(C(C)C)occ2)=O)CCC(NC(C2CC2CF)=O)C(C)(C)C1 C1(C(N2CCN(CC)C(C)C2)=O)CC2(CCC2)CN1C(=O)CCCCCF C(=O)(C1=CC2C=CC(C1)C2)NCC1CCN(C(CCCC)=O)CC1O N1(C(CCn2ccc(C)n2)=O)CCN(C(c2ccc(C#N)[nH]2)=O)CC1C1CC1 C1(CCC)CN(C(c2sccc2CO)=O)CCN1C(C1CC(F)(F)CS1)=O c1(OC)cncc(C(N2CC(NC(=O)CCNC(c3cnoc3)=O)C2)=O)c1 C#CC1CCN(C(C2CC(O)CN2C(c2cccc(N(C)C)c2)=O)=O)CC1 CC1=C(C(=O)N(C)CC2CCCN(C(c3[nH]ccc3C)=O)C2)S(=O)(=O)CCO1 CCC(C)(CNC(c1occc1CN(C(c1ccccc1)C(=O)O)C)=O)OC C1(C#N)(C(=O)NCCn2ccc(C(NOCCCOCC)=O)c2)CC(=O)C1 O=C(CCC(=O)N1CCOCC1)NC1C=CCN(c2ncccn2)C1 C12(NC(c3nccc(C)n3)=O)CCOCC1CN(C(C1(O)CC(F)(F)C1)=O)C2 Cc1ccnc2c(C(=O)NC3(CO)CN(C(c4cnn(C(C)C)n4)=O)C3)cnn12 C1(CNC(C(C)N(C(c2cc(CO)on2)=O)CC)=O)CC2(CC2)CO1 N1(C(C2=C(C)OCC2)=O)CCC(C2CCN(C3CCCc4ccc(Br)cc43)C2)CC1 c1(C(=O)NCC(CO)NC(COC(C)=O)=O)ccc2c(c1)CC(C)O2 N1(C(C(C)OC2CC2)=O)CCC=C(C(=O)NCCC(C2CC2)C2CC2)C1 Cc1cn2cc(C(=O)NCCN(C)C(C3CC3c3ccn(C)c3)=O)sc2n1 CC1(C(N2CC=CC(NC(c3cc(Cl)nc(Cl)c3)=O)C2)=O)COC(=O)OC1 C1(C(=O)NCC(C)(C)NC(C(C=C)OC)=O)CC2COCC2C1 C(=O)(CC(C)(C)C(=O)NC1CC2(C1)CN(C(C1CCC1OC)=O)C2)OC N1(C(c2c(C)csc2)=O)CCCC(CN(C)C(C2CC3CC3C2)=O)C1 N1(C(CCC#C)=O)CC(NC(=O)CCOc2ccccc2C(C)C)CCC(O)C1 CN1CCCC(N(C(=O)C(Cn2cncn2)NC(c2ccc(F)cc2)=O)C)C1 C12(CNC(c3cnc(CCC)s3)=O)CCC1CN(C(=O)C=NOC)C2 C1(C(N2CCC(c3nc(N(C)C)n[nH]3)CC2)=O)(CC)CCCCN1 N1(C(c2c(OC)c(F)ncc2)=O)CCCN(C(c2ccc(Cl)cc2)=O)CC1CO N1(C(CCC)=O)CCC2CN(Cc3ccn(C)n3)CC12 N1(C(c2c(COC)noc2)=O)CC2CC(C1)N(C(=O)Cc1ccno1)C2 Cc1ccnc2nc(C(=O)NCC3CC(O)CN3C(=O)CCC3CC3(F)F)nn12 c1(OC)ccc(O)cc1C(=O)N.C1(O)(CC)CN(C(=O)CC2CC(C)C2)C1 Cc1ccccc1C1CC(C)N(C(=O)CCc2cn(C)cn2)C1 CC1(C)CC(C)(C(=O)NC(CO)C2CC2)CN1C(c1ccccc1Cl)=O Cc1ncc(CC=O)s1.N12CCCC1C1(CC1)C2=O.C1(C=O)CN(C=O)C1.N CS(=O)(=O)CC(=O)NC(C1CCCC1)CNC(c1cc(O)cs1)=O N1(C(c2n(CC)ncn2)=O)CCC(CO)C(NC(c2ncc(N(C)C)cn2)=O)C1 c1(-c2cn(C(C(CC)C)COC)nn2)ccc(Br)c(O)c1 C(C(O)C(=O)NC1(C)CN(C(=O)CCCC2CCC2)C1)SC C1(CNC(c2cccc(NC)n2)=O)CN(C(=O)CC)CC(C)(C)C1.C(N)=O N1(C(C2N(C(CNC(c3ccc(C)nc3)=O)=O)CCC2)=O)CCC(O)(CF)CC1 c1(C(=O)NCC(CNC(C(CCC#C)O)=O)F)sc2ccc(C)cc2c1C C1(CC)COC(C)CN1C(=O)C=CC1CCN(C(=O)CC=C(C)C)CC1 c1(CC)cc(OC)cc(C(=O)N)c1.c1(C=O)cccc(C(C)C)c1.C1CC1.C C1(C(N(CCC(=O)NC)C)=O)CCCN(C(=O)C(C)(Cl)Cl)C1 C1(F)(CNC(c2cc(C)sn2)=O)CCCN(C(=O)CC2CCC(F)(F)CC2)CC1 C1(CC=O)CCN(C)C1=O.C(=O)(C(C)(C)CN(C)C)N1CC(CC=C)C1.N CCS(=O)(=O)Cc1cn(CC(C)(C)CC2CCOC2)nn1.C1CCC(=O)O1 Cc1nn(C)c2c(N3CCC(C)(CO)C3)nc(=NCC(Cl)Cl)[nH]c12 CC(CN(C)C)CCC(=O)NC1C2CC1N(C(=O)CC1CCCO1)C2 C#CCCCCCC(=O)N(C1CCCCCC1)CCNC(=O)C(CC)OC Cc1cccc(C=O)n1.c1(C(N(CCC)C(C)C)=O)cc(C(F)(F)F)cn1C.N N1(C(=O)CC2CCCC2O)CCCC2(CCCN2C(c2ccc(O)nc2Cl)=O)C1 c1(CCCCC)ccc(C(=O)NC2CCC(C)C2)o1.C1(C(=O)N)(C=O)CC1 N1(C(C2(CC)CC2)=O)CC(C2CCCN(C(=O)C(C)Nc3ccc(Br)cc3)C2)C1 N1(C(C(c2ccc(C)o2)C)=O)CCN(C(=O)CC(C)n2cccn2)CC(C)C1 C12(CNC(C(C)SCC)=O)CCCC(CN1C(c1cc3ccccc3[nH]1)=O)C2 C1(C(=O)NC)CCCC1N=c1[nH]c(=NCCOC2CCCC2)[nH]c2cccc(F)c12 C(=O)(CCC(F)(F)C(F)(F)F)N.CCCC(C)NC(=O)COc1ccn(C)n1 N1(C(C(C)SC)=O)CCC(C(C)NCC(=O)Nc2ccncc2)C1 c1(C(c2nnnn2CC(F)F)NC2(C)CCSC2)c(F)cccc1F N1(C(c2cccc(C(C)C)n2)=O)CC(NC(c2cnn(C3CC3)c2)=O)CC(C)C1 c1(OC)c(CC(N2CC(NC(C3CC(C)C3)=O)C3(CC3)C2)=O)cccc1Br C(C)(CC(=O)NCC(n1cc(Cn2cnc(-c3ccccc3)c2)nn1)C)SC C1(CNC(CSCC)=O)CC2COCC2N1C(c1ccc(Cl)c(F)c1O)=O c1(OCCN(C)C(C2CN(CC(C)(C)O)C2)=O)ccc(C(C)(C)C)cc1 C(C)(C)(CC(C)(C)O)NC(C(C1CN(C(CC(CC)C)=O)C1)OC)=O C1(CC(=O)N)COCC2(CCC2)O1.CC(C(=O)NCCCN(CCC)C)C(F)F c1(OC)ccnc(OC)c1C(=O)NC1CC(NC(=O)C(C)C(C)(C)C)C1 c1(CC(C(=O)OCC=CBr)O)c(F)cccc1Cl c1(OC)cc(C(N2CC(F)CC2CNC(C23COCC2C3)=O)=O)c(F)cn1 N1(C(COCc2n(C)ncc2)=O)CCCC12CN1CCC2CC1 CC(CCC(=O)NCCC(C)CCNC(c1cncc(C2CC2)c1)=O)N(C)C C1(CNC(CCOCCCOC)=O)CCC(C)CN1C(c1scc(C)c1C)=O c1(NC(C(CCC)C)C)cc(NCc2cncnc2)nc(C)n1 c1(NC(c2nc(C(C)NC(C3CCCOC3)=O)oc2)=O)cc(C#N)ccc1O C1(C(=O)NCCCCCN(C)C(C2C(F)(F)C23CC3)=O)COCC1(C)C c1(C(=O)NC(CNC(c2c(C)n(C(C)(C)C)nc2)=O)C)ccc2c(n1)CCO2 C1(NC(C=COCC)=O)CN(C(c2cc(OC(F)F)n(C)n2)=O)C(C)(CC)C1 C1(C(=O)NC(CNC(C(C)N(C)C)=O)CO)CC2CC1CC2(F)F c1(C(N2CC(NC(c3c(CC)c[nH]c3)=O)C(C)C2)=O)ccccc1C#CC1CC1 CCCCC(C)CCC(=O)NC(CN(C)C)C(=O)NC(CO)C(=O)N(C)C c1(NC(=O)NC2(C#C)CCCC2)cc(C(=O)NC)cc(Br)n1 c1(C(C)C)nnnn1CC(=O)NC(C)CNC(c1nccn1C(F)(F)F)=O C1(C(N(CCC(=O)OC)C)=O)CC(N(C)C)CCO1.C12CC(C1)N2 Cc1nncc(C(=O)NC2CCCCC2C)c1C.C1(C(F)(F)F)(C=O)CCC1.N c1(N2CCC(C(CC)C)CC2)ncnn2c(C#N)ccc12 C1(C(N2CC(NC)C2)=O)C2CC1(c1ccc(OC(F)F)cc1)CO2 N1(C(c2cc(C)c(C)o2)=O)CC(CNC(C2(C3CC3)CCC2)=O)CCC1C O=S(=O)(C1CCCN(c2cc(C(F)F)nc(Cl)n2)C1)N1CCCC1 C=CC1(CC(=O)N(C2CN(C3CC3)C2)C)CN(C(=O)CC2COC(=O)C2)C1 c1(C(N2C(C)CC(NC(Cc3ccc(C(C)=O)cc3)=O)C2)=O)ccc(F)c(Cl)c1 C1(C(N(C2CN(C(c3cc(COC)no3)=O)C2)C)=O)COc2ccc(Cl)cc2C1 N1(CC)CC(C(N2CCCC(C(=O)Nc3ccccc3)C2)=O)CC1=O C1(C(N(CCC)C)=O)CCCCN1C(=O)C1CC1.C(C)(C)(C=O)OCC.N N1(C(CC(C=C)C)=O)CCC2(CC1)CC(C)N(C(=O)C=Cc1cncs1)C2 CCC(C(=O)NCC(C)(C1CC1)NC(=O)C(C)=C1CCCC1)SC C(CC(C)C(=O)NC(CNC(c1cc(CCCO)on1)=O)CO)OC c1(CNC(C(=O)NCC(C2CCNCC2)C)=O)cccc2[nH]ccc12 c1(C(=O)NC2CCCC(NC(COCCCC(C)C)=O)C2)cncc2[nH]ccc12 CCC(CC(=O)NC1(CO)CCCN(C(=O)CC)C1)C(F)F.C(=O)(C(C)(C)C)N n1(CC(N2C(CCNC(C=COCC)=O)CCCC2)=O)cccc([N+](=O)[O-])c1=O c1(C(C(=O)N(C(C)CNC(C2CCCC2)=O)CC)=O)ccc(F)c(F)c1 CCC(CNC(=O)CCC(C)NC(C1C=CC1C(=O)OC)=O)(CC)CO N1(C(C=C(C)C)=O)CC(C)(C(=O)NC2CC(C(F)F)C2)C1 N1(C(c2ccc(Cl)cc2C(F)(F)F)=O)CC2CN(C(C3CCC3)=O)C2C1 CN1CCC(F)(CNC(C2(C)CCN(C(c3nc(=N)cc[nH]3)=O)C2)=O)C1 C1(NC(CC2N(C)CCC2)=O)CC2(CCCCN2C(=O)CCC2CCCCO2)C1 C1(NC(C(C)N(C(C2CC(F)(F)C2)=O)CC)=O)CCCCC1(C)C C1COCCC1C=O.c1ccccc1C1(C(F)(F)F)CC1.CC(C)(C)OC=O C1(NC(C(C)Oc2ccccn2)=O)CN(C(C2CCCC2)=O)C2(CCCCC2)C1 N1(C(CC2C(C)C2)=O)CCC2(CCN(C(=O)C(c3cscn3)N(C)C)C2)C1 C1(C(N(C(C)CNC(c2cnc(C)s2)=O)CC)=O)CCc2nn[nH]c2C1 c1(C(N2CCCCC2Cc2ccccc2Cl)=O)ccn2cccc2c1 C1(CC=O)CC(O)C12CCC2.CC1CC=CCC1C(=O)N(C)CC1(C)CC1 c1(NC(C2CC23CCN(C(c2ncccc2O)=O)C3)=O)ccc2ccncc2c1 C1(C(=O)NCCCCNC(=O)CC2NC(=O)CNC2=O)(OC)CCCCCC1 C1(NC(COCC(=O)OC)=O)CCC(C(=O)NC2CCCOC2)C1 c1(N(C)C)ccc(N)c(C(N2CCCC2)=O)c1.C(=O)(CCN(CC(F)(F)F)C)N c1(C(N2CCC(CC3CCC3)C2)=O)[nH]nc2ncc(-c3cc(F)ncc3F)cc12 C1(NC(C2CCN(C)CC2)=O)CCCCN(C(C2C3CC4C(C3)C24)=O)CC1 N1(C(C=CCCC)=O)CCC2(C1)c1[nH]cnc1CCN2C(c1cc(C)c(C)o1)=O c1(OC)ccc(C(C)NC(=O)C(c2ccc(-c3nn[nH]n3)cc2)C)cc1Br Cc1c(C2N(C)CCN(c3ncc(C4CC4)cn3)C2)[nH]c2ccccc12 C1(CN(C(CN(C2CC2)CC)=O)C)CCCN(C(=O)CC2CC(S)C2)C1 N1(C(C(C)=C2CCC2)=O)CCC(C)C(C)C1.n1(C2(C=O)CC2)cc(Cl)cn1.N c1(C(N2CCN(C(CN(CC)CC)=O)C(CC(F)F)C2)=O)cc2cccnc2[nH]1 Cc1cc(C)c(C(=O)NC(CO)CCCCNC(C2(C)CC=CCO2)=O)cc1C c1(C(N(C2C(C)CCC2)CC2CC2)=O)ncc(O)cc1F C(c1ccc2[nH]ccc2c1)=CC(=O)N(CCNC(=O)CCC(C)(C)F)CC c1(CC)ccc(Oc2ccc(C(C)(C)C)cc2)cc1.C1(C#N)C(=O)CS1 c1(CC)cccnc1-c1nc(C2CN(C)CCO2)nn1Cc1cccc(F)c1 Cc1nc2ccc(C(=O)NC34CCN(C(=O)Cc5csc(=N)[nH]5)CC3C4)cc2[nH]1 N1(C(C(c2ccccc2)C)=O)CC2CC1CN2Cc1ccc(C(N)=O)cc1 c1(C(N(CC=O)C(N2CCCC2)=O)=O)ccccc1.C1CC(=C2CCC2)C1.O S(=O)(=O)(c1ccc(Br)cc1NC)NC1CCN(C(CCSC)=O)C1.C1(C)CC1 CC1(C)CC(CC(=O)NCc2ccc(C)cc2)CO1.C(=O)CCn1ccnc1.N Cc1ccc(C(C)CC(=O)NC2CC2NC(=O)Cc2conc2C)cc1 N(C(=NCC)NC1CCN(C=O)CC1)CCOC.C(C)(C)C.C(CC1CC1)N C1(C(=O)NC(C(N2CCC(C)(CC)C2)=O)CC2CC2)CC2CCCC2C1 N1(C(C23CC(NCc4cc(Br)c[nH]4)(C2)C3)=O)CCCCC1c1ccccc1 CCCCCCCCCCCC(=O)N1CC(F)(C(=O)Nc2cccc(C)c2Br)C1 N1(C(C2(COC)CN(C(=O)CC3CC=CCN3C)C2)=O)CCCCCC1C c1(C(=O)Nc2cc(F)c(F)cc2C(F)F)cc2ccc(Br)cn2n1 CC1CCN(C(=O)Cn2cnnc2)CC1NC(c1ccc(OCCF)cn1)=O Cc1ccc(C(N)C(N2CCC(NC(c3ccnc(OC4CC4)c3)=O)C2)=O)cc1 c1(C(=O)NC2CCC2O)ccc2scc(Br)c2c1 N(C(=NCCc1ccc(Cl)nc1)NCC1(C)CCC(C)CC1)C(CC)C N1(C(C(C)(C)Br)=O)CCC(F)(CNC(c2ccccc2)=O)CC1.C(C)(C)C.O c1(C(N2CC(NC(CC=C(C)C)=O)C(C)C2)=O)ccc(=O)n(C2CC2)c1 C=CC1(CC(=O)NC2CCCC2COC)CN(C(=O)CN)C1.c1ccccn1 c1(N2C(CN(C(CN(C)Cc3ccccc3)=O)C)CCC2)ccnc2ncnn12 c1(C(=O)NC2(CCC(=O)NC(CCCC)C)CCCC2)ncc(C)cc1C C1(C(=O)NC2CC(CNC(CC(C)SC)=O)C2)Cc2c(F)cccc2O1 Cc1cccc(Br)c1C(C=O)NC(=O)COCCN(C)C.C1CCC(=O)N1 c1(CN2CCCC(c3n(C)ncc3)C2)cccc(F)c1C(=O)O c1(C(C)O)ccc(CNC(c2nnnn2Cc2ccco2)C2(C)CCC2)cc1 N1(C(c2cc(OC)nn2C)=O)CCC2(C1)CN(C(C1CCCC1(F)F)=O)C2 c1(C(=O)NC2CCC(NC(c3ccc(C)o3)=O)C2)cnn(C)c1S(N)(=O)=O C(=O)(C1Cc2ccc(F)cc21)NC1(C)CCCN(C(C(C)OCCOC)=O)C1 C1(COC)(CNC(=O)Cc2ccco2)CCCN1C(C1CCSC1)=O C1(CNC(CCOCCN(C)C)=O)CCCCN1C(c1cccnc1)=O c1(C(N(CCC)C(C)C)=O)cc2cc(-c3c[nH]nc3C)ccc2o1 C(CNC(=O)C(C(C)C)n1ccnc1)(C(C)(C)C)NC(Cc1c(C)ocn1)=O C1(C(=O)NCC(CNC(c2cc(N(C)C)ncc2)=O)O)CC2C=CCC(C1)C2 C(C)(C)(CCCF)NC(C1(CC)CN(C(=O)CCn2ccnc2C)C1)=O N1(C(c2c(C)nsc2)=O)CCCC(C)(CNC(C2CCC(O)CC2)=O)C1 CC1(C)OCCOC1CNC(c1nnnn1CC(F)F)CCC1CCCC1 C1(CNC(c2cc(C)nn2C)=O)CN(C(=O)COCCCN=[N+]=[N-])CCN1C C(=O)(C[SH](=O)=O)NCCCC.C(=O)CCC=O.C(C)(C)(C)OC.C1CC1.N C1(C=C)(C(N2CCC(CC#C)C2)=O)CCN(C(c2cc(C)ncn2)=O)C1 C#CC1(O)CCN(C(C)C(=O)N(C2CCN(C(=O)C=C(Cl)Cl)C2)CC)CC1 C1(CCC(=O)N(C(C(N)=O)C2CCCC2)C)CCCCN(C(=O)C)C1.C1CC1.O N1(C(c2ccc(NC(N(C3CCCC3)C)=O)cc2)=O)CCNC(=O)C1(C)C Cc1ccncc1C(=O)NCCCCC1CN(C(c2coc(N(C)C)n2)=O)C1 C1(C(c2nnnn2C(C)C)(C)NC2(COC)CCOC2)CC2CCC1CC2 C(CCC(C(=O)N(C)Cc1cc(C)on1)NC(=O)CC1COCCO1)OC c1(OCC)cccc(C(=O)N(C)CC2CCCN(C(=O)C(O)C3CC3)C2)c1 c1(CC2C(CNC(C(N3CCCC(CC)C3)=O)=O)C2)nc2ccccc2s1 C1(C(=O)NCC2(C#C)CCC2)CC12CCN(C(=O)C=Cc1cncn1C)C2 Cc1cccc(C(=O)NC2CC3C(NC(=O)C(C)(O)C4CCC4)C3C2)c1C c12cc(C)cc(C)c1NC(=O)C(=O)NC2.C1(CC)CCOC1C(=O)OC c1(C(=O)NCC(C)CN(C(=O)C=CS(C)(=O)=O)C)cccn2nnnc12 C1(N(C(C(C2CCN(C(C3CC4C=CC3O4)=O)CC2)C)=O)C)CCC(F)(F)C1 c1(C=O)cc(F)cc(Cl)c1.C1(NC(Cc2nc(CC)sc2)=O)CCCCC1C.N N1(C(c2c(C)n(CC3CC3)cc2)=O)CCC2(CCCN2C(=O)CCC2CC2)CC1 CC(C)CC(C)(C)C(=O)N1CC(NC(c2cccc(Cl)c2Cl)=O)C(C)C1 C1(C(=O)NC)CCN(C(=O)CC2(NC(C3CCCN3C)=O)CC2)C1 N1(C=O)CCN(C(=O)C(C)N2CCC2)CC1.c1(C(C)OC)nc(CCC=C)cs1 C1(CNC(CC(CCC)O)=O)CN(C(c2cccc(O)c2F)=O)CCC12CCC2 CCC(C)(C)C(O)C(=O)NC(C)(CNC(C1CC1C1CCCCC1)=O)C1CC1 C1(NC(c2c(C)cno2)=O)CC2CC(C1)N(C(C1(n3cccc3)CCCC1)=O)C2 CN1C(=O)CCC1C(=O)NC1CCC(NC(C2CCNC(=O)C2)=O)CC1 c1(C=O)cc2c(ncn2C)s1.Cc1nccc(C(=O)NCC2(F)CC(C)C2)n1 C1(COC)CCN(C(C2CCN(C)C2=O)=O)CC1.C1(C=O)CCCNS1(=O)=O.N N1(C(C2CC(NC(C3CC(C#N)(OC)C3)=O)C2)=O)CC(C)(C)C2CCCC12 C1(CNC(C2(SCC)CC2)=O)(C)CCN(C(c2cccc(F)c2)=O)C1 Cc1ccc(CCCC(=O)NCCC2(C)CCN(C(c3csc(Cl)c3)=O)C2)cc1 N1(C(C)=O)CCOCC1C(N1CC(F)(C)C1)=O.c1(C2(C=O)CC2)ccsc1.N Cc1nc2nnnn2c(C)c1CCC(=O)N(CCCN(C)C(C1(C)CC1F)=O)C n1(C(C)C)nccc1C(=O)N(CCCN(C)C(C1CCN(C)C1)=O)C c1(C(=O)NC2C3CN(C(C(C)C(C)(C)C)=O)CC32)ccc2c(n1)COCC2 C1(NC(CC(CC)NC(=O)CN=[N+]=[N-])=O)CCOCC1(C)C Cc1ccc2[nH]c(C(=O)NCC3CC4CC4N3C(=O)C(C)C(F)(F)F)cc2c1 C(=O)(C1CCc2ccccc21)NC1C(NC(C(N=S(C)(C)=O)=O)=O)C1 C1(NC(C(C)CC(F)F)=O)CCCCN(C(c2cc3occc3n2C)=O)CC1 CCC(CC(C)C)C(=O)NC(C)(CNC(c1csc(C(F)(F)F)c1)=O)CO C1(C2CCCOC2)CC1.c1(CCNC(C2(OC)CCC2)=O)n[nH]cc1C(=O)N C(=O)(CCS(=O)(=O)C(F)(F)F)N1CCCC1.C1(CC(=O)N)CCC(C2CC2)O1 N1(C(C2C(=C)C2)=O)CCC(NC(C2CC3CCCC(C2)C3)=O)C12CCC2 N1(C(CCSc2n(C)nnn2)=O)C2CCC1C(CNC(=O)Cc1c[nH]nc1O)C2 C(=O)(C1=CCCSC1)NCC1N(C(CNC(C)=O)=O)CC1 N1(C(C(C)c2ccco2)=O)CCC(C)(CNC(=O)C(O)C2CCC2)C1 N1(C(C(CC=C)C(C)C)=O)C(C)CC2CN(C(=O)CCCN3CCCC3)CC12 c1(C(N(CC(O)CN(C)C(C2CCC(O)CC2)=O)C)=O)cccc2nsnc12 C1(NC(=O)NC(CC)COC)CCCN(C(=O)N(C)C)C1 C1(CN(C(c2cn(C3CC3)nn2)C)C)Cc2ccccc2O1 c1(C(=O)NC2CN(C(=O)C=Cc3ccc[nH]3)CC2O)cccc(Br)c1[N+](=O)[O-] N1(C(c2ccc(C(C)=O)[nH]2)=O)CCCCC(N(C(=O)C=Cc2cscn2)C)C1 Fc1ccc(F)c(-c2ccc(CNCc3cc(I)ccc3)cn2)c1.CC(F)(F)F.O Cc1cc2ccc(C(=O)NC(C)CNC(=O)C(c3ccc(F)cc3)CO)cn2c1 Cc1ccc2ncc(C(=O)NC(C)CC(C)NC(=O)CN(C3CCC3)C)n2c1 CC(C)CC(C(=O)NCC1COCCN1C(c1sccc1Br)=O)N(C)C CC1CCN(C(c2ncccc2O)=O)CCN1C(=O)Cc1cncn1C Cc1ccc2c(c1)CCN(c1ccnc(NCCNC(C3CCC3)=O)n1)C2 C(=O)(C#CC1CCCCO1)N1CCCC(C)(CNC(c2c(COC)ccs2)=O)C1 CCCC(C)(O)CC(=O)NCC1=CCN(C(C2(c3ccccc3C)CC2)=O)CC1 CCCS(=O)(=O)CC(=O)N1CC(NC(=O)C(F)(F)c2csc(C)c2)C(F)C1 Cc1nccn1CCN(C(=O)C(C)CNC(=O)CSc1cn[nH]c1)C c1(C(=O)NCC2CC(F)(CNC(C(C)c3ccsc3)=O)C2)ncccc1F CC1CN(C)CC(C(N2CC(C)C2C(=O)NCC2(F)CC2)=O)O1 c1(-n2cc(C(CCC)NC(=O)CC(C)CF)nn2)ccc(N)c(C)c1 S(=O)(=O)(c1ccc(NCC2CC2(Cl)Cl)cc1Br)N1CCC(C=C)(CO)CC1 C1(=CC(=O)NC2CCN(C(c3cc(C)n(CCO)n3)=O)C2C)CN2CCC1CC2 c1(C(=O)NCC2C(NC(CC3CCCN(C)C3)=O)CCC2)c([N+](=O)[O-])cnn1C C1(OC)CC(C)CN(C(=O)CC2CC(NC(=O)CCCNC(C)=O)C2)C1 c1(C(=O)NC2C(C)N(C(=O)COCCO)CCC2)cnc2c(Cl)cccn12 c1(C(N(CC(CNC(c2cc(CC)no2)=O)(C)C)C)=O)cccc(C=O)c1 C(=O)(C(C1(O)CCC1)NC(=O)CCNC(=O)CO)NCC(C)O C(C(F)(C(=O)NCCP(C)(C)=O)C(C)C)NC(C(CC)OC)=O Cc1csc2ccc(C(N3CCC(NC(c4cccc(O)n4)=O)C3(C)C)=O)cc12 c1(C(=O)O)nccnc1C(N1CCN(Cc2cn(C3CCOC3)nn2)CC1)=O Cc1cc(C)[nH]c(=NCC2CC3CCC(C2)N3C(=O)Cc2cnoc2)n1 c1(C(=O)NC2CC(NC(c3c(C)n[nH]c3)=O)C(O)C2)ccc2cccc(F)c2n1 Cc1cc(F)c([N+](=O)[O-])cc1C(N1C(C(N2CC3CCCC3C2)=O)CC2CC12)=O N1(C(C(C)(C)CF)=O)CC2CCCC(NC(c3cncc(F)c3)=O)(C2)C1 c1(OCCNC(C)C(C)(C)O)cccc(Cl)c1Cl C1(C)CC(F)(F)CN1C(=O)Cn1nnc(=N)[nH]1.Cc1cnc(C(=O)N)c(F)c1 c1(-c2ccc(OC)cc2)ccc(SCC(O)COc2ccc(CO)cc2)c(O)n1 C1(C(=O)NC)CCC(C2CC2)CC1.C1(F)CN(C(=O)C(=Cc2c[nH]cn2)F)C1 Cc1ccnn1C(C)C(=O)N1CC(C(C(=O)OC(C)(C)C)N(C)C)C1 N#Cc1ccc(Br)c(C(N2CCC3CN(C(c4c(Br)cncc4Br)=O)CC23)=O)c1 C(=O)(C1CCc2nccn21)NCCCCCN(C(c1cc(OC)c(Cl)s1)=O)C c1(C(=O)NCC(CC=C)NC(=O)C(=Cc2ccccn2)C)ccccc1O c1(C(=O)NCC2(F)CCC(NC(CCCC)=O)C2)cc(F)cc2cc[nH]c12 C1(NC(C(C(C)C)NC=O)=O)CN(C(c2ccc3occc3n2)=O)CC2(CC2)C1 c1(NC2CC(CNC(C(C(C)O)C)=O)C2)ccc(S(C)(=O)=O)cn1 C#Cc1cccc(C(N2CCC(C)(CC(=O)NC3CCCC3CF)C2)=O)c1 C=CCCC(C(=O)NCCc1ccccn1)NC(=O)C(O)C=C N1(C(Cc2cc(C)no2)=O)C(C)CN(C(=O)C(N2C(=O)CCC2=O)C)CC1C C1(C)CC(F)(F)CN1C(=O)C=O.Cc1ccc(F)cc1C(=O)N.CC(F)F.C Cc1cc(N)cnc1C(N1CCC(C(=O)NCC2CCCCN2C)(CO)C1)=O N#Cc1cc(S(=O)(=O)NC2CCCN2CCCO)ccc1NCCCCO C1(CNC(C(CC)(C)C)=O)(CNC(c2c[nH]cc2Br)=O)CC2CCCC2C1 N1(C(CC(C)CF)=O)CC(F)(F)CC1(C)CNC(=O)C.C(=O)(C(F)(F)F)N c1(OC)ccc([N+](=O)[O-])cc1SCC(N1CC(CO)C(c2cccc(C)c2)C1)=O c1(C(=O)NC2CC(F)(CNC(C3(C=C)CCC3)=O)C2)n[nH]c(C)c1Cl c1(C(N2CCC(C(=O)NCC(C=C)C)CC2)=O)cccc2ccoc12 CCCCC(C(=O)N1CC(S(C)(=N)=O)C1)NC(c1cnc(OC)nc1)=O N1(c2ccc(Br)nc2)C2CCC1CN(Cc1nocc1Br)C2 C(=O)(C(CCSC)NC(N)=O)NC1(C2N(C(CCOC)=O)CCC2)CC1 N1(C(c2c(C)csn2)=O)CC2CCC(N(C(=O)CC3CC4CC4C3)C)C2C1 N1(C(=O)NCc2ccc(OCCC)nc2)CCCC2(CC2C(=O)O)C1 c1(C(C)OC(C2CN(c3ccc(C#N)cn3)C2)=O)cc(F)c(Cl)cc1Cl CC1(CNC(c2c[nH]c(=O)cn2)=O)CCN(C(C2CCCC(N(C)C)C2)=O)C1 N1(C(=O)OC(C)(C)C)CCC(NC2CCN(C3CC3)C2=O)C12CC2 C#Cc1cc(C(=O)N(CCO)C(c2ccc(Br)s2)C)cc(F)c1 C1(CC)C(C(N2CCC(C)(N(C)C)C2)=O)CCN1C(C1CN(C(C)C)C1)=O C(CC(C)C)(C(=O)N1CC(CCO)C1)ONC(CC1C(C)=NNC1=O)=O Cc1nc2c(s1)CCCC2C(=O)NCCC1CC(NC(c2ccc(F)s2)=O)C1 c1(C(=O)NCC23N(C(CC(C(=O)OC)C)=O)C(CC2)CC3)cc2ccccc2[nH]1 CC(C)CCCCC(=O)N1CCC(C2CC2)(NC(=O)COCC2CCCO2)C1 c1(C(=O)NC2CCN(C(C(CC)=CC)=O)CC2F)cc(Br)cc([N+](=O)[O-])c1 Cc1ccc(C2(NC(=O)CCN3CCOCC3CC(=O)O)CCC2)cc1 c1(CNS(C)(=O)=O)cn(CC(=O)NCc2cncs2)nn1 Cc1cccc(F)c1CC(=O)N(C1CCCC1)CC.C1(CC(=O)N)CCC(C)C1 C1(C(=O)OC)C(O)C(O)CN1C(C)=O.c12ccc(cc1)NC(=O)CN2 CC(O)C(C)(CNC(=O)NC1(C#N)CC1(C)C)Cc1ccccc1 Cc1nc(N(CC(C)CNC(c2ccnc(CO)c2)=O)C)[nH]c(=N)n1 c1(CNC(N2C(C)(C(=O)NC(C(CC)C)CO)CC2)=O)ccc(Cl)cc1Cl c1(-c2cn(CC3N(C(c4cnc(C)n4C)=O)CC3)nn2)cc(F)c(Cl)cc1Cl CN1CCc2ccccc2C(NC(c2csc3ccccc23)C(=O)O)C1=O c1(C(C(=O)OC)NC(C2CC(C)C(C)N2)=O)cc(Br)ccc1Cl c1(C(=O)NCC(C)CNC(C2CCOC2(C)C)=O)cc(N)cc(O)c1 C(C1OCCc2sccc21)N(C(C(C)Sc1ccc(F)c(F)c1)=O)C O=C1COc2cc(C(N3CC4CC4(NC(=O)CN4CCCC4=O)C3)=O)ncc2N1 c1(C(=O)NC(C2CCCN2C(c2csnn2)=O)C)cc(C(N)=O)cs1 N1(C(CSCC#C)=O)CC2CCCC2(CNC(c2ccccc2Br)=O)C1 c1(NC(C2C(NCc3cncc(OC)c3)C2)=O)cncc(Cl)c1C C=CCC(C(=O)OCC)NC(=O)CCN(C(=O)CC1CCCC1)CCO N1(C(CCC(CC)OC)=O)CCC2(CC2)CC1C(=O)NCc1noc(C(C)C)n1 N1(C(c2c(C)c[nH]c2)=O)CC(O)CC1C(N1CCN(CC(F)(F)F)CC1)=O C1(CC)CCC(C(=O)NC2CCC(NC(=O)COCCCN(C)C)C2)O1 c1(C(N(CC(CC)NC(c2cnn(C)c2SC)=O)C)=O)cc2c(s1)CCCCC2 c1(C(N2CCC(C)C2C)=O)csc(S(C)(=O)=O)c1.c1(CC(=O)N)cnccn1 NC(=O)CN=c1[nH]c(=NCC2CCCC23CCC3)c2cccc(F)c2[nH]1 N1(C(C(CSC)O)=O)CCCC(CNC(C2CC=CCC2C)=O)C1 CC(CC(C)(C)C)C(=O)NCC1CN(C)CCN1C(c1ncc(Cl)c(N)c1Cl)=O C1(NC(COC)=O)CCC2(CCCN(C(=O)Cc3ccc(OC)cc3F)C2)C1 C(C)(CCCC(C)C)NC(CNC(c1cc(OC)ns1)=O)=O C12(NC(CNC(=O)NC)=O)CCCC1N(C(c1ccc(O)nc1Cl)=O)CC2 N1(C(C2N(CCC)C(=O)CC2)=O)CC2CC(C1)CN(C(=O)CCc1ccon1)C2 C1(CC)CC(CC(=O)NCC2(CCNC(c3ccccc3Cl)=O)CC2)CCO1 C1(NC(C2(C)CCOCC2)=O)CC1C1CCN(C(C2C(F)(F)C23CC3)=O)CC1 C1(F)(C(N(C)Cc2ccccc2CNC(=O)CCF)=O)CC12CCCCC2 C=CCC(C)(C)CC(=O)NC1CC12CCN(C(=O)CCSC(F)(F)F)C2 N1(CC(=O)NC2CN(C(COCCSC)=O)C(C)(C)C2)Cc2ccccc2C1=O C1(C(N2CCC2)=O)OCCOC1c1ccccc1.C(=O)(COCC(=O)N)OC C#CCCC(O)C(=O)NCCOC1CCN(C(c2c[nH]nc2C(F)(F)F)=O)CC1 C1(O)(C(=O)NC2CN(C(CC=CC)=O)CC2CCC)CC2CCC1C2 c1(C(=O)NCCCCNC(CSC(C)C)=O)nn(CC(F)F)cc1[N+](=O)[O-] C1(C(=O)NCC=CCC(=O)N(C)Cc2cnn[nH]2)CC(C)(C)CN1C c1(C(=O)NCC2(F)CCCN(C(C=CCC)=O)C2)c(Cl)ccc2c[nH]nc12 C1(CC(=O)NC2(C)CCCCC2)CCCS1(=O)=O.C1(C=O)CC1C(F)F.N c1(OC)cc(CS(C)(=O)=O)ccc1NC(=O)C(N1CCSC(C)(C)C1)=O C1(C#N)(NC(Cc2ccc(SC)cc2)=O)CCN(C(c2ccc(Br)cc2I)=O)C1 c1(CC)ccc(C(N2CCCCC2CNC(=O)COC2CCCCC2C)=O)cc1 c1(C(c2nnnn2CCCOC)NC(CC=C)(C)C)ccccc1F CC(C)(C#N)CC(=O)NCCN(C(=O)CC1CNC(=O)C1)CC1CC1 Cc1nn(CC(=O)NCC(CC(C)C)NC(=O)C=Cc2ccccc2)c(C)c1Cl C(=O)(CCCCC(C)CC)Nc1ccc(F)c(CO)c1.C=C1CC2(C1)C(=O)NC2 C1(NC(C2(C(F)(F)F)CC(=C)C2)=O)CCN(C(=O)C=Cc2cc[nH]c2)CC1 C(=O)(CC(C(C)C)NC(c1ccn(C(F)F)n1)=O)N(CC(CC)O)C Cc1ccc(F)c(C(=O)NC2CC(C(C)NC(=O)C(C)N3CC(C)C3)C2)n1 Cc1cc(NC(=O)C(c2ccco2)NC(=O)Cc2ccsc2C)cc(O)c1 N(C1c2ccccc2CC1NC(c1c(Cl)nn(C)c1Cl)=O)C(CC)=O C1CC2CN(C(c3cc(N)nc(Cl)c3)=O)CC12.C(CO)(C(=O)NC)NC(N)=O Cc1sc(C=O)nc1O.N1(CC(C)C)CCN(C(C2(O)CC(F)(F)C2)=O)CC1.N c1(C(=O)NCCC2CCN(C(C3CC4CCC(C3)S4)=O)CC2)c(O)cccc1Cl c1(C(=O)NCC2C(NC(CCC)=O)C2)cccc(C(F)(F)F)c1C C(=O)(C1=CCCSC1)NCC(CNC(c1nn(C)c(C2CCCCC2)c1)=O)F C=CC1(NCc2csc(C)c2OC)CCCCC1 c1(C(N(C2CCN(C(=O)C(F)F)C2)CCC)=O)cnc2nc(O)ccc2c1 N1(C(C23C4C5C6(C)C4C2C6C53)=O)CCC2CC(C)(C)C12.C(=O)C1=COCC1.N Cc1ccc(F)cc1C(N1CC(CNC(C23CCC(F)(CO2)C3)=O)C1)=O C1(CO)(NC(C2CCc3c(ccc(OC)c3)C2)=O)CCCc2ccccc21 C1(C(=O)OCCCN(C)C)CN(Cc2ccccc2)CC1Cc1ccccc1 N1(C(C(COCC)C)=O)CCCC(CO)(NC(c2cc(F)ccc2OC)=O)C1 c1(C(=O)NCC(C)NC(=O)Cn2nccn2)ncn(C(C)C)n1 c1(C2C(C(C)Nc3c(C)n(C4CCNC4)nn3)C2)c(F)cccc1Cl c1(C(=O)NCC2N(C(CCSc3n(C)ccn3)=O)CCC2)cc(Cl)cc(Cl)c1 CCCCCC(O)C(=O)N1CC(C)(C)C1C1CCN(C(=O)CC(O)COC)CC1 c1(OC)ncnc(OC)c1C(N1CCCOC(CNC(C2(O)CCOC2)=O)C1)=O Cc1ncc(N2CCOCC(C(=O)NC(C)Cc3ccccc3Cl)C2)nc1C CCC(C#N)(CC)C(=O)N(CCCCNC(c1cnc(OC(C)C)c(Cl)c1)=O)C Cc1c(Cl)ccnc1C(N1CCOC(CNC(c2cc(N)ccc2Cl)=O)C1)=O CCCC(C(=O)N1CCCCC1CCN(C)C(C1(Br)CC1)=O)NC(C)=O C(=O)C(O)CC(F)(F)F.c1(OCC)ccccc1OCC(=O)NC1CC1.N CC(C(=O)NC)C(C)S(C)(=O)=O.C1CN(C(C2CCC(=O)C2)=O)CCC1(F)F c1(CC(=O)N(C2CN(C(C3CC4C=CC3O4)=O)C2)C)cc(Cl)ccc1[N+](=O)[O-] C(=O)(CC(F)(F)C(F)F)NCC(C)(C)CNC(C1CC12CC2(F)F)=O Cc1nccc(C(=O)NC(C)(CNC(=O)CCOc2ccccc2)CO)c1N N1(C(c2cc(C)cc(O)c2)=O)CC2CC(C1)N(C(=O)Cn1cnc([N+](=O)[O-])c1)C2 c1(C(=O)NC2CCC(NC(c3c(SC)scc3)=O)C2)cccc(C)c1F C(=O)(C(O)CCNC(C1CCCCO1)=O)NCC(NOC)=O C1(C)(C=O)CCCCC1.C(=O)(CCC1CCC1)NCCCNC(=O)OC.N N1(C(C2(NC(C(CC)C#N)=O)CCOCC2)=O)C2CCC1CN(C)C2 C(=O)(C(O)C=C)N(CC)C.C1(COC)(C)CC1C(=O)N(CCC)C.O CCCS(=O)(=O)C(C)C(=O)N1CC(CNC(=O)CC)(OC)C1.CCCCOC N1(C(c2cncc(C)c2)=O)CCCC(C2CN(C(C3(P(C)(C)=O)CC3)=O)C2)C1 c1(C(N2CC(C)(NC(C3CCCS(=O)(=O)C3)=O)C2)=O)cccc2c1COCC2 C1(CNC(C(C)=C2CC2)=O)CC(F)CN1C(=O)C(c1ccc(C)cc1)F Cc1csc(Cl)c1C(=O)NCC1CN(C(=O)CC(C)C2CCCCC2)C1 S(=O)(=O)(c1cc(F)c([N+](=O)[O-])cc1Br)N1CC(C)C(C)(C(=O)OC(C)(C)C)C1 C(=O)(CC(C)C(=O)N1CCCC(NC(c2ccc(C(C)C)c(C)c2)=O)C1C)OC Cc1noc2cc(C(=O)NC3CCCCC3)ccc12.C1(C(=O)N)CC1C(C)(C)C C(C(=O)N1CCC(CNC(C2CCCN2CC)=O)CC1)(C(C)C)SCC C1(C(N2CC(CC(C)NC(=O)CCC3(O)CCC3)C2)=O)CCC(=O)O1 CC1CN(C(=O)CCC(N)=O)CCC1CNC(c1sccc1C#N)=O CCCCCCCC(=O)NCCCCCC(=O)N1CC(Cn2ccnn2)C1 C12(CCNC(C(C)NC(C)=O)=O)CCC(CC1)C2.C1(C=O)SCC=C1C.N N1(C(C2C(OC)(OC)CC2)=O)Cc2occ(C=O)c2C1.C1(C)(CC)CCOC1.N C(=O)(CC1=CCOCC1)NCC1(C)OCCN(C(CCc2cnn(C)n2)=O)C1 CCCC(CC)C(=O)N1CCC(N(C(=O)Cc2ccn(-c3ccccc3)n2)C)C1 C(c1ccc(C)c(C)c1)=CC(=O)N(CCN(C(C1C(CC)OCC1)=O)C)C c1(C(=O)NC23CCN(C(c4cccc(O)c4)=O)CC2C3)cc(Br)n2c1CCC2 c1(C(=O)Nc2cc(C)ccc2)c(N)sc2c1CCC2.C1(C)(CC=O)CC1(F)Cl.N c1(OC)ccc(NC(CCC(C)C)c2nnnn2CCC2(C)CC2)c(Cl)c1 C1(F)(C(=O)NCc2ccn(C)n2)CCN(C(C2CC2F)=O)CC1 Cc1cc(=NCCCC2CC2)[nH]c(=NCCC2COCC(C)O2)[nH]1 c1(NC(C2CC3CC3N2C(c2ccncc2C(F)(F)F)=O)=O)cc(Br)ccc1I C(=O)(CC1=CCN(C(=O)CCCn2cncn2)CC1)NCC(CC)O C1(C)CCN(C(C23CC(C)(CO2)C3)=O)CC1.Cc1nn(C)cc1CC(=O)NC CP(C)(=O)CC(=O)NCc1ocnc1C(=O)NOCC(F)(F)F n1(CC)ncc(Br)c1C(=O)NC(C)C(CO)NC(=O)C(C)CCOC N1(C(CCc2c(C)nn(C)c2)=O)CCC2CC1CN(C(c1ccoc1)=O)C2 c1(CNC(C(CC2CCC2)NC(c2c(C)con2)=O)=O)nnn(C)c1C C1(C(N2CC(c3c(C)nn[nH]3)C2)=O)CN(C(=O)COCCC(C)C)CC1(F)F c1(C(N2CCCC3(CNC(=O)CCn4ccnc4)C2C3)=O)cc(Cl)c(F)cc1O C1(CC(=O)NC2(CCNC(c3cc(Cl)ccn3)=O)CC2)CSc2ccccc2O1 N1(C(C2CCC(SCC)CC2)=O)CCCC(O)C1.C(=O)CC.C(=O)C1CC1.N n1(CCC)cc(C(C(=O)NC2(C)CC2)N(C)Cc2ccccc2CC)c(C)n1 N1(C(c2cc(SC)oc2C)=O)CC2C3CCC(C2C1)N(C(C1CC12CCC2)=O)C3 Cc1ccc2nc(COc3nnc4ccccn34)cn2c1 C(c1ccc(Cl)cc1Cl)=CC(N1CC2(CN(C(c3ccc(C)cc3I)=O)C2)C1)=O C1(C(=O)NCC(CCNC(CNC(N)=O)=O)O)COc2c(F)cc(F)cc2C1 C1(n2cnnn2)(CC(=O)NCC=CC)CCOCC1.C(=O)C(O)c1ccsc1.N c1(C(=O)NC2C(CC(=O)NCC(CC)(C)C)CCCC2)cc2cnccc2[nH]1 O=C(C1CCCc2ccccc21)NCC1CN(C(C2(C3CC3)CCC2)=O)CC1O C1(NC(C2C(C)CCO2)=O)CC2CCC1CN(C(C1(C#N)CC1(C)C)=O)C2 n1(CC)nc(C(=O)N(CC)C)c(Br)n1.C1(CC=O)CC=CCC1.C1CCC1 C(=O)(C1CCCc2nn[nH]c21)N1CCC(CC=C)(NC(c2cc(C)ccn2)=O)C1 Cc1cc(F)ncc1C(N1CCC(NC(=O)CC2(C)CC2(Cl)Cl)C(C)C1)=O N1(C(C2N(CC)CCOC2)=O)C2CCCC1CC(NC(=O)Cc1cn[nH]c1)C2 N1(C(CCCCOCCC=C)=O)Cc2ccccc2C(c2cccs2)C1 c1(OC)ccc(CC(=O)NCC(C(C)(C)C)NC(c2coc(C)c2)=O)cn1 N1(C(C(C)CC2CC2)=O)CC2CCN(C(c3ccc(Cl)c(Cl)c3O)=O)C(C2)C1 C1(CC(=O)N(C2C(OC)COC2)C)C2CCCC2N1C(c1ccsc1)=O N1(C(C(C)C2CC2)=O)CCN(C(C2(c3ccno3)CCC2)=O)CC1c1cn[nH]c1 Cc1nc(N2CCC(C(C)NC(c3cncnc3C(C)C)=O)CC2)[nH]c(=N)n1 C1(C(N(C2(C(=O)NCc3nc[nH]n3)CC2)C)=O)CC2C=CC1O2 c1(NC(C)=O)ccc(CC(=O)NC2CN(C(C3(O)CC3)=O)CC2O)cn1 C(=O)(C(COC)CC(C)C)N1CC(CC=C)(C(N2CCC(C)(N(C)C)C2)=O)C1 c1ccccc1F.C(CC(=O)N(C1C(=O)N1)CCN(C)C)OCCCOC c1(CN(C(CCOCCCNC(CSCCCC)=O)=O)C)nncn1C c1(N2CCN(C3CCCN(C(c4c(C)nc[nH]4)=O)C3)CC2)ncc(C#N)cc1Cl c1(C(=O)NCC2(COC)CN(C(=O)CC3=CCCC3)C2)nccn2cnnc12 C1(NC(C(CC=CC)C)=O)COCCN(C(c2cc(C(C)=O)on2)=O)C1 C1(C(=O)NC23CC(NC(=O)CCc4ncc[nH]4)C(OC2)C3)CCc2cnnn2C1 C1(C(=O)NC(C(C)NC(CCN(CCC)C)=O)C)CCC(C)(C)C1 c1(C(=O)NC(C)CC(C)NC(c2coc(O)n2)=O)nn(C)cc1N Cc1ccc(C(=O)NC2(CF)CCN(C(=O)Cn3ncnn3)C2)c2ncccc12 Cc1ccc(Cl)cc1C(=O)N(C1CCC(NC(C2CCC(C)C(C)C2)=O)CC1)C c1(C(=O)NC2CC(C)(NC(Cc3ccc(C)cc3)=O)C2)ccc([N+](=O)[O-])s1 CCC(CCC(=O)N1CCOCC1CCNC(=O)C=CCN(C)CC)OC c1(OS(c2c(C)scc2)(=O)=O)ccc2ccc(Cl)c(C)c2n1 C1(NC(c2c(C)[nH]c(C#N)c2)=O)CN(C(c2n[nH]c3c2COC3)=O)CC1C1CC1 c1(NC(=O)OC)ccc(C(=O)NCCNC(=O)CC2C=CCCC2)s1 C1(OC)CN(C(=O)C(=Cc2cccs2)C)CC1NC(C12CCC(CC1)O2)=O CP(C)(=O)c1cccc(C(N2CCCCC(NC(C34CC(C3)C4)=O)C2)=O)c1 C1(F)(C(=O)NC(c2ncc(C)[nH]2)CC)CCCN(C(c2csnc2Cl)=O)C1 c1(C(=O)NCC(C(C)(C)C)NC(=O)C(O)c2ccsc2)c[nH]c2cccnc12 C1(C2CCN(C(=O)C(F)F)C2)(NC(C2CCn3cncc3C2)=O)CC1 Cc1ccc(Br)c(C(=O)N(c2nccc(C)n2)C(C2CCCNC2)C)c1.C(C)(C)O c1(CCC(=O)N(CCC#C)C)nc(O)c2c3c(sc2n1)CC(C)CC3 CC1(C)CC(C(=O)NCC2CCCCN(C(=O)CS(=O)(=O)C3CC3)C2)CNC1=O N1(C(C(C)SC)=O)CCC(CNC(c2cnn(C3CC3(F)F)c2)=O)C1 c1(CCN(C(=O)CCCCCC#N)C)cccc([N+](=O)[O-])c1 C1(N(C(CCC)=O)C)CC2CCC(C1)N2C(=O)CCc1c[nH]c(C)c1C(C)=O CC(C)CC(CNC(C1(N(C)C)CCC1)=O)NC(c1nn(C)cc1Cl)=O C1(NC(c2cn(CC(CC)O)nn2)=O)C2CC1N(C(=O)Cc1ccnn1C)C2 C#CCC(C(=O)OC)NC(=O)C(C)(C)NC(=O)COCC(=O)NCC C1(C(=O)NCC2CC(C)(C)CN2C(=O)CC2=CCCCC2)CCCCC(F)(F)C1 CCCCC(CNS(=O)(=O)CCC1CCCO1)CCC C1(C(N(C(C=O)C2CC2)C)=O)CCC(F)CC1.C1(C(=O)OC)(C)CCC1 N1(C(c2c(C)nsc2)=O)CCCC2(CCN(C(c3cccc(O)c3C)=O)C2)C1 CCC(C)(C)CC(=O)N1CC(NC(=O)CC2CCC(C3CC3)O2)C(F)C1 c1(SC)cc(C(=O)NCCC2(C)CCN(C(C3CC3C3CC3)=O)C2)c(C)o1 N1(C(c2ccnc(C)n2)=O)CCC2CCN(C(c3cccc4occc34)=O)CC12 C1(F)CCN(C(C2(CC(F)F)CCC2)=O)C1.CC(C)(C)C(=O)NCC(=O)N c1(SCCNC(c2ccc(C(=O)OC)o2)C(C)(C)C)ccc(C)cc1 C#Cc1cnn(C)c1C(=O)NC(CNC(=O)CC1CCN(C)CC1)CCCC C12(CC)CCC(C(=O)NC(C)Cn3cc(-c4cccc(C#N)c4)nn3)(CO1)C2 CCCCCCN(CC)C(c1ocnc1C(F)(F)F)=O.C(=O)(C)N.C(C)=O C#CC1(NC(C2(NC(=O)CC3CCC(C#N)C3)CCC2)=O)CCCCCC1 C1(NC(=O)C=C2CC2)CCN(C(C2CCS(=O)(=O)CC2)=O)CC1CO c1(C=O)cc(O)cc(C#N)c1.N1(C(C2C(OCC)C2)=O)CCC(C)(C)C1.C C1(O)(CCNC(c2ncc(N(C)C)nc2)=O)CCCN(C(=O)C(F)C(C)(C)O)C1 c1(NC(CC)=O)cncc(C(N2CC(F)(C)C2)=O)c1.C1(C(=O)N)CCCCC1O C=C(C)CC(C(=O)NC(C)(C)C#CCC)NC(c1nn(C)cc1Cl)=O C(CC(O)C(F)F)NC(c1cc(CNC(=O)C=CC(F)F)[nH]n1)=O c1(OC)cc(N)c(Cl)cc1C(N1CC(NC(=O)CCCC(C)(C)C)CC1(C)C)=O C1(C(=O)N)CC2(CCCCC2)CO1.C(=O)(C#CC(=O)NCC1COCC1)N(C)C c1(OC)ncccc1C(=O)NCC(C)NC(c1c[nH]nn1)=O.C1CNC(=O)O1 C(=O)(C(C)(CC1=CCCCC1)NC(c1ccc(OCCF)cc1)=O)OC N1(C(c2ccc(CC)[nH]2)=O)CCCC(C)(C(=O)N(C2COC(C)(C)C2)C)C1 CCC(C(=O)NC1(C(=O)N(CC)CC2CCCO2)CC1)SC C1(C(C)N2c3cc(ncn3)C2=O)CC2CCC1CC2.C(C1CCCC1)=NC(N)=O N1(C(C2C(C)CCO2)=O)CCCCC1CN(C)C(C1CCCN1C=O)=O c1(C=O)cccc(S(C)(=O)=O)c1.C(C(O)C(=O)NCCCN(CCC)C)SC Cn1c(O)nc2c(-c3nc(C(F)F)nn3CCF)cccc12 N1(C(c2cccc(C)n2)=O)CC2CCCC(NC(c3cnc(O)c(F)c3)=O)C2C1 c1ccc(C#N)cc1.C(CC(C(=O)N)NC(C1CC(=C2CCC2)C1)=O)=CC c1(CC)cccc(C(=O)NC(CNC(=O)C=C2CCC2)C(C)C)c1N CCCCCC(F)C(=O)N1CCCCC(CCC(=O)NCC(C)(C)CC(F)F)C1 C1(NC(CCC2CC(OC)C2)=O)CCN(C(c2cc([N+](=O)[O-])c[nH]2)=O)C12CC2 CCC(CC)(C(=O)NC1CCC1NC(=O)Cn1cnnc1O)c1ccccc1 N1(C(C2(OCC)CCOC2)=O)CCC(C(=O)N(CC(=O)OC)C)C(C)(C)C1 c1(C(N2CCCNC(=O)C2CCO)=O)cc([N+](=O)[O-])ccc1NC=O CC1(CCCN)C2=NC3=NNC3=CC=CC=CN(S(=O)(=O)C1)CC(C)C2 c1(C(=O)NCCC(C)N(C(c2cnc(C)[nH]2)=O)C)sc2ncccc2c1Cl CC(C)C(F)(F)CC(=O)N1CC(NC(=O)C=CC2CCCC2)CC12CCC2 c1(C(=O)N)cnc(O)c([N+](=O)[O-])c1.Cc1cccc(C(N2CCC(C)(C)C2)=O)c1 N1(C(C(=Cc2cccc(Cl)c2)C)=O)C2CCC1CC(NC(=O)C)C2.[SH](C)(=O)=O N1(C(C2CC(OC)C2)=O)CC(C(=O)NCCN2CCC2)C(C2CC2)C1 C(C(C)(C)CNC(=O)COCCOC)N(C(c1nnsc1N)=O)CC Cc1noc(C)c1Cn1cccn1.C1CCN(C(=O)C(C)(F)F)C1.C1CCS1.N c1(C(N2CC(C)(CNC(c3c(C)n[nH]c3)=O)C2)=O)cc2c(cc1Cl)NC(=O)C2 N1(C(C(C)(C)OC)=O)CCC2C(C1)CN2C(C1CC2CCC(C1)C2)=O C1(NC(C2CC(CC)C2)=O)CN(C(C2(CO)CCOCC2)=O)CC1S(C)(=O)=O N1(C(CCC#C)=O)CCC(C2CCOCC2)(CNC(C2OCCC2C)=O)C1 N1(C(C2(OC)CCSC2)=O)CC2(COC(CNC(c3n[nH]c(C)c3Cl)=O)C2)C1 C1(F)CC(C=O)C1.C1(CC)CCCC1.C(C(=O)N)=CCOCCOC N1(CC(=O)NCC2CCC2)C(=O)CNC1=O.C(=O)C(O)CC1CCCCC1.C N1(C(C(n2cc(Cl)cn2)C)=O)CCC(O)(C(C)NC(C2CCCCO2)=O)C1 C1(CC(=O)N(C(CC)C2CC2)C)N(C(c2cc(OC)n[nH]2)=O)CCC1(C)C c1(C(=O)NC2(C)CCC2)cc([N+](=O)[O-])ccn1.C1CC(F)(F)C1.C(=O)(C)N CC(Cc1cnc[nH]1)C(=O)N(CCCNC(=O)C)CCO.c1n[nH]c(=N)s1.S C1(NC(C2CCCCS2(=O)=O)=O)CN(C(=O)Cc2ccccc2F)CC12CCC2 C(c1cncnc1O)=CC(N1CC(CCNC(=O)Cn2nccn2)OCC1)=O C(C)(C(=O)N1OC2CCC1C2)N(C(c1cnc(C)s1)=O)CCN(C)C C1(CNC(c2ncn(CC)n2)=O)CC(C)(C)CN1C(C1CCCC12CC2)=O c1(C(=O)NC(CC)C(=O)NCC(O)CC2CCCC2)ncccc1F c1(SC(C(N2CC(NC(C#CC(C)C)=O)C(C)C2)=O)C)ccc(C#N)cc1 C1(CNC(NC(c2ccc(F)cc2Cl)C)=NCCF)CC2(CCOCC2)CO1 N1(C(CCC2(C)CCCC2)=O)CCCC(C)(NC(c2nc(OCC)oc2)=O)CC1 Cc1c(C(N2CC(N(C)C(c3cc(C4CCC4)on3)=O)C2)=O)csc1Br N#Cc1c(F)cc(C(=O)NC2CCOC2)cc1F.C1(CC=O)CS(=O)(=O)C1.C C1(C(=O)NCCCN(c2ncc(C(=O)OC)cc2Cl)CC)CCc2nnnn2C1 C1CN(C(c2nnn(C(C)(C)C)n2)=O)CCN1C.C1(C(=O)N)(NC(C)C)CC1 c1(C(=O)NCC(CCCC)NC(=O)C(O)C2CC2)ccc2c(c1)C(=O)OCC2 N1(C(CCc2scc(C)n2)=O)CCN(C(c2cccnn2)=O)CC2CCCCC12 Cc1ccc(S(=O)(=O)N2CCCC2)cc1NC(c1c[nH]cc1C1CC1)=O C(=O)(CC(C)C(F)(F)F)N1CC2(CC(NC(C(C3CCOCC3)C)=O)C2)C1 CC1C(NC(=O)CNC(c2ccoc2)=O)CCN1C(c1ncnn1C)=O C(=O)(C(CNC(=O)CCc1ncccn1)C(C)C)N(C(C)CO)CC c1(C(N2CC(N(C(=O)CC3(O)CCCCC3)C)C2)=O)cccc2c1OC(C)(C)C2 Cn1cc(Br)c(C(=O)NCC2CC(NC(C3CCC3)=O)C23CCC3)cc1=O CN1CC(O)CC1C(N1CC2CC2(NC(=O)C=CC2CC2)C1)=O CC(=NOCc1nc2ncc(Br)cn2n1)c1ccc(F)c(C(F)(F)F)c1 CC(C)CCCCC(=O)N1CC(NC(=O)Cc2cccc3occc23)CC(C)C1 c1(CC(C(=O)NC(C2CCCN(c3cnc(F)cn3)C2)C)C)ccc(F)cc1 Cc1cc(Cl)nc(N)c1C(=O)NCCC1CCN(C(=O)CC)CC1.CC(N)=O.S N1(C(c2ccn(C)n2)=O)CCC2(CC1)CCN(C(C1CC3CCC(C1)C3O)=O)C2 CC1CC(C(=O)NC2CCOCC2)CN(C(C2CCCCCN2C)=O)C1 c1(C(=O)NCC(c2ccc(F)cc2)NC(CCC=C=C)=O)cc(C)n[nH]c1=O C1(C(N2CC(CCNC(c3cc(F)c[nH]3)=O)(OC)C2)=O)CCc2nnnn2C1 N1(C(c2n(CCC)nc(C)c2)=O)CCC(C)C(NC(c2nsnc2O)=O)C1C N1(C(COC2(C#C)COC2)=O)CCC(O)(C(C)NC(c2ocnc2C)=O)CC1 N1(C(c2ncc(C(F)F)s2)=O)CCCN(C(C2CC2F)=O)CC1 CC(C)(CC(F)C(=O)NCCC1CCCC12CC2)NC(=O)Cn1nccn1 n1(CCCC)nc(C(=O)N(CCNC(C2COCCO2)=O)C(C)C)ccc1=O c1(CNC(C(C(OCC)Oc2ccccc2)O)=O)ccccc1C(F)(F)F C1(CNC(c2c(C)oc(C(C)C)n2)=O)COCCN(C(c2[nH]cnc2C#N)=O)C1 N1(C(C2CCCCN(C(c3c(OC)scc3)=O)C2)=O)CCCC(C2CC2)CC1 C1(CC(=O)NCc2scc(COC)c2)(C(=O)O)CCN(C)CC1 C#Cc1cc(NC(=O)Nc2nc(-c3ccc(N(C)CCO)cc3)cs2)cnc1C N1(C(c2cnc3ccsc3c2)C(=O)NCC)CCC2(CC1)CC(C(=O)OC)CO2 C1(C#CC(=O)NCCC2CCN(C(c3nc(OC)ccc3F)=O)CC2)(CC)CC1 C1(NC(c2cnc(C)s2)=O)CCCCC1C(=O)NC1(C2CCCCO2)CC1 CC1CC(NC(c2ccc(=O)oc2)=O)CCN1C(=O)C=Cc1cccc(N)c1 Cc1nc(O)nc(O)c1CC(=O)NC(C)CNC(C1CC2C=CC1C2)=O C1(CC(N)=O)CN(CC2CCC(F)(F)C2)CC12CC2 c1(C(=O)NC(CCC)CC(=O)NC(c2c[nH]ccc2=O)C)cc(C#N)ccc1C c1(C(=O)NCCCCCNC(C=Cc2ccc(C)s2)=O)cccc(F)c1C Cc1onc(-c2ccsc2)c1C(N1CC(C)C(C)C1)=O.C1(C)(C=O)C=CCC1.N N1(C(CONC(c2cnc(C)o2)=O)=O)CCC(C)C(CO)C1 c1(CC)ccccc1C(=O)NC(CO)C(=O)NC12CC(C)(C1)C2 C12(CNC(C3(C=C)CCC3)=O)CCCC(CN1C(C1CC1C1CC1)=O)C2 C1(C(=O)N)CC2C(C1)C2(F)F.c1(OC)ccccc1C(=O)C(=O)NCCCO c1(NCC2(OC)CC2)ccc(S(=O)(=O)NCC(C)C(F)F)cc1F c1(OC)ccc2oc(C(=O)NCC(CO)NC(c3cn(C)cn3)=O)c(C)c2c1 c1(C(N2CC(NC(C3(O)CCSCC3)=O)C2)=O)ccc(Br)c(O)c1 c1(CC)oc(C(=O)NCCCC(C)NC(=O)CCC(=O)OC(C)(C)C)cc1C C(=O)(CC(C)C(C)C)NC1(C)CC(NC(c2c(C)cnn2C(C)C)=O)C1 C1(C(=O)NCC2CCCSC2)CC=CC(n2cc(-c3ccc(CO)cc3)nn2)C1 Cc1nc(Cl)sc1Cc1nnnn1C1CC(F)(F)C1.C1(CC)CC(C)(C)CO1.N C1(CC(=O)NCC(C)C#N)CCC(NC(=O)C(C)n2ccnn2)C1 c1(C(=O)NC2(c3cn(-c4ccccc4F)nn3)CCC2)cc(Cl)c(Cl)c(Cl)c1Cl Cc1cn2cc(C(=O)NC3CC(C)CN(C(=O)CC(=O)N(C)C)C3)ccc2n1 C1(CCCNC(C2CC2(F)F)=O)CCCN1C(c1cnc(CC2CC2)s1)=O Cc1ccc(CCNC(c2cnc3ccc(C(=O)O)cn23)=O)c2ccccc12 CC(C)CC(CNC(=O)Cc1ccc(F)nc1)NC(C1(CO)CCCC1)=O C(=O)(C(F)CC(C)C)N(c1ccccc1)CC#C C1(CC)CCCN(C(C2CCC2C)=O)C1C(=O)N(CC(C)(C)C#N)C N1(C(C2CC(C)N2C(c2coc(N(C)C)n2)=O)=O)CCC(CCF)CC1 CON(CCC(=O)N1CCC(N2CCC2)C1)C(=O)C1(F)CCC(C)CC1 CCC(C)(O)C(=O)NCC(Cc1ccccc1)NC(=O)CCNC(=O)NC C(=O)(C(C)(C)CC(C)(C)C)N1CC2CC(NC(COC(CC)(C)C)=O)CC2C1 C1(CCC)CN(C(C2CC2C(N)=O)=O)CCN1C(c1ncoc1C)=O C(c1ccn(C)c1)=CC=O.C(=O)(CCc1ccoc1)N.C(CC)N(C(C)=O)C N1(c2ncnc(CC)c2F)CCC2CCC(C1)N2C(=O)Cc1cc(C)no1 c1(CC)ccc(C(=O)NC2COCCN(C(c3c[nH]nc3CC)=O)C2)c(F)c1 CC(C(=O)NOCC1(c2cn(CCCC(=O)O)nn2)CC1)n1ccnc1 c1(NCCCN(C(C(CCC)OCC)=O)CCC)nc(Cl)nc2c1CCC2 Cc1cnc(C)c(C(N2CCCC(C)C2CNC(c2coc(Cl)n2)=O)=O)c1 C(=O)(C(C)(C)CC(C)(C)C)N1CC2OCC(NC(C(C)SC)=O)C2C1 C1(CN(C(C2(CC)CCC2)=O)C)CCN(C(=O)CCC2CCC(C)O2)CC1 c1(OC(C(=O)NCC(C)(C)NC(C(C)n2cnnn2)=O)(C)C)ccccc1 N1(C(CSCC=C)=O)CCN(C(c2cccc(Cl)c2C)=O)CC1CCO N1(C(C2(C)CC2)=O)CCC(C2(NC(C3CCC3c3nc(S)n[nH]3)=O)CCC2)CC1 N1(CCNC(C2(CC)CC2)=O)CCCN(C(=O)CC2CCC(=O)NC2)CC1 c1(N(CCC(C)O)C)nc2ccc(Cl)cc2c(=NCCC(C)C2CCCCC2)[nH]1 c1(NC(c2c(C)nc(NC(c3noc(C)c3C)=O)s2)=O)ccc(Cl)c2cc[nH]c12 c1(NC(CC(C)NC(=O)COCC2CC2)C)ncnc(O)c1Br C(c1ccc(O)cc1)=CC(=O)NCC=CCNC(C(C(C)C)OC)=O C1(C(N2CCC(N(C(=O)CCc3ncc[nH]3)CCC)CC2)=O)CCC(C)(O)CC1 c1(C(C)NC(=O)NC(C)CC(F)F)cc(C(C)(C)C)ccn1 C1(OC)CCC2(C(N3CC(C(N)=O)(C)C3)=O)CCC12.c1(C(=O)N)cocn1 N1(C(CSCCC)=O)CC2(NC(=O)Cc3cccc(Br)c3)CCC1CC2 Cc1c(O)c(=O)ccn1CC(N1CCCC(CNC(=O)C(C)S)C1)=O.C(C)C N1(C(CCc2c(C)n(C)nc2)=O)CC(NC(=O)C(C)(C)COC(C)C)CC(C)C1 C(=O)(C1=CC(C)(C)C1)N1CCCC(CN(C)C(c2ccc(OCF)cc2)=O)C1 C(N=c1[nH]c(Cl)ncc1Cl)C1C(C)(C)CN(C(C2(O)CCCC2)=O)CC1 c1(C(=O)NC2CCCC2C(=O)Nc2cccc(Br)c2F)cccc(Cl)c1[N+](=O)[O-] c1(CC(=O)NCC2COCCN(C(CSCC)=O)C2)ccc2c(c1)CCCO2 C(=O)(C1=NNC(=O)C1)N(C)CCC1CCCCN1C(=O)CCc1ccsc1 c1(C(CNC(C2C(C=C)OCC2)=O)NC(=O)C(C)COC)cccc(Cl)c1Cl Cc1cc(C(=O)NCCCc2cn(Cc3nc(C(=O)O)cs3)nn2)ccn1 c1(CC(=O)NC(C2CCN(C(CCC(C)OC)=O)C2)C)cc(OC)ccc1OC c1(CC)cccc(F)c1C(=O)NCC(C)(CNC(C1C=CCC1)=O)OC c1(NC(C(=O)NC(C2CCCCC2)CCC)=O)c(N(C)C)cccc1I c1(NC(C(C)(c2ccccc2)NC2CC2)=O)cccc2cnccc12 N1(C(C2C(C)OCCC2)=O)CCc2nc[nH]c2C12CCN(C(=O)C(O)C1CC1)C2 N1(C(COC(CC)C)=O)CCN(C(C2(CC)CCC2)=O)CC1CC CC1C(NC(c2cc3c(s2)CCC3)=O)CC2CCC1N2C(=O)CC1CSC1 C(=O)(CCN(OC)C(=O)C1=CCOCC1)N1C(C)CCC(OC)C1 N(C(=NCC1=CCCOC1)NC(C1CC1)C1CC1)C1C(C)(C)C1(C)C c1(C(N2CC3CC3C2)=O)ccnc(P(C)(C)=O)c1.CC(C(=O)NC)C(C)(C)C C=CCN(OC)C(=O)C1CCN1C(=O)Cn1cnnc1 C1(CCC2N(C(C3N(CC)CC3)=O)CCC2)CCCCN1C(C1CCCC1)=O C1(C(=O)NC2C3CN(C(C#CC(C)C)=O)C(C3)CC2)CCc2ccc(F)cc2O1 C(CNC(=O)C(C)(C1CC1)OC)(C(=O)N1CC(C)(CF)C1)OC Cc1cccc(C(=O)NCCC2CN(C(C3CN(C)CC(C)O3)=O)C2)c1C#N C(=O)(C1=CCN(C(=O)C(C)N2CC(C)C2)C1)N1CCN(CCOC)CC1 c1(NC)c(C(=O)NC2CN(C(c3ccnc(C)c3)=O)CC2C)sc2nccnc12 Cc1oc2cc(C(N3CC(NC(=O)C(C)CO)C(F)C3)=O)[nH]c2c1C C(=O)(CCC(=O)NCC(c1ccccc1)NC(C1C=CCC1)=O)NCC CC(C)C(C(=O)NCC1CCOC1C(=O)NCC1(CO)CCCO1)C(C)C n1(CC)c(C(N2CCCC(NC(C3(CCF)CC3)=O)C2)=O)nc2ccccc12 C1(C(=O)NCC2OCCN(C(C3CN(C)C(=O)N3)=O)C2)CC(=O)NC(=O)C1 C1(CC)CN(C(=O)CCc2cc(Cl)no2)CCC1.c1(C=O)nc[nH]c1C(C)(C)C C(C(COC)CC(=O)N1CCCC(CCNC(C2(CF)CC2(F)F)=O)C1)OC CC(CCC(=O)NCC1CSCCO1)NC(=O)CCc1csnn1 C#CCC(C)C(=O)NCCC1CCCCN1C(=O)Cc1nnc(S)n1C C1(C)(NC(C(C=CCCC)O)=O)CCN(C(C2(N(C)C)CCCSC2)=O)CC1 N1(C(C2CN(C)C(=O)N2)=O)C2CCC1CN(C(=O)Cn1ccc(=N)[nH]1)CC2 CC1CC(CNC(c2cc(Cl)n(C)n2)=O)CCN1C(C1CCSC1)=O C1(C(N(CC(C)O)C)=O)OCCC1NC(C1(CC2CC2)COC1)=O C1(C(N2C(CCC=C)CCC2)=O)CCCCC1NC(C1(C)CC(F)(F)C1)=O CC1(C)CCCC1(C)NC(=O)C(Cc1ccoc1)NC(=O)CC1CCOC1(C)C N1(C(COCCCCC)=O)CCC(C(C)(C)C)(C)C1.C1(C(=O)N)CC(=O)C1 C(CCCCCNC(=O)CCC(=O)C1CC1)N(C)C(C1C=CC=CC=C1)=O Cc1nc(C(N2CCCC(CCNC(C3CC34CC4)=O)C2)=O)c(=O)[nH]c1C c1(OC)ccc(C)c2c1CCN(C(c1cc(CC#N)ccc1F)=O)C2 C1(C#N)(C=O)CCSCC1.Cc1ccc(CCNC(=O)C(C)CC2CC2)cc1.N CC(C)C(C(C)NC(=O)CN1CCOCC1)NC(=O)Cn1ncc(Br)n1 CC(CS(C)(=O)=O)C(=O)N1CC2CC(C1)N(C(c1nc[nH]c3ncnc1-3)=O)C2 c1(C(N(C)Cc2c(CNC(CCC#C)=O)cccc2)=O)cccc2ccncc12 CCCC(C)CC(=O)NCC(C(C)C)NC(c1ccc(-c2ccccc2)cc1)=O N1(C(c2n[nH]c3c2CN(C(C(C2CCC2)OC)=O)C3)=O)CC2(COC(C)(C)C2)C1 Cc1ncnc(C)c1OCC(=O)NC1COCCN(C(=O)CNC=O)C1 c1(CC)oc(C(=O)NCC2(NC(C3CC3F)=O)CCC2)cc1C c1(C(=O)OC)cc(C=O)n(CCN(C)C)n1.CCN.C1CC1.C(N)=O C1(CNC(=O)CCOC2CC2)CCC(NC(c2ccsc2Cl)=O)CC1 N1(C(=O)CCc2cnc[nH]2)CCCC(C2CN(C(c3cc(Br)c[nH]3)=O)C2)C1 N1(C(C2N(CC)CCCC2)=O)CCC(C2CCCN(C(=O)C(C)N3CCC3)C2)C1 c1(OC)ccccc1C(c1nc(C)c(C)s1)NCCc1nc(C)c(C)s1 N1(C(=O)NCc2ccc(C)cc2)CC2CN(C(=O)Nc3ccc(CO)cc3)CC12 N1(C(C(C)Cc2cnc[nH]2)=O)CCCCC1CN(C)C(C1CC1(F)F)=O C(c1cccs1)=C(C(=O)N)C.C1(C(C(=O)N2CCC2C)OCC)CCOCC1 c1(SC)cc(C(N2CC(O)CC2CNC(=O)Cc2cc[nH]c2)=O)oc1C CC(C)CC(C)CNC(C1(c2ccc(Br)cc2)CCNC1)=O C12(NC(C3CCCC(N(C)C)C3)=O)CCCC1(F)CN(C(=O)C(C)(C)C)C2 c1(C(=O)NC(CC)CN(C)C(c2ccc(C)cc2F)=O)cnc2sccn2c1=O Cc1cc(C(=O)NCC2CCN2C(c2c(C)nn(C)c2C)=O)nc(C)c1 CC1CCC(CO)(CNC(=O)Cn2cc(-c3ccc(N(C)C)cc3)nn2)CC1 C1(C)(n2c(CN(C(COC)=O)C)nc(-c3cscn3)n2)CCS(=O)(=O)C1 CC1CCN(C(c2ccoc2)=O)CC1N(C)C(c1cc(N)ccc1F)=O C1(O)(C(=O)NC(C2CC(NC(C3CC=CCO3)=O)C2)C)CCCCC1 C(CCCC(=O)NC1CCOC1C(N1CCC(CN=[N+]=[N-])C1)=O)(OC)OC C(=O)(N=c1ccn(CCOC)[nH]1)C1(C(C)NC(CCN(C)CC)=O)CC1 C(C(C)(C)C)NC(COCCC#C)=O.c1(CCC=O)nc(C(C)C)no1.C c1(NC(=O)NCC2CC2C2CCC2)cc(Cl)nc(Br)c1 N1(C(CC(CC)C2CC2)=O)CCC2(C1)CN(C(=O)CC1CCCS1(=O)=O)C2 Cn1cc(NCC2CCCC(O)C2)c(OC(F)F)n1 C(C(C(=O)NCC(=O)NC)n1cc(C(C)C(OC)OC)nn1)OCC CC(C)C(C(=O)NCC1CCC1)NS(C)(=O)=O.C1CCCCO1.C(=O)C CC1CC2(CCN(C(=O)CCOc3cccnc3)CC2)CN1C(C1CC1F)=O O=C1CCC(C(N2CCC(NC(=O)CCSc3ccccn3)C2)=O)C1 Cc1ccc(CC(N2CCC(NC(C3C(F)(F)C34CC4)=O)CC2)=O)cc1O N1(C(C=CC)=O)C2CCCC1CN(C(C1CCCCN1CC)=O)C2 c1(OCC(=O)NCCNC(C(n2ccc(C)n2)C)=O)cc(Cl)ccc1Br C1(C#N)(C(N(C(C)C(=O)N)C2CC2)=O)CC(=O)C1.C(C(C)(C)C)=CC N1(C(c2nc(C(C)C)oc2)=O)CC(NC(C2CC(N(C)C)C2)=O)C(O)C1 Cc1[nH]c2ccccc2c1C1CCN(c2cc(Br)cnn2)C1 c1(C(C)=O)c(NC2C3CN(C(=O)Cc4cc(C)ccc4OC)CC23)ncnc1Cl CC(C)CC(=O)C(=O)N1CC(NC(c2ccc([N+](=O)[O-])o2)=O)CCC1C C1(C(N(C2CCCC2(F)F)C)=O)CN(C(=O)OC(C)(C)C)CC(F)(F)C1 c1(C(C(=O)NC2C(CNC(CSCC)=O)COC2)C)cccc(Br)c1 C(CC1=CCN(C(c2c(C)ccnc2C)=O)CC1)NC(C(C(C=C)C)C)=O N1(C(CN(CCC)C(c2ccc(CO)cn2)=O)=O)CCOC(C(N)=O)C1 c1(C(COC(C2C(C)(CC)C2)=O)=O)c[nH]c2ncc(Br)cc12 C1(NC(c2cnc(C)s2)=O)CCCC12CN(C(=O)CN(C)C(=O)C1CC1)C2 Oc1cc(C2CC2)nc(CNC(=NCCN2CCCOCC2)NC2CCCC2)n1 c1(CC(=O)NC(C2CCN(C(c3ccc(CO)o3)=O)C2)(C)C)ccc(F)cc1Cl N1(C(CCCCCNC(Cc2c(C)scc2)=O)=O)CC(=O)N(C)CC1C c1(C(=O)NC(c2ccccc2)CNC(CC2CC(OC)C2)=O)nscc1C C(=O)(CCCCCC#N)N1C(CN(C(CSCCN(C)C)=O)C)COCC1 CC(C)C1=NOC(C(N2CCC(O)(C(=O)NC3CCC3)CC2)=O)C1 CCC(C)(C)C(C)CC(=O)N1CCCC(NC(c2ccsc2C)=O)C1C c1(C(N(CC)C2CC2)=O)ccc(-c2ccncc2)s1.C(C)(C(=O)N)OCC c1(C(N2CC(CC)C(NC(C3CC3(Cl)Cl)=O)C2)=O)cccc(C)c1C C#Cc1cn(C)nc1C(=O)NC1CCN(C(c2cc(N(C)C)ccn2)=O)CC1F N1(C(C(C2CN(C(c3ccc(=N)[nH]n3)=O)C2)OC)=O)CCNC(=O)C1C CC1CCN(C(=O)CC(C)(C)CN(C)C)CC1NC(C1(O)CCOCC1)=O N1(C(c2cn(C(C)C)nn2)=O)CCC(NC(=O)CO)C(F)C1.c1ccccn1.C Cc1ccc(NC(c2cc(CNC(=O)C(N3CCOC3=O)C)nn2C)=O)c(O)c1 Cc1cc(Br)cnc1C(=O)NC1CN(C(c2cccs2)=O)C2CC12 C1(N(C)C)(CNC(CNC(CNC(CC)=O)=O)=O)CCC1 C1(C(C=O)C)CCCN(C(C2(C3CC3)CC2)=O)C1.C1(C(=O)OC)C=CCC1.N c1(CCC(=O)N)ccc(O)c(F)c1.C1CC(O)CN1C(=O)C=Cc1cocn1.C S(=O)(=O)(c1ccccc1)N(C1CCCCC1NC(=S)N1CCOC1)C C12(NC(c3oc(CC)c(C)c3)=O)CCN(C(c3ccoc3C)=O)CC1C2 Cc1nc2ccccc2n1CC(=O)N(CCC(C)NC(=O)C1=CCCOC1)C N1(C(c2cc3c(s2)CCC3)=O)CCC2C(CCCN2C(C2(O)CC(F)(F)C2)=O)C1 Cc1cc(=O)ccn1CC(=O)NCC1C(C)CCCN1C(=O)C#CC(C)C CC(C)CCC(=O)NC(C1CCN(C(c2ncccc2N)=O)C1)C C#CCCCCCCC(=O)NC1CC(CNC(C2CCCSC2C)=O)C1 C(=O)(C1=C(C)CCCC1)N1CCN(C(C2C(C=C)CC2)=O)CC1c1ccccc1 C(=O)(C1=CS(=O)(=O)CCC1)N1CC2(CCCO2)C1.CCC(CC(=O)NC)C(F)F N1(C(=O)C=C2CCCC2)CCCC(N(C(=O)C=Cc2cscn2)CCO)CC1 N1(C(c2cn(CCC(C)C)nn2)=O)CCCC(C)(CNC(c2ccsc2)=O)C1 c1(C(=O)NC(CN(C(c2n[nH]c3c2COC3)=O)CC)C)cc2c(cn1)OCCO2 c1(C=O)cc(C(C)C)nc(O)c1.C1(N(C(C2CC2)=O)C)CCCCC1.COC C(=O)(C1=CC(O)CCC1)NC1CCC(NC(CNC(C(CC)CC)=O)=O)C1 Nc1ccc(Cl)c(C(=O)Nc2cccnc2C2(C(=O)N)CC2)c1.C1(C)CC1 C1(C(N2CCC(OCCNC(C3(CCC)CCC3)=O)CC2)=O)CCC(O)CN1C c1(C(CNC(C=C)=O)NC(=O)COCC2CCCO2)cccc(C)c1 c1(NC(C2N(C(c3c(COC)cccc3)=O)CCOC2)=O)c(F)cc(I)cc1F C1C(C)CCCN1C(c1n[nH]c(C(C)(C)C)n1)=O.n1(CC)ccnc1C(=O)N c1(C(N(CCC(=O)N(C2CC(C)(C)C2)C)CC=C)=O)ccc([N+](=O)[O-])[nH]1 C1(NC(C(CC=C)C)=O)CCC12CN(C(c1cc(C)nc(O)c1)=O)C2 Cn1cc(C(=O)NCC(O)C)c2cccc(Cl)c12.C1(C=O)CC1C(F)(F)F.N Cc1cccc(C2CCCN2C(=O)Nc2ccccc2OC(F)F)c1 C(C(C)(C)C)N(CC(=O)N(CC(=O)NC(CN(CCCC)C)C)C)C CC1COc2ccc(C(N3CCOC(CCNC(=O)C#CC4(C)CC4)C3)=O)cc21 CCC(C)(C)CCCC(=O)NCc1n[nH]cc1C(=O)N(C)CCN(C)C c1(C(N2C(CC(=O)NCCn3c(C)cnn3)CCC2)=O)nnn(C)c1N C1(C(=O)N)CC2C=CC1N(C(=O)C(=O)C(C)C)C2.C(=O)(CCC1CC1)OC N1(C(COCCCCC)=O)CC2(NC(C3OCCOC3C)=O)CCCC2(F)C1 C1(CNC(CC2N(C)C(=O)CC2)=O)CN(C)CCN1C(C12CSCC1C2)=O C12(NC(C(=CC3CCCC3)C)=O)CC1CN(C(c1ccc(F)s1)=O)C2 c1(C(=O)NCCN(C(=O)CC(C)(F)F)C)coc(S(C)(=O)=O)c1 C1(C(=O)NCc2nc(C(C)C)on2)CN(C(c2ccc(O)cc2)=O)CC1C C1(CC)CCCN1C(c1cn(C(F)(F)CO)nn1)=O.C(C=O)OCCSC.N c1(CC(=O)NCC2CCC(C(=O)Nc3ccccc3CO)CC2)ccnc(F)c1 CCCCC(C)C(=O)NCC1CCCCN1C(c1ncc(F)cn1)=O N1(CC(=O)N(C(C)C)C(C)C)CCCC(CC)C1.C1(C=O)CC1(C)C(C)C CCS(=O)(=O)CC(=O)NC1CCC(NC(c2c(C)cccc2O)=O)C1 N1(C(C(C)=C(CC)C)=O)CCC(O)(CCNC(c2cnc(O)c(F)c2)=O)CC1 c1(CC)cc(C(N2CCC(N(CCO)Cc3cnon3)CC2)=O)nn1C CC(C)C(O)CC(=O)N1CCC(=CCNC(C2CCC2C(F)F)=O)CC1 c1(OC)cc(C(N2CC(O)CC2C(N)=O)=O)cnc1-c1ccc(O)c(CO)c1 c1(CC)cccc(C)c1CNC1(C)CCOCC1 C1(CNC(C(CSC)C)=O)CC(C(=O)Nc2cnccc2C2CC2)=NO1 C1COCCN(C(c2cnc(N)c(N)c2)=O)C1.C1(CCOCC)(C=O)CCC1.N c1(CC)nc(N(C2CCN(C(=O)CN3CC4CCC3C4)C2)CC)cc(C)n1 N1(c2cc(-c3ccc(OC)cc3)nnc2C)CC(F)(F)CCC1C C1(OC)CN(C)C(C)(C=O)C1.C1C2CCCC12.c1(C=O)ccnn1C(F)F.N c1(C(=O)NCC2N(C(C(C=CC)O)=O)CC2)cnc(C)c(Cl)c1Br Cc1nc(C(=O)NCCCCNC(C2(c3ccc(Br)cn3)CC2)=O)c(C)o1 N(C(=NCCC(=O)NC)NCC1COC(C)(C)O1)C(CC)C(F)F c1(C(N2C3C(NC(C(CCC#C)O)=O)C(CC3)C2)=O)onc2c1CCCC2 C1(C(C(=O)NCCCC)NC(=O)CCc2nc[nH]n2)CC=CCC1 C(=O)(CCCC(C)(C)C#N)N1CC(Cn2cc(CCC(C)O)nn2)OCC1 C(=O)(C(CNC(=O)CC1(CSC)CC1)C(C)C)N(C(COC)C)C c1(N2CC3(OCC(C)C3)C2)ccc(Br)c(S(=O)(=O)NC2CC2(C)C)n1 CC1COC(CO)CN1C(=O)Cc1cnn(C)c1.C(=O)CC1(N(C)C)CC1.N C1(C(N2CC(OCC(=O)NC(c3cc[nH]n3)C)C2)=O)CC2C=CC1O2 C#CC1(O)CC(C(=O)NCC2(NC(=O)CC(C)c3ccncc3)CCOC2)C1 C=CC1CN(C(=O)CN2CSCCSC2)CC1NC(c1cnc(C(C)C)nc1)=O C1(CCC)CC(C(=O)NC2CC(F)(C)C2)CCO1.C(=O)(CC=C(C)C)N N1(C(CC2CCCN(C(C3C(C=C)OCC3)=O)C2)=O)CC2CCC=CC12 C1(C(N(CCC(=O)NCC(CSC)C)C(C)C)=O)CC2CCC2C1 c1(CCCC)cn(C(C)C(=O)NCC2CCOC2C)nn1 C1(CNC(c2c(F)cccc2Cl)=O)(CO)CC12CCN(C(=O)C(F)(F)CO)CC2 Cc1oncc1S(=O)(=O)N1CCSCC1C(N1CCN(C2CCC2)CC1)=O C1(C)CCCN1C(c1cn(C)nc1C=O)=O.C1(CCC)CC1C(=O)NC C1(C)(C(=O)NC(C)CNC(=O)C(C)(F)F)CCC(F)(F)C1 C12(NC(C(CC=CCC)C)=O)CCCC(NC(=O)C(C)O)(C1)C2.CCCCCC CC1CCC(NC(c2cc(Cl)nn2C)=O)CN1C(=O)Cc1n[nH]c(=N)s1 C1(C(=O)N)CC2(CCN1C(=O)CCC(CF)CF)CC2.c1(COC)n[nH]c(C)n1 N1(C=O)CC(C)C1.C1(CC(=O)N(C(C=O)C2CC2)C)CCC(=O)C1.C C1(C)(OC)CCCN(N2CCC(c3n[nH]c(C)n3)CC2)C1 C1(NC(CCCC=C)=O)CCCN(C(=O)Cc2cn(C)cn2)C1CC CC1CCC(C(=O)CNC(=O)C)N(C=O)C1.C(C)(C)C.CCS.CC c1(C(N2C(C(=O)NCC(C)(C)O)CCC(O)C2)=O)cc2cnccc2[nH]1 C1(OC(C)(C)C)N(N2CC(c3ccc(Br)cc3)C2)CC12CCOCC2 C(C(C)(C(=O)N(CC(C)C(C)(C)C)C)NC(=O)C(C)c1cc[nH]n1)SC C1(c2n(CC=C)nnn2)(NCc2ccno2)CC2CC(=C)CC(C2)C1 c1(C2N(C(c3cn(C)nn3)C(=O)NC(c3ccccc3)C)CCC2)ccc(Cl)cc1 N1(C(CCC=C(C)C)=O)CCN(C(=O)CCN(CCC(C)(C)C)C)CC1C(F)F C1CCC(C)(C)CN1C(c1ccc(=O)oc1)=O.Cc1cc(C)c(CC(=O)NC)s1 CCCCC(C(=O)NCCC1OCCC1(C)C)NC(C1CC(O)C1)=O CC1(C)OCCC1(O)C(=O)NCC1CCC(C(=O)NOC2CC3CCC2C3)C1 C1(C(N2CC(CC=C)(C(=O)NCCC(O)C3CCC3)C2)=O)CSCC(=O)N1 c1(C(=O)NCC2N(C(C(CC)OC)=O)CCC(C(C)C)C2)cccn2cnnc12 C1(OC2CN(C(Cc3c(C)occ3)=O)C2)CCN(C(c2ccon2)=O)CC1 CCC(CCC(=O)NCC1CC1C(=O)NC(CO)C(C)O)OC CC1(C)CC(NC(C2CC(=C3CCC3)C2)=O)CN1C(C12CSCC1C2)=O N1(C(C2=NOC(CNC(c3ccncn3)=O)C2)=O)CC(C2CC2(F)F)C1 N1(C(C(CCO)N(C)C)=O)CC2CC(C1)N(C(=O)CCNS(C)(=O)=O)C2 c1(SC)c(C(=O)NC2CCC(F)(CNC(C3CC4CC4C3)=O)C2)cnn1C N1(C(CCCCC#C)=O)CC2(CCC2)CC1CNC(c1ccc2c(n1)CCC2)=O C#CCCC(O)C(=O)N(CCCCNC(=O)CC(C(F)F)c1ccc(F)cc1)C O=C(CC1=CCN(C(=O)Cc2ccc[nH]2)CC1)NC1CC2CC3C(C2)C13 c1(CNC(CS(CC)=O)=O)ccc2c(c1)CCC2NC(=O)C(C)(C)C1CC1 C#CC1CN(C(C2CCN(C(=O)CNC(C)=O)C23CCC3)=O)CCN1C n1(CC)ccnc1C(=O)NC(C)CC1CN(C(=O)CSc2ccccc2)C1 N1(C(CCN(C)CCO)=O)CC(N(C)C(c2ccccc2CO)=O)C(F)C1 c1(C(N2CCC(O)(CNC(C(COCC)C)=O)C2)=O)nccc2[nH]ccc12 c1(C(=O)NC(CNC(CCCC=C)=O)C)ccc(C)nc1C1CC1 C1(CNC(C(C)N2CCC2)=O)CN(C(c2cncc(Cl)c2Cl)=O)CCC1(F)F N1(C(C(C)OC2CCCCC2)=O)CC(=O)NCC1C(=O)N(C(C)C(N)=O)C C12(CNC(c3c(C)c[nH]n3)=O)CCCC1CN(C(C1CCCCO1)=O)C2 c1(C(N(C)CC2(O)CCN(C(C=CCC)=O)C2)=O)cc(OC)c(F)c(F)c1 N1(C(c2cc(C)ns2)=O)CCOC(C(=O)NOCC(F)F)C1 N1(C(C(C)(N(C(=O)C(=O)C2CCCC2)C)C2CC2)=O)CCOC2CC12 N1(C(c2ccc(OC)nn2)=O)CCN(C(=O)CC2CCC2)CC(C)(F)C1 C1(O)(CN(C(C(=O)N(C)C)=O)C)CCN(C(=O)CS(N)(=O)=O)C1 C1(C(=O)NCCC(CC)O)CN(C(=O)CCC2CC(C)C2)CC1(F)F C1(CN(C)Cc2cc(-c3ccccc3)c(OC)c(Cl)c2)CC2(C1)CC1(CCC1)C2 CCCC(CNC(c1ccc(=O)n(C)n1)=O)C(=O)NCc1nc(C)c(C)o1 c1(C(N2CCN(C(c3cccc(C4CC4(F)F)c3)=O)CC2)=O)cccc(Cl)c1 C1(CNC(CCC(CC)OC)=O)CCC2(CC1)CCN(C(C1CCO1)=O)CC2 Nc1ccc(C(=O)NC2CCC(NC(C3CCS(=O)(=O)C3)=O)C2)c(O)c1 N1(C(CCNC(C(C)(C)C)=O)=O)CCCC(C2CCCN(C(=O)C=C3CC3)C2)C1 C(=O)(C(C)(CC#C)NC(=O)CCc1nc(C)no1)NCCCCCC#C c1(C(=O)NCCC2CCN(C(C3C4CC4C4CC34)=O)CC2)coc2c1CCCC2 N1(C(C(C)=C2CC2)=O)CCCC(C2CCN(C(c3c(C)cc(C)nc3O)=O)C2)C1 Cc1cc(N(CC(C)CNC(C2CCCC(O)C2)=O)C)nc(Cl)n1 N1(C(c2c(C)[nH]nc2C(F)(F)F)=O)CC2CC(N(C)C(c3cncn3C)=O)C1C2 N1(C(C(C)(C)SC)=O)CCC(C2CCN(C(c3nnc(O)nc3O)=O)C2)C1 CCC(CCOC)C(=O)N1CCOCC(NC(=O)C(C)SC(F)(F)F)C1 CC(C)(C#N)CCC(=O)NCC(C(=O)N1C(CO)CC2OCCC12)C(C)(C)C Cc1n[nH]c(C)c1CCC(N1CC(C)(NC(c2ccc(Cl)cn2)=O)C1)=O c1(OC)cc(C(=O)NCC2COCC2NC(c2cc(Cl)c[nH]2)=O)cnc1O C1(NC(c2cnn(CC)c2C)=O)CCC(C)(C(N2CCCC2C(N)=O)=O)CC1 C1(CCNC(c2cc(C)ncc2)=O)CN(C(c2c[nH]ccc2=O)=O)CCS1(=O)=O c1cc(Br)c([N+](=O)[O-])s1.c1(C(=O)NCCC2CCCN2)cc(Cl)cc(Cl)c1Br.C C1(C(N(CCNC(C2(c3c(C)cno3)CC2)=O)C)=O)CCC(C)(O)CC1 C(C1c2ccsc2CCN1C(c1ccc[nH]1)=O)NC(C(CCC)O)=O c1(NC2C(CC=C)CCCC2)ccc(S(=O)(=O)NCc2csc(C)c2)cc1C#N N1(C(c2cc(OC)no2)=O)CCN(C(=O)CC2(C)CCCC2)C(c2cn[nH]c2)C1 C1(CNC(C=CSC)=O)CC2CCCCC2N1C(=O)CCNC(C1CCC1)=O C(CCCCCC(F)(F)F)OC(C(c1ccc(F)c(Br)c1)(C)O)=O CCCC(C(C)C)NCc1ccc(CC(C)C)s1 C(=O)(C(F)CC(C)C)N1CCN(CC2CN(C(Cc3cccc(C)c3)=O)C2)CC1 c1(CCC(N2C(CCc3cn(CC=C)nn3)CCC2)=O)ccncc1Br C(C)(CNC(=O)OC(C)(C)C)(C(C)C)NC(CC(C)OC)=O Cc1cc(C(=O)NC2(C3CCN(C(=O)Cc4n[nH]c(=N)s4)C3)CC2)c(O)nc1C C1(CNC(c2sccc2F)=O)(CNC(C2C3COCC23)=O)CC1(F)F C1(CC(=O)NCC#CC(=O)NCC2(CF)CC2)CCCCCC1 N1(C(c2nc(C)[nH]n2)C(=O)NCC2CCCO2)CCc2cc(OC(F)F)ccc21 C1(NC(C2(C=C)CC2)=O)CCCC12CCN(C(C13CCC(C)(CC1)CO3)=O)CC2 C1(OCC)COCCC1CC(=O)NCC1CCCCN1C(c1ccon1)=O c1(C(=O)NCCCC(C)NC(=O)CN2CCOCC2=O)cnc2c(c1)CCCO2 Cc1ccc(N)cc1C(=O)NC1CCN(C(c2cnoc2)=O)C1C c1(OCC)ccc(C)cc1CN1CC2C(C1)N2C(=O)Cc1cccc(O)n1 c1(OC)ccccc1OC(C)(C)C.C1CCS(=O)(=O)NCCO1 C(=O)(C(C(C)C)NC(C)=O)NC(CN(C(C=C(CC)CC)=O)CC)CC c1(-n2c(-c3cc(C)ncn3)nc(COC)n2)cc(F)ccc1C C1(NC(CCCC)=O)CCN(C(=O)CC2CCCN2C)C(C)C1 N1(C(c2ccn(C)c2)=O)CCCC2CN(C(c3ccoc3Br)=O)CCC12 C1(C(=O)N)CN(C)CCN(C)C1.N1(C(CNC(=O)OC)=O)CC(O)(CC)C1 c1(OCC)cc(C(=O)NCC2CCCC2)ccc1C.C1(C(=O)N)CCCOCC1 N1(C(C2CCC(=C)CC2)=O)CCCC(C(C)C)C1.C1(C(C)(C)O)(C=O)CCC1.N Cc1occc(=O)c1OCC(N1CCC(CNC(=O)CN(C)C)C12CC2)=O Cc1ccn(CC(=O)NCC2CN(C(=O)C(C)CO)CC2(C)C)c(=O)c1 c1(CC(N2CCC(CNC(c3nc(OCC)oc3)=O)C2)=O)ccnc(F)c1 N1(C(C2N3C(C)CN(CC3)C2)=O)CC(NC(=O)Cc2cccs2)C2CCCCC12 c1(C(N2CC3CCN(C(=O)CC4CCC4)C3C2)=O)cc2c(nc1O)CCCC2O c1(C(N2CC(NC(C(C)CC(F)(F)F)=O)CC2(C)C)=O)ccc2nnn(O)c2c1 N1(CCNC(c2ccnc(C3CC3)n2)=O)CCCC(C2CCCCN2)C1 Cc1ncc(C(N2CCCC(CNC(c3ncccc3F)=O)C2)=O)c(C(C)C)n1 Cn1cc(I)c2c(NC(=O)CCOCc3ccccc3)ncnc12 c1(C(=O)NC2CN(c3nccc(Br)n3)CC2(F)F)cccc2cnccc12 c1(CC(N2C(C3(C=O)CC3)CCC2)=O)ccc(F)cn1.C1(CC)(CC)CCC1 N1(C(CC(C=C)C)=O)CCN(C(c2csc(Br)c2C)=O)C(CCO)C1 C1(CC(=O)N(CCC(=O)NCCSC)C(C)C)CC2CC2C1 N1(C(Cc2nc(Nc3nc(SC)c(Br)cn3)sc2)=O)CCn2nccc2C1 CCCCCC(=O)NCC1CCC(NC(c2nc(COC)no2)=O)C1 Cc1cc(C(=O)NCCCCCCNC(=O)CNC(=O)C2CC2)cn1C c1(CC)sccc1C(N1CCCC1C1(NC(C2CC(C)=NO2)=O)CC1)=O Cc1cc2cc(C(C)NCC3(F)CCN(C(C)(C)C)CC3)oc2cc1C N1(c2cc(OC)ncn2)CCC(CNC(C2CN3CCC2CC3)=O)C1(C)C C=C=CCCC(=O)NC1CC(C(C)NC(c2coc(C(C)C)n2)=O)C1 C(C(C)(C)CC(=O)NCCCCCNC(C1(CC(=O)OC)CC1)=O)OC C1(O)(CNC(CCc2onc(C)n2)=O)CCCN(C(C2CC2(Cl)Cl)=O)CC1 C(c1cccc(F)c1Cl)=CC(=O)NC1(C)CCN(C(c2ns[nH]c2=O)=O)C1 N#Cc1ccnc(N2CCSC(C(=O)Nc3cc(C(F)(F)F)ccc3Br)C2)n1 C(=O)(CCCC(=O)NC1CCCN(C(=O)C(C)(C2CC2)OC)CC1)OC c1(C2C(C(=O)NCC(CC)NC(c3cc(Cl)cs3)=O)C2)ccnn1C CCCC(C)C(C)N=c1nc2ncn(C)c2c(NCc2ccc(C(F)(F)F)s2)[nH]1 C(C)(CCCCNC(c1cc(Cl)ccn1)=O)NC(CC1(COC)CCCC1)=O c1(OC)ccc(C(N2CCCC(C)C2C)=O)cc1.C(=O)C(C)(C)O.C(C)C.N C#Cc1cc(C(=O)NCCCCCNC(C2CC3CCCCN3C2)=O)ccc1C C1(CNC(CC(=C)C)=O)CCCC1O.n1(CC(=O)N)nc(C(F)(F)F)cc1C c1(CC(N2CCC(N(C(Cn3c(C)nnn3)=O)C)C2)=O)c(F)cccc1F Cc1ccc(=NC(=O)N2CCN3CCCC3C2C(=O)O)[nH]n1 c1(C(N2CC(NC(c3ccsc3Cl)=O)C3(C2)CCC3)=O)ncnc2c1CCCC2 C(=O)(C(F)C(C)CC(C)(C)C)NC1C(C)CN(C(C2SCCCS2)=O)C1 N1(C(C2(CC)N(C(C=CC(CC)C)=O)CCC2)=O)CC2CCCCC12 C1(C)(C(N(CC(C)NC(CCSCCC)=O)C)=O)CCC(OC)CC1 CC1CN(C(c2cnsn2)=O)CCC1N(C(=O)COc1ccccc1Cl)C C1(NC(C(C)OC)=O)CCC(C(C)NC(=O)CC)CC1.C(=O)(C1CC1)N c1(CC)ccc(C)c(C(=O)NCCCC)c1.c1(C=O)cc(C)n(C(C)CC)n1.N N1(C(C2N(C(C)=O)CC(O)C2)=O)CCC2(CC1)CC2C(F)C(=O)O C1(CC(=O)NCCc2cc(C(N(C(CC#C)C)C)=O)no2)CC(=O)NC1=O C(c1ccncc1F)=CC=O.n1(CC)cc(Cl)cc1C(=O)NCC1CCCC1 N1(C(CN(CC)CC)=O)CCN(C(=O)C(=Cc2ccccn2)C)CC1CC(F)F C1CC(F)CN1C(c1cc(Cl)c[nH]1)=O.C(=O)(CC)N(C)C.c1(C=O)cccs1 N1(C(c2cc(SC)oc2)=O)CCC2(CC1)CC2CNC(c1nn[nH]c1C)=O.C CC(O)C(N=c1cc(NCC(N)=O)nc(C(F)(F)F)[nH]1)c1ccc(F)cc1F c1(C(C)NC(=O)CCNc2ccc(F)c(F)c2)cccc(S(C)(=O)=O)c1 N1(C(CCc2cc(C)on2)=O)CCCC(NC(=O)COC2CCCCC2)CC1 Cc1cc(C(=O)NCC#CCNC(=O)C2=NOCC2)c(O)nn1 C1(S(N)(=O)=O)(C=O)CC1.N1(C(C)C)CCN(C(=O)Cc2ccc(O)nc2)CC1 c1(C(N(CCCNC(c2cnsc2)=O)CC)=O)cccc(C2CC2)c1.CCO CCC(CC)(C(=O)N(CCCCN(C)C(c1cc(N)ccn1)=O)C)C(C)C c1(C(N(C(C)C(N2CC(=O)NC(C)(C)C2)=O)CCC)=O)ccc2occc2c1 N1(C(=O)Nc2ccccc2)CC2CC(C1)CN(CC(N1CCCC1)=O)C2 Cc1c(O)c(=O)ccn1Cc1nc(-c2ccoc2)nn1-c1nc(Br)nn1C CCCS(=O)(=O)CC(=O)NCC1CN(C(=O)CCN2CCN(CC)CC2)CC1C CC(C)CCCC(=O)N(C(C)CNC(c1ccc(N2C(=O)CCC2=O)cc1)=O)C C1(NC(C2(C)COC2)=O)CC2CCCC(C1)N2C.c1ncc(Br)cc1C(F)(F)F C12CCC(CC1)N(C(C1CC(CCF)C1)=O)C2.c1(CC(=O)NC)ccc(Cl)cc1 C12(CNC(C3CS(=O)(=O)C3)=O)CCC1CN(C(=O)CCc1ncccn1)C2 c1(CC)cc(C(=O)NC2CC3CC2CN3C(=O)CCCN2CCCC2)ccc1Cl CC1(NC(c2cnc(F)c(F)c2)=O)CCCN(C(C2CC3(C2)CC3(F)F)=O)C1 CC1(C)CCC(CNC(C2(C)CC2)=O)N(C(c2onc3ccccc23)=O)C1 Cc1ccc(N(C(=O)CCC2CCN(C(=O)CCc3cccs3)CC2)C)cc1F C#CC(C)(CC)NC(C1(C2CCCN2C(c2cnn(C)n2)=O)CC1)=O N1(C(C2(CCC=C)CC2)=O)CC2CC(NC(=O)Cc3cnns3)C1C2 N1(C(C2CN(CCOC)C(=O)C2)=O)CC2CCC(C2)C1.C(=O)(C1=C(Cl)CC1)N N1(C(C2C(=C)C2)=O)CCN(C(=O)CCCCNC(N)=O)CC1c1ccccc1 N1(C(c2cc(CC)n(C)n2)=O)CCC(C)(C)CC1.C12(C(=O)N)CCC(CC1F)C2 N1(C(c2c(C)oc(C(C)(C)C)c2)=O)CC2CC(NC(C3OCCC3C)=O)CC1C2 c1(CC(=O)NCC(CC)NC(=O)C(C(C)C)c2ccn(C)n2)cc(C)nn1C C(C(C)(C)CC(=O)N1CC(NC(=O)C(F)(F)C2(OC)CCCC2)C(C)C1)OC c1(OC)nccc2cc(NCC(O)COc3ccccc3Cl)ccc12 N(C1=CCCCC1)(C(=O)NC(C1(O)CCC1)C)CC c1(C(=O)NC2C(NC(c3nc(OCC)oc3)=O)COC2)ccc(Cl)c(N)c1 C(=O)(C1SCc2cccnc21)N1CCN(C2CCN(C(C(C)(C)C)=O)C2)CC1 C1(NC(CN(C2CC2)CC)=O)CCCCN(C(C2CC(=O)CO2)=O)C1 C1(NC(Cc2cn(CC)nc2)=O)CN(C(=O)CSCC(F)(F)F)CC1C1CC1 CC1CN(c2ccnc(N3CCC(c4ccccc4)C3)n2)Cc2cncnc21 c1(OC)c(C)cc(C(=O)NCCCCNC(c2coc3c2CSC3)=O)cc1Cl c1(-c2nc(C)[nH]n2)ccc(C(=O)NCC(c2ccc(C)s2)N2CCOCC2)cc1 N1(C(c2nc(COCC)sc2)=O)CCC(C)C(CN)C1.c1ccc(C#N)nc1 N1(C(CC2CCC(C)O2)=O)CCCN(CCNC(=O)Cc2nnc(O)s2)CC1 C1(C(=O)NC2(CC)CCCN(C(=O)C(C)(C)OC)C2)CCC2(CCCCC2)C1 c1(C(=O)NCC=C2CCN(C(C(C)SC)=O)CC2)ccc(OC(F)F)nc1Cl C12(C(N3CC(CNC(C(C)(Cl)Cl)=O)C(C)(C)C3)=O)CCCCN1CCC2 C(CCCCC(=O)NCCOCC(N1CCC(C(C)(C)C)C1)=O)=CC N1(C(c2c(CC)nns2)=O)CCC2(CC1)CC2NC(=O)CN1CCNCC1 C1(NC(CC2CN(C)C2)=O)CN(C(c2nc(=N)cc[nH]2)=O)CC12CCCC2 C1(C(N(C(CCCC)C)C)=O)COC2(C1)CN(C(=O)C=CC(C)C)C2 N1(C(CC2C(C)OC(C)C2)=O)CC2CCC(C1)N2C(=O)CCc1ncc[nH]1 c1(OC)ccc(CC(C)C(=O)NC)cc1.c1(C(NC)=O)cc(C)[nH]n1.C1CC1 C=C(Cl)C(C)(C)C(=O)NCC=CCNC(=O)C(F)C1CC1 N1(C(c2ccc(CCC)s2)=O)CC2CC(C1)C2NC(c1conc1CC)=O c1(N2CCN(C(c3cnn(C)c3C(F)F)=O)CC2)ncnc2c1c(Br)nn2C c1(-n2ncc(C)c2)ccc(C(=O)NCCCCN(C(=O)C=CCF)C)cc1 C1(C(N(CCC2CCN(C(C(COC)(C)O)=O)CC2)C)=O)CC2C(C1)C2(F)F N1(C(CCCC)=O)CC2(NC(C3CC(=O)N(c4ccccc4Cl)C3)=O)CCC1C2 C1(F)(CC)CCC(C(=O)NCC2(C(OC)OC)CCC2)C1 CC1=C(C(=O)NCCCCCCNC(C2(C)CCCS2(=O)=O)=O)CCCO1 c1(CC(N2CCCC(CNC(c3c(C(C)C)n[nH]c3)=O)C2)=O)c(F)cncc1Cl CON=Cc1ccc(C(=O)NCC(O)CNC(C2CC23CCOCC3)=O)cc1 c1(OC)cc(NC(=O)CC2CN(C(c3cc(F)cc(F)c3)=O)CCO2)ccc1O CC1C(=O)NC(=O)CN1C(=O)C=CC1CCCN1C(=O)C(C#N)C(C)(C)C C1(CCC)CN(C(=O)CN(C)C(C)C)CCN1C(=O)C=C(C)C(F)F C1(N(C(=O)Cc2nccn2C)C)CN(C(C2CCC(C)(C)O2)=O)CC1O C1(CNC(CCC(CC)C)=O)CCC2(CN(C(c3ccc(C)cc3C)=O)C2)O1 Cc1nn(C)cc1C(N1CC(F)(F)C1C1CC1)C(=O)NC1CCCCC1 C1(C(=O)NC(C)C(C)(C)NC(c2nnc(O)nc2O)=O)COc2ccccc2C1 c1(C(=O)NCCCN(C(c2c(C(C)C)con2)=O)C)ccc(C2CCC2)cc1 c1(C(CC(=O)N)C)ccc(F)cc1F.CC1CC(C#N)(C(=O)NCC=CC)C1 c1(OC)ccc(O)c(C(=O)NC2CC(C(=O)NCc3ccccc3I)C2)c1 Cc1ccc2sc(=NCC(C)NC(C3CCCCC34CCC4)=O)[nH]c2c1 C1(C(N(CC2=CCSC2)C)=O)CCC2CCC1N2C(c1occc1C1CC1)=O C1(OC)(C)CN(C(=O)C(C)Cc2cnc[nH]2)C1.C(=O)CN(C)C(N)=O.N Cc1c(C(N2CCC(N3CCC(N4CC(=O)NC4=O)CC3)C2=O)=O)cnn1C Nc1cc(-c2cn(C3CC(NC(C4CCCOCC4)=O)C3)nn2)ccc1Cl N1(C(CC2C(C)(C)CCO2)=O)CCC2CCN(C(C3CC3c3cccs3)=O)CC12 Cc1ccc(Br)c(C(N2CCC(SC(F)(F)F)CC2)C(=O)NC2CCOC2)c1 c1(C(N2C(C(=O)NC(C(=O)NC)C3CC3)C=CC2)=O)ccc(C)cc1O c1(N(CC(F)(F)Cl)C)nc(=NCCOCC(F)F)[nH]c2c1CCC2 C=CC(CC)CC(=O)N1CCC(C2CCCN2C(=O)C(c2ccc(F)cc2)F)C1 N1(C(C2=CC(C)(C)C2)=O)CCC(C2CCN(C(c3nocc3Br)=O)C2)C1 N1(C(C(C)(C)C#N)=O)CC2(CC(C(N3CC(N=[N+]=[N-])C3)=O)CO2)C1 C1(CSC)CCCC1NC(=O)CC1(NC(=O)CCc2csnn2)CCC1 C=CC(O)C(=O)NCC(CNC(c1sccc1-c1ccccc1)=O)OC C12(C(N3CCC(CN=[N+]=[N-])C3)=O)C(NC(c3ccsc3Cl)=O)C3CC1C2C3 Cc1ccc(CC(N2CCC(NC(=O)C3=CCSC3)C2C(C)C)=O)cc1O C1(CCNC(c2c(C)csc2)=O)CN(C(C23CC(C)(CCO2)C3)=O)CC(C)O1 C(=O)(CCC(=O)NC)N1C(C(=O)NCCN(C2CC2)CC)CC1C c1(SCC(=O)NC(C2CCN(C(c3ccc(Cl)o3)=O)C2)C)nnnn1C C1(C(N2CCC(N(CC)CC)C2)=O)CC12CCN(C(c1cc(Cl)c(Br)s1)=O)C2 N1(C(Cn2c(=O)sc(C)c2C)=O)CCC2CCCN(C(=O)O)C2C1.C(C)(C)(C)C=O N1(C(C2(OC(C)C)CCC2)=O)CC(C)C2(CC2)C1.C(=O)C(=O)N(C)C.N C(=O)(CCCCCC#N)N1C(C(N2C(CC)CC(C)C2)=O)CCC1C1CC1 C(=O)(C1OCCc2c(O)cccc21)NCCNc1cc(OC)cc2c1CCC2 N(C1C(=O)Nc2cc(Br)ccc21)C(c1ccc(CC)o1)c1nnnn1C1CCC1 C1(NC(CCn2c(C)ncc2)=O)CCC(F)(CNC(C2CC23CC3)=O)C1 Cc1cc(C(N2CC(NC(c3snc(O)c3Cl)=O)C3CC23)=O)c2c(C)noc2n1 n1(CC(=O)N(CC(CN(C(C(COCC)C)=O)C)O)C)ccc2ccccc12 Cc1c(C(=O)NCC2CCOC2)nnn1C(C)C.c1(CC(=O)N)cncnc1 CC1OCCN(C(c2ccoc2Cl)=O)C1C(=O)NCC1NC(=O)NC1=O C1(NC(CCCC=C)c2ccccc2)CNC2CCC1C2 c1(COC)cccc(C(=O)N(C2CCCC2)CC)n1.C1(CC=O)CCCO1.N C1(C2CCC(=O)NC2)(C(N2CC(NC(=O)CN3CCCC(CO)C3)C2)=O)CCC1 c1(C(N2C(C)CCN(C(=O)CCC3CC3(Cl)Cl)CC2)=O)ccc([N+](=O)[O-])cc1O Cc1cc(C(=O)NC2CCCCCC2NC(C2CCN(C)C(C)C2)=O)nc(O)c1 O=C1OC2CCCC2C1NC(C1(F)CCN(C(=O)C2=CCOCC2)C1)=O C1CN(C(C2CC2)=O)CC12CCC2.c1(NC)cccnc1C(=O)N.C(C)=O.C c1(C(=O)NCC(CNC(C(C)C(C)O)=O)S(C)(=O)=O)ccc(F)c(C#N)c1 C=C=C(C)CC(=O)NC1CC(NC(c2cc(-c3ccccc3)c[nH]2)=O)C1 c1(C(c2n(CCOC)nnn2)NCC2CC2(F)F)cccc(C(=O)OC)c1 C(c1ccccc1[N+](=O)[O-])=CC(=O)NCCCOCC.C1(F)(C=O)CCC1.N c1(-c2c(C(=O)NCCCCCC(=O)OC)csc2)ccc(O)c(F)c1F CC(C(=O)NCC1(F)CCCC1)S(N)(=O)=O.C(=O)CC(C)(C)N(C)C.C CC(C)(C)C(F)(F)F.C(=O)(CCC(=O)NC(CCOCCO)C=O)OCC N1(C(c2cnc(CC)s2)=O)CC(NC(c2cnc(O)n2C)=O)CC(C)C1 C1(NC(C2CC(N(C)C)C2)=O)CCC(F)C1.C12(C=O)CC(C#N)(C1)C2.C C(=O)(CC(C)(C)C(F)F)N1C(CCCNC(c2ccc(C)cc2C)=O)CCCC1 C(=O)(C1CCc2nnc(C)n21)NC(CNC(C=CC=CC)=O)CC CCC(CC(=O)NC(CNC(c1cc(CO)ccn1)=O)CCOC)C(C)(C)C C1(C=O)C2CC3C(C2)C13.C(C)(C(C)(C)C)=CC=O.c1(CCC)nc[nH]n1 c1(OC)ccc(NC(C2CCCN2C(c2[nH]cc(C)c2C)=O)=O)cn1 C1(NC(C(C)(C)c2sccc2Cl)=O)CCC(NC(=O)COCC(F)(F)F)CC1 c1(NCC2OCC(CNC(C3CC(C)OCC3)=O)C2)nccc(C#N)n1 CC1CCCCN1C(c1ccnc(C(F)(F)F)c1)=O.C(=O)(CN(C1CCC1)C)N C(=O)(CCCCC(F)(F)F)NCC(C)N(C)C(c1cc(C(N)=O)sn1)=O C1(NC(CCCC(=C)C)=O)C2COCC1CN(C(=O)C(F)C(C)C)C2 Cc1ncc(C(N2CC(CC(C)NC(C3(C)CCCCO3)=O)C2)=O)c(C)n1 CN1CC=CCC1CC(=O)NC1CCOC(C(N2CC(C3CCCO3)C2)=O)C1 N1(C(C(C)OC2CCCCC2)=O)CCC(C)N(C(c2ccc(Cl)cn2)=O)CC1 N1(C(C2=NOC(C)(C)C2)=O)CCCC12CCCN(C(=O)CCc1ccncn1)C2 N1(C(CC)C(=O)N2CC(C(C)NC(=O)Cn3nccn3)C2)CCN(CCO)CC1 Cc1ncc(CC(=O)NC2CC(NC(=O)CC3CCC(C)O3)C2)s1 N1(C(C(=O)NC(CCSCC)C)=O)CCC(C#N)(c2cc(F)cc(F)c2)CC1 C1(C(=O)NCCCCC#C)N(C(c2cc(C3CC3)on2)=O)CCC1(C)C CN1CC(NC(C23CC(CO)(CN2C(c2cnc(N)cn2)=O)C3)=O)CC12CCC2 c1(N2CC(CC)C2)ccnc(C2CCCC2)n1.C1(C=O)(COCC)CCCO1.N C(=O)(C(C)(C(C)C)OC)N1CCC(C(CO)NC(C(NOC)=O)=O)CC1 N1(C(CN(C(=O)OC)C)=O)CCC(C)C(NC(c2cc(Cl)c(Cl)n2C)=O)C1C C1(C#N)(C=O)CC(=O)C1.c1(C(=O)NCC(COCC)O)[nH]ccc1C N1(C(c2c(C)oc(C(C)C)n2)=O)CC2(CCN2C(=O)C(F)(F)C(C)O)C1 Cc1nc(CNC(=O)CC2CC(=O)NC2=O)oc1C(=O)Nc1ccccc1 C1(NC(c2n(CCC)ncc2)=O)CC(F)CN(C(=O)CC(O)C(C)C)C1 CC1(C)CCCOC1CNC(=O)CC1CCC(NC(c2ccc(Cl)s2)=O)CC1 C1(C2CCC2)(C(N(C2CCC2)C)=O)CC1.C1(C=O)CCCN(S(C)(=O)=O)C1 CCCS(=O)(=O)C(C)C=O.C1(CCC)CN(C(C2(n3cccn3)CCC2)=O)C1.N N1(c2cc(NC3(COC)CCOC3)nc(C(C)C)n2)CCc2nc(=N)[nH]cc2C1 c1(C(=O)OCC)sc2ncnc(NC3(CC)CCCC3)c2c1C C(CCC(F)(F)F)N(C)C(c1coc(CNC(=O)C(C)(C)O)c1)=O CCC(C#N)(CC)C(=O)NC1CCN(CCNC(=O)C(F)C(C)(C)O)CC1 c1(NC(C2CCN(C(C3C(C)(C(C)C)C3)=O)CC2)=O)cccc(F)c1C#N N1(CC)N=C(C(=O)N2C3CCC2CC(N(C(=O)C(C)OC)C)C3)CCC1=O Cc1ccc(C(=O)NCC(O)CN(C)C(C2CS(=O)C2)=O)s1 N1(C(CCCN=[N+]=[N-])=O)CC2(CC(NC(=O)C(F)(F)c3ccccn3)CO2)C1 c1(CC)nc(C#N)cc(=NCC2CN(C(=O)CC(C)n3ccc(C)n3)CCO2)[nH]1 C(CCCCC(=O)NCC(=O)NCC(=O)Nc1cc(O)ccc1C)=CC C1(C)CCCN1C(C1CC1)=O.c1(OC)ncc(C(=O)NC)s1.c1ccccc1 CCC(CNC(=O)C=Cc1nccs1)(CC)C(=O)N1CCC(COC)C1 c1(SC)ccc(CC(=O)NCC(=O)Nc2ccccc2)cc1.C1CC1(C)C OCC(CC1CCOCC1)CN=c1nc2sccc2c(NCCC2CCCO2)[nH]1 C(=O)(C(C)(C)n1cnnn1)N(c1nnc(C2CCC2)s1)C c1(C(N2CC3C(CNC(C4CCN(CC)CC4)=O)C3C2)=O)c[nH]c2cccnc12 C(CNC(C1(CF)CCC1)=O)(CC(F)(F)F)NC(C(C)=CC)=O c1(OC)cc(C(=O)NC2CC(CSC3CCCOC3)C2)cc([N+](=O)[O-])c1.O C(=O)(C(C)(O)C(C)c1ccccc1)N(C(C)CNC(=O)CCSC(F)(F)F)C C(=O)(N=c1cc2c(n[nH]1)CCC2)NC(c1nc(C)sc1)C c1(CC(CN(C)C(C2CC2[N+](=O)[O-])=O)NC(c2coc(C)c2)=O)ccccc1 c1(C(=O)NC2C(NC(c3c(C)ncnc3C)=O)CC2)cc2nn[nH]c2cc1F c1(C(=O)OC)ccc(C(N2CCN(C(C3(CSC)CC3)=O)CC2)=O)cc1Cl C(=O)(C(C)CF)NC(CN(C(c1ccc(Cl)o1)=O)CC)C N1(C(c2c(CC)cccc2)=O)CCC(F)(CNc2ncncc2C)CC1 O=C(C1CCc2snnc21)NC1CCN(C(C2(CO)CCCC2)=O)C1 C(C(C(=O)NCCCC(F)(F)F)C(C)(C)C)NC(c1c(C)n[nH]c1C)=O N1(C(c2c(O)cccc2Br)=O)CC2CN(C(c3cccc4sccc34)=O)CC2C1 C1(CC)CN(C(c2cnsc2)=O)CC1C(N1CC(C(=O)NC2CC2)C1)=O C(C)(C(=O)N(C)Cc1ncccn1)(C1CCCC1)NC(C1(CC=C)CC1)=O CP(C)(=O)c1ccccc1C(=O)NCC1CCN1C(c1cnc2ccccn12)=O c1(C(=O)NCC(CC)(C)NC(=O)CCOC2CCC2)cc2cccnn2c1 C1(NC(CCSC)=O)C2CC3CN(C(c4ccc(C(F)(F)F)c(N)c4)=O)C1C3C2 Cc1oc(S(N)(=O)=O)cc1C(CC1N2CC2C1)=O.C1(C(=O)N)CC1C1CCCC1 C(CCCCCC(=O)N(C1CCCCN(C(=O)CCc2ccnn2C)C1)C)SC Cc1nc2ccccc2nc1C(=O)NC(CNC(=O)C)CC(C)C.CC(N)=O.S c1(NC)cc(Cl)ccc1C(=O)N(C1CCC(NC(=O)CC2CCCOC2)CC1)C C(=O)(C1Cc2ccccc21)N1CCC(C(N(CC)Cc2ncc[nH]2)=O)C1(C)C C(=O)(C1=CCC(NC(=O)C(C)(C)C(C)C)C1)NCCc1ccnc(C)n1 C(C)(C)(C(=O)NCC1COCC1NC(=O)CC1C=CCCC1)SC C(=O)(CC(C)(C)C(F)(F)F)NC1(CO)CN(C(C(C(=O)OCC)F)=O)C1 Cc1nc(C(N2CC(NC(C3CC3F)=O)CCC(O)C2)=O)c2ccnc-2[nH]1 C#CCCC(O)CCNC(C1CCN1C(c1cc([N+](=O)[O-])n[nH]1)=O)=O C1(NC(C(c2ccc(Cl)cc2)(C)O)=O)CCC(NC(C2CCCC(=O)O2)=O)CC1 CC1CN(C(c2cncc(F)c2Cl)=O)CCC1NC(=O)Cc1ccnn1C N1(C(C(CC)c2ccccc2)=O)CCC2C1CCN2C(c1cnsn1)=O N1(C(CCCCOC)=O)C2CC=C(C(=O)N(C(C)CC(C)C)C)C1CC2 C1(NC(c2c(Nc3c(OC)cncn3)cccn2)=O)CC(S(C)(=O)=O)C1 CCC(C)(C)CC(=O)NCC(C)CNC(c1ccc(C(=O)OC)c(Br)c1)=O c1ccc(CC(N2CCC2C(N2CCOC(C(N)=O)C2)=O)=O)cc1.C(=O)OC.N O=C(C#CC1CCNCC1)N1CCC2CCNC2C1 C(=O)(CCCC(C)(C)NC(=O)C(C)n1cccc1)NCC1(CC)CCOCC1 c1(C(C)C)nc(NCCC=CBr)cc(=NC(CCO)C2CCC2)[nH]1 C1(O)(CNC(c2c(C)noc2C)=O)CCCN(C(c2cncc(O)c2)=O)C1 C1(C(N2CCC(O)(CCC)CC2)=O)CC2(CCN1C(=O)C(C(C)O)N(C)C)CC2 CC1CC(C(=O)NC2(C)CCCN(C(=O)CSS(C)(=O)=O)C2)=NO1 Cn1cc2ccc(C(N3CCC4(NC(=O)CSc5nc[nH]n5)CC4C3)=O)cc2n1 C1CN(C(c2cn(CC(F)(F)F)cn2)=O)CCO1.NC(=O)CSCC(=O)N.C c1(OC)cc(C(=O)NCCCCNC(=O)C(C)SC(F)(F)F)cnc1OC N1(C(C2C(=C)C2)=O)CCCCC1c1n[nH]cc1C(=O)NCC1C2CCCC12 N1(C(c2n(C)ncc2Cl)=O)CC2(CNC(=O)CC3(C)CCCO3)CCC1CC2 Cc1cc(C)c2[nH]cc(C#N)c(=NCC3CCN(C(C4(C)CCC4)=O)C3)c2c1 c1(C(N2C(C)CCC(NC(c3csc(Cl)c3)=O)C2)=O)ccc(S(C)(=O)=O)cc1N CCCCCC(C)CC(=O)N1CC(OCCNC(c2cnccn2)=O)C1 C1(C(=O)NC2CC(N(C(c3c(OC)scc3)=O)C)C2)CCCC(OC)C1 C(CC(C(=O)NC1CCCC(NC(C2CCC2C#N)=O)C1)OC)OC CC#CCC(C(=O)N1CCC1c1ccccc1)NC(C1(C2(O)CCC2)CC1)=O C1(C(=O)NC(C#C)(C)C)CSCCN1C(=O)Cn1cccc1 C12(COC(COc3cn(C)nc3)=O)CC(CO)(CO1)C2 c1(C=O)nn(C)c2c1CSCC2.C12CCC(CC1)C2.C(C(=O)N)NC(=O)NC Cc1nc(CNC(=O)C#CC(C)C)oc1C(=O)NC1CCOC(C(C)C)C1 N1(CC(=O)OCC)CCN(C(c2cccnc2Cl)=O)C(CC#N)C1 c1(C(=O)NCCC2(CNC(C(C(C)O)C)=O)CC2)cccc2nncn12 C(=O)(C#CC(C)(C)CNC(C1CC2CCC1CC2)=O)NC(CCC)C(=O)OC N1(C(C(CC)(CO)OC)=O)CCCCCC(NC(=O)Cc2cncc(C)c2)C1 Cc1ccc(CCC(=O)N2CC(CNC(C3(N(C)C)CCCC3)=O)C2)s1 C1(O)(CC)CCN(C(c2cc(Cl)nn2C)C(=O)NC2CC(C(=O)OC)C2)CC1 N(C1CCCc2occc21)Cc1ccc(OCCC#C)cc1 N1(C(C2CC(O)(CC#C)C2)=O)CCC2CN(C(=O)CCCCCOC)CC12 C12(C(N3CCCC(CNC(c4cc(CCCO)on4)=O)C3)=O)CCC(CC1)CC2 S(=O)(=O)(c1c2ccccc2nn1C)NCc1ccc(C)cc1N1CCOCC1 Cn1[nH]c(C2CCCN2C(c2n[nH]cc2C(=O)O)=O)nc1=N Fc1cc(CN2CCCC3(CCC3)C2)c(F)c(Cl)c1F C1CCN(C(=O)CC)C12CC2.c1(NCC)ccc(C(=O)NC2CC2C)[nH]1 C=CCC(CNC(=O)C(CC(=C)Cl)NC(=O)C1=C(C)OCC1)CC(C)C C(CC)(C(=O)N(C1(CC(=O)NC2CC2CC(C)(C)C)CC1)C)OCC Cc1cc(N)ccc1C(=O)NCC1(O)CCN(C(c2ccc(Cl)nn2)=O)CC1 Cc1cccnc1C(=O)NCCC(C(C)C)NC(c1cnn(C2CCC2)c1C)=O c1(OCC(=O)NCC(CNC(COCCC)=O)C)ccc(F)nc1 N1C(=NCCCC)N2CC(S(=O)(=O)C(C)C2)C1.C#Cc1cccc(N(C)C)c1 C1(C(=O)NC(C(=O)OCC)CO)CCC2(CC1)CC(Nc1ccc(Cl)nc1)C2 c1(-c2cn(C3CC(C(=O)NCCc4n(C)nnc4)C3)nn2)cnc(C(=O)O)n1C n1(CC(=O)N(C)CC)ccc2cc(Br)c(Cl)cc2c1=O Cc1ncc(C(N2CCC(F)(CNC(C3CCCC34CCC4)=O)CC2)=O)c(O)n1 C1(C(=O)NC(c2ccc(C)cn2)C)CN(C(c2ccncc2O)=O)C2(CCC2)C1 C1(CNC(c2n(C(CC)(C)C)nnn2)(CC)CC)CC(=O)N(C)C1 N1(C(C(CC)OCC)=O)CCOCC(C)(CNC(=O)Cc2cncc(F)c2)C1 C1(C(=O)N)(COC)CCOCC1.C1CC(C)N(C(=O)Cc2csc(=N)[nH]2)C1 C(CC(C)C(=O)NC1(C)CC(C(=O)N(CC(Cl)Cl)C)C1)OC c1(C(=O)NC(CC2CN(C(C(COC)(C)OC)=O)C2)C)cc2c(cn1)OCCO2 c1(C2C(C(=O)NC34C(CN(C(CCC)=O)C3)C4)C2)ccc(C(F)(F)F)cc1Cl C(CCC1CCC1)(C(=O)NCCC1CCSC1)NC(C(n1ccc(C)n1)C)=O C1CCCN1C(=O)C.c1(C=O)ccc(CS(C)(=O)=O)o1.[SH](C)(=O)=O.CC C(=O)(C1=NOC(CNC(=O)C(=O)NOC)C1)NC(C=C)(C)CC C12(C(=O)NCCC#C)C(NC(=O)C(O)C=C)C3CC1C2C3 c1(OCCNC(C2CC2NCc2csc(Br)c2)=O)ccccc1 C1(C(N2CC(OC(CC)=O)C2)=O)CN(C(=O)C(C(C)(C)C)OC)CCN1C CC(C)C(F)(CNC(=O)C(C)N(C)C)C(=O)N(C)CC1(O)CCC1 C1(CC=C)(NC(=O)CCc2cnn[nH]2)CCCN(C(=O)C(O)C(C)(C)C)C1 CN1CCN(C(=O)C2=CCCCO2)C(CNC(=O)Cc2cc[nH]c(=N)c2)C1 Cc1cc(F)c(NC(C2CCN(C(c3scnc3Cl)=O)CC2)=O)cc1F CN=C1SC(CC(=O)N(CCCC(C)O)C)C(=O)N1C C1(CNC(C(=O)NCC2(C(=O)OC)CCCO2)=O)CC2CCC1N2 c1(OCC(N2CCC(N(C(C3OCCOC3C)=O)CC)C2)=O)ccc(F)cc1F CCCCCC(C(=O)NC1(c2ccccc2)CCN(C(C2(F)CC2)=O)C1)C(C)C N1(C(C(c2cncnc2)C)=O)CC2(CCC(CNC(=O)CCN3CCC3)O2)C1 N1(CC(=O)NC(CCC(C)CO)C(=O)O)CCC2(CC1)CCC(F)(F)CC2 N1(CC=C)C(=S)NC(c2cn(-c3ccccc3)nn2)C2=C1C(C)N(C)C2=O CCCCC(C(=O)N1CCCC(N(C)C(C2CNC(=O)C2)=O)C1)C(C)C C(C(C)(C)C(C)(C)C)NC(C(C)NC(C(CC=C)NC(C)=O)=O)=O N1(C(Cc2c(C)nc[nH]2)=O)CC2CCC2(CCNC(C2(CO)CCC2)=O)C1 c1(-c2nc(C(C)NCCCc3cccc(Cl)n3)on2)ccc(F)cc1 c1(C=O)cccc(C(F)F)c1.C1(CC#C)(C(=O)NC23CC(C2)C3)CCCC1 N1(C(c2scc(Cl)c2Cl)=O)CCCCC1c1ccc(C(F)(F)F)cc1 C1(NC(C2CCC(C)C(C)C2)=O)CCCCC12CCN(C(c1cc(O)cs1)=O)C2 C1(CC(=O)NC2CCC2CNC(C2CC(Cl)(Cl)C2)=O)CN2CCN1CC2 C1(C(N(C2CCN(C(c3ccnn3CC)=O)C2)CCC)=O)CC2(C1)CC(F)C2 C(N=c1[nH]c(Cl)nc2c1COCC2)C1(O)CCCN(C(C(C)(C)C2CC2)=O)C1 C(=O)(C(F)C(F)(F)F)NC(CN(C(=O)C(C1CC1)C1CC1)C)(CO)CO N1(C(C=CC(CC)C)=O)CCC(C)(NC(c2coc(N(C)C)n2)=O)C1 c1(C(=O)NC(C)C(C)NC(c2csc(CCP(C)(C)=O)n2)=O)ccccc1 Cc1cc(Br)oc1C(=O)N(C)CC1(NC(=O)COCC(C)C)CC1 C(CC(C)C(=O)N1CCC(N(C(=O)CCn2nc(C)nc2C)C)C1)=CCC CCCC(F)C(=O)NCC(CC1CC1)C(=O)NCCC1CCCCC1 N1(C(c2nc(CCC)sc2)=O)CCN(C(C2(C(C)C)CCC2)=O)CC(O)C1 c1(C(=O)OCC)cc(C(N2CCC(CCNC(C3CC3F)=O)C2)=O)[nH]c1C c1(C(N2CC(CCCCNC(CCCCC)=O)C2)=O)ccc(OC)cc1C(F)F CC1(NC(C2CC2(C)C)=O)CCC(NC(c2cc(O)nc(O)c2)=O)CC1 C12(CNC(c3ccc(F)cc3)CC(=O)Nc3ccncn3)CCC(CC1)C2 C(C)(C)(C(=O)N1CCCC1)NC(=O)NCC=C.c1cnn(C)c1.C(=O)C c1(C(N2CC(C(C)(C)O)C2)=O)cnnc(C)c1.C1(CCC)CCCC1C(=O)N C(=O)(C1=NOC2COCC12)N1C(CC)C(C(=O)N(C)Cc2ccccc2C)CC1 C1(NC(C=CC)=O)COC2(CCCN(C(c3ccc(S(C)(=O)=O)o3)=O)C2)C1 C(=O)(C1=CCCOCC1)NC1(CC(=O)NC2C(C)C2C)CCCCC1 c1(CNC(C2(C)CCC(C)CC2)c2n(CCSC)nnn2)c(C)nn(C)c1Cl c1(SCCC(=O)N(C(CNC(C23CCC2C3)=O)C2CC2)C)ccccc1Cl C12(C(=O)NCCC(C)N(C(CC(C)c3ccco3)=O)C)CC(C)(CCO1)C2 CC(C)CC(O)C(=O)N1CCCC(N(C(=O)CC2CCC2C)C)CC1 N1(C(CCCC(=C)C)=O)CC2CCCC1(CNC(c1ccc3c(c1)OCO3)=O)C2 C1(C(=O)NC(C23CC(CO2)C3)C)CC2CCC1CC2.C1(C)(C=O)CC1(F)F N1(Cc2c(C)ccnc2)CCC(C2CCN(C(C3CCC(F)C3)=O)CC2)C1 C1(C(=O)NCC=CCOC)CC(C)(C)CCN1C(=O)CC(C)(F)F C1(C(=O)NCC(C)NC(C2CCOC2(C)C)=O)CCCCCCC1 Cc1cc2scc(CC(N3CCN(C(C4(C)CCCOC4)=O)CC3CO)=O)c2s1 c1(C(N2CCC(C=CC(=O)NC(C)CS(C)(=O)=O)CC2)=O)cnn2ccccc12 CC1CCC(S(C)(=O)=O)CN1C(C1CCCCC1)=O c1(C(N2CCC(CC(=O)NC3CCCCC3)CC2)=O)c(F)cccc1I N1(C(CC2(OC)CCCC2)=O)CC(C)C(C)(C)C1.C1(C(=O)N)CN2CCC1CC2 C1(C(C)NC(CSCC#C)=O)CCN(C(C2(F)CCCC2)=O)C1 c1(C=O)cccc2sncc12.Cc1cnc(C(=O)NCC2(CC)CC2)c(C)c1.N C1(N(C)C(c2csc(Cl)n2)=O)CCC(NC(C2CC2(c2ccccc2)C)=O)CC1 N1(C(C2CCCCN2C(c2cccc(O)c2Cl)=O)=O)CCc2ccccc2C1 c1(C(N2CCC(NC(CC(C)F)=O)C2C)=O)cc2cc(Br)cnc2s1 C1(NC(C23CC(C(C)(C)C)(C2)C3)=O)CCSC12CN(C(C1CCCOC1)=O)C2 C1(NC(C(=CC2CCCC2)C)=O)CCCC(C(=O)NC(c2sccc2C)CO)C1 c1(CCC(=O)NC2CCN(C(C(CC)OC)=O)C2C)ccc2[nH]ccc2c1 C1(NC(C(CC)(C)O)=O)CCN(Cc2cc(OC)c(O)c(Cl)c2)CC1(C)C c1(C2(C(=O)NC(C(C)NC(c3ccnn3C)=O)CO)CCC2)ccc(F)cc1F N1(C(C(CC)(C)F)=O)CCC2(CC1)CC2NC(C1CC2CC2C1)=O CC1=C(C(=O)NC(C2CCOC2)C)CCC1.c1(CC(=O)N)nocc1C(C)C c1(CC)noc(C(=O)NCC(C2CC2)NC(=O)C(C)(C)C2CC2)c1C c1(C(=O)NCC(CC)Nc2ncc3ccnc-3[nH]2)ncnc2c(C)csc12 N1(C(c2cnc(CC)s2)=O)CC2(CC2)CC1CC(=O)NCCc1cn(C)nn1 c1(C(N(CCNC(=O)CC2CCCC2C)CC)=O)ncc(Cl)cc1O CC(C)(CC(=O)NCCC1(O)CN(C(C2C3CCCC23)=O)C1)C1CC1 C1(C(=O)N)CCN(C2CC2)S1(=O)=O.c1(NC)ccc(C(=O)N(CCC)C)nc1 Cc1ccc(CNC(=O)C(=O)NC(C)C(c2ccccc2)C)nn1 N1(C(c2cscn2)=O)CCCC2(C1)CN(Cc1ccc([N+](=O)[O-])c(Br)c1)CCO2 c1(NCC2CC(C)(O)C2)cc(NCC2(CC3CCC3)CC2)ncn1 c1(CC(=O)NC(CNC(C(C)NC(CC)=O)=O)CC(C)C)n[nH]c2c1CCCC2 c1(C(N(CC(CN(C(C(c2ccn(C)c2)C)=O)C)O)C)=O)cc2ccncc2[nH]1 N1(C(Cc2c(CC)cccc2)=O)CCC(NC(c2ccnn2C)=O)CC(C)(C)C1 N1(C(C(C(C)C)O)=O)C2CCC1CC(NC(=O)Cn1cccc1)C2 Cc1ccc(F)c(C(=O)NC2CC(NC(=O)Cc3ccc(O)nc3)C2)c1 CCCC(CC(=O)OC)C1(CNCCOCC)CCC1.c1ccn[nH]1.C(=O)N c1(C(=O)NCC2CC3CCC2N3C(c2cc[n+]([O-])cc2)=O)cc2c[nH]cnc-2n1 Cc1cc(C)c(CCN2C(=O)NC(Cc3cnn(C(C)(C)C)c3)C2=O)c(C)c1 Cc1[nH]nc(C(=O)NCC=CCNC(=O)CCCc2cccnc2)c1F CCC(C)C(C(=O)NCC(C)N(C(=O)Cc1c(C)noc1C)C)N(C)C Cc1ccnnc1C(N1CCCC(C(C)NC(c2ccc(CO)cc2)=O)C1)=O C1(C(=O)NCCCC2CCCN2C(C2CCCSC2)=O)C2CC3C(C2=O)C13 Cc1nn(C)c(F)c1C(N1CCC(O)(C)C1)=O.c1(CC=O)ccc(F)cc1F.N N1(C(C(CCOCC)NC(=O)CCC(C)(C)C)=O)CCOCC2(CCC2)C1 C1(C(N(C(CC)CO)C)=O)CCCN1C=O c1(SC)ccc(N)cc1C(N1CCCC(NC(=O)CC(C)(C)C)C1C)=O C1(CC)(CC)CCCN(C(c2ccsc2C)C(=O)NCC2CCCO2)C1 Cc1ccc(C)c(CN2CCC(CNC(=O)CCC3CCOC3)C2)c1 c1(N2CC(CC)(CC)SCC2)nc(NCCC(=O)N(C)C2CC2)c2ncsc2n1 c12cc(Br)ccc1NC(C1CCCO1)c1nnnn1C2.c1(CC)ccccc1O C1CCCCC1.C1(C(c2n(CCC)nnn2)NC)CCN(C)C1=O.[SH](C)(=O)=O C1(N(C(CCN(C)CC)=O)CC)CCN(C(c2c[nH]nc2C2CCCO2)=O)C1 CCC(CNC(=O)CN(C)C)N=c1[nH]c(C2CCCC2)nc(=N)[nH]1 N1(C(C2(CCCC)CC2)=O)CCN(C(c2cc(C)oc2C)=O)C(c2cn[nH]c2)C1 C=CC1COCCN1C(c1ccc(CNC(C2CC(CC3CC3)C2)=O)o1)=O CC(C)CC(O)C(C)C(=O)N1CC(CF)(NC(=O)C(C)Cc2cnco2)C1 c1(C(=O)NC2CCN(C(CC(C)F)=O)CC2C)ccn2cccc2c1 CC1CN(C(C2CCN(C(c3cc(O)nn3C)=O)C23CC3)=O)CC1(F)F CC1CC(C=O)CN1C(=O)CC.C(C(F)(F)F)=CC=O.C(C)(C)C.CC CC1CCC(NC(=O)Cc2csnn2)CN1C(=O)Cc1cncs1 N1(C(CNC(C)=O)=O)CCOCC(CNC(=O)C(C)n2cncn2)C1 n1(CC(=O)NCC2N(C(C(C3CC3)OC)=O)CCOC2)cnc([N+](=O)[O-])n1 Cc1nccc(CNC(=O)CC(C)CNC(C2(N(C)C)CCCC2)=O)n1 c1(CC(N2CC(O)(C(C)NC(c3ccnnc3)=O)C2)=O)cc2ccccc2nc1O CC(CC(=O)NC(C)CCCCNC(=O)CCc1ccc(CO)cc1)C(F)F C#CCC(C)(C(=O)N1CC(CC)CCC1C)NC(C1CC(C)=NO1)=O Cc1nc(N2CCOCC2)c(CNCc2ccccc2C)s1.C(=O)N.C1CC1 C1(O)(CNC(C2C(C)CCO2)=O)CCCN(C(c2ccc(F)cc2F)=O)C1 CCC(C)C(O)CC(=O)N(C1CN(C(C2CCOC2)=O)C1)C C(=O)(CCCC(C)NC(C1C=CC1C(=O)OC)=O)NCCC#CCC c1(Oc2ccc(C)cc2)nnc(C)c(C)n1.c12cn(nn1)CC(C)NC(=O)CO2 Cc1ccc(C2(F)CN(C(=O)C(=O)Nc3cccc(I)c3)C2)cc1 c1(COC)cncc(C(N2CCC(NC(=O)C=Cc3ncc[nH]3)C2)=O)c1 C1(NC(CCN2C(C)CCCC2)=O)CCN(C(=O)Cc2csc(=N)[nH]2)C12CCC2 N1(C(C(C)NC(C)=O)=O)CC2CN(C(=O)CCc3ccc(C)cc3)CC12 n1(CC)nc(C(=O)NC2CC2)ccc1=O.c1(C(=O)N)cnnn1-c1ccccc1 C(=O)(C(C)S(N)(=O)=O)NCCN(C(c1c(OC)nccc1)=O)C N1(C(c2cc(CC)n(C)n2)=O)CCN(C(=O)CC2(C)CC2(F)Cl)CC(C)(C)C1 CC1(C(N2CCC3(NC(=O)CS)CC3C2)=O)COC(=O)OC1.c1ccc(Cl)cc1 Cc1cc(F)c([N+](=O)[O-])cc1S(=O)(=O)N(C(c1ccccc1)C(=O)O)C C1(C(=O)NC2CC(NC(C3(C#C)CC3)=O)C2)CCCC2(C1)CC2(F)F C1(CC(=O)NCC(C)(F)F)CCN(C(=O)CSc2ccc(N)cc2)C1(C)C Cc1cc(Br)ccc1S(=O)(=O)NC1CC1C(=O)N=c1[nH][nH]cc1C c1(C(N2CC(CC)OCC2)=O)c(C)c(C)cc(C)c1C.C(C(C)C(=O)N)OCC c1(C(c2n(CCCSC)nnn2)NCCO)nnc2n1CCCC2.C1CCCO1.C C1(CC)OCCC1C(N1CCCC1CNC(=O)Cn1ccnc1C)=O N1(C(c2c(CC)nccn2)=O)CC2(CC(NC(C3CCOC3)=O)c3nccn32)C1 C1(C(=O)NC(C)CCN(C(=O)CN(C)CCO)C)CCCc2ccccc2C1 O=C(CCCOCC(=C1CN(C(=O)Cc2ncc[nH]2)C1)F)N.c1ccccc1.C Cn1nnc2ccc(C(=O)NCC3CC3NC(c3cc[nH]n3)=O)cc12 C1(NC(c2c(C)ncnc2)=O)CCN(C(C23CCCN2CCC3)=O)CCC1CO CC(C)C(C)(Cc1ccccc1)C(=O)N1CC2CC(CNC(=O)C3=CCC3)C2C1 N1(C(COC(C)C)=O)CCCC2(CCCCC2NC(=O)C(=O)NCC(F)F)C1 Cc1cc(C(=O)NC2CC(C)N(C(=O)CCCc3nnc(C)n3C)C2)c(C)[nH]1 N1(C(C=C(CC)CC)=O)CC2CCC(NC(c3cccn(C)c3=O)=O)(C2)C1 c1(CC(=O)N(CC(C)N(C(C=CC(CC)C)=O)C)C)c(C)cc(O)cc1C N1(C(c2nccnc2CNC(C2(F)CCNCC2)=O)=O)CCC2(CCOC2)C1 c1(C(=O)NCC(C)(CO)NC(CCc2ncc(C)[nH]2)=O)ncnc2c1CCCC2 CCC(C)CN=c1nc2sccc2c(NC2CCC(F)(F)C2)[nH]1 C(C(=O)N1CCC(CNC(=O)Cc2cscn2)(OC)C1)(C(C)(C)C)OC N1(C(C(COC)(C)C)=O)CCN(C(c2cc(Br)no2)=O)C2CCCCC2C1 c1(CC(C)C)cc(C(N2CC(CO)C2)=O)cc(O)n1.C(=O)(CN=S(C)(C)=O)N C1(C(=O)NC2(C3CCCCN3C(c3csc(O)n3)=O)CC2)CC12CCCCC2 CC1CN(C)CCN1C(=O)NCCCc1ccn(C)n1 c1(C(N2CC(CN(C3CC(CN(C)C)C3)C)C(C)C2)=O)ccc2c(c1)OCC2 C1(c2n(C)ncc2)CN(C(=O)CSc2cn[nH]c2)CC1.C1(C)(C(=O)N)CCOC1 Cn1nc2c(c1C(N1CC3CCC1CN3C(=O)CCN1CCCCC1)=O)CCC2 C1(C2CCCN(C(C3CC34CC4)=O)C2)(NC(c2cc(CCC)on2)=O)CC1 c1(NC(C2CCCN2C(=O)CN)=O)cccc(F)c1Cl.[SH](=O)(=O)c1nccs1 c1(CNS(CCc2c(C)ncs2)(=O)=O)cccc(C2CC2)c1 c1(CC)c(C(N2CCC(CNC(=O)C=CS(C)=O)(O)C2)=O)[nH]c2ccccc12 Cc1c(C(=O)NCCCCN(C)C(C2(c3ccno3)CC2)=O)cncc1Br Cc1cc(C(=O)NCCC2CCN(C(C3CC(C)OC3C)=O)CC2)cc(N)c1 Cc1ccc(C(=O)NC2CC3(C2)CC(C(=O)N(C)CC2CC2)C3)c(C)c1 Cc1ccc(O)c(CC(=O)NC2CCC(C)N(C(C3CCC34CCC4)=O)C2)c1 N1(C(c2cnn(C(CC)C)c2C)=O)C2CCC(C2)C1CNC(c1cncnc1)=O CC(c1ccccc1Cl)=CC(=O)NCC1CN(C(c2cc(O)no2)=O)CCC1C C(=O)(CS(=O)(=O)c1ccccc1F)NCCCC(C)NC(Cc1nc(C)oc1)=O Cc1sc(-c2ccccc2)nc1C(=O)NC1CC1.c1(CCC=O)nc(=N)[nH][nH]1.N CC1=C(C(=O)N(C)CC2(NC(=O)C(C)C(C)(C)C)CC2)Cn2ncnc2N1C c1(C(=O)NC2(CNC(C3N(C)C(=O)NC3)=O)CCCC2)cc2c(s1)CCC2 c1(N2CCCCC(SCC)C2)ccc2c(n1)OCCC2=O c1(CNC(=O)NC2C(C)(CC)C2)cccc(Cl)c1O C(=O)(C(C)(F)C(C)(C)F)N1CC(CC(C)NC(c2ncn(CC)n2)=O)C1 c1(C(=O)NC(CNC(COCCC)=O)CO)nn2c(c1C)OCCC2 N1(C(C(C=C)O)=O)CC2(CCCC2NC(c2ccc(F)c(OC)c2F)=O)C1 Nc1cncc(C(N2CCCC(NC(=O)COCC(N3CCCC3)C)C2)=O)n1 C1(C(N(C2CN(C(C(n3ccc(C)n3)(C)C)=O)CC2O)C)=O)CCC=CCCC1 CCC(CCCC(=O)NC1(C)CCC(=O)N(C)C1)NC(=O)CN=[N+]=[N-] C(=O)(CCC[N+](=O)[O-])N(CC(C)NC(c1ccc(C)n1C)=O)C N(C1CCc2cc(CNC(c3ccon3)=O)ccc21)C(CC1CCN(C)CC1)=O c1(C(N(C(C2CCC2)C)CC)=O)cc(CNC(c2ccncn2)=O)ccn1 C1(C(N(C(CSC)C)C)=O)N(C(=O)Cc2ccoc2C)CC12CCCC2 N1(CC)CCOC(C(=O)N(CC(O)CNC(c2ccc(C(C)=O)o2)=O)C)C1 C1(C(=O)NC(CNC(C2(C)CC2)=O)C2CC2)CCc2ccnn2C1 c1(C(N(CCC(N)=O)C)=O)ccccc1-n1cc(-c2ccns2)nn1 C#Cc1ccc(F)cc1C(=O)NC(C(C)NC(C1(C#C)CCC1)=O)C(C)C S(=O)(=O)(c1ccc([N+](=O)[O-])c(Cl)c1)N1CC(NC(C2CC=CCC2)=O)(C)C1 C1(C)(NC(C=C)=O)CCN(C(=O)C(c2ccc(OC)cc2)C)C1 Cc1ccc(CNC(=O)COc2cccc(F)c2F)c(N(C)C)c1 C(=O)(C1=CCCCC1P(C)(C)=O)N(C(CNC(c1cc(CC)c(F)cc1)=O)C)C CC1CC(NC(=O)C(F)CC2CCCC2)CCN1C(C1CC(N=[N+]=[N-])C1)=O CC(C)S(=O)(=O)c1ccc(CNc2ccc(C(C)(C)C)cc2)cc1 N1(C(c2ccc(OC)cc2N)=O)CCCN(C(C2CC(=O)NC(C)C2)=O)CCC1 S(=O)(=O)(c1cccnc1NC)NCC1(C)C=CCCC1.C1NC(=O)CC1(C)C C12COC(C(=O)N)(C1)C2.C(CC(O)CNC1(c2ccccc2)CC1)OCC c1(OC)cccc(CC(=O)NCC2CCC(c3ccccc3)O2)c1Cl n1(CC)ccnc1C=CC(=O)NCC1CCCCN1C(=O)CCO.C(N)=O.N c1(C(=O)NCC2N(C(c3ncc(CC)s3)=O)CCCC2)occ2c1CCOC2 c1(OC)nscc1CNC(=O)CC1(NC(C2CC(C)C2)=O)CCC1 Cc1cc(-c2ccc(CN3CCN(c4ccccn4)CC3)s2)cc(O)c1 N1(C(c2cccc(CNC(C=CCCC)=O)n2)=O)CCC(N(C)C)C1(C)C CS(=O)(=O)c1ccc(C(N2CCOC(CC(=O)NCCN3CCOCC3)C2)=O)cc1 c12cc(C)ccc1O2.c1(CNC2(C(=O)NCC)CC2)c(C)noc1C N1(C(c2cc(C)n(C)c2)=O)CCC(C)CC1C(=O)NCC1CCCCN1C O=C(CC(F)(F)Br)NCCN(C1CCCCC1)C(=O)CC1(CO)CC1 CN(CCCC(=O)N1CC2C(NC(=O)CC(C)(C)O)C2C1)N=O N1(C(c2c(C)c(Br)sc2)=O)CC2(COC(CNC(c3ccon3)=O)C2)C1 C1(SC)CCCC1NC(C)(C)C.C12CCC(C1)n1nnnc1N2 N(S(=O)(=O)N1CCC2(CCCCC2)CC1)C1CC(C[Si](C)(C)C)C1.CCO Cc1cc(C(=O)NCC(C)N(C)C(C2CC(F)(F)C2)=O)c2c(c1)CCC2 N1(C(CC2N(C(CN(C(=O)OC)C)=O)CC2)=O)CC(CO)C1(C)C CC(C(=O)NC12CC(NC(c3cnc(N(C)C)cn3)=O)(C1)C2)C(C)(C)C c1(CC)ccc(C(=O)N)cc1F.C(=O)(C(C)N(C)C(C)=O)NC.C1CC1.C c1(CCC(=O)NC2CC(C)(NC(CN(CC)CC)=O)C2)c(C)n[nH]c1C c1(OC)cccnc1C(=O)N(C(CNC(C12CC1C2)=O)C1CC1)C C1(NC(CN(C)CC)=O)CS(=O)(=O)C12CCN(C(c1cc(N)ccc1Cl)=O)CC2 C1(NC(C(C)=C(CC)C)=O)CCCC(CC(=O)N(C)CC2CCOC2)C1 N1(C(C2(CC)CC2)=O)CCC2C(C1)CN2C(=O)C.c1(C=O)ccc(Cl)cc1Cl CC1(C)CCN(C(=O)CSC(F)(F)F)C1C.C1(C)(C=O)CCC(F)(F)C1.N Cc1cc(C(N2CCC(NC(C3(F)CC3c3ccccc3)=O)C2C)=O)cc(F)c1 C(C(CC(F)(F)F)NC(=O)C(F)CC1CCCCC1)NC(c1cncs1)=O c1(-c2nc(-c3ccc(F)c(Cl)c3)nn2CC2CCCO2)ccc(F)cc1.CCC N1(C(c2cc3c([nH]2)CCCC3)=O)CCN(C(C2(Br)CC2)=O)CC2(CC2)C1 c1(C(=O)NCC2C(NC(C3(CC)CCC3)=O)CCC2)cccc2nn[nH]c12 N1(C(CC=C)=O)CC(n2cc(C(O)Cc3ccccc3)nn2)(C(=O)OCC)C1 C=CC(C)CC(=O)NCC12CC(NC(c3cn(C)nc3SC)=O)(C1)C2 c1(NCCC2(C(C)(F)F)CC2)cc(=NCCCCCCCN2CCCC2)[nH]cn1 N1(C(CCN(CC)CC)=O)CCOCC1CC(=O)NCc1cc(CO)[nH]n1 C1(NC(C2(CC#C)CCOC2)=O)C2CC1N(C(=O)C(O)CC1CCOCC1)C2 N=S(=O)(O)c1ccc(-c2cncnc2C(N2CCCCC2CO)=O)cc1 c1(C(=O)NC2C=CCC(C(N3CCCC(C)C3CO)=O)C2)ccc2nccn2c1 N1(C(CNC(C(C)SC(C)C)=O)C)CCN(C(=O)CC2CC(F)(F)C2)CC1 C=CCCCC(C)(C)C(=O)NC1CC(CCC(=O)NC(C2CC2C=O)C)C1.O Cc1c(C(=O)NCC(C)C(F)C(=O)N2CCOC(C)C2C)cncc1F CC1CN(C(C2CC2c2ccccc2)=O)CC1NC(c1cnnn1C)=O C1(NC(CC=C=C)=O)CCCN(C(c2cc(N3CCCC3)cc(Cl)c2)=O)CC1 Cc1cc(Cl)c(C)c(C(=O)NC2CC(C)N(C(c3ncsc3C)=O)C2)c1N C1(NC(CNC(c2ccc(C)s2)=O)=O)CC2CC1CN(C(=O)CC(C)O)C2 C1(C(N2CC(CC=C)(NC(c3ccccc3SC)=O)C2)=O)CCCC(C#N)C1 Cc1ccc(-c2nc(CC3C=CCC3)n(Cc3ccc(Br)cc3)n2)cc1 c1(NC(CN(C(c2cncc(OCC)c2)=O)C)C)nc(C)ccc1C(=O)OC C(CC(=O)NC(c1nc[nH]n1)CO)(C(C)CC)NC(C(CCC)=CCC)=O C(=O)(C(O)C(C)c1ccccc1F)NCCOC.C(=O)C(C)=C1CCC1 C1(C(=O)NCCOC2CN(C(C(C)P(C)(C)=O)=O)C2)CCC2(CCCC2)CC1 Cc1nc2ccccc2c(C)c1CC(=O)NC1CCN(C(c2cnc(Cl)[nH]2)=O)C1 CC1(C)Cc2cc(C(=O)NCC3CC(NC(C45CCCCC4C5)=O)C3)sc2C1 c1(OC)cccc(C(C(=O)NC2CCC(NC(C3CC(O)C3)=O)C2)OC)c1 OC1CCc2cc(Br)c(NC3CC(c4ccccc4Cl)C3)nc21 CCC(C)C(C(=O)NCC1(CO)CCN(C(c2cc(C)c(O)nn2)=O)C1)OC Cn1c(C(N2CCC(CF)(NC(c3ccc(=O)n(C)c3)=O)C2)=O)ccc1C#N N1(C(Cn2c(C)ccn2)=O)CC2COCCC2(NC(C2CC(=C3CC3)C2)=O)C1 C1(CNC(CSCCOC)=O)CC2(CO1)CN(C(c1[nH]ccc1C)=O)C2 CC1(C)CN(CC(=O)O)CCO1.N12CCC(C(NC(=O)C(F)(F)F)C1)NC2=O CC1CN(C(c2cnc3scnc3c2)=O)CC(C)C1NC(=O)CS(=O)(=O)C1CC1 C=C(C)CCCN=c1nc(N2CCc3c(O)noc3C2)c2c([nH]1)CSC2 C=CC(C)CC(=O)NCC(C(=O)NCCC1CCN(C)C1=O)N(C)C CCCC(C)(CC)C(=O)NCCC(CC)(CC)NC(c1ccnc(C(F)F)c1)=O c1(CCC(N2CC(C)(C)C(NC(c3cc[nH]n3)=O)C2)=O)cc2ccccc2o1 c1(C(=O)NC2(C)CC(NC(c3scc(C)c3)=O)C2)cc(C2CCOCC2)nn1C N1(C(c2cn(CC)nc2)=O)CCCC(NC(c2ccc(Br)nc2O)=O)C1C Cc1ccc(O)cc1C(N1CC2CC2(CNCc2cccc(Cl)n2)C1)=O N1(C(CCCOC(C)C)=O)CCC(F)C(NC(=O)CCc2nccn2C)C1 C(=O)(C(CO)NC(c1sccc1F)=O)NCCN(C)C(=O)C1CC1 c1(C(=O)NCCCC(C)(C)NC(c2c(C)c[nH]n2)=O)ccc(=O)n(C)n1 c1(C(=O)NC2CCCN(CC(=O)N(C)CC)CC2)cccc2ccnn12 N1(C(c2cncc(C)c2C)=O)CCC2(CCCN(C(=O)CSC(C)C)C2)C1 C(N=c1[nH]c2c(c(=NC(C)C3CCCO3)[nH]1)CSC2)c1c(C)non1 Cc1cc(C(=O)NCC2COCCN(C(=O)CC34CCCC3C4)C2)ccc1F CCCCC(C)CCC(=O)N1CC(O)(CCNC(c2ccnn2CC2CC2)=O)C1 N1(C(Cc2cnc(C)s2)=O)CC(CNC(c2cccc(N(C)C)n2)=O)C(C)C1 N1(C(C(n2ncc(C)c2)C)=O)CCCC(NC(=O)COCCC(C)C)C1C C(=O)(CC(=O)NC(Cc1ccoc1)C(=O)NCC(CC1CC1)CO)N(C)C Cc1nc(N)c2c(C)c(C(N3CCC(NC(C4CCSC4)=O)CC3)=O)sc2n1 C1(NC(=O)OC(C)(C)C)CCC(C(N2CCCCC2C(C)(C)C)=O)OC1 CCCCC(C(=O)NC)NC(C1CC(O)CN1C(=O)CCS(C)(=O)=O)=O c1(CC(N2CCCC(NC(c3c(CC)onc3)=O)C2C)=O)ccc2n[nH]cc2c1 N1(C(Cc2cn(C(C)C)nn2)=O)CCC(NC(C2CCCN2C)=O)CC(C)(C)C1 Cn1cc(C#CCNC(=O)C(c2cn(C)nn2)NC(=O)Cn2ccnc2)cn1 Cc1nc(C)c(C)c(=NCC(C)N(C(=O)C=Cc2cnc(O)nc2O)C)[nH]1 C#CCC(C)(C)C(=O)N(C)CC1C2CN(C(c3cnoc3C(C)C)=O)CC12 C12(NC(c3cncc(SC)c3)=O)CCCC(NC(c3cccnn3)=O)(C1)C2.O C1(C=O)C2CCCCCCC12.CC1(C)CC(C)(C(=O)NC)C1.C12CC(CO1)C2 c1(C(=O)NCCC(C)N(C(=O)C#CC(C)(C)C)C)ccc(Br)c(Cl)c1F O=S(=O)(c1ccc(=NCCCCc2nccs2)[nH]c1)N1CCC2(CCCCC2)C1 N1(C(c2nccc(C)n2)=O)C2CCCC1CN(C(c1cnc3[nH]cncc1-3)=O)C2 c1(C=O)cc(O)cc(=O)o1.c1(C(=O)NCC(C)CO)cc(C(N)=O)ccn1.N c1(NC(C)=O)nnc(N2CCCC(C(F)(F)F)C2)n1C.N12CCN(CC1)CC2 c1(N2C(N(CC(=O)N(CC)CC3CCNC3)C)COCC2)cc(S)nc(C)n1 Cc1cc(F)ccc1CNCc1ccc(C(F)F)o1 Cc1ccc(CC(=O)NCCNC(=O)CC2CCS(=O)(=O)C2)cn1 N#CC1CN(C(C2CC23CCN(Cc2cccc(-n4cncn4)c2)C3)=O)CCO1 N#CC1(C(=O)N(CCNC(c2cn[nH]c2)=O)C2CC2)CCC(=O)CC1 c1(CC(N2CC3C(C(=O)NC4(CC)CCNC4=O)C3C2)=O)ccc(Cl)c(Cl)c1 N1(C(c2c(COC)cc[nH]2)=O)CCOC(C)(CNC(=O)C2=CCCS2)C1 Cc1nc2c(o1)CCCC2CC(=O)N1CC2C(CNC(=O)Cc3nc[nH]n3)C2C1 C1(NC(c2cc(C)n(C)n2)=O)CC2CN(C(C3CC(C(C)C)=NO3)=O)CC12 C1(OC2CN(C(C(CC)OC)=O)C2)CCN(C(=O)C(C)OCCC(C)C)CC1 C(N=c1[nH]c(=NCCN(C)CC)c2cccc(F)c2[nH]1)c1ncc(CC)s1 c1(C(=O)NC(CCOC)CNC(c2c[nH]nc2C)=O)cccc2oc(C)nc12 C1CN(C(c2cncc(C(F)F)c2)=O)CC1(C)C.CN1CCC(C)(C(=O)NC)C1 Cc1c(C(=O)NCC(C)(C)CNC(C2CCCN2CCC(C)C)=O)cncc1N c1(C(=O)OC)nc(C)c(S(=O)(=O)NC2CC(c3nncn3C)CC2O)s1 CCCC(C(=O)NC1(CNC(C2(Cl)CC2(C)C)=O)CCC1)c1ccccc1 c1(C=O)nc(Cl)c(=O)[nH]c1N.C(C(C)C(F)(F)F)NC(C(C)(C)C1CC1)=O.N c1(C(N(CC(N2CCN(C(CCC#C)=O)CC2)=O)C)=O)ccc2nnc(S)n2c1 N1(C(c2cc(C)c(Cl)s2)=O)CCN(C(C2CC2C)=O)C(CF)C1 Cc1ccccc1C(=O)NC1CCCC1CNC(=O)Cc1ccccc1 N1(C(C=CC=CC)=O)CCCN(C(=O)Cn2ccc([N+](=O)[O-])n2)C(C)C1 C(C)(CO)(C(=O)NCC1CC1)NC(C)=O.C1(CC(C)C)(C=O)CC1.C c1(C(=O)NC(C(=O)NCCCC2(C)CC2)C2CCC2)c[nH]c(=N)o1 Cc1ccc(C(CNC(=O)C(C)(Cl)Cl)NC(C2CC(n3ccnc3)C2)=O)cc1 c1(C(N2CC3CN(Cc4c(C)ccc(Cl)c4)C3C2)=O)cc2cccnc2s1 C(=O)(C1=CCN(C)C1)N(CCC(C)NC(=O)C(C)(C)C1CC1)C N1(C(C(COC)(C)OC)=O)CC2CCC(C1)C(NC(=O)CCCCCSC)C2 Cc1ccc(CNC(C2CCC(C)N2C(=O)CCn2cnc(=N)[nH]2)=O)c(O)c1 C(CCCCCNC(=O)CC1CCCO1)NC(CC1N(C(C)=O)CCC1)=O c1(CC)onc(C(=O)NCC(O)CCNC(C2CCC(CC)O2)=O)c1C C1(C(N2C(C)(C(=O)NCCC3C(C)C3)CCC2)=O)CC(=O)C12CCC2 Cc1cc(NC(=O)C(O)CCNC(c2cnc(O)c(C)c2)=O)c(O)c(C)c1 N1(C(=O)OCC)CC(C)N(Cc2coc(NCc3ccccc3)n2)CC1C c1(C(=O)NCC(C)N(C(CC(CC)OC)=O)C)csc2ncnc(O)c12 c1(C(=O)NCC2C(C(=O)NC(COCC)(C)C)CCO2)cn(C)nc1 C1(OC)CCN(C(c2cc(C(F)(F)F)cc(O)c2)=O)CC1(C)OC c1(C(=O)NCCOC2CN(C(c3cncs3)=O)C2)ccc(F)c2[nH]ccc12 C(=O)(C1CCCc2cncn21)NCC1CC(NC(c2c[nH]c(=O)cn2)=O)C1 c1(C(=O)NC(CCOC)CNC(=O)C(c2ccccc2)O)c[nH]c(=N)cc1C C12(NC(c3cc4sccc4[nH]3)=O)CCC(CC1)N(C(=O)C=CC1CCOCC1)C2 C1(C(N2CCCC(C(C)N)C2)=O)C2CCC1C(F)(F)C2 C(=O)(C(C(C)O)NC(=O)C(c1cncnc1)C)NCc1ccc(CC)o1 C1(C(N(CCCNC(C23CCCC2C3)=O)CC)=O)CC2CC(=O)C1O2 C(=O)CCC(=O)N1CC2CC2C1.C(CCC=CC(=O)N)=C(C)C.CC.N(C)C c1(CC(=O)NCC(CNC(CCOCC)=O)OC)csc(C2CC2)n1 c1(C(=O)NC(CCNC(C(C)CF)=O)(C)C)cc2cccnc2s1 C1(C(N2CC(O)C(O)C2)=O)CN(C(C2CC2c2ccccc2Cl)=O)CCN1 N1(C(C(CC)(C)C)=O)CCCN(C(=O)CN(C(=O)COC)C)CCC1 c1(NCc2nc(C)on2)ccccc1.N1(C)CCC(C=O)CC1.C(=O)C(C)(F)F CP(C)(=O)CCC(=O)NC1CCCC1NC(=O)C=Cc1cncs1 O=C(C1=CCN(C(=O)CC2CC3C=CC2C3)C1)N1CC2CCCC2C1 C1CCCCC1.C(c1ccccn1)=CC=O.C1(O)(CC#C)CC(C(=O)NC)C1 c1(C(=O)NC2(C)CCN(c3nnc(C)s3)C2)cc2c[nH]cnc-2n1 c1(CCC(=O)N2CCC2c2cccc3ncccc23)cnc2n1CCCCC2 c1(-c2cn(C3CN(C(CC4C(C)(C)CCO4)=O)C3)nn2)cc(Cl)ccc1Cl C(c1cc(F)c(O)c(F)c1)=CC(=O)N.N1(C(C=C2CCN(C)C2)=O)CCCCC1 CCCCCCC(C)C(=O)NCC1(OC)CCN(C(c2ccnnc2O)=O)C1 C1(c2nnn[nH]2)(Nc2cccc(OCC#N)c2)CCOC(C(N)=O)C1.C1CC1.C c1(C(=O)NC(C2CN(C(=O)CC3CCC(=O)N3)C2)C)ccc2ccoc2c1 n1(CC)nc(C(=O)NC(C(=O)NCCN2CCC2)C2CCC2)cc1O N1(C(C=C(CCC)C)=O)CCC(NC(=O)CC(=O)OCC)C(C)C1 C12(NC(C(CC(=O)OC)C)=O)CCOCC1CN(C(c1cncc(Cl)c1)=O)C2 C=CCCCCCCC(=O)NC(C1CCOC1)CNC(c1nnsc1C)=O Cc1nc(-c2nc(CC(C)(C)CO)nn2Cc2cncc(F)c2)c(C)s1 C1(O)(C(C)NC(=O)COC(F)(F)F)CCN(C(C2C=CC=CC=C2)=O)C1 N1(C(CC2(CSC)CC2)=O)CC(NC(=O)CCN2CCC2)CC1C C=CCC(F)(F)C(=O)N1CC(NC(=O)C2=CCCOC2)CC(O)C1 N1(C(COCC=C)=O)C2CCC1CC(n1cc(-c3ccc(C(=O)O)cn3)nn1)C2 c1(CC(=O)N(CCN(C(C(C2CC2)SC)=O)C)C)cncn1C1CC1 c1(C(=O)N)nc(O)nc(O)c1.C1(C)(NC(C2CN(C(CC)=O)C2)=O)CCC1 C1(C)(CC)CC(C(=O)N)CCO1.C1CN(C(=O)CCN(C)CCO)C(C)(C)C1 c1(C(=O)NC(CC=C)CNC(=O)CSC)cncc2sccc12 CCC(C)(C)C(O)C(=O)NCC1CN(C(c2cc(-c3cccs3)[nH]n2)=O)CC1O C1(NC(c2cc(C(N)=O)[nH]n2)=O)COCCC1NC(=O)CSC1CC1 C1(CCC)(C(=O)NC(C2CN(C(=O)CCC3CCCC3)C2)C)CC(=O)C1 Cc1nc(C)c(C(=O)NC2CCC(C(=O)NOCCF)CC2)s1 Cc1nc(-c2ccccc2)oc1C(=O)NC12CC(C1)C2.C(=O)CC1CC1.N Cc1cn2ccnc(C(N3CC(NC(=O)C=Cc4ccccc4)CC3C)=O)c2n1 C1(C(=O)NC(CN(C(CCCC)=O)C)C)Cc2ccccc2O1 N(C)(C1=NS(=O)(=O)c2ccccc21)CC=O.C(C=O)OC(C)=O.C1CC1.N Cc1ccc(C)c(C(=O)NC)c1C.N1(CC=O)CCN(C2CC2)C1=O.C1CC1 CC1(C(=O)NCCC2(O)CN(C(=O)CC3(C#N)CC3)C2)CC=CC1 N1(C(COCCCCC)=O)CCC2C(C1)NC(=O)CN2C(=O)C(C)P(C)(C)=O C1(CCN(C(c2cc(C)on2)=O)C)CCCCN1C(C1CCN(CC(C)C)C1)=O N1(C(C2CC3(CC(=O)C3)C2)=O)C2CCC1CN(C(=O)CCc1cncnc1O)C2 N1(C(c2c(NC)nc(C)cc2)=O)CCC2CCC(C1)N2C(=O)C(C)CS(C)(=O)=O c1(C(=O)NCC2COCCN(C(C(CC#C)C)=O)C2)cc(F)cc2cnccc12 c1(C(=O)N)c(F)c(C)cc(N)c1F.C(=O)CS(=O)(=O)C1CC1.C(C)(C)OC C1(N(C)C(c2cnc(Cl)s2)=O)CCN(C(c2cncc(C(N)=O)c2)=O)CC12CC2 N1(C(CCc2nc(C)sc2)=O)CC(NC(=O)CO)C2(CCC2)C1 c1(C(N2CC(CCCCNC(C3C(C)OCC3)=O)C2)=O)cc(O)ccc1OC(F)F N1(C(c2c(C)nco2)=O)CCC2(CNC(C3CC4CC4C3)=O)CCCCC12 c1(C(N2C(CC)COC(C)C2)C(=O)NCCCOC)cnc2ccc(C)cn12 C(=O)(C1=CCN(C(c2cccc(CC)n2)=O)CC1)NC(CCC(=C)C)C Cc1ccc(O)c(C(=O)NC2CC(CNC(c3c(C)ncnc3O)=O)CC2O)c1 C(=O)(C(C)CC(=O)OC)N(CC(N1CCC(OCC(N)=O)C1)=O)CCC Cc1nc2ccc(-c3nc(NC(=O)NCc4ccn5cnnc5c4)cs3)cc2[nH]1 c1(C(N2CC(CNC(C(C(C)C)N3CCCCC3)=O)C2)=O)ccc([N+](=O)[O-])n1C O(Nc1nc(NC(C2CCN(C(=O)NC(C)(C)C)O2)=O)cs1)c1cccc(C)c1 c1(CS(=O)(=O)NCCC(=O)NC(C)C)ccc(C(=O)O)cc1 N1(C(COCc2c(C)ncs2)=O)CCC(C)N(C(c2cocn2)=O)CC1 N1(C(C2CCC2)=O)CCC(C2CC2)C1.c1(C=O)cnc(C(C)(C)C)o1.CC.O c1(OC)ccccc1C(O)C(=O)NC(CNC(=O)CC12CC(C1)C2)CO C(=O)(CCCCCN=[N+]=[N-])NCCN(C(c1cccnc1OCCO)=O)CC N#CC1CN(Cc2cnnc(Cl)c2)CC1NC(C1(F)CCCC=C1F)=O C1(NC(c2cn(C)nc2)=O)CCC2CN(C(c3ccn(C4CC4)n3)=O)CC2C1 C(=O)(C1CCc2ccc(Cl)nc21)NCC(CNC(C)=O)O C(C)(C)(C(C)C)NC(CCCc1onc(CC)n1)=O.c1(C(=O)N)ccc(N)cn1 Cc1cc(N)c(C(=O)N(C2CN(C(=O)CC3CCCOC3)C2)C)cc1C C12(NC(CCc3ncc(C)[nH]3)=O)CCC(NC(C3CC=CCC3)=O)(CC1)C2 N1(C(C(C)SCC)=O)CC(C)(C)CCC1CNC(=O)Cc1cncnc1 N1(C(C(C(C)C)NC(N)=O)=O)CCCC(N=c2[nH]cnc3cnn(C)c23)C1 c1(C(=O)NCCc2c(OC)nccc2)cc(S(=O)(=O)N(C)C)ccc1Cl N1(CC(N2CC(F)(CNC(C34CCC(CC3)C4)=O)C2)=O)CCCCCC1=O n1(CC)nnc(C(N2CC3CC2C3NC(=O)COC2(C)CCCC2)=O)c1C Cc1cc(N2CC3CCC(C2)C3O)ncc1S(=O)(=O)NCC1CCNC(=O)C1 N1(c2c(C(=O)OC)c(Cl)ncn2)CC(NC(=O)CC2CCSCC2)CC2(CC2)C1 C(=O)(C1=CC2(CN(C(c3cnc(S)nc3)=O)C2)OC1)NC(C1CC1(C)C)C c1(C(=O)NC2CCC(N(C(=O)C(N)=O)C)C2)ccc(Br)cc1O N#CC1CCC(C(=O)NCc2cn(CC(=O)NCC=CCl)nn2)CC1 C1(CNC(=O)CC2OCCO2)CCCCC1NC(=O)CCCc1cccc(Cl)c1 c1(CNC(c2nc(OCC)oc2)=O)ccccc1.C1(C=O)COCC(C)O1.C CCCCCC(O)CC(=O)NCC1=CCN(C(c2ccc(Cl)cc2C)=O)CC1 c1(CC(=O)NCC2(NC(c3c(C)ncs3)=O)CCCC2)oc2ccccc2c1C N1(C(c2c(C)nsc2C)=O)CCC2CC1CN(C(=O)COCC1CCCCO1)C2 N1(C(CCCOCC=C)=O)CC2CCC1C2.C1(C(=O)N)CCC(=O)N(C2CC2)C1 c1(C(CC)OC)cn(CCNC(c2ocnc2C(C)C)=O)nn1 N1(C(CCSCCC)=O)CCC2CC2(C(=O)Nn2cnnc2C(=O)OC)CC1 C12(CCCC(C=C)C1)c1nnnn1Cc1ccc(cc1)N2.C1(CC=C)CCOCC1 CCC(CC)C(F)C(=O)NCCCCC(=O)NC(C)(CSC)CO C(C1(C)CCCc2ccccc21)(c1n(CC)nnn1)NCC(C)(C)c1ccsc1 C1(C)(CNC(CC=CC)=O)CC(OC)CN1C(=O)CSS(C)(=O)=O CC(C)CC(CO)CN=c1[nH]c(=NCc2nnc(O)n2C(C)C)[nH]c2c1SCC2 CC1CCCC1.N1(C(COC)=O)CCC(C(F)F)C1.C1(C=O)(C(N)=O)CC1 N1(C(C2C(C(C)C)C2)=O)CC23CCCCC2(C1)CN(C(C1(C)COC1)=O)C3 CC1(C)CC1(C#N)C(=O)NCc1ccc(C(=O)NCCCc2ccncc2)o1 c1(OC(c2cnn(CC)c2C(F)(F)F)=O)cccc2c1CCCC2 CCCC(C)(C)CC(=O)NC1CC(C(=O)N2CCN(CC)C(=O)C2)=CC1O C1(N(C(=O)CSC)CC)CCCN(C(=O)CSCC(N)=O)CC1 Cc1nsc(N)c1C(=O)NC(CNC(=O)CC(C)Cc1ccc(Cl)cc1)CO c1(C(=O)NC(CC)CNC(=O)C(F)=CC2CC2)sc2cccc(F)c2c1Cl C(=O)(C1CCCn2cnnc21)NCC(C1CCCC1)NC(C(CCC)O)=O CCCCC(C)C(=O)N(CCCC(=O)NCc1cn(CCC)nn1)C C1(CC)CN(CC)CCN1C(C1(C)CN(C(c2c[nH]c(=N)o2)=O)C1)=O c1(CC)ncc(C(=O)NCCCCCN(C)C(c2cccc(Cl)c2Cl)=O)c(C)n1 c1(C(=O)NCC2N(C(C3N(CCCC)CCCC3)=O)CCC2)cc(C)ccc1C c1(C(=O)OC)cccc(-c2cn(CC3(C)CC4(CC4)C3)nn2)c1F c1(NC(c2ccccc2)c2nnnn2C2CCOC2)ccc(SCC2CC2)cc1 n1(CCC(=O)NC(CN(C(C2CC(C#C)(O)C2)=O)CC)C)ccc(O)nc1=O C1(C(CNC(c2ccc(C)[nH]2)=O)(C)C)CCN(C(C2(C)CCNC2=O)=O)CC1 c1(CC(=O)N(CCCCNC(C2CC(C)OCC2)=O)C)nc([N+](=O)[O-])n[nH]1 C1CN(C)CCN1C(=O)C(F)CC1CCC1.C(=O)(CCC(=O)N)N(C(C)C)C.C c1(C(N2CC(O)(C(C)NC(=O)CSc3ccccc3)C2)=O)cc(Br)cn1C N1(C(CC(=C)C)=O)CCCCC1C1CCCN(C(c2cc(CCC)n(C)n2)=O)C1 CC(C)CC(C(=O)N1CCCC1C(C)(C)NC(c1cn(C)nc1Cl)=O)N(C)C CC1CCC(CNC(C2CCN(Cc3cncn3C)C2)=O)O1 O(NC(=O)C(F)(CNC(c1ccc(O)cn1)=O)C(C)C)CCC(C)C C(=O)(CC(O)CCC)NCC(CC=C)NC(c1cccc(OC(C)C)n1)=O C1(C)(CNC(c2c(CC)[nH]cc2)=O)CCC(NC(c2cccs2)=O)CC1 Cc1nnc2n1CCCC2Nc1nc(N(CCCCC(C)C)C)c2c(n1)COC2 Cc1nc2n(c1CC(=O)NC1CC(C)CN(C(=O)C(=O)N)C1)CCCC2.C1CC1 N1(C(c2ccc(CNC(CC(C)(F)F)=O)o2)=O)CC2CCCCC2C1 c1(NC(N2CC([N+](=O)[O-])C2)=O)ccc2c(ccn2Cc2ccccc2)c1 Cc1ccc(Cl)c(Cc2noc(CC3COC(=O)C3)n2)c1 c1(C(=O)NC(CC)CNC(=O)CC(C(C)C)C(C)C)nn(C)cc1S(C)(=O)=O c1(CNC(=O)CN(C(C2CCOCC2)=O)C2CC2)n[nH]c2c1CCC2 C1(F)(C(N(C(CC)CC)CCO)=O)CCN(C(=O)CC2CCC(C)O2)CC1 C1(c2cn(Cc3cocn3)nn2)(C(=O)Nc2n(C(C)C)ccc2)CCCOC1 Cc1nc2n(n1)CCN(C(=O)CC1CCCN1C(=O)CC1CC(N(C)C)C1)C2 N1(C(C(C)C(F)(F)F)=O)CCCC(F)(CNC(c2ncnc3cc[nH]c23)=O)CC1 C12CCCC1CCN2C(c1coc(C)c1)=O.c1(OC)ccc(C(=O)NC)c(N)c1 N1(C(CC(CC)C2CCC2)=O)CC2(CO)CC1(CF)C2 C(C)(CCC(=O)N1CCC(C(=O)NOC(c2ccccc2)C)C1C(C)C)OCC Cc1c(O)nc2ccccc2c1C(=O)NCCCNC(=O)Cn1cc(C#N)cn1 N1(C(c2cc(OC)no2)=O)CC2COCCC2(NC(=O)Cc2ccsc2)C1 CC(C)(C)CC(C(=O)N1CCC(CCCO)CC1)NC(C1CC(F)C(=O)N1)=O c1(C(N2C3(C(=O)NCC(COC)(C)CO)CC3CC2)=O)c[nH]c2cnccc12 Cc1nc[nH]c1CC(=O)NCC(O)CNC(=O)CCCF c1(OC)cccc(-c2cn(C(C)CNC(=O)C(C3CCC3)C3CCC3)nn2)c1Cl c1(C(C)C)ccc(N)c(C(=O)N(CC(C)NC(=O)CN2CCCCCC2=O)C)c1 CC1=C(C(=O)NCC2CCN(C(=O)CC3CCSC3)C23CCC3)SCCO1 N1(C(C(CC#C)C)=O)C2CCCC1CC(NC(c1c(OC)noc1C1CC1)=O)C2 C1(CNC(C(=O)NC2C(CC(=O)OC)CCC2)=O)CCC2(CCNCC2)O1 C(=O)(C1Cc2ccccc21)NC(c1c(C)ccnc1)C.C12CC(C1)NC(=O)C2 C(=O)(CC(O)CC(C)(C)C)NC1C(NC(C2(C)CCC(C)CC2)=O)CCC1 c1(OCC)ccc(C(=O)NC2CN(C(=O)CCCC3CC3)CCC2F)cc1C C1(CNC(C(=O)NCC)=O)C(C2CC2)CCN1C(=O)Cc1cnccc1C Cn1nncc1C(N1CCC(N2CC=CC2)C1)C(=O)NC1CC1 N1(C(c2cnc(C)n2C)=O)CC(NC(c2cnc(C(F)(F)F)cn2)=O)C2(CC2)C1 c1(C(N2C3CCC(CCNC(c4[nH]cc(C)c4)=O)(C3)C2)=O)c(Cl)ccc(C)c1O N1(C(C(C)SC)=O)CCC(NC(=O)COC(F)F)C(F)(F)CC1 c1(C(c2nnnn2CCCOC2CC2)NCC(C2CCC2)OC)cncnc1 C1(S(C)(=O)=O)(C=O)CCCCC1.CCCCCC(=O)NCC1CC(F)(C)C1.N C12(NC(CC(=C=C)C)=O)CCOC(CNC(=O)CCN(C)CCO)(C1)C2 c1(CC(=O)NCCC(C)NC(=O)C(C)C2CCCC2)ccc(F)c(Cl)c1 S(=O)(=O)(c1ccc(C(=O)NC2CCCCCN(C(=O)CC(C)O)C2)cn1)NC N1(C(c2c(C)onc2)=O)CC2CC(NC(=O)Cc3cccc(Cl)c3Cl)C(C2)C1 CCC(CC(=O)N1CCC(CNC(c2cc(Cl)c[nH]2)=O)C1(C)C)CC(F)(F)F CC1(C)CN(C(=O)CCOC2COC2)C(C)CO1.C(=O)(C(C)(C)C(N)=O)N CS(=O)(=O)C1CN(C(c2ccoc2)=O)CC1NC(=O)C1CC1.C(=O)(C)N CC1(C(=O)NCCCCCn2cc(-c3cscn3)nn2)CCC(=O)C1 N1(C(c2cc(C(CC)CC)no2)=O)c2cc(C(=O)OC)ccc2CC1C C(C1c2ccsc2CCN1C(=O)CC1CSC1)NC(Cc1c(C)noc1Cl)=O CC(c1cccc(Cl)c1)=CC(=O)NC(C)C(CO)NC(=O)CCc1ncccn1 c1(CNC(=NCCc2onc(C)n2)NC(C)C2CC2)cnn2ccn(C)c(=O)c12 c1(C(=O)NC2C(C)CN(c3nnc(C#N)s3)C2)cccc(F)c1Cl N1(C(=O)CCCCCF)CCCC(C2CCN(C(c3cccnc3S)=O)C2)C1 CC(C)(CCCNC(=O)C(CO)C(F)(F)F)C(=O)N1CC(C)(CO)C1 CCC(C(=O)NCC1(CC(C)C)CC1)OC C1(C(N2CC(OCC)C2)=O)CCN(C(c2sc(O)nc2C)=O)C1C c1(CC(=O)NCC(CNC(=O)CC2CCCC23CC3)CO)ccccc1F C1(C(=O)NC2CC(NC(c3c[nH]c(=NC)s3)=O)C2)CCc2ncnn2C1 C1(CCC)(NC(=O)CO)CCCN(C(C2CCC(C)O2)=O)C1.c1ccc(Cl)cc1 N1(C(c2cc(C)sc2)=O)CCCC2C1CCCN2C(c1nccc(C(F)F)n1)=O C(C)(C(C)COC)(c1n(C(CC)(C)C)nnn1)NCCC(=O)NCC(=O)NC C(=O)(C1=NOC(C(=O)N(CC(C)CNC(=O)Cc2ccccc2)C)C1)OC N1(C(c2cc(C(=O)OC)oc2C)=O)CCN(C(=O)CS)C2CC12.C1CCCC1 C(N=c1ncc(C(F)F)c[nH]1)C1C(NC(=O)CCCCc2cnn[nH]2)CCC1 C1(CC(=O)NC2CN(C(C(C)OCC#C)=O)C2)CCCC(C)(C)C1 c1(-c2cn(CCCC)nn2)nnc2n1CCN(C(=O)C(O)c1ccsc1)C2 Cc1cc(CNC(=O)C=Cc2cn[nH]c2)oc1C(=O)N(CC(C)O)CCF CC12CCC(C(=O)NCC(O)C)(CO1)C2.C(=O)(C(F)(F)c1csc(=N)[nH]1)N CC(C)C(CN(C)CCN(C)C(=O)OC(C)(C)C)NC(C1CCCO1)=O C1(OCC)CC(NC(=O)C(=O)NC(c2cn(C)nn2)C)C12CCCCC2 C1(C(=O)NCC(CC)n2cccn2)CC2CCC1N2C(=O)Cn1cccn1 c1(C(N2CC3C(NC(c4ccc(Cl)o4)=O)CC(C3)C2)=O)c[nH]c2ccc(Cl)cc12 C1(N(C(COCC(=O)OC)=O)C)C2CN(C(C3CC=C(C)CC3)=O)CC12 C1(N(C)C(C2CC3C=CC2O3)=O)CCCN(C(=O)C=Cc2cc[nH]c2)CC1 C1(c2scc(CC)n2)COCCN1C(c1ccsc1Cl)C(=O)NCC1CCOC1 c1(C(=O)NCCc2ccsc2)ccc2c(c1)CCN(S(=O)(=O)CC1CC1)C2 CC(C)(CNC(c1coc(CNC(c2ncc(F)cn2)=O)c1)=O)CCCO c1(CC)cc(C(=O)NC2CCN(C(=O)C(n3cc(C)cn3)C)C2)nn1C Cc1nn2c(C)cccc2c1C(N1CCCCC(NC(=O)CC2CC=CC2)C1)=O C(=O)(C1=CCC(F)(F)CC1)N1C(C)CC(NC(c2ccc(F)c(C)c2N)=O)C1 CC1(C)C(NCc2csc(-c3ccccc3)n2)CCC1O C(=O)(C(C)C(C)NC(=O)CCC1(C)CCCN1C(c1nccnc1N)=O)OC CC(CCNC(=O)NCC(C1(O)CCOC1)(C)C)S(C)(=O)=O CC(c1ccc(F)cc1F)=CC(=O)NCCC(O)CNC(=O)CCc1cnc[nH]1 C(CCCCCC(=O)NC(C)CCCNC(c1ccno1)=O)SC C=CCCCCCCCCC(=O)NC1(C2CCCN(c3ncc(Br)cn3)C2)CC1 N1(C(CC(CNC(c2c(CC)ncnc2)=O)(C)C)=O)CCC(C)(C#N)CC1 CCCCCC(CC)C(=O)NCC1(F)CC(CNC(=O)C(F)C(C)(F)F)C1 C12(NC(c3c(C)csc3)=O)CC1CN(C(c1cnc(C3CCC3)s1)=O)C2 C1(C(=O)NCC(CC)(O)CC)C2CCC(C2)N1C(C1CC2(C1)CC21CC1)=O C1(C(=O)NC(C)CCN(C)C)CCC(C)(C)N(C(C2(C#N)CC(=O)C2)=O)C1 C1(F)(C(NOCCCC(=O)OC)=O)CCCN(C(=O)C(C)(C)N2CCCC2)C1 C1(C(=O)NC(C2CCCCN2C(=O)CCN2CCC2)C)(CC)CC(C)(C)C1 c1(CC)ccc(F)c(C(=O)NC(C2CCCN2C(C2CNC(=O)N2)=O)C)c1 CCCC(C)CC(=O)N(CCC(=O)NCCN1CC(CF)C1)C C=CCCCCCC(=O)NCC1CN(C(c2cccn(C)c2=O)=O)CC(C)(C)O1 N1(C(CS(C)(=O)=O)=O)Cc2ccnn2CC(NC(c2cc3cccnn3n2)=O)C1 N1(C(C(CC)C#N)=O)CC2(CCC2)CC1CNC(c1cccc(O)n1)=O CC(C)CC(C)(O)c1cn(C2CC3(C(=O)NCCc4cnn(C)c4)CC23)nn1 C1(NC(C(c2ccccc2Cl)C)=O)CCC(NC(c2cnc(Cl)[nH]2)=O)CC1 CC(F)(F)CC(=O)N1CCC(c2n[nH]cc2CNC(c2ccnnc2O)=O)C1 O=S(=O)(c1ccc(C(F)F)c(Br)c1)N1CCCC1c1cc(C2CC2)on1 C1(NC(=O)Cc2ccc(Cl)s2)CCC2(C1)CN(C(c1ccnc(Cl)c1)=O)C2 CC1CCC(C(N)=O)CN1C(C1CCOCC1NC(c1cncs1)=O)=O CCC(C(=O)NCC(c1ccccc1)(C)OC)N(C)C CC(C)CCCC(=O)NCC1COCCN1C(c1cnn(C)c1)=O C1(C(=O)NC2C(NC(C(C)(C)SC)=O)C2)CCN(C(=O)N(C)C)CC1 c1(OC)cc(C(=O)NCc2ccc(C(=O)NC3CCCC(C)C3)cc2)ccn1 C1(C(N(C(C)C)CC)=O)(OC)CCN(C(c2cnn(C)c2N)=O)CC1 c1(OC)ccc(C(=O)N(CCN(C)Cc2sc(C)nc2C)C(C)C)cc1O Cc1ccc(C(N2CC3CC2CCC3NC(C2CC23CC3)=O)=O)c(F)c1Cl c1(C(=O)NC(C)CCCCNC(c2ccc(Cl)s2)=O)ccc2nn[nH]c2n1 c1(CN2C(C(=O)NCC(CC)Oc3cccc(C)c3)CCC2)ccc(Cl)c(F)c1 C(=O)(CCC(N)=O)NCC(C)CNC(C1CC(=O)N(O)C1)=O N1(C(CCC2CCC(C)O2)=O)CC=C(C(=O)NCC(C)(F)C(C)(C)F)CC1 Nc1c(Cl)ccc(F)c1C(=O)NC.C1CN(C(C2C=CCCC2)=O)C2(CCC2)C1 c1(CCC(=O)NCC(CCC)NC(=O)C(C)CCOC)cccc(C)c1 C(C(F)(F)C(=O)NC1CN(C(=O)Cc2ccccc2Br)C1)N(C)C C1(NC(c2c(OC)oc(C)n2)=O)CCCCCN(C(=O)COC(C)C)C1 N1(C(C2CCc3nccn3C2)=O)CCCC2(C1)CN(C(C1(O)CCOC1)=O)C2 C1(F)(C(=O)OCC)CN(C(=O)C(N2CCN(CCOC)CC2C)=O)CC12CCC2 N1(C(COCC)=O)CCC(NC(C2(CC)CC2)=O)C1c1cccc(Br)c1 C(=O)(C(CC)(CC)O)NCC(C)N(C(c1cc(C2CCOC2)[nH]n1)=O)CC N1(C(CSSC)=O)CCCC2(C1)CN(C(C1(C)CC(C#N)C1)=O)CCO2 CN1C2CCCC1CN(C(c1ccc(CNC(=O)CC3CC3)cc1)=O)C2 C(=O)(C1=CCCSC1)NCC(N(C(C12CC(OC)C1C2)=O)C)C1CC1 C1(NC(C(C)CC2CC2)=O)CCSC12CN(C(=O)Cn1cc(C3CC3)nn1)C2 C1(CC=C)(NC(=O)CC2C(=O)NN=C2C)CCCN(C(c2nonc2N)=O)C1 c1(C(=O)NC2C(C)CN(C(=O)C(F)(F)CO)C2)cc(N)cc(O)c1 C12(NC(=O)C=C(Cl)Cl)CCCN(C(C3(CCN4CCCCC4)CC3)=O)CC1C2 C(c1cccc2ccccc12)=CC=O.C(C)(C(=O)NCC(O)C)OCCC=C.N C=C1CCN(C(=O)Cc2ccc(C#N)cc2)C(C(=O)NCC(F)Cl)C1 C1(COC(c2ccn(C3CC3)n2)=O)CC12CCOC2 c1(C(N2C3CCN(C(c4occc4Br)=O)CC3C2)=O)cccc2nccnc12 CC(C)(C)C(CC(=O)NCCC1CCCCO1)NC(=O)CCC1(C)CC1(F)F N1(C(CC2N(C(c3c(C)c(=O)cc[nH]3)=O)C3C2CCC3)=O)CCN(C)C(C)C1C C=C(Br)CCCNC(CCC=C(C)C)c1nnnn1C1CCCCC1 c1(NC(C2(C)CCCN2Cc2cncc(F)c2)=O)nccc(Cl)c1Cl CCC(C)CCCCC(=O)N1C(C(=O)NC(c2cn[nH]c2)C)CCC12CC2 C1(NC(C(CC)CC)=O)C(C)CN(C(c2cnoc2-c2ccc(C)o2)=O)CC1C Cc1csc2cc(C(=O)NCC(C)CN(C(=O)CCOc3cccnc3)C)[nH]c12 N1(C(CCOCC)=O)CCC(C2CC2NC(=O)C(C)CSC)CC1 C1(OC)CC(NC(=O)CCc2ccc(F)cc2)CN(C(=O)C(F)n2ccnc2)C1 Cc1cc(C)n(CCCC(=O)N(C)CC2CCN(C(C3CCC3CF)=O)C2)n1 c1(C(N(C2CCN(C(C3(C)CCC3)=O)C2)C)=O)cc(C2CC2)oc1C1CC1 c1(CNc2c(C(=O)NC3C=CC(CC)C3)n(C)nc2)c(OC)cccc1F N1(C(C(C(CC)C)N(C(=O)Cc2cccnc2O)C)=O)CCC2(CC1)CN(C)C2 Cc1nc(=N)[nH]cc1C(=O)NCCN(C(=O)CN1CCC1C)C(C)C N1(C(Cc2ccn(C)n2)=O)CC(=O)NCC1c1ccccc1 C1(NC(C2(OCC)CCOC2)=O)CCN(C(=O)CC(C)(C)C2CCCCC2)C1C CCCCCC(O)Cc1nc(C2CSC2)nn1CC1CCSC1 Cc1c(-n2nc(Cc3cccc(Cl)c3)nc2CCCc2cscn2)cccc1Cl Oc1ccc2nc(Cc3nc(-c4cncn4C(F)F)no3)oc2c1 Cc1ccc2c(O)c(C(N3CC4(NC(c5nccn5C)=O)CC3C4)=O)cnc2n1 c1(CC)noc(C)c1C(N1CC(COC)C(C)C1)C(=O)Nc1ccccc1.O CC1(C)CCC(C(=O)NC2CCCC2NC(c2cc3n(n2)CCC3)=O)CO1 N#Cc1ccncc1C(=O)NC(C(N1CCC(CO)C(O)C1)=O)C1CCCO1 Cc1ccc2c(c1)CC(C(=O)Nc1ccccc1OCC(N)=O)O2 c1(C(=O)NCC2CC2NC(C2C3COCC23)=O)cccc(N2CCCC2)n1 c1(C(N2CCC(N(C)C)(CC)C2)C(=O)NC2CCCC2)cc2ncccc2s1 N1(C(Cn2cnc(=N)[nH]2)=O)CCCC(C2CC2NC(c2nc(F)ccc2Cl)=O)C1 C1(C(=O)NC)CCN(C(=O)CCC2CCC2)C1C.c1(CC(=O)N)n[nH]c(C)n1 C(=O)(CC(F)(F)C(F)(F)F)N1CC(CC(C)(O)CN)C1 Cc1cc(C(=O)NC(CCN(C)C(C2(F)CC=CCC2)=O)c2cccs2)nn1C CC1(C)CCC(CNC(C2C=CCN2C(c2ns[nH]c2=O)=O)=O)O1 C1(O)(CC)CCN(C(c2ccc(C(N)=O)s2)=O)CC1.N=c1[nH]c(CC(=O)N)cs1 CC1CCn2ncc(C(N3CCC(CNC(C4CCCNC4=O)=O)CC3)=O)c2C1 C1(CNC(c2nc(C)sc2)=O)CC2CCC(C1)N2C(C1OCC2COCCC12)=O CCCC(C)(C)C(=O)N1CC(CNS(=O)(=O)C(F)(F)F)C(F)(F)C1 C1(CNC(CC2C(C)C2)=O)CCCCN1C(=O)CCS.C1CCS(=O)(=O)C1 CC(c1ccccc1F)=CC(=O)NCC1CCCC(NC(=O)Cc2cnns2)C1 CC(C)C(O)C(=O)NC(c1ccccc1)C(=O)NCCC1CCCOC1 C(=O)(C1CCCc2ccccc21)NCCCN(C(=O)C(C)(C)C1CCOC1)C c1(CC)nc(=NCC2CCCCN(C(=O)CCc3cncn3C)C2)s[nH]1 c1(OC)cccc2c1C(C(=O)NCC=CCNC(=O)C1=CCCSC1)CC2=O CCCCC(C(=O)NCC(C)CC(=O)NC(C)(C)CC1CCC1)N(C)C C1(NC(COCCCCOCC#C)=O)CN(C(c2cccnc2Cl)=O)CC1(C)C C(=O)(CCCCCCCS(C)(=O)=O)NC1CCN(C(c2nc(CC)oc2C)=O)C1 C(=O)(C(=O)N=S(C)(C)=O)NC(C(C)C)C(C)NC(c1occc1Br)=O C1(C)(C(N2CC(CNC(CC(=C=C)C)=O)C(C)(C)C2)=O)CC(C(C)C)=NO1 Cc1ncc(C(=O)NC2CCCCC2c2ccc(Cl)cc2)cn1 S(=O)(=O)(c1ccc(C)cc1C)NCCC(=O)NCC(COCC)O c1(C(N2CCC(NC(C3(CCCC)CC3)=O)C(F)C2)=O)cncc2ccsc12 C1(CC)CCCC1C(N1CC(C)(CCC(=O)NC2CC3(CC3)C2)C1)=O c1(CC)cccc(OC)c1NC(=O)NCC(c1ccc(C(F)(F)F)cc1)C c1(NC(C2CCS(=O)(=O)CC2)C)cccc(P(C)(C)=O)c1 c1(CC)cccc(C(N2CCC(CN(C(=O)C(C(C)O)N(C)C)C)C2)=O)c1N N1(C(C(COCC)N=[N+]=[N-])=O)CCC(C)N(C(=O)CSc2n[nH]c(O)n2)CC1 C(=O)(CCC(C)NC(=O)NC1(c2ncco2)CC1)OCC c1(C(=O)NC2CN(C(C3C(CC)C3)=O)CC2SC)c(Br)ccc2n[nH]cc12 C1(CC)(CNC(=O)CCn2cc(CCS(=O)(=O)N(C)C)nn2)CCCCO1 C(C(=O)NN1CCCC1C(N1CCC1(CO)CO)=O)=C(CC)CC C=CCCCC(=O)N(CC(C)(C)CNC(=O)C(=O)NCc1ccc(F)cc1)C c1(CC)cc(C)ccc1C(=O)NC1CC(NC(=O)CCF)CC1O N1(C(c2c(C)nc(CC(C)C)s2)=O)CCN(C(C2(C)CC2Br)=O)CC1C c1(NC)ccc(F)cc1C(N1CCC(C)C1CNC(=O)CN=S(C)(C)=O)=O C(C)(C)(C(=O)N(CC(O)CN(C)C(c1ccn(C2CC2)n1)=O)C)OCC Cc1csc2c(C(=O)NCC(CO)NC(c3ccc4c[nH]nc4c3)=O)ncnc12 C1(CC(=O)NCCCCCCNC(C=CC(CC)C)=O)CC2(CCCC2)CO1 C1(NC(c2cccc(O)c2F)=O)CC2(CCN(C(=O)C)C2)C1.C1CC(F)(F)C1 N1(C(=O)CCc2nc[nH]n2)CC2CN(C(c3sccc3F)=O)CCC2(CO)C1 Cc1ncc(C(N2CCN(C(c3cccc4ncnn34)=O)C(C)C2)=O)cc1C#N c1(C(=O)NCc2cc(C(N(C(CC(CC)C)C)C)=O)n[nH]2)n[nH]c2c1COC2 C1(C(NOCC#C)=O)CCN(C(c2cc(Cl)ns2)=O)C1(C)C c1(C(C)=O)cc(C(=O)NC2CCCC2NC(=O)Cc2ccc(O)nc2)ccc1O C1(C(=O)NCC2C(C(=O)NCc3cc(C)on3)C2)COCCN1C S(=O)(=O)(c1ccc2ccccc2c1)N1CC(C(N2CCN(CC#C)CC2)=O)C1 C(=O)(C(C)(CC)CC)N(CCOCCC(=O)NC(CCC)C(=O)N(C)C)C CCC1=NOC(C(=O)N(C)CC2CCN(C(c3cnc(Cl)s3)=O)C2)C1 C1(C(N2CC(NC(C34CC(C3)C(C(F)(F)F)O4)=O)C2)=O)C2CCCCCC12 C1(C(=O)NCC(C)CN(C)C(C2(C)CCC(=O)C2)=O)CCc2nncn2C1 C1(F)(CNC(C(C)=C2CC2)=O)CC(NC(=O)C(c2ccc(Br)s2)=O)C1 CC(C)C(C(=O)N1CCC(C)(CNC(=O)CC(C)(O)C2CC2)C1)N(C)C c1(C(=O)NC2C(NC(=O)Cn3cccn3)CCC2)ccc(NC=O)cc1F.C c1(C(=O)NC(C(C)NC(=O)CSC(F)F)C)cnoc1-c1ccc(Cl)s1 C1(NC(CSCC#C)=O)CCN(C(=O)Cc2nc(C)c(C)s2)CC1C c1(CCCCC)cn(CC2CCCC2NC(=O)C(C)(F)F)nn1 c1(CC)c(C(=O)NC2CCCC(C)C2)cccc1C.c1(CC=O)cc(C)on1.N Cc1cc(C(=O)NCCC2CC2)nc(O)n1.C1(CCCC=O)CCCC(=O)N1.N c1(C2(C(N(CCCCCn3cc(C(C)N(C)C)nn3)C)=O)CCOC2)ccccc1 c1(C(=O)N)cc(O)cc(Cl)c1Cl.C1(OC)CC(C)N(C(c2onc(C)c2C)=O)C1 CCC1=C(C(=O)N2CCC(CNC(=O)CN3CC=CC3)C(O)C2)SCCO1 c1(CC)cc(CC)nc(N2CCCC2CNC(=O)CC2(COC)CC2)n1 C1(CNC(c2n(CCCOC)nnn2)c2cnco2)(OCCO)CCCOC1 C(=O)(C1=C(F)CN(C(C2CNC(=O)O2)=O)CC1)N(C1CCCC(O)C1)C Cc1ncc(C(=O)NCCc2cc(C(N3CCC(O)C(F)C3)=O)no2)c(=N)[nH]1 C12(CNC(C(C)NC(C(C3CC3)OC)=O)=O)CCN(CC1)C2 C(=O)(C(N=[N+]=[N-])C(C)C)N1CCCC(C)C1.c1(OCC)cccnc1C(=O)NC CCCC(CCO)NC(=O)CCOCCN(C(=O)CC1CCCC(C)O1)C Cc1noc2cc(C(=O)N(C(C)CNC(=O)C(C)(C)C(C)O)C)ccc12 N1(C(C2CCC(=O)C2)=O)CC2CC(NC(c3ccsc3C(F)F)=O)CC(C2)C1 C1(NC(C(C)c2ccco2)=O)CC2CCCC(C1)N2C(=O)C#CC1CC1 C(=O)(C(O)CCNC(=O)CN(C)C(=O)C1CC1)N(CC(C)(C)CO)C c1(C(N2CCC(C(=O)OC)CC2)C(=O)NCCC)ccc(CC(C)C)cc1 CCCCCC(F)C(=O)N(C)CCOCCNC(C1(C)CC(O)CN1C)=O C#Cc1cccc(C(=O)NC23CCN(C(c4occc4C(C)C)=O)CC2C3)c1C c1(CCC(=O)NC2CCC(CCNC(c3ccns3)=O)C2)cnc(O)[nH]1 Cc1cc(CNC(C2CN(C(C3CC(F)C3)=O)CC(C)O2)=O)cc(C)n1 c1(CC)cnsc1C(=O)NC(C(=O)N(CCN(C)C)CC)c1cccs1 c1(C(=O)NCC2CCCCN2C(C2(Br)CC2)=O)cnc(O)c(F)c1 C(=O)(C1=CCCCCC1)N1CCN(CC2CN(C(c3c(CC)scn3)=O)C2)CC1 c1(C(=O)NCC(CC=C)NC(=O)CCC(C)SC)cc2c(cc1F)NCCC2 N1(C(C=C(C)C(F)F)=O)CCCCCC(NC(c2coc(C)c2)=O)C1 C1(CNC(C=CC(=O)OCC)=O)CCCCN1C(C1OCCC1C)=O.C c1(C(=O)Nc2cccc(-c3c(OCC(=C)C)cccc3)n2)cc(C)cc(C#N)c1 C1(CC(=O)NCCCN(C)C(C2(C#N)CC2(C)C)=O)CCCNC(=O)C1 Cc1c(F)ccc(C(N2CCN(C(c3ccnnc3)=O)C(C(C)C)C2)=O)c1C#N C1(C2CCC2)(C(=O)NCC(CC)NC(=O)CCc2cc(Cl)cs2)CC1(F)F Cc1nc(O)nc(C)c1C(N1CCC(C(C)NC(=O)C#CC(C)(C)C)C1)=O C1(C)(CC(=O)N(C2CCN(CC34CCCC3C4)CC2)CCC)CC(F)(F)C1 c1(C(=O)NC(C)CNC(C2(C)CC2(F)F)=O)cnn2cnnc2c1 Cc1cc(C#N)ccc1C(N1CC2CCC(C1)C2NCc1cc(O)ccc1O)=O N1(C(C(CCC)O)=O)CCCC(C)(CNC(=O)CCC(C)Sc2ccccc2)C1 c1(OC)cccc2ncnc(NC3CC(C)N(C(C4CCCC(C)(C)C4)=O)C3)c12 CC(C)CC(C)(O)C(=O)N1CC(n2cc(CCCO)nn2)C(C)C1 c1(OC)ccc(C(=O)NC)c(F)c1Cl.C1CCCCN1C(c1cc(C)c(C)[nH]1)=O c1(CC=C)ccc(OC(c2ccnn2C2CCS(=O)(=O)C2)=O)c(OC)c1 C1(C(=O)NCC(C#C)(C)C)CN(C(=O)CCCN2CCCC2)CCN1C C1(C(N2C3CC(CC(NC(CC(CC)O)=O)C3)C2)=O)CCc2n[nH]cc2C1C N1(C(C(C)CN2CCOCC2)=O)CCC2(CC(NC(c3scnc3Cl)=O)C2)C1 c1(CC(=O)OC)ccccc1CN=C(NCc1ncnn1C)NCc1cccs1 c1(C(=O)NC(C(C)NC(C(C)=C2CCC2)=O)C)c(Cl)nsc1Cl c1(C(N(C(C)C(=O)NC2CN(C(=O)C3CC3)C2)CC)=O)[nH]cc(C)c1C c1(C(=O)NCC2C(NC(CCC(C)OC)=O)CCC2)ccc(F)c(C#N)c1 C1(CNCc2nc(C(=O)O)on2)CCCN(C(=O)Cc2cnc[nH]2)C1 C(=O)(CC(C)(C)CN(C)C)NC(CCCC)CNC(C1(SC)CCOCC1)=O CC1CCc2c(sc3nc(C(C)NCCc4ccc(C#N)cc4)nc(O)c23)C1 N1(CC(c2ccccc2)(C)C)C(=O)CCN(Cc2cccc(C(F)F)c2)C1=O C12(NC(C(CC)SC)=O)CC(CO)(C1)OC21CN(C(c2cccc(N)c2C)=O)C1 c1(C(N2CCC3C(NC(c4ccc(C#C)cn4)=O)C32)=O)cc(N)c(O)c(F)c1 C(CCN(C)C)(C(=O)N1CCC(F)(COC)C1)NC(CCSCC)=O Cc1cccn2c(C(=O)NCC(c3cc(Cl)cc(Br)c3)O)nnc12 c1(C(=O)NCC(C2(O)CCN(C(c3ccnnc3)=O)C2)C)cc(C(F)F)ccn1 c1(C(=O)NC2CN(C(c3c(C)cnc(F)c3)=O)CC2C)nc2cnccc2s1 c1(C(N2CCC(CC(=O)NC3C(C)(C)C3)CC2)=O)c[nH]c2cccnc12 C1(NC(C(C)=C2CC2)=O)CN(C(=O)CSC2CC2)CC1n1ccnn1 c1(C(=O)NCCNC(c2cc(N(C)C)ncc2)=O)cc(Br)c(F)cc1Cl CC1C(NC(c2csc([N+](=O)[O-])c2)=O)CCCN1C(=O)CCCCO c1(OC)ncccc1C(=O)NC1CN(C(=O)Cn2cc(C#N)cn2)CC1C c1(CN2C(C(=O)Nc3c(CCC(N)=O)cccc3)CC2)cc(Cl)cc(Cl)c1 c1(OC)ccc(C=CC(=O)N(C(C)CNC(C2CCCCC2O)=O)C)cc1 N#CC1CCC(N=c2[nH]c(=NCC3CC34CCOCC4)c3ncccc3[nH]2)CC1 C(CN=c1cc(Cl)nc(C(F)(F)F)[nH]1)N1C(c2cc(F)cc(F)c2F)CCC1 N1(C(C(c2c(C)cccc2)C)=O)CC2CCC1C1CN(c3ncc(Br)cn3)CC21 c1(NC(C2C(C)(C)N(C(c3c[nH]ccc3=O)=O)CC2)=O)ccc2c[nH]nc2c1 c1(C(=O)N)cc2ccccc2s1.O=C1CC(CC(=O)NC2CCCC2C)C(=O)N1 C1(CC)CCN(C(=O)Cc2cnccn2)CC1.N1(C(=O)NC)CCC(C(=O)N)C1 N#CC1(CS(=O)(=O)N(CCO)CC2CC=CCC2)CCOCC1 CC1(C)CCC(C(=O)NCC(Cl)=CCl)CN1C(=O)C1=CC2C=CC1C2 C(=O)(CCC(=O)NC1CCN(C(c2snc(C)c2N)=O)C1C(C)C)NCC c1(CC)ccccc1OCC(=O)NCCCCN(C(=O)Cc1nnc(O)s1)C c1(C(N2CCC2C(N2CCC3(CCCO3)CC2)=O)=O)cc(F)c(F)c(Br)c1F c1(C(=O)NC2(C)CCN(C(c3nccnc3C(N)=O)=O)C2)nc[nH]c2ncnc1-2 N1(C(CC=CCC)=O)CCC(C(=O)NCc2n[nH]cc2C)(C(C)C)C1 N1(C(CC2(OC)CCC2)=O)CC2(CCC(NC(c3cccnc3O)=O)C2)C1 N1(C(C(CC)(CC)OC)=O)CCC2(CCC2)C(NC(=O)CC(=O)O)C1.C(C)(C)C c1(C=O)ccc2c(c1)NCC2.C1(NC(C2CC(SC)C2)=O)(C)CCCCC1C.N C(c1c[nH]nc1C)=CC=O.C1(CC(N2CCCC2CC)=O)(OCC)CCCC1.N C12(CNC(C(C)n3cnnn3)=O)CCC1CN(C(=O)CCc1csc(=N)[nH]1)C2 N1(C(C(C(C)C)F)=O)CC(CO)C2(C1)CN(C(C1CN=C3N=CNN3C1)=O)C2 CCCC(C(O)C(=O)NCCCn1cnnc1)NC(=O)CN(C(=O)COC)C C(=O)(C1=CCC(NC(c2cnn(C)c2N)=O)C1)NC(CCCCC)C c1(-c2cc(C(=O)NC3C(NC(c4c(C)n[nH]c4)=O)CC3)no2)ccc(Cl)cc1Cl CC(CCCc1ccccc1)NC(=O)CS.c1cccs1.C1(C)CC1.C1CC1.N C1(CNC(Cc2cn(C)nc2)=O)CCN(C(C2CCCC23CCC3)=O)C12CCC2 Cc1cc(Cl)ccc1C(=O)NC1(CNC(C2C3CCC23)=O)CCOC1 c1(C(=O)NC(CC=C)CNC(c2cnc(Cl)s2)=O)ccc2nnn(O)c2c1 N1(C(CC(=O)NC)=O)CCCCC2(CCN(C(=O)CC3CCCCO3)C2)C1 CCCCCCC(C)C(=O)NCC(CC(=O)N(C)Cc1nnnn1C)OC C(CCCC)NC(C(C)NC(=O)OC(C)(C)C)=O.C1(C=O)CC(=O)N1.N C(=O)(C(CN=[N+]=[N-])NC(=O)CC1CCSC1)NCCCCC1C(C)C1 n1(CCCC)cc(C(=O)NCC(=C2CN(C(=O)Cn3ccsc3=N)C2)F)nn1 N1(C(c2n(C)c(S)nn2)=O)CCC(C)(C)C1CNC(=O)C(c1ccc(Cl)cc1)O N1(C(C(C)N=[N+]=[N-])=O)CCCC(O)(CCNC(=O)C(c2cnn(C)c2)O)C1 c1(OC(C)C(=O)NCCC2COCCN2C(c2cn[nH]c2)=O)cccc(Cl)c1 C1(CNC(=NCCSCC=C)NC2CCC2)CCC2(CCCOC2)O1 C1(n2cc(-c3cncc(Cl)c3)nn2)(C=O)CC(F)(F)C1.C1(CC)CCC(C)C1.N S(=O)(=O)(c1ccc(Cl)nc1)N1CCC(CNC(c2c(CC)cccn2)=O)C1 C(=O)(C(F)(F)C(C)(C)O)NCCC(C)(C)NC(=O)CCCc1nccs1 N1(C(c2cc(C(C)=O)sc2)=O)CCCC(F)(CNC(=O)C=CBr)CC1 c1(OC)ncc(C(=O)NC2(C)CN(C(c3cscn3)=O)C2)cc1Cl CCC(C(C)O)NC(=O)CN(C(=O)CC1OCCCO1)C C(=O)(C1=C(C)OCCS1(=O)=O)N.C1(NC(c2nc(CC)oc2)=O)CCCCCC1 c1(OC)ccccc1C(N1CC(C)(CCC(=O)NC2CC(=O)N(O)C2)C1)=O Cc1ccc(O)cc1C(N1CC(O)(CNC(c2csc3cncn23)=O)C1)=O Cc1nsc(C(N2CC(NC(=O)CC3SC(=N)NC3=O)CC2C)=O)c1N c1(C(=O)NCC2N(C(c3ccnc(OC)n3)=O)CCCC2)ccc(Cl)c(C#N)c1 c1(NCc2ccc(OCc3ccc(F)cc3)cc2)nccc2cc[nH]c12 c1(N2CC(NC(c3ccccc3OC(F)F)=O)C(F)CC2)ncc2cn[nH]c2n1 N1(C(C2N(C(CC3CC(=O)OC3)=O)CC2)=O)Cc2cccnc2C1 N1(C(c2ncc(N)nc2)=O)CCCC(CC(N2CC3(CO)CC3(CO)C2)=O)CC1 c1(N2CCC(N(C(=O)CN3CCOCC3)CC)C2)nc(CC(C)C)nc(Cl)c1C N1(C(c2cc(CO)[nH]n2)=O)CCN(C(c2cc(C3CCC3)no2)=O)C(CF)C1 C1(CSC)CCC(NC(=O)Nc2ccc(CCC(F)(F)F)cc2)CC1 N1(C(C(C(C)C)OCC)=O)CC2CC(NC(c3c(Cl)cnn3C)=O)C(C2)C1 c1(NCc2nc(C)c(C)o2)ccc(-c2ccc(F)cc2)c(F)c1 C#CCC(CC#C)NC(C1(C(C)C)CCN(C(=O)CCc2conc2C)C1)=O C1(NC(C(c2cn(C(C)(C)C)nc2)=O)=O)CCN(C(C2(CF)CC2)=O)CC1O C(=O)(C(Cl)=CCl)N(CCCCNCC(=O)NC(CCO)C1CCC1)CCO c1(C(=O)Nc2cc(C)cc(Cl)c2)cc2ncc(-c3cnn(CCCO)c3)cc2[nH]1 c1(CC)nn(C)cc1C(=O)NCCN(CC(C)O)C(=O)C.c1ccncc1 c1(C(N2CCCC(NC(=O)CC3(O)CCC3)C2)=O)cccc(I)c1F N1(C(C2CC(C#N)C2)=O)CC2(CC(NC(C3C=CCC3)=O)CO2)C1 C=CCCC(F)(F)C(=O)NCCCC1(CNC(C2(O)CCC2)=O)CCCC1 c1(CN2CCC(C(C)C(N3CCC(C)(C)C3)=O)CC2)ccc([N+](=O)[O-])cc1Br CCCCN=C(NCCCc1ncn(C)n1)NCC(C)(F)F c1(CSC)c(C(N2CC(NC(=O)C(O)C(C)C)C(C)C2)=O)oc2ccccc12 C(=O)(CCC(C)(C)C#N)NCC(C)N(C)C(C1CC1C(C)(F)F)=O C1(CNC(C(C)C2CC2)=O)CC2CCC1N2C(=O)CCc1nc(C2CC2)no1 C1(CNC(CC=CC)=O)C(O)C(O)CN1C(=O)Cc1c(C)noc1Cl C12(C(N(CCOC)CC)=O)C3C4C1C1C2C3C41C.C1CCCC1.C(=O)C c1(C(N(CCCC)C)=O)ccc(OCCOC)cc1.C(=O)(C(CCO)N(C)C)N C(=O)CC(C)(C)CN(C)C.n1(CC=C)cccc1C(=O)NC1C=CCC1.C C1(C(=O)NCCCN(C(c2csc(Cl)n2)=O)CC)COCCN1C(C)=O N1(C(c2c(N)ccc(O)c2)=O)CCCC(C2CC2NC(c2ccns2)=O)C1 N1(C(C(C)OC2CCOC2)=O)CCC2(C1)CN(C(c1cccnc1C(F)F)=O)C2 c1(C(=O)NCCN(C(CCC=CCC=C)=O)CC)ccc(F)c(CS)c1 N1(C(CC(C)C2CCCO2)=O)CCCC1(C)CNC(c1cncn1C)=O N1(C(C2C(C)C2C)=O)CCCC(CO)(NC(=O)Cc2nc(C3CC3)cs2)C1 N1(C(C2C(CC)CCO2)=O)CC2(C1)CN(C(=O)C(C)=CCO)CCO2 Cc1cc(C(N2CCN(CC(C)NC(=O)C(F)C(C)(C)O)CC2)=O)cnc1C C1(NC(c2c(C#N)ccs2)=O)CN(C(=O)CCCC2CCC2)CCC1F CC(C(=O)NCC1COCCN1C(=O)C1=CCCC1(C)C)C1=CCCC1 c1(CC(=O)N(CC(CC)NC(=O)Cc2cccn2C)CC)cnn2c1CCCC2 c1(C(N2CCCC(NC(c3cc(OC)nc(F)c3)=O)C2)=O)cc(F)c(N)c(F)c1 c1(C(=O)NCC(C)NC(c2c(C(C)C)cnn2C)=O)nc2ccccc2cc1Cl CC#CCC(C(=O)N1CC(F)CC1CO)NC(=O)C=CCO N1(C(C(C)N(C(c2ccc(COC)o2)=O)CC)=O)CCCC(O)(CO)C1 C1(C(=O)NCC2C(=O)NC(=O)N2)CCCCCCN1C(=O)CC12CCCC1C2 C(=O)(C(C)(C)C(C)NC(c1ncc(F)cc1F)=O)N(CC(=O)NCC)C N1(C(C(Cc2ncn(C)c2)O)=O)CCN(C(c2cnc(O)c(F)c2)=O)CC1CO c1(C(=O)NCC(C)(C)NC(Cc2c(Br)ccc(C)c2)=O)ccc2nc[nH]c2c1 CCC(C#N)(CC)C(=O)NC(C)(C)CCC(=O)OC C(=O)(C1=CCCCO1)NC1(C)CCN(C(C2(C)CCSCC2)=O)C1 Cc1nnc2n1C(C(=O)NCC(O)CNC(=O)C(C)(C)O)CC2.CC(F)(F)F C1(NC(=O)CC2CC(NC(C3CC4(CCC4=O)C3)=O)C2)CC2(CCCC2)C1 Cc1ccc(C)c(C(=O)N(CCCN(C(=O)CCc2ccc(F)nc2)C)C)n1 c1(C(N2CCC(F)(CNC(c3[nH]cc(C)c3)=O)C2)=O)ccc2cnccc2c1 CC1NC(=O)CCC1N=c1[nH]c(N2CCc3ccc(Cl)cc3C2)nc2c1SCC2 C(N=c1[nH]c(N2CC=CC2)nc2c(F)cccc12)C1C(=O)NCC1 C(C)(CO)(C(=O)N(CC(O)C1CC1)C)NC(C1N(C(C)C)CCC1)=O c1(CC)ccc(NC(C2CCN2Cc2ccc(C)nc2)=O)cn1 N1(C(Cc2c(C)non2)=O)CCC2CCN(C(C34CCC(CC3)C4(C)C)=O)CC12 n1(CCOCC)nnnc1C(C)(C1CC1)NCCc1ccno1 c1(CC)cc(C(=O)NCC2CCN(C(C3CCCN(C(C)=O)C3)=O)C2)oc1 N1(C(c2nn(C(CC)CC)c(C)c2)=O)CCCC(O)C1.C(=O)(C(C)=CC(C)(C)C)N C1(C)(C(=O)NC(CNC(C)=O)C(F)(F)F)CC(C(F)(F)F)=NO1 c1(C(=O)NC(C2CN(C(=O)CC3CSC3)CCO2)C)cn(C)nc1Cl Cc1cn(C)cc1C(N1CCCC(CCCCNC(=O)CCNC(N)=O)C1)=O c1(CC(C(=O)O)NCc2c(F)ccc(Br)c2F)coc2cc(F)cc(F)c12 c1(OC)ccc(Br)cc1S(=O)(=O)NCC1CN(Cc2ccc(C)c(F)c2F)C1 N(C(=NCCC(=O)NC(=O)N(C)C)NCC1CCOC1C)CC(C)C N1(C(c2nc(CNC(c3c(CC)[nH]cc3)=O)oc2)=O)CCC(C2CC2)C1 C(=O)(C(CC)CC(C)C)NCCN1CCN(C(c2c(CC=C)cccc2)=O)CC1 C1(NC(c2c(C(C)C)n(C)nc2)=O)CN(C(c2cc(N)cc(F)c2)=O)C(C)(C)C1 C1(CC)(CC)CC(NC(c2c(C)ncn2O)=O)CN1C(=O)CN(C)C(C)C Cc1ccccc1NC(=O)C(C)N1CCC1CNC(=O)CC1COCCO1 Cc1[nH]nc(C(=O)NC2(CCNC(=O)CC3CCCCC3C)CC2)c1C c1(-c2scc(OC)c2)nc(CCOC)nn1C1CCCCC1C CC1=CCN(C(=O)CCC2(NC(C3CC3C#N)=O)CCC2)CC1 C=CCCC(F)(F)C(=O)NC(C)CCC(=O)NCCC1CC=CC1 C1(C(=O)NC)CCC(CNC(c2cc(-c3ccc(Cl)s3)on2)=O)CC1 C1(CN=[N+]=[N-])COC2(CCN(C(=O)C(N3CCSC3)=O)CC2)C1.C(=O)(C1CC1)C c1(OC)cc(C(N2CC(NC(c3nncn3C)=O)C(C)C2)=O)c(F)cc1N Cc1ncn(C)c1C(=O)NCC1C2CC1N(C(C1CCCC3CC13)=O)C2 Cc1cc(C(=O)NCCCCC(=O)N2CCC(c3nc[nH]n3)C2)ncc1F C1(C)(C(N2CC(CCCCNC(c3c(OCC)ccs3)=O)C2)=O)CCCC1C c1(C(=O)NC2CC(C(N3C(C(=O)NC)CC3)=O)C23CCC3)cccc2[nH]ncc12 C1(C)(CN(C(CC=C)=O)Cc2ccsc2)CC(O)CN1.c1cnc(C)c(Br)c1 C1(CNC(C(C)(O)C2CC2)=O)CN(C(=O)COCC(F)F)CC12CC2 C(c1ccc(F)c(C)c1)=CC(=O)NC1(CCC)CCN(C(=O)CSC)CC1 C(CCC(=O)N1CCCC1C(C)(C)CNC(C1(C2CCCO2)CC1)=O)N(C)C N1(C(=O)CN2CCCC2)CC(S(=O)(=O)C2CNC2)C1.c1ccccc1 CC(C)CS(=O)(=O)CCC(=O)NC(C)CCNC(C1CC12CCOCC2)=O c1(-c2cn(C3CC(C(=O)NCC(C)SC)C3)nn2)cc(C(=O)O)ccc1F N1(C(c2c(N)cc(F)cn2)=O)CCC2CC2(C(=O)NC(CO)CCO)CC1 C=CCC(C)C(=O)NCC(CCOC)NC(c1ccccc1COC)=O C(=O)(C1CCCc2sccc21)NC12C(CN(C(C3(C#N)CC=CC3)=O)C1)C2 C1(NC(C2N(C(CC3CC(SC)C3)=O)CC3(CC3)C2)=O)CCC(=O)NC1(C)C CCCC(CC)CC(=O)N1CCC(CNC(=O)CN(S(C)(=O)=O)C)C12CC2 Clc1ccc(C2(CNCc3c[nH]nc3-c3ccc(Cl)o3)CC2)c(Cl)c1 C(C1=CCN(C(=O)CCC2(O)CCC2)CC1)NC(C1CCCC(OC)C1)=O C12CN(C(=O)C(c3cc(F)ccc3C)(F)F)CC1CCO2.C(C(=O)NC)OCC C1(CCC)CN(C(=O)Cc2ccsn2)CCN1C(=O)CCCc1cncs1 c1(C(C)OCC)ncc(C(N2CC(CCC)C2)=O)s1.C(=O)C(C)(C)N(C)C C1(CNC(C(C(C)C)O)=O)CN(C(c2cc(C(F)(F)F)ncc2F)=O)CC12CC2 c1(CN(C(=O)CC2CCCN2C(C2CCC(F)C2)=O)C)cccc(F)c1 c1(OCCCCCC)cncc(OCCn2cc(C3CCCCC3O)nn2)c1 CCC(O)CC(=O)NC(CN(C)Cc1ccccc1)C(=O)NCC(C)CCO CC1CCCN1CC(=O)NCC1CC1CNC(c1ccc(Cl)s1)=O CC1(CCCO)CCCN1C(c1cnc(C(=O)O)o1)=O C1(CC)(NC(=O)C(C2CCCOC2)OC)CCCN(C(c2nc(O)sc2C)=O)C1 C1(CCNC(C(C)OCCCCCC)=O)CCCN(C(=O)C(F)n2cccn2)C1 CC1OC(C)CC1C(=O)NCC(=C1CN(C(=O)Cc2ccn(C)n2)C1)F c1(CC(c2n(CCOCC)nnn2)NC(c2cccnc2O)C)ccc(C)cc1 C#CC1(CNC(C2CC(NC(=O)CCOCCO)C2)=O)CCCC1.C Cc1ccc(NC(=O)C(N2CCC(N(C(=O)C(C)C(C)(C)C)C)C2)C)c(C)c1 C(=O)(C(C)C(F)(F)C(F)F)N(CC(CC)NC(c1cnn2ccccc12)=O)C CN(C1CCc2ccc(Br)cc21)c1ncnc(N(C)CCN(C)C2CC2)c1C#N O=S(=O)(CCC1CCc2ccccc21)NCc1ccc(Cl)cc1F c1(NC(C)C(C2CCCCC2)NC(c2cncc(Cl)n2)=O)cnc(C#N)cn1 C(=O)(C(C)(C)CCCCCC)N(CCNC(C(CCC#C)O)=O)CCC C1(C(=O)NCC2(NC(C3CCN(C(C)=O)C3)=O)CC2)CN2CCCC2CO1 CN1CCCC1C=CC(=O)NC1CCC(NC(=O)CSC)C1.c1ccncc1 CC1Cn2nccc2CN1C(=O)C(C)(C)CCNC(C1CCC(F)CC1)=O N1(C(CC2ON=C(C)C2)=O)CCC(F)(CNC(c2sccc2-n2ccnn2)=O)C1 C1(C(N2CCC2)=O)CCCCN1C(c1cccn1C1CC1)=O.C(=O)C(F)(F)F C1(C(N(C2CN(C(C3CSCCS3)=O)C2)C)=O)CC(C)(C)C1 C1(CN)CCN(C(C2(F)CCCC2)=O)CCC1(F)F C(=O)(C1CC(=O)N(C)c2ccccc21)N1C(CNC(COCCC=C)=O)CCC1 c1(C(N2C(CNC(CCS(C)(=O)=O)=O)COCC2)=O)n[nH]c2ccccc12 C1(C=O)CCCN1N=O.C=C(C)CCNC(C1CC1C(=O)NCCO)=O.N C1(CNC(C2(C)CCC(C)C2)=O)CC(C)(C)CN1C(=O)CCN(C)CCO c1(C(=O)NCC2(F)CN(C(Cc3cc(C)n(C)n3)=O)C2)ccnc2c1CCC2 O=CN1CCCC1C(N1CC(N2CCN(C(=O)C(F)C3CCC3)CC2)C1)=O Cc1cccc(CC(=O)N(CCC(C(C)(C)C)NC(C2CCNC2=O)=O)C)c1F C1(CCC(=O)Nc2ncc(Br)s2)CCCN(C(=O)NCc2ccco2)C1 C1CN(C(=O)C=O)C(C)(C)C1.C(C)(C)(C1(C(=O)N)CC1)OC.C(C)=O c1(-c2cn(CC(CNC(C(C(C)C)CO)=O)(C)C)nn2)cn2ccccc2n1 N1(C(c2c(OC)csc2)=O)CCCC(C(=O)N(CC(O)C(F)(F)F)C)C1 C1(C(N(Cc2cn(-c3c(C(=O)OC)cccc3)nn2)O)=O)CC12CC(C)(C)C2 C(=O)(C(C)(C)CC(C)(C)C)N1CCC2(C(NC(c3c(C)cc(O)nn3)=O)C2)CC1 c1(C=O)ccc(C)c(C2CC2)c1.CCC(C(=O)N)NC(N)=O.C1COCC1.C N1(C(c2n(C)ncc2)=O)CC2CCC(NC(C3CC=CC3)=O)CC2C1 C1(CC=C)(NC(c2ccc(OC)nc2)=O)CCN(C(C2(CC)CCC2)=O)C1.O c1(C(=O)NCCCCC(C)NC(=O)CCc2ccccc2)cc(Cl)c([N+](=O)[O-])[nH]1 C(=O)(CN=c1[nH]c(C)cs1)NC(c1cccc(C)c1)CNC(CC(=C)C)=O c1(NC(=O)N(CC(F)(F)F)CC2CC2[N+](=O)[O-])nc(C(F)F)co1 c1(C(N2CCN(C(CCCC#C)=O)C3C2C3)=O)ccc(C#N)c(O)c1 N1(C(CN(C(=O)OC)C)=O)CC2CCC1CN2C(C1CCc2ccnn2C1)=O C1(NC(C(C2CCC(C)CC2)CC)=O)CCN(c2ncc(O)cn2)C(C)C1 N1(C(=O)Cc2cccc(Br)c2)CCC2(CCN(Cc3ccnc(Cl)c3)C2)C1 c1(C(=O)NCC(CC)NC(=O)C(C2CCOCC2)O)ccncc1F c1(C(N(C2CCN(C(=O)Cc3cn[nH]c3)CC2)CCC)=O)nn(C)c(Cl)c1Cl c1(NC(NCC(C=C)(C)C)=NCCOCC)ccc2occc2c1 CC(C)CC(C)C(=O)N1CC(N2CCN(C(=O)C(c3ccccc3)=O)CC2)C1 N1(C(C2C(C)(C)CN(C(C34CC(F)(C3)C4)=O)C2)=O)CCCCC(C)(F)C1 C1(C=O)(CNC(C(C)SCCCC)=O)CC12CCC2.c1(C2CC2)cc[nH]n1 c1(OCC)cc(-c2nccn2CCC2CC2(F)F)c(-c2ccns2)c(Cl)c1O CCCC(F)C(=O)NCc1csc(C(=O)N(C2CC3CCC2O3)C)c1 C1(NC(C=CC=CCC)=O)CC(F)CN(C(c2cc(OC)ccc2F)=O)C1 Cc1cc(C(N2CCC(CO)(NC(=O)C=CC(F)(F)F)C2)=O)n2nccc2n1 C12(C(N3CCC(CC#C)C3)=O)COCC1CN(C(c1cccnc1C)=O)C2 C1(C)(C(N2CCC(CCNC(C(C)(C)F)=O)C2)=O)CC(C(F)(F)F)=NO1 c1(C(N2CC(C)CCC2)=O)ccc(S(N)(=O)=O)cn1.C1(C#N)(CC=O)CCC1.N N1(C(C(=Cc2ccco2)C)=O)CC(CC(N(C)CP(C)(C)=O)=O)C(C)C1 c1(C(N2C(CC)(CC)CC(NC(c3cnns3)=O)C2)=O)cnn2cccc(C)c12 C1(O)CCCN(C(=O)C=C2CCC(C)C2)C1.c1(C(C)C)ncc(C(=O)N)s1.C Cc1cc(-c2nc(-c3nc[nH]n3)nn2C(C)C(C)(C)C)c(F)cc1F C12(C(N(C)CC3OCCN(C(C(C4CC4)SC)=O)C3)=O)CCC(CC1)CO2 c1(C(N2CCCC(CC=C)(NC(C3CCSC3)=O)C2)=O)cc(F)cc(F)c1O N1(c2nnc(CC)s2)CCC2(CC1)OCCC2NC(=O)CCC.C(=O)(C1CC1)N C1(C(=O)NC(CCN(C(CCCOCC)=O)C)C)CCC(F)(F)CC1 C1(C(N(CCN(C(c2c(C)cc(CC)o2)=O)C)C)=O)C2C(=O)OCC12Br c1(NC(C2(O)CCN(C(C3CCC(=O)NC3)=O)C2)=O)cc(O)ccc1Br C12(C(N(CC(C(C)C)C)C)=O)CC3CC(C(=O)N1)C2C3 C1(C(C)C)CCC(NC(C2(C)CN(C(=O)C(CN(C)C)N(C)C)C2)=O)CC1 C1CCN(C(c2cnc(C)[nH]2)=O)CC1.CCCCOC(=O)C=CC(=O)N.C c1(C(N(C2CCN(C(c3c(CC)ncs3)=O)C2)CC)=O)cnc(F)c(C)c1 C(=O)(CC(C)CC(=O)NCC(C(C)(C)C)NC(C1CCCCCC1)=O)OC C12(C(=O)NCC3CCN(C(C4(CC=C)CCC4)=O)CC3)CCC(C1)OC2.C C1(CN=C(NCc2cnc(C)o2)NCC2CCCO2)COc2ccccc2C1 C1CN(C(=O)C(F)=CC2CC2)CCC1(F)F.C1(CC)CCCN(CC(=O)NC)C1 N1(C(C(C)SCCCC)=O)CCC(C(N2CC(O)(C(N)=O)C2)=O)CC1(C)C c1(C(=O)NCC(C2CCN(C(C3(C)CCCS3)=O)CC2)O)ccc2nncn2c1 CC1CCN(C(c2ccccc2C(C)(C)C)=O)CC1CNc1nccnc1C#N N1(C(CCc2cccc(OC)c2)=O)CC(NC(c2cc(Cl)ns2)=O)C(C2CC2)C1 C(=O)(C#CC1CCCO1)NCCC1CC(NC(C(C)(C)SC)=O)C1 C1(CNC(CC2C(C)C2)=O)CC2(CC2)CN1c1ncc(Cl)cn1 C=C(C)CCC(=O)N1CCC(N(C(=O)C=C(C)C2CC2)CCO)C1.C(C)=O N1(C(CCCCSC)=O)CC2CCCC2(C(=O)NCCC(C)C(F)(F)F)C1 c1(C(=O)NCCC2N(C(c3c(C)cns3)=O)CC(F)(F)C2)cc2c([nH]1)CCCC2 N1(C(c2cn(CCOCC)nc2)=O)CCCCC(NC(=O)CCC(C)OC)C1 c1(OCCC)c(OC)cc(CNCc2cccc(SC)n2)cc1Br N1(C(C)C(=O)NC2CCCC2)C(=O)CCC1=O.c1(C(=O)N)ccnn1CC(F)F O=S(=O)(CCNC(=NCC1CCC1(F)F)NC1CCCC1)C1CCOCC1 c1(OC)ccc(C(C)C(=O)NC(C)CCN(C(=O)C=Cc2ccoc2)C)cc1 c1(CCC=O)cnccn1.C(C)(C)(C1(C(=O)N(CCC)C2CC2)CC1)OC C1(NC(C2(C)N(C(C3CC(C)=C(C)CC3)=O)CC=C2)=O)CC2C=CCC(C1)C2 C1(NC(Cc2cn(C)nn2)=O)CCN(C(=O)Cc2cn[nH]c2)CC1CO c1(C(N2C3CN(C(C4(CN(C)C)CC4)=O)C(C3)C2)=O)cccc2c1OC(C)(C)C2 C1(CNC(COc2cc(C)on2)=O)CCC(N(C(=O)C(C)C2CCCC2)C)CC1 C1(CC(=O)NC2CN(C(c3ncccc3O)=O)C3CC23)CC2C=CC1CC2 c1(C(=O)NCCCCCCNC(C(CCC)(F)F)=O)cc2nccnc2[nH]1 N1(C(CS(C)(=O)=O)=O)CCC(NC(C2CCCN2C=O)=O)C12CCC2 C1(NC(C2C(CC)C2)=O)CC2CCC1N(C(=O)C=CC(C)(C)C)C2 CC1(C)NC(=O)N(CC(=O)NC2CCN(C(=O)C(O)C(F)F)CC2F)C1=O C1(O)(CC=O)COC(C)(C)C1.CC(Cn1cccn1)C(=O)NCC1CCC1 N1(S(C)(=O)=O)CCN(C(=O)CC2CCCN2C(=O)C(Cl)(Cl)Cl)CC1 C1(O)(CCNC(C(N2CCSCC2)C)=O)CN(C(=O)C=CCF)C1 CCC(CCC(=O)Nc1csnc1OC)NC(=O)C(C)CC1CCCC1 c1(OCCOCC)ccc(C(N2CC(C)C2)=O)cn1.C(=O)C(C)(O)CC.N C(CCN=C(NCC1CCOC1=O)NC1CCC12CCC2)OC C1(NC(C(C(C)C)NC(N)=O)=O)C2CC3C1C3C2C(N1CC(CO)C1)=O O=C1OC2CN(CCCC3CCNC3)CC2O1 c1(CN(C(=O)CC(N)c2ccccc2)C)cccc(Cc2ccccn2)c1 Cc1cc(C(=O)NCC2(O)CN(C(=O)C3=CC(C)CC3)C2)cc(C)c1Cl Cn1ncc(C(N2CCOC(C)C2)=O)c1C(F)F.C1(C)(CC=O)CC1(F)Cl.N C1(C=O)CC(O)CN1C(N)=O.C1(C(NC(C)C)=O)CCCN1C(C)=O.C C1(CCC(=O)NC(C)Cc2cnn(C)c2)CCN(C(=O)Cc2nccn2C)CC1 CCC(CCC(=O)N(C(C)CCNC(C1(n2cccn2)CC1)=O)C)OC C1CCN(C(c2cnc(C(F)F)s2)=O)CCC1(F)F.C(C)(C)(C(=O)N)OCC N1(C(C(C)N(C(C)=O)C)=O)CCC(CNC(=O)C)C(C)C1.C(C)(C)C.O C1(NC(=O)C#CC2CC2)CN(C(=O)Cc2ccc(C(F)(F)F)cc2)CC1C1CC1 CCC(CN(C)C)CC(=O)NC(C)CC.c1(C2(CC(=O)N)CCC2)ccccc1 C(c1ccncc1C)=CC(=O)N(CCN(C(CC=O)=O)C)C(C)C.CC.O c1(NC2CC(C)N(C(c3c[nH]c(Br)c3)=O)C2)ncc([N+](=O)[O-])cc1F N1(C(C2CC(OC)C2)=O)CCC(O)(CN(C)C(C2CCC(C)(C)C2)=O)C1 Fc1ccc(Cn2cc(COc3ccc(C4(F)CC4)cc3)nn2)cc1 c1(OCC(=O)NC(C(C)NC(=O)C(C)(F)F)C)cc(Br)cc(F)c1F C1(C2(NC(CCOCCN(C)C)=O)CC2)CCCCN1C(C1CCCCS1)=O Cc1ccc(Br)cc1CC(=O)NC1CCCCN(C(C2(C)COC(=O)C2)=O)C1 Cc1cc(Br)cnc1CNC(C1CCSC1(C)C)c1ccc(Cl)cc1 N1(C(C(C)CN(C)C(C2(F)CCCC2)=O)=O)CCC(CO)C(C)(C)C1 C#Cc1ccc(C(N2CCCC2c2ccsc2)C(=O)NCCOCC)cc1 c1(NC(=O)NCc2snc(-c3ccc(OC)cc3)n2)ccc2ncsc2n1 C1(N(C(=O)CC2(O)CCC2)C)CCC(NC(=O)Cc2sccc2Cl)C1 c1(SC)nccc(=NC(=O)C2CC3(CC3)CN2C(=O)C(C)(C)C)[nH]1 c1(C(N(CC(C)N(C(=O)CC(C)(C)O)C)C)=O)cn2c(Br)cccc2n1 CC1c2ccccc2CC1C(=O)NCCCCCCNC(=O)CCc1cncs1 C1(C(=O)NC2CC(OC(C)C)C2)CC2CN(C(=O)Cc3cnns3)CC2C1 c1(C(N2CCC(CC=C)(NC(=O)CC(C)OC)C2)=O)ccc(C#N)nc1O C#CCCCCCC(=O)N1CCC(N(C(c2cncc(F)n2)=O)CC2CC2)CC1 N1(C(C2(CC=C)CC2)=O)CC2CCN(C(=O)C(C)Oc3ccccc3C#N)C2C1 C1(NC(C23OCCC(C)(C2)C3)=O)C2CC3CN(C(c4cccnc4N)=O)C1C3C2 c1(OC)cc(Br)cnc1C(=O)NC1(CF)CCN(C(=O)C(C)C(F)F)C1 C1(C(=O)Nc2nnc(C(=O)OCC)s2)CCN(C(=O)CC)CC1.C1CCCC1 c1(CSC)c(C(=O)N)oc2ccccc12.c1(C(N2CC(C)C2)=O)nn(C)cc1Cl C1(OC)CN(C(c2cc(COC)on2)=O)CC1NC(C1CCOC(=O)N1)=O c1(C(=O)NCC2C(CNC(=O)CCC3CC3)C2)ccc2nc(Br)nn2c1 CC(C)(C)C(C)(C)C(=O)N1CCC(O)(CNC(=O)C(F)C2CCOC2)CC1 C1(CC(=O)NCCC2(C)CC2)CCCC1NC(c1cc(C(N)=O)co1)=O C(=O)(C#CC(C)(C)CNC(=O)OC(C)(C)C)NC1C(C)CCCCC1 C(=O)(CCCC(=O)N1C(C(=O)NCc2cncnc2)CCC1C(C)C)OC Nc1cccc(CC(=O)NC(Cc2ccccc2)CCNC(c2cc[nH]n2)=O)c1 CC1(C)C(NC(C2(O)CCOC2)=O)C1C(=O)NC1CCC1 C1(C(=O)NC2CCC(CNC(c3cncc(N(C)C)c3)=O)C2)CC12CCSCC2 Cc1nc(O)nc(C)c1CC(=O)NC1CC(O)CN(C(c2cn(C)c(C)n2)=O)C1 N1(C(c2c(OCC)ccs2)=O)CCC(CO)(NC(c2ncn(C)c2C)=O)C1 c1(C(=O)NCC2CC(OC)CN2C(c2nnn(C)c2C)=O)ccnc2cc[nH]c12 C(C)(CCC(=O)NCCCN(C)C)NC(C(C)N(C)C1CC1)=O C1(F)(C(=O)NCC2CC(CNC(c3coc(Cl)c3)=O)C2)CCCCC1 C1(C(=O)NC(C)CC2C=CCC2)CCC(n2cc(CCCC#N)nn2)C1 N1(C(=O)CCc2cnc(O)[nH]2)Cc2cccc([N+](=O)[O-])c2C1 C(=O)(CC1NC(=O)c2ccccc21)N1CC(NC(CC(=C)C)=O)C(C)C1 N1(C(C2C(C(=O)OC)C2)=O)CC(CC(=O)O)(NC(c2ccccc2)=O)C1 N1(C(c2c[nH]c(=NC)s2)=O)CCC2(CC1)CN(C(C1CC(C)(C)CO1)=O)C2 Cc1cc(C(=O)NC2C=CCN(C(c3ccnc4ncnn34)=O)C2)cc(=O)n1C N1(C(C(CC=CC)C)=O)CCCC(O)(CC)C1.C(=O)(CCCc1n[nH]c(=N)s1)N c1(CCC(=O)NCC2(NC(=O)CC3CCCOC3)CC2)ccc(F)nc1 C1(NC(C2C(COC)C2)=O)CN(C(c2ccc(Cl)cc2F)=O)CC2(CCC2)C1 Cc1cc(C#N)cc(C)c1CC(N1CCN(C(c2ccns2)=O)C(C(C)C)C1)=O c1(C2C(C)C2)ccc(CCC(=O)NC(CNC(=O)CC2(C)CC2)CO)o1 CC(C)(C)C(=O)NCCC(=O)NC.C1(O)CN(C(=O)CC(O)C2CCCC2)C1 c1(CCNC(CCCOCC=C)c2nnnn2CCCC)ccncc1C C1(C(=O)NCC(CC)O)CC(C)(C)CN1C(=O)COCC1CCCC1 C(=O)(CC(C)(C)CC(=O)NC1CC(F)CN(C(=O)CCF)C1)OCC C(=O)(C1=CC2(CCOCC2)C1)N1CCCC(CNC(=O)COC2CCCC2)C1 C1(NC(=O)CCc2cccnc2Cl)CN(C(=O)CCN2CCCC2)CC(F)(F)C1 C#Cc1ccc(F)c(C(N2CC(CCNC(C3CCCC(C)CC3)=O)C2)=O)c1 N1(C(c2cncc(-n3cnc(C(=O)OC)n3)c2)=O)CCC(C(=O)OC)C(CN)C1 c1(OCC(=O)NCC2(C)CCN(C(Cc3cc(C)[nH]n3)=O)C2)ccccc1C#N CC1=C(Br)CCN(C(c2ccc(-n3ccnc3)cn2)=O)C1 CC1CC(NC(=O)CC2CCN(C(=O)CCCCC3CC3)C2(C)C)CCC1(C)C C1CN(C(=O)C=C2CC2)CCC1C(F)(F)F.c1(C(C)=O)c[nH]c(C=O)c1.N C1(CN(C(C2(CC)CCCC2)=O)C)COCCN1C(c1nc(Cl)sc1C)=O C1(CCNC(CCC=C)=O)CCN(C(c2cnoc2C2CC2)=O)CCC1(F)F N1(C(C2C(COC)C2)=O)CC(O)(CC)C1.c1(N(CCC=O)C)ccncc1 N=c1ccc(C(=O)NCCCCCNC(=O)CSC2CC2)c[nH]1 C(=O)(CC(F)(F)C(F)(F)F)NCCC1CC(NC(c2ccc(C#C)cn2)=O)C1 C1(C)(CNC(CSCC(=O)OC)=O)CCN(C(=O)CNC=O)C1 c1(NC(N2CCN(Cc3cc(C)cc(=O)o3)CC2)=O)c(C)ccc2cnccc12 C1(N(C(C(C2(O)CN(C(CCC)=O)C2)F)=O)C)CCCC(O)C1 c1(C(N2CCC(CC)C2CNC(=O)CC(C)F)=O)c[nH]c2ncccc12 Cc1cc(=O)n(C)cc1C(=O)NC1CC(O)CN(C(=O)C2=CCCC2)C1 c1(C(=O)NC2CCC(C)N(C(=O)C=Cc3cc[nH]n3)C2)cc(O)c(O)c(O)c1 C1(C(N(CCC)CCNC(c2cc(C(C)C)nn2C)=O)=O)CCCCC12CCC2 c1(CCC(=O)NC2CCN(C(c3ccc(Cl)c(Cl)n3)=O)C2)ccc(F)cc1Br CCC(CC)C(=O)NCC(=O)Nc1ccccc1.CC(=O)NC1(CCC)CC1.N C1(NC(=O)CCc2cccc(F)c2)CC2(CCN(C(=O)Cc3cc[nH]n3)CC2)C1 C1CCCCC1.C1(C=O)C(Cl)(Cl)C12CC2.C1(N(CCC(=O)NC)C)CCCCC1 N1(C(CCCC#C)=O)CC(CNC(=O)C(=Cc2cnc[nH]2)C)C(C)(C)C1 c1(CC)cccc2c1NC(=O)C2NC(c1cc(=O)n(C)c(O)n1)=O C1(CCC)CN(C(c2c(C3CC3)noc2C)=O)CCN1C(=O)C(C)c1ccsc1 N1(C(C=CC(=O)N)=O)C2CCC1CC1(C2)N=N1.c1nc(C=O)co1.C1CC1 c1(C(=O)NCC(CO)NC(c2c(C)noc2)=O)ccc(C(C)(F)F)cn1 c1(C(C(=O)OC)(C)C)ccc(NC(C2CCC(C(=O)OC)C2)=O)c(OC)c1 CCCCC(F)C(=O)N1CCC(C2CCCN2C(c2scnc2Cl)=O)CC1 CCN=c1cc(C(=O)NC2CCC(N(C(=O)CCCOC)C)C2)cc[nH]1 C1(NC(CC(C)C2CC2)=O)CCCC(CNC(c2cnc(-c3cccs3)o2)=O)C1 CC(C)(CC#N)C(=O)N1CC2CC(C1)C2NC(C1CCCC(O)C1)=O Cc1cc(Cl)c(C(=O)NCC(C)(C)CCNC(c2ccn(C)c2)=O)cc1F C=CC(C(F)(F)F)NC(=O)N(C1CCCCC1)Cc1cnn(C)c1 C(CCC(C)(C)NC(=O)C(C)NC(C12CCCC1C2)=O)OC c1(C(=O)OCC(=O)Nc2ccccc2Br)ccc(F)c2[nH]ccc12 N1(C(CCCCOCC)=O)CC2CC1CN(C(c1ccnc(C3CC3)n1)=O)C2 CCCCCC(F)C(=O)NC1C2CC3C(C2)C13C(N1CCC(C2(C)CC2)C1)=O C1(C(=O)NOCc2cccnc2)(NC(=O)CON)CCOCC1 C(=O)(C#CC1(C)CCCO1)NC1C(C(=O)Nc2cc(C)c(F)cc2F)OCC1 c1(OC)cccc(-c2nc(CO)nn2C2CCCOC2)c1CO C1(C(=O)NOCCN2CCCC2=O)(CC#C)CCN(C(c2ccon2)=O)C1 c1(C(=O)Nc2nc(Cl)ncc2O)cc2cc(-c3cc(F)ncc3F)ccn2n1 c1(N2CC(CNC(C(c3ccc(OC)cc3)(C)C)=O)C2)ccc(F)cc1[N+](=O)[O-] Cc1ccc(C)c(C(C)C(N(C(=O)N(C2CCNCC2)C(C)C2CC2)C)=O)c1 C1(CNC(C(C)N(C(=O)C(COC)N(C)C)CC)=O)CCN(OC)C1 C(=O)(CC(C(F)(F)F)c1ccccc1)NCCOC1CCN(C(CCC#N)=O)C1 CN1CC(C(=O)NCCN2CCN(C(c3ccc(=O)n(C)n3)=O)CC2)CCC1=O Nc1[nH]c(=O)c(Cl)nc1C(=O)NCC1CCCN(C(C2CCCCN2N=O)=O)C1 C(CC(=O)NC1CC2CN(C(c3cnoc3C)=O)CC2C1)(C(F)(F)F)OC N1(C(Cc2c(C)occ2C(F)(F)F)=O)CCN(C(C2CCOC2)=O)CC(C)(F)C1 C12(NS(C3CC(CC(C)(C)C)C3)(=O)=O)CC3(C)CC(C)(C1)CC(O)(C2)C3 c1(C(=O)NC(CC)CNC(=O)C(C)C(F)(F)F)cc(C#N)cc(C)n1 CC1CN(C(=O)CC2CCCN(C)C2)CC1CC(=O)N(C)CCN(C)C Cc1ccc(C(=O)NC2(CNC(=O)CSCC(C)C)CCCCC2)c(C)c1 C1(CC)CN(C(c2ncccc2Cl)C(=O)Nc2ccc(F)cc2)C(CC)CO1 C1(NC(C23CCCC2C3)=O)CCN(C(C2CCCN(c3ccccn3)C2)=O)CC1 C1(C(=O)NC(CNC(c2cccc(Br)c2O)=O)CO)CCc2ccnn2C1 C(=O)(CS(N)(=O)=O)NC(C)CC(C)NC(=O)C(C#N)=CC1CC1 c1(CNCCCC(=C)Cl)cc(Br)c(OC)cc1C N1(C(C2C(C(C)C)C2)=O)CCC2(CCCC2)C1.C1(CC=O)CCCC12CC2.C C1(C(=O)NCCC(C)N2CCC2)CNC(=O)CN1C(=O)CC1CC(=O)NC1=O C(C)(CCC(=O)NCC(C(=O)NC1(CO)CCC(C)C1)OC)OC C(CC(=O)NCCN(C(=O)CCCC#N)C1CC1)(C(N)=O)NC(C)=O N#Cc1ccc(CNC(C2CCC(NC(C3CCSCC3)=O)CC2)=O)cn1 CC1C(NC(=O)C(F)(F)C2CCOCC2)CCN1C(=O)CC1CCC(F)(F)C1 C1(c2nnnn2CCSC)(NCc2cc(CC)on2)CCCC(C)CC1 c1(C(CNC(C2CC(COC)(CO)C2)=O)OC)ccc(SC(F)(F)F)cc1 C1COC(C)(C)CN1C(=O)C=CC(=O)N(C)C.C(CC(=O)NC)=CCC N#CC1(C(=O)NC2CN(C(c3ocnc3-c3ccccc3)=O)C2)CC2(CC2)C1 N1(C(CCc2c(OC)cccc2)=O)CC(OC)CC(NC(=O)C(C)CF)C1 c1(-c2cn(C3CC(CNC(C4N(C(C)=O)CCC4)=O)C3)nn2)ccc(C)cn1 C1(NC(C2N(C(C(C=C)(C)O)=O)CC(O)C2)=O)CCCCN(C)C1=O CC1CN(C(C2CC(C)(C)C2)=O)CCC1NC(=O)C(C1(O)CCCCCC1)(F)F N1(CC(=O)NCC(C)(C)C)CCC(CNC(=O)C(C)(C)C2CCC2)CC1 N1(C2CN(C(C3(CC)CCCC3)=O)C2)CC(NC(C2CCOC2=O)=O)CC1=O Cc1c(OCC(=O)NC2CC(C)CN(C(C3(C)CCCC3)=O)C2)cccc1Cl c1(OC)cc2[nH]c(C(=O)Nc3cnc(C4CC4)nc3)cc2c(OC)c1OC c1(C(C)(C)NC(C2CN(C)CC2O)=O)cc(Cl)cc(Cl)c1 C(=O)(CC(C)(C)C(=O)N1CC(OC)C(C(=O)NC(c2nccs2)C)C1)OC N1(CC)CC(C(N2CCN(CC(=O)N(C3CC3)C(C)C3CC3)CC2)=O)CC1=O c1(C(N2CCC(O)(CNC(CCC(C)=O)=O)CC2)=O)ccc2sncc2c1 N1(CCC)CCN(C(=O)CSc2ccc(-c3nccc(N4CCC4)n3)cc2)CC1 C1(CNC(CN(C)CCO)=O)C2CC2CN1C(=O)CCn1cncn1 CC(C)CC(C)(O)C(=O)N1CC(CNC(=O)CCN2CCOCC2=O)C2(CC2)C1 N1(C(C2Cc3c(C)[nH]nc3CC2)=O)CCC2(CC1)CCN(C(=O)C(C)CCO)C2 CC1CCC(NC(c2cnn(C3CCCC3)c2)=O)CN1C(c1ccoc1)=O N1(C(CCN(CCC)C)=O)CCC(CNC(C2C3CNC(=O)C23)=O)CC1 C1(C#N)(C(N2CCC(C(N3CCC(C(C)(C)C)C3)=O)CC2)=O)CC2CC2C1 c1(CNC(N2C(c3n(CC)ccn3)C(C)(C)C2)=O)cc(O)cc(O)c1 Cc1sc(C(=O)NC2(CNC(c3c(C4CCCC4)noc3C)=O)CCC2)nc1O C1(N2C(C(N(C(CC)C)CC)=O)CCC2)CCN(C2CCCC2C(=O)OC)CC1 N1(C(c2c(C)ccs2)=O)CC2CCN(C(c3cn(C)c(=O)nc3O)=O)CC2C1 N1(C(C(CC)(C)O)=O)CCC2(CC(C(=O)NCC3Cc4ccccc4C3)=NO2)C1 c1(C(=O)NC2(C)CCN(C(C(C)OCCC=C)=O)CC2)cnn2ccn(C)c12 Cc1ccncc1N(C(c1ccnc(F)c1)C(=O)NCC1CCCO1)C O=C(CCCCc1ccc(Cl)cc1)NC1CC1NC(=O)CCc1cscn1 Cc1ccc2c(c1)C(NC(c1ccc3n[nH]c(C)c3c1)=O)C(C)C2 c1(C(=O)NCC(CNC(=O)C=Cc2ccncc2)CO)ccc2scnc2c1 Cc1ccc2[nH]cc(C(=O)NCC3(O)CN(C(=O)C=Cc4c[nH]nc4C)C3)c2c1 Cc1cc(N)ccc1C=O.C1(C(N(CCCC(C)C)C)=O)CCN(C)S1(=O)=O.N Cc1nccc(Cl)c1C(=O)N(C1CCC(n2cc(CN(C)C)nn2)CC1)C Cc1c(Br)sc(C(N2CCN(C(c3cn(Cc4cnns4)nn3)C)CC2)=O)c1C c1(CCCC)nc(C(=O)NC2CC2NC(=O)C(c2cnn(C)c2)C)cs1 c1(C(=O)NCC2C(C)CCN(C(CCC(=C)Cl)=O)C2)c(F)cc(C)cc1Cl O=C(NNc1ccc(F)c([N+](=O)[O-])c1)NCCC(=O)NC1CCCCC1 N1(C(C2CCN(C(=O)Nc3c(CC)cccc3)C2)=O)CCN(C(C)=O)CC1C n1(CC(=O)N(CC)C)cnc2c1c(=O)n(C)c(=O)n2C.C(C=O)(C(C)C)SC C1(NC(Cc2cn(CC)nn2)=O)COCCC1C(N1CCOC(C2CC2)C1)=O C1(NC(CCCCC=C)=O)CCCCN(C(=O)C(CC=C)C(C)C)CC1 C=CCCCC(C)(C)C(=O)NC1CC1C.C1(=CC=O)CC2CCC(C1)N2C.N N1(C(C2(C)CCC(=O)NC2)=O)CCCCCC(NC(c2cccc(Cl)c2)=O)C1 C(=O)CS(=O)(=O)N(C)C.CC(Cn1cccn1)C(=O)NCC1(C)CCC1 c1(C(N2CCN(C(CC3(C)CCOCC3)=O)C3C2C3)=O)cc(Cl)c(Cl)cc1N c1(C(=O)NC2C(CC)CN(C(c3nccc(C)n3)=O)CC2)cc2cccnn2c1 c1(C(=O)NC(C2CCCN2C(c2ccco2)=O)C)cccc2nnn(C)c12 c1(CNC(C2N(C(c3cc(C)[nH]c3C)=O)C3C(C2)C3)=O)cccc(C)c1O CCC(C#N)C(=O)NC(C)CC(=O)NCCC(F)(F)F Cc1nc(CNC(C2CC2C(C)(C)F)=O)cs1 CC1=CCC(N=c2[nH]c(=NCC3CCN(C(C)(C)C)C3)[nH]c3cccnc23)CC1 C(=O)(C(CNC(=O)CCC1CCCC1)C(C)(C)C)N1CCCC(OC)C1C N1(C(c2cn(CC=C)nc2)=O)CCC2(CC1)CN(C(C13CC(C1)C3)=O)CC2C N1(C(C(C)(C)c2nccs2)=O)CC(NC(C2C3CCCCC23)=O)C2(CC2)C1 C(=O)(C(CCCC(C)C)NC(c1ccc(-c2cccc(C#N)c2)cc1)=O)OC c1(CCNC(CNC(CC2(C)CCOC2)=O)=O)ccc(O)cn1 c1(C(=O)NC(CCC)CNC(C2CCOC2(C)C)=O)ccc(O)cc1C CCC(C)CCCCC(=O)NCc1ccc(C(=O)NC2CCOCC2)nc1 c1(N(CCCN2CCC(O)CC2)CC)nc(C(=O)OC)cc(N)n1 c1(C=O)cc2ccc(F)cc2o1.C1(O)(CNC(c2cnc(O)o2)=O)CCC1.C Cc1ncnc(N2CC(F)CC2CNC(=O)C(C)Cc2ccncc2)c1F c1(OC)cscc1C(=O)N(C)CC1CCCN1C(=O)CC1CC(C)=NO1 C1(NC(COC)=O)CCCCC12CCN(C(c1cccc(F)c1SC)=O)CC2 CCC(CC(C)C)C(=O)NCc1ccc(C)cc1.c1(C(=O)N)cc(C)cc(C)c1 C(=O)(CC(=O)NCC(CNC(=O)CCc1ccon1)CO)OC C=CC1CCCC(NC(=O)CC2C(NC(=O)CNC(=O)OC)CC2O)C1 CC(C)(C(=O)N1CC(C(N)=O)(CNC(c2cc(O)no2)=O)C1)C1CCCO1 c1(C(N2CC(C)C(NC(=O)Cc3c[nH]ccc3=O)C2)=O)cc2ccc(Cl)cc2[nH]1 C1(C(=O)NCCCN(CC)CC)COCCN(C(C)Cc2cc(C)ccn2)C1 C(C(CC)N=c1[nH]c2cc(F)cc(F)c2o1)NC(C1(CC=C)CCOCC1)=O CC(CC(F)(F)F)C(=O)NC1CCC(NC(C2CN(C(C)C)CCCO2)=O)C1 c1(C(N(CC(C)(C)CNC(=O)CS(N)(=O)=O)C)=O)cn2cccc(F)c2n1 O=C1NC2(CN(Cc3csc(Br)n3)C2)Nc2ccccc21 c1(C(=O)NCC(CC(C)C)(C)NC(c2ccc(O)nn2)=O)ccc2ccoc2c1 C1(F)(CNC(C=C(C)CN2CCOCC2)=O)CCC1.C1(C=O)COC(=O)N1 C(C(C)CC(=O)N1CC(OC)C(NC(c2cc(C3(C)CC3)n[nH]2)=O)C1)OC C(=O)CC(C)(C(F)(F)F)N(C)C.N1(C(c2c(C)[nH]c(=N)s2)=O)CCCC(F)C1.N c1(NCCN2CCC(C)(C)C2)cc(S(=O)(=O)NCC(O)C(C)(C)C)ccc1C#N Cn1c(-c2nc(-c3ccc(C#N)cn3)no2)cc2ccc(Br)cc12 c1(-c2cc(CCC)on2)nc(-c2ccoc2)nn1CCc1ccncc1 C(=O)(CC(C)(C)C=O)OCC.C1(C=O)CCC2(C1)CC2(F)F.C1CC(C)C1 N1(C(C=C=C(C)C)=O)CC2CC(NC(c3nccn4cnnc34)=O)CC1C2 Cc1c(C(=O)NC(C)CCNC(=O)CCCCCN(C)C)[nH]c2c1CCCC2 C1(NC(c2csnn2)=O)(CF)CCN(C(c2ccnc(O)c2)=O)C1 c1(C(=O)NCC(C)NC(C2(Br)CC2(F)F)=O)c(Cl)ccc2c1OCO2 C1(C(=O)NOC2CCCCC2)(CC)CCN(C(C2CCCCO2)=O)CC1 C1(C(=O)N(C(=O)CN)C2CC2)CC(F)(F)CN1C(C1(CCCC)CCC1)=O CC(C)(CC(F)C(=O)N1CCC2(C1)CC2(F)F)NC(=O)CSc1cn[nH]c1 Cc1cc(CC(N2CCC(N(C(c3cnc[nH]3)=O)CC3CC3)CC2)=O)nn1C C(N=c1cc(C)nc(C)[nH]1)C1CN(C(C2C(CC)C2)=O)CC1(C)C C(C(C(=O)NC1CCC1)C(C)(C)C)NC(C=CCOCCOC)=O.C C1(CCNC(C(SC)SC)=O)CSCCN1C(c1cnn(CCO)c1N)=O C(=O)(CS(=O)(=O)C(C)C)NC(CCCNC(c1c(C)ncnc1C)=O)C N1(C(c2cn(CC)nn2)=O)CCCC1(C)CNC(=O)C(n1nc(C)cc1C)C C1(C(N2CC(C(=O)NCc3nncs3)(SC)C2)=O)CN(C)CC(C)O1 C1(CNC(=O)Cc2cnc[nH]2)CCCCN1C(c1cscc1C(F)F)=O c1(C(=O)NCC(CC)NC(=O)CCC2CC2C)c[nH]c2ccccc2c1=N C1(N(C)C=O)(C=O)CC1(C)C.C1(=CC=O)CCN(C)C1.C(C)(C)C.C N1(C(c2cc(C)c(C)nc2)=O)CC2(CCCC2)C1C(=O)NCc1cnccn1 c1(OC)csc(C(=O)NC)c1.C12CC(C1)C2.C(=O)C(C)CC1CCCCC1 c1(CCNC(CCN(C(=O)C=CC(C)CC)CC=C)=O)cnnn1C C1(C(N(CC(C(=O)NC(c2cccs2)CC)C)C)=O)CC2CC1CC2=O C(=O)(C(C)(C)CCC#N)N1CCCCC(NC(C=Cc2cncc(OC)c2)=O)C1 CCCCCC(C)NC(=O)CONC(C1(CC)CC(C)(C)C1)=O C(C(C)C(=O)N1CCCC1CCNC(C1(c2ccccc2)CC1(F)F)=O)OC c1(SC)nc(C)c(C(=O)N(C)C)s1.C1CCCC1.C1(C=O)(C(F)F)CCCO1 C(=O)(N=c1ccc(C#N)c(C)[nH]1)c1cc(OC)c(C)cc1 n1(CCNC(CCCC(c2ccc(C)cc2C)=O)=O)cc(P(C)(C)=O)cn1 C1(NC(C2C(CC)OCC2)=O)(CF)CCN(C(C2(CC#N)COC2)=O)C1 CCC(CNC(c1cnn2c1OCC2)=O)(CC)C(=O)NC1CCN(CC)CC1C C1(CC=C)(NC(=O)CC2COCCO2)CN(C(C2CC2CC)=O)C1 C(=O)(C(CC)C(C)C)NCC1(C)CC(NC(CC(=C)I)=O)C1 CCCC(O)(CCC)CC(=O)N(CCCN(C)C(c1snc(Cl)c1Cl)=O)C N1(C(c2cc(C)c(Br)cc2)C(=O)NCc2cccs2)CCOC2(CCOC2C)C1 C1(NC=O)CCCCC1C(=O)O.C1C2CN(CC(F)(F)F)CC12.C1CCOCC1 c1(CC)cc([N+](=O)[O-])ccc1C(N1CCCC(NC(=O)C(CC)CC)C1C)=O Cc1nc(C)c(C(N2CC=CC2CNC(c2cccs2)=O)=O)nc1C N1(CC(N2C(c3n(C)nc(I)c3)CCC2)=O)CCN(C(=O)O)CC1=O.C(C)(C)C c1(C(=O)NC(C=CC(=O)NCC(CCC)C)(C)C)cccc(C)c1C#N N1(c2nc(C)nc3c2c[nH]n3)CCC2(CCCN(C(C3(F)CCCCC3)=O)C2)C1 C(=O)(CCC(=O)N(C)C)NC(CCC)CNC(c1cnn(C2CCC2)n1)=O C1(C(N2CC(CC)N(C(=O)CCC3CCC(=O)N3)CC2)=O)CCC2(CCC2)CC1 Cc1nnc2n1CC(C(=O)N(C)CC1(NC(=O)C(C)C#N)CC1)C2 Cc1cc(O)c(CN2CCCC(c3nnc4ccccn34)C2)cc1C CN1CCC(C)(C(=O)NCC2(F)CN(C(C3(C4CCC4)CCC3)=O)C2)C1=O C1CCCCC1.C(=O)(CCNC(=O)C=CCO)N(C)C1CC1.C(N)=O.C O=C(C#CC1CCCOC1)NCCC1COCCN1C(=O)C(=O)NCC(F)F CCC(C)(CNC)C(=O)N1CCN(CCOC(F)F)C(=O)C1.c1cn(CCO)nn1 c1(CNC2C(C(=O)NC(c3ccccc3I)CO)CCC2)cc(F)c(F)c(F)c1 N1(C(CCCc2c(C)ccs2)=O)CCC(CCNC(=O)C#CC(C)C)CC1C c1(C(=O)NC(c2ccc3c(c2)CCC3)C)cc(F)c(Br)cc1Cl C1(CC(=O)C(C2CCCCC2)=O)CC(C(C)(C)C)=NO1.C(CC)N(CC)C C#CCCCC(C)C(=O)NC1(CNC(=O)C=C2CCC(C)(C)CC2)CC1 C1(CNC(CCN(C(CCC)C)C)=O)C2CN(C(=O)Cc3cc(OC)no3)CC12 Cc1cnc2n1C(C(=O)N1CCC(CNC(c3ccc(CO)cn3)=O)C1)CCC2 N1(CC(=O)NC2(CNC(c3cncc(O)c3)=O)CCOC2)CCCCCCC1=O Cc1cc(=NC(CNC(c2ccnnc2Cl)=O)C2CCC2)c(C#N)c[nH]1 C12CCC(CC1n1cc(CCN(C)C)nn1)C2.C1(CC(C)C)(C=O)CCCC1.N C1(C(=O)NC(CC(C)C)CNC(=O)C#CC(=O)N(C)C)Cc2nncn2C1 C(C(C)(C)CC(=O)NC1CCCCNC1=O)NC(CC1CN(C(C)=O)C1)=O CC(C(=O)NC1CCN(C(=O)CSCCC#N)C1(C)C)S(=O)(=O)C1CCOCC1 N1(C(c2cc(F)cc(F)c2)C(=O)NC(CC)C)CC(C)(CO)CC1(C)C N1(C(CSCCOC)=O)CC2CC(NC(c3ccccc3)=O)CC2C1.C(N)=O O=C(C1=CCCSC1)NCC1CN(C(=O)C2=CCC2)CC1C(F)(F)F O=C1CCC(C(N2CC3CC2C3NC(=O)C(c2cccc(Cl)c2)(F)F)=O)CN1 c1(C(=O)OCC)cnn(C)c1OC(=O)CN(C)Cc1cnns1 c1(C(N(CC(C)NC(=O)C(c2ccccc2)SC)CC)=O)cnn(CC)c1Cl C1(F)(C=O)CCC(=O)CC1.C1(N(C(=O)COC2CCOCC2)C)CCCCC1.N N1(C(=O)CCOCC2CC2)CC2CCN(C(=O)Cn3cc4ccccc4n3)C2C1 O=C(C1=COCCO1)NC1C=CCN(C(C23COC(CF)(C2)C3)=O)C1 N1(C(=O)C=Cc2ccccc2)CCN(C(c2cccc(O)c2)=O)C(C(F)(F)F)C1 S(=O)(=O)(c1[nH]c(=NCC2(C)CCC2)ccc1Br)N1C(C)CCCCC1 N1(C(c2c(COC)ncs2)=O)CC(NC(=O)CC)C2(CC2)C1.c1ccccn1 c1(C(=O)NC(CC)(C)CNC(=O)CCC(C)SC)ccc(Cl)c(OC)c1N N1(C(=O)CC2CCCO2)CCCC2(C1)CN(C(C1COCCO1)=O)CCO2 CC1(C)CC(NC(=O)CCc2ccoc2)CN(C(c2ccc(O)c(F)c2F)=O)C1 CN1CCN(C(c2coc(CNC(C3(C4CC4)CC3)=O)n2)=O)CCC1=O CC(C)(C)CC(O)C(=O)N1CCC(CNC(=O)C(=O)NC2CC2)C12CCC2 CCCC(CCC)C(=O)NC1CC2(C1)CN(Cc1cccc(Br)c1C)C2 c1(OCC)cc(C(=O)NC2CCN(C(c3c(Cl)n[nH]c3)=O)C2)oc(=O)c1.C c1(-c2nc(C(C)C3CC3)nn2CC2CCCC2(F)F)c(F)ccc2nc[nH]c12 N1(C(C(C(C)C)NC(C)=O)=O)CC2(CCCN(C(=O)Cc3cnsc3)C2)C1 Nc1cc(C(=O)NCc2nc(C)cs2)cc(Cl)n1.C(=O)(CCc1cnc[nH]1)N Cc1cnnc(-c2cn(Cc3ccc(C(=O)NCCC(C)CO)o3)nn2)c1 C(c1ccccc1)=CC(=O)NCC1CCOC1.c1(C=O)ccc(C(F)F)nc1.N N1(C(C(C)=C(C)C)=O)CCC(C(O)CNC(=O)COc2ccsn2)CC1 c1(OC)cccc(C(=O)NC2CCN(C(c3ccc(SC)s3)=O)C(C)C2)c1N c1(C2(C(=O)NCC3(F)CCN(C(c4cnon4)=O)C3)CC2)cccc(F)c1F CC1CN(C(C2CC3COCC3C2)=O)CCC1C(=O)NCC1CC1.C1CCC1.C C1(CNC(=NC)NCc2cc(C(C)(C)C)on2)CC2(C1)C(F)(F)C21CCC1 C1(NC(CCOC)=O)CCC(F)(CNC(C23CC(C2)C(C)O3)=O)C1 C(=O)(C1c2c[nH]nc2CN1C(c1cc(O)cs1)=O)NCC(C=C)O CC(C)C1=NOC(C(=O)NCC2CCN2C(=O)CC2CCCC(F)(F)C2)C1 C1(NC(CNC(CC)=O)=O)CCCN(C(=O)CCN2CCCC2=O)CC1F CCCC(CCC)C(=O)NCC(CC(=O)N1CCC1C(=O)N(C)C)OC C=CC(C)CC(=O)NCCC1(CNC(=O)C(C)Cc2ccc(F)cc2)CC1 C1(CNC(C2C(C=C)C2)=O)N(C(=O)CCN2CCCC2)CCCC1(C)C c1(C(=O)NC2CC(NC(=O)C=CCF)C2)ncn(-c2ccccc2)n1 C1(CNC(=O)CCC(F)F)CCC2(CCC2)C1NC(c1cn(CCO)nn1)=O C12(C(=O)Nc3n(C)ccn3)CCN(C(=O)CC3CC3)CC1C2 CCCC(C#N)C(=O)N1CCN(C(=O)C2=CCOCC2)C(CC2CC2)C1 CCC(CC(=O)NC1(CCCC(=O)NCC2CC3CCC2O3)CCC1)SC C(=O)(C1=NOC2COCC12)N1CCC(C(C)CNC(=O)Cc2ccon2)C1 C1(NC(CN(C)C(c2ccc(Cl)s2)=O)=O)(CO)CCSC1 c1(C(C)=O)cc(C(=O)N(C)CCNC(=O)CC2OCCOC2(C)C)c(C)nc1C Cc1cc(S(N)(=O)=O)cc(C(N2CCOCC(NC(=O)C(C)CO)C2)=O)c1C C1(C(N2C(CN(C(CC(=C)C)=O)CC)CCC2)=O)CCC(CC2CC2)CC1 Cc1cnc2cc(C(=O)NC(C3(O)CN(C(=O)C(C#N)C(C)(C)C)C3)C)ccn12 c1(C(N2C(C(=O)NC(C)Cc3ccnn3C)COCC2)=O)ccc2ccoc2c1 Cc1ccc(CC(C(=O)NCCCN(C(=O)C(C)C)C(C)C)N(C)C)cc1 Cc1cc(NC(C)COCC2CC2)ncc1S(=O)(=O)NCCC1SCCS1 N1(C(C(C(C)O)C)=O)CC2(CC(NC(c3cc(CF)on3)=O)CO2)C1 c1(C(N2CC(NC(C(C)C3CCCO3)=O)(CO)C2)=O)ccnc(Cl)c1O c1(NC(C(N2CCC(Cc3ccn(C)n3)C2)C2C(C)CC2)=O)ccc(Cl)cc1F CC1CN(C(=O)CSCC(F)(F)F)CCN1c1cc(C2CC2)nc(C2CC2)n1 c1(C(c2cccs2)NC(c2cccn2C2CCCC2)=O)cccc(Br)c1 C1(NC(c2c(C)con2)=O)CN(C(c2cnc(N(C)C)nc2)=O)CC1N=[N+]=[N-] c1(CC(=O)N(C(C23CC(CC)(C2)C3)=O)C2CC2)cnc(C)cn1 CCCCCCC(C)NC(C1(CNC(c2ccc(CO)cc2)=O)CC(C)(C)C1)=O N1(C(c2nc(C#C)sc2)=O)CCc2sc(CNC(C3CCC(C)O3)=O)nc2C1 CC1=C(C(=O)N)CCC1.c1(C(N2CCC(C(C)(C)C)C2)=O)ccc(=O)n(C)c1 c1(NC)ncccc1C(=O)NC1CCCC(NC(C2CCN(C(C)=O)C2)=O)C1 C(CCCNC(c1cnn(C2COC2)c1)=O)OC.c1(C=O)ccc(C(N)=O)[nH]1 N1(C(CC(CCC)O)=O)CCCC12CCN(C(=O)CN1CCCCC1)C2 C(=O)(C1=CC(C)(C)C1)NC(CC=C)CNC(c1csc(-c2ccsc2)n1)=O Cc1nc(C(F)(F)F)oc1C(=O)NC1CCC(NC(C2CC(C)C2)=O)C1 Cc1nc(NC(C2(C)CCCN2C(c2ncnn2C)=O)=O)nc(C)c1Br N1(C(c2cn(CC=C)nn2)=O)CC(NC(C2CC3CCCC3C2)=O)C2CCCC12 N1(C(C=CC)=O)CC(C(=O)O)CC12CCC2.C1CNC(=O)O1.NCCC N1(C(Cn2c(C)ncc2)=O)CCN(C(C2C(C)C2C)=O)C(CO)C1 Cc1c(Br)cnc(O)c1C(N1CC(CNC(=O)C(O)C(C)C)C(O)C1)=O Cc1c(C(=O)NC(C(C)NC(=O)Cn2nccn2)C(C)C)csc1Br C1(C(=O)NCC2N(C(c3cnn(C)c3Cl)=O)CCC2)CCC2CCCCN12 C1(C(=O)NC2(C(=O)NCC3(Cl)CCC3)C(C)(C)C2)CC12CCOCC2 C(C)(N=c1[nH]c(N(C)CCc2ccccn2)nc2cc[nH]c12)c1nnc(C)o1 N1(C(CN(CCC)C)=O)CCCC2(CCCCC2NC(=O)CC2CC2)C1 CCCCCCC(F)C(=O)N1CC2(CCN(C(C3(C#N)CCCO3)=O)CC2)C1 O=C(C1=C(Cl)CCC1)N1CC2(CCN2C(C2CC(O)C2)=O)C1 C(=O)(C1=CCCSC1)NCC(C)(C)NC(=O)Cc1ccc(O)cc1Cl c1(OC)ccc(C(N2CCOCC(NC(=O)C(F)(F)C3CC3)C2)=O)n2nccc12 CCCCCCC(C)C(=O)NC1CCN(C(C2CCC(C)CC2)=O)C1 Cc1cc(NC(C2(C)CCN2Cc2ccc(Br)cc2)=O)c(C)cc1Cl Cc1cc(=NCCc2ccc(F)c(Br)c2)[nH]c(=NCCN2C(C)CCCC2C)[nH]1 c1(CNC(CNC(N(C(c2c(C)cccc2)C)C)=O)=O)ccc(F)cc1F C1(C(N2CC(O)C2)=O)COCCN1C(=O)Cc1ccc(-n2ccnc2)cc1 C(=O)(C(C)(C)C(N)=O)NCC1N(C(C=CCCC(C)C)=O)CCC1C c1(SC)ccccc1C(N1CC(NC(=O)CSCC2CCCCO2)C1)=O C1(CC=O)CCCN(C=O)C1.CCCC.c1(CC(=O)N)ccoc1.C(C)(C)C Cc1ccc(C(C(=O)NC(C)C)N(C)Cc2ncn(C)n2)o1 CN=c1ccc(C(N2CC3CC3(C(=O)Nc3nc(Cl)ccc3C(N)=O)C2)=O)c[nH]1 N1(CC(=O)NC(C)C(CO)NC(=O)Cc2nnc(O)s2)C(=O)CCC1=O c1(C(N2CCC(CC(=O)N(C(C)C(C)(C)O)C)CC2)=O)cccc(O)c1F C1(C)(CC(N2CCC(CC)CC2)=O)CCS(=O)(=O)N1.Cn1ccc(CC=O)n1.N c1(CNC(c2onc(C)n2)=O)ccccc1CN(C(=O)CCn1cccn1)C N1(C(C(COC)OC)=O)CC2(CCC2NC(=O)CCc2cnc(O)[nH]2)C1 N1(C(C)C)CC(C=O)CC1=O.C(c1ccc(Cl)s1)=CC(N1C(CC)CCC1)=O.N N1(C(CC2CCN(C(C)C)CC2)=O)CCN(C(C2C3COCC23)=O)CC1CCO Cc1noc(C)c1.C1(NC(CSCC)=O)CCN(C(c2ccc(F)s2)=O)CC1.C C1(C(=O)NCCC2CCCCN2C(c2csnc2Cl)=O)COCC2(CCC2)O1 C1(c2cn(C)nc2)CN(C(=O)CCOCC2CCC2)CCN1C(c1ccsc1)=O c1(C(=O)NC2CCN(C(C#CC(=O)O)=O)C2)n[nH]c2ccc(F)cc12 C1(N(C(C2C(C)C2C)=O)CC2CC2)CCCN(C(c2ccncc2F)=O)C1 C1(CNC(C(C2CCCC2)NC(c2cn[nH]c2)=O)=O)CCCSC1.C1CC1.C C(=O)(CCC(=O)NN(C)C)NCCNC(C(C1CCOC1)OC)=O O=C(CCCC(F)(F)F)NCC1CN(C(=O)C(O)Cc2ccccn2)C1 C1(C(C)C)C(C(=O)Nc2ccc(Cl)cc2)CCN1C(=O)CSc1cn[nH]c1 CC(C)CC(C(=O)NCC(C)CO)ONC(=O)c1cnsc1 C1(NC(c2cn(CC=C)nn2)=O)(CO)CCCN(C(C2CCCN2CC)=O)C1 C1(CC)CCN(C(=O)CCSCC(N)=O)C1CNC(C1SCC=C1C)=O N1(C(c2ccnc(C)n2)=O)CC2CN(C(c3oc(CO)nc3C)=O)CC2(C)C1 N1(C(C(C)O)=O)CC2C(NC(C3CCN(C(=O)OC(C)(C)C)C3)=O)C2C1 C1(Cl)(C(N2C(CNC(C(N3CC(C)C3)C)=O)CC2)=O)CC1(F)F c1(C(N2C(CNC(C(c3scc(C)n3)C)=O)CC2)=O)nccc(C(F)(F)F)n1 C(=O)(CCCCCNC(c1cc(=O)n(C)cn1)=O)NC(CC(C)(C)OC)C c1(OC)cscc1C(=O)NC(C)CC1CN(C(c2csc(C(F)F)c2)=O)C1 c1(C(N2C(C)CN(C(COCC(C)C)=O)C(C)C2)=O)ccc2c(c1)COC2=O O=C(C(Cc1ccoc1)NC(=O)C(F)OC(F)(F)F)NCC1CCCSC1 N1(C(c2cc(C)c(C)s2)=O)CCCN(C(=O)CCCC(F)F)CC1 N1(c2n(C)c(C3COC4CCCC4O3)nn2)CCn2ncc(S(N)(=O)=O)c2C1 CCC(C(=O)N1CCCCC(NC(=O)C(C)(Cl)Cl)C1)C(C)(F)F c1(C(=O)NC(CC(C)NC(C2(CC=C)CC2)=O)C)cccc(C)c1O C1(NC(Cc2c(CC)cccc2)=O)CN(C(C2CC2c2ccco2)=O)CCC1F c1(OC)ncc(C(N2CCC3C(NC(=O)CC4CSCCS4)CC23)=O)cc1C C(CCC(C)C(=O)NC1CCC(C(=O)NC2(C(C)(F)F)CC2)C1)OC C1(C(=O)NC(CN(C(c2cc(C(C)C)nn2C)=O)C)C)CC2C=CC1C21CC1 c1(CN2CCN(c3ccc(NC(=O)C(F)F)cn3)CC2)cc(O)ncc1Br N1(C(c2c(C)con2)=O)CCC(CC(C)NC(c2cnoc2C2CC2)=O)CC1 C1(NC(C2(CC#C)CCCCO2)=O)CCc2[nH]c(=N)sc2C1 c1(C(=O)NCC=CCC(=O)N(CC(C(=O)NC)C)C)ccc(OC)nn1 c1(C(=O)NC(C2CN(C(=O)C)C2)C)cn(C)cn1.C1(C(=O)N)CCCCC1 C(=O)(CCCCC)NCC=CCNC(c1c(CC)n(C)cc1)=O.C(N)=O.N c1(CN2C(C(=O)NC(CCCC)CO)C=CC2)c(Cl)ccc(F)c1F c1(NC(C(C2CCOCC2)C)=O)cccc(-n2cccc2)c1 C1(F)(CNC(C(C(C)C)N(C)C)=O)CCN(C(c2ccncc2Cl)=O)CC1 C=CC1(CC(=O)NC(C)CNC(C2CCC2C(F)F)=O)CCCCC1 N1(C(C(CC)C)=O)CCC2(CC1)CCN(S(=O)(=O)c1ccc(OC)c(Cl)c1)CC2 c1(N(C)CC2N(C(CC(C)C3CCCCC3)=O)CCC2)ncc(C(C)(C)O)cn1 c1(C(=O)NCC2N(C)CCN(C(C3CCC(=C)CC3)=O)C2)cc2cnn(C)c2s1 N1(C(c2cc(C)c(Cl)s2)=O)CC2CCC(C1)N2C(=O)C(C)(C)S(C)(=O)=O c1(C(N(C)CC2CCCN(C(C3CCCCS3)=O)C2)=O)cccc2cc[nH]c12 C(C(=O)N1CCN(C(c2ccncc2OC(C)C)=O)CC1C)(C(C)(C)C)OC CC1OC2CCC1(C(=O)NCCC1CCC1)C2.N1(CC(=O)N)CCNC(=O)C1 C=CCN(OC)C(=O)C(C1CCCC1)NC(c1c[nH]nc1C(C)C)=O c1(C(=O)NCC(C2CCOC2)NC(CCOCC)=O)n[nH]cc1Br C(CC)(CC)(CC)NC(c1c(CC)nccc1)=O.c1(C=O)ocnc1C1CC1.N Cc1cccc(Cl)c1CC(N1CC(CNC(C2CC3(CCC3)C2)=O)C(C)C1)=O c1(C(=O)NC(c2cn(CC3CCOC3)nn2)CCC)cc(Br)sc1Cl C1(C(=O)NCCC2N(C(C=NOC)=O)CCOC2)Cc2cccc(C)c2O1 N1(C(C(C(C)O)C)=O)CC(NC(=O)CSC(F)(F)F)C(C)(C)C1 CCCC(C)(C)C(=O)NCC(C1CCCN1C(c1cc(F)cnc1O)=O)(C)C c1(C(=O)NCC(CNC(C(C)OC)=O)C)cccc([N+](=O)[O-])c1 CC1(CCC(N2CCC(NC(c3nncs3)=O)CC2)=O)CCC(=O)N1 C(=O)(CC1=CCCCC1)NCC(C(C)C)NC(CCC(=O)OC)=O CCC(C(=O)N(C(C)C(C)n1cccn1)C)NC(=O)C=CC(=O)OCC CC1CCN(C(=O)CCC2CCC2)CC1CNC(=O)CC1(N(C)C)COC1 n1(CC)ncnc1CNC(=O)C=CC(C)(C)NC(=O)CCC1CC1 CCC(C)(C)CC(=O)N(C)CCO.C(=O)(C(C)Cn1ccc(C)n1)N(CCC)C CCCC(CNC(=O)C(C)CC1CC1)C(=O)NCC(C)(CO)CO c1(C(=O)NC(C2CCCN2C(=O)CCC)C)cc2cccnc2cn1.C(C)(C)C.O c1(N2CCCC(NC(=O)OC(C)(C)C)(CO)C2)cc(C(F)F)nc2ncnn12 C1(C)(CC(=O)NC2(C(=O)NC(C(=O)OC)C)CC2C)CCOC1 C1CCN(C(C2(N(C(=O)C(C)=CC(C)(C)C)C3CC3)CCC2)=O)C1.CO c1(CNC(C2C(c3n(CC)ncc3)OCC2)=O)ccc(Cl)c(OC)c1 N1(C(c2nn(CC)c(O)c2)=O)CC(C)(C(=O)NCC2CC2(C)C)CC1(C)C c1(CC)cccc(C)c1C(=O)N(CC(C)CNC(=O)C(C)(C)F)C c1(C(N)=O)cccc(C(=O)NCCC2CCCN2C(c2nscc2N)=O)c1 c1(C(N(C)CCOCCN=c2[nH]cnc(=N)[nH]2)=O)cc2c(Cl)cc(Cl)cc2[nH]1 C1(CNC(CN(C)C(N)=O)=O)CC2CCCC2N1C(=O)CS.c1cccs1 Cc1ccnnc1C(N1CC=CC1CNC(C1CCCC12CC2)=O)=O CN1CCC(CCC(=O)N(CC(O)CN(C(=O)CCCc2ccccc2)C)C)C1 N1(C(CCc2c(C)nc(O)nc2O)=O)CCC2(CC1)CN(C(=O)C(C)C(C)O)C2 Cc1[nH]c(=N)sc1C(=O)NC(C)CN(C)C(C1CC(=O)N(C2CC2)C1)=O C1(C)(CCC(C)C)NC(=O)N(CC(=O)OCCOCCOCCO)C1=O C1(CNC(c2c(C)n(C)nc2)=O)CCC2CN(C(c3cc(F)ccc3N)=O)CC12 C=C1COc2c(C(=O)NCCN(CC(C)O)C(C3CCCCN3C)=O)cnn2C1 C(C(F)(F)C(C)(C)O)NC(C(CC=CC)NC(c1n[nH]c(C)c1Cl)=O)=O c1(C(N2CCC(N(C(c3ncc(C)nc3)=O)C)C2)=O)cc(Cl)cnc1O C1(NC(CN(C)C)=O)CCCCC12CCN(C(c1cnn(C)c1Br)=O)C2 c1(OC)ccc(CC(N2CC(N(C)C(c3ccoc3C3CC3)=O)C(O)C2)=O)cc1 C1(C(C)C)CN(C(=O)CCCCN(C)C)CCN1C(=O)C=Cc1ncco1 c1(C(=O)NCC2CC(CNC(C(C#N)C3CC3)=O)OC2)cnc2cccnn12 c1(C(=O)NC(C)C(C)(C)NC(C2C=CCC2)=O)cc2c(s1)CCC2 c1(C(N2CCCC(NC(CC3(COC)CC3)=O)C2)=O)cnc2sccn12 Cc1cccnc1C(c1ccc(F)cc1)NCc1ccc(CC2CC2)s1 C1(CC)CN(C(=O)C(N2CCCCC2)C)CC1C(=O)NCCC1(C)CCOC1 N1(C(c2cccc(OC)c2N)=O)CC2CCCC2(NC(=O)CS(=O)(=O)N(C)C)C1 C1(C)(CC)CC(C(=O)NC2CN(C(c3csnc3C)=O)C(C)(C)C2)CCO1 n1(CC(=O)NCCCOCCC)ncccc1=O.C(=O)(C(O)CN1CCCC1)N Cc1nn(C)cc1C(N1CCCCC1CC(=O)NC1(CO)CC1)=O C1(NC(COCCC)=O)CCCC(C(=O)NCc2[nH]nnc2CC)CC1 n1(CC)cc(C(N2CC(NC(C3CCOCC3)=O)C(O)C2)=O)c(C(C)(C)C)n1 c1(OC)ccc(C(N2CCC(O)(C(C)NC(=O)C)C2)=O)nc1Cl.C1(C)CCC1 C1(C(=O)OC)CC2(CCCC2)CN1Cc1cc(C2CC2)cc(F)c1 N1(C(c2nc(CC)sc2N)=O)CC(C2CN(C(=O)C(C)(CC)CC)C2)C1 C(=O)(C1CCCc2scnc21)NCC1CN(C(C(C)CC(F)(F)F)=O)C(C)C1 C1(C(=O)NC2C(NC(c3csc(C4CC4)n3)=O)COC2)CC2CCCCCC12 N1(C(C(C)n2cccn2)=O)CC2CC1C2NC(=O)Cc1ccc(CO)cc1 Cn1cc(C(N2CC3CC3(NC(C3CC34CCOCC4)=O)C2)=O)n(C)c1=O N1(C(C(C)O)=O)CCCC1C(C)NC(=O)Cc1cnc[nH]1 C1(C)(CC)CCCC(NC2(c3ccncc3)CC2)C1 C1(N(C)C(C2CC(C)(C)CCO2)=O)CCC2CN(C(=O)C(F)C(F)(F)F)CC12 C1(C(=O)OCC)CCC(NCC2(CS(C)(=O)=O)CCC2)CC1C C1(C)(C(N2CCC(CCOC)(NC(CSCC=C)=O)C2)=O)CCC(C)CC1 C=CC1(CC(=O)NC2CCC2NC(c2cc(-c3cnn(C)c3)[nH]n2)=O)CCC1 C=CCC(CC(C)C)C(=O)N1CC(C(C(=O)NC2(c3ccsc3)CC2)OC)C1 c1cc(C2CC2)ccc1C(=O)N(C1CCCN(C(=O)CN2CC(C)C2)C1)C.CO C1(O)(C(N2CCN(C(c3cnc(OC)nc3)=O)C(CF)C2)=O)CCC(C)(C)CC1 N1(C(C(C)(C)OC(C)C)=O)CC2CCCC(C1)N2C(=O)CCCCCN=[N+]=[N-] CC1CN(C(=O)CC(C)(C)O)CCN1C(C1C2CC(F)(F)CC12)=O C(=O)(C1=C(F)CN(C(=O)C(C2CCOCC2)O)CC1)NCC(C)O C12(C(=O)NC(CC)(C)CO)CC(CO)(CN1C(C1CNC(=O)N1)=O)C2 CCC(CC)CC(F)C(=O)NCC1CCC(C)CN1C(c1cnc(Cl)[nH]1)=O C(=O)(N=c1[nH]nc(OCC[Si](C)(C)C)cc1Br)NC1CN(C)CC1F C1(NC(=O)C2=COCC2)CN(C(=O)C(c2cccc(Br)n2)(F)F)CC12CC2 N1(C(c2c(N)nccc2)=O)CCCOC(CNC(=O)COC2COC2)C1 C(=O)(CC(C)C(=O)NC(CC(=O)N(C(C)C(C)C)C)C(F)F)OCC C1(C(=O)NCC2C(C(N(CC(N)=O)C)=O)C2)CCOCC1 C1(NC(CCNC(C2CC(SC)C2)=O)=O)CC2CC1C(O)C2O C1(C(N(CC(C)CNC(c2cnc(C(N)=O)s2)=O)C)=O)CCC(C)(F)CC1 N1(C(CCOCC)=O)CCC2CN(C(=O)Cc3ccc(C)cc3Cl)CC12 C(=O)(C1=CCCC1C)N1CCC(OCCNC(C(CC)CC2CCCC2)=O)CC1 N1(C(C=CC=O)=O)CCC(C=C)(C(=O)NC2CCN(C(C)=O)C2)C1.C C1(CNC(c2onc(C)n2)=O)CC2(CC2)CN1C(=O)CC1CC1 CCC(C(=O)N(CCCCCNC(c1cn(C(C)C)nn1)=O)C)OC C1(C(=O)NC2(C)CN(C(c3cnc[nH]c3=N)=O)C2)CC2CCC(C1)C2 Cc1ncccc1CCC(=O)NCC1(NC(c2cnc(S)[nH]2)=O)CCOC1 c1(C=O)cc2n(n1)CC(F)C2.C1(NC(CCC=CCC=C)=O)CCC(F)(C)C1 n1(C(F)F)cnc(=NC2CCNC3(CCCCC3)C2)[nH]1 c1(C(N(C)CC2(O)CN(C(=O)C(O)C(F)F)C2)=O)cc2cccnc2o1 c1(CC=O)cccc(C)c1C.c1(NC)nc(C(=O)NCCC2CCOC2)cs1.N C(=O)(C(CC)N(C)C)NCCC(=O)N(CCOCC#C)C N(C(=NCc1ccco1)N1CCC(CCOC)C1)CC(C(=O)OCC)(C)C N1(C(C(C)C)=O)CC(CO)C2(C1)CN(C(c1cc([N+](=O)[O-])n[nH]1)=O)C2 c1(C(=O)NC2(CNC(C=C(C)C3CC3)=O)CC2)ncc(C)cc1F c1(C(=O)O)ncccc1CN1CCC(CC2CC2)CC1 C1(CNC(Cc2n(C)ccn2)=O)(NC(C2CC3CC2CC3O)=O)CC2CCC1CC2 C1(C#N)(C=O)CC1(C)C.c1(CN(CC(C)(C)C)C)nn(C(C)(C)C)cc1Cl N1(C(N2C(C)CC(O)C2)=O)CCCN(c2ccc(F)cc2)CC1 C1(C)(C=O)CCCN(C(C2CC(=O)N(C(C)C)C2)=O)C1.C1(OC)CCCC1.C C(C(=O)NCCCN(CCO)C(C1CC12CCCC2)=O)(C(C)C)OCC c1(C(=O)NC2(C(=O)NCCc3nccs3)CCC2)cc(O)cs1 CCCCCCCCCC(O)C(=O)NC(C)CN(C)C(C1CC1(F)F)=O c1(C(N2C(CNC(c3cnc(C)[nH]3)=O)CCC2)=O)scc(C)c1Br N1(C(C2C(C=CC)CN(C(C)=O)C2)=O)CCCC12CCCCC2 Cc1ccc(C(N2CC(Nc3cc(Br)no3)C2)=O)o1 C(CC(C(C)(C)C)NC(C1(C)CCCO1)=O)N(C(C(C#C)(C)C)=O)C C1(NC(C(CCOCC)NC(c2cncc(C)c2)=O)=O)CCC(C)(C)C(C)C1 C1(N(C(=O)C)C)CCCN(C(C2CC2(C)Br)=O)CC1.c1ccc(C(N)=O)cc1.N N1(C(CCCCCC=C)=O)CCN(C(=O)CSC2CCOC2=O)CC2(CC2)C1 c1(NC2CN(C(C)=O)C2)cnc(F)cn1.C12CC(C1)CNC(=O)C2 N1(C(c2sc(C)c(O)n2)=O)CCC2(CC1)CC(NC(=O)CSc1nc[nH]n1)CO2 N1(C(C2(S(N)(=O)=O)CCC2)=O)CCC(C2(NC(C3CCSCC3)=O)CC2)C1 c1(C(=O)N)cccc2c1OCC2.C1(CC=C)(C(=O)NC2CC(C)C2)CC=CC1 N1(C(CC=CC=C)=O)CCCC(O)(CNC(c2c(OC)cccc2F)=O)CC1 Cc1nc2sccn2c1C(=O)NC1CC2CC1CN2C(=O)Cc1ccoc1 n1(CC)ncc(Cl)c1C(=O)NCC1C2CN(C(=O)CS(N)(=O)=O)CC12 Cn1[nH]c(=NCc2ccc(Br)c(Br)c2)c2c1CCOC2 N#Cc1cc(F)c(Cl)nc1NC(C1CN(C(=O)CSc2ccccc2)C1)=O C1(C(N2CC(C(=O)OC)(CC)C2)=O)C2CN(C(c3ccc(Cl)cn3)=O)CC12 N1(C(C(CN(C)C)NC(c2cc(CC)[nH]n2)=O)=O)CCCC(O)(C(N)=O)C1 c1(OC)cc(C(=O)NCC2CCCC2)cc(F)c1F.C(=O)CCO.C(N)=O.N c1(C(N2CCC(N(C)C(c3cn(C)nc3Cl)=O)C2)=O)cnc2c(cnn2C)c1 c1(C(=O)N)nc(C2CC2)oc1C.C1(CNC(C2C(CCC)C2)=O)COCC1 C1(OC)CN2CCCC2(C(=O)NC2CC(C)N(C(c3ccc4c(c3)CC4)=O)C2)C1 c1(C(CCOC)NC(CCC(C)(C)C)c2n(C)nnn2)cccc([N+](=O)[O-])c1 c1(NC(CCCN(C)C(c2cocn2)=O)=O)cccn(CC)c1=O c1(COC(C)C)cc(NC(=O)C(n2cnc(C(F)(F)F)n2)C)ccc1O C12(C(=O)NCCC(=O)N(CC(C)O)CCOC)CC(C1)OC21COC1.C C1(CCC(N2C(c3cn(CC(CC)O)nn3)CC2)=O)CCCN(S(C)(=O)=O)C1 Cc1[nH]nc2ncc(NC(C3CCC(NC(C4C=CC(=O)N=N4)=O)CC3)=O)cc12 C1(C)(CC)CCCN(C(=O)C(O)CNC(c2ccc([N+](=O)[O-])o2)=O)CC1 c1(C(N2CCN(C(C(C(C)(C)C)N(C)C)=O)C(CF)C2)=O)cc(F)c(F)cc1O N1(C(COC2(C#C)COC2)=O)CCCC(C)(C)C1.C1(C=O)CN(C(N)=O)C1.N c1(CC(N2C(CNC(c3c[nH]nc3C3CC3)=O)CC2)=O)cc(F)ccc1Cl c1(CCC(=O)NCC(CNC(CC(C)c2ccncc2)=O)F)ccc(Cl)cc1F c1(C(=O)NC(C(C)C)CNC(=O)C(C2(O)CCCC2)F)ccc[n+]([O-])c1 N1(C(CCC2CC(NC(=O)CCc3cncs3)C2)=O)CC=CC(O)C1 N1(C(c2c(NC(C)=O)sc(Cl)c2)=O)CCC(C)C(C)C1 Cc1occc1C(N1CC(O)(C(C)NC(=O)COc2ccon2)C1)=O C(=O)(N=c1[nH][nH]c2c1CN(C(=O)CC(O)c1ccccc1)C2)c1n[nH]c(C)c1C CCC(N=c1ccnc(C)[nH]1)C1(CO)CCCC1 c1(C(N2CCN(Cc3c(C)n[nH]c3C)CC2CO)=O)cc(Cl)cc2nc[nH]c12 CC(CC(=O)NCC1CN(C(=O)CCCN2CCOC2=O)C1)C(C)(C)C C1(C(N2CC(OCC)C2)=O)CC(C)(C)CCN1C(c1nccc(C)c1F)=O C1CC(C)N(C(=O)C=CC(c2ccccc2)=O)C1.N1(C=O)CC(C=O)C1.C C(=O)(C(C)(C)c1sccc1Cl)NCC(CC)NC(C1CCC(C)O1)=O C1(CC(N2CC(C)(NC(Cc3n(C)nnc3)=O)C2)=O)CCC(=O)NC1 c1(C(=O)NCC(C2CCC2)NC(C(C(C)O)N(C)C)=O)cccn2cnnc12 N1(C(c2cc(OC)c(Br)nc2)=O)CCCC2(CCCN2C(C2CC2C)=O)C1 c1(NC)ccc(C(=O)N)nc1.C(C)(C(=O)N1CCC(n2cnnn2)C1)C1(C)CC1 N1(C(c2cc(C)sc2)=O)CC(NC(c2ccc(-c3ncon3)cc2)=O)CC1C N1(C(c2cc(CNC(CC3CCC(C)O3)=O)ncc2)=O)CC2(CNC(=O)C2)C1 c1(Cn2cc(C3(C)CN(C(=O)Cc4ccc(F)cc4)C3)nn2)ccc(I)cn1 c1(C(C(N2CC(CCNC(CNC(CC)=O)=O)(O)C2)=O)(F)F)ccccc1F c1(C(N2CCC(NC(CCC(=C)Cl)=O)C(CC)C2)=O)n[nH]c2c1CC(C)(C)C2 Cc1csc2nc(CC(=O)NCCOCC)cn12.c1(C=O)cc(N)nc(Cl)c1.N c1(C(=O)NCC2C(NC(C#CC(C)C)=O)C2)cnc2ccc(F)cn12 C1(NC(CC2CC(=C)C2)=O)CCCC1NC(=O)C=C(Cl)Cl c1(C(N2CC(=C(CNC(c3c[nH]cc3Br)=O)F)C2)=O)cccc(C2CC2)n1 N1(C(c2c(OC)scc2)=O)CCCOC(CNC(=O)C=Cc2ccccc2C)C1 C1(CNC(CCc2nc(C)sc2)=O)CC2CN(C(C3C(C)(C)C3(C)C)=O)CC12 N1(C(C(CC)O)=O)CC(CNC(C2CN(C3CCN(C)CC3)C2)=O)C2(CCC2)C1 N#Cc1ccc(C(=O)NC2CC2CNC(C2COCCOC2)=O)nc1 Nc1ccc(NC(C2(C3CCCCO3)CCOCC2)=O)cc1[N+](=O)[O-] CCC1=NOC(CNC(C2(C)CCCN2C(c2cc(Cl)n[nH]2)=O)=O)C1 Cc1cc2c(C(=O)NC(C)(CNC(=O)COCC(F)F)CO)cccc2[nH]1 C1(C(C(=O)N(C(c2onc(C)n2)C)C)C)CCN(C(C2CCN(C)C2)=O)CC1 C1(CC(N2CCC2C2CCCCC2)=O)CCCN(C(c2sccc2Cl)=O)C1 C1(C2CC2)CCN(C(=O)C)C1.C1(C(=O)N)(CC)CC(C)(C)C1.CCC(C)C c1(C(N2CCC3C2C3)=O)cc(O)ccc1[N+](=O)[O-].c1(CC)cnoc1C(=O)N.C C(=O)(C1=C(Cl)CCOC1)N.C(=O)(C(F)C(C)C)N(CC)Cc1cnn(C)c1 Cc1cc(C(N2CCOC(CNC(C3C(F)(F)C34CC4)=O)C2)=O)nc(C)c1 N1(C(C=COCC)=O)CCCN(C(=O)CCC[N+](=O)[O-])CC1C C1(C(=O)N)CCCCCC1.C12(C=O)C=CC(CC1)C2.CC(O)(C1CC1)C1CC1 C(=O)(C(C)C(F)(F)F)NC(CC1CN(C(c2c(C)coc2C)=O)C1)C C1(C2CN(C(=O)CC3COCC3(C)C)C2)(NC(CCN(C(CCC)C)C)=O)CC1 Nc1cc(F)cnc1C(N1CC(O)CC1C(=O)NC(CO)CCO)=O c1(C(N(CC)CC)=O)cc(S(N)(=O)=O)cs1.C(=O)CC(C)C.C(N)=O O(N1CCC(CC(=O)NC2CCCC2)CC1)CC.C1(C(=O)NC)CC1C1CCCC1 C1(C(=O)NCC(COC)NC(=O)C(C)(O)C2CCC2)(N(C)C)CCCCC1 c1(C(=O)O)cc(CNC(C2(c3noc(C4CCC4)n3)CC2)=O)cc(F)c1 C=C(Cl)CC(C(=O)NC1CC2(C1)CN(C)C2)NC(=O)C(C)=C1CC1 Fc1cc(-c2ccc(Cl)cc2Cl)ccc1OC(F)(F)F C1CN(C(C2CC(=C3CC3)C2)=O)CC12CC2.n1(C(CC)C)ncc(C(=O)N)c1C CCCCC(F)C(=O)N(C(c1cccs1)C)Cc1ccc(F)cc1 C1(CNC(C(C)(C)C2CCCC2)=O)(CO)CCN(C(=O)C(c2ccccc2)O)C1 c1(OC)ccc(C(CSc2ccc(NC(C3(C)CNC3)=O)cc2)N(C)C)cc1 Cc1[nH]nc(C(=O)NCCNC(=O)C(O)C2CCCC2)c1I O(NC(=O)CNC(=O)CC1CCC1)CCC#C.N1(CCC(=O)N)CCOC1=O C#CCC(C)C(=O)N1CCN(C2CCN(C(c3cc(CC)on3)=O)C2)CC1 N#Cc1cc2c([nH]c1=NCC(C1CC1)Oc1cc(O)ccc1O)CCCC2=O C1(NC(C(C)Cc2ccccn2)=O)CCN(Cc2nccs2)CC(C)(C)C1 c1(C(c2ncnn2C(C)(C)C)NC(CCC)C2CCC2)nnnn1CCCSC C#CCCC(O)C(=O)N1CCC(CF)(NC(c2ccc(Cl)cc2Cl)=O)C1 C(C1CN(C(=O)C2=CCCC2)CC1C(N1CC(CS(C)=O)C1)=O)=CC N(C1C(=O)Nc2cccc(Cl)c21)C(c1n[nH]c(C(C)C)c1[N+](=O)[O-])=O C1(C(N(CC(C)NC(C(c2cccc(Cl)c2)SC)=O)C)=O)CCS(=O)CC1 CC1=C(C(=O)N2CCC(C3CC3)C2)CCS1(=O)=O.C(=O)CNS(C)(=O)=O c1(C(N(CC(CN(C(=O)CC2CSCCS2)C)O)C)=O)ccnn1CCF C1(C(=O)NC(C)CN(C(=O)C(C)OCC(F)(F)F)C)CC2CC2C1 C(=O)(CCC1=CCCCC1)NCCN(C(c1c(N)ccc(NC(C)=O)c1)=O)C c1(CC)nc(O)c(C(=O)NC2CCN(C(C3CCCCS3)=O)CC2F)cc1C N1(C(C(C(C)C)OCC(C)C)=O)CC2CCCCC2C1.C1(CC=O)CC1(Cl)Cl.N O=C(C#CC1CCC1)NCC(=O)NCC(=O)NCCc1ccncc1 c1(C(N2CC(CC(N3CCC(O)(CC)CC3)=O)C(C)C2)=O)cc2ncccc2[nH]1 S(=O)(=O)(c1ccc(Br)cc1NC(c1cccs1)CC)N1CC(CCC)OCC1.CCC c1(CN2CCC(CNC(N3CCc4sccc4C3)=O)C2)ccc2c(c1)COCC2 CC(O)C(C)(C)C(=O)NCC1CCN1C(C12CCC(CC1)CO2)=O Cc1ncncc1C(=O)NCC(C)N(C(=O)CN1CCCCC1=O)C N1(C(C2ON=C(C)C2)=O)CCN(C(=O)Cc2ccc(O)cn2)CC1C(C)C c1(C=O)c(C)cccc1F.C(CCC(=O)NC(C1CC1)C)NC(=O)OCC Cc1cc(F)ccc1CC(=O)NCC1CC1NC(C1CC(N(C)C)C1)=O C12(CNC(CNC(CC)=O)=O)CC1CN(C(c1[nH]ccc1C1CC1)=O)C2 c1(C=O)cc[nH]c(=N)c1[N+](=O)[O-].C(C(=O)N(C)CC1(C)CC1)N(CCC)C c1(C(=O)NC2CC(n3cc(C(COC)(C)O)nn3)C2)ccc2c(C)noc2c1 O=C1COc2ccc(NC(C3CN(C(c4ccncc4)=O)C3)=O)cc2N1 CC1COCCN1C(c1cnn(CCNC(=O)Cn2ncnn2)c1)=O N1(C(COc2c(CC)cccc2)=O)CCCCCC(NC(=O)C2CC2)C1 C(C(CC(C)C)C(=O)N1CCCC(C(C)C(=O)NCCNC2CC2)C1)OC.C c1(OC)ccccc1Nc1ccc(CNC(=O)CCN2CCOCC2C)cc1 C1(NC(c2c[nH]nc2Br)=O)CCCN(C(c2cc(C3CCOCC3)no2)=O)C1 C1(NC(CCCCN(C)C(c2cccnc2N(C)C)=O)=O)CC12CCCCCC2 N1(C(C(CSC)O)=O)CCC2CN(C(c3ncoc3C3CCC3)=O)CC2CC1 C1(C(N2CCOC(CCCNC(c3sccc3F)=O)C2)=O)(OC)CCC(C)C1 c1(C(N(C(C)CNC(=O)C(O)C2CC2)C)=O)ccc(-n2[nH]c(O)nc2=O)cc1 N#Cc1ccsc1C(N1CCCC1C(=O)NC1CC2C=CC1C2)=O n1(CC(C2CC2)OC)c(N(C2CC(C)(C)C2)C(C)C)nnc1COC c1(C(=O)NC(CC)CNC(c2cc(=O)cc[nH]2)=O)cnn2c1N(C)CC2 C(=O)(C(CN(C)C)C(C)C)N1CCC(NC(c2c(C)cno2)=O)(CF)C1 C(=O)(C(C(C)(C)C)N(C)C)N1CC(O)(CNC(C(F)OC)=O)C1 C(=O)(C(F)(F)C1=CCOCC1)N1CCC(F)(CNC(C(C(C)C)O)=O)C1 C1(CNC(C(C)OCC)=O)(OC)CCN(C(=O)C(C)=CC2CC2)CC1 C1(NC(c2cc(C)c(F)cc2)=O)CCCC12CCN(C(c1cnc(S)nc1)=O)C2 C1(C(=O)NCCCC(C)(C)NC(=O)Cc2cc(Cl)ccc2Cl)CCC2(CC1)CC2 CC1=CCCN(C(=O)C(O)C2CN(C(C3(C)CCNC3=O)=O)C2)C1 CCCCC(F)C(=O)NCc1ncc(C(=O)NC2CC=C(C)CC2)cn1 N1(C(C23CCC(OC)(CC2)C3)=O)CCCC2CN(C(=O)CC3COC(=O)N3)CC12 c1(C(=O)NC2C3CN(C(c4c(C)cnnc4)=O)C2CC3)cc([N+](=O)[O-])oc1C N1(C(C(C=C)(C)CC)=O)Cc2ccc(CNC(=O)CC3CCC(=O)NC3)cc2C1 CC1(C)CC(CNC(=O)C=Cc2ccc(F)cc2)N(C(C2CC2C)=O)C1 N1(C(C2CCC(CC)O2)=O)CCC2(C(=O)NC3C=C(C)CCC3)CCCC12 N1(C(CC2CCC(C)CO2)=O)CC2CCOC2(CNC(=O)Cc2cc[nH]n2)C1 CCCCCCCN1CCC(N(C(=O)Cc2nc(C)sc2C)C)C1 C1(O)(CCNC(=O)CC(F)F)CCCN(C(C2CCCCCC2)=O)C1 CCC(C)(CO)C(=O)N1CC(CNC(=O)Cc2ccccc2)C1.[SH](C)(=O)=O C1(CNC(c2cc(O)c(Br)c(O)c2)=O)CC(c2ccc3c(c2)CCO3)=NO1 C(CCCCCNC(=O)CC1(CSC)CC1)N(C(C1C(OC)C1)=O)C c1(Oc2ccc(NC(C34CCC(CN3)C4)C)cc2)ccc(C#N)cc1[N+](=O)[O-] c1(C(N(CC(CC)NC(=O)C(C)NC=O)CC)=O)ccc2nccnc2n1.O O=C1COC2(CCN(C(CC3CCOC3)C(=O)NC3CC(F)(F)C3)CC2)N1 C1(NC(C(C2CCCCC2)C)=O)CCCN(C(=O)CC2(CO)CC2)CC1 C(C(=O)NC1CCOC1)(C(C(C)C)C(C)C)NCc1cn(CC)c(=O)nc1O C1(C(=O)Nc2cnc(OC)c(C)c2)CN(C(=O)Cc2nocc2C)C2(CCC2)C1 C(CCC(CO)NC(C1CC(C)(C)CO1)=O)NC(CCOC(C)C)=O C1(C(=O)NC2C(OCC)CCC2)C2CC2CN1C(C1CC(=O)C1(C)C)=O C1(CNC(c2ccoc2Br)=O)CN(C(c2cncnc2)=O)C2(CCOCC2)C1 C#Cc1cncc(C(=O)NCC(CC)NC(c2scnc2C(C)(C)C)=O)c1 C1(NC(=O)C(F)=CCCF)CN(C(c2ncoc2C2CC2)=O)CCC12CCC2 C(=O)(C1c2ccccc2C(=O)OC1(C)C)Nc1c(C)c(-n2cnnn2)ccc1 C1(NC(C(c2ccoc2)NC(=O)CCn2ccnc2)=O)COCCOC1 c1(C(N2CCN(C(C3(O)CCCC3)=O)CC(CO)C2)=O)cc2cccnn2n1 C1(CC(=O)NC(C2CCCC2)C)COCCN1C(c1ccc(CF)cc1)=O C(C(CC(F)(F)F)NC(c1cccc(Cl)c1O)=O)NC(c1cc(C)no1)=O c1(C(N(CCNC(c2c(C)[nH]c(C(C)(C)C)c2)=O)C)=O)ccn2ccccc12 N1(C(COCCOC)=O)CC2CCC(C2)C1.c1(C=O)c([N+](=O)[O-])cnn1C.C C(C(C)(C)C(C)O)NC(C1(C)CN(C(c2cnc(C)o2)=O)C1)=O C12(CNC(C(C)CO)=O)CCC(CC1)N(C(c1cnn(C)c1C1CC1)=O)C2 C1(C(=O)NC(COC)(C)C2CC2)(CNC(=O)C(OC)O)CCCCC1 c1(OC)cccc2[nH]c(C(N3CC4CC3CCN4C(=O)C(O)C(C)C)=O)cc12 CC(C)(C#Cc1cn(Cc2ncon2)nn1)NC(C1(F)CCOC1)=O C12CC(CCO1)N(C(C1CC1C(F)F)=O)C2.O=C(C(F)CC1CCC1)NC C1(CNC(Cc2cc(C)sc2)=O)CCC2(CN(C(=O)Cc3cc[nH]c3)C2)O1 C1(C(=O)NC2(CNC(c3c(F)ccnc3F)=O)CCCC2)CC12CCSCC2 C(CCCC(C)(F)F)NC(C(C1CN(C(C2CC(OC)(OC)C2)=O)C1)O)=O C1(C(=O)NCC(C(N2CC3CC3(CO)C2)=O)OC)(CC)CCNC1=O CCC(C)(C)C(O)C(=O)N1CCC(C2CCCN2C(=O)Cc2ncc(Cl)s2)CC1 C1(C(=O)NC23CCC(n4cc(C(CC)O)nn4)(CC2)C3)CCc2ccccc2N1 C1(Cn2cc(C(C)(C)NC(C)C)nn2)CCN(C(C2CC2C(F)F)=O)CC1 C1(C(N(C2CN(C(c3c(SC(C)C)cccc3)=O)C2)C)=O)COCC(C)(C)O1 c1(C(=O)NCC(CN(C(=O)CC2CCCC2)C)O)ccc(F)c(Cl)c1F C(C(C)CC(=O)NC(C)(C)CCCNC(C1(COC)CCCC1)=O)OC c1(N2CCC(C)C(NC(c3ncc(Cl)s3)=O)C2)ncnc2cc(F)c(F)cc12 CC(CC(=O)NC1C=CC(C(=O)NC(CO)C(N)=O)C1)N(C)C c1(C(=O)NCC2C(C(=O)NCC=C=C)CCCC2)nnc(O)nc1O CCCCC(C(=O)N(C(C)C(N)=O)C)NC(=O)CCC c1(C(=O)NC(CC)CN(C)C(c2cc(CO)on2)=O)cc(C2CC2)ncn1 C1(OC)CN2CCCC2(C(=O)NCC=CCNC(=O)CCc2cn[nH]c2)C1 Cc1cccc2c(C(=O)NC3CCN(CCCNC(=O)C(O)C4CC4)C3)c[nH]c12 CC1CCC(NC(CS(=O)(=O)N2CCC(N(C(c3cnsn3)=O)C)C2)=O)CC1 C1(NC(C2=NOC(C)C2C)=O)CCC2(CCN(C(C3CCC3C(C)(C)C)=O)C2)C1 CCS(=O)(=O)CC(=O)N1CC(N(C(=O)Cc2ccc(Cl)c(F)c2)C)C(O)C1.CO c1(CC)onc(C(=O)NC(C)(C)C(=O)NC(C)CC2(O)CCC2)c1C C1(C(C)NC(C2(CO)COC2)=O)CN(C(c2ncccc2O)=O)CCO1 C(C)(C)(C(C)CC(=O)NC(C(C)C)C1CCC1)NC(c1cn(CCC)nc1)=O C1CC2CN(C(=O)Cc3cc(C(F)(F)F)co3)CC12.C(C)(C(=O)N)OCC C(=O)(C1=CCCC1C)NCCC1N(C(C(c2cn(CC)nc2)=O)=O)CCSC1 CC1C(C(N2CC(C(F)(F)F)OCC2C(=O)O)=O)C2CNCC2C(O)C1N=[N+]=[N-] c1(C(=O)NC(CNC(CCCC=C)=O)(C)CO)cc2ccc(OC)cc2nc1C c1(OC)ncc(N(C2CC3(CNC3)C2)C(=O)Cc2ccc(F)cn2)cn1 C(=O)(C(F)CCC(=O)O)N1CCC(CNC(C)=O)C1 C=C=CCCC(=O)N1CCCC1C(C)NC(=O)C(c1ccc(F)cc1)(C)F CC(CCC(=O)N(CCCN(C)C)CCNC(C1CCCCC1O)=O)N(C)C c1(C(=O)NC2CCN(C(CSCC)=O)CC2C)cccc2nccnc12 c1(OC)c(F)cc(F)c(NC2CCCN(C(C3(OC)CC3)=O)C2)c1[N+](=O)[O-] N1(C(C2CC2)=O)CCN(C(=O)C(C)Cc2ccco2)CC1CC(F)F.CCO C1(C(N2CC(C(=O)NCc3cncs3)C2)=O)COC2CCCCC12 C1(NC(C(CC=C)C)=O)CCCCC12CCN(C(=O)C(C1CCOCC1)C)CC2 C1(CC)(CC)CC(NC(=O)C)CN1C(=O)C(C)n1cncn1.CCCC(C)C.O c1(C(N2CCC(C(C)NC(=O)CCc3ncco3)C2)=O)nc[nH]c2nccc1-2 N1(C(Cc2ncc(C)o2)=O)CCN(C(=O)Cc2ccoc2)C2CC12 N1(C(COCCOC)=O)C2CCC1C(C)C2.C(=O)(C(F)(F)c1cccnc1)N c1(OC)ccc(Br)c(F)c1C(N1CCC(N(C)C(C2CC2(C)C)=O)C1)=O N1(C(C(c2cncn2C)N(C)C)=O)CC2CCN(C(=O)C(C)(C)CO)CC2C1 N1(C(CCCC(CC)NC(=O)CCn2cnnn2)=O)CCOCC(C2CC2)C1 CC1CN(C)CC(C(=O)NNC(=O)Nc2ccccc2-c2ccccc2)O1 c1(CC(C=O)C)ccc(C#N)cc1.Cc1conc1C(=O)NCCC1CCC1.N CCC(CC(=O)NC1(CCO)CCCCC1)NC(=O)C(C)c1ccco1 CCCCC(C(=O)N1CCCC1CNC(c1cc(F)cc(F)c1OC)=O)C(C)C c1(C(=O)NCC2(CNC(C3CC3Cl)=O)CCOCC2)cc(Cl)ccc1Cl C1(NC(=O)CCC2CC2)CC2CCC(C1)N2CCc1cccc(Cl)c1Cl CC1CN(Cc2cnc(C3CCCCC3)s2)CCC1(F)CO CC1(NC(=O)CCCNC(N)=O)CCCN(C(C23CCCC2C3)=O)C1 c1(C(=O)NC2C(CNC(C=CC(C)C)=O)C2)ccnn1CC(C)C O=C(N=c1[nH][nH]cc1Br)C1C2CCCC1CN(S(=O)(=O)c1ccc(F)cc1)C2 c1(OCC)cc(C)ccc1CNC(=NCCF)NC1CCC(C)(C)CC1 Cc1cc(C(=O)NC)c(C)n1-c1ncccn1.C1(C(N2CCC2)=O)CCC1(F)F C12(NC(COCc3c(C)cccc3)=O)CCN(C(c3ncccc3Cl)=O)CC1C2 Cc1nn[nH]c1C(=O)N(CCNC(C1CCC(=O)C1)=O)CC1CC1 N(C(=NCCn1cc([N+](=O)[O-])cn1)N(C)CC(=O)NCCOC)C(C=C)C c1(C(N(CCNC(C(CCCC)(C)F)=O)CCOC)=O)sc2ncccc2c1N Cc1cc(N2CCN(c3ccsc3C#N)CC2)nc(N(C)Cc2sccc2C)n1 Cc1nn(CCCNC(c2ccc(C(F)(F)C(F)(F)F)nc2)=O)c(C)c1Cl C(C(C)CC(=O)N1CCC(O)(CNC(=O)C(=Cc2cccnc2)F)C1)OC c1(OC)ccc(C(C)=O)cc1CC(N1CCOCC(NC(=O)C(C)(F)F)C1)=O C(=O)(CCCCCC#N)N1CCCC(CCNC(CC(COC)C)=O)CC1 c1(C(=O)NC2CCCN(C(C=C(CC)CC)=O)C2C)ccnc2cc(C)ccc12 C1CC2CC1CN(C(=O)C(CC)N(C)C)C2.C(C)(C(=O)N)OC(=O)OCC C(=O)(CCCCC1CC1)N(C1CCC(NC(CC2(OC)CCCC2)=O)C1)C C(C(CC(C)C)C(=O)N1CCC(COC)C1C)NC(C(CC)(CO)OC)=O C1(CNC(Cc2cn(CC)nn2)=O)CN(C(C2(C#N)CCCO2)=O)CCO1 C1(C(=O)Nc2c(CC)nn(C)c2)CCCCCN1C(=O)C(C)C1CCC1 C(=O)(C(C)C(=O)OC(C)(C)C)NC(C)CCNC(c1ccns1)=O C1(CNC(=O)Cc2cc(Cl)cs2)CCN(C(=O)CCC2CCCO2)CC1O C1(CCOC)CN(C(=O)Cn2nccc2C)CCN1C(C1C2CCCC12)=O S(=O)(=O)(c1[nH]c(=NCCCCS(C)(=O)=O)ccc1Br)N1CCC(OC)(OC)C1 c1(C(=O)NC2(C)CC(NC(CC3ON=C(C)C3)=O)C2)cc(Br)c([N+](=O)[O-])[nH]1 c1(C(=O)NCC(C)N(C(C2CC3(CC3)C2)=O)CC)cc(Cl)ccn1 C1(NC(C2N(C(CCc3ncn(C)c3)=O)CCC2)=O)CCCC(CO)C1 c1(CCCC(=O)NCCOCCN(C)C(C2CCCOCC2)=O)ccccc1Cl C(CCC(=O)NC1(C(=O)NC2CCC(C)C2)CC1)OCC=C CC1CCCN(C(=O)OC(C)(C)C)C1C(=O)Nc1ccc(C2CCNCC2)o1 c1(C(N2CCCC(C)C2CN=c2[nH]cnc(Cl)c2F)=O)n[nH]c2c1CCCCC2 N1(C(CCCNCCNC(C)=O)=O)CCC(c2ccccc2)C1c1cccnc1 C1(C(C)CO)CCN(C(=O)CC2(NC(C3CCSC3)=O)CC2)CC1 N1(C(c2nn(CC)c(O)c2)=O)CC2(C1)CN(C(=O)CCCCC(F)F)CC2CO Cc1sc(Br)c(C(=O)NC(C)CNC(c2c(C3CC3)cnn2C)=O)c1C c12ncnc(c1C)Oc1ccccc1C1CCN2C1.C(C)(=O)OCC C(=O)(CCCCCCC)N1C(C(C(=O)NC(CC=C)C2CC2)(C)C)CCC1 c1(CC(=O)N(CCNC(=O)C(C)CC(C)C)CC)c(C)[nH]c2ccccc12 C=C(Cl)CCC(=O)N(C1CCN(C(C2OC3CCC2C3)=O)CC1)CC1CC1 N1(C(C(COC)COC)=O)CCC2CCCC12C(=O)N(C1CC2(CCC2)C1)C C12(NC(C(CC)C(C)C)=O)CCCC1N(C(=O)CCC1CCCN1C)CCC2 N1(C(C2CCn3ccnc3C2)=O)CCCC(S(=O)(=O)N(Cc2ccccc2)CC)C1 O=C(CCCCC(F)F)NCC1(O)CCN(C(=O)C(F)CC2CCCC2)CC1 c1(OC2CCN(C(C3(C)CCCN3C(=O)CN)=O)CC2)ccc(F)c(F)c1F C1(CNC(C2(C3N(C(C(CSC)O)=O)CCC3)CC2)=O)CC12CCCCC2 N1(C(C)=O)CCCCC2(CCN(C(=O)CC3CCCCCC3(F)F)C2)C1 N1C(=O)CCC1CC=O.C1(O)(C(C)(C)C)CN(C(=O)C(F)=CC2CC2)C1.C C(=O)(CCCCC(F)(F)F)N1CC(C)CC(NC(C2CCN(CCC)CC2)=O)C1 c1(SC)cc(C)ccc1C(=O)NC(C1CCCC1)C.C1(CC=O)CC=CC1.N c1(C=O)cc(C)cc(C)n1.C1(OC)(C)CN(C(C2COCC2C(N)=O)=O)C1 CCC(C)(O)C(=O)NC1CCC(NC(=O)C(CCSC)NC(N)=O)CC1 C1(CC=C)(NC(c2cc(OC)no2)=O)CCN(C(C2C3(CC3)C23CC3)=O)C1 C1(CNC(=O)CC2C=CCCC2)CCN(C(c2ccnnc2)=O)C12CC2 C1(OCC)CCN(C(=O)C(=O)NC(c2ccccc2Nc2ccccc2)C)CC1 N1(C(C2(C)CCOCC2)=O)CCC2C(NC(c3cc(Cl)cs3)=O)CC12 C(C(C)CC(=O)N(C1CCN(C(=O)C(C)CC2CCCCC2)CC1)C)OC Cc1ccc(F)c(CNC(C23CC(CO)(CN2C(=O)C2=CCCC2)C3)=O)c1 C1(CC(=O)NCCNC(c2cn(C)nc2)=O)CC2C=CC1CC2 Cc1nccnc1C(N1CCC(N(C(=O)CCNC(C2CCOCC2)=O)C)C1)=O c1(C(N2CC3C(CN(C(C(CCC)OC)=O)C)C3C2)=O)ccc(C)c2c1CCC2 C1(NC(CCN(C)CCO)=O)CCN(C(=O)Cc2nncn2C(C)C)CC1O c1(C(N(C2CC(NC(C(c3cncnc3)C)=O)C2)C)=O)ccc2cn(C)nc2c1 c1(C(=O)NCCN(CCC)CCOCCn2cncn2)cc[n+]([O-])cc1 N1(C(CCN(CC)CC)=O)CC(C(N2CC(N(C)C)C(O)C2)=O)CCC1(C)C CC1CC(=O)NCC1C(=O)NC12CCOC(CNC(C3CC3F)=O)(C1)C2 C1(CC)CN(C(=O)CCOC)CCC1.c1(C=O)cnn(C(C)C)c1C.C1CC1 c1(SC(C)C(=O)NCCC2CCCN2C(=O)C=CC2(C)COC2)ccccc1 C1(NC(C(c2cn(C)nn2)NC(c2c(C)nc(C)o2)=O)=O)CCC(C#N)CC1 N1(C(C2CCN(C(c3c(C)[nH]cc3)=O)C2C)=O)CC2(CC(N(C)C)C2)C1 Cc1ccc(F)c(C(=O)NCCNC(c2ccccc2N2CCCC2=O)=O)c1F C1(C(=O)NCC(COCC)O)CCN(C(c2ccccn2)=O)CC1(C)C Cc1cc(C(N2CCSC(C(=O)NCC3CCCN3C)C2)=O)cnc1F C1(C(=O)NCCOCCCN(C(=O)Cc2nncn2C)C)OCC2CCCC1C2 C1(C(N2CC(C)(CF)C2)=O)CCCC(NC(c2cncc(F)c2)=O)C1 C(C1(O)CCc2ccccc21)NC(=O)C(=O)Nc1cnn(-c2ccc(Cl)cc2)c1 CCC(C)(CNC(=O)C(c1ccccc1)F)NC(=O)CC1CC(C)(C)C1 C1(C(=O)NC)CCCN(C(C2CC2(C)C)=O)C1.C(=O)CC(C1CC1)C1CC1 Cc1cc(C(=O)NCC2CCN(S(=O)(=O)c3ccccc3Br)C2)ncc1[N+](=O)[O-] C1(c2nnnn2CCC2CC2)(NCc2c(C)nc(Br)s2)CCN(C)C(C)C1 C(=O)(CCC(CF)CF)NCC1(C)CCN(C(C2N(C(=O)OC)CCC2)=O)C1 NC(=O)CC(O)C(=O)NCCOCCCNC(=O)CCF c1(C(N2CCC(C)(NC(=O)CCc3nncs3)CC2)=O)cnc2c(c1)NCC2 C1(CC)CN(C(=O)C2=COCCC2)CCC1NC(=O)Cn1ccccc1=O C1(NC(CCSC)=O)CC12CCN(C(c1ncc(F)cc1F)=O)C2 C(=O)(C(CO)C(C)(C)C)N1C(C(NOCCCC(=O)OC)=O)CC(F)C1 O(C1CCCc2ccccc21)CCCNC(=O)NCc1c(C(C)C)c(Cl)ncn1 N1(C(C2(C=C)CCN(C(=O)C(C)C3CCOC3)CC2)=O)CC2CCCC(O)C2C1 CCC(C)(CNC(=O)C(F)=C(C)C)C(=O)N1CC(O)(CO)C1 C12(NC(c3ccc(NCCO)cc3)=O)CCCC1CN(C(=O)CCCF)C2 CC1(C(=O)NC2CCCN(c3nc(CC4CC4)ns3)CC2)CCCS1(=O)=O N1(C(C#CC2(C)COC2)=O)C2CC=C(C(=O)N3CCCC(F)CC3)C1CC2 c1(C(=O)NCC2(OCC)CCC2)cc(Cl)cc(Br)c1N C(CS(=O)(=O)CCNC(c1nnnn1C1COC1)C1CC1C1OCCO1)OC CCCCCC(O)CC(=O)NCCOC1CN(C(C2(F)CCS(=O)(=O)C2)=O)C1 N1(C(CC2N(C)C(=O)CC2)=O)CCn2nc(CNC(=O)C(F)(F)CO)cc2C1 N1(CC2(C(=O)O)CCCOC2)CCc2cc(O)ccc2C1 CC(C)CC(C(=O)N1CC(C)(C)C1)ONC(=O)C(C)C1CCOCC1 C1(NC(CCC=CC)=O)CCCCC12CCN(C(c1ccc(N)c(O)c1)=O)C2 c1(CCC(=O)NCC(CNC(C(CC)O)=O)OC)nc2cccc(C)c2[nH]1 C1(C(N(C2CN(C(C3CC3)=O)C2)C)=O)CC(O)C1.C(C)(C)C.C(=O)N C(=O)(CC(C)C(F)F)NCC1(C)N(C(C(n2ncc(C)c2)C)=O)CCC1 Cc1ccc2c(C(=O)N(C3CCOC3C)Cc3ccco3)onc2c1 c1(NC(C2(C)N(Cc3c(OC)c(F)ccc3)CCC2)=O)cc(Br)ccc1[N+](=O)[O-] C1(CNC(c2cnn[nH]2)=O)CC(F)(F)CN1C(=O)C(C1CCCCCC1)O C(=O)(CC(C)NC(c1cocc1C(N)=O)=O)NC1C(CC)C1 c1(C(N2CCC(NC(c3ccc(F)o3)=O)C(F)C2)=O)c(Cl)ccc2c[nH]nc12 C=C=CCCC(=O)NC1(COC)CN(C(=O)C(C)OC)C1 c1(C(N2C3C(NC(CNC(C)=O)=O)C(C3)C2)=O)cc2ccc(Cl)c(F)c2[nH]1 C1(CCC)CN(C(=O)C=CC(C)CC)CCN1C(=O)CN1C(=O)CNC1=O c1(C(N2CCC(C(CNC(C=CC(CC)C)=O)C)CC2)=O)ncccc1N=[N+]=[N-] c1(-c2nccc(CN3CCC(c4ccc(OC)cc4)C3)c2)c(F)cccc1F C1CC2CCC(C1)N2C(c1c[nH]c(C(F)(F)F)c1)=O.CC(C(=O)NC)C(F)F C=CCC(C)(CC)C(=O)N(C)CCNC(c1csc(Cl)n1)=O Cc1ccnc(CNC(C2CC2C)=O)c1F.c1(C(=O)N)cn(C)c(=O)cn1 C1(C(N2CC3CC3C2)=O)COCCN(Cc2cc(Br)cc(I)c2)C1 N#Cc1ccccc1NC(N1CCOC(CC(N2CC3(CC3)C2)=O)C1)=O C1(C(=O)Nc2sncc2C(=O)O)CCCN(Cc2ccccc2C(F)(F)F)C1 c1(C(=O)NC(c2cn(-c3ccc(F)cc3)nn2)C)nc(Br)ccc1Br C1(C(=O)N)(CNC(C(C)NC(C)=O)=O)CCCC1.C1(C2CC2)CC1.C Cc1ccc(C(=O)NC(c2ccccc2)CNC(=O)C(C)C2CCC2)cc1C#N c1ncoc1C(C)C.C(C(=O)NC)(C1CC1)NC(COCCCOC)=O C#CC1(C(=O)NC(CN(C)C)CO)CCN(C(=O)CC2OCCCO2)C1 c1(C(C)CC(=O)NCC2CC2)ccccc1C(N)=O.C1CC1.C(=O)CO.C C(=O)(CCC(=O)NCCCCNC(c1cc(SC)n(C)n1)=O)NCCC c1(C(=O)NC2C=CCN(C(c3cncs3)=O)C2)[nH]nc2ncnc(O)c12 CCC(C(=O)NCC12CC(CO1)C2)C(C)C.c1(C=O)cn(C)nc1C(C)C c1(C(N(C)CC2N(C(C(C)SCC)=O)CCC2)=O)cc(F)cnc1Cl c1(C(=O)NCC(C2CCCN2C(c2nscc2N)=O)(C)C)cnc(C(F)F)nc1 C1(C(N(C(CNC(CC(C)C2CC2)=O)C)C)=O)CC2(CCCO2)C1 c1(C(N(C2CCCC2)CCCOC)=O)cc2c(C)ccc(C)c2[nH]1 C(=O)(C(C)(O)CCN(C)C)N1CCCC(C(=O)NCc2nc(C)c(C)o2)C1 C(=O)(CC(CC)C(C)C)N1C(C2CC2)CCC1.c1(OCC)cccc(CC=O)n1.N Cc1ccc(O)c(NC(=O)COCCNC(=O)CC2CCOC2(C)C)c1 Cc1cc([N+](=O)[O-])c(C(N2CCCC(C)(CNC(=O)CO)C2)=O)cc1Cl C(CO)(C(=O)Nn1nnc(C)c1C)NC(c1ccc(OC)o1)=O c1(C(N2C(C)(CNC(C3CCC(=O)N3)=O)CCC2)=O)ccc2nccn2n1 N1(CCC(CC)C2CCC2)CCOC(CCOC)C1 C1(C(=O)NCCC(CNC(C2CCC2(F)F)=O)OC)CC(F)(F)CS1 c1(OC)ccncc1-c1cn(CC2CN(C(=O)CCn3ccnc3)CCO2)nn1 S(=O)(=O)(c1cc(C)cnc1)N(CC(C(=O)NC)C)C.c1csc(C(F)F)n1.N Cc1cc(=NC(=O)C(=O)NC)[nH]o1.C1CN(C(C23CC(C2)C(C)O3)=O)CCN1C N1(CC2CC(OCC)C2)CCOC(C(F)(F)F)C1 c1(CN2CCCC(C(C)NC(C3CCC3)=O)C2)cc(Cl)cc(C#N)c1 c1(OC)c(C(=O)NC(CCNC(=O)CCS(C)=O)C(C)C)cnc2c1cnn2C N1(C(CC2(C=C)CN(C(C3CCCCC3CC)=O)C2)=O)CC2CCCC2C1 C1CC2(CCN(C(=O)C(F)(F)C)C2)CO1.c1(CC)onc(C)c1C(=O)NC C12(CNC(CNS(CC)(=O)=O)=O)CC1CN(C(c1csc(Cl)c1Cl)=O)C2 c1(C=O)cc(C(C)C)nc2onc(C)c12.CCS(=O)CC(=O)NCC1CCC1.N CCCC(CNC(c1cccc(OC)c1)=O)C(=O)N(C1CCCC1)CCC Cn1cc2c(n1)CCN(C(C1CC(n3cc(CSC4(O)CCSC4)nn3)C1)=O)C2 C(C1COC(C)(C)O1)=CC(=O)N(CC(C)C)C.N1(C(C)=O)CCCC(C=O)C1 C1(CCC(=O)NCC2CCCN(C(c3cc(Cl)no3)=O)C2)CCCC(=O)N1 Cc1cc(N2CCC(C(N3CCCC(NC(=O)CC(F)(F)F)C3)=O)C2)cc(F)c1 C1(NC(c2c(CC)n(C)nn2)=O)CCCN(C(=O)Cc2ncccc2C)C1CC C12CCC(C1)N(C(C1CC(=O)OC1(C)C)=O)C2.Cc1ccc(CC(=O)NC)cc1 C1(NC(Cc2nc(C(C)OC)sc2)=O)(CO)CCN(C(=O)Cc2ccsn2)C1 c1(C(N2CCOCCC2)=O)cc(C)c(F)c(C)c1.c1(CC)c[nH]cc1C(=O)NC C1(CC(=O)N(CC(C)NC(C2(CC(C)=O)CC2)=O)CC)CC2CCC1O2 N1(C(C23C4C5C6(C)C4C2C6C53)=O)CC(NC(=O)CO)CC12CCCOC2 c1(C(=O)NCC(C)NC(=O)CCN=c2[nH]ccs2)cc2cc([N+](=O)[O-])ccc2[nH]1 CCC(CC)C(C)C(=O)N1CC2CC(NC(c3cnc(S)n3C)=O)C1C2 CCC(C)CCNC(=O)N(C)C(c1ccccc1)C C(=O)(C1CCCn2nccc21)N1CC(CNC(Cc2cc(C)nn2C)=O)C(C)C1 Cc1nc2cc(C(=O)NC(C)CCN(C(=O)CC(C)O)C)ccc2n(C)c1=O C(C(C)(C)CN=[N+]=[N-])NC(c1scc(CNC(c2c(CC)cno2)=O)c1)=O C1(C)CCN(C)C1.C1(C(=O)OC)(C(=O)NCC(=O)NCC(=O)N)CC1 c1(C(N2CCC(F)(CNC(C3CNC(=O)O3)=O)CC2)=O)ccc2c(c1)COC2 C1(C(N2CCCCC2)=O)CCCCC12CC2.C(CC(=O)NC)NC(=O)OCC Cc1c[nH]cc(Br)c1=NC(=O)C1=CCCN(Cc2ccc(Br)nc2Br)C1 N1(C(c2nc(OCC)oc2)=O)CCN(C(=O)C(C)(C)CCF)C2(CCC2)C1 CC1CC(NC(c2cc(C3CCCC3)nn2C)=O)CN1C(=O)CC1CCOCC1 C(c1ccc(F)c(F)c1)=CC(=O)NCCCC.c1(C=O)c[nH]nc1.C(C)C.N CN=c1cc(C(=O)N(CC(C)NC(=O)CCCCc2ccc(F)cc2)C)cc[nH]1 N1(C(C2(OC)CCCC2)=O)CC2CCC1CN2C(c1cn(CCN(C)C)nn1)=O c1(C(N2CC(CNC(C3NC(=O)OC3)=O)OCC2)=O)ncc2[nH]ncc2n1 CC1(O)CCCN(C(=O)NCC23CC(C2)C3)CC1 C(N=c1nc(O)c(Br)c[nH]1)C1(C)CCN(C(c2cc(S(N)(=O)=O)co2)=O)CC1 N1(C(CSc2cn(C)nc2)=O)CC2CC(NC(=O)Cc3cc(O)nc(O)n3)C2C1 CC(O)C(F)(F)C(=O)NCC=C1CCN(C(C2(c3cccs3)CCCC2)=O)CC1 C(=O)(CCCC=O)N.C(CCC(=O)NCC1CCCC1)NC(C)=O.C(C)(C)C N1(C(c2ccc(C#C)cn2)=O)CCOCC(F)(CNC(C2(C)CCSCC2)=O)C1 C#Cc1ccc(C(=O)NC(C2CN(C(=O)C(=O)NCC)CCO2)C)cc1Cl N1(c2snc(C)n2)C2CCC1CC(NC(C1(F)CCOC1C)=O)C2 N1(C(C(C2CCOC2)OC)=O)C2CCCC1CC(NC(c1c[nH]c(=O)cn1)=O)C2 N1(C(c2n(CC)ccn2)=O)CC(NC(=O)CCC(=O)c2ccccn2)CCC1C c1(NCc2scc(C)c2)ccc(C(=O)O)cc1S(=O)(=O)N1CCSC2CCCC12 C1(C(=O)NC(C(C)C)CCNC(=O)C(C)(C)C2CCCO2)CCC2(CC1)N=N2 c1(C(=O)Nc2ncc(C(=O)OC)c(C)n2)noc2c1CN(C(=O)O)CC2.C1CC1 C1(C(N2CCC2)=O)CC2(C1)CC2F.C1(CCCC)(C(=O)NCCO)CCCC1 C1(NC(C(C(C)C)F)=O)CCC12CCCN(C(=O)Cc1n[nH]c3ccccc13)C2 C(=O)(C1=C(CC)OCCC1)NCCC(C)(CC)NC(CC(CCC)C)=O C(=O)(C1=NOC2COCC12)NC(C(C)C)(C)CNC(c1cc(CCCO)on1)=O c1(C(N2CCC(CNC(c3ccns3)=O)C2)=O)cncc(N2CCCC2)n1 C1(NC(CCCc2c(C)ccs2)=O)CCN(C(=O)C(C)CF)CC12CCC2 N1(C(CCCCCCC)=O)CC2CN(C(c3cccc(Cl)c3)=O)CCC2(CO)C1 c1(CC(=O)N(C2CN(C(COCCCOC)=O)C2)C)csc(C)c1 Cn1ccc(OCC(=O)NC(Cc2cn(CC3CCOCC3)nn2)C(=O)O)n1 c1(C(=O)NC2C(C)CCN(c3nccnc3C#N)C2)noc2c1CCCCC2 [N-]=[N+]=NC1(C(=O)NC2CCC(c3ccccc3)C2)CC1 CCC(CNC(=O)C(Cc1cn[nH]c1)NC(C1CCC2CC12)=O)C(C)(F)F c1(C(=O)NC2C(NC(C=CC(CC)C)=O)CCC2)cccc2scnc12 c1(NC(=O)NC2CCN(Cc3onc(N(C)C)n3)CC2)ccc(F)cc1F C1(C(=O)NCCCCN(C(c2ccc(CC(C)C)cc2)=O)C)OCCOC1(C)C Cc1oncc1S(=O)(=O)NC1CCN(C(C2CC2C2CC2)=O)C1 C1(C(=O)NCC(C)(C2CC2)NC(C2N(C)CCOC2)=O)CC1C1CCCCC1 c1(C2(NC(C3CC(O)CN3)=O)CC2)cccc(-c2ccc(O)cc2)c1 Cc1nn(C)c2c(NCCc3cccc(Cl)c3F)nc(=NCC3CCSC3)[nH]c12 N1(C(C(C=C)c2ccccc2)=O)CC2CN(C(C3CCC4(C3)N=N4)=O)CC2C1 c1(C(=O)NC2CC3(C(NC(C=C(C)c4cccs4)=O)C3)C2)c(C)cc(O)nc1C N1(C(C=COCC)=O)CCN(C(c2cc(Cl)ncc2O)=O)C(CC(F)F)C1 CC(C)CC(CC(=O)NC1CCCCN(C(c2ccc(O)nn2)=O)C1)CC(N)=O C(=O)(CS(=O)CCC(F)(F)F)N1CC(NC(c2cc(C3CCC3)on2)=O)C(O)C1 N1(C(C(CCC)C)=O)CC(CO)C2(C1)CN(C(=O)Cc1ccccc1COC)C2 C1(CC=O)COC2(CCC2)CO1.c1(CC)ncc(C(=O)NC(C)CCOC)[nH]1 Cc1cnc(C)c(C(N2CC3CC3(CNC(c3ncc(F)cc3N)=O)C2)=O)c1 C1CN(C)CCN1C(C1C2CC3C(C2=O)C13)=O.CC1CC1C1CC1C(=O)N.C c1(COC)nc(NCc2ccn(C(F)F)n2)cc(N2CCOC(CCO)C2)n1 C(=O)(C(F)C(=O)NC1(c2nccs2)CCC1)OCC c1(C(N2CCC(OCCNC(CCc3scc(C)n3)=O)C2)=O)[nH]cnc1C#N CC1CN(C(=O)C2=CCN(C(C3(C)CC3(F)F)=O)C2)CCN(C)C1 c1(C(=O)NC(CNC(c2c(C)nns2)=O)(C)C)ccc(Cl)cc1F Cc1cccc2c1OCCC2NC(=NCC1CC1)NCC1(F)CCOC1 Cc1cccc(C)c1CNCC(=O)Nc1ncc(CC2CC2)s1 C1(NC(CCCC)=O)CC(NCCOC(C2CCC2)=O)C12CCC2 CCC(C)(C(=O)N(C1CCN(C(c2ccc(Cl)o2)=O)CC1)CC(C)C)OC c1(NC(c2scc(C)c2C)=O)c(-c2cc3c[nH]nc3cc2C)ccc2c1OCO2 C1(C(N(C2CCN(C(=O)CCn3cccc3)C2)CC2CC2)=O)CCCC(=O)N1 C1(NC(C2N(C(C(CCC)F)=O)C(C)CC2)=O)CCn2cncc2C1 C1(CNC(=O)CO)CC(NC(=O)C(O)C2CCCC2)C(O)C1 N1(C(=O)Cn2cccn2)CCC(C(N2CCC23CCC3)=O)(CF)C1 C1(CNC(=O)C(F)CC2CC2)CCCCCN1C(=O)Cc1ccc(Br)cc1 C12(C(=O)Nc3cccc(-c4cn(CC)nn4)c3)CCCC1N(CC)CCC2.C(C)=O C(c1ccc(O)cc1Cl)=CC(N1CCNC(C(=O)NCC23CCN(CC2)C3)C1)=O C(=O)(n1ccc2c1CN(N1CC(O)CC(O)C1)CC2)OC C1(C(=O)NCC2(CO)CCOCC2)C2CC(C(O)C2O)S1(=O)=O C1(C)(C(N2CCC(NC(c3c(C)nsc3N)=O)C(CO)C2)=O)CCCNS1(=O)=O c1(C(=O)NC(CNC(c2nc(C)sc2)=O)(C)C)cc(=O)c2cc(O)ccc2o1 C1(CNC(C(CCC)C)=O)CCCCN(C(c2cc(N)nc(Cl)c2)=O)C1 O=C1CC2(CCC2)C(C(N2CC3(CCC3NC(=O)C3=NOCC3)C2)=O)CN1 CC(C)(C)C1CN1.c1ccc(N2CCCCC2)cc1.C(=O)(CCN1CCCC1)OC CC1CCCC(OCC(=O)N(CC(C)(C)C)C)C1.C(=O)C.C1(C=O)CCC1.N CC1(C)CCC(CO)N(C(=O)NCc2c(Br)cccc2Br)C1 CCC(CCCC(=O)N(CC(F)F)C1CC1)NC(=O)CC1CC1(C)C Cc1cccc2c(C(=O)NC34CC(CNC(=O)CCCCC(F)F)(C3)C4)coc12 C1(NC(c2ccn(CC#N)n2)=O)CN(C(C2CCS2(=O)=O)=O)CC12CCC2 N1(C(C(CCC)C)=O)CCCC(C)(NC(=O)Cn2ccc(Br)n2)C1 C(C(C)(C)CC1CN(C(c2ccoc2)=O)C1)NC(C)=O.CC1CC1C=O.C c1(C(C)=O)cc(C(=O)NC(C(=O)NCCC(C)N2CCCC2)C2CCC2)no1 Cc1cn2c(n1)CC(C(N1CCN(C(=O)CC(C)P(C)(C)=O)C(CCO)C1)=O)C2 C1(NC(C2C(C3C(C)C3)C2)=O)CC2CN(C(=O)C#CC(C)(C)C)CC2C1 C1(C(C)NC(CC=C(C)C)=O)CN(C(=O)C(=CC2CCCC2)C)CCO1 C1(CC)C(C(=O)NC2(CCF)CCC2)CCN1C(c1ncncc1C)=O C1(C(N(C2CCN(C(c3sccc3Cl)=O)C2)CCO)=O)CC2CCC1O2 C(=O)(C1=CS(=O)CCC1)NCC(C)NC(C1CC(F)(CO)C1)=O c1(C(N2CCC(N(C(=O)CC)CCC)C2)=O)ccc(C2CCC(=O)N2)cc1 c1(-c2ccc(SC)s2)cnc2c(C(=O)Nc3cccc(C(F)F)c3F)cccn12 c1(C(N2C(CNC(=O)C(F)CC3CCCC3)C=CC2)=O)cc(F)ccc1Br N1(S(CCOCC(=O)OC(C)(C)C)(=O)=O)CCc2n[nH]cc2C1C(=O)O c1(C(=O)NC(CCCNC(c2c(COC)cccc2)=O)C)cc(C)nc(C)n1 c1(-c2cc(C(N(CCCCO)CCCC)=O)ncc2)cnc(O)c(C)c1 CC(CC(=O)N1CCNC(C(=O)Nc2cc(O)nc(Cl)n2)C1)CC(C)(C)C Cc1c[nH]c2ncc(C(=O)N(C)C(c3cn(Cc4cccc(Cl)c4)nn3)C)cc12 C1(C(=O)N)C(C)(C)CCCC1(C)C.C1(NC(c2c(CC)scc2)=O)COCCC1 C(=O)(CC(C)(C)C)N1C(CNC(C(C)OCC#C)=O)CC1 C(C)(CCC(=O)N1CCC(C(O)CNC(c2cccs2)=O)CC1)OCC N#Cc1cn[nH]c1C(N1CCN(C(c2ccsc2C(F)(F)F)=O)CC1)=O C(=O)(C(C)(C)CCSC)NC(CC)(C)CNC(=O)CCc1nc(C)cs1 C1(NC(CN(C)CC)=O)COC2(CCN(C(c3ncncc3OC)=O)C2)C1 N1(C(CC2(N(C(CCN(C(C)=O)C)=O)C)CC2)=O)CCOC(C2CC2)C1 C1(C(N2CCC(C(F)(F)F)C2)=O)CC2(CCOC2)C1.C(=O)(CCC(=O)N)OC C1(C2CCN(C(C3(C)CC3(F)Cl)=O)CC2)(NC(CCSCC(C)C)=O)CC1 C1(C=O)CCCCC(=O)C1.C1CN(C(=O)Cc2csc(C3CC3)n2)C1.COC N1(C(C=C(C)C(C)C)=O)CCCC(C(=O)N(C(C)CO)C)CC1 O=C1CN(C(=O)CCC2CCCC2)CCN1CC(N1CC(O)C1)=O c1(CC(=O)NCC2CN(C(CCC=CC)=O)C(C)C2)ccc(F)cc1Br CCC(CC)C(C)C(=O)NCCCCCNC(=O)C(C)(O)C(C)C C(=O)(C1CCc2cccc(O)c21)NC1CCN(C=O)CC1 S(=O)(=O)(c1ccc(Cl)cc1)N1CC(N(C(=O)C(CO)OCC(=O)O)C)C1 C(C(=O)NCC1(C)CCCN1C(c1ccc(=O)oc1)=O)(C(C)C)OC c1(NC(CSCCC)=O)cccc(CNC(c2[nH]cnc2CC)=O)c1 C(=O)(C1CCCc2nc[nH]c21)N(C)CCNC(=O)Cn1cnc(C(F)(F)F)n1 CC1CN(C(=O)CCC2(C)CN(C(c3cnn[nH]3)=O)C2)CCC1(F)F N1(C(c2nc(-c3c(C)noc3)sc2)=O)CCCC(N(C)C)C1 N1(C(C2CC(=C)C2)=O)CCC2CCN(C(c3cc4cccnn4c3)=O)C2C1 c1(N2CCOCC(C(=O)Nc3ccccc3)C2)ncc2ccccc2n1 CC(C)(O)C(F)(F)C(=O)Nc1cccc(NC(c2c[nH]nc2C2CCOC2)=O)c1 C1(C)(NC(c2n(C)nnc2CNC(=O)C(C)(C)Cl)=O)C(C)(C)C1(C)C N1(C(c2n(CC)nnc2)C(=O)NCCOC)CCC(c2nncn2C)CC1 N1(C(c2ccc(C=C)cc2)=O)CC2CC(O)C1C2NC(c1cc(C)c(F)cn1)=O C1(N(C)C(c2cc(Cl)c(Cl)n2C)=O)CC2CCC(C1)N2C(=O)C1=CCCCCC1 c1(C(=O)NCC(C(C)C)NC(=O)C(C)C#N)ccc(O)nn1 C(c1ccc(O)cc1)=CC(=O)NC(CCOC)CNC(=O)Cc1ccno1 CCC(CCCC(=O)NCC1CCOC(C)(C)C1)NC(c1cccn1C(C)C)=O c1(C(=O)NC2CN(C(C=CCOC)=O)CC(F)C2)n[nH]c2c1CC(C)CC2 N1(C(c2cncc(C)c2)=O)CCCCC(CNC(c2nnn(C)c2C)=O)C1 C1(C(NC)=O)SC2C=CC1CC2.c1(C(N2CC3CC3C2)=O)cc(=N)[nH]c(Cl)n1.C c1(C(=O)NCCCC(C)NC(C2(C)C=CCC2)=O)cc(Cl)nnc1O C1(CCC)(C(=O)NC2(C(=O)O)CCNC2)CCNC1=O CC1(C)CCc2nc(C(=O)NCC3(F)CN(C(C4(C)CCCO4)=O)C3)ccc2C1 c1(C(=O)NCC(CNC(C(C(C)O)N(C)C)=O)C)coc(S(C)(=O)=O)c1 c1(C(=O)NCC(C)CNC(C2CS(=O)(=O)C2)=O)cc2ccc(Br)cc2[nH]1 c1(C(c2n(C(CC)(C)C)nnn2)NCC2COC(C)(C)C2)nc(Br)c(C)cc1F CCC(CCCC(=O)N(C)Cc1nccn1C)NC(=O)C(C)(C)C(N)=O C(=O)(C1CCc2sc(NC(=O)C(=O)N(CC(C)CC)C)nc21)OCC C(=O)(C1CCc2c(Cl)cccc21)NCC1CCN(C(c2nn(C)c(Cl)c2)=O)CC1 c1(NC(c2n(CCSC)nnn2)c2csnn2)ccc2cnc(C)n2c1 N1(C(C(C)NC(COC)=O)=O)CC=CC(NC(=O)Cc2nc(C)sc2Cl)C1 c1(OC)cnnc(C(N2CCCC2CNC(=O)CC2CCC(=O)N2)=O)c1 Cc1ccc(Cl)c(C(N2CCC(OCCNC(C3CCSCC3)=O)C2)=O)c1O c1(C(N2CCOCC2c2ccccc2)C(=O)NCCOCC)cn(C)nc1I C1(NC(=O)C=CCN2CCCC2)CCC(C(=O)NC2COC(C3CC3)C2)C1 N1(C(CC2N(C(C(C)(F)F)=O)CC2)=O)CCOCCC1C(N)=O c1(C2(C(=O)NC3CC(CNC(C4CC4Cl)=O)C3)CC2)ccc(Cl)cc1Cl N1(C(C(=O)NCC(C)=O)C)CCc2ccccc21 Cc1cc(=O)n(CCC(=O)NC2CC2C)cn1.C1(C=O)CCS(=O)(=O)C1.N C1(C(=O)NCCC(C(C)C)C)CN(C)CCN1C(=O)Cc1cnsc1 N1(C(C(C)CCO)=O)CCC(C2(NC(=O)Cc3ccc4ocnc4c3)CC2)C1 N12CCC3C(CCCN3CC1=O)C2.Cc1cc(=NCc2ccccc2)[nH]c(C)n1 CCCCC(C(=O)N1CCC(C(=O)NC2(CCC)CCNC2=O)CC1)C(C)C N1(C(CN(CCCCCC)C)=O)CCCC(F)(CNC(=O)C(C)CCOC)C1 Cc1nc(NC(C2CCCC2NCc2c(Cl)cncc2Cl)=O)ccc1Cl C(N=c1[nH]c2c(F)cccc2o1)C1CCC(NC(C2(F)CC3(CCC3)C2)=O)C1 c1(OCOC)ccc2c(c1CNCCC1CCN(C)CC1)OCO2 c1(CC)c(C(=O)N(C)CCOCCCNC(=O)C(O)CCSC)cccc1F c1(C(N2C(CNC(c3cccc(F)c3F)=O)CC2)=O)ccc2nc[nH]c2c1F c1(NC(C)=O)c(C(N2CCC(F)(C)C2)=O)cccc1C.C(=O)(C1=CCCC1C)N n1(CCC)cc(C(=O)NC(C)(CNC(C2CC(C)=NO2)=O)CO)nn1 C1(C(=O)NC2C(C)(C)N(C(C3CCCN3C3CC3)=O)CC2)CCC(N=[N+]=[N-])CC1 CC1(C)CC2(CO1)CN(c1cc(Br)ccc1S(=O)(=O)N1CCC=C(Br)C1)CCO2 C1(C(=O)NC2C=C(C)CCC2)CN(C(=O)C(=O)N(C)C)CC(C)O1 C=CCC(CC(=O)Nc1cnn(C)c1C(C)C)NC(=O)CN1CC2CC2C1 S(=O)(=O)(c1cc(C(N2CCC(C)CC2)=O)n(C)c1)NC.n1(CC=O)ncnn1 c1(C(N2CCC(N(C)C(C3C=CCCC3)=O)C2)=O)cccc(CF)c1 CC(C(F)C(=O)NCCNC(C1CC2(C1)CC(O)C2)=O)C(F)(F)F c1(C(=O)NC2C(C)CN(C(c3cc(O)ccc3N)=O)CC2)cn2cnnc2cn1 C(=O)(C1CC(=O)c2ccccc21)NCC(C)NC(Cc1c(C)n(C)cn1)=O C1(C(=O)NCc2onc(C)n2)CCN(C(=O)CCc2cn[nH]c2)C1C C1(O)(CC)CCCN(C(c2cc(C(N)=O)co2)=O)C1.C(C=CC=O)(CC)=C.C Cn1cncc(C(=O)NC2CCCC2C)c1=O.C1(CC=O)CCC(C)(O)CC1.N Cc1cc(NC(c2c(C)[nH]c(C(=O)NC(CO)C(C)C)c2C)=O)cc(Br)c1C c1(CC)cc(NC(=O)CC2CC(NC(c3cc(C(C)C)no3)=O)C2)n[nH]1 C1(C2CCC2)(C(N2C(CCNC(CN3CC(CC)C3)=O)CCCC2)=O)CCC1 N1(C(COc2c(OC)cccc2)=O)CCCC(NC(C2CC3(CSC3)C2)=O)C1C N1(C(c2c(C)[nH]nc2Br)=O)CC2CCC2(CCNC(=O)Cc2ccno2)C1 c1(CC)ccc(NC2CCC2SC)cc1S(N)(=O)=O c1(NC(C(CNC(=O)C=CC2(C)COC2)OC)=O)cccc2c1CCC2 C1(C(=O)O)CC2(CCCC2)CCN1CC#Cc1cncs1 N1(C(=O)Nc2cc(C(F)(F)F)cs2)CCCCC1C1(O)COC1 c1(C(N2C(C)CC(CNC(CCNC(C)=O)=O)C2)=O)cccc(F)c1Cl c1(CC)ccc(CC(=O)NC2(CCC)CC2)cc1F.C1(C)(C=O)CC(C)(C)C1 c1(C(=O)OC)ccc(F)c(C(=O)N(c2ccccc2Cl)CCOC)c1C C1(C(N2C(C(N(CCOCC=C)C)=O)CSCC2)=O)CCC=CCCC1 N1(C(Cn2ccnn2)=O)CC(C(F)(F)F)C(S(C)(=O)=O)C1.C1(C(C)C)CC1.C C=CCC(C(=O)NCc1nc(N(C)C)n[nH]1)NC(c1cncn1C)=O c1(C(=O)NC(CCCC)CNC(C2COCCN2C)=O)cc2n(n1)C(C)CCC2 c1(C(=O)NCC(CNC(c2cnn(C)n2)=O)CO)cc2c(cc1O)CCCC2 c1(C(C2CCCCCC2)NC(=O)Cc2cc[nH]n2)ccc(Cl)cc1.C1(CO)CN1 N(C1CSc2ccccc21)C(C12OC(C)C(C1)C2)=O Cn1c(CCNC(c2ccc(C)nc2)=O)noc1=O.C1(CC(=O)N)CSCCO1 c1(C(=O)NC2CCCC(N(C(=O)Cc3cnc[nH]3)C)C2)cnc2ccccc2c1 C1(c2ccccc2)N(Cc2cccnc2N2CCCC2)CCCC1(C)C c1(C(N2CCC(C3CCCO3)C2)=O)cc(S(=O)(=O)Nc2ncccn2)c[nH]1 c1(C(N2C(C)(C(=O)NC3(CC)CCOC3)C=CC2)=O)occ2c1CCC2 N1(C(CCCOC)=O)CCOC(CN(C(=O)Cc2csc(C3CC3)n2)C)C1 CCCN=C(NCC1Cc2ccccc2N(C)C1)N1CCC(C(F)(F)F)(CO)C1 N1(C(C2(C(=O)OCC)CC2)=O)CC=CCC1.C1(C(C(=O)N)O)CCCCCC1 C12(NC(C3C4(CC(OCC)C4)C3)=O)CCC(NC(=O)CC)(CC1)C2 Cc1cc(C)c(C=CC(=O)NC2COCCN(C(=O)C(C)CCO)C2)cc1C CCC(CNC(c1cccn2cncc12)=O)(CC)C(=O)N1CCCC(C)(F)C1 C1(NC(c2ccc(CC)s2)=O)CN(C(=O)C=C(C)C)C2CC12 c1(C(=O)OCCc2nc3ccccc3[nH]2)c(F)c(F)cc(Br)c1F N1(C(c2ccc(C#C)nc2)=O)CC2(CCOCC2)CC1CNC(=O)CC(C)CF N1(C(C(OCC)OCC)=O)CCC(O)C(C(N2CCSC(C)C2)=O)C1 c1(C(=O)OCC)cc(CN2CCC(C(=O)N3CCCCO3)(CC)CC2)ccc1O N1(C(C2C(NC(c3c(CC)ccs3)=O)CCO2)=O)CCC(O)C(CO)C1 C12(C(N3CCC(CCNC(=O)Cn4nccn4)C3)=O)CCCCC(=O)N1CCC2 c1(C(C)(C)C)cc(N2CC(CNC(c3ccc(C(F)(F)F)nc3)=O)C2)ncn1 c1(C=O)nc(C(C)C)oc1C.C1(C(=O)OC)(C(N2CCC2)=O)CC1(F)F.C Cc1ccc(F)cc1N(C)C(C1CCCS1(=N)=O)=O Cc1cnc(C(=O)N(CC(C)O)CCNC(C2CC(C)(C)C2)=O)cc1Br CCCC(CCCNC(=O)CCC(N)=O)NC(C1CC1c1ccccc1CC)=O c1(NC(=O)NCC2C(CN)C2(F)F)cccc(F)c1F.N1(C=O)CCCC1 N1(C(c2ccc(C)s2)=O)CC(CC(=O)N(CCO)CCO)C(C)C1 c1(OC)ccccc1CNC(=O)C(C)=CCNC(=O)CCCCSC C1(CCOC)(NC(c2n[nH]c(C)c2O)=O)CCN(C(c2cnc(O)s2)=O)C1 c1(N(CCNCC(C2CCCCC2)OC)C)cc(NC2(CO)CC2)ncn1 n1(CC=C)c(-c2cccc(OC)c2)nnc1S(=O)(=O)Cc1ccc(Cl)c(F)c1 c1(N2C(CC(=O)OCC)CCC2)ncc2sccc2n1.c12ccc(cc1)[nH]2 O=C(C#CC1CCCO1)NC1CN(C(c2ccc(O)nc2)=O)CC12CC2 N1(C(C(C(CNC(C(CC(C)C)=O)=O)C)F)=O)CCc2ncccc21 CN=c1nc(C(N2CCN(C(C3CCc4c[nH]nc4C3)=O)CC2C)=O)cc(C)[nH]1 c1(NC(COC)C(C)C)nc(N2CC3CC(C2)C3(C)C)c2ccccc2n1 C=CC1(C(=O)NCC2C3CCCC23)CCN(C(c2cnsc2)=O)CC1 c1(C(=O)NCC(CC)NC(=O)CCCn2cccn2)cc2cc(Cl)ccc2o1 Cc1nc(C(=O)N(C)CC2CC(F)CN2C(C23CSCC2C3)=O)cn1C(F)F c1(C(=O)NCCN(C(CCOC)=O)CC(C)O)cc2c(s1)-c1ccccc1OC2 C1(CC(=O)N(C2CCCN(C(=O)Cc3cnccc3C)C2)CC)C(=O)ON=C1C N1(C(Cc2c(C)n[nH]c2)=O)CC(C)(C)CC1CNC(c1cncs1)=O C1CCNC1.N1(C(=O)NC)CC(C=O)C1.C(=O)CC(C)C.C(=O)C.CC.N c1(C(=O)NC(C(=O)NC(CC#C)C(N)=O)CC(=C)Cl)cnn2ccccc12 c1(OCC)ccc(=NC(=O)CC2CN(S(=O)(=O)c3c(C)noc3C)CCO2)[nH]n1 C1(C(N2CCC2(C)C)=O)COC2(C1)CN(C(C1CC3(CSC3)C1)=O)C2.COC c1(CC)nnc(C)cc1C(=O)NC.C1CCN(C(=O)CCc2cnc[nH]2)C1(C)C N1(C(C2CCC(C)C2)=O)CCC2(CC1)CC(NC(=O)Cc1cc(F)ccc1F)C2 Cc1ncc(CC(=O)NC2(C(=O)NCCCS(C)=O)CC(O)C2)s1 N1(C(CC(C)C2CC2)=O)CC2CC1CN2C(=O)C(C)c1ccco1 N1(C(c2c(C)nc[nH]2)=O)CCOCC1CCNC(c1ccncc1Br)=O c1(NC(C(CC)C)=O)cc(C(N2CCCC2c2cc(C)on2)=O)ccc1C N1(C(c2cn(C)nc2)C(=O)NCCCOCC2CC2)CCC(F)(F)C(O)C1 c1(C(=O)NCC2OCC(CNC(=O)CCn3ccnc3)C2)ccc2sccc2c1 c1(N(C2CCN(C(=O)CC3CCCS3(=O)=O)C2)C)nc(Cl)ncc1F c1(CC(=O)NC2CCN(C(c3cc[nH]c3C3CC3)=O)CC2)nc2ncccn2n1 Cn1cc(N)c(C(N2CC(CO)(NC(=O)CCOC3CC3)C2)=O)n1 N1(C(CSCC=C)=O)CC(C)OC(C)(C)C1.c1(CC(=O)N)ccc(Cl)cc1Cl n1(CC(N2CCC(C)C2)=O)cc([N+](=O)[O-])cn1.CC(C=O)OCC(F)(F)F.N N1(C(Cn2c(C)nnn2)=O)CCC(C)C(NC(c2cccn3nnnc23)=O)C1C C(N=c1nc2[nH][nH]cc-2c(O)n1)C1N(C(COCc2cn(C)nc2)=O)CCC1 CC1(NC(c2cc(C(C)(C)C)ccc2O)=O)CCN(C(C2(C3CC3)CC2)=O)CC1 O=C(N=c1nc[nH]s1)NCC1(O)CN(Cc2ccc(OCCO)cc2)C1 c1(OC)cc(OC)c(C(=O)NCC(C)N(C)C(c2nocc2Br)=O)cc1N N=c1ncc(C(N2CCN(CCNC(=O)C(F)(F)CF)CC2)=O)c[nH]1 c1(C(=O)NC2CN(C(c3cc(NC(C)=O)ncc3)=O)CC2C)ccnc(Br)c1Cl CC1(C)C(C)(CN2CCC(C(=O)N3CCCO3)CC2)C1(C)C C=C(Cl)CC(C(=O)N(C1CCCCC1CC)C)NC(=O)C(F)C1CCCC1 Cc1cc(C(=O)N(CCC(C)(C)NC(=O)CCSCC2CCC2)C)nn1C C1(CNC(c2ccc[nH]2)=O)CCN(C(c2nccc3ccsc23)=O)CCC1(F)F N1(C(C(CN(C)C)(F)F)=O)CCC2CC2(NC(C2CC3(CCC3)C2)=O)CC1 CC1CN(C(=O)C=Cc2cncc(O)c2)CCCN1C(C1CCC(C)(C)OC1)=O CC(C)C(F)C(=O)N1CC(C(N)=O)(CNC(c2cccc(O)n2)=O)C1 CC1CN(C(=O)CC2C3CN(C(C4(O)CCOC4)=O)CC23)CC1O C#CCC(O)C(=O)N1CC2C(CNC(c3ccc(-c4ccncc4)s3)=O)C2C1 CC(C)(O)CC(=O)NCc1cccc(C(=O)NC(C(C)(C)CO)C2CC2)n1 c1(CC(=O)NC2C(NC(CC(=O)NCC)=O)COC2)cccnc1OC C(=O)(C(C)(O)C(C)(C)C)N.Cc1cnc(C=CC(=O)N(CC)C(C)C)[nH]1 C(=O)(CCCCCN(C(=O)CC(C)n1cccc1)C)NCC1N(CC)CCCC1 CC1CN(C(=O)Cc2c(F)cccc2F)CC(C)N(C(c2ccco2)=O)C1 c1(NC(C2C=CC(NCc3nc(Br)cs3)C2)=O)ccc2ccnc(O)c2c1 c1(C(N(C(C)C(=O)N(CCC(C)(C)C)C)CCC)=O)ccn(C)c(=O)c1 C(CC(=O)N1CCN(C)CC1)(C(F)F)NC(C(C(C)C)NC(C)=O)=O C(=O)(CC(F)(F)C(F)F)NC1CCCC(NC(c2scc(OC)c2)=O)C1 C(N=c1cccc(S(=O)(=O)NCC2(C)CCCCO2)[nH]1)C1(C(C)C)CC1 c1(CC=C)cccc(C(=O)NCCCOCCNC(=O)C(C)CF)c1 CC(=O)CCCCC(=O)N1CCC(O)(C(C)CNC(=O)COCCF)C1 c1(C(=O)NC2CCN(Cc3cccc(C)n3)CC2F)ccc2sccc2c1O C1(C(=O)NCC(CC(=O)N(CC)CC)O)CCCCC(=O)C1 c1(OC)c(C(N2CC(F)(C(=O)NCC3CCC4(CC4)C3)C2)=O)cnn1C Cc1nn(C(C)C)c(C)c1C(N1CC(CCO)(NC(=O)CC2CCCO2)C1)=O c1(OC)ccc(OC)c(C(c2nnnn2C(C)C)N)c1.C1CCC(C)(C)CC1.C N1(c2ccnc(NCc3cnc(CC)s3)n2)Cc2nccn2CC(C(N)=O)C1 c1(C(N(CCSC)CC)=O)cc(-c2cnc(N(C)C)nc2)cnc1Cl Cc1ccc(NC(=O)C(C(C)O)NC(C2CC2C2(C)COC2)=O)c(C)c1O c1(C(=O)NCC(CC)NC(=O)C(C)OCCOC)c(C)sc2ccccc12 N1(C(CC2ON=C(C)C2)=O)CC(NC(=O)CN(C)C(N)=O)CC1(C)C C1(C(=O)NC(C)CF)CC(O)(CNC(=O)C(CO)N(C)C)C1 c1(N2CCC3CN(C(c4n(C)ncn4)=O)CC32)ncnc2c1cc(I)n2C N1(C(c2c(CCC)[nH]cc2)=O)CCC(C)N(C(=O)C(C)COC)CC1 N1(C(c2c(C(C)C)occ2)=O)CCC(O)(C)CC1.C1(C=O)CCC1C(N)=O.N C=C(C)CC(C(=O)NCC(CC)CC(C)C)NC(=O)CC=C(C)C C(C(CNC(=O)C)C(F)(F)F)NC(CCCOCC=C)=O.c1nc(C)no1 c1(CC(N2CC=C(CCNC(C(CC)F)=O)CC2)=O)ccc2c(c1)CCCN2C N1(C(N(CC(C)(C)C)C)=O)CCC(O)(C(F)(F)CO)CC1 C1(C(N(C(C)CCNC(c2snnc2C2CCC2)=O)C)=O)CCCC(C2CC2)O1 N1(C(C2(NC(c3cn(CC=C)nn3)=O)CSC2)=O)CCC(C)(N(C)CC)C1 Cc1ccc(Cl)cc1C(=O)NC1CCCN(C(=O)CCCN2C(=O)CCC2=O)C1 Cn1cc(C(=O)N)c(O)nc1=O.N1CCN(C(C2CC(C)(O)C2)=O)CC1.C1CC1 N1(C(CC(=O)OCC)=O)CCCC(NC(=O)CCCOc2cccc(F)c2)C1 N1(C(COC2CCCC(C)C2)=O)CCC(C)(NC(C2CC=CCO2)=O)CC1 CCCC(C(=O)NC(Cc1cn(Cc2cc(F)ccc2F)nn1)C(N)=O)C(=O)O Cc1ccc(C2(CNCC(O)Cc3ccc(F)c(F)c3)CC2)c(C)c1 c1(C(N(CC(=O)N(C)Cc2c(C)cco2)C2CC2)=O)cnc(S)nc1 C1(O)(CNC(=O)NCC(C)CC(F)F)CCOC1(C)C C=CCC(C)(CC)C(=O)N1C(CC(=O)NCCCC(C)C)C2CCCC12 c1(OC)cccc(I)c1C(=O)NCCNC(=O)C(C)C(C)(F)F Cc1ccc(S(C)(=O)=O)cc1C(N1CCCC(C(=O)Nc2ccccc2Cl)C1)=O C1(C(=O)NCCN(C(C23CCC2C3)=O)CC)CNC(=O)N1 C1(C(=O)NC2(CC#C)CCC2)CCC2(CC2)N1C(C1CCC(N(C)C)C1)=O CCCC(C(=O)N1CCC(n2cc(CNc3cncc(OC)n3)nn2)C1)OCC C=CCC(CNC(C1CC(C)(O)C1)=O)NC(c1cnc(C(C)(C)C)o1)=O CCCCC(C)C(=O)NCC(C)(C)OCC(=O)NC(c1nc(C)oc1C)C C1(NC(c2ccc(CC)nc2)=O)CC2CC1N(C(c1c(Cl)n[nH]c1C)=O)C2 C1(C(N(CCCCOC)C)=O)CC(OC)CN1C(=O)C(O)CC1CCCC1 S(=O)(=O)(c1cccc(=NC(C)CS(=O)(=O)CC)[nH]1)NC(CC)COC O=C(C1=CCSC1)NC12CC(CNC(c3cc(CO)on3)=O)(C1)C2 CON=Cc1ccc(C(N2CC(CNC(=O)CC3CC(CF)C3)C2)=O)cc1 N1(C(c2cn(C)nn2)=O)CCC2CN(C(=O)Cc3cc(C4CC4)on3)CCC2C1 C1(CCNC(Cc2nc(C)sc2Cl)=O)CN(C(c2[nH]nnc2C)=O)CC(C)O1 CC1C(NC(=O)COC2CCCC2)CCN1C(c1cscc1C#N)=O c1(NC(C2N(c3ncc(C)cn3)CCNC2)=O)nc2c(s1)CN(C)CC2 C1(CC)CCCN(C(=NCc2cc(C)on2)NCC(=O)NCc2ccccc2)C1 C(N=c1[nH]c2ncc(Cl)cc2s1)C1CN(C(C=C(COC)C)=O)CC12COC2 C1(NC(c2n(C)ncc2)=O)CC(C(=O)NCCC(F)(F)F)C1(C)C C12(CNC(Cc3cc(C)no3)=O)CCC(CC1NC(c1cnc(S)nc1)=O)C2 c1(N(C)CC)ccc(C(N2CCC(NC(=O)CCC3CCC(=O)NC3)C2)=O)cc1 c1(CCC(=O)N(C(C)C2CC2)C(=O)C2CC2)ccc([N+](=O)[O-])cc1.N N1(C(C)=O)CCN(C(=O)CC2CCC=CCC2)C(C(F)F)C1.C1(C(=O)N)CCC1 C1(C(=O)NCC2COCCN(c3nnc(C4CC4)s3)C2)COc2cc(F)ccc2C1 C(C1=CCN(C(=O)C=CC2CC2)CC1)NC(CC1C(OC)COCC1)=O C(=O)(C(C(C)CC)N(C)C(c1cc(CC)n(C)n1)=O)NCCOCC#C C1(C(N2CCC(NC(C3(c4ccccn4)CC3)=O)CC2)=O)Cc2nnsc2S1 CCC(C)CC(=O)NCc1ccc(C(C)NC(=O)CCN2CCCC2=O)cc1 CCC(C)C(O)C(C)C(=O)N(CCCNC(=O)C(C)OCC(C)C)CCO Cc1cc(C(=O)NC(CNC(=O)C(C)(C)C(C)C)C2CC2)cc(N)c1 CC1(CNC(C2(O)COC2)=O)CC(F)(F)CN1C(c1ccoc1Br)=O C(=O)(C(F)(F)C(O)CC)N1CCN(C(C(CC)=CC)=O)C(c2cccc(Cl)c2)C1 CCCCCCCCCC(=O)NC(C1CN(C(c2cnc(Cl)n2C)=O)CCO1)C c1(C(N(CCNC(C2(C)CC3CC3C2)=O)CC)=O)c[nH]c2cc(F)ccc12 c1(OC)cc(NC(=O)CC2CCN(C(c3cccc(Br)n3)=O)C2)c(C)cc1Br c1(OC)c(C(N2CCCCC2CNC(=O)Cn2cnnn2)=O)cccc1Br c1(-c2nc(-c3c(OC4CCS(=O)(=O)CC4)ccc(Br)c3)on2)cc2n(c1)CCCC2 c1(CC)cc(C)c(C(N2CCC(O)(CC)C2)=O)o1.N1(CC=O)CC2CC2C1.N C1(CNC(CN(C2CCCC2)C)=O)C(O)C(O)CN1C(=O)C=C(Cl)Cl C1(CNC(c2cn(C(C)(C)C)nc2)=O)CC(O)CN1C(C1CCOCC1)=O C1(C(=O)NC2C(NC(c3n[nH]cc3Cl)=O)CCC2)Cc2nccn2C1 c1(OCC(=O)NC(CNC(c2cc(C)no2)=O)CO)ccc(Cl)cc1F C1(NC(c2ccoc2Cl)=O)C2CCC1N(C(c1cnc(-c3cccnc3)s1)=O)C2 N1(C(C2CSCN2S(=O)(=O)CC2CCOC2)=O)CCC(O)(CO)CC1 C1(N(C(=O)Cc2cnc[nH]2)C)CCCCC1NC(c1cc(C2CC2)ns1)=O C#CC1CCCCN1C(=O)CC1CN(C(c2csc(C#N)c2)=O)CC1C C#Cc1ccc(OCC(=O)NCC2CN(C(=O)CC)CCCO2)cc1.C(C)=O.N CC1Cc2c[nH]nc2C(C(=O)NC2(CCNC(C3(Cl)CC3)=O)CCC2)C1 N1(C(c2c(C)[nH]c(=N)s2)=O)CCC(NC(=O)C(C2CCOCC2)O)C(O)C1 C1(CC)CCCC(NC(=O)C(CC2CCC2)NC(=O)C(C)C2CC2)C1 CSC1=C(C(=O)NC2CC(C)C23CCC3)CCCC1.C(=O)CN(C)C(N)=O.N c1(C(N2CC3C(CNC(CCC(C)SC)=O)(CC3)C2)=O)cc2c(cc1Cl)OCO2 c1(CN(C)C(C2CCC2=O)=O)ncc(F)cc1F N1(C(c2cc(C)c(C)o2)=O)CCN(C(=O)Cc2ccn(CC(F)(F)F)n2)CC1C CCC(CC)CC(=O)NCC1(C(N)=O)CN(C(=O)C(F)(F)c2cncs2)C1 CC(C(=O)N(C1CC1)CC1CCCO1)c1nn[nH]n1 C=CC(CCC)CC(=O)NCc1nnn(C)c1C(=O)NCC1CCSC1 C(=O)(C(CCC(=O)N(C)C)N1CCC1)NC.C(C)(C)C.C1CSC(=O)N1 Cc1oc(-c2ccccc2)nc1C(=O)NC1CC(NC(C2CCCC(C)C2)=O)C1 CC(O)C(C)(C)C(=O)NCC12CC(NC(c3cccc(F)c3F)=O)(C1)C2 c1(-c2cncc(NCc3c(C)ncs3)c2)cc(N)c(Cl)c(O)n1 CN1CCC(NCc2cn(C3C=CCC(C(=O)NCC4CCOC4)C3)nn2)CC1 c1(C(C(=O)OC)NC(c2sc(C3CC3)nc2C(=O)O)=O)cccc(O)c1 N1(C(C(C)O)=O)CCn2ncc(CNC(C34CC(CO)(C3)OC43COC3)=O)c2C1 C1(N=c2cnc3cc(F)c(F)cc3[nH]2)(CNC(C2(C)N(C)CC(O)C2)=O)CCC1 N1(C(COC)=O)CCC2(CC1)CCN(C(=O)C(C)Cc1ccccc1F)CC2C C1(CNC(C2C(CC(C)C)C2)=O)CN(C(c2ccoc2C(C)C)=O)CCO1 N1(C(COC)=O)CCCC1CCNC(C1CC1c1ccsc1)=O N1(C(Cc2c(C)ocn2)=O)CC(NC(c2c[nH]cc(C)c2=O)=O)CC(O)C1 c1(NS(C2(CC=C)CC2)(=O)=O)cc(OCC)ccc1OC N1(C(CCNC(N)=O)=O)Cc2nccn2CC(NC(=O)CC2CC(C(F)F)C2)C1 N1(C(c2c(N)ccc(CC)c2)=O)CC(C2CN(C(C3COCCN3C=O)=O)C2)C1 c1(OC)cc(CN(C(C)C(=O)Nc2ccc(Cl)cc2)C)cc2c1OCCO2 CC(C)CC(C)CC(C)C(=O)NCCN(C(=O)Cn1ncnn1)C(C)C c1(CC(=O)NCCCN(C(C2CC3C=CC2C3)=O)CC)ccccc1O N1(C(C2CC=CC(n3cc(-c4ccns4)nn3)C2)=O)CCC2CCC(C1)S2(=O)=O C1CN(C(C2(N(C)C)CC2)=O)CCC1O.n1(CC)nc(C(=O)N)cc1C1CC1 C12(NC(C3N(C(C)=O)CSC3)=O)CCC1CN(C(=O)Cc1cc(F)ccc1F)C2 N1(C(CC2N(C)CCCC2)=O)CC(CN=c2cc(F)nc[nH]2)C2(CCC2)C1 c1(NCC(CCC)CCO)ccc(OC(F)F)c([N+](=O)[O-])c1 c1(CC(=O)NCCC(=C)CNC(c2c[nH]cc2Br)=O)ccc2nc(O)[nH]c2c1 c1(C(=O)NCCCCNC(CC2CC(C)(C)OCC2)=O)cccc2ncccc12 C1(NC(=O)C(F)CC2CN(C(C3CCC(O)C3)=O)C2)CCCC(O)CC1 C(CCCCC(=O)NC1(C(=O)N(C)Cc2nc(C)no2)CCN(C)C1)OC C1(NC(C(C)=C2CC2)=O)CCN(C(=O)C(=O)NC(C)C)CC1O C1(CN(C)C(C23CSCC2C3)=O)CCCN1C(=O)COCC1CCCC1 N1(C(C(CC)SC)=O)CCc2ccccc2C(N(C)C(c2cc(Cl)no2)=O)C1 C(=O)(C(CN)C(C)(C)C)N1CCC(c2occ(C(=O)OC)n2)CC1 C(C(C)CC(=O)NC(c1cncs1)C)NC(C(C)NC(N)=O)=O c1(N2C3CN(C(C4COC5COCC45)=O)C(C3)C2)ccn2c(Br)cnc2n1 N1(C(CC(C=C)C)=O)CCC(O)(CNC(C2COCCC2(F)F)=O)CC1 c1(C(N2C(C)CC(NC(c3cccnc3N)=O)CC2)=O)coc2ccccc12 c1(C(C(=O)NCC(C(C)C)NC(=O)Cc2cc[nH]c(=N)c2)C)cncc(F)c1 C(=O)(C1CCCc2c[nH]nc21)N.Cc1ncn(C)c(=O)c1C(=O)NCC1CCC1 C(=O)(CC1=CCN(C(=O)C(C)S(N)(=O)=O)CC1)NCCOCC N1(CC)CCC(N=c2[nH]c(=NCCCC3(C)CC3)[nH]c3c2CCC3)CC1 c1(C(N(C(CN)C2CC2)C)=O)cc(C(C)(C)C)on1.c1nc(C2CC2)ns1 CC1(C)CCCC(c2nnnn2C2CCCC2)(NC2CC2C2CCC2)C1 Cc1cnc(C=CC(=O)NCC(F)C)[nH]1.C1(C(=O)N)CCCN1c1cnccn1 N1(C(C(CCCCC)O)=O)CC2(CCN(C(C3CNC(=O)N3)=O)CC2)C1 c1(OC)cc(OC)c(NC(=O)NC(=O)C(C)OC(C)=O)cn1 c1(OC)cc(CN=c2[nH]cc(-c3ccc(OC(F)(F)F)c(F)c3)s2)cc(Br)c1O C1(CC)CCN(C(C2CC(CC3CC3)C2)=O)C1C(=O)N.CCS(C)(=O)=O c1(C(N(C2CCN(C(C=CC)=O)C2)CCC)=O)cccc(CCC)c1 c1(NCC2=CCN(C(=O)OC(C)(C)C)C2)ccc2ncnc(O)c2c1 c1(C(=O)NCC(C2CC2)NC(CCC)=O)c(Cl)ccc(Cl)c1O Cc1n[nH]c2cnc(C(=O)NC3CCC(C)N(C(=O)Cc4nc[nH]n4)C3)cc12 C(=O)(C1=CCCCC1)NC1CCC(C(=O)NCCCNC(=O)OC)CC1 N12CCC(CC1)OCc1cn(nn1)CC2=O.c1(NC)c(C2CCCC2)noc1C C1(NC(C2CCCO2)=O)(CO)CCN(C(c2cnsn2)=O)C1 C1(CCC)(NC(c2oncc2C)=O)CCN(C(=O)CC2CCN(C)C2)CC1.O Cc1ccc(C(N2CCC(C)(C)C(c3ccccc3)C2)=O)cc1S(=O)(=O)N(C)C C=C(C)CC(C(=O)N(CC(F)(F)CC)C)NC(=O)COCCC CCC(C)CCCCC(=O)NCC12CCC1CN(C(c1ncn(CC)n1)=O)C2 N1(C(c2c(C)nc(C)o2)=O)CCS(=O)(=O)C(CCNC(=O)C#CC2CCOC2)C1 CC1CCC(CNC(=O)Cc2cscc2Br)CN1C(c1cc(F)n[nH]1)=O N1(C(CCOCCOC)=O)CCCC(C(C)(O)C)C1.c1(C=O)cnc(S)nc1.N N1(C(Cc2cn(CC)nn2)=O)CCN(C(=O)C[SH](=O)=O)CC2(CC2)C1.C1CC1.N c1(CC)cc(Br)ncc1C(=O)NOC(c1ccccn1)C C(=O)CCCc1nc(C(C)(C)C)no1.C1(N(CC(=O)NCCC)C)CCCC1 n1(CC(=O)NCC2C(C)CN(C(C3(CCO)CC3)=O)CC2)cnc2c1CCCC2 N1(C(=O)COC2CCOC2)CC2CCC1CN2C(C1CC1C1CCCC1)=O CCCCC(C(=O)NCC1(F)CCCN(C(c2cc(C)[nH]n2)=O)C1)NC(N)=O C1(c2nnnn2C2(C)CC2)(NCc2ccc(OC)c(SC)c2)CCCC1C1CC1 Cc1cc(O)cc(=O)n1CCC(=O)NC1CN(C(=O)CC(O)C(C)C)C1 N1(C(c2ccc(CC)s2)C(=O)NCC)CC2CC1(C(=O)OC)C2.c1cccs1 CC(C)(CCNC(=S)NNC(c1ccc(OC(F)F)cc1Cl)=O)S(C)(=O)=O N1(C(CC2(O)CCCN(C)C2)=O)CC(C2CCCCN(C(=O)COCCO)C2)C1 CC1CN2CCC1CC2.C12(C=O)CCC(CC1)N(C(C1(C(F)(F)F)CC1)=O)C2.N C1(CNC(C2CN(S(CC)(=O)=O)C2)=O)CCCCN(C(=O)C(C)C2CC2)C1 C1(CC)CCCCCN1C(=O)C(COC)n1cc(-c2nccs2)nn1 Cc1nc(C)c(C(N2CCCC(C)C2)=O)c(C)n1.c1(C(=O)N)cc(C(N)=O)cs1 c1(C(=O)NC(CCNC(c2ncnc(OC)c2F)=O)C)csc2ncnc(O)c12 C1(C(=O)NCCCCOC)CSCN1C(C1CCC(=O)C1)=O CN1CCCC(N=c2ccc(Br)c(S(=O)(=O)NCC3CCNC(=O)C3)[nH]2)C1 c1(CC(=O)N(C(CC)C#N)C)c(C)[nH]c(-c2cccs2)nc1=O Cc1ccc2nc(C(=O)NCC(CO)NC(c3cc[nH]c3C(C)C)=O)cn2c1 c1(N(C2CCNCC2F)C(C(C)Oc2ccccn2)=O)ncc2c(n1)NC(=O)C2 c1(NC2CCCN(C(c3n(CC)ncc3Cl)=O)C2)cnc(C#N)c(C#N)n1 CCCCC(C)C(C(=O)Nc1ccc2c(c1)CCC2)N(CC(C)CO)C C(=O)(CN=S(C)(C)=O)NC1(CNC(CCC2CCC(C)O2)=O)CC(F)(F)C1 Cc1ccc(C=CC(=O)NC(CNC(=O)C(C)C2CCC2)CC(C)C)cn1 C1(C(=O)NCC2CCCN(C(C(CC)(F)F)=O)CC2)CCn2nccc2C1 CC(N=c1ccnc(N2CCN(S(=O)(=O)N(C)C)CC2)[nH]1)C1CC(F)(F)C1 N1(C(c2nc(C)n(C)c2)=O)CCC2(CC(NC(c3ccsc3)=O)CO2)C1 c1(C(C(=O)Nc2ccccc2)N(CCC)C2CC2)cnn(C)c1OC c1(OC)ccc(C(N)=O)cc1C(=O)NC1CCCN(C(c2cnc(Cl)[nH]2)=O)C1C C(C(C)(C)C1=CCCC1)NC(C(CC=CC)NC(=O)C(F)C1CCC1)=O c1(OCC)ccc(C(N2CCCC(C(C)NC(=O)C=CCF)C2)=O)cc1C C(CC(C(C)(C)C)NC(=O)CC)N(C(c1c(CC)[nH]cc1)=O)C.CC(F)(F)F CC(=O)CCN=C(NCC(c1ccc(F)cc1)N(C)C)NC1CCOC1 N1(C(c2cc(C)ns2)=O)CCN(C(=O)C(c2ccc(Cl)cc2)N(C)C)CC1C CC1=C(C(=O)NC(C(=O)NC(C(C)C)c2nc[nH]n2)C2(O)CCC2)CCCO1 N1(C(c2c(C)sc(Cl)n2)=O)CCN(C(c2ccc(CN(C)C)[nH]2)=O)CCC1C c1(C(=O)NC2CCN(C(CC(CC)C)=O)CC2)cc(Cl)cc([N+](=O)[O-])c1Cl C12(OC)CCC1CN(C(=O)CC1(NC(=O)CC3CCCC(=O)C3)CC1)C2 C1(CC=C)CCN(C(C2COC(=O)N2)=O)C1.C1(C(=O)N)CCCN1CCC(C)C c1(NCC(C)N(C(=O)Cn2nnc(C3CC3)n2)C)ncc(I)cn1 CC1=C(C(=O)N2CCN(C(=O)CN3CC4CC4C3)CC2c2nccn2C)CCC1 C(C)(C)(C(=O)NCC1CC1)OC(C)C.c1(C=O)cc(C(N)=O)c[nH]1.N c1(C(=O)NCCn2cc(CCN3CCCCC3)nn2)ccc(C(O)C2CC2)cc1 Cc1ccc(C(=O)NC2CCC(C)C2)c(N=[N+]=[N-])c1.C(=O)(CCn1ccnn1)N C1(C(=O)NCCCCN(C)C(=O)OC(C)(C)C)CC2CCC(C1)N2C N1(C(c2c(S(N)(=O)=O)n[nH]c2)=O)CC2CC(C1)C2N=c1[nH]c2ncc(Cl)cc2s1 N(C(=NCCNC(C)(C)C)NC1CCOC(c2cccs2)C1)C(CC)C C1(C=O)CS(=O)(=O)CC12CC2.c1(CC)cc(C(N2CC3CC3C2)=O)ncn1.C CCC(C)(CNC(C1CC1c1cccs1)=O)NC(c1cnc(C)s1)=O C(=O)(CC(C(F)(F)F)NC(c1cc[nH]c(=N)n1)=O)N1C(C(N(C)C)=O)C=CC1 C12(C(N3CC(NC(C4(COC)CCOCC4)=O)C3)=O)CCCCC1C2Br C1(C)(CC)CCCN1C(=O)C=CC1CC1.C(=O)(CC(C)(C)C1CCCCC1)O C1(CNC(c2ccc(OCC)cc2)=O)CCN(C(=O)C2=CCCSC2)CC1C C=C1CCC(C(=O)NC2CC(C(=O)N)C2)CC1.c1ccccc1C(F)(F)F.C CN1N=CC(CC(=O)NC(C(=O)NCC(c2ccccc2)O)C2CC2)C1=O C1(O)(CNC(c2c(CC)nccn2)=O)CCN(C(C2CC(CCO)C2)=O)CC1 C(CC(F)=C(F)F)NC(C1CCC(C2CC2)N1C(c1cnn(CCF)c1)=O)=O CCC(CCC(=O)NCC(CCOC)NC(c1ccc(OC)c(OC)c1)=O)OC c1(-c2nnc(C3C(OC)CCO3)o2)cnccc1C c1(C(N2C(C)(CNC(CCCCCSC)=O)CCC2)=O)cc([N+](=O)[O-])oc1C Cc1nc2c(o1)CCN(C(C1CCN(C(c3cn4ccc(Cl)cc4n3)=O)C1)=O)C2 CC(=O)CCCC(=O)N1CC(C(C)(C)O)(C)C1.c1(C=O)nc(Cl)sc1C(C)C c1(C(=O)NC2CCN(C(c3sc(C)c(O)n3)=O)C2)ccc(Br)cc1F Cc1nc2ccccc2cc1C(=O)NN(C)C(=O)N(C1CCCC1)C1CCCC1 c1(N2C(C3CCN(C(C(C)OCCOC)=O)CC3)CCC2)ccn2nccc2n1 c1(-n2cncc2)cccc(F)c1.C1(C(CC)O)CCCN1C(=O)CNC(=O)CS c1(C(N2CCC(C=C)CC2)C(=O)NC)cc(OC)c(OC)cc1C N1(C(CN(C(CSCC=C)=O)C)=O)CCC(C(=O)NC)C1C c1(CNC(C(C)OC2CCCC2)=O)cccc2c1CN(C(=O)CC=C(Cl)Cl)C2 CC(F)(F)C(C)(C)CNC(=O)C=CCNC(C1CCO1)=O N1(C(c2onc(C)n2)=O)CC(NC(c2cn3c(n2)CCC3)=O)CC2(CC2)C1 C1(CNC(C(C(C)C)n2cncn2)=O)CN(C(C2SCCS2)=O)CCCO1 c1(C(=O)N)ccnc2[nH]nnc12.C1(CC)CN(C(=O)CC2CCC(C)(C)O2)CCO1 C1(C)CCCN1C(=O)C=Cc1cn(C)nn1.c1(C=O)cncc(N)c1.COC CC1=NOC(C(=O)NCC(C)=CC(=O)NCC2CN(C(=O)OC)C2)C1 N1(C(C2C(C=C)C2)=O)CCN(C(c2csc(Br)n2)=O)C(c2ccccc2)C1 c1(CCC(=O)NCC(C2CCCC2)NC(C2CC3CCCC23)=O)cccc(F)c1F C1(NC(C(C)NC(CC)=O)=O)COc2ccccc2SC1 c1(C(N2CCC(CC)(NC(=O)C(C)S)CC2)=O)ccc2c(c1)CN(C)C(=O)N2 C1(NC(CC2(OCC)CC2)=O)CC=C(C(=O)N(CC(N)=O)CC)C1 N1(CC=C)CCC(NC(=O)CC(C)CNC(C2(OC)CCCOC2)=O)CC1 c1(OCCC(=O)NC2CN(C(C3CCC3)=O)CCC2CO)cccc(Cl)c1Cl c1(C(=O)NCCN(C(Cn2ncc(N)c2)=O)C2CC2)cc(F)cc(Cl)c1 CCCC(C(=O)NC(c1cc(C)no1)(C)C)NC(c1cc(OC)ns1)=O c1(NCC(C2CCCC2)C)nc(N2CC3CCC3(OCC(F)F)C2)nc2scnc12 O=C(C#CC1CCCCC1)NCC1CC2CCC1N2C(=O)COc1cccnc1 N1(C(C2C(SC)CCC2)=O)CC2(C1)CN(C(c1ccc(N)c(CN)c1)=O)CCO2 C(CN=c1[nH]c2ccc(F)cc2o1)C1CCC(NC(C(C)c2ccsc2)=O)C1 c1(C(=O)NCC2(NC(C(C)NC(C)=O)=O)COC2)cc(C)cc(Br)c1 C1(C(N(CCCNC(c2cccnn2)=O)C)=O)CCc2nc[nH]c2C1 C1(CCNC(CCC)C(=O)OC(C)(C)C)COc2ccccc2O1 CCC(CC(C)C)C(=O)N(CC(O)CNC(=O)C=CC(=O)N(C)C)C Cc1ccc(OCCCCNC2CCCC2(C)O)cc1 C(=O)(NN1CCCC1C(=O)NCCC1CC(F)C1)c1cc(CC)oc1C CCCCCC(C)CC(=O)NC1(COC)CN(C(c2ccc3oncc3c2)=O)C1 N1(C(c2c(C)n(Cc3ccc(F)cc3)nn2)=O)CCSC2(CCC2)CC1 Cc1cnc(C(N2CCCC2CN(C(C2CCCCC2C)=O)C2CC2)=O)c(O)c1 C(CCN=C(NCCc1scnc1C)NCC1CCNC1=O)OC C1(NC(CCc2onc(CC)n2)=O)CC(C)CN(C(c2cc(C)nc(C)n2)=O)C1 c1(C(=O)NCC(C(C)C)NC(=O)C(Cl)=CCl)cc2occ(Br)c2[nH]1 C1(C)(C(N2CCC(OCCNC(Cc3c(C)ccs3)=O)C2)=O)CCCCO1 CC1(C)CC=C(C(=O)NC2CCCCCN(C(=O)CC3CCCC34CC4)C2)CC1 Cc1cc(NC(C2CCN(C(c3coc(C(C)C)n3)=O)C2)=O)ccc1O c1(C(N2C(C(C)NC(c3c(CC)occ3C)=O)CCC2)=O)occ2c1CCC2 c1(OC)ccc(CCC(N2CCC(C(C)C)C2)=O)cc1.C1(O)(CC(=O)N)CCC1 N1(C(Cc2cnc(C)s2)=O)CCN(C(c2cccc(C)c2F)=O)CC1CCO C=CC1(C(=O)NC(CC2CC2)C(=O)NC)CCN(C(=O)CCCCC2CC2)C1 CC1(C)NC(=O)CC1C(=O)NC1CN(C(=O)CC2NC(=O)NC2=O)CC1.C c1(CNc2cccc(C(=O)Nc3ccnnc3)c2)cc(F)c(Cl)cc1F C(C)(CCC(=O)NC1CC(NC(c2c(C(F)(F)F)noc2C)=O)C1)OCC C1(CC)CN(C(c2cccn(C)c2=O)=O)CCC1NC(=O)C(c1cnn(C)c1)F C1(C2(C=O)CC2)CC(F)C1.C(C=O)C1CCCC1.C1(COCC)CCCO1 C#CC1CCCCN(N2CC3CC2CC3C(N)=O)C1 N1(c2ncnc(C)c2C#N)C2CCC1C(C)C(NC(=O)CC1CC=CC1)C2 CC(C)C(C)(O)C(=O)NCCCCC1CN(C(c2coc(C(F)(F)F)n2)=O)C1 C1(N(C(c2c(CC)oc(C)c2)=O)C)CN(C(=O)Cc2ccn(C)n2)CC12CC2 Cc1ccc(CC(=O)N)c(C)c1.c1(CCC(N2CCC2)=O)nc(C(F)(F)F)n[nH]1 N1(C(CN(C2CC2)CC)=O)CCCC(O)(CC)C1.c1(C=O)ncnc(O)c1Cl.N Cc1ccc(Br)cc1C(=O)NC1(CCO)CN(C(=O)CC(C)F)C1 C1(N(C(Cc2c(CC)con2)=O)CC)CC2CC1N(C(=O)CC1(C)CCC1)C2 Cc1c(NC(=O)C(C2CCCN(C(C3CC3C3CCC3)=O)C2)(C)C)cccc1F CCC(CC)C(O)CNC(C1(CCNC(=O)CC2CCSCC2)CC1)=O O=C(C1=CC2CCCCC12)NCC(F)CNC(c1ccc2c(c1)CCCC2)=O n1(CC(=O)NC2C3CCN(C(=O)CC(O)C4CCCC4)C23)cc([N+](=O)[O-])cn1 [SH](=O)(=O)c1ccccc1Cl.C(C)(C(C)C)N(OCC)CC1CC1.C1CCC1.N c1(-n2cc(C3(C)CN(C(c4cc(C(C)(C)C)on4)C)C3)nn2)ccc(F)nc1 c1(C=O)cc(F)c(F)c(O)c1F.CC1(C)CN(C(=O)C(F)C2CCC2)CC1C.N CC(C)CC(C(=O)NCC1CC(C)(C)CN1C(c1c[nH]nc1Br)=O)C(C)C C1(NC(CC(C)(C)O)=O)CC2CC1N(C(=O)C=CC(c1ccc(F)cc1)=O)C2 Cn1c(C(=O)NC2CC3CN(c4ncc(Br)cn4)CC23)cccc1=O Cn1ccnc1CC(=O)N(CCC(=O)NCC1(N(C)C)CC1)CC1CC1 N1(C(C2C(C)(C)OCC2)=O)CCCC2(CCN(C(C3CC(=C4CCC4)C3)=O)C2)C1 N1(C(C2(C(F)F)CC(=C)C2)=O)CCC2(CC1)CC2.CC(C)(C)C.C(=O)(C)N N1(C(CN(CCC)C)=O)CC2C(CNC(c3cc(Br)c(OC)s3)=O)C2C1 C(=O)(C1NC(C)(C)Cc2ccccc21)NCC1OCCN(CC)C1c1cnn(C)c1 c1(NC(=O)NC(C2CC3CC3C2)C(=O)OC)ccc(OC)cc1OC C12(C(=O)NC3CCN(C(c4ccco4)=O)CC3CO)CCCC(O)(CC1)C2 O(N(C(=O)C1CCCN(C(C2CCC2(F)F)=O)C1)C(C)C)CC c1(C(N2CC(N(C(c3nc(CC)oc3)=O)C)C2)=O)ccc(F)c(C2CC2)c1 Cc1nn(C)cc1C(C)C(N1CCC(NC(=O)Cn2cncn2)CC1)=O C(=O)(C(F)C(F)(F)F)N(C1CCN(C(c2nccc(C)c2F)=O)CC1)CC C(C1CCN(C(c2ccc(C)nn2)=O)CC1)=CC(=O)N.C(=O)(OC)NCC c1(N2CC3C(N(C)C(C45CCC(CC4)C5(C)C)=O)C3C2)cnc(C#N)c(C#N)n1 C1(C(N2CC3C(CO)C3C2)=O)CCCC(NCc2ccc(Cl)nc2)C1 c1(COCC)nc(C(=O)NC(C)(C)C(C)NC(c2cncs2)=O)cs1 Cc1ccc(C(=O)NCCC(C)CCNC(C2COCC(C)(C)O2)=O)c(F)c1 c1(C(N2CCC(CC(=O)Nc3ccnc(C)n3)CC2)=O)ccc2nccn2n1 C(c1ccc(F)c(F)c1)=CC(N1CCN(C(C2CCCC(F)(F)C2)=O)C2CC12)=O N1(C(C2(O)C(C)(C)C2)=O)CCCCC(NC(c2ccc(F)cc2)=O)C1.C(C)(C)C Cc1csc(=O)n1CCC(N1CC2C(CN(C)C(C3(C)CCOC3)=O)C2C1)=O c1(N2CCN(C(CNC(C=C(C)C3CC3)=O)C(F)(F)F)CC2)cncc(C#N)n1 N1(C(C=CCC(C)(C)NC(c2csc(O)n2)=O)=O)CC2(CCC(=O)O2)C1 CC1(C)CCN(C(=O)CCc2cc(Cl)no2)C1CNC(c1cnsc1)=O Cc1cc(N2CCC(NC(c3cnc4cccnn34)=O)CC2)n2nc(C)nc2n1 C1(C)(C(=O)NC(COC)CNC(=O)CCCSC)CCC(=O)C1 C1(NC(c2onc(C)c2C)=O)CCC2CCN(C(c3ccc(F)cc3Cl)=O)C1C2 CCC(C#N)C(=O)N(C1CC1)CC1CCN(C(=O)Cc2conc2C)CC1 N1(C(c2ccc(CC)o2)=O)CC=CC1(C(=O)N)COC.C1CC12CCC2.C C(C(O)CC(=O)NCC1CCCN1C(=O)C(c1ccc(Cl)nc1)(F)F)N(C)C c1(C(N)C(=O)N(CC(F)(F)F)CCO)ccc(Br)cc1 c1(CC(=O)N(CC(C)(C)CNC(C2(F)CC2)=O)CC)ccccc1.C Cc1[nH]nc2ccc(C(=O)NCC(C)CNC(C3(C)CCC(=O)C3)=O)c(Cl)c12 Cn1c([N+](=O)[O-])cnc1N1CCC2C1C2(F)F C12(C(=O)N)CCC(CC1F)C2.C(=O)(C1=C(C)CC1)NCC1CC(OC)C1 n1(CC)ncc(Cl)c1C(=O)NCCc1cn(C(c2ccnc(Cl)c2)(C)C)nn1 C(=O)(CC(C(F)(F)F)N1CCOCC1)N(CC(O)CNC(c1cnsn1)=O)C CCCCC(C)C(=O)OCCOCCOC1(C(=O)O)CC(CO)C1 N1(C(CN(C2CC(C)=NO2)CC)=O)CCN(C(=O)Cc2cccc(F)c2)CC1 C1(CN=C(NCc2cccc(OCC)c2)NC2CC2)Cc2ccccc2N(C)C1 CC1(C)CC(CNC(=O)CC(C)(O)c2ccccc2)CN(C(=O)C2=C(Cl)CC2)C1 N1(C(c2oc(C)c(CO)c2)=O)CCC=C(C(=O)NC2CCCC2CCO)C1 C(=O)(C(C)(C)NC(=O)C(CO)NC(=O)C(C)Cn1cccn1)OCC c1(C(N2C(C(=O)Nc3cn[nH]c3)CC(F)C2)=O)cccc2cc[nH]c12 C(=O)(C(O)C(C)(C)C)NC(C1CCN(C(CC(CC)C2CC2)=O)CC1)(C)C C1(CNC(c2n(CCC)nnn2)c2ncn(C)n2)CCCN(C)C1=O c1(NC(C(C2CC2)NC(C(CC)n2ccnc2)=O)=O)ccc(C(C)C)nc1 c1(-c2cncc(C(=O)NC)c2)ccc(C(=O)Nc2ccnnc2)c2[nH]ccc12 C(CN=C(NC1CC1)N1CCOC(COC)C1)Oc1ccc(F)cc1C(F)(F)F FC1(F)CCCC(NC(=NCC2C3COCC23)NC2CCC2)C1 Cc1ccc(C(N2CCN(C(C3CCS(=O)(=O)C(C)C3)=O)CC2)=O)c(Cl)c1C N1(C(c2ccnc(CO)c2)=O)CC2CCCN(C(=O)CCc3ncc[nH]3)C2C1 C1(NC(c2c(C)ccs2)=O)CC(NC(=O)CCOC2CCN(C)CC2)CC1O c1(C(N2C(C(=O)NC3CSC3)CC(C)C2)=O)c[nH]c2nccc-2c1 c1(OC)cccc(C(C)=CC(N2CCC2C)=O)c1.C1(C=O)CN2CCN1C(C)C2 C=Cc1cccc(CN2CC(CNC(=O)C(c3ccc(OC)cc3)=O)C2)c1 c1(OCC)ccc(C(N2CCC(N(C)C(C3CCCO3)=O)C2)=O)c(F)c1F c1(OC)cc(C)ccc1CC1CC1.C1(=O)CCC2CC2N1 N1(C(C23CCC(OC)C2C3)=O)CCOCC(C(N2CCCC(F)C2)=O)C1 CC#CCC(C(=O)NCc1cnc(CO)s1)NC(c1ccn(C(C)C)n1)=O c1(CNC(=NCC)NCCOC)cn(C)c2ccccc12.C1CC(C(F)(F)F)=NO1 C(=O)(CC(O)C(C)(C)C)N1C(CNC(CC(C)(C)c2ccccc2)=O)CC1 Cc1cnc2c(c1)NC(=O)CC(C)N2C(=O)Cc1cnns1 CCC(C)CCC(=O)NC(C)CNC(C12CCCN1CCC2)=O C1(CC)CCN(C(C2CCCN2C(N)=O)=O)CC1.CC(C(=O)N)OC1CCCC1 C(=O)(CCCS(C)(=O)=O)N(C)CC1N(C(C(SC)SC)=O)CCOC1 c1(C(=O)NC(CNC(c2[nH]cc(CC)n2)=O)CCOC)ncc(OC)cc1F c1(C(N2CC(CNC(C(CC)C#N)=O)C2)=O)cc([N+](=O)[O-])cnc1C C(N=c1[nH]c(C)c(C(N2CCC(COC(C)C)CC2)=O)s1)c1c(CC)cccc1 C1(CNC(C(CC2CCC2)NC(c2nocc2Cl)=O)=O)(CO)CC2CC2C1 C1CCN(C(=O)CC2(O)CCCC2)CC1(F)F.C(C)(C(=O)N)(C1CC1)OC.C C1(C(=O)NC(C)CCNC(=O)CCCNS(C)(=O)=O)CCc2nn[nH]c2C1 Cc1ccc2nc(C(=O)NC3CN(C(c4coc(C)n4)=O)CC3O)cn2c1 C1(C(N(C)CC2N(C(c3c(C)oc(Cl)n3)=O)CCOC2)=O)Cc2nnc(C)n2C1 C1(C)(CNC(C2(SC)CC2)=O)CCCN(C(C23CCCC2C3(F)F)=O)C1 CC(C)C(O)C(C)C(=O)NCC1(C)CCN(C(c2cc(O)ccc2F)=O)C1 CC1CC2(CC(C(N3CCC(C(=O)NCCC4CCN(C)CC4)C3(C)C)=O)C2)C1 c1(OC)cc(C(=O)NCC2CCC(NC(=O)CN3CCCCCC3)C2)ncn1 C1CCCN1C(=O)CCN1CCOC1=O.C1(C)(C=O)CS(=O)(=O)C1.COC N1(C(CC2C(CC)C2)=O)C(C(=O)NOC2CCN(C)CC2)CCC1C c1(OCc2cn(CC)nc2)cc(C(N2CCN(C(C)=O)CC2)=O)ccc1OC CC(C)CC(C)C(=O)NC1CC=CCC1C(N1CCC1(C)CCO)=O N1(C(c2c(C)cc[nH]2)=O)CCC2(CC(NC(=O)C3=CCC3)c3ccccc3O2)C1 C#CCCC(C(=O)NCCc1cncc(C)n1)NC(c1ncnc(O)c1F)=O C1(C(N2CC(F)(CO)C2)=O)CC2(CC2)CN1C(C1CCCC1O)=O c1(CCC(N2CCC(NC(C(C(C)C)C)=O)C2C2CC2)=O)nc2cnccc2[nH]1 Cc1cc(=NCC2CSCCS2)[nH]c(NC(c2ncccc2Cl)C)n1 c1(NC(C2CCN2Cc2ccnc(Br)c2)=O)cc(Cl)ncc1C(F)F N1(c2nnc(C(C)(C)C)o2)CC(NC(=O)Cc2csc(Cl)c2)C2CCCCC12 c1(C=O)ccnnc1O.Cn1nccc1CN(C(=O)CCC1CCC1)C1CC1.N Cc1[nH]nc(Cl)c1C(=O)NCC(C)CN(C)C(c1cc(C(C)C)[nH]n1)=O c1(CC)ccc(CCCC(=O)NCC2CCN2C(C2CCC(CC)CC2)=O)cc1 S(=O)(=O)(c1ccc2c(c1)S(=O)(=O)CC2)NS(CC(C1CCOC1)OC)(=O)=O C1(C(=O)NCC(CNC(C2(C(=O)NC)CC2)=O)C)CC(C2CCC2)C1 CCC(O)(CC(=O)N1CCC(C)C(NC(c2n[nH]c(C)n2)=O)C1)c1ccccc1 N1(C(C2CNC(=O)N2)=O)CC=CCC1C(N1CC(CC2CC2)C1)=O N1(C(c2ccc(N3CCN(S(=O)(=O)C(Cl)(Cl)Cl)CC3)s2)=O)CCc2nc[nH]c2C1 Cc1ccc(C(N2CC(O)(CCNC(C3CCCC(F)C3)=O)C2)=O)c(O)n1 N1(C(COC(CC)C)=O)CCCC(C)(CNC(c2cccc(C3CC3)c2Cl)=O)C1 N1(C(c2[nH]cc(C)c2)=O)CCC(C)C(CC(=O)NCc2cccc(F)c2)C1 CCC(C)C(=O)C(=O)NCCCOCCC(=O)NCCCSCCO C(=O)(CS(C)(=O)=O)NCc1scc(C(N(C2CC2C2CC2)C)=O)c1 N1(C(COCc2cc(C)on2)=O)CCC2CN(C(C3CCCOCC3)=O)CCC12 C(=O)(C(C(C)CC)NC(=O)CC=C(Cl)Cl)N(CC(=C)C)CC C1(C(=O)NCC2CCN(C(=O)C(C(C)C)OC)C2)(CC)CNC(=O)C1 c1(CCOc2cccc(NC(N)=O)c2)cccc2cc[nH]c12 CC1CCOC1CC(=O)NCCC1CCCN1C(C1CC12CC2)=O N1(C(c2c(F)ccc(C)n2)=O)CCN(C(=O)CN2CC=CC2)CC(O)C1 CCC(C(=O)N1CC(NC(c2nc(OC)c(C)s2)=O)C(C(F)(F)F)C1)C(C)C CC1CN(C(=O)CN2CC3CC3C2)CCCN1C(C1CCOC1C(F)(F)F)=O Cc1cc(Cl)nc(C(c2nnnn2C)NC(C)CCF)c1Br CC(CO)CCN=c1[nH]ccc(=NCC(C)C2CCCCC2)[nH]1 C1(NC(c2c(C)n(C)nc2)=O)CC(C)CN(C(C2(C)COC(=O)C2)=O)C1 C=C(C)C1OCCCC1C(=O)NC(C)(C)CC.c1(C(=O)N)cc(C(C)C)[nH]n1 Cc1cc(C)c(C(=O)NC2CC(CNC(C3CC(CCO)C3)=O)C2)cn1 Cc1c(CC(=O)NCC2CC2CC(=O)NC(C)Cc2ccncc2)ncn1C N1(C(C2CC(CN(C)C)C2)=O)CCN(C(=O)CS(N)(=O)=O)C(C2CCCC2)C1 Cc1cnc(C(N2CC(O)C(O)C2CNC(c2csc(C)c2C)=O)=O)c(F)c1 CCC(C)(C)CCCC(=O)NCC1CC(C(=O)N(CC(O)COC)C)C1 c1(-c2ncc(C(=O)NCC(CC)NC(=O)Cc3ccon3)s2)ccccc1Cl N1(C(C2CN(CC)C(=O)C2)=O)CCC(O)(C)CC1.C(c1ccncn1)=CC=O.N c1(C(N(C)Cc2c(CC)noc2)=O)ccc(S(=O)(=O)N)cc1.c1cc(Br)no1 c1(CNC(=O)CN2CC=CC2)cncc(C(N2CCCCC2CCO)=O)c1 CC1CC(OCCNC(=O)Nc2c[nH]nc2C2CCOC2)CC(C)(C)C1 c1(NC)ncccc1C(N1CCC(C2CCCN2C(=O)Cc2nc[nH]n2)CC1)=O C1(C(=O)NCC(=O)NCC(C)C)CC2(CC2)CN1C(=O)C(C)N(C)C C1(NC(C#CC(C)(C)C)=O)CC2CCC1CC2.C1(C=O)CCC(=O)N1C1CC1.N C(=O)(C(C(C)(C)C)N1CCNC1=O)N(CCCNC(c1cc(F)c[nH]1)=O)C C1(C(N(C2CC(C=O)C2)C)=O)C(C)OCCN1C(=O)CC1CCC(C)(C)O1 C12(C(=O)NCC(C(CC)C)CO)CCC(CN(C(c3ccn(C)c(=O)c3)=O)C1)C2 N(C1CCCc2cc(C(C)N)ccc21)C(C(c1cccc(C(C)(C)C)c1)(C)C)=O C(CC(O)C(=O)NC1(CC(=O)NC2(C)CCOC2=O)CC1)SC Cc1sc(C(N2CCCC2CNC(C2CCS2(=O)=O)=O)=O)cc1S(N)(=O)=O C1(CN(C(c2c(CC)csc2)=O)C)CN(C(c2oc(CO)cc2C)=O)CCO1 C1(C(=O)N)CC2C(C1)C2(F)F.CCC(C(F)(F)F)NC(c1ccc(C)s1)=O c1(C(=O)NCc2[nH]nc(C(C)O)n2)cc(NS(C)=O)ccc1F C1(C(N(CC(C)CNC(=O)Cn2cccnc2=O)C)=O)OC(C)(C)OC1(C)C C1(NC(C(n2ccc(C)n2)C)=O)CC12CCN(C(=O)C(c1ccc(C)s1)C)C2 CC1OC2(CO)CC1(C(=O)NC1(C)CCN(c3ncncc3Cl)C1)C2 c1(C(C)C)ccc(C=CC(=O)NCC(C)(O)CNC(=O)CCC=CBr)cc1 Cc1ccccc1-c1nc(C2CC2C2CC2)n(C2CCSCC2)n1 c1(CNC(C2CC(n3cc(CNC(CC)=O)nn3)C2)=O)csc2nccn12 C1(CNC(C(C)OCCOC)=O)CC(C)N(C(=O)CC)C1.C1CCOCC1 C1(C(=O)NCCC2CC(NC(=O)CC3CCCCC3)C2)OC2CCC1CC2 CCC(CC(=O)NC1CN(C(C2C3(CC3)C23CC3)=O)CC1C)CC(C)C N12CCn3nc(cc3C1)C2=O.CC(C)(O)CC(=O)NC1CCCC1OCC(=O)O Nc1cc(C(N2CCOCC(CNC(c3cc(Cl)no3)=O)C2)=O)c(F)cc1F Cc1c(Cl)ccnc1C(=O)NCC(C)NC(C1CCC(CN2CCOCC2)O1)=O C#Cc1ccc(C)c(NC(=O)C#CCNC(c2cc(Cl)no2)=O)c1 C1(NC(c2nnc(C)s2)=O)CCSC12CN(C(C1CC(C)OC1C)=O)C2 Cn1cc(C(=O)NCC2(C)CCCN2C(c2cc(C(F)F)nn2C)=O)c(Cl)n1 c1(-c2cn(C3CCC(CCCC)CC3)nn2)c(C)ccnc1C c1(OC)cc(F)c(C(=O)NC2(C)CCC2)cc1.C1(CC(=O)N)CCCC1C c1(C(c2nnnn2CC(F)F)NCCN2C(=O)CCC2)ccccc1I c1(C(N2CCC(N(C(c3cnc(C)[nH]3)=O)C)C2)=O)ccc(N)cc1Br N1(C(CCc2nnc(C)s2)=O)CCC12CCN(C(c1c(F)c(C)nn1C)=O)CC2 N1(C(c2cnc(C)o2)=O)CCC(C(=O)N(C2CCCCCC2O)C)=C(F)C1 CCC(C)(CO)C(=O)NC(CNC(c1ccc(OCCF)cn1)=O)CO N1(C(c2ccccc2)=O)CCC2(CC1)CCN(C(C1(CF)CC3(CCC3)C1)=O)C2 c1(C(N(CC(=O)NC)CC)=O)c[nH]nc1CCNC(c1cn[nH]c1)=O c1(C(=O)NC2CC(NC(C3=C(C)OCC3)=O)CC2O)ccc2nc[nH]c2c1 c1(N(C)C)cccc(C(=O)NC2(C)CCN(C(=O)CCOCC(F)F)C2)c1F c1(OC)c(N2CCCC(C3CCCCN3C(c3cc(Cl)no3)=O)C2)ncnc1C c1(C=O)ccc2c(c1)S(=O)(=O)N(C)C2=O.C(=O)(CC#N)N(CCC)CC.N Cc1[nH]nc2c1CCC(NC(N1CCOCC3(CC3)C1)=O)C2 C1(NC(Cc2n(C)c(S)nn2)=O)CC12CCN(C(C1CC=CC(O)C1)=O)C2 Brc1snnc1CSCCc1nnc(-c2ccccc2)o1 C(c1ccc(C)nc1)=CC(=O)NCCCCOC.C1(C#N)(C=O)CC=CC1.N C=CC(C)(C)CC(=O)NCC1CC(OC(C)(C)C)C1(C)C C1(CC(N2CCC2)=O)C=NN(C)C1=O.c1(CC)nc(CC)n[nH]1.C(=O)CC.N c1(CNC(CN(C2CC(C#N)C2)C#N)=O)cccc(-c2cscn2)c1 N1(C(C2(N(C)C)CCCC2)=O)CCC(C)(CC(N2CCC3CC23)=O)C1 N1(C(Cc2n[nH]c(=NC)s2)=O)CC2(CCN(C(C3(C)CCOC3C)=O)CC2)C1 c1(C(=O)NC2CCC(NC(COCCC)=O)CC2)c(F)c(F)cc(F)c1F C1(CCC(C)(C)NC(CCCOCCC)=O)CCCCN1C(c1nnsc1C)=O c1(C(C)C)nc(C(=O)NC2CC(F)(CNC(=O)Cc3ccco3)C2)cs1 C1(C(N(C(CC)CNC(C2CC2c2cccs2)=O)C)=O)COCCN1C c1(C(C(C)NC(=O)NC2CC(OC(C)(C)C)C2)O)c(Cl)cccc1Cl C1(C(C(=O)NCCCN(C(C)(C)C)C)OC)CCC(C(C)(C)C)CC1 N1(C=O)CC2CCC1C(C=O)C2.C1(C(N(CC)C(C)C)=O)NC(=O)OC1C N1(C(CS(=O)(=O)NC)=O)CCOC2(CCN(C(=O)C=CSC)C2)C1 C(=O)(C(F)C1=CCCCC1)NC1CC2CN(C(c3cc(N)nc(Cl)c3)=O)CC21 c1(CC)nocc1C(=O)NCC1CCC1NC(=O)Cc1cc(C)cs1 Cc1ncc(C=CC(N2CCN(C(=O)C=Cc3cncn3C)CC2C)=O)c(O)n1 Cc1ccc(=O)n(CC(=O)N(CC(C)(C)NC(C2CC2c2cncn2C)=O)C)c1 CCCC(O)CC(=O)N(C)CCN(C(c1cc(C(F)F)ccn1)=O)C(C)C CCC(C)C(C(=O)NCc1ccc(F)cc1Br)n1cc(C(C)(C)F)nn1 c1(C(N2CC(C3C(C(=O)NC)C3)C2)=O)cc2cccnc2[nH]1.C12CC(F)(C1)C2 n1(C(CC)C)nccc1C(N1CC(CC(C)(C)CNC(C2CCC2)=O)C1)=O C(C(C(=O)NCC(C)C)N(CC(=O)N(CC)CC)C)(C1CC1)OCC n1(CC(N2CCC(N(C(CC(C)C(F)(F)F)=O)C)C2)=O)ccc2cc(F)ccc12 N1(CCNC(=O)OCC)C(=O)CCN(Cc2ncccc2F)C1=O C1(CC)CN(C(=O)C(C)NC(=O)CC2CCCCC2)CCN1C(=O)C1=CSCS1 CC1CCc2c(C(N3CC(O)CC3C(=O)NCc3ccncc3)=O)n[nH]c21 c1(C(=O)NCC(C(C)C)NC(C23CCC2CC3)=O)c(O)nnc2c1COCC2 C1(C#N)(C(=O)NCCN(CCCCCC)C(=O)C(O)CSC)CC12CCOCC2 C(=O)(C(F)C(=O)NCc1cc[nH]c1C(=O)NC)OCC.c1cncn1C.C Cc1nccc(C(=O)N(C)CCN2CCN(C(=O)CC3CCC(C#N)C3)CC2)n1 CC1(C)CC(CNC(C2CC2(C)C)=O)CN1C(c1ccc(-c2ccco2)[nH]1)=O C(=O)(C(C)CCc1ccccc1F)N(CC(CNC(C1(CC)COC1)=O)C)C c1(C(=O)OC)cc(C(=O)NC2CCCCC2)cc(O)c1.C1(C(=O)N)CCCC1C C1(NC(C(n2ccc(C)n2)C)=O)CCc2ccccc2NC1=O Cc1noc2cc(C(N3CC4CCN(C(c5ncc(F)cn5)=O)C4C3)=O)ccc12 Cc1ccc(N(C)C(C)C)c(C(=O)N(C(C)C)C)c1.C(=O)C#CC(=O)N(C)C C1(NC(C(C)NS(C)(=O)=O)=O)CCN(C(c2ccno2)=O)C1 c1(CC(N2CCCC(N(C(C3(C)CC3)=O)CC)CC2)=O)cc(F)c(F)cc1F n1(CC)nc(C(N2CCCC(CNC(C3CC4CC4C3)=O)C2)=O)cc1O CN1CCC(=CC(=O)NC2CCC2C2CC2)CC1 c1(C(N(C(C)CCNC(=O)C=CC2CCCN2C)C)=O)cc(F)c(C)c(F)c1 c1(C(=O)Nc2scc(C(N3C(C)CN(C)CC3)=O)n2)cc(Br)ccc1C#N CC1CCC(O)(C(=O)NCC2CCCN(C(=O)C(C)C#N)C2)CC1 CC1(C)CC(CNC(=O)Cc2cnc[nH]2)CN(C(=O)C(F)(F)CO)C1 CON(CCC(=O)NCC(O)C1CC1)C(=O)c1cccc2c[nH]nc12 C1(NC(C2(C#C)CCC2)=O)(CNC(C2CCCC(=O)O2)=O)CCCCC1 C1(NC(C2N(C)CCC2)=O)CCC2(CC1)CCN(C(c1[nH]ncc1C#N)=O)CC2 C1(=CC=O)CCOc2ccccc21.C1(CC(=O)NCC)(C(=O)OC)COC1.N CCCCC(C(=O)NC1C2CC1N(C(=O)CC(=O)OCCC(C)C)C2)C(C)C C(C(C=O)CC)CN(CCN(CC=C)C)C(=O)NC N1(CC(=O)NCC(CNC(C(CC)n2nccc2C)=O)F)CCN(C)CC1 C1(COC)CC(CNC(c2cc(Br)n(C)c2)=O)N(C(=O)C2=CCCC2)C1 C1(N(C(c2c(OC)nccc2)=O)C)CCCCN(C(C2OCC2(C)C)=O)C1 N1(C(CC(C=C)(C)C)=O)CCCC(C2CC2)C1.C1(C(=O)N)CCC(=O)N1C1CC1 Cc1cc(C#N)ccc1C(N1CCC(NC(c2cnc(O)c(Cl)c2)=O)C1)=O C1(NCC(=O)NC2(C(=O)NCCC(C)(C)N(C)C)C(C)C2)CCOCC1 c1(C(N2CCC2)=O)ccc(S(=O)(=O)C2CC2)cc1.c1ccc(C=O)s1.COC C(=O)(CC(O)CN(C)C)NC(C(=O)NCCC(=C)C)CC1CCC1 C12(NC(CSCC=C)=O)CCC1CN(C(C1CC1)=O)C2.c1cccc(Cl)c1.S c1(CC)ccsc1C(=O)NCC1(F)CC(NC(=O)CCc2ccoc2)C1 C1(C(=O)NCCCCCNC(=O)C(O)Cc2cnc[nH]2)CC12CCCCC2 c1(C=O)[nH]c(C)nc1C.C=C(C)CC.c1(N(CC=O)C(C)=O)ccccc1.N C1(C(=O)NC2(CNC(C(C=C)O)=O)CCCC2)OC2CCC1CC2 N1(C(C2CCC(CNC(=O)COC3CCCOC3)CC2)=O)C2CCC1COC2 C1(CNC(CN(C(=O)CN2CCNC(=O)C2)CC#C)=O)Cc2nccn2C1 C1(C#N)(C(N2CCCC(C3N(C(CC=C=C)=O)CCCC3)C2)=O)CC2(CCC2)C1 CC(=O)CC(C)(C)CC(=O)NC(C1CCN(C(=O)COC2CCCCC2)C1)C CC(=O)CC(C)C(=O)N1CCOCC(C(=O)NC(c2nccnc2C)C)C1 N1(C(CCC(=C)C)=O)CC2COCCC2(NC(=O)CCn2nc(C)cc2C)C1 N1(C(c2ccc(CNC(=O)C3CC3)cc2)=O)CCCSCC1C1CC1 Cc1ncc(C(N2CCC=C(CNC(=O)CCC3(C)CC3(F)F)C2)=O)cc1N C1(NC(C=C(C)C)=O)COC2C(NC(=O)CCCCN(C)C)COC12 c1(C(=O)NCC2CCN2C(=O)CO)ccc(-c2ccncc2)o1.C1CCCO1 C1(F)(C(=O)NCCOC2CCN(C(C3(CO)COC3)=O)C2)CC=CCC1 c1(C(=O)NCC2C=CCN2C(=O)C2=C(Cl)CCC2)ccc2nc(S)[nH]c2c1 c1(CCCC=O)cc(F)ccc1F.C1(CC(=O)NCC2CC2)(CSC)CC1 c1(OC)ccc(C2CC2C(N2CC(C(C)NC(C3(C)CC3)=O)C2)=O)cc1 C1(C(=O)NC2C(C)OC2)(NC(C2CC2C(F)F)=O)CCCC1 c1(C(=O)NCC2N(C(CC(CC(C)C)O)=O)CC2)ccc2c(n1)NCCO2 N#Cc1ccc(S(=O)(=O)NCCOC2CCN(C(=O)CCCCCCBr)CC2)cc1 N1(CC)CCN(C(=O)COCCNC(=O)CC2(O)CCCOC2)CC1(C)C c1(-c2cn(C3CCN(C(C(CC)(C)OC)=O)C3)nn2)cc(F)c(C(=O)O)c(F)c1 N1(C(C)C(F)(F)F)CCN(C(=O)NCCCC(F)F)CC1 c1(C(=O)NCC2CCN(C(c3occ(C)c3)=O)C2)cnn2cc(Br)cnc12 N1(C(c2cc(C)ns2)=O)CCCC(C(C)C(=O)NCc2nnc(C)n2C)C1 c1(C(=O)NC2CN(C(C(CC)n3cccn3)=O)CC2SC)cn2c(n1)CCC2 C#CC1(F)CCN(C(=O)CCN(C(=O)CC)CC2CC2)CC1.C(=O)(CO)N C1(C(N(CCC(=O)N)CC#C)=O)CN(C(=O)Cn2nccc2C=O)CC1F CCC(C)C(C(=O)NCC(C(C)(C)C)NC(=O)CCCCCF)NC(N)=O C1(O)(CN(C)C(C2CC23CCC3)=O)CCCN(C(c2ccccc2)=O)C1 c1(COC)nsc(N(CCCN(C)C(C2CCCC2c2ccccc2)=O)C)n1 CS(=O)c1ccc(C(=O)NC(C2CCCN2C(c2[nH]ncc2C#N)=O)(C)C)cc1 N1(C(C(c2ccc(OC)cc2)(C)C)=O)CCC2(NC(=O)C(O)C(C)C)CCCC12 C1(CNC(CCN(CCCCC)CC)=O)CN(C(=O)CC2CC2CC)CC1O c1(OCCCC)ccc(C(=O)NCCCC(C)NC(=O)CC2CCC2)c(Cl)c1 C1(CC(=O)OC)CCN(C(c2nnc(C3CC3)s2)C(=O)NC2(C)CC2)CC1 C1(c2cn(CC(=O)O)nn2)COCCN1CCc1cn(C2CCC2)nn1 N1(CCNC(=O)OC(C)(C)C)CCCC(NCC2CNC(=O)O2)C1=O c1(C(=O)NC2CC(C)N(C(c3nccc4occc34)=O)C2)ccnc2[nH]ncc12 C(=O)(C(S(C)(=O)=O)CCC)N(C)CCN1CCN(C(c2cnc(O)s2)=O)CC1 Cc1cc(C(=O)NCC2(C)CCC2)nn1C(C)C.C(=O)C(O)C1CCC1.N CC1(C)CCC(CN=c2nc(-c3ccc(Cl)cc3)o[nH]2)CC1 C1(COC)COCCN1C(C1COC(CNC(=O)C2CC2)C1)=O c1(N2CCC(C(=O)NCC)C(OC)C2)ncc2c(C)ccc(Br)c2n1 C(CC)C(F)(F)F.N(C)(S(N)(=O)=O)C1CC1.CC(C)(C)OC=O.C=O C(C)(CCCCNC(c1cc(C(C)(C)C)n[nH]1)=O)NC(C=CC)=O N1(CC2(C)CCC(C)CC2)C(=O)CCN(CC(c2ccc(Cl)cc2)(F)F)C1=O Cc1cc(F)cc(C)c1C(N1CCC(CNC(c2cnc(Cl)cn2)=O)C(C)C1)=O c1(OC)ccc(C)c(C(=O)NC)n1.C1COCCN1C(=O)Cc1ccc(C)cc1 C1(C(=O)NC)CCCN(C(c2cnc(SC)s2)C(=O)NCc2ccc(Br)cc2)C1 C(CC(C(=O)NC1(c2nc(C)no2)CC1)NC(c1cccc(CO)n1)=O)SC C1(C)(C=O)CN(C(=O)CCC)C1.C(C)(C)C.C(C)C=CCC.C=CCO C1(CNC(CC(C)CF)=O)CCCCCN1C(=O)Cn1nc(C2CC2)n(C)c1=O c1(C(N(C(C(=O)OCC)C)C2CC2)=O)cc(C(F)(F)F)cc(F)c1 CC1CN(C(C2(c3cccc(N)c3)CCC2)=O)CC1NC(=O)C(O)C1CC1 C1(N(C(=O)C(C2CCOC2)NC(=O)CC(C)(C)N(C)C)C)(C)CCCCCC1 CC1CC(NC(C2(c3ccccc3)CC(O)C2)=O)CN1C(C1CCOC1)=O C(CN=c1[nH]c(=N)[nH]c(=NCc2coc(C3CC3)n2)[nH]1)c1ncc(CC)o1 c1(C(=O)NC23CC(CNC(CS(N)(=O)=O)=O)(C2)C3)c(O)cccc1Cl c1(N(CC(C)NC(C(CCSC)O)=O)C)nc(-n2cccn2)cc(C)n1 C1(COCC)(NCCCN(C)Cc2ccccc2)CCS(=O)(=O)CC1 c1(C(C(=O)NC2CCC(NC(c3ncn(CC)n3)=O)C2)C)ccc(F)c(F)c1 CC1CN(C)CCC1NC(=O)CN1CCN(C(c2ccoc2C2CC2)=O)CC1 C1(NC(=O)CC2COC3CC2C3)CC2CN(C(=O)CCc3cnoc3)CC2C1 Cc1cc(C(N2CCC2C(=O)Nc2ccc(-n3cccc3)cc2)=O)nc(C)c1 c1(C(=O)NC(CNC(CN(C)CC)=O)C(C)C)cc(C)c(N)cc1F c1(CC)nc(C(=O)NC)c(C)o1.C1CN(C(C2C(C)(C)C2(F)F)=O)CCO1.C c1(C(C)C)ccccc1NNC(=O)CCCCCn1cc(C2CC23CC3)nn1 C1(NC(C2C(C)CCC2)=O)CCSC12CN(C(c1csnn1)=O)C2 c1(CC(=O)NC2CN(C(CC(CC)CN(C)C)=O)CC2O)ccc2c(c1)CCC2 C(C(O)C(=O)N1CC(O)(CN(C)C(C2(C)CCCS2)=O)C1)N(C)C c1(C(N2CCCC(CCNC(C3C(CC)C3)=O)CC2)=O)c(C)cc(OC)cc1F N1(C(C2(CCC=C)CC2)=O)CCC(C(C)NC(=O)Cc2cccnc2Cl)CC1 CCCC(C(O)C(=O)NC1(C)CC(C)(C)OC1=O)NC(c1cscc1OC)=O N1(C(c2cn(CC=C)nn2)=O)CC2CC(NC(=O)C=CC3CCCCCC3)C2C1 C1(CC(=O)NCC(F)C2CCC2)CCCCN1C(c1cc(Cl)n[nH]1)=O.C1CC1 c1(N2CC(CNC(C(C)OCC)=O)N(C)CC2)ncc(C#N)cc1C C1=CN(Cc2c(F)cccc2)Oc2cncc1c2.N1CCCC1=O C1(NC(C(CCF)NC(CCSC)=O)=O)CC(N(C)C)C1(C)C c1(OC)cccc(F)c1C(=O)N(C)CC1CCCN(C(=O)C(C)n2ccnn2)C1 CC1(C)CN(C(C2CCOC2(C)C)=O)CCC1NC(c1cnc2[nH]cncc1-2)=O c1(CC(N2C(CNC(CC(C)OC)=O)C(C)CCC2)=O)cnc2n1CCCC2C N1(C(c2cc(CCC)ncc2)=O)CC2(CCNC(C3CC3(F)F)=O)CCC1C2 c1(C(=O)NCC(CC(F)(F)F)NC(C#CC(C)(C)C)=O)cnc2[nH]cncc1-2 CCC(O)CC(=O)NCc1ccc(C(N2CC=CCC2)=O)cc1 N1(C(CCC2N(C(C3CCC(=O)C3)=O)CCC2)=O)CCCC2(CCC2)C1 C1(C)CC(F)(F)CN1C(=O)CC1CCC(O)C1.Cc1ccnc(O)c1C(=O)N N1(C(c2c(OC)cncn2)=O)CCC(CNC(=O)CCS(C)(=O)=O)C(C)C1 c1(C2(C(c3nnnn3C)NC(C(C)C)C3CCC3)CCC2)ccccc1 N1(C(C(C(C)C)SC)=O)CC2CC(NC(c3cccc4oncc34)=O)CC(C2)C1 c1(OC)cc(C(N2CC(N(C)Cc3cc(O)ccc3Cl)C2)=O)cc(Cl)c1O c1(C(=O)NC2CCC(F)(CNC(c3ccc(C)cn3)=O)C2)cc(C)c(Cl)cn1 c1(C(=O)NC(C=CC(=O)NCC2CC(C#N)C2)(C)C)ncccc1Cl N1(C(C)C)CCC(CNC(C2(NC(=O)CCC3CC3C)CCC2)=O)CC1 c1(C(=O)NCCN(C(C=CCCC)=O)CC(C)O)cc(C)ccc1Br C1(C(=O)NCCC(=O)N(C(C)C=O)CC)C2CCC(F)C12.CC(C)C.N n1(C2CN(C(CCOCC)=O)C2)cc(CNC(=O)Cc2cccnc2)nn1 CC(C)(C#N)CC(=O)NC1(CNC(C2CCC(C)(C)CO2)=O)CCOC1 C1(C(=O)NCC2C=CCN2C(=O)C(O)CC(C)(C)C)(OC)CCCCCCC1 Cc1c(C(N2CCCCCC2(C)C)=O)oc2c(Br)cccc12 N1(CCNC(CN(C(COCC)=O)CCOC)=O)CCOC(C)C1 N1(C(=O)CCc2ncccn2)CCC2CN(C(c3cn(C(F)F)cn3)=O)CCC2C1 c1(C(N2C(C)C(NC(C3CCCN3C(N)=O)=O)CC2)=O)cnc(O)c(Cl)c1 C=C1CC(C(=O)NCC(O)CCNC(=O)C(F)F)(COC)C1 C(=O)(C(CC)C(C)C)N1CC(CC(=O)OC)(OC)C1.C1(C=O)CCOC1(C)C C1(CCC)CCC(NC(C23CC(CN2C(C2CC(=O)N(C)C2)=O)C3)=O)CC1 c1(NC(CC(CC)C)CO)nc(C(F)(F)F)c(S(N)(=O)=O)s1 C(=O)(C(O)CCS(C)=O)N1CCC(OCCNC(COCCCC)=O)CC1 N1(C(CC(=O)OCC)=O)CCN(CCN(C(=O)Cc2cc(C)[nH]n2)C)CC1 N1(C(COCc2n(C)ncc2)=O)CCN(C(C2CCC(F)(F)C2)=O)C2CCC12 Cc1cnc(O)cc1NC(=O)CCC1CCCN1C(=O)CCc1cccc(O)c1 c1(OC)nc(Cl)ccc1CN1CCSC(C(=O)Nc2cccc(CO)c2)C1 Cc1c[nH]c2ncc(C(N3CCCC3CCCNC(c3ccn(C)c3)=O)=O)cc12 N1(C(CC2CC(=C)C2)=O)CCC(C(=O)NC(c2ccn(C)n2)CC)(C(C)C)C1 Cc1cc(C(N2CCCC(CNC(=O)CC3CCOCC3)C2)=O)ccc1Cl C12(C(N3CCCC(NCc4ccc(C)c(C)c4)C3)=O)CC3CC(C1)CC(F)(C3)C2 N1(C(C2(C)C(C)CCC2)=O)CCCC2(NC(=O)Cc3ccc(Cl)s3)CC2C1 c1(CC)cc(C(=O)NC(C)C(C)C(=O)NCc2cc(C)no2)ccn1 N(C1CCCn2ncnc21)C(c1cc(CCNC(C2CC(CF)C2)=O)on1)=O N1(C(c2c(C)nc(C)s2)=O)CCC2CN(C(c3cnc4cc[nH]c4c3)=O)CCC12 C(=O)(CC(C)C(C)C)NCC1CCC(NC(C(COC)COC)=O)C1 C1(OC)CCCCC1C(=O)NCC.N1(CC(N2CCCC2)=O)CCC(F)CC1.O CCC(C(=O)NCC1CCCCN1C(c1c[nH]nc1-c1ccnn1C)=O)C(C)C N1(C(c2cccc(F)c2)=O)CC2(CCN2C(C2(F)CCCOC2)=O)C1 N1(C(c2c(C)ncs2)=O)CCC2(CC1)CCN(c1ncnc3cnn(C)c13)CC2 CCN=C(NCC1(c2ccccc2OC)CCC1)N1CCCC(C(C)C)C1 C1(C)(C(=O)NCc2cc(C(C)=O)sc2)CCCN(CCCCCO)C1 C1(OC)CCC(C(N2CCC(OCC(=O)NC3CCC3)C2)=O)CC1.C1CC1.C S(=O)(=O)(c1cnc(NCc2cc(C)ncn2)c(Cl)c1)N1CC(C)C=C(C)C1 N1(C(c2c(C)cn(C)c2)=O)CCC(c2cn(CC3CCCO3)nn2)C12CC2 C=C1CCN(C(c2ccc(CNC(=O)CCn3ccnc3C)cn2)=O)CC1 N1(C(C(C)OCC)=O)CCCC1(C)C.c1(C(C=O)n2cccn2)ccccc1.N N1(C(C2CN(C)C2)C)CCC(C(=O)NCCCN2CCCCC2)CC1 C#CC1CCCC(CNC(C2CCN(C(=O)CC(C)OC)CC2C)=O)C1 Cc1cc(C(=O)NCC2CCCCC2NC(=O)COC2CC2)cc(C)c1C C1(C(N(CCC(=O)N(CC(=O)OCC)C)CC#C)=O)CCSC(C)C1 n1(Cc2ccc(C)cc2)ccc2ccc(NC(=O)CSc3ncccn3)cc12 c1(C(=O)NCC2N(C(C(n3c(C)ccn3)C)=O)CC(O)C2)cccc2sncc12 Cc1cc(C)c(C(=O)NC2(CO)CCN(C(=O)C(C)CC3CCC3)C2)c(C)c1 C1(CNC(C(C)CF)=O)COCCN(C(c2ccn(-c3ccc(O)cc3)n2)=O)C1 C(CN=c1ccnc(N(C)CC2COC(=O)N2)[nH]1)c1cc(CC)no1 CCCCN(O)C(=O)C(C#N)CC1CCOCC1 N1(c2n(CC)c(C3CN(C)CC3c3ccccc3)nn2)CCc2nc(O)[nH]c2C1 Cc1ncc(NC(C23CC(NC(=O)C(F)F)(C2)C3)=O)c(C)n1 CC1CC(NC(C23CC4CC2C3C4)=O)CN(C(c2sc(Br)cc2F)=O)C1 N1(CC(=O)NC(C2CCCN2C(=O)C(C)N(C)C)C)CCN(C)CC1 Cc1cc(C(N2CC3(CCN3C(C3C4CCC(C4)C3C)=O)C2)=O)cc(=O)n1C C(=O)(CC(C)C(F)F)N1C(CC=C)(C(=O)NCCN2CCN(C)CC2)CCC1 N1(C(C2CC(=O)NC2)=O)CC2CCC1C2NC(=O)COC1CC=CC1 c1(C(=O)NCCN(CCC)C(c2cccn3nnnc23)=O)cc2sc(C)nc2[nH]1 c1(NCC2CC(C)N(C(=O)C3=CCCS3)C2)ncnc2c1nnn2CC1CC1 C(=O)(C1=C(SC)CCCC1)NC1C(NC(C(C(C)C)SC)=O)COCC1 c1(NC(C(CSC)(C)NC(c2ccc([N+](=O)[O-])[nH]2)=O)=O)cccc2ccccc12 N#Cc1ccc(NC(C2(F)CCN(Cc3ncccc3Cl)C2)=O)c(Cl)c1Cl N1(C(C2(COC)CC2)=O)CCC2CCCN(C(c3cc(C)cc(O)c3)=O)C2C1 Cc1cc(F)ccc1CNC(C1C=CC(NCc2ncco2)C1)=O c1(C(=O)OC)ccc(C(=O)NC2CCC(C)C2)[nH]1.C(=O)CC(O)C1CCCC1 C#CCC(C)(C(=O)N(CC(F)Cl)C)NC(c1cc(F)ccc1F)=O CN1CCN(C(c2cc(Cl)ccn2)C(=O)NCC2CCCO2)CC(O)C1 Cc1cc(COCC(=O)N(CC(C)C)C)no1.c1(C=O)[nH]ccc1C1CC1.N [SH](=O)(=O)c1cccc(F)c1.n12cc(C(=O)NNC(=S)NC)c-1n2.CC CC1(C(N2CCCOCC2)=O)CCN(C(c2ccc(NC=O)cc2)=O)C1 n1(CC(=O)N(C(C)C(=O)NC2(CC3CCC3)CC2)CCC)nccc1C CCC(C(=O)N(CC(F)(F)CO)C)NC(=O)C(C)C1CC1 CC1C(=O)NC(=O)CN1C(=O)CC=CCNC(=O)Cc1ccsc1 Cc1cc(Br)ccc1N(C(C1CCOCC1N)=O)Cc1ccccc1 CC1CCC(CCNC(C23CC(CN2C(=O)CC2CCCCO2)C3)=O)CC1 Cc1c(NC2CCN(C3CCOC3)CC2)ncnc1NC1CC(n2cccc2)C1 c1(OC)ccnc(C(N2CC(NC(c3cnn(CC(F)F)c3C)=O)C(F)C2)=O)c1 Cc1nccc(C(N2CC(O)(CNC(C3(CC(C)C)CC3)=O)C2)=O)c1O c1(C(N2C(CNC(Cn3ncn(C)c3=O)=O)C=CC2)=O)cncc2ccccc12 CC(=O)CCCC(=O)N1CCC(CNC(=O)Cc2cc[nH]n2)C1(C)C Cc1cncc(-n2nc(C3CN(C)CCO3)nc2CCn2nc(C)oc2=O)c1 c1(-c2n(CC(C)C)c(N3CCCC(C(F)F)C3)nn2)ccn2cncc2c1 C1(NC(C2CC(n3ccnc3)C2)=O)CCN(c2nnc(C3CC3)o2)C12CCC2 CP(C)(=O)COCc1cn(CC(C2CN(C(C3CC(F)C3)=O)C2)F)nn1 C(c1ccccc1)=CC(=O)N(CC(CC)NC(c1cc(C2CC2)nn1C)=O)C CCC(C)C(O)CC(=O)NC1(C(=O)NCc2nc(C)no2)CCCC1C C(C(CC(C)C)OC)NC(C1(CC)CN(C(c2cc(C)c(C)o2)=O)C1)=O Nc1c(C(=O)NC2CCC2NC(=O)C(O)Cc2ccc(Cl)cc2)ccnc1Cl C1(C)(CCNC(C2ON=C(CC)C2)=O)CCN(C(=O)CC2CCC(=O)CC2)CC1 n1(CC(N2C3C(NC(C(COC)OC)=O)C(CC3)C2)=O)ccc2cc(F)ccc12 N1(C(C2N(C(C(CO)OC)=O)CCOCC2)=O)CC(C)(C)OC(C)(C)C1 Cc1ccc(F)c(N)c1C(N1CCCN(C(c2ccc(Cl)cn2)=O)CCC1)=O C(=O)(C(C)(C)Cc1cnn[nH]1)NC(C)CC.c1(C(C=O)(C)C)cccc(F)c1.N c1(C(NOCC=C)=O)c(CNC(C2CCC(=O)CC2)=O)nnn1C C(=O)(CC(C)C(C)C(C)C)N1C(CNC(C2(OC)CC2)=O)CC(F)C1 C(=O)(C1=COCCO1)N1CCC(C2N(C(c3c(CC)scc3)=O)CCC2)CC1 CC(F)(F)CC(N)C(=O)N1CCCC(CC2CCCNC2)C1 N1(C(C=C(C)Cl)=O)CCC(C)(C)C(CNC(C23CC=CCN2CCC3)=O)C1 C1(NC(C2C(C)C2)=O)CC2CC(NC(C3CCC4(CCC4)O3)=O)CC2C1 CC1CCCCC1CNC(=O)C.c1(CC=O)ccco1.c1(C=O)ccsn1.N C1(CNC(C2(F)C(C)C2)=O)CC(NC(=O)Cn2ncn(C)c2=O)CC1O C12(CNC(C3CCC(C)C3)=O)CC(NC(=O)Cc3ccccc3F)(CO1)C2 c1(C(=O)NC2CCCC(NC(c3ncc(C)c(Cl)c3)=O)C2)cccn2nnnc12 C1(NC(c2ccc(CCCCCC)s2)=O)C=CCN(C(c2c(C)nsc2N)=O)C1 CCC(CCCO)NC(=O)CN(C1CC(C#N)C1)C(C1CCC(C)(C)C1)=O c1(OC)cc(C(=O)NCC2CC2CNC(C2CCOC2C)=O)on1 N1(C(C(C2CCCCC2)OC)=O)CC2CCC(C1)N2C(=O)CC1COC2CC1C2 c1ccc(Br)cn1.C1(F)(CNC(C(C)OCC2CC2)=O)CC(C=O)C1.N c1(C(=O)NC2CCN(C(c3ncccn3)=O)CC2CO)ccc2nc(Cl)nn2c1 Cc1ccc(CN(Cc2ccco2)Cc2ccc(C)o2)o1 C12CCCC1CCN2C(C1CC12CC2)=O.c1(OCC)ncc(Cl)cc1C(=O)N c1(C(=O)NC2CC(C)N(C(=O)CC3CC3)CC2)sccc1S(N)(=O)=O CN1CCN(C)C(C(=O)NC2CC(C(F)C(=O)NCCc3cscn3)C2)C1 c1(C(N(CCNC(COC2C(CC)CCCC2)=O)C)=O)oc2ccccc2c1Cl C1(CC)CCCCC1C(=O)NC(CNC(=O)Cc1ccc(C)nc1)CC c1(CC(C)NC(=O)C(C)NC(N)=O)ccc(Cl)s1 c1(C=O)ccc(CC(C)C)nc1N(C)CCN(C(C1CC=CCC1)=O)CC Cn1nccc1C(=O)N(CCCn1cc(Cn2ccnn2)nn1)C1CC1 c1(CCC)ccc(-n2nc(C(F)F)nc2Cc2cc(C3CC3)no2)cc1 C1(C)(NC(C(C)(C)CCl)c2n(C(CC)(C)C)nnn2)CCCC(F)(F)C1 c1(N(CCC(N2CCOCCC2C(C)O)=O)C(C)=O)ccc2nc(C)sc2c1 n1(CCC(C)C)cc(Br)c(NC(=O)NCC(C)SC(F)F)n1 C1(C(=O)NCc2cc(O)ns2)CCN(C(c2ncc[nH]2)=O)C12CC2 Cc1c(C(=O)NCCOCC(=O)N(C2CC3CC3C2)C)cccc1F N1(C(C2CC(OC)C2)=O)CC(NC(=O)C[SH](=O)=O)C(F)C1.C(C)(C)C.N Cc1noc(C)c1C=CC(=O)NCC1(O)CCN(C(C2CCC3CC23)=O)C1 N1(C(C2N(N=O)CCCC2)=O)CC2CCCN(C(c3cnoc3)=O)C2C1 C1(C(N2C(CCNC(CC(C)(C)O)=O)CSCC2)=O)CCCC(C)(C)C1 c1(C(N2CC(C(C(=O)NC(C)C(F)F)O)C2)=O)cc2cccnc2[nH]1 C(=O)CCCC(C)C.C1(CC=O)C(=O)NN=C1C.C(=O)(CC1CC1)OC.C c1(C(N2CCC(NC(C3C(CC)CCC3)=O)(CF)C2)=O)cn2c(n1)CCC2 C(=O)(CC1=CCCC1)N(CC(C)NC(C(C1CCC(F)(F)CC1)C)=O)C N1(C(C=CC)=O)CCC(OCCNC(C2CC2C(C)C)=O)C1 N1(C(C(C2CCCCC2)NC(Cc2c(C)nccc2)=O)=O)CC(=O)N(C)C(C)C1 Cc1nn2cc(C(=O)NCCC3CCCN3C(=O)C=CC(N)=O)nc2s1 C(=O)(CC(C)O)N(C1(CC(=O)NC(C(=O)NC(C)C)C)CC1)C CC1CN(C(C2CCN2C(C)(C)C)=O)CCC1CNC(=O)C(C)C(C)(C)C C1(C(=O)NCC2(C(=O)NCCN(C)CC)CC2)CC(C)C1 Cc1ccc(Cl)cc1C(N1C2CN(Cc3cc(Br)ncc3Br)CC12)=O N1(C(CC2C(CC)C2)=O)CC2CCN(C(=O)C3=CCCCC3)CC2C1 c1(C(=O)NCC(CC)NC(C(CC#C)C)=O)ccc(F)cc1O C1(CN(C)C(c2cccc(CN=[N+]=[N-])c2)=O)COCCN1C(c1sccc1F)=O Cc1c(C(=O)NC2(CF)CCN(C(=O)CC3CCCC3C)C2)ccc2cncn12 C1(NC(CC=CC=C)=O)CN(c2cc(-c3cccc(Cl)c3)ncn2)CC2(CC2)C1 C(c1cnc(C(C)(C)C)s1)=CC=O.Cc1cocc1C(=O)N.C1CCCC1.C Cc1ncnc(C(=O)NCCCNC(c2nccc(Cl)c2F)=O)c1C C1(C(N2C(CCC#C)CCC2)=O)(CC=C)CCCN(C(C2CCCC2)=O)C1 C1(C(=O)NC2CC3(C(C(N4CCC(C)C4)=O)C3)C2)CCCCCN1C C1(OC)CC(NC(=O)CCc2nc[nH]n2)CN(C(=O)C(=Cc2ccco2)C)C1 C1(C(=O)N)CCCN(C(C)=O)C1.n1(CC)ncc(C(N2CCCC2CCC)=O)n1 CCCC(CC)C(=O)NC1CCN(C(=O)COc2ccc(OCC)cc2)CC1F c1(CC)csc(-n2cc(C(=O)NC(C)(C)C)cn2)n1.C(=O)C.CC(C)C.N N1(C(C23CCC(OC)C2C3)=O)Cc2occ(C(=O)NCCCCCCO)c2C1 CN1CC(C(N2CC(NC(C3CCOCC3)=O)C(n3ccnn3)C2)=O)CC1=O C1CC(C(N)=O)=NO1.C1(C(=O)N)(COC)C=CCN1C(C1CCC1)=O.C c1(C=O)[nH]c2ccc(C)cc2c1Cl.C#CCCOCC(=O)NCCOCCC.N C(=O)(N1CC(n2cc(C3CCCO3)nn2)CO1)c1cn(CC)nc1C(F)(F)F C(CC(C)C)(C(=O)NC(C)(C)C(F)(F)F)NC(CC1CC(OC)C1)=O N1(C(C(CC)C#N)=O)CC23CCCC2(C1)CN(C(C1CCN(C)C1=O)=O)C3 c1(C(N2CC(CNC(c3cccc(C)c3F)=O)OCC2)=O)cc2cccnc2o1 Cc1ccc(Cl)c(C(=O)N(C2CCN(C(C3CCC(CN(C)C)O3)=O)CC2)C)c1 N1(C(C(CN(CC)CC)F)=O)CC2CC1CN2C(=O)C(=O)N(C)C c1(NCC(c2ccccn2)C)ncc(S(=O)(=O)NCC2=CCCCC2)cc1Cl C1(NC(CCCCCN(C(CCSC)=O)C)=O)C2CCC3C(C2)CC13 S(=O)(=O)(c1scc(OC)c1OC)NCC1(C(=O)OC)CCNCC1 c1(CNC(C(COC)N(C)C)=O)nnc2n1CCN(C(c1cccs1)=O)C2 c1(C(N2CCC(NC(c3c(COC)cccc3)=O)CC2)=O)cccc(C)c1N c1(C(N(CCCCNC(CC(C)SC)=O)C)=O)cc(C)nc2ncnn12 N1(C(C(CC=CC)C)=O)CCC2C(NC(=O)Cc3c(C)nn(C)c3C)C2C1 N1(C(C(CCC)C)=O)CCC(C2CC2)C1CNC(=O)C(C)NC(=O)CC C(=O)(CCCCCn1cc(CCC(O)C(=O)O)nn1)NCC(C)C1CCC1 N1(CC(=O)N(CCC)CC)CCCC(N(C)C)C1.C(C)(C1CC1)=CC=O C1(NC(c2ccc(Br)c(Cl)n2)=O)CCCN(c2nnc(-c3ccccc3)o2)CC1 C(=O)(CCP(C)(C)=O)NC(C)(C)C(=O)NCC(F)(F)F C1(NC(C2(CC)CC(C)(C)C2)=O)CN(C(C2CC2(C)C)=O)CCC1O c1(C(=O)NC2CN(C(c3c(C)cncc3)=O)C(C)CC2)ccc2nc(O)[nH]c2n1 c1(C(N2CCCC(C(N3CCC(OC)CC3)=O)C2)=O)ccc(C(F)(F)F)c(I)c1 Cc1[nH]nc(C(N2CC(NC(C3(C(C)(C)O)CCC3)=O)C(C(F)F)C2)=O)c1Cl C(=O)(CCC(F)(F)C(F)F)NC1CN(C(CCN(C)CCO)=O)CC(O)C1 N1(CCNC(C(C)N(C)C(c2cc(CO)[nH]n2)=O)=O)CC(C)(O)C1 Cc1ccc(F)c2[nH]c(C(=O)N(C(C)CN(C)C(c3ccc(Cl)cc3)=O)C)cc12 CC(C)CCCCC(=O)NCC(CC(C)C)NC(c1cnc(O)cc1O)=O c1(-n2c(C)cc(C(=O)NC3C(CC)CCC3)n2)ccc(F)cc1F n1(CC)ncc2cc(C(=O)N(CC(C)NC(=O)CCc3nncs3)C)cnc12 c1(OC)ccc(Br)c2c1CCN(c1nccnc1C(F)(F)F)CC2 N1(C(C(CC(C)(C)C)O)=O)CC(NC(=O)C(C)(C)CO)CC12CCCOC2 C1(C(=O)NCC2(C)CN(C(=O)CN3CCCC3)C2)CCC2CCC(=O)N2C1 N1(C(c2ncoc2C)=O)CCN(C2CC2)C(=O)C1.C(=O)(CCC(=O)N)NC.C c1(C(=O)NC2C(NC(CSc3cccc(OC)c3)=O)CC2)cc2occc2[nH]1 N1(Cc2n(C)cnc2)CCCC2(CCN(C(=O)C(=O)Cc3ccc(O)cc3)C2)C1 CCCC(CNC(=O)CCNC(=O)N(C)Cc1ccc(F)cc1)CCO c1(CN(S(C(CCOC)C)(=O)=O)C)cccc2[nH]ccc12 Cc1nc(N2CCCC(CNC(C3CCC(N(C)C)CC3)=O)C2)c(C)c(Cl)n1 CCCCCCCCCCCn1nc(C2CCC2)nc1-c1ccc(C2CC2)cc1 Cc1nccn1CCN(C)C(C1COC(CNC(=O)CC2COCCO2)C1)=O CC(CC(C)(C)CO)NC(=O)C(C1CCN(C(c2cc(O)nn2C)=O)CC1)C c1(N2CCC(CC=C)(NC(=O)C(F)CC)CC2)nc2c(cc1C#N)CCC2 c1(C(=O)NCC(C)(C2CC2)NC(C(C)Cn2ccnc2)=O)ncc(F)cn1 C(=O)(C(CC(C)C)ONC(c1cnc(C)cn1)=O)N1CCN(C(C#C)C)CC1 c1(C(=O)NCC(=O)NC)ccc(-c2ccc(C(N)=O)cc2)cc1 N1(CCC(=O)NCCC(F)Cn2cc(Cn3cccc3)nn2)CCCCCC1 Cc1ncc(C(=O)NC2CN(C(=O)C=CBr)CC2c2nccn2C)n1C c1(N2CCC(N3C(=O)OCCC3)CC2)cc[nH]c(=NCCC2=CCCCCC2)n1 C1(OC)CC(CNC(=O)Cc2cscn2)N(c2ccncn2)C1 C1(C(=O)NC)(COC)CC=CCC1.C1(O)CCN(C(=O)CC)C1.C(N)=O c1(C(=O)NCC23CCC(C2)N(C(C2CC(O)C2)=O)C3)cc2nccnc2cc1F C1(C2CC2)(C(N(C2CN(C(=O)CCOCC3CCCO3)C2)C)=O)CC1 N1(C(CCCC)=O)CC(CCNC(c2noc(CC)c2C)=O)C(C)C1 C1(CC#C)(C(=O)NCCn2ncnn2)CCN(C(C2CCN(C)CC2)=O)C1 N1(C(c2n(C)cc(Br)n2)=O)CC2CC1CN2Cc1cccc(Cl)c1Cl C1(NC(C2(CO)CC2)=O)CN(C(C2CC3(C2)CC3(F)F)=O)C2(CCCC2)C1 Cc1cc(=O)cc(CNC(=O)CCC2(NC(c3nccnc3C)=O)CCC2)[nH]1 CC(C)C(O)C(C)NC(c1ccccc1Cn1cc(C2(C3CC3)CC2)nn1)=O N1(C(=O)NCc2cccc(-c3nnc(C)o3)c2)CC2(CCCCC2)C1C(C)C CC(C)CS(=O)(=O)CCC(=O)N1CCC(NC(C2(C(C)(F)F)CCC2)=O)CC1C C#CCC(O)C(=O)N(C1CCN(C(c2ccnn2CC2CCC2)=O)CC1)CC C1CN(C(=O)CC2(C(F)(F)F)CC2)CCN1C(=O)C=O.CC(F)(F)F.CC N1(C(c2c(CCC)nns2)=O)CCN(C(=O)C(=O)NCC2CC2)C(C)CC1C N1(C(COC(CC)C)=O)CC2CC(C(=O)Nc3cncc(CO)c3)CC2C1 c1(CC)cc(C(=O)NC2CCN(C(c3cnc(C)c(N)c3)=O)C(C)C2)cc(O)n1 CCC(CCCC(=O)N1CC2CC1CN2C(C)C)NC(c1cc(C(C)=O)[nH]n1)=O c1(CC)ncc(S(=O)(=O)NC(C23CCC(CC2)C3)C(=O)OC)s1 N1(C(C2C(C)=CCS2)=O)CC(C(=O)O)C(N=[N+]=[N-])C1 C#CCCC(O)C(=O)NC1CC(NC(=O)CCN2CCCC2)C(O)C1 C1(C(=O)NCC2CCN(C)C2)CCN(C(=O)C2CC2)O1 C1(CNC(C(CC)(C)C)=O)CC2(CC(NC(=O)C(O)CC3CCCC3)C2)C1 CCC(C(=O)N(CC(C)N(C)C(c1ccn(CC(F)F)n1)=O)C)C1CCOCC1 C1(OCCC)CCCCC1C(=O)NC(CCN(C)C(c1[nH]nnc1C)=O)C(C)C C(=O)(C1=CCC(C)(C)CC1)N(CCCCCNC(C1C(C)OCC1)=O)C N(C(=NCCc1ccc(Cl)c(OC)c1)NC(c1cccs1)C)C1CC(OCC)C1 c1(C(=O)NCCCC(=O)NC(C)C)cncc(OC(c2ccccc2)C)c1 CC1CCC=C1C(=O)N1CCC(CNC(c2cn(CCC3CC3)nn2)=O)C1(C)C N1(C(C(=O)NC2(C)CCO2)=O)CCC(N)(c2cccc(C(F)(F)F)c2)C1 C12(C(=O)NCC3N(C(C=C(CC)CC)=O)CC(C)(C)C3)CCCCC1CCC2 N=c1[nH]cc(CNC(c2[nH]nnc2C2CCNC2)=O)s1 c1(C(N2CC(OC)CC(NC(C(CCOC)OC)=O)C2)=O)c(F)ccc(Cl)c1N C#CC1(C(=O)NCC(CO)C(C)C)CCN(C(c2nonc2N)=O)C1 c1(C(N2CCN(C(CSCC)=O)C3C2C3)=O)ccc2c(C)cc(O)nc2c1 C1(C(=O)NC2CCN(CCNC(CC(CC)CC)=O)CC2)CCC2(CCC2)OC1 CC1=CCN(C(=O)CC(C(F)F)n2ccnc2)CC1.C1(CC(=O)N)CCS(=O)(=O)C1 CCC(CC(=O)N(CCC(C)NC(=O)CN(C)C(N)=O)C)c1ccccc1 C1(NC(CCCN(C(C(C)CCN(C)C)=O)C)=O)COCC(C)(C)C1 CCC(C(=O)N)C(C)(C)CC.C1(C(N2CCC2C(=O)N(C)C)=O)CCCCC1.C CC1C(C(=O)NCCC2(O)CCN(C(c3cc4c([nH]3)CCCC4)=O)C2)=NOC1C C1CC(C)CCN1C(C1CC(=O)N(C)C1)=O.n1(CCC)ccc(C(=O)NC)n1 C(=O)(C#CC1(C)COC1)N(CCC)C1CC1.N1(C(CC)=O)CCCCC1C(=O)N c1(OCC)ccc(C2CN(C(=O)C(c3ccccc3)F)CCO2)cc1 c1(C(N2CCOCC(CNC(CC3CNC(=O)O3)=O)C2)=O)nc2ccccc2[nH]1 CC1(C)CC(CC(=O)NC)CN1C(c1ccc(Cl)s1)=O.C1CCC(C(N)=O)O1 CN1C(C(=O)N(Cc2ccc(F)cc2)Cc2ccco2)CCS1(=O)=O C1(NC(CC=C)=O)CCC2(CCCN(C(C3CS(=O)C3)=O)C2)C1 C1(N(C2CCN(CCSCC(F)(F)F)C2)C)CCN(C2CC2)CC1 CC1CN(C(C2CNC(=O)N2C)=O)CCCN1C(=O)Cc1cc[nH]c1 n1(CC)cc(NC(=O)C(=O)Nc2ccsc2Cl)c(=O)c(Br)c1 N1(C(C(C(=O)OC)OC)=O)CCCC1(C)C.c1(C=O)nnn(C)c1C(F)F.C N1(C(C(C)C(C)(C)C)=O)CC2(C1)OC(=O)NC2C.C1(C=O)CC1.CCOC c1(CCC)cc(C(=O)NC2CC(NC(C3CCOC3C)=O)C2)n(C)n1 c1(C(N2CCCC(CN(C(CC(CC)C)=O)C)C2)=O)c(C)nc2sc(C)nn12 C=C(C)CCCC(=O)NCC1CCN(C(=O)Cc2ccccc2C(N)=O)C1 CC1CN(C(c2cccc(O)n2)=O)CC1NC(=O)Cc1ccccc1I N1(C(C(CC)OC)=O)CCCC(F)(CNC(C2CC(=C3CCC3)C2)=O)C1 S(=O)(=O)(c1ccc(F)cc1F)NCCCC(=O)NCC1COc2ccccc2O1 C1(C(C)C)C(NC(c2cnn(C)n2)=O)CCN1C(c1cc(C#N)c[nH]1)=O C1(C(=O)NCC(C)Cn2cccn2)CC=CCN1C(c1nonc1N)=O c1(CC(N2CC(F)C2)=O)cccc2c1OCCO2.c1(C(C)C(=O)NC)ccc(Cl)s1 C1(C#N)(C(=O)NC(c2cn(C3COCC3C(F)F)nn2)C)CC12CCC2 C1CN(C(C23CCC(C)(CO2)C3)=O)CCC1(C)C.C(CC(=O)N)N(CC)CC N1(C(c2c(CCC)cccc2)=O)CCN(C(=O)C(C)OC2CCCC2)C(CF)C1 C1(NC(C(C(C)C)NC(=O)CCC2CCCCO2)=O)CCCC2(CC1)CC2 C1(OC)CCC12CC(C(=O)NC1C=CCN(C(c3cncc(C4CC4)c3)=O)C1)C2 Cc1nn(C)c(Br)c1CNC(C(F)(F)F)c1ncc[nH]1 S(=O)(=O)(c1ccc(C(F)F)s1)N(C)Cc1ccc(Br)cc1F c1(C(N(CCCNC(c2cnc(CC)[nH]2)=O)C)=O)oc(C)nc1CC c1(CC)ccc(C(=O)NCC(C)(F)CNC(=O)C(C)(C)C2CCCO2)[nH]1 C1(NC(C2(COC)CC2)=O)CN(C(c2ncoc2C2CC2)=O)CC1F C(=O)(C1CCCn2ccnc21)NCCCC(C)NC(c1c(C)n2c(s1)cnc2)=O C1(C(=O)NCC(C2CCCN2C(=O)CCOCCON)(C)C)CCC1(C)C C(=O)(C1=CCCSC1)NCC1CN(C(c2c(CC)[nH]c(=N)s2)=O)C1 N1(C(CCN(C(Cc2c(C)cnn2C)=O)C)=O)CC2(C1)CC1(CCC1)C2 c1(C=O)sc(C)nc1CC(C)C.Cc1csc(C(F)(F)C(=O)NC2CC2)n1.C c1(Cc2nc(C(C)OC)n(-c3ccc(Br)c(C)c3)n2)ccc(Cl)c(C)c1 c1(C(=O)NCC(CNC(=O)CC2CC(F)C2)OCC)occc1C CC(C)(C)C(=O)NCCCC(=O)N(CCNC(C1CCO1)=O)C.C1CC1 C1(C)(C(=O)NCC(CNC(c2ccc(C(C)C)o2)=O)F)CC2CCC1O2 Cc1nn(C)c(-n2cccn2)c1C(=O)N(C)CCNC(C1CC(C)C1)=O CC1CC(C#N)(C(=O)NCCCC(C)NC(c2ccccc2Br)=O)C1 N(C(=NCCCCl)NCCOC(F)F)CCN(C1C(C)CCCC1)S(C)(=O)=O C(C)(CCC(=O)NC1CCC(CNC(=O)CC2CCCCCC2)C1)SC C1(CC)CN(C(=O)C(C)N2CCC2)CCC1C.c1(C=O)cccc(C(C)C)n1.N c1(C(N(CCC(=O)N(CC#CC)CC#C)C(C)C)=O)cn(C)c(=O)n1C Cc1nc(Cl)nc(N2CCOC(C(C)NC(c3ncnc4sccc34)=O)C2)c1F N1(C(c2cc(C)c(C(F)(F)F)cc2)=O)CCCCC1C1CCCN1C(=O)CC#N C#CCCCC(=O)N1CCCC1C(C)NC(=O)CC1CC2CC2C1 c1(CC(=O)NC(CN(C(C2CC(F)(F)CS2)=O)CC)C)ccc(C)cc1F c1(C(=O)NCCC(CC)CC)cc(C)c(F)c(S(C)(=O)=O)c1.C(=O)C(C)C.N CC1CN(S(=O)(=O)CCC2(C)N=N2)Cc2ccccc2O1 C1(C)(CNC(C(C2CCN(C(C(CSC)C)=O)C2)(C)C)=O)CCCCCC1 CCCCCC(=O)NC(C)CC1CN(C(c2cnc(-c3cnn(C)c3)s2)=O)C1 C=Cc1cncc(C(N2C(C(=O)NCCC(F)(F)F)CC2C)=O)c1 c1(C(=O)NC(C(=O)NC(C=C)C2CC2)CCF)cnc(O)c(F)c1 c1(C(C)(C)C)ccc2c(c1)CN(N1CC(C#N)(CCC(=O)C3CC3)C1)CCO2 N1(C(=O)CCn2cccn2)CCOC2(CCN(c3nc(Cl)ncc3Cl)CC2)C1 C1(C(N(CC(C)(C)C)C)=O)CC(C)CC(C)C1.CC(C)C(=O)N(CC(=O)N)C c1(NC(C2CC23CN(C(C2CCC4(CNC4)O2)=O)C3)=O)c(Br)ccnc1Cl c1(C(=O)NCC2(O)CCN(C(C3CCCCC3O)=O)CC2)ccc(Cl)c(Cl)c1O Cc1noc(C(=O)NCC2C3CN(C(=O)CSc4cccc(Cl)c4)CC23)c1C c1(C(C=O)(F)F)ccc(Cl)nc1.C=C(C)CCNC(=O)COCC(=O)O c1(C(C)(C)C)cnc(C(=O)NCC2(c3ccc(O)cc3)CC2)nc1 N1(C(c2c(CCC)occ2)=O)CC2CCN(C(=O)CCn3cccn3)CC12 Cc1cnc2c(C(N3CC(C)C(F)(F)C3)=O)cccn12.C(=O)C(C)CN(C)C.N c1(C(=O)NC2CCC(CCNC(C=CCCC)=O)C2)ccc(F)cc1F N1(C(C2C(C(=O)OC)C2(C)C)=O)CCN(C(c2ocnc2C)=O)C(C)C1C C(=O)(CCC(C)(C)F)NC1C(NC(C(C)N2CCCC2)=O)CCOC1 C1(CNC(C(=O)N(CCC(=O)OC(C)(C)C)CC=C)=O)CCCN1C N1(C(C=C(NC(C)=O)C)=O)CC(NC(=O)Cc2sccc2Cl)C2(COC2)C1 C1(NC(=O)C2=COCCC2)CCC2CCN(C(=O)Cn3cncn3)C1C2 Cc1cc(C#N)c[nH]c1=NC(=O)N1CCC(C)(CC#N)C1 c1ccc(-n2cccc2)cc1.CC1CCC(N(C)CCNC(=O)C=CC=O)O1.N N1(C(C2(C=O)CC2)=O)CC2(CC2C(N2CCC(c3ccn(C)n3)CC2)=O)C1 C1(CNC(CNC(C)=O)=O)CCC1NC(=O)C(C)OCCC(C)C C1(CC(=O)NCC(CCC)(C)C)CCCN(C(=O)CC(C)SC)CC1 CN1CCCC1(C)C(=O)NC1CCC(n2cc(Sc3ccc(Cl)cn3)nn2)CC1 CCC(CCCC(=O)NC(COC)C1CC1)NC(C1CC1C(C)C)=O CCCCCC(O)C(=O)NC1(C)CC(NC(c2cnc(C)nc2C)=O)C1 Cc1ccc(C(N2CC3C(CNC(c4ccc(CO)o4)=O)C3C2)=O)cc1C#N c1(C(CCCNC(=O)NC2C(SC)COC2)C)cccc(C(F)(F)F)c1 Cc1cc(CCC(N2CCCC2CCNC(C2CCOCC2)=O)=O)n[nH]1 c1(C(N2C(C)CC(NC(=O)CC(C)(C)C#N)C2)=O)cc2ccncc2s1 N1(CCOCC(C)C)CCC(C)C(NC(c2ccncc2Cl)=O)C1 N1(C(CC=CC=C)=O)CC(C)C1C(=O)NC(C)Cc1ccccn1 CC(C)(C(=O)NCCCNC(c1ccsc1C(F)F)=O)n1cccn1 C(=O)(CN=S(C)(C)=O)N1CCN(CCN(C(c2nccc(C)n2)=O)C)CC1 n1(C(C)C)cc(C(=O)NCc2cnc(C(C)(C)C)[nH]2)cn1 CC(CC(=O)N1CC2CC1CN(C(c1cnn(C)c1C#N)=O)C2)P(C)(C)=O CC#CCCC(=O)NC1CC1CNC(c1ccc(C2(C)CC2(F)F)cc1)=O CCC(C)(C)C(O)c1nc(CCOc2ccccc2)nn1-c1ccn(C)n1 CC(C)C(C)C.C(=O)(C(CCC1CCC1)N(C)C)N.C1(=CC=O)CCSCC1 CC(C)CC(C(=O)NC1(CNC(=O)Cc2c(F)cccc2F)CCCC1)C(C)C C1(NC(c2n[nH]cc2-c2ccccc2)=O)CC2(C1)CC(NC(C1CC1)=O)C2 Cc1ccnc(NC(C2CC(O)CN2C(=O)Nc2ccc(F)c(Cl)c2)=O)c1Br n1(CC)nc(C(N2CC(NC(C3C(F)(F)C34CC4)=O)C(C)C2)=O)cc1O c1(C(=O)NC(CNC(c2cn(CC)nc2)=O)C(C)C)cn(C)c(=O)n1C C(=O)(C(C)C(O)CC)N1CCC(CCNC(c2n(CC#C)ccc2)=O)CC1 n1(CC)ccnc1CN(C(=O)CC1CCN(c2nc(-c3ccccc3)cs2)C1)C Cc1nc(C2CC2)sc1CC(N1CCOC(CC)C1)=O.C(=O)(C(C)(C)N(C)C)N N1(C(C(C)NC(C2COCC2C(N)=O)=O)=O)CC(C=O)C(C2CC2)C1.C c1(OC)cccc(C2CC2C(=O)N(CCCN(C)C(c2nc(C)nn2C)=O)C)c1 c1(N2CCCC(C)(OC)CC2)cc[nH]c(=NCCC2CCS(=O)(=O)CC2)n1 Cc1cc(C(=O)NC(C)C(CO)NC(C2(C)CC(C)C2)=O)cnc1O N1(C(=O)CNc2nccs2)CC23CCCC2(C1)CN(C(C1CS(=O)(=O)C1)=O)C3 CC1(C)CCCN(C(=O)C=Cc2ncc[nH]2)C1CNC(c1cc(Cl)ncc1Cl)=O Cc1nc(C(=O)NCC2CCC(O)C2)c(C)n1C.C(=O)(C(C)CC1CC1)N N1(C(c2cc(Cn3ncc(C)c3)on2)=O)CC(NC(C2CCOC2)=O)C2CC2C1 C1(C)(CC(=O)NCC2(C)N(C(c3ccc(C)[nH]3)=O)CCC2)CCS(=O)(=O)N1 c1(CC(=O)NC(CC)(C)CNC(=O)C(COC)OC)ccc(F)cc1C C(=O)(CC1=CCN(C)CC1)NC1C(CNC(C(=Cc2cccnc2)C)=O)C1 C(=O)(CCCOCC)NC1C(C(N(C(C)CN(C)C)CCC)=O)CC1 C1(C#N)(OC)CC(C(=O)NC2(CC(=O)NC3CCN(C)C3)CC2)C1 C1(C(N2CCC(C(C(=O)NCC(C=C)(C)C)F)C2)=O)CC(=O)C12CCC2 c1(CC(=O)NC(C(=O)N(CC)CC)c2ccco2)cccnc1F N1(C(C(C2CCC2)OCC)=O)CCCN(C(C2CCCN(CC(F)F)C2)=O)CC1 c1(SC)nn(C)cc1C(=O)NCCC1CCN(C(c2cnn(C)c2C)=O)C1 O(N1CCC(c2nnnn2CCCOC)(NCCCC2CCOC2=O)CC1)CC C(=O)(CC(C)C(F)(F)C(F)(F)F)NC(CNC(c1c(C)nnn1C)=O)C c1(CC(=O)NCC(CCO)c2ccccc2)cc2ccccc2s1 C=Cc1ccc(C(N2CCC(C3OCCC3NC(=O)C(C)CCCC)CC2)=O)cc1 c1(C(=O)NC(CNC(c2cc(C)n(C)n2)=O)(C)C(C)C)cccc2nn(C)cc12 NS(=O)(=O)c1cc(C(=O)N)c(Cl)c(F)c1.C12CC1CN(C(c1ccoc1)=O)C2 N1(C(C2(N(C(C(C)C#N)=O)C)CC2)=O)CC2C(C1)C2(F)F c1(C(N(C)CC2CCN(C(C(n3ncc(C)c3)C)=O)CC2)=O)occ2c1CCC2 c1(C(C(=O)NCC=CCNC(C(CC)C#N)=O)C)cc(C)cc(F)c1 N1(C(C2CCCC(NC(c3cn(C(C)C)nc3)=O)C2)=O)CCC(O)C(C)(C)C1 CC(C)(Cc1cccc(Cl)c1)C(=O)NCCC1CCN(C(=O)C(N)=O)C1 CCCC(F)C(=O)NCC(CC(=O)NCC(C)CC1CC1)OC N#CC1CC12CCN(C(c1coc(CNC(=O)C(C3CCCCC3)O)n1)=O)CC2 CCCC(O)CNC(=O)C(Cc1cnc[nH]1)NC(=O)CC1CC=CC1 CC1=NOC(C(=O)NCc2cc(C(=O)NCC(C)(O)C3(C)CC3)n[nH]2)C1 C1(C#CC(=O)N2CCC(C(N3CCC(N(C)CC)C3)=O)C2)(CC)COC1 CCCC(C)(O)C(=O)NC1CC(CC(=O)NCCc2[nH]cnc2C)C1 CC1(CNC(=O)CC2CCCC23CC3)CCCN1C(=O)CCn1ccnn1 Cc1nc(N2CCC(CF)(NC(c3cc[nH]n3)=O)C2)c2cc[nH]c2n1 c1(CNC2(C#N)C(C)CCC2)cc(S(C)(=O)=O)co1 C1(C(N2CCC(N(C(c3ccc(Cl)o3)=O)CC)C2)=O)COC(C)(C)C1 C1(N(C(CC2(C=C)CC2)=O)C)CC2CCC(C1)N2C(c1cnc(C(C)C)o1)=O N1(C(C(CCSC)O)=O)CC2(CCC2NC(=O)CN(C(=O)C(C)C)C)C1 N1(C(C(C=C)(C)CC)=O)CC(NC(c2cccnc2OCC)=O)C2CCCC2C1 N1(C(=O)CC2C=CCCC2)CCCC(CCNC(C2(C(F)F)CCCC2)=O)CC1 CC1=C(C(=O)NCC#CCNC(c2cnn(C(C)(C)C)c2Br)=O)CCCO1 Nc1cc(Cl)ncc1C(=O)NCC1(CC)CC1.C1(F)(C(=O)N)CC=CCC1 CCCCC(C)CCC(=O)NC1CC(NC(C2CC(Cl)(Cl)C2)=O)C(O)C1 C1(NC(C#CC2(C)CC2)=O)CN(C(=O)C(O)C2CCCC2)C2(CCCC2)C1 Cc1cc(C)cc(C=CC(=O)NC2CC(NC(c3occc3F)=O)C2)c1 Cc1ccc(C(=O)N(CC(C)NC(=O)CC(F)(F)C(F)F)C)c2c1NCCC2 c1(C(C)C)cc(=NC(C)CN(C)C(C2CC2C2CCCC2)=O)[nH]c(C(C)C)n1 c1(NC2CC(OC)C(OC)C2)ncnc(N2CCCN(CC(N)=O)C2)c1C c1(C(C(=O)NCCCOC)N(C2CCOC2=O)C)ccnc(Cl)c1OC CCCCCC(C(=O)NCC1(NC(=O)C2=C(Cl)CC2)CC1)C(C)C CC1CCN(C(=O)Cn2cc(CO)nn2)CCN1C(C1(C)CCN(C)C1=O)=O C12(C(N3CCC(N(CC#C)C(c4ncc[nH]4)=O)CC3)=O)CCCCC1OCC2 C1(C(=O)OC)CN(C(C23CNC(C)(CO2)C3)=O)c2ccccc2O1 C1(C(=O)OC)C(NC(=O)COC(C)C)CCCN1C(C1CCCO1)C CC(C)C(C(C)C)C(N)C(=O)N1CC(=O)Nc2ccccc21 Cc1ncc(CCC(N2CC(O)(C(F)C(=O)NCCC3(C)CCCO3)C2)=O)o1 c1(C(=O)Nc2ccc(N3CCN(S(=O)(=O)C4CC4)CC3)cn2)ccc(Cl)c(Br)c1 CC(C)(C)C(CO)C(=O)NCCOCCCNC(=O)CC1OCCC1(C)C C1(S(C)(=O)=O)(C(N2CCC(CC=C)C2)=O)CCC1.C1(C=C)(CC=O)CC1 N1(C(c2ccc(COC)o2)=O)CC2(C=C(C(=O)NCCO)CO2)C1.C1CC1 N1(C(C2CCCSS2)=O)CCC2CCC(C1)N2C(c1ncc(Cl)nc1Cl)=O C1(C2CC2)(NC(=O)Cc2ccsn2)CCN(C(c2cccc(F)c2F)=O)C1 Cc1ccc2c(c1)OC(C)CN2c1ncnc(=N)[nH]1 C1(NC(C(N2CC(C)C2)C)=O)CC(NC(c2sccc2F)=O)CC1O C#Cc1cn(C)nc1C(=O)NC(C)(C)C1CC1.c1(C=O)cc(C(C)C)on1 C1(CCNC(C2CCOC2)=O)CSCCN1C(c1ccc(N2CCC2)nc1)=O CC(C)C(F)(F)CC(=O)NCC1(O)CCCN(C(c2cnn3ccn(C)c23)=O)C1 C1(C(=O)NC(CCF)C(=O)NCCc2cncnc2O)CC2CCC1CC2 C(=O)(CC(C)NC(=O)C(c1cnn(C)c1)NC(c1ccsc1Cl)=O)NC c1(C(C)=O)cn(C)nc1C(F)(F)F.c12ccc(nc1)NC(=O)N2 Cc1ccc(C(N2CCCCC2CN2CCCC(C)CC2)=O)cc1C c1(C(=O)NC(C2CCN(C(C=CC=CC)=O)C2)C)n[nH]c2cc(Cl)ccc12 c1(SC)cc(F)ccc1C(N1CCCCC1C)=O.C(=O)(C(C)(C)c1cnsc1)N CC(C)C(C)CCNC(=O)CCOC1CC1.c1(CC(=O)N)ccc(F)cc1 C1(C(N)=O)(CNC(c2conc2C2CC2)=O)CN(C(C2CC2F)=O)C1 C12(C(=O)NCCOCC(=C)C)CC(CCO1)N(C(=O)Cc1ccoc1)C2 C1(CN(C(=O)Cn2ccnn2)CC)CCCCN1C(c1cccc(F)c1)=O N1(C(C2CN(C)C2)=O)CCC(S(C)(=O)=O)C1.C1(C)(C(=O)N)CC2(CCC2)C1 C(=O)(CC(C)(C)N(C)C)NCC1(CNC(CC2CCC(C)C2)=O)CCC1 Cc1cc(C(=O)NCCNC(C2(N3CCOCC3)CC2)=O)ncc1C#N C1(C=O)CCn2cnnc2C1.C1(NC(CC2(OCC)CCC2)=O)C2CCCC12.N C1(NC(C(C)OC)=O)CCCC(NC(=O)Cc2c(C)n[nH]c2C)C1 c1(C(N2CCC(CNC(C(C(CC)C)OC)=O)CC2)=O)ncsc1S(N)(=O)=O c1(OC)cccc(S(=O)(=O)N2CC(F)(F)C2c2ccc(F)cc2)c1 c1(C(N2CC(CC(=O)OC)C2)=O)ccon1.c1(C=O)cnn(C2CC2)c1.C Cc1nc(N2CCCC(NC(C3(CO)CC3)=O)C2C)ncc1Br c1(OC)ccc(C(=O)N(C)CC2(NC(=O)CCCC)CC2)cc1C(C)C.S CCCC(O)C(=O)N1CCC(C)(CNC(=O)CCc2nc(=N)[nH][nH]2)C1 c1(OC)ccc(-c2cncc(C(N3CCC(N(C(=O)C=CBr)C)C3)=O)c2)cc1 CC(C)CC(C(=O)NCCn1cc(C)nn1)N(C)C.C(=O)(CCCC1CC1)N n1(C(CC)C)ncc(C(N2CC(Oc3ccccc3Cl)C2)=O)c1C C1(NC(c2ccc(O)cc2)=O)CC2CCC1N(C(c1ncc(Br)cn1)=O)C2 Cc1cccc2[nH]cc(C(=O)NC(CCC3CCCC3)C(C)(C)C)c12 C12(NC(C(CCC)C)=O)CCOC(CNC(c3cccc(C4CC4)n3)=O)(C1)C2 CC1CN(C(=O)CCc2cncc(F)c2)CCC1NC(c1ccn(C2CC2)n1)=O c1(CN(CCNC(CNCCC=C)=O)CCOC)noc(-c2ccsc2)n1 N#Cc1ccc(Br)cc1CN1CC2C(C(=O)Nc3cc(C(N)=O)ccc3Cl)C2C1 N1(C(CCOC)=O)CCCCC1C(C)(C)CNC(=O)C(F)(F)C1(O)CCCC1 c1(C(C(=O)NC2CC(OC)C2)NC(=O)CN(C)C2CC2)ccnn1C C1(NC(C(=O)OCC)=O)(COC)CCCN(C(c2ccc(F)nc2C)=O)C1 C1(C(N(CC(=C)C)C)=O)CCC(C2CC2)N1C(c1ncc(OC)cn1)=O c1(C(=O)NC2C(C)(C)C(C(=O)Nc3ccc(O)c(F)c3)C2)cccn2nccc12 C1(C(=O)NC2CCN(c3n(C)ccn3)C2)OC2CC1CN(C(=O)O)C2.C(C)(C)C C1(N(C)C(c2ccco2)=O)C2CN(C(=O)C(C)(C)c3ccno3)CC12 C1(NC(CN2CC(C)CC(C)C2)=O)CCCC12CN(C(=O)COC)C2.C1CCC1 C12(C(N3CC(CCC)N(C(C4CCC5CCC45)=O)CC3)=O)C3CC(CC13)C2(F)F c1(OC)c(C(=O)NCC2CCN2C(C2CC2)=O)occc1=O.C1CCC1.C c1(N2CCN(C(c3nn(C)c(Cl)c3)=O)C(C(F)(F)F)C2)ncnc2c(Br)c[nH]c12 C1(C)(C(=O)NCC(N2CCOCC2)C)CCCCCC1.C(CC(=O)NC)=C.C1C(=O)N1 C1(CC(=O)NCC2(F)CN(C(c3c(C)onc3)=O)C2)CCC(=O)NC1 N1(C(CN(C)CC)=O)CC2(CCN(C(c3ccc(N)c(F)c3Br)=O)CC2)C1 C=CCC(C)(CC=C)NC(=O)C(c1ccccc1)NC(c1ccc(C)nc1)=O c1(CNC(C(=O)NCCOc2ccccc2Br)=O)ccccc1I c1(C(=O)NCCC2CCN(C(C(C(C)C)C)=O)C2)cc(=O)c2ccc(Cl)cc2o1 N1(C(c2c(CC)n(C)nc2)=O)CCCC(C)(C)C1CNC(=O)CC1CSC1 Cc1c(C(=O)N)cnn1C1CCCC1.N(S(=O)(=O)N(C)C)CC(N1CCC1)=O C(=O)(C(O)CC(C)C)NCCCN(CCCNC(c1cnc(CC)[nH]1)=O)C N1(C(CCCc2ccc(CC)cc2)=O)CCC2(CCCN2C(=O)C(O)C(F)F)C1 CC(C)CCC(F)C(=O)NCC(CNC(=O)C=Cc1cnccn1)CO C1(CC=O)OCCC1(C)C.C1(CNC(C2CC(CC)C2)=O)CC(F)C1.C c1(C=O)cc(C(F)(F)F)cc([N+](=O)[O-])c1.C1(C(N(C)CC)=O)C2CCC12.N C1(F)(CNC(C(C)OCOC)=O)CCN(C(C2(C)CCCC2)=O)CC1 O=C(C(F)CC1CN(C(=O)CN2CCCCC2)C1)NCCCC1CCCC1O C1(NC(c2ccsc2)=O)CC2CCC1(NC(c1ccccc1OCCF)=O)C2 CC(C)(C)C(CO)C(=O)N1CCC(C)(C)C(C(N2CC(O)C(N=[N+]=[N-])C2)=O)C1 c1(C=O)c[nH]c2cc(Cl)ccc12.C1(O)CCN(C(=O)CC2CS(=O)(=O)C2)C1.N c1(C(=O)NCC(CC=C)NC(=O)CC2CC3(CCC3)CO2)cc(C#N)ccc1C c1(C=O)ccc2c(c1)NC(=O)C2=O.C(C(C)C(=O)NCC1(C)CC1)OC C1(NC(c2cc(C)c(Cl)s2)=O)CCC2CCN(C(c3nccc4ccsc34)=O)C12 C12(CNC(CCCNC(C)=O)=O)CC(CN1C(C1COC(=O)N1C)=O)C2 N1(C(c2c(C)nccn2)=O)CCC2CCN(C(C3(O)CCCC3)=O)CC12 C1(CC(N2CCC(CNC(CC3(C#N)CCC3)=O)C2)=O)CCS(=O)(=O)C1 Cc1nn(C)cc1C(=O)NC1C2CC1N(C(C1CCCOC1)=O)C2 C#Cc1cnc(C(=O)NCC2COCC2)c(C)c1.c1(C=O)ccc(F)c(O)c1.N C1(N(C)C(c2ccc(Br)s2)=O)CN(C(c2c[nH]ccc2=N)=O)CC1O N1(c2sc(C(=O)OC)c(Cl)n2)CCC(NC(C2(C)CCCCCC2)=O)C(C)(C)C1 [N-]=[N+]=NC1CCCN(C(=O)C(CCF)NC(=O)CC2=CCOCC2)C1 c1(C(N2CCCC(CNC(=O)CC34CC(C3)C4)C2)=O)c(Cl)ccc(Cl)c1O CC1C(NC(c2ncccc2Cl)=O)CCCN1C(=O)COc1ccccc1O C12(C(=O)NCC(N(C(C(n3ncc(C)c3)C)=O)C)C3CC3)CC3CC1C2C3O N1(C(CC(C)C)C(=O)NCc2ccccc2)CC2CCCN2CC1CO C1(N(C(CC2(C=C)CN(C(=O)COc3ccsc3)C2)=O)C)CCN(C)C(C)C1 Cc1ccc(OCC(=O)NC2CN(C(C3(F)CCCN(C)C3)=O)CC2F)cc1F C1(NC(c2cnn[nH]2)=O)CCN(C(c2cncc(C(F)(F)F)c2)=O)CCC1CO CC(CC(F)(F)F)C(=O)N1CCC(C2CCCCN2C(=O)Cc2cn[nH]c2)CC1 C(C(C)N(C)N1CCSCC1)c1cccc(C)c1 C(=O)CC(C)(CN(C)C)C(F)(F)F.N1(C(C(CSC)O)=O)CCN(CC)CC1.N O=C1CCC(CC(N2CC(NC(c3cc(Cl)ccc3O)=O)C3(CC3)C2)=O)C(=O)N1 c1(C(N(CCN(C(C2CCCN(CC(C)C)C2)=O)C)C)=O)ccc([N+](=O)[O-])n1C c1(CC)cnc2ccccc2c1C(N1CC(NC(=O)CC2(CC=O)CC2)C1)=O c1(N(C)C)ccccc1C(=O)NCC1CCCN1C(=O)C=CC(N)=O N#CC1CCN(C(C23CC(CN2C(=O)CC2(O)CCCC2)C3)=O)C2(CC2)C1.C C1(CN(C(=O)CSCCO)CC)CCCCN1C(C1CC12CCCC2)=O N1(C(C2(CC=C)CC2)=O)CCCC(C(C)(O)C)C1.c1(C=O)cc(CCC)[nH]n1 C12(C(=O)NCC(CC)CC)CC(C)(C1)OC21CCC1.C1(CC=O)CCC(C)C1 c1(NCCC)cncc(C#N)n1.C1(C(=O)N)CCC12CCC2.C(C)(C)C.C=O C1(NC(Cc2c(Br)cc(C)s2)=O)C2CCNC2C1(C)C O=C(C#CCNC(=O)CCC1CCOC1)NCCC1CCCCC1 CCC(C#N)C(=O)NCC1CCN1C(=O)C(C)N(C)C c1(C(=O)NC(CNC(CCC(CC)C)=O)(C)C2CCC2)ccc2c(n1)CCCN2 N1(C(CC(=O)NC)=O)CCC(C)(C(N2CCCC2CC(=O)OC)=O)CC1 CCCCCC(F)C(=O)NC(CCC(C)C)C(=O)NC1CC(C)(OC)C1(C)C C1(CNC(CCS(C)=O)=O)(NC(c2occ3c2CCC3)=O)CC2CCC1CC2 N1(C(c2ncc(OC)cn2)=O)CCCC(NC(c2cc(F)ccc2Cl)=O)C1C c1(C(N(CCC)C)=O)cnc2c(cnn2C(C)CC)c1.C(CC(C)C(=O)N)OC C1(C(=O)NC2CC(=O)N(C3CC3)C2c2ccncc2)CC(O)(C2(O)CCC2)C1 C(=O)(C1CCCc2c[nH]nc21)N(C)CC1CCCN1C(C12CC(CO1)C2)=O C1(C2CCC2)(CNC(C2CC2C2CCCC2)=O)CCN(C(c2cn[nH]c2)=O)CC1 C(CCN(C)C)(C(=O)NC1CCN(CCO)CC1)NC(C(CC)O)=O C1(C(N2CCC(N3CCN(C(C=CC)=O)CC3)CC2)=O)CC(C)(C)CN1C C(C1CCN(C(C2CCCCS2)=O)CC1)=CC(=O)NCCCN=[N+]=[N-] O=C1CC(C(N2CC=CC2C(N2CC(F)C2)=O)=O)CCN1 Cc1ncc2n1CC(C(=O)N(CCC(C)NC(=O)CCCC(=O)N(C)C)C)CC2 C1(C(=O)NCC2CCCN2C(C2CCC(n3ccnn3)CC2)=O)CCC(F)CC1 C(=O)(CC=C(Cl)Cl)N1CC(CC=C)(NC(=O)CC2(C)CC2(F)F)C1 C1(O)CCOC1C.c1(CNC(C(C)OCCOC)=O)cc(C(=O)N)co1 c1(C(=O)OC2CC(CCC(=O)OC)C2)ccc2c(c1)NC(=O)C(C)S2 C#CCCCCCC(=O)N1CCCC(O)(CNC(=O)C(C)NC(C2CCC2)=O)C1 Cc1ccc(OCC(N2CCC(CNC(=O)O)C2(C)C)=O)cc1C.C(C)(C)C C1(NC(C(CC)N(C)C)=O)C=CCN(C(c2ncccc2N)=O)C1 C1(C)(C(N2C(C)(CC(=O)NCC#CC3CC3)CC2)=O)CCC(=O)NC1 C(CC(CC)(CC)NC(=O)C(C(C)C)OC)NC(c1n(C(CC)C)ncc1)=O C1(C(CNC(c2ncc(C(=O)OC)c(C)c2)=O)=O)C2CC3CC(C2)CC1C3 c1(C(N2CCCC(NC(c3cnc(C)[nH]c3=N)=O)C2)=O)cnc2onc(C)c2c1 C1(C(=O)NCC2CCC(NC(C(C)SC)=O)CC2)CCOC2(CCCCC2)C1 CN1CCn2cc(C(=O)NCC(C3(O)CN(C(=O)C(C)(F)F)C3)(C)C)nc2C1=O c1(C(N(CC(CNC(C(F)OC)=O)C)C)=O)cc(F)c(Br)c(F)c1N C=C(C)CN=C(NCc1cc2ccccc2s1)NCC1CN2CCN1CC2 c1(C(N2CC(CNC(CC3(C=C)CC3)=O)(OC)C2)=O)ncc(Br)cc1F N1(C(Cc2cnc(C)o2)=O)CCCC2CN(c3ccnc4nc(C)nn34)CC12 c1(C(C)(C)C)cc(C(=O)NC2CC(F)C2)on1.c1n[nH]c(O)n1.C(=O)C.C N1(C(C(C(=O)OC)OC)=O)CCC(C(=O)N(C)Cc2cc(C)on2)CC1C Cc1cc(O)c(C(N2CCC(C)C2CNC(c2cc3c(s2)CCC3)=O)=O)cc1F c1(C(N2C(CCNC(c3scnc3Cl)=O)CCC2)=O)ccc2nc(S)oc2c1 C1(C(N2CC3C(NC(C(C)N(CC)CC)=O)(C3)C2)=O)CCN(C)S1(=O)=O CC(C(F)C(=O)N1CCCC1CNC(c1cnoc1)=O)C(F)(F)F c1(-c2c(C(N(CC)Cc3ccncc3)=O)c[nH]n2)c(F)cccc1F c1(NC(CNC(=O)NCCC(CC)(F)F)=O)ccc(C)cc1C C1(NC(CC(OCC)OCC)=O)CCN(Cc2cccc(Br)c2Br)CC1O c1(C(=O)NC(CNC(C(C)n2cncn2)=O)C2CC2)cnc2ccccn2c1=O NC(=O)C(O)C(CC1(c2ccccc2)CC1)c1nc(-c2cccc(Br)c2Cl)no1 c1(C(C(=O)NC(CCOC)CNC(=O)CC2CCCCO2)=O)ccc(O)cc1 C(=O)(C(F)(F)C(C)O)NCC(C)CNC(c1ccc(CN(C)C)o1)=O c1(CCNC(COCC(=O)NC)=O)ccccc1.C1(C(=O)N)CCCCS1 c1(C(CC)O)nc(-c2ccnc(C(=O)OC(C)(C)C)n2)n(CC(C)O)n1 C=C1CC2(C1)CC(C(=O)NC(C)CCNC(=O)CC1CCC3CC13)C2 c1(CC=O)ccccc1.C(CCC)OC.C(C(C)(C)C)=CC=O.C(C)=O.N CC1(C)CN(C(=O)CNC(c2ccccc2Cl)=O)CCN(C(=O)C(C)(C)F)C1 c1(C(=O)NCC2(C)C(C)CN(C(CSCC=C)=O)C2)ccc(Cl)c(Cl)c1O C(CN=c1[nH]c(=NCC2CCOCC2(C)C)[nH]c2cccnc12)N(CCOC)C c1(CCC)ccc(N)c(C(=O)NCC(CCCC)NC(c2snc(O)c2Cl)=O)c1 CC(C)CC(C(=O)N1CCOC(C)CC1)ONC(C1(C)COC(=O)N1)=O Cc1ncc(C(=O)NCC2CN(C(C3CCC4CC4C3)=O)C2)c(C)n1 C(=O)(C1=CS(=O)(=O)CCC1)NCC(CN(C)C(C1C2CCOCC12)=O)O CC1(C)CN(C(=O)CC2CCC23CCC3)C(C)CO1.C1(CC=O)CC(=O)C1.N C12(NC(C3CSCC(=O)N3)=O)CCCC1N(C(=O)CCCCCF)CC2 C1(NC(c2cn(CCC)nn2)=O)CCN(C(=O)C(C(C)C)NC(N)=O)CC1O N1(C(C(C(C)C)O)=O)Cc2ccccc2C(NC(=O)C(C)(C)CC2CC2)C1 C(=O)(CC(C)C(F)(F)F)N1C(C=O)C=CC1.C1CCC(C(N)=O)CC1.COC C(=O)(CC(O)CCCC)NCc1c(C(=O)NCC2(CO)C(C=C)C2)n[nH]c1 C(=O)(CC(C)CCC=C(C)C)NCC1CCCN(C(C2N(CC)CC2)=O)CC1 C1CC2(CCN(C(=O)CS(=O)(=O)C3CC3)CC2)C1.c1(C(=O)N)cc(Cl)no1.C CCCCC(C(=O)NC(COC)C(=O)OC)NC(c1cnccn1)=O n1(CC2CN(C(C3C(CC)C3)=O)C2)cc(-c2cn(C)cn2)nn1 C1(CC)CCCCCCN1C(=O)CC(C)NC(=O)CCOCC1CCC1 C1(C(N2C3C(NC(c4ccnnc4)=O)CC(C3)C2)=O)CCc2nc(O)[nH]c2C1 Cn1ccc(C(=O)NCC2(C(=O)NC(CO)C3CCC3)CCCO2)cc1=O c1ccc(F)cc1C=O.C1(CC(=O)N(CC)CC)CCC(C)O1.CCO.CN C1(C(=O)NCC2(CNC(CC3CC(C)C3)=O)CCOCC2)CC12CCOCC2 c1(N2CCN(C(c3c(C)cnn3C)=O)CC2)ncc([N+](=O)[O-])cc1Cl c1(N(C)C(c2cnn(-c3ccccc3F)c2N)=O)ccc(OC(F)(F)F)cc1Br Cc1cc(C(N2CC(O)CC2CNC(C2CCC=CCC2)=O)=O)cc(C)c1F C#Cc1cccc(CC(N2CCC(C(F)CNC(=O)C(CC)CC=C)CC2)=O)c1 Cn1nc(C(=O)NCCc2cc(C(=O)Nc3ccsc3)no2)cc1F C(N=c1cc(C)n(C(C)(C)C)[nH]1)(C12COCC1C2(F)F)c1n(CC)nnn1 N1(C(CNC(C)=O)=O)CC(NC(c2ncc3c(F)cccn23)=O)C2CCCCC12 c1(CNC(C2C3CCC2(c2ccncc2)C3)=O)cccc(Cl)c1 C1CC2(CC2)CN1C(c1cc(O)nc(Cl)c1)=O.c1(C(=O)N)ccc(C2CC2)o1 C(=O)(CCC(C)(C)OC)N(CCC(C(C)C)NC(C(CC)N(C)C)=O)C C1(NC(C2=C(C)CCC2)=O)CC2CC1CN(C(=O)CCC(C)N(C)C)C2 C(=O)(C1=NNC(=O)CC1)NC(C)C(C)C.c1(C(=O)N)cn(CCO)c(=O)nc1O c1(CC)ccc(C)cc1C(=O)N(C)CC1CN(C(C2CC2F)=O)CC12CC2 N1(C(=O)Nc2ccc(OCCCC)cc2)CCCCc2ccccc21 c1(COCC(CN(C)Cc2scc(C)n2)O)ccc(F)cc1 Cc1cccc(C=CC(N2CCOC(C(=O)N(C(C)CO)C)C2)=O)c1 C(CCN=c1[nH]c(N2CC(=O)NC(C)(C)C2)nc2c1COC2)n1c(C)cc(C)n1 N1(CC(CC)OC)CCCC(COC)(NC(=O)Cc2ccc(Cl)s2)C1 C1(C(=O)OC)(CC)CCCN1C(=O)C(=O)NCC(C(F)(F)F)OC C1CC(C)(C)C1.C1(CC(N2CC(C(C=O)OCC)C2)=O)(OCC)CCC1 c1(OC)cccc(S(=O)(=O)CC(=O)NC(C)CC)c1.c1(C(=O)N)cn(C)cn1 C(CC(C(C)C)NC(=O)C(c1cccnc1)O)N(C(C(C)(C)OC)=O)C Cc1nc(NCC2CCC(F)(F)CC2)cc(NC2CCN(C3CC3)C2)n1 C1(CNC(CCCC)=O)CCN(C(=O)C(F)(F)CN2CCCC2)CCC1(F)F c1(CCC(=O)NC2CN(C(CC3(C#N)CCC3)=O)C2)cc2ccccc2[nH]1 N1(C(CC2C(C)CCCC2)=O)CCC(F)(CNC(c2[nH]cnc2C#N)=O)CC1 CC1CC(C(=O)NC2CC3(NC(c4nccc(Cl)c4F)=O)COC2C3)CCN1C C(=O)(C1=C(C)CCC1)N1CC(CCC)C(C(=O)NC(c2cnccc2C)C)C1 C(=O)(CC(C)C(C)C(C)C)N1CC(O)(CNC(C(Cc2c(C)cccc2)C)=O)C1 C1(CNC(C2OCC(C)(C)C2)=O)(CO)CCN(C(C2(Br)CC2)=O)CC1 c1(NCCC(CC)(C)C)ccc(S(=O)(=O)NCCCOc2ccccn2)c(Br)c1 C1(CNc2ccc(CC#N)nc2)Cc2ccccc2CN1 c1(N2C(CNC(C(C)OCCC(C)C)=O)CC3(CC3)C2)ncnc2ccccc12 N1(C(c2c(C)cccc2O)=O)CC2CCN(C(=O)C(C)(C)N(C)C)CCC2C1 CS(=O)(=O)c1ccc(C(=O)N)o1.C1(O)CCCN(C(=O)C=CC2CCOC2)C1 C1(CC)CN(C(=O)CC2CCCNC(=O)C2)CCN1C(=O)CS.c1cscn1.C c1(C(=O)OC)nc(=NC2CC(C)C2)cc[nH]1.C1(C=O)Cc2ccccc2S1(=O)=O.N c1(C(=O)NC(C(C(C)C)NC(c2cc(Br)c[nH]2)=O)C)cnc(C2CC2)nc1O N1(C(C=CC(C)NC(C2C(CCC)C2)=O)=O)CCCCCCC1 c1(C(=O)NC)cn(CC(=O)N)nn1.C(=O)(C(O)CN(C)C)N(CCCC)C Cc1ccccc1CCCO.c1(-c2cn(CC=O)nn2)ccc(F)cc1.C1CCC1(C)C.N c1(C(=O)NC2CC(N(C(CSCC)=O)C)C2)nn(C)c2c1CCCC2 Cc1cc(Cl)c(C(=O)NC(C2CCN(C(c3csc(C)n3)=O)CC2)C)s1 c1(C(C(=O)NC2CCN(C(C3(CC(F)(F)F)CC3)=O)C2)F)ccc(F)cc1 C12(NC(C3(NC(C(COC)N(C)C)=O)CC(CO)C3)=O)CC1COC2(C)C CC(C)CS(=O)(=O)CC(=O)N1CC(NC(=O)Cc2nc(=N)[nH][nH]2)CC12CCC2 c1(C(=O)NCC(C)N(C(=O)CC2CCCN2C)CC)ccc(=O)n(C)c1 C1(CNC(C(c2ccn(C)c2)C)=O)(NC(=O)CCc2ccncc2)CCCCC1 c1(C(=O)NC2(CCO)CN(C(CCCCC#C)=O)C2)cccc2c1CCO2 c1(CNC(C(CSC)C)=O)ccc(C)cc1F.c1(C(=O)N)cnc(Cl)c(N)c1 C1(C(=O)NC(C)CCNC(=O)CN2CCC2)(COC)CCCCO1 CC1CCC(C(=O)N(CC(C)C(C)(C)C)C)N(C(=O)C2=CCCC2C)C1 C1(CC=C)CCN(C(C2OCCC2c2ccccc2)=O)C1.C(=O)(C=C(C)C)N c1(C(=O)NCC(CCNC(CC2CC(C)(C)C2)=O)O)cccc(CO)n1 C(=O)(C1=NOC2(CCC2)C1)N1CCC(C(C)C(=O)NCC2CC23CC3)CC1 CCC(CC(=O)NC12CCN(C(c3oc(C)nc3C)=O)CC1C2)CC(C)C C1CCCN(C(c2cc(C(F)F)sn2)=O)C1.C1(C(N(C)C)=O)CCC1.C1CC1 CC(CCCN=c1c(C#N)c[nH]c2ccc(Cl)cc12)NC(=O)C=C1CCSCC1 c1(OC)ccc(C(C(=O)NCC(C)C)N(C)Cc2ccccc2OC(F)F)cc1 C1(NC(=O)CC2CC2)CC(C2CCN(C(=O)CCSCc3cccs3)C2)C1 CCC(O)C(C)C(=O)N1CCCC1C1CCN(C(C2(N=[N+]=[N-])CC2)=O)CC1 CCCCC(CNC(=O)CC1CCC2CC12)NC(=O)CSc1n[nH]c(O)n1 CC1(C(=O)NCC2=CCN(C(=O)C(F)(F)CCn3cccn3)CC2)CCC(O)CC1 N1(C(c2cc(C)sc2C)=O)CC(CNC(=O)CC(O)C2CCCC2)C2(CC2)C1 C1(CC=C)(NC(=O)CCc2nccn2C)CCN(C(=O)C(O)CC(F)F)CC1 CC(C)C1CC(NCc2cccc(OC(F)(F)F)c2)c2ccccc21 C=CC1(C(N2CCSC(CC)C2)=O)CCN(C(=O)Cn2c(C)ccc2C)C1 n1(CC(N2CC(C)(NC(c3c(N)ccc(CC)c3)=O)C2)=O)ncc2cccnc12 N1(C(C2(OC)CCCCCCC2)=O)CCC(NC(C2CCCS2)=O)C2(CCC2)C1 CC(CS(C)(=O)=O)C(=O)NC1CCOC(CNC(c2ccn3ccsc23)=O)C1 c1(C(=O)NCC2CC(NC(Cc3c(C)nc(S)s3)=O)C2)cnc2nccnc2c1 c1(C(=O)NCC(C)N(C(c2c(CC)non2)=O)C)cc(Cl)c(Cl)cc1O C1(C(N(C(C)C)C)=O)CN(CP(C)(C)=O)C1.Cc1nc(C=O)c(C)n1C1CC1 C1(C(=O)NC(C)CC(C)C)(OC)CCC(C(C)(C)C)CC1.c1(C=O)cnsn1 c1(OCOC)cccc(S(=O)(=O)NC(c2ccccc2NS(C)(=O)=O)C)c1 CCCC(C(=O)N(C1CCN(C(=O)C(CO)c2ccccc2)CC1)C)NC(N)=O C1(CNC(c2nc(C(C)C)sc2)=O)CCN(C(c2ccnc(Cl)c2O)=O)C12CC2 n1(CCN(C)C)cc(C(=O)NC2CCC2NC(C2CC(Cl)(Cl)C2)=O)nn1 C(C(C(=O)O)NC(=O)C(CC1CCOC1)NC(=O)OC(C)(C)C)OC c1(C=O)ccc(O)cc1C(F)F.Cc1csc(CCCC(=O)NC2CC2C)n1.N CCCCC(CN=c1cc(Cl)nc(-c2ccccn2)[nH]1)NC(=O)C(C)CN(C)C CC1(CC(=O)NCc2cn(C3CC3)cn2)CCN1C(=O)CC1CCC1 CC1C(C(=O)NC2CC2)=Cc2ccccc21.C(=O)(CN(C)C(=O)C1CC1)N Cc1ncc(C(=O)NCc2nc(C(=O)NC(C3CCCO3)C)co2)o1 CC1CCN(C(=O)C)CCN1C(C1CS(=O)(=O)CN1C(C)C)=O.c1nncs1.S N1(C(C(CC)OC)=O)CCC(O)(CN(C)C(c2cccn2C(C)C)=O)C1 C1(C(N2CC(NC(CSCCN(CC)CC)=O)C(F)C2)=O)OCC2CCCC12 c1(NCC(=O)NCC2C(NC(c3c(C)cns3)=O)C2)ccc(F)cc1Br O(P(C)(=O)CNC(C1CC(N(C(=O)C(CC)N(C)C)C)C1)=O)CC c1(C=O)c(OC(F)F)cccc1F.Cc1ccc(C=CC(=O)N(CC)CC)o1 c1(C(=O)NC2CCN(C(C(C)C(F)(F)F)=O)C2C2CC2)ccc2ccncc2n1 C(C(C)(C)C(C)O)NC(CC1CC(NC(C(C)NC(CC)=O)=O)C1)=O c1(C(=O)NC2CCN(C(c3ncc(C)c(C)c3)=O)C2)c(N)cc(F)cc1Br C1(CN(C(=O)C(C2CC2)C2CC2)C)CCCCN1C(=O)CC.C1CCCOC1 c1(C(N(CC(O)CN(C)C(C2(N(C)C)CC2)=O)C)=O)cc2sccc2[nH]1 N(C(=NCCc1ccc(F)cc1)NCC(F)(F)Oc1ccccc1)CC1(C)CC1 CCCCCC(CC)C(=O)NC1CCC(F)(CNC(c2ccc(CC)cn2)=O)C1 N1(C(C(SC)SC)=O)CCCCCC1C(=O)NCC1CC12CC2 C1(NC(C(c2nccc(C)c2)(C)C)=O)CCN(CC23C4C5C6C4C2C6C35)CC1O c1(CN2C(C(=O)NCC3CCSCC3)CC3CC32)c(O)ccc(F)c1F c1(C(=O)NC(CNC(CNS(CC)(=O)=O)=O)C2CC2)ccc(C)cc1N C1(N(C(C2C3C=CSC23)=O)CCc2ccccc2)CCC2(CC1)CNC2 CON(CCO)C(=O)C1(CNC(c2cccc(Cl)c2)=O)CCC1 C12(CNC(CN(C)CCO)=O)CCCC(CN1C(=O)CCCn1ccnn1)C2 c1(CN2C(CC(=O)Nc3ccc(C(F)F)nc3)COCC2)cnc(Cl)c(F)c1 C#CCCCCCC(=O)N1CC2CC(C(=O)NC3CCCCCC3F)CC2C1 C1(C(=O)NC(c2cn(Cc3ccno3)nn2)CCC)CCCN1C.C1CO1 c1(CC(=O)NC(C)CNC(=O)CN(C)C2CC2)ccc2c[nH]nc2c1 c1(C(N2CCCN(C(C(C=C)(C)O)=O)CC2)=O)ccc(F)c(C)c1Cl CC(C)(C)CC(=O)N1CC2CC1C2C(=O)NCC(O)CO C(CCCCCN=c1ccnc(CO)[nH]1)NC(C(c1ccc(F)cc1)CC)=O CON(Cc1ccccc1)C(=O)CCCNC(c1c(C)noc1C)=O N1(C(C(C)(C)NC(=O)NCC)=O)CCOCC(NC(c2cccnn2)=O)C1 N1(C(C2CC(=C)C2)=O)CCCCCC(NC(C2CC2C)=O)C1 c1(OC)c(C(=O)NC2(C)CCC2)csc1Cl.C1(C(=O)N)CC1.C(C)(C)C C(=O)(C1=CC2C=CC(C1)C2)N(C1CCCN(C(=O)C(C#N)(CC)CC)C1)CC c1cc(C)ccc1C.C1(CC(=O)OCC)CCC1.C1(=O)CCOC(=O)N1 C1(CC(N2CCC(NC(C(C(C)C)NC(C)=O)=O)C2)=O)Cn2ccnc2NC1=O C1(CC)CN(C(c2cc(C)n(C)n2)=O)CCN1C(=O)C.C(F)(F)C(F)(F)F C(=O)(CCC(=O)N1CCCCC1C1CCN(C(=O)CCc2nncs2)CC1)NC N1(C(c2c(OC)n[nH]c2)=O)CCN(C(=O)C(O)C2CN(CC)C2)CC1CSC c1(CC(=O)N)cc(F)ccc1O.O=C(CCCCNC(=O)C1CC1)NCCCO c1(CC(=O)NCCCN(C(=O)Cc2cnn(C)c2)C)coc2ccccc12 C1(C(N2CCN(C(CCCCC)=O)CC2)=O)CCCN(S(N)(=O)=O)C1 CS(=O)(=O)c1ccc(C(N2CC(C(=O)Nc3ccc(Cl)nc3Br)C2)=O)cc1 C1(NC(C(C2CCCC2)NC(C)=O)=O)CCCN(C(C2CCC=CO2)=O)C1C c1(CC(=O)NCC2CC(NC(c3cn(C)c(O)n3)=O)C2)cncc2ccccc12 N#Cc1cnc(N2CC(C(N)=O)(CNC(=O)C3=CCC3)C2)cn1 c1(CC)ccc(C(=O)NCC(CC)NC(C2CCCSS2)=O)cc1 N1(C(c2c(C)snc2)=O)CCN(C(C2CC2F)=O)C(C2CC2)C1 C(=O)(C(O)CC(N)=O)NCC(C(=O)NC1CCC(C)CC1)CC1CCCC1 c1(OC)nc(C(=O)NCCC2CCC2)cc(O)n1.C1(CC=O)CCCCC1O.N N1(C(CC=CCC)=O)CC(C2CCN(C(=O)CN3C(=O)CCC3=O)C2)C1 C1(NC(CC(C=C)C)=O)CCC(O)CN(C(c2cn(C3CCOCC3)nn2)=O)C1 C1(C(C)NC(C)=O)CCCCN1C(=O)CNC(C1CCCC1)=O.C1CC1.C C1(NC(CCc2ccc(OC(C)C)cc2)=O)CCN(C(=O)C(C)(C)O)CC1C N1(C(C=CCCC)=O)CCN(C(c2ccc(C3CCC3)nc2)=O)C(C)CC1C C1(CC=C)CC2CCC(C1)N2C(=O)C(C)(C)CCS(C)(=O)=O.C(=O)C=C C#CCC(C)(C(=O)NCC(c1ccccn1)C)NC(c1ccc(Cl)o1)=O N1(C(c2ncc(NC)nc2)=O)CCC(C)(C)C1.C1(C=O)CCC1.[SH](C)(=O)=O CCN=C(NCC(CO)N(C)C)N1CCCC(OC)C1 c1(C(N2CC(C)(NC(=O)CC3CCCO3)C2)=O)cc2ncccc2[nH]1 CCCC(C)(CC)C(=O)NCCCN(CCCCNC(=O)CC(C)SC)C Cc1cc(C)cc(C=CC(N2CC3CC2C3C)=O)c1.C1(C=O)CCSC(C)C1.N c1(N2C3CC(CN(C(c4cc(SC)oc4)=O)C3)C2)cc(Cl)nc(S(C)(=O)=O)n1 c1(-c2nc(C)[nH]n2)ccnc(-c2noc(CC3CCN(S(C)(=O)=O)CC3)n2)c1 O=C(C(O)C(F)(F)F)NCc1ccc(C(=O)NC(CC2CCCC2)CO)cn1 C(=O)(CCCC(F)F)NCC(CN(C(CNS(NC)(=O)=O)=O)C)O CC(C)(C)C#CC(=O)N1CCC(N(C(c2cc(O)nc(O)n2)=O)C)CC1.C1CC1 N1(C(CC=CCC)=O)CCOC(C2CN(C(C3CC=CC3)=O)C2)C1 CCC(CCCC(=O)NCC1CCOC1C)NC(c1nsnc1O)=O N1(C(C=C(C)C2CC2)=O)Cc2ccc(CNC(=O)C(F)C(C)C)cc2C1 CC1CC(C(=O)NCCN(C)C(=O)C2CC2)N1C(C1(C)CCCC1)=O Cc1scc(C(N2CC(NC(c3ccc(O)nc3)=O)CC2C)=O)c1Br C1(C(N2C(CN=[N+]=[N-])CC2)=O)CC2(CCN(C(C3(F)CCCC3)=O)C2)C1 N1(C(c2cn(CCCC)nn2)=O)CC(CNC(=O)C#CC(C)(C)O)CC12CCC2 c1(C(N2CCC(CNC(CC3C(C)(C)CC3)=O)C2)=O)c(O)nnc2c1CCCC2 C(=O)(CCn1cncn1)NC(C(=O)OCCC)C.C(=O)C(F)n1ccnc1.N C#CCC(C(=O)N(C1CCN(C(=O)C=Cc2ncc[nH]2)C1)C)C1CC1 C1(NC(N(C)Cc2nc(-c3ccccc3)no2)=O)CCCN(CP(C)(C)=O)C1 Cc1nnc(CCCNC(=O)CC2CC(NC(=O)CN3CCCC3=O)C2)n1C c1(C(N2CCC(O)(CCNC(C(C3CC3)OC)=O)C2)=O)nccc2c1NCCC2 c1(CC)c(Cl)nc[nH]c1=NCC1(C)CCN(C(c2nc(Cl)c(Cl)s2)=O)C1 CCC(CC(=O)NC1(C)CN(C(=O)C(F)CC2CCC2)C1)c1ccccc1 c1(CC(=O)NC(CN(C(Cn2c(C)cnc2)=O)C)C)c[nH]c2cnc(Cl)cc12 O=C1NC2(CCC2)C2(CN(C(c3cc(-c4ccc(Cl)cc4)on3)=O)C2)O1 C1(N(C)C)CCCC(C(N2CCC(N(C(=O)C(F)n3ccnc3)C)CC2)=O)C1 C1(C=O)CN2CCN1C(C)C2.c1(SC)ccc(C=CC(=O)NCC#CC)cc1.N C1(CSC)COC2(C1)CN(C(=O)C=CC(F)F)C2.C(C(C)C)NC=O c1(-c2c(C(N3CCCC(C#C)C3)=O)scn2)cc2c(C)cccc2[nH]1 CCCCCS(=O)(=O)CC(=O)NCC1CC(NC(C2CC3(CC3)CO2)=O)C1 C1(NC(c2sccc2Cl)=O)CCN(C(=O)Cc2cccc(C(F)F)c2)CC(O)C1 C1(C(=O)NC2C=CCN(C(=O)CCc3ccc(F)cc3)C2)CS(=O)(=O)CCO1 c1(C(=O)NCCCNC(C2CCCC(C(F)(F)F)O2)=O)ccn2ncccc12 Cc1cc(C(=O)Nc2cnn(C)c2C(N)=O)nn1C(C)(C)C N1(C(c2cc3cnccc3o2)=O)CC2CCCCC2(NC(C2CC(O)C2)=O)C1 CC(C)(C)C(C(=O)NC1(C)CCSC1)NC(c1cc(N)cc(F)c1)=O C1(C(NOCC2CC(=C)C2)=O)(NC(=O)C(C)C(F)F)CCCCC1 c1(OC)ccnc(C(=O)NCC2CCCC2NC(c2nccc(C)c2F)=O)c1N C(=O)(CC(O)C(C)(C)C)N1CCC(C)C(c2ccccc2)C1 Cn1ncc(CC(C(=O)NC2CC2(C)C)NC(c2cc(Cl)cs2)=O)c1O C1(C(=O)NCC(C(C)C)NC(CCc2cncc(C)c2)=O)CC2(C1)CC2(F)F c1(NCC)c(C(=O)NC(C)CNC(c2cc(OC)ccn2)=O)cccc1F N1(C(CC(=C=C)C)=O)CCOCC(NC(=O)C(C(C)C)c2cnc(C)s2)C1 C=C(C)CN=C(NCC(C)(C)C1CC1)N1CCCC2(CC2)C1 C(=O)(C1CCCn2nccc21)N1CC(CCCCN(C(=O)C(F)=CC2CC2)C)C1 CN1CCCCCC1C(=O)NCCCC1CN(C(=O)CC(F)(F)Cl)CCO1 Cc1cc(C(=O)N(C2CCN(C(C3CC(C#N)C3)=O)C2)CCF)ncc1CO c1(CC(NOC(CC)C)=O)cccc(CC2CC2)c1 C(=O)(CCCS(N)(=O)=O)NC1CN(C(CCCc2onc(CC)n2)=O)C2C1C2 N1(C(C#CC(=O)N(C)C)=O)CCCC2C(CCCN2C(c2cccs2)=O)C1 n1(CC=O)ccc2ccccc12.c1(CC(=O)NCC2(C)CC2)ccc(O)cc1 c1(CCC)cc(=NCC2CN(C(c3ccc4[nH]ccc4c3)=O)CC2C)[nH]c(Cl)n1 c1(C(N2CC(=C(CNC(Cc3n(C)ncc3Cl)=O)F)C2)=O)cnc(Cl)cc1Cl C1(NC(CC2OCC(C)(C)C2)=O)CCC(C)(CNC(=O)C)CC1.c1nccs1 c1(C(=O)NCC2(CNC(=O)CCc3cc[nH]n3)CC2)ccc(CF)cc1 c1(CNC(C)=O)cccc(NC(=O)Nc2ccc(C3(C)CC3)cc2)c1 CCC(C(=O)NCC(=O)OC)N(C)C(c1conc1C(C)C)=O C(=O)(C(C1=C(C)C=CCC1(C)C)N1CCN(c2nc[nH]n2)CC1)NCCOC N1(C(c2c(OC)cncc2)=O)CCC(NC(c2cnn(CCF)c2)=O)C12CC2 C(C1=CCN(C(c2cc(C)n(C)c2C)=O)CC1)NCC.C12CCC(CC1)C(=O)N2 c1(C(CCNC(C2C(CCC)C2)=O)=O)ccoc1C(C)C.C(C)(C)C.O C12(CNC(CC(C)C)=O)CCC(C1)N(C(=O)CN1CC=CC1)C2 C1(CNC(C2CC(=C(F)F)C2)=O)C2CN(C(c3ccc(=O)oc3)=O)CC12 N1(C(c2n(C)cc(C#N)c2)=O)CCC(N=[N+]=[N-])(C(N2CC(F)(CF)C2)=O)C1 C1(CNC(=O)NCCC2COC(C)(C)O2)CC2CCCC(C1)C2 N1(C(c2c(C)cc(C)[nH]2)=O)CCOCC(F)(C)C1.C1(CCC=O)CC(F)(F)C1.N C1(NC(c2c(C)cnnc2)=O)COC2(C1)CN(C(=O)CC1CCCCC1(C)C)C2 Cc1cc(C(N2CC(NC(=O)C=CC3CCOC3)C2)=O)c(C)o1 CC(C)(C)C#CC(=O)N(CC(=O)NCCOC1CC1(F)F)C1CC1 N1(C(C2CCC(NC(c3n[nH]c(CC)c3C)=O)CC2)=O)CC(O)CC(C)(C)C1 Cc1cc(C)nc(-c2cn(C(C)C(=O)NC3(C4CN(C(C)C)C4)CC3)nn2)n1 Cc1cc(C(=O)OC(c2ncc(C)o2)C)cc(S(C)(=O)=O)c1C C1(C)(NC(C2CCCCN(C(c3cc(C)nnc3O)=O)C2)=O)CN2CCC1CC2 c1(C=O)cnn(C)c1C1CC1.C1(NC(C2C(OCC)C2)=O)CCC1.C c1(CC(=O)NCCNC(c2ccc(OC)nn2)=O)cccc(C)c1C N1(C(CC(COC)(C)C)=O)CCC2CCN(C(=O)CC3COCC3O)CC12 C1(CC)CCC(C)CN1C(=O)CCCOCCO.c1(C(C(=O)N)C)ccn(C)c1 c1(NCC(C)OC)ncnc(N2CCC(c3cnccn3)C2)c1C Cc1ccc(C(=O)NCC2CCC(C)N(C(c3nn(C)cc3C)=O)C2)c(C)c1 c1(SC)c(C(N2CCCC2C(C)NC(=O)CCCCCC2CC2)=O)cccc1F CCCCC(C(=O)Nc1ccc(O)c(C)c1)NC(C1CCCCNC1=O)=O Cc1ccc(=N)[nH]c1C(N1CCCCC1CN(C(=O)C#CC1(C)CC1)C)=O Cn1ncc(CN2CC3CC2C3C(N2CCOC(c3ccccc3)C2)=O)c1Cl C1(C=O)CCc2cc(C)ccc2O1.C1(c2nc(C)cs2)CCN(C(=O)CC)C1.CC=O C#CCCCCCC(=O)NC1CCC1NC(=O)CCn1c(C)c(C)sc1=O n1(COC)ccc(C(=O)NC2CCCC2NC(c2cccn2C)=O)n1 CC1CC(NC(C2(C(F)(F)F)CC(F)(F)C2)=O)CN(C(c2ncccc2N)=O)C1 C1(C(=O)NC(CC#C)(C)C)CCC(C)(C)N(C(=O)C(CC)C(F)(F)F)C1 C1(CNC(c2cc(C)n(C(C)(C)C)n2)=O)CCN(C(C2C(C)C2C)=O)CC1 C=C(Cl)CC(C(=O)NC(COC)CCOC)NC(C1CC(C)(F)C1)=O c1(C(N2CCN(C(C(C)n3ccnn3)=O)CC2C(F)F)=O)n[nH]c2ccccc12 C1(NC(C2(CC#C)CC2)=O)COC2(C1)CN(C(=O)C(c1cccc(Br)c1)O)C2 C1(C(=O)NCC2(NC(C(CC)SC)=O)CCCCC2)CCCCN(C)C1=O C12CC(C)(CCO1)C2.Cc1cc(CNC(C2CN(C)CCO2)=O)oc1C=O.N C1(CNC(C(c2c(C)cccc2)C)=O)CC2(CCC2)CN1C(C1(CO)CC1)=O c1(C(N(CC(CC)NC(=O)C(C2CC2)C2CC2)C)=O)cccc(=S)n1O C(C)(N=c1[nH]c2c(c(=NC3CC=CC3)[nH]1)CCCC2)c1cc(OC)c(F)cc1 C12(C=O)CCC(CC1)C2(C)C.C=C(C)CCNC(=O)C(C)(C)N1CCCC1.N N1(C(C(C)N2CCC2)=O)CCCCC1CCNC(=O)CC1(C(F)F)CC1 N1(C(=O)C2=CCCOC2)CC2CCC(N=c3ccnc(CO)[nH]3)CC2C1 C=CCCCC(C(=O)N(C1CCC2(CC1)CC2)C)NC(=O)CCn1cnc(=N)[nH]1 CC(C)CC(CC(C)C)C(=O)NC1CN(C(=O)C(C)N(C)C)CCC1(C)C N1(C(c2c(CC)nc[nH]2)=O)CC(O)CC1C.N1(C(C(=O)N)=O)CCCC(C)C1 C(c1ccc(Br)c(Cl)c1)=CC(=O)NC(C)C(C)NC(C1CN(C)C1)=O c1(CN=c2c(C#N)c(-c3ccccc3)cc(C)[nH]2)ccc([N+](=O)[O-])cc1[N+](=O)[O-] C1(C(N2CCC(NC(C3C(=C)C3)=O)C(C)C2)=O)CC2CCC1CC2OC C1(NC2(c3ccc(Cl)cc3)CCC2)CC12CCC1(CC2)OCCO1 CCC(C)(C(=O)N1CCC(N(C)C(c2cnco2)=O)CC1)OC C1(C(C)C)CN(C(c2[nH]nnc2-c2ccccc2)=O)CCN1C(=O)CCC1CC1 C1CCCC2(CC2)C1.Cc1noc(C)c1CC(=O)NC1(C(=O)N)CC(F)(F)C1 C1(NC(CCC2N(C(c3c(C)nsc3C)=O)CCCC2)=O)CCOC(C)(CC)C1 CC(C)C(O)C(C)C(=O)N1CCC(C)(CNC(=O)C(C)NC=O)C1 C1(NC(c2ccc(C#C)nc2)=O)C2CC(O)C1N(C(C1(F)CC1)=O)C2 C1(C(=O)NC2C(C)(C(F)F)C2)C=CCCN1C(=O)CCOCC1CC1 C1(C(=O)OCC2OCCC(C)(C)C2)CN(C(=O)O)CC2(CC2)C1.c1ccccc1 c1(C(N2CCC(NC(C3(C(=O)OC)CC3)=O)C(F)C2)=O)c(Cl)cc(Cl)cc1Cl c1(C(=O)NC(C)CNC(C2CC=CC2)=O)cc2cccc(Cl)c2[nH]1 C1(N(C(C2(C)N(C(c3nc(CC)sc3)=O)CC=C2)=O)C)CC(C)CC(C)C1 C(=O)(C1=C(C)OCCC1)NC1CCCCN(C(C(C=C)(F)F)=O)C1 CC1COCC(C(N2CCC(NC(=O)CCn3cccc3)CC2)=O)O1 c1cccc(F)c1.C(=O)(CC)N(C)CC1(C)CC1.C(=O)(COC(F)F)N C(=O)(CCCC1CC1)N.C1(CC)CC2(CCC2)C1.C1(O)(C(C=O)F)CCCC1 C(=O)(C(CCCN)Sc1nc[nH]n1)NCC(C)(C)NC(=O)OC(C)(C)C c1(C(N2C3CC(NC(c4nc(CC)sc4)=O)C(C3)C2)=O)ccc2c(c1)CCN2C C1(CC)CN(C(C2CCC2COC)=O)CCC1.C1(CC(=O)N)CC(C)OC1C C1(NC(C(C2CCOC2)OC)=O)C(C)CCN(C(C2C3COCC23)=O)C1C n1(CCC(=O)NCC2N(C(c3n(C)ncc3)=O)CC2)nc(O)c2c1CCCC2 c1(CNC(=O)Nc2cccc(NC(CC)=O)c2)c(C)cccc1[N+](=O)[O-] C1(COC)(C)CCNCC1.c1(CC(=O)N)ccc(Cl)c(Br)c1.c1nnn(C)n1 c1(CC=O)cc(C)[nH]n1.C1(C(N(CCC)CC)=O)CCC(C(F)(F)F)O1.N c1ccc(C)c(S(C)(=O)=O)c1.C1(Cc2n(CC)nnn2)CCSC1(C)C.C1CC1 c1(C(N2CC(CCNC(=O)CC3CCCCCO3)OCC2)=O)ccc(O)cc1F C(=O)(CCC1=CCCCC1)N1C(C(N(C)CC2(C)CC2)=O)CC(O)C1 C(CCCCC(=O)NC1CC(O)C1)n1cc(COC)nn1 C1(CNC(C(CC)(C)CC)=O)CC12CCN(C(C1(n3cncn3)CC1)=O)CC2 Cc1onc(-c2cccs2)c1C(=O)NCC1CCCN(C(C2CCCOC2)=O)C1 C1(NC(C2(SCC)CC2)=O)CCN(C(=O)CCCCn2ccnn2)C12CC2 C1(C(=O)NC2C(C(=O)NCc3n[nH]c(C)c3C)CC=CC2)CN(C)CC(C)O1 CCC1=C(C(=O)NCC(CC)NC(C2CC2C(F)(F)F)=O)CCCO1 C=C(C)CCC(=O)NC(C)CCCCNC(=O)CCn1ccnc1C N1(C(Cn2c(C)c(Cl)cn2)=O)CCC2C(CCN2C(=O)C=CCn2cncn2)C1 CC(C)(C#N)CCC(=O)NC1CCCN(C(=O)Cc2ccc(Br)c(F)c2)C1 c1(C(C(=O)OC)(C)C)c(Cl)nc[nH]c1=NCC(C)(C)NC(c1cnn2c1CCC2)=O N1(C(C(CCC)O)=O)CCN(C(C2C3CCC2(c2cccs2)C3)=O)CC1C1CC1 c1(C(N2CCN(C(CNC(C3CC3[N+](=O)[O-])=O)=O)CC2)=O)c[nH]c2cnccc12 Cc1cc(NC(=O)CC2CCN(C(c3c(C)nn(C)c3C)=O)CC2C)cc(Cl)c1 C1(NC(c2cnc(C)[nH]2)=O)CN(C(c2nc(C(F)(F)F)cs2)=O)C(C)(C)C1 C1(C(=O)NCCC(C)C)C2CCN(CC2)S1(=O)=O.N1(CCC=O)CCCCC1.N c1(CC)cc(C(=O)N(C)CCNC(c2cc(C)nc(C)c2)=O)cn(C)c1=O C1(C(N(CC(O)C2CC2)C)=O)CCOCC1NC(C1CCCC(=O)C1)=O C(=O)(C1=CCCOCC1)N1C(C)CCC1C(=O)NC1CCC(=O)NC1 Cc1onc(CO)c1C(=O)NCCCN(CCO)C(c1cc(=O)cc[nH]1)=O Cc1ccc(C(=O)NCCCCC(C)NC(=O)Cc2ccc(Br)s2)nn1 O=C(CCCC(F)(F)Br)NCC1CC(NC(C2(CC3CC3)CCC2)=O)C1 C12(CNC(c3cc(C)ncc3)=O)CCCN(C(c3cncc(Cl)c3Cl)=O)C1C2 CC(c1ccco1)=CC(=O)NCC(O)C(=O)NCC1CCCC1N(C)C Cc1nccn1CCC(=O)NC(C)CCNC(c1c[nH]nc1-c1ccccc1)=O Cc1cc(C(=O)NCCCCNC(=O)C(c2ccccc2)C)cc(C)c1 c1(CN2CCC(N(C)C(c3scnc3C(F)(F)F)=O)C2)cc(Br)cc(F)c1F C12(CC)CCC(CC1)C2.c1(C=O)cc(C2CC2)on1.O=C(COCCCF)N C1(NC(C=Cc2c(C)cccc2)=O)CN(C(c2cnn[nH]2)=O)C2CCCC12 N1(C(c2c(C)cns2)=O)CC(CNC(C2(Br)CC2)=O)C2(CCC2)C1 c1(NC(CCC2CCN(C(CC(C=C)C)=O)CC2)=O)cnc(C)nc1C CN1CCC(NC(=O)NC2CC(Cn3cncn3)C2)C(C#N)C1 c1(C(=O)NC2C(NC(C(CC)F)=O)COC2)cnn(C(C)C)c1Br C1(CC)(CNC(=O)C(C)CC)CCC(=O)N1.c1(C=O)cocc1C(N)=O CC(C)(O)C(C)(C)C(=O)NCCOCCNC(=O)CN1CCC(O)CC1 C1CCOC1.C1(CC)CC1C(=O)N(CC(C)O)CCNC(=O)CO.C C(c1cc(Cl)ccc1)=CC(=O)N(C1CCCC(NC(CC(=O)OC)=O)C1)C.O C12(NC(C3(C)CCN(C(COc4cn(C)nc4)=O)C3)=O)CCN(CC1)CC2 C1(NC(C2CCCC(O)C2)=O)CCS(=O)(=O)C12CN(C(C1CCOC1)=O)C2 C1(CNC(c2cc(OC)no2)=O)CN(C(=O)C(C)CC2CC2)CCN1C c1(C(C)C)ocnc1C(=O)NC(C)C(C)NC(c1cnn(C2CCC2)c1)=O c1(C=O)cccc(S(=O)(=O)CF)c1.CC(C)CNC(=O)CSC1CC1.N c1(C(=O)NCC2CC(C)N(C(c3ccc(C(F)F)s3)=O)C2)cccc2nonc12 C(=O)(CC1=NNC(=O)C1)NCCOC1CN(C(C2CCN(C)C(=O)C2)=O)C1 CC(C)S(=O)(=O)C(C)C(=O)NCC1CN(C(c2ncc3ccccn23)=O)CC1O C1(C(=O)NC(C)C#N)CCC2(CN(S(=O)(=O)CC3CCC3)C2)O1 C(C(C)C(=O)NCc1ccn(C2CC2)n1)N(C(C(C)OCCC=C)=O)C c1(OC)ccc(N)c(C(=O)NCC(C)NC(=O)C=CC2CCCN2C)c1 c1(C(=O)NCC2C3CN(C(CCSC)=O)CC32)cccc(S(C)=O)c1 C12(CNC(CCCCCC)=O)CCCC1N(C(c1cn(C)[nH]c1=N)=O)CC2 CN1CC(N(C)C(C2(NC(=O)CCN(C)C)CC2)=O)CCC1=O c1(C(N2CCC(N(C(c3c(C)ocn3)=O)CCO)C2)=O)ccnnc1C(F)(F)F C(=O)(CC(C)C(C)(C)NC(C1COC(=O)N1)=O)NCc1ncc(CC)[nH]1 C1(NC(Cc2c(C)cco2)=O)CC2CCC1N2C(C1COCCO1)=O C1(C(=O)NCCN2CCN(c3c(C)c(Cl)ncn3)CC2)CCC2C(CC1)C2(F)F Cn1cnc2nc(Cl)[nH]c(=NC3CCCCN(C(c4ccc(F)nc4)=O)C3)c12 C1(C(N2CC(CCNC(CC(C)(C)O)=O)OCC2)=O)CCCCN1S(N)(=O)=O C1(NC(c2ccc(F)cc2Cl)=O)CN(C(=O)C=CCF)Cc2ccnn2C1 c1(C(C(=O)OC)C)ccc(NC(=O)NCc2ccc(C)c(C)n2)c(C)c1 C(=O)(C(O)CCC(C)C)NC1CCC(NC(CCc2c(C)noc2Cl)=O)CC1 c1(CC=O)c(C)nn(C)c1C.C(CCCNC(c1ccoc1C1CC1)=O)OC C1(C(N(C2CCCCC2)CC#C)=O)COCCN(CC2CCC(OCC)CC2)C1 N1(C(C(C=CC)O)=O)CCC(C)C(CNC(C2CC2C(=O)OC)=O)C1 c1(C(N)=O)cccc(C(=O)NC(Cc2cccc(Cl)c2)CO)c1 C1(O)(CNC(CC2CC(NC(C(C)CN(C)C)=O)C2)=O)CC2CCC1C2 Cc1nc(CC(=O)NC(C(=O)NC(C)CCCO)C2CCC2)cs1 c1(CC(=O)NCc2ccc(OC)nc2NC(C)C)cnc2cccnn12 C1(C(=O)NCC)(C(N2CCC2)=O)CCSC1.C1CCOC1.C(=O)(CO)N N1(C(C(CC)O)=O)CCN(CC2CN(C(=O)COCC3CCOC3)C2)CC1 N1(C(CC(C=C)C)=O)C2CCC1CC(NC(c1noc3c1COCC3)=O)C2 C1(C(C=O)(C)C)CCCN(C(c2ncn(C(C)(C)C)n2)=O)C1.C1(C(C)=O)CC1 C1(CNC(=O)C=Cc2cc[nH]c2)CCCC(NC(=O)CO)C1.C1CC=CC1 C1(NC(C(CC)(C)C)=O)CN(C(c2cccc(C)c2F)=O)C2(CCOC2)C1 c1(C(N(CCNC(CC)=O)C2CC2)=O)nsc2ccccc12 C1(NC(CC(C)(C)O)=O)CN(C(C2COC(=O)N2)=O)CC1(C)C C#CCC(C(=O)NC1CCCCC1C(=O)NCCC1CC=CCC1)C1CC1 C1(NC(CC(C=C)CC)=O)CCC2(CC1)CC2Nc1ncncc1I c1(OC)ccc(Cl)c(F)c1C(=O)NC1CCN(C(C2OCCO2)=O)CC1O N1(C(c2ccc(CC)cc2N)=O)CC2(CCN(C(=O)CC(C)n3cccn3)C2)C1 c1(C(N(C)CC2CCCN(C(C=C(C)C)=O)C2)=O)cc(Br)cc(C)c1F CCC(CC(F)(F)F)C(=O)NC1CCCC(NC(=O)CCn2cnnn2)C1 C1(NC(CCCC(N)=O)=O)CN(C(=O)CCCC(F)F)CC1C1CC1 c1(C(N2CCC(O)(CN(C(=O)C(C)(C)CO)C)CC2)=O)cc2cc(F)ccc2[nH]1 c1(C(=O)NCCC(C)NC(=O)Cc2nc[nH]n2)ccc2c(c1)OC(F)(F)O2 C1(C(=O)N)COCCN1C(C)C.c1(CCNC(CC(=O)OC)=O)ccccc1Cl C1(NC(c2c(C)ccc(C)n2)=O)CCSC12CN(C(=O)CCCN(C)C(C)C)C2 C(C)(C)(C(C)NC(c1ccco1)=O)NC(C1CC1)=O.N1(CC)CCCCC1 c1(C(=O)NC(C)CNC(=O)C(Cc2ccccc2)C2CC2)ccnn(C)c1=O c1(OC)ccc(Br)c(N)c1C(=O)NCC(C)N(C)C(c1ccc(O)nn1)=O c1(NC(c2nc(C)sc2C)CC)cccnc1OC(F)(F)F c1(Cc2n(CCOCC=C)c(N3CCC(F)C3)nn2)ncc(F)cc1F c1(-c2ccc(C(=O)NCC3CN(CC=O)C3)o2)ccc(Br)cc1.[nH]1ccnn1.C c1(C(=O)NC2CCN(C(c3c(CC)ncnc3)=O)C2)ccc(OC)c2ccnn12 C(=O)(C1=NOC(c2ccccc2)C1)N1CCC(C(C)NC(CCC(C)(C)C)=O)C1 CC1(C)Oc2ccc(NC(=O)CCc3cnccn3)cc2O1 C1(CNC(=O)NCC2(C)CCCC2)CCCCC1n1cccn1 C1(CNC(C2(C)C=CCCC2)=O)CCCCN(c2ccncn2)C1 Cc1cn2c(n1)CC(C(=O)NCCCCC1CC1)C2.C1(C(=O)N)CC2CCC2C1 c1oc(C)c(C)c1S(C)(=O)=O.c1(C(C)NC)cn(Cc2ccc(C=O)o2)nn1 N1(C(CC(=C)C)=O)CC23CCCC2(C1)CN(C(=O)C1=CN(C(C)=O)CC1)C3 CCCCC(CC)CC(=O)N1CCC(O)(CNC(c2scc3c2CCCC3)=O)C1 N1(C(COCCC=C)=O)CCC2(CC1)CCN(C(c1sccc1C1CC1)=O)CC2 N1(C(C2(CC(C)C)CC2)=O)CCC(C)N(C(=O)C(O)C2CCCC2)CC1 c1(NCC(CC=C)(C)CO)ccc(S(=O)(=O)NC(CO)CC(C)(C)C)c(Cl)c1 C(CN=c1ccc(F)c(C)[nH]1)NC(C(CCC)CCC)=O O=C(CCCC(F)(F)CO)NC1CCC2CN(C(c3cc(O)cs3)=O)CC2C1 N1(C(c2c(C)occ2)=O)CCCC(O)(CN(C)C(c2cc3scnc3[nH]2)=O)C1 C(C)(CCC(C)(C)C)(c1nnnn1C1CCCCC1)NCc1c(C)c(Cl)ccc1 N1(C(c2cccc(CC)c2O)=O)CC2CC(C1)CN(C(C1(CF)CC(=O)C1)=O)C2 C1(CNC(C(CC)n2cccn2)=O)(OC)CCN(C(C2(C3CC3)CCC2)=O)CC1 C1(CC=C)CCCCN1C(C1CCCCC1NC(=O)CN1CCOC1=O)=O Cc1c(F)ccc(Cl)c1C(=O)NC1CN(C(=O)COCCOCCO)C1 c1(CC)c(NC(CNC(C2(C)CC(O)CN2C)=O)C2CCC2)ncnc1Cl N1(C(c2cc(C(C)(C)O)on2)C(=O)N)CC(C)(C)OCC1C.C(=O)(CC)OC C(=O)(C(CNC(=O)CC(=O)OC(C)(C)C)C(C)(C)C)NC1CC(C)C1 O=C(CCCCC(F)F)N1CCN(C(c2ccc([N+](=O)[O-])o2)=O)C(CCO)C1 C(CNC(=O)C(C)c1ccsc1)(C(=O)NCC1=NOCC1)OC C1(C(N2CCCC(C(C)C)CC2)=O)N(C(C2CC(C)(C)CO2)=O)CC12CCCC2 CC1C(C(=O)NC2CN(CCF)C2)CCCN1C(C1CCC1)=O C(CC(=O)NCC(CO)C1CC1)(C(F)(F)F)NC(CC(C)(C)OC)=O C1(CNC(CCN(CC#C)C(c2sc(F)cc2C)=O)=O)CCCCN(C)C1 C(=O)(C(C)C1=CCCC1)N1CC(C)N(C(=O)C(=O)NCC2CC2)CC1 N1(C(C(CCN(C)C)O)=O)CCN2CCN(C(C3CCC=CCC3)=O)CC2C1 c1(C(=O)NCC(C)NC(=O)CCc2cnco2)ccccc1OC1CC1 C1(CN(C(C(C2CCOC2)OC)=O)C)CCN(C(=O)C=CC=C(Cl)Cl)CC1 c1(OC)ccc(C(=O)NCC2CCN(C(=O)CC3(O)CCCC3)C2)cc1F.C C1(NC(CC2(C=C)CC2)=O)CCCCN(C(c2ccc(CS(C)(=O)=O)cc2)=O)C1 N1(C(c2cc3ncccn3n2)=O)CCC2(CC1)CN(C(C1CCS(=O)CC1)=O)C2 N1(C(C(C)OCC=C)=O)CCN(Cc2ccc([N+](=O)[O-])cc2)CC1C#N N1(C(C(CC)O)=O)CCC2CN(C(c3cc(C)cc(Br)c3F)=O)CC2C1 N1(C(c2c(CC)cccn2)=O)CCC2(NC(=O)CCCC3CCC3)CC2C1 CC(C)C(=O)C(=O)NC(C)C(=O)NCCOc1cnn(C)c1 Cc1cc(=O)oc(C)c1C(=O)NC.c1nccc(O)n1.C(=O)C=C1CCC1 C1(C(=O)NC2CC(C)(NC(C(C)n3cncn3)=O)C2)CCOC2(CCC2)C1 N1(C(C(Cc2cc[nH]n2)NC(c2cc(CC)no2)=O)=O)CCOC(CCO)C1 CC1CN(C(C23CSC(C2)C3)=O)CCCN1C(C1CC(=O)NC1(C)C)=O Cc1cc(Cl)ncc1CC(=O)NC1COCCN(C(c2cccn2C(C)C)=O)C1 C1(NC(=O)C(O)CN2CCCC2)C=CCN(C(=O)CN2C(=O)CCC2=O)C1 C1(c2nc(-c3ccc(OCC)cc3)nn2C2CCC2)CCc2c[nH]nc2C1 C(=O)(C(F)C(=O)NCCN(C(C1(C)CCCCO1)=O)CC)OCC c1(CN2CC3(CC(C(=O)NCC4(Br)CCC4)C3)C2)cc(F)c(Br)c(F)c1 C1(CNC(c2c(C)c[nH]n2)=O)CN(c2ccc(C(C)=O)cn2)CCC1(F)F Cc1cccnc1CCNC(=O)COC1CCN(C(C2CCC(=O)N2)=O)C1 C1(CNC(C(CC)OC2CCCCC2)=O)CN(C)CCN1C(=O)C.C(C)(C)C c1(CC)c[nH]nc1C(=O)NC(C)C=CC(=O)NCCC1CCSC1 c1(OCCCC)ccc(CNC2CCC(C(=O)Nc3ccncn3)CC2)cc1 C1(C(N(CC(N2CCC2(C)C)=O)C(C)C)=O)CC(=O)NC1(C)C.COC N1(CC)CCC(NC(=O)C(O)C2CN(C(c3cc(C)no3)=O)C2)C1 C12(NC(CC3N(C(CSCC=C)=O)C4CCC3C4)=O)CC3CC(CC1C3)C2 CC1(C)CN(CC(N2CCCCC2)=O)CC1NC(C1CCC(F)(F)CC1)=O CC1(C(=O)OCc2nnc(C3CC3)n2-c2ccccc2)CCS(=O)(=O)CC1 C1(C(=O)NC2C3CN(C(=O)CN4CC5CC5C4)CC23)C2CCC3C(C2)CC13 c1(C(N2C(C)CC2C(=O)NCc2cnn(C)c2O)=O)cnn2ccccc12 C1(C(=O)NCC2(NC(C3CC(=O)C3)=O)CCC2)COc2cc(F)ccc2C1 Cc1ccc(Cl)cc1C(N1CC(N(C)C(c2cc(O)cs2)=O)C(C)(C)C1)=O c1(CC)nc(CCNC(=O)CNC(=O)C(C)(C)OC(C)=O)n[nH]1.C N1(C(CN(CC#C)C(c2ccn(C)c2CC)=O)=O)CCSCC1C N1(C(C(CCSC)N(C)C)=O)CCCC(O)(CNC(=O)C(c2ccccc2)=O)C1 CC1C(NC(C2(C)CC2C)=O)CCCN1C(c1cn(-c2cccc(Cl)c2)nn1)=O Cc1ccc(C(=O)NC2(CCO)CN(C(=O)CN3C(=O)CN(C)C3=O)C2)cc1O C(C)(C(C(=O)NCC1CCC1)SC)SC.c1(C(=O)N)c(C2CC2)noc1C Cc1ocnc1C(N1CC(c2ccccc2)C1CO)C(=O)NC(C)C n1(C2CCCN(C(C=CC)=O)C2)cnc2c1CCN(C(C1CC(=O)N(C)C1)=O)C2 c1(CNC(C=C(C)C)=O)nn(C)c2c1CN(C(=O)Cc1cn(C)nc1Cl)CC2 Oc1ccc(C(c2nnnn2-c2ccccc2Cl)NCCC2CCCC2)cn1 c1(CC)cccc(CC)c1CC(=O)NC1CCC1.C1(C#N)(C(=O)N)CCSCC1 CC(C)(C#N)CC(=O)NCCC1CCCN(C(c2cnc(S)nc2)=O)C1 Cc1ccncc1C=CC(=O)NC1CC(CNC(=O)CC2CCC(C)C2)C1 CCC(CC)(CO)C(=O)N1CC2CCCC2(CNC(C2CCC2)=O)C1.C(C)=O.N Cc1nc2ccccc2nc1C(c1nnnn1C)NC(C)Cc1ccccc1Cl C1(NC(c2c(C)scc2)=O)CC(NC(=O)C(C(C)C)n2cncn2)CC1O C1(C(N2CC(O)(C(F)C(N3CCOCC34CC4)=O)C2)=O)CC2(CCCO2)C1 C(=O)(CCCC(=O)N)NC(C)C.C1(O)CCN(C(=O)CC2CCC(=O)O2)C1.C c1(OC)cc(OC)cc(N2CCC(NC(C3CCC(OC)CC3)=O)CC2)c1 C=CCC(CNC(c1[nH]nnc1C)=O)C(=O)NC(CC1CCCC1)CO N1(C(c2n(C)nc(C(F)F)c2)=O)CC2(C1)CN(C(=O)CCS)CCO2.CC(N)=O C=C(C)CCNC(C1(C(F)(F)F)CC1)=O.C1(C(C=O)C)CCC(=O)N1.N C(C(C(=O)NCc1ccc(Cl)cn1)C(C)C)NC(C1C(CC)N(C)CC1)=O C1(CNC(Cn2c(C)ncc2)=O)CCN(C(c2cc(Cl)c[nH]2)=O)CC1 c1(C(=O)OC)nsc(=NC2CC(C)N(C(=O)CCc3ccccc3Cl)C2)[nH]1 CCCCS(=O)(=O)CC(=O)NCCCOCCCNC(=O)CCCCOC N1(C(CC2(COC)CCC2)=O)CC(C(N2CCOC(C3CC3)C2)=O)OC(C)C1 c1(C(N2C(C)CC(NC(c3c[nH]c(=N)o3)=O)C2)=O)cc(Cl)c(Br)cc1F c1(C(=O)NCC(C(C)(C)C)NC(C2CC3CC3C2)=O)ccc(N)cc1F N1(C(CCCC(C)O)=O)CCCC(C2(NC(=O)C=Cc3ccc(Cl)nc3)CC2)C1 c1(C(=O)NC(CC(C)NC(C2(OCC)CCCC2)=O)C)nc2cccnc2s1 Cc1cc(Br)c(S(=O)(=O)NCCC(CCO)C(=O)O)c(Br)c1 c1(CNC(CNC2CCN(C(CC(C)SC)=O)CC2C)=O)cc2ccccc2o1 C1(COC)(C)CCCN1C(C1CCNC(=O)C1)=O.c1(C(=O)N)ccc(Br)o1 C1(C(=O)NC(Cc2cc(C)[nH]n2)C)CC2CCN(C(C3CNCCOC3)=O)CC12 C(=O)(C(CC)N(CCCOC)CC1CCOCC1)NCCC c1(OC)cc(CCC(N2CCC2(C)Cn2cc(C(C)O)nn2)=O)ccc1Cl c1(CC)c(C(=O)NC2CCC2CC(N2CC(C(=O)OC)C2)=O)cnn1C c1(CC)cccc(C)c1CNC1(C(c2nnnn2C2CCCC2)SC)CCOC1 CC(C)CC(C(=O)N1CCN(C(=O)C=C2CCSCC2)C2COCC12)C(C)C Cn1nccc1C(=O)NC1CCC(CCNC(=O)C(C)(C)C2CCC2)C1 C(C(F)(F)C(=O)N(CC(C)(C)NC(=O)C(C1CCOCC1)O)C)N(C)C N1(C(CCCOCCC)=O)CCC(NC(=O)Cc2cnsc2)C2(CCC2)C1 Cc1sc(C)c(C(=O)NC2CCN(C(c3ccc(Cl)cc3Cl)=O)C2)c1C#N C12(NC(=O)CCN3CCC3)CCN(C(c3c(O)cccc3F)=O)CC1C2 N1(C(Cn2c(C)c(O)c(=O)cc2)=O)CCC2CCN(C(c3cnc(S)[nH]3)=O)C2C1 C=CCC(C)(C)CC(=O)NC(CCC)CC(=O)N(C1CCOC1)C1CC1 Cc1ncc2n1CCC(C(=O)NCC(C)N(C)C(c1ccccc1C(C)O)=O)C2 Cn1cnc(CNC2CCCC2Cc2ccc(O)cc2)c1Cl N1(C(C(c2c(OC)cccc2)O)=O)CCN(C(=O)CO)C(C)C1.C1(F)CC1.C c1(CC(=O)NCC(CC)NC(c2ccccn2)=O)c(C)nn(C(F)F)c1C.N CC(C)CCC(F)C(=O)N1CC=CCC1C(=O)N(C)CCC1CCOCC1 c1(C(N(C2CCCN(C(c3cnco3)=O)C2)C)=O)cnc(-c2ccccc2)cn1 c1(CC)cc(C(N2CCCC2C)=O)n(C)n1.C12(C=O)CCCC1(C(N)=O)C2.C O=C(C1=CCCCO1)NCC1CCCCCN1C(=O)Cn1nc(Cl)ccc1=O c1(C(N(C)CC2(NC(C(C)NC(CC)=O)=O)CC2)=O)coc(CO)c1 Cc1cc(NC(=O)CN2CCN(C(=O)Cc3cccc(Br)c3)CC2)nc(Cl)c1 C(=O)(CC(C)(C)CNC(c1cc(CO)[nH]n1)=O)NCC(C(C)O)O c1(C(C)C)nc(=NCCCCC(C)NC(c2cc3ccccc3[nH]2)=O)s[nH]1 N1(S(C)(=O)=O)CCCC1C=O.C1(O)(CC)CN(C(=O)C)C1.C1(C)CCC1 CS(=O)(=O)c1ccccc1C(O)CNCc1cccc(I)c1 Cc1c(NC(=O)CN(C)Cc2nnc(C)s2)c(O)nc(=O)n1-c1ccccc1 CC1CCc2sc(C(N3CCC(CNC(c4cnc(Cl)[nH]4)=O)CC3C)=O)cc2C1 C(Cc1cc[nH]n1)(C(=O)N=c1ccn(C(F)F)[nH]1)NC(=O)CC1CC1 C(=O)(CCC(C)C)NCCn1ncc(C(=O)NC(COCC)C)c1 CC1CCC(=CC(=O)NC2(CO)CN(C(c3ccccc3)=O)C2)CC1.C(C)C.N N1(C(c2ncn(CC)c2)=O)CCC2(CCN(C(C3CN(C(C)C)CCO3)=O)C2)C1 c1(C(N2CCC(CN(C(=O)C(F)(F)CC3CC3)C)C2)=O)cnc(S)nc1 C(CCC(C)C(=O)N1CCC(C)(C)C1CNC(c1cc(Cl)ncc1O)=O)OC C1(C(=O)NCCCOCCC=O)(CC)CCCCO1.C1CC1.C(=O)C1CC1 N1(C(CNS(CCCC)(=O)=O)=O)CCCC(N(C)C(c2cnc(C)cn2)=O)CC1 Cc1cnc(C#N)nc1N1CCOC(CNC(=O)C(F)C(C)(C)O)C1 N1(C(c2c(C)ccc(N)c2C)=O)CCC2(CCN(C(=O)Cn3ccnc3C)C2)C1 C(CCO)(C(C)C)NC(C1(C(C)NC(=O)CCC2CCCO2)CC1)=O c1(CNC(N2CCCC(C(C)=O)C2)=O)csc2ccc(Br)cc12 C1(C(N2CC(OC)C(NC(=O)CCn3cncn3)C2)=O)CCOC(=O)CC1 CC1(C)CCCCC1(C)NC(=O)CCc1cccnc1 C=C(C)C1OCCCC1C(=O)NC1(C)CCN(C(C2(c3ccnn3C)CC2)=O)C1 C(=O)(C(F)CC(CC)CC)N1CCC(C(=O)NC(C#C)CC)(C(C)C)C1 CC1(O)COCCN(C(=O)C(C2CCC2)NC(C2CN3CCN2CC3)=O)C1 N1(c2snc(CCC)n2)CCCC(N(C(=O)CC(C)(C)C=C)C)CC1 N1(C(c2cn(C)nc2)=O)CCN(C(c2cc(CC3CC3)on2)=O)C2COCC12 C1(NC(c2n(CCCC)nnn2)C2(n3cccn3)CC2)CC2(CCCC2)C1 C(=O)(CCS(C)(=O)=O)N(C)C.c1(OC)ccccc1CC(=O)NC1CCCCC1 C1(C(N(C)Cc2cn[nH]c2)=O)CC(O)CN1C(C1CSCC(=O)N1)=O Cc1cc(C(=O)NC2C3CN(C(=O)Nc4c(C)cccc4Cl)CC23)cc(F)c1 CCCCCC(C(=O)NCC1(C)CC1)C(C)C.c1(C=O)cncc([N+](=O)[O-])c1.N CCC(CC)(CC)C(=O)NC1CN(C(c2cn(C)ccc2=O)=O)CC2CC12 C1(C(=O)NC(CCCOC)c2nn[nH]n2)C2CN(Cc3ccccc3)CC12 c1(COC)cc(C(=O)NCCCC2COC(C)(C)C2)n(C)c1 C1(C(=O)NCCN(C2CCCC2)C(c2ccc(C(C)C)s2)=O)CN(C)CC1C C1(NC(C(C)OCCOC)=O)CCC(C)(C)CC1.c1(C(=O)N)cncs1 Cc1cc(Cl)nc(N)c1C(=O)NCC(CO)NC(c1ccc2nn[nH]c2c1)=O CCC(CCC(=O)N1CCN(C2CN(C(=O)C(C)OCCOC)C2)CC1)OC C(=O)(CC(C)(C)CC(F)F)NC1C(SC)CN(C(=O)CSC(F)F)C1 c1(-c2nc(SCC(=O)NCC3CC(F)(F)CO3)on2)cccc(Cl)c1 C1(CCC)(CO)CCCN1C(C1CC(F)CN1C(=O)CCNC(C)=O)=O CC(C)C(C(=O)N1CCCC(O)(c2ccc(Cl)cc2)C1)C(C)C C1(C(=O)NC2C=CCN(C(CN3C(C)CCC3C)=O)C2)CCC2(CC1)CC2(F)F c1(C(=O)NCC(CO)NC(C(C)NC(c2ccoc2)=O)=O)ccn(C)n1 c1(C(=O)NCC2C(C)CCO2)ccnc(CNC(=O)C(C)(O)C2CCC2)c1 Cc1cc(-c2nc(COC(C)C)nn2Cc2cccs2)nnc1C Cc1cncc(C(=O)NCCC2CCOC2)n1.C(=O)CC(F)(F)F.C(=O)(C)N CCCCC(=O)C(=O)N1C(CC(N2CC(N(CCC)CC)C2)=O)C2CCCC12 C(C1=CCCN(C(=O)CCC(N)=O)C1)NC(C1(OC)CNC(=O)C1)=O CC(C)(CNC(C1CC(=O)CCO1)=O)CC(=O)NCC1CC12CCC2 n1(CC(N)=O)nc(-c2cnn(CCO)c2)nc1-c1nc(Cl)sc1Cl C1(CNC(C2(C)CC(C)C2)=O)CCC12CCN(C(=O)CC#N)CC2 c1(C(N(CCNC(C2(C=C)CCOCC2)=O)C)=O)ncnc2cc[nH]c12 Cc1coc(C=CC(N2CCCCC2CNC(=O)Cc2cc[nH]n2)=O)n1 c1(CC)nocc1C(=O)N(CCCNC(=O)CC1CN(C)C1)CCO C1(C(=O)Nc2c(N(C)C)cccc2)CC2CCC1N2C(=O)CC(Cl)Cl C1(C)(C=O)CCC(=O)NC1.C(=O)(CC(C1CC1)C1CC1)N1CC(CC)C1.N CCCC(C(=O)NCC1(F)CCC1)N(C)C.c1(C=O)nn(C)cc1C=O.N N1(C(C(c2ccccc2F)OC)=O)CCC2(CCC(C(=O)O)CC2)CC1 c1(C(C)C#N)cccc(C(N2CCC(O)(C(N3CCCC3C(N)=O)=O)C2)=O)c1 N1(C(C2C(C)(C)C2(F)F)=O)CCCCC(C2CN(C(=O)CC3CC=CC3)C2)C1 C(CO)(C(F)(F)F)NC(=O)C(=O)NCC1(F)CCC1 c1(C(N2CCCN(C(c3c(CC)[nH]cc3)=O)CCC2)=O)ccc(Cl)c2occc12 C1(C(=O)NCC2CC(CNC(C3ON=C(CC)C3)=O)C2)CC12CCCCC2 C12(CC(=O)NCc3c(SC)cccn3)CCC1CN(C(=O)C(F)F)C2 c1(C(=O)NC2CN(C(=O)C3=COCCC3)CC2O)ccc2c(c1)CCCC2 C1(N(C(c2ccccc2)=O)CC)CCCN(C(=O)C(c2ccc(F)cc2)F)C1 C(=O)(C1=C(C)OCCS1)NCCC(=O)N(c1cnn(-c2ccccc2Br)c1)CC c12cn(C(=O)OC)c(n1)OC(OC)CCNC(=O)N2.C(C)(C)OCC C1(C)(C(=O)NC2CC(C3CCN(C(CCSC)=O)C3)C2)COc2ccccc2O1 c1(C(=O)NC2C(NC(C=COCC)=O)COC2)ncncc1C c1(CNC(C(=O)NCC(N2CCCC(C)C2)(C)C)=O)cnn2c1OCCC2 Cc1nc2cc(CN3CCOC(C(=O)OC(C)(C)C)(CO)C3)ccc2n1C1CC1 C1(C2N(C(CCOC(C)=O)=O)CCC2)CCCN(C(C2(O)CCC2)=O)C1 C1(NC(C(C)NC=O)=O)CC(NC(C2(CO)CC(C)(C)C2)=O)CC1O C(=O)(CCCCc1cnn[nH]1)NC(CCNC(C1CC(C(C)C)C1)=O)C C1(C(=O)N(C2CCCCC2)CCO)CN(C(C23CCN(CC2)C3)=O)CCC1(F)F C1(CNC(C(=O)NCCC(N)=O)=O)CCCCN(C(=O)C(F)C2CCC2)C1 N1(C(C(C)Oc2ccccn2)=O)CCCC(N(C)C(C2CC=CCO2)=O)CC1 C1(OC(C)C)CCN(C(C2CCC2CNC(C2CC2(F)Cl)=O)=O)CC1 C1(C(N(CCC(C)NC(c2cccc3cncn23)=O)C)=O)CC2CCC(C1)N2C C(=O)(C(F)C(C)C)N1CC(C)(NC(CCCOCC=C)=O)C1 Cc1nc(O)sc1S(=O)(=O)NCC(=O)OC1(c2ccccc2)COC1 C1(NC(Cc2c(C)ccs2)=O)CC2CC(NC(=O)Cn3cnnc3)C1C2 Cc1nc2c(Cl)cccc2cc1C(=O)Nc1c(C)cc(C#N)cc1Cl Cc1c(Cl)ccnc1C(=O)NC1CC2CC(NC(c3ncc(F)cn3)=O)C2C1 c1(C(=O)N)cnc2c(n1)CCCC2.N1(C(C(CC)NC(C)=O)=O)C(C)C2CC1C2 C1(C(=O)NCC2=CCCN(C(C(CC#C)O)=O)C2)CC1C1CCOCC1 C(=O)(C1=NOC2COCC12)N1CCCCC(N(C(=O)C(C2CCCCC2)F)C)C1 C#Cc1ccc(C(N2CCN(C(C)CNC(c3ccncc3)=O)CC2)=O)nc1 N1(C(c2cc(OCC)ns2)C(=O)NCCCSC)CCC2(CC(=O)N(C)C2)C1 C1(NC(=O)CCN2CCOC2=O)C2COCC1CN(C(=O)COCC)C2.CCO.O c1(CC)nn(C)cc1C(=O)NCC(C)OCC(=O)N(CC(C)C)C Cc1ncc(CN(C)C(c2csc(CNC(=O)CC3(C)CCOC3)c2)=O)s1 N1(C(C(C)N2CCC2)=O)CCC2C(CCN2C(c2cccc(C(F)F)c2F)=O)C1 C(=O)(C(CCC)C(=O)OCC)NCCCCNC(C1(CC#C)CC1)=O CC(C)C(O)C(C)(C)C(=O)NC1COCC1NC(c1ccnn1C1CCCC1)=O CC1(C)C(CNC(=O)C)CCN1C(c1cnn(C2CCOCC2)c1)=O.CCF.O c1(-c2nc(-c3ncc(NC)nc3)on2)ccc2c(cnn2C)c1 N1(C(CNC(NCC)=S)=O)CC2COCC(C1)N2C(c1ccc(C)c(C)c1)=O C1(C(N2CC(NC(C3CN(C)C3)=O)C(CO)CC2)=O)CC2OC(C)(C)OC2C1 C1(NC(C2(CO)CC(C)(C)C2)=O)CC2(CCN(C(c3cccc(Cl)c3)=O)C2)C1 N1(C(Cc2onc(C)n2)=O)CCN(C(c2ccc(Cl)cc2F)=O)CC12CC2 N1(C(c2c(C)nc[nH]2)=O)CCC2(CCCN2C(c2ccc(Cl)c(F)c2N)=O)C1 N1(C(CC(=O)NCC)=O)CCC2CCN(C(=O)C=CC3(C)COC3)CC12 C#CC1COCCN1C(=O)NCCC1CCC2(CCC2)O1 CC1(NC(=O)C(F)=C2CCCC2)CC(NC(=O)COC(F)(F)F)C1 c1(OC(C)C)cccnc1C(N1CC(N)CC1C)=O CC1(C(=O)NCCC2CCCN(c3nc(C4CCCC4)ns3)C2)CCC(F)(F)C1 c1(C(=O)NCC2CC(NC(C(CCCC)O)=O)C2)c(C)cc(N(C)C)cc1C C#Cc1cc(Br)cc(OC(F)(F)F)c1C=O.C1(CS(C)(=O)=O)CC(F)(F)C1.N C1(C(=O)NC2CC(NC(c3nc(Cl)cs3)=O)C2)CCOC1c1ccccc1 C1(C(=O)O)(CC)CCCN(C(C2(C)CCN(C(c3cnn4c3OCC4)=O)C2)=O)C1 C(CNC(=O)C(F)F)(CC(=O)NC1(C(O)CO)CCC1)OC N1(C(C(C)=C(C)C)=O)CCC(C2CCCN(C(c3cccc(Cl)c3C)=O)C2)CC1 Cc1nc2c(N3CCC(CNC(C4Cc5ccccc5C4)=O)CC3)ncnc2s1 C1(OC)COc2c(C(=O)N(C(C)CNC(=O)CC#N)C)cnn2C1 N1(C(C2ON=C(C)C2)=O)CCC(C(=O)Nc2cccnc2C)C(C)(C)C1 C1(CC(=O)NC(CCNC(C(CC)Sc2ccccc2)=O)(C)C)CCC(=O)N1C N1(C(c2nn(C)c(F)c2)=O)CCC2(C1)CN(C(=O)C(F)=C1CCC1)C2 C1(C(=O)NCCOCCN(C(=O)C=C2CCOCC2)C)CCN(C)C1=O C(=O)(CCCC(C)C)NCc1cn(CC(=O)N(C23CC(C2)C3)CC)nn1 Cc1ncc(C(=O)NCC2CC(C)CCN2C(=O)CCCF)c(Cl)c1Br c1(OCC)cccc(CC(=O)NCCC2CCCCC2)c1.C1(C(=O)N)CCCO1 C1(NC(c2c(CC)con2)=O)CCN(C(c2scnc2CC)=O)C(C2CC2)C1 N1(C(C2(C#C)CC(=O)C2)=O)CCC2(CC1)CC2C(=O)NCCc1cc[nH]n1 C12(C(=O)NCC3(C(=O)O)CC3(F)F)COCC1CN(Cc1ccccc1)C2 c1(CC)ccc(C(=O)NC2CCCCC2NC(=O)Cc2cc(OC)no2)cc1Cl Cn1nnc2c(NC3(C)CC(NC(=O)CN4CCCCC4)C3)ncnc12 C1(N(C(N2CCC(C=C)C2)=O)CCN(C)C)CS(=O)(=O)CC1N1CCCCC1 CC1CCC2(CC1)CCN2C(=O)C(Cc1cnc[nH]1)NC(=O)C(O)C(C)(C)C C(=O)(C1=C(Cl)CCCC1)NCCN(C(=O)Cc1ccc(Cl)nc1F)CC C(C1=CCN(C(C2CC2c2ccncc2F)=O)CC1)NC(c1nnn(C)n1)=O O=C(C1=CCCSC1)NC12CC1CN(C(c1csc(-c3ccc(F)cc3)n1)=O)C2 C1(C(=O)NC2CCCC2CN(C)C)(NC(C(C)OCC)=O)CCOCC1 c1(C=O)cc(C#N)ccc1C.Cc1cc(COCC(N2CC=CC2C)=O)on1.N C1(NC(CC(=O)Nc2nccs2)=O)CN(C(c2ccccc2)=O)CC1F c1(C(N2CC(C(C)NC(c3c(C)cccc3)=O)OCC2)=O)c(C)cc(=O)oc1C c1(N(C(C2CCN(C(C3OCCN(CC)C3)=O)CC2)=O)CC)ncc(Cl)c(O)n1 c1(CC(=O)NCCCCNC(C2(F)CCCOC2)=O)coc2ccccc12 C1(OC)CC2CCC1(OCCC1CCC1=O)CC2 CC(C(=O)N1CCC1C(=O)NCCOCCC(C)C)c1ccsc1 C(=O)(C(F)C(C)(C)O)N1C2CC(C1)C2.CC(CCOc1ccccc1)C(=O)N c1(CC)ncc(Br)cc1NC(C1CCCCNCC1)=O N1(C(C2(O)CCNC2)=O)CCc2nc[nH]c2C1c1ccc(F)cc1 C1(CC(N2CC(C(=O)NC)C2)=O)CC2(C1)CN(C(=O)CN1CCCC1C)C2 N1(C(C(C)=CC)=O)CCN(C(=O)C(C)C(C)C)CC1 C1(C(N2CC(OC)(C)C2)=O)OCCOC12CCC2.c1(C=O)ccc([N+](=O)[O-])s1.N Cc1cc(F)cc(C(=O)NCC(O)CCNC(c2c(N)cc(Cl)nc2Cl)=O)c1C c1(C(=O)NCC2N(C(C(=O)NCC)=O)CC(OC)C2)ccccc1.CC C1(CC)CC(C(=O)NC2(CNC(C3CC(CC)=NO3)=O)CCC2)CCC1=O C1(CC(=O)NCC(C(C)C)NC(c2ccc(=O)oc2)=O)CCC(F)(F)CO1 c1(C(=O)NCC2N(C(=O)CC3CC3)CCN(C)C2)nnc(O)c2ccccc12 C1(SCCCN(C)Cc2n(CC)cnn2)CCS(=O)(=O)C1 CCC(=O)CCC(=O)N1C(C(=O)NCc2ccncc2Cl)CCC1C1CC1 C#CCC(C(=O)NCCCCSC)NC(=O)CCCN(C)C(C)C C1(NC(c2cn(CCC)nn2)=O)CCCCCC1C(=O)NCCc1nncs1 N1(C(c2ccnn2C)=O)CCCC(C2CN(C(=O)CN3CC(C)(C)C3)C2)C1.CS c1(OCC)ccc2cc(C(=O)NCCCCNC(=O)C(F)OC)[nH]c2c1 C1CN(C(=O)CNS(=O)(=O)N(C)C)CC1N=[N+]=[N-].C(C(=O)N)N(CC)CC c1(C(=O)NCC2(O)CCN(C(C3(CC#C)CC3)=O)C2)c(C)oc(C)c1Br C1(C(C)(C)C)(CNC(=O)Cc2ccco2)CCN(C(c2ccc(O)cc2)=O)C1 c1(OC(C)C)ccc(C(=O)NCCCCNC(=O)CCC(C)CN(C)C)cc1F N1(C(C(=O)N(C)C)=O)CCC2CN(C(=O)Cc3cccc(F)c3F)CCC12 c1(OC)c(C)cc(Br)c(C)c1NC(=O)Nc1ccc(OCC(C)C)nc1 C(=O)(C(CC)C(F)(F)F)NC(CCN(C(C(CCC)F)=O)C)C(C)C C1(O)(CNC(c2c(C)scc2)=O)CCCN(C(=O)C(O)C2CC2)CC1 N1(C(C(C(CC)(C)C)OC)=O)CCCC2(C1)CN(C(c1ccc(C)c(F)c1)=O)C2 N1(C(C(C)Cc2ccccn2)=O)CCCCC1CNC(c1cnn(C)n1)=O CC1NC(=O)CCC1c1noc(CCCCCCCNC(=O)NC(C)(C)C)n1 C12(COC)CCOC1CN(C(=O)Nc1nn(C)cc1S(C)(=O)=O)C2 C1(NC(C=CC(C)C)=O)CCC2(CCCN(C(=O)Cc3cnnn3C)C2)C1 C1(CNC(C2COCCN2Cc2cnco2)=O)CCc2ccccc2O1 C1(C)(CC)CCCN(C(=O)C=CC2CCN(C(c3cc(C)nn3CC)=O)CC2)C1 N1(C(c2cc(C(F)F)on2)C(=O)NC(C(=O)OC)C)CCOC(C(C)C)C1 Cc1cnc(NCCOCCCO)c(S(=O)(=O)N(C)Cc2scnc2C)c1 C1(CNC(c2ncoc2C)=O)CCC2(CC2)CO1.C1(C(=O)N)CCNC1=O C1(O)(CCNC(CSCC=C)=O)CCCN(C(=O)C(F)OC(F)(F)F)C1 c1(NC(c2nc(N(C)C)nc(O)c2)=O)c(Cl)cc(Cl)c2nsnc12 C(c1ccco1)=C(C)C(=O)NCCCN(C(C1CCC(C)C1)=O)C(C)C c1(-c2scc(C(N3CCC(NC(CNC=O)=O)(CF)C3)=O)n2)c(F)cccc1F C1(CC(N2C3CC(C3)C2)=O)CC(C)(C)C(=O)N1.C1(NC)CC(C=O)C1.CC CC1=C(C(=O)N2CC(C(F)(F)F)C(C)C2)CCC(C)(C)C1.C(=O)C=CCO C=CC(C)(C)CC(=O)N1CCC(O)(CN(C)C(c2nc(Cl)sc2Cl)=O)C1 N1(C(CN2CCC(C)CC2)=O)CC2(CC2)CC1C(=O)Nc1cnnc(O)c1Cl C1(C(N(C2CN(C(c3cc(Br)c(C)c(Br)c3)=O)C2)C)=O)CCC2CCC(=O)N2C1 c1(C(=O)NCC2(C)CCC(NC(c3c[nH]c(Br)c3)=O)C2)cc([N+](=O)[O-])n[nH]1 C(C)(CCC(=O)NCC1CCCC(NC(=O)CN(C)C2CC2)C1)SC c1(NC(Cc2cnc(C)o2)=O)cccc(NC(c2cc(C)n(C)c2)=O)c1 c1(NC(N(C(CC)CO)CC)=O)ncc(C)c([N+](=O)[O-])c1C c1(NC(=O)NC2CC23CCCC3)cccc(C2(F)COC2)c1 N1(CC(=O)NCCCN(C(CNC(C)=O)=O)C(C)C)CCCC1C c1(C(=O)NC2CN(C(c3cc(SC)c(C)o3)=O)CC(O)C2)ccc(C)c(C#N)c1 C1(C)(C(=O)NCCC(C)F)CC(O)CN1C(c1nc(Cl)cs1)=O N1(C(C(c2n(C)cnc2)O)=O)CCCC(Cn2cc(C(O)C3CC3)nn2)C1 CC(C)(CC(=O)N1CC(NC(c2ccc(CC3CC3)cc2)=O)CC(O)C1)C(F)F C1(NC(=O)NCCCCc2nn[nH]n2)CCCCC12CCOCC2 C1(COC)(NC(=O)C(C2CCC2)NC(=O)C(C)N2CCCC2)CCCC1 C(=O)(C(CCF)NC(=O)COCCNC(=O)C(C1CC1)SC)OC Nc1cnc(C(=O)Nc2ccc(-c3ccccc3)nc2)cn1 C(=O)(C1=CCC(C)CC1)NCCC(C)NC(c1cc(C(F)(F)F)cc(C)n1)=O c1(C(N(CCCNC(c2c(CC)nn[nH]2)=O)C)=O)cc2ccc(F)cc2nc1C C(=O)(C(O)CC(C)(C)C)NC1(CO)CN(C(CC(C(C)C)OCC)=O)C1 C(=O)(CCC1CCc2ccccc21)NCC(C)N(C(c1c(CC)non1)=O)C C1(CNC(Cn2c(C)nnn2)=O)CN(C(=O)CCCOC(=O)C(C)C)CCC1C CCCCCCCCc1cn(CCOCCNC(=O)C(C)C2CCCO2)nn1 C(C1CCCCCC1)=CC(=O)NC1(C)CN(C(C(c2n(C)ccc2)=O)=O)C1 N1(C(C2CCCC(CC)C2)C(=O)NC(C)C)CCC(OC)C(C)(C)C1 C(=O)(CCCCC#N)N(C(C)CNC(C1CN(C(C)C)C1)=O)CC CCCC(CC)CC(=O)N1C(CNC(C2CCC(C)C2)=O)CC2COCC12 Cc1cc(Br)ccc1C(C)(C)C(=O)N1CC(C)(NC(=O)C(C)CF)C1 c1(CC(N2C(C)CC(NC(c3cn(C)cn3)=O)C2)=O)cc2cc(Cl)ccc2[nH]1 CC1CC(NC(=O)CCCC(=O)C2CC2)CCN1C(=O)C(C1CCOCC1)F Cc1cc(=NC(=O)c2n[nH]cc2NCc2ccc(F)c(F)c2Br)[nH]c(Cl)n1 C12(CC(=O)NCCN(C)CC)CCC1CN(C(c1coc(C)c1)=O)C2 N1(C(CNC(CNC(C(CC)C)=O)=O)=O)CC(C)OC2(CCC2)C1.CC(=O)NO c1(NC(C(C)NC(CC)COC)=O)ccccc1C#Cc1ccccc1 N1(C(CCC(C)SC)=O)CC2CCC1C1CN(C(c3cc(O)cc(=O)o3)=O)CC21 CC1(CNC(=O)CN(C(=O)CC2CCOCC2)C2CCC2)CCC(=O)N1 C(C(C)(C)C#CC(=O)N)NC(c1c(C)oc(C#N)c1)=O.C12CCC(O)(CC1)CC2 c1(C=O)coc2c1CS(=O)(=O)C2.C1(NC(CSCC)=O)CC(C)C1(C)C c1(C(=O)NC2CCN(C(c3n[nH]c(CC)c3Br)=O)C2)cc(N)cnc1Cl c1(C(C(=O)N(CCCCNC(c2cc(C)[nH]n2)=O)C)=O)c[nH]c2cc(F)ccc12 CC1OC(C)C(C(N2CCCCC2C2CCN(CCn3cncn3)C2)=O)C1C N1(C(c2cnc(CC)s2)=O)CC2=C(C1)CN(C(=O)CC(O)C1CCCC1)C2 S(=O)(=O)(c1ccc(Cl)cc1)NCC(=O)NC(COCC=C)C(=O)OC n1(CCCC)nnnc1C(CCC1CCCCC1)NCC(C)OC N1(C(=O)CCc2ccsc2)CC2CC2(C(=O)NCCC2CCCC2)C1 c1ccc(F)cc1.c1(OC)ccc(C(=O)NC(C)C)o1.c1(C(=O)N)cscn1 S(=O)(=O)(c1ccc(=NCCOc2ccccc2Br)[nH]c1)N1C(CCCC)CCC1 CN(CC(C)(O)C1CCCCC1)N1CCC(O)(c2cccc(F)c2)C1 CON1CC(C(N2CCC(C(C)NC(C3CC(C)(C)CO3)=O)CC2)=O)CC1=O C1(C)(CCNC(CSC)=O)CN(C(C2CCCN2C(=O)C(C)C)=O)C1 c1(CNC(N2CCN(Cc3cnc[nH]3)CC2)=O)nc2ccccn2n1 c1(C(=O)NC(C)CCN(C(=O)COC2CCN(C)CC2)C)cc2cccnn2n1 C(CCCCC(=O)NC(C1(O)CCN(C(=O)C=C2CCN(C)C2)C1)C)OCC C(=O)(C(C)(CC)CCCCC)N1CCC(N(C(=O)C=C(C)C(F)F)CC#C)CC1 N1(C(C2(CC)CC2(F)F)=O)CCOC(CN(C(=O)C(c2ccncc2)C)C)C1 CC1(CCc2ncc[nH]2)CCN(CC(=O)N(C)C)C1 N1(C(Cn2c(C)ccn2)=O)CCCC(CNC(=O)CCC2(C#N)CCC2)C1 c1(C(=O)NC2CN(C(CC(CCC)CC)=O)CC2C)cccc2c(C)[nH]nc12 C1(CN)(NC(c2c(F)cc(F)c(F)c2F)=O)C2CC3CC(C2)CC1C3 O=C1CCC(C(=O)N2CCCCC2CCNC(c2ccc3snnc3c2)=O)=NN1 C1(c2n(CCCSC)nnn2)(Nc2cccc(Br)c2)CCC(C)CC1.C1C(C)N1 C1(CNC(C(CC)=CC)=O)CN(C(=O)CS(=O)(=O)NC)CCC12CCOC2 c1(OC)ncccc1NC(=O)CCc1cccnc1.C1(NC(=O)C)(C)CC1 CC(CC(F)(F)F)C(=O)NC1(C)CC(C(=O)NCC2CC3OC2C2CC32)C1 C1(C(N2CCC(c3cccc(C)c3)C2)=O)CCc2ncnc(C)c2C1 CCC(C)C(C(=O)NC1(C)CCC(C)(C)C1)N(C(=O)C#CC(C)(C)C)C N1(C(c2cn(CCCC)nn2)=O)CCC(N(C)C(c2nnccc2C)=O)C(C)C1 CC(C)CC(C(=O)N1CCCCCC1)NC(C1CC(F)C(=O)N1)=O c1(C(=O)NC(CCCNC(CCCCC#C)=O)C)cnc2c(cnn2C)c1 n1(CCC(=O)NCC2C(NC(C(C(C)C)(C)O)=O)C2)cnc2sccc2c1=O c1(-c2onc(-c3c(Br)ccc(C)c3)n2)ccc(S(=N)(=O)N(C)C)cc1 N1(C(CCC2CCN(C(c3nn(C)c(=O)cc3)=O)C2)=O)CC2CCC(C1)C2O Cc1ccc(C#N)cc1C(N1CC(C)C(C)(C(=O)NCC(F)CO)C1)=O C1N2N=C(C(C)C)C=C1NC(=O)C1CC(=O)CN1C2=O.C(C)(C)(C)OC CC1CN(C(C2CC3CCC(C2)O3)=O)C(C)CN1C(=O)CC1CC(F)(F)C1 CCC(CC#N)N=c1[nH]c(=NC(C)c2cnn(CC)c2)[nH]c2cc[nH]c12 C1(C(=O)NCC(C)NC(=O)CCSc2cccc(Cl)c2)CCCCC12CC2 c1(CN(C)C)cc2sccc2[nH]1.c1(C(N2CCCC2)=O)cc(-c2cn(C)nn2)on1 C1(CC=O)CC2(CC2)CN1C(=O)CCn1cncn1.CC1(C)CC(C(O)C)C1 C(CC(C)C(=O)N1CC(CC)(NC(=O)CC2CCCCC2C)C1)=CC C1(C(N(CC=C)CC=C)=O)CC2C=CC1N(C(c1nccnc1OC)=O)C2 CCCC(CC)CCC(=O)NCC(=O)NCC(N1CCN(C)C(=O)C1C)=O c1(OC)ccc(C(=O)O)cc1CN1CCCN(c2ncc(F)cn2)CC1 C1(NC(c2ccc(OC)s2)=O)CC(NC(=O)CC2OCCO2)C12CCC2 c1(C(N2CCC(NC(C)=O)C(c3ccccc3)C2)=O)cnn(C)c1S(N)(=O)=O Cc1cc(CC(N2CCN(C(=O)CN(C)C(C)C)C(C(C)C)C2)=O)ccc1Cl Cc1cnc(F)c(C(=O)NCC2(C)CCCN2C(c2ccc([N+](=O)[O-])[nH]2)=O)c1 C(CC(=O)N(C)CC1(O)CCOC1)(C(F)(F)F)NC(c1n(OC)cnc1C)=O c1(N2C(CNC(C3C(C)CC(C)O3)=O)C(C)CC2)ncc2c(n1)CCOC2 C1(CNC(c2ncc(C3CC3)o2)=O)CCN(CCO)CC1O.c1cccnc1.C CCCCC(CNC(C1CCOC1)=O)NC(c1cc(C)nn1C1CCC1)=O CCC(C)C(C(=O)NC)N(C)C(C1CC(=O)OC1(C)C)=O.C1(O)CCN(C)CC1 C#CCC(C(N)=O)NC(=O)CCOC1CN(C(C2CCN2C)=O)C1 c1(C(C)=O)ccccc1C.N1(C(C(=O)NCCCCCO)C2CC2)CCC(CC)(CO)C1 N1(C(CCOC)=O)CCCC2(CNC(C3(C)CCCS3)=O)CCCCC12 N1(C(C(C)SCC)=O)CCC(CC(=O)NCc2noc(C)n2)C1(C)C N1(C(c2c(-n3ccc(C)n3)cccc2)=O)CC2CCN(C(c3nncs3)=O)C2C1 n1(C(CC)C)ccc(=NC(=O)CC2CN(C(=O)C(C3CCCCC3)F)CCO2)[nH]1 c1(C(N(CCn2cc(CC3CC3)nn2)C2CC2)=O)ccc(C)c(Cl)c1F.C C1(NC(c2cnc(CCC)s2)=O)COC2(CCN(C(c3cc(Cl)ns3)=O)C2)C1 CC1CC(CC(=O)N(CCCCN(C)C(c2cccc(Cl)c2)=O)C)C(C)O1 c1(CCC)nc(C(=O)N(CCCNC(=O)CC2C=CCCC2)C(C)C)cs1 c1(CC)nnc(CN(C(=O)CCN(C)C(c2scnc2Cl)=O)C)o1 C(=O)(CC(CC#N)c1ccccc1)NCCCCN(CCCCOC)C c1(NC(C)C)ncccc1C=O.C1(CC)CSCCN1C(C12CC(C)C1C2)=O.N c1(C(N2CCN(Cc3cscn3)CC2)C(=O)NCCC)cc(OC)c(F)cc1F N1(C(c2cc(C=O)sn2)=O)CCN(C(C2CC2)=O)CC1CS(C)(=O)=O.CO C1(C(=O)NCC(c2ccccc2)NC(c2cn(CC)nn2)=O)COCCOC1 c1(OC)ccc2oc(C(=O)NC3COCCN(c4ncc(F)cn4)C3)cc2c1 C1(C(=O)NCC(C)(C2CC2)NC(C=CSC)=O)CCN(CP(C)(C)=O)CC1 N1(C(Cc2nnc(C)o2)=O)CC(CO)C2(C1)CN(C(C1(C)CCCCCC1)=O)C2 C1(C(N(CCN=[N+]=[N-])CC)=O)CCN(C(=O)C(C)(C)C(C)O)C(C)(C)C1 C1(O)(CC(N2CCCC(NC(=O)CC3CCCC3)C2)=O)CCCCCC1 c1(C(N2CCC(NC(c3ccnc(C(C)C)n3)=O)C2)=O)c(O)nnc2c1CCC2 Cc1ccncc1C=CC(=O)NCC(C)(CO)NC(C1CC12CCOCC2)=O C1(C(C)(C)C)(C=O)CCNC1.C(C(=O)N)N(C)CC.C1CC1.C(C)(C)C Cc1nc(C2CCC2)sc1CC(=O)NCCCCNC(c1nc(Cl)cs1)=O C1CCCN(C=O)C1.C1(N(C(=O)OC(C)(C)C)CC)CCN(CC(C)C)C1 C1(C(=O)OCC)(C(=O)NCCOCCN(C)C)CC1C N1(C(c2c(C)nn[nH]2)=O)CC2CCC1C1CN(C(C3CCC(=O)NC3)=O)CC21 C1(CC(N2CCC(N(C(=O)CCC(N)=O)CCC)C2)=O)CCC2(CCC2)O1 C1(C(=O)NC(c2cc(Cl)cc(Cl)c2)CO)COCCN(C(C2CC2(F)F)=O)C1 n1(C(CCC)C(=O)OC(C)(C)C)ccc(=NC(=O)NCCC2(OC)CC2)[nH]1 C1(CNC(CC2CC(=O)C2)=O)CC2CCCC2N1C(c1cc(C2CC2)on1)=O c1(OC)cc(C)c(C(N2CCC(=CC)CC2)=O)cn1.C1(C=O)(C=O)CC1.N CCCCCCC(CC)C(=O)NCC(C)CN(C(=O)CCCCSC)C c1(OC)cncc(CCC(N2CC(NC(=O)Cc3ccc(Cl)nc3)CC2C)=O)c1 N1(C(CCC=CC(C)C)=O)CC2CCN(C(=O)CC3CCSCC3)C2C1 C1(NC(C(C)OCCOC)=O)CCCC12CN(C(c1ccc3occc3n1)=O)C2 c1(NC2C(SC)COC2)nc(N2CCC(C3(C)CC3)C2)c2c(n1)CCS2 C=C(C)CC(C(=O)NCc1cc(C2CC2)[nH]n1)NC(=O)C(C1CCOCC1)F C(=O)(C1=CCC(F)(F)CC1)N(C1CCCN(C(=O)Cc2cnc[nH]2)CC1)C N1(C(c2c(C)c[nH]n2)=O)CCC(C2CCN(C(=O)Cn3ncn(C)c3=O)C2)C1 O=C(CS(=O)(=O)NC1CC1)Nc1ccc(C2CCC2)cc1 C1(C(N(C2CCCN(C(C3CC(F)(F)C3)=O)C2)CC)=O)COc2ccccc2C1 c1(C(=O)NCC(CCC)NC(=O)CC2CCC(C)CC2)cc(C)nc(O)n1 C1(NC(C2(C(N(C)C)=O)CC2)=O)CCC(C)C1.c1(C=O)cc(Cl)nn1C.C C1(C(=O)NCC2(NC(C(C3CCCCC3)N(C)C)=O)CCCC2)CCC(O)CC1 C1(NC(C(C=C)(C)CCOC)=O)CC2CCC(C1C)N2C(=O)C(C)O.C1CC1 N1(C(C=CCC)=O)CCCC(C)C1CNC(c1cc(OC)no1)=O C12(CNC(CCN(C(=O)Cn3nccn3)CC#C)=O)CCCC1C2 C1(CNC(c2nncs2)=O)CCC2CN(C(c3cnc(F)c(F)c3)=O)CCC2C1 CCC(CN(C)C)CC(=O)NC1CCCN(C(C2CC2(F)F)=O)C1C CC1CCC(C)(C)CC1(c1nnnn1CCOC)NC1CC1 c1(CC(=O)NCC(CO)NC(C(C)NC(N)=O)=O)ccc2c(c1)ncn2C N1(C(C=CC(=O)OC(C)(C)C)=O)CC2OCC(NC(c3cnc[nH]3)=O)C2C1 N1(C2CCN(C(C(C)=C(CC)C)=O)C2)CCC(NC(C2CCCN2C)=O)CC1 C1(NC(CCn2ccc(C)n2)=O)CCCCC1CNC(=O)C(C)(C)C1CCCO1 C1(NC(c2cn(CCCC)nn2)=O)CCC(CC(=O)NC2CCN(CC)C2)CC1 Cc1cc(C)n(C(C)C(=O)NCC23CC2CN(C(c2cc(Cl)ns2)=O)C3)n1 N1(C(CSC)=O)CC(CNC(=O)C(C)Oc2ccc(Cl)cc2Cl)OC(C)(C)C1 N1(C(=O)NCc2ccnc(Br)c2)CCCC2(COC2)C1 CON(CCC(=O)NCC1CCCC1N(C)C)C(=O)CCCCCC(C)C C1(NC(C)CCc2ccccc2F)CC2(C1)CC(C)(C(=O)O)C2 C(=O)(C(O)C1=CCCCC1)N1CCC(C(N2CCC(C)(N(C)CC)C2)=O)C1CC N1(C(CC(=O)OCC)=O)CCCC2CN(C(c3cccc4c3OCC4C)=O)CC12 C1(C)(CC)C=C(C(=O)N(CCCNC(=O)Cc2nnc(C)o2)CCO)C1 c1(OC)ccc(C(=O)NCCN(C(c2cnc(Cl)s2)=O)C2CC2)cn1 c1(COC(C)C)nnc(-c2ccn(-c3ccccc3F)n2)n1C C1(NC(=O)NC23COC(CNC2=O)C3)CCCC1C1CCCC1 c1(CC(=O)NCC(CC)(C)NC(=O)C(C)=CC(C)(C)C)cc(C)ccc1Br O=C(O)CCCNC(=O)CC1CC12CC2.C(=O)C1=CCC1.C=O.C=O.N c1(C(=O)N)ccc(N)c(N)n1.C1(C(C)C)OCCC1C(=O)NCCC1CCC1 C(=O)(CCC(=O)N1CCCC(CNC23CC2CN(Cc2ccccc2)C3)C1)NC N1(C(CC2(C)CCCO2)=O)CCCN(CCNC(c2cnn3c2OCC3)=O)CC1 C1(CCC=C)(C(N2CCC(OCCF)C2)=O)CN(C(C2CCCC2)=O)C1 C1(CNC(C2CC2c2ccccc2)=O)CCCCC1.C1(C=O)CC(F)(F)C1 N1(C(c2nncc(CCC)c2)=O)CCN(C(C2(C)COC(=O)N2)=O)CC(C)C1 C1(C(C(=O)NCC(C)(C2CC2)NC(=O)CCF)OC)CC(F)(F)C1 c1(NC)cnc(C(N2CCC(C(C)C)C2)=O)cn1.c1(C=O)ocnc1C1CC1.N c1(OC)ccn2ccnc2c1C(=O)NC1CCCN(C(=O)CC2CC23CC3)CC1 c1(C(=O)NCC2(O)CN(C(C3C(C)CCS3)=O)C2)coc2c1COC2 c1(NC(C2(F)CN(C(c3c(C)cc(Cl)nc3)=O)C2)=O)cccn2cncc12 C(c1ccc(F)c2ccccc12)=CC(=O)NC(C(CC)C)C(N)=O C1(NC(COCCOC)C(C)(C)C)CNCCC12CCOCC2 N1(C(=O)COc2ccc(F)cc2F)CCc2cc(Cl)c(F)cc21 C1(NC(CC2CN(C)C2)=O)CC2CC1N(C(c1c[nH]cc1C(C)(C)C)=O)C2 C(CCCN1CCC1)NC(=O)NC1C(CC(C)C)C1 c1(C(c2n(CCOC)nnn2)NC2CCCOC2)cc(Cl)cnc1F C1(C)(CNC(C(C)(C)c2sccc2Cl)=O)CCCN(C(C2(CCF)CC2)=O)C1 C1(C(=O)NCC(C2CCCN2C(=O)C=CC2CCC2)(C)C)CCCC(CF)C1 C1(CCOCC)CC(O)CN1C(=O)C(C)=CCN.C1(=O)NCCN1 c1(CC(=O)NCCCN(C(CC(=C)C)=O)CCO)nnc(S)n1C N1(C(COCC)=O)CC=CC1C(=O)NC1(C(F)(F)F)CC1 c1(C(C)=O)c(CCC(=O)NC23CC(C2)N(C(=O)C(=O)N(C)C)C3)c[nH]c1C C(Cc1cnc[nH]1)(C(=O)NCC(O)CO)NC(=O)CCc1nccs1 c1(OC)ccc2cccnc2c1C(N1CC2C(NC(=O)COC(C)C)C2C1)=O Cc1nc2ccccc2nc1C(N1CCC(O)C1C)=O c1(C=O)ccc(S(N)(=O)=O)o1.C1(S(N)(=O)=O)(C)CCC1.CC(C)(C)CC C1(CNC(C(CO)OC)=O)CN(C(=O)C)CC1(F)F.C1(CC=O)CCCC1 C1(NC(C(C)n2ccnn2)=O)C2CC(NC(c3cnc(Cl)s3)=O)CC12 CC(CC(C)NC(C1CC1(C)Br)=O)NC(C1CC1(F)F)=O c1(OC)ncc(NC(C2C=CC(NCc3snnc3C)C2)=O)cc1Cl Cc1c(C(N2CCC(CF)(NC(c3ccc(Br)o3)=O)C2)=O)cccc1N c1(CC)ccc(NC(=O)C(C2CC2)NC(C23CSCC2C3)=O)cc1 C1(N(C(C2CCCC2CF)=O)CC)CCCN(C(=O)CC(C)C)CC1 C(=O)(CCn1cccn1)NC(C(=O)OCC)C.c1(CCC=O)cc(C)on1 C1(F)(C=O)CCCN(C(=O)CN2C(=O)CNC2=O)C1.C12(CC)CCC(CO1)C2 N1(C(C(C)O)=O)CC2CCCN(C(C3CCC(C)N3C(=O)O)=O)C2C1.C(C)(C)C C1(C(=O)N)CCC12CCCO2.c1(C(C)C)n[nH]cc1C(=O)NC1CC(F)(C)C1 C1(C)(CNC(c2n(CC)c(O)nc2)=O)COCCN(C(c2cccc(C)n2)=O)C1 c1(C(N2CCC(c3cn(CCC=C)nn3)CC2)=O)ccc(OC)cc1Cl Cc1cc(NC(=O)C(CC2CCC2)NC(c2cnc[nH]c2=N)=O)c(C)c(C)c1 CCC(CC(=O)NC1CC(C(F)(F)F)C1)N(C(=O)Cn1cnc(C#N)n1)C CCC(CC)C(C(=O)NC1CC(=O)N(C2CN(CCCOC)C2)C1)OC c1(OCC)nc(N2CCN(C(c3cnc(Cl)cc3I)=O)CC2CC)ncc1C CC1CN(CC23CCC(CC2)O3)CC(C)N(C(=O)OC(C)(C)C)C1 Cc1cc(N2CCC(C)C2CNC(=O)C(O)C2CCCC2)n2nc(C)cc2n1 CC1CN(C(=O)CCc2ccccn2)CCCN1C(C1CCNC(=O)C1)=O N1(C(C2C(Cl)(C(=O)OC)C2)=O)CCc2ccc(C(C)=O)cc2CC1 C1(CCC=C)CCCN(C(=O)CC2C3CN(C(=O)CCn4ccnc4)CC23)C1 N1(C(c2c(CC)noc2)=O)CC(NC(=O)CO)CC12CCC2.c1ccc(O)cc1 c1(C(=O)NC(Cc2cn(CCOC)nn2)C(=O)OC)cnccc1Br N1(C(C(C2(C)CC2)NC(c2c(C#C)c[nH]n2)=O)=O)CCN(C2CC2)C(C)C1 c1(COC)nc(=N)[nH]cc1C=O.c1(C(N2CC3C(C3)C2)=O)cc2cscc2s1.N C(=O)(C#CC1CCCOC1)NCC1(C)CCCN1C(=O)Cc1csc(S)n1 CC(C)C(O)CC(=O)NC(C)CCCNC(=O)C=CC1CCC1 CC12CC(C(=O)NC3CC34CCN(C(=O)Cn3ccccc3=O)C4)(CCO1)C2 C=C(Cl)CC(C(=O)N(C)CCc1cnn(C)c1)NC(=O)C(C)Cn1cccn1 N#Cc1cn[nH]c1C(=O)NC1CCCN(C(=O)CCCc2cccc(Br)c2)C1 C1(O)(C(=O)NC2CC(NC(C3CCCOCC3)=O)C2)CCOCC1 N1(C(=O)C(O)Cc2ccccc2)CC2(CCOCC2)c2cc(C(F)(F)F)ccc21 CC1=C(C(=O)NCC(CC(C)C)NC(C2CC2(c2ccccc2)C)=O)CCCC1 C1(C(N(CCCC)C)=O)CCCC(NC(C2CC3(CCO2)CC3)=O)CC1 c1(C(N2CCC(C(N3CC(COC)OCC3)=O)C2)=O)cc(C)c(Br)cc1C c1(C(=O)NC(C)CNC(=O)C(C)(C)c2ccns2)ccnc2ccncc12 CCC(C)C(=O)N1CSCC1NC(=O)OC1CCN(C(=O)O)C1.C(C)(C)C c1(CN(C)C(=O)NC2CCCC2c2ccccc2)cc(Cl)no1 c1(CCCNC(=NCC=C)NCCc2cnc(C)cn2)ccc2c(c1)OCCO2 c1(N(C)CCO)ncc(C(N2CCCC2CC(C)(C)C)C(=O)NCCC#N)cn1 c1(N(CCOCCN(C)C)C)ccc(S(=O)(=O)N2CCOC3(CC3)C2)cc1C#N CCS(=O)CC(=O)NCCNC(C1CC(F)C(=O)N1)=O.c1ccc(Cl)nc1.C CC1CNc2ccc(C(N3CC(NC(=O)OC(C)(C)C)C(C4CC4)C3)=O)cc2O1 Cc1cc(C(=O)NC2CC2)nc(N2CCCCC2)n1.c1(CC(=O)N)nc(C)no1 CC1CCC(F)(F)CN1C(=O)C(c1cccnc1)NC(=O)CC#N N1(C(C(C2CCCOC2)OC)=O)C2CCC1CN(C(=O)CS(=O)(=O)N(C)C)C2 CCCCCCCCC(CO)NC(c1cccc(Br)c1SC)=O c1cc(F)ccc1Cl.c1(NC(N2CC3C(C3)C2)=O)cccc(Cl)c1Cl.O=CC1CC1 CC1(C)COCCN(C(C23CC(F)C2C3)=O)C1.c1(C=O)cnc(C2CC2)nc1O.N Cc1ccc(NC(=O)C(CC2CCCC2)NC(=O)C=CC2(C)COC2)cn1 C1(CC)CN(C(=O)C(Cc2ccccc2)C(F)(F)F)CC2(CCCOC2)O1 N1(C(c2c(C)ccc(F)c2)=O)CC(CNC(=O)CC=O)OC(C)(C)C1.C1CC1 c1(CNC(c2n(CC)nnn2)c2ccnn2C)nc2c(s1)CC(C)CC2 C(CC(C)CC)(C(=O)Nc1cnc(CCC)nc1)NC(CCC#C)=O c1(C(C)(C)C)cc(=NCC2(C(C)(C)C)CCN(C(c3cnns3)=O)C2)[nH]cn1 S(=O)(=O)(c1cccc2nonc12)N1CCC(O)(CC(N2CC(O)C(F)C2)=O)CC1 C1(C)(N(C)C)CC(C(=O)NCC2CC2NC(=O)CCC2CCCOC2)C1 C(CC)(CCCC(=O)N1CC(F)(F)C1C1CC1)NC(C(CCC)=CCC)=O C1(CN(C(C2N=C(C)SC2)=O)C)CCCN(C(=O)C(C)CSc2ccccc2)C1 N1(c2nnc(CCC)s2)CCC2(CCCC2NC(c2ccc(Cl)cc2F)=O)CC1 Cc1cscc1CNC(c1n[nH]cc1C)c1nnnn1C1COC1 n1(CC(N2CCC(O)C2)=O)cnc([N+](=O)[O-])c1.c1(COC)cc(CC=O)no1.N N1(C(Cc2cc(C)n(C)n2)=O)CCOCC(C(=O)NC2CC3CCCC3C2)C1 CC12CC(C(N3CC4C(NC(c5csc(Br)c5)=O)C4C3)=O)(CCO1)C2 CCCCC(C)C(=O)NC1C2CC1N(C(=O)CCCOc1cccc(C)c1)C2C C1(C(=O)NCC(CN(C)C)O)COCCN(C(=O)CNC(N)=O)C1 N1(CC)CCN(C(C2CCCN2C(=O)C(n2ccc(C)n2)C)=O)C(C)C1 CC1(C)CN(c2nnc(C(F)F)o2)C1C1CCN(C(C2(F)CC2)=O)CC1 c1(C(N(C(CCNC(C2N(C(C)=O)CC(O)C2)=O)C)C)=O)ccc2nncn2c1 C1(O)(CC#C)CC(C(=O)NCC2CN(C(N)=O)C2)C1.CC(C)=CC=O C1(C(CC)CC)CCN(C(=NCCCN2CCOCC2)NC2CC2(F)F)C1 N1(C(c2c(C(C)C)noc2)=O)CC(NC(=O)Cn2cc(C3CC3)cn2)C(O)C1 C1(SCC)CCCC(N=c2[nH]c(=N)[nH]c(=NCCC3SCCS3)[nH]2)C1 C1(C2CC2)(NC(Cc2ccc(C)cc2)=O)CCN(C(=O)CO)C1 O=C1CC(C(=O)NC23CC(NC(=O)C(O)CC4CCOCC4)(C2)C3)=NN1 c1(OC)ccc(C)c(NC(C2CC(c3cn(C4CCOC4)nn3)C2)=O)c1 c1(OC)cc(C(=O)CCC(=O)N(C2CCN(C(C3CCCO3)=O)C2)CC)ccn1 C1(N(C(C(=O)NC2CCCC2)c2ccon2)C)CCC2(CCCCC2)CC1 C=CCC(F)(F)C(=O)NCC1(F)CN(C(C2CC2c2ccoc2C)=O)C1 N(C(=NCCSC)N1Cc2cccc(F)c2C(C)(C)C1)CC1C(C)C1 C1(OC)CC2CC1CN(C(C1CCC(C(C)C)N1C(=O)CCCC1CC1C)=O)C2 c1(-c2cn(CCCCOC)nn2)cc(NC(=O)C(CCSC)NC=O)ccc1F N1(C(c2ccc(CC)[nH]2)=O)CCC=C(C(=O)N2CC(CC(F)(F)F)C2)C1 CC#CCCCC(=O)N(C)Cc1ccccc1CNC(=O)C(CC)OCC C1(C(=O)NCC(CNC(c2ccc(Br)cn2)=O)O)C2CNC(=O)C12 C=CC(O)C(=O)N(CC(=O)NC(C)(COC)CC)CC1CC1 C(=O)(C1CCCc2c[nH]nc21)NC(C)CN1CCN(C(=O)CN=S(C)(C)=O)CC1 Cc1ccc(CNC(C2CCCN2C(=O)C(F)(F)F)=O)cc1.C(C=O)C(C)C N1(C(c2ccc(C)[nH]2)=O)CCC(C2CC(NC(C3CC3(Cl)Cl)=O)CCO2)CC1 N1(C(C=CC=CCC)=O)CC2CCC1C1CN(C(=O)CC3COCC3O)CC21 Cc1cccc(C(=O)NNC(=O)NCCCOc2ccc(C(=O)O)cc2)c1 C1(C(=O)NC(CN(C(CCCCCCCC)=O)C)C)CC2(CCCCC2)S1(=O)=O CCCCCCNC(=O)C(CN(C)C)N(C)C.c1(C=O)ccc(C(=O)CC)cc1 CC1CN(C(c2ccc(OCC(F)(F)F)cc2)=O)CCCN1C(c1cnns1)=O N1(C(C(C)SC)=O)CCC(CO)C(NC(c2cn(C)c(=O)cn2)=O)C1 C12CCC(CC1)N2C(=O)CN(CC(C)(C)C)C.CC(CC(=O)NC)N(C)C N1(C(COCCCOC)=O)CCN(C(=O)CC(C)(O)C2CC2)CC1C N#Cc1ccc(N(CC=O)C(=O)CCF)cc1.C1(CC=O)CC=CCC1.C1CCC1 C1(C(=O)NC(c2cc[nH]n2)C)CCN(C(c2ncccc2Cl)=O)CC1 c1(N2CCCC(CC)C2)ccncc1S(=O)(=O)N1CCCOC1.C=O CN1Cc2cc(C(c3nnnn3C3COC3)NCCOC(=N)O)ccc2C1=O c1(C(=O)NC2C(CNC(C(C=C)(C)CC)=O)COC2)ccc2oc(O)nc2c1 N1(C(=O)CCOCC2CCCO2)CCC2C(C1)C2(F)F C1(NS(C)(=O)=O)CCC(CNC(=O)CSCCc2ccccc2)CC1 n1(CC(=O)NC2CC(NC(C3(C)CC(C)OCC3)=O)C2)cnc2ccccc12 c1(C(c2nnnn2C2CCCC2)NCCOCCC=C)ccncc1CC C1(C(C(=O)NC(C2CCCN2C(c2ccc(O)cc2)=O)C)(C)C)CCCN(C)C1 Cc1cc(C#N)ccc1C(N1CCC(C)(NC(C2CCCS2(=O)=O)=O)CC1)=O C1(c2n(C)ncn2)COCCN1C(=O)NCCCc1ccnn1C c1(C(N2CC(COC)N(C(=O)C(O)CC3CC3)CC2)=O)ccc2c(c1)OCO2 N1(C(CCNC(C)=O)=O)CCC(N(C)C(c2ccc(C)c(C)c2)=O)C(C)C1 C1(C(=O)N)SC2C=CC1CC2.C(C)(CCC(=O)NCC1(O)CC(C)C1)OC C1(CC=C)(NC(=O)C(C)C(C)O)CCCN(C(c2nc(C)nn2C)=O)C1 c1(CCC(N2C(C3CCN(C(C(CC)C)=O)C3)CCC2)=O)ccccc1C(N)=O CCS(=O)(=O)c1ccc(CNC(=O)NCC2(C#N)CCCCC2)cc1 C(=O)(C1=C(Cl)CCCC1)NC1(CO)CCN(C(c2cn(CCOC)nc2)=O)C1 CCCCC(F)C(=O)NCc1ccc(C(N2CC(C)C(F)C2)=O)o1 C1(C2CC2)(CNC(=O)CCC(F)F)CCN(C(C2(O)CC3CCC2C3)=O)C1 Cc1nc2c(cnn2C(C)C)cc1C(=O)OCC(=O)C(C)C C(=O)(C(C)(C)C(=O)N1CC2(CCN2C(=O)CNc2nccs2)C1)N(C)C C1(C)(OC)CC(NC(=O)CC2CCCCN(C(C3CCC3C)=O)C2)C1(C)C N1(C(c2ccc(C)cc2O)=O)CC2CCN(C(c3n[nH]cc3[N+](=O)[O-])=O)CC2C1 c1(CC(N2CC(C)C(NC(=O)Cc3cccn3C)C2)=O)ccn2cncc2c1 c1(C(=O)NC(CN(C(=O)CC(F)(F)Cl)CC)C)cnc2c[nH]nc2c1 C1(C(=O)NCCc2ncc(C)nc2)CCN(C(=O)CCCn2cncn2)CCO1 N1(C(C(C)N(CCC)C(C2CC(C#N)C2)=O)=O)CCCC(O)(CO)C1 c1(C(=O)NC(C(C(C)C)NC(c2nc(C)sc2C)=O)C)cccc2nc(Cl)cn12 Cc1oc(C2CC2)nc1C(=O)N(CC(C)NC(c1c[nH]nc1C1CCOC1)=O)C c1(OC)cncnc1C(=O)NC(C1CC=CCC1)C(N1CCC(OCCF)C1)=O C1(CC)C(NC(c2cc(O)nc(OC)n2)=O)CCCN1C(=O)Cn1ccnn1 n1(C(CC)C)ncc(C(=O)NC(C)(C)CCCNC(C2CCC(=O)N2C)=O)c1C C1(O)(C(C(=O)N(CC(C)(C)NC(C2CC2(F)F)=O)C)F)CCCC1 c1(NC(COCCC=C)=O)ccccc1.c1(C=O)cc(C)nn1C(C)(C)C.N c1(C(=O)NC(C=C)C)ccc2nc(-c3ccc(OCC)c(C)c3)cn2c1 CCC(C)(C(=O)N1CC(C)(NC(C2CCC(=O)O2)=O)C1)C(F)F c1(OC)ccnc(C(N2C3CCC2(CNC(c2ncn(C)n2)=O)CC3)=O)c1.O C1(C(C)NC(c2ccc(Br)s2)=O)CCN(C(=O)CCCn2cccn2)CC1 c1(C(N2CCC2)=O)cc(Cl)n(C)n1.c1(CC=O)ccccc1.CC(=O)NCC c1(CNC(c2cc(C)ccn2)CCC)ccc(C)nn1 Cc1nnc2n1CCC2(C)C(=O)NC(CNC(c1coc(CO)c1)=O)C1CC1 Cc1cc(C(=O)N(C)CC2CCCN(C(=O)C(C)(C)C3CCCO3)C2)sc1C CCCCCC(F)C(=O)N1CCC2(CC(NC(c3cnco3)=O)C2)C1 N1(C(C(C)OCC)=O)CC(CNC(=O)C=O)OC2(CCC2)C1.c1ncc[nH]1 C(=O)(C(C)S(=O)Cc1noc(C2CCC2)n1)N(c1c(C)cccc1)C1CCC1 C(CCCCC(=O)N1CCN(C(=O)Cc2cccc(C)c2)C(CO)C1)OC c1(OC)cnc[nH]c1=NCC(c1ccccc1F)NC(=O)C(C1CCOCC1)O c1(C(=O)NCc2cn(C3CN(C(C4C(C)C4)=O)C3)nn2)cc(Cl)c(Cl)[nH]1 C#Cc1ccc(C(=O)N(CC(CC)NC(=O)CC2CC3CC3C2)C)cc1F N1(C(COCCC=C)=O)CCN(C(=O)C(F)=C2CCCC2)C(CS(C)(=O)=O)C1 c1(OC)cnnc(-c2nc(CC(C)OC)nn2C2(C)CCCCC2)c1 N1(C(c2c(CCC)occ2)=O)CC(NC(=O)CCF)CC(F)C1 c1(C(=O)OC)cn(C)nc1C(=O)NC.c1ccccc1F.C1CC1.C(=O)C C1(C(N(C(C)C2CC2)C)=O)CCN(C(=O)C(O)CC2CCCC2)CCO1 c1(N2CCCC(CSC)C2)nc(NC2CC3CCC2O3)c2ncn(C)c2n1 N1(C(c2scc(C(=O)Nc3c(C)cc(I)c(F)c3)n2)=O)C2COCC1CC(F)C2 C(=O)(C(C)CCc1cccc(F)c1)NCC1(OC)CN(C(COC)=O)C1 c1(C(N2CCN(C(C3C(C=C)C3)=O)C(CO)C2)=O)c(F)cc(OC)cc1F N1(C(C2CCN(CC)CC2)=O)CCC(NC(=O)CCC(N)=O)CC1C1CC1 C1(C=O)(CNC(C2CC=CC(O)C2)=O)CC12CCC2.C1CCC2(CC2)C1.N C(=O)(C(C)(C)CC(C)C)NCC(CNC(c1cnn(C)c1C)=O)OC c1(C(N2CCC(CN3CCCC3)CC2)C(=O)NCCC)cc(Cl)ccn1 C1(OC)(C)CCN(C(c2cc(C(C)(C)C)on2)=O)CC1.C(=O)CC1CC1.N c1(CN(CC(CN)O)CC(O)CO)cc(Cl)ccc1Oc1cccc(Cl)c1 Cc1cccc(CC(=O)NC2(CC(=O)Nc3nc(C)cs3)CCC2)n1 c1(C(=O)N)cccc(C(F)(F)F)c1.c1(C(=O)NC(C2CCOC2)C)cscn1 c1(C(N2CCN(C)C(C3CC3)C2)C(=O)NC(CC)(C)C)cc2cc(Cl)ccc2o1 c1(C(N2CCC(NC(c3ccc(C)c(CO)c3)=O)C2)=O)ccc2cn(C)nc2c1 C(=O)(C1=NOC2(CCOC2)C1)N.CC1(C)CCCCC1.C12(CC=O)CC(C1)C2 c1cn(C)nc1C(F)(F)F.CCCCCCn1nnnc1C(C1(C)CSC1)NC C12(C(N3CCC(CC(=O)NCc4c(C)nc(C)s4)C3)=O)CC(C)(CCO1)C2 C1(N(C(C2C(C)(CC)C2)=O)C)CCC2CN(C(=O)CCc3cncs3)CC12 c1(CC)ccc(F)cc1C(c1nnnn1C1CCOC1)NCCCOC(C)C c1(NC)cncc(C(=O)NCC=CC)c1.N1(CCC=O)CCCS1(=O)=O.N C1(CCC(=O)OC)CN(C(=O)C(=O)NC2(Br)CCCC2)CCO1 C1(C(N2CCN(C(c3n(CC)ncc3)=O)C(C)C2)=O)CCCN(S(N)(=O)=O)C1 Cc1cc(C(=O)NCC2CCCCN2C(=O)C(O)Cc2cnc[nH]2)nnc1O Cc1nc(C2CCCN2C(=O)C(C)Cc2ccncc2)n[nH]1 C1(NC(C(c2ccc(C)o2)C)=O)CCC(NC(C2CC(CF)C2)=O)CC1 c1(C(=O)NC(Cn2cc(-c3cn(CC)nc3)nn2)C)c(OC(F)F)cccc1F N1(S(c2cccc(CC(=O)OC)c2)(=O)=O)Cc2nccn2CC(CO)C1 N1(CC)CCC(c2ccc(F)cc2)(C(=O)O)CC1.S1(=O)(=O)CCC2CN1C2.C N1(C(c2ccc(F)s2)C(=O)NC2CC(F)(F)C2)CCC2(CCSC2)C1 c1(CC(=O)NCC2(O)CN(C(c3[nH]cc(C)c3)=O)C2)ccc2c(c1)ncn2C CCC(C)(CNC(=O)CCc1cnoc1)NC(=O)CCc1nccn1CC N1(C(C(C(C)C)O)=O)CCC2(CC1)CCN(C(C1CN(C)CCO1)=O)C2 C1(CNC(C2C(C)=C2)=O)CCCC12CCN(C(=O)CCC1CCC(=O)N1)CC2 N1(C(c2sc3c(c2)CC(C)CC3)=O)CCC(N=c2ccnc(C(=O)N(C)C)[nH]2)C1 N1(C(C=CCCC)=O)CC(CNC(c2ccc(F)cn2)=O)C(C)(C)C1 C1(C2CCCCC2)(C(=O)NC2C(F)CCN(C(c3cnc(N)c(Cl)c3)=O)C2)CC1 c1(OC)cncc(C(N2CCC(NC(c3c(C)noc3C)=O)C2)=O)c1C c1(C(c2ccc(CN(CCC(C(C)C)O)C=O)cc2)=O)cc(Cl)ncc1Cl c1(NCCCNC(C2(C)N(C)CC(O)C2)=O)cc(C(N)=O)ccc1[N+](=O)[O-] c1(C(=O)OC)ccc(NC(=O)NCc2cn3c(C)cccc3n2)c2c1CNC2=O N1(C(CCC2(C)CN(C(=O)Cc3cncnc3O)C2)=O)CC2(CCCO2)C1 C1(CCC=C)CCN(S(=O)(=O)Nc2cc(Br)ccc2Br)CC1 C1(CC(=O)NCCCCCNC(C(C)(F)c2ccccc2)=O)CN2CCN1CC2 c1(C(N2C(C(=O)NC(C(=O)OC(C)C)C)CC2)=O)ccc2c(n1)OCCO2 C1(OC)CCC12CC(C(=O)NCCC1CCC1)C2.C(=O)CC(C)c1ccco1.N C1(F)CCN(C(=O)C(C)(C)n2ccc(C)n2)C1.c1(CC)ncc(C(=O)N)[nH]1.C c1(CC(=O)NC(C(C)C)CCN(C)C(C2CC(O)CN2C)=O)ccc(C#N)nc1 N1(C(Cc2cc(C)no2)=O)CC=C(CC(=O)N2CCN(C)C(CO)C2)CC1 c1(C(=O)OC)ccc(Br)cc1NC(=O)C(=O)NC1CCCC1n1cccn1 C(CCO)(C(F)F)N(C(CN(CCC)C(C1OCCC1C(C)C)=O)=O)C C1(C2CC2)(C(N2CC(COC)OCC2)=O)CN(C(=O)CCC2CCCN2C)C1 C1(NC(c2c(-c3ccc(Cl)cc3)n[nH]c2)c2nnnn2CI)CCC2(CCC2)C1 CCCCC(C)C(=O)NC1CCN(CCNC(=O)C(n2cc(Cl)cn2)C)CC1 c1(C(=O)NCCCCC(CO)NC(C2C(=C)CC2)=O)cc2c(cc1Cl)OCCO2 c1(OCC)ncc(NC(=O)C(C(C)C)NC(c2[nH]nnc2CC)=O)cn1 c1(CNC2CCCC(C(N3CCC(C#C)CC3)=O)C2)cc(Br)cc(C)c1O N1(C(C(CN(C)C)(C)C)=O)CCN(C(C2(c3cccc(F)c3)CC2)=O)CC(O)C1 C1(CCC)CCCN(C(C2CCCN(C(=O)CC3CC3(F)F)C2)=O)CC1 c1(C(=O)NC2CCN(C(C(C(C)C)O)=O)C2)ccc([N+](=O)[O-])cc1Cl N1(C(C=C(C)CNC(c2nonc2C)=O)=O)CC2CCOC(=O)C2C1 c1(CC(CC)N(CC)Cc2cnn(CCF)c2)ccccc1 c1(C(=O)NC(C)CNC(C2CC2(C)C(F)F)=O)ccnc2ccnn12 C12(C(N(C(C)CN(C)C(c3cn[nH]c3)=O)C)=O)CC(CO)(C1)OC2C C(=O)(CCN(OC)C(=O)C(C)C1CCOC1)NC1(C#C)CCCCCC1 C1(N(C(N(CCCCC=C)C)=O)C2CC2)CCCN(c2ccccc2)C1=O Cc1nc(C)c(CCC(=O)N(CC(O)CNC(C2(O)CCOC2)=O)C)c(O)n1 Nc1cncnc1C(=O)NC1(C(=O)NCC#CCCO)CCSC1 N1(C(C(=O)NC(C)C)C2=NOC3CC23)C2CNC(=O)CC1COC2 C#Cc1cc(C(N2CCCC(N(C(=O)CN3CC=CC3)C)CC2)=O)cc(N)c1 C1(CC)CCOC1C(=O)N(CCCCN(C(=O)C(C)OC1CCCCC1)C)C CCC(CC)CCC(=O)NC(CNC(c1cnco1)=O)CO Cc1cc(C)c(C(=O)N(CC(C)NC(c2c(C)nc(C)n2O)=O)C)c(O)c1 C1(NC(c2cscc2Cl)=O)CC2(C1)CN(C(=O)C(F)(F)CO)C2 c1(SC)ccccc1C(=O)NCCN(c1ccccc1)C(=O)CC#N c1(C(N2CCCC(NC(CCCOC(C)C)=O)C2)=O)cc(N)cc(O)c1F Cc1[nH]nc(Cl)c1C(=O)NC1CC2(C1)CC2.C1(C=O)CCN(CC(C)C)C1.N CC1CN(C(=O)CC2(O)CCCOC2)CC(C)N(C(c2ccon2)=O)C1.N(C)(C)C c1(OC)ccc(-n2nc(C3CCCCC3)nc2C2(C)CCOC2C)cn1 N1(C(c2[nH]cc(C)c2)=O)CC2CC(C1)C2NC(=O)C(c1ccc(C#N)cc1)C C1(C(N2CCC(F)C2)=O)CCC2(CCC2)CC1.c1(C(N)=O)cc(C(=O)N)c[nH]1.C Cc1nc(NCC2CCCCC2NC(C2(n3cnnn3)CC2)=O)cc2nncn12 C1CCCCCC(=O)N1.c1(SC)nccn1C1CC1.c1cn(C(C)C(=O)NC)nn1 C1(NC(C(F)=CC)=O)CCCC(N(C(=O)CCn2cc(Br)c(C)n2)C)C1 C(=O)(CCCC(F)(F)F)NCC1N(C(CC(CC#N)c2ccccc2)=O)CC1 N1(C(C(COCC)N=[N+]=[N-])=O)CC2(C(=O)NCCCP(C)(C)=O)CCC1CC2 C1(CNC(=O)CCn2cccn2)COCCN(C(c2ccc(O)nc2)=O)C1 C1(CNC(c2c(C)n[nH]c2)=O)Cc2ccccc2CN1C(C1CC12CC2)=O C1(CNC(C2CCCC(NC(C=C(C)C)=O)C2)=O)CN2CCC1CC2 C1(N(C(C(C)n2cccn2)=O)CC2CC2)CCN(C(C2CCSC2)=O)C1 c1(OC)cnccc1C(=O)N(C)CC1(O)CN(C(c2cccc(O)n2)=O)C1 C=CCC(CNC(C1CCC1CF)=O)NC(c1cc(-c2ccncc2)no1)=O c1(C(CNC(CC(=O)NC2CC2)=O)NC(=O)CO)cccc(Cl)c1 Cc1cc(CCC(=O)NCCCCn2cc(CN(C)CCO)nn2)no1 C1(NC(=O)CCCC2CC2)COC2C(NC(c3cnc4c(c3)COC4)=O)COC12 C1(C(=O)N)Cc2cc(F)ccc2O1.c1(C(=O)NCC(C)C)ccc(C#N)c(F)c1 C(CSC)(CN=c1[nH]c(=NCC2CS(=O)(=O)CCO2)[nH]c2cc[nH]c12)OC C1(C(=O)NC(C2CN(C(=O)C=CC(N)=O)CCO2)C)CC2C=CCC(C1)C2 c1(OC(C)C)ncccc1C(=O)NC(C1CCCN(Cc2ccccc2)C1)C C1(C(C(=O)NC(CC(C)NC(CC(=O)NCC)=O)C)O)COC(C)(C)O1 c1(C(=O)NCC(C)(C)NC(C2OCCN(C(C)C)C2)=O)[nH]nc2cnccc12 N1(C(C)C)CCCC1CC(=O)N(C)CC1CCCN1C(C1CC(CF)C1)=O N1(C(C(C)OCCC(C)C)=O)CC(O)(CN(C(=O)C(c2cnccn2)C)C)C1 c1(CC(=O)NC(CNC(c2[nH]cc(CC)n2)=O)C)ccc2c(c1)CCC2 c1(C(N2CC(N(C(=O)Cc3cn(C)nn3)C)C3(C2)CC3)=O)cc2ncccc2o1 N1(C(C23CC(CC(C)C)(C2)C3)=O)CCN(C(c2ncc[nH]c2=O)=O)C2(CCC2)C1 CCC(CCC(=O)N1C2CCC1C(CNC(c1csc(COC)c1)=O)C2)OC c1(CC)onc(C)c1C(=O)NCC12CC1CN(C(c1nccnc1O)=O)C2 c1(C(=O)NC(CC)CNC(C2C=CC=CC=C2)=O)c(F)ccc2[nH]ccc12 N1(C(=O)Nc2c(CC)cccc2)CCC(COC)C(C)C1 CN(C(=NCC1CN(C(N)=O)C1)NC1CC1)CC(c1ccc(Cl)s1)O c1(C(=O)NCC2N(C(c3c(C)ccnn3)=O)CCC2C)c(C)ccc2nonc12 c1(OC)cc(C(c2nnnn2CC(F)F)NCC2CC23CC3)cc(OC)c1C C(C(F)(C(=O)NC(C1CC=CCC1)CO)C(C)C)NC(c1nc(C)oc1)=O N1(C(COC(C)=O)=O)CC2CCCC(CNC(c3sccc3C#N)=O)(C2)C1 Cc1occc1C(=O)NCCCN(C(=O)CC1(c2ccon2)CC1)C1CC1 C(=O)(C(C)(CC#C)NC(=O)C(COC)C)NCCC(=O)NCC#C.O C(=O)(CC1=CCCCC1)NCC(CN(C(C(C(C)(C)C)SC)=O)C)C C1(C(N2CC(C(C)NC(c3cnn(C4CC4)c3)=O)C2)=O)CCC(=O)N(C)C1 CC(C)(C)[Si](C)(C)OC1CCCC1Oc1ccnc(Cl)c1F N#Cc1cccc(C(c2ccccc2)NCC2CCC3CCCC23)c1 C1(C(N(CCCO)CC)=O)CC=CCC1NC(=O)C(c1ccnn1C)C C(C(C(=O)N(CCCn1ccnn1)CC)NC(=O)C(C)C1CCC1)SCC c1(C(C(N2CC=CC(NC(=O)CSC3CCCCO3)C2)=O)=O)cc(Cl)cc(Cl)c1 C1(C)(CC)CC(NC(c2ccncc2Cl)=O)CN1C(=O)C(F)=CC1CC1 C1(O)(CN(C)C(c2csc(CO)n2)=O)CCN(C(c2cnn(C)n2)=O)CC1 C#CC1(OCC(=O)NC(CNC(c2ccoc2C(C)C)=O)CC)COC1 N1(C(CC(C)O)=O)CC2COCC2(C(=O)NCC=Cc2ccccc2)C1 C1CCC2(CN(C(C3CS(=O)(=O)CCO3)=O)C2)O1.C=C1CC(C(=O)NC)C1 c1(C(N2CCC(CNC(COCC)=O)(CO)CC2)=O)ccnc2ccc(F)nc12 c1(OC)ccc(-c2cc(C(=O)N(C3COC3)Cc3ccccc3)no2)c(Cl)c1 N1(C(C2(F)CCN(C(C(CSC)O)=O)CC2)=O)CCc2cccc(F)c21 C(=O)(N=c1ccn(CC(C)C)[nH]1)C1OCCC(NC(c2ccc(COC)o2)=O)C1 C1(C2CC2)(NC(C2(C(N3CCCC(C(C4CC4)=O)C3)=O)CC2)=O)CCCC1 c1(C(=O)NCCCNC(c2cc(CC)sn2)=O)cc(C)nnc1O C(CCC(=O)NC(C)CC(C)O)NC(C(C)=C1CCCC1)=O c1(CNC(CCC(C)(C)[N+](=O)[O-])=O)cccc2c1CCN(C(c1ccoc1)=O)C2 CC1(C)CC(NC(c2nc[nH]c2C(C)(C)C)=O)CN(C(c2cccc(N)c2)=O)C1 Cc1c(CCC(=O)N(C(CNC(=O)C=CCO)C2CC2)C)cnn1C C(=O)(C(C)CCCC(C)C)NC(CC)CCC(N1CC2OCC(CO)C2C1)=O CCCCC(CCCC)C(=O)NCC1CN(C(=O)C2=COCCC2)CC1(C)C CCC(CC(=O)NC1CCCCN(C(=O)CCOC)CC1)C(F)F C1(C=O)CC(O)CN1C(=O)CC1CCN(C)C1=O.C(=O)(COCC)OC c1(C(N(C(CC)C(=O)Nc2cnc(F)nc2)C)=O)cccc(=O)n1C CC1(C(=O)NCCCCNC(c2ccc(F)o2)=O)C=CCC1 N1(C(C(C2CC2)NC(CCN(CC)CC)=O)=O)CC(CO)OC(CO)C1 N1(CC(=O)O)CCN(CC(=O)Nc2cc(NC3CC3)ncn2)CC1=O C1(NC(C2C(=C)C2)=O)COC2(CCN(C(=O)CCCCCNC(C)=O)CC2)C1 N1(C(c2cc(C)oc2C)=O)CC2OCCN(C(=O)Cc3cc(Br)cs3)C2C1 N1(C(c2ccc(OC)o2)=O)CCC2(C=C(C(=O)N3CCCC(C)(CO)C3)C2)C1 C1(NC(=O)CCc2cnccn2)CC2(CCCN(C(C3CC3(Cl)Cl)=O)C2)C1 c1(OC)ccc2c(C(=O)NC3CCN(Cc4nc(C(C)OC)no4)C3)cnn2c1 N1(C(C2N(CC)CC2)=O)CCC(C(C)NC(=O)CC2CC(F)C2)CC1 C1(CC)CCCN(C(c2cc(C)cs2)=O)C1C(N1CCC2(CSC2)C1)=O C1(C(N2CCC2)=O)CC2OC(=O)OC2C1.Cc1c(C(=O)N)cnn1C1CCC1.C Cn1ncc2c(NC3CC3C(=O)Nc3cc(F)cnc3Br)ncnc12 C1(NC(c2nnn(CC)c2C)=O)CC2C1CCN2C(=O)Cc1ccccc1SC C1(C(N(C2CCN(C(=O)CC3CCOC3(C)C)CC2)CC)=O)CN2CCCC1C2 C(CCCCC(=O)NC(C)Cc1cnc[nH]1)NC(C1C(CC(C)C)C1)=O Cc1nnccc1C(N1CCCC1CCCNC(C1(F)CCCOC1)=O)=O CC1CCN(C)c2ccccc2N1C(=O)C(c1nn[nH]n1)C1CC1 C1(C(=O)NCC(C)N(C)C(C2(C=O)CC2)=O)C2C3CC4C1C1C2CC3C41 Cc1ccc(F)c(C(=O)N(C(C)CNC(=O)CN(S(C)(=O)=O)C)C)c1F c1(C(=O)NC2CCCCC2NC(C2CCCCC2)=O)ccc([N+](=O)[O-])nc1 C1(C(=O)NC(C)CC(C)(C)O)(CC)CCCN1C(C1CN(C)C1)=O N1(C(C(C)NC(=O)NC2CCCC2)=O)CC(C)CC(C)(C)C1.c1c(Cl)cnn1C Cc1cc(NC(C2CCCS2)=O)ccc1NC(c1occ2c1CCC2)=O C1CC2(CC2)C(=O)O1.C1(C(=O)N)(NC(C(C)OCC=C)=O)CCCCC1 N1(C(N(C)C)=O)CCCC(C(=O)NCCC2CCN(C(=O)CC)C2)C1.C1CC1 Cc1cc(Cl)c(C(=O)NCC#CCNC(=O)C=Cc2cnc[nH]2)cc1[N+](=O)[O-] CC1(C)CCC(C)(C(=O)NC2CCC2NC(C2CC(n3cccn3)C2)=O)CC1 Cc1cc2c(cc1C)OC(C(=O)N)C2.C12CC(C1)N(C(=O)CCC1CC1(Cl)Cl)C2 N1(C(CC2CC(C=O)C2)=O)CCC2(C1)CN(C(C1CCSC1)=O)C2.CC(C)C.O C1(C)(c2nc(-c3ccc(C)o3)nn2-c2cccc(C#N)c2)CCNC(=O)C1 N1(C(C2(COC)CCCC2)=O)CCCC(NC(c2coc(C)n2)=O)CC1 Cc1c(Br)ccc(C(=O)NCC2CCC2NC(=O)C(C)Cn2ccnc2)c1N C1(N(C(=O)CCC2CC2)C)C2CN(C(=O)CC34CCCC3C4)CC12 c1(C(=O)NC2(C)CCN(C(C(CC(C)C)C)=O)C2)ccn2ncccc12 C(=O)(CCC)N1CCC1.C(=O)(CCO)N(C)CCOCC(F)F.C1CCCO1 C(C)(C)(C(C)NC(c1[nH]nnc1CC)=O)NC(COCCCC#C)=O c1(C(=O)NC(CN(C(C=C(CCC)C)=O)C)C)cccc(Cl)c1C N1(C(CCN(C)C)=O)CCN(C(c2ccc(N3CCCC3)cc2)=O)C2CC12 c1(C(N(CCNC(c2coc(Cl)n2)=O)C2CC2)=O)cc2c(F)cccc2s1 N1(C(C(C)(C)C)=O)CCC2C(CCCN2C(c2ccn3ncccc23)=O)C1 c1(N2C(CNC(=O)CCF)CCC(C)(C)C2)nc(Cl)nc2sccc12 C1CC(F)(F)C1.c1(C(C(=O)N)N(CC=CC(=O)OCC)C)cscc1Br Cc1n[nH]c(C)c1CC(N1CC(CNC(c2cc(Cl)n(C)n2)=O)C(C)C1)=O c1(C(C(=O)NC(C(=O)OC)C)Nc2ccccc2)sccc1Cl.c1cncs1.C c1(C(N2C3C(NC(c4scc(C(N)=O)c4)=O)C(C3)C2)=O)ccnc2ccncc12 c1(C(C)(C)C)ccc(NC(=O)CC2CCN(C(c3cnsn3)=O)C2)c(I)c1 c1(NC(c2c(Oc3c(C)nccc3)cccc2)=O)ccc(C#N)nc1 C1(C(N(C)CC2(N(C)C)CC2)=O)CSCCN1C(=O)C(F)=CC1CC1 C1(C(=O)OC)CC12CC(S(=O)(=O)N(c1cn3ccccc3n1)C)C2 N(C1CCCc2ccoc21)C(CC(C)(C)NC(C1C(C=C)OCC1)=O)=O c1(C(=O)NC2(CNC(c3ccncc3O)=O)CC2)cnc(O)c2cnccc12 C=CCC(C(=O)N1CCC(C)C1CNC(C1CCN1C(C)(C)C)=O)N(C)C CCCCC(C(=O)N1CCC(C(=O)NOCC(F)F)(n2cccn2)CC1)C(C)C O=C(CC1CCCN1C(=O)CO)N=c1ccn(CCC(=O)O)[nH]1.C1CCC1.C c1(NCC)cccnc1.C(CC)C(=O)N1CCCC1.C(=O)C.C(=O)C1CC1.N C1(NC(C2CCN(C(c3c(C)n(C)cc3)=O)CC2)=O)CC(CO)C12CCC2 C1(C(N2C(C(N(CCCC)CC(N)=O)=O)CC(=O)C2)=O)CCCC12CCC2 CN1CCN(C)CC(NC(C2COCCN2C(=O)C(F)n2ccnc2)=O)C1 C(=O)(C1=C(C)N(C)c2ncnn2C1C)NCCN(C(=O)C(=O)N(C)C)CC N1(C(C(C)=CC)=O)CCCCC1C(C)NC(c1cc(CN(C)C)c[nH]1)=O C1(C)(C(=O)NC2CN(CC)C2)C=CCN1C(=O)COCCSC c1(C(N(CCCN(C(c2nccc(OC)c2)=O)C)C)=O)coc2ccc(F)cc12 c1(C(=O)NCCC(=C)CNC(c2cncs2)=O)cccnc1OCC(C)C c1(C(N2CC(CC(=O)OCC3C(OC)CCC3)C2)=O)cc([N+](=O)[O-])n[nH]1 c1(NC(CCC(=C)C)C)cc(N2CCC(OCCF)C2)nc(C(C)C)n1 c1(C(N2CCC(N(C(C=C(C)Cl)=O)C)C2)=O)cc2n(c1)CCCC2 CC1CCN(C(=O)COCCCF)CC1N(C)C(C1C2COCC12)=O c1(NCC(CC)(C)O)ccc(S(=O)(=O)NCC(C)OC(C)(C)C)cc1C#N C(CN=C(NCCF)NC1CCCC(c2cccc(Cl)c2)C1)c1c(C)nn(C)c1 c1(C(N2CCC(NC(c3c(CC)cccc3)=O)C(O)C2)=O)ccc(S(C)=O)cc1 C1CC2(C1)CN(C(c1n[nH]c3c1COC3)=O)C2.C1(C(=O)N)(CSC)CC1.C C(C(C)CC(=O)NCC1(COC)CCN(C(C2CCSC2)=O)C1)OC N1(C(c2n(C)cc(C)n2)C(=O)NCc2ccco2)CCCCC(C)C1 C(CN=c1[nH]nco1)(N(C(c1c(OC)cc(O)nc1)=O)C)C1CC1 CN1CCOC(C(N2CCC(F)(CNC(c3cnns3)=O)C2)=O)C1=O c1(C(=O)NCCC(C(C)C)NC(C2CCCOC2)=O)cccc(C(F)(F)F)c1F N1(c2c(C)c(F)c(Br)cc2)NC(=O)C2CCCC2S1(=O)=O C#Cc1ccc(C(N2CCCC(N(CCF)C(C3CC(N(C)C)C3)=O)C2)=O)cc1 Cn1cc2c(n1)CCC(C(=O)NCC1(F)CC(NC(c3ncccn3)=O)C1)C2 c1(CC(=O)NC2(C3CCN(C(c4cc(O)no4)=O)C3)CC2)ccc2n[nH]cc2c1 c1(C(=O)NC(CC)(CNC(=O)C2=C(C)OCC2)CC)cnc([N+](=O)[O-])n1C N1(C(C(CCC)=CCC)=O)CC(C(=O)NC(c2nc[nH]n2)C2CC2)CC1(C)C c1(C(N2C(CNC(CC3(CN(C)C)CCC3)=O)CC2)=O)cnc2cccnn12 C(=O)CCCc1nccs1.C1(CNC(=O)C=CC(=O)NC2CC2)CCC1 N1(C(CN(c2ccccc2)C)=O)CC2(CC2)CC1C.C(=O)(C(F)n1ccnc1)N CC(C)CCC(F)C(=O)N1CCC(C(C)C(N2CC3CCC3C2)=O)CC1 N1(C(C(CC)NC(C)=O)=O)CCN(C(C2CSC2)=O)C(CC(F)(F)F)C1 N1(C(C(C)(C)OC(C)C)=O)CC2(CCN2C(C23CCCN2CCC3)=O)C1 CC1CN(C)CC(C(=O)NC(C)C(C)C(=O)N2CC(CC(C)(C)C)C2)O1 C12(C(=O)NC(CCC)CC)CCC(NC(C3CC(C(C)C)=NO3)=O)(CC1)C2 c1(NCCC2CCN(C(C(C)C)=O)C2)ncnn2c(Br)ccc12 c1(CC)ccccc1C1CC(=O)N1.N(C(=NCC)NC1CC1(C)OC)C(C)C C(=O)(C1CCCc2c[nH]nc21)NC(CC)(C)CNC(C1CC2(CCCC2)C1)=O CC(C)CC(C)CC(=O)N(C)CCOCCN(C(=O)C=Cc1ccco1)C C(=O)(CC1=CCCC1)N1CCN(C2CCN(C(=O)CN3CC4CC4C3)C2)CC1 CC(C)CC(CCO)NC(=O)C(Cn1cncn1)NC(=O)CO.c1nc[nH]n1.C C(=O)CC(O)C(C)CC.c1(C(N(CC)Cc2cnn(C)c2)=O)c(C)nnn1C c1(SC)nc(NCC(CO)C(C)C)cc(O)n1 c1(C(=O)NC2C(NC(C(C)CC3CCC3)=O)CCCC2)c[nH]c2ncccc12 CC1(C2CN(C(C3CSCCN3C(=O)CCc3nc[nH]n3)=O)CCO2)N=N1 C1(NC(C(=Cc2ccncc2)C)=O)CCC(C)(C)CC1C.c1(C=O)n[nH]cc1F.N Cc1c(C(N2CCCC23CN(C(c2cn(C)cn2)=O)C3)=O)ccc(F)c1[N+](=O)[O-] N1(c2ccnc(NC(c3ccccc3N(C)C)C)n2)CCOc2cccc(F)c2C1 C(C)(CCOC)NC(C1(CCOC)CC1)=O.c1(C=O)ccn(C(C)C)n1 C1(NC(C2COCCO2)=O)CC1C1CCN(C(=O)C2=CSCS2)CC1 c1(C(=O)NCC(CNC(COCCC(C)C)=O)CO)cnc2ncnn2c1O C(=O)(CCN(OC)C(=O)C(F)CCC)NC(C1CCOCC1)C#C C#CCCCCCCC(=O)NCC1CN(C(=O)CSCC2CCCCO2)CC1C CC1CN(C(c2csc(-c3ccoc3)n2)=O)CC(C)C1NC(c1cccs1)=O N1(C(c2c(C)snc2)=O)CCC2CN(C(C3(O)CC3)=O)CC2C1 C(Cn1cncn1)(C(=O)N(C(C)C(=O)N(C)C)C)NC(CSCC)=O CC1C(NC(c2cnc3c(c2)NCC3)=O)CC2CCC1N2C(=O)Cn1ncnn1 CCCCC(C(=O)N(CCCCNC(=O)CCN1CCCC1=O)C)C(C)C C(C)(C(=O)NCCC1CC(C)=NO1)(N(C(CC)=O)C)C1CC1 C1(NC(C=C2CCC(C)CC2)=O)CC(O)CN(C(C2(C(F)F)CC2)=O)C1 N1(C(c2c(C)nc(O)nc2C)=O)CCC2CC1CN(C(=O)CC1CC(C)(C)C1)C2 N1(C(C=C(CC)C)=O)CC2(NC(=O)Cc3sc(C)nc3C)CCCC2(F)C1 c1(C(N2CC3(COC)CC2(CO)C3)=O)cc2c(C)cccc2o1 C(=O)(C(CC=CCl)c1ccccc1)NCC(CNC(COCCSC)=O)C c1(NCC2C3CN(C(C(C(CCC)CC)O)=O)CC32)ccc([N+](=O)[O-])c(OC)c1 c1(C(=O)NCCCCC2CN(C(CC)=O)C2)cc(C)c(Cl)cc1OC c1(C(=O)NC2CC(NC(c3ccc(OCCF)cc3)=O)C2)ncnc2sccc12 N1(C(c2n[nH]c(C)c2C)=O)CCC2(CCC(N3CC(N(C)C)C3)CC2)C1 C1(C(N2CCCC(NC(C=CC3COC(C)(C)O3)=O)C2)=O)CC2(CCCCC2)C1 CC1CCC(=CC(=O)NCCC(C)CCNC(c2c[nH]c(C#N)c2)=O)CC1 c1(C=O)nnn2ccccc12.C(C)(C)(C)OCCNC(C1C(C(C)C)C1)=O c1(CNC(C(C=C)(C)CC)=O)n[nH]c2c1CN(C(=O)CNC(=O)CCC)CC2 CC(O)C(C(=O)NCC1CCC(C)(C)O1)NC(C1CC2CC2C1)=O C1(NC(CCn2c(C)csc2=O)=O)CCN(C(=O)CC(C)F)C12CC2 c1(C(=O)OCC(N2CCN(C(CC(=C)C)=O)CC2)=O)cc(F)cc([N+](=O)[O-])c1N c1(C(=O)NCCCC)cccc(OC)c1.C1(C=O)CCNC1=O.C(=O)C.N C(C)(O)(CN=c1ccc(Br)c(S(=O)(=O)NCC2CCC2)[nH]1)c1c(C)cc(Br)cc1 c1(OCC=C)ccc(Cl)nc1C(=O)NC.C1CCN(C(C2(O)CCC2)=O)C1.C N1(C(c2c(NC(CCC=C(C)C)=O)cnc(F)c2)=O)CCc2sccc2C1 C12(C(=O)NCCCc3cn(C)nc3)COCC1CN(C(C1CC1(Cl)Cl)=O)C2 c1(N(CCC)CCNc2nonc2C(C)C)cc(=O)n(C2CCCCC2)c(O)n1 N1(C(C=C(C)C(C)(C)C)=O)CCN(C(=O)CSc2ccncc2)CC1CC(F)F CC(CC(=O)NC1(CF)CCN(C(=O)CCc2nccn2C)C1)C(F)(F)F C1(C)(C(=O)NCC(C(C)O)C)CN(C(=O)CCC2CCCCO2)C(C)(C)C1 C1(Cl)(C(=O)OC)CC12CCN(C(=O)NCC1CCN(CCO)CC1)CC2 C1(C(N(C)CC2N(C(C(C=C)OC)=O)CCC2)=O)CCC(F)(F)CC1 C1(OC)CN(C(=O)Cc2cccc(Cl)c2)C(C)(C)C1.C1(C(=O)N)CCCCC1O C1(c2ccccc2)CC(NCc2ncoc2C2CC2)CCO1 C1(C(N2CC(COC)(C)C2)=O)C2CCCCCC12.C1(C(=O)N)(CCO)CC1 CCC(C)(CNC(=O)CC1CCSC1)C(=O)NC1CCCOC1 c1(CC)occ(C)c1C(N1CCC(N(C(C2COC(C)(C)C2)=O)CC)C1)=O N1(C(CC(CC)CC)C(=O)Nc2ccccc2C)CC(O)CC2(CCCC2)C1 CC(C)(C)C#CC(=O)NCC(CC(F)(F)F)NC(C1(CF)COC1)=O c1(NC(C2CC23CCN(C(c2cccc(O)c2)=O)C3)=O)ncc(Cl)nc1Br N1(C(c2cc(C(C)C)on2)=O)CCN(C(C2CC3C=CC2C3)=O)CC1CC#N Cn1cc(C=CC(N2CCNC(CCO)C2)=O)nn1 CN1N=C(C(=O)N2CCC(NC(=O)CCN3CCCCC3)C2C2CC2)CCC1=O c1(CC(=O)N(C2CCCC(N(C)C(c3cnsc3)=O)C2)C)cccc(F)c1F c1(C(N2CC(C(=O)NC3CC(C(=O)OC)C3)(CF)C2)=O)cc(C)ccc1C C=CCC(C)(C)C(=O)NCCC(Cc1ccccc1)NC(c1ccc(F)s1)=O C(C(C)(CC(C)C)NC(c1cc(C)c[nH]1)=O)NC(CCN(C(CC)CC)C)=O CC1CN(C(=O)CSCC2CCCCO2)CCC1N=c1ccnc(S(C)(=O)=O)[nH]1 C1(C(N2C(CNC(c3cccnc3O)=O)CC(C)(C)C2)=O)CC2CCCCCC12 CCCC(O)CC(=O)NCC1CC2(CC(NC(c3ccc(Br)o3)=O)C2)C1 C12(CCN(C)CC1)c1nc2no1.C1CC2(CC2)CN1.CC c1(C(N2CC(N(C(C3(C#C)CC3)=O)C)C2)=O)cc2cccc(C)c2[nH]1 N1(C(C=CCCC)=O)CC2CCC2(NC(c2cc(OC)nc(F)c2)=O)C1 C1(F)(CNC(CNC(CCC)=O)=O)CCC1.C(=O)(C(F)CC1CCCC1)N c1(C(=O)NC(CC)CN(C(=O)COCCCOC)C)cc2sc(C)nc2[nH]1 C12(C(N3C(C)(C(=O)N)C=CC3)=O)CCCC1C2(F)F.C=CC1CC1(CO)C N1(C(C(C)(C)OC)=O)CCCc2cc(OC)c(Cl)cc21 c1(N(CC(C)NC(c2ccnc(O)c2)=O)C)nccc(C#N)n1 C(=O)(C(F)(F)C(C)O)NCC(C)N(C(c1nc(C)n(C(F)F)c1)=O)C N1(C(=O)NCC(C)(C)c2cccs2)CC2CCOC2(CO)C1 CS(=O)(=O)CCC(=O)NC1CCN(C(c2cccc(F)c2N)=O)CC1F c1(CC)ccc([N+](=O)[O-])cc1C(=O)NCCCC.C1(CC=O)CC(=O)NC1=O C1(NC(CCC(=C)Cl)=O)CN(C(=O)Cc2csc3nccn23)C2(CCCOC2)C1 C1(O)(C(C)C)CCN(C(=O)C(CCF)NC(=O)C(O)C2CCC2)C1 C1(C)(CNC(C(C)OCC)=O)CCCN1C(=O)CC1CSCCS1 Cc1oc(Cl)nc1C(=O)NC.c1(C=O)cnc(-c2ccco2)s1.C1(CC)CC1 c1(NCC2(C)CCN(C(c3n[nH]c(C)c3C)=O)C2)ncc([N+](=O)[O-])cc1Br C1(C(=O)OC)CCc2nc(NC(C3(COC(C)C)CC3)=O)ncc2C1 c1(C(=O)NC(C2CCCN2C(=O)CO)C)ccnn1C1CCC1.C1CCOC1 Cc1ccc(C(N2CCC(C(C)NC(c3n[nH]c(C)n3)=O)CC2)=O)c(N=[N+]=[N-])c1 C1(NC(C23CC(C)C2C3)=O)COC2(CCN(C(c3ccc(F)o3)=O)CC2)C1 N1(C(CNC(CC(C)(C)C)=O)=O)CCC(C)(C)C1CNC(c1cn[nH]c1)=O CC(=O)CCCC(C)C(=O)N1CC(C(=O)NOC(CO)C(C)C)CC1(C)C C(C(=O)NCC(C)CO)(C(C)(C)C)SC.c1(CCC(=O)N)cc(C)cc(C)c1 C1(NC(CCC(=O)N(C(C)C)C)=O)CN(C(C2C3CCC(F)(F)C23)=O)CCC1C c1(NC(C(=O)N(C2COC(C)(C)C2)C)=O)cccc(C(N2CCC(O)C2)=O)c1 N1(C(C(C=C)OC)=O)CCOCC1CCNC(c1ccc[nH]1)=O N1(C(C2(N)CC(c3ccccc3)C2)=O)CCCCC1C1CCCO1 N1(C(CC)=O)CC(O)CCC1C(=O)N(C)CCN1CCCCC1 c1(OC)cc(C(=O)N(CCCNC(C2CCC2(F)F)=O)C)c(OC)cc1Cl c1(C=O)ccc(C#N)c(O)c1.CC(CNC(=O)CC)C.c1(C=O)ccoc1.N c1(C(=O)NCCCN(C(=O)C(O)C(F)(F)F)C)c(F)cncc1Cl C=CCC(C)(C)C(=O)NC(C)C(C)NC(=O)CNS(=O)(=O)CCCO C12(CNC(C(CSC)O)=O)CC(CCO1)N(C(c1ncnc3cc[nH]c13)=O)C2 C1(C(=O)NC(CCCC)COC)CC2CC1CN(C(=O)COC(C)=O)C2 C1(C(CNC(C=CCOC)=O)(C)C)CCCCN1C(c1cc(Cl)n[nH]1)=O N1(C(CC2C(C)(C)C2(C)C)=O)CCC2(CCCN(C(=O)Cc3ccon3)C2)C1 CCCC(C)(C)C(=O)N1CC(NC(C2CCCN(C(=O)C(C)C)C2)=O)C(F)C1 C1(C(C)C)CN(C(=O)Cc2ccccc2F)CCN1C(=O)CC1(C)CC1 N1(CC(=O)NC(C)(C)CCNC(=O)CC2CCCO2)C(=O)CCCC1=O C(=O)(CC(C)(C)C=O)OC.C12CC1CN(C(c1cnc(C(C)(C)C)[nH]1)=O)C2.N C1(NC(c2c(CC)nns2)=O)CC2CC(C1)N(C(C1CC1(C)C)=O)C2 Cc1c(C(=O)OC(C)(C)C)sc2ccccc12.c12ccccc1CN(C=O)C2C C1(C(=O)NCc2occc2C(N2CCC(CCCO)CC2)=O)CC2(CCO1)CC2 c1(C(N2CCCC(CNC(=O)CCc3cnn[nH]3)C2)=O)ccc(Cl)cc1Cl N1(C(C2CC(C(=O)OC)C2)=O)CCC(F)(C)CC1.C(=O)C(Br)=C(C)C.N c1(C(=O)NCCCC(C)(C)NC(C(CC=C)CC)=O)cc(P(C)(C)=O)cs1 C1(C(=O)NC(CCC)c2nn[nH]n2)CCCC1CNC(=O)CN1CCCC1C C1(NC(c2n(CC=C)nnn2)c2ccc(CC3CC3)s2)CCc2nc(C)cn2C1 Cc1nc(O)c(C(N2CCCC(N(C(=O)COC(C)C)C)C2)=O)cc1Br Cc1onc(O)c1C(N1CCCC(C(C)NC(c2cnn(C)c2C)=O)C1)=O c1(CC)nn(C)cc1C(=O)N.C1(CCC)CN(C(C2(Cl)CC23CCC3)=O)CCO1 C1(CCCC)CCCC1NC(=O)C=CCNC(C)=O c1(C(N2C3C(NC(C(CC#C)O)=O)(CCC3)CC2)=O)cc(S(N)(=O)=O)cnc1C c1(C(=O)NC2CN(C(=O)Cc3ccno3)C2)cncc2cccnc12 O(N(CC)C(=O)C(C1CCCO1)NC(=O)C=Cc1ccccc1)CC CC1(C)CC(n2nc(-c3ccoc3)nc2-c2cnn(-c3ccccc3)c2)CCO1 C1(NC(COC(C)C)=O)CCC2(CC1)CCC2.c1(C=O)sc([N+](=O)[O-])cc1Cl.N CC1CC(=O)NCCN1C(C1(NC(C2CCCCNC2=O)=O)CCOCC1)=O Cc1cc(NCC2CC(C)CO2)c(F)cc1[N+](=O)[O-].c1(C(=O)N)ccnc(F)c1 c1(OCC)ccc(F)cc1C(N1CCN(C(=O)C)CC1)=O.C(=O)(CC(C)F)N Cc1nc2cc(C(=O)NC3(CO)CCCN(C(C4(C)CCOC4)=O)C3)ccc2o1 C1(CNC(CC(=C)C)=O)(NC(=O)CCN2CCOC2=O)CCCCCC1 C(=O)(C(F)C(C)(C)O)N(CC(CC)NC(c1cnsn1)=O)C N1(C(C(C2CN(C(=O)CC3CCCC3)C2)OC)=O)CCC(COC)C(O)C1.C N1(C(C2C(CNC(=O)Cc3ncccn3)CC2)=O)CCCN2CCCC2C1 S(=O)(=O)(c1cccc(Cl)c1F)NC1C2(CCN(C(C(C)(O)C(F)(F)F)=O)CC2)C1 C1(CC=C)C(NC(=O)CONC(=O)CC2(C)CCOC2)CC1O N1(C(c2nc(C(C)OC)sc2)=O)CCC2(CCC2NC(=O)C2=CCCOC2)CC1 Cc1cc(=NC(=O)C(=O)N2CCC(Nc3nc(C)nc(C)c3F)CC2C)[nH]o1 C1(CC(=O)N(CCCCO)CCC)CN(C(=O)CCC(C)CC)CC12CC2 N1(C(c2c(C)noc2)=O)CCCCC1.C1(C=O)CC1C=O.C(C)(C)C.CC.N c1(C(N2CCC3(CCN(C(C=CC=C)=O)C3)C2)=O)cc([N+](=O)[O-])c(F)cc1N.CC C1(C(N2C(CN(C(=O)Cc3ccoc3)C3CC3)CCC2)=O)CCn2nncc2C1 C1(CC)CN(C(C2(CCF)CCC2)=O)CCN1C(c1ccc(C(=O)OC)o1)=O C1(CCNC(C2(O)CCN(C(c3ccccn3)=O)CC2)=O)CCc2nccn2C1 C(=O)(C#CC(C)(C)O)NC(C)C(CO)NC(=O)C(N1CCCCC1)C C1(CNC(C(CC=C)NC(C2CC2(F)Cl)=O)=O)CCCC2(CC2)C1 N1(C(Cc2c(C)non2)=O)CCCC(C2CCN(CCN3CCOC(C)C3)CC2)C1 C(=O)(C(O)CC(F)(F)F)N1CC(C)(C)C(C(N2CC3CCCC3C2)=O)C1 N1(C(C(C)P(C)(C)=O)=O)CC(NC(=O)CCSC(F)(F)F)C2(CCC2)C1 [N-]=[N+]=NCCCC(=O)NC1CN(C(=O)C2=CCOC2)CC1F CC1CCN(C(=O)C2=CCCS2)C(C)C1NC(=O)Cc1cnn(C)c1 Cc1oc(Cl)nc1C(N1CCC(N(C(=O)C=Cc2ccccn2)C)CC1)=O C12(C(=O)NCC3(O)CCN(C(CCC=C)=O)CC3)CCOC1CS(=O)(=O)C2 C1(CC=C)(NC(c2ccn(CC3CC3)n2)=O)CCN(C(c2occc2Br)=O)C1 C1(NC(C(C2CCN(C(C(COC)C)=O)C2)C)=O)CC(C)(OC)C1(C)C c1(C(N(C2CCN(C(C(COC)COC)=O)C2)C)=O)ccc(F)c2cnccc12 N1(C(C(C)(C)OCC)=O)CCC(C2CC2)C1.c1(C=O)cc(C2CCC2)[nH]n1.N c1(C(N(CC(CNC(C(COC)N(C)C)=O)(C)C)C)=O)ccnc2[nH]nnc12 c1(C(C(N2CCC(NC(C=C(C)Cl)=O)(CF)C2)=O)O)c(C)cccc1C c1(C(N2C(C(=O)OC)CCC2)C(=O)NCCCC2CC2)csc(Br)n1 CC(C)(CNC(=O)CC)C(F)(F)F.C1(C)CN(CC(F)F)C1.C(C)(C)C CCC(CC)CC(=O)NCC1(O)CCN(C(=O)C(C)C(O)CC)CC1 N1(C(CC2C=NN(C)C2=O)=O)CCCC(F)(C(=O)NC2CCCC(N(C)C)C2)C1 Cc1onc(CO)c1C(=O)N(CC(C)NC(=O)CC1CCOC(C(C)C)C1)C CC1CC2CC2CC1C(N1CC(CNC(C2CCOC(C)(C)C2)=O)C1)=O CCCCC(C(=O)NC(CCC)C(C)(C)C)NC(=O)CCc1ccc[nH]1 N#CCCCC(C(=O)NCC1CC1)N(CCCO)C1CC1 C1(c2n(CCOC)nnn2)(NCc2ncc(Cl)n2C)CCC(C)(C#N)C1 C1(C(C)(C)C)(CNC(c2occc2Cl)=O)CCN(C(=O)C=CC2CCC2)C1 N1(C(CCCCCN(C)C)=O)CC2(C(=O)NC3CC34CCCC4)CCC1CC2 C(c1ccc(F)cc1F)=CC(=O)NCC1OCCN(C(C2C(C)(C)CC2)=O)C1 c1(C(N2C3(C(N4C(C(C)O)CC4)=O)CC(C)(C2)C3)=O)cccc2[nH]ncc12 c1cncc(Cl)n1.C1(NC=O)(CO)CN(C(=O)C)C1.c1(C=O)ccccc1.N c1(NCCC(C)CO)ccc(S(=O)(=O)NC2CCn3cnnc3C2)cc1F C1(C)(C(=O)NC2C(C)CN(C(C34CC(C)C3C4)=O)C2)C(C)(C)C1(C)C N1(C(c2cn(CCC)nc2)=O)CCCCC1CNC(C1CC=CC1)=O C=CC(CC)CC(=O)N1CCN(C2CCCN(C(c3cocn3)=O)C2)CC1 C1(CC(=O)NC2CC(CCNC(C3CC4(CCC4)C3)=O)C2)CCCCC1F N1(Cc2ccc(C)o2)CCC2(CCCC2C(N2CCC(Br)C2)=O)C1 c1(N(CC(=O)N(C)C)C)nc2ccsc2c(=NCC(=O)NCCS(C)(=O)=O)[nH]1 C(=O)(CC(O)C(C)CC)N1C(C(N(C2CC(=C)C2)C)=O)CC(F)(F)C1 c1(C(=O)NC(C2CCN(C(=O)CC3CC3)C2)C)[nH]c2ccccc2c1Cl c1(NCCC(N2CC(C(C)NC(CC3C(C)C3)=O)C2)=O)ccccc1 c1(CC(CC)NC(C2CC(n3cc(-c4csc(CO)c4)nn3)C2)=O)ccc(Cl)s1 CCC(CC(C)C)C(=O)OC1CCN(COC(=O)Nc2ccccc2)CC1(F)F C1(C(=O)NCCC(COC)O)CN(C(C2CCC2(OC)OC)=O)CCO1 c1(OC)ccncc1C(=O)NCC1CCN(C(C2CC(C)OC2=O)=O)CC1 c1(C(N2CC=CC2)=O)ccc(O)c(C(C)C)c1.c1(OCC)nc(C=O)co1.N C(=O)(C(F)CC(C)(C)C)NCCCCCN(C(C(C(C)C)C1CCC1)=O)C(C)C c1(OCCC)ccccc1C(=O)N(C1CCN(C(=O)CC2CCOC2)C1)C C1(C(N(C(CC)CNC(=O)COCCN(C)C)C)=O)CNC(=O)N1 Cn1cc(C=CC(=O)NCCCCNC(C2(O)CC2(C)C)=O)cn1 C(=O)(CC(C)(C1CCC1)C1CC1)NC(C1(C)CC1)C.c1(C=O)ccno1 CC(C)CC(O)C(=O)NC(CC(=O)NCCN1CC=CCC1)C(C)C N1(CCC)CCCC(C(=O)NCC2CCN(C(=O)CN)C2)C1.[SH](C)(=O)=O c1(C(=O)NC2CCS(=O)(=O)NC2)nc2cnccc2s1 CC1(C)C(CNC(=O)C=Cc2cc(Cl)sc2Cl)CCN1C(C1CC1C#N)=O C1(NC(c2c(C)cco2)=O)CC2(CCCCC2)C1.C(=O)CC1(N(C)C)CC1.N c1(C(N2C(CN(C(CCC=CC)=O)C3CC3)CCC2)=O)cnn(C)c1Br Cn1cccc1C(=O)NCCOC1CN(C(c2n[nH]cc2F)=O)C1 c1(C(=O)NCCC2CC(NC(=O)COCCF)C2)ccc(CO)cc1 C1(C(=O)OC)CCSC12CN(S(=O)(=O)CC(C1CCCC1)OC)C2 c1(C(=O)OC)ccc(O)c(C(N2CCOC(C(C)NC(=O)C(C)CO)C2)=O)c1 c1(C(N2CCC(NC(C(=O)OCC)=O)C(F)C2)=O)c(Br)ccc2ccccc12 N1(C(C(CC2CC2)NC(CCc2n(C)cnn2)=O)=O)CC2(C=CCO2)C1 c1(C(N(CC(=O)NCCC(O)C(C)C)CC)=O)ccc(=O)n(C)n1 N1(C(C(Cc2cn[nH]c2)NC(C(CC)N(C)C)=O)=O)CC2CC(OC)C(C2)C1 c1(CC(=O)N(C2CN(C(c3ccn[nH]3)=O)C2)C)ccc(C(F)(F)F)cc1.CC c1(C(=O)NC(C)C(C)NC(C2CC(OC(F)F)C2)=O)cc2c(s1)CCCCC2 C1(C)(C(N(C(C#C)C)C)=O)C=CCN1C(c1nc(O)sc1C)=O c1(C(=O)OC)cncc(C(=O)NCCNC(C2SCCC2C)=O)c1C c1(CC(=O)NCCNC(C2CN(C(=O)Cn3cccn3)C2)=O)csnn1 c1(N2CCC(O)C2)ccnc(C(C)C)n1.c1(C(CN)SCC)cnn(C)c1.C C=CCC(C(=O)N1CC2CCC(C1)C2NC(=O)CN1CCCC1C)C(C)C c1(C(=O)NCCC(=C)C)ccc([N+](=O)[O-])[nH]1.C(=O)(CC)N.[SH](=O)(=O)CC N1(C(c2cc(CCC)on2)=O)CCC2CC(C(N3CCC(C)C3(C)C)=O)C2C1 c1(C(N2C(C)C(C)N(C(c3cnc(Cl)[nH]3)=O)CC2)=O)c[nH]c2cccc(Cl)c12 C(=O)(C(F)C(C)C)NCC(CC=C)NC(=O)CCCCN1C(=O)CCC1=O C(=O)(C(C(F)(F)F)C(F)(F)F)N(C1CCCC(C)C1C)CC(C)(C)C S(=O)(=O)(C1CCN(c2ccccc2)C1)N1CCN(C(C)=O)CC1 C1(C(C)(C)CNC(=O)CCc2cn[nH]c2)CCN(C(=O)C)CC1.C(=O)(C)N c1(OC)ncnc(C)c1C(N1CCCCC(NC(=O)Cc2c(C)n[nH]c2C)C1)=O N1(C(C=C(COC)C)=O)CC(F)CC1CN(C(=O)C(C1CCCCCC1)C)C C1(NC(c2c(F)cc(C)c(F)c2)=O)CCCC12CCN(C(c1n[nH]cc1C)=O)C2 C(CCN=c1[nH]c2cc(F)ccc2o1)N(C)CC1CCCCN1C(=O)C(C)(C)C c1(N(CCOC)C)ccnc(NCCCN)n1.C12(CC1)CN2.C(C)C C1(N(C(COCCC)=O)C)CN(C(c2cccs2)=O)CCC1C.C(=O)C1CC1.N N1(C(c2cnc(CC)nc2C)=O)CCC2(CCN(C(c3ccc(F)cc3)=O)C2)C1 N1(C(C(CC)(C)CC)=O)CC2CCC1C1CN(C(=O)Cc3cncc(O)c3)CC21 c1(C(C)=O)cc(C(N2CCCC2CN(C(C2CCCOC2)=O)C2CC2)=O)no1 N1(C(Cc2n(C)ncc2)=O)CC(C2CC2)(C(=O)NCCOC2CCOC2)C1 Cc1nn(C)c(N)c1C(=O)NCc1cc(C(N2CCC3CCCC23)=O)n[nH]1 C1(CNC(c2cccc(C#C)c2)=O)CN(C(c2cccnc2F)=O)CCC1(C)C N1(C(COCCCCC)=O)CC(CNC(=O)C(C#N)CCC)C2(CC2)C1 Cc1[nH]c(C#N)cc1C(N1CCN(C(C2COCCN2C)=O)C(C2CCC2)C1)=O c1(C(=O)NC2(CC=C)CCCN(C(=O)Cn3nccn3)C2)cc(F)cc(C=C)c1 Cc1cc(C(N2CCCC2C(C)(C)NC(=O)COC(F)F)=O)c(F)cc1N N1(C(CCC)=O)CCC(C(=O)NC(C)CC)CC1.C(c1nc(C)cs1)=CC=O.N CCCCCC(O)CC(=O)NC1CC2CN(c3ccnc(C4CC4)n3)CC2C1 c1(C(=O)NC2(C)CCN(C(C3(CF)CC3(F)F)=O)C2)cc(F)cc(F)c1N C1(CC(=O)NCC(C(C)C)(F)F)CN(C(c2cncn2C2CC2)=O)CCC1C N1(C(C(=O)NCC)=O)CCCC2CN(C(c3ccc(C(F)F)s3)=O)CCC12 CCC(C(=O)NC1CC1CC(=O)NCC1CC(F)(CO)C1)N(C)C C1(C(=O)NCCCN(C(C2CC(C)=NO2)=O)CC)CCc2ccccc2O1 c1(OC)cc(CCNC(=O)NCCCCOC)ccn1 C(=O)(CCC(C)C#N)NCCC1(C)CCN(C(Cc2nc(C)sc2)=O)C1 Cc1oc(C)c(C(N2CCC2CNC(c2ccc(C3CCCCC3)o2)=O)=O)c1C N1(C(C=CCN(C(C(C)S(N)(=O)=O)=O)C)=O)C2CCC1CC(=O)NC2 c1(NCC(C)C(C)(F)F)cccc(N2CCN(C(=O)N(C)C)CC2)c1Br C1(NC(C2CN(C(=O)C3CC3)C2)=O)CCN(C(=O)c2ccc(Cl)cc2)O1 CN1CCC(C(=O)NC2(C)CC(C(=O)NCC3CCSCC3)C2)C1 c1(OC)cc(CC(=O)NCC(CCNC(=O)CC(C)F)OC)on1 C=CC(C)(CCOC)C(=O)N(C)CC=CC(=O)NCC1(OC)CCCCC1 c1(OC)cc(CN2CC3CC3(C(N3CCN(C)C(C)C3)=O)C2)c(Br)cn1 N1(C(CC(=O)OC)=O)CCC2CC(NC(=O)C(n3cc(Cl)cn3)C)CCC2C1 CC(C)(C#N)CC(=O)NC1CC(C(=O)NC2(CCCF)CC2)C1(C)C C1(C(N2CCC(CC)(NC(C3CCC(CC)O3)=O)C2)=O)CC(F)(F)C1(C)C c1(CNC(C2CC(=C)CN2S(=O)(=O)CCCCl)=O)cccc2[nH]ccc12 C1(C(N(C2CC(C=O)C2)C)=O)CC(C(C)C)=NO1.C1(C)(COC)CCCC1 c1(OC)c(S(=O)(=O)NCC)cc(Br)c(C)c1[N+](=O)[O-].c1(C(=O)N)ccnn1C CCCC(C(=O)N(CC(c1nn[nH]n1)C)C)NC(=O)CCC(C)OC C(=O)(C(F)C(=O)N1CCCC(CCNC(c2conc2C)=O)C1)OCC C1(CCC(N2CC(OC)C2)=O)NC(=O)NC1=O.C1(C2CC2)(CC=O)CC1.C C(=O)(C(N=[N+]=[N-])C(C)C)NC1CCCC(C(=O)NCC(CCC)(C)O)C1 C1(C(N2CC(CC)OCC2)=O)CCC2CC2CC1.C(C(=O)N)NC(=O)OCC c1(CC(=O)N(CC(CN(C(C2CCN(CC)C2)=O)C)O)C)ccc(C)c(F)c1 c1(OC)nc(C(=O)NC2CCN(C(c3cccc(Cl)c3C)=O)CC2F)cc(O)n1 C1(C(=O)NC(C)CCCCNC(=O)C(C)(C)c2ccsc2)CC2(C1)CC(F)C2 N1(C(C(=O)NC)C)C2CCC1CN(C(c1cscc1C)=O)CC2 N1(C(C(=O)Nc2ccccc2)=O)CC(NC(C2CC2c2ccoc2)=O)C(O)C1 N1(C(COCc2cccc(OC)c2)=O)CCN(C(C2(F)CCOC2C)=O)C(C)C1 NS(=O)(=O)c1ccc(CCc2noc(CC3(CO)CC3)n2)cc1 CC1CN(C(C2(c3cccs3)CCOCC2)=O)CC1NC(=O)COC.C1CC1 C(=O)(C(CC(F)F)N(C(=O)Cc1ccn(C)n1)C)N(C1CCCN(C)C1)C C(CCCCCC(=O)N(C(CNC(C1CC1c1ccccn1)=O)C1CC1)C)SC c1(NC(C2N(Cc3ncc(C)nc3)CCC2)=O)ccc(F)cc1C(F)(F)F c1(C(C)O)nnc(N2CCC(CC3CC3)CC2)n1CC(=O)NCC(F)F Cc1ccc(F)c(CN2CCCC2C(=O)Nc2ccc(CO)cc2)c1Br C1(C(=O)NC(c2ccc(OC)c(F)c2)C(F)F)CCC2(COC2)OC1 C1(C#N)(C(=O)NCC(CNC(c2nc(C)sc2C)=O)C)CCCCC1 c1(CC)nn(C)c(C(=O)N(C(C)C2CC2)C)c1Cl.c1(CC=O)sc(O)nc1O C(=O)(NNc1ccnc2cc(Cl)ccc12)N1C(C)C(C(F)(F)F)CCC1 Cn1ncc(-c2nnc(SCC3CCN(C4CCCCC4O)CC3)o2)c1Br c1(C(N2CCCC(NC(CC3(C)CCOC3)=O)C2)=O)ccnc2c1CCC2 Cc1c(C(N2CCC(N(C)C)C(NC(c3cc[nH]c3)=O)C2)=O)ccc2c1OCO2 c1(OC)cc(C(N2CC3CCC2CN3Cc2cccnc2F)=O)ccc1[N+](=O)[O-] C(=O)(CCC(F)F)N(CCC(C)C)CC.c1(CC=O)ccccc1.C(=O)CC.N c1(C(=O)NCCN(C(C)(C)C)C(C2CC3CC3N2)=O)cccc(Cl)c1O C1(C(=O)NCC2(NC(C3COC(=O)O3)=O)CCCCC2)CCc2nccn2C1 Cc1nc(O)c2ccc(C(=O)NCCCNC(C34CC(CO3)C4)=O)cc2n1 c1(NCC)ncc(C(=O)NCCC2CC(NC(C3CCC3)=O)C2)cc1Cl C1(F)CCCN(C(=O)CN2CC3CC3C2)C1.c1(CCC)ccc(C(=O)NC)cc1 C(CN=c1nc(C(C)(C)C)nc[nH]1)(C1CC1)NC(c1cc(CCC)nn1C)=O C1(F)(CNC(c2[nH]cc(CC(C)C)c2)=O)COCCN(C(=O)C(N)=O)C1 CCC(C)CC(=O)NC1(C(=O)NC(CC)C(=O)NCCO)CSC1 C(C(COC)CC(=O)N1CC(CC(=O)NCCC2CC=CC2)C(C)C1)OC C1(C(=O)NC2(C)CN(C(C3(C(N(C)C)=O)CC3)=O)C2)CCC(F)(F)CC1 N1(C(C2(CC(=O)OC)CC2)=O)CC(NC(C2CC2(F)F)=O)C(C)C1.C Cc1cc(Cl)cc(C(=O)NC2C3CC2N(C(=O)CC2CC(F)(F)C2)C3)c1C n1(C2(C)CC2)nnnc1C(CC1CCOC1)NCCOCCC1CC1 Cc1nc(C(C)(C)C)ncc1C(=O)NC1CCC(=O)NC1c1ccccc1 c1(CC)nc(C(C)C)ccc1C(=O)NC(c1cn(Cc2nccs2)nn1)C c1(C(=O)NCCNC(C2C(C(C)(C)O)C2)=O)ncoc1C(F)(F)F Cc1ccn2ncc(C(=O)N(C)CC3CCN(C(=O)CN(C4CCC4)C)C3)c2n1 C1(C=O)CC2CCCC(C1)C2=O.c1(OC)cc(C(=O)NC(C)(C)C)c(F)cn1 C1(CNC(CC(C)NC(c2cc(Cl)no2)=O)=O)(CO)CC2CCC1C2 C(=O)(C1=NN2CCCN=C2N1)NC1CC(C)(CNC(C(C)OC)=O)C1 Cc1nccc(C(N2CCC(CNC(c3c(Cl)cncc3Cl)=O)C23CC3)=O)c1N N1(C(C(C)S(N)(=O)=O)=O)CCC2(CC1)CCN(C(=O)CC1CCN(C)C1=O)C2 C#Cc1cccc(C(=O)NCC(N2CCOC(c3ncno3)C2)=O)c1 C1(C(=O)NC(Cc2cc(C)[nH]n2)C)CCN(C(=O)c2occc2C2CC2)O1 c1(C(N2CCN(C(C(CC)NC(N)=O)=O)CC2CCO)=O)nccc2occc12 CCCC(CNC(C1CNC(=O)N1)=O)C(=O)N1CCC(CN(C)C)C1 c1(C(N2C3CC(CNC(CCOC(C)C)=O)(OC3)C2)=O)cnn2ccncc12 C1(C(=O)NCCCCNC(C(C)c2ccsn2)=O)CC(C2CC2)=NO1 C(=O)(C#CC1CCCCC1)NCc1c(C(=O)NC(C)CO)n(C)nn1 c1(C(=O)NCCCC(C)(C)NC(CC(C)F)=O)c(Cl)cccc1S(C)(=O)=O N1(C(C(C(CC)C)N(C(=O)Cc2cnccc2C)C)=O)CC2(COC(=O)C2)C1 C1(C=O)CC2(CCOCC2)C1.O=C1CCC(C(=O)NCC2(F)CC(C)C2)O1 c1(C(N2CC(N)(c3nn[nH]n3)C2)=O)c(F)cc(Cl)cc1Cl N1(C(Cc2c(C)nc(S)s2)=O)CC2(NC(=O)COc3cccc(F)c3)CCC1C2 C(=O)(C1=NOC(CNC(=O)CN(C2CCC2)C)C1)N(C(C(C)C)C)C CC1(C)CC(CC(=O)Nc2ccc(F)cc2)CN1C(c1cnc(=N)[nH]c1)=O S(=O)(=O)(c1cc(F)ccc1F)N1CC2(N(C(C3CC4CCC3O4)=O)CC2)C1 N#CC1CCCCC1S(=O)(=O)N1CC(N)CCC1c1ccccc1 CS(=O)(=O)c1ccc(SCC(=O)NC2CCC2)cc1.C(=O)(C#CC1CCCC1)N Cc1cnc2c(C(N3CC(NC(=O)C(C)C(C)(C)C)CC(F)C3)=O)cnn2c1 c1(CC(=O)NC2C(C)CN(Cc3noc(C4CCC4)n3)CC2)c[nH]c2cnccc12 c1(C(=O)NCCC(C(=O)NCC2(CCOC)CC2)O)nnc(O)nc1O C1(CC(=O)NCCC(O)CNC(c2c[nH]nc2-c2ccc(Cl)s2)=O)COCCO1 C1(COC)CCCN(C(=O)CC(C)n2cc(-c3ccnc(C)c3)nn2)C1 N1(C(c2ccn(C)c2)=O)CCOC2CN(C(C3CC4CC3CO4)=O)CC12 N1(CC(=O)NC(C2CC=CCC2)C(=O)NCCCCOC)CCOCC1=O C1(NC(=O)NCCCN(C)CC2CCCCC2)CCOC1C1CC1 N1(C(CC(CC)OC)=O)CCC(NC(=O)C(=Cc2cccnc2)F)C12CC2 C1(C(=O)NC2CC(NC(C(c3cn(C)nc3)(C)C)=O)C2)CCCN1N=O N1(C(c2cccc(C)c2)=O)CC2C3CCC(C2C1)N(C(=O)CC1CCCCC1)C3 C1(CCN(CC)Cc2nnc(C)o2)CCN(C(=O)CCC2CCOCC2)CC1 c1(OC)cc(Br)cnc1NC(C1CC(C)CN1Cc1c(C)n[nH]c1C)=O Cc1nn(CCN(C)C)cc1-c1nccn1C1CCCCC1C C1(C(C)(C)C)CNC(=O)CN1C(=O)CCCn1cc(C(C)(O)CCO)nn1 O=C1CC(C(=O)NCc2ocnc2C(N2CCC(n3ccnn3)C2)=O)CO1 c1(-c2n(-c3c(C)cccc3Cl)nc(C3CC3C)n2)ccc2[nH]c(C)c(C#N)c2c1 C12(NC(=O)Cn3ccnn3)CCCCC1N(C(=O)C(C1CCC1)C1CCC1)CC2 c1(OC)ncc(NC(=O)C(n2cc(CCN(C3CCCCC3)C)nn2)C)cc1Br c1(C(N2CCOC(Cc3cccnc3)C2)=O)cc2ccc(-c3ccncc3)cc2[nH]1 C1(NC(c2ccc(C(F)F)o2)=O)CC2CN(C(=O)Cc3ccc(O)cc3)CC12 N1(C(CCNC(CC(C)n2cccc2)=O)=O)CCOCC1CC(N)=O C1(CNC(Cc2cc(COC)on2)=O)CN(C(c2ccncc2Cl)=O)CCO1 C(CC(C(=O)N1CCOC(CN=[N+]=[N-])C1)NC(=O)Cc1c(C)noc1C)=CC c1(OC)ccc2[nH]cc(C(=O)NCC3CCCN3C(=O)C(F)F)c(=O)c2c1 c1(CC(=O)NC(CC(C)NC(=O)C2=NOCC2)C)ccc(Cl)c(Cl)c1 C=C(C)CC(C)C(=O)NCC(O)CNC(=O)CN(CCCCCC)C c1(C(=O)NC(CNC(C(CC=C)CC)=O)(C)C(C)C)cc2n(c1)CCSC2 C=CCC(CC=C)C(=O)NC(C1CC1C(=O)NCc1nc(C)co1)C C12COCCN1C(=O)CN(C(C1CCC(=O)O1)=O)C2.C(C(C)(C)C(=O)N)OC.C c1(C(N(C(CNC(=O)CCc2ccccc2O)C2CC2)C)=O)csc(Cl)c1Cl C1(CC(N2CCC(N(C(=O)CCOCC3CC3)C)C2)=O)CCCCCC1(F)F c1(C(N2CCN(C(CS(CC)=O)=O)CC2C2CCCC2)=O)ncnc2ccsc12 Cc1sc(Br)cc1C(=O)NCC1CC(O)CN1C(=O)CC1CCOC1 C=CCCC(C)(C)CNC(C1(F)CN(C(=O)C(C)COC(C)=O)C1)=O C12(CNC(CCC(CC)C)=O)CCC(CC1)N(C(=O)C(O)CC1CC1)C2 CN1CCN(C(C2CC3CCC(C2)N3C(=O)C(N)Cc2cscn2)=O)CCC1=O CC1(C)CCCC(CNC(C2CCN(C(c3cc(O)nc(O)n3)=O)CCO2)=O)C1 c1(OC)ncc(Cl)c(C(N2CC3CC(C2)C3NC(=O)CCn2cncn2)=O)c1Cl C1(C2(O)CCOC2)(C(=O)NCCC(CNC(c2ccc(C)n2C)=O)O)CC1 N1(C(c2n[nH]cc2Br)=O)CC2=C(C1)CN(C(C1(F)C3CCCC13)=O)C2 CC1CN(Cc2ccccc2Br)CC(C)O1.C12CCN(CC1)C(=O)Cn1cc2nn1 c1(C(=O)NCC2CCCC(NC(C3(CC)CCC3)=O)C2)ccc(N)cc1Br C1(C(=O)NCCCN(C(=O)C(C)OC2CCCCC2)CC)CC(C)(C)C1 N1(C(C=C(C)Cl)=O)CCc2ccccc2C(N(C)C(C2CCN(C)CC2)=O)C1 C1(CCNC(Cc2cnc(C)s2)=O)COCCN1C(C1CCC(=O)N1C)=O c1(CC)cncc(C(=O)NCC(C)N(C(=O)C(c2ccccc2)F)C)c1 C(CCCCCC(=O)N1CC(N2CCOC2=O)C1)NC(CC1N(C)CCCC1)=O CC(C)C(CCN(C)C(c1ccc(C(F)F)o1)=O)NC(C1(F)CCOC1)=O C#CCCC(=O)NCC(CNC(c1ncoc1-c1ccc(C)s1)=O)OC c1(C(N2CC(C)N(Cc3ccccc3)CC2)=O)cc(Br)cc2[nH]ccc12 CC(C)C(O)CC(=O)NCCC(C)(C)C(=O)Nc1ccc(F)cc1O C1(NC(C2C(CC(C)C)C2)=O)CN(C(C2(C#N)CC=CC2)=O)CC12CCOCC2 C1(NC(c2ccc(COC)cc2)C)CC(C#N)CC1O C1(C)(COC)CC(NC(c2nocc2Cl)=O)CN1C(c1cscn1)=O N1(C(COC)=O)CCOC2CN(C(c3cnc(OC)cc3C(F)F)=O)CC12 C1(N(C(=O)CC)CCC)CCN(C(=O)C(F)CC2CCCC2)C1.C(=O)(CO)N c1(CN2CC(OC)C(NC(c3c(C)cccc3F)=O)CC2)cc(I)cc(I)c1O C(=O)(N=c1[nH][nH]c2c(Cl)cccc12)C1(C)CCN(C(C(CCCCC)C)=O)C1 C1(NC(C2(C)CC2)=O)CCC(C(N2CCN(c3cccnc3)CC2)=O)CC1 O=C(CCCc1cnccn1)NCC=CCNC(C1CC(CC(F)F)C1)=O c1(N2CCC(NC(C3=NOC(C)(C)C3)=O)C(O)C2)nc(O)c2ccc(Cl)cc2n1 CCC(CC)C(C)C(=O)NC(CC)CC(=O)NCC1(C)CC2CCC1C2 CCCCCS(=O)(=O)CC(=O)N(C(CNC(=O)CCN1CCCCC1)C1CC1)C Cc1cccc(C2(C(=O)NCC3CCN3C(=O)C(C)CN(C)C)CC2)c1 c1(C(N(C(C)CN(C)C(C2CC2(C)C)=O)C)=O)cc(C(F)F)cs1 Cc1ncncc1C(=O)NCC(C(C)C)NC(c1ccc(-c2ccco2)[nH]1)=O c1(CNC(C2(CCC)CC2)=O)nnc2n1CCN(C(C1(O)COC1)=O)C2 N1(C(CSCC#C)=O)CC2(CNC(=O)C(C3CCOC3)OC)CC1CO2 c1(C(N2C(CNC(=O)C=C3CC3)CCC2)=O)c(O)cccc1Cl c1(COCC)nc2ccccc2c(=NCC2CCOC(C(C)C)C2)[nH]1 Cc1ccc(C=CC(N2CCC(N(C)C(C3COCC(C)O3)=O)CC2)=O)cn1 N1(C(CC2CCN(C)C2)=O)CCC(C)(NC(=O)CCOCCN(C)C)C1 n1(C(COC)C)nc(-c2ccoc2)nc1C1CCC1C(F)(F)F.COC c1(CC(=O)NCCCN(C(CNC(=O)OC)=O)C)cccc(Cl)c1Cl c1(CCC(=O)NCC2(NC(C(CC)n3ccnc3)=O)CCC2)ccc(Br)cn1 C(C(F)(F)C(=O)NC1CCC(N(C(=O)CC2CCCN2C(C)C)C)CC1)OC c1(CC)ccc(NC(C2COCCC2)=O)c(C)c1.C1(CC(=O)N)CCCC2CC12 c1(NC)cc(C(=O)NC2CC(c3cccc(C(=O)OC)c3)C2)nc2ccccc12 c1(C(N2C(CC(=O)NCc3ccc(C4CC4)nn3)CC2)=O)cc(O)cc(F)c1 N1(C(c2cc(C)sn2)=O)CCC(C2N(C(c3cn(C)[nH]c3=N)=O)CC2(C)C)CC1 N1(C(CN(C(=O)OC)C)=O)CCCC2(NC(c3csc4nnsc34)=O)CC2C1 c1(CC(=O)NCC(C2CCN(C(=O)C(O)c3cnc[nH]3)CC2)C)cnccc1Cl N(C(=NCC(C)(C)n1ccnc1)N1CCC2(CC(C(F)F)=NO2)C1)C(COC)C C12(NC(c3nncs3)=O)CCN(C(c3ccnc(-n4cccn4)c3)=O)CC1C2 N1(C(C2OCCC(C)C2)=O)CCC(C)(CNC(c2cc(C3CCC3)[nH]n2)=O)CC1 C1(N(C(C(C)OCCC=C)=O)C)CCN(C(C2(CC(C)=O)CCC2)=O)C1 C#CCC(O)C(=O)N(C(C)CN(C(=O)C(=Cc1cccnc1)C)C)C C1(C(=O)NC2C(CCOC)CCC2)CCN(C(C2CC=CCC2C)=O)CC1C c1(OC)ccc2[nH]cc(CN3CCC4(CC4C(N4CC(O)CC4C)=O)C3)c2c1 C(=O)(CCC(=O)NC1C2CC(NC(C3CCOCC3)=O)CC12)NC Cc1ccc(C)c(CC(N2CCC(CNC(=O)C(C)(Cl)Cl)C23CC3)=O)c1 CC(CC(=O)NCC1CCCCC1)C(C)(C)C.C(=O)C(F)(F)F.C(=O)(C)N c1(C(=O)OCC)cncs1.C1(CC)CCN(C(=O)C=C2CCC(C)C2)C1.N c1ccc(Cl)c(Br)c1N.c1(CN(CC)CC)cnc(Br)s1.C(=O)(C)N.CC N1(C(c2n(C)ccn2)=O)CCC2CN(C(=O)C(c3ccc(F)cc3)=O)CCC2C1 CC(C)C(CCN(C(=O)CSC(C)(C)C)C)NC(=O)Cc1ccsc1 C(c1ccccc1Cl)=C(C)C(=O)NC1CCC(N(C)C(C2SCCC2C)=O)CC1 C#CCC(C)(C(=O)N1CC(C(=O)NC)C1)NC(=O)C(C)C1CCOC1 c1(C(=O)NCC(N2CCN(C(CCCCCC)=O)CC2)C)ncnc2cc[nH]c12 c1(OCC)cccc2c1CN(CCc1ccc(Cl)nc1)C2 C1(C)(CNC(c2c(C)cns2)=O)CCN(C(C2(F)CC=CC2)=O)CC1 c1(C(C)=O)ccc(F)cc1NC(=O)C(CC(C)C)N1CCNCC2CC12 C1(NC(N2C(CNC(=O)OC(C)(C)C)CCC2)=O)CCC(F)(F)C1 c1(C(=O)NC2CC(NC(C3N(CC)CC3)=O)C(O)C2)cc(C)nc(O)c1 c1(Oc2ccc(NC(N(CCCC3CCOC3)C)=O)cn2)ccc(Cl)cc1Cl Cc1cc(C(N2CC3CC(NC(=O)C(C)(C)CO)C2C3)=O)cc2nc[nH]c12 N1(C(c2c(CC)csc2)=O)CC(CNC(C2CS(=O)(=O)C2)=O)CC(C)C1 c1(SC)cc(N2CC3CC2C3C(=O)Nc2ccc(OC(F)F)cn2)nc(C)n1 C(=O)(C#CC1CCCC1)N1CCCCC(C(=O)NCC2N(C)CCOC2)C1 C(=O)(C1=NOC2(CCC2)C1)N1CCOCC(C)(CNC(C2CC2F)=O)C1 c1(N2CCC3(C(COC)C3)CC2)nc(=NCC(C)OC)[nH]c2ccccc12 N1(C(c2ccc(CC)c(C)c2)=O)CC(C)N(C(c2ccsc2OC)=O)C(C)C1 N1(C(C2(NC(CCOCC)=O)CCCC2)=O)CCCC1(C)CO C1(NC(C2CCC(CC)O2)=O)CN(C(c2cc(O)ccc2C)=O)CC2(CC2)C1 C1(NC(c2c(C)n[nH]c2)=O)CN(C(C2COCC2(C)C)=O)C2(CCCCC2)C1 O=C(C1=COCCO1)NCc1nc(C2CCCN(C(=O)C(=O)N)C2)n[nH]1.C1CC1 Cc1cc(C#N)ccc1C(N1CC=CC(C(=O)N(C)CC2(F)CCCC2)C1)=O C1(C(N2CCC2)=O)(OC)CCCC(C)(C)CC1.C1(C=O)C2CC3C(C2=O)C13.C CC1(C(N2CC(F)(C#N)C2)=O)CCCN1C(=O)Cc1ccsn1 CC(C)C(C(=O)ON)C(=O)Nc1cccc(NC(c2cnccn2)=O)c1 N1(C(CC(C)F)=O)CCC(N=[N+]=[N-])(C(=O)N(C)CC2OCCC2(C)C)C1 c1(OC)cncc(CCC(=O)N(CC(O)CNC(=O)CC2CC(C)C2)C)c1 CC(C)CCC(O)C(=O)N1CC2CC2C1C(N1CCC(O)(CO)C1)=O N1(C(CN(CC)CC)=O)CCCCC1C1CCCN1C(c1ccc(C2CC2)s1)=O S(=O)(=O)(c1cc(C)ccc1F)NCC.C1(c2nnnn2C(C)C)CCOC(C)C1 N1(CCCc2onc(C)n2)CCC2(CC1)COC(CNC(=O)C=CC1CC1)C2 CC(C)CC(CC(=O)NCC1CCCC1N(C)C)NC(C1CCCCS1)=O c1(OC)cnc(C(N2CC(OC)C(NC(C3CC34CC4)=O)C2)=O)c(F)c1 Cc1cccnc1CC(=O)NCC(CC(=O)NCC(F)(F)CC1CC1)C1CCC1 C1(NC(c2[nH]c(=NC)sc2)=O)CCc2nc(C(F)(F)F)cn2C1 N1(CC(=O)NCC(C)N(C(=O)C)C)CCCC(C(N)=O)C1.c1ccccc1.S Cc1nnc2n1CC(C(N1CC3(C1)CN(c1nnc(CO)s1)C3)=O)C2 Cc1cnc(N(C)CCN2CCCC2)c(S(=O)(=O)NCC2CC2C2CC2)c1 c1(OCC)ccc(C(N2CCC(C(=O)Nc3ccc(F)c(Cl)c3)C2)=O)cc1C#N C1(c2n(CCOC)nnn2)(NCC(C)(C)c2ccsc2)CC2(CC2)C1 CC(C)(C)C(O)C(=O)N.c1(C2(C(N3CC(O)C3)=O)CCCC2)ccc(F)cc1.C Cc1nc(CC(=O)N(CCCCN(C)C(c2c(C)ncn2C)=O)C)sc1C c1(C(N2CCC(NC(c3c(OC)nccc3)=O)C(O)C2)=O)ccc2nsnc2c1 N1(C(c2c(CNC(Cc3cc(C)no3)=O)c[nH]n2)=O)CCSC(C)(C)C1 CCCC(C)(O)CC(=O)N1CCC(n2cccn2)(C(N2CC(O)(CO)C2)=O)CC1 C1(NC(c2cnc(OC)s2)=O)CN(C(=O)C(C)CCCC(C)=O)CC2(CCC2)C1 C12(CNC(c3[nH]c4cc(C)oc4c3)=O)CCCCC1N(C(=O)CCCCO)CC2 C1CCC2(CN(C(C3CC(O)CN3C(N)=O)=O)C2)O1.CC1CC1C(=O)N.C CCCC(C(=O)N(CCC(=O)NC1CCN(CC)C1)C)C(C)C c1nnnn1C1CCCC1.C=CCCOCC(=O)NC1CC1C.C(=O)C.N CCCCC(O)C(=O)NC(CCOCCO)C(=O)NC1CCCC(C(N)=O)C1 N1(C(c2ccc(C)nn2)=O)CCN(C(=O)C(F)(F)c2csc(Cl)c2)CC(O)C1 Cc1nc(C)c(C(=O)NC2CCOCC2NC(c2c(Cl)noc2C)=O)[nH]1 Cc1nc2nccc(C(N3CCC(NC(c4ccoc4Br)=O)C(C)C3)=O)n2n1 C(=O)(CC(C)CC(C)(C)C)N(CC(C)(C)NC(c1ccc(CCC)c(N)c1)=O)C C(CC(C(C)C)c1ccccc1)NC(C(=O)NC(C#C)C)=O CCC(C)CCC(=O)NC1(C2CCCN2C(=O)C)CC1.c1(C=O)cc(C)on1.N CC(C(=O)NCC(CC1CC1)C(=O)NCCC1(O)CCC1)C(C)(C)C c1(C(=O)NCC(CC)NC(c2ccn(C)c2)=O)cccc(Cl)c1 C(=O)(N1CC(O)C(O)CO1)C1CN(C(C(COC)OC)=O)CC12CCC2 CCCC(C(=O)NCC(=O)NCC(N1CCC(NC(C)=O)C1)=O)N(C)C c1(-c2nc(NC(CN(C)CC3(C)CC3)=O)sn2)ccc(Br)cc1 c1(CC(=O)N(C2CCCN(C(=O)C(C)O)C2)CC)c(C)cnn1C.CCC(C)C Cc1cccc(C2(NC(C3CCC(c4ccccc4)C3)=O)CC2)c1C C1(NC(c2ccc(SC)cc2Cl)=O)CC12CCN(C(c1cnn(C)c1C)=O)CC2 CC(C)(CC(=O)N1CCCC(NC(=O)Cc2cnc(C3CC3)[nH]2)C1)C1CC1 C12CC1CN(C(c1ccccc1OC(F)(F)F)=O)C2.C(CC(=O)OC)C1(C)CC1 Cc1nc(C(=O)NC2(C3CCCN3C(C3CC(C#N)C3)=O)CC2)c2ccccn12 c1(OCCC)cccc(C(=O)NCC2CCC(NC(C3COC3)=O)CC2)c1 N1(C(C(=O)NCCC(=O)OCC)C2CC2c2ccco2)CCOC(CF)C1 CC1C(C(F)(F)F)CCN1C(=O)C=O.S(=O)(=O)(C(F)(F)F)NCCC.C Cc1cccc2c1CCOC2C(=O)N(C)CC1CCCN1C(c1cnc(O)o1)=O c1(C(=O)NC(C(C)NC(CCCCC=C)=O)C)cc(F)c(F)cc1Cl c1(C(C(=O)NCCCCC(C)NC(c2occ(C)c2C)=O)O)ccc(Cl)c(F)c1 c1(C(=O)NC(CN(C(C2ON=C(C(C)C)C2)=O)C)C)cc2oc(Br)cc2[nH]1 C1(C=O)CCOC(C)(C)C1.C(=O)(CNC(=O)C)NCCOC.CC.O N(C(=NCCC1OCCCC1(C)C)NC1CCN(C2CCCC2)C1)CCOCC Cc1cc(C(=O)NC(C2CCCN(Cc3ccc(O)cc3O)C2)C)cc(F)c1 CC1(C)C(=O)NCC1.c1(C(NCC(=O)N)=O)cc([N+](=O)[O-])c[nH]1.C1CC1 C1(C(C)C)(CNC(N(CCC#C)Cc2ccccc2)=O)CCN(C)CC1 C(=O)(C(C)C(C)C1CCCC1)NC(CNC(Cc1cnc(C)[nH]1)=O)(C)C c1(C(N(C(CC)CNC(=O)C(F)CC2CCCCC2)C)=O)cnc(O)n1CC c1(OC)ccc2c(c1)CC(C)CC2Nc1nc(C)ncc1F C12(NC(C(N3CCC(C)CC3)=O)=O)CCCC1N(C(C1(C)CCC(=O)NC1)=O)CC2 C1(CC)CN(C(=O)CN(C)Cc2ccccc2)CCC1NC(c1[nH]cnc1C)=O CC1(C)CCC(OC(C23CCC(CNC=O)(CC2)C3)=O)CO1.C(C)(C)C C1(COC)(NC(c2cnc(C)o2)=O)CCCN(C(c2ccc(Cl)[nH]2)=O)C1 c1(OC)cccc(C(=O)NC(C)C(C)NC(=O)CC2CNC(=O)C2)c1N N1(C(C2C(NC(C(CN(C)C)N(C)C)=O)CC2)=O)CCC(N=[N+]=[N-])CC1 C1(C(=O)NC2CN(C(C)C)C(=O)C2)CC2CCC(C1)N2C(=O)Cc1cnsc1 c1(C(=O)OC)nc(C(=O)N(C2CC(NC(=O)CC3CC=CC3)C2)C)co1 C12(C(N(C3CCCCC3)C)=O)CCCC1CN(C(c1cnc(C3CC3)o1)=O)C2 Cc1cc(C(=O)NC(C)(CNC(=O)CCCC2CCCC2)C2CC2)cc(O)n1 N1(C(CNCc2[nH]c(=NCC)sc2)=O)CC(CCC(=O)OC)Cc2ccccc21 C1(CCOC)(C(=O)NC)CCN(C(C2CC2[N+](=O)[O-])=O)CC1.C1C=CCOC1 CC1OC2(C)CC1(C(=O)NCC1CCCCN(C(c3ncc(Cl)cc3Cl)=O)C1)C2 CCS(=O)(=O)CC(=O)NC(C)CCC.n1(CC=O)nc(C2CC2)n(C)c1=O.N c1(OCC)cc(NC(C2CN(Cc3cccc(O)c3F)CCS2)=O)ccc1Br c1(C(N(CC(CC)NC(=O)CC(C)F)C)=O)ccc2cnc(C3CC3)n2c1C C(=O)(C1Cc2ccc(F)cc21)N.C1(NC(C2CC(N(C)C)C2)=O)CCCC(C)C1 CC1CN(C(c2ccc3ncc(Br)n3c2)=O)c2cccc(Br)c2O1 C(C1=CCN(C(C2(CF)COC2)=O)CC1)NC(C(C)Cc1ccccc1F)=O n1(CC(=O)NC2C3CN(C(Cn4c(C)cnc4)=O)C2C3)nc(O)ccc1=O C1(C(=O)NCCC(C)NC(c2csc(-c3ccoc3)n2)=O)(CC)CC1(F)F CC1(C)C(CC(=O)NOCc2ccncc2)CCN1C(=O)CC1CSC1 Cc1nc(C)c(C(=O)NCC(C)C2CC2)s1.c1(C=O)ccnc(C(C)(C)C)c1 C=CCCC(c1nnnn1CCCCCC)NCCNC(c1cccn1C)=O C(c1nccs1)=CC(=O)NC1CCCC1CNC(=O)C(O)Cc1ccccn1 CC1CCN(C(C2CC(C)(O)C2)=O)C1C(=O)NCC(C)(O)C1(C)CC1 c1(C(N(C2CN(C(c3cc(F)c(F)cc3N)=O)C2)C)=O)noc2c1CCCCC2 c1(C(=O)NC2CN(C(c3c(OC)nn(C)c3)=O)C3C2C3)ccc(=O)n(C)n1 CCCCCCCCCC(O)C(=O)NC1CC2CC(NC(c3nncs3)=O)CC12 CCCCCCCC(=O)NC1(CCO)CN(C(=O)CCN2CCNC(=O)C2)C1 C(=O)(C(O)CC(C)C)NCC1CC(OC)CN1C(=O)C(C1CCCC1)OC c1(C(N(CCN(C(C2CCOC2CN)=O)CC)CC)=O)nccc(O)c1 N1(C(CC(C(C)C)O)=O)CCC(=O)NC2CN(C(=O)CN=S(C)(C)=O)CCC12 c1(N(C)C(C2CN(C(=O)C(F)OC(F)(F)F)C2)=O)cnc2sccn2c1=O CC1CN(C(c2cn(C)nc2O)=O)CCC1CNC(=O)CC1CCC2(CC2)CO1 c1(C=O)sccc1OC(F)F.C(C(F)(F)F)NCC(=O)N.C1(CC)CCCC1 c1(OC)cccc(C(C)C(=O)N)c1.C1C=CCN(C(c2cc(C(N)=O)cs2)=O)C1 c1(C(N2C(C(=O)NCC3(C)CCCC3)COCC2)=O)ccc2c(Cl)ccnc2c1 C=CCC(F)(F)C(=O)NCCC1(CNC(c2ncn(C(C)C)n2)=O)CC1 C1(NC(CCCC)(C)c2nnnn2C2CCOCC2)CCCC(C)(C)C1 N1(Cc2c(OCCOC)nccc2)C2CCC(C(=O)O)C1CCC2OC c1(CC(=O)N(CCC)CCNC(c2nnc(CC)o2)=O)cccc2cnccc12 C=CC(F)(F)C(=O)NC1CCCCC1NC(c1cn(-c2ccccc2)nn1)=O C1(C)(C(=O)NC2CCN(C(c3ccc(CC)cc3F)=O)CC2)CCCCC1(F)F C(=O)(C(CC1CC1)OC)NCC1N(C(CC=C)=O)CC1 c1(CC)cncc(C(=O)NC2CC(CCNC(c3sccc3SC)=O)C2)c1 c1(C(=O)OCC)cc(Cl)ccc1Sc1ncc(N)c(C(C)C)n1 C1(C(N2CC(NC(c3ccn(CC)n3)=O)C(OC)C2)=O)CCC=CCCC1 S(=O)(=O)(c1c[nH]ccc1=NC1CC(c2ccccc2)C2CC12)N1CCC(OCC)C1 C1(O)(C(=O)NCCC(=C)C)CCCC(C)(C)C1.c1(C(=O)N)ccc2occc2c1 C(c1cccnc1C)=CC(=O)N.C(C(=O)NCCC1CCCC1)(C1CC1)OC Cc1cc(=N)[nH]cc1C(N1CCOCC(NC(=O)CC2CCC(=O)NC2)C1)=O N1(C(Cc2c(C)ccnc2)=O)CCC(NC(C2C=CCCC2)=O)C(O)C1 C(=O)(C(C)(C)Cc1cn(CCCNc2cc(Br)c[nH]2)nn1)OC c1(C(N(C(C)CNC(=O)CC2CCCC2)C)=O)cc[nH]c(=N)n1 CC(C)(CCC(=O)N1CCN(C(c2cc(Cl)ccc2Cl)=O)C2CCC12)[N+](=O)[O-] CCC(C)(C)C(O)C(=O)NC1CN(C(=O)CC=CC(C)(C)C)CCC1CO c1(C(N(C)CCc2ncon2)=O)cccc(CNC(=O)CCc2cncs2)n1 CCC(CCC(=O)NC1CC(=O)NC1=O)NC(c1ccc(OC)nc1)=O c1(C(=O)N)cccc2c1OCC2(C)C.C1(CNC(C(C)OCC)=O)CCCC1 c1(C=O)cc(Cl)cc(Cl)c1O.n1(CC)nncc1C(=O)NC12CC(C1)C2.C C1(C2CCCN(C(=O)CCCn3cc(-c4ccc(Cl)cc4Cl)nn3)C2)(OC)CC1 c1(C(N2CC(C)C(NC(C3(C#N)CC3)=O)CC2)=O)ccc2c(c1)COB2O c1cccc(S(C)=O)c1.C(CC(C(=O)N)NC(=O)OC(C)(C)C)OC(C)C c1(C(=O)NCC2(CNC(=O)C(O)C(F)F)CCCC2)cnc2ccoc2c1 Cc1cnc(C(=O)NC2C=CCN(C(=O)CCc3cncnc3)C2)cc1C C1CCCCN1C(=O)CC1NC(=O)NC1=O.c1(C(C)=O)cc(C(=O)NC)co1.C c1(C(N2CC(CCC)C2)=O)cc(C(F)F)cc(Cl)c1.C1(CC(=O)N)OCCC1C Cc1nc(CO)ncc1NC(=O)CCNC(=O)CN1CCCC1 N1(C(C2(CC)CCOC2)=O)CC2C(CC(=O)NCCCO)C2C1 N=S(=O)(CCNC(C1CCCC(F)(F)C1O)=O)c1cccc(Br)c1 C1(C(N(CCNC(C(CC)N(C)C)=O)C2CC2)=O)OC2CCC1CC2 c1(C(N(C(C)CN(C)C(c2cnc[nH]2)=O)C)=O)cc(F)c2c(c1)CCC2 c1(OC)ccc(OC)c(C(N2CC(NC(c3cncc(O)c3Cl)=O)CC2C)=O)n1 c1(C(N(CCC(C)NC(=O)CC(C)(C)C2CC2)C)=O)nn(C)cc1N N1(C(C(CC)N(CC)CC)=O)CC2(C1)CN(C(c1ccc(N)c(Cl)c1)=O)CCO2 c1(C(N(C(C)C)CCN2CSCCSC2)=O)ccc(C(=O)C2CC2)c(F)c1 c1(NCC(=O)OCC2CCN(C(C)(C)C)C2)cccc(C#N)c1 C#Cc1cnn(C)c1C(N1C2CCC1C(NC(C1C3C4CCC(C4)C13)=O)C2)=O N1(C(c2nn(C)c(C(C)(C)C)c2)=O)CCC(C2CN(C(=O)CC(F)F)C2)CC1 N1(CC(N2C(C(=O)O)CCC2CCC)=O)C(=O)SC(=Cc2ccc(F)cc2)C1=O N1(C(CC(CCC)C)=O)CC2CCCC2(C(=O)N(CC(C2CCCC2)O)C)C1 c1(C(N(CC(C)C)CC(=O)O)=O)ccn(C(F)(F)F)n1 O=C(CCC1=CCCCC1)N1CCCC1Cc1cn(CC2CCOC2)nn1 c1(OC(C(=O)NCC(CNC(CC2(C)CC2)=O)(C)O)C)ccc(F)cc1 C1(NC(=O)NC(CSCC=C)C(=O)O)CCC2CCC(=O)N12 Cc1nc(N2CCC2C=O)cc(C(F)(F)F)n1.c1cc(O)nc(OC(F)(F)F)n1.N C12(CNC(c3cnn(C)c3Cl)=O)CCC(CN(C(=O)C(O)C3CCC3)C1)C2 c1(C(N2CCC(NC(CCCCC#C)=O)C2C2CC2)=O)ccc(F)cc1C#N C1(NC(C(C)OC)=O)CCS(=O)(=O)C2(C1)CC(CN)C2.c1nccnc1C#N c1(C(=O)NC(C2CS(=O)(=O)C2)C)ccc2c(c1)ncn2C C1(CNC(=O)NCC2(CCOC)CCC2)CC2(C1)OCCO2 C1(OC)CCN(C(c2conc2C(C)NC(=O)C2=CC3C=CC2C3)=O)C12CCC2 Cn1cncc1C1CC1C(=O)NC1CC1NC(=O)CCOC1CCCC1 C1(C(N(CCF)CC)=O)CN(C(c2c(C)noc2C)=O)CC12CC2 CC1(C)CN(c2nnc(-c3ccccc3)o2)CC1NC(=O)CCC1CCCCO1 N1(C(c2cc(C(=O)OC)c(Cl)cc2)=O)CCc2ccc(C(=O)NCC#N)cc2C1 C1(C(=O)NC(c2nn[nH]n2)CC)(NC(C2CC(C)CO2)=O)CC(O)C1 c1(-c2cn(C3CC(S(C)(=O)=O)C3)nn2)csc2ccccc12 c1(C(N2CCC(CC=C)(NC(C3CCCOCC3)=O)C2)=O)ccc(OC)c(N)c1 c1(OC)nscc1NC(=O)C(C)N(C(=O)C=C(C)C(F)F)C(C)C C1(NC(c2ccn(COC)n2)=O)CC2CC(C1)N(C(c1nn(C)c(Cl)c1Cl)=O)C2 C1(CNC(c2c(CC)n(C)cc2)=O)CC(C(=O)NC(c2nccs2)C)=NO1 c1(C(N(CCN(C(=O)CC2CC3(CC3)CO2)C)C)=O)cccnc1Cl N1(C(c2n(C(CC)C)ncc2)=O)CCN(CC(C)(C)NC(=O)CC2CCC2)CC1 C1(N2C(CNC(N(CCC=C)CC)=O)CC2)CCS(=O)(=O)C1 C(=O)(C1=CC2(CN(C(C3(CCC)CC3)=O)C2)OC1)NC1CN(CCC)C(=O)C1 c1(CS(C)=O)cccc(C(=O)NC2CC2)c1.C12(C=O)CC(C)(CO1)C2.C Cc1cc(NC(c2ncccc2NCc2ccc(C(C)(C)C)nc2)=O)cnc1Br C(=O)(CC1COCc2ccccc21)NC(CCCC)CNC(C1(C)CC=CC1)=O c1(OC)ccc(CC(=O)NC(CNC(c2cccc(O)n2)=O)CO)nc1 C1(NC(CC(=O)NCC#C)=O)CCC(NC(c2ncc(CC)cn2)=O)CC1 N1(C(CC)=O)CCC(NC(c2ccn(CCNC(=O)Cc3cn[nH]c3)c2)=O)C1 c1(C(=O)NCC(C)(C2CC2)NC(=O)C(F)=CCCF)ccc2nncn2c1 c1(-c2ncc(C=O)s2)ccc(Cl)cc1.CC1CC(C(=O)NCCC2CCC2)C1.N N1(C(Cn2c(C)cc(C)n2)=O)CCC2C(CCCN2C(=O)Cc2ccsc2C)C1 c1(C(=O)NC(CC)CNC(c2ccc(Br)cc2)=O)cnc2ncnn2c1C c1(C(=O)OC)sc(CNCC2(C(C)(C)O)CC2)cc1N CCC(CC)CCC(=O)N1CC2(CCC2)CC1C(=O)NC1CN(CC)CC1(C)C N1(C(C2(C)CC(=C)C2)=O)CCOC(c2cn(CC3CCS(=O)(=O)C3)nn2)C1 C1(C(=O)NCc2n(CC)ncn2)CCCN1NC(=O)C(CN(C)C)N(C)C C(=O)(C(C(C)(C)C)NC(c1cccc(C#N)c1)=O)N(C(CC(C)C)C)C C1CN(C(=O)C=O)CC1C=O.c1cnns1.C(C)(C)C.C(=O)(NCC)O c1(COC)nccc(OC(C2C=CCN(C(=O)OC(C)(C)C)C2)=O)n1 N1(C(Cc2c(C)nc[nH]2)=O)CCC(N(C(=O)C=C2CCCCC2)C)C(C)C1 C1(C(N2CC(C(=O)OC)C2)=O)CC2CCC(C1)N2C(=O)CN(C)C Cc1cc(C(N2CC(NC(=O)COC3CCOCC3)CC(F)C2)=O)cc(F)c1 N(C1c2ccccc2CC1NC(=O)C(C)(C)O)C(c1ccc(CCC)s1)=O C1(NC(Cn2cc(CNC(C(C(C)C)F)=O)nn2)=O)CN(C)C2(CCC2)C1 c1(C(N2CC(NC(=O)CCC(F)(F)F)CC(C)C2)=O)cc2cccnc2nc1N C(=O)(NNc1cc(Cl)nc(Cl)c1)C1C(N)c2ccccc2C1 Cn1cnc(NC2(CNC(=O)CCSc3ccccc3)CCCCC2)cc1=O c1(NC)cncc(C(=O)NCC(C2CCCC2)NC(C2C3CCCCC23)=O)c1 C(=O)(CC(Cl)Cl)N(C1CCN(C(=O)CCc2cn[nH]c2)C1)CC#C c1(C(c2n(CCCCCC)nnn2)NC(COCC)C(C)C)ccc(Cl)cc1F c1(C(=O)NCCCCCNC(C(C2CC2)OC)=O)ccc(C(N)=O)nc1 n1(CC)cc(CCNC(=O)CCOCCOCC)cn1.C(=O)C1CC1 CC1Cc2cc(NC(C3CCN(Cc4cccc(O)c4)CC3)=O)ccc2O1 Cc1cc(-c2ncccc2C(=O)NC2CCC(F)(F)C2)cc(C)c1O C1(C(N2CCCCC(NC(Cc3c(C)cco3)=O)C2)=O)CCOCC12CCCC2 N1(C(CC(C)(F)F)=O)CC(C(=O)NC2CC3C=CC2C3)C(C)(C)C1 C#CC1CN(C(=O)C(C2CCOCC2)C)CCN1C(=O)Cc1cc(C2CC2)no1 Cc1cc(=O)ccn1CC(=O)NCCC(O)CNC(=O)C=Cc1cscn1 C1(C)(C(=O)NC2CN(C(C3CCC(CC)O3)=O)CC2(C)C)CCCCNC1=O c1(OC)ncc(C)cc1C(=O)NCC1COCCN1C(=O)CCOC(C)C CC(C)S(=O)(=O)c1ccc(NC(=O)NCc2cc(=O)cc[nH]2)cc1 C1CCOC(C)C1.c1(CC)ncoc1C(=O)NC(c1cnn(C)c1)C(=O)NC NC(=O)CCC(N)C(=O)N1CC2CN(S(=O)(=O)C(F)(F)F)CC12 C(=O)(C1CCc2c[nH]nc21)S(CC(C(=O)OC)C)(=O)=O.c12ccc(nc1)[nH]2 C(CC(C)(C)C(=O)N1CC2(C=CCO2)C1)NC(C1C(CC)CCC1)=O CCCCC(CNC(=O)Cc1ccc(Br)s1)NC(=O)CC1(O)CC1 C1(NC(C(F)=CC)=O)C2CC3CN(C(=O)CC=Cc4ccc(Br)cc4)C1C3C2 C1(C(N2CC(C(C)NC(=O)Cn3nccn3)C2)=O)COCC(C)(C)O1 c1(C(N2C(CC)CC(OC)C2)=O)ccc(O)cc1C.C(c1cscn1)=CC(=O)N c12cn(C)[nH]c-1nc(=O)[nH]2.c1(OCCCSC(C)C)cccc(F)c1 N1(C(=O)COC2CC2)CCOC2(CCN(C(=O)C(F)(F)C(F)(F)F)CC2)C1 CC(=O)CCN=C(NCC1(C)CCC(=O)N1)N1CCN(c2cccs2)C(=O)C1 C1(NC(CC(C)C)=O)CCCCC1CNC(c1cc(C2(C)COC2)no1)=O c1(C(=O)NCCN(C(c2coc(CC3CC3)n2)=O)CC)ccccc1 Cc1cc(C(N2CC3CC2(CNC(C2CC24CC(O)C4)=O)C3)=O)c(F)cc1F C1(C(=O)NC2(C(=O)NCc3c(C)nn(C)c3)CC2C)CC(C2CC2)=NO1 C1(NC(CCCOC)=O)CCC(C)N(C(C2CCOCC2)=O)C1 CCCC(CC(=O)NCCc1cnc(C)o1)NC(=O)C(C)(C)C1CC1 N1(C(C2(C=C)CCC2)=O)CC(C)CN(C(=O)Cc2cccc(C(F)F)c2)C(C)C1 CN1CCCC(CC(=O)NCCC2(C(=O)NC3(c4cccs4)CC3)CCC2)C1 c1(C(N(C(C)C)CCN(C(=O)C(C)C(C)O)C)=O)cc2ccccc2c(O)n1 CC1C(NC(=O)C(C)c2ccsc2)CCCN1C(=O)COc1ccccc1Cl C1(NC(=O)CSC2CC2)COCC1NC(=O)CC1CC=CCC1 c1(OC)nc(C(N2CCC(NC(=O)CC3(O)CCOC3)C2)=O)cc(O)n1 O=C1CCN(C(=O)CC2C=CS(=O)(=O)C2)c2ccc(Br)cc21 N1(C(C(C2CCC2)OC)=O)CC2CCCCC2(NC(c2cccc(C#N)c2)=O)C1 CC1=C(C(=O)NC2CC(NC(c3cnn(C(C)C)c3F)=O)C23CCC3)CCCO1 C12(CNC(Cc3n(C)cnc3)=O)CCCC1N(C(=O)CSc1nncs1)CCC2 N1(C(c2csc(C(C)(F)F)n2)C(=O)NCCCSC)CCCC12CC2 N#CCCCCCC(=O)NCc1ccsc1C(N1CC(n2ccnn2)C1)=O C1(CNC(C2C(C)C2C)=O)CC2COCC2N1C(c1ccn2ccnc2c1)=O Cc1cc(CN(C(c2cc(Br)c(Br)s2)C(=O)O)C)sc1Cl C=C=C(C)CC(=O)N(CCCNC(C1CCCCN1Cc1cccnc1)=O)C c1(C(=O)NC(C(=O)OC)C2CC2)cnc2cc(C3=CCCCC3)ccc2c1Cl N1(C(c2c[nH]c(=N)s2)=O)C2CCC1CN(C(c1ncc[nH]c1=O)=O)CC2 c1(C(N2CC(NC(Cn3c(C)c(Cl)cn3)=O)C3C2C3)=O)nc(O)nc(O)c1F Cc1cc(F)cnc1C(=O)NCCCC(C)NC(c1cccc(F)c1Br)=O c1(-c2nccc(CN(C(C(=O)NC)C)C)c2)ccc(O)c(OC)c1 C1(NC(C(CC)N(C(=O)C#CC2CC2)C)=O)CCCC(O)C1 CC(C)CC(CNC(=O)CCCCO)NC(=O)CC1CC(F)(F)C1 N1(C(C2CC(C)N2C(C2CCC3(CC3)C2)=O)=O)CC2C=CC1CC2 N1(C(c2c(C)ocn2)=O)CCCC(C2CCCN(c3nnc(C(F)F)o3)C2)C1 N1(C(COCC)=O)CCN(C(c2ccc(C3CC3)cc2)=O)C(CC#N)C1 c1(C=O)ccc(P(C)(C)=O)cn1.C1(NC(CCOCC)=O)CCC12CCC2.C N1(C(C(CCC)CC)=O)CC(C2CN(C(c3ccc(OC)cc3F)=O)C2)C1 Cc1[nH]c2ccnn2c(=O)c1CC(=O)OC1C=CS(=O)(=O)C1 Cc1noc(C(=O)NC2CCCC2CNC(=O)C(C)C)n1 C1(CC)CN(C(c2n[nH]cc2C2CCC2)=O)CCO1.CC(C(C)(C)C)=CC(=O)N C1(C=C)(C(=O)NC(C2CCOC2)C#C)CCN(C(c2c[nH]nc2Cl)=O)CC1 c1(C(=O)NCC(C(C)(C)C)=O)ccc2nc(Br)nn2c1 CC1(C(=O)NC2CC(O)CN(C(=O)CCCC3CC3)C2)CCC2CC2C1 C(=O)(C(CC(F)F)N(C)C(c1cnc(O)c(C)c1)=O)NCCC=CCCC n1(CC(=O)NC2CN(C(=O)C(C3(O)CCCC3)F)CC23CC3)cc(F)ccc1=O CC(C)(C)CCCC(=O)NC1CC2CCC1CC2NC(=O)Cc1ccc(O)cn1 C1CC2(C1)CS(=O)(=O)C2.N1(C(C(=Cc2ccco2)C)=O)CC(N(C)C)C(O)C1 c1(C(N2CCC(C(C)NC(c3ccnc(OC)n3)=O)C2)=O)cc(C)c(C)cc1Cl Cc1nn(C)c2[nH]c(=NC3CCCN(C(C4OCC4(C)C)=O)C3)c(C#N)cc12 c1(CNC(=O)Nc2ccc(-c3ccc(O)cc3)cc2)cc(F)c(O)c(F)c1 c1(NC(CC(C)NC(=O)OC(C)(C)C)=O)ccccc1C1CCOC1 C(=O)(C1Cc2c(Cl)cccc21)NC1(CNC(COCC#C)=O)CCOCC1 N1(C(c2c(C(=O)OC)scc2)=O)CCOC(C)C1.c1(C=O)csc(C(F)F)n1 c1(C(=O)OCC)c(NC(=O)C(=O)NC)sc(C)c1C.C12CCCC1CCC2 N1(C(CCCC)=O)CCC(O)(C2CCN(C(C3(OC)CCS(=O)(=O)C3)=O)CC2)C1 C12CC(CN1C(C1CC3C=CC1C3)=O)C2.N1(CCC=O)CCCC1=O.COC N1(C(CN(C(C(C)NC(CC)(C)C)=O)C(C)C)=O)CCOCC1CO CCC(CC(=O)N(CC(O)CNC(=O)CCNC(c1ccsc1)=O)C)C(C)C C1(NC(C=NOC)=O)CCC(C)(C)CC1CNC(c1ccnc2c1CCO2)=O C1CN(C(=O)CC2(O)CC2)CC(C)(C)O1.c1(OC)cc(F)ccc1C(=O)N C1(OC)CC(C)N(C(=O)CC2CC2(F)F)C1.c1(CC=O)c(C)noc1C.N c1(OC)ccc(CC(=O)NCCC(C(C)C)NC(c2c(CO)noc2C)=O)cc1F N1(C(CC2CC(C)C2)=O)CCCN(C(=O)Cc2cccc3nonc23)CC1C C1(C(CNC(CN(CC)CC)=O)C)CCN(C(=O)Cc2ccc(O)nc2)CC1 N1(Cc2cc(OC)ncc2)CCCC(C)(C(=O)NC(c2cccc(Br)c2)C)C1 N1(C(=O)NC2CC3CCC2CC3)CCCC1C1CCCc2ccccc21 N1(C(C(C)CN(C(=O)CC2CCOCC2)C)=O)CC(C#N)(C(N)=O)C1 CCC(C(=O)NC1CC2CCC(C1)N2C(=O)C(C)(C)CC#N)C(F)(F)F c1(C(C)C(N2CC(NC(=O)C=CCO)C(C(F)F)C2)=O)ccc(F)c(Cl)c1 N1(C(C2CCC(C(F)(F)F)CC2)C(=O)NCCCOC)CCCCC1C#N C1(CCCC)CN(C(=O)C=NOC)CCN1C(c1cccc(O)c1Cl)=O C1(NC(C(CC(F)F)N(C(c2cc(CC)n(C)n2)=O)C)=O)CCn2nccc2C1 C1(N(C2CCN(C3CC3)C2)C(c2cnn(C)c2)=O)CCC2(CC1)CNC2.CC.O c1(C(C)OC)nc(C(N2CC(O)(CCNC(=O)NCCCl)C2)=O)cs1 Cc1ccncc1CC(=O)NC1CCN(C(c2ccn(-c3cccnc3)n2)=O)C1 O=C(CCS(=O)(=O)Cc1cccs1)NC12CC(C1)C2.C1(F)(C=O)CC1.C c1(OCC)cnc(C(N2CCC(F)(CNC(C3CCOC3)=O)C2)=O)cn1.C N1(C(c2nc(CCC)oc2)=O)CC(CNC(c2csnn2)=O)OC(C)(C)C1 S(=O)(=O)(c1cnc(NCCC2CC=CCC2)c(Cl)c1)N1C(C(C)C)OCC1 CCC(C)(CCNC(=O)CC1CC1(C)C)NC(=O)Cc1coc(C)n1 C1(C(=O)NC(C2N(C(c3c(C)c(O)ccc3)=O)CCC2)C)CC2CCC1C21CC1 CCCC(O)CC(=O)NC1CCCCC1NC(=O)Cn1ccc(C)n1 C1(C2CC2)(CNC(c2[nH]nc(OC)c2Cl)=O)CCN(C(=O)CCC(F)F)C1 N1(C(C(=C(C)C2CC2)F)=O)CCCCC1CC.n1(C(C(=O)N)C)cnc(C#N)n1 n1(CC(=O)NC2CC(n3cc(-c4c(C)nccc4)nn3)C2)cc2ncccc2n1 CC(O)CCCCCC(=O)NC1CC(CNC(c2cnc3c(c2)COCC3)=O)C1 N1(C(c2cc(C)n(C)n2)=O)CCC(NC(c2cc(C(C)C)n(C)c2C)=O)C(C)C1 C(=O)(C1CCS(=O)(=O)c2ccccc21)N(CCCCNC(C(C=C=C)C)=O)C CC(C(=O)N1CCC(F)C(NC(=O)Cn2nnc(C(C)(C)C)n2)C1)C(F)(F)F C1(NC(c2ccc(F)cc2)=O)CCN(C(c2cnn(CC(F)(F)F)c2)=O)CC1O Cc1nc(CSc2nnc(CC)o2)nn1C.C(=O)N(C)C c1(C=O)ccc(F)c(O)c1.c1(C(=O)NC(c2ccccc2)C)cc(C)ccn1.N C1(CCNC(c2c(CC)occ2)=O)CCCCN1C(=O)CSC(F)(F)F N1(C(CCc2cc(C)on2)=O)CCN(C(C2CC(O)C2)=O)CC(C)(C)C1 c1(C(=O)NC2C(C)CCN(C(C3(C)CC(C)C3)=O)C2)cc(F)c(F)c(C#N)c1F N1(C(=O)NCc2ccc3cc[nH]c3n2)CCOc2ccc(F)cc21 N1(C(CC(C)c2ccco2)=O)CC(C)(C)CC1C(N1CC(O)(C(N)=O)C1)=O CCC(C(=O)N(C)CC1(O)CCN(C(=O)Cn2ccc(C)c2)CC1)C(F)(F)F c1(C(=O)NCCS(CC#C)(=O)=O)cccc2c(N)cccc12 N1(C(c2c(CNC(C(CCCC)O)=O)nnn2C)=O)CCC12CCC(C)CC2 C1(C(N2CC(N(CC(=O)OC)C)C2)=O)CCOCC1.C(=O)(CC1CCCO1)N N1(c2nc(C)cc(OC)n2)CC2CCC(C1)C2C(=O)NCCc1scnc1C C1(CNC(C2CC(=C)C2)=O)CCC2(CN(C(=O)CC3(C)CC3(F)F)C2)O1 C1(OC)CC(CNC(=O)CS)N(C(=O)C(C)n2ccnc2)C1.C(C)(C)C c1(CNC(C(N)=O)CO)cc(F)c(F)cc1Sc1ccccc1 N1(C(CCC)C)CC(C(=O)NCCNC(=O)Cn2cncn2)CC1=O N1(C(c2ccc(C)nc2C)=O)CCOCC(C)(CNC(C2(Br)CC2)=O)C1 C1(C(N2CCCC(NC(C3(CF)CC(F)(F)C3)=O)CC2)=O)CCCC12OCCO2 C1(CN(C)C)CCN(C(=O)CSCCNC(=O)COC2CCCC2)C1 C1(CC)CCCN(C(=O)CC2CCCC2O)C1C(N1CCC(CC(C)C)C1)=O N1(C(CC=CC=C)=O)CC2CN(C(=O)CCC34CCC(CC3)C4)CC2C1 C1(NC(C2N(C)C(=O)CC2)=O)COC2(CCN(C(C3CCC3)=O)CC2)C1 c1(C(=O)NC(C)C(C)(C)NC(=O)C=CS(C)=O)cccc(S(N)(=O)=O)c1 C(CN=c1[nH]nc(C2CC2)s1)C1CCC(NC(c2cccc(=S)n2O)=O)C1 C1(C(=O)NCc2nc(C(C)C)nn2-c2ccccc2F)(CSC)CCCCCC1 c1(CC(N2CCN(C(C(C=C=C)C)=O)CC2CC)=O)ccc2cnccc2c1 C(C(C)(C)CN(C(=O)C(C)c1ccsc1)C)NC(C1(SC)CC1)=O C1(CNC(C(=O)N(C2CC(OCC)C2)C)=O)CCCC1(C)C C1(C(=O)NCC2(N(C)C)CC2)COCCN1C(=O)COc1nn(C)cc1Br N1(C(c2c(CNC(C3Cc4nccn4C3)=O)c[nH]n2)=O)CC(O)(C2CC2)C1 C=CCCCCCCCCC(=O)NCC(C)CNC(C1(CO)CC1)=O c1(C(N2C(C)CC(NC(c3c(C)ccc(O)c3)=O)C2)=O)cnc2c(c1)COCC2 C(CCCC(C)NC(C1CCC1(C)C)=O)NC(C1(C)CC(=C)C1)=O c1(CC)cn2c(n1)CCC(C(=O)N(C)CCO)C2.C1(C)(C=O)CCCS1.CC c1(C(=O)NC23CC2CN(C(C2CC(F)C2)=O)C3)ccc(F)c2cccnc12 C(=O)(CC1=CCOCC1)N1CC(NC(C2CCN(C)CC2)=O)C(CC(C)(C)C)C1 c1(C(=O)N)ccc2nnc(O)n2c1.CC1=NOC(C(=O)NC2CC(F)(C)C2)C1 c1(CCC(=O)NCC2CC3CN(C(c4ccccc4)=O)CC23)ccc(Cl)cc1Cl C1(O)(C(=O)NC2CC(CCNC(CCC=CC)=O)C2)CCCC(C)(C)CC1 C1(C(=O)NC)CCN(N2CCCC(C(=O)NCCOC)C2)CC1 C1(CNC(C(C)NC(=O)CC2COCC2O)=O)C(C)(C)C1(C)C C1(C)(CC)CN(Cc2ccc(-c3ccccc3)c(Br)c2)CCO1 CC1CN(C(C2(S(C)(=O)=O)CCC2)=O)CC(C)N(C(=O)C=CC2CCOC2)C1 c1(OCC)ccc(NC(=O)CC2(NC(C3CCC(F)CC3)=O)CC2)cc1 c1(C(=O)NC2C(NC(C(Cn3ccc(C)n3)C)=O)C2)cc2nccnc2cc1C N1(C(C)C)CCN(C(C23CC(CO)(CN2C(c2csnn2)=O)C3)=O)CC1=O C1(NC(C(C=CC)O)=O)CCN(C(=O)COc2cccc(Br)c2)CC1(C)C N1(c2nc(C)cc(C)n2)CCC2(CCN(C(=O)C(C)NC=O)C2)CC1 C1(C(=O)N)CCS(=O)(=O)C1.C(C(C)(C)C)N(C(CCN(C)CC)=O)CC O=C(Cc1cc(C(F)F)cc(F)c1)N=c1cc(C2CCCCN2C(=O)CO)[nH][nH]1 C(=O)(C(O)CCSC)NC1CC(N(C(C2(CC=C)CC2)=O)C)C1 Cc1nnc2sc(C(N3CCC4OC(=O)OC4C3)=O)c(N)c2c1C CC(CC(F)F)C(=O)NC1CC12CC(NC(C1(C(C)(C)C)CCCCC1)=O)C2 N1(C(c2ccc(CC)o2)=O)CCc2sc(CNC(=O)CCNC=O)nc2C1 c1(C(N2C(C)CN(C(C3(C)CC4(CCC4)C3)=O)CC2)=O)ccc(S(N)(=O)=O)s1 Cc1cccc2c(C(=O)NCC3CCN(C(C4CC=CC4)=O)C3(C)C)coc12 CCC(CN(C(=O)CN1CCCC1)CC)NC(C1(C2CCCO2)CC1)=O Cc1cccc(C)c1CC(N1CCC(NC(=O)C(F)(F)C2CC2)C1)=O C1(C(=O)NCC2CCC2)C2CN(C(=O)CC3CC3)CC12 c1(C(N2CCC(C3OCCO3)C2)C(=O)NC(CC)C)cnn(C2CCCC2)c1 C1(NC(CC(C)CF)=O)CC2(CCN(C(=O)C(c3ccc(F)cc3F)=O)C2)C1 N1(C(C2C(NC(CN(C)C)=O)COCC2)=O)CC2CCCC(C2)C1 C12(NC(C3(C)CC4CC4C3)=O)CCC(CN(C(=O)CCc3ccccc3Cl)C1)C2 c1(NC(C2(C)CCN(C(c3c(CCC)nco3)=O)C2)=O)cccc(O)c1F C#Cc1cccc(C(=O)NCCN(C(=O)C(C)C2CCOC2)CC)c1 C1(C(=O)NCC(CNC(=O)CC2(C)CCC2)OC)CN2CCCC1C2 CCC(C)C(C)C(=O)NCCCN(CCCNC(c1csc(Cl)c1)=O)C C1(CC)CN(C(c2cn(CCO)nn2)=O)CCC1NC(C1(C)CCNC(=O)C1)=O C1CCN(C(c2cnn(C)c2C(F)F)=O)C(C)C1.c1(OC)cccnc1C(=O)N C1(C(N2CCCC(N(C(C(CCC)O)=O)CC)C2)=O)CCc2cnn(CC)c2C1 C1(C)(CC(=O)NCCCN(C(=O)CCC)C(C)C)CC1(Cl)Cl.C1CCOCC1 CC(CC(=O)NOC1CCC(O)C1O)N(C)C(c1sccc1F)=O CC=C=CCCN=c1[nH]c(N(C)CCc2cccc(C#N)c2)nc2c1CCCC2 c1(C(N(CC(C)N(C)C(C2CCS(=O)(=O)C2)=O)C)=O)cc(Br)cnc1N c1(C(=O)NC(C(C)C)CNC(C2CCCSC2)=O)cc2c(ccn2C)[nH]1 N1(Cc2c(OC)nsc2)CCC2(CCCN(C(=O)C(C)(C)C(F)(F)F)C2)C1 c1(CC)nc(C)c(C(N2CCOC(CCCNC(C3SCCS3)=O)C2)=O)o1 N1(C(CC(COC)(C)C)=O)CCOC2(CCC(NC(=O)CC3CCC3)CC2)C1 c1(C(=O)NC(CNC(c2cc(-c3ccc(C)s3)[nH]n2)=O)C)n[nH]c(C)c1[N+](=O)[O-] C1(C(N(CC(O)CNC(=O)Cn2cnnn2)C)=O)CCCC12CC2 N1(C(CCCNC(C)=O)=O)CCCOC(CNC(=O)Cc2cnccc2C)C1 c1(OC)cncc(CNC(=O)NCc2cnn(CCO)c2)c1 c1(C(=O)NCC(C)N(C(=O)CC(C)C(C)C)CC)ccc2c(c1)COC2 c1(OC)nc(C)ccc1C(=O)NC1CC(C)N(C(C2CC3CC3C2)=O)C1 c1(C(N2CCCC(NC(C=NOC)=O)C2C)=O)coc2cc(C)ccc12 N1(C(C=C(C)C2CC2)=O)C2CCC1C(NC(=O)CC=CC(C)(C)C)C2 Cc1ccc2c(c1)CC(C(N1CC(C)(C)CC1)=O)S2.C(C=C(Cl)Cl)=CC=O.C C1(CNC(CN(C(C)C)C)=O)CCC(C)CN1C(=O)COCC(C)(C)C C1(C(N(C)CC2CN(C(C(C)OCCCC)=O)C2)=O)CC(c2cccnc2)=NO1 N1(C(c2nc(CNC(c3cc(C)c(O)cc3)=O)oc2)=O)CC(=O)NC2(CC2)C1 C1(NC(CC(C)(C)OC)=O)CCN(C(C2(C(C)(F)F)CC2)=O)CCC1CO C12(C(N(CCNC(Cc3cc(C)nc(O)c3)=O)C)=O)CCCCC1C2(F)F c1(C(N2CCCC(Nc3cc(COC)ncn3)C2)=O)ccn2ccccc12 Cc1c(C2(CNC(C3(C(F)F)CC4(CC4)C3)=O)CC2)cccc1F C(C(C(C)C(C)C)NC(c1ccc(N(C)C)c(F)c1)=O)NC(CC=C=C)=O CCCC(C(O)C(=O)N1CCC1CF)NC(=O)C(O)CC(N)=O C(=O)(CC(F)(F)C(F)F)N1CC(NC(C2(c3cn(C)nc3)CCCO2)=O)C1 C1(NC(C(CC)O)=O)COC2(CCN(Cc3cc(Cl)ccc3F)CC2)C1 C1(CNC(Cc2n(C)cnn2)=O)COCCN(C(c2c(F)cncc2Cl)=O)C1 C=CC(C)(CCOC)C(=O)NC(CC(=O)N(C)CCC)C(C)C CC1(C)CCCC(c2cn(C(c3cc(Cl)sc3Cl)CCc3ccsc3)nn2)C1 C1(COC)(OC)CCN(C(C2(NC(=O)Cc3ncccc3F)CC2C)=O)C1 c1(COCC)nc(N(CC(C)NC(c2c(C)nn(C)c2C)=O)C)cc(C)n1 Cc1nc(CNC(C2CCO2)=O)oc1C(=O)NC(C12CCC(CO1)C2)C c1(C(=O)NCC(CC=C)NC(c2ccc(Cl)c(C)c2)=O)ccc(N)c(N)n1 C1(NC(CC(n2ccc(C)n2)C)=O)CCCC(N=c2nn[nH]n2C)C1 C(=O)(C1=C(CC)N(C)C(=O)N(C)C1c1ccc2c(c1F)CCCN2)OC CN1CC(O)CC1(C)C(=O)NC1C=CCN(C(=O)C2=CCOCC2)C1 C1(NC(c2c(CC)oc(C)c2)=O)CCCN(C(c2c(C)[nH]c(C)c2C)=O)CC1F C1(NC(C2NC(=O)OC2)=O)CC2(C1)CN(C(c1n[nH]c(C3CC3)c1Br)=O)C2 c1(OC)cc(Br)c(CNC(=S)NNC(=O)CC#N)cc1OC c1(N(C2CCN(C(C3OC(C)CC3C)=O)CC2)CCOC)ncnc2scnc12 C1(CCCNC(CCN(CC=C)C(C2CCOC2C(C)C)=O)=O)CCCC1O O=C(N=c1[nH][nH]c2cc(Cl)ccc12)C1CC(F)(F)CN1Cc1cc(O)cc(F)c1 C1(C)(C(=O)N)Cc2cc(Cl)ccc2C(=O)O1.Cc1nc(C(=O)NC2CCC2)co1 C1(CC(=O)N(C(C)CNC(c2cccnc2C)=O)CC)COc2ccccc2O1 C(C1CCOCC1)=CC(=O)NC(CC)CNC(=O)C=CC(C)CC Cc1nc2c(C(N3CCN(C(c4c(C)ccnc4O)=O)CC3)=O)ccnc2[nH]1 N1(C(c2ccn(C3CC3)c2)C(=O)NCCCSCC)CCOC2C(O)CC12 Cc1ocnc1C(=O)NCC1(CN(C(=O)C(C)(C)c2cccnc2)C)CC1 C1(CC(=O)N(c2cnc(C)nc2)CCN2CCOCC2)CN(C=O)CCO1 C(C)(CC(=O)NC(C(=O)N1CC(N2CC(F)C2)C1)C1(C)CC1)SC C1(NC(CC(CNC(C2OC3CCC2C3)=O)OC)=O)CCCCN(C)C1=O c1(CC)cc(C(N2CCC(C(O)CO)CC2)C(=O)NC2CCC2)cc(F)c1 C1(CNC(c2cc(C(=O)OC)on2)=O)CCCN(C(C2(F)CCCCC2)=O)C1 CCC(CC(=O)N1CC2CC1C2NC(C1(OC)CCCC1)=O)OC C(c1ccco1)=C(C)CNCCCC(C)NC(=O)CCOC(=O)CO CC(CCCCNC(=O)CCC(=O)c1ccc[nH]1)NC(C1CCNC(=O)C1)=O C1(C(C)NC(COCCSC)=O)CCCCN1C(c1cnn(C2CC2)c1C)=O C1(C2CC2)(CNC(=O)CCc2cn[nH]c2)CCN(C(=O)C2=NOCC2)C1 c1(C(N2CCN(C(=O)Cc3ccco3)CC(O)C2)=O)cc2n(n1)CC1(CC1)C2 c1c(C(=O)N(CC(O)C)C)cnn1C(C)(C)C.C1(C=O)CCC(=O)N1C.CC C(=O)(C1=CC2CC(C1)CC2O)N1CC(CCNC(CN(C)C(N)=O)=O)OCCC1 C=CCC(C)(C)CCNC(=O)CC1(C=C)CN(C(=O)CCCC)C1 C1CCC2CN(C(=O)Cc3cnc(C4CC4)[nH]3)CC12.Cc1csnc1C(=O)NC c1(C(=O)NC2CCN(C(CNC(C)=O)=O)CC2CO)nccc2nn[nH]c12 C1(C(=O)NCc2cc(C)ns2)CCCN1NC(=O)C1(C)CCCCO1 C1(NC(CCc2cnc(C)s2)=O)CN(C(c2csnn2)=O)CC(F)(F)C1 C(C)(C(C(=O)NOCCC1CC1)C(C)C)NC(CCC)=O N1(C(C(C)SCC)=O)CCN(C(C2(CCOC)CCN(C)CC2)=O)CC12CC2 CCC(C(=O)NC1CC2CCC1CN2C(=O)COCC1CCCC1)C(F)(F)F Cc1[nH]c2ncnc(NCC3(O)CCCN(C(C4CC4(Cl)Cl)=O)C3)c2c1C N1(C2CN(C(=O)CN3CCCC3COc3ncccn3)C2)CCC(NO)CC1 C1(NC(=O)NCC2(F)CN(C(C)=O)C2)CCCC(c2ccccc2)C1 C(=O)(C(F)(F)C(F)(F)F)N1CCCCCC1.c1(NC(C)=O)nc(C(=O)N)cs1 CC(C)CC(CN=c1[nH]c(=NCCC(F)F)[nH]c2c1COC2)OC(C)(C)C C1(F)(CNC(C(=O)N(C)C)=O)CCN(C(c2cnco2)=O)CC1 c1(C(N2CCN(C(C3C(C)(C)C3)=O)CC2C(F)F)=O)ccnc2ccc(F)cc12 N1(C(C23CCC2C3)=O)CCCCC1Cc1cn(CCCO)nn1 N1(C(C(=O)N(CC(C)Nc2ccccc2)C)=O)CCSC2CCCC12 N1(C(C)C)CC(CNC(=O)N)CC1=O.C1CN(C=O)CCO1.C(C)(C)C.C Cc1cc(NC(C2CCN(CC(F)F)CC2)=O)ccc1C(C)C C1(CNC(C2C(C(C)C)C2)=O)CC2(CCN(C(c3cc(Cl)no3)=O)CC2)CO1 O=S(=O)(c1ccc(NCCC(O)C2CC2)c(Br)c1)NC1COc2cccc(F)c21 N1(CCN2CCC(c3cccc(C(=O)O)c3)C2)CCC2NCCC12.c1ccncc1 C1(NC(CCC2CCCN(C(CS(=O)(=O)NC)=O)C2)=O)CC(C)N(C)CC1C c1(C(=O)NCC=CCNC(c2ccc(C(C)=O)cc2)=O)cc(Cl)nnc1O c1(C(=O)NCC(C)CN(C)C(c2ccc(O)cc2O)=O)csc2cncn12 CCC(N=c1[nH]c(=NC(C)c2ncn(C)n2)[nH]c2cc[nH]c12)C1CCC1 N1(C(CC(=O)NCC)=O)CC(NC(c2ccc(Cn3cccn3)o2)=O)CC1C c1(C(=O)NC2CCC(NC(c3ccc(CF)cc3)=O)C2)ccn2ccsc12 Cc1[nH]nc2ncc(C(=O)NCC(C(C)C)NC(C3CC4(C3)CC4(F)F)=O)cc12 N1(C(=O)C(O)CC2CCCC2)CC2(CC(NC(C34CCCC3C4(F)F)=O)CO2)C1 c1(C(N2C(CNC(c3[nH]nnc3C3CC3)=O)COCC2)=O)cc(O)ccc1Cl c1(OC)cc(O)cc(CCC(=O)NC2CC2CNC(c2cncnc2C)=O)c1 Cc1ccc(CN(C(=O)NC)Cc2cccs2)s1.c1nc(-c2cccs2)no1.C C(=O)(C(C)(CNC(C1CCC2(CC2)C1)=O)CC)N(CCC(N)=O)CC N1(C(c2ncccc2O)=O)CC2CC(NC(C3CC(C(F)F)C3)=O)C(C2)C1 c1(OC)cc(C(=O)NC2CCCC(NC(c3cscc3C)=O)CC2)cc(F)c1 CCC(C)(O)C(=O)NCCC1(O)CCN(C(=O)CCC(=O)c2cccs2)C1 C1(C(N2CCCC(NC(c3ncc(NC)nc3)=O)CC2)=O)CCc2nn[nH]c2C1 C(=O)(C(CCC1CC1)NC(C1CC1Cl)=O)NC(CC)C(C)C C1(CCC=C)CCCN(C(=O)COC(C)(C)C)C1.c1(C(C=O)C)ccnn1C.N c1(C(C(N2CC(CNC(C=C(CC)C)=O)OCC2)=O)C)c(F)cccc1F Cc1ccsc1C(=O)NCC(C)(O)CNC(=O)C(C)Cn1ccnc1 c1(N(C)C)cc(C(=O)NC2CCCC2NC(C2(C)CC(C#N)C2)=O)ccn1 CCCCCCC(CNC(=O)C(=O)NC1CNCCOC1)CC Cc1cccc(-c2cn(CCCC(=O)N3CC(N4CCC4)C3)nn2)c1C C1(NC(C2(C#C)CN(C(c3cccc(F)c3O)=O)C2)=O)C2CCC3C(C2)CC13 c1(C(N2CC(CCCCNC(C(n3cc(Cl)cn3)C)=O)C2)=O)cc(O)nn1C N1(C(C)C)CCCC(CC(=O)NCC2CCCC2NC(=O)CC2CCOCC2)C1 C(=O)(CCCCC(F)F)N1C(CNC(C(C(C)C)(C)O)=O)CN(C)CC1 C(=O)(N1CCCc2nncn21)C1C(F)(C(=O)OCC)C1 CCC(CC(F)(F)F)CS(=O)(=O)Nc1cc(Br)cnc1O C(=O)(C1CCCc2nc[nH]c21)NCC(CC)NC(=O)C(F)CC1CCCCC1 C12(C=O)CC3CC(C(=O)N1)C2C3.n1(COC)ccc(C=O)n1.C(C)C(C)C.N C1(CNC(C(c2c(C)cccc2)(C)C)=O)CCN(C(C2SCCCS2)=O)C1(C)C N1(C(=O)C2=CCOC2)CCC(F)(CNC(C2(Br)CC2(F)F)=O)CC1 c1(C(N2CCC(NC(c3cnc(C)nc3)=O)C2)=O)cc(S(N)(=O)=O)co1 C(=O)(CC1CCc2ccccc21)NC1(CO)CCCN(C(C=CSC)=O)C1 C1(NC(c2nnc(C)s2)=O)CC2(C1)CN(C(C1CCC(O)C1)=O)C2 C(C1=CCN(C(c2occc2C(=O)NC)=O)CC1)NC(CC1CCC(CC)O1)=O C(=O)(CCC(CC)CCCC)NCC1N(C(C(C=C)O)=O)CCCC1 C(=O)(C1=CCC2(COC2)OC1)N(C)CCOCCNC(C1CCCCC1F)=O c1(CCC)ncc(C(C(=O)NCCCSC)N(C)C(C2CCOCC2)C)s1 C#CCC(CC(F)F)C(=O)NCC1OCCC1C(N1CC(C(C)OC)C1)=O Cc1cc(C)n(C(C)C(=O)NC2(CN(C(=O)CCC(N)=O)C)CC2)n1 C1(NC(C2CCC(CNC(Cc3ccc(C)s3)=O)O2)=O)CC2CC1C(O)C2O c1(C(N(CCCn2cc(C(CC)OC)nn2)C2CC2)=O)cc2ccc(Br)nc2[nH]1 c1(OC(F)(F)F)cccc2c(N3CCCC4CC34)nc(Cl)nc12 c1(C(N2CCCC(C)C2)=O)coc(S(C)(=O)=O)c1.c1(C2C(C=O)C2)ccsc1.N Cc1cc(C(N2CC(N(C(=O)CCN3CCCS3(=O)=O)C)C2)=O)cn(C)c1=O CCCC(CCCNC(=O)CC(O)CN(C)C)NC(=O)Cn1c(C)csc1=O N1(C(CCCC)=O)CC(CNC(C2(C(=O)OCC)CCO2)=O)C(C)C1 Cc1nc2c(N3CC4C(NC(c5ccc(C)n5C)=O)C4C3)ncnc2s1 CC1(F)CN(C(=O)COc2ccccc2Cl)CC1(C)Br c1(C(F)(F)F)cccc(C2CN(Cc3cnn(C4CC4(F)F)c3)CCO2)c1 C1(CSCC(COC)C)CC(C)(C)C(=O)O1 C1(C=O)CCCCCN1C.C1(C(=O)NCC(=O)OC(C)C)CC2(CC2)C1.C N1(C(Cc2c(C)ncs2)=O)CC(NC(=O)CC2(C)CCOC2)CC12CCC2 N1(C(C2CC(=O)NC2)=O)CC2OCCN(C(c3cc[nH]c4nccc3-4)=O)C2C1 c1(C(N(CCOC)CCNC(=O)C(C)(C)SC)=O)cc(Br)nn1C O=C(O)C1CN(S(=O)(=O)Cc2cccc(Cl)c2Br)c2ccc(Br)cc21 N1(C(=O)CCc2ccoc2)CC(C(N2CC(F)C(F)C2)=O)CC(F)(F)C1 C1(NC(c2c(C)ccs2)=O)CN(C(=O)CCc2ccc(O)nc2)CC2(CCC2)C1 C1(NC(c2c(C(C)=O)cccc2)=O)COCCN(C(c2nccc(C)c2F)=O)C1 N1(C(C(C)N2CCC2)=O)CC(NC(c2cnn3c2CCC3)=O)CC12CCC2 N1(C(CC(C)C)=O)CCCC1C1CCCN1C(c1ccc(=NCC2CC2)[nH]c1)=O c1(C(N(CCNC(C(C)Cc2ccccc2)=O)C)=O)ncccc1Br O=C(C1=Cc2ccccc2OC1C(F)(F)F)N1CCCC(C2COC2)C1 C1(OC)COCCN(C(C2CN(C(=O)C(C)C3CC3)CC2OC)=O)C1 C1(NC(C2C(C=C)OCC2)=O)CC2CC(NC(c3ccnn3CC#N)=O)CC2C1 Cc1oc(CO)cc1C(N1CCC(C)C1CNC(=O)Cn1ccc(Br)n1)=O C1(C(=O)OCc2cnc(-c3ccc(Cl)s3)s2)CCCC(C(F)(F)F)C1 C(=O)(CCCCC(F)F)NCC(C)CN(C)C(c1cc2n(n1)CC(F)C2)=O c1(-c2ccc(CC)o2)ccc(NC(C2(C)CCCC2N)=O)cc1 N1(C(C(C#N)C2CC2)=O)CCCCC(CNC(=O)C=Cc2cscn2)CC1 Cn1cc(C=O)c(C2CC2)n1.c1(C(N2C(C3CC3)CCC2)=O)cc(C#N)c[nH]1.N C1(NC(c2c(C)[nH]cc2)=O)(CO)CCCN(C(=O)CC(C)C(F)F)C1 N1(C(c2c(C)nc(C)s2)=O)CCN(C(=O)C(C)C(F)F)C(C(C)C)C1 CCC(CC(=O)NCC1(C2(O)CN(C(=O)Cc3cnnn3C)C2)CC1)CC(C)C C1(C=O)COC2(C1)CN(C(C1(C(C)(C)O)CC1)=O)C2.C(CCC)SCC.N C=CCC(F)(F)C(=O)N1CC(NC(C2CC2c2ccc(F)nc2)=O)C(C)C1 N1(C(C(C(C)C)O)=O)CCC2(CCC(NC(c3cc(C(N)=O)co3)=O)C2)CC1 N1(C(c2c(C)nc(C)o2)=O)CCC(C(=O)NCC2(C)CCC2)C1(C)C N1(C(c2cnc(C(C)O)s2)=O)CCC(F)(CNC(=O)CCC(=O)N(C)C)C1 N1(C(Cc2c(C)ccs2)=O)CCC(CCNC(=O)C=Cc2ncc[nH]2)CC1C C(C(C(C)C)N(C)Cc1nncn1C)(OC)OC c1c(C)cc(C)cc1C.C(=O)(CCNC(=O)N)NC1CC(C(=O)OC)C1 CCC(C)(C)C(C)NC(c1cnc(N2CCN(C)CC2)nc1)c1nnnn1C N1(C(COCCN(C)C)=O)CCCC2(NC(=O)CC3=CCOCC3)CCCC12 C1(CNC(CC(C)CN(C)C)=O)CN(C)CCN1C(=O)Cc1cccc(Cl)c1 c1(C(N2CC(COC)C2)=O)cccc(F)c1.C(c1ccc(Cl)s1)=CC=O.N n1(CC)cc(C(N2CC(C)C2)=O)c(C(C)C)n1.C(=O)C(F)Cc1ccccc1 Cc1nc(C)c(C(N2CCCC(CCNC(=O)CSC(F)(F)F)C2)=O)o1 Cc1cc(CN(C)C(C2(NC(=O)Cc3cccnc3)CC2C)=O)no1 Cc1c(C(=O)NC2(C)CC2)sc2[nH]cnc(=O)c12.C1(CCC=O)CCC(C)O1 N(C1CCCc2c[nH]nc21)C(CNC(c1c(Cl)cccc1[N+](=O)[O-])=O)=O C(N=c1[nH]cnc(C)c1C#N)C1CCC(CNC(CCC(=O)NCCC)=O)CC1 CC1CCCN(C(=O)C=Cc2ccncc2)C1CNC(c1n[nH]c(=N)[nH]1)=O N1(C(C2(C)C=CCC2)=O)CCCC(C)(CNC(=O)Cc2ccc(Cl)s2)C1 CCC(C)CC(=O)C(=O)N1CCCC(F)(CNC(=O)CC(C)c2ccco2)C1 N1(C(C2(C)CC2(F)F)=O)CCN(CC2(NC(C3CCCCC3)=O)CC2)CC1.C N12CCCC(C1)C2=O.N1(C)CCC(F)C1.C1(N(C(C)=O)CC)CC1C=O C1(C)(C(N(C)CC2CCN(C(CCOC)=O)CC2)=O)CCCCNC1=O N1(C(Cc2n(C)c(S)nn2)=O)CC2CC3CC2C1C3NC(C1CC=CCC1)=O c1(C(=O)NC(C(CO)NC(C2CC(C)N(C)C2)=O)C)cc2sccc2n1C N1(C(C)=O)CC(C)CN(C(=O)Cn2nnc(=N)[nH]2)CC1C.C(C=O)NC(C)=O.N n1(CCC)cc(C(=O)NCCC2CCCCC2)cn1.C1(CC=O)CCC(C)O1.N c1(OC)cc(F)c(F)cc1C(=O)NC(C)C.C1(C)(C(=O)N)CCC12CCC2 O=C(C1=CC2C=CC(C1)C2)NCc1ccc(C)cc1.c1nccs1.C(=O)C.N C1(CCC(=O)OCC)CCCN(N2CC(C)CCC2c2cccnc2)C1 N1(C(C=CC(CC)C)=O)CC=C(C(=O)NCC(O)CC(C)(C)C)C1 Cc1cc(CCNC(=O)C(N2CCC(Oc3ccccc3)C2)=O)on1 N1(C(C(C)C(F)F)=O)CC(NC(c2cnn3c2CCC3)=O)C2(CCC2)C1 C=CCC(CC=C)C(=O)NC1CCN(C(c2c(Cl)ccnc2C)=O)CC1CC Cc1cc(NC(C2OCCC2C(C)C)=O)ccc1NC(=O)CCc1ncco1 C1(C(=O)NC2C=CCN(C(=O)CC3C=CCCC3)C2)Cc2nccnc2C1 C1(CCC)CN(C(=O)C(C)(C)SC)CC1C(N1CC(OC)CC1CO)=O C1(CC=O)CN(C(=O)C(O)C2CCC2)CCN1C(c1cnc(C2CC2)[nH]1)=O.C N1(C(=O)NCc2c(C)c(Cl)ccn2)CCC(N=c2cc[nH]cc2Cl)CC1 O=C(C1Cc2ccc(Cl)cc21)NCCCC1CCCN1C(c1ccc(CO)o1)=O C(=O)(C(C)(C)C(C)(F)F)N1C(CNC(c2cnc(C(C)(C)C)nc2)=O)CC1 C1(C)(C(=O)N)CS(=O)(=O)C1.C1(CC)OCCC1C(=O)NC1CC1C C1(C(=O)NC(c2n(C)cnn2)CO)COC2(C1)CN(C(=O)C(C)(C)Cl)C2 c1(C(C(=O)NC2(CNC(C3CCCSC3)=O)CCCC2)O)ccc(Cl)cc1Cl C1(C=O)C2CC(CN(C(=O)C=C3CCC3)C2)N1C(C1CC1(F)Cl)=O.CC N1(C(C(C=CC)O)=O)C2CCC1CC(CNC(c1ncc(Br)cc1O)=O)C2 c1(C(=O)NC2CCN(C(c3c(OC)c[nH]n3)=O)CC2F)ccc(C)c(Cl)c1F C1(CC)CCN(C(C2CCCN(C(C)C)C2)=O)CC1.C1(C=O)CC(=O)N(C)C1.N CC1CCN(CC(=O)OCC(c2csnn2)=O)CC1C N12CCC(CC1)CC2.c1(OCC(=O)NCC=O)cccc(F)n1.c1cccs1.N N1(C(CCOCCOC)=O)CCC(NC(c2ccnc(O)c2)=O)C1(C)C CCCCN(C)N1CCN(c2n[nH]c(C)c2Cl)CC1 N1(C(Cc2cc(C)[nH]n2)=O)CC(NC(c2cccc(C(C)C)c2)=O)CC(C)C1 Cc1ccc(CCC(N2CC(CCNC(=O)CN(C)C)OC(C)C2)=O)cc1C CC1N(C(=O)C=CCNC(=O)CC2CCCC3CC23)CCOC1(C)C c1(NC(C(N2C(C#C)(C)CCC2)=O)=O)ccc(C(=O)OC)c(F)c1C CCC(CCC(=O)NCC(O)CC(F)(F)F)NC(=O)C(O)C(C)(C)C C1(C(=O)NCCCN(C)C)(NC(c2c(C)ccs2)=O)CCOCC1 C1(C(=O)NC2CC(C)OC2=O)CN(C(C2(C)CC2(C)C)=O)CC1C1CC1 C(=O)(C(CS(C)(=O)=O)NC(=O)CCCCNC)OCC C(=O)(CC1CCc2ccccc21)N1C(CNC(=O)CCOC2CC2)CCCCC1 CCCC(C)CC(=O)NCCC1(NC(=O)C(C)Cc2ccc(OC)cc2)CC1 N1(C(c2ccc(CC#N)cc2)=O)CCCC2(CCCN(C(=O)CC3CCC3)C2)C1 C1(CNC(c2noc(CC)c2C)=O)CCN(C(C2CC2F)=O)C1(C)C C1(NC(CCOC)=O)CCOC12CCN(C(c1c(S(C)(=O)=O)cnn1C)=O)CC2 c1(C(c2nnnn2C2CCCC2)Nn2cc(CCCC)nn2)ccc(OC)cc1 c1(C(=O)NCC2CN(C(CCCSC)=O)CC23CC3)cc2cccnc2[nH]1 c1(NC(C(C)OC)C(=O)O)cc(C#N)ccc1[N+](=O)[O-] NC(=O)CCCC(=O)NCCNC(C1CC1)=O.N1(C(C2CC2)=O)CCCC1 N1(C(C2C(c3n(C)ncc3)C2)=O)CC(C)CC(C)(C)C1.C(=O)(C)N.C1CC1 N1(C(C2CSCCN2C(c2cc(O)ccc2O)=O)=O)CCc2c(F)cccc2C1 C(=O)(C(O)CC(C)C)NCC(CNC(c1c(CC)nc(C)s1)=O)CO C1(CC)CC(C(=O)NC2CCCC2(F)F)CCN1C(C1C2CCC(F)C12)=O CC1C=C(C(=O)NCCCCC2CCN(C(=O)CCOCC(F)F)CC2)CC1 O=C(C1=CCCCCC1)NCC1CC1NC(c1cnc(C2CC2)[nH]1)=O N1(C(c2c(C)n(CC(C)C)nc2)=O)CCCC2(CCN(C(=O)C(C)C3CC3)C2)C1 c1(CCC)ccc(N)c(C(N2CC(CNC(=O)C)C(C)C2)=O)c1.CC(N)=O c1(C(C)NC(C(C2CCC2)NC(C(C)=C(C)C)=O)=O)ccc(O)nc1 Cc1cnc(C(=O)NCC2CCCN(Cc3ccc(I)c(O)c3)C2)cc1Br N1(C(c2cc(NCCC3CCCC3)co2)=O)CCC(C=O)CC1.C1(F)CCC1.N c1(C(=O)NCCC(O)CO)cccc(S(=O)(=O)NC)c1.c1nc(C2CC2)no1 C(=O)(C(F)(F)C(O)CC)N1CCC(C(CNC(C(CC)O)=O)(C)C)CC1 C1(NC(c2n(C)nc(Br)c2)=O)CN(C(C2(C)CC3(CC3)C2)=O)CC1C1CC1 c1(CN(C2CN(S(CC)(=O)=O)C2)C=O)cc(Cl)n(C)n1 CCCCC(CC)CC(=O)NC(CCCC)CC(=O)NC12CC(F)(C1)C2 C(CN=c1cccc(S(=O)(=O)N(C)CCN(C)C)[nH]1)N1CC(C)CC(C)C1 Cc1cncc(OCC(=O)NCCCN(C(=O)C=Cc2ncco2)C)n1 C1(C)(C(N2CCCCC(Nc3nccc(C(=O)OC)n3)C2)=O)CCCCC1(F)F CCC(CC(=O)N1C(C(N2CCCC(CN(C)C)C2)=O)CC1C)C(C)C C=CCC(CC=C)C(=O)N1CCCC1CC1CCCCN1C(=O)C(O)CC(N)=O N1(C(C(CCC)N(C)C)=O)C2CCCC1CC(NC(=O)CC1CCNC1=O)C2 C1(C(N(C2CCNC2c2ccccc2)C(C)C)=O)CN(C)NC1=O c1(C(=O)NC2C(CNC(CCOC(C)=O)=O)CCCC2)cc(F)c(C)cc1F N1(C(C(C2CCN(C(c3cncs3)=O)C2)F)=O)CCn2nncc2C1 N1(C(Cc2cc(CC)nn2C)=O)CC2CCCC(C1)N2C(C1CC2(CSC2)C1)=O C1(NC(Cc2c(C)occ2)=O)(CF)CCN(C(C2(C)CCC(C)C2)=O)C1 CC1CC(CCNC(=O)C=CCC(C)(C)NC(=O)C2=COCC2)CCO1 N1(C(C(C(CC)C)NC(c2ccc(F)cc2)=O)=O)CCOCC2(CC2)C1 CC(O)CC(C)NS(=O)(=O)C1CC1c1cccc(Cl)c1.c1ccccc1.C(=O)O N1(C(CCC)=O)CCCC(C(N2CCC(N(C)C(C3CC=C(C)CC3)=O)C2)=O)C1 C(C)(C(O)C(=O)N(CCC)C1CC1)SC.c1(C=O)coc(C2CCCCC2)n1.N CC1CCN(C(C2CCCN(C(=O)C3=NNC(=O)C3)CC2)=O)C1(C)C C1(NC(C(CC#C)C2CC2)=O)(CO)CCN(C(=O)CCOc2cccnc2)CC1 c1(OC)ccccc1N1CCC(NC(=O)C(C)(C)c2ccccc2)C1=O Cn1nccc(C(=O)NC2CCOCC2NC(=O)CCCC2CCC2)c1=O c1(C(N2CCCC2)=O)ccc2c(c1)OC(C)(C)C2.C(CO)(C(=O)N)NC(C)=O CCCC(C)C(=O)NCCC1CCN(C(=O)C(c2ccc(OC)cn2)(F)F)C1 C1(NC(C(C)c2cncs2)=O)CCCN(C(c2ccc(C(F)(F)F)o2)=O)C1C c1(OC)ccc(CCNC(C2CC2C(=O)N)=O)cc1O.c1cc(Cl)cc(Cl)c1 C1CN(C(=O)C(O)Cc2cnn(C)c2)CC1N(C)C.C(C)(C(=O)N)=C(C)C C(=O)(C(CC(C)C)ONC(=O)C=Cc1cncs1)NC(CCOC)(C)C C12(C(C)C)COC(C(=O)N(C3CCC3)C)(C1)C2.C1(C=O)CC(=O)N(C)C1.N N1(C(CC(C)C(F)F)=O)CCC(C(=O)NCC2(C(C)(C)O)CC2)C12CCC2 c1(OC)cc(Br)cnc1C(N1CC(CCn2cc(C(O)C(C)(C)C)nn2)C1)=O C1(OC)CN(C(C2CC(F)(CO)C2)=O)C(C)(C)C1.CCC(C)C.C(=O)C.N C(C(CC(C)C)C(=O)N1CC2CC1C(F)(F)C2)NC(C1C(CCC)C1)=O C12(C(N(C(C)Cc3cnccn3)C)=O)CCCC1(C(N)=O)C2 CC1CN(C(c2cc(Cl)cnc2F)=O)CCN1C(=O)CNS(C)(=O)=O C1(C)(NC(CCOCC(C)C)=O)CCCN(C(C2(C)CCC3CC3C2)=O)C1 N1(C(Cc2cc(CC)nn2C)=O)CC(C)CN(C(=O)CC2CC(=O)C2)CC1C O(NC(=O)C(F)CC(C)(C)C)C(C(=O)Nc1cncc(C#C)c1)CC(C)C N1(C(c2ccc(C)nn2)=O)CC(C2CN(C(C3CC4(CCCO4)C3)=O)C2)C1 CCCC(CCC)C(C)NC(=O)NCC1(CCOC)CC1 c1(OC)[nH]c2ccccc2c1CNC(=O)N.CC(C)N(C)C=O.C(C)(C)C n1(CCC)cccc1C(=O)NCC1(C)CN(C(C2CNC(=O)C2)=O)C1.O C1(C)(NC(C(C)NS(C)(=O)=O)=O)CCCN(C(C2CCCO2)=O)C1 Cc1ccc(-c2ccc(NCC3CCC(C(C)(C)C)CC3)nc2)cc1C(F)(F)F c1(C(N2CCCC(NC(c3c(C)n[nH]c3C)=O)C2C)=O)cncc2cnccc12 O=C(C1=NN(c2ccc([N+](=O)[O-])cc2)C(=O)C1)NC1CNC2CC12.c1cccs1.C C(C(C)CCCC(C)C)NC(C1(CNC(COC)=O)CC12CCC2)=O C(c1ccncc1)=CC(=O)N(C(C(=O)NCCC(C)(C)OC)C)C CC(C)C(F)(F)CC(=O)NCCCCC1(NC(=O)C)CC1.C1CC(F)(F)C1 c1(C(C)NC(C(=O)NC(Cc2ccc(CC)cc2)C)=O)cc(Br)ccc1F c1(C(=O)N)cc(Cl)c2c(c1)OCCCO2.CC(CCO)NC(=O)CN(C)C1CC1 C1(C(=O)NC23CC(CNC(CCCSC)=O)(OC2)C3)CC(=O)NC1(C)C c1(OC)cnc2[nH]c(C(N3CCC3C)=O)cc2c1.C1(C=O)CCN(C)C(=O)C1.N C(=O)(C(F)CCC(C)(C)C)N1CCC(C)C(NC(=O)CC2CC(=O)NC(=O)C2)C1 Cc1cn2c(CCC(=O)NC3CCCCC3NC(c3n[nH]cc3C)=O)csc2n1 C=CCC(C)(O)C(=O)NC1CCN(C(=O)C(C)CO)C1 Cc1nn(C)c(Cl)c1C=CC(N1CCN(C(c2nnn(C)c2N)=O)C(C)C1)=O C(C(CCCCNC(=O)C(c1cnccn1)C)C(=O)O)c1cc(OC)c(Cl)cc1 C=CCC(C(=O)NCC1CCOC1)C(C)(C)C.C1(C=O)CCN(C2CC2)CC1.N CC12C3C4C1C1C2C3C41C(=O)NC1(C)CCN(C(=O)CC2CC=CCC2)C1 Cc1ccc2[nH]c(CNC(C3CC(=O)N(c4cnn(C(C)C)c4)C3)=O)cc2c1 C1(C(=O)NCc2cc(F)cc(F)c2)CCC2(CN(C)C2)O1.c1c(O)cccc1Cl N1(C(C(COC(c2ccc(OC)nn2)=O)N(C)C)=O)CCCC12CCOCC2 CC1(CO)CCCN(C(=O)C(Cc2cn[nH]c2)NC(=O)C#CC2CCC2)C1 CC(C)CC(O)CC(=O)NCC1(O)CCN(C(=O)CCC2CC(C)(C)CO2)CC1 C1(C(=O)NC(C)C(=O)NC2CC2)CN(C(=O)CCCC2CC2)CC(C)(C)C1 Cc1nc(C(C)C)oc1C(=O)NCC1(C)CCCC1.C1(C=O)COCC1(C)C C1(C(=O)NCCNC(C(C)OCC)=O)CCCC2(CC2)C1 CCC(C(=O)NC1(C)CN(C(C2(NC(C)C)CC2)=O)C1)OC CCCCCC(O)C(C)C(=O)NC(CNC(c1ccnc(S)c1)=O)C1CCC1 C(c1cccc(Br)c1)=CC(=O)NCC1N(C(C)=O)CC=C1 C1(NC(CCCC#CC)=O)CN(C(=O)C(C)(C(C)C)NC(C)=O)CC2(CC2)C1 N1(C(C(CNC(C(C=C)(C)O)=O)CC2CC2)=O)CC2CCC(C1)C(=O)N2 CC1(CCNC(C23CCC2CC3)=O)CCN(C(C2(C)CCCO2)=O)CC1 C1(C(=O)NCCC)(CCOC)CCN(C(C2CCCC3(CC3)C2)=O)CC1 C(CN=C(NCC1CCOC1)N1CCCC(CC2CC2)C1)N1CCC(OC)CC1 C1(C(=O)NCC(CNC(C2(COC)CC=CC2)=O)OC)CN2CCN1CC2 C1(CC)CNC(=O)CN1C(C1CC(C)CN(C(=O)CC(C)O)C1)=O c1(C(=O)NCC(c2cccc(Cl)c2)NC(CCC(=C)Cl)=O)ccnc2ncnn12 N1(C(c2cc(C)ns2)=O)CC(NC(C2OCCCC2(C)C)=O)C(C)(C)C1 c1(Nc2scc(C(N(C)CCC3OCCO3)=O)n2)ncncc1F N1(C(c2ccc(OC)c(Br)n2)=O)CCOC2CN(C(=O)Cc3noc(C)n3)CCC12 CC(C)(CS(N)(=O)=O)C(=O)NC1CCOCC1.c1(C=O)ncoc1C1CC1.C Cc1cc(NC(=O)CCC2CC2(F)F)ccc1NC(=O)C=CC1CCOCC1 C1(C2CCC(=O)NC2)(C=O)CCC1.c1(OCC)nc(C)cc(C(F)(F)F)n1.O c1(OC)cc(-c2cnc(C3CCCN3C(=O)C(C)(C)C)[nH]2)c(OC)cn1 C1(NC(C2(NC(=O)CCc3cncs3)CCN(C)C2)=O)CCCN(O)C1=O C1(NC(c2cc(CC)[nH]n2)=O)CC(NC(c2ccc(C)cc2)=O)C12CCC2.O n1(CC)c(C)nn(CC(=O)NCC(F)C)c1=O.C1(CC=O)CCNC(=O)C1.N N(C(=NCCF)NC1CC(F)(F)C1)CC(N1CCOCC1)=O n1(CC)nc(C(=O)NC(C2CN(C(=O)C(C)(C)C)C2)C)ccc1=O Cc1ncn(O)c1C(=O)NCCOC1CN(C(c2ccnn2C(C)C)=O)C1 Cc1nc2ccc(C(=O)N(CC(C)NC(=O)CCc3ccn(C)c3)C)cc2o1 c1(NCC2C(NC(c3ccc(C(C)(C)C)cn3)=O)CCC2)ncnn2cccc12 C1(C(N2CC(F)(CNC(c3c(C)onc3)=O)C2)=O)CCSC(C)C1 N1(C(C(C)c2cccs2)=O)CC2CCCC1C2CNC(=O)CCc1cncs1 c1(N2CCN(C(C3CCN(C)C3)=O)CC2C#N)ncnn2cc(Br)cc12 C1(c2nnnn2CC)(NCC(CC)C)CC(n2cncn2)C1 CCC(CC)(CO)C(=O)N1CC2CCC(C1)N2C(C1CCCSC1)=O N1(C(COC(CC)C)=O)CCOC2(C1)CN(C(c1ccc3cnccc3c1)=O)C2 C1(C(=O)Nc2cn(CC(F)(F)F)nn2)CCCN(C(=O)Cc2cccc(F)c2)C1 C1(C(N(C(C)C2CC2)C)=O)CC2CC1CN(C(C1CSC1)=O)C2 Cc1cccc(C(C)(C)C(=O)N2CC(OCCNC(C3CC4CC3C4)=O)C2)c1 CCCCC(O)C(C)C(=O)NCC1CC(OC)CN1C(c1cn(C)nn1)=O C(=O)(CCCCN=[N+]=[N-])N1CC(C(=O)NCC(C(C)C)C(C)C)OCC1 Nc1c(C(=O)NC23CCC(C2)N(C(=O)CS)C3)nc(O)nc1O.CCNC=O C1(C=O)CN(C(c2cncc3[nH]ccc23)=O)C2(CCC2)C1.C1CC1C(F)(F)F.N C1(CC)CC(C(=O)NC(C)C(C)(C)NC(C2CC(O)C2)=O)CC(=O)N1 N1(C(COCc2c(C)ncs2)=O)CCOCC(C)C1.C1(C)(C=O)CC2CC2C1.N C1(C(N(C(C)CNC(=O)C(C)OCCC(C)C)CC)=O)OCCOC1C C1(C(N(C(CN(C(C)=O)C)C)C)=O)(NC(=O)C(C)O)CCN(C)C1 C1(CCNC(=O)CNC(=O)C2CC2)CCCN(C(=O)Cn2cccn2)C1 Cc1occc1C(=O)NC(CNC(=O)CC(C)C1CC1)CO Cc1cc(C=CC(N2CC(F)(C)C2)=O)c[nH]c1=N.c1(C(=O)N)c(F)cccc1F C(=O)(CCCCCl)N1CC(C)(C(=O)NCc2ccccn2)C1 C1(C(C#C)NC(=O)CCN(C(=O)C(SC)SC)CC)CCCCC1 N1(C(c2cn(C(C)C)nc2)=O)CC2(CNC(=O)C=C3CC3)CC1CO2 C1(NC(CC2(C(=C)F)CCC2)=O)CC2CCC1N2C(=O)CCn1cnnn1 C(=O)(CS(=O)(=O)CCOC)NCC(C1CCCC1)NC(C(CCC)O)=O c1(C(N2CCC(COC)(NC(=O)CC3CC3)C2)=O)cc2cccc(C)c2o1 N1(C(CN2CCN(CC)CC2)=O)CCC(NC(c2ncc(C)cn2)=O)C(F)C1 N1(C(c2cnc(CCCC)s2)=O)CCC(F)(CNC(c2[nH]c(C)nc2C)=O)C1 c1(OC)ccc(C(=O)N(CC(C)NC(C2CC3CCC3C2)=O)C)cc1Cl C12(NC(c3c(C)ccc(C)n3)=O)CCC(CN(C(c3cnc(C)[nH]3)=O)C1)C2 Cc1ncsc1C(=O)NC(C(=O)NC1CC(CN(C)C)C1)C1CCCO1 C1(c2n(CCOC)nnn2)(Nc2cc(C)c(C)c(C)c2)CCCC2CN(C)CC12 C1(CCOC)(NC(c2cnnc(Cl)c2)=O)CCN(C(=O)C)CC1.CC(N)=O.S c1(C(N(CCN(C(C)C)C(C2CC(C)N(C)C2)=O)C)=O)cccc(N)c1F C(=O)(C(F)(F)C(C)O)N(CCCCCCNC(C1(OC)CCOC1)=O)C Cc1nc(NC(c2cc(-c3c(F)ccc(F)c3C)ccn2)=O)cnc1C#N CC(C)(C(=O)NCC1CC(NC(c2ccc(CO)o2)=O)CC1O)C(N)=O Cc1ccc(CCC(=O)NC2C=CCN(C(=O)C=Cc3cc(C)no3)C2)cc1 C1(C(=O)N)(CNC(=O)COCC2CCCOC2)CCCCCC1.c1cccs1 C1(C(NOC(C)C)=O)CN(C(=O)C(CO)N(C)C)C(C)(C)C1 C1(C(=O)Nc2c(C)ccnc2)CC2CC1CN(C(=O)Cn1ccnc1C)C2 C1(CC#C)(C=O)CCCO1.c1(C(N(CC)C2CC2)=O)cc(C(F)F)no1.N Nc1ccc(F)cc1C(N1CC(CCCCNC(c2cn(C(F)F)cn2)=O)C1)=O c1(C(=O)NCCSC2CCCC2)ccc(-c2ccsc2)cc1 N(C(=S)NC1CCc2cccc(F)c21)c1c(Br)ccc(OC)c1 C(CC(=O)NC1CC(F)(C)C1)(C(C)C)OCC.c1cnn(C)c1.C(=O)C C(C(N)C(C)C(C)C)NC1(c2n(Cc3cccc(OC)c3)nnn2)CCC1 CC1(C)CC(C(=O)NC2(c3ccccc3)CC2)CN(C(=O)C=CC2CCC2)C1 c1(CC)ccc(F)c(C(=O)NC2COCCN(C(C3CC(=O)N(OC)C3)=O)C2)c1 Cc1nc[nH]c1CCNC(=O)C(C1CCCC1)NC(=O)C(C)n1cccn1 C1(NC(=O)CC2CCCC2)C=CCCC1C(=O)NC1CCCNC1=O CCCCCC(CC)C(=O)NCC(C1CC1)NC(=O)C=CCO Cc1nc(NCCN=S(C)(C)=O)cc(=NC(C)CS(C)=O)[nH]1 c1(C(=O)NC(C(C2CCCCC2)NC(COC)=O)C)cccc(F)c1C c1(NC(CCNC(C2CCCN(CC)C2)=O)(C)C)cc2nncn2cn1 CC(F)(F)C(F)C(=O)N1C2CCC(C2)C1C(=O)NCC1(C2CC2)CCC1 Cc1ccncc1CC(=O)NCC(C1CC1)NC(=O)C(=O)NC1CC1 c1(C(=O)NC2(C3CCCN3C(=O)C3=CC4CCC3C4)CC2)cccc2ccoc12 C(=O)(C(O)Cc1cnc[nH]1)N1CC(N(C(C)(C)C)C(C2(C)CNC2)=O)C1 N1(C(C2(CC)CCOCC2)=O)CCOCC(NC(c2c(C)cncc2C)=O)C1 c1(C(=O)OCC(=O)Nc2cc(Br)cs2)cc(Cl)cc(Cl)c1 c1(NC(N(C(CC)C)C)=O)ccc(Br)c2nc(C)ccc12 c1(OC)ccc(F)c(C(=O)NCCC)c1N.c1(C=O)cccc(C(F)(F)F)n1.N C1(C)(CNC(c2cnc(SC)s2)=O)CCCC1.C(C1CCCO1)=CC=O.N c1(SCC2(C(=O)NCC(C)N(CC)CC)CC2)ncn(C)n1 C1(C2CC2)(CNC(C(CC)C)=O)CCN(C(=O)C2=NOCC2)C1 c1(C(=O)NC2CC(CC(=O)NC(CC(C)C)(C)CO)C2)ccc2[nH]ccc2n1 C(C)(CO)(C(=O)N(CCNC(C1CSCCS1)=O)C1CC1)OC C#CCCCCCSCC.C(C)CC(F)F CCS(=O)(=O)CC(=O)NC1CCCCCC1C(=O)NCC(C)CC(F)(F)F c1(C(N2C(CNC(c3c(Cl)ncc(C)c3)=O)CC2)=O)ccnc2ccc(N)cc12 N(C1CC2(CCNC2)Oc2ccccc21)c1ncc(NC(CC)=O)cn1 [N-]=[N+]=NC1CCC(NC(=O)CC2CCN2C(=O)CCC(N)=O)CC1 c1(C=O)cnc(C)cn1.N1(C(CNC(CC2(OCC)CCC2)=O)=O)CCCC1 CC1=CCC2CN(C(C3(C)CCCN(CCS(C)(=O)=O)C3)=O)CC2C1 c1(C(=O)OC)ccc(NC(C2CCN(S(=O)(=O)CCBr)C2)=O)nc1Cl N1(C(c2cnc(C)nc2)=O)CCOCC(NC(=O)Cc2sccc2Cl)C1 C1(CCC)CCC(NC(C2CCN2C(C2C(C)C2C)=O)=O)CC1 n1(CCOC)ccc(=NC(=O)C2CN(C(=O)CC3(C)CCC3)CCO2)[nH]1 C(c1ccc2c(c1)OCCO2)=CC(N1CC(C)N(C(=O)CC2CCOC2)CC1)=O C1(C(=O)NCCCN(C(c2cc(O)ccc2)=O)CC)Cc2nnc(C)n2C1.O N1(C(C(CC)NC(C)=O)=O)CCC2C1CCN2C(C1CCC(CC)CC1)=O C1(Cn2cc(CN(CC)CC)nn2)CCCCN(C(C2(C#N)CC2)=O)C1 N1(C(c2ccc(CO)o2)=O)CC=CC(NC(C2(c3ccc(F)cc3)CC2)=O)C1 c1(Cn2c(CSC)nc(-c3ccc(C)cc3)n2)ccc(Cl)cc1Cl C1(CC#C)CCN(N2CCCN3CCCC3C2)C1 Cc1nsc(N(C)CC2CCN(C(c3nccn3C(C)C)=O)C2)c1C#N c1(C=O)cn(C2CC2)c(C)cc1=O.C1(NC(C(C2CC2)OC)=O)COCC1.C C1(C(=O)OC)CN(C(c2ccc(C)nc2C)C(=O)NC2CC2)CC1(C)C c1(C(=O)NCC(C(C)C)NC(C=C(C)C(F)F)=O)cn(C)nc1C(C)C CC1(C)C(C(=O)NCC2CCCC2)CCS1(=O)=O.C1(C#N)(C=O)CC=CC1 CC(C)(C)CC(F)C(=O)N1CCC1CC(=O)NC1CC(CCF)C1 c1(C(=O)NC2(CNC(CC3CN(C)C3)=O)CC2)nccnc1N N1(C(c2ccc(CC)o2)=O)CCCC(CC(=O)NC2CC(F)(F)C2)C1 C#Cc1cccc(C(N2CCC(NC(=O)CP(C)(C)=O)CC2)=O)c1C C1(NC(c2nnn(CC)c2C)=O)CN(C(=O)CCC2CCC(=O)NC2)CC12CC2 C1(NC(=O)NC2CCC(CC(=O)OC)C2)CN2CCC1(C)CC2 C1(OC)CC(C(=O)NC2(CCNC(=O)CC3CCCN(C)C3)CC2)CC1 C1(c2n(CCCSCC)nnn2)(NCC(C)C2CCC2)CCC(=O)NC1 CN1CCOC(C(=O)NCC2CN(C(c3cc(Cl)n(C)n3)=O)CCCO2)C1=O c1(C(C)C(=O)NC(C)C(C)NC(c2c[nH]c(=N)s2)=O)cn(C)c2ccccc12 C12(NC(CN(C(C3C(C(C)C)CCO3)=O)CC3CC3)=O)CCC(C1)OC2C C(CN=c1[nH]c(C)cc(=NCCC=CBr)[nH]1)N1C(=O)CC(OC)C1 C1(C(=O)NCCO)CC2OCCC2N(C(c2ccccc2Cl)=O)C1 c1(C(N2CCC(CNC(C(C(C)C)O)=O)CC2)=O)cc(Cl)cc([N+](=O)[O-])c1O N1(C=O)CCCC(C=O)C1.C1CCCN1C(=O)C(C)C.C(C)C.CCSC c1(C(N2CC(C(C)NC(=O)CC3CCOC(C)(C)C3)C2)=O)cccc2[nH]ccc12 C1(CC(=O)NC2CC(C)(C(N3CCC(CCCC)C3)=O)C2)CCC(C)(C)O1 CCC(CC)CC(F)C(=O)N(C(CCN(C(=O)CC(C)=C(C)C)C)C(C)(C)C)C c1(C(=O)NCC(CC(=O)N(CC(F)F)CC#C)C)cc2occc2[nH]1 Cc1cn2c(n1)CCC(C(N1CCC(CF)(NC(C3CCCC3)=O)C1)=O)C2 c1(C(N2CCC(C(F)(F)F)(OC)CC2)C(=O)NCCC)cc2nccc(Cl)c2s1 N1(C(C=C(C)c2ccco2)=O)CC(C(N2CCCC(F)(F)CC2)=O)CC12CCC2 C(CN=c1cc(C)[nH]c(=NCC=C(C)C)[nH]1)(C1CCOCC1)OCC c1(C(=O)OC)cc(=NC(=O)C2CCCN(C(=O)C(F)(F)Cl)C2)[nH][nH]1 N1(C(Cc2n(C(C)C)ncc2)=O)CCC2(CCC(NC(C3(C4CC4)CC3)=O)C2)C1 C(C)(CCC(=O)NC1(C)CC(NC(c2ncoc2C2CCCO2)=O)C1)SC CC1CC1C1CC1C(=O)NCCN1CCN(Cc2sncc2Br)CC1 CC1COC(C)(C)CN1C(c1cc(CNC(C2CCC3(CC3)C2)=O)no1)=O N1(C(C(COC(C)=O)C)=O)C2CCC(C2)C1C(N1CCC1c1ccccc1)=O Cc1ccc(Cl)cc1C(N1CC(NC(c2cc(C3CCC3)no2)=O)C(O)C1)=O Cc1cccc(CC(=O)NCC2(C(F)F)CCN(C(c3cnns3)=O)C2)c1Cl C1(C(N(CCNC(CC(=C)C)=O)C)=O)NC(=O)CC1C NS(=O)(=O)c1ccc(CCNC(C2CCN(C3CCCC3O)CC2)=O)s1 C1(CNC(CC2C(CC)C2(F)F)=O)CCCCCN1C(=O)C=C1CCC1 N1(C(c2cc(CC)c(F)cc2)=O)CC(NC(=O)CCC2CC(C)C2)C2CCCC12 N1(CC)CCOCC1CC(=O)NCC1(F)CN(C(=O)CCCc2ccccc2)C1 C(=O)(CCCCc1cnn[nH]1)NCCC1CN(C(C(F)OC)=O)C1 N1(C(Cc2cc(C)on2)=O)CCSCC1CCNC(=O)CCN1CCC1 N1(C(c2occ(C)c2)=O)CCCC2(CCN(C(C3CCCCC3(F)F)=O)C2)C1 N1(C(c2c(CC)occ2)=O)CC2CN(C(c3ccc(Cl)o3)=O)CC2(C)C1 C(C)(C)(CC(C)C)NC(c1ccc(OC)nc1)=O.C1(N(CC=O)C)CCCC1 C(=O)(C1=CC2CCCC12)NCC1=CCN(C(C2CC(C)(O)C2)=O)CC1 Cc1cccc(C(=O)N(C(CC(F)F)C(=O)N2CC3CC2C3)C)c1C#N C1(CC(=O)NC2C(NC(COCC(C)C)=O)COCC2)CCCCCC1(F)F C(N=c1[nH]cnc2ccccc12)c1ccnc(C(F)(F)F)n1 c1(C(N2C(C)C(NC(=O)CC3(O)CCOCC3)CCC2)=O)ncnc2sccc12 C(CC(C)C)(C(=O)N1CC(CO)C(O)C1)NC(c1cc(CC)on1)=O c1(OC)ccc(C(=O)N)nc1.C1(C(C)C)CCN(C(=O)C(C)(C)C2CCOC2)C1 C=CCC(F)(F)C(=O)NC(C)C(C(C)C)NC(c1cc(C(F)(F)F)ccn1)=O C1(C(N2CC(NC(CNC=O)=O)C(O)CC2)=O)CCC2(CCC2)CO1 c1(CCN(C(CNC(C)Cc2cccnc2)=O)C)cccc(C(=O)O)c1 C(C(CCN=c1nc(N2CCCC(C(=O)N(C)C)C2)cc[nH]1)C(C)C)OC c1(C(N(C=O)Cc2cn(CCC)nc2)C#N)ccc(Cl)cc1F CC1C(=O)CCC(C(N2CCCC2CN(C)C(C2CCC(F)C2)=O)=O)C1(C)C CC1SCCCC1C(=O)NCC1(NC(c2cn(CC(F)F)cn2)=O)CCC1 c1(C(N(C(C)CCNC(=O)CC2CCCCN2C)C)=O)cnn(C)c(=O)c1 c1(C(N2CCN(C(=O)COCC(F)(F)F)CC2)=O)c(O)ccc(Cl)c1F c1(CC)ccc(C(N2CCCC(C(N3CCC3CC)=O)C2)=O)nc1 C1(NC(c2cc(C(N)=O)[nH]c2)=O)CC2CC(C1)N(C(=O)CCC1CCOC1)C2 n1(C(C)C)ncc(C(=O)NCC2CC(F)CN2C(=O)C(O)C2CCC2)c1N C(=O)(CCCS(N)(=O)=O)N1CC2C(CNC(C(c3ccc(C)cc3)=O)=O)(C2)C1 N1(C(=O)NCC2(CC)CCCCO2)CC(O)CCC1C C(=O)(C(CCC)C(C)C)NCC1CCC(C(NOCC=C)=O)CC1 c1(N2CC(c3[nH]nc(O)n3)C2)ncnc2ccccc12 C(CCCCC(=O)NCC1(O)CN(C(c2csc(Br)c2)=O)C1)SC CC1CCN(C(C2CNC(=O)O2)=O)CCN1C(=O)CNS(=O)(=O)C1CC1 c1(OC)cc(C(=O)NCC2CC3(C2)CN(C(=O)CC)C3)ccc1O.C(C)=O n1(CC)nccc1-c1cn(C2CC(C(=O)NCCc3cnc[nH]3)C2)nn1 c1(C(=O)NC2CN(C(CN(c3ccncc3)C)=O)C3C2C3)cnc2n1CCC2 S(=O)(=O)(c1cccc(Br)c1Cl)NCCC1(C)CC1(F)Cl c1(CC)[nH]nc(C(=O)NCC(C(C)C(C)C)NC(=O)C2=CCCCC2)c1[N+](=O)[O-] Cc1ncc2n1CCC(C(N1CCC3CN(C(=O)CCC(F)(F)F)CC13)=O)C2 N1(C(C2(CNC(c3n[nH]c(C)c3O)=O)CC(=C)C2)=O)CCCC(C2(C)CC2)C1 CC1(C)CC(C(N2CCOC(C#N)C2)=O)N(C(c2ccc(C#N)s2)=O)C1 C1(NC(C(C(=O)OC(C)(C)C)F)=O)CCC(N=[N+]=[N-])CC1 N1(C(c2n[nH]c(C)c2Br)=O)CCN(C(=O)C(N)=O)C(CC(C)(C)C)C1 N1(C(C(C)CO)=O)CCOC2CN(C(C3(F)CCCCC3)=O)CC12 Cc1c[nH]cc1C(=O)NCC(O)CN(C)C(c1conc1C1CCC1)=O CC(C)(C(=O)N1CC2C(CNC(=O)C(c3cccc(Cl)c3)(C)C)C2C1)C(F)F c1(N(C)C)ncc(C(=O)NC2CCC2CNC(=O)CCc2cscn2)o1 C=CCC(C(=O)NCC(C)NC(c1nn(C)cc1C(C)=O)=O)C(C)(C)C C#Cc1ccccc1NC(C1CC12CCN(Cc1ccc(C)[nH]1)C2)=O c1(C(=O)NC(C(=O)OC)C)conc1CNC(C1CC1(Cl)Cl)=O C1(C(=O)NC2CCCN(C(=O)CC=C(Cl)Cl)CC2)CC(c2ccccc2)=NO1 N1(C(C(CC)n2cccn2)=O)CCC(CO)(CNC(c2[nH]cc(C)c2C)=O)CC1 C(=O)(C#CC1CCCOC1)N1CCC(CN(C(c2cn(CC)nc2C)=O)C)C1 c1(C(=O)Nc2cn(CCNC(C(CC)C)=O)nn2)cccc(NC(C)C)n1 C1(CNC(CCC#CC)=O)CN(C(c2ccc(O)nn2)=O)C2CCN1C2 c1(C(N(CCCN(C)C(c2ncccc2Br)=O)C)=O)cc(N)cnc1Cl C1(C(N2CCC(NC(C3ON=C(C)C3)=O)C2C2CC2)=O)CCC(C(N)=O)CC1 N1(C(COCC(C)(C)C)=O)CCN(C(=O)CCc2ccccn2)C(C2CCC2)C1 C1(C(=O)NC2CC(C)N(C(C3CCC4(CCC4)O3)=O)CC2)CN=C2N=CNN2C1 c1(C(N(C(C)CCNC(C2CN(C)C(=O)N2)=O)C)=O)cnn(C)c1C#N c1(CN2CC(NC(c3nc(C)c(Br)cc3)=O)C(O)C2)cccc2ccccc12 C(CC(C(C)C)NC(c1ccnc(OC2CC2)c1)=O)N(C(c1c(C)nc[nH]1)=O)C N1(C(=O)CC2(CO)CCC2)CC(CCO)c2ccccc21 c1(C(N(C)CC2COCCN2C(=O)C#CC(C)(C)C)=O)cc2c(nn1)CCCO2 C(C(=O)NC1COCC1NC(=O)Cc1n[nH]c(=N)s1)(C(C)C)SC C1(C)(CNC(CC(=C=C)C)=O)CCCN(C(c2cc(Br)c(C)cn2)=O)C1 Cn1cncc1CN(C(c1ccc(F)s1)C(=O)NCC1CCCO1)C Cc1oc(C#N)cc1C(=O)NCC1(O)CCC1.C(=O)C(C)SC(F)(F)F.N c1(C(N2CCN(C(C(COC)COC)=O)C(C)CC2)=O)c(N)sc2c1CCSC2 N1(C(C(COCC)NC(C2CC3(CC3)CO2)=O)=O)CC(C)C(F)(F)C1 c1(OC)cccc(CNC(=O)NCCNS(N)(=O)=O)c1Br c1(CC)nc(-c2cc(Cn3cc(Br)cn3)on2)n(C(C)C2CC2)n1 c1(CC)sc(C(N2CCC(CC(C)NC(c3c[nH]c(=NC)o3)=O)CC2)=O)cc1C N1(C(C(CCC)N(C)C)=O)CCC(CNC(c2ccoc2Br)=O)C12CC2 C1(C(N(CC(C)O)C)=O)COCCN(c2ccc(C(=O)C3CC3)cn2)C1 CC1CNC(=O)CN1C(=O)C(Cc1cc[nH]n1)NC(c1cccc(CO)n1)=O c1(C(=O)NC2CCN(C(C(C)C#N)=O)C2(C)C)ccc2oc(=O)oc2c1 CC(C(C)C(=O)N1CC(NC(=O)CCC2CC2)C(C)C1)S(C)(=O)=O C(CCCC(=O)N1CCC(N(C(C2CCCC2SC)=O)CC)CC1)OCC c1(SCC(=O)N(c2cncc(Cl)n2)C(N2CCOCC2)=O)cn2c(n1)CCCC2 c1(CC(=O)NCC(CC)(C)NC(=O)C=CC(F)(F)F)ccc2nonc2c1 C(=O)(C(O)C(C)(C)C)N(C)CC1CCN(C(=O)Cc2ccccc2)C1 N1(C(C2(C)CC2(F)Cl)=O)CC2CC(NC(c3cn4c(n3)COCC4)=O)CC2C1 c1(C(N2CC(NC(c3c(C)cnn3C)=O)CC2(C)C)=O)cc2cc(Cl)cnc2[nH]1 C(CC(C)C)(C(=O)N)NC(c1cc(C)nnc1)=O.c1ccccc1CC(=O)N(C)C C1(NC(c2c(CC(C)C)cccc2)=O)CCCC2CN(C(C)C)CC12 N1(C(C=Cc2ccc(C)s2)=O)C2CCC1CN(C)C2.C12CC(C1)C(=O)N2 c1(C(=O)OCCCC(N)=O)cc([N+](=O)[O-])cc([N+](=O)[O-])c1 c1(NC(CCCC)CC)ccc(S(=O)(=O)N2CCOC(C(N)=O)C2)cc1C#N C(CC(C(=O)NC1CC2CCC1O2)NC(=O)C(F)OC(F)(F)F)OC CCCC(C)(O)C(=O)NCC1(O)CCCN(C(=O)Cc2ccc(C)cc2)C1 c1(C(N(CCNC(C2CC3CC3C2)=O)CC)=O)nnn2c1CCCC2 C=CC(CC)CC(=O)NCCC(C)CCNC(c1cc(C(F)(F)F)cc(Cl)c1)=O C1(CC)CN(C(=O)CC=CC(C)(C)C)CC1C(=O)N(C1CCC1C)C C1(C(N2CC(CNC(c3n[nH]cc3F)=O)C2)=O)(COC)CCCCC1 c1(C=O)ccc2cc[nH]c2c1F.C1(C(C)C)(CC)CC1C(=O)N.C1(CC)CC1 c1(C(=O)NCCC(C)N(C)C(c2cccc(F)c2Br)=O)ccc(F)c(N)c1 c1(C=O)cn2c(n1)SCC2.CC(C)(C)CC(=O)NCCCOCCOCC Cn1cnc2[nH]c(=NCC3CC=CC3)[nH]c(=NC3CCCN(c4ncc[nH]4)C3)c12 C1(OC)C=CCN(C(=O)C(C)N(C)C(c2cn(C)cn2)=O)C1 Cc1noc(C)c1C(C)C(=O)N(C(C)CNC(c1nc(Cl)cs1)=O)C c1(C(N2CC(NC(C3CCC(CCCC)CC3)=O)C(C)C2)=O)cc(O)cc(O)n1 N(C1COc2ccccc21)C(CCN(C(c1cc(C)c(C)nn1)=O)CCO)=O c1(C(=O)NCC(CNC(c2ncn(C(C)C)c2)=O)O)ccnc(F)c1 c1(C(N2CC(NC(CCC(=C)Cl)=O)C(O)C2)=O)c(F)ccc(C)c1F c1(OC)ccc(-c2cc(CN3CC4CC(C3)O4)ccc2OC)cc1OC C1(OCC(=O)NC2(C(=O)NCCOc3nnc(O)o3)CC2)CCCCC1 CC1(C)CCN(C(=O)C2=C(Cl)CCC2)CC1C(=O)NCCC(C)(O)C1CC1 c1(CC)c(C(=O)NC(CNC(=O)Cc2ncoc2C)C2CCC2)nn[nH]1.C C(C(CC(F)(F)F)NC(=O)COCCc1ccccc1)NC(C=C(C)Cl)=O CC1(CNC(C2CCCC23CC3)=O)CC(F)(F)CN1C(=O)CN1CCSCC1 N1(C(c2c(NC)ccc(F)c2)=O)CC2CCC1C(NC(=O)C(C)C(C)COC)C2 c1(CC(N2CC(C)(CNC(c3cocn3)=O)OCC2)=O)coc2ccc(F)cc12 C1(NC(C(c2c(C)cccn2)(F)F)=O)CN(C(=O)C(C)(C)C2CC2)CC1N=[N+]=[N-] C1(C(=O)NC2CCCN(C(C3(C)CCC(=O)C3)=O)C2)CCc2nc(O)[nH]c2C1 C1(CC(=O)NCCC(C)C)CCCC2(CCC2)O1.C1(C=O)CC2(C1)CC(O)C2 C(=O)(C1=CCCC1(C)C)NCCC(C)(C)CNC(c1ccc(Cl)nc1N)=O N1(C(c2c([N+](=O)[O-])cc(C)c(Cl)c2)=O)CCc2ccc(F)cc2C1C(C)C c1(C(=O)N)cc(F)cc(Cl)c1O.C1(C)(CC)CCCN1C(=O)C(F)CC1CC1 Cc1ccc(-c2cn(C(C)C(c3ccccc3)NC(=O)CC3CCC3)nn2)nc1 C(=O)(Nn1ccccc1=O)C1(C#C)CN(C(=O)CCCC(F)(F)F)C1 Cc1cc(C(=O)NCCN(C(=O)C(F)CC(C)C)C(C)C)cnc1C N1(C(CCOCCCOC)=O)CCN(C(=O)Cn2ccccc2=O)C(C)CC1C CCC(C)(CCNC(=O)CCSC)NC(C1(CC(F)(F)F)CC1)=O N1(C(C2C(OCC)C2)=O)CCCCCC1CNC(=O)CC1(C)CCC1 Cc1cc([N+](=O)[O-])cc(C(=O)NC(C)CCNC(=O)Cc2cn(C)nn2)n1 c1(NS(CC)(=O)=O)ccc(C=O)cc1.C12CC(C1)C2.c1(C=O)ocnc1C.N C1CN(C)CCN1C(C1CC1(F)F)=O.c1(C(=O)OC)nccnc1C(=O)N.C N1(C(C(C(C)C)N(C)C)=O)CCC(CNC(=O)CC2CC(F)(F)C2)C1(C)C C1(C(N2CCCCC2C)=O)(CC)CCN(C(c2ccc(C#N)s2)=O)C1 c1(C(N2CC(O)(C(C)NC(CCCC#CC)=O)C2)=O)cnc2c(c1)COC2 CC1CC(C(=O)N2CC3(CC(NC(C4(C)CCC(F)(F)C4)=O)C3)C2)=NO1 Cc1ccc(C(N2CCN(C(=O)C3CC3)CC2)=O)cc1S(=O)(=O)N1CCOCC1 C12(NC(C(C)OCC)=O)CCC(C1)OC2.c1(C=O)c(C)noc1C(C)C C(CC(CC)C(=O)NCC(=C1CN(C(=O)Cc2ccsc2)C1)F)=CC(C)C c1(OC)cccc(CCN=C(NCCF)NC2CCCC(C(C)C)C2)c1F Cc1c(I)cc(CN2CC3CN(C(c4ccncc4O)=O)CC3C2)cc1I Cc1noc(CCC(N2CCCC2C(c2ccccc2)SC2CCC2)=O)n1 c12nocc1OCCOC2=O.C1(=O)CO1.C1(CC)CCC1 N1(C(c2c(F)ccc(C)n2)=O)CC(F)(F)CC1(C)CNC(C1(C)CSC1)=O c1(OCC)ccc(S(=O)(=O)N2CCCOC(c3ccccc3)C2)cc1C(=O)O CC(CN=c1[nH]c2c(c(=NCc3ccco3)[nH]1)CCC2)c1ccc(Br)cc1 C(C)(C)(CCCNC(=O)CSC1CC1)NC(CC(C)n1cccc1)=O C(CSC)(C(=O)N(CC(=O)NOC(C)(C)C)CCOCCO)OC C(=O)(CCCCNC(C1(C(=O)N(C)C)CC1)=O)NCC(C)(C)C#N N1(C(CC2N(CC)CCC2)=O)CCCC2(C1)CN(C(=O)Cn1ccccc1=O)C2 C1(NC(COCC(=C)C)=O)CCCCCN(C(=O)COC2CC2)C1 C(=O)(N=c1nc(CC)[nH]s1)NCC(COCC)(C)C c1(CNC(c2c(C)[nH][nH]c2=N)=O)cc(C)n(-c2cccc(F)c2)c1C c1(Cc2nnnn2C(C)C)cnccc1C(F)F.C(C=O)(C1CCOCC1)OC.N n1(CC=O)nc2n(c1=O)CCCC2.n1(COC)ccc(C(=O)NC(C)CC)n1.N c1(C(=O)NC2(CNC(CN3CCN(C)CC3)=O)COC2)cc2ccccc2n1C N1(C(c2ccc(C)c(Br)n2)=O)CCc2[nH]c(=N)[nH]c(=N)c2C1 C(CCC(C)C)NC(c1nc(C(C)OC)oc1)=O.c1(CCC=O)ccn(C)n1.N N1(C(CC(C(C)C)C)=O)CC(C2CCCCN(C(C3(O)CCCCCC3)=O)C2)C1 C1(C(=O)NCc2ccnc(C)n2)COCCN(C(=O)CCc2ccco2)C1 N1C(=O)CN(CCC(C)(C)C#N)C1=O.c1(C2C(C=O)C2)ccco1.CC(C)C.O N1(Cc2cc(OCC)c(OC)c(Cl)c2)C2CNC(=O)CC1CC2 C1(NC(C=CCN(C)C(c2ccc(CF)cc2)=O)=O)C(=O)NCCC1C c1(CC)ccccc1NC(C1CN(C(C)=O)C1)=O.C12COCC1NC2=O C1(C(N2CCC(CCNC(C(CC)(C)O)=O)CC2)=O)CC2(C)CC1CO2 N1(C(C(C)O)=O)CCC(NC(c2coc(Cc3ccccc3)c2)=O)C(F)C1 N1(C(c2cc(CCC)nn2C)=O)CCC2CCN(C(C3(C)CC4(CC4)C3)=O)CC12 C1(C(N2CCN(C(c3cnnc(O)c3)=O)C(C(F)F)C2)=O)CCn2cnnc2C1 Cc1nn(CC(=O)NC2CC(C)CN(C(=O)C3=CCCS3)C2)c(C)c1Cl Cc1cn2c(n1)CC(C(N1CCC(NC(c3coc(Br)c3)=O)C(C)(C)C1)=O)CC2 c1(C(C(=O)N)O)cccc([N+](=O)[O-])c1.c1(CC)ccc(C(=O)NC(C)CO)[nH]1 c1(CC(N2CCCN(C(C3C(C)CC3)=O)CC2CO)=O)cc(F)cc([N+](=O)[O-])c1 Cc1cccc2nc(C(=O)NCC(C)CNC(c3ccc(Cl)c(F)c3O)=O)cn12 c1(CCNC(C2C(C(N)=O)OCC2)=O)cc(Br)cc(Br)c1 c1(C(N(C)CC2N(C(C(C=C)O)=O)CCCC2)=O)c(C)nc2ccnn2c1C C1(C(C)C)N(C(c2nccnc2Cl)=O)CC12CCN(C(C1CC(=O)N1)=O)CC2 NC1CC2(C1)C(C(=O)NC1CCN(CCSc3ccccc3)CC1F)C2(F)F C1(CNC(Cn2nnc(C)n2)=O)CC2(CC2)CN1C(=O)C1=NOC(C)C1 c1(OC)ccc(N(C(=O)C(C)(C)Oc2ccc(Cl)cc2)C(C)C)cc1OC C1(C2CCN(C(=O)C(C(C)C)OCC)C2)(NC(C(C)=CC)=O)CC1 c1(C(=O)NC2C(F)CCN(C(CCC(CC)OC)=O)C2)cn(C)c2ccccc12 CC(C)CCC(F)C(=O)NCCN(C(C1CNC(=O)O1)=O)C(C)C N1(C(C(C)C)=O)CCC2(CCC2CNC(C2(C(C)(C)C)CCCC2)=O)CC1 N1(C(C(CC)C(C)C)=O)CC2(CCC(NC(c3sc(C)cc3Cl)=O)CC2)C1 Cn1nc([N+](=O)[O-])cc1C(N1CCSCC1CCNC(=O)CC1(O)CCC1)=O c1(C(=O)NCC(CN(C(C=CC(CC)C)=O)C)O)ccc2cc[nH]c2c1 Cc1nc2ccc(Br)cc2c(N2CCC(C3CCCO3)CC2)c1C N1(C(C2(C3CC3)CCC2)=O)CCC2(CCN(CCCOc3ccccc3F)C2)C1 CCCCC(CC)C(=O)N1CC(NC(=O)COCc2ccc(C)cc2)CCC1C C1(C(N2C(C)(CNC(C(F)OC)=O)CCC2)=O)CNc2ccccc2O1 C1(C(N2CCC(C(=O)NC(C3CN(C(N)=O)C3)C)CC2)=O)COCCC1(F)F c1(NC(C2CC(C)CN2C(c2cc(Br)ncc2Br)=O)=O)cccc2ncccc12 C1(NC(c2c(CC)con2)=O)CC12CCN(C(=O)C(C)(COC)COC)CC2 C1(CNC(C2N(CC)CC2)=O)CCCCN1C(C1(c2ccsn2)CC1)=O C1(NC2CC(C)SC2)CC2CCCCC2N1CC(=O)Nc1c(Cl)cc(Cl)cc1Cl N1(C(C(CSC)(C)C)=O)CC(CNC(=O)C(c2cccnc2F)(C)C)CC(C)C1 c1(C(N(C2CCCCC2)C)=O)ccc2cc[nH]c2c1.N(C)(S(N)(=O)=O)CC=O.N C1(C=O)C(=O)N2CCC(CC2)CN1.C(C)(C)(C)OC.C(=O)(C)N.C=O C(CC(=O)N(CCNC(c1ccco1)=O)C1CC1)NC(c1ccco1)=O c1(NC(N2CC3COCC2C3)=O)ccc(S(=O)(=O)Cc2ccccc2)cc1 C1(CNC(CN(C)CC)=O)CC(O)C(O)CC1C(=O)N.n1(CC)cccn1 Cc1ccc(S(=O)(=O)N2CCC(n3c(=O)oc4ccccc34)C2)nn1 Cc1ccc(C)n1CC(=O)N(CCC(N1CC2CC2(C(N)=O)C1)=O)CCO C1(NC(c2nnc(C)s2)=O)CCC(C)(CNC(c2csc(Cl)c2)=O)C1 C(=O)(C1CSc2ccccc21)N1CCN(C(c2c(C)nc(CC)s2)=O)C(C)C1 N1(C(c2c(C)nsc2N)=O)CCC(C)C(F)(F)C1.C1(C(=O)N)CC(C2CC2)C1 c1(Cn2c(-c3cccc(N4CC(O)C4)c3)ncc2)cc(F)ccc1F N1(CC)CCCC(NC(=O)C(Cc2cnc[nH]2)NC(=O)CC2CCOC2)C1 c1(C(C=O)O)cccc([N+](=O)[O-])c1.CC1(CNC(C2(C)CC2)=O)CC1.N N1(C(c2cncc(N(C)C)n2)=O)CCC2CN(C(c3csc(F)c3)=O)CC12 N#Cc1ccc(CS(=O)(=O)NC2CC2C(N2CCOC3CC23)=O)cc1 C1(NC(=O)C2Cc3ccccc32)CN(C(=O)C=CBr)C2(CCOCC2)C1 c1(C(N(C(C)C2CC2)C)=O)ccc2c(c1)N(C)CC2.CC(CC=O)C(C)(C)C.N C#CCC(C(=O)NC1CC1C(=O)N(C)CCOC)N(C)C=O.C(C)(C)C CCCC(CC)N=c1[nH]c(=NCCc2ccc3c(c2)COC3)c2ccccc2[nH]1 C(CCC(O)C(=O)NCc1nn[nH]n1)NC(C=C(C)C(C)C)=O N1(C2CN(C(C(CSC)O)=O)C2)CC(NC(c2ccnn2CC(C)C)=O)CC1=O C(=O)(C(CCC(C)C)NC(=O)CC1CC(F)C1)NC1CC(C)(CC)OCC1 Cc1cccc2ncc(C(=O)NCC(C)CNC(C3CCC(C)C(C)C3)=O)n12 N1(C(c2nn(C)c3c2CCC3)=O)CCC2(CCN(C(=O)Cc3nc(=N)[nH][nH]3)C2)C1 C1(NC(C2(N(C)C)CCCOC2)=O)CN(C(=O)CC(F)F)Cc2nccn2C1 c1(C(=O)NCC2CN(C(CCc3n(C)cnc3)=O)CC2O)c(F)cc(F)cc1F N#Cc1c[nH]ccc1=NC(CNC(=O)C=C1CCC1)c1ccccc1 C1(CCNC(CCN(C(c2ccc(C)[nH]2)=O)C)=O)CCCC2CC12 c1(N(C(N2CCN(C(C(C)OC(C)=O)=O)CC2)=O)C)ccc(F)c(F)c1 C1(OC)CC(NC(c2cc(Br)c[nH]2)=O)CN(C(C2CC3CCCCC23)=O)C1 C1(C(=O)NCCn2ccc(C(=O)NC3CCCC3CCO)c2)CCC=CCCC1 c1(C(=O)NCCNC(C2C(C)CCS2)=O)ccc([N+](=O)[O-])cc1N.C1CC1.C CCCC(CNC(c1ccc(C)s1)=O)NC(=O)CNC(=O)C.C(C)=O c1(CC(N2C(C)CCC(NC(C=CSC)=O)C2)=O)cccc2ccccc12 C1(C(=O)NCC(CNC(CC(C)(F)F)=O)(C)C)Cc2cc(F)ccc2O1 Cc1cc(C(=O)N(C2CCCCC2NC(=O)C2=NNC(=O)C2)C)cc(C(F)F)c1 c1(C(=O)NC(CN(C)C(C2CC2(C)Br)=O)(C)C)ccoc1Br CCC(C)CCCC(=O)NC1CC2CN(C(c3cccc4nccn34)=O)CC12 C1(NC(COC(CC)(C)C)=O)CCOC(C(=O)NC(C)(CSC)CO)C1 c1(C(=O)NC(C)C(CO)NC(C2CCCN2C)=O)coc2c1CS(=O)(=O)C2 CC(C)CCC(C(=O)NCCNC(=O)N(C)C)NC(C1CCO1)=O C1(N(C(=O)Cn2cccn2)C)CN(C(C2CC(C(F)(F)F)C2)=O)CC1F C1(C(=O)NC(C#C)C(C)C)CCCN(C(C2C3CN(C)CC23)=O)C1C C1(C)(CNC(c2ncn(C)n2)=O)CCCN(C(=O)CCc2ccc(O)nn2)C1 CC1(C)CN(C(C23CCCC2CCN3C(=O)C#CC2CCCC2)=O)CC(C)(C)O1 C(C(O)(C=O)C(F)(F)F)NC(=O)OC(C)(C)C.c1(C2CCCC2)ccccc1F N1(C(C(C)SC)=O)CCC(C2CCOCC2)(CNC(c2sccc2C)=O)C1 C1(CC(=O)NCC2CN(C(c3[nH]c(C)c(C)c3C)=O)C2)CCC2(CCCC2)CC1 C1(NC(C2CC=CC(NC(c3cccn3C3CC3)=O)C2)=O)CCc2n[nH]cc2C1 C12CCC(C1)N(C(=O)C=CC1CC1)C2.Cc1nn(-c2ccccc2)nc1C=O.N c1(C(N(C(C)C)CCNC(=O)COc2ccccc2F)=O)ccc2cnnn2c1 CC1CN(C)CC1NC(=O)CC1(C)CCN(C(C2(C#N)CC(=O)C2)=O)C1 Fc1cccc2c1CCC2N1CCN(Cc2ccc3nc[nH]c3c2)CC1 Cn1cc(NC2CC(C(=O)Nc3ccc(Cl)cn3)C2)c(C(F)F)n1 c1(C(N2CC(CNC(CC(CC)SC)=O)C2)=O)cn(C)c(C)c(Br)c1=O c1(C(=O)OC)cc(C(N2CCC(C)C2)=O)ccc1C.C1(C)(C=O)CC1(C)C.C c1(CC)nnc(C)cc1C(N1CCCC(NC(C2(C)CCOCC2)=O)C1)=O C1(C(=O)NC)CN(CC(=O)NCc2ccc(F)nc2C)c2ccccc2O1 [N-]=[N+]=NCCCCCC(=O)N1CCCC1CNC(c1ccc2c(c1)CCCC2)=O C1(C2CCCC2)(NC(C(CN(C(c2c(OC)nsc2)=O)C)C)=O)CC1 C1(C(=O)NCC2CCCOC2c2ccccc2)NCCC12CCCCC2 C(C(C)C)(C(O)C(=O)N1CCCC(C)(C)C1C(N1CC2CC(C1)N(C)C2)=O)OC c1(CNC(C(c2ncccc2F)C)=O)ccc(S(N)(=O)=O)cc1 N1(C(C(Cc2cccc(Cl)c2)NC=O)=O)CCN(C(=O)CC2CC2)C(CF)C1 c1(OC)cc(C(=O)NC2CN(Cc3ccc(OC)cc3)CC2F)c(Cl)cn1 CC1CCC(NC(c2cc(C(N)=O)ccc2F)=O)CN1C(C1C2CCC(=O)C12)=O Cc1ccc(Cl)c(C(=O)NC23CCC(CC2)C3)c1.C1(C#N)(C=O)CC1(C)C.N N1(C(c2cnc(C(N)=O)s2)=O)CC(NC(=O)Cc2cccnc2O)C(C2CC2)C1 C1(=CC(=O)N)CCCCCC1(F)F.c1(SC)ccccc1C(N1CC(CO)C1)=O C1(NC(c2c(C)n(CC(C)C)nc2)=O)C(C)CCN(C(=O)CO)C1C.C1CC1 c1(C(N2C(CNC(c3cncc(N)n3)=O)CC(OC)C2)=O)cnc2c[nH]nc2c1 C1(NC(C2CNC(=O)N2)=O)CC2CCC1(NC(c1cc[n+]([O-])cc1)=O)C2 N1(C(CC(COC)NC(C2(C)CC(=C)C2)=O)=O)CC(=O)N(C)CC1C N1(C(C(n2ccc(C)n2)C)=O)CCC(C)(C)C(CNC(=O)CC(C)(C)C)C1 c1(C=O)cc(C2CC2)nnc1O.C1COCC1.CC(C)(C)COCC(=O)NC C1(NC(C(CSC)OC)=O)CC(CC(=O)NCCc2ccco2)C1(C)C C(=O)(CS(F)(F)(F)(F)F)NCC1CCN(C(C(C)N(C)C)=O)C1 O=C1CC2CCCC2(C(N2CCC(F)(c3ccccc3Cl)CC2)=O)C1 c1(C(=O)NC(C#C)C(C)C)c(CNC(=O)CN2CCSCC2)nnn1C N1(C(C)=O)CCCCC1.C(C(=O)N(CC(=O)N)CC#C)OCCOCC#C C1(C)CCN(C(C2CC2C(F)(F)F)=O)C1.c1(C(C)C)noc(CCC(=O)N)n1 C(C(O)C(=O)NCc1ccsc1C(=O)NCCc1noc(C)n1)=CC C(C(C)(C(F)(F)F)NC(C1COCC1N)=O)OC c1(OCC=C)ccc(Cl)nc1C(N1CC(C(C)NC(C)=O)C1)=O c1(CNC(C2CN(C(C)=O)C2)=O)ccccc1.c1(C(NC)=O)c[nH]c(=N)o1 N1(C(c2n(C(C)C)ccn2)=O)CCC2(CCC2)C(CNC(=O)C=C(Cl)Cl)C1 C(=O)(C(CC(C)C)C(C)C)N1CC(F)CC(NC(c2c(C)nc(Br)o2)=O)C1 N1(C(C(C)SCCCC)=O)CCN(C(=O)CCO)CC1CC(F)(F)F.C1COC1 Cc1cnc2nccc(C(=O)NC3CN(C(=O)Cc4ccnn4C)CC3C)c2c1 CC1(C)OCC(C=CC(=O)NC2CN(C(=O)Cc3cnns3)C(C)(C)C2)O1 CC(C)CC(O)C(=O)N1CC(NC(c2ccc(Sc3ccccn3)cc2)=O)C(F)C1 C1(C(=O)NC(C)CNC(=O)CNC(=O)C(C)(C)C)CCC(C)(C)OC1 N1(C(C(C2CCOCC2)OC)=O)CCC(NC(=O)C(O)CC(N)=O)C(O)C1 Cc1nn(CCC(N2CCCN(C(c3coc(N(C)C)n3)=O)CC2)=O)c(C)c1C Cc1cccn(CC(=O)NCC(C)(F)CNC(C2CC3CC(=O)C2C3)=O)c1=O c1(C(N2CCCC2)=O)ccc(S(=O)(=O)CF)nc1.CC1(C)CC(O)(C(=O)N)C1 CC1CCC(NC(=O)C#CC(=O)N(C)C)CN1C(=O)CC1CCC(C(C)C)CC1 N1(C(CC(C)=C(C)C)=O)CCCC2(CCN(C(=O)COC3CCC3)CC2)C1 C1(CNC(Cc2c(C)nc[nH]2)=O)CCC2(CCC2)C1.C(=O)(CCn1cccn1)N C1(C(N2CC3CCN(C(Cc4c(C)scc4)=O)CC32)=O)CNC(=O)CC12CCC2 N1(C(CC)=O)CCC2(CCCN2C(c2cc(S(N)(=O)=O)c(C)o2)=O)C1.CC=O.N C(N=c1nc(N(CCCCN(C)C)C)c2c([nH]1)CCC2)c1c(CC)nns1 CCCCCC(O)CC(=O)N1CC(O)(C2CCCN2C(c2cc[nH]c2CC)=O)C1 C1(CNC(C=CC2N(C)CCC2)=O)(CO)CCN(C(=O)CCC(F)(F)F)CC1 C(=O)(CC(C)(C)N(C)C(c1conc1C)=O)NCCN(C(C)C)CC CC1C(NC(C2CN(S(C)(=O)=O)C2)=O)CCN1C(c1cnc(O)o1)=O C1(C(=O)NCC(C2CCCN2C(C2(F)CCCC2)=O)(C)C)CC2(C1)CC2F C1(=CC(=O)NC(C2(O)CCN(C(C(CC)(C)C)=O)C2)C)CCC(C)(C)CC1 C12(NC(C(CN(C)C)O)=O)CC1CN(C(c1ccc(OCC(F)F)cc1)=O)C2 Cc1n[nH]c(C)c1C(C)NC(=O)C(CNC(c1cccc(F)c1)=O)N(C)C c1(C(N2CCC(N(C(=O)Cn3cccc3)CC)C2)=O)[nH]c(C2CC2)nc1C C1(NC(c2n(CCCC)ncc2)=O)CN(C(=O)CC)CC(F)(F)C1.C(N)(=O)N c1(C(=O)OC)nn(C)nc1C(=O)NC1CCCCC1.C(C(C)C)=CC=O N1(C(CCC(CC)NC(c2ccn(CCC)n2)=O)=O)CCC2(C1)CN(C)C2 C(=O)(C1=CS(=O)(=O)CCC1)NC(CCCCNC(=O)CCC1CCCC1)CO C12(C(N3CC(CN(C)C(c4cc([N+](=O)[O-])n[nH]4)=O)C3)=O)CC=CCN1CCC2 C(C)(CCCCN=c1[nH]cncc1C)NC(c1sc(C)c(O)n1)=O CC1CN(C(C2(O)COC2)=O)CCN1C(=O)CCc1csc(=N)[nH]1 N1(C(CNC(c2c(C)occ2)=O)=O)CCN(C(C2CC=CCC2)=O)CC1C C(=O)(CC(C)C(F)F)NCCOC1CCN(C(c2cnc(SC)s2)=O)C1 c1(C(=O)NC2C(NC(C(CCC)C(C)C)=O)CCC2)cc2cc(Cl)ccc2n1C CC1(C)CC(F)(F)CN1C(=O)CC1CC2(CC2)CO1.c1(C=O)cc(Cl)cnn1 c1(NC(c2c(-c3c(OC)ccc(C)c3)ncc(Cl)c2)=O)cccc(C#N)c1OC C1(OC)CN(C(=O)C=Cc2nccn2CC)CC1.C1(C(=O)N)CC2C=CC1O2 c1(CNC2CC(NC(c3cnc(O)cc3O)=O)C2)c(F)ccc(Cl)c1Br C(=O)(C(C)(C)Oc1ccccc1)NCC(C)NC(=O)COC(F)F c1(CNC(C(COC)C)=O)nc2c(s1)CN(C(=O)C(C1CC1)OC)CC2 C(N=c1nc2cn[nH]c2c[nH]1)C1C(OC)CCCC1(C)C CCCCCC(O)C(=O)NCC(C)NC(C1CC2CCC1C2)=O N1(C(CSC(CC)C)=O)CCCC(N(C)Cc2nc(C(C)C)no2)C1 CC(C)S(C)(=O)=O.C1(C=O)CC12CCOCC2.CC(C=O)NS(C)(=O)=O.N c1(C(=O)OCC)cc(=NC(=O)C2CCC(NCc3cnc(O)nc3O)C2)[nH][nH]1 c1(C(N2C(CNC(CCCOCC)=O)CCCCC2)=O)cc2cn[nH]c2cn1 N1(C(C23CCCC2C3)=O)CC(C)N(C(C2(CCN(C)C)CC2)=O)C(C)C1.C N1(C(CCOC)=O)CC2(CC1C)CC2(F)F.c1(C(=O)N)ccc(C(C)C)nc1C C1(NC(C2CC(OC)C2)=O)CCCC(NC(C2CCN(CC(C)C)C2)=O)C1 N1(C(C(C)(O)C2CC2)=O)CC2(CNC(C3CC(C4CC4)=NO3)=O)CC1CO2 c1(N2C3CC(CNC(C(CC)OCC)=O)CC2CC3)nc2c(C)cccc2o1 CC(=O)C(C)(C)CC(=O)N(C(C)C(=O)NCC1(F)CCN(C)C1)C1CC1 c1(C(=O)NC2CCCCN(C(c3cc(CC)ncn3)=O)C2)ccc(C#N)c(Cl)c1 c1cc(C)c(C(=O)N(CC(O)CN(C)C(c2cc(C3CC3)no2)=O)C)cn1.C c1(OC)cc(C#N)ccc1C(N1CCC12CCN(C)C2)C(=O)NC1CCOC1 Cc1ccnc(C(=O)NCC(N2CCCC2)=O)c1.c12cc(ccn1)C(=O)NC2 Cc1nn(C(C)C)cc1C(C(=O)NCCC1CC1)N(C)CCOC=C N1(C(C(=O)NC(C)C)=O)CCCC1C1CCCN1C(=O)Cn1ccnn1 C(=O)(CCCC(N)=O)N(CCC)CCn1cc(C)cn1 C1(C(C)NC(c2c(C)ncs2)=O)CCN(C(=O)CC2CC3CCC2O3)CC1 c1(C(=O)NC2C(NC(COC(C)C)=O)CC2)cccc(-c2nnco2)c1 N1(C(C2(C(C)NC(C(C)=CC=C)=O)CC2)=O)CCN(CCOC)CC1 C(=O)(C(C)CC(C)CC)NCC1(C)CCCN(CC=CC)C1 c1(OC)cc(CC(=O)NC2CCN(C(c3oc(C)cc3C)=O)CC2F)ccc1C c1(CNC(NC(CCC=C(C)C)C)=NCCCC)cccc2c1OCCCO2 C=CC(C)(C)CC(=O)NC(CNC(c1ccc(-c2ccc(F)cc2)[nH]1)=O)CC c1(C(N(C2CCN(C(=O)C(CO)OC)C2)CC)=O)ccnc(OC)c1 N1(C(c2c(C)cccc2C)=O)CCOC2(CCN(C(=O)C(O)c3ccco3)C2)C1 Cc1c(F)ccc(N)c1C(=O)NC1CC(NC(C2(C)CCC2)=O)C12CCC2 Cc1nc(C)c(C(N2CC(C)(C(=O)NCCC3NC(=O)NC3=O)C2)=O)s1 C1(C(N2CCC(CNC(C=C(CCC)C)=O)C2)=O)CC2CCC1CC2OC C1(NC(CC(CC)C2CCC2)=O)CCN(C(=O)CNC(C2CCCC2)=O)CC1O C(=O)(C(F)C(=O)NCC1(CNC(C2CCC2)=O)CC1)OCC.C Nc1nccn2ncc(C(N3CC4CCC4(CCNC(=O)C4CC4)C3)=O)c12 N1(C(C2C(CC)N(C(=O)C(C)C(O)C(C)C)CCC2)=O)CC2CC(C1)C2(C)C c1(C(C(=O)OC)NC(C2CCCO2)CC)ccc(Br)cc1 c1(C(C)OC)nc(C=O)cs1.c1(C(NC)=O)cnc(C(F)(F)F)s1.C1CC1 C(=O)(CCS(C)(=O)=O)N1CCCC(CN(C)C(c2cncc(C3CC3)c2)=O)C1 C(=O)(C1CCCn2ncnc21)NCC(CNC(c1nsnc1O)=O)O C1(NC(c2cccc(CC)c2N)=O)COC2C(NC(=O)C3=CCC3)COC12 CC1(C)CCC(C)(NC(=O)CN(C(c2ncccn2)=O)C2CC2)C1 N1(C(C2CN(C(C3CC(=C)C3)=O)C3(C2)CCC3)=O)CCc2cccnc2C1 N1(C(=O)Nc2cccc(NC(C)=O)c2)CCOc2cccc(Br)c21 N1(C(Cn2c(C)ccn2)=O)CC2CC(C1)N(C(=O)C(C)n1cncn1)C2 C1(C(=O)NCC(CCCC)NC(=O)COCCF)CC2COCC2C1 C(=O)(C1CCCc2ncc(C)n21)NC1CCN(C(c2c(CC)n(C)nn2)=O)CC1 C1(CC(=O)NC2CC(O)C2)CN(C(c2ccc(-n3cncn3)cc2)=O)CCO1 C=CCCC(C)(C)C(=O)NCC1(OC)CN(C(C2CCSC(C)C2)=O)C1 C#Cc1cc(C(=O)NCCC2(O)CCN(C(C3COC(=O)O3)=O)C2)cc(F)c1 CN1CCC(C)(C(=O)NCCCCNC(=O)CC2CC=CCC2)C1 N1(C(CCCCC#C)=O)CCC2CN(C(=O)CNC(=O)CC)C2C1 CCC(C#N)(CC)C(=O)N1CCCC(O)(CNC(=O)C(C(C)(C)C)OC)C1 c1(NCC2CCN(c3c(C(C)=O)cccn3)CC2)ccc2c(n1)CCC2=O CC1(C)CCCCC1=CC(=O)NC1COCCN(C(=O)CC2CC=CC2)C1 C(=O)C(=O)N=S(C)(C)=O.C1(C(N2CCCC2)=O)CC2C=CC1C21CC1.CO.C C1(C(=O)NCC2CCSC2(C)C)(OC)CCC12CCC2 N1(C(CCC(N)=O)=O)CCCCCC(NC(c2ccc([N+](=O)[O-])nc2)=O)C1 C#CCCCCCC(=O)NCCC1CCN(C(C2CC3(CCO2)CC3)=O)C1 Cc1nc(N2CCN(C(c3cn(CC(F)F)nc3C)=O)CC2C(C)C)cc(O)n1 C1(F)(C(N2CCC(N(C(=O)C#CC(C)C)CC)CC2)=O)C(C)(C)C1(C)C C(=O)(C(C)C(C)COC)NCCCN(C(C=CC)=O)CCC C1(O)(CNC(CCC(=C)C)=O)CCCN(C(C2CC3CC2C3)=O)C1 C1(C(=O)NCCC2(NC(CC(C)C3CC3)=O)CCC2)CC(C)N(C)C1 C1(NC(C(COCC)C)=O)CCN(C(c2c(C)ncn(C)c2=O)=O)CC1(C)C C1(CCNC(c2c(CC)nns2)=O)CCN(C(=O)CC2CCCN2C)CC1(F)F C1(F)(C(=O)NCCN2CCCC(C)C2)CCN(C(=O)C(c2ccccc2)O)CC1 C12(CNC(Cc3c(C)ccnc3)=O)CCCC1CN(C(C1CCC1C)=O)C2 CCC(CC(=O)NCC1CC1C(=O)NCc1ncc(C)cn1)SC C1(C(N(CCNC(C2(CC(F)F)CCC2)=O)CC)=O)CCC2(C1)N=N2 C=C(NC(=O)Cn1cc(C(C)(C)NC(=O)OC)nn1)C(=O)NC(C)C C(=O)(C1=NOC(C)(C)C1)NC1CN(C(COc2ccc(C)cc2C)=O)C1 c1(C(=O)NCCOCCNC(CSC)=O)ccc2c(c1O)OC(C)(C)C2 C(CC(O)C(=O)NC(C)C(=O)OC)NC(C1N(CC)CC1)=O N1(C(C(C#N)C2CC2)=O)CC2CC1C2NC(=O)CNC(N)=O N1(C(C2N(C(Cn3cnc(C)n3)=O)C(C)C2)=O)CCN(C(C)(C)C)CC1 CCC(O)CC(=O)N1CCN(C(=O)CN(C)C(c2cnc(CC(C)C)[nH]2)=O)CC1 CC(C)CC(CC(=O)N1CCN(C)C(C)(C)C1)NC(C1(O)CC(CF)C1)=O N1(C(c2c(OC)csc2)=O)CC(C)(CNC(c2ccccc2)=O)CC1(C)C.S CC1CN(C(c2ccc(N)c(N)n2)=O)CCC1NC(c1cccn(O)c1=O)=O c1(OC)ccc2[nH]cc(CC(=O)OCC(=O)NCC3CC3)c2c1 C1(NC(=O)C2=COCC2)CCCCN(C(C23CC(C(F)(F)F)(C2)C3)=O)C1 N1(C(c2ccc(S(C)(=O)=O)[nH]2)=O)CCC2(CC1)CN(C(C1(F)CCC1)=O)C2 CCCCCCCCC(=O)NC(Cc1ccoc1)C(=O)NC1C=CC(C)(C)CC1 N1(C(COc2c(C)ccc(C)c2)=O)C2CCC1CC(NC(=O)CSC(F)F)C2 N1(C(c2nccc(CC)c2)=O)CC(NC(c2nnsc2SC)=O)CC(F)C1 C1(CNC(CCCCOC)=O)CN(C(c2csc(=NC3CC3)[nH]2)=O)CC(C)(C)C1 c1(CN(C)C)cccc(CN2CCN(C(=O)NCC(F)C3CNC3)CC2)c1 C(N=c1nc(Cl)[nH]s1)c1cncc(OC)n1 Cc1cc(C(=O)NC(c2ccccc2)C(=O)O)c2c(c1)C(C)CCN2 C1(NC(COc2cccc(C#C)c2)=O)CN(C(=O)CC(C)(O)CCC)CC12CCC2 Cc1nc2cc(C(=O)NCCC3CN(C(=O)C=CCF)CC(C)O3)[nH]c2s1 C(=O)(C1=Cc2ccccc2C1O)N1CCC(NC(c2n[nH]c3c2COC3)=O)CC1 CC1CCC(NC(c2ccnc(CO)c2)=O)CN1C(=O)NCCN(C)C N1(C(C(CC=C)OC)=O)CCN(C(=O)Cc2ccsn2)CC1C(C)(C)C c1(OCC)ccccc1C(C1CC1)NC(c1ccc(NC(C)=O)cc1)=O Cc1nc(NCC2CCC(NC(C3CCCC3)=O)C2)c2ccsc2n1.N(C)(C)C Cc1cc(Br)cc(F)c1C(N1CCCC(C)(NC(c2cccnc2)=O)C1)=O Cc1cc(C(=O)N(C)CCNC(c2cccc(OCC(F)F)n2)=O)ncc1Cl CCC(C)C(C(=O)N1CC2(CC2C(=O)NC)C1)NC(c1nocc1C)=O N1(C(C2(CCCC)CC2)=O)CC2(CC(C(=O)NC3CN(CCC)C3)CO2)C1 C(C(C)(C)C(F)F)NC(=NC)NCCC(C)(C)C#N CCCCC(CC(=O)NCCc1ncon1)NC(=O)C(C)(C#N)CC c1(C(N(CCn2cc(C3(O)CCOCC3)nn2)CC)=O)cc2cccnc2[nH]1 C(=O)(N1CCCc2nccn21)c1c(CNC(CC2ON=C(CC)C2)=O)ccs1 CC1C(=O)CC1C(=O)NCCN(C(C1CC(F)C1)=O)CC1CC1 C1(C(=O)NCC2(CN(C(=O)C3=CCCCCC3)C)CC2)Cc2ccccc2C1 C1(CNC(C2C(C)C2)=O)CN(C(c2ccnc(N3CCCC3)n2)=O)CCN1C CC1(C)CC(C(=O)NC2CC(F)(CNC(c3ccc(O)nc3)=O)C2)CCO1 N1(C(C(=O)NCc2ccc(C(C)SC)o2)=O)CCCC(CC(=O)O)C1 N1(C(C2CCOCCN2)=O)CC2C(C(F)(F)F)(CCS2(=O)=O)C1 CC1CCCc2ncc(C(N3CCN(C(C4CCC(C)(C)OC4)=O)CC3)=O)n21 c1(C(=O)NC2CC(F)(CNC(C(CC#C)O)=O)C2)scc2c1OCCO2 Cc1nc(CSCCC(=O)NC2(C)CC2)cs1.c1(C=O)sccc1C(C)C C1(CNC(c2ncncc2Cl)=O)(NC(C2CC(O)C2)=O)CC2CCC1C2 CC1CCCc2c(C(=O)N(CCCNC(C3CNC(=O)N3C)=O)C)cnn21 c1(C(N(C2CCN(C(=O)COCCCF)C2)CC)=O)cc2cc(F)ccc2s1 N1(C(CCCSC(C)(C)C)=O)CCC(O)(CNC(=O)CC2(C)CCCCC2)C1 N1(CC(=O)NC(c2ccccc2)C)CC2CC(NC(C3CCCC3C)=O)CC1C2 [N-]=[N+]=NC1CN(C(=O)CCC2CC2(F)F)CC1NC(=O)CCc1cnoc1 C1(NC(CC(CC)OC)=O)C2CCC1N(C(c1cn(CC=C(C)C)nc1C)=O)C2 c1(C(N2C(CNC(C3C(C)(C)C3(F)F)=O)COCC2)=O)ccnc2ccnn12 C(=O)(C(C)CCCC(C)=O)N1C(C=O)C(C(C)=O)CC1.CCC.C(=O)(OC)N c1(NC(C)=O)ccc2c(c1)CCN(C(=O)NC(CC(F)(F)F)C1CC1)C2 N(C(=NCCC1OCCC1(C)C)N(C)CCn1cc(Br)cn1)C(COC)C c1(C(N(C(CCNC(C(C)n2ccnc2)=O)C)C)=O)cc(F)cc2ccncc12 C1(C(=O)NCc2cncc(O)c2)COC2(C1)CN(C(=O)CCc1ncccn1)C2 C12(NC(c3c(Cl)ccc(C)c3)=O)CCCN(c3ncc(I)cn3)CC1C2 C1(NC(c2cc(SC)oc2)=O)CC2CCC(C1)N2C(c1c(C)cc(F)cc1C)=O c1(C(CC)C(=O)N2CCCC2CN(C)C(C2CC(CCO)C2)=O)cccc(Cl)c1 CC1CN(C(C2(NC(C3CCC4(CCC4)C3)=O)CCSC2)=O)C(C)C1C C(C1CCc2ccccc21)N(C(C(C1CCCC1)OCC)=O)C Cc1ncc(C(N2CC(NC(=O)C(C3CC(F)(F)C3)O)C(C)(C)C2)=O)cc1C#N N12CCCC(C(F)(F)F)(C1)N(C1CCC1)C(=O)C2.c1(C(=O)O)ccc(Br)cc1 N1(C(CC(C)CNC(c2ccc(C3CC3)cc2)=O)=O)CCCC2(C1)N=N2 C1(CC(N2CCC(F)(CNC(C#CC(C)C)=O)C2)=O)CC(c2ccccc2)=NO1 C1(CN(C(=O)C(CO)NC(N)=O)C)CCCCN1C(c1csnc1Cl)=O CC(C)(C)C(c1ccco1)NC(=O)C(N1CCC(Nc2ccccn2)C1)=O CC1=C(C)CC(C(N2CC3CC2CN3C(C2(F)CCCC2)=O)=O)CC1 CC1(NC(c2ccsc2C#N)=O)CCCCC1C(N1CCC(N2CCC2)CC1)=O c1(C(=O)NCCC2(C)CC2)cccc2ccsc12.C(=O)(C(O)c1cnc[nH]1)N C(=O)(N1CCCCCO1)C1CCN(C(C(C(C)C)NC(N)=O)=O)C1 c1(C(N(CC(=O)NC2CCC(N(C)C)C2)C2CC2)=O)ccc2cc[nH]c2c1 n1(CC(N2CC(NC(CCC(C)OCC)=O)C(C)C2)=O)cc(C#N)c(O)nc1=O CCC(COC)C(=O)N(C)CC1CCN(C(c2ncoc2C2CC2)=O)CC1 N1(C(C(CC)O)=O)CCN(C(c2scc(C)c2Br)=O)C(CCO)C1 c1(C(=O)NC2CCC(CNC(c3c(C#C)c[nH]n3)=O)C2)cc(F)cc(Br)c1F CC1CN(C(=O)CCC2CCC(=O)N2)CC2(CCN(C(=O)CCC(N)=O)C2)O1 N1(C(C2CCC(C=O)C2)C(=O)NCCOC)CCC(O)C1.C(C)(C)C.O C1CCC(C)N(C(C2CC(N(C)C)C2)=O)C1.c1(SC)ccc(C(=O)NC)cc1 S(=O)(=O)(c1cnc(NCC2(C)CSC2)cc1C)NC1CCN(CC)CC1C N1(C(C(C)(C)N(C)C)=O)CCOC(CC(=O)NCC2CCCO2)C1 N1(C(c2ccccc2Br)=O)CCCCC1CNC(C1(O)CCOC1)=O C1(C(N2CC3C(CNC(C=Cc4c(C)ncs4)=O)C3C2)=O)CC2(CCOCC2)C1 N1(C(c2c(CC)cco2)=O)CCCC2(CC(NC(c3cc(C)c[nH]3)=O)CO2)C1 C1(C(=O)NC(COC)C(N2CCCN(CCO)CC2)=O)CN(C)CCN1C c1(C(C=O)CO)ccc(Cl)cc1.n1(CC)ncnc1C(=O)N(C(C)C1CC1)C.N N1(C(C(=O)NC(C)C)=O)CCCC(CC(=O)NC2(C)CCCC2O)CC1 C1(C(=O)NC(C)C(CO)NC(=O)Cc2cn[nH]c2)CCCCC12CCC2 C1(OC)CC(C)(C)CCC1NC(=O)C(CC(C)C)NC(C)=O c1(C(=O)NCC2CCN(C(c3c(C)snn3)=O)C2)cnccc1.CC(F)(F)F.O N1(C(c2ncc(OC)cn2)C(=O)NCCC2(C)CC2)CCC12CCC(C)CC2 C(=O)(C(C1CN(C(c2cnns2)=O)C1)OC)NCC(=O)OCC#C C1(COC)(CNC(c2cnc[nH]2)=O)CCCN1C(=O)CCO.C(N)(=O)N c1(CC)c(C(=O)NCCCCNC(=O)COC(C)(C)CC)cccc1C.O Cc1cc(C)c(C(=O)NC(C2CCCN(C(=O)Cn3nccn3)C2)C)cc1Br C1(C(=O)NCCn2c(CC)nnc2)CCCC(C2CC2)O1 N1(C(CCNC(=O)OCC)=O)CCC(CNC(c2cccs2)=O)C1(C)C C=CCCCC(=O)NCC1CCC1NC(c1cncc(C(C)=O)c1)=O Cc1sc(C(N2CC3=C(C2)CN(C(=O)C(O)C2CCC2)C3)=O)cc1[N+](=O)[O-] C12(C(N3CC(NC(c4c(C)cccc4)=O)C(C)C3)=O)CC(C)(C1)OC21COC1 N1(C(CC2N(C)CCCC2)=O)CCC2(CCCC2NC(=O)C=Cc2cnc[nH]2)C1 c1(C(=O)NC(C(C)(C)O)C(=O)NCCCN2CC=CC2)ccn2nccc2c1 C(=O)(CC(O)CC)N1CC(CC=C)(NC(=O)C(F)(F)c2cnnn2C)C1 c1(CC)ncccc1C(=O)OCC1CC2CC2C1 N1(C(Cn2c(C)c(Br)cn2)=O)CCC2C(C1)CN2C(=O)C(C(C)C)C(C)C C(=O)(CC(=O)NCC1CC(NC(=O)CCO)C1)NCC.C1CC1.C C(=O)(C#CC1CCCO1)NC12C(CN(C(CN(CC)CC)=O)C1)C2 c1(C(N2CC(C)(C)C(NC(=O)C(F)CC3CC3)CC2)=O)cc2cccnc2cn1 CP(C)(=O)CCC(=O)N1CC(=O)NCC1C(=O)NCCc1cc[nH]n1 N1(C(CCCCCN(C)C)=O)CC2(CCC(CNC(=O)CCOC3CC3)CC2)C1 O(S(=O)(=O)c1cc(C)cc(C)c1)c1nc(C)c(C#C)c(C)c1I N(C1CCCc2ccc(C)cc21)Cc1cn(C(CC)C)nc1 C1(C(N(C2CC3CCC2O3)C)=O)CN(C(=O)Cc2cncn2C)CC12CC2 N1(C(CSc2n(-c3ccc(C)c(C)c3)ccn2)=O)CCC2(CC1)CCS(=N)(=O)C2 N1(C(c2c(OC)cccc2)=O)CCN(C(=O)C(O)c2cnc[nH]2)CC1CC(F)F CC(C)C(F)(CNC(C1CC2(CC2)C1)=O)C(=O)NCC(C)(C)n1ccnc1 c1(OCOC)ccc(C(N2CCOC(CCNC(=O)C(C(C)C)SC)C2)=O)cc1 C1(CNC(C(C)(C)OC)=O)CC(NC(=O)Cc2ccccc2Br)CC1O N1(C(c2ccn(CC)c2C)=O)CC2(CCCC2)CC1C(=O)O N1(C(CN(C)CC)=O)CCCN(C(=O)Cc2c(Cl)cccc2Cl)CC1C C#CCCC(C(=O)NCC1(C(=O)O)CCC1)NC(C1CC(C)(C)CN1C)=O C(CC1CCc2ccccc21)NC1CCC2CN(C)CC21 CCC1=NOC(C(=O)NC2(CC(=O)NOC(C)(C)CO)CC2)C1 c1(OC)ccc(C(=O)NC(C)C(C)NC(=O)Cc2nc(C)sc2C)c(C)c1 C1(C(N2CC(NC(c3nc(C)n(C)n3)=O)C(C)C2)=O)Cc2ccc(F)cc2O1 N1(C(C(CSC)OC)=O)CCN(C)CC1C(=O)NC1CC(=O)NC(=O)C1 C1(C(N(C)CC2CCN(C(=O)C=Cc3ncc[nH]3)CC2)=O)CCn2cnnc2C1 Cc1cncc(C)c1C(N1CC(OCC(=O)N(C(C)C(C)C)C)C1)=O CCCCCC(C)CC(=O)NCCCC(C)(C)NC(c1cnc(N(C)C)s1)=O N1(C(CC(C)CNC(c2ccc(O)nn2)=O)=O)CCC(F)(F)C(O)C1 C(CCC1CC1)(C=O)NC(c1n(CC#C)ccc1)=O.C(C(C)C)C1CCC1.N c1(NC)ccc(C(N2CCC(C)C2CNC(=O)C(O)C(C)C)=O)cc1 C(CCCCCCC(=O)N1CC2CCC(C1)N2C(=O)CC1CC1(C)C)SC CC(O)CCCCCC(=O)N1CC(NC(=O)COC2CCC2)C(C)(C)C1 O(N=C1CCCCCC1)CC=O.CCCCCNC(C1CCN1S(C)(=O)=O)=O.N N1(C(C(=O)Nc2scc(C)n2)C)CC2CCC(C1)N(C)C2 c1(C(N2CCC(N(C(C)=O)C3CC3)C2)C(=O)N)cc(Br)nn1C.C1CCC(C)C1 C(=O)(C1CCCc2nccn21)N1C(C(C)NC(CCn2c(C)ncc2)=O)CCC1 C1(C(N2CC=C(CCNC(C(C)CO)=O)CC2)=O)Cc2ccccc2CO1 c1(OC)ccccc1Oc1ccc(NS(=O)(=O)CCc2cccnc2C)nc1 C(=O)(C1CCOc2ccccc21)NC1(C2CN(C(C(C)C3CCC3)=O)C2)CC1 c1(C(N2CC3CC(NC(C=CCN(CC#C)C)=O)C3C2)=O)csc2ccccc12 c1(C(N2C(C)(C(=O)NCCSCC)CCC2)=O)cccn2nccc12 C(=O)(C(C(C)C)C(C)C)NCC1CC(OC)CN1C(=O)CC1=CCOCC1 C(=O)(C#CC1CCOC1)NCCC1(O)CN(C(c2c(OC)cccc2C)=O)C1 Cc1cc(Br)ccc1C(N1CC(n2cc(C(NS(N)(=O)=O)(C)C)nn2)C1)=O c1(C(N2CC(N(C(C(n3ncc(C)c3)C)=O)C)C2)=O)cc2c(cnn2C)nc1C C(=O)(C(C(=O)NC1(CCCC(=O)N2CCC2CC(C)(C)C)CCC1)OC)OC C(=O)(C#CC12CC3CC(CC(C3)C1)C2)NC1C=CCN(C(CCC(C)C)=O)C1 C1(F)(C(N2CCC(O)(CC)C2)=O)CCCCCC1.C(C(C)(C)C(=O)N)OC(C)C C(c1ccc(F)cc1F)=CC(N1CCC(NC(CC2ON=C(C)C2)=O)(CF)C1)=O S(=O)(=O)(c1cnc(NCC(C)C(C)C)c(Cl)c1)N1CCC(CC)(CC)CC1 Cc1nc2cc(C(=O)NC3CC3NC(C3CCCC3)=O)cc(Br)c2o1 CCCCC(CCC)NC(=O)C(C)(C1CCC1)NC(c1cscc1CC)=O C=CCCC(C)N=c1cccc(S(=O)(=O)N2CCc3cccnc3C2)[nH]1 C#Cc1ccc(C(N2CCC(C)C(CC(=O)NC3(CO)CC(F)(F)C3)C2)=O)cn1 C#CC1(C(=O)NCC(O)C2CC2)CN(C(c2coc(CC)n2)=O)C1 C(=O)(CCC(C)CN(C)C)NCC1N(C(CC(CC)C2CCC2)=O)CCC1 N1(C(C(C)OCC=C)=O)CCC12CN(C(c1ncc(Br)cc1N)=O)C2 C(c1ccccc1)=C(CC)C(N1CC(NC(=O)CSc2ccccn2)C(C)C1)=O CC(C(=O)NN1CCCC1C(=O)NC(c1ccc(F)cn1)C)n1ccnn1 S(=O)(=O)(c1ccc(NNC(=O)N2CC(S(=O)(=O)Nc3ccccc3)C2)nc1)NC C1(CC(=O)NC(CCCC=C)C)CC2(C1)CN(C(c1nonc1N)=O)C2 C1(NC(c2c(CC)nco2)=O)COC2(C1)CN(CC(C)CC)C2 c1(OC)cc(CN2CC(NC(c3c(C)ccnc3Cl)=O)C2)cc(O)c1OC N1(C(C#CC2(C)CC2)=O)CCCC2CCN(C(=O)C=CSc3ccccc3)CC12 C12CCC(CC1n1cc(C(C)(C)C(=O)O)nn1)C2.CCC(C=O)NC(C)=O.N c1(C(N2CCC(NC(C(C)C#N)=O)C2C)=O)ccc2cc(F)ccc2n1 C1(NC(C(C)(C)CCNC(=O)CCC2CC2(C)C)=O)CN2CCC1(F)CC2 CCC(C)(C)C(O)C(=O)N1CC2COCC2(C(=O)NC(C)CCC(C)C)C1 Cc1ccccc1CC(C)C(=O)N(C)C(c1cn(CC2(F)CCOC2)nn1)C C=CCCCCCCNC(C12CC(C)(CN1C(=O)C#CC(C)C)C2)=O Cc1nc(Cl)ccc1C(=O)N(CC(C)NC(=O)C=Cc1ccc(=N)[nH]c1)C c1(C(=O)NC(CNC(C(C)SCCCC)=O)C(C)(C)C)c[nH]cc(C)c1=O C(C)(C(=O)NC)(C(C)C)OC.C(c1c(C)coc1C)=CC=O.C1CCCCC1 N(C1CCc2cc(Br)c(Cl)nc21)C(C(=O)NC(CCC(C)C)C)=O N1(C(=O)CCc2cc[nH]n2)CCCC2(C1)CN(C(c1ccc(F)cn1)=O)C2 N1(CC(=O)NCC#CCNC(CC2OCC(C)(C)C2)=O)CCCCCC1=O C(=O)(C(C(=O)OC(C)(C)C)C1CC1)N1CCC(NC(c2scc(C)c2)=O)C1 N1(C(C2CN(C)C2)=O)CC2CCN(C(c3ccc(C(F)(F)F)[nH]3)=O)C2C1 C(C#Cc1cncc(C(=O)O)c1)NC(C(CN)N(C)C)=O c1(C(=O)NCCN(c2ccnc(C#N)n2)CC)ccnc2nccnc12 N1(Cc2cn(CC)nc2)CC2CN(C(C34CC5CC(CC3C5)C4)=O)CC2C1 C1(O)(CC(=O)NC2CC(C(N3CCCC3c3ccccc3Br)=O)C2)CCCCC1 Cc1cc(C(=O)NCC2CCC(NC(=O)CSC(C)(C)C)CC2)sc1C C1(CC(=O)NC(C(C)NC(Cn2c(C)cc(C)n2)=O)C)CN2CCN1CC2 c1(C(=O)NCCC(C)NC(=O)CCC2(C)CC2(F)F)ccccc1F CC1CN(C(=O)C=Cc2ccn(C)c2)CC1CNC(c1ccc(Br)cc1)=O C(=O)(C1COc2ccc(Br)cc21)NCCCCNC(CC(C=C)C)=O C1(C(=O)NCC(C2CCC2)O)(NC(C2CCC(OC)C2)=O)CCN(C)C1 c1(N2C3CC(CNC(C4(C5CC5)CC4)=O)C2CC3)ncc2c(n1)COC2 c1(NC(=O)NCc2cc(C)sc2C)cc(C(=O)N(C)C)nc(Cl)n1 N1(C(c2cc(C)c(O)cc2)=O)CCn2cc(C(N3CCSCC3)=O)nc2C1 c1(C(N2CCC(NC(C(CC#C)O)=O)(CC)CC2)=O)ccn2ccnc2c1 C(=O)(CCCCC(=O)c1ccc(F)cc1)N(CCNC(c1c(CC)nc[nH]1)=O)C CC(CCO)C(=O)NCc1ccccc1-n1cc(-c2ccc(C(=O)O)s2)nn1 c1(OCC#N)ccccc1-c1cnc(C(=O)NCCO)nc1.C1CCC(N)CC1.C Cc1nc(NCC2CCCC2NC(c2cccn2C)=O)ncc1[N+](=O)[O-] C#CCC(O)C(=O)NCCOC1CCN(C(=O)C(=Cc2cnn(C)c2)C)C1 c1(C(N(C(CCNC(C(C)OCCC(C)C)=O)C)C)=O)cncc(C#N)c1 Cc1[nH]c2ncccc2c1C(=O)NCCOCCNC(C1SC2C=CC1C2)=O N1(C(c2c(C)c[nH]n2)C(=O)NC(=O)C2CC2)CCN(CCC2CCOC2)CC1 c1(NC(C2CC2NCc2ccc3nonc3c2)=O)cc(F)cc(F)c1Cl CC1CCN(c2ccc(S(=O)(=O)NC3CCCCC3)cn2)CCC1(F)F C(=O)(C1=CCCOC1)NC(CCC)CNC(C1CCCC(O)C1)=O C1(NC(c2cc(CC)oc2C)=O)CN(C(=O)C(C)(C)CSC)CC1C1CC1 c1(C(=O)NC2CCCC(NC(CCCC(=C)C)=O)C2)cnc2c(c1)COC2 C1(NC(C(F)=C(C)C)=O)CN(C(=O)CCc2n[nH]c(=N)s2)Cc2nccn2C1 N1(C(C2(S(N)(=O)=O)CCC2)=O)CCC(C2CCN(C(=O)C=C3CC3)CC2)CC1 CC1(C)CCN(C(C2CCC(=O)O2)=O)CC1C(=O)NCC1CSC1 C(=O)(CC1NC(=O)c2ccccc21)N1CC(N(C(C(=Cc2cnc[nH]2)C)=O)C)C1 C1(C(=O)NCC=CCC(=O)NCCCC(=O)NC)OCCC1(C)C N1(C(C(CN(C(C2CCN(CC)C2)=O)C)C)=O)CC(C)(C)C1C(=O)OC CCCC(C)CC(=O)N1CC(C(C)NC(c2cc(CO)oc2C)=O)C1 c1(C(=O)NC(CCNC(C2N(C(C)=O)CCOC2)=O)C)cc2c(o1)CCCC2 C=CC(C)(O)CC(=O)NC1(C(N2CC3(CCC3O)C2)=O)CC(F)(F)C1 N#CC1CC2(CC(C(=O)OCc3ccc(Cl)cc3I)C2)C1 C1(NC(c2n(C)c(S)nc2)=O)CC1C1CCCN(C(c2ccnnc2Cl)=O)C1 CCCCC(C)(F)C(=O)NC1CC2CC1CN(C(=O)CCC(F)F)C2 CS(=O)c1cccc(-c2ccc(C(N3CC(C)(O)C3)=O)nc2)c1 c1(C(C)C)cccc(C(=O)NCCCC2CCCN2C(=O)CC2CCOC2)c1 c1(C(=O)NCCCN(C(COCCC#C)=O)C2CC2)cc(CC)n(C)n1 CCCC(C(=O)N1CC(N(C)C)C(CNC(C2COCCO2)=O)C1)OC N1(C(c2ncn(C)n2)=O)CCC(CO)C(NC(=O)C(O)CC2CCOCC2)C1 N1(C(CC2C(=O)NC(=N)S2)=O)CC2CCCC1C2CNC(=O)C1=COCCC1 c1(C(=O)NC2CCCN(C(CC(CC)CC)=O)C2)cc(Br)cc2[nH]ccc12 C1(NC(C2ON=C(CC)C2)=O)CN(C(=O)C2=CCCOC2)Cc2nccn2C1 C(=O)(CC(C)C(F)F)N1C(CCC(=O)N(C)Cc2cccc(C)n2)CCC1 C#Cc1cccc(C(=O)NCC2C3CN(C(c4cccc(OC)c4)=O)CC23)c1F N1(C(C(C)CN(C)C)=O)CCN(C(c2ccc(N)cn2)=O)CC1CO N1(C(CCN(C)CC)=O)CC2CCC(C1)C2CNC(=O)C(C)(CC)C(N)=O CCC(C)CCC(=O)N1CCC(CO)(NC(=O)CC23CCCN2CCC3)C1 C1(CC(C)NC(=O)C=CC2CCCO2)CCN(C(=O)C(C)(F)F)CC1 N1(C(C2(C#C)CC2)=O)CCCC2(C1)C(NC(=O)CCCc1nccs1)CCN2C C12(NC(C(=O)N(C)C)=O)CC3CC(C1)CC(C3)C2.C1(C=O)CNC(=O)N1.C C(=O)(C(C)C(C)(F)F)N(CCNC(=O)CC1CC1C1CC1)CC c1(-c2cn(CC(C)NC(C3CC(=C)C3)=O)nn2)cc(F)c(N)c(F)c1 N=c1nc(N2CCN(Cc3nc[nH]n3)CC2)[nH]c(=NCC2(C(F)(F)F)CCC2)[nH]1 c1ccc(C)c(F)c1.C(C)(C(C(=O)NC(CC1CC1)C(=O)N)N(C)C)OC CC12CN(C(c3c[nH]c4nc(Cl)ccc34)=O)CC1CN(C(c1n[nH]cc1F)=O)C2 C=CCC(CC)C(=O)N1CC(CC(N2CC3CC2CS3=O)=O)C(C)C1 C1(C(N(C2(C(=O)NC(CC)(C)CC)CCC2)C2CC2)=O)CCC(N=[N+]=[N-])C1 C1(N(C(C(CC)NC(N)=O)=O)CCSC)CCN(C(=O)COCCF)CC1 CC(C)C(F)(F)F.C1(C=O)CC(=O)N(C2CC2)C1.CCC=O.C(=O)(NC)N CC1(CNC(c2ccc(N)cn2)=O)CCCN1C(=O)CC12CCCC1C2 c1(C(N2CCN(CCNC(CCOC)=O)CC2)=O)cnc2cccnn12 C1(C(=O)NC(c2ccccc2)C)CCN(C(=O)C(N)=O)C12COC2 C1(C(C)(C)O)CCCN(C(=O)C(F)(F)C2CC2)C1.c1(C(C)C)oncc1C(=O)N C(C(CC(F)(F)F)NC(=O)CCC)NC(COCCCC#C)=O.C1CCOCC1.O C(N=c1[nH]c2cccnc2s1)C1CCCC(NC(C(C)(O)C2CC2)=O)C1 C1(C)(NC(C23N(C(CCCC#CC)=O)CC(C2)C3)=O)CCCC(C)(C)C1 Cc1ccccc1-c1nc(-c2cc(C)c(Br)s2)n(C2CSC2)n1 CC1CC(=O)NC1C(N1CCC1)=O.c1(C(N(CC=O)CC)=O)ccccc1 c1(C(C(N2C(Cc3cn(CC(COC)O)nn3)CCC2)=O)(F)F)ncccc1F Cc1nc(C(=O)NCC2CC2)cn1C(F)F.C(C1CCCCC1)=CC=O.N c1(CNC(c2c(I)ccc(OC)c2)=O)cc(C)c(C)cc1OC Cc1ccc(OCC(=O)NC23CC2CN(C(c2cnc(C)cn2)=O)C3)c(C)c1 N1(C(C(CCC)C)=O)Cc2ccccc2C(NC(=O)CC(C)(C)CN(C)C)C1 N1(C(C=CC)=O)CCC2(CC1)CC(NC(C1CCC3C(C1)C3(F)F)=O)C2 c1(C(=O)NCC(CC=C)NC(=O)Cn2ncnn2)cccc2c1CC(=O)N2 c1(C(=O)NCC(C)C)cc2ccncc2[nH]1.C1(C=O)NC(=O)CC1C(F)(F)F C(=O)(C(C(C)(C)C)NC(c1sc(F)cc1C)=O)N(C)Cc1onc(CC)n1 Cc1cc(C(N2CCc3sccc3C2)C(=O)NCC2CCOC2)c(C)cc1Br c1(OC)ccc(C(N2CCN(C(c3cc(N)cnc3C)=O)C3CC23)=O)nc1OC CCCCC(O)C(C)C(=O)NC(CNC(=O)CC1(C)CCCCC1)CO C1(C(=O)NC2(CNC(c3cnc(C)o3)=O)CC2)CCC12CCCO2 C1(C(=O)OCC)CC(F)(C)C1.C1(CC=O)CCC1.C(C)(C)C.C=O Cc1nc(Cl)ccc1C(N1CCC(O)(C(N2CCC(O)C(F)C2)=O)C1)=O C1(NC(C2=C(C)CCC2)=O)CCCCC12CCN(C(C1CCSCC1)=O)C2 c1(C(N2C(C(N3CCC(C)(O)C3)=O)CC3CC32)=O)cc2cccnc2nc1O N1(C(C2(C)CCCN(C(C)C(N)=O)C2)=O)CCCC2(C1)CN(C)C(=O)O2 c1(OCC(N2CCN(C(c3sc(F)cc3Cl)=O)C3C2C3)=O)cccc([N+](=O)[O-])c1 C1(NC(CCOCCC)=O)CCC(NC(=O)C(C)C)CC1 CCC(C)CCCC(=O)N1CC(CNC(c2cc3c([nH]2)CCCC3)=O)CC(C)C1 N1(C(C(CC)n2cncn2)=O)CCC(CO)(CNC(=O)Cc2cccs2)CC1 c1(OC)ccc2c(=NCCC(C)SC)[nH]c(=NCC=CC(C)(C)C)[nH]c2c1 c1cccc(O)c1Cl.C12(C(=O)NCCNC(=O)C(F)(F)F)CC1CN(C)C2 N1(C(C(CC)OC)=O)CCC2CC12C(=O)NC(CN1CCCC1)CO c1(C(N2CC(CCNC(C3C(CC(C)(C)C)C3)=O)C2)=O)cnn2ccsc12 C1(C(C)C)(CC)CC1C(=O)NC.C1CCN1C(C1CC(N(C)C)C1)=O N1(C(CNC(CNC(c2nc(CC)sc2)=O)=O)=O)CCC(C2CCCC2)C1 C=CCC(C)(CC)C(=O)N1CCC(CNC(c2cnn3c2OCC3)=O)C(O)C1 C(C(Cc1ccccc1)C(F)(F)F)NC(=O)NCC12CCC(CC1)C2 c1(C(=O)NCC(CC)NC(C2(C)COC(=O)C2)=O)c[nH]c2nccc(Br)c12 C1(CC)(CC)CCCN1C(c1coc(CNC(c2cn(CC)cn2)=O)c1)=O c1(NC(CC=C)C)ccc(S(=O)(=O)N(C2CCCN(CC)C2)C)cc1Br Cc1oc(C(=O)N(C)CC2COCCN2C(=O)CSc2nnnn2C)cc1CO c1(C(N(CCC(C)NC(CCC(=C)C)=O)C)=O)ccc2c(c1)C(=O)CCN2 S(=O)(=O)(CC(=O)NC(C1CC1)C)NC.C1(CC=O)CC2(CC2)CO1.C c1(CC(N2CC(C)C(CCNC(=O)C=CBr)C2)=O)c(O)ncnc1O c1(NC(C2CC3(CC3)CN2Cc2ccc(Cl)c(F)c2)=O)cnc2ccc(Cl)nn12 C1(C(N2CC(OCC(=O)NCCO)C2)=O)Cc2nccn2C1.CCC(F)(F)F c1(C=O)c(C(F)(F)F)oc(C)c1C.C1(OCC)CC1C(=O)NCCC.N N1(C(CCSCC)=O)CCC2(CC1)CC(NC(=O)CC1CCCCC1(F)F)CO2 CC1CC=C(C(=O)N2CCCC2CNC(=O)C=Cc2ccn(C)c2)CC1 C(=O)(CCCCCNC(N)=O)NC1C(CNC(COC(CC)C)=O)C1 C(CCCCCCC(=O)NC1COCC1NC(=O)C(O)Cc1ccccc1)SC c1(CC)nnc(N2CCCC(CCC3CCCCC3)C2)n1CC(C)C C(=O)(C1Cc2ccc(F)cc21)N(C1CN(C(c2c(C)nc(C)s2)=O)CC1O)C C1(OCCOC)CCN(C(C2CCN(C)C2)C(=O)NCC(F)F)C1 c1(OCC(=O)NCC2CC(NC(c3ccc(C)o3)=O)C2)c(Cl)cccc1Cl Cc1nc(S)sc1CC(=O)N(CC(C)NC(C1(C2CCC2)CCOCC1)=O)C C1(C(N2CC(CN(C)C(C3CNC(=O)O3)=O)OCC2)=O)CC2C=CC1CCC2 O=C(O)C(CC1CC(F)(F)C1)NC(c1ccoc1Br)=O c1(-c2ncn(CC)c2)nc(CCn2cncn2)nn1C1CSC1 N1(C(c2cc(CC)ncn2)=O)CCCN(C(=O)C(CO)N(C)C)C(C)C1 CCCC(CCC)CC(=O)NC1(C)CCN(C(C2(O)Cc3ccccc3C2)=O)C1 CC1CCN(C(C2CC3(C2)CC3(F)F)=O)CCN1C(c1cc2cccnc2[nH]1)=O n1(CC)c(N2CCN(Cc3ccc(F)cc3)CC2)nc2c(N)ncnc12 c1(OC)cc(-c2nc(COC(C)C)nn2-c2ccc(Br)cc2C)cnc1Cl C1(C(=O)NC(c2cccnc2C)C)(CC)CCN(C(=O)CC(C)COC)CC1 c1(CC)cc(=NC2CCCCN(C(=O)Cc3nc(CC)n[nH]3)C2)[nH]c(COC)n1 Cc1[nH]c2c(C(N3CCC(C)(NC(=O)C(C#N)C4CC4)CC3)=O)cccc2c1C N1(C(c2c(CC)ocn2)=O)CCC(C)C(NC(c2cnc(-c3ccco3)s2)=O)C1 c1(CN2CCCC(C(C)(F)F)C2)cc2cc(I)ccc2[nH]1 N1(C(COc2cc(C)on2)=O)CC(NC(C2(C)CCNC2=O)=O)CC12CCCC2 C=CCC(C(=O)N(C1CCCCN(C(c2cc(C)n(CC)n2)=O)C1)C)C(C)C N1(C(=O)CSC(F)F)CCCN(C(C23CC=CCN2CCC3)=O)CC1CO N1(C(CC=C)=O)CCC(C)C(NC(c2ccn(C3CC3)c2C)=O)C1 Cc1csc(C(C)NC(c2coc(CNC(=O)Cc3cn(C)cn3)n2)=O)n1 C1(C(=O)NC(CN(C(COC(CC)CC)=O)CC)C)CCCOCC1 Cc1ccc(C(=O)NC2CCN(C(=O)C(C)P(C)(C)=O)CC2(C)C)cc1C#N c1(N(C2CCN(C(=O)COC3CCCCC3)CC2)CCO)nc(Cl)nc2c1SCC2 c1ccc(C=O)cn1.C(C)CN(C(=O)C)C.C1(C=O)(C(C)C)CC1.CC CC1(C)C(NC(C2CCN(c3ccccn3)CC2)=O)CCN1C(=O)CO c1(CC)c[nH]c(C(=O)NCC(C)(O)CNC(=O)Cc2cnn(C)c2)c1 Cc1ccc(C)c(CC(N2CCCC(CNC(c3cc(=N)[nH]c(Cl)n3)=O)C2)=O)c1 C(=O)C1=NOC(C)(C)C1.c1(C(=O)NCC(C)OC)cncc(C2CC2)c1.N N1(C(C)=O)CC(O)CC1C(=O)NCC1(NC(C2CC(O)C2)=O)CCC1 CCCC(C)CC(=O)NC1CC(CO)N(C(=O)Cc2ncn(C)c2C)C1 c1(C(N2C(CNC(CSCC)=O)C3CCC2C3)=O)cc2c(Cl)ccnc2s1 C1(n2cc(C(C)(C)CO)nn2)CC2CCC1(NC(=O)CSC(F)(F)F)C2 Nc1cc2[nH]c(O)nc2cc1C(=O)Nc1nc2cnc(Cl)cc2s1 C(=O)(CC(C)(C)C#N)N.c1(C(=O)OC)ncoc1CCC(=O)N(C1CCCC1)C N1(C(C2(C#N)CC2)=O)CC2CCC2(NC(=O)COCC(F)(F)F)C1 CCC(C)(C)C(=O)C(=O)N1CC(C2CC2)(C(=O)NC)C1.C1CC(C)(C)CCO1 c1(C(=O)NC2(CNC(C=CC)=O)CC2)nc(OC(C)C)ccc1Cl N1(C(=O)CCCF)CC2CCN(C(C3(c4ccc(Br)cc4)CC3)=O)CC12 N1(C(c2n[nH]c(CC)c2Br)=O)CCN(C(=O)Cn2cnnc2)C(COC)C1 CCCCC(C(=O)N(C1CCCN(C(=O)CCCC(=O)NC(C)C)C1)C)N(C)C Cc1cc(OCC(=O)N)ccc1C(C)C.C12CC(C1)C2.C(=O)C(C)C#N.C N1(C(C(=O)NCCC(CC)(O)CC)C(C)C)Cc2ccccc2C1=O c1(C(N(CCCC)C)=O)[nH]nc([N+](=O)[O-])c1Cl.c1(CC=O)coc(C(F)F)n1.N CCCC(O)C(=O)N1CCC1CNC(C1CCN(C2CCSC2)CC1)=O c1(CN(C(c2ncnn2C)C(=O)NC2(C)CC2)CCC)cccc(Cl)c1 c1(C(=O)NCC2C=CC(NC(CC(CC)O)=O)C2)ccc(C(N)=O)c(Cl)c1 c1(C(=O)NC(C)C(N2CCC(Oc3cccc(C#N)c3)C2)=O)ccc(F)c(Br)c1 c1(C(=O)NCC2(C)N(C(C3C(=C)C3)=O)CCC2)ccc(OC)c2ccsc12 C1CCCN(C(=O)C2=C(Cl)CC2)CC1.C(C)(C=O)N(C=O)CC.C(C)(C)C C(=O)(CCCCCC#N)N(C)Cc1ccc(CNC(C2CC2(C)Br)=O)cc1 N1(C(C2(OC)CCC2)=O)CC2C(C(=O)O)(C1)CS2(=O)=O Cc1ccc(C)c(CNC2CCC(Cl)CC2)c1 c1(CCNC(=O)OC)cn(C2CN(C(C3CC4CCC34)=O)C2)nn1 N1(C(c2c(C)[nH]c(C(C)(C)C)c2)=O)CCC(N=c2ccnc(Cl)[nH]2)CC1C C1(CNC(c2c(C)nc(O)[nH]2)=O)CN(C(c2cnc(Cl)s2)=O)C2CCN1C2 CCCCC(C)C(=O)NCCN(CCOCCO)C(c1ccccc1C)=O C1(NC(c2cc(Br)cs2)=O)CCN(Cc2cc(O)ccc2Br)CC1F c1(C(=O)NCCCCn2cc(CCCSCC)nn2)cc(Br)ccc1Cl C12(C=O)C(=O)C3CC1C2C3.c1(C(=O)NC(C)CCC2CCCO2)cocc1.C CCC(C)C(=O)C(=O)NCC(C(=O)NC1(C)CCCC1(C)C)N(C)C C(CC(C)C)(C(=O)N(C(CC(F)F)C(=O)NCCCCN=[N+]=[N-])C)OC C=C1CCN(C(=O)C(COC)N(C)C)C(C(=O)NCCC2(CO)CCC2)C1 c1(C(N(CCC(C(C)C)NC(C2(C(F)F)CC2)=O)C)=O)ccc2ocnc2c1 c1(CS(C)(=O)=O)ccccc1NC(=O)NCCc1conc1Br C1(CN(C(=O)C(F)CC2CC2)C)CN(C(c2cc(Cl)n(C)n2)=O)CCO1 c1(C(C(=O)NCCCC)N(C(C)CSC)C)cc(F)c(F)c(F)c1F C1(NC(C(C)CBr)=O)CN(C(=O)Nc2ccc(C(F)(F)F)cc2)CC1(C)C CCC(C)(CO)C(=O)NC1CC(OCC(N2CCC23CC(C(N)=O)C3)=O)C1 C1CCC(C2CC2)C1.CCC(F)(F)C1(C(=O)NCC2CC2CC=O)CC1.N CC1(C#CC(=O)NCC(C)(O)CNC(c2cncc(C(C)(F)F)c2)=O)CC1 c1(C(N(C2CCN(C(=O)CCC3CCCC3)C2)C)=O)ccc(=O)oc1 N1(C(c2cc(F)c(O)c(F)c2)=O)CCCC1C1CCCN1C(=O)Cc1ccco1 c1(C(=O)NC(CNC(CC)=O)CCOC)cc(OC)c(Br)s1 N1(C(c2ccc(CC(C)C)s2)=O)CC2CC(NC(=O)C=CC3CCCCC3)C2C1 N1(C(C)=O)CC2CC1CC2NC(c1csc(Cc2cccc(Cl)c2)n1)=O N(C1CCCn2cnnc21)C(C1N(C(C(C)N2CCCC2)=O)CC(N=[N+]=[N-])C1)=O c1(N(C)C)nccc(=NC(=O)C2CC(NC(C3CNC(=O)C3)=O)C2)[nH]1 c1(C(N2CCN(CC(C)(C)NC(C(COC)OC)=O)CC2)=O)c(C)cccc1N C12(NC(c3cnc(-c4ccsc4)cn3)=O)CC3CC(F)(C1)CC(F)(C3)C2 Cc1ccc2c(c1)SC(C(=O)NC(C)(C)C1CC1)C2.C1(C=O)C2COCC12.N C1(CCOCC)(C(=O)N)CCN(C(=O)C(F)CC2CC2)CC1.c1ccccc1 N1(C(C(c2ccoc2)NC(C2C(=C)C2)=O)=O)CCCN(C=O)CC1 c1(C(N2CC3C(C)C3C2)C(=O)N(C(C)C)C=O)cccc(F)c1.C(C)(C)C C1(C)(C(N(CC(C)C(=O)NC2(CCO)CCC2)C)=O)COCCO1 N1(C(c2cc(Br)c(Cl)s2)C(=O)NCC=C)CC(C)OC(C)(C)C1C c1(OC)cccc(CCC(=O)NCC(C)(C)C)n1.C1(C=O)(C(N)=O)CCC1.N c1(CC(N2CCC(CN(C(C3(CC)CCCC3)=O)C)C2)=O)ncn(C)c1C c1(C(=O)NC(C(C)C)CCN(C)C(C2CC23CCC3)=O)ccnc2c1ncn2C C1(C(=O)NC2(C)CN(C(C(CCC)OCC)=O)C2)CC2COCC2C1 c1(C(N2CCCCC(CNC(C34CCC3C4)=O)C2)=O)c(F)ccc(F)c1Cl c1(C(c2n(C)nnn2)NCc2cccc(SC(F)(F)F)c2)cc(F)cnc1Cl Cc1conc1CNC(=O)C(=O)N(C1CCCCC1)C C12(NC(=O)CCc3cc(Cl)no3)CCCC1CN(C(c1ccc3c(c1)CC3)=O)C2 C(N=c1cc(Cl)nc[nH]1)C1(O)CCCN(C(c2ccc(C(N)=O)[nH]2)=O)C1 Cc1ncnc(N2CCN(C(=O)NC(C(C)C)C(F)F)CC2)c1F C12(CC(=O)OC)CC3CC(CC(C3)C1)C2.C(=O)NNC(=O)Cc1nc(C)cs1 C(=O)(C1CCc2c[nH]nc21)NC1(C(=O)NCCC#CCC)CCC(C)(C)C1 c1(C(C(=O)NC(CC)C)N(C)Cc2cc(C)ccc2F)ccc2cccnc2c1 c1(C(N2CC3C(CNC(C(C)N(C(C)=O)C)=O)(C3)C2)=O)cc(O)ncc1F C1(OC)COCCC1CC(N1CCC(N(C)Cc2cccc(C(F)(F)F)c2)C1)=O Cc1ccc(C(=O)NC2C3CN(C4CCCN(C)C4=O)CC23)c(F)c1Cl C1(OC)CC(CNC(c2csc(Cl)c2)=O)N(C(C2CCCN(C=O)C2)=O)C1 C1(F)(C(=O)NCCC(C)NC(c2occ(C)c2)=O)CCS(=O)(=O)C1 c1(C(C(=O)N(CC(C)N(C(C=O)=O)C)C)(F)F)nc2ccccc2n1C.CC.N C(=O)C(C)P(C)(C)=O.N1(C(CNCC#C)=O)CCC2CC12.C(C)(C)C.C C(=O)(C#CC(C)NC=O)NCC(C)N(C(=O)CN(C)C)C.C(C)(C)C C(=O)(CC(P(C)(C)=O)P(C)(C)=O)N.CC1(C)CCCC1C(N1CCC(O)C1)=O Cc1ccncc1C(=O)NC(C1CC(NC(=O)C(C)C(F)F)C1)C c1(C(=O)NCC2(C)C(C)CN(C(C(C)CN(C)C)=O)C2)cccc2ccnn12 c1(C(=O)OCC)cccc(C(N2CCOCC2C(=O)N)=O)n1.c1ccc(Br)s1 CCCC(C)C(=O)N1CC(C)CC1C(=O)NC(c1ccc(O)nc1)C c1(CC(=O)N)cc(C(F)(F)F)ccn1.Cn1cc(CC(N2CCC(C)C2)=O)cn1 O=C(C(C(=O)Nc1ccccc1)C1CC1)NCCCC1CCCN1 c1(C(=O)NCC2CN(C(CC(C)N(C)C)=O)CC2O)nn(C)c2ccccc12 N1(C(C2CC2c2ccco2)=O)CCCC(F)(C(=O)NC2CCOCC2)C1 c1(N2CCC3CN(Cc4ncc(C)cc4F)CC32)ncnc2c(C)cccc12 N1(CCC)CCCC1CNC(=O)COCCNC(C1CCC1C)=O C(=O)(C(C)(O)C(C)c1ccccc1)N1CC(CN(C)Cc2ccn(CC)n2)C1 c1(C(N(C(C)CNC(c2cc(C)oc2C)=O)CC)=O)cc(F)c(C)cc1N Cc1c(CC(=O)NC2CC23CC(NC(c2cnc[nH]2)=O)C3)cccc1Br c1(OC)cc(Br)cc(S(=O)(=O)NC(c2ncc(Cc3ccc(Cl)cc3)s2)=O)c1 C1(NC(=O)CN2CC3CC3C2)CCCCCC1NC(c1ccn2c1CCC2)=O NC(CC(F)F)C(=O)NC1COC(C(F)(F)F)C1 n1(CCC(=O)N)cnc2c(cnn2C)c1=O.N1(C(C2(CC)CC2)=O)CCC(O)C1 C1(NC(C2CCC(NC(C)=O)CC2)=O)CCC2CCN(C(=O)C(C)(C)O)C1C2 C1(C(=O)O)CC2(CC2)C1.C1(NC)CCCO1.N#CC(C1CC1)N.C1CC1 C12(C=O)CCCC1(C(N1CCC(CC)C1)=O)C2.C(=O)C(C1CC1)C1CC1 c1(CC(=O)NCC(C)NC(=O)C(=O)NCC(F)F)cccs1 Cc1ccc(C(=O)N)c(N)c1C.C1(CC=O)CC12CC2.C1CC1.CC=CC CCCC(CC(C)C)C(=O)NCC1(NC(=O)C(=Cc2cn(C)nn2)F)CCOC1 OC1CC2CC1CC2CNC(c1ccccc1)CNc1ccccc1 CCC(CC(=O)NCC1(C)CCCC1)CC(F)(F)F.C1(C(=O)N)CCC(=O)C1 N1(C(CC(CCC)O)=O)CCC2CCN(C(c3csc(C)c3OC)=O)C2C1 C1(CN(C)CC)CCN(c2nnc(C3C=CCC3)n2C)CC1 Cn1ncc(Cl)c1C(=O)NCC(O)C(N1CCCC(CF)C1)=O C1(C(NOCCOC)=O)CCCC(NC(=O)CN2CCNC(=O)C2)CC1 c1(C(=O)NC(c2cc(OC)c(OC(F)F)cc2)C)ccc2cnoc2c1 c1(C(C(N2CC(CNC(C3CCCC(N(C)C)C3)=O)C2)=O)O)ccc(Cl)cc1Cl C1(C)CC(F)(F)CN1C(=O)C(F)=C1CCCC1.C1(CC)CC1C(=O)N.C C1(F)(CNC(c2cnc(C)[nH]2)=O)CCC(NC(C2CCS(=O)(=O)C2)=O)C1 N1(C(=O)OC(C)(C)C)CC(CNCc2c(F)cc(Cl)cc2F)OC(C)(C)C1 n1(CCCC)nc(C(=O)NC2CN(C(C3CCSC(C)C3)=O)C2)ccc1=O C1(C(=O)NC(CC=CC)C(=O)NCC(O)CCOC)CC(C)(C)CCO1 C12(C(=O)OC)CCCC1(C(=O)NC1CCC1)C2.c1(C=O)sc(=N)[nH]c1C.N c1(CC)c(C(=O)N(C2CCCN(C(C3CCCCS3)=O)C2)C)[nH]c2ccccc12 c1(C(=O)NC2CCN(C(c3cccc(Br)n3)=O)CC2F)cc(Br)cc2[nH]ncc12 C=CC(O)(C(=O)NCC(CC)NC(c1cccs1)=O)C(F)(F)F c1(C(=O)NC2C(NC(COC(C)=O)=O)CC2)cc(-c2cc[nH]n2)ccc1F Cn1cc(Cl)c(C(N2CC=CC2CNC(=O)C=C2CCCC2)=O)n1 c1(C(N2CCN(C)CC2Cc2ccccc2)=O)c(N)n(C)c(=O)n(C)c1=O C(=O)(C1c2c[nH]nc2CN1C(=O)C(CCC)C(C)C)N1CCCC(C#C)(O)C1 Cc1nnc(N2CC3CCC(NC(C4CCC(C)CC4)=O)CC3C2)c(C#N)c1C C(=O)(C1CCCn2nccc21)N1CCC(F)(CNC(C2C3COCC23)=O)CC1 C1(C)(C(=O)NCC(C)C)CC(O)CN1C(=O)CC1COCCOC1 Cc1cc(Cl)cc(CN2CCCC(CNC(=O)C(CO)c3ccccc3)C2)c1O c1(OC)cccc(F)c1C(N1CC2CC1CN2C(=O)CCC1CCOCC1)=O CC(C)CC(O)C(=O)N1CCN(C(=O)CCCn2cncn2)C(CF)C1 C1(NC(C2CCC3CC23)=O)CN(C(=O)CCc2nnc(-c3ccsc3)o2)CC1O N1(C(C=CC(=O)OC)=O)CC2CCC1C(C(=O)NCCc1ccc(Br)s1)C2 C1(CNC(C(C)Cc2ccncc2)=O)CCN(C(=O)Cc2cccc(F)c2)CC1 CC1OCCC1(F)C(=O)NC1CN(C(=O)COCC(F)(F)F)C1 N1(C(C)=O)CC(O)CC1C(=O)N.C1CC(C)N(C(c2cn(C(C)C)cn2)=O)C1 C1(C(=O)NCC2C(CC(N3C(CC(C)C)CC3)=O)C2)CCN(C)CC1 c1ccc(Cl)cc1.CC1CCC(CC(=O)NC23CC(C2)C3)C1.C(=O)(C)N.C C(CC)C(C)CNC.n1(CCC)ccc(C(N2CCCC2C2(C=O)CC2)=O)n1 c1(CC)cccc(F)c1C(=O)NCC1(NC(C2CCOC2C)=O)CCCCC1 c1(CN2CCC(C(=O)Nc3ccc(C)c(Br)n3)C(O)C2)cccc2cc[nH]c12 C=C=CC(C)C(=O)N1CCC(N2CCN(C(c3ccncc3O)=O)CC2)CC1 c1(C=O)ccc(F)c(N2CCOCC2)c1.C1(C(=O)N)(COC)COC1.C(C)C c1(N2CCCC(CNC(C)C)C2)nc2cc[nH]c2c(=NCC(C)C(C)C)[nH]1 c1(CC(=O)NCC(C)NC(c2cn(CC(C)C)nc2)=O)cccc(Cl)c1Cl N1(C(C(C)OCCCCCC)=O)CCC(N=c2cc(C)nc(CC)[nH]2)CC1C Cc1ccc(Cl)cc1C(N1CCC(N(C)C(c2ccc(C#N)s2)=O)C1)=O C12(CNC(C3C(=C)C3)=O)CCC(NC(=O)Cc3csc(C)n3)(CO1)C2 C1(N(C(=O)Cn2cnnn2)C)CCC(NC(=O)CC2CC(C)(C)C2)C1 C1(NC(CCCOCC=C)=O)COCCC1(CC=C)OC N1(C(c2c(NC)cnnc2)=O)CC2CCC2(CNC(=O)C(C)COC)C1 N1(C(CC(C)N(C)C)=O)CC2CCC(C1)C2NC(C1CC2(CCCO2)C1)=O c1(C(C)NC(C23CC(OC)C2C3)=O)ccc(C)cc1.c1(C(=O)N)n[nH]cc1F C(=O)(CCCCCOC)N1CC(OC)(CNC(c2cccc(N(C)C)n2)=O)C1 c1(C(=O)N)sccc1S(C)(=O)=O.CN1CC=CCC1CC(N1CC(C)C(O)C1)=O c1(CNC(C2(OC)CCC2)C)cc2c(O)cccc2s1 C#CCCC(C(=O)NCC(Cl)=CCl)NC(=O)CC1CCC(=O)N1 c1(C(N(C2CN(C(COCC=C)=O)CC23CC3)C)=O)sc2cncn2c1C c1(-c2ccc(C)cc2Br)cccc2c1CCCC2=O CCC(C#N)(CC)C(=O)NCc1cc(C)c(C(=O)NCC(C)(C)OC)o1 N1(C(C2(C)CC(F)C2)=O)CC(NC(=O)C(C2CC2)C2CC2)CC2(CCC2)C1 C(CCCC(=O)NC(C1CC(NC(c2sccc2CC#N)=O)C1)C)OC C(CC(C)C)(C(=O)N1CCC(NC(=O)CCc2nccs2)CC1)NC(C)=O CCC(C)C(C(=O)N1CC(CNC(=O)CN(C2CCCC2)C)(O)C1)N(C)C c1(C(C(=O)N)(F)F)cc(F)ccc1F.CC1(NC(=O)CC2CCOC2=O)CCC1 CC1C(NC(c2cnn(C3CCC3)c2)=O)CC2CCC1N2C(c1ccoc1Cl)=O c1(C=O)ccc(C#N)cc1C.Cc1cccc(C(F)(F)C(=O)NCC2CC2)c1.N C(=O)(C1=NOC2COCC12)NCCCCC(=O)NCC1CCCC12CC2 C(=O)(C(CCC(N)=O)NC(c1cccc(F)c1Cl)=O)N(C)CCc1nn[nH]n1 c1(OC)cc(C(=O)NCC2(C)CC(NC(=O)C)C2)ccn1.c1nccn1C c1(C(=O)NC2CCN(C(C3N(CCC)C(=O)CC3)=O)CC2)cc(C)cnc1OC c1(CC(=O)NCCNC(c2ncoc2C2CC2)=O)ccc(S(N)(=O)=O)s1 c1(CNC(C(CC)(C)C)C)cnc2c(C(N)=O)cnn2c1 Cc1cn(-c2ccccc2)nc1C(=O)NC(C)(C)CCNC(C12CCC1C2)=O C1(CNC(C2C(OC)CC2)=O)CC12CCN(C(c1ccnnc1)=O)CC2 C#CCC(C)(C(=O)NCC1CC2C=CC1CC2)NC(=O)C(O)CC(C)C CC(C)C(C)CC(=O)NC(c1ccccc1F)CNC(=O)C(C)(C)C#N N1(C(CN2CCCC(CC)C2)=O)CCCC(CO)(NC(c2ccccc2F)=O)C1 c1(-n2c(-c3c(C)nc[nH]3)nc(COc3cccc(F)c3)n2)cccc(C#N)c1 c1(C(=O)NCC2(OC)CN(c3ncnc(CC)c3F)C2)coc2c1C(O)CCC2 c1(C=O)ccnc(C)c1.C(=O)(C(C)CNC(=O)C(C)N(C)C)OCC.N N1(C(CCCCCn2cc(C(C)(C)C)nn2)=O)CC2(C)COCC2(C)C1 c1(N(CCCN(C(C(C)n2cccn2)=O)C)C)nc2ncc(Cl)cc2o1 C1(CC(N2CC3CNC(C3)C2)=O)NCC2CCCC12 C(C(CC(C)C)NC(C1CC(Cl)(Cl)C1)=O)NC(C(n1ccc(C)n1)(C)C)=O C(CCCCCNC(=O)C(CO)NC(N)=O)N(C)C(c1cc(CF)on1)=O c1(C(=O)N)nccc(C#N)c1F.C1(CNC(CCOCCOC)=O)CCCC1 Cc1scc(C(=O)NC(C2CCCC2)CO)c1Br N(C(=NCCCc1nccs1)N1CC(C)c2ccccc21)Cc1cc(C)on1 CCC(O)C(C)C(=O)N1CCCN(CCNC(=O)CSc2ccc(Cl)cc2)CC1 c1(C(=O)OC)cc(C(=O)NCC2CCC2)no1.c1(C(=O)N)cc(C)c[nH]1 c1(OC)ccc(C(=O)N)c(O)c1.C12(CC(N3CCCC3)=O)CCC(C)(C1)OC2 N1(C(C2CCN(C(CCN(C)C)=O)C2)=O)CCOCC(CO)C1 Cc1cc(C(=O)NC2CN(Cc3cccc([N+](=O)[O-])c3)CC23CC3)c(F)cc1F C(=O)(CCC(F)(F)F)NCC1C(CNC(=O)CC2CCC(O)C2)C1(F)F C1(NC(CN(S(C)(=O)=O)C)=O)CCCC1.c1(C=O)csc(C2CC2)n1.C C(=O)(C(C=O)C(C)C)N1CCCCCC1.C1(CC)CN(CC(=O)N)C1.C(C)(C)C c1(OC)cc(C(N2CC(NC(=O)C3=C(C)CCC3)C(F)C2)=O)c(Cl)cn1 N1(C(C2CCCN(C(C)=O)C2)=O)CCCC(C)(C)C1.C(=O)C(C)S(C)(=O)=O.N C1(NC(C2CC(C)(C)OCC2)=O)CCC2(CC1)CN(C(C1(O)CCOC1)=O)C2 C1(C(=O)NCC(CC)CCO)N(C(c2cnn(C)c2OC)=O)CCC1(C)C C1(CC=O)CC2(CC2)CO1.CC1(C(=O)NCCn2ccnn2)CC1(Cl)Cl.C C(c1nc2ccccc2s1)=CC(=O)NCCC1CN(C(C(CCS(C)=O)O)=O)C1 c1(C(N(CCNC(C(CC)C)=O)C(C)C)=O)ccnc2cc(F)cnc12 c1(C(N2CCC(c3nc(C)no3)(CO)C2)C(=O)NCCSC)ccc(F)cc1C C1(CCOC)(NC(c2c[nH]nc2Cl)=O)CCN(C(=O)Cn2cc(CO)nn2)C1 CC1CN(C(=O)COc2c(Cl)cccc2Cl)CCN1C(C1C(C)(C)C1(C)C)=O Cc1ccc(C(N2CCN(CCNC(c3cc(Cl)ccn3)=O)CC2)=O)c(I)c1 N1(C(C(C)(C)SC)=O)C2CCC1C(NC(=O)CNC(c1ccsc1)=O)C2 C1(CNC(C2(NC(=O)CCn3cnnn3)CCC2)=O)CC12CCOC2 C(=O)(CC(F)(F)CC)NC1C(CNC(c2cc(CC)oc2C)=O)CCC1 N1(c2n(CCCOC(CC)C)c(CN3CCCC3=O)nn2)CCC(OC)CC1C N1(C(c2cc(C3CC3)cs2)=O)CC2CCC1CN2C(C1CCCCS1(=O)=O)=O O=C(N=c1cc[nH]c(CCO)c1)C1CN(C(=O)CC2(O)CCC2)CCC1O Cc1cccc(C(=O)NCC(=O)NC2CCCC2NC(=O)C2=CCOC2)c1 C(=O)(C1CCc2scnc21)N1C(CNC(c2cnn(C)n2)=O)CC(C)(C)C1 N1(C(CCNC(C)=O)=O)CC2CCC2(CNC(=O)CC2CCN(C)CC2)C1 N1(c2nccc(=NCCC3ON=C(C)C3)[nH]2)CC2CCN(C)C(=O)C2C1 N(C1CCCc2n[nH]cc21)C(c1ccc(CNC(C(C(C)C)OC)=O)cn1)=O C(c1cncc(O)c1)=CC=O.C1(F)CCC1.C(C)(C(=O)N)NC(CC)=O.C c1(C(N2CC(NC(c3cnc(CC)[nH]3)=O)C(O)C2)=O)c[nH]c2nccc(Cl)c12 Cc1cc(NC(N2CCC(Nc3ccc(N)cc3)CC2)=O)cnc1O N1(C(C2CN(C)C(=O)C2)=O)C(C(=O)N(C2CCCCCC2O)C)CCC12CC2 C(C)(N=c1[nH]c(N2CCC(c3nncs3)C2)nc2c1CSC2)c1nc(CC)sc1 c1(CC)ccc(CC=O)cc1F.C12CC(C1)N(C(c1csc(C(C)=O)n1)=O)C2.N N1(C(c2cn(CCC)nn2)=O)CCCC2(C)CC12.N(S(=O)(=O)NC)CC=O.N C1(C=O)CCC(=O)CC1(C)C.C1(C)CCCC1.C(C)(C(=O)NC)OCC=C.C N1(C(c2c(C)cn(C)n2)=O)CC(NC(C2(C3CC3)CC2)=O)CC12CCCC2 C(=O)(C1=CC2C=CC1C2)NC1(C)CC(C(=O)NCCc2cscn2)C1 c1(NC(C(=O)N(C)CC2C(C)C2)=O)cccc(N(C)C)c1 c1(OCC)nc(C(=O)N(C2CCN(C(=O)CC(C)c3cccnc3)C2)CC)co1 Nc1cccc(C(N2CCN(C(=O)Cc3ccccc3Cl)C3CC23)=O)c1Cl N1(C(C(F)=CC)=O)CCC2CN(C(c3cccnc3C(F)(F)F)=O)CC2CC1 c1(C(N(CC(CNC(COCCCCCC)=O)O)C)=O)cnc(C)nc1 C(=O)(CCCC(C)NC(C1CC(C)CC(=O)N1)=O)N(CC(=C)C)CC(=C)C C1(c2n(C(C3CCC3)Nc3nccn3C)nnn2)(NC)CCCN(C2CC2)C1 N1(C(C=CCOC)=O)CCC2CCC(NC(c3[nH]nnc3-c3ccnn3C)=O)C12 N1(C(CC)=O)CCN(C(C2(C(C)C)CNC(=O)C2)=O)CC(C)(C)C1.C=CCO C#CCCN=C(NCC1CCC2(C1)CC2(F)F)N1CCC(C2(O)CC2)CC1 C(=O)(CCCN(C)N=O)NCC(CC(C)C)NC(c1cccc2ccsc12)=O C(C1=NOC2CC12)c1nnnn1C1CC1.c1(SC(c2cccs2)C)cccc(N)c1 c1(NC(N2C(c3cccc(C)n3)CCC2)=O)ccc(Cl)cc1C c1(C=O)[nH]nc2ncnc(O)c12.c1(SCC)ccc(C(=O)NC2CCC2)cn1.N N1(CC2(CC)CC2)CC2(CNc3cc(C(=O)OC)no3)CCC1C2 C1(C(=O)N)CCCC2(CCC2)O1.c1(C(C)(C)C)ncc(C(=O)NC2CCCC2)[nH]1 O(C=C(C#N)C(=O)NCC1CCC(NC(C2CCCO2)=O)C1)CC C=CCC(C)(C)CC(c1nnnn1CCCC)NC1CN(c2ccc(Cl)cc2)C1 C1(S(C)(=O)=O)(C=O)CCOCC1.Cn1ncc(C(=O)NC(C)C(C)(C)C)c1Cl c1(C(N2CCC(C#N)(NC(=O)CC3CCOCC3)C2)=O)ccc2[nH]nc(I)c2c1 N1(C(C(C)C(C)O)=O)CC(O)(C2CCN(C(C3(F)C(C)(C)C3(C)C)=O)CC2)C1 C(c1ccncc1)=C(C)C(N1CCC(F)(CNC(=O)Cc2cnn(C)c2)C1)=O c1(OC)cc(C#N)ccc1C(=O)NC1CC(C)C1.C1(C=O)CCC(C)(C)CC1 C1(c2n(CC(=C)C)nnn2)(NCc2nc(C3CCCCC3)no2)COCCC1C c1(C(=O)NC2(C)CN(C(CS(CC)=O)=O)C2)cc2c(Cl)cncc2s1 CC1CN(C(C2CN(C)C2)=O)CC1NC(C1CC2C=CC1O2)=O N1(C(CCC=C(C)C)=O)CC(C)C(C)(C(=O)NCc2noc(C(N)=O)n2)C1 CCC(CC)CC(CNC(=O)NC(C)CCc1ccc(Br)cc1)CC c1(C(N(C(C)CNC(C2CC2(C)C)=O)C)=O)cc2cc(Br)cnc2[nH]1 C1(CNC(C(CC)OCC)=O)C(C)CCCN1C(=O)C1=CCOCC1 N1(C(c2cnc(OC)s2)=O)CCC2C(C1)CN2C(=O)C(C)N1CCC1 N1(C(c2cnn(C)c2F)C(=O)NCC=C)CCC(OC)C(C)C1 c1(C(N2CC3C(CC(=O)N(CC(O)CO)CC)(CC3)C2)=O)cnn2ccccc12 c1(CC)n[nH]cc1CNC(c1cc(CNC(=O)C2CC2)[nH]n1)=O CC1(C)CN(C(=O)CC(C(F)F)n2ccnc2)C(CNC(=O)CO)CO1 CC1CC(CNC(C2CCC2NC(c2coc(C3CC3)n2)=O)=O)CC(C)C1 c1(CNC(=NCC2CC2)NC2CCC2)nc2c(s1)CCCCC2.N1(CC)CCCC1 C1(C(N2C(CC)(CC)CC(NC(C34CSCC3C4)=O)C2)=O)Cc2ccccc2O1 N1(C(C2CN(C)C(=O)N2)=O)CCN(C(C2CSC2)=O)CC1CC1CC1 C1(CN(C)C(C2CC3(C2)CC3F)=O)CCCCN1C(c1cnn(C(F)F)c1)=O C1(C2CCC2)(C(N2CC(C3N(C(C(C)(F)F)=O)CCC3)(O)C2)=O)CC1 n1(CC#C)cccc1C(=O)NCC(C(=O)NC1(CO)CC(C)C1)OC N1(C(c2c(C)cc(C)[nH]2)=O)CCC12CN(C(=O)CC(C)c1cccnc1)C2 N1(C(=O)NC2CCN(c3c(C)cccc3)C2)Cc2cc(Br)ccc2CC1C CC1(CC(=O)NC2(C(=O)O)CC(c3cn(Cc4ccns4)nn3)C2)CCCCC1 C=C(C)CCCC(=O)N1CCN(C(c2cc(Cl)ccc2Br)=O)C(CO)C1 c1(C(N(C(C(=O)NCC(CC)CC)C2CC2)C)=O)ccc2cccnn12 CC(C(=O)N(C)CC1(O)CCN(C(=O)CN2CC3CC3C2)C1)C(F)(F)C(F)F Cc1cn2c(C(N3CC4CC3CN4c3cc(C#N)nc(C4CC4)n3)=O)cnc2s1 c1(CC)[nH]nc(C(N2CCCCC(N(C)C(C3CCSCC3)=O)C2)=O)c1[N+](=O)[O-] C(=O)(C1CCc2cc(Br)ccc21)N(CC(C)NC(=O)CCCN(C)C)CC N1(C(Cn2ccc(C)n2)=O)CCN(C(C2CC(O)C2)=O)C(C)C1 CN1CC(NC(=O)CC2CCN(C(=O)Cn3[nH]cnc3=N)C2(C)C)C(F)(F)C1 N1(C(Cc2cc(OC)no2)=O)CCCC(CCNC(c2n[nH]c(C)c2C)=O)CC1 c1(OC)cc2ccccc2cc1C(c1nnnn1C1CC1)NC1(C)CC(F)(F)C1 CC(N=[N+]=[N-])C(=O)N1CCN(C(=O)CNC(=O)CCn2ccnc2)CC1 c1(N(C(CNC(CC(n2ccc(C)n2)C)=O)C)C)nc(Cl)nc2[nH]ccc12 N1(C(c2c(C)sc(Cl)n2)=O)CCC(NC(c2ccc(F)nc2F)=O)C(C)C1 CC1(CC(=O)NC2CC(CNC(c3ncc(C(F)F)s3)=O)C2)CC1(F)Cl C1(CC(N2CC(CNC(C(C)(C)c3cccnc3)=O)C2)=O)CCC(F)(F)C1 N1(C(C(COC)C)=O)CCC(C)(NC(=O)CCn2nc(-c3cccs3)oc2=O)C1 C(C(=O)N1CCCC(CNC(C2(C)CC=CCC2)=O)C1)(C(C)(C)C)SC C1(NC(c2cc(CNC(c3c(C)cc(C)s3)=O)nn2C)=O)CCC=CCCC1 C(=O)(N1CC(C)(O)CO1)C12CC(NC(c3c(C)nco3)=O)(C1)C2 c1(C(=O)NCC2CCN(C(CC(CC)C)=O)C(C)C2)cnc2[nH]cc(C)c2c1 C1(C(C(=O)NC(CC=C)(C)C)C)CCN(C(=O)CNC(=O)CC(C)C)CC1 CN=c1ccc(C(N2CCC(NC(=O)CCCc3cncs3)C(F)C2)=O)c[nH]1 S(=O)(=O)(c1ccccc1)N(CC(N1CC(C)N(C(C2C=CCCC2)=O)CC1)=O)C C12(NC(=O)Cc3cccnc3)CCOCC1CN(C(c1ocnc1C1CC1)=O)C2 Cc1noc(C(=O)NCc2ccnc(OCCO)c2)c1I c1(N2CC(NCc3cn(CC)nc3)C(F)C2)ncc2cn[nH]c2n1 C1(C(C)(C)CO)CCN(C(=O)C(n2cc(Br)cn2)C2CC2)CC1 C1(NC)CCCC(C(F)F)CC1.c12cnc(cc1OC)[nH]c2=O Cc1cncc(C=CC(=O)NC2(C)CC(NC(=O)Cc3cnn(C)c3)C2)c1 CCCC(C)(CC)C(=O)NC1CCCCN(C(=O)Cc2nc(F)c(F)cc2F)C1 C1(C(=O)NCC(CN(C(COC(CC)C)=O)C)C)CC(c2ccccc2)=NO1 N1(C(CSSC)=O)CCCC2(NC(c3cc4c(C)n[nH]c4cn3)=O)CCCC12 CCCC(C(=O)NCCc1cnc(C)cn1)NC(=O)CC(C)N(C)C C(=O)(CC1C(=O)N(C)c2ccccc21)NCC(CC=C)NC(c1coc(C)c1)=O Cc1cc2occ(C(=O)NCCC3CCOC3)c2cc1C.C(=O)(CC1(C)CC1)N c1(NC(=O)NCC(CC)(C)Cl)c(OC)nc(C)nc1OCC c1(C(=O)NC(C(C)(C)NC(c2n(CCC)nc(C)c2)=O)C)ccc(Cl)cc1C c1(OC)nc(Cl)cc(C)c1C(N1CCN(c2nccnc2-c2nn[nH]n2)CC1)=O N1(C(COCC(C)C)=O)CCN(C(c2cnc3[nH]cncc2-3)=O)CC(C)C1 C12(C(=O)NCc3c(CNC(COCC)=O)cccc3)CCCC1CCC2 C(N=c1[nH]c(=NC2CC(C(F)(F)F)C2)[nH]c2ccsc12)c1c(C)cccc1C Cc1ccnc2nc(C(=O)NC3CCN(C(=O)CS(=O)(=O)N(C)C)C34CC4)nn12 C1(CC=C)(NC(=O)CS(=O)CC)CCN(C(=O)CC2CC3(CC3)C2)C1 c1(C(=O)NC(CSCC)C(=O)NC(C)CCCC(C)C)cccc(C)c1O C1(CC(C)C)(C(=O)NCC2CCN2C(C2CC2c2ccsc2)=O)CCC1 CC(CC1CC1)C(=O)NC1(CCC(=O)N(C)CCC2CCCC2)CCC1 CC#CCC(C(=O)N1CCCC1CN(C)C)NC(c1cc(=N)[nH][nH]1)=O C1(C=O)COC2(CCC2)C1.c1(C(=O)NCCC2CC2)ccsc1C(F)F.N Cc1cc(C)c(S(=O)(=O)N2CCOCC(O)C2)c(C)c1 Nc1ccc(C(=O)NCC2(NC(C3C=CCC3)=O)CC3CCC2CC3)c(F)c1F n1(CC(=O)N(C2CCCN(C(C3C(C)C3)=O)CC2)C)ccc2nc(O)nc(O)c12 Cc1ccc(-n2cc(C3(F)CN(C(=O)C(C)(C)C#N)C3)nn2)cc1Cl c1(C(N(CCOCCCNC(C(CC)(C)CO)=O)C)=O)ncc2[nH]ncc2n1 C=CCC(CC)C(=O)NC(C)(CNC(=O)Cc1cc(C2CC2)nn1C)C(C)C C=CCCCCCCC(=O)N1CCCC(CC(=O)NCC23CCN(CC2)C3)C1 Cc1nc2ccc(N(C(c3cccc(C(N)=O)c3)C(=O)NCCSC)C)cc2s1 c1(C(N2CC(C(=O)Nc3c(OCC)nccc3)(OC)C2)=O)ccc(F)cc1O Cc1cc(C)n(CC(C)Nc2ccc(O)cc2)n1.c12nnnn1NC2CC1CC1 Cc1c(Cl)c(C(N2CCN(C(C3CC(OC(F)F)C3)=O)CC2CO)=O)nn1C O=C(CCCC(F)F)NCC(O)CNC(c1ccnc(N2CCCCC2)n1)=O c1(CCNC(C2CCCCC2)CCC)nnc2n1CCOC2 c1(C(=O)NCC(CC)NC(C2CC(C)C2)=O)c(C)oc2ccc(OC)cc12 C(=O)(C(C)C(C)C)NC1(CCC(=O)N(CC#C)C)CCCC1 c1(C(C)NCCC2(C)CC2(F)Cl)c(F)cccc1Br c1(C(N2C(CC)C(C(=O)N)CC2)=O)cccc(F)c1F.C(C)(C)CCCN(C)C Cc1cccc(C(C(=O)NCc2cccs2)N(C2CCN(C)C2=O)C)n1 C1(NC(CCCCCCC)=O)CCS(=O)(=O)C12CN(C(=O)CC(=O)OCC)C2 c1(C(=O)NC(CNC(c2ccc(C)c(O)c2)=O)CO)n[nH]c2cc(Br)ccc12 c1(CC)nn(C)cc1O.C1CC(C=O)CO1.C(C)(C)(C=CC(=O)N)SC.C N1(C(c2cnc[nH]2)=O)CC(CO)C2(C1)CN(C(c1cnc(O)nc1O)=O)C2 C1(OC)CC(C(=O)Nc2nnc(Br)s2)N(C(=O)CCc2ccco2)C1 N1(C(C(=O)NC(C(C)C)Cc2ccc(Cl)cc2)=O)C2COCC1CC(F)C2 C1(CNC(=O)NCCOCCOC)CC2c3ccccc3C1c1ccccc12 c1(C(=O)NCC(C)N(C(Cc2cncc(C)c2)=O)C)cccc2cccc(F)c12 C1(C(=O)NC2(CNC(c3cnc(=N)[nH]c3)=O)CC2)OC2CCC1CC2 C1(C(N(CCC(C)C)C)=O)CC(NC(c2ccn(C)c2)=O)C12CCC2 N1(C(COc2cn(C)nc2)=O)CCC(C(=O)NC2CCSCC2)C1C1CC1 CC1(C)CC(NC(C2CC(F)C2)=O)CCN(C(c2ccn3cncc3c2)=O)C1 C(=O)(C#CC(C)(C)C)NC1CCC(N(C(c2cc(C(C)C)no2)=O)C)C1 CC1(CNC(=O)CC(c2cccc(F)c2)O)CCCN(C(C2CC2(F)F)=O)C1 Cc1nc2ncnn2c(N2CC(=C(F)C)C2)c1C.C1(CCC(=O)N)NC(=O)NC1=O C1(C)(CCNC(C(C)OCC=C)=O)CCN(C(=O)C(O)CC2CCCC2)C1 C1(NC(=O)CCOCC2CC2)CN(C(C2CN3CCC2CC3)=O)CC2CCCC12 CN1CCCC(CC(=O)NCCN(C(c2ncncc2Br)=O)C2CC2)C1 c1(NC(CC(CNC(C(CC)(C)OC)=O)C)=O)cc(C)c(O)cc1C c1(C(=O)NC2C(C)N(C(=O)CCCC3CC3)CC2)cnc2cc[nH]c2c1 c1(C(N(CC(CNC(c2cn(CC)nn2)=O)O)C)=O)cnc2sc(C)cn12 CCC(CNC(=O)NCCOc1c(F)cccc1Cl)(CN(C)C)CC C1(NC(C2CC(C)C2)=O)COCCN(C(=O)C(N2CCOCC2)C)C1 C(C1CCCCC1)=CC(=O)NC(C1CN(C(=O)C(F)n2ccnc2)C1)C N1(C(C2(C#N)CCC2)=O)CCN(C(c2csc(Br)c2)=O)C2CC12 Cc1nc(CC(N2CCC(N(C(=O)CSCC(C)C)CCO)C2)=O)c(C)s1 N1(C(CCCCCOCC)=O)CCC(C2CC2)C1CNC(=O)C(F)(F)C1CC1 CCCC(CC)CC(=O)NC1CCCCC1NC(c1ccc(NC(C)=O)cc1)=O CCC(O)C(C)C(=O)NC(C)CN(C(=O)C(N1CCOCC1)C)C Cc1cc(-c2nc(CC3CC(F)(F)C3)nn2C(C)C)c2cnn(C(C)C)c2n1 C1(CN(C(c2[nH]cc(CC)c2)=O)C)CC(F)CN1C(=O)CCC1CC1(F)F C1(OC)CCC(C)(C(=O)NC2CCN(C(=O)CC(C)SC)CC2)CC1 C1(NC(c2c(C)onc2)=O)CN(C(=O)NCCCl)CCC1(F)F c1(OCC)ccccc1C(F)(F)C=O.c1(CC=O)csc(C)c1.C(C)CC.N C1(C)(CNC(C2CC(CC)C2)=O)CCN(C(=O)CCc2cncnc2O)C1 N1(C(c2[nH]cc(CC)c2)=O)CCC(C)C(CNC(=O)Cc2cccc(C)c2)C1 C1(OC)CCC12CC(C(=O)NCC(C)(C)C)C2.c1(C(=O)N)cc(C#N)[nH]c1C C1(F)(C(=O)NC(c2nccn2C)CC)CCCN(C(=O)CC(O)CC)C1 N1(C(C(C)C(C)(C)C)=O)CC(NC(c2cncc(Br)c2)=O)CC2(CC2)C1 C=CC(C)(C)C(=O)N1CC(O)(CC)C1.C(=O)C(C)CO.C(C)(C)C.C=O.N C1(C(N(C)Cc2cnc(C)s2)=O)CC=CC(NC(C2COC(=O)N2C)=O)C1 CCC(CC)C(=O)N(CC(O)CNC(c1ccc(Br)o1)=O)C c1cnc2ccc(F)cn12.C1(N(C(C)(C)C)C(c2cccs2)=O)CC(NC=O)C1.C N1(C2CCN(CC=C)C2=O)CCCC(NC(=O)C(C)CCN(C)C)CC1 C12CC(C1)N(C(=O)C=C(C1CC1)C1CC1)C2.C(C=O)N(CCOC)C.N CC(C)CC(O)C(=O)N1CCC(C(=O)NCC(=O)NC2CCOC(C)(CC)C2)C1 C1(NC(CC(c2c(C)noc2C)C)=O)COCCN(C(=O)CCn2cncn2)C1 N1(C(CCSCCCC)=O)CC(O)(C2(C)CC2)C1.c1(CC(=O)N)ccccc1Cl C1(C(N(CCCN(C(C2(CC#C)CCC2)=O)C)C)=O)CCCC1SC CCCCC(=O)C(=O)N1CC(O)C(O)C1CNC(=O)C(CCC)OCC c1(CC(N2CC(C)(NC(=O)Cc3ccoc3)C2)=O)coc2ccc(F)cc12 c1(OC)cnncc1CNC(=O)C(=O)Nc1cccc(Oc2ncccn2)c1 c1(C(N(C(C)CNC(C2(C(C)(F)F)CC2)=O)C)=O)nn(C)c2c1CCC2 C1(C(=O)NCCN(C(=O)Cc2ccc(Cl)cn2)C)CCC2(CC2)C1 c1(C(=O)NCC2(NC(C(C)C3CCCO3)=O)CC2)n[nH]c(C(C)(C)C)n1 c1(C(=O)NCC2CC(NC(CC3CCC(C)C3)=O)C2)cccc2nc(CO)[nH]c12 N1(C(C2C(C)CC2)=O)CCCN(C(=O)C(C)(C)CC2CC2)CCC1 C1(NC(C23CC(C)C2C3)=O)CC2CC1N(C(=O)Cc1ccc(F)cn1)C2 C(N=c1[nH]c2cccc(F)c2s1)C1N(C(C2C3(CC(C)(C)C3)C2)=O)CCC1.[nH]1cccn1 c1(NC(N(CCC(C)NC=O)C)=O)nn[nH]c1C(F)(F)F.C(C)(C)C.O CN1CC(C(N2CCCC(C)(CNC(c3coc(CO)c3)=O)C2)=O)CCC1=O c1(C(=O)NCCCCN(CCCNC(CCC=C)=O)C)c(C)cc(Cl)cc1C C12(CC(=O)N(CCCN(C)C)C)CCC(CC1)OC2.c1cn(C(C)(C)C)nn1 CCC(CO)(C(=O)NC1CCN(CCNC(C2CCCO2)=O)CC1)OC C1CC(C)(C)CN1C(c1ccnc(C(N)=O)c1)=O.CCC(C)(C(=O)NC)OC C1(C(=O)NCC2CC(OC)CN2C(=O)CCC2CC2C)CCCC(C)(C)CC1 C(=O)(C(F)CCC(C)C)NCCC1(NC(c2cc(C)n(C)c2C)=O)CCC1 c1(SCc2nc(-c3cccc(C4CCC(=O)N4)c3)sc2)snc2c(Cl)cccc12 c1(C(=O)NCCC2CC(NC(C=NOC)=O)C2)cccc(NC(=O)OC)c1C c1(COC)cc(C(=O)N(CCC(=O)NCC2CC(O)C2)C(C)C)ns1 C(=O)(C(Cc1ccccc1)C(F)(F)F)NC1C2CN(C(CC(=O)OC)=O)CC21 c1(CCNC(NNC(c2c(C)nc(=N)[nH]c2C)=O)=O)ccc2c3c(cccc13)CC2 C1(C(N2CC(CNC(COCCCC)=O)C3(C2)CC3)=O)CCc2nncn2CC1 CC#CC1CCN(C(=O)C=CC2CCCN2C(=O)C(C)=C2CCCC2)C1 Cc1ccc(C(=O)N)c2c1CCC2.C(=O)(C(O)(C(F)(F)F)C1CC1)N1CCC1.C c1(CC(=O)NCCCN(C(C(C)OCCCC)=O)C)ccc(Cl)c(Cl)c1 C1(O)(CNC(c2cnsc2)=O)CCCN(C(=O)CC2C=CCC2)C1 N1(C(C2=C(C)CC2)=O)CC(CC(=O)NC2CCC(O)C(O)C2)C2(CC2)C1 C1(C(N2CC(N(C(=O)CCc3cccs3)C)C(F)C2)=O)(CC)CC(F)(F)C1 C1(C)(CC)CC1C(=O)NCC(C1CCCC1)C1CCCC1 CCCCC(O)C(=O)N1CC(NC(=O)C(COC)NC(C)=O)C2CC2C1 CC#CCCCC(=O)N1CCN(C(=O)CCC2OCCO2)CC1CO C1(C(=O)NCC2CCN(CCN=[N+]=[N-])C2)CCCC(C(=O)O)C1 N1(C(CC(C)C(F)F)=O)CCC2(C1)CN(C(c1ccc(F)cc1O)=O)C2 C(CC(C(C)(C)C)NC(=O)COC)N(C(C1C(=C)C1)=O)C.c1ccncc1 C12(C(=O)NCc3cc(CC)on3)COCC1CN(C(=O)CC(C)O)C2 N1(C(Cc2cn(CC)nc2)=O)CCCN(C(c2cc(C)n(C)c(=O)c2)=O)CC1C CCCCCCCCC(=O)NCCC1CCCN1C(=O)CC1CC=CCN1C C1(C2(NC(C(C)NC=O)=O)CC2)CCCCN1C(c1n[nH]cc1Cl)=O C1(NC(c2ccnc(C)c2N)=O)CCCCCN(C(=O)CCC2CCC2)C1 c1(C(N(CCCNC(C2CC=C(C)CC2)=O)CC)=O)cc(C)cc(Cl)c1 C1(NC(C2C(C)(C)OCC2)=O)CC2CCC1N(C(C1CC=CCC1)=O)C2 C12(NC(CC)=O)COC(CNC(C3(COC)CCOCC3)=O)(C1)C2 C1(CNC(=O)C(F)n2cccn2)CCN(C(C2(c3cccs3)CCCC2)=O)C1 C(=O)(CCN=C(NCC1CCCC(C)(C)C1)NC1CCS(=O)(=O)C1)NC S(=O)(=O)(c1cnc(Cl)nc1)N1CCCC(C)(C(=O)Nc2n(C)ncc2I)C1 c1(C(N2CCCC(C(CNC(c3c(C)cno3)=O)(C)O)C2)=O)cc(=N)[nH]c(Cl)n1 C=CCC(CC(F)F)NC(=O)C(C(C)(C)C)NC(C1CCO1)=O N1(C(C(C2(OC)CCCCC2)(F)F)=O)CC2CN(C(c3cnns3)=O)CC2C1 c1(N2C3CN(C(C4C(CC)C4)=O)C(C3)C2)nc(OC)c(F)c(C)n1 C1(NC(C(C)n2cncn2)=O)CC(=O)N(C2CN(Cc3cnn(C)n3)C2)C1 C(=O)(C1=CCC2(COC2)OC1)N(C1CCN(c2ccc(OC(F)F)cc2)CC1)C S(=O)(=O)(c1cc(NC(N2CCCCC2c2nc(C)c(C)s2)=O)ccc1O)NC CCCN=C(NCc1ccn(C(C)C)n1)N1CCCC(n2ccnn2)C1 S(=O)(=O)(CCC(=O)N1CCC(NC(=O)CC2(C#N)CCC2)C(CO)C1)NC C1(C(N2CC3CC2(C(N2CC=CC2)=O)C3)=O)CC12CCOC2 c1(CN2CCCC(CC(=O)Nc3c(O)ccc(C)c3)C2)cccc2sccc12 N1(CC(=O)NC2(c3ccccc3)CC(OCC)C2OC)CCN(CC)CC1C#N c1(NCc2ncc(C)o2)[nH]c(=NC2CCCCC2N(C)C)nc2scnc12 C=CC(O)C(=O)NC1(CNC(C2CSCN2C(C)=O)=O)CCOC1 Cn1nc(CC(=O)NC2CC(C)(NC(C3CSCCS3)=O)C2)cc1Cl C(=O)(C(C)CCC(C)(C)C)N1CC(O)(CCNC(c2cccc(OC)c2C)=O)C1 C12(C(=O)NC(COC)CO)CC(CN(C(C3CC(O)C(F)C3)=O)C1)C2 CCCCCCCC(=O)N(C)CCN(C)C(C1CN2CCCN1CC2)=O C(C(C)(O)C)NC(C(=O)NCCOC)=O.C(=O)C(C)Cc1cnc[nH]1.N C1(NC(C2(CCC)CC2)=O)CN(C(c2csc(Cl)c2)=O)CC(C)(C)C1 Cc1c(OC(F)(F)F)cccc1C(=O)NCC(C)(C)CNC(C1CCCS1)=O C12(CNC(C(CCC)C)=O)CCCC1N(C(c1ccc(NCC)cc1Cl)=O)CC2 CC1C2CCCCC2CN1C(=O)C(CNC(=O)CCCF)CC1CC1 CC1CN2CCN1C(C(=O)NCCN1CCCN(C(=O)Cc3cnco3)CC1)C2 N1(C(c2cc(F)ccc2I)=O)CCC2(CCN(Cc3cccnc3F)C2)C1 c1(CC(=O)NC2C(C)N(C(=O)C(F)OC(F)(F)F)CC2)c(F)cccc1F C1(N(C(Cc2c(C)ncs2)=O)C)CCCC(N(C(=O)CSCc2cscn2)C)C1 O=C1NC2(C(=O)NC3CN(C(=O)CCSc4ccccc4)C3)CC3CC1C2C3 N1(C(CCCc2nnc(C)n2C)=O)CC(C)CN(C(=O)CC2(C)CCC2)C(C)C1 N1(C(c2c(C)cccc2)=O)CCC2(CC1)CC2C(=O)Nc1ccc(F)c(C)c1 c1(C(N2CCC(O)C2)C=O)ccccc1CC(F)(F)F.c1(CC)ccc(Cl)cc1.N C1(NC(C(C(COC)C)C)=O)CN(C(=O)C=C(C)C(C)C)CC2(CC2)C1 C(=O)(C(CC(C)C)C(C)C)N(CC)C1CC1.N1(C(C(C)C)=O)CCCC1C=O C1(NC(C(c2cnc(C3CCC3)[nH]2)N(CC)CC2CSCCO2)=O)CCCCC1 N1(C(C2(CNC(CC(CN(C)C)(C)C)=O)CCCO2)=O)C2CCC1CC(F)C2 C1(NC(COC(C)C)=O)CCN(C(c2cc(N(C)C)ccn2)=O)CC1O Cc1sc(N)c(C(=O)N(C)CCN(C(C2CCCCC2O)=O)C(C)C)c1C CC(C)(CS(C)(=O)=O)C(=O)NCCC1CCCN(C(=O)CCc2cccs2)C1 CC(C)CC(C)C(=O)NC1C=CCN(C(=O)CNC=O)C1 n1(C(CC(=O)NC)C2CC2)cnc2c(N3CCC4(CC3)CC4CO)ncnc12 Cn1ncc(I)c1NC(=O)C(=O)NCC(c1ccccc1)(C)F CCC(C(=O)OC)C(=O)NCCCC(C)NC(c1cccc(-c2nnco2)c1)=O N1(C(c2ccc(-c3ccc(C)o3)s2)=O)CCOC(Cn2cc(C(=O)O)nn2)C1 CCC(CC)(CO)C(=O)NCC12CC1CN(C(=O)C(c1ccc(F)cc1)O)C2 CCCC(CCCNC(C1(C(F)F)CCCCC1)=O)NC(=O)Cc1ccc(C)o1 C1(C)(C(N2CCC(CC)(CC)C2)=O)CC(O)CN1C(=O)CN1CCOCC1 N1(C(C(CC=C)(C)C)=O)CCOC2(CCN(C(C3CCOC(=O)CC3)=O)C2)C1 C12(C(=O)OC)CCN(C(=O)NC3Cc4cncn4C3)C1CCOC2 c1(C(=O)NC(CCOC)CNC(C2CC2CN(C)C)=O)oc(C)nc1C C(c1ccc(Cl)cc1)=CC(=O)NC1CCCN(C(C2C(c3n(C)ncc3)C2)=O)C1 C1(CNC(C=CCCC(C)C)=O)CN(C(C2(C)CC3CC3C2)=O)CCC12CCC2 N1(C(CC2(O)CC(C)(C)OC2)=O)CC2CC(C1)CN(C(=O)C(F)C1CCCC1)C2 N1(C(c2nc(OCC)oc2)=O)CCC(O)(C(C)C)C1.c1(C(=O)N)cscc1 Oc1ccccc1C.C1(CCNCC)CCC(OC2CC2)CC1 N1(C(C(C)(C)C2CCC2)=O)CCN(CCCCCNC(c2ccnnc2)=O)CC1 c1(CNC(COCC(C)C)=O)ccccc1.C1(CC=O)CCS(=O)(=O)C1 c1(C(=O)NC2C(NC(C(C)OC)=O)C2)ccc(C2CC2)c(Cl)c1 C(=O)(CCCCCCn1cc(C(C)(C)O)nn1)NC(c1ccc(OC)nc1C)C C1(C(N2C(C(CC)C)CCC2)=O)CC(O)CN1C(=O)C(c1ccn(C)c1)C Cc1cc(O)ccc1CC(=O)NCC(O)CN(C(=O)C(c1cnn(C)c1)O)C Cc1ncc(C(N2CCCC(C(N3CCCCC3C(N)=O)=O)C2)=O)cn1 N1(C(C(Cn2ccnn2)NC(CCC(CC)C)=O)=O)CCC(C)(C2CC2)C1 C1(NC(CCCN(C)C)=O)CC(C(N2CCCCCCC2)=O)C12CCC2 C=CCC(C(=O)N1CCCC(CC(=O)NCC23CC(CO)(CO2)C3)C1)OC c1(NC(=O)CO)cc(F)c(OC(F)(F)C(F)C(F)(F)F)cc1-n1cncn1 c1(C(N2CCN(C(C=C(CCC)C)=O)C3C2C3)=O)cccc2cnsc12 C1(COC)(NC(C2(n3ccnn3)CC2)=O)CN(C(C2CC2(C)SC)=O)C1 CCC(CC)(C(=O)NC(C)C(C)C(=O)NCc1cnc(C2CC2)[nH]1)OC C(=O)(CS(=O)(=O)C1CC1)N1CCC(NC(C2(N(C)C)CCCSC2)=O)C(O)C1 c1(C(=O)NC(C)CCCNC(C23C(=O)C4CC2C3C4)=O)cccc2nccn12 C1(NC(CNC(CCC(C)C)=O)=O)CC2CCC(C1)N2C(=O)CC1=CCCCC1 CC(CS(C)(=O)=O)NC(=O)C(C)(C)CN(C)C(C1CCCC(O)C1)=O C1(Nc2cc(OC)nc(CC)n2)CCC2CN(C(c3cnco3)=O)CC2C1 N1(C(CN(CCC)C)=O)CCC(C2CCN(C(=O)CCc3cc(C)on3)C2)CC1 C(c1ccc(F)c(Cl)c1)=CC(=O)NCC1CC1NC(C12CCC1C2)=O C12(C(=O)NC(CC)CNC(=O)Cc3ccc(Cl)cn3)CCC(C)(CC1)OC2 c1(CC)ccc(F)c(C(=O)N(CC(C)CNC(=O)CCc2ccoc2)C)c1 Cc1ccc(O)c(C(=O)NCCCC(C)(C)NC(=O)Cc2cc(C)on2)n1 Nc1cc(C(N2CCC(NC(C3CN4CCN3CC4)=O)C(O)C2)=O)ncc1F c1(CC(N2CCC(C(C)NC(C3CC3F)=O)C2)=O)ccccc1N1CCCC1 Cc1cc(C)cc(C2=CCN(CC(C3CCOCC3)F)CC2)c1 N1(C(CC2(COC)CC2)=O)CCC(F)C1.c1(C=O)cnn(C(C)(C)C)c1.N CC(CC(=O)N1CCC(C(N2CC(C3CCCO3)C2)=O)C12CCC2)C(C)(C)C c1(OC(C)C)ccc(Cl)c(C(=O)NC)n1.C(=O)C(C)CN(C)C.C1CC1.C C(CC(C(=O)N1CC(CO)CC1CO)NC(=O)C(C)CC)=CC c1(CC(=O)NC2CCCC(NC(c3c(CC)n(C)nc3)=O)C2)cccc(C)c1C N1(C(C(=O)NCCC23COC(CF)(C2)C3)=O)CCOc2c(Cl)cccc2C1 c1(O)ccc(I)nc1Cl.n1(CC(C)OC(=O)CC2CC2)cc(C2(O)CSC2)nn1 Cc1nn(C)c(C(N2CCC3C(NC(c4ccc(C(C)C)o4)=O)C23)=O)c1Br C(=O)(C#CC1CCCCC1)NC1CCCN(C(C(C)OCCC#C)=O)C1C C1(CNC(C2CN(C(C)C)C2)=O)CC(C(N2CCC(C(N)=O)C2)=O)CO1 CC(C(=O)N1CCN(C(=O)CN(C(=O)CS)C)CC1)C(C)(C)O.c1ccccn1 C1(C(N2CC(O)(CN(C)C(C3(C)CC=CC3)=O)C2)=O)(COC)CCCO1 Cc1nc(C)c(C(=O)N)nc1C.C1(CC=O)CCS(=O)(=O)C1.C1(CC)CCC1 c1(NC2C(C)C2)[nH]c(=NCCCC(C)(C)CO)nc2sccc12.c1ccccc1F N#Cc1ccc(N)c(C(=O)OCC2CCCC2(F)F)c1 Cc1ccc(CC(N2CC=CC2CNC(c2cc(Br)oc2C)=O)=O)c(C)c1 Cc1cc(C(=O)NCCCCC(C)NC(c2ccc(F)c(CO)c2)=O)cc(N)c1 CC1CN(C(=O)C(c2ccccc2)N2CCCC2)CC1NC(C1CC(F)C1)=O.C C1(NC(C(=CC2CCCC2)C)=O)C2CC1N(C(C1(C)CC1)=O)C2.C(C)C.O c1(C(=O)NCC2(O)CCN(C(C(=O)N(C)C)=O)C2)cc(O)cc(Cl)c1 C(=O)(C(C#N)C(=O)CC1CCCC1(F)F)Nc1ccc(OCC)c(Cl)c1 N1(c2cc(NC3C(SCC)CCC3)ncn2)CCc2c(C)cccc2C1 C1(C(=O)NCCOc2ccc(Oc3c(C)nsc3C)cc2)Cc2ccccc2S1 C=C(C)C(C)(O)C(=O)NCC1CC(O)CN1C(c1cnc(S)[nH]1)=O Cn1cnc2cncc(C(N3CCN(C(c4cccc(CO)c4)=O)C4CC34)=O)c12 C1(C)(CNC(CCC=CCC=C)=O)COCCN(C(=O)Cc2ccc(Cl)nc2)C1 c1(C(=O)NC(CCF)C(=O)NC2CCC(CCO)CC2)cn2c(n1)CCC2 C1(NC(=O)Cc2c[nH]nc2O)C=CCN(C(=O)COCC2CCCO2)C1 c1(OC)ccc(C(=O)NCC#CCNC(C2(F)CC=CCC2)=O)cc1O c1(C(N(C2CCCNC2)CC)=O)ccc(-c2nn[nH]n2)cc1 Cc1cc(C)c(C(=O)NC2CCN(C(c3cc(O)ncn3)=O)CC2F)c(Cl)n1 C1(CC(N2CC(CNC(c3c(C)cc(CO)o3)=O)OCC2)=O)CCCCC1(F)F c1(C(=O)NCCC(C)N(C(=O)CCN(CC(F)(F)F)C)C)ccc2c[nH]nc2n1 c1(COc2cccc(C=CC(=O)Nc3ccccc3Cl)c2)cc2cccc(F)c2[nH]1 N1(c2n(CC)c(C3CC3Cc3ccccc3)nn2)CC(c2ccsc2)OC(C)C1 C1(NC(CC2CC(=C)C2)=O)CCCC(C(=O)NC2CCC3(CCC3)C2)CC1 N1(C(C(=O)NCCCCc2scc(C)n2)=O)CC(C)C(F)(F)C1 c1(C(N2CCC(NC(CCC)=O)C2)=O)c(Br)c(C)nn1C(C)(C)C n1(CCC)cc(C(=O)NC(C)C(C(C)C)NC(c2cccc[n+]2[O-])=O)c(C)n1 C(C(N=[N+]=[N-])C(=O)NCCCC(C)C)OCC.N1(CC=O)CCN(C)C(=O)C1 c1(C(=O)NC(CNC(C=CCCC)=O)C2CCC2)ccc(C2CCCOC2)cc1 c1(C(N(C)CC2N(C(CCC)=O)CCC2)=O)ccnc(OCC)c1 C(=O)(C1=CC2(CN(C(=O)Cc3ccccc3)C2)OC1)N1CC(CC)OCC1CC C(N=c1[nH]c(=N)[nH]c(=NCC(C)N2CCOCC2C)[nH]1)c1c(C)cc(Br)nc1 CC(C)(CCNC(=O)CCCCCCN)CS(C)(=O)=O CC(C)(C)S(=O)(=O)CC(=O)N1C2CCC1CC(CNC(C1CCCO1)=O)C2 c1(OC)cc2cc[nH]c2cc1C(N1CCC(F)(CNC(=O)CCC(N)=O)C1)=O c1(C(=O)NCCCCC2CCCN(C(CCC)=O)C2)cc(F)cc2nn[nH]c12 c1(CCC)ncoc1C(=O)NCCOCCN(C)C(c1[nH]nnc1C)=O N1(C(c2ccc(Cl)c(F)c2)CNCc2cc(C)c(F)cc2)CC2CCC1C(N)C2 CC1CC(NC(C2(F)CC3(CCC3)C2)=O)CCN1C(=O)C=O.CC(F)(F)F.N CCC(O)C(F)(F)C(=O)N(CC(C)NC(C1(F)CCOCC1)=O)C c1(C2(NC(=O)Nc3ncon3)CCC2)ccccc1OC1CC1 CC1(C(N2CCC(C)(CC(N3CCC(CO)C(O)C3)=O)C2)=O)CC2C=CC1C2 c1(C(=O)NCCCN(C(CC(CC)C(C)C)=O)C)ccc2oc(S)nc2c1 Cc1nc(F)ccc1CNC(C1CCC1(C)C)=O.C(C1CCC1)=CC(=O)N NS(=O)(=O)c1c[nH]c(C(=O)NC2CC(C)C23CCC3)c1.C(=O)C1=CSCS1.N C1(C(=O)NC(=O)C(F)C2CC(NC3CCS(=O)CC3)C2)CCCC12CC2 N1(C(CCCOC)=O)C(C(=O)Nc2cncnc2C)C2CC(F)C1C2 S(=O)(=O)(c1ccc(C#N)c(NC2CC=CC2)c1)NC(C)C(C)n1cncn1 C1(C(=O)OCC)CCC(C)(C(=O)N(C2CCCCC2)C)C1.C(=O)CCC(N)=O C(=O)(C(CC)C(C)C)N(CCCCC(=O)NC(CCC=C)CO)C Cc1ncc(Br)cc1C(N1CCN(C(c2ccc(Br)c(N)n2)=O)CC1)=O c1(OC)ccc(OC)c(CC(N2CCC(Nc3ccc(SC)cc3)CC2)=O)c1 C1(C(=O)NCCC(=O)N(C)C)CC(F)(F)CN1C(=O)CCC1(C#N)CCC1 Cc1cc(F)ccc1C1CCCN1C(c1ccc(Cl)nc1O)=O c1(C(N2CCOCC(NC(=O)CC3CCC(F)(F)C3)C2)=O)cc(F)c(O)c(F)c1 C(C1OCCc2ccccc21)N(C(=O)NCc1c(F)cc(C)cc1F)C N1(C(c2c(OC)ncc(C)c2)=O)CCCC2C1CCN2Cc1cnc(Cl)nc1 c1(OC)cc(Br)ccc1C(=O)NC1CCCCN(C(=O)CC2(CO)CC2)C1 Cc1cncc(C(=O)NC2CCC(NC(=O)C(F)CC3CC3)C2)c1Cl CCC1=NOC(C(=O)NC(CC2CCCC2)C(=O)NCCC(C)(C)CC)C1 CC1=C(C(=O)N2CCC(C)C(CNC(c3scnc3C)=O)C2)CCCC1 N1(C(c2c(OC)c(C)cs2)=O)CCCC(NC(=O)Cn2cnccc2=O)C1C Cc1cc(C(=O)N(C)CC2(C)CC2)cc(Cl)c1.C1(C(=O)N)CCNC(=O)C1 N1(C(c2cncc(C#C)c2)=O)CCC2CCN(C(=O)CC3CCCSC3)CC12 CC1CCn2ncc(C(N3CCCC(N(C(=O)C=Cc4cnc[nH]4)C)C3)=O)c2C1 C1(F)(CNC(c2nn(C)c(C(F)F)c2)=O)CC(N=c2[nH]ccn3nnnc23)C1 c1(NC)cccc(C(=O)NCC(C)(C(C)C)NC(=O)C=CC2CCOC2)n1 N1(C(CN2CCC(N(C)C)CC2)=O)CCC(NC(=O)CS(N)(=O)=O)C(O)C1 CC1CN(C(=O)C(CC(F)F)NC(c2ccn(C3CC3)n2)=O)CC(C)(C)C1 c1(C(N2CC3C(C(=O)Nc4cncc(C)n4)(CC3)C2)=O)cccc2occc12 C12(CNC(C3N(C)CCC3)=O)CCC(CN(C(c3cc(Br)ccn3)=O)C1)C2 N1(C(C2C(C(N)=O)C2)=O)CCN(C(=O)CSc2ccccc2O)C(CC(F)F)C1 C1(NC(CC(CC2CC2)NC(C(C)=CCC)=O)=O)C=CC(C)(C)CC1 C1(NC(=O)CNC(C2CCC2)=O)CCN(C(C2Cc3nncn3C2)=O)CC1F Cc1nnc(CCC(=O)N(C2CCS(=O)(=O)C2)Cc2cccnc2)n1C C1(NC(c2c(CC)ncs2)=O)CN(C(c2csc(C)c2C)=O)CC1C N1(C(C2(C#N)C(C)C2)=O)CC=C(CC(=O)N(C)CC2CCN(C)CC2)CC1 N1(C(C(N2C(=O)CCC2=O)C)=O)CCC(C2(NC(=O)C3=COCC3)CC2)C1 CCCCCC(O)C(=O)NC1CC(CCC(=O)N(CC(C)C)CC(C)C)C1 N1(c2n(CC)c(C(c3cccnc3)C)nn2)CC(C(N)=O)CC(OC)(OC)C1 C(=O)(C(=O)N=S(C)(C)=O)NCC1N(C(C(CC)CO)=O)CC(F)(F)C1 c1(SC(C)C(=O)N(C(C)(C)C(=O)O)C)ccccc1 CC1CC(NC(c2cc(O)nc(O)c2)=O)C(=O)N1c1ccccc1 C(=O)(CCCCCC(C)(C)C)N1CC(OC)C(NC(C2(C)CCCNC2=O)=O)C1 CC(O)(C(=O)NC1CC(CCC(N2CCCC3OCCC23)=O)C1)C(F)(F)F C1(CC)COCC(C(=O)O)N1C(N1CCC(C)(c2nn[nH]n2)CC1)=O.C(C)(C)C CC1CN(C(=O)CCC(F)F)CCC1NC(C1CCN(c2ccccn2)CC1)=O CCCCC(CC)C(=O)N1CCC(NC(c2ccc(O)c(C)c2C)=O)C(CO)C1 c1(C(=O)OCC)c[nH]c(=NS(=O)(=O)c2ccsc2-c2ccccc2)cn1 C(C(C(=O)N(C(C)CSC)C)NC(=O)COCCOC)OCC c1(C(C(=O)NC)N(C)Cc2ccn(CC)n2)cccc(Cl)c1C.c1ccc(F)cc1 c1(-c2cc(C)c(NC(c3c(Cl)ccc(F)c3Cl)=O)nc2)ccn2ccnc2c1 CCCCC(CC)CCC(=O)N1CCN(C(=O)Cn2cc(CO)nn2)C(CO)C1 C1(C=O)CCC2(CCC2)CO1.c1(SCC)cncc(C(=O)NC2CCC2)n1.C Cn1nc2c(c1C(=O)NCc1cn(CCNS(C)(=O)=O)nn1)CCC2 C1(NC2CC(c3ccc(OCC)cc3)C2)COCCN(C)C1 c1(C(=O)NCC2C(C)(C)N(C(c3ns[nH]c3=O)=O)CC2)cccc2nccnc12 C#CC1(F)CCN(C(C2CCCCC2CNC(=O)C(C)(CC)CO)=O)CC1 c1(CC(N2CC(C(C)C)C(C(=O)N)C2)=O)ccc2c(c1)CC2.C1CCC(=O)NC1 N1(CC2CC(C)C2)CC2CCN(C(=O)CNC(=O)C(C)(C)C)CCC2C1 c1(C(n2cc(CC(C)C(=O)NC3CCCCC3)nn2)C)ccc(Cl)cc1 C=CC1(C(=O)NCC(C)N(C(c2ccc(N(C)C)cn2)=O)CC)CCCCC1 c1(CC)nccc(O)n1.c1(C(=O)NC(C=O)c2cccs2)ocnc1C1CC1.N c1(CNC(C2C(NC(C=C)=O)C2)=O)ccncc1OCC(F)(F)F N1(C(CN(C2CC(C#N)C2)C(=O)CCC2CCOC2)=O)CCCC(CCO)C1 C(=O)(C1CC(O)c2ccccc21)NCC1C(NC(=O)Cc2cccc(F)c2F)C1 N1(C(CN(S(C)(=O)=O)C)=O)CCC2(CCCN2C(c2cnc(O)o2)=O)C1 c1(CN(C(=O)C=Cc2ccnn2C)C)cccc(C)c1.C(=O)CCC1CCC1 N1(CCOc2c(F)cc(Br)cn2)Cc2cccc(F)c2C1 N#Cc1ccc(-n2cc(CNC(c3ccc(C(F)F)cc3)=O)nn2)c(Cl)c1 Cc1cc(N)sc1C(N1CCC(c2ccc(O)cc2)C1)=O c1(C(N2CCC(NC(Cc3c(C)n(C)nc3)=O)C(C)C2)=O)nn(C)cc1[N+](=O)[O-] c1(C(=O)NC2CCCN(C(Cc3nn(C)c(Cl)c3)=O)C2)c(F)ccc(N)c1F N1(S(=O)(=O)c2cccc(C(F)F)n2)CC(O)C(O)CC12CCCC2 CN1CC(O)CC1(C)C(=O)NCCCOCCNC(c1cc(Cl)no1)=O CC1CCCCCCN1C(=O)NCC1(C)CNC(=O)O1 N1(C(C(=Cc2ccncc2)C)=O)CCCN(C(=O)C(c2cccc(C)c2)O)CC1 N1(C(C2C(C(C)(F)F)C2)=O)CCC1(C)CC(N1CCCC1C1(C)CC1)=O C1(CNC(C=NOC)=O)CN(C(=O)C=Cc2cncn2C)CC1(C)C c1(C(=O)NCCC2(O)CCN(C(C(COC)C)=O)C2)cc2nc(F)ccc2o1 C(=O)(CS(=O)(=O)CCO)N.c1(C(=O)NC)ccc(C(=O)NC2CCCC2)cn1 c1(N(C)C)cnc(C(=O)OCC2CC(c3ccccc3)OC2=O)nc1 N#Cc1ccc(C(=O)NCC2CC2CNC(=O)CS(N)(=O)=O)o1 C(=O)(C#CC1CCOC1)NC1C(CNC(C=CC=CCCCCC)=O)C1 N1(C(C2CCCS(=O)(=O)C2)=O)CCc2nc(C)sc2C1.C1(O)(C(=O)N)CCC1 CCC(C(C)(C)O)NC(C1(C2CCCN2C(=O)CNC(=O)OC)CC1)=O c1(CNC(=O)NC2CCCN(c3nccs3)C2)ccc2cnsc2c1 C(=O)(CS(=O)CCC(F)(F)F)N(CCC(C(C)C)NC(=O)CCc1ccc[nH]1)C Cc1ccc(C(=O)NC2(CO)CCCN(C(C3CC3C)=O)C2)nc1C C1CCCCCN1C(=O)CC1CC(C)(C)C1.c1(COC)c(C(=O)N)cnn1C CCCC(C)CCCC(=O)NCC(C(C)C)NC(=O)CN1CCCNS1(=O)=O N1(C(C=CCCC)=O)CCC(CC(C)NC(=O)CC(C)n2cccc2)CC1 Cc1ncnc(C)c1C(=O)NC1CCOC1C1CCN(C(c2ccc[nH]2)=O)CC1 n1(CCCC(=O)NCCC2CSCCN2C(=O)C(F)F)c(O)nnc1O c1(CN(C)C)c(C(=O)NCC(O)CCNC(=O)CO)oc2ccccc12 Cc1cc(C(N2CC(O)(C(C)NC(=O)C=Cc3ccsc3)C2)=O)c(C)[nH]1 C(N=c1[nH]c(=NC(C)c2ccc(F)cc2F)[nH]c2c1CCC2)C1(CCOC)CC1 c1(CC(N2CC(CNC(C(C)SC)=O)OCCC2)=O)ncn2c1CCCC2 C12(C(N3CCOCC(F)(CNC(C(C)(C)CF)=O)C3)=O)CCCC(=O)N1CCC2 C12(C(=O)NCCCCN(C)C(c3cnc(Cl)s3)=O)CCC(F)(CC1)CC2 C1(C(N(C)CC2CCCN2C(c2csnc2Br)=O)=O)C2CCCOC12 N1(C(C(C)=C(CC)C)=O)CCCCC12CC(NC(c1cccc3nccn13)=O)C2 N1(C(N)=O)CCCN(C(C2CCN2C(c2cc(O)ncn2)=O)=O)CC1 C1(CNC(Cc2c(C)nccc2)=O)CCC2(CN(C(=O)C3=CCCCC3C)C2)O1 C1(NC(c2n(CC=C)ccc2)=O)C=CCN(C(c2ccnnc2)=O)C1 N1(C(C2CCC(C)O2)=O)CCC2(CC1)CCC2.C1(C)(C(=O)N)CC1C(F)(F)F C1(C)(CN(C(CC=CC=C)=O)C)CCCC1.C1(CC=O)CC(C)(C)CO1.N C1(CC(=O)N(CCC)C)COC(C)(C)CO1.C1(C=O)CC(F)(C=O)C1.C c1(C(N2C3CC(CN(C(CC=C=C)=O)C3)C2)=O)cc(OC)c(F)c(F)c1 N1(C(CCC2C(C)=NOC2=O)=O)CCCC2CN(C(=O)CCF)CCC12 CS(=O)C=CC(=O)NC1CCC(N2CCN(C(C3CC3C#N)=O)CC2)CC1 N1(C(COCCSC)=O)CC2CCC1CN2C(=O)CC1(CSC)CC1 C1(C(=O)OCC)CCCN(C(C(=O)NC2(C)CC2)c2ccsc2)C1 CC(C)CC(Cn1cc(C2CCOC2)nn1)NC(=O)C(C)N(C)C Cc1ccc(C(=O)NC2CC(NC(=O)CN)C23CCC3)c(C)n1.c1ncccn1 N1(C(C)=O)CCN(C(=O)CC2(O)CNC2)C(c2cccnc2)C1 O=C(CCCC(F)(F)C(F)(F)F)NC1C2CCC1N(C(=O)C=C1CCOCC1)C2 C(CCCC)(CC(=O)NC(C)C(C)n1cccn1)NC(c1c(C#C)c[nH]n1)=O C1(NC(C2N(CC)CCOC2)=O)CCC12CN(C(=O)C(C)(C)CCOC)C2 C(=O)(CC1=CCOCC1)N1CC(NC(c2ccc(NC=O)cc2)=O)C(F)CC1 CC(CC(=O)NCC(C)(C)CNC(c1csc(-c2ccccc2)n1)=O)C1CC1 c1(C(=O)NCC#CCNC(COC)=O)ccc(C)c(Cl)c1F c1(C(=O)NCCC)ccccc1Cn1cccn1.C(=O)C(O)Cc1cnc[nH]1.N c1(C(=O)NC2CCN(C(c3cc(C)ncn3)=O)CC2CO)cc(C)c(Cl)c(C)c1 CN1CCC2CCN(C(=O)C(F)CC(C)(C)NC(=O)C=CC3CCOC3)C2C1 C1(C(=O)NCC(COCC)C)CC12CCN(C(C1CC1Cl)=O)CC2 c1(CC(N2CC(CN(C(C(C)CC3CC3)=O)C)OCC2)=O)c[nH]c2ccccc12 C1(C)(CNC(C(C)(C)SC)=O)CN(C(c2nc(C)sc2C)=O)C(C)(C)C1 c1(C(=O)NCC(C)N(C(C(C)CO)=O)C)cccc2[nH]cc(C#N)c12 C(=O)(C(F)(F)CO)N.N1(C(C2CN(C(C3CCCCC3)=O)C2)=O)CCC(C)C1 C1(NC(C2(OCC)CCCC2)=O)CCN(C(=O)C=C(C)C)C(C)C1 C(C)(CN=c1[nH]n2cc(C)nc2s1)N(C(C(c1c(C)cccc1)(C)C)=O)C Cc1ccc(C(=O)NC(C)C(CO)NC(c2nccnc2O)=O)cc1C c1(CN2CC(F)CC(C(=O)N=c3[nH][nH]cc3Br)C2)ccc2c(c1)OCCO2 N1(C(CNC(C2(C)CC3CCC2C3)=O)=O)CCN2CCC1CC2 C12(CNC(c3cnc[nH]3)=O)CCCC1N(C(c1nc[nH]c3nccc1-3)=O)CCC2 c1(CC)ccc(C)c(C(N2CCCC2C)=O)c1.C1(CC(=O)N)CC2(CC2)C1 Cc1c(C(N2CCC3(CC2)CC3NC(=O)C2CC2)=O)cc(C(F)(F)F)cc1N c1(C(N2CCCC(C)C2)=O)cc(S(N)(=O)=O)c[nH]1.C(=O)(CCC(=O)N)NC.C N1(C(C2OCC(C)(C)OC2)=O)CC2CN(C(C3CCCC3)=O)CC2(C(F)(F)F)C1 Cc1ccc(C)c(C(N2CC(C(=O)NC)C(C)(C)C2)=O)c1.C1CC12CC2(F)F C1(C(=O)NC2(C)CCN(C(c3cc(C(C)C)n(C)n3)=O)C2)Cc2nncn2C1 c1(C(C)OC(c2ccc(C3CCCO3)nn2)=O)cccc2ccccc12 CC(F)(C(=O)N1CCC1CNC(=O)C)C(F)(F)F.c1(C=O)cccnc1.N N1(C(C(C)C(C)(C)O)=O)CCC2CN(C(c3cc4cc(Cl)ccc4o3)=O)CC2C1 N1(C(C(C)=CC)=O)CCN(C(C2Cc3cccc(OC)c3O2)=O)CC2(CC2)C1 C1(N(C(c2cnc(S)n2C)=O)CC)CCCN(C(=O)CC2CCN(C)C2=O)CC1 C(C1CCOc2ccc(Br)cc21)NC(=O)NC1CCc2n(CC)ncc2C1 N1(C(CCOCC#C)=O)CCC2(C1)CN(C(C1CN(c3ncc(F)cn3)C1)=O)C2 c1(C(=O)NC2C(NC(c3cccnc3)=O)CC2)ccnn1Cc1ccccc1 CC(C)CC(C(=O)NC(C1(C)CC1)C)NC(N)=O.C(=O)C=O.C(C)C Cc1ccc(Br)cc1N(C(=O)CC1CNC(=O)NC1=O)C C#CCCCC(C)C(=O)NC1CN(C(c2ccn(CC)c2C)=O)CC12CC2 Cc1ccc(O)cc1NC(=O)C(C)(C1CCC1)NC(c1ncc[nH]1)=O CC1(CNC(=O)C=CCNC(=O)CCNC(N)=O)CCC1 C1(NC(C(C)c2ncco2)=O)CN(C(c2c[nH]nc2-c2cccs2)=O)CC1O n1(CCCNC(=O)N(C2CC2)Cc2ccccc2OC(F)F)cnccc1=O C(C)(C(=O)NCCOCCNC(c1ncco1)=O)OCCOC C1(C)(C(=O)NC(CNC(c2cc(C)c(O)nn2)=O)C)CCc2ccccc2C1 C1(C(N2CC(O)(CNCCC=O)C2)=O)CCOCC1.C(C(F)(F)F)C1CC1 C#Cc1cn(C)nc1C(=O)NC(C)(C)CNC(c1oc(CC)cc1C)=O C1(OC)CC2CCC1CC2C(=O)NC1CCN(C(C2NC(=O)C3CC23)=O)CC1 C1(C(=O)NCC(C)CN(c2nc(CC)ns2)C)(OCC)CCC(F)(F)CC1 C1(C(=O)NCC(COC)O)CCCCCN1C(=O)CCCCNC(N)=O c1(C(=O)NCCn2cc(C(C=C)(C)O)nn2)c(C)nc(=N)[nH]c1C N1(C(CN)=O)CC(O)C2(CCCC2)C1.CCC(C)C(=O)NCC(N1CC(O)C1)=O C1(C(=O)OC)CCC(C(=O)NCCC(C)(C)NC(=O)CCc2nccs2)C1 CCCC(C(=O)NC1(CO)CCCN(C(=O)Cc2nc(C3CC3)n[nH]2)C1)C(C)C C(N=c1[nH]c2c(c(=NCC3CSCCO3)[nH]1)SCC2)c1c(Br)ccs1 C12(C(=O)NCCC(CNC(c3nnc4ccccn34)=O)O)CCCCN1CCC2 N1(C(C2C(C(=O)OC)C2)=O)CCCCCC1.c1(C=O)ncn(C(C)(C)C)n1.N c1(C(=O)NC(CC)C(=O)NCc2nn[nH]n2)cc(OC)ncn1 C(C(C)C(=O)NCC(CO)NC(=O)CC1(C)CCC1)OCC c1(C(N2CCC(NC(C(C)SC(F)(F)F)=O)CC2C)=O)cc2c(nn1)CCC2 c1(CC(=O)OCc2cccc(C)c2Br)cc(F)c(F)c(F)c1 Cc1cc(C)c(C(=O)N(CC(C)NC(C2(C)CCC(=O)NC2)=O)C)cc1N C(CNC(c1ccn(C)c1)=O)(C(=O)NCC1C2CCCC12)OC c1(C(=O)NC2C3(CN(C(c4ccc(C)o4)=O)C3)CC2)ccc(S(=O)C(C)C)cc1 CC1(C)CCN(C(C2(C)CCOC2)=O)CC1C(=O)NOCC=CCl C1(C(=O)NCCC2(NC(CN3CCC(C)C3)=O)CCCC2)CC2CCCC(C1)C2 CCC(C)CCCC(=O)N1CC(N(C(=O)CCC2CCC2)C)C(O)C1 c1(CC(=O)NCCC(O)C)cccc(OC(F)F)n1.n1(CC(=O)N)cc(Cl)cn1 C(=O)(CC(C)C(=O)NC(Cc1cnc[nH]1)C=O)OCC.c1(CC)ncc[nH]1.N c1(C(N2CC(N(C(Cc3cnc(C)[nH]3)=O)C)C(F)C2)=O)ccnc(Cl)c1N Cc1ncc(CCC(=O)NCCC2(O)CN(C(=O)C(C3CCC(=O)N3)C)C2)o1 c1(C=O)nc(=N)cc[nH]1.c1(CC)nnc(CN(C(=O)CC2(C)CC2)C)o1 N1(C(C2CCC(C)C2)=O)CC(C2CN(C(=O)Cc3ccc(C)c(F)c3)C2)C1.CO Cc1cc(C)c([N+](=O)[O-])cc1C(=O)NCC1CC1.c1(CCC=O)ccnn1C C1(C)(C(N2CCCC(N(C(CC(C)N(C)C)=O)C)CC2)=O)CCCCCCC1 C1(NC(c2cn(C)nc2Br)=O)(CO)CCCN(C(C2CCCC2(C)C)=O)C1 Cc1ncn(C)c1C(N1CCC(O)(CNC(C2(CF)CCOCC2)=O)C1)=O N1(C(C)=O)CCN(C(c2cccnc2OCCO)=O)CC1CC1CC1 C1(CC(N2CC(CC=C)(NC(C3CC3(C)Br)=O)C2)=O)COCCN1C C(=O)(C1=CCCN(C(=O)CC2CC2)C1)NC(CC)C(C)C N1(C(C2N(CCC)CCCC2)=O)CC2CCC(C1)N2C(c1cncc(CO)c1)=O N1(C(CC=C)=O)CCCC2(C1)C(NC(c1nccc(C(F)(F)F)n1)=O)CCN2C C1CC2(CCC2)C1.C1(C(=O)NC)(CC)CCNC1=O.C1(C)(C=O)CCOCC1 c1(C(N(CCC)CCNC(C23CC(O)C2C3)=O)=O)cn2cccc(Cl)c2n1 N1(C(C(C)N2CCCC2)=O)CCC(C)C1C(=O)NCC1(O)CC(O)C1 c1(C(=O)N)ccc(Cl)c(Cl)c1N.Cn1nccc1COCC(=O)NCC(F)C N1(C(C(CCC2CC2)NC(c2cc(C)oc2C)=O)=O)CCc2n[nH]cc2C1 N(C1CCc2c(Cl)cc(Cl)cc21)Cc1nc(C(C)C)on1 N1(C(C2=CCCC2C)=O)C(C(N2CCc3ncsc3C2)=O)C2CC(O)C1C2 N1(C(c2scc(C(C)=O)c2)=O)CC2CC1C2NC(c1occc1Br)=O c1(C(N(C2CCN(C(C3(C#N)C(C)C3)=O)CC2)C)=O)cc(F)c(Cl)cc1F CCCC(C)(CCC)C(=O)NC(C)C=CC(N1CC(C)(C)CCC1CO)=O Nc1ccc(-c2cn(Cc3ccc(C(N4CCC4C(F)F)=O)cc3)nn2)nc1 CCCCC(C)C(=O)NC1CC(CCNC(c2cnn(C)c2C(F)(F)F)=O)C1 N1(C(c2ccc(CC)o2)=O)CCC(NC(=O)C(N2CCC(O)CC2)C)C1(C)C c1(C(=O)NC2CC(N(C(c3c(C)c(Cl)ccn3)=O)C)C2)c(F)ccc2nc[nH]c12 C1(C)(C(N(CCN(C(C)C)C(c2ccc(Br)o2)=O)C)=O)CCC(C)C1 C=C1CCN(C(C2CCN(C)C2)=O)C(C(N2CCOC(C)(C)C2)=O)C1 CCCC(C)CC(=O)NCC1(O)CCCN(C(=O)CCC(=O)c2cccnc2)C1 N1(C(c2n(CC)ncn2)=O)C2CCC1C(C)C(NC(=O)C=Cc1ncc[nH]1)C2 C1(CC)CN(C(C2(C(C)(F)F)CC2)=O)CCC1.C(C)(c1cccs1)=CC=O N1(c2ncc(C)cn2)CCC(C2(NC(c3nc(C(C)C)ncc3Cl)=O)CC2)C1 c1(C(=O)NCCn2cc(C3C4COCC34)nn2)nsc2cc(Br)ccc12 C1(C(N2CC(O)C2)=O)CC(C)(C)OC1(C)C.n1(CC)nccc1C=CC(=O)N C(=O)(C1=CCC(NC(=O)NCC(N)=O)C1)OCC c1(CNC(c2c(OC)scc2)=O)cnn(C)c1C c1(CNC(C2(CC)CN(C(CNC(CC)=O)=O)C2)=O)ccc(C#N)o1 c1(-c2cccc(Cc3cc(C)c(Cl)nc3)n2)c(O)cc(Br)cc1F c1(-n2cc(CC(C)C(=O)O)nn2)ccc(C(=O)NCc2nc(Cl)cs2)cc1 C1(O)(C(=O)NCCC2(CNC(C3(C(C)C)CC3)=O)CC2)CCC1 c1(C(=O)NC2CCC(NC(c3c(C)n[nH]c3)=O)CC2)cccc2cccn12 C(=O)(C1CNc2ccccc21)N1CC(C)C(NC(C2(n3cncn3)CC2)=O)CC1 c1(C=O)ccc2c(c1)C(=O)NC2.Cc1nn(C)c(Cl)c1C(N1CC2CC2C1)=O.N CC1CCN(C(=O)Cn2cnc(C(F)(F)F)c2)C1.C1(C)(CC=O)CCCO1.C n1(CCOC(c2cc(Cl)c(Cl)c(Cl)c2)=O)nc2ccccn2c1=O c1(-n2c(-c3ccc(CC)cc3)nc(CCO)n2)ccc(OC(C)C)nc1OC CCC(C)(C)CCCC(=O)N1C(CNC(=O)CC2COCCO2)CC2CCCC12 C1(CC(=O)NCC2(O)CCN(C(C3CC(F)(F)C3)=O)C2)CC(C2CC2)C1 Cc1cc(C(=O)N(C)CCN(C(=O)C=Cc2cscn2)C(C)C)c(Cl)cc1F N(C1COc2c(Cl)cc(Cl)cc21)C(c1n(C(CC)(C)C)nnn1)C1CCCCC1 C1(NC(Cc2c(C)nsc2)=O)CCN(C(c2cc(N)c(Cl)cn2)=O)CC1C C(=O)(C(CCCCCC)NC(C)=O)NCC1CCN(C(CCCCC=CC)=O)C1 C1(C2CC2)(NC(C2C(CCC)C2)=O)CCN(C(=O)C(F)=C(C)C)C1 N1(C(CCOCCC)=O)CCC(C(F)C(=O)NCCc2scnc2C)C1 Cc1ccc(OCC(N2CC3(C2)CN(C(=O)C(C)(C)F)C3)=O)cc1C CCC(CCCC(=O)NCCc1cccc(C)c1)NC(c1cnc(C)cn1)=O C(=O)(CC(C)(C)CC(=O)N1CCN(CC2CN(C(=O)CC)C2)CC1)OCC.S c1(C(=O)NC2CC(C(=O)Nc3cnn(CC)c3C)C2(C)C)cc(C)cc(O)c1 C1(C(=O)NC(C)(C)CCF)CSCCN1C(c1cnns1)=O C(=O)(C(O)CC(C)(C)C)N.N1(C(c2c(C(=O)OC)csc2)=O)CCC(CF)C1 N1(C(c2cc(OC)ncc2F)=O)CC(C2CCCCN(C(=O)CC(C)SC)C2)C1 c1(C(=O)Nc2c[nH]nc2C(=O)NCCc2ccc(Cl)cc2)cc(I)ccc1F n1(C(C)C)cncc1C(=O)NC(CC1CC1)C(=O)NC1(c2nn[nH]n2)CC1 c1(C2C(C(=O)NCCN(C(=O)CSC(F)F)CCC)C2)csc(Br)c1 CCCC(C)(CCC)C(=O)N1CCC(NC(=O)CCC=C(C)C)C(CO)C1 N1(C(C(C2CN(C(=O)CC3CCCC3)C2)OC)=O)CCC(O)(CO)CC1 CCC1=C(C(=O)N2CCC(NC(c3nocc3CC)=O)CC2C)SCCO1 C#CCCCC(=O)NCC(O)CCNC(=O)C(CC)N1CCCC1=O c1(N2CC(CNC(CC(C)(O)C3CC3)=O)OCC2)c(F)cc([N+](=O)[O-])cc1F N(C(=NCc1ccc(F)cc1)NCc1nnc(C(C)(C)C)s1)C1C(C)C1 c1(CNC(C(c2cn(C)nc2)NC(C2CCCCS2)=O)=O)cccc(Cl)c1 C(CN=c1[nH]c(=NC(C)c2nncs2)[nH]c2c(F)cccc12)N(C(C)C)C1CC1 c1(C(N2CC(CC(C)(C)C)C(NC(C3CC(O)C3)=O)C2)=O)ccc2nncn2c1 C(=O)(C1CCc2nccn21)NCC1N(C(c2cc(OC)ncn2)=O)CCN(C)C1 c1(OC)nn(C)cc1C(=O)NC(CCN(C(=O)C(C)C1CCOC1)C)C(C)C c1(C(N2CCN(C(C3C(C)OCC3)=O)CC2)=O)cccc([N+](=O)[O-])c1Br C12(NC(C3CCN(C)C3)=O)CCC(CN(C(C3C4CCCC34)=O)C1)C2 c1(CCNC(=O)NCC(c2cnccn2)(C)C)cccc(Cl)c1Br c1(C(=O)NCCC2(O)CN(C(C3(CC=C)CCCCC3)=O)C2)ncncc1C#N N1(C(c2n(CCC)ccc2)=O)CCC2CN(C(C34CSC(C3)C4)=O)CC2C1 N1(C(C2(C=C)CCC2)=O)CCCOC(CNC(C2CCCCN2CC(F)F)=O)C1 Cc1nc(C)c(C(C)NC(=O)CC(O)CNC(C2CCCC2O)=O)[nH]1 c1(C(N2CCc3ncsc3C2)=O)coc2c1CN(C(C1CCCOC1)=O)C2 N1(C(c2ccc(N)cn2)=O)CCC2CCC12CNC(c1ccnc(CO)c1)=O N1(C(Cc2nc(C)oc2)=O)CCC(C2(NC(c3ccoc3C)=O)CC2)C1 Cc1cc(=NC(=O)C(Cc2ccoc2)NC(=O)CN2CC=CC2)[nH]n1C CC(C)CC(O)CC(=O)N1CC2C=CC1C(C(=O)NC1CC(=C3CC3)C1)C2 CC(O)C(F)(F)C(=O)NCCC1(NC(=O)Cn2cccnc2=O)CC1 c1(C(N(C2CCN(C(C3(CCCC)CC3)=O)C2)C)=O)cc(C)n(C(C)(C)C)n1 CC1(C)CC(C(=O)O)(NC(=O)Nc2nc(-c3cccnc3)cs2)CCO1 C1(NC(c2nncn2C2CC2)=O)CCCN(C(c2csc(Cl)c2)=O)CC1 C1(NC(CCN(CCC)C)=O)CCN(C(=O)C(C)(C)c2ccno2)CC1C Cc1ccnc(O)c1C(=O)NC(CC(=O)Nc1cccc(F)c1O)C1CC1 Cn1[nH]cnc1=NC(=O)c1cscc1-c1ccccc1-n1cccn1 CN1CCN(C(=O)C(=O)NCC2CCN2Cc2ccccc2)CCN(C)CC1 C=CC1(CC(=O)N(C)CCOCC)CN(C(=O)COc2ccccc2C)C1 C(=O)(C(O)CC(F)F)NC1C(NC(c2cccc(F)c2Cl)=O)CCOC1 CN1CCOCC1CC(=O)N(CCNC(=O)Cc1ccnc(O)c1)C.C1CC1 c1(C(N(C)CC2N(C(C(C)O)=O)CCC2)=O)cccc2ncc(Br)n12 CC1CN(C(=NCCF)NCc2nc(CS(C)(=O)=O)n[nH]2)CC(C)S1(=O)=O c1(C(N2CCC(=C)CC2C(=O)NOCC2CCCCC2)=O)ccc2cc[nH]c2n1 c1(CC(N2CCN(C(C(CC)N(C)C)=O)CC2CF)=O)ccc(C#N)cc1F c1(C(=O)NC(CNC(CNC(CC)=O)=O)C(C)C)c[nH]c2ccccc2c1=N N1(Cc2cccc(OC(C)=O)c2)CC(F)(F)CC1C(=O)N.c1c(Cl)ccnc1Br C(=O)(CCCC(F)(F)F)N1C(CN(C(=O)C=CC2CCOC2)C2CC2)CCC1 c1(NC(c2ccc(CO)cc2)=O)ccc(N2CCN(C(=O)C(F)Br)CC2)cc1 c1(C(=O)NC(C(C(=O)NC(C)Cc2cnc[nH]2)(C)C)C)ccc2c(c1)CCC2 c1(C(=O)OCC)nc(Cl)c(Cl)nc1NC(C1CCCCC1)=O.C(=O)C(C)O C=Cc1ccc(C(=O)NCC2(C(=O)Nc3cc(C)cc(Cl)n3)CC2)cc1 C(C(CO)(CO)NC(=O)Cn1cnnc1)N(C)C(C1CN(C2CCOCC2)C1)=O C(C)(CCC(=O)NC1(CF)CN(C(=O)C(O)CSC)C1)OC N1(C(Cn2nnc(=N)[nH]2)=O)CCN(C(c2cccc(Cl)c2Cl)=O)C(C2CC2)C1 N1(C(c2c(CC)nccc2)=O)CC2CN(C(=O)C=CC(F)(F)F)CC2C1 N1(C(C(C(C)C)O)=O)CCC2(CC1)CC2C(=O)NCc1cc(Cl)no1 C(=O)(C(CC(C)C)OC)N1CC(CC(=O)NCCCCCC)C(C)C1 C(C(CC(C)C)C(=O)N(C)C(C1CCCO1)C)NC(COC1(C#C)COC1)=O O=C(C(CO)C(F)(F)F)NCC1CCN(C(=O)CCN2CCOC2=O)CC1O N1(C(C(C)O)=O)CCC(C)CC1C(=O)NCCCSCCO c1(C(N2CCCC(CNC(N)=O)C2)C(=O)NCCCCCC)sc(C)cc1Br C1(C(=O)NC2CCC(CNC(=O)Cn3ncnn3)C2)CCc2nncn2C1 Cc1cc(C(=O)NC(C)CC)ccc1S(N)(=O)=O.C1(C(=O)N)CC1.C(C)C C(=O)(CCCN=[N+]=[N-])NC(CCC)CNC(C1(C)CCOCC1)=O C(=O)(C=C1SCC(=O)N1C)N1CCC(NC(C(C(C)C)F)=O)C1C(C)(C)C Cc1cc(CCC(N2CCC3C(NC(=O)Cc4ccc(Cl)s4)C23)=O)nn1C C1(C(N(CC(C)N(C)C(c2cnn(C3CC3)c2)=O)C)=O)CCCC2(CC2)C1 N1(C(C2=C(C)CCC2)=O)CCC2(CCC2NC(=O)CCS(C)=O)CC1 CC1CCN(C(=O)CCOCCCNC(=O)CCc2ccncc2)C1C C1CCN(C)CC1C#N.n1(CC(=O)NC(c2nc(C=O)co2)C)ccccc1=O.N Nc1cc(Cl)c(Cl)cc1C(=O)NCC1CCCN(C(=O)Cc2cccnc2)C1 C1(NC(=O)C(F)n2cccn2)(CO)CN(C(=O)C=CSCC2CC2)C1 N1(C(c2cc(C)sc2C)=O)CCN(C(c2c(C)nsc2Cl)=O)CC1c1cn[nH]c1 C12(C(=O)NCC(C)N(C)C)CCC(CC1)C2.c1(CC=O)ncc(F)cc1F.N Cc1cc(F)c(C(=O)NC2CC(NC(c3ccccc3Cl)=O)CC2O)cc1F c1(C(C(=O)N(CC(CC)NC(=O)CC)C)C)ccc(F)cc1F.CCN(C)C.O C1(CC(=O)N)CCC(=O)NC1.C1(CNC(=O)CCN2CCC2)CCC(C)C1 N1(C(c2c(CC)cco2)=O)CC(C)(C)CC1CNC(=O)C(CC)C(C)O c1(CCC(=O)NC2C(CNC(=O)C(Cl)=CCl)C2)ccc(Cl)cc1 N1(C(c2c(C)occ2)=O)CC2(C1)CN(C(C1CN(C)CC1C(F)(F)F)=O)CCO2 C1(C(N2CCC(CC)C2)=O)CC2CC1CC2NC(=O)Cc1cc[nH]c1 CC(C)CC(C)C(=O)NC1CCC(CNC(c2c[nH]cc2C2CC2)=O)CC1 c1(CC)nc2c(C)csc2c(=NCCC2CCN(C(C3(F)CCOC3C)=O)C2)[nH]1 c1(CN(CC(C2(C#C)CC2)=O)Cc2cnc(C)o2)ccccc1 C1(C(=O)NCC2C(C(C)C)C2)(NC(=O)Cc2ccoc2)CCCCC1 CC(Cc1ccnn1C)C(=O)NC(C)CN(C(=O)C=Cc1cscn1)C N1(C(CCN(C)CCO)=O)CCC(NC(C2CC3(CCCC3)C2)=O)C(C)(C)C1 C(=O)(CC(=O)NCC(C(=O)NCc1c[nH]nc1C1CC1)N(C)C)N(C)C CC(=O)C(C)CC(C)C(=O)N1CC(NC(=O)CCC(C)(F)F)C(O)C1 c1(C(N(CCCNC(Cn2c(C)ncc2)=O)C)=O)cccc2c(C)ccnc12 C(=O)(C1CC(=O)Nc2ccccc21)NCC12CCCN(C(C=CC)=O)C1C2 c1(CNC2C=CC(C(N(C3CCOCC3)CC)=O)C2)c(F)cccc1[N+](=O)[O-] C1(CC)CC(C(N2CCCC2(C)CNC(=O)C(c2cccnc2)C)=O)CCC1=O Cc1cc(C(=O)NC2CC(CCNC(c3ncn(C)n3)=O)C2)n(CCO)n1 c1(C(N(CCCNC(=O)C(C)(C)O)CC)=O)c(C2CC2)nn2ccccc12 c1(C(N2CCN(CC(=O)NCc3nccs3)CC2)=O)ncn2c1CCC2 N1(C(c2sccc2Br)C(=O)NCCOC)CCCCC1c1ccc(C)cc1 c1(CCC)nc(=NCC)s[nH]1.c1(C(C(=O)N(CCO)C)C2CC2)ccc(F)cc1 CCCCCC(O)CC(=O)NC1(CCNC(=O)C=Cc2nc(C)co2)CCC1 C1(SC)CN(C(c2csc(C(F)(F)F)n2)=O)CC1NC(=O)C(C)CO c1(CNC(C2CC3C(C2)C3(F)F)=O)c(Cl)cccc1Cl C1(C(=O)NCC(C)N(C(=O)CCF)CC)CCS(=O)(=O)C1 C1(NC(c2cn(C)c(=O)cc2)=O)CCN(C(=O)CC2CCOC2=O)CC(C)(C)C1 N1(c2nccc(OC3CCC(O)C3O)n2)CCC2(CC1)CC2 N1(C(C2C(CC)C2)=O)CCC(CF)(NC(c2ccnn2CC)=O)C1 C1(C(=O)NCCSCCOC)CCCC(NC(=O)CCC2CCCC2)CC1 CC1(C)CCC(C)N(C(C2CC2[N+](=O)[O-])=O)C1.C(=O)C(F)(F)C1(O)CCC1.N C(=O)(CC(CC)CC(C)C)N1C2C(NC(C3CN(C(CC)=O)C3)=O)C(C2)C1 C1(CNC(CCC(=C)Br)=O)N(C(=O)CSC(F)F)CCCC1(C)C C1(NC(c2cc(OC)ncc2)=O)CC2CC(C1)CN(C(=O)C(F)CC1CC1)C2 c1(C(N2CCCC(NC(C(CC)CC(C)C)=O)C2)=O)c(C)nn2cc[nH]c(=O)c12 N1(C(C(CCC)C)=O)CC(CNC(=O)CCCc2ccc(Cl)c(Cl)c2)CC(C)C1 c1(SC)ccc(NC(=O)NC2CCN(OC)CC2)cc1Br c1(OC)ccnc(C(=O)NC2(C)CCC(NC(=O)C(CSC)OC)CC2)c1O CCCCC(C(=O)NC(C(=O)NC1CC1CC)c1ccco1)C(C)C N1(C(C(C)C)=O)CCCCC1C1CCN(CCS(C)(=O)=O)C1 C1(NC(CC2(OCC)CCC2)=O)CCCCC1N(C(=O)C(C)OC)C Cc1cc2ncc(C(=O)NC3CC3CNC(c3ccnn3C)=O)cn2n1 Cc1ccc([N+](=O)[O-])cc1C=O.c1(C(N(CC(C)C)C)=O)coc(C2CC2)n1.N c1(C(N(C2CN(C(=O)CC3CCCOCC3)CC2O)C)=O)cnc2scnc2c1 c1(C(N(CC(C)NC(C2=C(C)CCC2)=O)C)=O)[nH]nc2c1CCC2(C)C c1(C(=O)NCC(C(=O)NC2(CC=C)CC2)O)ccn2ccccc12 C1(C(N2CC(CC(C)NC(C3(c4ccccc4)CC(F)C3)=O)C2)=O)CCCOC1 C1(C(=O)NCC(c2ccc(Cl)c(F)c2)O)CC(=O)C12CCCCC2 C12(C=O)C3C4C1C1C2C3C41C.C1(C(N2CCC(CC)CC2)=O)CCC(O)CC1.N C1(C(N(C(CCSC)C)C)=O)CC(C)CCN1C(c1cc(C)sc1C)=O N1(C(c2ccc(C)c(F)c2)=O)CCC2(CCCC2N=c2[nH]ccnc2F)CC1 C(=O)(C1=CC2(CN(C(C3COCC3C(N)=O)=O)C2)OC1)N(CC(C)(C)C)C N(C(=NCC(=C)C)NC1CCN(C(=O)C2CC2)CC1)CC(CCC=C)(C)C n1(CC)ccc(C(N2CC3CC2C3CNC(C2CCCN2C=O)=O)=O)c1C N1(CC)C(=O)NC(c2c(C(=O)O)nn(C)c2C#N)C(C(=O)OC)=C1CC(F)(F)F N1(C(c2cc(C#N)[nH]c2)=O)CCC(O)(CNC(=O)CCc2cnoc2)CC1 C1(C)(NC(C(C)N2CCC2)=O)CCCN(C(c2ccnc(C(F)(F)F)c2F)=O)C1 c1(C(=O)NC2(CNC(=O)CCc3cccs3)CC2)ocnc1C1CC1 c1(CC(N2CCCC2)=O)cccnc1O.C1(C(=O)NCCO)(CSC)CC1 c1(N(CC(CC=C)(F)F)C(=O)CN2CCN(CC)CC2=O)cc2n(n1)CCCC2 C(=O)(CC(C)C(C)(C)C)N(CC(C)O)CCNC(c1sccc1F)=O CC1(C)C(NC(c2cocn2)=O)CC1CC(=O)NCC1CSC1 Cc1ccc(C(=O)NCC2CC2NC(c2cncnc2C2CC2)=O)c(Br)c1 Cc1ccc(C(=O)NCC2C3CN(C(c4ccc(=N)[nH]n4)=O)CC23)cn1 C1N(C(c2cnn(CC)c2)=O)CC1(C)C.C(c1cc(C)no1)=CC=O.CO.C C1(F)(CNC(C(C=C)CC)=O)CCCN(C(C23CCCC2(C(N)=O)C3)=O)CC1 CC1CN(C(=O)CSc2cccs2)CCC1NC(c1scnc1C(F)F)=O c1(C(=O)NC2CCC(NC(C3(C)N(C)CCC3)=O)CC2)ncnc2c1cnn2C CCC(C)(C)CCCC(=O)N1CC(C)C(C)(C(=O)NC2CC(C)(C)C2)C1 Cc1nccc(C(=O)NCCOC2CCN(C(=O)CCc3nncn3C)C2)c1N CC(C)C(CC1CCCCC1)C(=O)NCCCCCNC(=O)CCn1cnnn1 c1(C(N(CC(C)CNC(C2(CO)CC2)=O)C)=O)n[nH]c2ccc(O)cc12 C=C(CNC(=O)C(C)C)CCNC(=O)C(C)Cc1ccco1.C(C)=O.N Cc1ccc(CC(C(N2CCC(C)C2CNC(=O)CCCF)=O)NC=O)cc1 N1(C(C2(C#C)CC2)=O)CCC2(CCN(C(=O)C(CO)C(C)C)C2)C1 C1(C(=O)NCC(C)(C)CCNC(c2ccc(C)o2)=O)(CC)CCCC1O.S C1(NC(CC(CC)(C)C)=O)CN(C(C2CCC(=O)C(C)C2)=O)CC2(CCC2)C1 c1(OC)ccc(F)c(C(=O)NC2CC(F)(CNC(C3(Cl)CC3)=O)C2)c1 C12(C(=O)NCC3(CCO)CCCC3)CCCC1CN(C(c1ccc(F)s1)=O)C2 C(CCCN=c1ccn2nccc2[nH]1)NC(CC1CCC(C)CC1)=O n1(C(C)C)ncc2c1CCCC2NC1CCCc2ccc(Br)cc21 c1(CN(C(=O)C(C)NC(=O)C(C)=CC(C)(C)C)CC#C)ccco1 CC#CCCCC(=O)NCC(CNC(=O)C(c1ccc(Br)cc1)C)OC N1(Cc2cc(C)[nH]n2)CCC(NC(c2cc([N+](=O)[O-])cs2)=O)C(O)C1 C1(C(=O)NC(CNC(=O)Cc2ccon2)C2CC2)CCCC(F)(F)CC1 O=C(CCCOCCc1ccccc1)NC1(CNC(c2cn[nH]c2)=O)CC1 C(CS(=O)(=O)NC(c1ccccc1)C(N)=O)(C1CCOC1)OC C#CC1(C(=O)NC(c2nc(C)cs2)C)CN(C(=O)CCc2cccnc2)C1 CC(F)(CNC(c1cnc(N2CCN(C=O)CC2)nc1)=O)C(=O)O.C1CC1F.N C1(CNC(c2c(C)snn2)=O)CN(C(=O)C=CCF)CC1C(F)(F)F O(NC(=O)CCn1cccc1)CC(=O)NCCCC(C)O c1(C(N(C)CC2CCN(C(C(C=C)OC)=O)C2)=O)ccc(F)c(OC)c1F Cc1cc(C(=O)N(C2CCCCO2)CCNC(=O)O)c(F)cc1Br.C(C)(C)C c1(C=O)cn(CC(F)(F)F)nc1C.C12CC(C1)C2.C1(C=O)CC1.CCO C(=O)(C1=CSCCO1)N(CC(O)CNC(C1CC1c1ccncc1Cl)=O)C(C)C N1(C(c2c(C#C)c[nH]n2)=O)CCC(C)N(C(=O)CCc2ccc(Cl)cc2Cl)CC1 C(=O)(C1=CCCSC1)N1C(CCC(=O)NC(CCC(=O)OC)C)CCCC1 Cc1cc(=NCC(O)CNC(c2c[nH]cc2C2CC2)=O)[nH]c(S(C)(=O)=O)n1 C1CC(=O)N1.C1(C)CCC1.C(=O)(C)NCC=CCSCC.C(C)O CCCCC(C)C(=O)N1CCN(C(C2(F)CCCC2)=O)C(C(F)F)C1 CCC(C(=O)N1CCN(C(C2CC(O)C2)=O)C(c2cccc(OC)c2)C1)C(C)C C1(CNC(C(C=C)(C)C)=O)CCN(C(=O)C(C)CN2CCCCC2)CC1(F)F CCC(CC)C(C(=O)N1CCC(C(=O)NC2COCC2SC)C12CCC2)OC c1(C(N2CC(C3CC3)CC2)=O)nnc2n1CCCCC2.C(C(=O)NC)=CCOC C1(NC(C(CC)n2cncn2)=O)CCCC12CN(C(c1cc(N)cc(O)c1)=O)C2 C(=O)CC(C)CC(C)(C)C.Cc1ccn(CC(=O)NCC2(C)CC2(F)F)n1.N C1(CNC(C(C)NC(C)=O)=O)CC(F)CN1c1nnc(CC(C)C)s1 C1(C(=O)NC(CN(C(C2CCCCC2)=O)CC)C)Cc2cccc(Cl)c2C(=O)O1 Cc1nc(O)nc(C)c1CCC(N1CC2CCC1C2NC(c1cnc(Cl)[nH]1)=O)=O N1(C(C2CCC(NC(=O)CN3CCSCC3)C2)=O)CC2CC1CC2O CC(C)(F)C(C)(F)C(=O)CC(c1ccc(Cl)cc1)n1cc(-c2cnccn2)nn1 c1(OC)ncc(NC(=O)CCCCCN(C)C(C2CC(O)C(F)C2)=O)cc1C C1(NC(CN(CC)CC)=O)C2CN(C(c3nccnc3C)=O)CC12 C(C)(CC(=O)NCC1CN(C(=O)CC2=CCCC2)CCC1(F)F)(C(F)F)N(C)C C=CC(C(=O)N1CC(OCC(=O)NCCC(O)COC)C1)OC N1(C(c2nccs2)=O)CCCC2(C1)CN(C(c1ncoc1C1CC1)=O)CCO2 O=S(=O)(c1cnc(NCC2CC2Cl)c(Cl)c1)N1CCCc2occc2C1 CN1CCCCC1C(=O)NCC1CCCN1C(=O)CC1(CO)CC1 c1(C(=O)NC(C)Cc2ccnn2C)ccnc(CNC(C2CCC(F)C2)=O)c1 Cc1nc2ncnn2cc1COC(C1CCc2nc(NC(C)(C)C)nn2C1)=O c1(C(=O)NC(C(C)NC(c2c(SC)csc2)=O)(C)C)ccc(C)cc1Cl c1(NCCC(C(C)C)C)cc(=NCC(c2ccco2)N(C)C)[nH]cn1 C1(C(N(C)Cc2ccoc2)=O)CCCCC1.C1(C=O)(C(=O)C2CC2)CC1.N C(=O)(CCCC(C)C)N(C(CN(C(c1c(CC)onc1)=O)C)C)C c1(C(=O)OC)cccc2c1N(C(=O)NC1CCCC1(F)F)CCNC2=O C1(CNC(C2(CC#C)CCCCC2)=O)CN(C(=O)C=CCCC)C2CCN1C2 N1(C(CCc2n(C)ccn2)=O)CCCC12CCN(C(c1cccn1C1CC1)=O)C2 c1(CNC(CC2(C)N(C(CC3C(C)=NNC3=O)=O)CC2)=O)ccccc1C#N C1(C(=O)OCC)(C(=O)N)CCC1.C1(C2CCCO2)(C=O)CCC1.C(C)C C=CC(C)(CCOC)C(=O)N1CCC(CCOC)(NC(=O)CC2CC2)CC1 C1(CC(N2CC(O)C2)=O)C2CC3CC(C2)CC1C3.C(=O)C(F)C(C)(C)O.CC Cc1[nH]cc(C(=O)NCC(C)(O)CNC(=O)C(C(C)O)N(C)C)c(=O)c1Cl Cc1ccnc(C(N2CCCC2CNC(=O)COCC2CCOCC2)=O)n1 C(CC(=O)NC1CCOC(C)(CC)C1)(C(C)(C)C)NC(C1C(=C)C1)=O C(c1cccc(F)c1)=CCC(N1CC(C)(NC(c2cc(C)[nH]c2C)=O)C1)=O C(=O)(C(C)(C)S(C)(=O)=O)N1CCC(C)(CNC(C(C)C#N)=O)C1 N(C(=NCc1ccsc1)N1CCCC(CCC(C)C)C1)C(CC)C CC1CCC(NC(C2CCCOC2)=O)CN1C(c1ccc(-c2ccccc2)o1)=O c1(C(=O)NC(CC#C)C(=O)NC(CC)C(=O)NC)occ2c1CCC2 O=S(=O)(c1ccc(N2CCC=C(Br)C2)c(Br)c1)NC1(c2cccnc2)CCC1 N1(C(CCC(=O)OC)=O)CC(NC(=O)C(C)c2cc[nH]n2)CC12CCC2 N1(C(CCC=CCC=C)=O)CCC(C2(O)CC(NC(=O)CCCC#N)C2)CC1 C=C(Br)CCC(=O)NC1CC1NC(c1cc(-c2cnn(C)c2)no1)=O CC1OCCOC1C(=O)NCCCCCNC(c1cccc(-c2ccco2)c1)=O C(CCC(O)C(=O)NC(C(N)=O)C1CCCC1)NC(c1ccc(C#C)o1)=O C1(C(=O)N(CC2CCCCC2)OC)(CC=C)CCCN1C(C1CCO1)=O N1(C(C(C2CCCCCC2)C)=O)CCc2nc[nH]c2C12CCOCC2 c1(C(C)O)ccc(C(N2CC3CC3(CNCc3ccc(Br)s3)C2)=O)cc1 N1(c2oc3ccc(C)cc3n2)CCC(C2CCCN(C(C34CC(CO3)C4)=O)C2)C1 C=CCC(C)(O)C(=O)N1CCN(CC(=O)N(CCCC)CCCO)CC1 C(=O)(C(C)CS(C)=O)N1CC(CC=C)(NC(c2oc(CO)cc2C)=O)C1 C1(NC(=O)Cn2cccn2)C2CCN(C(C3CSCCS3)=O)CC12 C1(C)(CC)C=C(C(=O)NC2CCC(NC(c3nc(C)ccc3O)=O)CC2)C1 CCCC(C(=O)NCC1CC12CC2)NC(c1snc(C)c1N)=O C1(C(=O)NCC(C)C(C)(F)F)CC(C)(C)CN1C(c1n[nH]c(O)n1)=O Cc1sc(C(=O)N(C(C)CNC(=O)CC(C)(C)c2ccc(F)cc2)C)nc1O C1(C(C)(C)CO)CCCN1C(=O)Cn1ccc(Br)n1 N1(C(C=CCC)=O)CCC2(CCCC2NC(=O)CCC2OCCO2)C1 c1(OC)ccc2c(C(N3CCC3C(=O)Nc3nccs3)=O)cccc2c1 N1(C(c2c(CC)non2)=O)CCCN(C(=O)C(C)Sc2ccccc2)C(C)C1 CC1(C)COC(C(=O)NCC2CC2NC(=O)CS)C1.c1ccc(Cl)s1 Cc1[nH]nc(C(=O)N(CC(C)O)CCNC(C2(C3CCCO3)CCC2)=O)c1F N1(C(c2cnnc(C)c2C)=O)CCC2(CCC2NC(c2ccc(O)nc2)=O)CC1 c1(C(=O)NCCn2cc(CC(=O)O)nn2)ccccc1CC(F)(F)F c1(C(=O)NC2COCC2NC(C2CCCCN2CC(F)F)=O)ncc2n1CCCC2 C1(C(C)NC(C2(NC(C)=O)CCC2)=O)CCCN(C(C2CC=CC2)=O)C1 C1(NC(C2(C(C)(C)OC)CC2)=O)CCCC(C(=O)NCC2CC2)CC1 N1(C(N(c2cccnc2)CC#C)=O)CC2CC3CC2C1C3 C1(C(=O)OC)CN=C2N=C(CNc3cnc4c(cnn4C)c3N)NN2C1 N1(C(=O)NC(c2ccc(C#N)cc2)CF)CCCC1C1CCCc2ccccc21 C(=O)(CCCCCOC)NC1(COC)CN(C(=O)CC2CCC(C)C(C)C2)C1 c1(C(=O)NCC(CNC(C(CN(C)C)(F)F)=O)(C)O)cc(N)ccc1O N1(C(C=C(C)C(F)F)=O)CC2CCN(C(C3CC3(Cl)Cl)=O)C2C1C C(=O)(C1CCc2cc(Cl)ccc21)NC(CN(C(=O)C(=O)NC(C)C)CC)C C=C=CC(C)C(=O)NC(c1ccccc1)C(N1CCCC1)=O.C(C)(C)C.C=O.N C(=O)(C(O)CC(F)F)N(C1CCCCCC1)CCNC(c1ccccc1O)=O C1(CNC(C(CC(C)C)C)=O)CCCC2(CN(C(=O)C(C)(C)CC(C)(C)C)C2)O1 N1(C(c2n(C)ccc2)=O)C2CCC1CN(C(c1cc3sccc3s1)=O)C2 c1(C(N(C2CN(C(CN3CCC(C)CC3)=O)CC2F)C)=O)ccc([N+](=O)[O-])[nH]1 c1(CC)c(-c2nc(CCOC3CCCCC3)nn2CC2CCCN2C)cnn1C c1(C=O)cccn(C2CC2)c1=O.CN1CCOCC1C(=O)NC(C)C(C)(C)C.N C12(C(N3CC4C(NC(C5CC6CC6C5)=O)(C4)C3)=O)CCCN1CCC2 c1(C(N(CCCCNC(CN(C)CC)=O)C)=O)ccc(-n2ccnc2)cc1 CC(CC(N)=O)C(=O)NCC(c1ccc(F)cc1)NC(c1ncn(C)n1)=O c1(C(C(=O)NC2CCC(NC(c3occc3F)=O)CC2)=O)ccc(F)c(F)c1F C1(C(NC)=O)CCC(S(C)(=O)=O)CC1.C1CCN(C(=O)Cc2cscn2)CC1.C c1(CC(N2CCC(NC(CC3CCC(C)O3)=O)CC2)=O)c(F)cccc1Br c1(CNC(C(N2CCC(C(N)=O)CC2)C2CC3C=CC2C3)=O)ccccc1F c1(CC(=O)N(C(C)CNC(=O)CCCc2ccncc2)CC)cnnn1C N1(C(c2c(C)nc[nH]2)=O)CC2CC(C)N(C(=O)CN3CCCCCC3)C2C1 N1(C(CSCC=C)=O)CC(O)CC1CNC(=O)CCn1ccc(C)n1 n1(CC)nncc1C(=O)NC(C(=O)NC(c1cnn[nH]1)C)C1(O)CCC1 c1(CC)c(C(=O)NC2CCCN(C(=O)C(C)(C)O)C2)cnn1C N1(C(C=CC)=O)CC(C)OC2(CCN(C(=O)Cc3ccccc3)C2)C1.C(C#N)O C(c1cnc[nH]1)=CC(=O)N(C1CCN(C(=O)C(O)Cc2cnc[nH]2)C1)C N1(C(CC(=O)NCC#C)=O)CCC(NC(c2cc(C)[nH]n2)=O)C(CO)CC1.C N1(C(CCC(C)CN(C)C)=O)CCC2CN(C(=O)C(C)(C)C(F)(F)F)CC12 CCC(CC(=O)NC1(CCOC)CCN(C(c2ncncc2Cl)=O)C1)C(C)C C(CCCCCCOC(C)=O)(c1n(CC)nnn1)NC1CCCC(F)C1 Cc1cc(Cl)c(C(=O)NCC(O)CNC(=O)C(C(C)C)N(C)C)c(Cl)c1 C=CC1(C(N2CCC(CNC(C3CC4(CCO3)CC4)=O)(OC)C2)=O)CCCCC1 C1(NC(c2cn(CCNC(c3cc(=N)[nH][nH]3)=O)nn2)=O)CC2C=CCC(C1)C2 C(=O)C(C)C(C)(F)F.Cc1cc(C(N2CCC(CO)C2)=O)nn1CC(F)(F)F.N c1(CN(C(=O)C2=COCC2)CC)ccc(C)cc1-n1cc(C)nn1.C1CCOC1 c1(C(=O)NC(C2CN(C(C3CS(=O)(=O)C3)=O)CCO2)C)n[nH]c2c1CCCCC2 C(=O)(C(O)CCCn1cc(C2CC3CCC(C2)C3)nn1)NCC1CC(=O)NC1=O C(C(C(=O)NCC#CCOC)N(C)C)OC c1(OC)cc(C(F)(F)F)[nH]c(=NC2CN(C(=O)C(C)(C)C(C)C)CC2C)n1 N1(C(COCC)=O)CCC2CC2(C(N2CC3(CCOC3=O)C2)=O)CC1 N(C(=NCCCC(C)(C)C1OCCO1)NCC1CCCC(F)(F)C1)CCC(=O)NC c1(C(N2CC(CC)(NC(=O)C(C)(F)c3ccon3)C2)=O)cccc2ccnn12 C=CCC(F)(F)C(=O)N1CCC(CNC(=O)CC(C)CCc2ccccc2)C1 C1(NC(CCC(C)OC)=O)CN(C(=O)CSCC(N)=O)CC1S(C)(=O)=O c1(CNC2CC(C(=O)Nc3cncc(CC)c3)C2)cccc2c1OCCO2 CCC(C)(C)CCCC(=O)N1CCCC2C1CCN2C(C1CCCCC1CC)=O N1(C(CCC#C)=O)CC2CC3CC2C1C3NC(=O)C=C(C)c1cccc(OC)c1 C1(C(N2CC(C(=O)OC)C(CO)C2)=O)CC2CCN(C(c3cnc(C)s3)=O)CC12 C1(F)(CNC(=O)C=Cc2cn[nH]c2)CC(N=c2[nH]c(Cl)ncc2C2CC2)C1 Cc1nnc(CN(C(=O)COCCNC(=O)CN2CC3CC3C2)C)o1 c1(N2C(CNC(C(CC)C(C)O)=O)CC3(CCC3)C2)nc2ccc(N)cc2s1 Cc1nc(Cc2ccccc2)sc1C(N1CCC1)=O.C1(C(=O)N)CC1.N(C)C Cc1ncc2c(n1)CCC(C(=O)NC(C)(C)C(C)C)C2.C(=O)(CCC(C)(C)F)N c1(C(=O)NC2C(NC(C(C)SC)=O)CCOC2)nccc2ncccc12 N1(C(CC(CNC(c2cc(OCC)no2)=O)C)=O)CCn2ncc(C)c2C1 C(=O)(CC(F)(F)C(F)F)NC1C=CC(CNC(C(CC)n2cccn2)=O)C1 O=C(Cc1ccsc1)NNC(=O)C1CCC(n2cccc2)CC1 C1(CC)(CC)CCN1C(c1conc1CNC(c1cc[nH]n1)=O)=O C(C(C)C(F)C(=O)NCCCNC(C)=O)NC(CCC(=O)NCC)=O C1(=CC(N2CCC(CC)(NC(C3CCOC3)=O)CC2)=O)CCOc2ccccc21 C1(C#N)(C(N2CC(OC)C(NC(C3CC3c3cncn3C)=O)C2)=O)CCSCC1 CCN=C(NCCN1CCOCC1C)NC1CC(c2nccc(C(F)(F)F)n2)C1 c1(SCC)cccc(C(=O)N(C2CCC(NC(c3ccc(OC)o3)=O)C2)C)c1 CC1(C)CC(C(=O)NC2CCCC2C=O)(CO)C1.c1ccc(C(N)=O)nc1.N Cc1cc2ncc(C(=O)NC3CC(C(N4CCCCC4C#N)=O)C3)cn2n1 c1(OC)cnc(NC(=O)CC2CCN(Cc3cnc(Cl)nc3)C2)cn1 CC1(C(=O)NCC2(F)CN(C(=O)CS)C2)CC2CC2C1.c1ccc(F)cc1 C(=O)(C#CC1(C)CCCO1)NC1(C)CC(NC(C2=NOC(C)C2C)=O)C1 Cc1cc(CC(=O)NC2(C#N)CCN(Cc3ccc(Br)cc3O)C2)cc(F)c1 C(C(C)(C)CCNC(C1(C)CC2(CC2)C1)=O)NC(c1c(C)onc1)=O C[Si](C)(C)c1ccc(CNC(N2CCSCC(CO)C2)=O)cc1 C(c1ccccc1)=C(CC)C(=O)NCC(c1ccccc1)CN(C)CC C1(NC(c2cccc(Cn3ccnc3)c2)=O)C=CCN(Cc2ccccc2Cl)C1 N1(C(Cn2ncc(C)c2)=O)CC(NC(c2c(C)cc(Cl)nc2N)=O)CC(C)(C)C1 c1(OC)ccc(O)cc1C(=O)NCC1(NC(c2ccc(F)cc2F)=O)CC1 c1(C(=O)NCC2C(C(=O)NC3C(CC=C)CCC3)CCO2)nnn(C)c1C C1(C2CCCC2)(C(N2C3CN(C(C(C)CN(C)C)=O)C(CC3)C2)=O)CCNC1=O c1(C(=O)NC2C(NC(=O)C=Cc3cc[nH]c3)CCCC2)cccn(C2CC2)c1=O c1(C(=O)NC(C)CCNC(C2(F)CC=CCC2)=O)cc2c(O)ccc(F)c2[nH]1 N1(C(CC(C)C2CC2)=O)CCCC(C2CN(C(C34CC(C3)C4)=O)C2)C1 C1(C(N(CCCCC(=O)N(C(C(C)C)C)C)C)=O)CCC2(CCC2)C1 N1(C(C(CCCC)NC(c2ocnc2C)=O)=O)CCOCC2(CCC2)C1 N1(C(C2(SC)CC2)=O)CCC(C(=O)NCCc2cccnc2O)C(C)(C)C1 C(=O)(C(C)CS(C)(=O)=O)N(C1CCN(CC(N2CCCCCC2)=O)CC1)CCC N1(C(C2C(CNC(c3ccn(COC)n3)=O)OCC2)=O)CCC2(CC1)CC2 c1(OCC)cccc(C=CC(=O)N)c1.C1(C(N(CCC)C)=O)CCCCC1 N1(C(c2cc(C)[nH]n2)=O)CCC2(NC(C3CN(CC(C)C)C3)=O)CCCCCC12 C12(NC(CCCSC)=O)CC(CO)(C1)OC21CCN(C(=O)CC2CC2(C)C)CC1 c1(CNC(C(C)N(C(=O)CC)CC)=O)cnc(C)o1 N1(C(CCC(C)OCC)=O)CCCCC(CNC(=O)C(O)CSC)C1 C1(C(=O)NC(C)CC(C)NC(=O)CC23CCCN2CCC3)CC2(CCOCC2)C1 C12(C(N3CC(NC(=O)C=Cc4cnc[nH]4)C3)=O)CCC(CF)(C1)OC2 Cc1n[nH]c(C)c1C(=O)NCCN(C(=O)C(c1cccc(Cl)c1)N(C)C)C C(=O)(C(C)CC(F)F)NC(CC#C)C(=O)N1CCC(COCC)C1 C(=O)(CCS(C)=O)N1CC(O)(C(C)NC(C(F)OC)=O)C1 C(C)(CC(=O)N(CCC(=O)N(C)OC)OC)C(CC)SC C=CC(C)(O)CC(=O)NC1CCN(C(c2sc(C)cc2OC)=O)CC1CC c1(C(N2CCC(N(C(=O)C(C)OCCC(C)C)CC)C2)=O)cc(O)n(C)n1 c1(C(N2CCC(NC(c3cc(C(F)(F)F)on3)=O)C2)=O)cc(Cl)ccc1O N1(C(c2[nH]c3cc(C)oc3c2)=O)CCC(C2CCCN(C(=O)C3CC3)C2)C1 N1(C(C23CC2C3)=O)CCCC(NC(C2(c3ccccn3)CC2)=O)CC1 C(=O)(C(CC)C(=O)OC)N1C(C=CC(=O)NC(CCCC)(C)C)CCC1 C1(C=O)CCC(C(N)=O)CC1.c1(C(N(C2CCC2)C)=O)cn(CC(N)=O)nn1 CCCCCC(=O)N1CCC(C(=O)NC(c2ncc(C)cn2)C)O1 c1(C(=O)NC(CNC(C(C(C)C)(C)O)=O)CC(F)(F)F)ccc2nsnc2c1 CC(C(C)(C)C)=CC(=O)NCC1CC1.c1ccccc1.C(=O)CC1CC1 N1(C(c2n[nH]c(C)c2C(F)(F)F)=O)CC2(CCN2C(=O)CC2CCCOC2)C1 C1(C(=O)OC)CN(C(C2CCCCC2C(N)=O)=O)C2(CCOCC2)C1 c1(OC)cccc(C(N2CCCCC2c2n[nH]c(C)n2)C(=O)NC2CCCC2)c1 C(=O)(C1=CCN(C(=O)C=CC2CC2)C1)NCC1C(C)C1 c1(C(N2C(C(N3C(C)(CCC)CC3)=O)CC2C)=O)cc2n(n1)CCC2 C1(CC=O)CCCN(C(C2CCCC(=O)C2)=O)C1.C1(C(=O)OC)CC1C.N C=CCC(CNC(=O)CCS(C)(=O)=O)C(=O)NCCCNC(=O)C(C)C CN1CC(NCc2ccc(Cn3ccnc3)o2)CCCC1=O CC(C)C(C)(O)CNC(C1CC(=O)CN1C(=O)COC1CCCCC1)=O c1(C(=O)NCC(C(C)(C)C)NC(C2CC3CC2CC3O)=O)ccc(F)cc1Cl C1(NC(c2ccn(CC)n2)=O)C2CC3CN(C(=O)CN4CCCC4)C1C3C2 Cc1cc(OCCC(=O)NCCCCN(C(=O)C#CC(C)(C)O)C)c(C)c(C)c1 c1(C(=O)NCCCCC(C)NC(c2cc(C)oc2)=O)cccn(C2CCC2)c1=O N1(C(C2(CCC)CC2)=O)C2CCCC1CC(CNC(c1ccn(C)n1)=O)C2.N c1(OC(CC(CNC(COCC#C)=O)O)=O)cc(C)cc(F)c1 N1(CCOC)CC(C(=O)NCC(C)CNC(c2c[nH]nc2C)=O)CC1=O c1(C(N2CC(OCCNC(CN(C)CCO)=O)C2)=O)csc([N+](=O)[O-])c1 CCS(=O)CC(=O)NC1CCCCC1CNC(=O)C=CCN1CCCC1 N1(C2CCC(NC(c3cc(C)ns3)=O)C2)CCN(C(c2cccnc2S)=O)CC1 CCC(C)C(C(=O)NC)NC(c1ccc(=O)n(C)c1)=O.c1c[nH]nc1C(C)C CCCC(CC)CCC(=O)NC1(C)CN(C(=O)C(c2cccc(OC)c2)O)C1 c1(C(=O)NC(CC=C)CNC(c2cc(C(C)=O)cs2)=O)c(C)ccnc1O C(CCC(=O)NCC(CNC(=O)C(C)NC(=O)OC)OC)=CCC=C C1(NC(C(C)=CC)=O)CC(NC(c2ccncc2N)=O)C12CCC2 C1(NC(C=C(CC)CC)=O)CC(C)CN(C(c2cncc(C#N)c2)=O)C1 C1(NC(CCCCNC(c2cnn(CC)c2C)=O)=O)CCC(C)(C)C(C)C1 C1(C2CC2)(CNC(C(CCSC)N(C)C)=O)CCN(C(c2cccc[n+]2[O-])=O)C1 N#CC1(C(=O)NC2CCCC2CNC(C2CCCC(=O)N2)=O)CCSCC1 c1(CNC2CC(CC(=O)Nc3cccc(Br)c3Cl)C2)ccc(Cl)cc1[N+](=O)[O-] N1(c2nnc(COC)s2)CC(NC(=O)C(c2cccc(Cl)c2)(C)C)C(C)C1 C1(N(C)C)CCCC1NC(=O)CCNC(=O)C.C(=O)C(C)(C)C1CC1.N Cc1c(NC2CCCCN(C(C)C)C2)ncnc1NC(c1ccsc1)C C(C(C)(O)CC(=O)NC1(CO)CCN(C(=O)CCCn2ccccc2=O)C1)OC c1(C(C=O)(C)C)ccc(F)c(F)c1.C(C(O)C(=O)NC1COCC1C)=CC N1(c2n(C)ncn2)CCC(NC(=O)NCS(C)(=O)=O)CC1 c1(OC)ccc(CN2CCOCC2CC(=O)Nc2cc(I)ncn2)c(C)c1C O=C(CCCN1CCCCC1)NCCC1(NC(c2cc(C(F)F)cs2)=O)CC1 C(=O)(CCCC(F)(F)F)N(CC(C)(C)C)CC.C(=O)C(O)CN1CCOCC1.N C12(NC(c3c(C)cns3)=O)CCC(CC1NC(c1cc(Br)cn1C)=O)C2 Cc1cc2sc(C(=O)NC3CC4CCC3C(NC(C3CCC(=O)N3)=O)C4)cc2s1 CC1(C)CCN(C(C23CCCC2(C(N)=O)C3)=O)CC1.C(=O)(CCc1cnc[nH]1)N CCC(N=c1[nH]c2ccc(S(=O)(=O)N(CCO)C3CC3)cc2s1)c1sccc1C n1(-c2ccc(NC(c3c(C)c(Cl)c(Cl)s3)=O)cn2)cc(S(N)(=O)=O)cn1 C#Cc1ccc(C(=O)NC2CC(C)(NC(=O)C(COC)CC(C)C)C2)cc1F CC1(Cc2ccc(Cl)cc2)CCCN1C(=O)COCCn1cc(C(C)O)nn1 C1(C(=O)NC(C2CCN(C(c3nc(C)n(C)c3)=O)C2)C)CC(C)(C)CCO1 N1(C(c2n(C)ncc2)=O)CCC(F)(F)C(CNC(=O)C(O)CC(C)(C)C)C1 C(C(CNC(c1cnc(SC)s1)=O)C(F)(F)F)NC(C1(CC#C)CC1)=O C1(CNC(C2(OC)CC(C(F)F)C2)=O)CN(C(c2ccns2)=O)CCN1C N1(C(c2n(C)nc(C)c2Cl)=O)CCC2(CCC(NC(C3C4CCCCC34)=O)C2)C1 c1(NC)cnncc1C(=O)NCC1CC(C)N(C(C2SCCS2)=O)C1 C1(N(C(=O)CC2CC3(CC3)C2)C)CCN(C(=O)C(c2cccnc2)O)CC1 N1(C(C2CN(CCC)C(=O)C2)=O)CCN(C(c2cc(F)ncc2OC)=O)C(C)C1 CCC(C)(CC)CN=c1cc(NCCCC2CC3CCC2C3)nc(C(F)(F)F)[nH]1 C(c1cccc(OC)c1)=CC(N1C(C(=O)NCCCOCC)CC2CC21)=O C1(CC(=O)N)CCCCC12CC2.CN1CCCC1C(=O)NCc1nc(C)cs1 C=C1CCC(C(=O)NCC(C2CCCCC2)NC(c2snnc2CCC)=O)CC1 C(=O)(C1=NOC2COCC12)N1C2CC(C(=O)NCC(c3ncc[nH]3)C)(OCC2)C1 c1(C(=O)NCC(c2ccco2)N(C)C)cccc(NS(=O)(=O)C(F)(F)F)c1 Cc1[nH]ccc1C(=O)NC(CC1CCCC1)C(=O)NC(C)CN1CCCC1=O CCCCC(CC(=O)N1CCN(c2ccncc2)C(C)C1)OC c1(CC(N2CC(NC(C(C)N(C)C)=O)C2)=O)c[nH]c2cc(Cl)ccc12 CC1CCN(C(c2ccc(NC(N)=O)cc2)=O)CCN1C(=O)C(F)CC1CC1 c1(C(COC(c2ccc(COC)[nH]2)=O)OC(C)C)ccc(C)cc1 CC(CC(=O)NCC1(O)CCN(C(C2CCC(C)(O)CC2)=O)CC1)C(C)(C)C C=CC1(C(=O)NC(C)CN(C)C(C2CCCS2(=O)=O)=O)CCOCC1 c1(C(N(C(CCNC(CC2(OC)CC2)=O)C)C)=O)cnc2c(c1)nnn2C C(=O)(CCCCCCSC)N1CCCC(C)(CNC(C(CSC)OC)=O)C1 CC1CCC(NCc2ccc(-n3cccn3)cc2O)Cc2ccccc21 S(=O)(=O)(c1ccc2c(c1)CCN2)NCC1(CC)CCCCO1 Cc1cccc(CC(N2CCC(CNC(=O)C(C)c3ccsc3)CC2)=O)c1C C(=O)(C1=CCCSC1)N1CC2C(NC(=O)Cc3cnccc3C(F)(F)F)C2C1 C(CC(C)C)(C(=O)NC(CO)C(C)NC(c1n[nH]cc1C)=O)OC C(=O)(CC(C)(C)C)N(CCCNC(C1CCS(=O)CC1)=O)CC.C(N)=O C12CCCC1(F)CN(C(=O)C=C1CCN(C)CC1)C2.C(CCC)(C(=O)N)=CCC c1(C(C)NC(N2CCC(N3CC(C)(C)C3)C2)=O)cc(F)ccc1F c1(C(=O)NCC23C(CN(C(CC(C=C)(C)O)=O)C2)CC3)c(C)ccc(C)c1C N1(C(c2n[nH]c(C)c2Cl)=O)CCC(CNC(C2CCC3CC2CO3)=O)C12CC2 C=C(C)CCC(=O)N1CC=CC(NC(c2nc(C)oc2OCC)=O)C1 C1(NC(C2(SCC)CC2)=O)CCC2CCN(C(=O)C(C(C)C)C(C)C)C1C2 C(CN=C(NC1CN(C)CC1O)N1CCC(C(C)C)CC1)OCC C1(C)(CC(=O)NC2CC(C)(C(N)=O)C2)CCN(C(C2CC=CC2)=O)C1 CC(C)(C)CN=C(NCC1(S(C)(=O)=O)CCC1)N1CCOC2(CCCCC2)C1 c1(-c2nc(-c3c(C)c(Cl)cnc3)n(CCC(C)C)n2)cc2ccccc2o1 C(=O)(C1CCCc2n[nH]cc21)NC(CC)(CNC(=O)CC1CC1(Cl)Cl)CC C1(CC(N2CCC(CC=C)(NC(=O)C(C)O)CC2)=O)CCn2cncc2C1 c1(CNC(c2c(CNC(c3ccco3)=O)cco2)=O)nnc(O)nc1O.C [SH](=O)(=O)c1n[nH]c2nc(C)cc(C)c12.c1(C(=O)OCC)nc(SCC)oc1C CCC(C)(C)C(C(=O)NC1CCCC(NC(c2cc(C)c[nH]2)=O)C1)OC c1(CC)ccc(C)cc1C(N1CC(NC(c2nc(Cl)cs2)=O)C(C)(C)C1)=O c1(C(CC(=O)N(CC(C)NC(c2cc(CC)no2)=O)C)C)ccccc1OC C(=O)(C(C)CCc1cccc(F)c1)N(CCNC(Cc1cn(C(C)C)nc1)=O)C C(=O)(N(CCC(=O)NCc1cncc(F)c1C)OC)C1C(C)(CC)C1 Cc1sc(C)c(C(=O)NCC2(C)CCCN2C(C2CCN2C)=O)c1C N1(C(C(C2CCC(=O)N2)C)=O)CCC(C)(C)C1.N1(CC=O)CC(=O)N(C)C1=O C1(NC(CSCCOC)=O)CC2(CCN(C(=O)C(C)(C)CCOC)C2)C1 N1(C(CC2(OC)CC2)=O)CCCC(C2CCCN(C(c3c[nH]nc3C)=O)C2)C1 C(=O)(CC1=CCCC1)NCCC1(OC)CN(C(=O)Cc2sc(C)cc2C)C1 Cc1cc(C(=O)N(C2CCN(CC(N3CCNCC3)=O)CC2)C)cn1C(C)C S(=O)(=O)(c1c[nH]ccc1=NC1CCSc2ccc(Cl)cc21)N1C(C(C)C)CCC1 C(=O)(C1=CCC(F)(F)CC1)NCC1CC(OC)CN1C(c1ccc(C)o1)=O c1(C(N2CC(C(N3CC(C)OCC3)=O)C(O)CC2)=O)cccc2c1CCN2C O=C1CC(C(=O)NCCC2(O)CCCN(C(C3(Cl)CC34CCC4)=O)C2)=NN1 c1(C(C)=O)c[nH]c(C(=O)NCCNC(=O)CSC2CCCCO2)c1 c1cnn(C)c1C#N.C1(C(C)N(CC(C)C)C=O)CN(C=O)C1.C(C)(C)C C(=O)C(O)C1=CCCCC1.C(=O)(CCc1cn[nH]c1)N.C(=O)(CC1CC1)OC C=CCC(C)C(=O)NCCC(C)CCNC(c1ccc(NC(=O)NC)cc1)=O C(CCCS(=N)(=O)c1ccccc1)NC(CCc1cc(C(C)=O)c(C)o1)=O CCC(O)C(C)C(=O)NCc1nc(C)c(C(N2CCCCC2CF)=O)o1 c1(CCC)cnnc(C(N2CCC(CNC(C3(C)CC3(F)F)=O)C2)=O)c1 C1(C(=O)N)CC2(CCN1C(C1CN(C(C)C)C1)=O)CC2.CCCCN1CCCC1 N1(CCNC(c2ccc(CNC(=O)Cc3ccsc3)o2)=O)CCCNC1=O c1(C(=O)N)cc(O)cc(O)n1.c1(C(N2CC(C(N)=O)(C)C2)=O)cncc(F)c1 CCCC(F)(F)C(=O)N(CCCOCCN(C)C(c1cnoc1C(C)C)=O)C Cc1cnn(CC(N2CCCC2C(C)(C)NC(=O)Cc2cc(C)on2)=O)c1 c1(C(=O)NC2CN(C(C(CC)F)=O)C2)cc(C(C)C)nc2ccccc12 c1(NC(C2CN(C(C=CC=CC)=O)CC(F)C2)=O)cc(Cl)c(Cl)cc1O C1(C(N2CCCC(C)C2)=O)CC(C(C)(C)C)=NO1.C(CC(=O)N)N(CC)CC c1(CC)ccc(NC(=O)C(C)(C)C2CCCN2C(C23CC(C2)C3)=O)cn1.C N1(c2cc(OCC)ncn2)CCC(C)C(NC(=O)C(C)SC(F)(F)F)C1 c1(C(=O)NC2(CC=C)CCN(C(=O)C(C)(C)C=C)C2)cc(C)c(C)cc1C CC1(C)CC(C)N(C(c2cnn(CC(F)F)c2)=O)C1.C1(C)(C=O)C=CCCC1.N C1(O)(CNC(c2c(C)noc2)=O)CCN(C(C2CC(=O)C2C)=O)C1 C(=O)(C(C)N(OC)C(=O)CN(C(C1CC(O)CN1C)=O)C1CC1)OC C(C)(C(N=c1ccc(C#N)n[nH]1)C(C)C)NC(C(=O)Nc1c(C)ccc(C)c1)=O c1(OC)ccc2ncc(C(N3CC4CC3CCC4C(=O)N(C)C)=O)n2n1 C(=O)(CCC(F)(F)F)N(CCC)C.c1(C(C)NC(=O)NCC=O)ccccc1 C=CCN=C(NCCc1cc(C)no1)N1CCC(c2ccccc2)(C(N)=O)C1 C(=O)(C1=CCC(C)CC1)N1C2(CNC(C(CC)(C)OC)=O)CC(C1)C2 C12(CNC(C3(C)COC3)=O)CCCC1CN(C(=O)C=Cc1ncco1)C2 C(=O)(C(C)(C)CC(F)(F)F)N1CCCC(CNC(C=C(C)C(F)F)=O)CC1 C1(C(N(C2CN(C(C(CC)N3CCCC3=O)=O)C2)C)=O)Cc2nnsc2S1 C(C)(CSC)(C=O)NC(CC1C(CC)C1)=O.C1CCCC1C=O.C1CC1 C1(NC(c2c(C)n(C)cn2)=O)(C)CCC(F)(F)CC1.C(=O)(C(C)n1ccnc1)N c1(C(=O)NC2C(NC(C(c3ccccc3C)OC)=O)C2)cc(C)c(C)cc1Cl c1(CC)[nH]c(C(=O)NC2CC(CNC(=O)Cc3cccs3)C2(C)C)nc1Cl c1(C(CN(CCCC(C)O)C)O)cccc(C#N)c1 c1(OCC(CNC(c2ccc(-c3nnc(C)nn3)cc2)=O)O)cccc(Cl)c1Cl N1(C(C(C)O)=O)CCC2(CC1)CC(NC(C1OCC3CCCCC13)=O)C2 N1(C(c2cc(C(=O)OCC)n[nH]2)=O)CC2CC1CCC2.c1(C(=O)N)snnc1C C1(C=O)C=CC=CC=C1.C1(CCOCC)(C(=O)NC2CCC2)CCCC1.N N1(C(C(CC)N(C)C)=O)CCC(C)(C)C(NC(C2CN(C)C2)=O)C1 c1(C(=O)NC(CNC(=O)C(O)C2CCC2)CO)ccc(Br)cc1.C1CC1.O N1(CC(C)C)CCCC1CSc1nc(-c2ccccc2)cs1 C1(C(=O)NC(C(=O)OC(C)C)C)CCN(C(C2CC3(CC3)CO2)=O)CC1O c1(COC(=O)NC2COC(=O)C2)ccccc1Br CCCCCCC(C)c1nc(-c2ccoc2)nn1Cc1cccc(OC(F)F)c1 S(=O)(=O)(c1ccc2nnn(O)c2c1)Nc1ccc(C)cc1C(=O)N(C)C CCCC(CCC)C(=O)N1CCN(C(C2(S(C)(=O)=O)CC2)=O)CC(O)C1 Cc1nc2c(s1)CN(C(=O)Nc1cc(C)n(C3CCCCC3)c1C)C2 c1(C(N2C(C(N3CCC(=O)NCC3)=O)C=CCC2)=O)cc2ccccn2n1 N1(C(C23CC(COC)(OC2)C3)=O)CCCCC(CNC(C2CCC2)=O)C1 C1(C)(NC(Cc2c(C)noc2C)=O)CCN(C(=O)CC2COC(=O)C2)CC1 C1(NC(=O)Cn2cc(C3CC3)cn2)CC2(C1)CC2C(=O)NC(CO)CCO O=C1CC2CCC(CN1)N2C(c1csc(CNC(=O)Cn2ccnc2)c1)=O C#CC1CCCN1C(=O)CCOCCN(C(=O)Cc1cnccc1C)C C1(C)(CC(=O)NCC(CNC(C(C)OC)=O)CO)Oc2ccccc2O1 N1(C(c2c(C)ccc(F)c2)=O)CCC2(CC1)CN(C(=O)C(C)CC1CCCO1)C2 C(=O)(C1=CC(O)CC1)N1CCC(NC)CC1.C1(CC=O)CCC1.C(C)=O.CC c1(C=O)ccn(CC(F)F)c(=O)c1.C1C=CCN1C(=O)Cn1nnc(=O)[nH]1.N C1(=CC(=O)N)C2CC3CC(C2)CC1C3.C1(OC)(C)CN(C(=O)C(C)C)C1 C12(C(=O)NC3C(C)N(Cc4ncnn4C(C)(C)C)CCC3)CCCCC1OCC2 C1(C(N(CCC)C)=O)Cc2nnc(C)n2C1.CC(C(=O)N(C)CC)=C1CCC1.O N1(C(=O)C=CCO)CC2=C(C1)CN(C(C1CCC1Cc1ccccc1)=O)C2 N1(C(c2nc(C(N)=O)sc2)=O)CCN(C(=O)CC2CCOC2)C(CF)C1 Cc1n[nH]c(C)c1S(=O)(=O)N1CCc2sc(C(=O)Nc3cncc(Br)c3)cc2C1 CCC(CC(=O)NC1CC(NC(c2cccc(F)c2SC)=O)C1)C(C)C N1(C(COCCC=C)=O)CCC(N(C)C(c2csc(C)c2OC)=O)C(C)C1 C1(NC(c2ccc(SCC)nc2)=O)CCCCCN(C(=O)Cc2conc2C)C1 c1(OC)cncc(C(=O)NC(C(=O)NCc2cnns2)C2CC2)n1 c1(C(N2CC(CNC(C3CCC(C)O3)=O)OCC2)=O)csc2nccn12 c1(C(=O)NCCN(C(CCC=C)=O)CC2CC2)ccnc2cc[nH]c12 C=CC(CC)C(=O)N1CCC(Cn2cc(-c3cccc(Cl)c3)nn2)CC1 N1(C(c2cccc(N(C)C)c2)=O)CCC2C(CCN2C(=O)C2=CCSC2)C1 Cc1oc(S(N)(=O)=O)cc1C(=O)NC1CC1.c1(C=O)nc(C(C)C)oc1C CC(C)C(CNC(=O)CCCNC(c1cnc(Cl)n1C)=O)C(C)C c1(C(=O)NCCC(C)N(C(=O)CN2CCOCC2=O)C)cc2ccncc2[nH]1 CC(CC1CCCC1)C(=O)N(C)CCNC(C12COCC1C2)=O c1(C(=O)NCC2COCC2NC(C2(Cl)CC23CCC3)=O)cc2ccccc2s1 c1(C(N2CC(CC)N(C(C3CC4(CCO3)CC4)=O)CC2)=O)cc2c([nH]1)CCCC2 C(=O)(C(C#N)C(C)(C)C)N(C(C)C(=O)NCC1(CCO)CCC1)CC N(C)(S(=O)(=O)N(C)C)CC=O.CCCCCCNC(c1c[nH]c(=O)cn1)=O.N C1(C(=O)OC)(OC)CCC(SC2CN(C(=O)C=C(C)C)C(=O)CO2)CC1 CC(C)CCC(=O)NCCn1cc(CNC(C2(C)CCCCO2)=O)nn1 O=C1CCc2ccc(C(N3CC4C(NC(C5C6COCC56)=O)C4C3)=O)cc21 C1(C=O)CCC2(CCCCC2)C1.c1(CC)oncc1C(=O)NC1(C)CCOC1.N N1(C(c2c(C)n(C(C)(C)C)nc2)=O)CCCN(C(=O)C(C)C#N)CC1C c1(N(CCN(C(C)C)C)C)cc(Cl)c(O)nn1.C1CC(C)(C)C1C(F)(F)F Cc1nc(C)c(C(N2CC(c3nocc3C)C2)=O)s1.C12CCCN1C2=O c1(N2CCCCC(CO)C2)nccc(=NC2CN(C3CC3)C2)[nH]1 N1(C(CC(OCC)O)=O)CC(C(=O)N(CC(F)F)C(C)C)CC(C)(C)C1 N1(C(CCSCCC)=O)CC(CNC(=O)C(O)CC)CC(F)C1 c1(NCC2C(C(F)(F)F)CCN(C(=O)C3=CCC3)C2)nc2cc(Br)ccc2o1 C1(C(N(C(C(=O)N(CC(CN(C)C)O)C)C2CC2)C)=O)CNC(=O)N1 Cc1cc(C(=O)NC2(CC)CC2)cn1C.c1(C2C(C(=O)N)C2)cccc(Cl)c1 Cc1nccc(Cl)c1C(N1CC(C)OC(C(F)(F)F)C1)=O.C(=O)C=CCO.N c1(CC(=O)NCC#CCNC(C=CCN(C)CC)=O)ccc(Br)cc1 C1(C(CCO)NC2CC(CNC(=O)OC(C)(C)C)C2)CCCCC1 c1(CC)cccc2c(C(N3CC(NC(=O)COCCCOC)CC3C)=O)c[nH]c12 c1(OC)cc(Cl)cc(CN2CCC(C(=O)NC(c3cccc(Br)c3)CO)C2)c1O c1(C(N2CC(NC(CC(=C=C)C)=O)C3C2C3)=O)csc2ccccc12 c1(OC)nccnc1NC1CCN(Cc2ccnn2C2CNC2)C1 CC(C)(CF)C(=O)NCC(Cc1ccccc1)NC(C1C=CCCC1)=O c1(CC=C)ccc(OC(=O)CN2CCC2C2CCCCCC2)c(OC)c1 CCCCCC(F)C(=O)N1CC=CC1(C)C(=O)NCC(CO)C(F)(F)F C#Cc1cc(C(=O)N(C(C)CN(C(=O)CCSC)C)C)ccc1Cl CCCCC(CC)CC(=O)N(CCC(=O)NC(C)CC(F)(F)F)CCO C(=O)(C(C)CC1CCC1)NC1(CC(=O)NC(C#C)CC)CC1 Cc1[nH]c(=NCc2ccc(OCC(F)F)cc2)ccc1CO CN1CCC2CCN(C(=O)C(=O)NCc3cccc(SC(F)(F)F)c3)C2C1 N1(C(C2(C)CCCN(CCc3n(C)ccn3)C2)=O)CCCC12CCCNC2=O C1(NC(C(C2CCCCCC2)OC)=O)(CO)CCN(C(=O)CC(=O)N(C)C)C1 C(=O)(CC1CC(=O)Nc2ccccc21)NCCCCCNC(=O)CCC(F)(F)F C(=O)(C(CC)CC(C)C)NCC1CCN(C(c2c(CCC)n(CCO)nc2)=O)C1 C12(C(=O)NC(C)CC3CCC3)CC3CC(C)(C1)CC(C)(C3)C2 CC(C)(C)C(CNC(C1CC(=O)CS1)=O)C(=O)N1CC(=O)NC2(CC2)C1 c1(OC)ccnc(C(=O)NC(CN(C(=O)Cc2ccno2)C)(CO)CO)c1F Nc1ccccc1CCCC(=O)N1CC(=C(F)CNC(=O)C=CBr)C1 N1(C(c2c(C)ccs2)=O)CCCC(CNC(c2cc(Cl)ccn2)=O)CC1 CCCCC(C)CCC(=O)N1CCN(C)C(CNC(C2CC(=C3CC3)C2)=O)C1 C1(C(=O)NCCC(C)(C)c2ccccc2)CCCC(N=c2cncc[nH]2)C1 N1(C(CNC(CC)=O)=O)CCN(C(C2C=CCC2)=O)C(c2ccncc2)C1 C1(NC(C=CCN(C(=O)C(c2ccccc2)F)C)=O)CC2CC1CC21CC1 C1(C(N(CCCC)CCCC)=O)CCN(C(c2cc(C)cc(Br)c2)=O)CC1O N1(C(c2cc(OC)nc(C)c2)=O)C2CCC1C(C)C(NC(C1CC=CCO1)=O)C2 C1(CC=C)(NC(c2cc(CC)no2)=O)CCN(C(=O)Cc2csnn2)C1 c1(OC)cc(C)c(COC(c2cccnc2N)=O)cn1 c1(C(N2C(CCCNC(C3C(=C)C3)=O)CCC2)=O)cnc2c(c1)ncn2C c1(OC)ccc(C(=O)NC2(C(=O)O)CCC(C)CC2)cc1[N+](=O)[O-] N1(C(c2cc(C)nc(C)c2)=O)CCC(C(=O)NCCc2cnc(C)[nH]2)C12CCC2 c1(N(C)C)cc(NC(c2cc(F)cs2)=O)ccc1Cl C(=O)(N1CCC(C(=O)NCc2cc(C)ncn2)O1)c1[nH]cc(C)c1 N1(C(C(C)Cc2cnc[nH]2)=O)CCCCC1.c1(CC(=O)N(C2CC2)C)nccs1 C12CC1CN(C(=O)CCc1csc(=N)[nH]1)C2.C1(CC(C)C)(C(=O)N)CCCC1 CCS(=O)(=O)CCn1cc(NC(CNC=O)C2CC2)cn1.C(C)(C)C.O C1(N(C(c2c(CC)ncs2)=O)C)CCN(C(=O)CCC2CCCC2)CC1C N1(C(C(COC)OC)=O)CCC(C(=O)NCC2CCC(C)CC2)=C(F)C1 C1CC2(CCC2)CN1C(=O)C1=CCCC1.c1(C(=O)NC)cc(-c2ccoc2)on1 C1(CC(=O)NC2CCN(C(c3ccc(C(N)=O)o3)=O)C2)NC(=O)CNC1=O c1(OCC(=O)NC(CN(C(CC(CC)OC)=O)C)(C)C)c(C)cc(C)cc1C c1(C(NCCCNC(C2(O)CCC(CC)C2)=O)=O)cccc2nc(O)[nH]c12.C CC(=O)C(C)CC(C)C(=O)N(C(C)C(N1CC2CCCC(C1)N2C)=O)C Cc1nn(C)c2c(NCC(C)(C)CO)nc(N3CCC(CC(F)(F)F)C3)nc12 Cc1nc(=N)[nH]c(C)c1C(=O)NC.C1CC2CCC1N2C(=O)CCn1ccnc1 Cn1ncnc1CCNC(=O)CC1CC(NC(=O)CCc2nc[nH]n2)C1 c1(CN(C)C(c2cccn3c(Br)cnc23)=O)ccc2cnccc2c1 CN1CCN(C2(c3ncon3)CC2)CC1.C1CCN(C(c2cn(C3CC3)cn2)=O)C1 O=C(C1=CCSC1)NCC1OCCC1C(=O)NCCCN1CCCCC1 c1(OC(C)C)nccnc1-c1nc(-c2cncc(Cl)c2)n(COC2CCOC2)n1 c1(C(=O)NC2C(Nc3ncnc(CC)c3F)CCCC2)ccc([N+](=O)[O-])c(OC)c1 C1(CNC(c2ccc(C(=O)O)c(Cl)c2)=O)CCN(C)CC1(F)F.C[SH](=O)=O N1(C(CCc2c(C)c[nH]c2C)=O)CC2CCN(C(=O)C(=O)c3ccco3)CC2C1 N1(C(CCC=C)=O)CCC(OCCCNC(c2scnc2CC)=O)CC1 N1(C(C=C(CC)C)=O)CC(N(C)C(c2cc(CC(C)C)nn2C)=O)C2(CC2)C1 C1(NC(C2(CN=[N+]=[N-])CCC2)=O)COC2(C1)CN(C(=O)C1=CCSC1)C2 C(=O)(C(CCC(N)=O)n1cc(-c2cccs2)nn1)NCCCOCC N1(C(c2cnc(CNC(Cn3c(C)ncc3)=O)nc2)=O)CCCC2(CCCC2)C1 N1(C(C(N2CCCC(O)C2)C)=O)CCC(O)(CCNC(=O)C2=CCCSC2)CC1 c1(C(N(C(C)CNC(C2(C)CCN(C)CC2)=O)C)=O)n[nH]c2c1CC1CC21 Cc1cc(C(N2CCC(C(F)(F)F)C(NC(C3COC3)=O)C2)=O)n2nccc2n1 C1CS(=O)(=O)CC1.c1cn(C)nc1C=O.CC(F)(F)F.C(=O)C.COC C(=O)C1=CC2CC=CCC12.c1(NC(=O)NCC#CC)ccccc1.O=C1CN1 N1(C(CN(C(C(CCSC)O)=O)C2CC(C#N)C2)=O)CCC12CCCSC2 C(=O)(CC(C(F)F)n1cccn1)NC1CN(C(COCCCOC)=O)C1 N1(CC(=O)N(C)CCOCC)CCOCC1=O.C1(O)(C(C=O)F)CCCC1.N N1(C(c2cc(C(F)F)[nH]n2)=O)CCCCC(C(N2CCC2C2CCC2)=O)C1 c1(C(N(C2CCN(C(C3(N(C)C)CC3)=O)C2)CCC)=O)ccc(CO)nc1 c1(C(N2CCCC3(NC(CCOCC)=O)C(C2)C3)=O)ccc(Cl)cc1[N+](=O)[O-] c1(CNCC2(F)CCN(C(C(OC)OC)=O)CC2)ccc(O)c([N+](=O)[O-])c1 Cc1cc(C(=O)NC(CC2CCCC2)C(=O)NCCP(C)(C)=O)c(C)[nH]1 CCCCC(CC)CC(=O)NCc1cc(C(=O)NCCC#CCO)co1 c1(C(C)=O)c[nH]c(C(N2CCC(C(C)C(=O)NCCCc3cccs3)C2)=O)c1 C1(CC(C)C)(C(=O)NCC(CC)NC(c2n[nH]c(C)n2)=O)CCNC1=O N1(C(=O)COCCc2ccc(Cl)s2)CCCN(C(C2CCC(F)C2)=O)CC1 c1(C(=O)NCC(CC)N(C)C(c2cnn(C)c2C)=O)sccc1C#N c1(CC)ccc(C(=O)NC2(CNC(=O)C(C)O)CC2)c(O)c1 C1(C)(C(N(CC(CN(C)C(c2cccc(Cl)n2)=O)O)C)=O)CCNC(=O)C1 S(=O)(=O)(c1[nH]c(=NCCc2cccs2)ccc1Br)N1CCC(C)(C(N)=O)C1 C(=O)(C(O)(CC)c1ccccc1)N1CC(O)(CNC(COC(CC)C)=O)C1 N1(C(C(C)n2cccn2)=O)C2CCC1CC(NC(=O)CN1CCNC(=O)C1)C2 c1(C(N2CC3CC3(C(=O)NCC3CCOC3)C2)=O)cc(Br)cnc1O C1(CNC(=O)CCN2CCC(F)C2)COCCN1C(c1n[nH]cc1C1CCC1)=O CC(CC(=O)NCC1CN(C(=O)CCC(C)(C)C#N)C(C)(C)C1)C(C)(C)C c1(C(N(CCC)CC)=O)cccc(C(N2CCCC2CC(=O)OC)=O)c1 N1(C(C(C)OCC#C)=O)CC(C(=O)NC(C(C)C)C2CCC2)C(CC)C1 N1(C(C2C(CCC)C2)=O)CCOC(CNC(=O)Cn2ncn(C)c2=O)C1 C12(OC)CCC(C=O)(CC1)CC2.c1(CC=O)ccn(C(F)F)n1.CC(C)C.N c1(C(N(C)C)=O)oc2ccccc2c1C.n1(CC#C)cccc1C(=O)NC1CC1 c1(N2CC(C)c3c(cncn3)C2)nc(=NC2CCSC2)[nH]c2c1CCCCC2 N1(C(c2cc(CNC(CC(C)N(C)C)=O)no2)=O)CCC(O)(CO)CC1 C1(NC(COCCC(C)C)=O)CS(=O)(=O)CC1NC(c1scnc1Cl)=O c1(C(=O)NCCC2N(C(C3C(C)C3)=O)CCOC2)c2c(cc3c1CCC3)CCC2 C1(CCC)(NC(=O)C)CCCN(C(=O)C(C)CN2CCCCC2)C1.CC(N)=O.S C1(C(=O)OCC)CCCCN1C(C1CCN(C(c2cccc(O)n2)=O)CC1)=O C1(NC(=O)C(c2ccc(F)cc2)F)CC12CC(NC(C13CC(C1)C3)=O)C2 Cc1ccc(CNC(=O)CC2CCC(C)C(C)C2)c(O)n1 c1(OC)ccc2c(c1)N(C(=O)CCc1cc(F)ccc1F)C(=O)C(C)=NN=N2 c1(OCC#CCNC(N(C(C)C)CC)=O)csc(C)c1 c1(NC(C(c2occc2C)N(CC(=O)N(C)C)CC)=O)ccc2c(c1)OCCO2 c1(C(=O)NC2COCCN(C(CC(C=C)C)=O)C2)coc(S(N)(=O)=O)c1 N(C(=NCc1csc(C(C)C)n1)N1CCCC(NC(=O)N(C)C)C1)C(C=C)C C(=O)(N1CCC(C(=O)N(C)CC2CCOCC2)O1)c1n(CC#C)cnn1 C1(CC(C)NC(CCc2c(C)ncs2)=O)CCN(C(c2cocn2)=O)CC1 Cn1c(NC2CC(NC(=O)CCC3CC(F)(F)C3)C23CCC3)cc(O)nc1=O Cc1ccc(SCCC(=O)NCC(O)CNC(=O)CC)cc1.CCN(C)C.O c1(C(=O)NC(CC(C)NC(CCC=C=C)=O)C)c(CC)nc2ccc(Cl)cn12 CC(C)(C)C(=O)NCC(O)CNC(c1ccc(Br)s1)=O C1(CC)C(=O)N(C)CCN1C(C12CC1CN(C(=O)Cc1cccnc1F)C2)=O C(=O)(C(C(C)C)NC(C1CC2(CC2)C1)=O)NC(c1nnc(C)o1)C C=CCC(CNC(=O)CCc1cnc(O)[nH]1)NC(=O)C(C)c1cccs1 CC1(CNC(C2CCCC(C)(C)C2)=O)CCN(C(c2cc(Cl)cc(Cl)c2)=O)CC1 C1(CCF)(CN(C)CCOCCC(=O)O)CC(O)C1 c1(N(C)Cc2cncs2)nc2c(c(=NCc3ccccc3)[nH]1)CCC2.[SH](C)(=O)=O Cn1cc(Br)c(C(=O)NC2CCC2NC(C2C=CCCC2)=O)cc1=O N1(C(COCCOCC)=O)CCC(C2CC2)C1.C1(C)(CC(=O)N)CCC1 c1(C(=O)OC)cc(CN(C2CCCS(=O)(=O)C2)C)n(C)c1C C1(C(C(=O)NC2(C)CC(NC(CCOCC)=O)C2)O)CCCCCC1 CCCC(CCCNC(c1cc(Cl)c(Cl)n1C)=O)NC(C1CN2CCC1CC2)=O N1(C(C(C2CCOCC2)OC)=O)C2CCC1C(C)C2.C(=O)(CCSC(F)(F)F)N C(C)(C(=O)N(CCCNC(C1CC1(C)Br)=O)CCO)=CC C12(C(=O)NCC3N(C(C4CCN(C)CC4)=O)CCC3)CCC(F)(CC1)C2 C(CCN(C(=O)Cc1cccs1)C)(C(C)(C)C)NC(c1c(OC)c[nH]n1)=O c1(C(N2CCCC(C)(C)C2)=O)ccc2c(c1)C(=O)NC2.C1(C(=O)N)CCC(O)C1 CCC1=NOC(C(=O)N(C2CCN(C(c3nc(Cl)sc3C(C)C)=O)CC2)C)C1 c1(N2CC3CC(NC(=O)C(c4cccnc4)O)CC3C2)ccc(Br)cc1[N+](=O)[O-] C=CCC(C)C(=O)NC1C=CCCC1C(=O)NCc1cnc[nH]1 c1(OC)ccc(C(C)(C)C(=O)NCC(C(C)C)NC(c2nsnc2O)=O)cc1 c1(C(N2CC(CNC(C(C)N(C)C)=O)C3(C2)CCC3)=O)c(F)ccc2ccoc12 c1(C(N)=O)ccc(C(=O)NC2CC(O)C2CC=O)o1.C1CN(C(N)=O)C1.N C1(NCc2cnn(C)n2)COc2ccccc2OC1 c1(C(CN(C(=O)CN2CCCC(C)(C(F)(F)F)C2)CC)=O)ccc2occc2c1 N1(C(c2ccc(C)o2)=O)CCC(F)C(NC(C2CCCC(O)C2)=O)C1 N1(C(C=CCN(C)CC)=O)CCCC(N(C)C(C2CCCCC(=O)N2)=O)CC1 C(=O)(C1=CCCCO1)NCC1CN(C(CN2CC(C)C2)=O)CC1c1cncn1C C1CC2(CC2)CN1C(=O)CC1OCCO1.O=C(CCCOC1CCOCC1)NC CCC(CC)CC(F)C(=O)N1CC2(CCN(C(c3cc(N)cc(C)c3F)=O)C2)C1 N1(C(=O)CC2(n3cccn3)CC2)CCC2CCN(C(C3CCC3)=O)CC2C1 Cc1ccc2c(C(=O)NC3(C)CC(NC(=O)C)C3)ccnc2c1.C1CCCCO1.S C(=O)(C1CCCc2ncnn21)N1CCOCC(NC(c2ccon2)=O)C1 c1(C(N2C(C(CNC(C(C)NC(N)=O)=O)(C)C)CCC2)=O)cccn2nccc12 C(=O)C(C)(C)S(=O)(=O)C1CC1.C1(O)(C(N2CC(C)CC2)=O)CN2CCC1CC2.N N1(C(C2N(C(=O)NC)CCC2)=O)CC2C(NC(=O)CCn3cccn3)C2C1 N1(C(CC(=O)NCC#C)=O)CC(N(C(=O)CCC2CC2(F)F)C)C(O)C1 CC1CN(C(=O)C2=CCCCO2)CCC1CNC(=O)C=CC1CCCC1 S(=O)(=O)(CCC(=O)N(CCC(C)NC(=O)C)C)NC.c1ccc(F)c(Cl)c1.O c1(NC2CC(C(N)=O)OCC2)ccc(C(F)F)cc1F c1(NC(c2c(NC(C=COCC)=O)nc(Cl)cc2)=O)cnnc2ccccc12 CC(C)CC(C(=O)N1CCC1CNC(c1ccccc1C(F)F)=O)n1ccnc1 C1(C(=O)NC2C(NC(C3(C)CSC3)=O)CC2)C=CCCC1 Cc1cn2c(C(=O)N3CC(n4cc(-c5cnn(C)c5)nn4)CO3)c(C)nc2s1 N1(C(c2cncc(C)c2)=O)CCC2CN(C(=O)C=Cc3ccoc3)CCC12 N1(C(C2CCC(CCCC)CC2)=O)CC2(CCCCN2C(C2(CCO)CC2)=O)C1 N1(C(c2ccccc2)C)CCC(C#N)(NC(=O)NC(c2cc(F)ccc2Br)C)C1 C(=O)(C(C)(CO)NC(=O)C(C1CCCCC1)F)NC(c1nnc(C)o1)C C(CC)(CCC(=O)NCc1ccnn1CC)NC(C(CC)SC)=O C(=O)(C1OCCn2ccnc21)N1CCC(CNC(C2(COC)CCCC2)=O)CC1 Cc1nn(C)c(Cl)c1C(=O)NC1CC1.N1(C)CCN(C(=O)C)CC1.C1CC1 c1(C(C(=O)NC)N(CC)CC)ccccc1.C1CN(C(C2(C)COC2)=O)C1 c1(C(=O)NC(CN(C(CCCC)=O)CC2CCOCC2)C)cnn(COC)c1C N1(C(C)=O)CC(NC(c2cc(F)c(Cl)cc2Cl)=O)CC2(CCC2)C1 C1(CNC(CCC=CC(C)C)=O)CCCN(C(c2cc(-c3ccco3)cs2)=O)C1 c1(NC(C2C(NC(c3ccc(Br)c(F)c3)=O)C2)=O)c(F)cc(Br)cc1Br N1(C(C2N(CC)CCC2)=O)CCCC(C2CN(C(c3c[nH]c(=N)o3)=O)C2)C1 C12(C(=O)NC(c3cccs3)Cc3ccccc3)COCC(COC1)O2 C1(NC(Cc2ccc(C)c(O)c2)=O)CN(C(=O)Cc2cnn(C)c2)CC1C1CC1 C(CC(C)C(=O)NCC(C(=O)N1CCCC1C(C)O)N(C)C)=CCC c1(C(C)C)nc(NCCC(=O)NC(C)C)cc(=NC(C)c2ccc(C)c(F)c2)[nH]1 c1cccc(C)c1Br.C(=O)(CC(C)C)O.c1(CNC(=O)OC)ccc(C)cc1 c1(C(=O)NC(CNC(C(C=C)O)=O)CO)c(Cl)ccc(Br)c1F C(N=c1[nH]c(N2CCC(C3CC3)C2)nc2c1CCC2)c1c(Br)cn(CC)n1 C(CC(=O)NCC(C)CCO)(C(C)CC)NC(c1nc(CC)oc1)=O c1(CC(=O)NC(C)CCNC(=O)C=C2CCOCC2)cc(Cl)n(C)n1 CC(C)C(CNC(C1CCCCC1C1CC1)=O)N=c1ccc(C#N)c[nH]1 CC1CN(C(c2ccc(=N)[nH]c2)=O)CC1CCNC(c1csc(O)n1)=O c1(C2(C(N3C(c4ncc(C(=O)OC)cn4)CCC3)=O)CC2)ccc(Br)c(Cl)c1 C1(CC=O)CN(C(=O)CN2CCC(F)CC2)CCO1.C1(C(=O)OC)CC(C)C1 CC1(NC(=O)Cn2cc(Cl)cn2)CCN(C(c2nccc(C(F)(F)F)n2)=O)C1 CC(C)CCC(O)C(=O)N1CCCN(C(c2cccn(C)c2=O)=O)CC1C N1(C(C(C)C(C)(F)F)=O)CCC2(C1)CN(C(=O)CCS(C)(=O)=O)CCO2 N1(CCC(C)(C)OC)CC(CO)CCC1C c1(N(C(CNC(Cc2c(SCC)cccc2)=O)C)C)cnc(C(=O)O)c(C)n1 CCCC(C)(C)CC(=O)NCC1CC(C(N2CCC(NC(=O)CC)C2)=O)CO1 C(CCC(O)CO)NC(c1c(CCNC(CC(C)C2CC2)=O)n[nH]c1)=O C1(CNC(=O)C(O)CC(F)(F)F)CC2(CCN(C(=O)CC(F)(F)C(F)F)C2)CO1 c1(N(C)C)ncc(NC(=O)CN(C(C2OCCC2(C)C)=O)CC2CC2)cn1 N1(C(CC(C)SC)=O)CC2CCCC1C2CNC(c1cncc(C)c1)=O C(=O)(C(CN(C)C)N(C)C)N(CC(CC)NC(=O)C=CC1CC1)C c1(CN2CCN(C(CC3CNCC(C)O3)=O)CC2)ccc2ccoc2c1 C1(C(=O)NC2C(C(N(C)CC3CCCCO3)=O)OCC2)CN2CCC1CC2 C(=O)(C(O)C(C)c1ccccc1F)N1CCC(CNC(C=C(CCC)C)=O)C1 c1(C=O)cncc(C(F)F)c1.C1(C(NCC(C)(C)C)=O)C(F)(F)C12CC2 Cc1ccc(CNC(=O)C2CC2)c(F)c1F.C12CN(CC1O)C(=O)CN2 C1(C2CN(C(CC=CC)=O)C2)CN(C(C2CCC2OCC)=O)CCO1 C1(c2ccccc2)(NC(C)=O)CCN(C(=O)NCC2(C)CCC(=O)NC2)CC1 CCC(C)C(O)C(=O)N1CC(N(C)C(C2CCC2)=O)C1 c1(C(=O)NC2CCC(C(=O)NC(c3ccc(C)cc3)C)C2)ccc2ccoc2c1 C1(NC(C(CC)O)=O)CCN(C(=O)C=Cc2c(C)coc2C)C12CC2 C(CC(C(F)(F)F)C(F)(F)F)NC1CC(C)CC(C)C1 Cc1cc(C)c(CNC(=O)CC(C)CNC(c2ncsc2C)=O)s1 N1(C(c2n(C=C)ncc2)=O)CC(C(=O)NC23CCC(C2)OC3C)CCC1C N1(C(C2C(CC)N(C)CC2)=O)CC2(COC(CNC(c3cccs3)=O)C2)C1.O C1(C(C)(C)NC(C(C)OCCC=C)=O)CCCN1C(c1cc(Cl)cs1)=O C(N=c1[nH]c2c(c(=NCCCC3CCCCC3)[nH]1)COC2)C1(S(C)(=O)=O)CCC1 Cc1c(Br)c(C(=O)NC2CC2CNC(C2(C#N)CCSCC2)=O)nn1C Cn1cnc(C#N)c1C(=O)NCc1cn(Cc2cnc(C(F)(F)F)s2)nn1 c1(OC)ncc(Cl)c(=NCC2CN(C(C3CC3C)=O)CC2C(F)(F)F)[nH]1 C1(C=O)CC(F)C(=O)N1.N1(C(C)=O)CCCC1C(=O)N(C(C)C)C.CC=O CC(=O)CCCC(=O)NCCCCC1CCCN(C(=O)CC(C)C)C1 C1(C(N2CC(C(N3CC(CO)CC3CO)=O)(SC)C2)=O)CCC(O)CN1C C1CN(C(C2CC3(CCC3)CO2)=O)CCC1(F)F.C(C(=O)N)N(CCOC)C.C N1(C(C(C)OCC)=O)CCN(C(=O)Cc2ccc(Cl)c(C(=O)OC)c2)CC1C CC(C)S(=O)(=O)c1ccc2nccc(C(N3CCC(C)(N4CCC4)CC3)=O)c2c1 c1(C(N2CC(CN(C(C(C)OCC=C)=O)C)C2)=O)ccc(C)c2c1CCC2 C1(CN(C)C(C2CC2)=O)CCN(C(c2conc2C(F)F)=O)C1.C1CCC1 C(=O)C1=NN(C2CC2)C(=O)CC1.N1(C(COCC(C)C)=O)CCCC(C)C1.C C1(C(=O)Nc2cccc(NC(=O)CC3CC(F)C3)c2)CC2OC1C1CC21 c1(OC)cc(N(C)C)ccc1C(N1CCCC1CC)=O.C1(C=O)C2CCCC12.N c1(OC)ncnc(C(N2CCCC2CNC(=O)C=CS(C)=O)=O)c1F CC(C)(C)C(CNC(c1cnns1)=O)NC(c1cn(-c2ccccc2Cl)nn1)=O c1(C(=O)NCC(C)CN(C)C(c2nc(=O)n(C)[nH]2)=O)ccc2occc2c1 C1(C(N2CC(C)C2)=O)C(C)(C)C1(C)C.C(C)(C)OCC=C.C(=O)C.N C1(NC(C(C)(C)CF)=O)CCC2CN(C(c3cc(C(F)(F)F)cs3)=O)CCC2C1 c1(COC(c2c(C)cc(F)c(Cl)c2)=O)cccc2c(C)coc12 CC(C)(C(=O)NC1CCCC1NC(C1(CF)CC1)=O)C(F)c1ccccc1 C(CC(C(=O)N=c1cc(C)n(C)[nH]1)NC(=O)C(O)C(C)(C)CC)=CC C(C(CC)(CC)NC(=O)CC1CCOC1(C)C)NC(Cc1nc(CC)sc1)=O C1(CN(C(CCC2(NC(C3C(C)CC3)=O)CCC2)=O)C2CC2)CCCC1O C=CCC(C(=O)N1CC2(CC(CC(=O)NC(C)(CC)CC)C2)C1)C(C)C Cc1[nH]c(C)c(C(=O)NCCCCCCNC(=O)CCC2(C#N)CCC2)c1C c1(C(=O)NC2CCC(N(C(=O)CN3CCCNC3=O)C)C2)ccnc2ccnn12 CC1(C(=O)NCC2CCC2NC(c2ccnn2C(F)F)=O)CCNC1=O c1(-c2ccc(SC)o2)nc(CCN(C)C)nn1Cc1cccc(C)c1 C(=O)(CCCCC#N)N(C1CCCN(C(c2cn(C)nc2C(F)F)=O)C1)CCO C(=O)(CCN=c1[nH]ccs1)N1CC2C(NC(=O)CC3CS(=O)(=O)C3)C(C2)C1 C#CC1CCN(C(C2CCN2Cc2ccc(C#N)cc2)=O)CC1 CC1CCN(C(C2CCC3(C2)N=N3)=O)C(C)C1NC(=O)C=O.c1ccccc1.N C1(NC(=O)CSCCc2ccc(Br)cn2)CC(CO)C(CO)C1 C(c1cccc(F)c1)=CC(=O)NCCN(C(CC(C)F)=O)CCCN(C)C C1(OC)CCCCN(CC(=O)NCCOCCN(C)C(C2CC2F)=O)C1=O N=c1nc(CC(N2CC(CCNC(c3n[nH]cc3C)=O)C2)=O)[nH][nH]1.C(C)=O C(c1nc2ccccc2s1)=CC(=O)NC(C)(CNC(=O)CNC=O)CO N1(C(c2cc(C3(C)CC3)on2)=O)CCCC(NC(c2ccc(F)c(N)c2)=O)CC1 Cc1cccc(NC(=O)CC2CCCCN2C(=O)C(C)CC(C)C)c1C C1(C=O)CCS(=O)(=O)C1(C)C.N1(C(C2(CC=C)CCCC2)=O)CC2CC2C1.C CC1(C2CCN(C(c3ccc(-n4ccnc4)c(F)c3)=O)C2)CC1 CCCCCC(CC)C(=O)NC(C)CCCNC(c1ncc2cc(Cl)ccn12)=O CCC(C(=O)N1CCC(C)(C)CC1C(N1CCC(F)(CO)C1)=O)C(C)(C)CC C12(NC(=O)CCc3ccoc3)CCN(C(C3CCC4(CC3)CC4)=O)CCC1C2 CC1CN(C(c2cccc(Cl)c2)=O)CCC1N(C(=O)Cc1ccon1)C C1(NC(C(n2cnc(C#N)n2)CC)=O)CCCC2(CNC(=O)C2)C1 c1(C(=O)NCC(C)NC(C=Cc2c(C)cccc2)=O)n[nH]c2c1CC1CC21 C(=O)(CC(C)(C)CN(C)C)NCC(CC(=O)NC(CCC)CC)O Cc1noc(C)c1CNC(=O)CCCCNC(=O)CC(C)(C)C c1(SC)nc(=NC(C)CNC(c2ocnc2C(F)F)=O)s[nH]1 N1(Cc2ccc(CC)cc2)CC2(CC2)CC1C(=O)NC(c1ccccn1)C C(=O)(CC(C)C(=O)NC(C)CC(C)NC(=O)C=Cc1cccnc1C)OC Cc1cc(CC(=O)NCC(F)CNC(=O)CCOC2COC2)ccc1CO c1(C(=O)N)c(O)ncc2c1CCC2.C1C=CCN1C(C1CCOC1C1CC1)=O.C Cc1c[nH]c(C(=O)N(CC(O)CNC(c2ncoc2C2CC2)=O)C)c1 c1(C(N2CCOC(c3ccc(Cl)s3)C2)C(=O)NCC=C)cc(Cl)ncc1Cl N1(CC)CCCC(C(=O)NC)C1.C1CCCC1.N1(CC=CC=O)CCOCC1 c1(C(=O)NCC(CNC(C(C)C2CC2)=O)O)ccc(N(C)C)cc1F C1(C(N(C2(C#C)CC2)C)=O)C2CC2CN1C(C1(C2CCCCO2)CC1)=O Cc1ccc(C(C)C(O)C(=O)N(CCN(C(=O)C(C)(C)F)C)C(C)C)cc1 N1(C(CCC2CCN(C(C(C)OC)=O)CC2)=O)CCCCCC1C CCCC(C)(O)C(=O)NOC(CC(C)C)C(=O)NC12CCC(C1)C(O)C2O N1(C(C2C(C)(C)C2NC(=O)C=CC2CCCC2)=O)CCCC2COCC12 C1CN(C(=O)C)CC1(C)C.c1(C=O)ccc(N)cc1.C(C(=O)N)SCCC.C C(=O)(C(C)C(=O)N(CCCC(=O)NC(C)CCn1cncn1)C)OC CCCC(CCCNC(c1cc(C)cc(C)n1)=O)NC(=O)Cc1cn(C)nn1 n1(C(CC)CC)nc(C2CCOc3ccccc32)nc1-c1ccsc1 C(C)(C(C(=O)NCC1CCCCC1)N(C)C)OC.c1(C(C=O)O)ccccc1.N c1(CSCC(c2ccc(Cl)c(Cl)c2)C(=O)OC)ccc(F)c(Cl)c1 CN1CCCN(C(=O)CCN(CCCO)C(c2ccsc2)=O)CC1=O c1(NC(CC2(C)CN(Cc3ccccc3C(=O)O)C2)=O)cc(O)c(Cl)cc1Cl N1(C(CCCSC)=O)CC(NC(c2cnnc(C)c2)=O)C2CC12 Cc1cc(CNC(c2c(Cl)sc(Cl)c2Cl)c2nnnn2C2CCCC2)cnc1F C12(CNC(Cn3c(C)cnc3)=O)CCC1CN(C(c1ccncc1C(F)F)=O)C2 N#CC1(C(=O)NC2CC(NC(c3cnn(-c4nccs4)c3)=O)C(O)C2)CCCC1 C(C(=O)NC1CC(C(=O)Nc2cnccn2)C1)(C(C)C)OC c1(C(N(CCC(=O)NCCc2c(C)nc[nH]2)CCO)=O)cc(C)n(C)n1 C12(C(=O)NC(CC)C3CC3)CC(CN(C(=O)C3=CCCOC3)C1)C2 N1(C(c2c(C)nns2)=O)CCN(C(=O)CC2CCCCCC2)C(CCO)C1 C12(NC(CC=CC=C)=O)CCCC1N(C(=O)C=Cc1cccc(CO)c1)CCC2 c1(-n2cc(C3C(C(=O)NC(C(=O)OC)C4CCC4)C3)nn2)ccc(C)nc1 CN1C(=O)CCC1CC(N1CCC2CC12C(=O)NCc1ccnc(O)c1)=O c1(N2C(CCNC(Cc3ccc(CCC)cc3)=O)CCC2)ncnc(Cl)c1CC C=CCCC(C(=O)NCCCOCC1CC1)N1CCC(c2cnn[nH]2)C1 Fc1cccc2nc(N3CCOC4(CC4)C3)[nH]c(=NCC3(CF)CC3)c12 CC(C)(C)OC(=O)NCCNC(C)(C)C1CCC1 c1(C(C)Nc2n(CC)nnn2)nn(CCC(C)C)c2ccccc12.C1CCCC1 c1(SCC(=O)NC)cccc(NC(c2nnnn2C(C)CC)(C)C)c1.CCF C1(=CC(=O)NC(C)CNC(C2CCCC(=O)O2)=O)CC2CCC(C1)N2C CCC(CC(=O)NCCCCN(CCCNC(c1cnc(C)[nH]1)=O)C)C1CC1 C1(F)(CNC(C2C3CCCCCCC23)=O)CC(N=c2[nH]cnc3cc(Br)sc23)C1 N1(C(CC2CC(=O)NC2)=O)CC2CCC(CNC(c3ccc(F)cc3)=O)C2C1 C1(CC(=O)NCc2cnc(C)n2C)CN(C(c2csc(Cl)n2)=O)CC12CC2 C(CC1=CCN(C(=O)C(C)OC(C)(C)C)CC1)NC(c1c(C)nc(C)s1)=O C(=O)(C(C)C(C)NC(=O)C(C)SC(C)C)N(CC#C)CC N1(C(CCn2c(C)cc(C)n2)=O)CCN(C(=O)C=Cc2ccco2)CC1C1CC1 N1(C(C2CC(C(C)C)C2)=O)CCN(C(=O)CC2(O)CCOC2)CC1CO Cc1c(C(=O)NCCC(C(C)C)NC(=O)C2CC2)cccc1S(N)(=O)=O CN1CC(C(=O)NCCCNC(C2(n3ccnc3)CCCC2)=O)CC1=O c1(NC(C2CC23CCN(C(c2cccc(F)n2)=O)C3)=O)cc(Cl)cc2[nH]ccc12 C1(C(N2CC3C(NC(c4cccc(OC)n4)=O)(CC3)C2)=O)CCn2nncc2C1 N1(C(C(C(C)C)NC2CCCCC2)=O)CCN(CP(C)(C)=O)CC1 c1(C(=O)NC(CC)C)ccc(=NCc2ccc(C)nc2Br)[nH]c1 c1(C(=O)NC2(C)CC(NC(c3snc(Cl)c3Cl)=O)C2)cnn2c1OCC2 c1(C(=O)NCCC(=C)CNC(=O)CC)oc(CC(C)C)nc1C.C(C)=O.N N1(C(CSCCC)=O)CCC(C2CCN(C(=O)C(N3CCOCC3)C)C2)CC1 CN1C(=O)CCCC1C(N1CC=C(CNC(=O)C=Cc2cccnc2)CC1)=O c1(NCc2ccc(F)cc2Cl)ccc(Cl)c2ccncc12 c1(SC)nc(Cl)c(C)c(=NCCNC(C2CC(n3cnnc3)C2)=O)[nH]1 c1(C(=O)NC(CC)C)c(NC(c2cc(O)ccc2[N+](=O)[O-])=O)sc2c1CCCC2 N1(C(C(C(C)C)F)=O)CCCC(NC(=O)CNC(c2ccc(O)cc2)=O)CC1 C(=O)(C(C)S(C)(=O)=O)N1CC(N2CCN(C(C(COC)OC)=O)CC2)C1 Cc1cc(C)n(CC(N2CCC(CNC(=O)C)CC2)=O)c(=O)n1.C1CCOC1.O CCCCCO.C1(=O)C(C)N2CCC2CN1C.C1(=O)C(C)N1 C(CCCCCO)NC(=O)NC(C1(C)CC1(Cl)Cl)C Cc1nnc(C(CCC2CC(F)(F)C2)NC(CN(C)C)Cc2ccccc2)n1C C1(C)(C(N(CC=C)CCC)=O)CCCN1C(c1ccsn1)=O CC1CCN(C(c2ccccn2)=O)CC1CNC(=O)C(=O)C1CCCC1 C1(NC(C(C)OC2CCCCC2)=O)CC2CN(C(C3(O)CC(C)(C)C3)=O)CC2C1 c1(OC)cnc(C(=O)NC2CCCC(NC(=O)CCc3ccc(C)nc3)C2)cn1 c1(CC(C(=O)NC(C(C)O)CO)NC(C2CCNC(=O)C2)=O)ccccc1F C1(NC(c2c(CC)onc2C)=O)CCN(C(=O)Nc2ccc(SC)cc2)CC1F O=C(C1Cc2ccccc21)N1CCC2C(CCN2C(=O)Cc2cnoc2)C1 C1(C(N(CCNC)C)=O)CC12CCN(C(c1ccc(Br)cc1Cl)=O)CC2 Cc1ccc(C(=O)NCC2CCCC2)cc1[N+](=O)[O-].C1(CC(=O)N)CC1(C)C C=CCC(CC(F)F)NC(C1(C)CCN(C(c2cc(OC)cnn2)=O)CC1)=O C1(CCNC(C(C)=CCN)=O)CCCC12CN(C(=O)CCNc1cccnc1)C2 Cc1cc(CN2CCC(CNC(=O)CCC3CC(F)(F)C3)C2)n[nH]1 N1(C(CC(C)OC)=O)CCC(CNC(=O)C2=NOC(C(C)(C)C)C2)C12CC2 c1(CCc2cn(CCNC(CN(CC(C)(C)C)C)=O)nn2)cccc(O)c1 c1(C(=O)NC(CC2OCCN(C(CCOCC)=O)C2)C)cc(C)c2n[nH]cc2c1 C1(C(N2CC(F)(C(=O)OC)C2)=O)COCCN1C(=O)C(C)c1ccco1 C1(C(N2C(C)(CNC(c3ccc(C)c(O)n3)=O)CCC2)=O)CCC2(CCC2)CO1 Cc1ccc(C(N2CC(C)(C)CC2CNC(=O)C=Cc2ccncc2)=O)nc1C c1(-c2ccc(CN(CCCC(=C)C)C)s2)cc2c(cc1OC)OCO2 N1(C(c2c(CNC(c3c(OC)ccs3)=O)c[nH]n2)=O)CCCCCC1CO CCC(CC)CCC(=O)N1CC(OC)CC(NC(c2ccn3nnnc3c2)=O)C1 c1(CC(=O)NCC(C2CC2)NC(C2CCN(C)CC2)=O)cccc2ccncc12 N1(C(C(COC)COC)=O)CCC(NC(C2CC2(C)C(F)F)=O)C(C)(C)C1 C1(NC(COCC)=O)CCCC12CCN(C(=O)CCCn1cccn1)C2 C#Cc1cnn(C)c1C(=O)NC1CCCN(C(c2ccc(COC)o2)=O)C1C C1(NC(C(CSC)(C)C)=O)CCN(C(=O)CCN2CCCC(C(N)=O)C2)CC1O C1(NC(c2c(C)nco2)=O)CN(C(c2ccc(Br)c(Cl)c2)=O)C(C)(C)C1 C(C)(N=c1[nH]c(=NCC2(CO)CC2)c2ccccc2[nH]1)c1ccc(C)o1 C1(C=O)CN(C=O)C2(CCC2)C1.N1(CC=O)CCCC1.C(C)(C)C.CC.N C1(C(=O)NC2(C(=O)NC(C(=O)OC)CCF)CCOCC2)CCCCCN1C C(=O)(C(CC(C)(C)C)O)N1CC(C=C)(CC(=O)NC2(CC=C)CCCC2)C1 C1(NC(c2cc(C)c(C)s2)=O)(CO)CCCN(C(=O)C(C)O)C1 c1(C(=O)NC(CSCC)C(=O)NC(C(N)=O)C2CCCC2)ccncc1N c1(NC(C2C(NC(c3c(C)cc(Br)cn3)=O)C2)=O)ccc(C#N)cc1Br C(=O)(CCCCC(C)(C)C)N1CCC(C(=O)NC(COC)C(C)C)OCC1 c1(OC)cc(C)cc(C(=O)NC2CCN(C(=O)Cc3ccc(C)nc3Cl)C2)c1C C1(CNC(C=NOC)=O)CN(C(=O)CCCc2nnc(C)n2C)CC12CC2 C(=O)(N1CC(n2cc(CO)nn2)CO1)NC(c1c(OC)nccc1)=O N1(C(CC2(CC=C)CCCC2)=O)CCOC2(CCN(C(C3OCCC3C)=O)C2)C1 CCC(O)CC(=O)NC(C(=O)NCCOCCCF)C(C)O C1(C(=O)NCC(C(=O)NC(CCC)CO)OC)CC(F)C(=O)N1 c1(C(N2CC(C(C(=O)N)O)C2)=O)ccncc1C1CC1.C1(O)(CC)CCCCC1 N1(C(C2(OCC)CCOCC2)=O)CCCC2CN(C(=O)C(C)C3CC3)CCC12 N1(C(c2c(C)ccs2)=O)CCN(C)C(CNC(=O)Cc2nc(C)c(C)[nH]2)C1 N1(C(CCCC(C)=O)=O)CC2CCOC2(CNC(c2ccc(Cl)o2)=O)C1 C1(C(=O)NC2CN(C)C2)CC2CCN(Cc3ccsc3Br)CC12 c1(SC)ccc(O)c(C(=O)NCCC2CCCN(C(=O)CN3CCCCC3)C2)c1 C1(NC(=O)NCC2CCC(C)O2)CCC(C(=O)OC(C)(C)C)CC1 Cc1c(C(N2CCC(NC(C3(C(N)=O)CC3)=O)CC2)=O)cc(F)cc1Br c1(CC(=O)NC(C2CCCCN2C(c2cccnc2O)=O)C)c(Cl)cccc1Cl c12nccc(n1)CN1CCC2C1.C(CCN)(C(F)F)SC c1(COC)cccc(C(=O)NC(C)CN(C)C(C2CCC(=O)N2)=O)c1C c1(N(Cc2ccccc2)CC)ccc(C(=O)NC(=O)Cc2nccs2)cc1F N1(C(C(CC)C#N)=O)CC2CCC1CN2CC(=O)NC C(CCCCCNC(c1ccnc(Br)c1)=O)n1cc(CCN(CC)CC)nn1 c1(C(=O)NCC(CC)NC(=O)C(O)CCn2cncn2)ccn(CC)c1C c1(CN2CC(C(=O)Nc3ncc(I)cc3C(F)(F)F)C2)cc(F)cc(F)c1O C1(C(=O)NCc2c(C)nn[nH]2)CC(NC(=O)CC#N)C(O)C1 C1(CC)CN(C(C2CCC2(OC)OC)=O)CC1n1cc(C(CC)OC)nn1 C=CCCCC(C(=O)N(C)Cc1nc(C)cs1)NC(=O)CCc1cn[nH]c1 CC(C(=O)N(C)C)S(=O)(=O)N1CCC(N2CC(F)C2)C1 C1(CC)CCOCCN1c1nnc(-c2c(C)ccn2C)n1CC O=C(CC(C(F)F)N1CCOCC1)NC1CCN(C(=O)Cc2nc[nH]n2)C1 N1(C(C2CC(OC)C2)=O)CCN(C(C2(C(F)(F)F)CCC2)=O)CC12CCC2 C1(CC(N2CCN(C)C(C)(C)C2)=O)OCC2CCN(C(c3ccc(F)s3)=O)CC12 C1(COC)(NC(c2ccncc2Cl)=O)CCN(C(=O)COCC(C)C)C1 N1(C(c2c(C)occ2)=O)CCCC(C2CCN(C(=O)CC(C)C(F)F)C2)C1 C1(C(=O)NCC(=O)OC(C)C)(NC(CSCCCC)=O)CCOCC1 C12(NC(CCSc3n(C)nnn3)=O)CCCN(C(=O)C#CC3CC3)C1C2 N1(C(C2CC(OC)C2)=O)CCN(C(C2CN3CCCC2C3)=O)C2CC12 C12CCC(CC1)CO2.C1(O)(C=O)CCOC1.O=C(COCC1CC1)NC c1nc(C2CC2N)cs1.n1(C2CC(C(=O)OCC)C2)cc(C2CCOCC2)nn1 N1(C(c2c(C(C)C)scn2)=O)CC2CCCN(C(=O)CC3COCC3(C)C)C2C1 C(=O)(CC(C)(C)CC(F)(F)F)N.N1(C(C(C)=C2CCC2)=O)C2CCC1CC(C)C2 c1(OC)cnc(C(N2CCC(CC3CCN(C(=O)C(C)(C)F)CC3)CC2)=O)cn1 CC(COCc1ccccc1)N=c1[nH]c2cccnc2s1 c1(CC(=O)NC2C(NC(C(CSC)C)=O)CC2)ccccc1SC c1(CN2C(C(=O)N(CCO)C3CC3)C=CC2)cc(Br)cc(F)c1O c1(C(=O)OCc2cc(C)c(F)cc2)c(O)cc(C)oc1=O N1(C(Cc2ccc(C(N)=O)cc2)=O)CC2CC(C1)N(C(=O)CC1(C)CC1)C2.S C1(NC(CC2CC(=C)C2)=O)CCCCC1NC(=O)C(C)=NOCC#N c1(C(N2C3(CNC(CC(CCCC)O)=O)CC(C2)C3)=O)c(Cl)cccc1[N+](=O)[O-] N1(C(c2ncc(N(C)C)nc2)=O)CCCCC(CNC(=O)CC(C)(C)O)CC1 C(=O)(CC(CC1CC1)NC(c1ccsc1Cl)=O)NC1CC(CCOC)C1 C1(CC(=O)N(C)C)CCN(CCF)CC1.C1CCN(C(=O)Cc2ccn(C)n2)C1 Cc1ccc2cc(C(=O)N(C3CCC(NC(c4cnc(Cl)[nH]4)=O)C3)C)cn2c1 Cc1nc(-c2ccccn2)[nH]c(=NCC(C)CN(C)C)c1C c1(CC(=O)NC2CCN(CCN3C(=O)CNC3=O)C2)ccccc1.C(C)C.C CC(C)(C)CNC.C1CCC(C(F)(F)F)C1.C(C=O)=CCN(CC#C)C.C c1(NC(C(N2CCC(C(C)C#N)CC2)=O)=O)cccc2snnc12 C(=O)(CN=c1[nH]c2ccccc2s1)NC1CCC(CCNC(=O)C=CC2CC2)C1 N1(C(C2CCCS2)=O)CCC2CCCC12C(N1CC2CC1C(F)(F)C2)=O C1(C(=O)Nc2cccc(C(F)(F)F)n2)CC(O)CCN1C(c1ccc(Br)cn1)=O C1(C(=O)NCCC(C)CO)C(C)CCN1C(=O)CCOCC(C)(C)C c1(C(=O)NCCC2N(C(COc3cn(C)nc3)=O)CCSC2)cc(F)cnc1Cl N1(C(CCCCOC)=O)CC2(CCCC2NC(c2ocnc2C2CC2)=O)C1 N1(C(CCN(C(CSCCCC)=O)CC)=O)CCN(CCO)C(=O)C1 c1(C(N2CCCC2)=O)cccc2nccnc12.C1(C(=O)NC2CC2)CCS1(=O)=O CC(CC1CCCC1)C(=O)NC1CCN(C(c2sccc2-n2cccc2)=O)C1 N1(C(C(C(=O)OCC)(C)C)=O)CCN(C(C2(CF)CCC2)=O)C2(CCC2)C1 O=C(CCCCOCc1ccccc1)NC1CN(C(c2ncoc2C2CC2)=O)C1 c1(CC(=O)NCC2(Nc3c(Br)cnc(C(C)C)n3)CC2)ccc2ncsc2c1 c1(SCC(=O)N(C2CCN(C(C3(F)CC=CCC3)=O)C2)C)ccccc1[N+](=O)[O-] C(=O)(C1=CCCSC1)NCC(N1CC(C)OCC1)c1cccs1 c1(C(N2CCC(C)(NC(c3cc(C(N)=O)no3)=O)C2)=O)ccc2sncc2c1 c1(-c2c(OC)cccc2)cc(C(=O)NCc2nonc2C)c2c(C)noc2n1 C12(C=O)CCC(C1)S(=O)(=O)CC2.c1(N(C)C)ccc(C(=O)N)cn1.C(C)CO c1(C(=O)NC(CCCNC(CCCOCC)=O)C)coc2cccc(Br)c12 N1(C(CCn2cc(C(c3ccccc3)C)nn2)=O)CCC(CN(CC(C)=O)C)C1 N1(C(CCCNC(=O)OC)=O)CC(C)CCC1CNC(c1cc(C)on1)=O N1(CC)CCC(NC(=NCC2CCCCO2)NCc2cc(C(F)(F)F)sn2)CC1 N1(C(COCC(=O)OC)=O)CCC2CCC(C1)N2C(C1(C)CCCC1C)=O CC1(NC(C2CNC(=O)N2)=O)CCCN(C(=O)CS)C1.c1(C(C)=O)ccccc1 S(=O)(=O)(c1ccc(NCCCF)c2cnccc12)NCC(C1CC1)SC c1(C=O)cc([N+](=O)[O-])c[nH]1.C1(CNC(CNC(CCC)=O)=O)CCOCC1.C Cc1ccc(C(N2CC(C(O)C(=O)Nc3ccccc3C3CC3)C2)=O)nn1 C12(C(=O)NC(C(=O)NC(C)C)C)CC1CN(C(C1C=CCS1)=O)C2 c1(C(=O)NC23CN(C(c4c(C)ccc(C)n4)=O)C(C2)C3)cnc2n1CCCCC2 C1(NC(COCCOC)=O)CN(C(=O)C(=O)NCC2CC2)CCC1C c1(C(N(C)Cc2ccc(F)c(Cl)c2Cl)=O)ccc2[nH][nH]c(=N)c2c1 N1(C(C2CCCN(C(c3cnc(SC(C)C)s3)=O)C2)=O)CCCC(N(C)C)CC1 c1(C(=O)NC2(CO)CCN(C(C(CC#C)C3CC3)=O)C2)ccc(Br)c(N)c1 N1(C(C2N(C(CC3C(C)C(=O)CC3)=O)CC(C)C2)=O)CCC(F)(F)CC1 Cc1noc(C)c1CNC(=O)C(=O)NC(c1ccc(Br)cc1)C C12(C(=O)OC)CCCC(C(=O)OC)(CC1)C2.C1(=O)C(C)(CC)CN1 C1(C)(CC(=O)N(CCC#C)CCO)CCN(C(=O)Cc2csc(C)c2)C1 N1(C(C(CCCC)F)=O)CCCC12CCC(NC(=O)C=Cc1cc[nH]n1)CC2 C1(CC)(NC(c2cnc(O)s2)=O)CCCN(C(=O)CCc2ccncn2)C1 C12(C(N(C3CN(C(c4nc(C(C)C)sc4)=O)C3)C)=O)CCCC(C1)OC2 C1(CC(=O)NC2CCCN(C(c3c(C)[nH]cc3)=O)CC2)CC2(CCOCC2)CO1 N(C1COc2cc(Cl)ccc21)c1cc(NCc2ccc(C)o2)nc(C)n1 c1cc(F)ccc1F.C1(C(=O)NCC(=O)N(C(C)C2CC2)C)CCCC(F)C1 c1(-n2cc(C(C)(C)NC(c3cc(Cl)no3)=O)nn2)c(F)cccc1[N+](=O)[O-] c1ccc(F)c(F)c1.C1(CC(=O)NC(CC=CC)CO)CCCN(C(=O)NC)C1 c1(N(C)Cc2ccncn2)nc(N2CCC3(CC2)CC3CO)nc2sccc12 CC(C)(C)CC(O)CC(=O)NCC#CCNC(=O)Cc1cccnc1Br C(CCCCCNC(=O)CC1CCN(C)C1)NC(Cn1ncc(CC)c1)=O C1(C(N2CC(C)(C(=O)NC3(CC)CC3)C2)=O)CCC(C2CC2)C1 C=CC(CCC)CC(=O)N1CCOC(CC(=O)N(C)Cc2cccc(O)n2)C1 c1(C(=O)OC)cc(CN2CCOC(c3ccccc3)C2)ncc1Br C(=O)(C(C)(C1CCC1)NC(=O)CCc1ccco1)NC(C)CO c1cc(Br)ccc1Cl.c1(C(=O)NCC2(O)CNC2)ccc(C(F)(F)F)cc1F.C C1(C(N(CCCNC(C2CCCSC2)=O)C)=O)CNC(=O)CC12CCC2 c1(CC(N2CCCCC2)=O)c(C)cccc1F.C1(C(=O)N)(COC)CCOC1.C c1(-n2cc(CCC(C)=O)nn2)ccc(C(=O)NCCC2CCNC(=O)C2)cc1 C(=O)(CC(C)C(C)(C)C)NCCN(CC(C)O)C(c1ncn(CC)n1)=O C1(C(N2CC(NC(=O)C(=O)NC3CC3)CC(OC)C2)=O)CCc2nncn2CC1 C1(CC)CN(C(=O)C(COC)NC(C)=O)CCN1C(=O)CCCc1ccsc1 C1(C=O)CC2CS(=O)(=O)CC(C1)C2(F)F.C1(C=O)CC(C)(O)C1.CCCC.N c1(OC)c(C)ccc(F)c1-c1cc(C(N2CCOC(=O)C2)=O)ccn1 N1(C(C2(CC#C)CCCOC2)=O)CCC2C(CCCN2C(=O)C2CC2)C1 CCCCC(=O)NCc1c[nH]c(C(=O)C(Cl)(Cl)Cl)c1 N1(C(CN(C)C(N)=O)=O)CCN(C(c2c(O)ccc3nc[nH]c23)=O)CC(C)(F)C1 c1(C(=O)Nc2cccc(C(=O)OC)c2)ccc(S(=O)(=O)N(C)OC)cc1 c1(OC)cc(C(=O)NC(C)C)ccc1C#N.c1(C(C=O)(C)C)ccc(Cl)cc1.N C1(NC(c2c(OC)nc(C)cc2)=O)CC2CC(C1)CN(C(c1nncs1)=O)C2 C1(CC)CN(C(c2ccc(C3CC3)cc2F)=O)CCC1NC(C1(C)CCC1)=O Cc1c(C(=O)N(C)CCNC(=O)CCC(=O)NC)nn(C)c1N.c1ccccc1 Cc1ccc2nonc2c1C(N1CCCC(N(C)C(c2cnn(C)c2)=O)C1)=O C(N=c1cc[nH]cc1[N+](=O)[O-])C1CN(C(C2CC23CCOCC3)=O)C1 CCCCCCCCCC(=O)Nc1ccc(N2CCNC(=O)C2)cc1 Cc1nn(CC(=O)NCC2CCC2NC(C2CC2(F)F)=O)c(C)c1Cl CCCC(C(=O)N1CCN(C(c2nncn2C2CC2)=O)C(CO)C1)S(N)(=O)=O Cc1cccc(S(C)=O)c1NC(c1cn(C2CCOCC2)nn1)=O CCCCC(CC)C(=O)N(C1CCN(C(=O)COc2ccc(Cl)cc2C)C1)CC CCC(CC)(CC)C(=O)NCC1CC(C(=O)N(C)Cc2cnc[nH]2)=NO1 c1(CCC)nc(C)c(C(=O)NC2CCCC2)s1.c1(C=O)ccn(C2CC2)c1C.N C1(F)(C(=O)NC(CC)CN(C)C(c2cc(Cl)nn2C)=O)CCC(C)CC1 C1(NC(CCn2c(C)cc(C)n2)=O)CC(F)CN(C(=O)C=Cc2ccncn2)C1 c1(C(=O)NC(C)CN(C)C)ccc(CNC(=O)C(N2CCOC2=O)C)cn1 c1(C2CC(=O)NC2)ccccc1.C1(O)(C(CNC(=O)CO)=O)CCN(C(=O)CO)C1 c1(C(=O)NC2CN(C(C(CSC)O)=O)CC23CCC3)nnc(O)c2ccccc12 c1(C(N2CCC(C(C)NC(COCCCC)=O)C2)=O)cc2occc2s1 CC1(C)C(CC(=O)NC2CSC2)CCN1C(=O)C=Cc1cscn1 c1(C(N2C(CNC(CC(C)F)=O)CCC2)=O)cccc(OCC(F)F)c1 C=C(Cl)CCC(=O)NCC(C1CCOC1)NC(=O)C=C(C)CCC CC1CCCCC1n1nc(-c2ccc(Cl)nc2)nc1-c1ccnn1C c1(C(N(C)CCn2cc(-c3ccc(Cl)nc3Cl)nn2)=O)cc2n(n1)CCCC2 c1(CC)noc(CC)c1CC(=O)NCC12CC1CN(c1nnc(C(F)F)s1)C2 c1(C(N2C(C(N3CCC(OCC(C)C)C3)=O)CCC2)=O)ccc(CO)nc1 C1(NC(COCCC#C)=O)CC2CC1N(C(c1[nH]c(C3CC3)nc1C)=O)C2 c1(C(=O)NCC2(C)N(C(c3n(CC)c(O)nc3)=O)CCC2)scc2c1OCCO2 Cc1ccc(CN2CCCC(C)(C(=O)NCCCN3CCCC3)C2)c(C)n1 CC1CCN(C(c2cc(O)no2)=O)CC1NC(=O)C(F)(F)C(O)C1CC1 c1(OC)nscc1C(N1CCCC1C(C)NC(=O)C(=O)NC)=O.C1CC1 c1(C(N(C2CN(C(C=O)=O)C2)C)=O)cc2n(c1)CCS(=O)(=O)C2.CC.CO C1(C(N2C(C3(C(N(C)CP(C)(C)=O)=O)CC3)CCC2)=O)CC2(CCO1)CC2 C(C1Cc2ccccc21)NC(C1CCN(C(=O)Cc2ccoc2)CC1)=O c1(C(=O)NCCC2CN(C(C(C(COC)C)C)=O)C2)sc2[nH]cnc(=O)c2c1C C1(C(=O)NC(c2n(C)ccn2)C2CC2)COCCN(CCC(=O)NCCN)C1 c1(OC)ncc(NC(=O)C(C2CC=CCC2)NC(c2cn(C)cn2)=O)cn1 C1(CCC(N)=O)CCN(C(=O)CC2CSCCS2)CC1 Cc1c(NC(N2CCCC(C(=O)Nc3ccc(CO)c(Cl)c3)C2)=O)cccc1Cl c1(N(C)C)cc(Cl)cc(Cl)c1C(=O)OCC(C1CCOC1)=O CCC(O)C(C)(C)C(=O)NCC1CC(C)(C)CN1C(c1cccc(N)n1)=O N1(C(c2cc(OC)cc(Br)c2)C(=O)NCC(C)C)CCC(S(C)(=O)=O)C1 N1(C(C(C)(C2CC2)OC)=O)CCCCC2(CCN(C(=O)C=CC(C)C)C2)C1 C(c1ccccc1C)=CC(NOCC(=O)NC(CC=C)C)=O C1(C(=O)NC(CCSC)C(=O)NC(c2cccc(C)c2)C)C2CCC(F)(F)C12 N1(C(C2(CCNC(CN(CC)CC)=O)CCCC2)=O)CCC2(CCOC2)C1 N1(C(CCOCC)=O)CCC2(CCCC2)CC1.n1(CC(=O)N)cc([N+](=O)[O-])cn1 CCC(N=c1[nH]c(=N)[nH]c(=NCC(CSC)OC)[nH]1)c1ccn(C)n1 CCC(C(C)CN(C)C)NC(C1C=CCCN1C(=O)COC1CC=CC1)=O Cc1ccn(C(C)(C)C(=O)NCCC(O)CNC(=O)Cc2sccc2C)n1 N1(C2CCC(COC)C2)Cc2cccn2C(C)C1 CC1CN(c2nc(C(F)(F)F)ns2)CC1NC(c1coc(C(F)F)c1)=O C1(NC(C2C(C)(C)C2(F)F)=O)COC2CN(C(C3CCCCCC3)=O)CC12 Cc1cnc(NC(C2CN(C(c3ccccc3F)=O)CCS2)=O)c(I)c1 C=CCCCCCCCC(=O)NC12CN(C(=O)C(CCC)OC)C(COC)(C1)C2 C1(CNC(c2nc(C)oc2)=O)CC(C)N(C(c2ccc(=N)[nH]n2)=O)C1 C12CN(C(C3(C#N)CCCC3)=O)CC1CCO2.Cc1ncc(C=CC(=O)NC)s1 C1(CC(=O)N(C)CC2CC2C#N)CCCC(NC(C2CCCC2O)=O)C1 CCCC(C(=O)NC1(c2nc(C)no2)CC1)NC(=O)C=C(C1CC1)C1CC1 C(=O)(CC(O)(C(F)(F)F)c1ncco1)NCCN(C(C(C(C)O)(F)F)=O)C c1(NCC2(CNC(c3c(C)nn[nH]3)=O)CCC2)ccnc2ncnn12 Cc1cc(C)n(CC(=O)NC(C)C(CO)NC(c2cncnc2)=O)c(=O)n1 C1(CCNC(c2ccc(C(C)=O)nn2)=O)CCCN(C(=O)C=C(Cl)Cl)CC1 N1(C(C(c2ccccc2F)C)=O)CCCC12CCN(C(=O)CC1(C)CCCO1)C2 C(C)(C)(C(C)CC(=O)NOCC1CC1)NC(C(COC)OC)=O c1(C=O)[nH]nc2ncccc12.C1(CNC(c2cnc(C)o2)=O)(C)CC12CCC2.N c1(OC)ncc(C(=O)NC(C)C(CO)NC(c2ccnn2C2CCC2)=O)cc1Cl c1(OC)cncc(C=CC(=O)NC2CC(C)CN(C(C3CCC(=O)N3)=O)C2)c1 c1(OC)ccc(OC)c(C(=O)NC2CC(O)CN(C(=O)CC(F)(F)F)C2)c1O C(=O)(CCP(C)(C)=O)NC(C)CC.C(=O)CCC1CN(C=O)C1.C(C)(C)C c1(OC)cccc(C)c1C(N1CCC(O)(C)C1)=O.C(=O)(CCCn1ccnc1)N C#CC1CCN(C(C2CCCCC2CNC(C2C=CCCC2)=O)=O)C1 C#CCC(CC#C)C(=O)N1CCN(C(=O)C(c2cscn2)N(C)C)CC1C(C)C C(=O)(C(C)(C)C(=O)NC1CCC12CCC2)OC.C1(C)CCCC1.C(=O)C.C C(=O)(C#CC(=O)N1C(CNC(=O)CSc2nc[nH]n2)CC2CC12)N(C)C C#Cc1cnn(C)c1C(=O)NCCCC(C)(C)NC(=O)CCCCN(C)C N1(C(COCCOCC#C)=O)CC(F)CC1CNC(=O)C(C(C)C)S C(=O)(C(C)(C(C)C)OC)NC1C(CC(N2CCN(C(=O)OC)CC2)=O)CC1 c1(N(C(=O)CCC2CCCN2C(c2cc(C(N)=O)co2)=O)C)cccn(C)c1=O Cc1cc(=NC(=O)CCOCCCNC(=O)C(C)(C)CNC(N)=O)[nH]n1C c1(OC)ccc(C(N2CC(NC(=O)C(C)CN(C)C)C2)=O)nc1.CCC(C)C N1(C(c2[nH]cc(C)c2)=O)CC2CC2(C(=O)Nc2cccc(N(C)C)c2)C1 N1(C(C2(COC)CCCCC2)=O)CC(NC(C2NC(=O)OC2C)=O)CC(F)C1 C#CCC(CC#C)C(=O)N1CC2CC(NC(=O)Cc3c(C)nn(C)c3C)C1C2 Cc1coc(C)c1C(N1CCC(O)(CC)C1)=O.c1(C(=O)N)cccc(N(C)C)c1 C1(C(=O)NCCC2CCN(C(c3[nH]cc(C)c3C)=O)C2)CCOCC1(C)C c1(CC(N2C3C(NC(c4ccc(C(N)=O)nc4)=O)C(C3)C2)=O)ccc(Cl)cc1Cl N1(C(C2N(CCC)CCC2)=O)CCC(NC(=O)CN2CCC(O)CC2)C(F)C1 N1(C(=O)OC)CCCCC1.C1(C=O)CC2CC2N1C(c1cc(C(C)=O)on1)=O c1(C(=O)NC(C)CNC(C2CCCOCC2)=O)cc2c(F)cccc2[nH]1 CCC(C)C(=O)C(=O)NCC1CCN(CCOCCOC)C1.C12CC1C2 C1(C(N2CCNC(c3ccc(C(F)(F)F)cc3)C2)=O)Cc2cc(O)ccc2CN1 Cc1ccc(C(=O)NC2CCC2NC(C2(C3CC3)CC2)=O)c(C)c1Br C1(NC(C=CC(=O)OCC)=O)COCC1C(N1CC2(CC2)C1)=O CCCC(C(O)C(=O)NCCC1=CCOCC1)NC(c1coc(C)n1)=O CCC(=O)CCC(=O)N1CCC12CN(C(=O)C(F)C(F)(F)F)C2 N1(C(C=CC(CC)C)=O)CC(CNC(C2(Cl)CC2)=O)CC12CCOCC2 CC(C)(C#N)CCC(=O)N1CCC2CC12C(=O)NOCCC(F)(F)F CC1CCC(C)N1CC=O.C1C2CC1N(C(C1CC(=O)C1C(C)(C)C)=O)C2.N C(=O)(CCCCC=CC)NC12C(CN(C(C3(C)CC(=C)C3)=O)C1)C2 C(=O)(CS(=O)(=O)CC(=O)N1CCCC1CC)OC.C1(C)(C(=O)N)CC1(F)F c1(C(N2CCSCC2C)C(=O)NC(C(=O)OC)C)cc(Br)ncc1OC c1(NCC)ccccc1C(=O)NC(C1CCCN(C(c2cccc(C)c2)=O)C1)C c1(C(N(C2CCN(C(=O)Cc3ncn(C)c3C)CC2)CC#C)=O)nc(C)nn1C C1(C(=O)NCCCN(C(c2ocnc2C2CC2)=O)CCC)CC1C1CCCC1 N1(C(C2(OC(C)C)CCC2)=O)CCCCC1.C(=O)(C(C)(C)c1cnc[nH]1)NC.C C=CCC(C)(C)CC(=O)NC(CN(C(=O)C(C=C)CC)C)(CO)CO N1(C(c2nc(C)oc2)=O)CCN(C(C2C(C)(C)OC2(C)C)=O)CC2CCCCC12 C1(C#N)(OC)CC(C=O)C1.c1(C(N(C(C)C)C)=O)ccc(C(C)(C)C)cn1.N C1(NC(C(c2nc(C)sc2)=O)=O)CCCCN(C(c2cnn(CCO)c2C)=O)C1 C1(C(N(CC#C)CCO)=O)CN(C(C2(C)CSC2)=O)CC(C)(C)C1 C1(NC(C2(C)CC3CC3C2)=O)CN(C(c2cnc(S)[nH]2)=O)C2(CCCC2)C1 c1(N2CCC(C(c3ccccc3)C)C2)nccc(=NC2CC3COCC(C3)C2)[nH]1 CCC(CCCC(=O)N1CC(C)N(C)C(C)C1)NC(c1ccn(C)c(=O)c1)=O C1(C)(CNC(C=C(C)Cl)=O)CN(c2ncc(C(C)(C)O)cn2)CCO1 N1(C(C(COCC)C)=O)CCC2(CCC2)C(NC(c2ccnc3c2CCC3)=O)C1 c1(OC)ccc(CN2CCN(C(C3CCCC3C)=O)CC2C)c(C)c1 c1(C=O)cc(F)c(Cl)c([N+](=O)[O-])c1.C1(C)(CN(C(=O)CCF)C)CCCC1.N C1(NC(C2CCC(C(N)=O)C2)=O)CC2COCC(C1)N2C(C1CC(O)C1)=O.C Cc1ncn(C)c(=O)c1C(=O)NC1C2CN(C(c3cc(Br)cs3)=O)CC12 C(=O)(CC(C)P(C)(C)=O)N1CCC(NC(C(CN(CC)CC)F)=O)(C)C1 CN1CCN(C(=O)CN2C(=O)CNC2=O)C(CNC(c2cccc(Cl)c2N)=O)C1 c1(C(N(C)Cc2ncc(Cl)cc2Cl)=O)ccc2c(=O)n(C)c(S)nc2c1 N1(C(CC(C)F)=O)CCC(C(C)C(=O)NC(C)(CO)C2CCC2)CC1 N1(C(CS(=O)(=O)NC)=O)CCC2CCC(NC(=O)C=C(C)C(F)F)C12 c1(CCC)ccc(C(=O)CCC(=O)N(C(C(OC)OC)C(C)C)CCOC)cc1 c1(C(=O)NCC(C2N(C(CC3ON=C(C)C3)=O)CCC2)(C)C)cnncc1C c1(NC(c2c(NCc3cc(OC)c(C)cc3)cncc2)=O)nc(Cl)c(Br)cc1I C1(C(N(CCCN(C(=O)C2=C(Cl)CC2)C)C)=O)CCCCCS1(=O)=O c1cccc(C)c1O.N1(Cc2c(C(=O)OCC)ccs2)C(C(=O)N)CC2CC12 N1(C(C(C)OC)=O)CC(NC(c2cc(NC3CC3)ncc2Cl)=O)C2(CC2)C1 Cc1ccc(C(=O)N(C)CC2(O)CN(C(=O)CNc3ccccn3)C2)cc1 N1CC(C)(C)C1C1CCN(C=O)CC1.c1(C(=O)OC)c[nH]nc1.C(C)(C)C.C Cc1nc(O)nc(O)c1CC(=O)NC1CCC1C.C(=O)(CCCN1CCCC1)N CC1(O)CC2CC1CC2NC(=O)CC1CCCN(C(=O)CC2COCC2O)C1 c1(C(=O)NCCN(C(C(C)OCCC=C)=O)C)cc(-c2csc(C)n2)c[nH]1 C(=O)(CCS(=O)(=O)CC(C)C)NC1CCC(NC(C2CCCC(OC)C2)=O)CC1 N1(C(C2(Br)CC23CCC3)=O)CCN2C(CCS2(=O)=O)C1 C1(NC(C2COC2)=O)CN(C(c2ccc(C3CC3)cc2F)=O)CC12CCOCC2 c1(OC)ncc(NC(=O)C(C(C)(C)C)OC)cc1C.C1(=O)C(O)CCN1 N1(C(c2n(C=C)nnc2)=O)CC2CCCCC2(NC(=O)CC2C=CCCC2)C1 CC(C)CC(C)(CNC(=O)C(C)Oc1ccccc1F)NC(c1nocc1Cl)=O c1(C(=O)NCC2C(NC(=O)C=CC3CCC3)CC2)ccc(=O)n2c1CCC2 c1(C(=O)NC(C(=O)NCC(CO)OC)CC2CCCC2)cc(C#N)ccc1C c1(C(N2C(C(N(CCC)C3CC3)=O)CCCC2)=O)coc2c1COC2 C(c1ccc(Cl)cc1F)=CC(N1CCC(C)(C)C1C)=O.C1(C)(C=O)CCCO1.N C(=O)(CCCC(N)=O)NCC(CC)(C)NC(=O)CCc1cccnc1F c1(C(N2CC(NC(C3CCCS3)=O)C3(C2)CC3)=O)ccc(F)c2ccsc12 c1(NC(c2c(-c3ccc(OCCCC)c(F)c3)ncs2)=O)cc(F)cc(F)c1Cl N1(C(CSSC)=O)CCC2CCC(NC(c3cc(O)nc(O)n3)=O)C1C2 C1(C(=O)NCCOC2CN(C(=O)Cc3ccsn3)C2)CC2(CCCO2)C1 C1(CNC(=O)C(=O)NCC2(c3cccc(F)c3)CCCC2)CCC2CCCC2O1 CC(C)CC(C)(O)C(=O)N1CC(CNC(=O)COCC)C(O)C1.CCO.O C1(CC(=O)NC(C=CC(=O)N(CC(CC)O)C2CC2)C)COCCO1 c1(CC)cc(N2CCNCC2)nc(C(F)(F)F)n1 CCC(CC)(CCNC(C1CCC2CC1CO2)=O)NC(c1cocn1)=O C(C(CNC(=O)C(n1ccc(Br)n1)C)C(F)(F)F)NC(CCC(=C)C)=O CC1CC(=O)NC1C=O.c1(CC=O)cn(C)nc1C(F)(F)F.C1CC(C)C1 N1(C(c2c(CC)nccc2)=O)CCC2(CNC(c3cc(C)ns3)=O)CCCCC12 c1(CNC(c2cscc2F)=O)cnn2c1CN(C(=O)C=Cc1ccccn1)CC2 C1(C(N2CCC(C(C(=O)NC3CC(OC(C)C)C3)F)C2)=O)CC2(CCC2O)C1 Cc1nn(CC(=O)NC2CCC3CC2CN3)c(C)c1Br CS(C)(=O)=NC(=O)C(=O)NCC1CCCN(C(C23CCC(F)(CO2)C3)=O)C1 c1(C(=O)NCC23CCCC2C3(F)F)cc2ccnn2cn1 Cc1ncc(S(N)(=O)=O)cc1C(N1CC(NC(=O)CCC2CCC2)C(C)C1)=O CN1CCCCC1CCC(=O)N1CC(NC(=O)COCC2CC2)C1 c1(C(N2CCC(C(C)C(=O)NCCCC3CCOCC3)C2)=O)ccccc1O CCC(C#N)(CC)C(=O)NCC(C)(C)NC(=O)Cc1ccsc1Cl CC(CCCCO)NC(C12CC1CCN2C(=O)COC1(C)CCC1)=O CCC(C)(CCNC(=O)COc1cccc(O)c1)NC(c1nn(C)cc1Cl)=O O=S(=O)(N1CCC(CC(F)F)CC1)N1CCOC(CCn2ccnn2)C1 c1(NC(C2CC(F)CN2C(c2cccc(O)c2F)=O)=O)ccc(Cl)cc1Cl C12(CNC(CCC=CC)=O)CCCCC1N(C(=O)C=CCF)CC2 C#CCCN=C(NCC(F)(F)C(C)(C)O)NCC1CCN(CCOC2CC2)CC1 CC(CCN=c1[nH]cnc(Cl)c1Br)NC(=O)CC(C(F)F)n1ccnc1 c1c(C)nn(C)c1C.Cc1c[nH]cc1C(=O)NCC(C1CCCC1)NC(=O)C N1(C(CC=CC)=O)CCC(C(N2CCC(N3CC(O)C3)C2)=O)(CF)C1 CCC(C)(F)C(=O)N1CC(O)(CCNC(=O)CNC(C2CCC2)=O)C1 N1(C(C(C)NC(=O)NC)=O)CCC2(NC(c3ccc4c[nH]nc4c3)=O)CCCC12 C(=O)(CC(O)CC(C)C)NCCC(C(=O)Nc1cc(C)cc(F)c1)(C)C C=C=CC(C)C(=O)N1CCC(C(CO)NC(c2cn(C)cc2C)=O)CC1 C1(CC)CCCC2CC12.N1(C(C2(C=O)CC2)=O)CCCC1.C1(C(=O)N)CC1 C(=O)(C1CCCn2nccc21)NC1CN(C(Cc2c(C)nn(C)c2)=O)CC(O)C1 N1(C(C(CC(=C)C)OC)=O)CCC(C(=O)NC(C)COC(C)C)=C(F)C1 C(=O)(C(F)(F)CCn1ccnn1)N1CC(NC(C2C(C3C(C)C3)C2)=O)C1 CCC(C)(C)C(O)C(=O)NCc1cc(C(=O)NC2CC2C2CCC2)ccn1 c1(CN2CCC(CCNC(c3c(C)ccnc3)=O)C2)cc(F)cc(F)c1 C1(CNC(CCc2cncc(C)c2)=O)CN(C(=O)C=Cc2ncc[nH]2)CCCO1 N1(C(CC(COC)COC)=O)CC2CC1CN(C(c1ccnn1CCOC)=O)C2 C(c1cnn(C)c1)=CC(=O)NC1CC(NC(C(C=CC)O)=O)C1 c1(C(N2CC(C(C)NC(C(CC=C)(F)F)=O)C2)=O)cc2ccc(Br)cn2c1 c1(OCC)ccc(N)c(C=O)c1.C(C)(C)C(F)(F)F.C1CC1.C(=O)C.N N1(c2cn(C)nc2)CCCC(NC(C2CCOCCN2)=O)C1=O c1(NC(C=CC=CCC)C)nccc(=NCc2n[nH]c(C)n2)[nH]1 CCC(F)(C(=O)OC)C(=O)N(CC(C)NC(=O)C(O)CN(C)C)C N1(C(C(C)N(C(=O)CC2CCCOC2)C)=O)CCC(C)(O)CC1 CS(=O)(=O)C(C)C.C(=O)CC.C(=O)(C=CC(F)F)N.C1(C=O)CCC1 c1(NCc2ccc(CSC)o2)cc(NCCCC2CCS(=O)(=O)C2)ncn1 c1(CC)cc(C(=O)NCC(C)CNC(=O)CC(=O)NC2CC2)ccc1Cl C(=O)(CC(C)(C)C(=O)N1CCCC(NC(C2CCc3c[nH]nc3C2)=O)C1)OC c1(C=O)cnn(C)c1C.CCC(C)CNC(=O)CN(C)C(c1ccsc1)=O.N c1(C(=O)NC2C(OC)CN(C(C3CCCS3)=O)CC2)c(O)ccc(F)c1Br Cn1cnc(C=CC(=O)NC2CCC(O)C2)c1.C1(C=O)CC(C(F)(F)F)C1 c1(C2CCN(C(C3CN(c4nccc(OCC(F)(F)F)n4)C3)=O)C2)cccc(F)c1 C1(NC(Cc2cccc(C#N)c2)=O)CCN(C(C2COCCO2)=O)CC12CCC2 c1(C(N(C2CN(C(=O)Cc3cnc[nH]3)CC2O)C)=O)ccc(C=O)cn1.C(C)C C1(NC(c2nn(C)nc2Br)=O)COCCN(C(=O)CN2CCCC2)C1 FC1(F)CCOCC1CN(C=O)Cc1ccc(OC2CCCCC2)cc1 C1(C(=O)NC(C(C)NC(c2c(OC)n[nH]c2)=O)(C)C)CCC2(CCC2)O1 C(CN(C(=O)C(F)F)C)(CO)(CO)NC(C(C)OC1CCCC1)=O N1(C(CCC2N(C)CCC2)=O)CC(NC(c2sccc2C2CC2)=O)CC1(C)C CC(C)C(O)CC(=O)N1CCN(C(c2c[nH]nc2Br)=O)CC1C C(N1CCC(C2(C(F)(F)F)CCC2)CC1)N1C(=O)CC(OC)C1 Cn1c(C(=O)NC2CCCN(C(C3CCOC(C)(C)C3)=O)CC2)cc2occc12 Cc1cc(F)ccc1C(O)C(=O)NC1CCCC(NC(=O)Cn2cnnn2)C1 N1(C(C(C)CC(F)(F)F)=O)CCC2(CC1)COC(CNC(=O)CCCC1CC1)C2 N1(C(C2CN(C(C)C)C2)=O)CC2CC3CC2C1C3NC(C1CC2CC1CO2)=O c1(OC)ccc(CNC(N2CCC(c3ccc(C#N)cc3)C2)=O)c(C)c1 c1(C(=O)NC2CC(CNC(C(C)n3cccc3)=O)C2)cccc[n+]1[O-] N1(CC(C)C)CCCC1C(N1CC(CCNC(=O)COC(F)F)C1)=O C#Cc1cn[nH]c1C(=O)NC1CCC1CNC(c1cccc(CC)n1)=O CCC(C)(C)CC(=O)NCC(C(C)C(C)C)NC(c1cc(C(N)=O)c[nH]1)=O c1(C(=O)NC(CCCNC(c2c(CC)nn[nH]2)=O)C)cc(Cl)ncc1N c1(CC(=O)N(CC)C)ccc(S(C)=O)cc1.c1(C(C)OC)nc(C=O)co1.N c1(CC(=O)NC(C2CCCN(C(CCC(=C)Cl)=O)C2)C)c[nH]c2cccc(Cl)c12 NC1CCC2(CCC2)N(S(=O)(=O)CCC2CCOCC2)C1 n1(CC=C)c(N2CCC(NC(=O)OCC)C2)nnc1C(C1CCCCC1)C N1(C(=O)CCCC2CC2)CCC2CCN(C(c3cc(-c4ccoc4)[nH]n3)=O)C2C1 c1(C(=O)NC2CCN(C(c3c(C)con3)=O)C(C)C2)n[nH]c2ccc(O)cc12 C1(C(=O)NCC2N(C)CCCC2)CC12CCN(Cc1ccon1)CC2 CC(C)(C)CC(O)CC(=O)N1CCCCC1CNC(=O)CC(C)(C)C C1(C)(C(=O)NCC(C)(C)NC(CCc2n(C)ccn2)=O)CC2CCC1O2 c1(OC)cncc(NC(=O)CC2COCCN2Cc2nccnc2Cl)n1 c1(C(=O)NC2CN(C(CCOCCOC)=O)C(C)CC2)c[nH]nc1S(N)(=O)=O c1(C(=O)Nc2ccc(-c3ccsc3)cc2)ccnc2c(C(F)(F)F)cccc12 Cc1ccc(CC(=O)NC2CCC23CN(C(=O)C=Cc2cnc[nH]2)C3)c(C)c1 c1(C(N2CC(NC(COCC(=O)NC)=O)C2)=O)cc(-c2ccccn2)ns1 C(=O)(C(CNC(=O)C(C1CCCCC1)F)C(C)C)N(CCCCO)CC N1(C(CC(C)(C)C#N)=O)CCCC(C)(C)C1CNC(c1cc(F)n[nH]1)=O CC1CN(C(=O)CCF)CCC12CCN(C(c1csc(-c3ccco3)n1)=O)CC2 C1(C(=O)NC2CC(NC(CC3(N(C)C)COC3)=O)C2)CCOC1(C)C C(=O)(C1=CC2C=CC(C1)C2)N1CCC(C)(C(=O)NC2(C)CC(C)C2)C1 C(=O)(C1=NOCC1)NCC1(CC)CC(C)(C)C1.C(=O)C(C)(C)C(C)O.C Cc1c(C(=O)NC2CN(C(=O)CC(C)(C)F)C2)sc2[nH]cnc(=O)c12 Cc1[nH]c(C)c(C(N2CCC(Cn3cc(CN(CCO)CCO)nn3)C2)=O)c1C Cc1cc(NC(C2CC(F)(F)CN2c2ncc(C(F)(F)F)cn2)=O)ccc1I N1(CC)CCC(C=O)CC1.C1(C(=O)NC)CCCC1.C1(C2CC2)CCCO1.C C1(N(C(=O)C(=O)Nc2nccs2)C)CC(O)(C)C1.C(=O)(C)N.C1CC1 C1(C=O)CCCCC(C)(C)C1.c1(OC)nc(C)cnc1C(=O)NC1(C)CCC1 CN1CCOc2c(C(=O)NC3(CNC(=O)CSC(=N)N)CCOCC3)cccc21 c1(C=O)ccc(S(N)(=O)=O)c(N)c1.C(C)(CCC(=O)NC1CCC1C)SC C(=O)(CC(C)C(F)F)NCC(CNC(CC1(OCC)CC1)=O)F C(=O)(CC(C)(C)Cc1ccc(Cl)cc1)NC1C(CNC(CC(C)C)=O)CC1 N#CCCCS(=O)(=O)NCC1CNC(=O)C1 C(=O)C(F)(F)C(O)C1CC1.c1(C=O)c[nH]nc1C1CCC1.C(C)C1CCC1.N C1(C(N(c2ccccc2)CCCC)=O)CC(C)N(C(=O)Nc2cc(C)nn2C)C1 CCC(O)C(C)C(=O)N1CCOC(C(C)NC(C2C(C)(C)C2(C)C)=O)C1 N1(C(c2c(C)[nH]cc2)=O)C2COCC1CC(NC(=O)C(C)OC1CCOC1)C2 C1(C(=O)NCC2C(NC(=O)CCc3ccccc3)C2)CC12CCC(F)(F)CC2 C1(C(N(CCNC(C)=O)C)=O)CC12CC(NC(C1CC(C)C1)=O)C2 C1(C(=O)NC(C2CC=CCC2)C(=O)N(CC(N)=O)C)CC1C1CCCC1 CC(C)(C)C(O)CNC(=O)C(Cn1cccn1)NC(=O)C=CCF C1(CC)CC2CCC(C1)N2C(=O)C(CCSC)NC(=O)C(C)N(C)C(C)=O N1(C(C2(CC)CC2)=O)CCC2(CC2)C1.c1(CC=O)nc(C2CC2)cs1.CO Cc1cc(C(N2CC(CNC(c3cc(C(C)C)no3)=O)C3CC23)=O)cc(O)c1 N1(C(C(CCC#C)O)=O)CCC2CN(C(=O)COc3ccccc3C#N)CC12 N1(C(c2cc(COC)oc2C)=O)CC2CCCC(C1)N2C(=O)C(C)C(F)F C1(CCCNC(c2cc(OC)ns2)=O)CN(C(c2cncc(C)n2)=O)CCO1 C1(NC(=O)CN2CCSCC2)CC2CCC1CN2C(=O)CCC1CCCO1 c1(CN2CCC(F)(C(=O)Nc3n(C)nnc3)C2)cc2c3c(c1)CCCN3CCC2 NS(=O)(=O)c1ccc(CNC2(c3cc[nH]n3)CCOCC2)o1 N1(C(C(C2CCC2)OCC)=O)CCC2(CCC2)C(C)C1.C1(O)(C=O)CC1.N CON(CCC(=O)N1CCC12CCCCC2)C(=O)C(C)c1cncnc1 C1(C(=O)NC2(C)CCN(C(c3cnc(C)nc3)=O)C2)CCc2cnn(C)c2C1 c1(C(=O)NC(c2ccccc2)CNC(CCC)=O)oc(C(F)F)cc1C.C1CC1 C12(NC(C(F)=CCC)=O)CC1CN(C(c1cc(C(C)CC)no1)=O)C2 C1(C(N2C(C(=O)OC)CC(O)C2)=O)CC2CCN(CC(N3CCCCC3)C)CC12 c1(CC)c(C(=O)NCC2(O)CC(C)C2)cn[nH]1.C(=O)CCCC1CCC1 C1(NC(CN(CC)CC)=O)CCC2(CCN(C(c3cc(C)co3)=O)CC2)C1.C C1(Cc2c(C)oc(-c3ccccc3)n2)CCN(C(=O)CCCC#N)CC1O N#Cc1c[nH]c(C(=O)NCC2CC(O)CN2C(c2cnccn2)=O)c1 C(N=c1cc(NCCC(C)P(C)(C)=O)nc(C(F)(F)F)[nH]1)c1cnc(C)[nH]c1=N C1(C(N(CCNC(C2CCCSC2)=O)CC)=O)CCc2c(ncn2C)C1 Cc1ccc(C)c(C(N2CCN(C(=O)Cn3nnnc3C)CC(O)C2)=O)c1N c1(OCCCC)ccc2cc(C(N3CCC3C3CCC3)=O)[nH]c2c1 c1cnn2c1CN(C(c1cnc(C#N)s1)=O)CC2.C1(C(NC)=O)(N(C)C)CC1.C c1(C=O)ccc(Cl)c(C)c1.N1(C(C)=O)CCC(C)(C(=O)NCCCC(C)C)C1.N N1(C(c2c(C)c(Br)cnc2)=O)CCC(C2CCN(C(=O)CNC=O)C2)C1 c1cc(Cl)cc(Cl)c1.n1(CCOCCNC(C2CC2(Cl)Cl)=O)ccnn1.C c1(C(N(CC(C)NC(C2CN3CCC2CC3)=O)CC)=O)cc2ccc(O)nc2s1 N1(C(CC#N)=O)CCC2(CC1)CCN(C(=O)C1CCCc3ncnn31)CC2 c1(CC=O)ccc(C(F)(F)F)cc1.c1(C(=O)NCCCC)cnn(C(C)C)n1 C1(CC(=O)N(CCCCCCC)C)CN(C(=O)C(CC2CC2)OC)CC12CC2 CC1CCN(C(C23CC(C)C2C3)=O)CCN1C(C1CCN(C2COC2)CC1)=O CC1CN(C(C2CCCS2)=O)CCN(C(C2CCC(C)CC2)=O)C1 C1(NC(CCC(C)(C)OC)=O)CN(C(=O)CC2(CO)CC2)C2(CCOC2)C1 C1(NC(COC)=O)CN(C(=O)Cn2cnc(-c3ccccc3)n2)CCC1CO c1(C(=O)OC)ccccc1-c1cccc(CNC(c2cccnc2)C)c1 N1(C(C2CCCN(C(C)C)C2)=O)CC=C(CNC(=O)CCN2CCOCC2)CC1 C1(C(=O)NCCN(C(c2cnc(CC)[nH]2)=O)C)C2CCC(C2)S1(=O)=O C(=O)(C#CC1CCC1)NCC1(C(=O)Nc2c(OC)ncnc2)CC=CC1 C1(NC(C(CC(C)C)O)=O)CC2CC1CN(C(c1cnc(-c3cccs3)o1)=O)C2 Cc1ccc2[nH]c(=NC3CC(NC(=O)C(F)n4cccn4)C3)sc2n1 CCCC(CC)CC(=O)NC(c1ccccc1)CNC(=O)CN1CC=CC1 N1(C(c2c(CC)cncc2)=O)CC2CC3CC2C1C3NC(c1ccnnc1O)=O CCC(CC(=O)N(C1CC(NC(=O)CC2COCCN2C)C1)C)SC c1(OCC)cnc(C(=O)NC2CN(C(c3cccnc3O)=O)CC2SC)cn1 c1(C(N2CC(NC(c3ccc(C=C)cc3)=O)C3C2C3)=O)[nH]c2ccccc2c1Cl CC(CCCN=c1cc(Cl)nc[nH]1)NC(=O)CC1CC=CCN1C Cc1cc(C(F)(F)F)nc(=NCC(CNC(c2nc(Cl)sc2C)=O)C(F)(F)F)[nH]1 N1(C(c2cn(C)[nH]c2=N)=O)CC2CC(NC(=O)CCO)C2C1.c1ccc(F)cc1 N1(C(c2c(C)nc(O)[nH]2)=O)CC2CC(CNC(c3n[nH]c(C)c3O)=O)C2C1 c1(C(=O)OC)cncc(CC=O)c1.C(c1cnc(C)s1)=CC=O.CC(O)CC.N C12(CNC(C(C=C)(C)O)=O)CC(CCO1)C2.C(c1ccccc1)=CC=O.N C12(CNC(C(C)O)=O)CN(C(=O)C(C)(C)Cc3ccccc3)CC1CCO2 c1(OC)cc(C(=O)NCC2CC(C(=O)NCCc3cc(C)[nH]n3)C2)[nH]n1 c1(C(=O)NC(CC)(CNC(c2nc(C)n(C)c2C)=O)CC)ccc2snnc2c1 C=CC(C)(C)CC(=O)NCCOCCN(C)C(c1nc(Cl)cs1)=O CCC(C)CCCC(=O)N1CC(OC)CC1CCNC(c1ccc(F)cn1)=O N1(C(c2c(C)nc(CC)o2)=O)CCOCC(CNC(=O)C=C2CC2)C1 C(=O)(C1=CCCC1C)N1C(CC)C(NC(=O)CC(C)(C)OC)CC1 c1(C(=O)NC2CC(CC)(CC)N(C(c3ncsc3C)=O)C2)cc2ccncc2o1 C(=O)(CCCCCCC(C)=O)N(C(CCNC(C(C)OCC)=O)C)C C1(NC(CC(=O)OC)C2CCC2)(COC)CCN(C=O)C1.C(C)(C)C.O C(=O)(C1=C(C#N)CCC1)N1CCCC(NC(CC(C(C)C)C)=O)C1C C(=O)(C1CCc2scnc21)N(C)CCNC(=O)C=C1CCOCC1 C1(COC)CC(C)N(C(=O)Cn2cc(C)cn2)C1.c1(CC=O)ccsc1.N C(=O)(C#CC1CCOC1)NC(CC1CN(C(c2ccc(NC)cc2Cl)=O)C1)C c1(C(=O)NC(C2N(C(Cc3c(C)scc3)=O)CCCC2)C)cc(F)cc(F)c1N c1(C(N2CCN(C(c3cc(OC)no3)=O)CC2C2CC2)=O)cn2cc(C)sc2n1 C1(CCOC)(NC(C2CCC3CC3CC2)=O)CCN(C(C)=O)CC1 C1(N)CS(=O)(=O)C2CN(C(=O)CC3CC34CC4)CC12.c1cncc(Cl)c1.CC Cc1nc(NC(C2CC2C(=O)Nc2cnc3[nH]ccc3c2)=O)nc(Cl)c1Br N1(C(C=CC)=O)CC2(CCN2C(=O)C(C)NC(C2CCC(=O)N2)=O)C1 C1(c2n(C(CC)(C)C)nnn2)(NCc2cc(C)cc(Br)c2)CC2CC1CC2(F)F CC1(C)CC(C)(C)c2cc(NC(=O)NCc3sccc3Br)ccc21 N1(C(CCC=CCC=C)=O)CC=CC(C(=O)NCCc2cnn(C)c2C)C1 c1(C(=O)NC2C(C3CCN(C(CC)=O)CC3)OCCC2)cnn2cc[nH]c(=O)c12 CS(=O)(=O)C1(C(=O)NC2CC(CNC(=O)Cc3nncs3)C2)CC1 c1(C(c2nnnn2C)NC(C)C(O)Cc2cccc(Br)c2)ccc(Cl)c(Br)c1 C1(CNC(c2cn(C(C)(C)C)nn2)=O)CCCCN(C(c2occc2F)=O)C1 C(=O)(CC(F)(F)Cl)N1CCC(C(C)(C)NC(c2cc(CC)sn2)=O)C1 C1(C(=O)Nc2c(C)c(Cl)ccc2)C2CCCC2CN1C(=O)CCCF C(C)(C(C(=O)NCC(C)CC1CCC1)C(C)C)NC(C(=O)NCC)=O C(=O)(CC(C(F)F)NC(C1(C)CCC(=O)CC1)=O)N1CC(n2ncc(C)c2)C1 C(=O)(C1=CC(O)CC1)NCCc1cncc(C)n1.C1(CC=O)CCCC(=O)C1.N N1(C(CSC)=O)CCC(C2CC2NC(c2ccc(N3CCCCC3=O)cc2)=O)C1 C(=O)(C(C)(C)C(F)F)NC1C(CC)N(C(c2cccc(Br)c2OC)=O)CC1 N1(C(CCC2CCCN(C)C2)=O)CCC(C2(O)CCN(C(C3(C)CC3)=O)C2)CC1 N1(C(CC(C)CN(C)C)=O)CC2CC1CN2C(=O)C(C)(O)CCc1ccccc1 c1(C(C)=O)cccc(OC(C)C(N2CCCC2)=O)c1.C1(C#N)(C(NC)=O)CC1 C1(CC)CCC(O)(C(=O)NCCC2(NC(=O)C3CC3)CCC2)C1 CCCCC(CNC(=O)C(C)(C)C#N)NC(=O)C(C(C)C)NC(N)=O Cc1cn2nc(N3CCCC3CN(C(=O)Cc3csnc3C)C)sc2n1 N1(C(c2ccc(CC3CC3)cc2)=O)CCC(O)C(C=O)C1.c1ncn(C)n1.CN c1(C(=O)NC(CN(C(=O)CC2(O)CCOC2)C)(C)C)cnccn1 c1(NC(CNC(c2ccn(CCC)n2)=O)CO)ncnc2c1c(Br)nn2C CC1CCCC=C1C(=O)NCCN(C(c1cnsn1)=O)Cc1ccccc1 N1(CC(=O)Nc2ccc(C)cc2)CCN(C(c2cc(C)no2)=O)C(C)C1 N1(C(C2C(C#C)C2)=O)CCC2(CCCN(C(C3(OC)CCCOC3)=O)C2)C1 c1(C(C2CCOC2)NC(C(C)C)=O)ccccn1 c1(NC(C)=O)cc(Cl)ccc1C(N1CCOCC(NC(c2cc(Cl)c[nH]2)=O)C1)=O c1(N(CCN(CCN(C)C)C)C)ccnc(C(C)C)n1.C1C2CCC(F)(F)C12.N C1(C(=O)NC2C(NC(=O)OC(C)(C)C)COCC2)C2CS(=O)(=O)CC12 N1(C(C2C(C)CCO2)=O)CCC(C)(NC(c2nccc(C(F)F)n2)=O)C1 C(C)(C)(C(=O)N)NC(=O)OC.c1(-n2cccn2)cc[nH]n1.C1CCC1.C=O Cc1cc(C(N2CC3(NC(=O)Cc4scnc4C)CCC2C3)=O)c(Cl)cc1N CC1CC(NC(c2ccc(O)cn2)=O)CN(S(=O)(=O)CCCl)C1 c1(C(=O)NCC23C(CN(C(C(c4cn(C)nc4)=O)=O)C2)C3)nnn2c1CCCC2 c1(C(=O)N(Cc2ccccc2)CC2CCCO2)cnc2[nH]nnc2c1 C1(C(=O)NC(CN(C(=O)C=Cc2cccs2)CC)C)CCOC(C)(C)C1 N1(C(C2CCN(CC)CC2)=O)CCC(C2CC2)C1C.c1(CC(=O)N)nonc1C CCC(C(=O)N1CCC(N(C(=O)CCC(C)C)CCOC)CC1)C(C)C c1(NCc2c(S(C)(=O)=O)scc2)nccc(=NC2CC3C(C2)C3(F)F)[nH]1 c1(-c2cccc(C)c2)nc2c(s1)CC(C(=O)NCC1CN(C)C1)CC2 CC1(C)CC(NC(=O)C(F)F)CN(C(=O)CC2CCCC(C)(C)C2)C1 O=C(C1CCCc2nc[nH]c21)NC1CCCCCN(C(=O)Cc2ccno2)C1 c1(C(N2C(CCNC(c3scc(C)c3C)=O)CCC2)=O)ccc2c(c1)ncn2C C(CC(=O)N1CCN(C(=O)CCn2cc(Cl)cn2)CC1C1CC1)(C(C)C)OCC c1(C(N(C2CCN(C(C3CC(C#N)C3)=O)C2)C)=O)cnn(C)c1F Cc1cc(C(=O)NCC2CN(C(C3SCCCS3)=O)CCC2C)c(O)nc1C CCC(CCCC(=O)N(C)Cc1cnc(C)cn1)NC(c1ccnc(C)c1C)=O C1(CNC(COCC(C)C)=O)COCCN(C(=O)COCC2CC2)C1 c1(C(N(CC(CCC)C)C)=O)ccc(C#N)c2ccccc12 C1(NC(CC(CC)(F)F)=O)CCCCC12CCN(C(=O)CCc1ccon1)C2 c1(C(N(CC(C)(C)NC(Cc2nc(C)sc2)=O)C)=O)ccc(C(F)(F)F)nc1 CCC(C)(CNC(=O)Cn1[nH]cnc1=N)C(=O)N(CCCC(O)CO)C c1(C(=O)NCC(CC)NC(C2(C3CCC3)CC2)=O)c[nH]c2nccc(Br)c12 C12(CCNC(COCCOC)=O)CCC1CN(C(C1SCCS1)=O)C2 C1(F)(C(=O)NCCN(C(C2CCC(C(CC)(C)C)CC2)=O)CC)CCCCCC1 N1(C(COCCCC)=O)CCC(C2CCCN2C(=O)C(C)Cn2cccn2)CC1 CC1CCCc2ncc(C(N3CCN(C(C4OCCOC4(C)C)=O)CC3)=O)n21 c1(C(C)=O)ccc(C(=O)NCCCCNC(=O)C2=CC(C)CC2)c(F)c1 C(=O)(CS(=O)(=O)C1CC1)N1C(CC)C(NC(=O)C)CC1.c1csc(C)n1.S C1(CC(=O)N(CCC(=O)OC)C)C=CC(NC(=O)CC(C)F)C1 C1(C)(C(=O)NCCNC(C(CC#C)O)=O)CC2CCC1CC21OCCO1 N1(C(CCCC#C)=O)CCC(C(=O)NC2CCCCCC2(C)C)=C(F)C1 C1(C(=O)NC(CCC)(C)CO)CCN(C(=O)CC(O)C(C)C)CC1C c1(C(=O)NCC(O)CNC(=O)C)cc(Br)c([N+](=O)[O-])[nH]1.c1ccccn1.N N1(CCC=O)CCOCC1=O.c1(CC)cnc(CC(=O)N(C2CCCC2)CC)[nH]1.N Cc1nc2c([nH]1)CN(c1cc[nH]c(=NCCC3CCC4CC34)n1)CC2 Cc1ccc(NC(C2(NC(=O)CC(C)C(C)C)CCC2)=O)c(O)c1 Cc1c(CN=c2[nH]c(C(=O)NCc3ccc(Br)cc3)cs2)cccc1Cl N1(C(C(c2ccn(C)n2)(C)C)=O)CC2CN(C(=O)C(C)(C)c3ncco3)CC2C1 c1(NC(C2CCN(C(C)=O)CC2)=O)ccc2c(c1)CCC2NC(C)=O c1(C(N2CCC(CNC(CCC(=C)C)=O)CC2)=O)nccc(C)c1O N1(C(c2c(COC)cco2)=O)CC(=O)N(C)CC1c1ccccc1 C(CC1=CCN(C(c2cc(F)cs2)=O)CC1)NC(=O)C=Cc1cncc(F)c1 C=C1CC(C(N2CCC(CCNC(=O)CC)C2)=O)(C(F)F)C1.CC(F)(F)F CC(C)C(O)(C(=O)NCCCNC(c1ccc2c(n1)CCCC2)=O)C(F)(F)F O=C(CS(=O)(=O)CCO)NCC.C1(C(N2CCCC2)=O)CCC(=O)N1C1CC1 Cc1ccc(-n2nc(-c3ccoc3)nc2C2CC(=O)N(CC(F)(F)F)C2)cc1Br CCCC(CCC)CC(=O)NC1CCC(CCNC(C23CCC(CC2)CC3)=O)C1 N1(C(=O)C(O)CN2CCCC2)CCN(C2CCN(C(C3CCO3)=O)C2)CC1 C1(CCC=C)(C(=O)NC2CC(=C3CC3)C2)CN(C(C2CCN(C)C2)=O)C1 c1(N2CCC(S(=O)(=O)NC)C2)nc(N2CCOC(CCF)C2)c2sccc2n1 c1(N2CCN(c3ccc(C)cn3)CC2)nc2ccc(Br)cn2n1 n1(CCCOC)nccc1CNCCC1CCC(N)C1 c1(CCC(=O)NC2C(NC(Cc3ncc(C)[nH]3)=O)CC2)cccc(C#N)c1 C1(C(=O)NC2CC(CC)(CC)C2)CCCCCC1NC(C1CC(C)C1)=O.C Cc1cn(C)nc1C(N1CCC(NC(=O)C(=Cc2cccnc2)F)C1C1CC1)=O Cc1c(Br)cnn1CC(=O)NCC(n1cc(-c2ncoc2C(F)F)nn1)C C1(C(N(CCCC)CC(N)=O)=O)CCC2(CC2)N1C(=O)CC(C1CC1)C C(C(=O)NC(C1CCCN1C(c1csc(CC)n1)=O)(C)C)(C(C)C)SCC N1(C(C2(C)CCN(C(CCc3cn(C)nc3)=O)C2)=O)CCCC(O)(CO)C1 CCCCC(C(=O)NCCC(C)N(C)C(c1sc(C)cc1Cl)=O)C(C)C N1(C(c2nnc(CC)s2)=O)CCC(NC(c2cn(CCOC)nn2)=O)CC1C Cc1cc(N2CC(NC(=O)C(=O)Nc3ncc[nH]3)CC(C)(C)C2)n2ncnc2n1 N1(C(CNC(CCC)=O)=O)CCCCC1C(N1CCCC(OC(=O)NC)C1)=O Cc1cccc(N2CCCC(NC(c3ccc(OCc4nc[nH]n4)cc3)=O)C2)n1 c1(C(=O)NCC2CCCN(Cc3cccc(Br)c3)C2)ccc2cc[nH]c2n1 c1(C(=O)NC2(C#N)CCN(C(C(CC)CC)=O)C2)ccc2c(c1)c(C)nn2C C1(CNC(C(C)=C2CC2)=O)C2CN(C(=O)CC3CC4CC4C3)CC12 c1(NC(c2csc(C(N3C4CCC3COC4)=O)n2)=O)ncc(Br)c(O)n1 Cc1cc(C)c(C(N2CC3(C2)CN(C(C2CC(C4CC4)C2)=O)C3)=O)cn1 C(c1ccccc1)=C(CC)C(N1CCOCC1CNC(c1csnc1OC)=O)=O N1(C(c2cc(C(N)=O)ncc2)=O)CCC2CN(C(=O)C(O)C(F)(F)F)CC2C1 N1(C(CC2(C=C)CC2)=O)C(C)CC2CN(C(c3c[nH]nc3C)=O)CC12 O=C(C(O)C(F)F)NC1CCN(C2CCN(C(c3cccnn3)=O)CC2)CC1 CC(C)C(C)CN(C(=O)C(C)CN(C)C(c1c[nH]c(C(N)=O)c1)=O)C N1(C(c2n(C)c(O)nc2)=O)CCC2CCC12CNC(=O)C(F)(F)c1ccccn1 C1(C(=O)NCC(C(C)C)NC(C2CCN(OC)CC2)=O)CCCCC12CCC2 N1(C(C(CN(C)C)NC(C(C(=O)OCC)F)=O)=O)Cc2ccc(C)nc2C1 C1(=C(C(=O)NCCNC(C(C)c2ccco2)=O)F)CCCCC1 C1(C(=O)NC2(CCCC(=O)NC3(CCF)CC3)CCC2)CC2(CC(=O)C2)C1 c1(C(=O)NC(CC=C)CNC(=O)C(C)C(F)(F)F)cc(F)c(F)c(F)c1F N1(C(C2CC(F)(F)C2)C)CCCC(NCc2cn(-c3ccn(C)n3)cn2)C1 CC1(C)C2CCC(CC(N3CC4(CCCC4NC(=O)CCCC#N)C3)=O)C1C2 C1(NC(Cc2scc(C)c2)=O)CN(C(=O)CCC(C)C)Cc2nccn2C1 CC1(C(=O)NCCC2CCCC2O)CCN(C(=O)CCOC2CCCC2)C1 C1(C)(NC(c2c(OC)cccn2)=O)CCN(C(=O)C=CC(C)C)CC1 c1(CNC(c2c(C)cc(C)[nH]2)=O)ccc2c(c1)CCCC2NC(c1cscn1)=O C1(C(N(CC(O)C)C)=O)CCN(S(C)(=O)=O)CC1.C(=O)(C(O)C1CCC1)N N1(C(CN(C)C)=O)CCC2CN(c3ccc(F)c(C#N)n3)CC2CC1 c1(C(=O)NC2C(C)CN(C(=O)CCOC3CCCC3)C2)ccn2ccnc2n1 C(=O)(C(C)C(C)(C)C)N(CCNC(c1cnc(C)n1C(F)F)=O)C(C)C c1(C=O)cc(N)c(O)c(F)c1.C1(NC(C(CN(C)C)O)=O)CCC(F)(C)C1.N c1(OC)ccc(C)cc1C(N1CC2(NC(=O)CCn3ccccc3=O)CC1C2)=O n1(CC(N2C(C)CCC(CNC(CC3(C)CC3)=O)C2)=O)ccc2ccc(Cl)cc12 c1(C(=O)NCC2N(C(CC3OCC(C)(C)OC3)=O)CCC2)cc2sccc2cn1 c1(C(=O)NC2CC(NC(C3C(OC)C3)=O)C2)ccccc1CN(C)C C1(C)(CC)CN(CCNC(=O)Nc2cccc(Cl)c2)CCN1C(C)=O C1(CC)CCCCN1C(C1(SC)CN(C(=O)CC2CCC(=O)N2)C1)=O C1(NC(C2(CC)CC2(F)F)=O)CN(C(=O)CCNC(=O)CO)CC1C c1(C(N2CCCC(N(C(=O)C=Cc3ccc[nH]3)C)C2)=O)nccc2ncncc12 C1(C(=O)NC2CC(CNC(C3CCCO3)=O)C2)(OCC)CCCC1.C c1(NC(COc2cccc(C(C)=O)c2)=O)n[nH]c2c1CCC(C(C)(C)C)C2 c1(C(N2CCC(OCCNC(C(CCCC)C)=O)C2)=O)ccc(P(C)(C)=O)cn1 c1(OCCC(=O)NCC(CO)NC(C2CC2C(F)F)=O)cccc(Cl)c1Cl c1(C(N2CC(c3cn(CCCc4nnc(C)o4)nn3)C2)=O)cccc(Cl)c1Br C1(NC(C)=O)CN(C(=O)CC2CC(c3ccccc3)C2)C(C)C1.C(=O)(C)N O=S(=O)(c1ccc2nc(N3CCC(C(=O)O)C3)sc2c1)NCc1ncc(Br)s1 C1(C(=O)NC2CN(C(C(CCSC)OC)=O)C2)Cc2ccccc2C1(C)C c1(C(C)C)cc(C(N2CCC(n3cc(CCC(N)=O)nn3)C(O)C2)=O)ccc1F c1(C2C(C=O)C2)ccccc1.CC(C)(C)C=CC(=O)NC(C)(C)C1CC1 c1(OC)cc(NC(=O)CC2CCC2)ccc1C(C)C.C(=O)C.C(C)=O.N N1(C(C(C)OCCOC)=O)CC(O)CC1.c1(CC=O)cc(C2CC2)on1.C C1(C)(C(=O)N)CC2CCC(C1)S2.n1(CC=C)ccnc1C(=O)NC(C)CCC Cc1cc(C(=O)N(C2CCN(C(=O)C(=O)N(C)C)C2)C)cc(C)c1Cl C1(C=O)C2CC1N(C(=O)Cc1ccccc1C)C2.C(=O)(CC1CCCC1)OC.N c1(CC)nn(C)cc1C(=O)N.C1CC(F)CN1C(=O)C(C(C)C)c1ccncc1 c1(C(N2CC(C)(NC(Cn3c(=O)ccc(C)c3)=O)C2)=O)ccc2c(c1)OCCN2 CC1(C(=O)Nc2ccccc2-c2cc[nH]n2)CCCN(C(c2ccccc2)=O)C1 C12(C(=O)NCC(C3CC3)NC(c3c(CC)cc[nH]3)=O)CCC(OC)C1C2 c1(C(C)NC(=O)NC2(C)CC2C(F)(F)F)ccncc1Br C(CN(C(C)C)N1CC(C(F)(F)F)OC(C)C1)c1onc(-c2c(C)cccc2)n1 N1(C(C=CCC(C)(C)NC(=O)CC=O)=O)CC(S(C)(=N)=O)C1.C1CC1.N c1(C(=O)N)ccc(C)c(Cl)c1F.C#Cc1cn(C)nc1C(N1CCC(O)(C)C1)=O c1(C(=O)NCC2CN(C(C3CC(O)C3)=O)CCO2)ccc2c(c1)B(O)OC2 C12(C(=O)NC(c3cccc(C)n3)C)CCCC1CCN2C(c1csnn1)=O C1(CC)CCN(C(c2csc(F)c2)=O)C1CNC(=O)CN1CCC(C)C1 c1(CNC(C2N(C(CCOCCC)=O)CC(OC)C2)=O)ncccc1OC c1(OC)ccc(C)cc1CC(N1CCCC1C)=O.C12(C(=O)N)CCC(CC1F)C2 C12(NC(CCC(=C)Cl)=O)CCCC1CN(C(=O)Cc1ccn3cncc3c1)C2 Cc1cc2ncc(C(=O)N(C3CCC3)C)c(C)n2n1.C1(C)(C=O)CS(=O)(=O)C1 N1(C(C2CCN(C(c3ncn(CC)c3)=O)C2)=O)CC(O)CC(O)C1 c1(CNCC(CC)CC)ccc(Oc2cccc(F)c2)cn1 c1(C(N(CCn2cc(C(CC)(C)O)nn2)C)=O)cc(C)cc(O)n1 Cc1cc(Cl)ccc1C(=O)N(CCCNC(C1CC1(F)Cl)=O)CCO N1(C(c2[nH]cc(C)c2)=O)CC2(CC(NC(=O)CCN3CCC3)C2)C1 Cc1cc(C(N2CC(CNC(C3CCCS3)=O)CC23CCC3)=O)ccc1[N+](=O)[O-] Cc1nnc2cc(NC3CCN(C(=O)C(C)(C)CC(C)(C)C)CC3C)ncn12 C1(CN(C(c2ccnn2C)C(=O)NCC=C)C)COC(=O)O1 N1(C(C2(CC)CC2(F)F)=O)CC2(C1)SCCC2NC(c1cnsn1)=O C1(C)(NC(c2c(C)cc[nH]2)=O)CCCCC1C(=O)NC1(c2cccs2)CC1 C1(CNC(c2c(C)oc(Cl)n2)=O)CCCN(C(=O)CCCc2cccnc2)CC1 C(c1cccc(Cl)c1)=CC(=O)NCCC(=C)C.c1(C(=O)N)occc(=O)c1 C1(C)(CNC(c2cnn(C)c2Cl)=O)COCCN(C(C2CSC2)=O)C1 c1(SC)cc(C(=O)NC(C)CN(C(=O)C(F)C(C)C)C)cc(Cl)c1 CCC(CNC(=O)CC1CC1(Cl)Cl)(CC)NC(=O)CC1CCC(=O)C1 N1(C(C(C)c2ccco2)=O)CCC2(CCN(C(=O)CO)C2)C1.C(F)(F)C(F)(F)F O=C(C1=CS(=O)(=O)CCC1)NC12CC1CN(C(C1(CC(F)F)CCC1)=O)C2 c1(C2(C(=O)NC3C(NC(C4C(C)CCC4)=O)CCC3)CC2)ccc(Br)cc1 n1(CC(C)O)cc(CSCCNC(c2ccn(C(C)(C)C)n2)=O)nn1 C1(C(=O)NCC2N(C(c3cc(COC)no3)=O)CC2)C2CN(C)CC12 C(=O)(CC(C(=O)N1CC2(CCC2)C1)N(C)C)OC.C12(C=O)CC3CC1C2C3.C N1(C(CC(c2scc(C)c2)O)=O)CCC2(C1)CN(C(c1cnc(C3CC3)o1)=O)C2 Cc1ccnc2sc(C(=O)NCC(O)CN(C(=O)CC(C)N(C)C)C)c(C)c12 CC1=CCC(C(=O)NCC2CCN2C(c2cnc(N(C)C)nc2)=O)CC1 Cn1cc2c(n1)CCCC2C(=O)NCC1CC1NC(=O)CCSC1CCCC1 Cc1cc(C(=O)NC2COCC2CNC(=O)CCCN(C)C)cnc1O c1(C(=O)NC2CCCCC2)cccc(F)c1Cl.c1(C(=O)N)scnc1C(F)(F)F c1(CC)nnc(C)cc1C(N1CCC(N(C)C(c2cnc(OC)c(Cl)c2)=O)C1)=O CC1CN(C(=O)COCc2ncnn2C)CCCN1C(C1CCCCC1O)=O N1(C(C2(C)CCNC2=O)=O)CCC2(CCCN2C(c2cc(Cl)ccc2F)=O)CC1 c1(C(=O)NCCN(C(=O)C(F)C2CCOC2)CC)cccc(N)c1 c1(C(=O)OCC)cccc(N(C)C(c2csc(CC3CCOCC3)n2)=O)c1 c1(C(=O)NC2CN(C(C3=C(C)OCC3)=O)CC(O)C2)cccc2c1oc(=O)n2C CC1C2C(CCN2C(C2(n3cnnn3)CC2)=O)CN1C(c1cnncc1O)=O C1(NC(C2(C#C)CCCC2)=O)CCC2(CCN(C(=O)CC3CCCN3C)C2)C1 c1ccc(C)cc1.C(=O)(CCn1cccn1)NC(CN(C(=O)CO)CC)C Cc1cn2cc(C(=O)NCC3CCN3C(=O)CCC(O)C(C)(C)C)ccc2n1 C(=O)(C(C(C)CC)O)N(CC1CCN(C(C(CCC)NC(N)=O)=O)CC1)CC Cc1oc(C(=O)OCC(F)(F)C2CC2)cc1Br CP(C)(=O)c1ccccc1C(=O)NC1C=CCN(C(=O)C#CC2CC2)C1 C(=O)(CS(C)(=O)=O)N(C1CCN(C(=O)CCn2cc(Br)cn2)C1)CC N(S(=O)(=O)N(C)C)(CC(c1cccc(C)c1)=O)CC1CCOC(C)(C)C1 N1(C(C(C)(C)n2ccnn2)=O)C2CC1CN(C(C1CC3(CC3)CO1)=O)C2 c1(NC(C2CC(F)CN2C(c2cc(F)c[nH]2)=O)=O)c(C(F)(F)F)cccc1Cl N1(C(C(C)C2CC2)=O)CC(O)(C2(C)CC2)C1.C(=O)(CCC(=O)c1ccccn1)N C1(C#N)(C(=O)NCC(C)(C2CC2)NC(c2cc(C)[nH]c2)=O)CC2CC2C1 Cc1nccc(C(=O)NC(C2CCN(C(C3CC34CC(O)C4)=O)C2)C)n1 N1(CC(=O)NCC)CCC(CN2CC(C)OC(C)C2)C(C)C1 c1(C(N2CC(N(CC=C)C)C2)=O)cnc(CNC(=O)C(CC)SC)nc1 C1(CC)CC(F)(F)CN1C(c1nc(C(C)(F)F)cs1)=O.CC1C(C=O)C1C.N N1(C(C(COC)C)=O)CCN(C(=O)C(c2ccc(C)cc2)(C)C)CC1CC(F)F c1(OC)ccsc1C(=O)NCC(C(=O)N1CCC(CN=[N+]=[N-])C1)N(C)C c1(OC)ccc(C(N2CC3(C2)CN(C(=O)Cc2cnns2)C3)=O)cc1C N1(C(COC(C)=O)=O)CCC(C)(C)C1.c1(CC=O)csc(-c2ccc(C)o2)n1 c1(C(=O)NC(CC)CNC(C2C=CCC2)=O)ccnn1CC1CCC1 N#Cc1cc(C(=O)NC2CN(Cc3c[nH]c4ncc(Cl)cc34)C2)cc(F)c1F C1(C(N2CC(OCC(=O)NC)C2)=O)CCCC1NC(C1CC(=O)N1)=O C(CC(C(=O)NC1CC(OCC)C1)NC(=O)Cc1cnn(C)c1C)=CC C=CCC(C)C(=O)N1C(C(=O)Nc2ccc(OC(C)(C)C)nc2)CC2CC12 N1(C(CCC(c2ccc(C)cc2)=O)=O)CCC2CCCC12CNC(=O)C(C)C CC(CNC(C1CCCC1O)=O)C(=O)NCCOC1(C)CCCC1 c1(C=O)ccc2c(c1)COC(C)(C)O2.C1CC(C)C1.C(C=O)OCCOC.N CC1C(NC(c2cncs2)=O)CCN1C(C12CC(F)(C1)C2)=O C=CCCCCC(=O)N1CC(C(F)(F)F)C(CNC(=O)Cc2ccccc2O)C1 c1(OC)ccc(S(N)(=O)=O)c(OC)c1C(=O)NCCC1CCOC1 C1(C(N2CC(C(=O)OCC)C2)=O)CCN(C(=O)CN2CC=CC2)C1 C#CCC(C)C(=O)N1CC(O)(C(C)NC(C2CN(S(C)(=O)=O)C2)=O)C1 c1(C(=O)NC(CN(C(c2n(CCCC)ncc2)=O)C)C)ccc2nnc(S)n2c1 C(C(C)C(F)C(=O)NC1(C(=O)OC)CC(C)C1)NC(C(CC)CN(C)C)=O C12(C(=O)NCC(CC)(C)Cl)COC(C1)C(NC(=O)C(C)=NOCC#N)C2 N1(C(C2N(CC)CCOC2)=O)CCN(C)CC1C.C1(C(=O)N)COCC(C)(C)O1 c1(OC)ccc(Cl)cc1C(N1CCSC(C(N2CCC(O)(C(F)(F)F)C2)=O)C1)=O C#Cc1c[nH]nc1C(N1CC(CF)(NC(C2CC(CF)C2)=O)C1)=O c1(C(N2CC(CCO)(OC)C2)=O)c(F)cc(C)cc1Cl c1(CC(=O)NCCCN(C(C(C=C)c2ccccc2)=O)CCO)cccc(O)c1 c1(NC(C2CCN(C(CC3(C#N)CC3)C(=O)NC3COC3)C2)=O)cccc(F)c1 N#CC1(C(N2CC=CC(NC(C34CC3C4)=O)C2)=O)CC2CCC1C2 N1(C(C=CC(C)NC(C2CCC(=C)CC2)=O)=O)CCOC(C2(C)N=N2)C1 N1(C(C=C(CC)C)=O)CCn2c(CNC(=O)C(C)CC3CCCC3)nnc2C1 C1(NC(CCC=CC)=O)CC2CN(C(=O)CNC(=O)CCCCC)CC2C1 O=C1CN(Cc2cnc(-c3ccc(C(F)(F)F)cc3)s2)CCN1 N1(C(C(C)O)=O)CCCCC(N(C)C(c2ccc(NC(C)(C)C)cc2)=O)C1 C1(NC(c2ccnc(C(F)F)c2)=O)CCCCC1NC(c1cc[nH]n1)=O C1(NC(CC(C=C)C)=O)CCC12CN(C(c1ocnc1CC)=O)C2 CC1=CCC(C(N2CCCC2C(=O)NCC2=CCCCC2)=O)CC1 C1(NC(C(CC)COC)=O)CCCCCC1C(=O)NC1(C(=O)N(C)C)CC1 C1(C(N2CCC3CC32)=O)C2CC3C(C2=O)C13.C1(COC)CC1C=O.C c1(C=O)ccc(O)nn1.c1(C(=O)NC2CCC2)cc(=O)n(-c2ccccc2)[nH]1.N c1(CC(=O)NCCN(C)C(C23CCC(C2)C3)=O)nc(C2CC2)cs1 C=CC(CC)CC(=O)NCc1cc(C(=O)NC2CC(C(C)(C)C)C2)n[nH]1 c1(CCC(=O)NCCC(C)N(C(=O)Cc2ccsc2Cl)C)ccc(F)cc1 c1(-c2nnc(OC(CSC(c3ccc(Br)cc3)CC)OC)s2)ccc(Br)cc1F c1(NC(CC2CCN(C(C(C)=O)=O)C2)=O)cc(S(=O)(=O)NCCO)ccc1O C(=O)(C1=COCCO1)NCC(C)N(C(c1ccc(CC#N)cc1)=O)CC C12(NC(CNS(C)(=O)=O)=O)CCC1CN(C(C1CS(=O)C1)=O)C2 c1(NC(CCCC(=O)N(C)CC)=O)cc(F)c2c(c1)C(=O)C(C)O2 CC1(O)CCC2(CCN(C(=O)C(=O)NC3CCNCC3(C)C)C2)CC1 C1(C(=O)NCc2n(C)ncc2C2CC2)COCCN(c2ncc(O)cn2)C1 c1(C(N2CC(C)(C)OCC2CNC(=O)CO)=O)ccc(S(N)(=O)=O)c(Cl)c1 CC(C)C(C)CC(=O)NC1CCOC1C1CCN(C(=O)CC2(C#N)CCC2)CC1 C(C(C)(C)CCCO)N(C(CCC=CC)C)CC.CC=C c1(C(=O)NCC(C)(CO)NC(C2CCC(=O)C2)=O)cccc(C2=CCOCC2)c1 c1(C(N2C(C(=O)NCc3ccnc(Br)c3)CC(C)C2)=O)cccc2occc12 C1(CNC(CCCC)=O)CC2CCC1N(C(=O)C(c1ccc(F)cc1)C)C2 C(C(C(=O)N1CC(C)(CCO)C1)C(C)C)NC(C(CCC)N(C)C)=O Cc1ncc(NC(C2(NC(C3CCCCS3)=O)CC2(C)C)=O)cc1Cl c1(NC(c2n(CC=C)nnn2)c2ncc(CC)s2)ccc(N2CCOC2=O)cc1 N1(C(CSCCCC)=O)CC2CCN(C(c3cn(C4CC4)nn3)=O)C(C2)C1 N1(C(CC(CC)O)=O)CCOCC(CNC(C2CC3CC3C2)=O)C1 c1(C(=O)NCc2ncc(C)s2)cnc(-c2ccccc2N(C)C)cn1 C1(NC(C2CCC(N(C)C)C2)=O)CCC(NC(C2(C)CSC2)=O)CC1 C(c1cc(F)c(F)c(F)c1)=CC(N1CCCC(C(N(CC#C)C)=O)C1)=O O(C1CCCc2ccccc21)CCSCC(CC)NC(=O)C(C)(CC)C(F)F Cc1cc(F)ccc1C(=O)N(C1CCCN(C(=O)C(c2ccnn2C)O)CC1)C C1(CNC(C2N(C(C)=O)CSC2)=O)CN(C(=O)C(F)=CCCF)CC1(C)C N1(C(C(C)N)=O)CC2CCC1CC2.n1(CC=O)cnc([N+](=O)[O-])c1.[SH](C)(=O)=O C1(CNC(=O)C2=COCC2)CC2COCC2N1C(=O)C(F)(F)c1cccnc1 Cc1nn(C)c(N)c1C(N1CCC(C(F)C(=O)NC2CC(CO)C2)C1)=O CC(C)(C)C(C(=O)NC)N1CCNC1=O.C1(CC(N2CCC2)=O)CCC1C1CC1 N1(C(C(C)NS(CC)(=O)=O)=O)CCC(C2CCCN(C(=O)CO)C2)C1 C1(C(=O)NC2CCCC(NC(Cn3cnc(=N)[nH]3)=O)C2)CCn2c(O)nnc2C1 c1(C(C)NC(=O)NC(c2ncccc2F)C)nc(O)c2ccccc2n1 c1(NCC(=O)NCC2OCCN(C(=O)OC(C)(C)C)C2)cncc(Cl)c1Cl C1(C(=O)NCC(CNC(=O)CSc2ccccn2)OC)CC(O)CN1C CC1CN(C(c2cc(C(F)(F)F)ncn2)=O)CCN1C(=O)CCSC(F)(F)F C(=O)(CC1=CCOCC1)N(CCCOCCNC(c1cccc(C(C)C)n1)=O)C C1(C(C)NC(c2ccc(-c3cc[nH]n3)s2)=O)CN(C(C2CCC(=O)O2)=O)CCO1 c1(C(N2CCC(c3cn(C(CC)C)nn3)C2)=O)cc2cccc(F)c2[nH]1 c1(C(=O)NCc2c(C)c(Cl)c(Cl)cc2)cc2cc(F)ccc2o1 C(N=C(NCC1CCCCO1)N1CCCC(CC2CCOC2)C1)c1ncn(C)n1 c1(C(=O)NCC2(NC(C3C(C)OCCC3)=O)CCOCC2)ccc(F)c(O)c1 C1(C(=O)NC(C)(CO)CO)CCCN(C(C2CCCC(C#N)C2)=O)CC1 S(=O)(=O)(c1[nH]c(=NCC2CC2C2CCC2)ccc1Br)N1CCN(C(CC)=O)CC1 Cc1ccc(C(=O)NCCCCCCNC(c2ccnn2CCF)=O)cc1CO C1(CCNC(CN(C)C(N)=O)=O)CC(F)(F)CN1C(=O)CCC(C)(F)F C12(NC(c3c(CNC(=O)C(=C4CCCCC4)F)ccs3)=O)CCCCC1C2 c1(OC)cncc(C(=O)N)n1.C12CC(C1)C2.c1(C=O)cnc(C(C)(C)C)[nH]1 C#Cc1cc(C(N2CCC(NC(=O)Cn3cc(Cl)cn3)C2)=O)cc(Br)c1 Cc1cc(C(N2CC(CCNC(=O)CCCc3cccs3)C(C)C2)=O)cn1C N1(C(c2nc(C)sc2)=O)CCC(NC(c2ccn(CC(F)F)n2)=O)C(C)(C)C1 c1(C(=O)NC2CC3CC(NC(CC=C)=O)C2C3)cnc2n1CCCC2C c1(N(C(C(C)NC(C2CN(C(=O)CCCN=[N+]=[N-])C2)=O)=O)C)ccc(F)cc1Cl Cn1c(=O)oc2c(C(=O)NC3(C)CN(C(C4(C)CC=CCC4)=O)C3)cccc12 C1(NC(C(CC2CCCC2)NC(=O)Cc2ccco2)=O)CCC=CCC1 C1(NC(c2cc(OCC)ncc2)=O)CC2CC1N(C(c1c(Cl)n[nH]c1C)=O)C2 c1(C(N2CCC(CNC(CNC(CCC(C)C)=O)=O)C2)=O)cc2ccsc2n1C CC1(C)COCC1CC(=O)NCC1COCC1NC(c1ccccc1)=O CCCC(CC)CC(=O)NCC1CC2(CC2)CN1C(=O)C=CC1CCCO1 N1(C(C(C(CNC)O)C)=O)CCCN(Cc2ccccc2)C(=O)C1 c1(C(N2CCN(CCC#C)CC2)C(=O)NCCSC)ccc(Cl)c(F)c1 C(=O)(CC1=CCCCC1)N1CCCC(NC(c2c(C)cco2)=O)(CO)C1 Cn1cnc2ccc(NC(=O)CC3COCCN3Cc3cc(Br)co3)cc2c1=O [N-]=[N+]=NCC(F)CCNC(=O)CC1(NC(=O)CC2CCC3CC23)CCCCC1 C1(C(N2CCC(OCC#C)CC2)=O)N(C(C2CCC(O)CC2)=O)CCCC1(C)C N1(C(c2cc(C)c(Cl)s2)=O)CCC2CN(C(=O)CCCC3CCCC(=O)N3)CC12 c1(OC)ccc(C(F)(F)C(=O)NCC(C)CNC(C2COCCN2C)=O)nc1 c1(C(N(CC(CN(C(C(C2CC2)OCC)=O)C)O)C)=O)cn2cnnc2cn1 c1(OC(C)C)ccc(C(N2CC(CN=c3[nH]nco3)(O)C2)=O)cn1 C1(NC(CNC(CCC)=O)=O)CCN(C(=O)CCC(=O)C2CC2)C1C(C)C C(=O)(C(F)(F)C(F)F)NC1CC(NC(c2n(C)cc(Br)c2)=O)C1 C1(NC(CCc2c(C(=O)OC)nco2)=O)C(C)CN(C(c2ccc[nH]2)=O)CC1C C(=O)C1CCCn2ccnc21.c1(CNC(C(=O)NCC)=O)cccc(C)c1.N N1(C(C(C)Cc2ccnn2C)=O)CCN(C(=O)COCc2nc[nH]n2)CC1CO C1(C)NC(=O)NC1=O.CCC(C(=O)NCc1csc(C(=O)NC)c1)NCC CC(CC(C)(C)O)NC(C1C=CCN(C(c2cc(=O)cc[nH]2)=O)C1)=O c1(C(=O)OCC)c(NC(=O)CNC(=O)CCC)sc(C)c1.C(C)=O C12CCCCC1C2.CC1(OCC(=O)N)CN(C(c2coc(C(N)=O)c2)=O)C1.C C1(C(N(C2CCCCC2(C)O)C)=O)CC(O)C(O)CC1CNC(=O)CCN=[N+]=[N-] c1(CC(=O)NCC(CC)NC(c2cc(F)c[nH]2)=O)cncc(F)c1 C1(CNC(CC(=C)Br)=O)(NC(=O)CC2C(=O)ON=C2C)CCOCC1 c1(CN(C(=O)CC(Cl)Cl)CCNC(C2(COC)CC2)=O)ccccc1 C1(C)(c2cn(C(C)C(=O)O)nn2)CCN(C(=O)CC2CC3CCC2(C=O)C3)CC1 C1(n2cc(-c3c(C)cn(C)n3)nn2)CON(C(=O)CCC2CC(C)(C)CO2)C1 c1(C(C)C)ncc(-c2cn(C3(C(=O)NC4(CC(C)C)CCOC4)CC3)nn2)o1 Cc1cn2c(n1)C(C(=O)N)CCC2.C1(C)CN(C(C23CC4CC2C3C4)=O)CC1C.C c1(C(N(CC(C)C)C)=O)c[nH]c2ccncc12.c1(COC)cccc(C=O)c1.N c1(C(CC)C)cccc(NC(c2nnnn2CCCSC)C2CC2)c1 CC(C)CC(O)CC(=O)N1CCC(CCNC(=O)C(C)C(C)(C)C)CC1 N1(C(C(CCCC)C)=O)CCCC2(C1)CN(C(=O)C(F)(CC)C(=O)OC)C2 c1(OCCCOC)ccc(NC(=O)CCCCCC2OCCO2)cc1OC c1(C(=O)NC2C(CC)CN(C(c3ccsc3)=O)CC2)c(C)cc(C)nc1C C1(O)(CNC(c2n(C)nc(C3CC3)c2)=O)CCCN(C(C2CCCOC2)=O)CC1 c1(C(N2CCC(NC(C3C(C)(C)C3)=O)CC2)=O)ccc2oc(=N)[nH]c2c1 C1(CN(C(CSCC(C)C)=O)C)CCCN(C(=O)CCc2cccc(Cl)c2)C1 c1(-c2ccc(C)o2)cnc2ncc(C(=O)Nc3cn(C)nn3)n2c1 CC1(C(N)=O)CN(C(=O)CC2CCN(Cc3cccs3)C2)C1 C1(NC(CCc2cc(C)no2)=O)CC(CC(=O)N(C2CCOC2)CCF)C1(C)C CCC(O)CC(=O)NC(Cn1cncn1)C(=O)NCC1(C(C)C)CC1 c1(C(N(C2CC(NC(C3(C)C(C)C3)=O)C2)C)=O)cnn(C)c1Br CS(=O)(=O)C1CCN(C(C2CC2NCc2cccc3ccccc23)=O)CC1 c1(CCNCCn2cc(C(O)CC3CCCN3)nn2)cc2cccnc2[nH]1 C(=O)(CC(C)(C)COC)N(C(CNC(C1(CC)CCOC1)=O)C)C C1(CC(=O)N(CCCOCCNC(=O)CCc2nc[nH]n2)C)CCCNC1=O c1(CN(C)C(C2(O)CCN(C)C2)=O)cccc(O)n1.c1ccc(CC(=O)O)cc1 c1(C(C)NC(CC2(CC=C)CCCC2)=O)ccc(C)cc1.c1(C=O)cn[nH]c1.N C12(C(C)C)CNCC(C(N3CCOCC3CC3CCOCC3)=O)(C1)C2 C1(O)(CNC(C2(NC(CC3(C)OCCO3)=O)CSC2)=O)CCCC1(C)C c1(C(=O)NCCNC(c2ncsc2C2CC2)=O)cnn(C2CCOC2)n1 C1(C(=O)NCC2OCCCN(C(c3c(C)nccc3)=O)C2)Cc2cccnc2C1 c1(C(=O)NC2CCN(C(C(C(=O)OC)C)=O)CC2)cc(F)cnc1C n1(CCC#C)c(N(C2CC(C(C)C)C2)C)nnc1-c1cccc(OCCOC)c1 C1(C(CNC(c2c(CC)noc2)=O)(C)C)CCN(C(C2CC3CCC2O3)=O)CC1 C1(CNC(C(=O)Nc2ccc(COC(C)C)nc2)=O)CCC12CCNCC2 C(=O)(C1CCc2c(Cl)cccc21)N(CCNC(C1Cc2ccccc2O1)=O)CC C(=O)(C(F)CC(CC)CC)N(C(C)C(=O)NCC1CCN(C(C)C)C1)CCC c1(OCC(=O)NC2CC3CN(C(COCCCC)=O)CC32)ccc(Cl)cc1C#N CC(CC(=O)N1CC(NC(=O)C(C)(C)Cc2ccccc2)C1)C(F)(F)F C1(CCC)CN(C(=O)Cn2cccc(C)c2=O)CCN1C(=O)CC(C)(C)O C1(CNC(C=C(C)C(C)(C)C)=O)CC(C)N(C(=O)CCc2cnn[nH]2)C1 C1(NC(COCCC)=O)CCCC(NC(C2CC(n3ccnc3)C2)=O)C1 C1(NC(c2n(C=C)ncc2)=O)CC2CC(NC(=O)C=Cc3ncccc3C)CC12 c1(OC)cc(F)c(Br)cc1NC(C1C(O)CCN1C(c1n[nH]c(C)n1)=O)=O c1(C(N2CC(CNC(c3c(C)nsc3)=O)C(C)C2)=O)nc(C(F)(F)F)ccc1F S(=O)(=O)(C1CC1)N1CCC(COC(c2ccn(C(F)(F)F)c2)=O)C1 c1(C(=O)NC(CNC(CC(C)F)=O)C2CCC2)cccc(C2CC2)n1 Cc1nn(C)c(C(=O)OC(C)(C)C)c1Cl.c12ccc(cn1)N(C)CCNC2 C1(C(=O)NC(CNC(C=C(C)C(F)F)=O)C(C)C)CCC(F)(F)CO1 C1(C(=O)NC(C)CNC(c2cc(Cl)c(Cl)s2)=O)Cc2cc(Cl)ccc2O1 CC(CC(N)=O)C(=O)N1CCCC1CNC(=O)CC1(C)CCOCC1 N1(C(C(c2cccc(C)c2)F)=O)CCC(O)C(N(C(=O)CC2CCOC2)C)C1 c1(-c2occ(C(N3CC(N(C)C(c4ccncn4)=O)C3)=O)n2)ccccc1Cl N1(C(CC(CC)(F)F)=O)CCC2CCN(C(c3cc4sccc4[nH]3)=O)C2C1 c1(C(c2n(Cc3nnn(C)n3)nnn2)NCCC2CCCOC2)cccc(Cl)c1 Cc1c[nH]c(C(N2CCC(C(C)(C)C(=O)NC(C)CN3CCCC3)C2)=O)c1C Cc1nc(-c2ncc[nH]2)sc1C(=O)NC1CN(C(=O)C(C)C)C1.CCN(C)C C1(CC(=O)NCC(C)CN(C(=O)COCC2CC2)C)CCC(=O)N1 N1(C(C(C2CCN(C(C(C)n3cnnn3)=O)C2)(C)C)=O)CCC(C)(O)C(O)C1 N1(C(C(C(C)C)N=[N+]=[N-])=O)CC=C(CC(=O)N2CCC23CCSCC3)CC1 c1(C(=O)NC2CC3(C2)CN(C(=O)C(c2ccccc2)O)C3)ccnc2c1OCO2 C1(NC(C(C)(F)F)=O)COCCN(C(c2ccc(OCC(F)(F)F)cn2)=O)C1 Cc1cc(Cl)c(C(=O)NC2(C)CCCCC2)cc1N.C1(C(=O)N)CCCS1(=O)=O CCCCC(=O)C(=O)NC(C(=O)NCC12CC(F)(C1)C2)C1CCCC1 N1(C(c2ncn(CCNC(=O)CC3CCCSC3)c2)=O)CCOC(CC2CC2)C1 Cc1cc(Cl)cc(C(=O)NCC2CC(F)CN2C(=O)C2=CCCSC2)c1N C(CC(=O)NOCCC(F)F)(C1CC1)NC(C(C)C1(O)CCC1)=O C(c1ccc(C(F)F)o1)=CC(=O)N(CCCC)C.C12(CC=O)CCCC1C2.N c1(C(c2nnnn2C2COC2)NC(c2ncccc2Cl)C)ccc(Cl)cn1 C1(C)(C(NCCC)=O)COC(=O)OC1.c1(C(C=O)N(C)C)ccccc1.CC N1(C(C(CC)F)=O)CCOC2(CCC(NC(C3CC3C#N)=O)CC2)C1 c1(C(N)=O)cnc(Cl)[nH]c1=NCC(O)CNC(C1CCCCS1(=O)=O)=O C(=O)(C1=CC2CCCc3cccc1c32)NC(CS(C)=O)c1ccccc1 c1(C(=O)NC23C(CN(C(C(COC)(F)F)=O)C2)CC3)sc([N+](=O)[O-])cc1Cl CCCCC(COC)(c1nnnn1-c1ccc(Cl)cc1F)NCC(F)CO C12(Cc3nc(C)sc3)CC1CN(C(c1c(C)noc1C(F)(F)F)=O)C2 CN1CC2CC1CN2C(c1ccoc1CNC(=O)CC1CCOCC1)=O N1(C(CCCSc2ccc(OC)cc2)=O)c2nccn2CCC1C(F)(F)F N1(C(C2CC(=C)C2)=O)CCN(C)C(CNC(=O)C(CCC)NCC)C1 C1(C(=O)NC(C)C=O)C2CC3C(C2)C13.C1(C=O)CC1C1CCC1.C1CC1.N c1(OCC)ccc(C(N2CCC(C)(NC(=O)C(F)CC3CC3)C2)=O)cc1 CCCCCCCN(C1CCN(C(=O)CCc2cc(C)no2)C1)CC C1(NC(Cc2cccc(C)c2)=O)CC2CC(C1)N(C(c1ccc(O)c(Cl)n1)=O)C2 C12(C(=O)NCC3N(C(C=CC(CC)C)=O)CC=C3)CCC(CO)(CC1)CC2 c1(C(N(CC(C)C)C)=O)cnc(C(C)(C)C)s1.c1(C(C=O)SC)ccccc1.N Cc1ncc(Cl)cc1CC(=O)N.C1(CC(=O)N(CC)C2CC2)CCCCC12CC2 CC(C)CC(F)(F)C(=O)NCC1CN(C(c2ccc[n+]([O-])c2)=O)CC(C)(C)C1 N1(C(C=CC=O)=O)CC(F)(F)CC1C=O.CCN(C(C)C)C(C)C Cn1cc(C(=O)Nc2ccc(C3CCC3)cc2)c(C(=O)O)n1 C1(C(=O)NCC(CC(C)C)NC(=O)Cc2cnsc2)C(F)(F)C12CCC2 CC1CN(C(C2COCCO2)=O)CC(C)N1Cc1cn(C(C)CO)nn1 C=CCC(C(=O)N1CCC2(CC2C(=O)NCc2ccoc2)C1)C(C)C N1(C(C(CC=C)(C)C)=O)Cc2n[nH]cc2C1C(=O)NCCC1CCC(=O)N1 N1(C(C(=O)Nc2c(OC)cc(F)cc2)=O)CCC(C2(C)CC2)CC1 c1(C=O)cc(Cl)nnc1O.N1(C(C(C2CCC2)OCC)=O)CCC(O)(CC)C1.N C(C(C(=O)N(CC(C)CNC(c1cc(F)cs1)=O)C)NC(C)=O)OC CCCCC(O)C(C)C(=O)NCCCCNC(=O)CC1CCC(C)(O)CC1 c1(-c2scc(NC(N3CC(C)CC(CC)C3)=O)n2)cc2ccccc2o1 C1(CC(=O)NCC2C(CNC(c3[nH]cc(C)c3)=O)C2)CCCCC1(C)C CC(C)(C)C(CO)CN=c1cccc(S(=O)(=O)NC2COc3ccccc3O2)[nH]1 c1(C(C(=O)NCC(CC)NC(=O)CSc2cccc(C)c2)C)ccncc1C N1(C(C2(SC)CCC2)=O)CC(CNC(=O)Cc2nonc2C)C(O)C1 c1(N(C)Cc2cocn2)nc(=NC2CCN(S(C)(=O)=O)C2)[nH]c2c1CSC2 CC1(C)CN(C(=O)CC2(C)CCC2)CC1CNC(=O)CCCn1cncn1 c1(-c2ccc(CNCc3ccc(OC)cc3OC)nc2)cccc([N+](=O)[O-])c1F C(=O)C(C)(C)C(=O)N1CCC(N(C(=O)C)C)C1.C(=O)CN(C)C.CC.O C(=O)(CCC(C(C)C)NC(C1(C)CCCO1)=O)NCc1ccc(C)o1 c1(CN2CCC(C)(C(=O)Nc3cc(C)nc(F)c3)CC2)ccc2c(c1)OCCO2 C1(CC)CN(C(C2C3CCC(F)C23)=O)CC1C(N1CC(F)(C(=O)OC)C1)=O C1(C(N2CC(O)(C(=O)N)C2)=O)(CSC)CC(C)(C)C1.C1CC(Cl)(Cl)C1 N1(C(COCC=C)=O)CC2CC3CC2C1C3NC(=O)C1=CCCCCC1 c1(OC)ncc(C(N2CCCC(CN(C)C(c3ncccc3Br)=O)C2)=O)cc1F c1(OC)ccc(CC(=O)NC2(C)CCC(NC(c3cncn3C)=O)CC2)c(Cl)c1 C1(CC(=O)NC2CC2c2ccsc2)(OC)CN(C(=O)CC2CCCSC2)C1 Cc1c(C(C)C(N2CCCC2c2cc(C3CC3)on2)=O)cccc1Br Cc1onc(C(C)C)c1C(=O)NC1CC1C.C(=O)(CCSC(F)(F)F)N n1(CC=O)c(=O)oc2ccccc12.c1(SC)c(C(=O)NCC(O)C)cnn1C.N C1(C)(CNC(c2c(Cl)cn(C)n2)=O)COCCN(C(=O)C)C1.C(=O)C1CC1 N1(C(C2C(=C)C2)=O)CCOCC1CC(=O)NCCN=S(C)(C)=O C(CCC(=O)N(C1CCCCC1)Cc1cc(C(N)=O)co1)NC(C)=O C1(C=O)CC2(CCCCO2)C1.C(C(C)(C)C)=CC(=O)N(C(C)C)CC.N c1(C(=O)N)cccn2cnnc12.N1(C(C)C)CC(C(=O)NCC2CCC2)CC1=O C1(C(=O)NC2C(OC)C3(C2)CCC3)CC2C=CC1N(C(C1(C)CCC1)=O)C2 C(=O)(C(CNC(c1nc(C)ccc1F)=O)CC(C)C)NC(C=C)C1CC1 C1(C(=O)N)CC2CCC1CC2.c1(C(=O)NC2CCCC2)cc(C(F)(F)F)ccn1 C(=O)(C(C)CC(C)C(C)=O)NC(CC(=C)Cl)C(=O)NCCC1CCCC1 c1(-c2nc(CC(CC)C)nn2CCOc2ccc(Cl)cc2)cc2cnc(Cl)cc2s1 CC1CCCC(CCN2CCC(CNC(c3ccc(OC(F)(F)Cl)cc3)=O)C2)C1 C1(C(N(CCNC(=O)CC2CCCO2)Cc2ccccn2)=O)CC(=O)NC1 c1(NC(C2CC3CC3N2Cc2c(O)cccc2F)=O)ccc2c(Cl)n[nH]c2c1 C1(C(=O)NCC2(OC)CN(C(c3ncsc3C)=O)C2)CCOC(=O)CC1 C(=O)CC(C)(C)C1CCCCC1.C1(NC(C2(COC(C)C)CC2)=O)CCC1 C(CC(=O)N1CC(C)OC(C)(C)C1)(CC(C)C)NC(c1c(C)noc1)=O c1(C(N2CC(N(C(C(N3CCCCC3=O)C)=O)C)C2)=O)ccnc(C(C)(F)F)c1 c1(C=O)cc([N+](=O)[O-])c[nH]1.C(=O)(CC(O)CNC(c1cnnn1C)=O)OC.C c1(CC)cccc(NC(C23CC2CCN3C(C2CC(N=[N+]=[N-])C2)=O)=O)c1O Cc1oc([N+](=O)[O-])cc1C(N1CCOC(CC)C1)=O.C(=O)CN(C)C(N)=O.N N1(C(COCCCC#C)=O)CCC(C(F)(F)F)CC1CNC(=O)C(=O)NC C12(c3n(C)ncc3)CCC(C1)C2C(N1CCC(NC(C2CCOC2)=O)C1)=O CCC(CC(F)(F)F)C(=O)NCc1nnc(C(=O)OCC)s1 c1(NC(C2CC(CCNC(Cc3ccc(C)o3)=O)C2)=O)cncc(F)c1 C1(C(C)(O)CNC(c2csc(C3CC3)n2)=O)CCN(C(=O)C(F)(F)CO)CC1 CN1CCC(C)(C(N2CC=C(CNC(=O)CCc3nncn3C)CC2)=O)C1=O CC(C)(C)C1=NOC(C(=O)NNC(=O)NCC2CCCN(C(C)(C)C)C2)C1 C1(C#N)(C(=O)N)CC12CCC2.CCCCN(C(=O)C(=O)NCC1CC1)C CC(C)CC(CC(=O)N1CCC1)NC(=O)C(C)S(N)(=O)=O.C(=O)(N(C)C)O C1(C(=O)NCC2CCN(C(c3ccc(C(C)=O)o3)=O)C2)CCS(=O)(=O)N1 CCC(C(=O)NCCCOCCNC(c1cc(C(C)(C)C)n[nH]1)=O)C(C)O c1(C(C)(C)C)ncc(C(=O)NC2(C3CCCN3C(=O)Cn3nccn3)CC2)o1 C=CC(C)CC(=O)NCCC1(NC(C23CCCC2(C(N)=O)C3)=O)CCC1 C1CC(=O)NC1(C)C.C1(C(NCC)=O)C2CN(C=O)CC12.C(C)(C)C.C C(=O)(CC(C)CC(=O)N1CCC2C(C(=O)NCC3CC4CCC3O4)C2C1)OC C(=O)(CCC(C)NC(=O)C(C)NC(=O)CC1CC(F)C1)OC CCC(O)C(C)(C)C(=O)NC(C)CN(C(=O)C=C(C)c1ccccc1)C N1(C(CC=CC=C)=O)CCC(C(N2CC(OCCF)C2)=O)C(C)(C)C1 C(=O)(CCCC(C)(C)NC(=O)C(c1cncnc1)C)N1CC(C(=O)NC)OCC1 N1(C(C2C(CCOC)C2)=O)CCC(C)N(C(=O)CNS(=O)(=O)N(C)C)CC1 c1(OC)cc(C(N2CC(NC(c3ccc[nH]3)=O)C3CC23)=O)cc(OC)n1 c1(C(N(CCCCNC(C2CC(C)C2)=O)C)=O)c[nH]nc1C1CCOCC1 N1(C(C2CN(C(C)C)C2)=O)CCOCC(NC(=O)CN(C)C2CC2)C1 n1(CC)ccnc1C(=O)NC1CC(F)(C)C1.C(=O)CC.[SH](C)(=O)=O.N c1(C(=O)N)c(S(N)(=O)=O)cnn1C.CC(O)C(C)C(=O)NC1CCC(C)CC1 C1(C(=O)Nc2cn(CC#C)nc2)CCN(C(c2nccnc2C)=O)C1C(C)C CC(O)(C(=O)N1CC2CCC2(C)C1)C(F)(F)F.c1(CCC(=O)N)ccc(F)cc1 N1(S(CC#N)(=O)=O)CCCC(C(=O)Nc2c(O)cccc2F)CC1 c1(OC(C)C)nc(C(N2CCC2)=O)cc(O)n1.C(=O)C(F)(F)CC1CC1.C c1(C(C(=O)NCC(CC)NC(=O)Cc2nncn2C)O)ccccc1 N1(C(C(C2CCCCC2)OC)C(=O)NC2(C)CC2)CCc2cccc(O)c2C1 CN1CCCCC(CNC(C2C3CC3CN2C(c2c[nH]nc2Cl)=O)=O)C1 N1(C(c2c(C)cns2)=O)CC(CNC(=O)CCc2cncn2C)C(F)(F)C1 C(CN=c1[nH]c2c(c(=NCCCc3ccccc3C)[nH]1)CC(C)CC2)NC(C)=O Cc1cc([N+](=O)[O-])cnc1NCC1CC2CCC(C1)N2C(=O)Cc1[nH]cnc1C C1(C(=O)NCCCOC)CC12CCN(C(=O)Cc1ccccc1Br)C2 N1(c2cc(NCc3cc(C)[nH]n3)nc(C(C)C)n2)CCC(C2CCN(C)CC2)C1 c1(C(N2C(CC=C)(C(=O)N(CC3=CCCOC3)C)CCC2)=O)cccc(=O)n1C Cc1nc2nc(=N)[nH]n2c(C)c1CCC(=O)NCc1csc2cccc(F)c12 c1(CC(N2CCCC(N(C(C3CC(C)(CC)C3)=O)C)C2)=O)ccc(Cl)cc1F C12(C(N(C3CN(C(c4c(C)n(C5CC5)cc4)=O)C3)C)=O)CCOC1CCOC2 C1(NC(C)=O)CCC12CN(C(=O)CC(C)(C)C)C2.c1ccc(Cl)cc1.C(=O)N Cc1nc(N2CCCC2(C)CNC(C2CC3CCC2C3)=O)ccc1C#N c1(CN2CCC(CC(=O)Nc3cc(O)nc(Cl)n3)C2)ccccc1[N+](=O)[O-] N1(C(CC2(NC(C(CCC)OC)=O)CC2)=O)CC2CCC(C1)N2CC C1(NC(c2c(C)nsc2C)=O)CCN(C(c2cc(C(N)=O)cs2)=O)CC1O C(CC(C)C)(C(=O)NCC1CCCC1)NC(=O)OC.C1(C(=O)N)CC1C O=C(CC1OCc2ncccc21)NCCCCCCNC(C12CCN(CC1)C2)=O Cc1ccc(C(N2CC(O)CC2(C)C(=O)NCC23CCN(CC2)CC3)=O)cc1F C1(C(=O)NCC2CCC(=C)CC2)CCCC(NC(=O)C(CO)OC)CC1 c1(C=O)cccc2sncc12.N1(C(C(C)NC(=O)NC)=O)CC2CC2(C)C1.N N1(C(COCCCOC)=O)CCCC(CN(C(=O)Cc2sc(O)nc2O)C)C1 c1(C=O)cncc(CC=C(C)C)c1.C(C)(C(C)C)NC(CSCC)=O.N C1CC2CC1CC2O.N1(C(CC2(NC(C)=O)CC2)=O)CCC2CC12C(=O)N.C C(CCN=C(NCCn1cc([N+](=O)[O-])cn1)NCC(C)(C)C)c1n(C)ncc1 CC1(C)CCN(C(=O)C(O)Cn2cncn2)C(C(=O)NCC2CNC(=O)O2)C1 c1(C(=O)NC2CCN(C(CCSC)=O)CC2CO)cc(S(N)(=O)=O)cnc1C N1(C(C(C)(C)Cc2ccccc2)=O)CC2CCCCC2(CNC(C2COC2)=O)C1 N1(C(COCCOC)=O)CC(NC(=O)C(C)S(C)(=O)=O)C2CCCCC12 C1(OCc2cn(C(C)C)nn2)CCCN(C(=O)Cc2nnc(S)n2C)C1 C=CCC(CNC(=O)CCCC1CCCC1)NC(C1CC(F)C1)=O C(CC(=C)C)(C(=O)N(C)C)NC(c1n(CC#C)cnn1)=O.c1cc(=O)cc[nH]1 N1(C(CC)=O)CC(C(=O)NC(CC)CCO)(SC)C1 C(CCCCCN=[N+]=[N-])NC(C(C)OCC1CCC1C(=O)NCC(F)(F)F)=O N1(CCCNC(=O)CCc2csnn2)CCCC1.C1(C(C(=O)N)O)CC(F)(F)C1 Cc1cc(Oc2ccc3[nH]cc(Br)c3c2)ncc1[N+](=O)[O-] c1(CCC)ccc(CNC(=O)CC2CN(C)C2)cc1.N1(CC=O)CCOCC1 CCC(CC(F)(F)F)C(=O)N1CC(NC(=O)CNC(N2CCCC2)=O)C(C)C1 c1(C(=O)NC(C2CCN(C(C(COC)O)=O)C2)C)cccc(CO)c1 C#CCCCCC(=O)NC1(C)CCN(C(=O)CC2COC(=O)C2)CC1 C(=O)(N=c1cc(Cl)n(C)[nH]1)C1CCN(C(CCc2c(C)c[nH]c2C)=O)CC1O CCC(C)(C(=O)NCCC(O)CNC(c1cc(Br)n(C)c1)=O)C(N)=O C1(CN(C(C2C(C)CCO2)=O)C)CN(C(c2ccccc2Br)=O)CCO1 C=CCC(CC)C(=O)NC1CN(C(c2nn(CC)cc2Br)=O)C1 C1(O)(CN2CCC(OC)CC2)CC2CC1CC21OCCO1 CC1C(NC(C2(NC(=O)CCOCC(C)(C)C)CCC2)=O)C2CCN1CC2 c1(CC(N2CCC(NC(C3CC(OC)C3)=O)C(O)C2)=O)c[nH]c2c(F)cccc12 C(=O)(C(C)(C)CC)NC1CN(C(=O)OC)C1.C1(C(=O)N)CCCC(=O)CC1 Cc1csc(Cl)c1C(=O)N(C)C.C1(O)CN(C(=O)C)C1.c1(C=O)ccncc1 c1(C(=O)NCCOCCNC(C(CC)(C)F)=O)ccc(C#N)cc1C C1(CC)CN(C(=O)CN(C(=O)C(N2CCOCC2)C)C2CCC2)CCS1 c1(C(N2CCN(C(c3[nH]c(=NC)sc3)=O)CC2C(C)C)=O)ccc2n[nH]cc2n1 Cc1c[nH]c(=NCCC2(N(C)C)CN(C(=O)CC(C)C)C2)nc1CO.C(N)(=O)N C1(CC)CN(C(=O)C(C)N(C(=O)CC2CCOC2C)C2CC2)CC(C)O1 c1(C=O)ccc([N+](=O)[O-])cc1F.C1(CC)(OC)CN(C(=O)C=O)C1.C(C)C.N C=C(C)CCCC(=O)N1CCC(N(C(=O)COCc2cccc(F)c2)CCC)C1 c1(C=O)csc(-c2nc[nH]n2)n1.C1(C2(C(NC(C)C)=O)CC2)CCCO1.CC c1(-c2ccc(CN3CCC(C(=O)OC)(N(C)C)CC3)s2)cnc2ccc(Br)cn12 C1(NC(C(CC)O)=O)CN(C(=O)CCN(CC(F)(F)F)C)C2CCCCC12 C1(C(=O)NC23CC(C(N(CC(F)(F)CO)C)=O)(C2)C3)CC2CCCC2C1 c1(C(=O)NCC(C(=O)NC(CCC)CO)O)cc2cccnn2c1 C=CCCC(C(=O)NCC1(CN=[N+]=[N-])CC1)NC(=O)CCc1cncn1C N1(C(c2cc(C)ns2)=O)CC(NC(C2CC(F)(CF)C2)=O)CC(O)C1 C1(N(CC)Cc2ccncc2)C2CN(C(=O)Cn3ccnn3)CC12 C12(Nc3nccc(OCC)n3)CCC(C(=O)N)(CC1)C2.C(CC1CC1)CO N1(C(COc2cc(C)on2)=O)CCCC1C=CC(N1CCCC1CC(N)=O)=O CCC(C)(C(=O)N1CCC(CCCNC(=O)C2=C(C)OCC2)CC1)C(F)F N1(C(c2c(O)ccc(C)c2)=O)CC2CCC(NC(C3(O)CCCCC3)=O)CC2C1 N1(C(C(C)OCCC(C)C)=O)CCCCC(NC(c2c(C3CC3)cnn2C)=O)C1 c1(C(N(C(c2cscc2C)C(=O)NCCOC)C)C2CC2)ccc(F)cc1 Cc1noc2ncnc(N3CC4(CC4)CC3CNC(C3(O)CCC3)=O)c12 c1(CC)cc(C(=O)N(C)CCN(C(c2cncn2C)=O)C(C)C)on1 Cc1ccc2c(c1Br)CN(c1nc(=N)[nH]c(=NC(C)c3[nH]c(C)nc3C)[nH]1)CC2 CCCCC(C)C(=O)NC1CCCCN(C(=O)Cc2ccnc(F)c2F)C1 c1(C(N2C(CCCNC(C(CSC)(C)C)=O)CCC2)=O)coc2c1COC2 N1(C(Cc2ccc(OCC)cc2)=O)CCC(NC(C2CCCO2)=O)C(F)(F)CC1 C1(CN(C(c2c(C)snc2)=O)C)C2CN(C(=O)C(C)C(C)C)CC12 C1(C(=O)NCC(CNC(=O)C2=CCCC2)CO)CC2(CCO1)CC2 N1(C(CC2(OC)CN(C(=O)CNc3ncccn3)C2)=O)CCCC2(CCOC2)C1 C1(OC)CN(C(=O)C(C)=C2CCC2)CC1NC(C1CCCO1)=O CN1CC(O)CC1C(N1CCCC1CC(N1CC(CO)CC1CO)=O)=O C1(C=O)CCN(S(N)(=O)=O)CC1.C1(CN(CC)CC)CCS(=O)(=O)N1 C(c1ccccc1)=CCC(=O)NC(C1CCCN1C(c1nccnc1O)=O)(C)C Cc1cc(C)cc(C=CC(=O)NCC2CCN(C(C3CC3F)=O)C23CCC3)c1 c1(C(=O)NC(CNC(=O)Cc2cccc(O)c2)CO)ccc(=O)n(C2CC2)c1 C1(CNC(C2C(C)(C)CCCC2)=O)CN(C(c2ccoc2)=O)CC12CCC2 c1(C(N2CCCC(N(C(C(CC(=C)C)C)=O)C)C2)=O)ccc(NC)c([N+](=O)[O-])c1 N1(C(c2cc(OC)ncc2)=O)CCOC2CCN(C(C3CCCOCC3)=O)CC12 C1(C(=O)NC(CC(C)C)CNC(=O)CCc2cc[nH]n2)Cc2cccc(F)c2O1 N1(C(c2c(CC)ccs2)=O)CC(C2(NC(=O)C(c3cccnc3)C)CC2)C1 C1(CNC(CN(C(C)=O)C)=O)CC(C)(C)CN1C(c1cncc(Cl)c1)=O N1(C(COCC(C)C)=O)CCOC2CN(C(c3cc(F)c(F)c(F)c3)=O)CC12 C1(C(=O)NC(CCC)C2CCC2)C2CCN(C(C3(F)CC=CCC3)=O)CC12 c1(C(N(C2CCN(C(c3c(C)ccc(OC)n3)=O)C2)C)=O)ccc(F)c(Cl)c1N Cc1oc(C(C)(C)C)cc1C(=O)N.n1(CC(N2CCC2)=O)ncc(Cl)c1C.C N#Cc1cccc(CNC(=NCC2CC2)NC2CC(c3ccccn3)C2)c1 N1(C(Cn2nnc(C)n2)=O)CCC(CO)C(NC(=O)Cc2ccco2)C1 c1(C(n2cc(CNC(=O)C(C)C#N)nn2)CC)ccccc1C(F)(F)F C1(C(N(CC(=O)N(CC(=O)N(C)CC)CC)C)=O)CCC(=O)N1 C1(C(C)C)CCCN(C(C2(NC(=O)C=Cc3cncs3)CCOCC2)=O)CC1 C1(C(=O)NC2C(CNC(CCc3n(C)cnn3)=O)CCC2)CC12CCOC2 C1(NC(C=C(C)C(F)F)=O)CCC12CCN(C(C1CCCN1N=O)=O)CC2 c1(NC(C2N(C(c3cc(C)nn3C)=O)CC(C)C2)=O)ncc(Cl)nc1C#N Cc1nc(C(C)NC(=O)C(C)C)sc1NC(C1CCCO1)=O S(=O)(=O)(CC(=O)N(CCCC)C)N(CC)CC.C(=O)(CCCc1nccs1)N CC1=C(C(=O)NC2(c3ccccc3)CCN(C(=O)CCCC3CCC3)C2)CCC1 N1(C(c2ccc(C(C)(F)F)cn2)=O)CCCC(O)(CCNC(=O)CCCC#N)C1 N1(C(C(CC=C)C)=O)CCN(C(=O)CCNS(=O)(=O)c2cccs2)CCC1C C1(C(=O)N)CCSC(C)C1.c1(C(=O)NCC(C)Cn2cccn2)coc(C)c1 Cc1nc(CC2CC2)oc1C(=O)NC12CC(C1)N(C(c1ccc[nH]1)=O)C2 c1(OC)ncccc1C(=O)N(C(C)CNC(=O)CC1CC(F)C1)C Cc1cc(C)c(C(=O)NCC2(C)CN(C(=O)CC3CCCCO3)CC2C)c(C)n1 c1(CC)nonc1C(=O)NC(CO)C(=O)N(C(C)C(C)(C)O)C c1(NCC(C(C)C)(C)NC(C2C3CCC2CC3)=O)ncc(Cl)c(O)n1 C1(CC(=O)OC(C)(C)C)CC(NCc2cnc(C(C)C)nc2)C12CCC2 C(CN=c1[nH]c(Cl)ncc1Br)(C1CCCCC1)NC(C=C(CC)CC)=O C1(CC=O)CN2CCN1CC2.C1(NC(c2cc(OCC)n[nH]2)=O)CCCCC1.N C1(NC(Cc2cc(C)n(C)n2)=O)CCN(C(=O)CN2CC3CC3C2)C1(C)C CC(C)CCCCC(=O)N1CC2CC(NC(=O)C=CC(N)=O)CC1C2 C1(CCOC)CN(C(=O)CC)CCN1C(c1cc(C2CC2)[nH]n1)=O.C(C)=O.N N1(Cc2cnc(C)s2)CCN(C(N2CCCCCC2)=O)CC1 c1(N2CCN(CCCc3cccc(OC)c3)CC2)ccc(C)c(F)c1 c1(OC)ccc(C)c(OC)c1C(=O)NC1CCCC1.c1(CC=O)[nH]cnc1C.N C12(NC(c3c(OC)n[nH]c3)=O)COC(C1)CC2.c1(C=O)ccccc1C1CC1 CN1N=C(CC(=O)NCCCCNC(C2(C)CC2Br)=O)CC1=O CC1(C)C(C(=O)NCC2(O)CCN(C(=O)C(O)c3cnc[nH]3)C2)C1(C)C c1(NC(=O)NC2CC3(C2)CC3(F)F)nc2ccc(C(F)(F)F)cc2s1 c1(C(=O)NC(C(=O)NC(c2ccco2)CO)C2(O)CCC2)cc(=O)cc[nH]1 c1(C(C)CC2CCC2)nc(CC2CCCCC2)nn1-c1ccc(C(C)(C)C)cc1 CC1(C)CCC(C(=O)NC2CC(CCNC(=O)Cc3cccc(F)c3)C2)OC1 C(=O)(C(C)CC(N)=O)NC1CN(C(c2cccc(OC(C)C)c2)=O)CC1O C1(NC(c2nccc(C)n2)=O)CCN(C(=O)C(C)(C)C(C)O)CC(C)(C)C1 Cc1nn(C)c(C(N2CC3CC3(NC(=O)C(C)CC(F)F)C2)=O)c1[N+](=O)[O-] C1(C)(C(N2CC(CN(C(CC(=O)OCC)=O)C)C3(C2)CC3)=O)CCCCCCC1 N1(C(CC2CCCC(=O)C2)=O)Cc2n[nH]cc2C1C(=O)NCC1OCCCO1 O=C(CC1=CCN(C(c2cccnc2S)=O)CC1)NC(CCO)C1CCC1 c1(NCc2scc(Br)n2)[nH]c(=NCCSCC2CCOC2)nc2scnc12 n1(CC)cc(C(N2CC(NC(=O)CCC(=O)O)C(C)C2)=O)c(C(F)(F)F)n1 c1(C(=O)OC)cc(NC(c2cc(Cl)nc3ncccc23)=O)c(C)c([N+](=O)[O-])c1 C1(CN(C(c2c(CCC)nco2)=O)C)CCN(C(c2cnoc2C2CC2)=O)CC1 C1(C(=O)NCC2COCC(C)O2)COC2(C1)CN(C(=O)C(C(C)O)N(C)C)C2 N1(S(=O)(=O)c2ccn(CC(F)(F)F)n2)CC2C3COCC3C2C1 N1(C(C(CC=CCC)C)=O)CCC(C2CN(C(=O)C=C3CCC3)C2)CC1 C=CC(C)CC(=O)N1CCC(C(C)C(=O)NC(c2noc(C)n2)(C)C)C1 C(=O)(CCC=O)NCCCOCC.C(C)C(C)C.C1(CC=O)CCCCO1.N C1(C(=O)NCC(C)(C)NC(CC=CC)=O)CCC(OC(F)(F)F)C1 C(CO)(C(=O)NC1CC(C=O)C1)OC(C)(C)C.C(=O)C(F)=CC1CC1.N c1(NC(CCC(C)NC(c2ncccc2F)=O)=O)cccc([N+](=O)[O-])c1 c1(OC)ccc(Br)cc1S(=O)(=O)N1CC(C(=O)N)C1.c1(C2CC2)cccc(Cl)c1 Cn1cnc(=NC(=O)C2(C)CCN2C(=O)Cc2cc(Br)cs2)[nH]1 CC(CCC(C)(C)C)C(=O)NC1CN(C(c2cscn2)=O)CC2CCCC12 CC(C)C(C)(C)C(=O)NCCC1CCC(NC(c2ccc(Cl)s2)=O)C1 CCCC(CNC(c1cc(CO)on1)=O)C(=O)NC(C)(CO)CCC C(=O)(C#CC1CC(F)(F)C1)N1CCCN(C(C2N(C(C)=O)CCCC2)=O)CC1C c1(C(=O)NC(CC)(C)CNC(C2(F)CC2)=O)cc2ccccc2[nH]1 c1(C(=O)NCC2N(C(C3C(CC)C3)=O)CCC2)ccc2nc(C)oc2c1 c1(C(C)(C)C)ccc(CNC(=O)NCCc2ccccc2)cn1.C(N)(=O)N C12(CNC(C(C=C)OC)=O)CCC(CN(C(=O)C(c3ccn(C)n3)C)C1)C2 C1(C(N2CC(O)(CNC(=O)CNC(=O)C3CC3)C2)=O)CC12CCCCC2 c1(C(CO)NC(=O)NCCC2C(C)C2)cc(Br)ccc1F c1(C(C(=O)NCC(CNC(Cc2c(C)non2)=O)O)(C)C)cccc(Br)c1 C1(C(N(CC(=O)NCCCC)C2CC2)=O)CC1(C)C(C)C c1(C(=O)NC(CC)CNC(c2nc(C(C)C)oc2C)=O)cc2c(ncn2C)s1 N1(C(c2c(O)nnc(C)c2C)=O)C2CCCC1CC(NC(=O)Cc1cscn1)C2 CC(CN=c1[nH]c(N(C)Cc2ccc(F)cc2)nc2c1COC2)N1CCCC1 N1(Cc2c(OC(CC)C)cccc2)CCC(O)C(C(N2CCCCC2CO)=O)C1 c1(CC)nc(C)c(C(N2CCC(C)(C)C2)=O)o1.C(=O)(CCC1CC1(Cl)Cl)N C1(O)(CN(C(CCCOC)=O)C)CCN(C(=O)C)C1.n1(CC=O)cncn1.N C(=O)(C(C)S(N)(=O)=O)NC(C1CCN(C(=O)C(C)O)CC1)C.c1ccncc1 Cc1nn(C)cc1CC(=O)NCC(C)CN(C)C(c1ncsc1C1CC1)=O Cc1nc2cc(NCC3(Br)CC3)ccc2n1C(CO)CO C1(NC(=O)CC2CSC2)CCCC2CN(C(c3cnc4cccnn34)=O)CC12 CCC(C)(COC)C=O.C(C)(c1cnn(C)c1)=CC(N1CCCC(CC)C1)=O.N N1(C(CCC(C)OC)=O)CCC(C(=O)NCCc2ncccc2C)C12CC2 c1(N(CC(=C)C)C)cc(S(=O)(=O)NCc2nn(C)nc2Br)ccc1C#N Cc1ccc(C(C)C)c(OCC(=O)NCC=CC)c1.C(=O)C(C)C(C)O.N N1(C(c2c(C)cno2)=O)CCN2CCOCC2(CNC(=O)C2=NNC(=O)CC2)C1 Cc1cc(S(=O)(=O)NC(=O)C(c2cc3ccccc3o2)C)ccc1[N+](=O)[O-] C(=O)(C(C)(C)C(=O)NC)OCC.c1(C(N2CCCC2)=O)cccc(F)c1C c1(C(N2CC3C(NC(c4csc(Cl)c4Cl)=O)C3C2)=O)ncnc2c1CCC2 c1(NC(C2NCCN(C(C(N)=O)=O)C2)=O)c(F)cccc1Cl N1(C(C(C)C(C)(C)C)=O)CC2CCC(NC(C3CC4CCC(C3)S4)=O)CC2C1 c1(C(N2CCN(C(c3cc(O)cc(=O)o3)=O)C3(CC3)C2)=O)cnc2[nH]ccc2n1 C(=O)(C(CCc1ccccc1)CC(C)C)NC(CNC(CCSC)=O)(C)C N1(C(C2(C#C)CC2)=O)CC2C(CN(C(=O)CSc3ccccc3)C)C2C1.O N1(C(C2CCC(OC)CC2)=O)CC2CCCC2(C(N2CCC(C(C)(C)C)C2)=O)C1 N1(C(Cc2n(C)cnc2)=O)CCC(C2CCCN(C(=O)C(C)(Cl)Cl)C2)C1 c1(C(N2CCCC(NC(=O)COCC3CCCC3)C2)=O)ccnc(O)c1F C=CCC(CNC(c1cc(C)no1)=O)NC(c1cnn(CC(C)C)c1)=O CCC(C)(C)CC(=O)NC1CCN(C(c2cc(SC)oc2C)=O)C2CC12 N1(C(C2C(CC)C2)=O)CCC(C)(CNC(=O)CC2(O)CCCCC2)CC1 c1(NC2CC(CNC(C=CC)=O)OCC2)ncnc2c(-c3ccccc3)nsc12 c1(COC)cccnc1NC(c1ccncc1Cl)c1nnnn1C(C)(C)C C1(NC(c2ccc(CN(C)C)cc2)=O)CCN(C(c2ccon2)=O)CCC1(F)F C1(NC(c2ccc(C3CCCCC3)s2)=O)CCC2CC1CN2C(=O)CCF CCC(C(=O)NCC1(F)CC(NC(=O)C=Cc2cncs2)C1)n1ccnc1 c1(C(C2(n3ccnn3)CC2)Cc2n(CCCC)nnn2)cccc(Cl)c1 N1(C(c2ccc(Br)s2)=O)CC2CN(Cc3cc(OC(F)(F)F)ccc3F)C2C1 c1(-c2ccc(-c3n(C(CC)CO)ccn3)s2)cc(OC)c(C(=O)OC)cc1Br c1(C(N(C(CCNC(C(CC)NC(N)=O)=O)C)C)=O)cnc2[nH]c(=N)sc2c1 CC(C)CC(CN)CC(=O)N1CC2CCC1CN2C c1(C(=O)NCCOCCC(=O)NCc2ccccc2)ccncc1Cl.C1CC1 c1(CC=O)csc(-c2ccc(C)o2)n1.C(C=O)N(C(=O)O)C.C1CC1.CC c1(C(N2CC=CC(NC(CCNC(=O)NC)=O)C2)=O)cccc2nccnc12 C1(C=O)CCCCN1C(=O)CCC.C=CCCCNC(C1CC(F)(CO)C1)=O.N C1(CNC(CC2CC(C)(C)OC2)=O)CC12CCN(C(=O)C(C)(C)C1CC1)CC2 C=CC1(C(=O)NCC(N)=O)CCN(C(c2ccoc2Cl)=O)CC1 c1(C=O)c(S(C)(=O)=O)cnn1C.Cc1conc1C(=O)NCC1CC1C C1(CC(N2CC(OC(CC)=O)C2)=O)C(NC(=O)CC2CCCSC2)CC1O CC1(C)C(NC(=O)C)CC1C(=O)NCc1ncc[nH]c1=O.C1CC=CC1.O N1(C(c2ccc(C)nc2)=O)CC(CNC(=O)CC2CCCCC2O)CCC1C N1(C(c2c(NC)scn2)=O)CCOC(C)(CNC(=O)CC)C1.[SH](C)(=O)=O N1(C(C(C(C)C)SC)=O)CCC2(CCCN2C(c2cnn(C3CCC3)c2)=O)C1 c1(CN2CCC(NC(C)=O)C2)ccc(-c2ncc(F)cn2)cc1F C(=O)(C(C#N)CCC)NC(CC=C)C(=O)N(C)Cc1ccccc1F c1(C(=O)N)cc(C)nc2onc(C)c12.c1(SC)ccc(C(=O)NC(C)CCC)s1 C(=O)(CC1CCCc2oc(C)nc21)NC1CCCN(C(C(C)=C(CC)C)=O)CC1 CC1C(NC(=O)COCC2CC2)CCCN1C(=O)CCCc1ccncc1 C(CCC(C)C(=O)NCc1ncoc1C1CN(C(=O)CSC2CC2)C1)OC C1(NC(C(COCC)NC(=O)C(SC)SC)=O)CCOC1(C)C C1(CC(C)NC(=O)CC2CC2C)CCN(C(C2(O)CC2)=O)CC1 c1(CC(=O)Nc2nc(CC(=O)NCC3CCCS3)cs2)ccc(O)cc1 c1(OC)ccc(C(CNC(c2sccc2C2CC2)=O)NC(=O)CS)cc1 CN1CCC(NC(=O)C(C2(O)CCC2)NC(=O)CC(C)(C)C2CC2)C1(C)C C(C)(CCC(=O)NCCC1CC1)OC.n1(CC=O)nnnc1-c1ccsc1.C C1(C(=O)NCCNC(=O)Cc2cc[nH]c2)CCCC2(CCOCC2)O1 c1(C(=O)NCC(CNC(c2cc(CO)ccc2Cl)=O)CO)cc2cccnn2c1 C1(Br)(C(=O)NCCC(C)N(C(=O)CCc2ccon2)C)CC12CCC2 N(C(=NCCCC(F)(F)F)N1CCC2(C)C(C1)C2(Cl)Cl)CCCOC N1(C(C=C(C)c2cnn(C)c2)=O)CCC2CN(C(c3ccc(F)cn3)=O)CC2C1 C1(N2CCN(C(CC(CC)SC)=O)CC2)CN(C(=O)CCC(C)(C)OC)CCCO1 C(=O)(C(CCF)NC(=O)CC(C)F)Nc1cn(CCC)nc1 N1(C(C(CC)O)=O)CCCC(CNC(c2cccc(Br)c2)=O)C1 CCC1=C(C(=O)N2CCN(C(=O)C(C)(F)C(C)(C)F)CC2C)CCCO1 C1(C(=O)NCC(C)N(C(c2nc(C)sc2)=O)C)CCCN1N=O C(C(O)CN=C1NCC2(CCN(C(c3ccccc3)=O)C2)N1)N(C)C C1(CC(C)C)CC(c2nc(-c3cc[nH]n3)nn2-c2cnn(C)c2)CC(=O)N1 Cc1ccc(C(C)C(=O)NC(C2CCN(C(=O)C(c3ccc(Cl)s3)C)C2)C)cc1 C1(c2nnnn2C(C)(C)C)(Nc2c(C(=O)OC)csc2)CCN(C(C)=O)C1 N1(CC)CC(NC(=O)CC2CC(NC(c3c[nH]nc3CC)=O)C2)C(C)C1 O=C(CCCC(F)F)NC(c1ccccc1)CNC(c1cc(O)ncn1)=O N1(CC(=O)NCC=CCC(=O)NCC#CC2CC2)CCOCC1=O C(c1ccncc1C)=CC(=O)NC.N1(C(C2(COCC)CC2)=O)CCCC1 C(=O)(C(C)(C)CC(=O)N1CCC(C)(C)C1C(=O)N)OC.N1(C(C)=O)CCCC1 O(NC(=O)C1c2c[nH]nc2CN1C(c1nocc1Cl)=O)C(CC)C c1(C(=O)NCCCCNC(c2cc(C(=O)OC)no2)=O)cc(OC)c(Cl)s1 c1(C(N2CC(C(=O)Nc3ccnc(Cl)c3Br)C2)=O)c(Cl)cc(Br)cc1Cl C(=O)(C1CCCc2ncc(C)n21)N1CCC(N(C(c2c(C)c(Cl)ccn2)=O)C)C1 N1(C(c2c(CCC)[nH]cc2)=O)CC(F)(F)CC1C.C1(C=O)CC1C(C)C.N C1(C)(CC)CCN(C(C2CCN2C(=O)Cc2cnc(C)s2)=O)CC1 c1(C(c2n(CC)nnn2)NCC(=O)OC(C)C)sc(C)c(Br)c1C C=CC(C)CC(=O)N1CCC(N(C(=O)CCF)CCC)C1 C1(C(=O)NCCCCN(C)C)(NC(=O)C(C2CCOCC2)=O)CCC(C)(C)C1 Cc1c(CNC2CCCCC2C(=O)N(C)C)nc2ccccn12 N1(C(=O)COC2CCC2)CC(CN=c2[nH]nc(O)s2)C2(COC2)C1 C#CC(CCC)NC(c1ccoc1CNC(c1cc(C(C)C)on1)=O)=O c1(C(N2CC(CCNC(C(C)NC(C)=O)=O)C2)=O)sc2cccnc2c1Cl C1(C(N(CCCCCCNC(C2CN(C)C(=O)C2)=O)C)=O)CCN(C)S1(=O)=O C1(C)(C(=O)OC)CCN(C(=O)NCCN2CC=CC2)C1 CC1c2ccc(Cl)c(Cl)c2CCN1N1CCCC1Cc1cccc(Cl)c1 Cc1cnc(C(N2CCCC(CCNC(C3CN(C)C(=O)N3)=O)C2)=O)nc1 n1(CC)c(C)nn(CC(=O)NCCC(C)NC(C2OCCC2C(C)C)=O)c1=O C1(C(=O)NC(C)CN(C)C(c2cn(CCN(C)C)nn2)=O)CCC(F)(F)C1 C1(COC)CN(C(=O)Cc2cccc(F)c2)CCN1C(=O)C(C)Cn1cccn1 O=C(CCCc1ncco1)N1CC(F)(CNC(C2(CF)CC2(F)F)=O)C1 C1(C(=O)NC(CC)(CNC(=O)CC2CC=CCC2)CC)OCCOC12CCC2 C12(C(N3CC(NC(c4c(C(C)C)con4)=O)C3)=O)CCCCN1CCC2 c1(CC)cccc(C(=O)NC2C3CC(NC(c4cccnc4)=O)CC23)c1O C1(CNC(N2CC(CN(C)C)C(CO)C2)=O)C2Cc3ccccc3C12 C(=O)(C1=CCCOC1)NCCC(=O)NC(C)(CO)C1CCCC1 Cc1cc(C(=O)NC(C)(C)C2CCC2)cc(C(F)F)c1.C(=O)(C#CC(C)C)N Cc1ccc(C(F)C(=O)NCCc2cnc(NC(=O)CC3CCCCO3)s2)cc1 c1(CC)ncccc1C(=O)NC(C)(C)CC(=O)NCCC1CCN(C)C1 c1(NC(C2N(C(C(CO)OC)=O)CCC2C)=O)cccc(F)c1C C(=O)(C(CC)CC(F)(F)F)N(CC)C.c1(CC)nc(C)ncc1C(=O)NCC C(CC(C)C)(C(=O)NCc1[nH]ccc(=O)c1O)NC(C1CCC(OC)CC1)=O c1(C(N(CC)CC)=O)cccc([N+](=O)[O-])c1.C12(C=O)CC=CC(C1)OC2.N c1(C(CC)C)ccc(C(=O)NC2CC23CC(NC(=O)CC)C3)c(O)n1.C1CC1 C1(C(=O)NC(c2cn(-c3ccc(F)c(F)c3)nn2)C)Cc2ccccc2S1(=O)=O Cc1ccc([N+](=O)[O-])cc1C(N1CC(C)(CC(N2CCN(C)CC2CO)=O)C1)=O C1(C(=O)N)CC2(CCOCC2)CO1.N1(C(C2(CC=C)CC2)=O)CCC(C2CC2)C1 c1(C(C(=O)NCC(C)(C)OC)NC(c2cscn2)=O)ccccc1 Cc1cc(C(=O)NC2CCC(C)C2)ccc1C(F)(F)F.c1(C=O)cnn(C)n1 c1(OCC(CO)CC2CCC2)cccc(Cl)c1 c1ccc(Cl)cc1.C1(C=O)C2CCC(=O)C12.C1(CSCC=O)CC(F)C1.C C=C1CCN(C(C2C=CC=CC=C2)=O)C(C(=O)NCCCC(C)CO)C1 C(=O)(C1=CCS(=O)(=O)C1)N1CCCC(CC=C)(NC(=O)CCCC(C)=O)C1 C(c1ccncc1)=CC(=O)N(CC(O)C)C.c1(C=O)csc(C(F)(F)F)c1.N c1(C(N2C3C(C(=O)NCC(=C)C)C(C3)C2)=O)c(NC)cccc1[N+](=O)[O-] CC1(CNC(c2c(Br)cnn2C2CCC2)=O)CCN(C(c2cnc[nH]2)=O)C1 c1(CNC2C(C(N3CCC(N(C)C)C3)=O)CCC2)c[nH]c2nccc(Cl)c12 Cc1cc(C)c(C(N2CC3CN(C(=O)C=Cc4cccs4)CC3C2)=O)cc1Br C1(NC(c2scc(OC)c2)=O)COC2(C1)CN(C(C1CS(=O)C1)=O)C2 N1(CC(N2CC(COC)N(C(=O)Cc3cscn3)CC2)=O)CCCCC(O)C1=O C12CCC(C1)OC2.C(=O)CCN(CC(N)=O)C.C(C=O)N(C)C(=O)CCC c1(C(N2C(C)CCC2CO)=O)n[nH]c2c1CN(Cc1c(O)cc(F)cc1F)CC2 N1(C(CN(C)CC)=O)CCC(O)(CC)C1.c1(C=O)ccccc1SC(F)(F)F.N c1(C(=O)NCCC2CSCCN2C(c2cccnn2)=O)c[nH]c2cccc(F)c12 c1(C(=O)NC(C)CCN(C)C(C2(CF)CCOCC2)=O)cc2sccc2n1C C12CCN(CC1)C(=O)NC2.C1(C(N(C(C)CN(C)C)CC)=O)CSC1 c1(CC)ccoc1C=O.c1(CC(=O)N(CC(C)C)C)ccn(C2CCCC2)n1.N C1(CNC(c2c(C)noc2)=O)CN(C(c2cnn[nH]2)=O)CCO1 CC1CN(C(=O)C(N2CCCC(C(=O)NC3CC3)C2)=O)Cc2c[nH]nc21 N1(C(C(C)(C)SC)=O)CCCC(C2CCCN(C(c3cc(F)c[nH]3)=O)C2)C1 C1(C(=O)NCCC2CCCN2C(=O)CSc2ccccc2)CC(=O)N(O)C1 c1(C(CCC#N)NC(c2ccc(CCC)cc2)C)cccc(S(C)(=O)=O)c1 c1(C=O)cccc(N)c1.C(C)(C)(C(=O)NCC1CCCC1)SC.C1CC1.C C(=O)(C1CSc2ccccc21)N1CCC(CC=C)(NC(c2ccoc2Cl)=O)C1 C=CCC(C(=O)N(C1CCC(NC(C23CC(C2)C(C)O3)=O)CC1)C)C(C)C C1(NC(=O)CCc2cc(Cl)no2)CC12CCN(C(C1CC1[N+](=O)[O-])=O)CC2 c1(C(N2C(CNC(C3CC(C)C3)=O)CC2)=O)cccc(Oc2nccs2)c1 N1(C(c2sc(C)c(O)n2)=O)CCCC2CN(C(c3ncc[nH]c3=O)=O)CCC12 CCC(C)(O)CNC(=O)CC1(NC(C2CN(C(C)C)C2)=O)CC1 CCC(C)(C(=O)N1CC(C(F)Cn2cc(C(O)CO)nn2)C1)OC N1(C(CC#N)=O)CCC(CNC(c2c[nH]c3cc(Br)ccc23)=O)C(F)(F)CC1 C(c1cccc(Cl)c1)=CC=O.Cc1cc(CCC(=O)NC2C=CC(C)C2)no1.N Cc1scc(CNC(C2CN(C(C3CC(=O)CS3)=O)CCO2)=O)c1C c1(C(=O)NC(C(C)NC(C2CCNC2=O)=O)(C)C)ccc(C#N)c(O)c1 C1(C(C)NC(C2CCCN2C(=O)CO)=O)CN(C(=O)C(C)(C)C)CCO1 N1(C(CC2CCN(C)C2)=O)CC2(CCCN(C(c3nn(C)nc3Br)=O)C2)C1 c1(C(=O)NCCC(=C)C)c[nH]c2c(CC)cccc12.C(=O)(C(O)CC1CC1)N c1(C(=O)OC)cnc(N2CCCC2CNC(C2CCSC(C)C2)=O)nc1 c1(C(N2CCCN(C(C=CC=CCC)=O)CCC2)=O)ccc2nccc(C)c2c1 CCCC(CC)CCC(=O)NC(CN(C)C)C(N1CCC2(CCC2)CC1)=O C(=O)(C(CC)CC=CCC)N1CCCC(C2N(C(CCC=C)=O)CCC2)C1.C(CC)=C Cc1cc(C(=O)NCC2CN(C(=O)CC3(CO)CC3)CCCO2)c(C)cc1Cl C1(C(=O)NCC(C)CNC(c2csc(N)n2)=O)CCC(=O)NC1 CCCCC(C(=O)N1CC(C(N2CC(F)(CC)C2)=O)C(F)C1)N(C)C C1(NC(CN(CCCCCC)C)=O)CN(C(c2c[nH]cc2C2CC2)=O)CCC1O C1(NC(CCC2CCC(C)O2)=O)CN(C(c2cc(C(F)F)cs2)=O)CC1CO CCCC(CNC(C1CC2(CCCO2)C1)=O)C(=O)NCC1(CO)CC(C)C1 CC1CC(NC(c2csc(C(F)(F)F)n2)=O)CN(C(C2CCCC2C2CC2)=O)C1 c1(C(N(CC(=O)NCCc2onc(CC)n2)CCO)=O)cnccc1C#N C=CCC(CNC(=O)C(C)OCCCC)C(=O)NCCN(CC(F)F)C C1(NC(=O)CC23CCCC2C3)C=CCN(C(=O)Cc2ccsc2)C1 C1CC2(CC2)CN1C(=O)CN1CCCCC1=O.c1(C(=O)NC)ccnc(Cl)c1Cl c1(C(N2CC(OC)C(NC(=O)COC(F)F)C2)=O)ccn(C)c(=O)c1 C(=O)(C#CC1CCC1)NCc1cc(C(=O)NCC(C(=O)NC)O)no1 CC1(C)NC(=O)OC1CNC(C1CCN1C(C1CC(=O)CS1)=O)=O C1(C=O)CNC(=O)CN1C(=O)Cc1n[nH]c(C)n1.C1(CC=C)(C)CCCC1.N c1(N(CCCCC(=O)Nc2nnc(CCCCC)s2)C)cccc(C#N)c1.C(C)=O N1(C(C(C(=O)OC)C)=O)CCN(C(=O)COCCCF)C(COC)C1 n1(CC)ncc2c(N3CCN(C(=O)C(C(C)C)SC)CC3C)ncnc12 N1(C(C(CC#C)NC(=O)CCCCCOC)=O)CC2(CCC2)OCC1C CC1OCCC1N=c1cccc(S(=O)(=O)NC(CN(C)C)CCO)[nH]1 c1(C(N(C)CC2CCN(C(c3c(C)nns3)=O)C2)=O)ccc2c(O)nncc2c1 c1(CC=O)ccc(C)c([N+](=O)[O-])c1.C1(CC#C)(C(=O)N)CCOC1.C(C)CO CCC(C)C(C(=O)NCC1CC(F)CN1C(C1CCCC1)=O)OC C(=O)(CC(C)CCC)N(C1CCN(C(=O)C2=CCOCC2)C1)CC#C C1(OC)CN(C(=O)CCN(C)C)CC1C(=O)NCCCS(C)=O c1(-c2c(C)ccs2)c[nH]c2ccc(C(=O)Nc3c(C)ccnc3Cl)cc12 n1(CCC)cncc1C(C(=O)NC1COC1)N(C1CC(C(N)=O)C1)C Cc1cccc(Br)c1C(C(N1CC(F)C(F)C1)=O)NC(C1CCO1)=O c1(-c2nnc(N(CCC)CCC)n2CC(C)C2CC2)ccc(Cl)cc1OC(C)C N1(C(CNC=O)=O)C2CCCC1CN(C(c1c(F)cc(F)cc1Cl)=O)CC2 N1(C(C(=O)NCc2ccc(OC)cc2Cl)=O)CC(N)CC2(CC2)C1 C1(C(C)C)CCN(CC(O)COCc2ccc(Cl)cc2)C(C(N)=O)C1 CC1(C)CN(C(=O)C(c2cccs2)NC(=O)C2=CCCSC2)CC1O c1(C(C(=O)N(CC(C)NC(C2CC2c2ccccc2)=O)C)C)cncnc1 c1(COC)nc(N2CC(OCCNC(=O)C)C2)cc(Cl)n1.c1ccccc1Cl C1(C(N2C(CC(N3CCC(COC)C3)=O)CC2)=O)(CC)CCCCCC1 c1(C(N2CCCC(C(C)NC(c3c(C)occ3)=O)C2)=O)ccnn2ccnc12 C1(C=O)COC2(CCC2)CC(=O)N1.CCC.C(C)C.C=O.CC=CC N1(C(C2CCC(CNC(=O)C=Cc3cscn3)CC2)=O)CC2COCC(C2)C1 N1(C(Cc2nnc(C)s2)=O)CCC(C(C)(C)CNC(=O)C(=O)N)CC1.C1CC1 c1(OC)cc(C)cc(C(N2CCCC(N(C(=O)CSC)C)CC2)=O)c1N c1(C(N2C(C(N3C(CCC)CCC3)=O)CCCC2)=O)cccc(F)c1N c1(OC(C)(C)C)cc(CNC=O)ccn1.C1C(CN=[N+]=[N-])C1(C)C.CC.N O=C1CCc2cc(C(N3CCCC3CN=c3ccnc(Br)[nH]3)=O)ccc2N1 C(=O)(C1=C(Cl)CCCC1)NC(C)CNC(c1ccc(Cn2ccnn2)cc1)=O CC1(C)CCCN1C(C1CC(Cl)(Cl)C1)=O.c1(C(=O)N)cnn(-c2ccccn2)c1 c12ccnc(c1C)N2.c1(CC(N2CC(CC)OCC2)=O)c(F)cccc1Cl C(=O)(C1CCCc2n[nH]cc21)NCC(C(C)C)NC(CNC(=O)OC)=O C1(CCC(=O)O)(NC(=O)CCc2ccc[nH]2)CCOC1 N1(C=O)CC2(C1)SCCC2OC(C)(C)C.C1(C=O)CC12CC(C(F)(F)F)C2 C(=O)(CC(O)CCS)NC(CC)(CNC(c1ccn(C2CC2(F)F)n1)=O)CC Cc1cc([N+](=O)[O-])ccc1-n1cc(CN=c2[nH]cncc2Cl)nn1 N1(C(C(CN(C)C)O)=O)CCC(NC(=O)CCCn2ccccc2=O)C12CC2 N#CC1(CNC(=NCCC2CCCS2)NCc2ccco2)CCCCC1 c1(N(C(=O)NCC(C)N(C)CC)C)ccc2[nH]ccc2c1 C1(CC(N)=O)CCN(C(=O)C=CC(C)CC)CC1.c1(CC)nocc1C(=O)N C1(C(N(C)Cc2cccc(C)c2)=O)CN(C(c2csc(C)n2)=O)CC(C)(C)C1 c1(C(=O)Nc2c(C)cc(NC(c3cc(=O)cc[nH]3)=O)cc2)cn(C)c(C)cc1=O c1(C(=O)OC)ccc(C(C)NCc2cn(C3CCOC3)nn2)cc1C N1(C(C(C(C)C)O)=O)CCCN(C(C2(Cc3ccccc3)CC2)=O)CC1 c1(NS(Cc2c(C)noc2)(=O)=O)nc2c(s1)CCCCCC2 C(=O)(C(C)CC(C)(C)C)NC(C(C)C)C(=O)N(CC(C)C#N)C Nc1cc(F)c(C(=O)NC2CC2NC(c2ccc(CO)c(Cl)c2)=O)c(F)c1 O=S(=O)(C1Cc2ccccc2C1)NCC1SCCS1 C#CCC(C)(C(=O)NC1CCCC(C#C)C1)NC(=O)C(=O)NCC(F)F N1(C(CCCC)=O)Cc2ccccc2C(CNC(c2nnc(O)nc2O)=O)C1 c1(C(=O)N)cc2c(Cl)cccc2[nH]1.Cn1ccnc1CC(=O)NCC1CC1C CCS(=O)(=O)c1ccc(CC(=O)NC(C)CCN(C)C(c2nocc2Cl)=O)cc1 C(=O)(C1=CCCSC1)N1CC(C)C(CNC(C2(F)CCN(C)CC2)=O)C1 C1(NC(NCC(C)(C)C)=NCC2(C(C)(F)F)CC2)COc2ccccc2C1 N#Cc1ccc(NC(C2CC(O)CN2c2ncnc3sccc23)=O)cc1Cl C1(NC(C2(C)CC2(F)F)=O)CN(C(c2cccc3sncc23)=O)C2CCCCC12 c1(CCCCCC)nc(-c2cc(C)nn2C)n(CCS(C)(=O)=O)n1 N#Cc1ccccc1-c1cn(CCCCCC(=O)N2CC3(C=CCO3)C2)nn1 N1(C(CC(CC)(C)C)=O)CCC(C2(NC(C34CCC(CO)(CC3)C4)=O)CC2)CC1 O(N=C1CCCCCC1)CC(N1CC(C2(NC(CCCOCC)=O)CC2)C1)=O Cc1cnc(F)cc1C(c1nnnn1CC(F)F)NCC1CSCCS1 N1(CCCC)CCC(C2CCN(C(c3n[nH]cc3C)=O)CC2)C1 C1(OC)CN(C(C2CCCC(C)C2)=O)CC1NC(=O)COC(=O)CO c1(C(N(C2CCCN(C(=O)C(C)C3CCC3)C2)CC)=O)ccc(C2CC2)nc1O Cc1cc(C(=O)NC2CC2NC(c2ccc3nccn3c2)=O)c(O)c(Br)c1 CC(CC(N)=O)C(=O)N1CCC(N(C)C(C2CC(=O)N(C)C2)=O)CC1 Cc1ncc(C(=O)NCC(C)(C2CC2)NC(C2C(C)C2C)=O)[nH]1 c1(OC)ncc(NC(C2CCN(Cc3ccsc3)CC2)=O)cc1F Cc1c(Br)c(NC(=O)NOC(C)O)nn1C C1(C#CC(=O)N2CCC(O)C(NC(=O)C(C)(C)C)C2)(CC)COC1.C(C)C.O N1(C(c2ccc(-c3cncn3C)cc2)C(=O)NCCCSC)CC2CCC1CC2 C(CCCCC(=O)NCC1CC(CC)CCN1C(=O)CC(C)N(C)C)OCC C(CCCCC(=O)N1CCC(NC(c2scc(C)c2OC)=O)C1)=CC c1(CC)nc(C)c(C(N2CC(CNC(=O)C(C)(O)COC)C(C)C2)=O)s1 c1(C(N2CCC(C3CCCN3C(=O)C=CBr)CC2)=O)ccc2c[nH]nc2c1 Cc1ncc(NC(c2sccc2CNC(=O)CC(C)c2ccco2)=O)c(C)n1 C=CC1(C(N2CC(=O)NCC2C)=O)CCN(C(c2ccc(C)s2)=O)C1 C#Cc1cn(C)nc1C(=O)NC1(CC(N2CC(=O)NC(CC)C2)=O)CCC1 Cc1c(C(=O)NCCC2(C(=O)NC(c3cnc[nH]3)C)CCC2)cccc1O C1(CC(N2CCCC2)=O)(OC)CCCC1.S(=O)(=O)(C(F)F)N1CC(C=O)C1.C C12(CNC(C(C=C)O)=O)COCCN1CCN(C(c1ccc(C(C)C)nc1)=O)C2 C1(C(N(CC=CC=O)C)=O)CCCC(C)CC1.C1(C(=O)OCC)CCC1 N1(C(=O)CC2CCN(Cc3ccc(Cl)cc3F)C2)CC(F)(F)C(F)(F)C1 c1(C(N2CCC(CN(C(=O)C(O)C3CCCC3)C)C2)=O)cc2cc(O)ccc2[nH]1 C#CCCC(O)C(=O)NCC1C2CN(C(c3cn(CC(O)CC)nn3)=O)CC12 c1(C2C(C(=O)N)C2)cccc(S(C)(=O)=O)c1.c1(CC)cccc(-n2cnnc2)c1 Cc1cc(C(=O)NC2(CCCNC(C3CCC(C(C)C)CC3)=O)CC2)nn1C c1(CC(=O)NC2C(C(=O)NC(C#C)(C)C)CC2)cccc(F)c1 c1(C(N2CCC(C)(NC(C3CCC(CC(C)C)CC3)=O)C2)=O)ccc(Br)cc1F N1(C=O)CCC(S(=O)(=O)N2CCOCC2)C1.c1(CN)cn(CC2CC2)nn1.C c1(-n2ccc(CN(CCCCC)C(C)C)n2)ccc(Cl)cc1 N1(C(c2cncc(SC)c2)=O)CC2CCC1CN2C(C1CCC2(C1)CC2(F)F)=O N1(C(c2ccc(C)s2)=O)CCOC2(CCCN(C(c3ccc(N)c(F)n3)=O)C2)C1 c1(CNC2CCC(C(=O)NCCN(CCO)CCO)C2)cc(Cl)ncc1Br c1(CC(=O)NCCCCCNC(c2cccc(CCC)c2)=O)c(C)cccc1F C1(C(N(C2CCN(C(c3occ(C(=O)OC)c3)=O)C2)C)=O)CCc2n[nH]cc2C1 N1(C(CCCC(=C)C)=O)CCCC2CN(C(C3(C)COCCO3)=O)CC12 c1(C(=O)NC2CCN(C(=O)C(F)n3ccnc3)C2)occ2c1CCOC2 N1(C(C(CC)(O)c2ccccc2)=O)CCOCC(NC(=O)C(F)(F)C2CC2)C1 N1(C(C(C)=C(CC)C)=O)C2CCC1CC(N(C)C(c1ccsc1)=O)C2 C1CCN(C(=O)CC2CC3CCC2C3)CC1.c1(CC)ccc(C(=O)NCC)s1.O c1(C(=O)N)cc(S(N)(=O)=O)c[nH]1.CC(C)CCC.C1(CC=O)CCCC(=O)N1 c1(C(=O)NCC(=CC(=O)NCC(C=C)O)C)ccc(OC)nn1 N1(C(C(Cc2ccc(F)cc2)N(C)C)=O)CC2(C1)CN(Cc1ccccc1)C2 C1(C(N2CCCC(C(N3C(C#C)CC3)=O)C2)=O)CCCCCN1C c1(CC(=O)NCCCCCC)cc(Cl)ccc1OC.C1(C)(C(=O)N)CC2CC2C1 Cn1c(C(N2CC(O)(CNC(=O)CSc3nc[nH]n3)C2)=O)cnc1S c1(C(C(=O)NC2(C)CN(C(C(CC#C)C)=O)C2)C)ccc(OC)c(F)c1 N1(C(C(=O)NCC)=O)CC2CC(NC(=O)CCC(=O)Nc3nccs3)CC1C2 C1(C(F)(F)F)(C=O)CCCCO1.C1(NC(CCOCCOC)=O)CCCC1.C Cc1cccc(Cl)c1CC(N1CCN(C(C2CC3C=CC2CC3)=O)CC1CF)=O c1(C(N(C2CCC(NC(C=Cc3occ(C)n3)=O)C2)C)=O)cc2ccncc2[nH]1 c1(CC(=O)NC2C(C)(C)CN(C(C3CCC(=O)N3)=O)C2)c[nH]c2nccc(Cl)c12 N1(C(CCC(C)O)=O)CC2(CCC(CNC(=O)C(F)OC(F)(F)F)O2)C1 Cc1ccc2nsnc2c1C(=O)NC.C1CCCN(C(=O)C(C2CC2)C2CC2)C1 CC(C)CC(C(=O)N(CCC(=O)NC12CCC(CC1)C2)CC1CC1)C(N)=O S(=O)(=O)(c1cccc(-c2cnsc2)c1)N(C1CCNC1)C(C)C C1(F)(CNC(C(CC)(F)F)=O)COCCN(C(c2cccc(S(C)=O)c2)=O)C1 C1(C(=O)NCC(C)CN(C)C(C2(C(C)(C)O)CC2)=O)CC(=O)N(O)C1 C1(CNC(CSCCC)=O)CN(C(C2CCC2)=O)C(C)(C)C1.N(C)C.C c1(C(N(C2CCN(C(=O)CC3CC3)CC2)C)=O)cc(F)c(O)c(Br)c1 C1(OC)CC2(C1)CN(C(=O)CC(C(C)C)NC(=O)C(C)CO)C2 CCCCC(=O)NC1CCN(C(C2C3CN(C)CC23)=O)C1.C(C)(C)C.C(=O)N N1(C(C(C)NC=O)=O)CCCCC(CCC(=O)NCC(c2cnn(C)c2)C)C1 C(=O)(C1=CCN(C(=O)CCC2CC2)CC1)N(C1CCOC1)CC CC(=Cn1ccnn1)C(=O)NC(C)CC1CCN(C(c2csnc2C)=O)CC1 C1(C(=O)Nc2ccc3sncc3c2)CCCC12CCN(Cc1nc(Br)cs1)C2 C1(NC(C2ON=C(CC)C2)=O)CC(F)CN(C(=O)CC(COC)COC)C1 c1(OC)ccnc(OC)c1C(N1CC2(NC(C3CCCCC3O)=O)CC1C2)=O C1CN(C(=O)Cc2ccc(O)nc2)CC1C(F)(F)F.S(C(F)(F)F)CC(=O)N Cc1nc(CN(C(=O)CC(C)C)C)oc1C(=O)Nc1ccccc1.N(C)(C)C c1(CC)nonc1C(=O)NCCC(C)C.c1(C(=O)N)conc1C1(C)COC1 c1(C(=O)NCC2CC(NC(C3(C)CCC(C)C3)=O)C2)ccc2nc[nH]c2n1 C12(CNC(CCCN(CCCC)CCCC)=O)CC(CN1C(c1ccco1)=O)C2 Cc1c(C(N2CC(C)CCC2c2ccccc2)=O)cc(S(C)(=O)=O)cc1Br N1(C(c2cc(CCC)ncc2)=O)CCN(C(=O)CCC(=O)OCC)C2CC12 C(CCC(C)C)NC(C1CC(O)(CC)C1)=O.c1(CCC=O)cnc(C2CC2)o1 CCCCC(O)CC(=O)NCCOC1CCN(C(C2CC(C(C)C)=NO2)=O)CC1 Cn1nc2c(c1C(N1CCCC(NC(c3ccccc3Br)=O)C1)=O)CCCC2 Cc1cc(NC(=O)CCCCN(C)C)ccc1NC(=O)CCc1ccccc1C#N C1(NC(CC2CC(C)C2)=O)C2CC3C(C2)C13C(N1CC(F)(CF)C1)=O c1(NCC2CC(NC(=O)CC3CCCCCC3(F)F)C2)nccc(Br)c1[N+](=O)[O-] C1(C(=O)NCCc2ccncc2F)CCCN(C(=O)CC(F)(F)F)CC1 C1(F)(C(=O)NC(C2CCCN2C(c2ccc(O)cn2)=O)C)CCCN(C)C1 c1(NC(C2N(C(CCN(C(C)=O)C)=O)CC3(CC3)C2)=O)cnc(Cl)c(C#N)c1 O(NC(=O)C1CCCc2c[nH]nc21)CC(=O)N(C)C Cc1cc(C(=O)NC(CCC2CCC2)C(=O)NC2CCNC(=O)C2)nn1C CC(C)CC(O)CC(=O)NCCN(C(c1ccoc1)=O)Cc1ccccc1 Cc1ccc([N+](=O)[O-])c(C(N2CCSCC2C(N2CC(F)(F)CC2C#N)=O)=O)c1 C1(COC)CCN(C(=O)CC(C)CNC(C2C3CCCC23)=O)C1(C)C Cc1ccccc1C1(C(N2CCC(NC(C3(C)CCNC3=O)=O)C2)=O)CC1 N1(C(CCC2(NC(CCCCC#C)=O)CCCC2)=O)CCC2CC1C(=O)O2 C1(CN(C)C(=O)Nc2cnn(-c3ccc(Cl)cc3)c2)CCCCC1O C1(NC(=O)CCOc2ccccc2O)CCCCCC1NC(C1(Br)CC1)=O C1(NC(COCC(=O)NC)=O)CC2CCCC12.C1(CC=O)CCCCC1O.N CCCCC(O)C(=O)NCC1(C)CCN(Cc2ccc(F)cc2C(=O)O)C1 Cc1ccn2nc(-c3nc(-c4ccc(Cl)s4)nn3C3CCOC3)nc2n1 C1(OC)CC(NC(c2ccnn2C2CCOCC2)=O)CN(C(C2C=CCC2)=O)C1 CC(N=c1[nH]c(=NCc2ccsc2)[nH]c2c(F)cc(F)cc12)c1nccc(O)n1 c1(C(=O)NCCN(C)C(C2CCCC2(F)F)=O)cc(F)c(F)cc1Cl Cc1ccc(SCC(=O)NCCC(C)N(C(=O)C2=COCC2)C)cc1 N#CC1(C(=O)NCC(CO)NC(=O)Cc2ccccc2Br)CC2CC2C1 CCCC(C(=O)NC(C(=O)N(CC(C)(C)O)C)C(C)O)OCC c1(C(=O)NC2(CCC)CCN(C(C(CC)CC)=O)CC2)ccn2c(O)nnc2c1 C1(O)(CNC(=O)C2CCc3ccccc32)CC(N=c2nc(C(F)(F)F)[nH]s2)C1 CCS(=O)(=O)CC(=O)N1CC2CC1CN2C(c1sccc1OC(F)F)=O N1(C(c2cc(NC(C)=O)ncc2)=O)CC(NC(C2(CO)CC2)=O)CC(O)C1 Nc1nccnc1C(N1CCC(C(=O)NC2CC(O)C(O)C2)C1)=O C#CC1(F)CCN(C(=O)C(CNC(=O)C(CC)CCC)CC(C)C)CC1 N1(C(CC=C=C)=O)CC(OC)CC1(C)CNC(c1cc(CSC)ccn1)=O n1(CC#C)cnnc1C(=O)NCC1CC(C(N2CCC(CC)C2)=O)C1 Cc1nn(C)c(C)c1C=O.C1CC2(C1)CN(C(c1cnc(CC(C)C)[nH]1)=O)C2.N C#CCCCCCC(=O)NC(C)CCCC(=O)NCC1CCCCN1C C(=O)(N=c1[nH][nH]cc1C)C1CC(NC(CCCC#C)=O)C1 c1(C(=O)NC2(COC)CN(C(=O)CSC)C2)cc(C(C)C)oc1C CC1(NC(=O)COC2CCC(F)(F)CC2)CCC(C(=O)O)CC1 CC1(C)CCC(C(=O)NCC2CN(C(c3nocc3C(C)(C)C)=O)CC2O)C1 C1(NC(C2(N(C)C)CCC2)=O)CC(CO)N(C(=O)C(c2ccc(Cl)s2)=O)C1 Cc1cc(C(=O)NC(C(=O)NC2CCCC2)C(C)(C)C)cc(C)c1.N(C)C.C C12(CNC(Cc3n(C)ncc3)=O)CCC(CC1)N2C(C1CC2CC(=O)C1C2)=O C(C1=NOC2CN(C(c3ccc(Br)o3)=O)CC12)NC(COCC#C)=O C1(C2CCN(C(=O)CCCC3CC3)C2)(NC(=O)CC2CC2)CC1 Cc1oc(-c2ccccc2)nc1C(=O)N(CC(C)(C)CNC(c1cccs1)=O)C C(CCCC(=O)NC1CCCC(NC(c2ccncc2CC)=O)C1)OCCC=C Cc1ccc(O)cc1C(=O)NCC1(NC(c2c(Cl)cnn2C)=O)CCOCC1 C(CC(C)(C)CC(=O)NCC1COCC1NC(=O)CC1CCCCO1)OC n1(CC(N2CCCC2)=O)nc(O)ccc1=O.Cn1ccc(C(C)(C)C(=O)NC)n1 C1(C(=O)NCC2CN(C(Cc3cc(C)sc3)=O)C2)CCCN(CC(C)C)C1 c1(C(N2CC(F)(CNC(CN(C(COC)=O)C)=O)C2)=O)cc(=O)cc[nH]1 c1(C(=O)NC(CCOCC)C(=O)NCCC(Cl)Cl)cc2ccccn2c1 C1(CNC(C(Cn2cccn2)NC(CSCC)=O)=O)CC2(CCO1)CC2 N1(C(C2CCCN(CCC)C2)=O)CCN(C(C2(Br)CC2)=O)CC1C(C)C CCCCCCCN(C(=O)C(C)N(CCC)C(C1CC2CCC2C1)=O)C Cc1[nH]c(-c2ccco2)nc(=O)c1C(=O)OCc1cnoc1CCO.C1CC1 C1(C(=O)NCCc2cncc(C)n2)CN(C(=O)COC(C)C)C(C)(C)C1 c1(OC)cc(CC(N2CCCC2CCNC(C2CC2(C)C)=O)=O)ccn1 O(NC(=O)Cn1cc(CNC(=O)C(CC)N(C)C)nn1)CC(=O)OCC CCCC(CCCNC(C1CC(F)C1)=O)Nc1ncc(C(F)F)cn1 N(C1COc2ccccc21)C(C1CCCCN1Cc1ccncc1O)=O C(=O)(CCCC(=O)N1CCC(CCN(C(=O)CC2(C)CC2(F)F)C)CC1)N(C)C N1(C(c2cc(C)nnc2)=O)C2CCC(C2)C1C(N1CCNC(=O)C1C(C)C)=O N#Cc1cn(CC(=O)NC2COCC2NC(C2(C)CC2(F)F)=O)c(=O)nc1O N1(C(c2ccc(CC)nc2C)=O)CCC2(CC(NC(c3ccoc3)=O)CO2)C1 c1cccc2c(Cl)c[nH]c12.C1(OC)CC(OC(C)(C)C)CN(C(=O)N)C1.C=O C1(C(=O)NC2CC(=C)C2)CN(C(C2C=CC(C(=O)O)C2)=O)C2(CCC2)C1 N1(C(c2c(C)onc2C2CC2)=O)C2CCC1C(C)C(NC(=O)C1=COCCO1)C2 C(C1=NOC2CCCC12)NC(C1CC(CNC(C2C(CC)OCC2)=O)C1)=O c1(CCC=C)ccc(C(=O)NC2CCCN(C(C3(CC)CCNC3=O)=O)C2)cc1 C1(N(C(C)=O)C2CC2)CCS(=O)(=O)C1.Cc1c[nH]nc1C(=O)N.C1CCC1 N1(C(C2C(C)CCCC2)=O)CCN(C)C(CNC(c2n[nH]cc2Cl)=O)C1 C1(C(=O)N=S2(=O)CCC2)CCc2nncn2C1 c1(OCC)ccc(C)cc1C(=O)NCC(C)NC(C1(C)CCCO1)=O CC(C)(C)CC(CNC(C12CC(c3ccccc3)(C1)C2(F)F)=O)CO c1(NC(C2(N3CCOCC3c3ccccc3)CCC2)=O)cccc(-c2nn[nH]n2)c1 C=CC(C)CC(=O)N(C)CC1CN(C(C2CCN(C(N)=O)CC2)=O)CCO1 Cc1cccc(Cl)c1CC(N1CC2(CCN2C(=O)CN2CCOCC2)C1)=O c1(CC)cc(Cl)ccc1C(N1CC(NC(C23CC(CN2CC)C3)=O)CC1)=O C(=O)(C(O)CC(F)(F)F)N(C)CC1CCCCN1C(c1cocn1)=O C1(COC)CN(C(=O)C(C)NC(C)=O)CCN1C(=O)CN(C)C1CC1 c1(C(N2CC(NC(CC(CCC)C)=O)(CO)C2)=O)cc(N)c(F)cc1C CCCCCC(O)CNC(C1(NC(c2n[nH]c(CC)c2C)=O)CCC(C)(C)C1)=O C12(NC(c3cnc(CC)[nH]3)=O)CCCC1N(C(=O)C1=CCCCC1)CC2 c1(C(N2C(C(=O)NCCC)CCC2)C(=O)NC(C)C)ccc(C(F)F)cc1Cl Cc1c(F)ccc(C(=O)NCC2(F)CCC2)c1N.C1(CC=O)CCCNC1=O.N N1(C(C(N2CCC(C)C2)=O)=O)CC(NC(=O)CC=C(Cl)Cl)CC1CO c1(CN2C(CC(=O)Nc3cnsc3)CCC2)cnc2ccc(F)cn12 c1(C(N(C2CCN(C(C3C(C)C3C)=O)C2)CCC)=O)[nH]cc2c1CCC2 c1(NC(=O)NC(C)C(=O)NCC(F)(F)F)cccc(=Nc2ccccc2)[nH]1 c1(CNC(NCC2CCC(F)(F)CO2)=NCCCCl)cccc2cccnc12 c1(CC(N2CCCC(C(=O)N(CCF)CC3CCCO3)C2)=O)ncc(F)cn1 c1(C(C(=O)NCC2(n3cc(Cn4cccn4)nn3)CC2)(F)F)ccccc1Br c1(C(N(CC(C)N(C(CN(C)CC)=O)C)C)=O)cncc(S(C)(=O)=O)c1 Cc1cc(S(N)(=O)=O)oc1C(=O)NCC1CC1.c1(C=O)cc(Cl)ns1.N C1(CCOCC)(NC(c2cnc(CO)s2)=O)CCN(c2ccnc(C)n2)C1 CN1N=C(CC(=O)N2CCC3CCC(NC(=O)C=Cc4ccncn4)C23)CC1=O O=C1CCC(C(N2CCC(NS(=O)(=O)CCBr)C2)=O)CN1 N1(C(CC2(CC)CC2)=O)CCC(n2cccn2)C1.c1(C=O)cnn(C(C)C)c1.N c1ccc(Br)cc1C(N)=O.N1(C(C)=O)CC(Oc2ccc(Cl)cc2)CC1C=O.N c1(CN2CCCN(C(c3n(CCOC)ncc3)=O)CC2)c(OC)cc(Cl)cc1F C(=O)(C(F)C(F)(F)F)N1CCC(N(CC(=O)NC)C)C1 c1(N(C(=O)CN2CSCC2=O)CC)ccc(C)nc1 c1(CNC(CC(C)(C)n2cc(C(CCC)=O)nn2)=O)cncc2sccc12 C1(C#N)(C(=O)NCC(CNC(Cc2c(C)n(C)nc2)=O)F)CC2CC2C1 c1(OC)cc(O)ncc1C(=O)NC1CCC1C.C(=O)(CC(C)n1ccnc1)N C=CCC(C(=O)N1CCCN(C(=O)CCc2ccc(C)c(C)c2)CC1)C(C)(C)C Cc1cc(S(=O)(=O)N2CC(F)(F)CC2C(=O)Nc2c(Br)cnn2C)c(C)cc1Cl N1(C(=O)NCCOC2CCC(CC)CC2)CCCC2CC3(CCC12)OCCO3 C1(C(N2CCN(C(c3nccc(C#C)c3)=O)C(CO)C2)=O)CCn2ccnc2C1 N1(C(c2nn(CC)c(C)c2)=O)CCCC2(NC(=O)C)CC2C1.C(=O)C1CC1.N N1(C(C(CC)O)=O)CC(OC)CC(NC(=O)CCCCCOC)C1 CC1=C(C(=O)NC(C)C(C)NC(c2sc(C)c(Br)c2C)=O)CCCC1 C1(CC(N2CCC(F)C2)=O)CCC2(CC1)CC2.n1(C(C)C(=O)N)cc(Cl)cn1.C c1(C(=O)OCC)cc(C(=O)N(C2CCN(C(C3CCC(C)O3)=O)C2)C)on1 C1(C=O)CCC(C2CC2)C1.c1(CC=O)cn(C)nn1.C1(C(N(C)C)=O)CCC1 N(C1c2ccccc2CC1NC(=O)C=CCO)C(C1CC(SC)C1)=O S(=O)(=O)(c1ccc(NCc2coc3ccccc23)c(Br)c1)NCC(C)C#N Cc1cnc(NC2COCC2NC(=O)CC(C)C(C)C)nc1SC(C)C c1(C(=O)NC2CC(N(C(c3cc(OC)n(C)n3)=O)C)C2)cccc(F)c1F C(=O)(C1=COCCC1)NC(CC)CN(C(=O)CSC(C)(C)C)C N1(C(CC2(OC)CCCC2)=O)CC(NC(c2cc(C3CC3)ncn2)=O)CCC1C C#Cc1ccc(C(c2nnnn2C)NC2CC3OCCCC23)c(F)c1F c1(C(=O)NC2CN(C(c3[nH]c(=NCC)sc3)=O)C(C)C2)ccc2c(c1)CNC2=O CC(CC1CCCC1)C(=O)NCC(C)CC1(C)OCCO1 C(CNC(=O)CCC(C)OCC)(CC)(CC)NC(C(C=C)C)=O C1(NC(C2C(=C)C2)=O)CN(C(=O)CN2CCCCC2=O)CC1F C1(C(=O)NCC2ON=C(C)C2)(NC(=O)CC(C)n2cccc2)CCN(C)C1 c1(OC)cccc(F)c1CN1CCOCC1CC(N1CC(O)C(O)C1)=O c1(C(=O)NCC(=C2CN(C(C3OCC(=O)C3)=O)C2)F)ccccc1F C(c1cc(C)cc(C)c1)=CC=O.N1(CC)CCCC1C(=O)NC1CC(F)C1 c1(CC(C)C)ccc(C(=O)NCCCCCn2cc(C(O)C(C)(C)C)nn2)cn1 C(=O)C1CCc2cc(Cl)ccc21.CC1(C(=O)NCC2CC2)CS(=O)(=O)C1.C C1(CCNC(C=C(C)C)=O)(NCC)CCC1.CC(C)(C)C.C(=O)(C)N c1(C(=O)NCC2N(C(C=CCC)=O)CC(O)C2O)cc(O)nc2ncccc12 N1(Cc2cn(CC)nn2)CC(Cn2ccnc2C)CCC1=O c1(C(=O)NCC(C2CCN(C(CCC(N)=O)=O)CC2)F)ccc2c(c1)CCCC2 N1(C(C2(CC)CCCCO2)=O)CCn2c(CNC(c3cc(Cl)no3)=O)nnc2C1 c1(OC)ccc(Cl)cc1C(N1C(C)C2CC1C2NC(=O)CC(C)C(F)F)=O C1(N(C(c2c(C)ccnc2)=O)C)CCCN(C(C2(c3cccs3)CC2)=O)CC1 N1(C(COC(CC)C)=O)CCN(C(c2cnc(C(C)(C)C)o2)=O)CC1CO C1(NC(C=COCC)=O)CC(NC(=O)CCCc2cnccn2)C12CCOCC2 Cc1cc(NC(C2CN(C(c3ncccc3F)=O)C3(CCC3)C2)=O)c(O)cc1F c1(N(C(C(=O)NCC(C=C(C)C)(O)CO)=O)C)c(OC)cnc2ccccc12 C=C1CC2CC1CN2C(C1CC1C(C)NC(c1cnc(C)cn1)=O)=O N1(CC)CCCC(ONC(=O)CSCCNC(=O)CC(C)N(C)C)C1 C(=O)(C1CSc2ccccc21)N1CC2C(NC(C3CCC(CC)CC3)=O)(C2)C1 c1(C(N2CCC(CNC(c3cc(OC)ns3)=O)CC2)=O)ccc2nnn(O)c2c1 CC1(C)CCC(CC(=O)NCC2CN(C(=O)Cc3ccc(F)cc3)CC2O)C1 Cc1nn(C)cc1C1=NOC(C(=O)NC2CC(C)C2)C1.C(=O)C.C(C)(C)C.N C(C(=O)NCC1CCC(C(N2CCC(C)(F)C2)=O)CC1)(C(C)C)OCC Cc1c(C(=O)N(C(C)C)C)cnn1C(C)(C)C.C(=O)C(C)(C)n1cccn1.N C1(C(=O)OC)CC2COCC(C1)C2NCC(c1ccco1)N(C)C.C1CN1 N1(C(CCCC#C)=O)CC2(CNC(c3cncn3C(C)C)=O)CCC1CC2 C12(NC(c3[nH]cc(C)c3)=O)CCC(CC1NC(=O)Cc1ccco1)C2 N1(C(CCOC)=O)CCC2(NC(=O)CC(O)CN(C)C)CCCCCC12 CCC(C)C(O)CC(=O)N1CCCC1(C)C(=O)NCC1CCC(C)(C)O1 N1(C(CCC(CC)C)=O)CCCC12CCN(C(=O)C(CC1CCCC1)OC)C2 Cc1cnc(N2CCCC(C3(NC(=O)C(O)C4CCC4)CC3)C2)nc1S(C)(=O)=O N1(C(C(C)C2=CCCC2)=O)CC2CCCN(C(=O)CCOc3cccnc3)C2C1 C1(CC(=O)NCCCN(C)C(C2CCCCC2C(N)=O)=O)CCCS1(=O)=O Cc1ccnc2c(C(=O)N)cnn12.C(C1CCOC1)=CC(=O)N(C(C)C1CC1)C N1(C(CC)=O)CCCC(C(=O)NCC2CCN2C(=O)CCSC)C1 C1(NC(C2CC(C)OC2C)=O)CC2CC(C1)N(C(=O)Cc1sc(O)nc1O)C2 CCC(C)(CNC(C1CC(=O)CN1C(=O)CC1CCCSC1)=O)CC CC(C)C(O)C(C)(C)C(=O)N(CC(=O)NC(c1ccc(O)cc1)C)C1CC1 C1(CCC)(NC(C(CC#C)C)=O)CCCN(C(c2cc(CC)nn2C)=O)C1 c1(C(=O)NCC(C)NC(=O)C)ccccc1C(=O)N(C)C.c1ccccc1F c1c(C)nn(-c2ccccc2)c1Cl.CCC(C)(C)C(=O)NCCOCCN(C)C c1(OC)cccc(C=CC(N2CCC(NC(=O)C3CC3)C23CC3)=O)c1OC C1(C(N2CC(N(C(=O)COc3nc(O)nc(O)n3)C)C2)=O)CCc2nncn2C1 c1(OC)ccc(CN2CCC(C(=O)NCc3ccc(C)cn3)C2)cc1[N+](=O)[O-] Cc1nccc(OC2CC(NC(=O)Nc3ccnc(Oc4ccccc4)c3)C2)n1 C(N=c1[nH]cnc2ccsc12)C1C(NC(c2[nH]c(C)c(C)c2C)=O)CCC1 C1(CNC(C(C)Cc2ccco2)=O)(C)CC12CCC2.c1(C(=O)N)cscn1 N1(C(c2c(C)cncc2)=O)CCC2(CCCN(C(C3CCCCNC3=O)=O)C2)C1 C1(CC=C)(NC(C2CC(C#C)(O)C2)=O)CCN(C(C2CCCCN2CC)=O)CC1 C1(C(N(C)CCO)=O)(CNC(=O)Cn2cccn2)CC2(CC2)C1 C1(C(=O)NC2CC(OC)C2)CC(NC(=O)CCOC)C1(C)C.C1CC1 C1(C(N(CCNC(C2CCC(F)(F)C2)=O)CC)=O)CCCS(=O)(=O)C1 C1(C(=O)Nc2cccc(NC(=O)C=Cc3cnc[nH]3)c2)CCC2COCCC2C1 C1(O)(C(C)NC(C)=O)CCN(C(C2(C(F)(F)F)CC(F)(F)C2)=O)C1 Cc1ccccc1N=Nc1ccc(NC(=O)NC(C)CS(C)=O)c(C)c1 c1(NC(CCc2cn(C)nn2)=O)ccccc1C(N1CCOCC1)=O CC1(C)CN(C(NC2=C(Cl)C(C)(C)OC2=O)=O)CC2(CCOC2)O1 C(=O)(C(C)CCCC(C)=O)NC(CC#C)CC(=O)N1CCC2(CC1)CC2 Cc1cccc(C(C)NC(=O)C(c2cccs2)NC(=O)C(Cl)Cl)n1 C(C(C(C)(C)C)NC(=O)CCc1cccnc1)NC(c1c(C)cc[nH]1)=O C(=O)(C(F)(F)C(CC)NC(=O)CN1CCCC(C(=O)O)(CC)C1)OCC C1(NC(c2onc(C)n2)=O)COC2(C1)CN(C(C1CC1(c1ccccc1)C)=O)C2 c1(-c2cn(C)nc2)cccc(NC(=O)Cc2ccco2)c1 c1(C(N2C(CNC(c3cc(CC)on3)=O)CC2)=O)cc(Br)sc1C Cc1cc(C(=O)OC(COC(C)(C)C)C(C)(C)C)c(Br)s1 N1(C(C(C=C)O)=O)C2CCCC1CN(C(=O)C(C1CCCC1)OCC)C2 C1(CNC(C2CCC(C)C2)=O)CC2CCC1N2C(=O)C(C)(C)c1cccnc1 CP(C)(=O)CCC(=O)N1CCOCC(CNC(=O)CC2CCCS2(=O)=O)C1 N1(C(CN(C(C(N2CC(C)C2)C)=O)C2CC2)=O)CCOC(C)(C2CC2)C1 Cc1nc(F)ccc1C(N1CC2C(NCc3ncccc3Br)C2C1)=O N1(C(CCc2nc(=N)[nH][nH]2)=O)Cc2n[nH]cc2C1C(=O)N1CCCC2(CC1)CC2 c1(NC(C2(C=C)CCN(C(=O)Cc3cncc(C)c3)C2)=O)ccc2occc2c1 C1(NC(=O)COCc2ccnc(O)c2)COC2CN(C(=O)C3=CCCCC3)CC12 c1(C(N(C2CCC(NC(C3CNC(=O)N3)=O)C2)C)=O)cnn2c(Br)cccc12 C1(NCc2cnc(C)s2)CN(C(c2ccc(Cl)cc2)=O)CCC1(F)F CCCCCCC(=O)NC1(CO)CCN(C(c2csc(Br)n2)=O)C1 C=Cn1cc(C(C(=O)Nc2ccccc2)N(C2CCCC2C)CCCOC)cn1 c1(C=O)c(F)ccc(C(F)(F)F)c1F.C1(CCNC(CCOC)=O)CCCC1.N c1(C(C)NC(C(=O)OC)CC2CCCOC2)cc(C)cc(C)c1 N1(C(C2(C)CCCO2)=O)CC2(CCC(NC(=O)Cc3cncnc3)CC2)C1 c1(OCC)nc(C)ccc1C(=O)NC.C1CCCC1.C(=O)CC=C(C)C C1(NC(C(C(C)C)c2cnn(C)c2)=O)CCN(C(=O)C=CBr)C12CCC2 C1(C(=O)NC2(CNC(Cc3c(C)n[nH]c3C)=O)CCCC2)CCCC(=O)CC1 N1(C(CCNC(=O)OC)=O)CCCC(N(C(=O)C=Cc2cncn2C)C)C1 C1(O)(C(=O)NCC23CC(C(F)F)(C2)C3)CCCCC1O c1(NCC2(OC)CCCCC2)cc(=NCc2cc(=O)cc[nH]2)[nH]c(C(F)(F)F)n1 O=C(C1=CC2C=CC1C2)N1CC(NC(=O)C(F)(F)F)CC(F)C1.C1CN1 CC1C(C=CC(N2CCCCC2CNC(=O)C(F)C2CCC2)=O)C1(Cl)Cl Cc1oc(CNC(c2ccc(OCc3cccs3)cc2)=O)nc1.C(N)(=O)N c1(CC)cc(C(=O)N(CCCNC(=O)CCCC(=O)N(C)C)C)cc(N)c1 c1cc(C(=O)N(C2CCOC2)C2CC2)n(C)n1.C(C)(C(=O)N)=C(CC)C.C c1(NC(N(C(C)Cc2cccc(F)c2)CC#C)=O)ncccc1Cl C1(CNC(CCC(C)C)=O)CN(C(C2CC3(C2)CC(CO)C3)=O)CCC1C c1(NC(N(C(C(=O)OCC)Cc2ccccc2)C)=O)cnc(Br)c(Br)c1 n1(CC(N2CC(C3OCCN(C(CC(C)(C)SC)=O)C3)C2)=O)cnc([N+](=O)[O-])n1 c1(OCC(=O)NCCC(CNC(=O)C(C)(C)C)OC)ccc(Cl)cc1F C(C(=O)NC(C)C=CC(=O)N(C(C)CN(C)C)C)OC(C)C C1(CNC(C=CC)=O)COC(C(F)(F)F)CN1C(c1ccns1)=O c1(N2CCCC(C(C)NC(C(C)(C)OCC)=O)C2)nc(C(C)C)ccc1C#N N1(C(C(C)=C2CC2)=O)CCC2(CC1)CC(NC(=O)C(C)C(F)(F)C(F)F)CO2 c1(C(=O)NC(CCCC)C(=O)NCCC(O)CC)ccc2c[nH]nc2c1 N1(C(c2[nH]cc(C)c2C)=O)CCCC(C)(C)C1CNC(=O)CC1CC=CCC1 N1(C(C(=O)NC2CN(C)C(=O)CC2)=O)CC2C(C(F)(F)F)(CCCS2(=O)=O)C1 c1(OC)ccccc1NC(=O)COC(=O)C(C(C)C)n1ccnc1 Cn1ncc2nc(O)c(C(=O)NCC3COC(C)C3)cc12.C(=O)C.CC#N.N C1(C(=O)Nc2cnc(OC)nc2)CCCCCCN1C(c1c[nH]ccc1=O)=O N1(C(COC(C)C)=O)CC2(C(N3CCC(C)(C#N)CC3)=O)CC1CCO2 c1(C(=O)N)ccc(Cl)cn1.C1(C(N(C)CCOCC)=O)(C(F)F)CCCO1 C(=O)(C(CC(F)F)NC(C1(S(C)(=O)=O)CCC1)=O)OC N#Cc1ccc(C(N2CC(CC(F)C(N3CC4(CC4)C3)=O)C2)=O)s1 N1(CC(=O)NC2(C(N3CCC(CO)C3)=O)C(C)(C)C2)CCC(F)CC1 CN1CC(C)(C(=O)NCC(F)CNC(=O)CC2(O)CCC2)CC1=O C1(C(=O)NCCOCC=C)CC2CCC(C1)N2C(=O)C(CC)N(C)C Cc1ccc(Cl)c(CNC2CCCCC2c2cccc(C)c2)c1 c1(CC)ncc(Br)cc1NC(c1sccc1NC(c1ccnnc1O)=O)=O C1(C(C)NC(c2nccs2)=O)CCCN(C(c2cc(C(=O)O)n[nH]2)=O)C1 N1(C(C(CC=C)CNC(C2CC2C(F)(F)F)=O)=O)Cc2ccncc2C1 C1(CNC(c2c(C)cc(C)o2)=O)CN(C(c2cnc(C(F)F)cn2)=O)CCN1C c1(C(N2CCC(OCC)C(C)C2)=O)cc(C#N)c(O)nc1C C1(C=O)CC2(CCC2O)C1.C(CCC)N(CC)CC.C(=O)(Cc1ccoc1)N C1(C)(C=O)Cc2ccccc2C(=O)O1.CCC(C(=O)NC1CC(F)(C)C1)OC.N C=CCC(C)(C)CC(=O)NCC1CCCCC1.N1(CC=CC=O)CCOCC1.N CC(C)(CCCN=c1nc(C2CC2)[nH]s1)NC(=O)CNC(=O)C1CC1 C1(C(N2CCC(n3cc(CC(CO)CO)nn3)C2)=O)CC1C1CCC1 c1(C(N(CCn2cc(-c3cnc(O)nc3)nn2)CC)=O)n[nH]c2cccc(Br)c12 C(=O)(C#CC(C)(C)C)NCC1(COC)CCN(C(C2(C)CCCC2C)=O)C1 c1(C(C)C)cc(C(=O)NCc2cc(C(=O)NC3C(C)C3(C)C)on2)on1 C1(C(N(CC(C(=O)N2CC(OCCCCC)C2)C)C)=O)CCC2(CCC2)C1 C(C(C(C)C(C)C)NC(c1scnc1C)=O)NC(c1c(C)noc1)=O.C1CC1.C N1(C(CCCN=[N+]=[N-])=O)CC2CCC(NC(=O)C(F)(F)F)CC2C1 C=CCCC(C(=O)NCC1(C)CC1(C)C)NC(=O)CP(C)(C)=O c1(OC)ccc(Cl)c(C(=O)NCC2CC3CN(C(=O)C(C)O)CC23)c1F N1(C(c2c(O)cc(C)nn2)=O)C2CCC1C(C)C(NC(=O)C(O)C(C)(C)C)C2 CCC(CC(C)C)C(=O)NCC1(F)CCCN(C(=O)C(C)(C)CC(C)C)C1 N1(C(c2c(CC)n(C)nn2)=O)CCC(C)C(CC(=O)NC(C)C(C)(C)OC)C1 c1(C(=O)NCC2CC(C)N(C(=O)Cn3nnc(=O)[nH]3)C2)cnc(Cl)c(N)c1 c1(CNC(c2sccc2C#N)C)cccc(COCCO)n1 c1(C(=O)NCC2C=CCN2C(c2cnn[nH]2)=O)cc(=O)n2nccc2[nH]1 C(C(CC(=O)N(C)CC1CCC(C)CC1)NC(=O)C(COC)N(C)C)OC c1(C(=O)NCCCN(C2CC2)Cc2cc(C)no2)nnn(-c2ccccc2)c1C CCC(C(=O)N(CC(F)Cl)C)N(C)C(C1C=CCS1)=O C(C)(CCC(=O)NC1C2CC1N(C(C1CC(C=O)C1)=O)C2)OC.C(C)(C)C c1(C(N2CC3C(CNC(C4(C(C)(F)F)CC4)=O)(C3)C2)=O)ccc(Cl)nc1O CC1C(C)N(C(=O)C(F)F)CCN1C(=O)CSc1nc[nH]n1 c1(C(N2CCCCC2c2cn(Cc3nccs3)nn2)=O)coc(=O)c(Cl)c1 C(=O)(CC(O)C(C)C)NC(C(=O)NCCN(C(CC)C)C)C1(C)CC1 Cc1cc(Cl)ncc1C(=O)NCC1(C(N2CCC3(CC2)CC3)=O)CC1 C1(NC(c2nc(C(C)NC(c3cscc3Cl)=O)oc2)=O)CCC(C2CC2)C1 C1(NC(C2CN(C)C2)=O)COC2(CNC(=O)C(O)C3CCCC3)CC1C2 c1(C(N2CCC(COC)C2)=O)cnc2c(F)cccc2c1.C1(C(=O)N)CC(C)C1 C1(C(C)C)CN(C(=O)Cc2cccnc2)CCN1C(c1n[nH]cc1Cl)=O Cc1nccnc1C(=O)NC(C1(O)CCN(C(c2ccnn2CC(F)F)=O)C1)C C(=O)(C1CCCc2nn[nH]c21)N1CC(NC(c2cncc(SC)c2)=O)C1 N1(C(c2n[nH]c(C)c2C)=O)CCCC(CO)(CNC(C2CC3(CC3)CN2C)=O)C1 N1(C(CN(CCC)C)=O)CCCC(C(C)(C)C(=O)NCC2CC3CC3C2)C1.C N1(C(c2ccc(OC)nc2)=O)CC(CC(=O)O)CC12CCOCC2 CC(CC(=O)NCCCN(C(=O)C=Cc1nccs1)C)NC(C1CCCC1)=O N1(C(c2cc(C)c(O)cc2)=O)CCC2C(C1)CN2C(=O)C=CCO Cc1ccnc(C(N2CC(NC(c3cnc(C(C)(C)C)o3)=O)C(C)C2)=O)n1 C(=O)(C1=CC2(CCN(C(C3CCCO3)=O)C2)C1)N1C2(C#C)CC(C1)C2 CCC(C)C(C(=O)N(CC1CCCCC1)OC)NC(=O)C1CCc2c[nH]nc21 N1(C(C(CC#C)(C)CC)=O)CCC2(CCC2NC(c2ccnc(OC)c2)=O)CC1 Cc1cccc(CC(=O)NCC2CN(C(c3c[nH]c(C#N)c3)=O)CCO2)c1 C1(N(CCC)C(=O)Nc2ccncc2)CCN(Cc2c(C)noc2C)CC1 C1(C)(CC(=O)NCC(C(=O)NC)C)CCN(C(C2CN(CC)CCO2)=O)C1 N1(C(C(CC)(C)CO)=O)CC(CO)C2(C1)CN(C(c1oc(C3CC3)nc1C)=O)C2 CCC(F)(F)CC(=O)NCC(O)CNC(=O)C(C)(C)n1cncn1 C1(c2n(CCCCCC)nnn2)(NC2COC(C(F)F)C2)CCCOC1 c1(C(=O)NCC(CNC(c2c(C)cccc2C)=O)CO)noc2ncccc12 c1(C(=O)NC2CC(NC(CCC(C)N(C)C)=O)C(O)C2)c(F)ccc(Cl)c1F N1(C(C=CCC)=O)CC2CCOCC2(NC(c2cnc(C(=O)OC)cn2)=O)C1 c1(SCC(=O)NCC(CO)NC(=O)CCCCc2ccccc2)ccc(F)cc1 C1(C(=O)NC(CC#C)C(=O)N2CC(CF)C2)CCN(C)C(=O)C1 Cc1ccc(C(N2CCCC(CCC(=O)NC3(CC(N)=O)CC3)C2)=O)cc1F c1(C(N(CCCCNC(C2C(C)C2C)=O)C)=O)cnnc2ccccc12 C1(C(=O)NCC(C)N(C)C(c2cnc(C(C)(C)C)[nH]2)=O)(CC)CCOC1 Cn1cc(C(=O)C(=O)NC(c2ccccc2)CNC(C2CCC(C)O2)=O)cn1 CC1(C(=O)N(CCNC(C2CCC3CC23)=O)C2CC2)CCC(F)(F)CC1 C(CCC(=O)NC1CC(c2cccs2)(CNC(=O)C)C1)SC.c1nccs1.N N1(C(NNC(c2cc(C#N)oc2)=O)=O)CCOCC(F)C1 C1(C(C)(C)C)C(NC(=O)CC2OCCC2(C)C)CCN1C(=O)CCc1cocn1 CC(CC(=O)N(C)CCNC(C1(O)CCCC1)=O)C(F)(F)C(F)(F)F C1(C(=O)OC)CC(O)CN(C(C)=O)C1.C1(OCC)C(O)CCO1 N1(C(C2(C)CCCOC2)=O)CC2OCC(NC(=O)CCCC(F)(F)F)C2C1 CC1(C#CC(=O)NCC(CO)NC(=O)Cc2ncc(Cl)s2)CCCO1 N#CC1CCCN(C(C2CCCCN(C(c3cscc3Cl)=O)C2)=O)C1 Cc1cc(C)c(-n2cc(CN(O)C(=O)c3cn(CC(F)(F)F)nn3)nn2)c(Br)c1 c1(CC)nc(Cl)nc(N2C3CCC2CN(C(C2CC4(CCOC4)C2)=O)C3)c1C#N c12cc(nc(O)c1)C(c1cc(C)n(C)n1)c1nc-2no1.C(C)C N1(C(COCCC#C)=O)CCC(C(CO)NC(=O)CCC(C)OC)CC1 c1(C(N(c2ccncn2)C)=O)cnccc1C#N.C1CCNCC1F C1(CNC(=O)C(C2CCCCCC2)O)CC2(CC2)CN1C(C1CCCC1)=O N1(C(c2c(C)cc(Br)c(N)c2)=O)CCC2C1CCCN2C(=O)C(C)(C)F C(=O)(C1=NNC(=O)CC1)NCC12N(C(C3CCC(CC)O3)=O)CC(C1)C2 C1(C(N(CCCN(C(Cn2c(C)nnn2)=O)C)C)=O)CCCCC1C1CC1 CCC(CCC(=O)N1CC(F)(F)CC1CO)NC(=O)Cc1cnnn1C C(=O)(CCCCCSC)NC(CCNC(C(C(C)C)OC)=O)C C1(C(N2CCCCCC2)=O)(CC)CCN(C(=O)C(N2CCOCC2)C)C1 c1(CCC)ccc(NC(C2CC(F)CN2C(C2(C)CC2)=O)=O)cc1 C1(C(=O)NCC(CNC(=O)C=CC2CC2)OC)CC2CCC(C1)C2O N1(C(C2CC(=C)C2)=O)CCOC(CC(N2CCC(N3CCC3)C2)=O)C1 N1(C(c2ccc(C(=O)OC)nc2)=O)C2CCC1C1CC1C2.C(=O)C=C1CCC1 C(=O)(C(C(=O)NC(C)CC)C(C)(C)C)OCC.c1(C=O)cncc2nc[nH]c12 Cc1cc(C(N2CCCC(C)C2CNC(=O)CC(F)(F)F)=O)c2c(c1)CCC2 c1(C(N)C(=O)N2CC(N(C=O)CCO)C2)ccc(NC(N)=O)cc1 C1(C(=O)NC2CC3CN(C(C4(CCOC)CC4)=O)C2C3)CCc2nncn2C1 N1(C(C2CC(CC)(C)C2)=O)CCC(N(C)C(C2CN(C(C)C)C2)=O)C(C)C1 C(C(CC(=O)NC(c1ncccn1)C)NC(=O)C(C)C(F)F)OC CC(C)CC(C)C(=O)N1CC(NC(c2cc(O)ncn2)=O)C(c2cncn2C)C1 c1(CC(C)C(=O)N2CCC(CNC(C3(C)CC3C)=O)C2)ccc(C#N)cc1 C=CC(C)(CCOC)C(=O)NCc1ccc(C(=O)N)cc1.c1(CC)scnc1C Cc1ccc(C(=O)NC(c2ccccc2)C(C)NC(c2ccc[nH]2)=O)cn1 c1(C(=O)NCC(C)NC(C(C)Sc2ccccc2)=O)ccc2sc(O)nc2c1 CC1CN(C(=O)C2=NOC(C)C2)CCN1C(c1cc(-c2ccccc2F)on1)=O C1(OC(c2nc(C3CC3)sc2Br)=O)CCCN(c2cc(N3CCOCC3)ncn2)C1 N1(C(c2ccc(C#C)c(F)c2)=O)CCN(C(c2csc(C)n2)=O)C2CCCCC12 N1(C(CN2C(C)CCC2)=O)CCSCC1CCNC(=O)COc1cccc(Cl)c1 c1(C(=O)NC23CC(NC(=O)Cn4cccnc4=O)(C2)C3)sc2ccccc2c1Cl N1(C(C2CC(O)C(F)C2)=O)CC2(CC(CO)CO2)C1.C12CCCCCC1C(=O)N2 c1(C(C)=O)cc(C(=O)NC(c2noc(Cc3ccccc3)n2)C2CC2)cs1 Cc1cccc2nc(N(CC(C)NC(C3CCCCS3)=O)C)sc12 c1(OC)cc(C=CC(=O)N)sn1.C1C2CN(C(=O)Cc3csc(C)n3)CC12 N1(C(C2(CCC=C)CCCC2)=O)CC2CC2(NC(c2c[nH]nc2OC)=O)C1 C1(C(=O)NCC2(CCC)CC2)CC=CC(NC(c2cc(O)[nH]n2)=O)C1.C c1(CCC)ccc(S(=O)(=O)NCc2ccc(N3CC(CN)C(F)(F)C3)nc2)cc1 C1(c2nnnn2Cc2cccs2)(NCC(=O)OCC2CC2)CC2CCC1C2 c1(CCC=O)c(Cl)cccc1Cl.CCCCCCNC(=O)COCC1CCC1.N Cc1ccnc2c(C(=O)NC34CCCN(C(=O)OC(C)(C)C)CC3C4)cnn12 C(=O)(C(CC(C)(C)C)O)N(CC(C)N(C(C1CCC(SCC)CC1)=O)C)C c1(OC)cc(OC)c(C(=O)Nc2cnc(Br)c(F)n2)cc1OC C1(C=O)CCCC2(CC2)C1.Cc1nc(C2CC2)[nH]c1C(=O)NCCC1CCC1 c1(NC(Cc2[nH]c(=NCc3cc(C)c(Cl)cc3)sc2)=O)ncccc1[N+](=O)[O-] CC1CC(C)N(C(c2cc(O)nc(C3CC3)n2)=O)CCN1C(=O)CC1CC1 C(=O)C(C)P(C)(C)=O.c1(COC)cc(C(=O)NC2CC(O)(C)C2)no1 C1(NC(Cc2cc(C)no2)=O)CCC(C)(C)C1.c1(C(=O)N)csc(C(F)F)c1 c1(CC)nn(C)c(Cl)c1C(=O)N(C)CCNC(=O)C(C)(Cl)Cl N1(C(CCc2scc(C)n2)=O)CC2CCC(C1)N(C(=O)Cc1ccn(C)n1)C2 C1(NC(=O)CCc2cnn[nH]2)CCN(C(C2(CS(N)(=O)=O)COC2)=O)C1.C O=C(CS(=O)(=O)Cc1ccc(Cl)s1)N1CCC(Oc2ccc(F)c(Br)c2)C1 C1(CSCc2ncc(C(=O)OC)nc2)Cc2cc(OC)c(OC)cc2C1=O Cc1cnc(C(N2CCCC2CC(=O)OC)C(=O)NC2CCOC2)o1 C1(C)(C(=O)NCCCNC(CN(C)S(N)(=O)=O)=O)CCC2(CC1)OCCO2 O=S(=O)(c1ccc(Br)cc1NCC=CCl)N1CCC(F)(CO)C1 c1(NC(C2(NC(CCCCOC)=O)CCC2)=O)ccc(O)c(OC)c1 C1(C(=O)NCC2C3CN(C(C(C(C)C)C)=O)CC32)CCC(N=[N+]=[N-])CC1 N1(C(Cc2c(C)occ2)=O)CC(C)OC2(CCN(C(=O)C3=C(Cl)CCC3)C2)C1 C1(NC(C(C)NS(CC)(=O)=O)=O)C=CCN(C(c2cccc(Br)c2)=O)C1 N1(C(COCCC)=O)CCC(C)(CNC(=O)C(CC)N)CC1.c1ccco1.C N1(C(CCOCC(C)C)=O)CC2CCCC2(NC(c2cc(N)ccn2)=O)C1 CC(C)(C)S(=O)(=O)CC(=O)NCc1ccsc1Br C1(NC(=O)CCc2cc(F)ccn2)CCC2(CC1)CCN(C(C1CCOC1)=O)C2 c1(OC)ccc2cccnc2c1S(=O)(=O)N1CCC(C)C(F)(F)C1 [SH](=O)(=O)c1cccc(Cl)c1.C1(OC)(CN)CCSCC1.C1(C)(CC)CC1(F)F N1(C(c2csnn2)C)CCCC(NC(c2cn(C)nc2C2CCC2)=O)CC1 c1(CC)nc2sc(C)cn2c1C(N1CC(NC(c2oc(C)cc2C)=O)C1)=O Cc1ccc(C)c(C(N2CC(=O)NCC2C)C(=O)NC2(C)CC2)c1 c1(CC)noc(CCCC(=O)NC2CC2NC(C2CC3CC3C2)=O)n1 CC(C)CCN=C(NCCCOCC1CCC(C(N)=O)O1)NC(C)C CC1CCN(C(=O)CN2CCN(C3CC3)C2=O)CC1NC(=O)CCN1CCCC1 C1(NC(C2(C)C=CCC2)=O)CCCCN(CC(c2ccc(F)cc2F)O)C1 C#CCC(C(=O)NC(C)CC1(O)CCC1)NC(c1nccn1C)=O CCCCCS(=O)(=O)CC(=O)NC(C)(C)CCCNC(=O)C(C)(C)CCC N(C(=NCCc1ccc(F)cc1)NCc1ccsc1Br)CC(O)CF N1(C(C(C2CCCCC2)OC)=O)CCC2C(CCN2C(=O)CCNC(N)=O)C1 c1(-c2cn(CCCNC(c3nccc(C)c3F)=O)nn2)cc(F)c(F)c(F)c1 c1(C(N2CCCC(C(C)NC(=O)Cc3nccn3C)C2)=O)cc(O)c(F)cc1N c1(C(N2C(C(N3C(C(C)C)C(C)(C)C3)=O)CC2)=O)c[nH]c2ncccc12 c1(-c2cn(C(C(=O)NCc3c(SC)nn(C)c3)C)nn2)ncc(Cl)cc1F c1(C(N2C3C(NC(C=C4C(C)(C)CCCC4)=O)C(C3)C2)=O)ccc2[nH]ccc2c1 CC(C)(CC(F)F)C(=O)N1CCCC(c2ccc(F)c(O)c2)C1 c1(C(=O)NC(C)C(C)NC(C2(CO)COC2)=O)ccc(CO)nc1 N1(C(C2CC(OC)C(OC)C2)=O)CC2(CCCN(C(C3(OC)CCOC3)=O)C2)C1 c1(C(=O)NC2CC(N(C(c3cc(CC)on3)=O)C)C2)c(OC)ccnc1O C1(CNC(C(C)(C)CO)=O)CC(NC(=O)Cc2csc(Br)c2)C12CCC2 c1(CC(C(=O)NCCC(C)F)NC(C2CC2(F)F)=O)cnn(C)c1O c1(OC)cncc(C(=O)NCC2CC(O)CN2C(=O)Cc2nc[nH]n2)c1 CCC(Cc1cccc(C)c1)C(=O)NCC(C)CNC(C1CN(C(C)C)C1)=O c1(C(=O)NC(CNC(c2nc(C)oc2C)=O)CC(C)C)ncc(Br)cc1N N1(C(CC=C)=O)CC2CC1CN2C(=O)C=Cc1cnc(C(C)(C)C)s1 CC(C)CC(C)CC(=O)N1CC2(CC2)CC1CNC(c1occ2c1CCC2)=O c1(C(=O)NC2(C)CN(C(=O)CCCCC3CC3)C2)ccc2cnccc2c1 c1(C(=O)NC2CN(C(C=CC(=O)NC)=O)C2)cc(N)c(C)cc1Cl c1(NC(=O)NCCc2cc(C)c(Br)cc2)c(C)ccnc1C#N c1(OC)cc(=NC(C)Cc2c(OC)cccc2Cl)[nH]nc1OC c1(C(=O)NCC(CC)NC(C2CC(N(C)C)C2)=O)oc2ccc(C)cc2c1C C12(CNC(C(C)Cn3cccn3)=O)CC(NC(=O)C=C(Cl)Cl)(CO1)C2 C1(C)(C(=O)NC(CNC(C(=Cc2cccs2)C)=O)C)CCC(C)C1(C)C C1CC2(CC2)CN1C(=O)CC.C1(C(=O)NC)(OC)CCC(C)C1.CC(F)F C1(C)(C(N2CCC(CC(=O)OC)C2)=O)CCCN(C(C2(CCO)CC2)=O)C1 C#Cc1ccc(CCC(=O)N(CCCCN(C(=O)C(C)(C)C)C)C)cc1 C1(NC(c2cnc(CCCC)s2)=O)(CC)CCCN(C(C2CCCN2C=O)=O)C1 Cc1nc(C(=O)NC2CCCC(NC(C3(N4CCOCC4=O)CC3)=O)C2)c(C)o1 N1(C(C(COC)C)=O)CCCC(CCC(=O)N(CC(C)(C)C)C(C)C)C1 C1(N(CC(F)F)C)CCN(C(=O)CC2(c3ccccc3)CC2)CC1 C(C)(N=c1nc(C2CC2)[nH]s1)C1CCN(C(C(C)Sc2ncccn2)=O)CC1 Cc1nc2c(N(Cc3cccc(C#N)n3)CC3CCSCC3)ncnc2[nH]1 S(=O)(=O)(c1cc(Cl)ccc1Cl)N1CC2C(C(=O)Nc3cccc(OC)c3I)C2C1 c1(C(N2CC3C(C)(C)C3C2)=O)cc2ccc(-c3cnn(C(F)F)c3)cn2c1 N1(C(C(C2CCCC2)OC)=O)CCC(OCCC)CC1.C1(C)(C=O)CC1(F)F.N Cc1cccc(N)c1C(=O)NCC1CCN(C(c2cccc(C(C)C)n2)=O)C1 C1(C(=O)NC(CCCC)CNC(=O)Cc2c[nH]nc2O)CCCC1P(C)(C)=O c1(C(=O)Nc2cc(OC)c(Cl)nc2)cccn2c(-c3cnccc3C)cnc12 C(=O)(C(=O)N(CC(C)CCOCCOC)C)NCC(C)C.C(=O)(C)N N1(C(C2CCCN(C)C2)=O)CC2CCN(C(=O)C(F)OC(F)(F)F)CCC2C1 CN1CC(C(=O)NC2(C)CCN(C(c3ncccc3Cl)=O)CC2)CCC1=O C12(CNC(C(C(C)C)O)=O)CCC(CC1)CN2C(C1CCC1)=O c1(NC(CC2OCCN(C(c3cc(CC)on3)=O)C2)=O)ccc2c(O)n[nH]c2c1 n1(CC)nc(C(N2CC(NC(C3CCC(F)CC3)=O)CC2C)=O)c(C)n1 c1(CNC(N2C(C)(C(C)C)CC2)=O)cnn2c1NCC2 N1(C(=O)Cn2nnc(C3CC3)n2)CCOCC1C1CC(F)(F)C1 N1(C(C2CCCN(C(CC)=O)C2)=O)CCN(C(c2ccnn2C(C)C)=O)C(C)C1 CC(C)(N=[N+]=[N-])C(=O)N1CC(C(=O)NCCCCC(N)=O)C(F)C1 Cc1cccc(C)c1CC(=O)NCCC1CCC1.n1(CC=O)ncn(C)c1=O.N C(F)(c1ccccc1)=CC(=O)NCCC(C)NC(C1(c2ncco2)CC1)=O N1(C(=O)CC2C=CCC2)CC2CC(N=c3[nH]c(Cl)ncc3F)C2C1 O=C(C1=CCCN(Cc2ccc(C(F)(F)F)nc2Cl)C1)Nc1nnc(Cl)cc1Br c1(C(=O)NC2CC(CNC(CCC(C)(C)F)=O)C2)cc([N+](=O)[O-])ccc1Br Cc1ncncc1C(N1CCC(CC(=O)N(CC(C)(O)C2CC2)C)CC1)=O C1(C(N2CC(COC)(C)C2)=O)CCC12CCCO2.c1(CC=O)c(C)n[nH]c1C C(=O)(C(CC(C)C)C(N)=O)NCCOCCC(=O)N(CC(=O)NC)C S(=O)(=O)(c1cc(I)ccc1C)NCc1c(CC)ccc(OC)c1 C1(NC(COCCCCC)=O)CC(O)CN(C(c2cnns2)=O)C1 c1(CNC(=O)NC2CCS(=O)C2)ccc(-c2cscn2)cc1 N1(C(=O)CSC(F)(F)F)CCC2CN(c3ccc([N+](=O)[O-])cc3Br)CC2CC1 C#CCCC(O)C(=O)NCCCCNC(c1c(C2CCCC2)noc1C)=O c1(OC)ccc([N+](=O)[O-])c(S(=O)(=O)NCc2cnc3c(c2)COCC3)c1 c1(OC(CC)C)ccc(C(N2CC(C(C)NC(=O)C(F)C(C)C)C2)=O)cc1 N1(C(CC2CC(OC)C2)=O)CCN(C(=O)CSC(C)C)C(C2CC2)C1 c1(NCC(=O)NCC=CCC(=O)NC(C2CCCC2)C#C)ncccn1 CCCCCC(O)CC(=O)NC(CNC(=O)CS(=O)(=O)CC(C)C)CCCC C(=O)(C(C)(C)C(C)(C)C)NCCC1(C)CCN(C(CCC)=O)C1.C(N)(=O)N C1(C(N(CCC)CCC)=O)OCCC1.C(=O)C.C(=O)C.C(=O)C1CC1.N C1(OC)CCCC(CC(N2CC(F)CC2CNC(=O)C(C)C2CC2)=O)C1 C(C(C(=O)NCCC1(C)CCCO1)NC(C1CC(C)C1)=O)OCC C(=O)(C#CC1CCCO1)N(CC(C)O)CCNC(=O)Cc1ccc(C#N)nc1 C1(CNC(=O)C2=CCCC2)CCCCN(C(=O)CC2CCC(C3CC3)O2)CC1 C1CCN(C(=O)CN2CCCNS2(=O)=O)CC1C.C(C(=O)N)=CC=CCC.C CC(C)C(O)CC(=O)NCc1ncoc1CCNC(c1cc(Cl)ccc1)=O.C C(CC(=O)NCCOC1CCOC1)(C(F)F)NC(C(CC)(F)F)=O c1(CNCC23C(CN(C(=O)C(F)F)C2)C3)cc(O)ccc1[N+](=O)[O-] CCC(C)(F)C(=O)NCC1(C(C)(C)O)CN(C(=O)Cc2csc(C)n2)C1 C=CC(O)C(=O)NC1CCCC1NC(=O)CCNC(=O)OC(C)(C)C C1(CCC=C)(C(=O)NC2CCN(C(=O)CSc3n[nH]c(C)n3)C2)CCCC1 CC1CCN(C(=O)C(C)N2CCC2CNC(C2(O)CCOCC2)=O)CC1 CC1=CCC(C(=O)N(C2CCCCC2NC(=O)CCN2CCC(O)CC2)C)CC1 c1(C(N2CC(NC(c3cc(CC)ncn3)=O)C(C)C2)=O)ccc(Br)nc1O c1(C(C)C)nc(N2CCC3CC3C2)cc(N2CCC(CN(C)CC3CC3)CC2)n1 CCC(O)C(C)C(=O)NCC1(NC(=O)C(C)n2cccn2)CCOC1 C(=O)(CCC(C)(C)C#N)NC(CCC)C(=O)NCc1nnc(C)o1 C1(NC(c2n(C)cnc2)=O)CS(=O)(=O)CC1N=c1cc[nH]cc1C#N C(=O)(CCCCC#N)NC(CC=CC)C(=O)NCC(CO)CC(C)C C1(C(N(C2CC3CCC(C2)N3C(=O)CSC2CC2)C)=O)Cc2ccccc2O1 N1(Cc2nc(CCCC(C)C)on2)CCCC2(CC(CO)CO2)C1 C(=O)CC(C)C(F)F.Cc1c(C(=O)NC(C)C(C)C)cnn1CCN(C)C.N C(C)(CCC(=O)N1CCC(N(C(=O)Cc2cccc(O)c2)CCO)C1)SC C1(CC)(NC(C2CCCCC2NC(c2cc[n+]([O-])cc2)=O)=O)CCCCCC1 c1(C(=O)NCC2(NC(c3ccco3)=O)CC2)ncncc1Cl.[nH]1cccn1.C N1(C(C(CC)(C)O)=O)CC(C(=O)N(CC(C)C(F)(F)F)C)CCC1(C)C C(=O)(CC(CC)CCCC)N(CC1CCN(C(CCCC)=O)CC1)CC C12(CNC(Cc3c(C)noc3Cl)=O)CCCC1N(C(C1CC1C)=O)CC2 C=CCC(CC)C(=O)NCCCCCC(=O)NC(C)C(F)F C1(C(=O)NCCN(C(c2n(C=C)ncc2)=O)C2CC2)CCc2nc(C)sc2C1 CCCCC(O)C(C)C(=O)N1CC(NC(c2cc(Cl)c[nH]2)=O)CC1(C)C c1(C(=O)N)ccc(O)nc1C.C(CC(=O)NCCCOCC(C)C)NC(C)=O CCCC(O)C(=O)NCC#CCNC(c1ccc(OC(C)(C)C)nc1)=O C1(CNC(c2cnsn2)=O)CCC(NCc2ncccc2Cl)CC1 C1(CC=O)CCC(C)(C)CO1.Cc1nn(CC(F)F)cc1C(=O)NC1CC1.C c1(N2CCC(OC)C(F)C2)nc(=N)[nH]c(=NCc2cnn(CC(C)C)c2)[nH]1 FC1(F)C2(CC2)C12CC(CNC(=NCCC1CCCO1)NC)C2.C1CCCCO1.S C1(C(N(CC#C)C)=O)CC2(CCC2)C1.c1ccccc1.C1(CC=O)CCCO1 N1(C(CCCCOC)=O)CCC2(CCOC2)C(CNC(c2n[nH]c(C)n2)=O)C1 N1(C(C(CC#C)CC#C)=O)CCOC2(CCN(C(c3c(C)nsc3N)=O)CC2)C1 C1(NC(C2CC(C)(C)C2)=O)CCCC(NC(C2CC2)=O)CC1.c1ccco1.N C1(C=O)COCCN1CC(F)(F)F.c1(C(=O)NCCC)n[nH]cc1C1CCC1.N c1(CC)cnc(C(N2CCOCC2CN(C(=O)C(C2CC2)SC)C)=O)nc1 c1(C(=O)NC2(CF)CN(C(CCNC(C)=O)=O)C2)ncc(N)cc1C N1(CC(=O)N(CCC)CC)CCN(C)C(=O)C1.c1(C(=O)N)c[nH]c(=O)cn1 [SH](=O)(=O)c1ccccc1.C(C)(CC)N(C(C=C(COC)C)=O)C.C(=O)CC.N Cc1ccc([N+](=O)[O-])c(C)c1C(=O)NC1COCCC1NC(=O)C(C)N(C)C C#CC1CCC(NC(c2coc(CNC(C3(CCC=C)CC3)=O)c2)=O)C1 N1(C(Cc2[nH]c(=NC)sc2)=O)CCCCC(CN2CCN(C)CC2)C1 c1(OC)ccc(S(N)(=O)=O)cc1C(N1CC(CO)C1)=O.C(=O)CNC=O.N c1(CNC(C2(CNC(c3csnc3Cl)=O)CC(=C)C2)=O)ccc(CO)cc1 C1(C(N(C)C)=O)CCCC1NC(=O)C(F)(F)c1nccs1 c1(OC)cc(C(=O)NCC2(C)CN(Cc3ccc(OC)nc3)C2)c(Br)cn1 O=C1CC2(CCCN(C(=O)NC(c3ccc(F)cc3)C3CC3)C2)CN1 C(C(=O)N1CC(F)(CNC(=O)CC(C)O)C1)(C(C)(C)C)SC C1(C(=O)N)(COC)CCC(=O)N1.C(c1cnc(C)s1)=CC=O.CC(O)C c1(OC)cc(C(N2CCCC2C(C)NC(C23CCC(C2)C3)=O)=O)cc(F)c1F C(=O)(CCC(C)(F)F)NC(CNC(C1(OC)CCSC1)=O)C1CC1 C(=O)(CS(=O)(=O)C1CC1)NC1C(CNC(CSC)=O)CCCC1 Cc1oc(C(=O)NCC2COCC2)cc1-c1ccccc1.C(=O)(C)N.C1CC1 c1(C(N2CCCC(C)(O)CC2)=O)cn2ccc(-c3cc(O)c(F)c(F)c3)cc2n1 N1(C(c2nc(C)sc2C)=O)C2CCC1CN(C(c1cnn3cccnc13)=O)C2 CC1(C(N2CCC2CO)=O)CCCN1C(c1nc(C(c2ccccc2)=O)cs1)=O c1(C(N(CCNC(c2cc(C)nnc2O)=O)C)=O)cccc2occc12 C12(C(c3n(CCCOC)nnn3)NC3CC=CCC3)CCC(CC1)OC2 c1(OC)ccc(C(N2CCC2CNC(=O)Cc2ccns2)=O)cc1Cl C=CCN=c1[nH]cc(C(=O)NCCN(C(=O)C(C)OCC)CC(C)O)s1 CC1CCN(C(=O)OC(C)(C)C)CC1C(c1nnnn1C)N.CCC.C(N)=O CC1CCC(CC(=O)NCC2CCC(NC(c3cc(C(F)F)no3)=O)C2)OC1 C(CC(CO)C(C)C)NC(c1sc(Br)nc1C)c1n(CCCOC)nnn1 C1(C(=O)NCCCCN2CCCC2)CC(O)CN1C(=O)CC1CCC(O)C1 C1(C(N2CCC(NC(C3(C)CCN(C)CC3)=O)C2)=O)Cc2cncn2C(=O)N1 c1(CC(N2C(CNC(c3c(C#C)c[nH]n3)=O)C=CC2)=O)c(C)nc(C)nc1C c1(C(=O)NCC(C)CNC(C2(F)CCOC2)=O)ccc(O)c2ccccc12 N1(C(C(C(C)(C)C)C2CCC2)=O)CCC(C2(O)CN(C(=O)CC3CCCC3)C2)CC1 O=C(C(O)CC(F)(F)F)N1CCCN(C(c2ccnn2C2CCCC2)=O)CC1 CN=c1cc(C(=O)NCC2CCCC2NC(c2cscc2F)=O)cc[nH]1 c1(NC(c2c(N)cc(CC)c(F)c2)=O)ccc(N=S2(=O)CCCC2)cc1 Clc1cc(C(c2nnnn2C2CC2)NCc2ncc(-c3ccccc3)[nH]2)cnc1Br C1(CC)CCCN1C(=O)C(=O)NCC.c1(CC=O)c[nH]nc1O.C1CCC1.C N1(C(CCC=C)=O)CC(CNC(=O)C(c2ccccc2Cl)C)OC2CCCC12 c1(OC)cc(C)c(NC(=O)CN2CCN(C(=O)CCC(C)OC)CC2)cn1 N1(C(C#CC(C)C)=O)CC2CN(C(=O)Cc3cnccc3Cl)CCC2(CO)C1 C1(NC(C2C(=C)C2)=O)(C)CCC(F)(F)CC1.n1(C(CC=O)C)nc(C)cc1C N1(C(CCC2(C)N(C(CN(C3CCC3)C)=O)CCC2)=O)CCC2(CCC(O)C2)C1 N1(C(C(C)=CC)=O)CCCC(CCC(N2CCC(CC(C)(C)C)C2)=O)C1 c1(N2CCC(C)(CNC(C3C(C4C(C)C4)C3)=O)CC2)ncnc2c1nnn2C c1(NCCOCCCCNC(C(=O)N(C(C)CO)C)=O)ccccc1 C1(NC(C2CCC(CC)O2)=O)CC(C(=O)NC)C12CCC2.c1nccc(C)n1 O=C(CCC1=CCCCC1)NCC1N(C(c2cnc(O)o2)=O)CCCC1(C)C C1(C(=O)NCc2cn(CC#C)nc2)CCOCCN1C(=O)CC1(OC)CCC1 Cc1coc(C)c1C=CC(N1CCOC(CCNC(c2snc(O)c2Cl)=O)C1)=O C(CC(C(=O)N(C1CN(C(C2CC(C)(O)C2)=O)CC1O)C)OC)OC C1(c2cccnc2)(C(c2ccccc2)N(CC(C2(C)CC2)O)C=O)CCCCC1 CC(C)S(C)(=O)=O.N1(C(=O)NC)CCC(C=O)CC1.C1(C=O)CNC(=O)C1 C1(CNC(C(CSC)O)=O)CCCN(C(C2(C#N)CCCC2)=O)C1 C1(NC(=O)Cn2cccn2)CCCCC1NC(C1CC12CCCC2)=O C1(O)(CNC(C(CC)OC)=O)CCCN(C(c2ccc(C(N)=O)cn2)=O)C1 Cc1ncnc(C)c1OC(C1(C)C2CN(C(=O)OC(C)(C)C)CC12)=O c1(OC)cccc2scc(C(=O)NCC(C)NC(=O)CCC3CCN(C)CC3)c12 C1(NC(C(C)c2cncs2)=O)CCCCC1NC(=O)C=Cc1cccs1 c1(C(=O)NC2(C)CC(NC(C(CC)Oc3ccccc3)=O)C2)cccc(O)n1 c1(C(N2CCC(N(C(Cc3cn(C)nc3)=O)CCO)C2)=O)cnccc1C(F)F N=c1[nH]nc(CCCC(=O)NCC2CN(C(=O)C=CC3CCCC3)C2)s1 c1(CNC(C2CN(C(=O)C3CC3)CCC2O)=O)ccc(F)cc1C(F)(F)F C1(C(N2CC(C)(C)C(NC(=O)C)CC2)=O)Cc2c[nH]cc2S1(=O)=O.C(N)=O.N c1(C=O)ccc2nc(S)oc2c1.c1(CC)oc(C(=O)NCC2CC2)cc1C.C C1(O)(CN(C)C(C2(O)COC2)=O)CCCN(C(=O)C=CSc2ccccc2)C1 Cc1cc(F)c(C(N2CCC(NC(C3CC(F)(CO)C3)=O)C(C)C2)=O)cc1F CC1(NC(=O)C(c2cccnc2)NC(c2cnsn2)=O)CC(O)(CO)C1 C1(CNC(CC(CC)C2CC2)=O)C(C2CC2)CCN1c1nc(CC)ns1 C1CCC(C)(C)O1.C1(CCC=C)(C(=O)N)CN(C(=O)CN(C2CCCC2)C)C1 C12(NC(CNC(C)=O)=O)CCCCC1CN(C(c1ccccc1)=O)C2.C(N)=O.N C1(C)(NC(c2c(CC)cno2)=O)CCCCC1C(=O)NCC1=NOC(C)C1 c1(COc2cc(I)cc(OC)c2[N+](=O)[O-])cc([N+](=O)[O-])cc2ccccc12 c1(C(=O)NC2(C(N3CCC3C3CCCCC3)=O)CC2)coc2ccccc12 C1(CNC(C=C(C)C)=O)CN(C(c2ccc(CN3CCCC3)o2)=O)CC1C c1(CC)ccc(C(N2CC(CC(F)C(=O)N3CCC(CC4CC4)C3)C2)=O)o1 c1(OC)cc(O)ncc1C(N1CCCC1(C)C)=O.n1(CCC(=O)N)cnc(=N)[nH]1 O=C1COCC2(CN(C(C3CC(NC(C4(CF)CCOCC4)=O)C(O)C3)=O)C2)N1 C(=O)(NNC(=O)Cc1ccc(C#N)cc1)N(C1C(C)CCCC1)c1ccccc1 C1(NC(c2ccc(CC)[nH]2)=O)CN(C(c2ccnn(C)c2=O)=O)C(C)(C)C1 C1(NC(c2c(O)nc(=N)[nH]c2)=O)CC2CCC(C1)N2C(C1CCCCS1)=O C1(NC(C2CCC(CC)O2)=O)CCCN(C(c2ncc(C(C)(C)C)o2)C)C1 Cc1c(C(=O)N(C2CN(C(=O)C(C)C(C)(C)C)CC2O)C)cccc1Br C1(CNc2cccc(SCC)c2)CC2C=CC1CC2 CCCC(CNC(C1CCC1OCC)=O)C(=O)NCCC1CCOC1(C)C c1(C(=O)NC(C2CC=CCC2)C(=O)N(CCCC(C)O)C)cc(CO)ccn1 N1(C(C2(C#C)CC(=O)C2)=O)C2CCC1C(C(N1CCCC(CO)CC1)=O)C2 C1(C2CC2)(NC(CCC2CCCN(C(COC3(C)CCC3)=O)C2)=O)CCOC1 C(C)(CO)(C(=O)NCC1(NC(=O)C(N2CCOCC2)C)CC1)OC CC1CCC(C)(NC(C2OCCC2NC(=O)C(C)(C)O)=O)C1 C1(NC(=O)CCOC2CN(C(c3sccc3Cl)=O)C2)CC(O)(CO)C1 c1(C(C)(C)C(=O)NC(C(=O)O)C2(C)CC2)cc(Cl)ccc1F C(C)(C(C(=O)O)NC(C1CCC1(C)C(=O)O)=O)OC Nc1c(C(=O)NCC2CCC(NC(c3csnn3)=O)C2)cccc1Cl c1(CNC(=O)NCC2CC(OC)C2(C)C)ccc(Br)cc1Cl C(=O)(CCCCC(C)(C)C)N(C(CCNC(Cc1c(C)cco1)=O)C)C N1(C(CC2C(C)CCC2)=O)CC(CNC(C2CCCCC2)=O)C(F)(CO)C1 C1(NC(CCCOC)=O)CC2CC1N(C(C13CCC(C)(CO1)C3)=O)C2 Cc1c(C(=O)NCCC2(O)CCCN(C(=O)C=C3CCC3)C2)nn(C)c1N Nc1cc(C(NC2CCCc3cnccc32)=O)c2c(c1)OCCO2 C1(CNC(C(c2cnn(C)c2)NC(C(C)C)=O)=O)CC(C)(C)CCO1 N1(C(CC(CC)O)=O)CCC2(CCCN2C(c2ccc(N(C)C)cc2F)=O)CC1 c1(OC)cc(F)c(C(=O)NC)c(F)c1.C1CN(C(C2CCC(C)CC2)=O)CCO1 C(=O)(C1=CSCS1)NC1(C)CC(NC(C2CSCC(=O)N2)=O)C1 C1(C)(NC(Cc2c(C)nc(S)s2)=O)CCC(NC(=O)CCC2CCCN2C)CC1 c1(CC(=O)NC2CN(C(c3n[nH]cc3[N+](=O)[O-])=O)CC2(F)F)ccc(F)c(Br)c1 Cc1cc(C(N2CCC3(C2)CN(C(=O)C(C)(C)c2cnsc2)C3)=O)c(N)c(Cl)c1 c1(C(C)(C)C)cccc2c1OCC2C(=O)NCc1ccnc(N2CCOCC2)c1 C1(CCC(=O)N(CC(C)O)CCNC(c2cc(C)oc2)=O)CCN(C)CC1 c1(OCC)c(F)c(C=O)cc(F)c1F.C1(CC=O)CCC12CCC2.C1CC1.N NS(=O)(=O)c1n[nH]cc1C(N1CCCC(F)(CNC(C2CC2F)=O)C1)=O c1(OC)cccc(C(N2CC=CC(NC(c3ccc(CSC)o3)=O)C2)=O)c1 c1ccsc1C(N1CCCC1C1CC1)=O.c1(CC=O)nc[nH]n1.CC(=O)N.C Cc1ccc(C(C)C(=O)NC)o1.C1(C#N)(CCC(=O)N)CCC1.C1CCC1 Cn1ccc(CNC(=O)SC2(C)CCN2C(=O)OC(C)(C)C)n1 CC(C)C(F)C(=O)N1CC(O)CC1CNC(c1cn(C2COC2)nn1)=O C1(NC(C(F)=CC)=O)CCN(C(=O)Cc2cccc(COC)c2)CC1O CC1(F)CCCCN(C(C2CCC(CNC(=O)Cc3cn[nH]c3)O2)=O)C1 N1(C(CCCCC#C)=O)CCN(C(=O)Cn2ccc(Br)cc2=O)CCC1C Cc1cc(F)c(F)cc1C(=O)NC1CCCC1C(=O)Nc1ccc(Br)nc1C N1(C(C(CCC)n2cccc2)=O)CCN(C(=O)Oc2cccnc2C)CC1C#N c1(C(=O)NC2CCN(C(CSCCC)=O)C2C)nnc2ccccc2n1 CCC(C)CC(=O)C(=O)N1CCC(C(N2CC3CCC3(CO)C2)=O)O1 C1(C(C)NC(C(C2CC2)OCC)=O)CCN(C(=O)C(C)=CC2CC2)CC1 c1(OC)nc(N2CCCC2)c([Si](C)(C)C)cc1-c1ncccc1C(=O)NC1CC1 CCC(CC(F)(F)F)C(=O)N(CC(C)NC(C1(n2cnnn2)CCOCC1)=O)C N1(C(c2cc(-c3nc(C)sc3)oc2)=O)CCC(NC(=O)C(C)O)CC(C)(C)C1 C12(NC(c3cc(OC)cc(Cl)c3)=O)CCC(CC1)N(C(c1ccc(Cl)cn1)=O)C2 C1(c2c(N(CCOC(C)=O)C)c[nH]n2)CCCN(C(=O)OC2CCOC2C)C1 N1(C(C2C=CC(NC(C3CCC3)=O)C2)=O)CC2COCC2C1 N1(C(CCN(C(CC)CC)C)=O)CCC2(CC1)CCN(C(c1c[nH]c(=N)s1)=O)C2 C1(C)(CNC(C(CCCC)C)=O)COCCN(C(c2cc(C)c(F)cc2N)=O)C1 C1(C(C)C)(C(N2CCC(C(C)C(=O)NCCN(C)C)C2)=O)CCCC1 c1(OC(C(c2ccc(Br)c(Cl)c2)OC)=O)ccc(S(=O)(=O)NC2CC2)cc1 C1(NC(CC(=C=C)C)=O)CN(C(=O)CCN(CCCCC)C)CCC1C c1(OC)ccc(C(=O)NCC2(C)CCCN(C(C3CC3C)=O)C2)c(Cl)n1 C#Cc1cc(C(=O)NCCC(C)CCNC(C2(F)CC3(CCC3)C2)=O)ccc1C C1(C(=O)NCC(C)(C)OCC(N2C3COCC2C3)=O)CCCCCC1 CC1(C)CN(C(=O)CCCCNC(=O)C=CC2CC2)C1C1CC1 N1(C(CCc2cnn(C)n2)=O)CCCC2(NC(C3CCOC(C)(C)C3)=O)CC2C1 Cc1ccc(F)cc1S(=O)(=O)N1CCC2CN(C(c3ccncc3Br)=O)CC12 C(=O)(C(CC(F)F)NC(=O)CCCn1cncn1)N(CC(O)C1CC1)C C12(C(=O)NC(C)CCO)CC(CN1C(C1CN(C)C(=O)N1)=O)C2 C=C(F)C1(CC(=O)NCCC2CN(C(=O)C)CC(C)O2)CCOCC1.C(C)C.S N1(C(C2N(C(CCC(C)C)=O)CCC2O)=O)CC(C(N)=O)CCC1C c1(C(=O)NCC2(F)CN(C(C3(Cl)CC34CCC4)=O)C2)cc(CO)ccc1Cl N1(C(C2N(C(C(CC(C)C)=O)=O)CCCC2(C)C)=O)CC2CCC(C1)C2C#N N1(C(C2(C(CC)(F)F)CC2)=O)CC2(CCN(C(C3CC3F)=O)C2)C1 c1(C(=O)NC2CN(C(c3c(CC)c[nH]n3)=O)C(C)C2)c(Cl)nc2sc(C)cn12 C1(C(N(CCCNC(C(CCCOC)C)=O)C2CC2)=O)CC2OC(=O)OC2C1 N1(C(C(CN(CC)CC)F)=O)CCCC2CN(C(=O)Cn3cccn3)CC12 C1(C(=O)NC(c2c(C)nccn2)C)C2CCCC2CN1C(c1csc(Cl)n1)=O c1(N2CCC(OCC)C2)nc(=NC)[nH]c(=NCc2ccco2)[nH]1 c1(C=O)cc2cc(F)ccc2o1.C1(CC(=O)N(C(C)C2CC2)C)CC1(Cl)Cl.N Cc1cc(C)c(C(=O)NC)cn1.C12CC(CO1)C2.C1(C=O)CC(N(C)C)C1 C(C(=O)NC1CCCC1)(C1(OC)CCC1)N(CCOC)Cc1cccs1 N1(C(CC=C=C)=O)CC(C)CN(C(c2ccc(OC)c(Br)c2)=O)CC1C c1(OC)ccc(C(=O)NC2CN(C(=O)C3CC3)CC2c2nccn2C)nc1Cl N1(C(c2cnsc2)=O)CCC2(CC1)CN(C(C1CCC1F)=O)C2 N1(C(c2c(=N)[nH]cnc2)=O)C(CC(=O)NCC2CC3(CCC3)C2)C2CCCC12 C#Cc1ccc(OCC(N2CCC(N(C)C(C3C4CCC3CC4)=O)CC2)=O)cc1 N1(C(CCNC(C(C)N(C)C)=O)=O)CCC(C)C(C)(C)C1 N1(C(CN2CC(C)(OC)C2)=O)CCC(CF)(NC(=O)CC2COC(=O)C2)C1 C1(C(=O)NCC(C)OCC#C)CC12CCN(C(c1ccc(O)c(C)c1)=O)C2 N1(C(C2C(C(C)(F)F)C2)=O)CCC2C1CCCN2C(c1ccc(CF)cc1)=O c1(CC(C)NC(=O)CCN(CCCO)C(C2CNC(=O)C2)=O)cnn(C)c1 C(CCCCC(=O)NC(C1CC=CCC1)C(=O)N(C)CC)=CCCC N1(CC(N2C(C)C(C(F)(F)F)OCC2)=O)C(=O)c2cccc([N+](=O)[O-])c2C1=O C(=O)(C(CCF)NC(c1cncc(O)c1)=O)N(CCCC#C)C c1(CNC(C2CCCSC2)=O)nnc2n1CCN(C(c1cnc(C3CC3)s1)=O)C2 Cc1c(NC(=O)NCC2CCCN(CCc3ccccc3)C2)cccc1N N1(C(C(CC)O)=O)CCC(CCC(=O)NCC2CCOC2)CC1 c1(NC2CC(c3nccc(OC)c3)C2)cc(=NCC2CCCN(C)C2=O)[nH]cn1 C(=O)(C(CC(C)C)NC(C1CSCC(=O)N1)=O)N(CCCO)CC C1(CNC(CCC2CC(OC)C2)=O)CC2COCC2N1C(c1cnn(C)n1)=O c1(-c2cccc(CCC)c2)nc(C(CC)OC)nn1C1CCCc2ccccc21 CCCC(CC)CCC(=O)N1CCC(C)(C(N2CC(C)CC(C)(C)C2)=O)CC1 C(=O)(C(O)CCC(C)C)N1CC(NC(c2c(OCCOC)nccc2)=O)C1 Cc1nn(C)c(Cl)c1CC(=O)NC(CNC(c1cc(Cl)ns1)=O)CO C1(NC(C(CC2CC2)NC(C2(C#C)CCCC2)=O)=O)CN2CCC1(F)CC2 N1(C(COC2(C)CN(C(C3CCC(CC)CC3)=O)C2)=O)CCC(C)(C)CC1.O c1(C(N2CCC(C)(C(=O)NCc3c(C)nn(C)c3)CC2)=O)n[nH]c2c1CCCC2 N1(C(CCSCCCC)=O)CC(F)(F)CC1C(=O)NCCN(C)C1CC1 C12(C(=O)OC)CCC(C(=O)NCC(c3ccc(F)cc3)F)(COC1)C2 c1(OC)cc(C(=O)NC(CCNC(=O)CCCN=[N+]=[N-])C(C)C)cc(C)n1 c1(NC(C2N(C(C(CCC)OC)=O)CC2)=O)nc(-c2ccc(Cl)cc2)ncc1C Cn1ncc2nc[nH]c(=NC3CC(NC(c4cc(CO)on4)=O)C34CCC4)c12 c1(NCC2C(C(C)C)OCCC2)ccc(S(=O)(=O)NCc2sccc2Br)cc1Cl c1(C(=O)NC2CN(C(Cn3nnc(C)n3)=O)CC(F)C2)ccc2ncsc2c1 N1(C(C(C2CCCOC2)OC)=O)CCn2c(CNC(=O)CSC)nnc2C1 N1(CC(C)CC(F)(F)F)C(=O)CCN(CC2CS(=O)(=O)CCO2)C1=O N1(C(=O)CSCc2cccs2)CC2(CCN(C(c3ccc4sccc4c3)=O)C2)C1 CCC1=CCCCCC1.C1(CC(=O)NC(C2CC2C(=O)N)C)C=NN(C)C1=O N1(C(C(CC)n2ccnc2)=O)C(C(=O)N(CC(C)O)C)C2CC(O)C1C2.C1CC1 CC(C)C(O)C(F)(F)C(=O)NCC1CCC(NC(=O)C=CCO)CC1 Cc1c(C=O)cccc1[N+](=O)[O-].C12CCC(C=O)(CC1)C2.C(C1CC1)C1CC1 C(C(=O)N(CC1CCCCC1)OC)C1C(NC(C(CC#C)C2CC2)=O)CC1O c1(C(=O)NCC2C(NC(C(C)OCC)=O)CC2)c(C)ncnc1C C(=O)(C#CC1CCCCC1)N1CC2(CC(NC(c3c(C)n(C(C)C)nc3)=O)C2)C1 c1(C(=O)NC(CCCNC(CC=C)=O)CCC)cc(=O)c2cc(F)ccc2o1 N1(C(C(C)N(CC(=O)NC2(C)CCOC2)C)=O)CC(C)(OCC2CC2)C1 S(=O)(=O)(C1CN(C(=O)CCC2(C)CC2)C1)N1CCN(CC2C(C)CCCC2)CC1 c1(OC)ccc2[nH]cc(F)c(=Nc3ccccc3NS(C)(=O)=O)c2c1 c1(C(=O)OC)ccc(CC(=O)NC(CO)C(C)NC(C2CCSC2)=O)cc1 c1(C(=O)NCC)cccc(OCCC)c1.C1(C)C(C)(C)C1(C)C.C(=O)N c1(OC)ccc(C(=O)NC2CC(OCC(=O)NC3OCC3(C)C)C2)cc1 N1(C(CSCC(C)C)=O)CC(NC(C2CCCCC2O)=O)C(C2CC2)C1 c1(OC(CC)C)cc(C(=O)NCC(C(C)(C)C)NC(=O)C(C)O)ccn1 C1(C(=O)NCCCn2cc(C3N(C)CCC3)nn2)CC(S(C)(=O)=O)C1 CN1CCCN(C(=O)C(C(C)(C)O)NC(c2n[nH]c(O)n2)=O)CC1=O n1(C(C)C)nc(C2CC2)cc1C(N1CCCC1C1CC1)=O.C1(C=O)CCOC1.N S(=O)(=O)(c1ccc2[nH]c(=O)ccc2c1)N1CCCC(OCC#C)C1 Cc1ccnnc1C(=O)NC1CN(C(=O)C(CCN(C)C)N(C)C)CC1C c1(OC)cc(CN2CC3CC2CN3C(=O)CSC)cc(OC)c1OC C#Cc1cnn(C)c1C(N1CC(C(=O)NC2(C)CC(=C)C2)C(F)C1)=O c1(C(=O)NC(CC=C)C(=O)NC)nc(C)cc(Cl)c1OCC C1(NC(c2cc(CC)nn2C)=O)CCCCN(C(=O)C(C)(C)C2CCCCO2)C1 C(=O)C1=NOC(C)(C)C1.C1(COC)CCCN1C(=O)CC.[SH](C)(=O)=O.C CON(CCC(=O)NCC1(O)CCC(C)CC1)C(=O)C(C)(F)C(C)(C)F CCC(C)CCC(=O)NC1COCC1NC(c1cnn(C2COC2)c1)=O N1(CC)CCC(CO)C(c2ccccc2)C1.c12ccc(cc1)N(CC)C(=O)N2 C(CC)(CC(=O)N(CC(C)OCCOC)CC)NC(C(C)NCC)=O C=C(C)C(CC(=O)NC1(CNC(c2ccncc2C)=O)CCCCC1C)OCC c1nnc2n1CCN(C(C13CC(C)C1C3)=O)C2.CC(C(=O)NC)OC1CCCC1 CCC(CCCC(=O)NC(C1(CO)CC1)C)NC(=O)CCCC(OC)OC c1(C(=O)Nc2ncc(-c3c(C)noc3)cn2)cc(O)nc(O)n1 CC1(C)COCC(CC(=O)NCC2CC2NC(=O)C=CS)O1.c1ccco1.C C(CC(C(=O)N)NC(=O)Cc1cccc(F)c1)OCC.C1CCOC1C1CC1 C=C(C)CCC(=O)N1CCC(CCNC(=O)C(c2ccc(Br)s2)=O)CC1 c1(OC(C)C)ccccc1C(=O)N.C1(O)CN(C(=O)Cn2ccsc2=N)C1.C N1(C(CN(C)CC)=O)CCOC(C(=O)NC(c2ncc[nH]2)C)CC1 CC(O)CS(C)(=O)=NC(=O)c1coc(N2CCNCC2)n1 n1(CC=O)nc(C(F)F)cc1C.C1(OC)CN(C(=O)Cc2cc(Cl)cs2)C1.C Cc1nc(-c2ccccc2)sc1C(=O)NCC(O)CNC(=O)C(Cl)=CCl c1(C(=O)NC2CC(CCNC(COCCC=C)=O)C2)nccc2[nH]ccc12 N1(C(c2cccc(CNC(C3C(CC)OCC3)=O)n2)=O)CC(C)C(C)C1C N1(C(c2c(C)nc(-c3ncc[nH]3)s2)=O)CC2CC(NC(=O)CC(C)(C)C)C(C2)C1 C1(C(N(C2CCN(CC)C2)C)=O)CC(C)CCN1C(=O)Cn1cccn1 N1(C(Cc2c(C)noc2C)=O)CC2CC1CN(C(c1cc(Cl)cc(Cl)c1)=O)C2 C#CCCC(O)C(=O)NCc1csc(C(=O)OC)c1 c1(C(N(C2CCN(C(c3c(OC)c(C)sc3)=O)C2)C)=O)ccc2c(c1)CC(=O)N2 c1(C(=O)NC2CCCN(C(C3C(C)C3)=O)C2)ccnc(O)c1Br C(CCCC)(CC(=O)NOCC(=O)OC)NC(C(CC=C)CC)=O C1(OCC)CC2(C1)CC2C(N1CCC(C)C1)=O.C1(C)(C=O)CNC(=O)C1 Cc1ccn2cc(-c3nc(-c4nccs4)nn3CC3CCC3)nc2c1C c1(C(=O)NC2C(NC(=O)C=CCN3CCCC3)CC2)cc(C2CC2)ncn1 C12(CC(=O)NC(C(C)(C)C)c3ccccc3)CC3CC(CC(C3)C1)C2 c1(C(N(C(CNC(C2C(CC)OCC2)=O)C)C)=O)ccc([N+](=O)[O-])o1 C1(CNC(Cc2nc(CC)sc2)=O)CC2CCC1N2C(C1CC1(C)Br)=O Cc1ccc([N+](=O)[O-])c(OCCCNC(C2(n3cc(Br)cn3)CC2)=O)c1 C1(CC(=O)N(CC(C)CO)C)C2CCCC2N1C(=O)C(C)(O)C1CC1 Cn1cc(C(=O)NCCC2CN(C(c3csc([N+](=O)[O-])c3)=O)CCO2)ncc1=O C1(C(=O)Nc2ccc(OCC)cc2)CCC(C)N(C(=O)CC)C1.C(=O)CO.N c1(CN(C(C(C)N(C(C)=O)C)=O)C)ccccc1.C(c1cscn1)=CC=O.C N1(CC)CCCCC1C(=O)NC(C)CCNC(c1coc(C(C)(C)C)n1)=O N1(C(C2(OCC)CCCC2)=O)CCC(C)(C)C1.C(C1CCCN1C)=CC=O.N C1(CC)CCCCN(C(c2cc(CNC(C3CCOCC3(C)C)=O)on2)=O)C1 C(=O)(CCCS(C)(=O)=O)N1CCC(CNC(C(C)Cn2ccnc2)=O)C1 N1(C(c2cccc(C)c2C)=O)CCC2(C1)CN(C(C1C(C)(C)C1(C)C)=O)CCO2 CCC(CC)CCC(=O)NC(C1CCCC1)CNC(c1cnc(CC)nc1O)=O C1CC2(CCCCC2)C1.c1(C=O)ccc([N+](=O)[O-])[nH]1.CS(=O)(=O)NCC=O.N c1(C(N(CC(C)OC)C)=O)n[nH]c2c1CN(C(C1(C)CCC(C)CC1)=O)C2 C=CCC(C(=O)NC1CC=CCC1C(=O)NCCCC1C=NNC1=O)OC c1(OCC(N2CCN(Cc3cc(C)nc(C)c3)CC2)=O)cc(Br)cc(F)c1F c1(C=O)cncc(S(N)(=O)=O)c1.CC(C(=O)NC1CCOC1)S(N)(=O)=O.C c1(C(N(C(CNC(=O)C=CC2CC2)C2CC2)C)=O)cc(Cl)ccc1O C1(C(=O)NC2CC(OC)CN(C(COCC=C)=O)C2)CCn2ncnc2C1 CC(C)C(C)CCNC(c1ccnc(N(C)C)c1)c1nnnn1C(C)(C)C C(=O)(CC1=CCCC1)N.CC1CCN(C(=O)C(=O)N(CCC(C)C)C2CCC2)CC1 Cc1cccn2cc(C(=O)NC(C(C)NC(=O)Cn3ncnn3)C(C)C)nc12 CCCC(CC)CC(=O)N(CC)CC1CCCN1C(c1cnc(C(C)OC)s1)=O CN1CCc2[nH]nc(C(=O)NC3(C)CCN(C(C4CCS(=O)(=O)C4)=O)CC3)c2C1 Cc1nc2c(F)cccc2c(C(N2CCC3(C2)CN(C(=O)C(C)CF)C3)=O)c1O C1(NC(c2cnc(OCC)s2)=O)C2CCN(C(C3CCCC(O)C3)=O)CC12 CC#CCCC(=O)NC12COC(CNC(=O)CCn3nc(C)nc3C)(C1)C2 c1(CC(=O)N(CC=C)CC=C(C)Cl)cccc(C)c1.C(C)(C)C.C=O c1(CC(=O)N(C)CCOCC)ccc(Cl)c(F)c1.C1(C=O)SC2C=CC1C2 CC1=C(C(=O)NC(CNC(=O)CCCn2cccn2)CO)SCCO1 CC1CN(C(=O)C=Cc2cncc(O)c2)CCC1CNC(=O)CCc1ccsc1 Cn1nc(C(=O)NCC2CC2)c2c1CCCC2O.C1(C(=O)N)CC1(C)C(F)F CCC(CC(F)F)C(=O)N1CCN(C(C2(F)C(C)(C)C2(C)C)=O)CC1CO c1(C(N2CCC(O)(CNC(c3cc[nH]n3)=O)C2)=O)cccc(F)c1C1CC1 CC1(C)CCCC(C(=O)NCCCCC2CN(C(c3cc4ccsc4s3)=O)C2)C1 CC(CCC(C)(C)C)C(=O)N1CC2CC2C2CC12 C(CC(C)(C)CC(=O)NCC(CC1CC1)C(=O)N)OC.C1(CC)OCCC1(C)C c1(NC(C2=NOC(C)C2C)=O)nc2cc(C#N)ccc2n1C C(=O)(CCCCc1ccc(C(C)(C)C)cc1)NCCC(C)NC(=O)C1=CCOC1 Cc1ccc(NC(C2CC(N)C2)=O)c(C(F)(F)F)c1.c1ccc(C(=O)O)cn1 N1(C(CNC(CCC)=O)=O)CC2CCC1CN2C(C1CC(n2ccnn2)C1)=O c1(C(=O)NC(CCCNC(C(CCSC)O)=O)C)cc2c(C)cccn2c1 C(=O)(C#CC1CCCC1)N(C1CN(C(=O)CCCC2CCC2)CC12CC2)C N#Cc1cc(C(=O)NC2CC3CC(C2)N(C(c2ccoc2)=O)C3)ccc1[N+](=O)[O-] c1(C(C)N(C(=O)CC2CCCOC2)C)cn(CC(=O)O)nn1 c1(C=O)ccc(S(C)(=O)=O)c([N+](=O)[O-])c1.C1CCCC1.C(C=O)=CC=C.CC n1(CC)ccc(CC(N2CC(O)(c3cn(-c4ncc(C)s4)nn3)C2)=O)n1 C1(C(C)C)CC(NC(=O)C(CN(C)C)NC(=O)CC#N)CO1 CN1CCCCC1CC(=O)NC1(CC(=O)NC2CC(C#N)C2)CCCCC1 C(CC(C)(C)C(=O)NC(c1ccc(CNC(=O)C2=CCC2)cc1)C)SC C(CCC1CCC1)(C(=O)N1CCC(C=O)C1)NC(c1cc(COC)[nH]n1)=O Cn1ncc(=NC(=O)C2(C)CCCN2C(c2ccc(F)c(C#N)c2)=O)[nH]1 C1(CNC(CC=C)=O)CCC2(CO1)CC(NC(=O)C(c1ccccc1OC)O)C2 C1(C(=O)NCC2N(CC)CC2)CCC(CNC(=O)C(SC)SC)O1 c1(OC(C(=O)NCCC(C)NC(CC2(C=C)CC2)=O)C)cccc(Cl)c1 c1(N2CCN(C(CN(C)C)=O)CC2)ccc(S(=O)(=O)NC2COCC2O)cc1Cl CC(CC(=O)Nc1ccc(CO)cc1O)C(C)(C)NC(=O)CC1(C)CCOCC1 C(=O)(C(CC(N)=O)NC(=O)CSC(F)F)NCCCC(C)(F)F C(=O)(C(CNC(c1cc(C)c(N)cn1)=O)CC(C)C)N1CC(O)(COC)C1 C1(CC)CN(C(c2cc(C#N)c[nH]2)=O)CC1C(=O)NCc1cnc(C)cn1 CC1CN(c2nccc(Br)n2)CCN1C(c1cc(C(C)(C)C)ccc1O)=O N1(C(C(C(C)C)C(C)NC(c2ncn(C)n2)=O)=O)CCC2(COC(=O)N2)C1 Cc1cc(C(=O)NC(c2cncnc2)C)c(C)n1-c1cnccn1 N1(C(CCC(CCCC)O)=O)CCC2CC(NC(=O)C=CCO)CCC2C1 N1(C(C=C(C)c2cccnc2)=O)CCC(C2(NC(=O)CN(C3CCC3)C)CC2)C1 C(=O)(C1CCCc2nncn21)N(CCCCNC(C(C(CC)CC)OC)=O)C C(=O)(C(CS(=O)(=O)c1ccccc1)N1CC23CCC2(COC3)C1)NCCOC [N-]=[N+]=NC1CNC(C(N2CCN(CC3CCCC3)CC2)=O)C1 C1(CCC(=O)N(CCCCCNC(c2ccoc2)=O)C)CCCC(O)C1 Cc1cc(C(=O)NC2CCN(C(c3cc(C)sn3)=O)C(C)C2)nc(C(F)(F)F)n1 c1(C(=O)NCCCNC(C2(C)CC3CCC2O3)=O)cc2cc(Cl)cc(Cl)c2[nH]1 C1(NC(C2CCC(NC(CC)=O)C2)=O)CCN(C(=O)CC(CC)SC)C(C)C1 N1(C(C=C=C(C)C)=O)CCOC(C(=O)NCCc2cncc(C)n2)CC1 c1(OC)cc(CNC(C2CC(C)N2C(=O)CCn2cncn2)=O)ccn1 C1(C(N2CCC(N(C(CCC=C(C)C)=O)CCO)CC2)=O)CCCC(F)(F)C1 C1(NC(C2C(C(=O)OC)C2)=O)(CF)CN(C(C2COCCO2)=O)C1 Cc1cc(=O)n(C)cc1C(=O)NC12CCN(C(c3cnc4n3CCC4)=O)CC1C2 C12(NC(C(C=C)OC)=O)CCC1CN(C(C1(C3CCCO3)CCC1)=O)C2 c1(C(=O)NCC(CCCC)NC(=O)C#CC2(CC)CC2)nc(C(C)C)ncc1Cl c1(C(=O)NC(C2CCCN(C(CCOC(C)=O)=O)C2)C)ncc(F)cc1F C1(CNC(COCCCCCC)=O)CCC2(CN(C(=O)C(CC)C(C)C)C2)O1 CC(C)C(O)CC(=O)NC(C)(C)CCC(=O)NCCNS(N)(=O)=O CCCCCCC(C)(CC)C(=O)N1CC2CCCC(C1)N2c1ccc(C#N)nn1 C=C(Br)CC(C)(C)C(=O)N(CCCNC(=O)COc1ccc(CC)cc1)C c1(CC(C(=O)O)NC(C(c2ccc(Br)c(Cl)c2)C)=O)cc(Cl)ccc1Cl N1(C(C2CC(C)(F)C2)=O)CCOC(C2CN(C(=O)CC3CC3)C2)C1.C1CC1.N C(=O)CCC(C)C.C1(C(=O)NCc2cc(CC)n[nH]2)(C)CC(C)(C)C1.N Cc1cc(C(N2CC(NC(=O)CCOC3COC3)C(C)(C)C2)=O)c(C)cn1 c1(OC)ccc(C(=O)NCC2=CCCN(C(c3ccc(CO)o3)=O)C2)c(C)n1 C(=O)(C1=C(F)CN(C(C2CSC2)=O)CC1)NC(CC(C)O)C C1(C)(C(=O)NCCCNC(c2c(C)onc2-c2ccncc2)=O)CCNC(=O)C1 C1(NC(C2CSCCS2)=O)CC2CC1CN(C(=O)CCOCC1CCC1)C2 C(=O)(C1=CCCC1C)N(C)CC1(O)CN(C(C2CCN(CC)C2)=O)C1 c1(C(N2C(C)CC(CNC(=O)Cc3ncccc3F)C2)=O)ccc(N)c(O)c1 CCC(F)(C(=O)OC)C(=O)NC1CCN(C(c2ccon2)=O)C(C)C1 C1(CCOC)(NC(=O)Cc2cn[nH]c2)CCN(C(=O)CC2CCOC2=O)C1 C=CC(C)(CC)C(=O)NCC1C(O)C(O)CN1C(=O)CCn1cccnc1=O Cc1cc(CNC(=O)NC2C=C(C#N)CC2)ncn1 C(=O)(CS(=O)(=O)CCO)NC(CC(C)NC(C1(CC#C)CCCCO1)=O)C c1(CN(C)C)cnn(Cc2cccc(OC)c2)c1CC.N1(CCC)CCCC1 C1(C(N(CCCC)C(C)CC)=O)CCOCC1NC(=O)CN1C(=O)CCC1=O C=CCCCC(CNc1nc(CC)cc(SC)n1)c1ccccc1 C(=O)(C(C)C(F)F)N1C(C(=O)NC2(C(=O)OC)CC2)CC1 N1(C(C(COC)(F)F)=O)CC2CC(NC(c3cc(C(F)F)ccc3Cl)=O)CC1C2 c1(NC2CN(C(CCOCc3ccc(C)cc3)=O)C(C)C2)cc(C)nc(C)n1 N#CC1(c2cccc(Cl)c2)CCN(C(c2ccc(C(F)(F)F)c(I)c2Cl)=O)CC1 c1(CC=O)ccccc1S(N)(=O)=O.C(=O)(CCSC(F)(F)F)N(CCC)CC N1(C(c2c(OC)n[nH]c2)=O)CCN(C(=O)CC(O)C(C)C)C(CSC)C1 Cc1ccc(-c2cncnc2NC(=O)C(Cc2ccccc2)C2CCCC2)cc1 Cc1cc(C(C)C(=O)NCC(C)(O)CNC(=O)CSC(F)F)cc(F)c1 C(C(C)(O)CC(=O)N1CCCC1CN(C(=O)CCC(C)(F)F)C)OC CC1(C)NC(=O)CCC1NC(C1CCN1C(=O)C=Cc1cocn1)=O C1(C(=O)N)CNC(=O)CC12CCC2.N1(C(C=C(C)C(F)F)=O)CC(C)CC1(C)C C1(NC(CC(C)c2ccco2)=O)CCC(C)N(C(c2ccc([N+](=O)[O-])[nH]2)=O)C1 C(=O)(N=c1ccn(CCc2ccncc2)[nH]1)NC1C(C)CN(C2CC2)C1 c1(C(C(=O)NCc2ccco2)N(C(CC)(C)C)C)cc(Cl)cc(OC)c1OC N1(C(c2n(CC=C)ccc2)=O)CCOCC1CNC(c1ccsc1C(F)F)=O Cc1cc(C)n(CC(N2CC(=O)CC2C(=O)NCCC2CCN(C)C2)=O)n1 C1(CNC(c2n(CC=C)ccc2)=O)CCCC2(CN(C(c3ccoc3Cl)=O)C2)O1 c1(C2(C=O)CC2)ccccc1.C1(C)C(=O)N(C)CCN1C.C1(O)(C)CNC1 CC1CCCC(C(N2CCC2C(=O)Nc2ccc(NC(=O)C(C)C)nc2)=O)C1 C1(N(C(CC2(OC)CCOCC2)=O)C)CCN(C(C2(C(N)=O)CC2)=O)CC12CC2 C1(CC=C)(NC(=O)CCCC2CCC2)CCN(C(c2cccc(C(F)F)c2)=O)C1 C=CC1(CC(=O)NC2(CCO)CCCCC2)CN(C(c2nccs2)=O)C1 c1(C(=O)NCC(C)N(C(CC(=C)C)=O)C)cn(-c2ccccc2)nc1C N1(C(C2(C(=O)OCC)CCCC2=O)=O)CC(OC)C(C2CCCC2)C1 C1(C#N)(CC(N2CCC(N(C(C3CCCCC3F)=O)CC)CC2)=O)CCCCC1 c1(C(=O)NCCN(C(c2c(OC)nccc2)=O)C(C)C)sc2nccnc2c1N C1(F)CCN(C(C2(C)CC(C)=NO2)=O)C1.C1(C(F)(F)C=O)(OC)CCCC1.N C1(NC(CCc2onc(CC)n2)=O)CN(C(=O)CCOC(C)=O)CC1F N1(C(C(C)(C)CC2CC2)=O)CCC2C(C1)CN2C(c1cc(Cl)ns1)=O Cc1cc(CC(=O)NC(C2(O)CN(C(=O)CCC3CCC3)C2)C)n[nH]1 c1(C(=O)NC2C(NC(=O)Cc3ccncc3Cl)C2)ccc(Br)c(O)n1 C1(C(N2C3(CN)CC(CC2)C3)=O)NCCC12CCCC2 N1(C(c2c(C)nc(CO)nc2)=O)CC2CCCC2(N=c2[nH]ccn3nnnc23)C1 c1(CNC(COCC(C)C)=O)nn(C)c2c1CN(C(C1CC3CC3C1)=O)CC2 Cc1cncnc1C(=O)N(CCC(=O)NC(C)Cc1nccn1C)C c1(NC(C2OCC(C)C2)=O)ccc(-n2cc(-c3ccc(CO)nc3)nn2)cc1 N1(C(C(C)OCC=C)=O)CCCN(C(=O)CN2CCN(C)C(=O)C2)C(C)C1 Cc1cc(C(=O)Nc2ccnn2Cc2ccc(F)cc2)cc2nn[nH]c12 N1(C(c2c(C)n(C)nn2)=O)CCC(CNC(=O)COCC2CCOC2)CC1C N1(c2cc(OC)ncn2)CCS(=O)(=O)C(CCOC(=O)C(C)O)C1 C1(NC(c2n(C(C)(C)C)nnn2)(C)CCC2CC2)CCC(C(F)F)CC1 c1(OC)ccc(C(=O)NC(C)CC(C)Nc2nccc(CC#N)n2)cc1 C(=O)(C(C)CCC(C)(C)C)NC(COC)C(=O)NCCC12CCCC1C2 S(=O)(=O)(c1c[nH]c(C(=O)N(C2CCCN(C(c3cn(C)cn3)=O)C2)C)c1)NC N1(C(C(C)CN(C)C(C2CCNC2=O)=O)=O)CC(F)(F)C(F)(F)C1 c1(C(=O)NC(C2CCN(C(=O)COCC(F)(F)F)C2)C)ccc(O)nn1 Cc1[nH]nc(C(=O)NCC2CCCC2NC(c2cocn2)=O)c1O C(=O)(C(F)CC(C)(C)C)N1CC(CCC)N(C(c2cccc3oncc23)=O)CC1 C1(CCC)CN(C(C23CC(C)(CO2)C3)=O)CCN1C(c1cc([N+](=O)[O-])n[nH]1)=O CCN=C(NCCOc1cccc2ccccc12)N1CCN(C)C(C(C)C)C1 c1(CC)cccc(C(=O)N(C(C)CN(C)C(c2cc(C(N)=O)[nH]n2)=O)C)c1F C(C(F)(F)F)(C1CC1)CCC1CN(CC(n2cc(Cc3ccccc3)nn2)C)C1 C(CCC(=O)N(CC(C)N(C)C(C)=O)C)=CC.c1(CC(=O)N)csc(C)n1 CC1CC(C)(C)CCC1NC(c1cc(CNC(=O)O)on1)=O.C(C)(C)C c1(OCC)ccccc1CCC(=O)NCC12CC1CN(C(C1CCC1C)=O)C2 C(c1cc(Cl)cc(Cl)c1)=CC=O.c1(CC)c(C(N2CC3CC2C3)=O)ccn1C.C N1(C(CCC(=O)Nc2ccc(CO)cc2)=O)CC(C(N2CC(O)C2)=O)CC(F)C1 C(=O)(CCCCCNC(=O)Cc1cccnc1)Nc1c(CC)nccc1 C12(NC(c3cc4ccccn4n3)=O)CCCN(C(=O)COC3COC3)CC1C2 N1(C(CCCSC)=O)CC(CNC(C2(N3CCOC3=O)CC2)=O)C(O)C1 C=CCC(C)C(=O)N1CCC(CCNC(c2cn(CC=C)nn2)=O)CC1 C(=O)(C1=CCCS1)N1CC(CCCCNC(c2ccc(C3CCCO3)[nH]2)=O)C1 O=C1NC2CCCC1CN(c1nccc(=NCc3cccc(F)c3)[nH]1)C2 N1(C(c2c(C)con2)=O)CCN(C(c2cc3cnccc3o2)=O)C(C)C1C C1(NC(C(CC)CC)=O)CC2CC(NC(c3cnnn3C(C)C)=O)C2C1 N1(C(c2cc(CNC(c3c(C(C)C)ocn3)=O)nn2C)=O)CC(C)OCCC1C C1(NC(CNC(C)=O)=O)CC2CCCC12.c1(C(=O)N)cc(C)n(C2CC2)n1 C1(C(C)O)CCN(C(=O)C(N2CCN(CC(O)C3CC3)CC2)=O)CC1 C(=O)(CC(C)(C)C(=O)OC)NC(CC#C)CC(=O)NCC(C)(C)CSC C1(F)(C(=O)NCCCN(C(=O)CS)C(C)C)CCOC1C.c1ccc(Cl)cc1 C(=O)(CC(C)CC(C)(C)C)NCCC1N(c2nnc(C(C)C)o2)CCC1 N=c1[nH]c(C(=O)NCC=CC(N2CC(n3cnnn3)C2)=O)cs1 c1(C(C)C)cccc(Cl)c1NC(N1CCCN(C(=O)C(C)(C)C)CC1)=O c1(C(N=c2cc(C)o[nH]2)=O)cc2ccc(-c3ccc4c(c3)CC4)cn2c1 Cc1nn(C)nc1C(=O)NC(C1CC(NC(c2cccnc2)=O)C1)C C1(C(=O)NC2(C(F)F)CC(NC(CCC#C)=O)C2)C2CCCCC12 C1(C(N2CCC(C)(NC(C3(n4cnnn4)CC3)=O)C2)=O)CCCC2(C1)CC2(F)F CN1CCN(CCNC(C2CC(=O)N(C3CCC3)C2)=O)C(c2ccccc2)C1 C1(C(N2CCC(N(C(CC(C)O)=O)C)C2)=O)(OCc2ccccc2)CCOCC1 N1(C(CSCCCC)=O)CC2CCC2(CC(=O)N(C)Cc2cnc[nH]2)C1 c1(OC)ccc(C(=O)N(C(C)CCNC(=O)CCCCCSC)C)c2sccc12 CCC(C)(CNC(=O)CC1CC1)CC.C1(N(CCC=O)C)CC(C#N)C1.C Cc1c(C(N2CCCC(CNC(c3cccc(Cl)c3)=O)C2)=O)c(C(F)F)nn1C Cc1cc(C(=O)NC(C)(C)CNC(c2csc(-c3ccccc3)n2)=O)ccn1 C1(COC)(NC(C2CCCC(C)C2)=O)CCN(c2nccc(C(C)(C)C)n2)CC1 N1(C(c2noc(CC)c2C)=O)CC2CCC(C1)N2C(=O)CCC(CC)OC c1(CC(C(N2CC3C(CNC(C=CCC)=O)(C3)C2)=O)C)ccc(C#N)cc1 c1(C(=O)NCC2(F)CCN(C(CCc3nc(C)c(C)o3)=O)C2)cccc(F)c1F c1(C(=O)NCc2scc(CNC(C(CC)C)=O)n2)scc(C)c1OC c1(C(=O)NCC(CC)(CC)NC(=O)C(CCO)N(C)C)c(C)cccc1[N+](=O)[O-] CC(C)(CC#N)C(=O)N1CCC(NC(C23CC2CCC3(F)F)=O)C(O)C1 C1(C(C)(C)C)CCN(C(c2c[nH]c(=N)s2)=O)C1.C(C)(C(=O)N)OCC=C N1(C(C2CN(C(C)=O)C2)=O)CC2CCCC1C2.C(=O)C1=NNC(C(F)(F)F)C1.N c1(NCC=CCNC(CC2CC(C)(C)OC2)=O)ncc2c(n1)COC2 C1(CNC(=O)Cc2cnc[nH]2)CCN(C(=O)CCc2cccc(Cl)c2)CC1CO C1(CCCNC(C=C(C)CNC(=O)COc2ccccc2)=O)CCOC1=O CC(C)CC(C)C(=O)N(C)CC1(O)CN(C(c2cc(Br)n[nH]2)=O)C1 C12(C(=O)NCC(CO)NC(c3cccc(C(C)=O)c3)=O)CCC(CC1F)C2 C(=O)(C1Cc2c(Cl)cccc21)N1CC(N(C(CC=C)=O)C)C2(C1)CC2 c1(C(=O)NCC(C2CCN(C(C(CC#C)(C)C)=O)CC2)F)noc2c1CCCC2 c1(C(N(CCNC(=O)C(F)C(C)C)CC)=O)ccc2c(c1)CCOC2(C)C C1(C(=O)NCCCn2ccnc2)CCN(C(=O)c2cnc(S)nc2)O1 C(=O)(CC(F)(F)C(F)F)N1CC(NC(Cn2cnc(=N)[nH]2)=O)(CF)C1 C1(C(C)(C)O)(CNC(=O)CCc2ccc[nH]2)CN(C(C23CCC2C3)=O)C1 CC(C)CS(=O)(=O)CCC(=O)N1CCCC(C)(NC(=O)Cn2nnc(=O)[nH]2)C1 C(=O)(CS(=O)CC)N(CCNC(C(CC)OCC)=O)C N1(C(CCC2CC(NC(C3(CC#C)CCCO3)=O)C2)=O)CCN2CC(F)CC2C1 CC(C)C(C(=O)N1CC(C)(CO)C1)C(C)NC(=O)C=C1CCCCC1 N1(C(C2CCCN(C(C)=O)C2)=O)CCOCC(NC(=O)CCOC(C)=O)C1 C1(C)(C(N(C2CCC(NC(=O)CS)CC2)C)=O)CCC(=O)NC1.c1ncc[nH]1 N1(C(c2c(C)n(C)nn2)=O)CCC(C(N2CCOC3(CC3)C2)=O)C(C)C1 C(=O)(CCCCCCCCC1CC1)NC1Cc2n(C(C)C)ncc2CC1 C1(Sc2ccccc2)CCN(C(=NCCCc2nc[nH]n2)NCc2cccs2)C1 C1(CNC(C(CC)CN(C)C)=O)C(C)CCCN1C(c1ccc(F)cc1C)=O C1(C(=O)NC(C#C)(C)C2CCOC2)CCN(C(=O)C2CCOC2C(C)C)O1 Cc1cc(C(N2CCC3(CC3C(=O)NC3CCC=CCC3)C2)=O)cc(F)c1 c1(C(=O)NC2CCN(C(c3n(C(C)C)nnc3)=O)C2)ccc2cnoc2c1 c1(NC(N2CCCC(O)(C(F)(F)F)C2)=O)ccc2c(c1)OCC2 CON(C)CCCNC(C1(C)C=CCN1C(=O)CO)=O c1(C(=O)NCC2CCC(NC(C3CCCC(=O)O3)=O)C2)cc2occc2s1 CCC(O)CCCN=c1ccc(S(=O)(=O)NCC(C(C)C)OC)c[nH]1 C#CCCCC(C)C(=O)NCC(CC(C)C)NC(=O)CCNC(c1ccco1)=O N1(C(C(C=C=C)C)=O)CC2=C(C1)CN(C(c1ccc(Cl)c(F)c1F)=O)C2 C1(NC(C(CC)C)=O)CC2CCC(C1)N2C(c1cccc(Br)c1F)=O CCC(C)C(C(=O)NC1CC2CN(C(c3cnoc3C3CC3)=O)CC12)OC C#Cc1cnc(N2CC(NC(=O)C=Cc3ccccc3)CCC2C)nc1 c1(OCC)cc(CCCNC(=O)COc2ccccc2C(F)F)ccc1F c1(C(=O)NC(C2CCCN2C(C2CC2F)=O)C)cc(OCF)cc(F)c1 c1(C(=O)NCC23C(CN(C(c4cc(C)cc(N)c4)=O)C2)C3)cc2c(ncn2C)[nH]1 c1(C(=O)NCC2CCN(C(C3CCC3CF)=O)CC2)n[nH]c2c1COC2 N1(C(=O)CC(c2ccc(F)cc2)O)CCC2(C1)CN(C(C1CC=CC1)=O)CCO2 C(=O)(CCC(=O)NC1(C)CCC1)NCCCOC.c1(C=O)ccnn1CC Cc1nc(=NC2(CNC(=O)C3CCCn4nccc43)CCC2)s[nH]1 c1(CC=O)cnn(C2CCCC2)c1.C(C(=O)N1CCC1)(C1CCC1)OCC.C c1(OC)cc(C(N2CCCCC2CCNC(=O)CC2CC2)=O)c(N)c(Br)c1 c1(C(=O)NCC2CC(C(F)(F)F)CN(c3ccncn3)C2)cnc2cc[nH]c2c1 C1(C(=O)NC(c2nc(C)no2)CO)(CC)CCCN(C(C2CN3CCC2C3)=O)C1 c1(C(=O)NCCC(C)NC(C2Cc3cccnc3C2)=O)nccc2ncccc12 C(CN(C(=O)Cc1nccn1C)C)(CO)(CO)NC(COCCCOC)=O Cc1nccn2c(C(=O)NNC(=O)c3ccccc3Cl)cnc12 c1(C(c2ccccc2)=O)ccccc1NC(C1CC2(C1)N=N2)=O c1(CCC(=O)NCC#CCNC2CCN(C(CC)=O)C2)cccc(C(=O)OC)n1 c1(OC)ccc(C(=O)NCCCOCCNC(C2COC(C)CO2)=O)cc1Cl C1(CNC(C(CC)N(C)C)=O)C(C)CCCN1C(c1scnc1C)=O.C1CC1.C c1(C(CNC(=O)C=C(C)Cl)NC(CCC=C)=O)ccc(Br)cc1 c1(C(=O)NCC(CC=C)NC(C2CC(=O)NC2)=O)cc(F)ccc1C.C1CC1 CC1CN(C2CC3CCC(C2)N3C(c2ccc(O)cc2)=O)CCC1(O)C(F)(F)F Cn1ncc2c1CC(C(=O)Nc1cnc3n1CCNC3)C(C(F)(F)F)N2 C(=O)(C(C)(C)CCNC(C1C2CC(=O)CC12)=O)NCC(C(CC)C)O C(N=C(NCC(F)F)N1CCC(NC(=O)NCC2CC2)C1)c1c(C)noc1 C1(OC)CCC(N=c2[nH]c3c(c(=NCCc4c[nH]c(=N)s4)[nH]2)CSC3)C1 C(=O)(C1=CSCCO1)NCC1N(C(COC(CC)(C)C)=O)CCOC1 C1(C(C)C)CC(NC(=O)C(C)NC(C2(O)CCOC2)=O)CO1 c1(C(N2CC(O)(CNC(c3cc(C)c(C)s3)=O)C2)=O)ccc(OC(F)F)nc1Cl C1(Nc2cc(NC(CF)CF)nc(C)n2)CCOC2(CCS(=O)(=O)CC2)C1 Cc1cc(C(=O)NC2CC(NC(=O)CN3CC4CC4C3)C2)n2nc(C)cc2n1 c1(NC(C23CC(NC(c4ccccc4CO)=O)(C2)C3)=O)ccc(Br)cc1O n1(C(CC)C)ncc(C(=O)NCC2CC2(C)C)c1-n1cc(CCNC)nn1 C(CCC(=O)NC(C)C(c1ccccc1)NC(c1c[nH]cc1C)=O)N(C(C)=O)C c1(C(=O)NCC2(O)CN(C(C3C(C(C)C)OCC3)=O)C2)ccn2ncnc2c1 C=C(Br)CCC(=O)NC1CN(C(c2ccc(-c3ccco3)[nH]2)=O)CC1C C1(C)(C(NCCN2CCCC2)=O)CCCN(C(c2ccc(C)c(F)c2)=O)C1.CC c1(C(N2CC(OCC)(CNC(=O)CC3CCCC3C)C2)=O)ccccc1.O c1(C(C)=O)cc(C(N2C3CCC2(CNC(c2cc(C)cs2)=O)CC3)=O)ccc1O c1(C(N2CC(CC(C)NC(c3n[nH]c(O)n3)=O)C2)=O)ccn2nncc2c1 N1(C(C(C)(C)CF)=O)CC2CN(C(C34CCC(CF)(CC3)CC4)=O)CC2C1 c1(CN2CCCC(CC(=O)Nc3c(C)n[nH]c3)C2)ccc(F)c(C)c1F N1(C(c2c(C)nc(CC)s2)=O)CCC2CCCC12.c1(C(=O)N)cn(C)c(=O)n1C C12(C(=O)Nc3c(C)cccc3C)CCCC1N(C(C1CC=CC1)=O)CC2 N1(C(C=C(COC)C)=O)CCC(N=[N+]=[N-])C1.C1(C)(C(=O)N)CCC(C)C1(C)C N1(C(C2C(C(=O)N)C2)=O)CC2OCCC2C1.C1(C=O)CCC2(CC2)C1.CCO C1(NC(C(CC)C)=O)CCN(C(=O)Cc2occc2C)CC(O)C1 O=C(C1OCCn2ccnc21)NC1CCCN(C(C2CN(C3CCC3)C2)=O)C1 c1(CCC(=O)NCC2C(CNC(C3C(=C)CC3)=O)C2)ccc(F)cc1F N1(C(CC(CNC(C2CC2(C)C)=O)OC)=O)CC2CC(O)CC1C2 c1(C(N2C(C)CC(CNC(c3ccc(F)o3)=O)C2)=O)cnn2ccccc12 Cc1ccc(N2CCC3(C2)CC3(F)F)c(S(C)(=O)=O)c1 N1(C(Cc2ccc(OCC)cn2)=O)CC(C)(C)OCC1C.C1(C=O)CCCS1.N c1(N(CCCCCC)C)cc(N2CCCC(CN(C)C(C)C)C2)nc(C(C)C)n1 Cc1nsc2ncc(-c3nc(CCC(C)C)nn3Cc3ccncc3)cc12 CCCC(C)CC(=O)NCC1(OC)CN(C(C2CN3CCC2CC3)=O)C1 c1(C(=O)OC)ccc(=NCC(C)NC(=O)CC23COC(C)(C2)C3)[nH]c1 c1(CCC)nc(C(=O)N(C(C)CCNC(c2cscc2SC)=O)C)co1 C1(C(=O)NCC(=O)NCC(CC)NC(C2(C)CC2(C)C)=O)CCOCC1 C(=O)(CC(C)CNC(c1cc(C2CC2)on1)=O)N(C1CCN(C)C1)CCC CC1CN(C(c2cc(C3CC3)no2)=O)CCC1CNC(C1CC2(C1)CC2F)=O N1(C(=O)CC2CCN(C(C3CC34CCOC4)=O)C2)CC(O)C2(CCCC2)C1 c1(CNC(C(CC)C)=O)ccc(CNC(=O)CC2CC=CCC2)cc1 CC(CN(C)C)CN=c1nc(N2CCC(C3CCOC3)CC2)c2c([nH]1)CCC2 c1(C(N2C(CNC(CCCN(C(C)=O)C)=O)CCC2)=O)sc(C(C)C)nc1C CS(=O)(=O)C1CCCCN(C(=O)CCC(F)(F)C(F)(F)F)C1 C(C1CC1)(C1CC1)=CC(=O)N.c1(C(C)C)cc(C(=O)NC(C)CCC)on1 CC1(NC(=O)COc2ccc(F)nc2)CCN(C(=O)Cn2cnccc2=O)C1 Cn1c(O)ncc(C(=O)NC23CC2CN(C(c2sccc2SC(F)F)=O)C3)c1=O C1CN(C(=O)Cn2cc(Cl)c(C)n2)C2(CCC2)C1.C(=O)(C(C)C(=O)N)OC c1(C(N2CCN(C(C3C(C)OCC3)=O)CC2)=O)ccc(S(N)(=O)=O)c(F)c1 N1(C(C(CCCC)(C)F)=O)CC2(C1)CN(C(C13CC4CC(CC1C4)C3)=O)CCO2 N1(C(c2n(C)ncc2)=O)CCN(C(=O)CCC(C)(F)F)CC1CC(F)(F)F CON(CCC(=O)N1CCN(C(C)(C)C)CC1)C(=O)C(F)C1CCOC1 C#Cc1cc(F)c(C(=O)NC2CC(NC(c3conc3CC)=O)C2)cc1F c1(OCC)c(Cl)cc(NC(=O)C(c2cnn(C)c2)C)cc1Cl C12(C(N3C4CC(CCC4)C3)=O)CC3CC(C(=O)N1)C2C3.C(C=O)(C(C)C)SC Cc1ccc2occ(C(=O)NCC3(F)CCC3)c2c1.C(=O)CCCS(C)(=O)=O.N Cc1ncc(C(N2CCC(NC(=O)CC3CCCCC3)C(CO)C2)=O)cc1C#N c1(C(N)=O)c(F)cc(CNCc2ccc(-c3cc(Cl)c(F)cc3F)s2)cc1F c1(C=O)cc2c(Cl)c(F)ccc2[nH]1.CC(CC(=O)NCC1(CC)CC1)N(C)C C1(NC(C(C2CC(F)(F)C2)OC)=O)CCC2CCN(C(c3cnnn3C)=O)C12 CCCC(CCC)=CC(=O)N(C1CC1)CC1CCCN1C(=O)CCCOCC c1(NC(CC2N(C(C3(CC=C)CC=CC3)=O)CCC2)=O)ccccn1.C(C)C.O CC1(C)CCN(C(c2ccncc2F)=O)CC1CNC(=O)CC1(O)CCOCC1 c1(C(C)NC(=O)CNC(c2cc[nH]n2)=O)nn(C)cc1O CCCC(C(=O)N(CCCNC(c1noc(C2CC2)c1C)=O)C)OCC c1(C(=O)NCC2CC(C)NC2)n[nH]c2ccc(F)cc12 Cc1cc(Cl)cc2cc(C(=O)NCC3CC3C)[nH]c12.C1(C(=O)N)CSCCS1 CC(c1ccccc1OC(F)F)=CC(N1CCCC(c2ncc[nH]2)C1)=O C1(C(N2CC=CCC2)=O)C2CCC1(C)C2(C)C.n1(C(C)(C)C)cc(C(=O)N)nn1 c1(OC)ccc2[nH]c3c(c2c1)CN(Cc1ccc(-c2cncn2C)cn1)CC3 N1(C(CC(CN(C)C)C(F)F)=O)CCC2CN(C(C3(CCF)CCC3)=O)CC2C1 Cc1nnc2n1C(C(=O)N)CC2.c1(C(N(CC)C2CC2)=O)cc(O)c2sccc2c1 CC1(C(=O)NC2CCCC2)CC(C2CC2)=NO1.C12(CC=O)COC(C1)C2.N c1(C(=O)NC(C)(C)CCNC(=O)CC2CCOC2=O)ccccc1Cl c1(CC(N2CCC(C(N3CCC(C)(CN)C3)=O)CC2)C)ccc2c(c1)OCO2 N1(C(c2c(C=C)cnn2C)=O)CC(C)C2(CCC2)C1.c1(C(=O)N)cnc(C)n1C Cc1cc(N2CCC(NC(Cc3ccco3)CO)C2=O)n(C)n1 c1(N(C)CCC2CCCC2)nc(N2CCC(c3nc[nH]n3)C2)nc2c1cnn2C CC(C)C(C(=O)NCC(C)CN(C)C(C1(C)CCCNS1(=O)=O)=O)C(C)C O(N=C1CCCCCC1)CC(=O)NC1CN(C(C2CCC(=C)CC2)=O)C2C1C2 C1(CC=C)(C(=O)N(CC(C)(C)NC(C2(F)CCC2)=O)C)CCOCC1 C1(NC(=O)CC2C=CCC2)C2CCC1CN(C(=O)CCOCc1ccccc1)C2 C(=O)C(C)S(=O)(=O)C(C)C.C12(CC)CN(C(=O)CNC=O)C(C1)C2 C=CCC(C(=O)OCC)NC(C1CCCN(C(=O)C(C#N)CC)C1)=O c1(OC)cccc(Cl)c1CC(N1CC=CC(NC(=O)CCc2cnco2)C1)=O C(c1csc(C(F)(F)F)c1)=CC=O.c1(C(N(CC)C2CC2)=O)cncs1.N c1(CNc2ccc(OC)cc2C2CC2)cc(OC)c(N)c(Cl)c1 c1(C=O)cn(C)c(=O)n1C.c1(OC)ncccc1CC(=O)NCC(C)C(C)C.N CC(C(=O)NCC(C)(CO)NC(c1cc(-c2ccns2)on1)=O)C(F)(F)F c1(C(=O)NCC2(C(F)F)CCN(C(CCC(C)OC)=O)C2)ccc(Cl)cc1F C1(CC)OCCC1(C)C.c1(CNC(C(C2CC2)SC)=O)cc(C(=O)N)cs1 N1(CCNC(c2c(C)ccn2C)=O)CCCN(C(C2CC2CF)=O)CC1 CC(N=c1[nH]c(=N)[nH]c(=NCC2CCC(C)(C)O2)[nH]1)C1CCC1 c1(CC)nc(C)n(C)c1C(=O)NCC1CN(C(c2ccsc2)=O)CC1O c1(OCC=C)cccnc1CNC(=O)CC1CC1.C(C)(C)C.C=O.C c1(SC)ccc(Cl)c(C(=O)NC2(CNC(c3ncccn3)=O)CCOC2)c1 N1(CC(=O)N(C(c2cccs2)=O)C)CCC(OCCCO)CC1.c1cccnc1.O Cc1ncc(F)c(N2CC3CC3(CNC(=O)CCc3cccc(O)c3)C2)n1 C=C(Cl)C(C)(C)C(=O)N1CCCC(CN2CCN(C(=O)C(O)C(C)(C)C)CC2)C1 C1(CNC(C2CCN(CC)C2)=O)CCN(C(=O)CC2CC2)CC1(F)F C1(CCNC(CCN(C2CCOCC2)C)=O)CCN(C(C2(C)C=CCC2)=O)CC1 C1(C(N(C)CCOCC2CC2)=O)CC(O)CCN1C(c1ccc(F)cc1)=O Cc1cc(Br)ccc1C(C)NC1(c2ccc(OC(F)F)cc2)CCOC1 C(=O)(CCCCCCNC(C12CCOCC1C2)=O)N1CCC(C(=O)OC)C1 c1(OC)cnc(C(=O)N)cn1.C1CCC(C)N(C(=O)CNS(N)(=O)=O)C1.C C12(NC(C(C)NC(=O)CSC(F)(F)F)=O)CCC(CC1)C2(C)C CCN=c1[nH]c(C(N2CCC(C)(NC(C3C(C)(C)C3(F)F)=O)C2)=O)cs1 c1(C(=O)NCC(CN(C(Cc2c(C)scc2)=O)C)O)ccc2[nH]c(=N)oc2c1 Cc1ccc(CN(C(=O)C(=O)NCCc2sccc2Br)C)o1 c1(CNC(C2N(Cc3n(C)ccn3)CCSC2)=O)ccc(O)cc1Cl O=C1Cc2ccccc2N1CC(=O)N1CC(O)(CNC(C2CCSC2)=O)C1 c1(CN2C3CN(C(c4scc(CC)n4)=O)CC2CC3)c(OC)cccc1[N+](=O)[O-] O=C1CCCCC(C(N2CCCC2CC(=O)NCCCc2ccco2)=O)C1 C(=O)(C1CCCn2c(C)cnc21)N1C(CNC(c2n(CC)c(O)nc2)=O)CCC1 C1CCC=CO1.C(C=O)N(CC(=O)NCC)C(C1CC1)=O.C(C)(C)C.O c1(CC(=O)NCC2(NC(C=CC)=O)CC2)cccc([N+](=O)[O-])c1 N1(C(=O)O)CC(C(=O)N(CCC#CCO)CCO)OC(C(F)(F)F)C1.CC(C)C N1(C(C2C(=C)C2)=O)CCC(C(=O)NC2(COCC)CCCC2)CC1 N1(C(C2(OC)CCCOC2)=O)CCC2(CC1)CCN(C(=O)CCC(C)SC)C2 c1(C(C)C(=O)NC2CC(NC(=O)CCC3CCCN3C)C2)ccc2c(c1)OCO2 C1(C(=O)NCCC(C)N(C(c2ccc(SC)s2)=O)C)CCC(C)=C(C)C1 c1(C(=O)NC2CCC(CNC(=O)CC(O)C3CC3)CC2)cnc2c(c1)OCCN2 O=S(=O)(c1cnn(C2CCCCC2)c1)NC1(CN2CCOCC2)CCCCC1 N1(C(=O)CCN2CCOCC2)CCCC(CCCN2CCCCC2)C1 C1(C(=O)NCCC(CC)(CC)NC(=O)C(O)P(C)(C)=O)(OC)CCCCCC1 c1(CC(N2CC(C(=O)NCCc3ccsc3)OCC2)=O)ccc2c(c1)CCCC2 CCCS(=O)(=O)CC(=O)N1CC2C(CNC(c3cc(F)c(F)cc3O)=O)C2C1 Cc1cc(C(C)C(N2CCCCC(NC(c3cnccc3C)=O)C2)=O)cc(F)c1 CC1(C)CN(C(=O)C=C2CCCCC2)CCC1NC(C1CC12CC(F)(F)C2)=O C1(CNC(CC2CN(C(C)=O)C2)=O)C=CCC1.C(=O)(C(C)(O)C1CC1)N C1(C(N(C(CNC(C2CCC=CO2)=O)C2CC2)C)=O)CC12CCOC2 c1(C(=O)N)cc(F)cc2nn[nH]c12.N1(C(c2n(CC)ncn2)=O)CC(C)C(C)C1 C#Cc1ccc(C(=O)NC2CCN(C(=O)CC(C)(C)F)CC2CC)nc1 C1(CNC(C(C(C)O)N(C)C)=O)N(C(=O)C=Cc2cscn2)CCC1(C)C c1(COC(C)C)ccc(C(N2CCOCC2c2cnn(C)c2)=O)cc1 CS(=O)c1cccc(C(=O)NCCC2(CNC(=O)C3=CCCO3)CC2)c1 c1(C(N(C2CCC(NC(C3CCC3)=O)C2)C)=O)cc(F)cc2c1CCC2 C(C)(C)(CC(N)=O)NC(C(CC1CN(C(c2scc(C)c2)=O)C1)F)=O CC1CCOC1C(=O)NCCC1(CNC(c2nocc2Br)=O)CC1 c1(C(=O)NC2CN(C(c3cn(CCOC)nc3)=O)C(C)C2)cccn2nncc12 c1(C(=O)OCC)nc(Br)ccc1NC(=O)CSc1ccccc1SC c1(NC(C2C3(CCN(Cc4sc(C)c(Br)c4)C3)C2)=O)ncc(C#N)cc1I C1(NC(CC=C(C)C)=O)CCN(C2CCN(C(=O)C(C)O)C2)CC1 c1(C(N2CC(C=C)C(NC(c3cnsc3)=O)C2)=O)ccc2c(c1)COC2=O Cc1cc(C)n(CCNC(C)Cc2cc(-c3nn[nH]n3)no2)n1 CC1CCN(C(=O)CONC(=O)OC(C)(C)C)CC1.C(=O)CCn1cncn1.N C1(CNC(C2(OC)CCOC2)=O)CCCCN(C(=O)Cc2ccsc2C)C1 N1(c2ncc(CCC)cn2)CCC2(CCCN(C(=O)CN3CCOC3=O)C2)CC1 c1(C(=O)NC2CCN(C(=O)Cc3nc[nH]n3)CC2O)noc2ccc(F)cc12 Cc1nc2cc(NC(=O)CC3CN(C(c4ccc(F)nc4F)=O)C3)ccc2s1 C1(C(=O)NC2(CC#C)CCOCC2)COCCN(C(C2(C)COCCO2)=O)C1 Cn1cc(C(N2CCC3CCCC(C2)N3C(C2(C)CC2)=O)=O)n2cncc2c1=O C1(C(N(C2CCCC2)CCCNC(CC=CC)=O)=O)SC2C=CC1C2 c1(OC(C(COCC=C)NCC)=O)ccnc(N=[N+]=[N-])c1 c1(C(N2CC(N(C(C(CC)OC)=O)C)C3(C2)CC3)=O)ccc2c(c1)S(=O)(=O)NC2 C1(CC(=O)NCC2C(NC(CC=C)=O)COC2)CCC(C)(C)O1 C1(OC)(CNC(=O)CC2CCCC2O)CN(C(c2csc(O)n2)=O)C1 S(=O)(=O)(c1cc(F)cc(Br)c1)Nc1c(C(=O)OC)ccc(Br)n1 N1(C(c2c(OCC)scc2)=O)CCC2(NC(=O)C(C)OC)CCCC12 c1(-n2cc(-c3occn3)nn2)cccnc1N1CCCCC1 C(=O)(C#CC1CCOC1)N1C(CCN(C(c2nc(CC)sc2N)=O)C)CCCC1 N1(C(C(C)C2CCC2)=O)C2CCC1CC(CNC(=O)CC(O)C1CC1)C2 c1(C(=O)OC)nsc(=NCC2(F)CCN(C(c3ccc[nH]3)=O)CC2)[nH]1 c1(CC)cc(=NC(C)(C)CN(C)C(c2ccccc2F)=O)[nH]c(COC)n1 c1(OC)ccc(C)c(C(=O)NC2CC2)c1.c1(C=O)ccccc1-n1cccn1.N C1(C)(NC(CCC(C)NC(=O)CN2CCCCC2)=O)CCC2(CC1)CC2 c1(C(=O)NC2CCCC(NC(c3n(C)nnc3)=O)CC2)cnn2c1NCCC2 C12(NC(C(CC)N(C)C)=O)CCCC1CN(C(=O)CC(C)(C)CN(C)C)C2 N1(CC(=O)NCCC2CN(C(=O)C(O)CF)CCO2)CCCNS1(=O)=O CC(C)(C)CCCC(=O)NCC1CCC(NC(c2c(C3CC3)cccc2F)=O)C1 Cc1cc(C(N2C3CCC2C(CNC(c2cn(CCF)nn2)=O)C3)=O)cc(F)c1 c1(CCC(=O)NC)cc(F)cc(F)c1.C1CC2CCC1N2C(=O)C(F)C(F)(F)F C1(C(=O)NCC2C(NC(c3cc(CC)on3)=O)C2)CC2OC1C1CC21 c1(CCC(=O)N(C2CC(NC(C3(C)CC3)=O)C2)C)ccccn1 C(C(C)C)(C(O)C(=O)N1C2CCC(C(N3CCN(CCF)CC3)=O)C1CC2)OC N1(C(C2(C)CC2Br)=O)CC2(CCC(CNC(c3cc(Br)co3)=O)O2)C1 n1(CC(=O)NCC(=O)NC(c2cccs2)C)cccn1 N1(C(Cc2ccn(C)n2)=O)CC(NC(=O)CC(O)c2ccccc2)C(C)(C)C1 C(=O)C(F)(F)CC(C)C.N1(C(c2cn(CC)nc2C2CC2)=O)CC(C2CC2)C1 C(=O)(CCC(=O)CC)NC(CCC)C(=O)N(C)CC1CC1C C1(F)(CNC(CS(N)(=O)=O)=O)COCCN(C(c2ccc(C(O)CF)cc2)=O)C1 CC1CCC(CCC(=O)NCC2CCC(NC(=O)Cc3cncnc3)C2)O1 Cc1cc(O)ncc1C(N1CCCCC1C1(NC(C2CC(F)(F)C2)=O)CC1)=O N1(C(C(CSC)O)=O)CCC(NC(=O)C(C)Sc2nncn2C)CC1 N1(C(C2(C=O)CCC2)=O)CCCC(C)(C)C1.c1(CC=O)cc(Cl)n(C)n1.C c1(C(=O)NC(C2CN(C(c3nc(C)sc3)=O)C2)C)ncc(F)cc1F C=CC(C)(C)CC(=O)NC1CCN(C(c2nc(C(F)(F)F)cn2C)=O)C(C)C1 C(=O)(C#CC1CCC1)N1C(CNC(C2CCC(C(N)=O)CC2)=O)CCC1 C1(C(=O)NCC(C#C)CC)CC(=O)CN1C(c1ccn(COC)n1)=O C1(C(=O)NC(c2ncccn2)CC)COC(CNC(=O)CCc2cnco2)C1 Cc1scc(C(=O)NCC2CC(NC(C3CCC3C(C)(C)C)=O)C2)c1C c1(C(N2CC(F)(F)C2C2(OC(F)F)CC2)C(=O)O)cc(F)c(F)c(F)c1 c1(C(N2C(CC(=O)NC(C#C)C(C)(C)C)CCC2)=O)cccc2[nH]ncc12 C1(C2CC2)(C=O)CC(=O)C1.c1(C(C)C)ncc(C(=O)N)o1.C1CCC(CC)C1 C1(C(N2CCCC(NC(C(C)OCC#C)=O)(CO)C2)=O)CCc2nnc(O)n2C1 CC1CC(NC(C2CC3C(C2)C3(F)F)=O)CCN1C(=O)Cc1nnc(O)s1 CC(C)(O)C(C(=O)NCCn1ncccc1=O)NC(C12CCC(C1)C2(C)C)=O C1(C(N(C)C)=O)CCC(C(=O)N)CC1.C1(O)(CC)CN(C(c2sccc2Cl)=O)C1 c1(C(=O)NC(C(C)NC(c2ccon2)=O)(C)C)cc(C2CCOCC2)nn1C C1(C(=O)NC(CC)CNC(C2CCCCC2)=O)CCc2ccccc2C1 c1(C(=O)NC(CNC(c2c(C)csc2)=O)C)ccc2[nH]c(=N)[nH]c2c1 C1(C(N2CCC(CN(C(=O)COCC(F)(F)F)C)C2)=O)Cc2ccccc2N1 Cc1nc(C(N2CC=C(CCNC(c3cocn3)=O)CC2)=O)c2n1CCCC2 c1(C(=O)NCC2CC(C)N(C(=O)CCCN(C)C)C2)cc(N)nc(Cl)c1 C1(C(C)C)CCC(C(N2CCC(O)(C(F)F)C2)=O)N1C(=O)CC1CC=CC1 c1(C(=O)NCc2c(CCNC(=O)C(=Cc3c[nH]cn3)F)ocn2)ccncc1Cl c1(C(C)(C)C)cccc(C(=O)NC2CC(NC(C3CCC3(F)F)=O)C2)c1 c1(CC)ccc(C(N2CC(NC(C34CC(F)(C3)C4)=O)CC(F)C2)=O)cc1.C NC(=O)CCC(=O)N1CCOC(Cn2cc(-c3c[nH]nc3C(F)(F)F)nn2)C1 C(=O)(CC(C)(C)C(C)=O)NC(C(N1CCC(COCC)C1)=O)CO N1(C(=O)NC2CC(OC(C)C)C2)CCN(C)C(C(N2CCCC2)=O)C1 c1(CNC(C2CCN(C(C(CC)=O)=O)C2)=O)cncc(C#N)c1 c1(-c2cn(CC3CCC(NC(C(COC)(C)O)=O)C3)nn2)ccc(Cl)c(OC)c1 C(CN(C)C)(C(=O)NCc1cncs1)NC(C=C(C)C1CC1)=O c1(C=O)ccc2nnc(C)c(C)c2c1.C1(C)CCC1.C1(OCC)CC1C=O.N S(=O)(=O)(c1cccc(=NCC(C)C2CCC2)[nH]1)NCC1(OCC)CCCCCC1 c1(C(N2CCOCC(NC(C3(F)CCC3)=O)C2)=O)sc2ccccc2c1Cl c1(C(N(C2CN(C(CCc3c(C)noc3Cl)=O)C2)C)=O)ccc2c[nH]nc2c1 c1(CCN2CCC(N(CC#C)C(C3C=CCCC3)=O)CC2)ccc(F)c(F)c1 c1(C(N2C(C(N3CCC(CC#C)CC3)=O)CC2C)=O)ccn2cncc2c1 C1(C)(CNC(C(=Cc2cccs2)C)=O)CCN(C(=O)CC(O)c2ccccc2)C1 O=C(CC(C(F)(F)F)NC(C1CC12CC2)=O)NCc1ncc(CO)[nH]1 C1(NC(Cn2cnc(C(C)=O)n2)=O)CC(C)N(C(c2nc(Br)c[nH]2)=O)C1 C1(CCOC(N2CC(O)(CSCC)C2)=O)CCCCC(=O)N1 c1(CN2CCC(N(C(c3cccc(OC)c3O)=O)C)C2)ccc2ccccc2n1 C12(C(=O)NC3CC(CC)(CC)C3)CCN(C(c3cnc(C)[nH]c3=N)=O)CCC1C2 CC(CC(=O)N(CCC(=O)NC(C1CCCOC1)(C)C)C)n1ccnc1 C1(C)(C(C)O)CCCN1C(=O)CCCCNC(=O)CCOCC(F)F c1ccc2oc(O)nc2c1.C12(C(=O)NCCCNCC)CC(CC)(CO1)C2.C c1(CN2C(C(=O)NCC3COC3)CSCC2)ccc(-n2cccn2)c(Cl)c1 C1(C(=O)O)(COC)CN(S(=O)(=O)CC(=O)OC)CCO1 C1(CC)CN(C(=O)C(=O)N(C)C)CCN1C(=O)C1=CCCC1C c1(C2CCN(C(C(=O)NCC(CC)CC)=O)C2)ccc(O)nc1 C(=O)(C(C)(CSC)NC(c1cc(C)on1)=O)NC1(CC=C)CCC1 C=C(C)CC(C(=O)O)NC(c1occc1CNC(=O)C(C)C(F)(F)F)=O CC1(C)CCCC(C(N2CCC3CC23C(=O)NC2COCC2CO)=O)C1 C1(C(N(C)CC2COCCN2C(C2CCCCC2)=O)=O)CC2CCC1CC2 C(C(C(=O)N(C1CCN(C(=O)Cn2cnnc2O)C1)C)NC(=O)N)OCC N1(CC)CCOCC1C(N1CCCC(CNC(C2CC2)=O)C1)=O.C1CCC1.C C1CC12CCN(C(c1coc(C3CCCC3)n1)=O)CC2.C1(C(=O)NC)(C=O)CC1 N1(C(c2ccc(SC)cc2)=O)CCN(C(c2sccc2C2CC2)=O)C(CF)C1 n1(COC)ccc(NC(=O)C(CO)NC(N)=O)n1 c1(C(N2CCCC2CC(C)O)C(=O)NC(C)C)csc2cc(Br)ccc12 Cc1cc(=NCCCC(C)NC(=O)C(C)NC(N)=O)[nH]c(-c2cccs2)n1 N(C1CCCc2c1cnn2CCO)C(c1csc(-c2cnccn2)n1)=O Cc1cnncc1C(=O)NC1(C)CC(NC(C2CC2(c2ccccc2)C)=O)C1 C1(C)(CCC(=O)NC2C(CC=C)CCC2)CCCN1C(=O)CC1CC=CCC1 Cc1cnc(-c2cn(C(C)C(=O)NCCNC3(Cl)CC34CCC4)nn2)c(C)c1 N1(C(c2cc(OC)ns2)C(=O)NCCSC)CCOC(C)(C(F)F)C1 N1(C(C(C)CCO)=O)CCC2(CCOC2)C(CNC(c2ccc(=O)oc2)=O)C1 c1(C(N2CC(CCCCNC(C(C)SC(F)(F)F)=O)C2)=O)ccc2occc2c1 Cc1ncccc1C(N1CCOC(C(C)NC(=O)Cc2c(Cl)cnn2C)C1)=O Cc1cc(N(CCCCN(C)C(C2CC2(C)Br)=O)C)c(F)cc1[N+](=O)[O-] Cc1ccc(C(F)F)cc1C(N1CCCCC(NC(=O)C=CC2CC2)C1)=O c1(OC)cncc(CNC(c2cccc(-c3ccc(F)cc3)c2)C)n1 C1(C(=O)NCCC(C(C)C)OC)COCCN(C(C2(O)CCCCC2)=O)C1 C1(CC#C)(C(=O)NC(CCO)C(F)F)CCN(C(=O)Cn2cncn2)C1 C#CCCCCCCNC(=O)CC(C)(C)CNC(C1CCCCC1O)=O CC1(C)OCCOC1C(=O)NCC=CCNC(=O)C(c1ccc(F)cc1)=O C1(NCc2ncc(C)nc2)CCN(C(=O)CCCNC2CCCCCC2)CC1C Cn1nc2c(c1-c1cn(CCC3CN(C(c4cnsc4)=O)C3)nn1)CCCC2 Cc1cc(=NC(C)c2cc(C(F)(F)F)n[nH]2)[nH]c(=NCCC(C)O)[nH]1 N1(C(C(C)=CC2CC2)=O)CCCCC(C2CN(C(c3c(C)nsc3C)=O)C2)C1 C1(F)(C(=O)NCC(CSC)(C)O)CCCN(C(=O)CCc2ccnc(C)n2)C1 c1(OC)ccnc(NC(=O)CC2CN(C(=O)CCC(C)N(C)C)CC2C)c1 c1(CCC(=O)NCC(c2ccc([N+](=O)[O-])cc2)C)ccc(F)c(F)c1F N1(Cc2onc(-c3c(C)cncc3)n2)CCC2(O)CCCCC2C1 C12(CNC(C3(COC)CC3)=O)CCC(C1)N(C(C1CCNC1=O)=O)C2 c1cccnc1C1CC1.C1(C(=O)NCC(=O)NCC(=O)N)CCC2(CC2)C1 c1(NC(=O)CC2CC3CN(C(=O)CN4CC=CC4)CC23)ccc(F)cc1CO C(=O)C(C)CC(C)C.CC(C)(C)C.C1(C=O)(C(=O)N(C)C)CC1.CCO c1(CC)cc(C(=O)NC(C2CCN(C(C3CSC3)=O)CC2)C(C)C)nn1CCO C(=O)(C(C)(C)C)N1CCCC1.C(=O)(CC(C)NC(=O)C)NC.C(C)=O.O N1(C(C(C(C)O)C)=O)CC(C2CCCN(C(c3cc(Cl)c(Cl)n3C)=O)C2)C1 CC(C(=O)N1CC(=C(F)CNC(c2cnc[nH]2)=O)C1)C(C)(C)C c1(C(=O)NC(C(C)NC(c2c(C)c(F)ccc2)=O)C)cnc2c(c1)NCC(=O)N2 c1(OC)ccc(C(N2CC(NC(=O)CN(C)CCO)CC2(CC)C)=O)nc1Cl c1(CCNC(COC2CC(NC(C3C(C)CCC3)=O)C2)=O)cccc(F)n1 C1C(CC)(CC)C(=O)N1.c1(CNC(C2CC(CC)OCC2)=O)cccc(O)c1C CCC(C)C(C(=O)N1CC2(CC2)C1)N(C(=O)CC1(N(C)C)CCC1)C C1(OC)CN(C(c2sccc2C)=O)CC1NC(c1cncc(C(C)=O)c1)=O N1(C(c2c(C)c[nH]n2)C(=O)NC2(C)CC2)CCCCC1CCOC(C)(C)C C(=O)(C(CC(F)F)NC(=O)C(O)C=C)N(C(C=C)C1CC1)C N1(CC)CCCC(C)(NC(=O)CCC(c2ccc(OC)c(OC)c2)=O)C1 Cc1ccc(CC(N2CCN(Cc3ccc(O)cn3)C3CC23)=O)c(F)c1 CCC(CC)(CCOC)C(=O)Nc1ccc2ncsc2c1 c1(C(N2C3CN(Cc4nnc(CC)s4)C(C3)C2)=O)ccc2nc(O)oc2c1 c1(C(=O)NC(CNC(C2CC(C)OCC2)=O)(C)C2CC2)cnc2n1CCCCC2 C1(C)(COC)CCCN1C(=O)CC1CC(C)C1.C(=O)C(C)C.CCC(C)C c1(OC)cc(CC(=O)N(CCCNC(=O)CC(C)O)C)cc(Cl)c1 C(=O)(CC(C(F)(F)F)P(C)(C)=O)N1CCCC(F)C1.Cn1cnc(C(=O)N)n1.C c1(C(N2CC(O)(C(C)C)C2)=O)cc2c(o1)CCCC2 CCCC(C#N)C(=O)NCC1CCC(C(=O)NCc2cnccc2Cl)CC1 C1(CN(C(=O)C(c2ccccc2)C)CC)CCCN(C(=O)C=O)C1.C1CC1.N C1(N(C(c2c(C)nns2)=O)C)CCCN(C(=O)COc2cccc(O)c2)CC1 C=CCC(F)(F)C(=O)NC(C)CCNC(=O)C(C(C)C)n1cc(Br)cn1 O=C1CC(C(N2CCC(CNC(c3ccccc3)=O)CC2)=O)C2CCCCC2N1 c1(C(=O)NC2(CN(C(C3(C=C)CCOCC3)=O)C)CC2)ccc2snnc2c1 [SH](=O)(=O)c1ccccc1.N1(C(C(C)=C(C)C)=O)CCC(NC(=O)CC)C1(C)C C(CC(F)F)(C(=O)NC1CC(N2CCCC2)C1)NC(c1c(C#C)c[nH]n1)=O c1(C(=O)OC)ccc(C(N2CC3CC3(C)C2)=O)cc1C.C1(C=O)CC12CC2.N c1(C(=O)Nc2ccc3ocnc3c2)n[nH]c2c1CN(C(=O)CCC(F)(F)F)CC2 C1(C(N2CCC3C(C2)CN3Cc2ccccc2)=O)C2CCC3C(C2)CC13 c1(C(=O)NC(C2CCCCN2C(=O)C=Cc2ccoc2)C)ccc2[nH]ccc2c1 C=CC1CCCC(Nc2cc(NCC3CCCC3)nc(C)n2)C1 C1(NC(C2C(C=C)OCC2)=O)CC2CC(NC(c3n[nH]cc3CC)=O)CC12 O=C(C#CC1CCCOC1)NCC1CC(O)CN1C(c1cc(CCCO)on1)=O C=CCC(C)(C)C(=O)NCC1CN(C(c2sccc2OC)=O)CCC1C C1(O)CCC1.c1(C=O)c[nH]nc1C.C(C(=O)N)N(C=O)CC.C(C)(C)C N1(C(Cn2ncc(C)c2)=O)CC2CCN(C(=O)CCOC3CC3)CC2C1 C(CC(=O)NC1CC(CNC(c2cc(C)cnc2C)=O)C1)(C(C)C)OCC Nc1cccc(C(=O)NC2CCC(NC(c3ccnn3C3CC3)=O)C2)n1 C1(F)(C(=O)NC2(c3c(C)ccc(Br)c3)CC2)CCC(C)(C)CC1 C1(CNC(=O)C2CC2)CC2CCCCC2N1C(=O)Cc1cc(F)ncc1Br c1(C(=O)NCCC(C)NC(c2c(C)nc(CC)s2)=O)nc(OC)ccc1C N#Cc1ccccc1C=CC(N1CC2(CCN(C(C3CCCOC3)=O)C2)C1)=O C(C(CC)(CC)C(=O)N1CC(c2ccon2)C1)NC(C(CCCC)O)=O CC1CCN(c2nnnn2CC2CCCCN(C)C2)C1(C)C c1(OC)cccc(OC)c1OCCNC(C1CCCN(CCC(F)(F)F)CC1)=O C1(C(N2CC(C)(NC(CC3CCN(C(C)=O)CC3)=O)C2)=O)CCCC2(CCC2)O1 C(CCC(N)=O)(C(=O)N1CCN(C(C2CC2(C)C)=O)CC1CCO)N(C)C c1(C(N2CCC(F)(CNC(C3CCC3(F)F)=O)CC2)=O)cnc2ccccn12 CCC(C)C(C(=O)NCCCC(=O)NC)N(c1ccc(OC(C)(C)C)cc1)C c1(C(N2CCC(C)(NC(=O)C(O)CN3CCCC3)C2)=O)coc2ccccc12 CCCC(C(=O)N(C(C)C(=O)Nc1ccccc1OC)C1CC1)NC(N)=O CC(C(=O)NC1(CC=CC(=O)NCC(C)(F)F)CCC1)C1(O)CCC1 c1(OC)ccc(Br)c(CC(N2CCCC2c2cn(CC(O)C(F)(F)F)nn2)=O)c1 C(=O)(CCC(N)=O)NCC(CC=C)NC(c1ccc(CC=C(C)C)cc1)=O C(=O)(C(C#N)C(C)C)NC(CC)C(=O)Nc1cccc(F)c1F c1(C(=O)NCCCCCC)ccc([N+](=O)[O-])n1C.C1(CC(=O)N)CC(C)(C)CO1 O=C1CCC(CCC(=O)NC2CCC2NC(=O)Cn2cccc2)=NN1 C1(NC(=O)NCC(CO)C2CCOC2)CCC(F)CC1 N(C1CCc2ccccc21)(CCCOCCOC)Cc1ccccc1 c1(C=O)cnc(Cl)c(I)c1.C(=O)(C(Cl)(Cl)Cl)NC(=O)NC1CC(C)C1 N1(C(c2c(C)nns2)=O)CC(C(=O)N(c2nccs2)C)CC2OCCC12 c1(CCC(=O)O)ccc(N2CC(C(F)F)C3(CC3)C2)c([N+](=O)[O-])c1 C1(NC(CC(C)(C)OC)=O)CCC2CCN(C(=O)C(C)Cc3ccc(C)cc3)C12 N#Cc1ccnc(-c2ccc(Cl)s2)n1 C=Cc1cnn(C)c1C(N1CCC(CCNC(C2(OC)CCCOC2)=O)CC1)=O CCCC(C(=O)N1CC(F)CC1CNC(C1(COC)CCCO1)=O)OC C1(CC(=O)NC(CCCNC(c2cn(C(C)C)nc2)=O)C)CC(=O)NC1=O C(=O)(C1=CCCCC1)NC1CC(F)(CNC(C2(CC#C)CCOC2)=O)C1 C1(NC(c2cc(O)ccc2Cl)=O)CC2CC(NC(C3CCC4(CC4)C3)=O)CC2C1 C(=O)(C1CCCc2n[nH]cc21)N1CCCC(C)(NC(C23CCCCC2C3Br)=O)C1 Cc1ccc2[nH]c(C(N3CC(NC(C4CC4C)=O)CC34CCCC4)=O)c(Cl)c2c1 S(=O)(=O)(c1ccc(Br)cc1N1CCC(C)(C)C1)N1CCn2c(C)ncc2C1 c1(C(=O)NCC2CCCC(NC(c3ccco3)=O)C2)nccc2ncccc12 C1(C=O)CC(=O)N(C2CCCCC2)C1.Cc1ccc(C(N2CC(O)(C)C2)=O)o1.N c1(NC(C(=O)NC2CC(C)(NC)C2)=O)cc2c(C)cccc2[nH]1 c1(C2(C(=O)NCC(CC)NC(c3[nH]c(O)nc3C)=O)CC2)cccc(F)c1 C(C(CC(C)C)C(=O)NC(C)(CNC(c1ccc2nn[nH]c2n1)=O)C(C)C)OC c1(NC(=O)CSC2=NCCS2)ccc(C2CC2(F)F)cc1 Cc1nc(Br)oc1C(=O)NC1(CNC(C2CN(C)C2)=O)CC1 C1(N(C(C2C(NC(C3(COC)CCCC3)=O)CCO2)=O)C)CCOCC1C C1(N(C(C(CSC)OC)=O)CCF)CCCN(C(=O)CCSCC(N)=O)C1 c1(C(N2C(CNC(C3CCC(C)O3)=O)CCC2)=O)cc2c([nH]1)CCCC2 N1(C(c2c(C=C)cnn2C)=O)CC2CCCC2(NC(=O)CCC)C1 c1(CC)cc(C(N2CC(NC(=O)CCSc3ccccc3)C2)=O)n[nH]1 N1(C(COCC)=O)CCCC2CN(C(c3ccc(C(C)(F)F)cc3)=O)CCCC12 c1(C(=O)OCC)cccc(C#CCNC(=O)NC)c1.C1(C)COC(=O)C1 N1(C(CC(C)n2cccc2)=O)CCC(CCC(=O)NCC(=O)N(C)C)CC1 N1(CC)CCN(C(=NCC(O)(C=C)CC)NC(c2ccc(F)cc2)CF)CC1=O c1(C(N2CCN(C(C3CC3)=O)CC2C2CC2)=O)ccc(P(C)(C)=O)o1.CCC c1(OC)ncccc1C(=O)NCCC(C)(C)CNC(=O)CC12CCCC1C2 N1(C(C2CC(SC)C2)=O)CC2(NC(C3CCCC(O)C3)=O)CCC1CC2 C1(F)(CNC(C2C3COCC23)=O)CCCN(C(=O)CCSC2CCCC2)C1 S(=O)(=O)(c1ccc(N2CC3CSCC3C2)c(Br)c1)NC1C(N(C)C)CCCC1 CCC(CC(=O)N1CC2C(C(=O)NC3CN(c4ncc(F)cn4)C3)C2C1)C1CC1 CCCC(C(=O)NOC1CCCC1)NC(=O)C#CC1CC1 CCCCCC(C)CC(=O)NCC1(F)CN(C(c2cccc3c2CCCC3)=O)C1 C(CCC(=O)NCC1CC(NC(c2cnc(C3CCOC3)s2)=O)C1)N(C)C C1(NC(CC2(N(C)C)CCC2)=O)CCCC(NC(=O)CC2(C)CCCCC2)C1 C(CCCC(=O)N1CCC(NC(=O)C(C)CSC)CC1)OCCC=C c1(NC2(CC)CCN(C(C3CC(CCC)OCC3)=O)CC2)cc(=O)n(C)c(O)n1 Cc1cc(C(N2CC(C(=O)NOC(CO)C(C)C)C(F)C2)=O)c(C)nn1 C#CCC(CC(=O)N(C1CCCNC1=O)C)NC(=O)C(C)(C)CN(C)C C#Cc1cncc(C(=O)N(CCCC(=O)NC2(CO)CCC(C)C2)C)c1 CC1=CCC(C(C)NC(C)CCc2ccc(I)cc2)CC1 CC(C)CCC(=O)NC1CC(CNC(=O)CNC(c2ccncc2)=O)C1 C12(CNC(CC)=O)CC(NC(C3(CC)CCC3)=O)(C1)C1(CCOCC1)O2 Cc1ccc(N(C)C(C)C)c(C(=O)N(C)CC)c1.C12(CC(=O)N)CCCC1C2 C(N=c1[nH]c2c(c(=NCCOCCC3CC3)[nH]1)CSC2)c1cc(C(C)(C)C)no1 C(C)(c1ccccc1C)=CC(=O)NC1CCCN(C(c2ncn(CC)c2)=O)CC1 N1(C(c2ccc(=O)oc2)=O)CCN(C(=O)Cc2csc(Cl)c2)C2CCCC12 C(=O)(CC(C)C(C)(C)C)NC(CC(=C)Cl)C(=O)NCCCCC(F)(F)F CCC(C)C(O)CC(=O)NC(C(=O)NCCn1nc(C)nc1C)c1cccs1 Cc1ccc(F)cc1NC(C1CC12CCN(C(c1cncc(O)c1)=O)C2)=O Cc1c(Cl)cnn1CC(=O)NC1CCC1.C1(C=O)CCN(S(C)(=O)=O)CC1.C c1(C(=O)NC2C(OC)CN(C(C3(CCCC)CC3)=O)C2)nccc(N)c1Cl Cc1cc(C(=O)NC2CCCCC2)c(N)c(F)c1.c1(C(=O)N)cn(C(C)C)nn1 C(=O)(C1=C2CCCN=C2NN1)N1CCCCC(NC(C2COCCO2)=O)C1 CCCCCC(O)C(=O)NCCC(C)N(C(=O)CNc1nccs1)C c1(N2CCC(CC)CC2)nc2cc[nH]c2c(=NC2CC(C3CC3)C2)[nH]1 c1(CC=O)cccc(O)c1.CCCCCCOC(C)C(=O)NC1CCCC1C.N N(C1CCc2ccccc21)C(C1=CC(O)C(NC(C2(C=C)CCOCC2)=O)C1)=O N1(C(c2c(C)nsc2)C(=O)NC(C)C)CC2(C)C(=O)NC(=O)C2(C)C1 C1(NC(C(CCSC)NC(=O)CCCNC(C)=O)=O)CC2(CCCO2)C1 CC1CC(NC(=O)C(=O)N(C)C)CN(C(C2(c3cccc(F)c3)CCCC2)=O)C1 c1(CC(=O)N(CCC)CC)cncc(C#N)c1.C(=O)C(C)(C)C.C(=O)CC N1(C(C(C)=CC2CC2)=O)CCC2CCN(C(c3cc(C(N)=O)c[nH]3)=O)C2C1 c1(C(=O)NCC2(NC(=O)CCCC3CCCCC3)CCC2)cc2ccccn2c1 N1(C(C(c2ccoc2)NC(CCOCC)=O)=O)CCCC(CO)C1C N1(C(C2C(C)CCCC2)=O)CC=C(CC(=O)NCC(C)(O)C2(C)CC2)CC1 c1(CC=CCC(=O)NC2CC(CNC(=O)C=CBr)C2)ccccc1 C1(NC(C(CC)c2cccnc2)=O)CC(OC)CN(C(C2CNC(=O)C2)=O)C1 C(CC1=CCC2CC1C2(C)C)NC(NC1CC(NCCCC)C1(C)C)=NC(C)C CCC(C#N)(CC)C(=O)N1CCCCC(C(N2CCCN(C)CCC2)=O)C1 C1(C(=O)NC2C=CCN(C(c3c[nH]c(=N)o3)=O)C2)CCC2(CCOCC2)C1 CC1CN(C(c2cccc(CF)c2)=O)CC2(CCN(C(=O)CC=C(Cl)Cl)C2)O1 S(=O)(=O)(c1ncc2ccccn12)NC(c1cccc2nc[nH]c12)=O N1(C(c2c(CC)[nH]nc2Cl)=O)CC2(C)CN(C(c3cnnc(Cl)c3)=O)CC2(C)C1 c1(C(N2C(C)CCC(NC(=O)CCN)C2)=O)cc2c(ncn2C)s1.[SH](C)(=O)=O C1(NC(C2(C)CC(=C)C2)=O)CCN(C(c2cnn(C)c2Cl)=O)CC1CC C(c1ccc(C)c(Cl)c1)=CC(N1C2CC(C2)C1)=O.C(C=O)N(CCOC)C.N c1(CCC)nsc(N)c1C(=O)N.C1CCCC(N(C(=O)C=Cc2cn[nH]c2)C)C1 N1(CC)CCC(CC(N2CCC(c3nn[nH]n3)C2)=O)C1(C)C.c1(C(=O)N)ncccn1 N1(C(CCCN(C(C)C)C)=O)CCC(C)(C)C(C(=O)NCCc2cnn[nH]2)C1 O(P(C)(=O)CNC(=O)C(Cc1cnc[nH]1)NC(C1CC(C)(C)CO1)=O)CC c1(C(N2CCN(CCNC(c3c(OC)c[nH]n3)=O)CC2)=O)cc2ncccc2o1 CCC(=O)CCC(=O)N1CC(OC)CC1C(=O)NC1(C2CCCCO2)CC1 C(=O)(C(CC)CCCC)NC12CN(C(CC(C=C)(C)C)=O)C(CC1)C2 C(CC(O)CC(=O)N(C(C)CNC(c1cnc(CC(C)C)[nH]1)=O)C)SC C=C(C)C1OCCC1C(=O)NC(CC(=O)NC1CC(=C2CC2)C1)C(F)F CC1CN(C(C2(N3CCOC3=O)CC2)=O)CCN1C(=O)CC1(O)CCCN(C)C1 CCC(C)CC(C)NC(C1(NC(=O)CN2CCN(C)CC2)CCN(C)C1)=O c1(NC(C2CC(NC(CC(C)Oc3ccccc3)=O)C2)=O)ccccc1Br N1(C(C(C(C)C)C)=O)CCC2(C1)CN(C(=O)CCCc1ccncc1)C2 N#CC1CN(C(=O)CC2CCCN(C(c3cc(O)nc(O)n3)=O)CC2)CCO1 c1(C(=O)NC2CN(C(c3onc(C)n3)=O)CC2(C)C)ccc2c(c1)CCCCN2 N1(C(c2n(CC)ccn2)=O)CCC2CCC(C1)N2C(c1cc(C)no1)=O N1(C(CCc2ccco2)=O)CCc2nc(O)[nH]c2C1.C(=O)(COCC=O)OC.N c1(NC(C2CC2C(F)F)=O)cncc(CO)c1C.C1(SC)CC(C=O)CC1O c1(C(N(C2CCN(C(C3CC3Br)=O)C2)CC)=O)cc(F)cc(Cl)c1 CCCC(C)(O)CC(=O)N1CCC(NC(=O)Cn2ccnn2)C(C)C1 N1(C(COCCC)=O)CCCN(C(C23CCC(C(F)(F)F)(CC2)C3)=O)CC1C C1(C(N(CCS(N)(=O)=O)C)=O)CN(C(c2ccc(Cl)o2)=O)C2(CCC2)C1 N1(C(C2(O)CC(C)(C)C2)=O)CC(NC(=O)CC(C)(C)C2CCCCC2)CC(O)C1 c1(NC(c2cc(C)cn3c2ncc3)=O)ccc2c(c1)Cc1ccccc1-2 c1(NC(C2CN(C(=O)COC3CCCC3)CCC2O)=O)cc2c[nH]nc2cc1Br C1(CC(N2C3CCC2CC3)=O)CCC2(CC1)CCN(C(C1CC1F)=O)CC2 C1(C(N2CCN(C(=O)CO)CC2)=O)(NC(C(CC)N(C)C)=O)CCN(C)C1 Cc1cc(N(CC2=CCCOC2)C)nc(=NCCc2c(F)cccc2Cl)[nH]1 C=CC1OCCC1C(=O)N(CC(O)CNC(=O)Cc1cc(Br)nn1C)C C=C1CN2C(=O)CCC2(C(=O)NC2CCC(C)C2)C1.c1(CC=O)cnoc1.N C(=O)(CCCC(C)(C)C)NCC1N(C(=O)CC2CCCNC(=O)C2)CCN(C)C1 C1(C(N2CCC(O)(CNC(CCN(CCC)C)=O)C2)=O)CCC(F)(F)CC1 N1(C(c2cccc(OC)c2)=O)CCCC2(CC(NC(=O)Cc3cncs3)CO2)C1 C1(CNC(c2cc(OCC)no2)=O)CN(C(=O)C(F)=C2CCCC2)CC1C c1(OCC)ccc(CCC(=O)N(C)CCN(C)C(c2[nH]c(C)nc2C)=O)cc1 C(CCCC(=O)NCC1CC1(F)F)N(C)C(C1CCN1C(C)(C)C)=O CC1=NNC(=O)C1CC(=O)NC1CN(C(c2cccnc2)=O)CC1C.C(C)(C)S CCCC(CC)C(=O)NCC1(F)CCC(CNC(=O)CS(C)(=O)=O)C1 Cc1[nH]c(C(C)(C)C)cc1.N1(C)CC(=C(F)C)C1.C(=O)CCC1CC1(Cl)Cl C12(CC)CCC(C1)N(C(c1cnn(C3CC3)c1)=O)C2.C1(C(=O)N)CC1(F)F Cc1cc(C(=O)NC(C)CC(C)NC(c2cnn(C)c2C#N)=O)c(C)cc1Br C#CCCCCC(=O)NC1(C)CCC(NC(C2(C)CCCS2(=O)=O)=O)CC1 c1(C(=O)NCC(CC)NC(=O)CSS(C)(=O)=O)c(C)c2ccccc2oc1=O c1(OC)cccc(C=CC(=O)N(C2CCC(NC(c3csc(Cl)n3)=O)C2)C)c1 c1(OCC)cc(C(=O)N)cc(F)c1.C1CN(C(=O)CN2CC3CC3C2)CC1C Cc1noc(C)c1CCC(=O)N(C(C)CNC(=O)C(c1ccccn1)O)C C(=O)(C(CC(C)C)NC(=O)CC1COCC(C)O1)NCc1scc(CC)n1 N1(C(c2cc(C(C)C)sc2)C(=O)NC2(C)CC2)CCCC(C(C)C)(CO)C1 CP(C)(=O)C1CCC(NC(=S)NC(c2ccccc2Br)CF)C1 c1(N(C2CC3CC2CN3)C(C(N2CCCCC2)C)=O)ccc(C(=O)N(C)C)cc1 CC(C)CC(C(=O)NC(c1ccccc1F)CNC(=O)CC)C(N)=O.C(C)C.S c1(C(=O)NCC(CNC(C(C)=C(CC)C)=O)F)cc(C(F)(F)F)n[nH]1 C1(NC(c2ccc(OCF)cc2)c2n(C)nnn2)CCC(C2CC2)C1 c1(C(N(CCN(C(=O)CO)CC)CC)=O)[nH]cnc1C.C1CCCOC1.C c1(C(=O)NCC2COCCN2C(C23CCC(C2)C3)=O)cc(O)cc(F)c1 C1(C(=O)NCCNC(C(CC)SC)=O)CCN(C(=O)Cn2ccnn2)CC1.C N1(C(c2ccc(C(=O)NC)cc2)=O)CCc2sc(-c3cccnc3C)cc2C1 C(=O)(C1=CCCOC1)N1C(CNC(C(C2CC(F)(F)C2)OC)=O)COCC1 C1(NC(CCC#CC)=O)C2CC3CN(C(c4cc(F)c(O)c(F)c4)=O)C1C3C2 Cc1cc(C(=O)N(C2CCC(NC(=O)C=CC3CCCCCC3)C2)C)ccc1Cl N1(C(CC(CC)C)=O)CC(NC(c2cc(C)n(-c3ccccn3)n2)=O)CC(F)C1 N1(C(c2nc(C)oc2)=O)CC2CC1C2C(N1CCCC1CC1CCC1)=O C1(C(N2CCCC(NC(C3CC(O)C3)=O)C2)=O)OC2CCC1CC2 C1CN(C(C2CCC(F)(F)C2)=O)CCCO1.Cc1cc(COCC(=O)N)no1.C C1(CCOC)CN(C(=O)C(C)CCN(C)C)CCN1C(=O)CC1CCCC1 C1(C)CN(C(=O)Cc2ccc(C(C)=O)cc2)CCO1.C(C=O)N(CC)CC.N N1(c2cc(COC)ncn2)C2CCC1CN(C(c1nc[nH]c3ncnc1-3)=O)CC2 C(=O)(CCC(N)CCC(=O)NCCc1ccc(NS(C)(=O)=O)cc1)OCC c1(CNC(=O)NC(c2c(CCC)nns2)C)ccc2cc[nH]c2n1 N1(C(Cn2c(C(=O)OC)cnc2)=O)CCCC(C)(CNC(=O)CNC=O)C1 CCC(CC)CC(F)C(=O)NC(CC(C)C)C(=O)NC1CCN(C(N)=O)C1 c1(OC)csc(C(=O)NC2CCC(CC(N3CC(n4cnnn4)C3)=O)C2)c1 c1ccccc1Cl.n1(C2CN(C(C3C(=C)CC3)=O)C2)cc(-c2cnn(C3CC3)c2)nn1 c1(C=O)cc2c(s1)CC(C)(C)C2.c1(CC)cc(C(N2CC=CC2C)=O)ncn1 CCC(C)N(OC)C(=O)C(C)CNC(=O)C(C)NC(N)=O CC1CN(C(C2CC(C)(C)C2C(F)(F)F)=O)CC1C.c1(C=O)cc(Cl)on1 C1(C(=O)NCC(CC)(CC)NC(=O)CN2CCCC2C)CCC2(CCOCC2)O1 CCCC(=O)O.c1(C=O)csc(C2CCCN2C(C(C)(C)C)=O)n1.C(C)(C)C C1(NC(c2c(CC)nn(C)c2)=O)CCCN(C(=O)Cc2ccc(Cl)cn2)CC1 Cc1noc(C(C(C)C)NC(N2CCC(N3CCOC3=O)C2)=O)n1 C1(NC(C(C(=O)OCC)(C)C)=O)CC2CCCC2C1.c1(C(=O)N)cscc1 CCC(CC(=O)NCCOCC(=O)NCC1CC[Si](C)(C)C1)C1CCC1 N1(C(C2C(C=C)C2)=O)CC(NC(C2CN(S(N)(=O)=O)C2)=O)C(C)(C)C1 C1(NC(C(C)CC2CCC2)=O)CN(C(c2ccncc2F)=O)Cc2ccnn2C1 N1(C(C(N)=O)=O)CC(CNC(c2cn3cnnc3cn2)=O)OC2(CCC2)C1 CC(CCC(=O)NCCC1CC(F)(F)CN1C(c1ccnn1C)=O)S(C)(=O)=O Nc1cnc(Cl)cc1C(N1CCN(C(C2CCC(O)C2)=O)C(CF)C1)=O C=CCCCC(C)(C)C(=O)NC1CC(OCC(=O)NCC(=O)NCCO)C1 C1(C=O)CC(C)(C)OC1=O.C12(CCNC(C(C)SC)=O)CCC(CC1)C2.N N1(C(C(CSC)(C)C)=O)C2CCC1C(F)C(NC(C1CC3CCCC3C1)=O)C2 C=CCC(C)(CC)C(=O)N(C)CC1CCN(C(=O)CSc2cccc(C)c2)CC1 C1(NC(=O)COC2CCCCC2)C=CCN(C(=O)CCc2nc[nH]n2)C1 Cc1cc(=NC(=O)CC(c2ccccc2)NC(c2cccc3cc[nH]c23)=O)cc[nH]1 CCC(CNC(C1CCC(=O)N(C)C1)=O)(CC)C(=O)NCC(C)(C)C(C)O C(=O)(C(C#N)C(C)(C)C)NCC(C(=O)NC(CO)CCCO)OC c1(C(=O)NC2CN(C(CCc3c(C)ncs3)=O)C2)c(N)cccc1F C1(C(=O)NCCN(C(c2cnn(CCCC)c2C)=O)C)C2CS(=O)(=O)CC12 C(C)(C)(C(C)CC(=O)N1CCC(C)(CO)C1)NC(CCOC(C)C)=O C(=O)(CC1CS(=O)(=O)c2ccccc21)N1C2C(NC(c3c(C)cns3)=O)C(C2)C1 CC(C)C(F)(F)CC(=O)NC1CN(C(=O)CC(C)O)CC12CCC2 CCCC(CCC)C(=O)NCC(C)(C)CNC(C1CC2COCCN2C1)=O N1(C(C(C(CNC(C(CCOC)(C)C)=O)C)F)=O)CCC2(C1)CN(C)C2 CC(C)(C#N)CCCC(=O)N1CCN(C(=O)CCN2CCNC(=O)C2)C(CF)C1 C(=O)(C(F)C(C)(C)O)NC1C(NC(C2CC(OC)CN2C=O)=O)C1.O C1(C(=O)NCCF)CCCN(CCC2(O)CCCC2)C1 N1(C(C2CCC(C)CC2)=O)CCN(C(=O)C2CC2)CC1CCO CC1CN(C(=O)CCc2cc(F)cc(F)c2)CCCN1C(=O)CC#N Cc1cc(C)c(C)c(S(=O)(=O)NCC(N2CCc3c(CN)cccc3C2)C)c1C C1(C(=O)NCC2OCCC(NC(=O)Cc3cncs3)C2)CCC2(CCC2)OC1 c1(C(=O)NC2CC(CC(=O)NC3CC3O)C2)nccc2[nH]ccc12 c1(C(=O)NCC(CC(C)C)NC(C(CC)c2cccnc2)=O)cc(F)cnc1O C1(C(=O)NC(CNC(C2(OC)CCC2)=O)C2CC2)CCn2cncc2C1 c1(CCC(=O)NCC2CC2NC(=O)Cc2ccccc2F)csc2ccccc12 C1(NC(CS(CC)=O)=O)CC2CCC1CN2C(=O)CC1CSC1 N1(C(C2(CC=C)CC2)=O)CCOC2(CCN(C(c3nonc3N)=O)CC2)C1 C1(C(=O)NCC(COC(C)C)O)C(C2CC2)CCN1C(=O)CCCC1CCC1 C=CC(C)(O)CC(=O)N1CC(OC)C(NC(=O)Cc2ccccc2C)C1 c1(C(=O)NC(CCNC(c2ccc(OC)cn2)=O)C)cnc(C)nc1C c1(C(N(CCCNC(C2CC3CCC2C3)=O)CC)=O)nccc2c1NCCC2 N1(C(c2cccc(F)c2F)C(=O)NCCCSCC)CC(C)(C)CC1(C)C.O CCC(C(=O)N1CCC(F)(C(=O)NCC2(C)CCCC2)C1)C(C)(C)CC CCCCC(C(=O)NCCC1(C)CCN(C(=O)CNC(=O)OC)CC1)N(C)C O=S(=O)(c1ccc(=NCc2ccc(F)c(Br)c2)[nH]c1)NC1CC(C2CC2)C1 C(CC(O)CC(=O)N1CCN(C(=O)C(C)(C)C(=O)OC(C)(C)C)CC1C)SC C1(C#N)(CC(=O)Nc2nn(C)c(C3CCCCC3)c2)CCS(=O)(=O)CC1 CCC(C)(C)C(=O)C(=O)N1CCC(C(=O)NCCC(C)C(F)F)C(O)C1 Cc1ccc(F)cc1C(=O)NCCCC1CCCCN1C(C1CCC(=O)N1)=O N1(CCC(=O)CNC(c2ccccc2)Cc2ccncc2)CCOCC1 Cc1nc(N2CCOC(CNC(=O)CCc3cnc[nH]3)C2)c(C)c(Cl)n1 C1(NC(c2c(C)noc2)=O)CCN(C(c2cccc(Br)c2Cl)=O)C12CC2 C(=O)(CC(CNC(c1ccc(F)cn1)=O)C1CCC1)N(C1CCC(O)CC1)C N1(C(C(C)C)=O)CCC(CNC(C2(Br)CC2)=O)C1(C)C N1(C(c2c(COC)ncs2)=O)CC(C)N(C(c2cc(N(C)C)ccn2)=O)CC1C c1ccc(C)c(N2CCCS2(=O)=O)c1.CCCC(C(=O)N)NCCSCCOC C1(CCNC(c2cc(C)sc2)=O)CCCN(C(C2CCCSS2)=O)C1 c1(CN2C(CC(N3CC4CCCC4C3)=O)CCC2)cccc(O)c1Cl C1(c2nc(C(C)C)on2)CC(C)CCN1C(=O)NC1CCC(SCCO)CC1 c1(OC)cc(C(F)F)c(C(N2CCOCC(C)C2)=O)cn1.C(=O)(C(C)C(F)F)N C1(CC(=O)NCC2CCCN2C(=O)Cc2ccsc2Cl)CC2CCC1C2 N1(C(Cc2cn(C)nn2)=O)CC(NC(=O)CC2=CCCC2)CC(C)(C)C1 C1(CC(=O)NCCNC(=O)Cn2nnnc2-c2ccccc2)(CO)CCOCC1 c1(C(=O)NC(C)C(C)(C)NC(c2ncccc2O)=O)cc(C(F)(F)F)ccn1 c1(C(N2C(CCNC(c3n(C)nc(O)c3)=O)CCCC2)=O)c[nH]c2ccccc12 N1(C(CSC(C)C)=O)CCN(C(=O)CC2CCC(O)C2)CC1c1ccccc1 c1(OC)ccc(C(=O)NC2CCOCC2NC(=O)CCCn2cncn2)nc1N Cc1noc(Cl)c1CC(=O)N(C)CC1CN(C(=O)C(C)CN(C)C)CCO1 C1(CNC(CCC#CC)=O)CC2(CN1C(c1cccc([N+](=O)[O-])c1)=O)CC2(F)F c1(C(=O)NCC(CC=C)NC(c2cnc[nH]2)=O)c(C(F)(F)F)cccc1F N1(C(COC(CC)CC)=O)CCC2CCN(C(c3ccncc3)=O)C2C1 C12(CNC(NCC(CC)Nc3ccccc3)=NC)CCCC(NC)(CC1)C2 c1(NC(C2C(CCC)CNC2)=O)ccc(C(F)(F)F)c(C)c1 C(CCCC(=O)N1CCC(C)(CCNC(=O)CC(F)(F)Cl)C1)OCCC=C N#Cc1nc(Br)cnc1NC(C1CC2CC2N1Cc1cccc(Br)c1F)=O c1(CC)noc(C(N2CC(CC(C)NC(C3C(C)C3C)=O)C2)=O)n1 c1(C(=O)OCC)cc(C=O)[nH]n1.CC(C)C1CC1.N1(CC=O)CC(C)C1 c1(CC(=O)NCC2(OC)CN(C(CSCCCC)=O)C2)ccccc1Br CCS(=O)c1ccccc1C(=O)NC1CC1NC(c1ccc(C)cc1OC)=O c1(C(=O)NCCC(CCNC(c2cn(CC)nc2)=O)C)sccc1S(N)(=O)=O c1(C(=O)NC2COCC2NC(C2(O)CCSC2)=O)ccc(F)cc1C(F)F c1(C(N(C2CN(C(c3cnc(CC)nc3)=O)CC2O)C)=O)nc(OC)ccc1Cl c1(C(N2CCCC(C)(NC(C(CC)C)=O)C2)=O)cc(O)nc2[nH]c(=N)ccc12 N1(C(C)CO)CCC(C(=O)NCCc2nc(-c3ccccc3Cl)no2)CC1 C1(C(=O)NC2C=CCN(C(Cc3cn(C)nc3)=O)C2)CS(=O)(=O)CC12CC2 C#CCC(C(=O)N(CC(C)(C)C(=O)NCCC(CCC)SC)C)C1CC1 c1(C(=O)NCC(CNC(c2scc(OC)c2)=O)F)cn2c(C)cccc2n1 C1(O)(CN(C(CN(CC)CC)=O)C)CCCN(C(C2(CF)CCOCC2)=O)C1 N1(C(C2C(=C)CC2)=O)CCC(C)(CCNC(=O)CCCc2ccccn2)C1 Cc1cc(C(=O)NC2CC=C(C(=O)NC3(c4noc(C)n4)CC3)C2)cc(C)n1 N#Cc1cccc([N+](=O)[O-])c1NC1CC(NC(c2c[nH]cc2Br)=O)C12CCC2 C1(C(=O)NC2(CCOC)CCN(C(=O)C)C2)Cc2ccccc2S1.C(C)(C)C Cc1ccc2c(C(N3CCCC(NC(C45CCC4C5)=O)C3)=O)ccnc2c1 C1(NC(Cc2c(C)cc(Br)cc2)=O)CN(C(=O)CC#N)CCC1(C)C C1CC2(C1)CN(C)C2.C(CC1CCOCC1)(C=O)NC(C(C)N(C(C)=O)C)=O Cc1nc2n(n1)CC(C(=O)NC1CC(C)C1)CC2.c1(CCC(=O)N)nncn1C C12(NC(c3ccc(C)cc3)=O)CCN(C(c3nnn(C)n3)=O)CC1C2 c1(NC(C2CCCC(NC(c3n(CC#C)cnn3)=O)C2)=O)ccc(O)c(C)c1 CCCCCC(C)(C)C(=O)NCCCN(CCCNC(C1CC1C1CCC1)=O)C N1(C(C(C2CCOCC2)OCC)=O)CCOC2(CCC(C(=O)OC)CC2)C1 N1(C(CCOC(C)C)=O)CCC(CCCCNC(=O)CCNC(=O)C=CCl)CC1 NS(=O)(=O)N1CCCCC1C(N1CC2CCC1CN2C(=O)CCn1cccc1)=O N1(c2c(C#N)cccn2)CCN(N2CC(C(=O)NCc3ccccc3)C2)CC1 c1(C(N2CC(O)C2)=O)n[nH]c2c1CC(C)CC2.C(=O)(C(C)(C)C1CCC1)NC.C c1(C(=O)OC)[nH]c2ccccc2c1CN1CC2CC2(C(N2CCCC(O)C2C)=O)C1 C1(CNC(c2ccc(COC)o2)=O)CCN(C(C2OCCC2(C)C)=O)C1.O Cc1cc(C=CC(=O)NC2CC(C)C2)ccc1F.C1(C=O)CC(C)(C)CO1.N CCC(C)C(O)C(=O)NCC1(F)CCCN(C(=O)COCCOCCO)C1 C(C)(C)(C(C)CC(=O)NCc1ncccc1F)NC(CC(CC)C)=O c1(C(=O)NC2C(NC(C3(O)CCC(C)CC3)=O)CCC2)cc2sccc2cn1 N1(C(C(CC)(C)COC)=O)CCC(C2CC2)(CNC(c2cnc(Cl)s2)=O)C1 CC(CCC(=O)NC1C2CCCC12)NC(C12COCC1C2)=O C1(CC#C)(C(N2CC(CNC(=O)CCC(=O)OC)C(C)C2)=O)CCCCO1 C1(C(=O)NCC2N(C(c3cccc(CC)n3)=O)CC(O)C2)CC(C)(C)CN1C CCC(C(=O)NCC(N1CCN(C(c2cc(C)c(Cl)s2)=O)CC1)C)C(C)C C12(C(=O)NCC3N(C(C(C)NC(=O)C4CC4)=O)CC3)CCCN(CC1)C2 C1(CNC(C(C=C)O)=O)CC(C)(C)CN1C(=O)CN1CCS(=O)(=O)CC1 Cc1c(C(N2CCN(C(=O)C(C)N3CCC3)CC2C)=O)cncc1Cl C1(CCNC(C(CC)OCC)=O)CSCCN1C(c1ocnc1C)=O C1(C(N2CC3CC3C2)=O)CNC(=O)C(C)(C)C1.CC(C(=O)N)OC1CCOC1 C=CCC(F)(F)C(=O)N(CC(C)CNC(=O)C(CC)C1CCOCC1)C c1(C(=O)NC(CNC(Cc2n(C)cnn2)=O)(C)C)cccc2ccsc12 c1(NC(=O)C(C2(O)CN(C(=O)C(O)c3ccco3)C2)F)cccc(C(N)=O)c1 N1(C(C(C)OCC=C)=O)CC(C)CC1C(N1CCC(C)(O)C1)=O N1(C(CC(COC)NC(c2cc(C)nc(C)c2)=O)=O)CCC2(CNC(=O)N2)C1 CCCCCC1CC1.CC(C(=O)N(C1CC1)C(=O)O)n1ccnc1.C(C)(C)C CS1(=O)=NCc2c(-c3c(Br)cncc3F)cccc21 N1(C(c2n(CC#C)cnn2)=O)CCC2(CCN(C(=O)C(C)(C)CO)CC2)C1 c1(C(N2C(C)C(C)CC2)C(=O)NC2CCOC2)csc2cc(Cl)ccc12 N1(C(C2(O)C(C)(C)C2)=O)CCOC(Cc2cn(C)nn2)C1.c1ccoc1C(=O)O N1(C(C2(CC#C)CCOC2)=O)CC(NC(=O)CCCc2csc(=N)[nH]2)C(C)C1 c1(C(=O)NCCNC(=O)C(=O)NCC(F)(F)F)c[nH]ccc1=O C1(NC(c2cc(CNC(=O)CC(F)(F)F)ccn2)=O)CCCC12CC2 N1(C(C(C)C)=O)CCC(NC(c2ccc(C(C)(F)F)nc2O)=O)C12CC2 C(=O)(C1=C(F)CN(C(C23CCC(C2)OC3C)=O)CC1)NCc1ncc(CC)s1 Cc1ncoc1C(N1CCCC1C(C)NC(=O)C=Cc1nccs1)=O C1(NC(C)=O)CCC(C(N2CCCC2C)=O)CC1.c1(C(=O)N)cnoc1C(C)C C1(NC(C2(C)CCN(C(c3c(C)c[nH]n3)=O)C2)=O)CCCC(O)C1O C(=O)(C(O)CC(N)=O)NCCC1OCCN(C(C(CC)C2CCC(=O)N2)=O)C1 c1(C(C)=O)cc(Cl)c(NC(=O)C(=O)NC(C2CCCC(C)C2)CC)c(Cl)c1 C1(NC(C(CCSC)O)=O)CN(C(c2ncccn2)=O)Cc2nccn2C1 C1(NC(c2c(Br)nc(C)s2)=O)CC2CN(C(c3ccoc3)=O)CC2C1 C1(C(=O)N)CN(C(=O)CC2C=CCC2)CC(C)(C)C1.n1(CC)ncc(C)c1C N1(C(CNC(=O)OC)=O)CCC2CN(C(=O)C=C(C)c3ccccc3)C2C1 C1(N(C(CCC)=O)CCF)CCCN(C(=O)C=Cc2ccc(Br)o2)C1 N1(C(C(CC)Cc2cn(CC(=O)NC)nn2)=O)CCC(O)(C(N)=O)CC1 CC(C)S(=O)(=O)C(C)C(=O)N1CC2CCC1CN2C(=O)C(C1CCOCC1)O N1(Cc2nn(C)c(CNC(=O)O)c2)CCC12CCS(=O)(=O)C2.C(C)(C)C N1(C(C2CC(C#N)(OC)C2)=O)C2CCC1CN(C(=O)CSc1ccncc1)C2 N1(C(C2C(OC)CCCC2)=O)CC2CN(C(C3(CO)COC3)=O)CC2C1 CC1CCC(NC(c2ccc(-c3ncc[nH]3)nc2)=O)CN1C(c1ccco1)=O C(=O)(C1=CCCCC1)NC(C1(O)CN(C(=O)CN2CCCC2CO)C1)C CC(C)C(C(=O)NCCC(C)(C)CNC(C1CCCC12CC2)=O)C(C)C C=CCC(C)C(=O)NC(C)CNC(C1CC(=O)N(c2cn[nH]c2)C1)=O c1(NC(c2n(C(C(=O)OC)C)nnn2)C(C)(C)C)cccc(-c2nccn2C)c1 c1(C(N2CCN(C(c3c(F)ccc(C)n3)=O)C(CF)C2)=O)c([N+](=O)[O-])cnn1C C12(C(N(CCCN(C(C3(CC#C)CC=CCC3)=O)C)C)=O)CCC(C)(C1)OC2 CC1CC2CN(C(=O)COCCN(C)C)CC2N1C(c1nocc1Br)=O c1(OC)ccc(O)c(C(=O)NCCC2CCN(C(=O)C(C)C(C)(F)F)CC2)c1 Cc1cnc(CNC(=O)C(C2CC2)NC(=O)CCOCC(F)F)s1 CC(C)CC(CNC(=O)CC1CC=CCC1)NC(=O)Cn1ncccc1=O c1(CC(=O)N(CCN(c2nccc(C(F)(F)F)n2)C)C2CC2)c[nH]ccc1=O C=C=CC(C)C(=O)NC1CCCC1(C)CNC(c1ccc(Cl)cn1)=O c1(OC)ccc(C)c(C(=O)NC2CCN(C(c3occc3F)=O)C(C)C2)c1 c1(C(=O)NC2C(CN(C(C(C3CC3)SC)=O)C)CCC2)c(C)csc1C C1(NC(CC(CC)NC(=O)Cn2nnnc2C)=O)CC2CCCC2C1 C(CCCC(=O)NCC1(OC)CN(C(=O)CCCC2CC2)C1)OC C1(CNC(CC(=O)OC)=O)CC(F)CN1C(c1ncc(C(F)F)s1)=O n1(CC(=O)NC2CN(C(c3ncc(C)cn3)=O)CC23CC3)c(C)cc(O)cc1=O C1(NC(C2CC2(F)F)=O)CC2CCC1N(c1ncc(Cl)cn1)C2 c1(C(=O)NCC2CCN(C(c3ccc(C)nn3)=O)CC2)ccc(C)c(Cl)c1Cl C1(C(=O)NC2(C)CC(NC(c3c(OC)c[nH]n3)=O)C2)CC2CCCCN2C1 CC(C)(C)S(=O)CCNC(c1csc(Cl)n1)c1nnnn1C1CCOCC1 C(CCO)(C(F)(F)F)NC(C(C)N(C(=O)C(O)CN(C)C)CCC)=O CC(C)CC(O)CC(=O)NC(C)CCCNC(=O)Cn1cnc([N+](=O)[O-])n1 c1(CCNC(C(C2CC2c2ccccc2)N(CCCCO)C)=O)nccn1C n1(CC)cccc1CCNC(=O)NCC(CO)C1CC1 c1(C(N2C(CNC(=O)CSc3nc[nH]n3)CC2)=O)nccc2[nH]ccc12 C(CCC(=O)N1CCC(C(F)C(=O)N(CC(C)O)CCF)C1)OC c1(C(=O)NC(C2CCN(C(=O)C(C)N3CCC3)C2)C)ccnc2c1CCO2 c1(C(C(=O)NCC(C2CCC(C(=O)OC)CC2)(C)O)C)cccc([N+](=O)[O-])c1 N(C(=NCC1CCCOC1)NCc1ccc(F)cc1)CC1COC(=O)O1 Cc1cc(Cl)c(C(=O)NCC2C(O)C(O)CN2C(=O)CCC)cc1F.C(N)=O Cc1nccc(C(=O)NC23CC(C(=O)NCC4CCCC(F)C4)(C2)C3)n1 c1(OC)ccc(C(=O)NCCCCCNC(c2cccnc2C)=O)cc1C(C)C c1(C(=O)NCCCCC(C)NC(C=C(CC)CC)=O)cc(O)cc([N+](=O)[O-])c1 Cc1cccc(C(=O)C=CC(=O)NC(C)(C)C)c1.c1(CC=O)cnco1.N c1(C(N(C2CCN(C(C=C(CC)C)=O)C2)C)=O)ccn2nncc2c1 Cc1nc(O)c(C(=O)NC2CC2CNC(=O)C2=CCSC2)cc1Br N1(C(c2c(CC)nc(C)o2)=O)CC(NC(=O)CC2COCCO2)C2CC2C1 N1(C(c2cnc(CC)[nH]2)=O)CC2(C1)CN(C(C1CC3CC(O)C(C1)C3)=O)CCO2 C1(N(C(C(C)(C)C)=O)CC(=O)NC2CCOCC2)CN(C(=O)CO)C2CCCCC12 C(=O)(C1=NNC(=O)C1)N1C(CCC(=O)NC(COC)COC)CCCC1 C1(F)(CNC(=O)COCC(F)F)CC(NC(=O)C(O)c2ccco2)C1 c1(C(N2CC3(C(C(=O)NC(COC)C)C3)C2)=O)ccc(OC)cc1C N1(C(C23C(C)(C)OCC2C3)=O)CCC2(CCCC2CNC(=O)C2=CCCC2)CC1 c1(C(=O)NCC(C(C)(C)C)NC(c2cccc(C#C)c2)=O)occ2c1CCOC2 CC1(C)CN(C(C2CC3C(C2)C3(C)C)=O)C(C)CO1.C(=O)(C(O)CC(N)=O)N CC1CC(=O)NCCN1C(=O)CC1N(C(c2cnc(=N)[nH]c2)=O)CCC1(C)C CC(C)CCCCC(=O)NC1(C(=O)NOCc2nc[nH]n2)CCCC1C Cc1cnc(CNC(=O)CCC2(N)CC2)o1 Cc1cc(C(=O)N)c2n[nH]cc2c1.C12CC(C1)N(C(=O)CC1SC(=N)NC1=O)C2 Nc1ccc(F)cc1C(=O)NC1(CCO)CN(C(=O)CC2CCCCO2)C1 CC1(NC(C2CC2CF)=O)CCN(C(C2(c3ccccc3Cl)CCOCC2)=O)C1 CC(C)(CNC(=O)CN1CCCC1)CC(=O)NCCC1CC2CCC1O2 Cc1oc(C#N)cc1C(=O)NC(C)CC(=O)N(C)CCc1ncon1 N1(C(COC2(C)CCCC2)=O)CCCC2C1CCN2C(=O)C(C(C)(C)C)C1CCC1 CC(C)CC(C)(O)C(=O)NCC12CCC(CC1)CO2.c1(C=O)cnc(S)n1C.N C1(NC(c2cc(C)sc2-n2cccc2)=O)CC(C)CN(C(=O)Cc2nc[nH]n2)C1 CCC(O)C(C)C(=O)N(C)CCN(C)C(c1ccncc1O)=O C12(NC(C3(NC(CNC(=O)OCC=C)=O)CC3)=O)COCC(C1)C2 C1(C#N)(C(=O)N)CC12CCOCC2.Cc1cn(C(C)(C)C(=O)NC2CCC2)cn1 N1(C(CNC(=O)NC)=O)CCC(CNC(=O)CC(n2nc(C)cc2C)C)C1 N1(C(C2(CCOC)CC2)=O)CCC(C(C)NC(=O)C(C)n2cccn2)C1 C(N=c1[nH]c2ccc(N)cc2s1)C1CCCCN(C(C2(C)CC2(F)F)=O)C1 C1(C(=O)N)CCn2nnnc2C1.c1(SCC(=O)NCCC2CC2)nnc(S)s1 c1(C(N(CCN(C(=O)CC2CS(=O)(=O)C2)C(C)C)C)=O)cc(C)n[nH]1 N1(C(c2c(CC)cno2)=O)CC(CNC(C2(C)CCCCC2)=O)OC2COCC12 C(=O)(C#CC1CCCCC1)NC1CCN(C(c2cc(C)c(C)o2)=O)CC1O c1(C(N(CCNC(c2c(C)ccc(O)c2)=O)C)=O)ncnc2c1c(Br)cn2C c1(C(=O)NC2CCN(C(CCC(=O)NCC)=O)C2C)c(C)nn(C)c1N CS(=O)(=O)CCCC(=O)N1CCCC1C1CC1.c1(C=O)cc(C(F)(F)F)no1.N c1(OC)ncc(C(N2CCC(C(=O)NCCC(C)C)CC2)=O)c(C(F)F)n1 C(=O)CS(=O)c1ccc(Cl)cc1.c1(OC)ncc(C(=O)NCC)c(C(F)F)n1.N C1(C(N2CC(C(=O)NC(CC)C)C2)=O)C=CCCC1 N1(C(C(CC)(C)C)=O)CCC2C(CCCN2C(c2onc(C)c2C)=O)C1 N1(C(CCC2CCC(C)O2)=O)CCCC2(C1)CN(C(c1cc(C3CC3)cs1)=O)C2 c1(CC(=O)NCC(CCCC)NC(=O)C(COC)CC)c(Cl)c(CC)nn1C Oc1cc(Br)c(I)cc1CN(C=O)CCc1ccc2c(c1)OCO2 C(C(CC(F)(F)F)NC(=O)CC1CCOCC1)NC(Cn1nnc(C)n1)=O c1(C(N2C(CNC(C3NC(=O)C(F)C3)=O)CCCC2)=O)ccc2c(n1)CCOC2 C1(C(=O)N)CCn2c(cnc2C)C1.C(=O)(CC(C)(C)C(=O)NCCC(O)C)OC c1(C(N2C(CNC(C=CCCC)=O)CC(F)C2)=O)ccc2cnccc2c1 c1(CC(=O)NCC2CCCCCN2C(c2sccc2Cl)=O)ccc2nc[nH]c2c1 C=CCCCCCCC(=O)NCC(C)N(C)C(c1ccc(N)c(F)n1)=O CN1CC2CCN(C(=O)C(C3CCCO3)NC(c3cc(Cl)n(C)n3)=O)CC2C1 Cc1nnc2n1C(C(=O)N1CC3CC1CN3C(c1conc1C(F)(F)F)=O)CC2 Cc1nc(CNC(=O)C(C)NC=O)oc1C(=O)NCC(O)C1(Cl)CC1 N1(C(c2c(C)nc(Br)cc2)=O)CCC=C(C(=O)N2CCC3(C2)CC3(F)F)C1 c1(OC)ccccc1CC.c1(C=O)cn(C(C)C)cn1.C1(C(=O)N)CC1(F)Cl CCC(O)(CC(=O)N1CC(CNC(c2nocc2Cl)=O)C(O)C1)c1ccccc1 CC1CCCCC1(CO)NC(=O)C(O)C1CN(C(=O)CCCc2cnn[nH]2)C1 CC(C)CCCCC(=O)N1CC2CC2(CNC(c2nocc2Cl)=O)C1 Cc1c(CNC(C2CCC(C)N(C(=O)CCCCC=C)C2)=O)cccc1F.C#CC C12(NC(c3c(CCCC)ocn3)=O)CCN(C(=O)CC#N)CCC1C2 N1(C(=O)Cc2csnn2)CCC2CC12C(N1CCC1CO)=O C(=O)(CC(C)(C)C(C)(F)F)N1C(C)CC(CNC(C(CC=C)(C)C)=O)C1 C=CCC(C(=O)NC(C)C(CO)NC(c1ccc(=O)oc1)=O)C(C)(C)C C(=O)(CCCCC(=O)N(N1CC(OC)C2(CCC2)C1)c1cn(C)nc1C)OC N1(C(CS(=O)(=O)NCC)=O)CCCCC(C2CN(C(c3ccc(F)cn3)=O)C2)C1 C(=O)(C(CO)C(F)(F)F)N1CCN(CC2(NC(C(C)C3CCCO3)=O)CC2)CC1 n1(CCC)ncc(C(=O)NCCCC)c1C1CC1.C(=O)(CN(C)C1CC1)N N1(C(C(Cc2cc(Br)sc2Br)NC(C)=O)=O)CC(O)(C2CCC2)C1 CC#CCCC(=O)NCC(C)N(C(C1CCC(CC)O1)=O)CC N1(C(C(CC=C)CNC(=O)CCOC)=O)CC(F)(F)CCC1C C#Cc1ccc(C(=O)NCCC2CC2)cc1.c1(C(C=O)(C)O)cccc(F)c1.N C(C(C)CC(=O)NC1(CNC(=O)CO)CCCCC1)OC.c1ccc(O)cc1 C1(C(N2C(CNC(C(CC)F)=O)CCC2)=O)CC(=O)N(c2ccc(C)cc2)C1 Cc1cnc(NC(CNC(C2CCS(=O)(=O)CC2)=O)C2CCC2)nc1C N1(C(CSCC#C)=O)CC2CC(C(=O)NCCOCC(F)F)C(C2)C1 CC1CN(C(=O)CC2CCCC2(F)F)CCN1C(c1nonc1N)=O C12(C(=O)NC3CCCN(C(C4(OC)CCCC4)=O)C3)CCCC(CCC1)C2O CCCC(CC)CCC(=O)N(CCNC(=O)Cn1nc(C)cc1C(=O)O)CC CC1CN(C(c2ccc(=N)[nH]c2)=O)CC1NC(=O)Cc1cc[nH]n1 CN1CCC(C)(C(N2CCC(CNC(=O)CCO)C2)=O)C1=O.C1CCCO1.C N1(C(C(C)N(C(=O)C)C2CC2)=O)CCC(C)C1(C)C.c1(OC)ccn(C)n1 C1(C(N2C(CCNC(=O)Cc3cn[nH]c3)CCC2)=O)CC2C=CC1CC2 c1(NC(C2CCC(NC(=O)C=CCBr)C2)=O)ccccc1-c1nn[nH]n1 N1(C(c2ccc(CC)cc2O)=O)CC2(CCN(C(=O)C=CC3CCOCC3)C2)C1 c1(OC)ncc(CN2CC3C(C2)N3C(=O)Cc2ccc(Br)cc2OC)cc1Cl C1(NC(CSCC#C)=O)CCN(C(c2cccc(O)c2C)=O)CC1C CCC(CCCC(=O)N1CC(CC2CC2)C1)NC(=O)Cc1cccc(C#N)c1 Cn1cc(C(F)=CC(=O)NCC2CCOC2)cn1.C1(C=O)CC(F)(F)CS1.N n1(C(CC)CC)ccc(C(=O)N(CCCCN(C(=O)C=Cc2ncc[nH]2)C)C)n1 C(C)(CC(=O)N1CC(C(O)C(=O)NC2CCOC2C2CC2)C1)SC C1(NC(C2CC(OC)C2)=O)CC2CC1CC2C(=O)NC1CCN(C)C1 N1(C(C(=O)NCCOC)=O)CCN(C(=O)C(C)n2ccnc2)CC1CO C1(C2(O)CCN(C(C3CCOC3C(F)(F)F)=O)CC2)(NC(CCCC#C)=O)CC1 c1(CNC(C(C2CC(CC)C2)N(C)CCC2CCOCC2)=O)scnc1C Cc1nn(CC(=O)N(C)CC2(O)CN(C(=O)CC3(C)CC3F)C2)cc1Br c1(C(N(CC)CC2CCCN2C(=O)C)=O)cnn(C)c1F.C=O.C1CC1 N1(CC(=O)Nc2ccccc2C(F)(F)F)CCCC(NC(c2ccoc2)=O)C1 N1(C(CCc2nnc(C)s2)=O)CCCN(C(c2cc3n(n2)CCC3)=O)C(C)C1 c1(N2CCOCC(CNC(C(C)N(C)C)=O)C2)nc(Cl)nc2c1S(=O)(=O)CC2 n1(CC)cnc2c(NCc3ccoc3)[nH]c(=NCc3ccc(CO)cc3)nc12 c1(C=O)ncccc1.N1(C(C(C2CCC2)OC)=O)CC(O)(CC)C1.C(C)=O.N N1(C(c2cc(OC)c(Cl)cc2Cl)=O)CCc2ccccc2C(NC(=O)C(C)O)C1 N1(C(C2OCCN(CC)C2)=O)CCCCC2(C1)CN(C(=O)C(F)(F)CC1CC1)C2 N1(C(COCC=C)=O)CC(C(=O)NC(C)COCC2CC2)(CC)C1 CCCC(C)(C)C(=O)N1CCCC(CNC(c2ncsc2C)=O)CC1 C(=O)C(C)(C)CS(N)(=O)=O.C1CCC(C)(C)CC1.C=C1CC(C)(C(=O)N)C1 c1(NC(=O)NCCCONC(=O)Cc2ncc(F)cn2)cc2ccncc2[nH]1 c1(OC)ccc(CC(N2CCC2CNC(=O)C=Cc2scnc2C)=O)cc1Cl C(=O)(CC(C(F)(F)F)NC(=O)OC(C)(C)C)Nc1cn(COC)c(=O)cc1 CC(C)C(O)C(F)(F)C(=O)NC1CC(CNC(c2cc3cscc3s2)=O)C1 S(=O)(=O)(c1ccc(NC2CCN(CF)CC2)c(C#N)c1)N1C(COC)CCOCC1 C1(NC(c2ccc([N+](=O)[O-])s2)=O)CN(C(=O)CNc2ncccn2)CCC1F C1(N(C(CN(C2CCCCC2)C)=O)C2CC2)CC12CCN(C(=O)C)C2.C1CC1 S(=O)(=O)(c1c[nH]ccc1=NCC1CCSC1)N1CCCC(CCC)CC1 C1(CCNC(c2c(C)nn[nH]2)=O)COCCN1C(=O)C(C1(O)CCCC1)F C=CCC(C(=O)N1CC(C(=O)NCC)C1)C(C)C.c1(C(=O)N)cccc(O)c1F S(=O)(=O)(c1csc(C(=O)NCCCCN(C)C(C2(O)CCOC2)=O)c1)NC C1(C)(C=O)CC(C)(C)C1.c1(C(C)=O)ccc(C(=O)NCCC2CCCC2)o1 c1(OC)cccc(C(=O)NC2CCC(NC(C3OCCOC3C)=O)CC2)c1F c1(C=O)nc(O)nc(O)c1F.c1(C(=O)OC)cn(CC(=O)N)nn1.C1CC1.C c1(C(=O)NCCC2(O)CCN(C(CSCC)=O)C2)c(C)nn(CC)c1C c1(OC)cnnc(C(=O)NCC2CCN2C(c2c(C)n[nH]c2C)=O)c1 N1(C(C(COC(C)C)NC(=O)C(C)N=[N+]=[N-])=O)CC2(CCC(=O)N2)C1 C1(C(=O)NC(C2CCN(C(C3(CC#C)CCCCO3)=O)C2)C)CCCC(=O)CC1 c1(CC(N2C3CC(NC(C(C(CC)C)C)=O)(C3)C2)=O)cc(F)cc2c1OCOC2 C12(CC(=O)NCCC3CN(C(=O)CN4CCC(CO)CC4)C3)COCC(C1)C2 C1(NC(=O)CC(O)CNC(C2CNC(=O)N2)=O)CC2CCC(C1)O2 c1(NC(C(=O)NCC(C)N(C(COC(C)=O)=O)C)C)ccc(O)nc1 C1(C(=O)NCc2nncs2)(COC)C=CCN1C(=O)C(O)C(C)C c1(OC)ccc(C(=O)N(C)CCNC(c2cc(O)cs2)=O)s1 C1(NC(c2n(CCCC)nnn2)C2CC=CC2)CCCC=C1Br C(CCN=C(NC(C)C)N1CCC(c2csc(C)c2)C1)OCc1cccc(OC)c1 CCC(CNC(c1oc(C)nc1C)=O)(CC)NC(C1OCCO1)=O CC1(C)CC(NC(C23CCC(F)C2CC3)=O)CN1C(c1cc([N+](=O)[O-])n[nH]1)=O c1(NC(c2c(C)oc(CNC(=O)CC3CCCSC3)n2)=O)cc(C#N)ccc1O C1(C#N)(C(=O)NCCCN(CCCNC(=O)C(C)(C)CO)C)CCCOC1 CC1C(N(C)C(C2CCCC2NC(=O)Cc2ccn(C)n2)=O)CCCC1C c1(CC(N)=O)ccc(C(N2CCCCC2CCNC(C2CSCCS2)=O)=O)cc1 C1(CNC(=O)OCCC)CCN(CC(N2CCCCC2CC)=O)CC1 C1(OC(C)C(=O)NC2CCCC2CNC(C2CCOCC2)=O)CCCCCC1 N1(C(C(C)=C2CCCC2)=O)CCN(C)CC1CNC(c1cn(C)cn1)=O N1(C(CSCCC)=O)CC(CC(=O)NC2CCC(=O)NC2=O)CC1(C)C c1(C(=O)NCCN(C2CCCCC2)C(C(C)O)=O)ncoc1CCC(F)(F)F c1(C(=O)NCC(C(C)(C)C)NC(c2c(C)nn[nH]2)=O)cc2ccccc2oc1=O C(=O)(C(C)CC(C)C)NCC1(COC)CCN(C(=O)CCN2CCCC2)C1 N1(C(C2C(C)C2C)=O)CCCC(C)(CNC(=O)CSc2cccc(Cl)c2)C1 c1(C(=O)NCCCCCN(C(C(OC)OC)=O)C(C)C)cnc2ccccc2c1 Nc1ccc(-c2nc(C3(C4CC4)CCC3)n(C3CCOC3)n2)nc1 C(C=O)(C(C)C)NC(=O)OCC.C1(CC)CN(C(=O)C)CCO1.CC.N c1(C(N(C)CC2(NC(c3n(C=C)nnc3)=O)CC2)=O)cn2cccnc2n1 C1(NC(c2ccc(C)s2)=O)CN(C(C2(C)CC3(CC3)C2)=O)CC1C C1(C(N2CCC(SC)C2)=O)C2CC3C(C2NC(=O)CC2CCCSC2)C13 C1(C(N2CC3CCC(CC3)C2)=O)C2CC(O)C(C2)N1C(=O)Cc1cccnc1F N1(C(c2ncn(C(C)(C)C)n2)=O)CCC(C)(NC(c2ccc(Cl)s2)=O)C1 Cc1c(CCC(N2CCC(CCNC(c3coc(O)n3)=O)C2)=O)cnn1C C1(O)(C(C)NC(=O)CCS(C)=O)CCN(C(=O)CC(C)(C)c2cccs2)CC1 CC(CC(=O)NC1CCCC1(C)NC(C1COCC1(C)C)=O)C(C)(C)C c1(C(N2CCC(C(C(=O)N(CC=C)CCO)F)C2)=O)ccc(C)n1C C1CCc2nc(C(F)(F)F)cn2C1.c1(C(=O)O)cccc(C(O)CNC(=O)N)c1 CC(C)CC(O)C(=O)N1CCOCC1CN(C)C(C1CC2(CC2)CN1C)=O C1(C(=O)N)CCN(C(C2CCCNC2)=O)C(C)(C)C1.C(=O)(C(C)C)NCC Cc1cc(-c2csc(=NCC3(O)CCOC3C)[nH]2)n(C)n1 C=CCC(C(=O)NCC(C)C(C)C)C(C)C.c1(CC=O)ccc(C(N)=O)nc1.N C1(C(N2CCC(CN(C(c3c(OC)c[nH]n3)=O)C)C2)=O)CCC2(CCC2)OC1 C(c1cnc(C)nc1O)=CC(N1CC(CNC(CCCC#C)=O)C2(C1)CC2)=O N1(C(C(c2cn(C)nn2)NC(=O)C(O)CN2CCCC2)=O)CCC2=C(CCCC2)C1 N1(C(c2c(OC)n[nH]c2)=O)CCN(C(=O)CCC(N)=O)CC1CC(F)F c1(CCOC(c2cnn(C3COC3)c2)=O)cc(Cl)cc(Cl)c1 C1(C(=O)NCCc2cnc(C)[nH]2)(C(C)C)CCN(C(=O)C(C)NC=O)C1 c1(C(=O)NCCCNC(C2C(C3(C)CC3)C2)=O)ccc(F)c(Cl)c1 c1(C(N(CCN(C(C2C(CCC)CCC2)=O)C)C)=O)nc(Cl)cc(N)c1Cl c1(C(=O)NCC2(C)CCN(C(C(C)=C3CC3)=O)C2)ccc(C(C)C)nc1O c1(OC)ccnc(OC)c1C(=O)NC1CN(C(C2(C)CC(C)=NO2)=O)CCC1F C1(NC(CC2CN(C)C2)=O)CCC2(CC1)CN(C(C1CCCC(F)(F)C1)=O)C2 C1(O)(CCNC(=O)CC2COCCOC2)CCCN(C(=O)CC2CC3(CC3)C2)C1 N1(C(CC)=O)CCCC(C(=O)NC(C)CN(C(=O)CCn2ccnc2)C)C1 C1(CCCC)CN(C(c2cncc(C#N)c2)=O)CCN1C(c1cccc[n+]1[O-])=O C(CCC(=O)N1CC2(C1)CC2(F)F)(C(C)C)NC(C1C(OC)CCC1)=O N12CCC(O)C(C1)C2=O.N1(C(=O)NCCOC(C(=C)C)=O)CCC(O)C1 C(=O)(CC1=CCN(C)CC1)N(C(CNC(C1C(C(C)C)CCO1)=O)C1CC1)C C1(C)(CNC(c2c(C)n(C)nc2)=O)CCCN(Cc2ccc(O)cc2Cl)C1 C1(C(=O)NCC(C)(CO)NC(c2cnn(CCO)c2)=O)CC12CC(F)(F)C2 CCCCCC(O)C(=O)NC12CCCC(NC(C3CCC(C(C)C)CC3)=O)(C1)C2 C(CCC(C)(C)C(=O)NCCCC1CNC1)OC N1(C(c2cccc(CN(C)C)c2)=O)CCC(C2CC2)(C)C1.C(=O)C1=CCCS1.N C=C(C)CCC(=O)N(C1CCCN(C(c2oc(C)nc2C(F)(F)F)=O)C1)CC CCCC(C#N)C(=O)N1CC(c2ccccc2)(NC(c2ncc[nH]c2=O)=O)C1 C1(CCC)CC(C(N2CC(C)(NC(c3cc(Cl)c[nH]3)=O)C2)=O)CCO1 N1(C(c2cnn(C)n2)=O)CCCC2CN(C(C3(S(N)(=O)=O)CCCC3)=O)CCC12 c1(C(=O)NC2C(C)(C)CN(Cc3ccccc3Br)C2)cnc2cccnn12 C1(C(=O)NCC2CC(NC(CCOc3ccc(C)cc3)=O)C2)CCOCC1(C)C Cn1nc(I)cc1S(=O)(=O)N1CCCCC1COC(=O)NC1CC1 C(C(C(=O)N1CC(CO)(CF)C1)C(C)(C)C)NC(CC(=O)OC)=O C(C1=CCCN(C(=O)C(F)(F)C(O)C2CC2)C1)NC(C(C)OCC#C)=O CC1(CNC(=O)COCCCF)CC(F)(F)CN1C(c1cnc2n1CCC2)=O C12(NC(C(CC=C)NC(C)=O)=O)CCN(C(c3ccc(=O)n(C)c3)=O)CC1C2 N1(C(c2nn(C)c(O)c2)=O)CCCC(C)(CNC(C2CC3CC(=O)C2C3)=O)C1 CN1CCCC1C=CC(=O)NCCc1ccc(C)cc1.C1(C=O)CC(C)(F)C1 N1(C(C2CCC(CC)CC2)=O)CC(C(=O)NCc2cnoc2)CC(C)(C)C1 CC1C(N=c2[nH]c(=NCCC34CC(CCO3)C4)[nH]c3c2CSC3)CCCN1C N1(C(c2ncn(C(C)C)n2)=O)CCC(C)(C(=O)NC2CCOCC2F)CC1 CC1Cc2cc(Cl)ccc2N1S(=O)(=O)c1cccc(N(C)Cc2cnn(C)c2)n1 N1(C(C2CC3(CN(C(c4cc(C)[nH]c4)=O)C3)C2)=O)CC=C(c2ccccc2)CC1 c1(C2(CNC(C(=O)NC(CC)CCOC)=O)CC2)c(OC)cccc1F C1(N(C(=O)Cc2ncc(C)o2)CC)CCCN(C(c2ccn(CC)n2)=O)C1.O C(=O)(C(C)(C)CC(C)(C)C)NC.N1(C(c2c(C(C)C)scn2)=O)CCC(O)C1.C Cc1nc([N+](=O)[O-])cn1CC(N1CC(NC(C2CCN(C)CC2)=O)C(C)(C)C1)=O c1(C(N2CC3N(C(c4nc(C)nn4C)=O)CC(C3)C2)=O)cnn2cccc(C)c12 c1(C(=O)NC2(CC=C)CN(C(C3CCCSC3)=O)C2)cnc(C)n1C N1(C(CCC=C=C)=O)CC(F)(F)CC1C(=O)NCCCCn1ccnc1 CC1(C)CC2(CC2C(=O)N)C1.C1CN(C(C2(C)CC(F)(F)C2)=O)CC12CC2 N1(CCC=O)CCC(F)C1.CCC(=O)N(CCCN(C)C)CC.CC(C)CO C1(C(=O)NCc2n(CCC)ncn2)C=CCCN1C(=O)COC1CCOC1 N1(C(CC(=O)OC)=O)CCN(C(=O)CC(C)c2ccncc2)C2(CC2)C1 N1(C(C(CCC(C)C)NC(c2nocc2Cl)=O)=O)CC2(C1)NC(=O)NC2=O C1(C(=O)NC2CC3CN(C(c4nc(C)n(C)c4)=O)C2C3)CCc2[nH]nc(O)c2C1 C1(CC(=O)N)N(C(C2CCC(C)(C)C2)=O)CCC1(C)C.CN(CC)C1CC1 c1(OC)cc(C(=O)NC2CC23CCC3)cnc1.C1(=CC=O)CCC(C)C1.N C(=O)(C(CN(C)C)NC(C1CCCOC1)=O)NCC(C)CO c1(OC)cc(CO)ccc1C(N1CCC1CNC(C1(CO)CC1)=O)=O N=S1(=O)CCC(C(=O)OCCCOc2ccccc2Br)CC1 CC(C)CC(C(=O)NCCN(C(C1CC1C1CC1)=O)C1CC1)c1ccccc1 c1(CCC(=O)N(C2CCN(C(=O)C(F)CC3CC3)C2)CCC)ccccn1 CC(C)CC(C(=O)N(CC(C)CO)C)NC(=O)C(C1CC1)C1CC1 c1(C(N(CCNC(C2CN(C)C2)=O)C)=O)cccc(-n2ccnc2)c1 CN1CCC(O)C(NC(c2ccc(-n3cc(CC(=O)O)nn3)cc2)=O)C1 N1(C(C2CN(C(CC)=O)CC23CC3)=O)CCc2nc(O)[nH]c2C1 N1(C(CN(C)C2CC2)=O)CC2CCC1C(C)C2.c1(C(=O)N)coc(N(C)C)n1 c1(SCC(=O)Nc2ccc(C)cc2C)nc(O)cc(C)c1C#N C=CC1CC(NC(=O)COCCNC(=O)C(C)(C)OC)CCO1 c1(C(=O)NCCCCNC(c2c(CC)n[nH]c2)=O)sc(C2CCCCC2)nc1C N1(C(C2(CC=C)CN(C(c3cccc(=O)o3)=O)C2)=O)CCC(C2=NOCC2)C1 C(=O)(C1CCC(N)c2ccccc21)NC(c1ccc(C)c(F)c1)C CC1CCCN(C(=O)CCN2CCCCC2)C1CNC(=O)C(C)(Cl)Cl N1(C(C=CC(=O)OC(C)(C)C)=O)CCc2ccccc21.n1(CC=O)ccnc1 N1(C(C(c2ccc(C)o2)C)=O)CCCC(CNC(c2ccncc2Br)=O)C1 c1(C(=O)NC23C(CN(C(c4c(C)coc4C(C)C)=O)C2)C3)c(F)cccc1F CCC(F)(F)C(C)(C)C(=O)N(C)CC1CCN(C(=O)CN2CC3CC3C2)C1 N1(C(CCC(=O)NC)=O)CCN(C(c2ncccc2F)=O)C(c2ccncc2)C1 c1(OCC(CNC(C2C(C(=O)OC)(C(C)C)C2)=O)O)ccc(Cl)cc1C c1(C(=O)NC(CN(C(C(CC=CCC)C)=O)C)C)cc(C)c2[nH]cnc2c1 N1(CC)CC(C(=O)NCCCCNC(=O)CONC=O)NC1=O.C(C)(C)C CC1=C(C(=O)NC(C2CC(NC(C3CC3(C)C)=O)C2)C)COCC1 C1(CNC(C(CSC)(C)C)=O)CC2(CCC2)CN1C(C1CCCCS1)=O c1(C(=O)NCC2(C(C)NC(C(CCOC)C)=O)CC2)ccc(O)nc1Cl c1(C(=O)NC(C2CCOC2)CNC(=O)CCN2CCOCC2)cccc(CO)n1 C1(CNC(C2=C(C)OCC2)=O)CN(C(c2ccc3c(c2)CCO3)=O)CC(C)(C)O1 c1(N(C)CC)ccnc(N2CCN(C(C3(O)CCCCC3)=O)CC2)n1 Cn1cc(C(=O)NC)c2cc(Cl)ccc12.C1(C(N2CCC2)=O)CC2COCC(C1)C2 c1(NCC2(C)CCS(=O)(=O)CC2)ccc([SH](=O)=O)cc1F.C1CCOC(C)(C)C1 c1(C=O)cc(C)sc1C.C(=O)(C(C1CC1)NC(=O)C)NC.C(C)(C)C N1(C(C2CCN(C(=O)c3ncn(CC)n3)O2)=O)CC=CCC(C)(C)C1 Cc1cnc(NC(=O)C(C2CCN(Cc3ncc(Cl)s3)CC2)C)c(Cl)c1 C1(OC)CC(C(=O)NC2(C)CC(F)(F)C2)C12CCC2.C(=O)CSC(F)F c1(NC(C(c2ccccc2)C)C)ncc(S(=O)(=O)NCCCCCCSC)cc1Cl c1(C(=O)NC2(O)CC(NC(CCCN(C)C)=O)C2)ccncc1.C(C)(C)C.C Cn1cc2c(n1)CCCC2C(=O)N1CCN(CCS(C)(=O)=O)CC1 C1(NC(COCC#C)=O)CC(NC(=O)C(c2ccccc2)O)CC1O C(=O)(CC(F)(F)C(F)F)NC(CC(C)C)CNC(=O)CC1COC(C)CO1 Cc1ccc(C(=O)NCC2CCN(C(C3(C)CCC(=O)CC3)=O)CC2C)c(C)c1 C1(NC(C2C(C(C)C)C2)=O)CCOCC1C(=O)NCCCC1CCCC1 C1(C(=O)N)CCCCC1(C)C.C(=O)(CCCN(C)C)NCCOCCOC c1(NC(N(c2ccc(-n3nccn3)cc2)C)=O)ccccc1CS(C)(=O)=O c1(OC)nc(-c2ccc(CO)c(C)c2)ccc1C(=O)NCCc1ccco1 N(C1CN(C(c2cscc2F)=O)CCc2ccccc21)C(C1N(C)CCOC1)=O C1(C(=O)N(C(C)C(C)C)C)(OC)CCN(C(c2ccncc2F)=O)C1 N1(C(C(CNC(C2CC3OC2C2CC32)=O)OC)=O)CC2C=CCC(C2)C1 CCC(CC)CCC(=O)NCC1CC(CNC(c2cnn(C)n2)=O)CO1 C=CCC(CC(=O)NCC(CO)C(C)C)NC(C1CN(C2CCC2)C1)=O C1(CNC(C=CC=CC)=O)CCN(C(=O)CN(CC(=O)N)C)CC1C N1(C(CCOCCOC)=O)CC(C(N2CCCC(C(=O)OC)C2)=O)OC(C)C1 c1(C=O)cnn(C)c1C1CC1.C(C)CCC.C1(C(=O)NC)(C(=O)N)CCC1 CC1CS(=O)CCN1C(C1CNC(=O)CN1C(c1ccc([N+](=O)[O-])[nH]1)=O)=O C12CC(C1)CCO2.Cc1cc(C(=O)NC)c(C)[nH]1.C1(CC=O)CCCC(C)O1 C(=O)(C1CN(CC2CCN(CC(C)O)CC2)Cc2c(C(F)(F)F)cccc21)OC c1(C(=O)NCC2(C)CC2)nc2n(c1Cl)CCCC2.c1(C(C=O)F)ccccc1 N1(CC2N(C(C(F)(F)Sc3cn(C)nc3)=O)CCC2)CCC(O)(C(F)(F)F)C1 c1(CC)ccc(C(=O)NCC(C)(CO)NC(C2CN(C)CCO2)=O)c(C)n1 c1(NC(C2(F)CCN(C(CCc3c(C)cccn3)=O)C2)=O)cc(Br)ccc1C C(=O)(CC1CC(=O)c2ccccc21)N(CCNC(Cc1c(C)nc(Cl)cc1)=O)C C1(C(=O)NCCOC2CN(C(C(CC#C)CC#C)=O)C2)Cc2c[nH]cc2S1(=O)=O N1(C(Cc2ccc(C)cc2)=O)C2CCC1CC(NC(=O)CCc1csc(C)n1)C2 N1(C(C2(CCOCC)CCCC2)=O)CCC(NC(=O)C(C)C)C2(CCC2)C1 C1(C(N2CCCC(Cc3nc(C)on3)C2)=O)CCC2(CCC2)NC1 N1(C(C(c2ccccc2F)OC)=O)CC2CC2(NC(c2ccnnc2O)=O)C1 c1(C(N2CCN(CCNC(C(C=C)O)=O)CC2)=O)nccc2ccccc12 CN1CC(O)CCC1C(N1CCC(N(C(=O)CS(=O)(=O)N(C)C)CCO)C1)=O C1(NC(CS(CC)=O)=O)CCC2(CCN(C(c3cncc(Cl)c3)=O)CC2)C1 C(CNC(C1CC(CC(F)F)C1)=O)(C(C)(C)C)NC(CNC(C)=O)=O Cc1oc2nc(Cl)ccc2c1C(=O)NCC1CCC1.c1(C(=O)N)ccn(C)c1C N1(C(C(C)(C)NC(=O)COc2ccsn2)=O)CCOCC(C2CC2)C1 C1(C)(C(=O)NC(C)CN(C)C(c2cc(Br)n[nH]2)=O)CC(C(C)(C)C)=NO1 C1(O)(C(=O)NCC2(CC(=O)NC3C(C)COC3)CC2)CCOC1(C)C S(=O)(=O)(C1CC(CF)C1)N1CCC(c2ccccc2)(C(=O)OC)C1 C1(NC(C(c2ccccc2F)C)=O)CCN(C(C2CC2C)=O)CCC1CO c1(N2CCC(CCC)C2)nnc(C(C)[N+](=O)[O-])n1CCS(=O)(=O)N(C)CC c1(CC(N2CC(CNC(C#CC3(C)CC3)=O)C(C)(C)C2)=O)c[nH]c2cnccc12 c1(C(N2C(C3CCN(C(C(CCC)F)=O)C3)CCCC2)=O)cn2cccnc2n1 CCCCCS(=O)(=O)CC(=O)NC1CC1CNC(c1cc(Cl)ccc1C)=O N(C(=NCCN1CCNC1=O)NCc1ccoc1)CC(C)(C)C C1(NC(CC(CC)C)=O)CCCN(C(c2c(F)cccc2Br)=O)CC1 C1(C(=O)NCC(COC)O)CN(C(c2cc(C)cc(O)n2)=O)CC1(F)F c1(CN(CCF)Cc2cnc(Br)c(Cl)c2)cc2ccccc2s1 N1(C(c2[nH]cc(C(C)=O)c2)=O)CCCC(CNC(c2coc(Cl)c2)=O)CC1 C12(OC)CCC1CN(N1CCOCC1C1CCC1)C2 CC1C(CO)CCN1C(=O)NCC1(C2CCCO2)CCC1 C12(NC(CN(C(=O)CSC3CC3)CC#C)=O)CCCC1OCC2 Cc1oc(C#N)cc1C(=O)NC(C(=O)N)c1ccoc1.c1cc(F)cc(F)c1.C c1(C(C)=O)ccc(C(=O)NOCC2CCCO2)cc1F N1(C(C(C)(C)OC)=O)CC(NC(c2cnoc2C)=O)C(O)C1.[SH](C)(=O)=O.N C1(N(C(C=CC(=O)OCC)=O)C)CC2(C1)CC2C=O.C1CCNC1.N C(=O)(C(C)(C)CC(F)F)N1CCC(C)CC1.c1(CC)ccc(N)c(C(=O)N)c1.C CCCCCC=CC=CC(=O)NC(C)C1CCC1.n1(CC(=O)N)cccn1 C1(CO)C(c2ccccc2)CCN1Cc1cnn(C2CC2)c1Cl C(c1ccc([N+](=O)[O-])s1)=CC=O.CC1(C)CCC(C(=O)N)OC1.C(C)(C)CC C(N=c1[nH]c2c(F)cccc2o1)C1C(C)(C)CN(C(=O)C(N)=O)C1 N1(C(c2c(C)cco2)=O)CC(NC(=O)C(C2CCCCCC2)C)C(C(F)F)C1 c1(N(CCC)CCNC(=O)C(c2cccc(Cl)c2)CC)nccc(C#N)n1 c1(OCCC)cc(F)ccc1NC(=O)C(=O)NC1CC(N(C)C)C12CCC2 C1(O)(C(=O)N)CCCC(C)(C)C1.CC(C)C(C(=O)N1CCC(C)(C)C1)N(C)C N1(C(c2ccc(SC)cc2)=O)CCCC2(CCN(CC#N)C2)C1 C(C)(C(=O)NCCC1(CNC(=O)C(C)OCC)CC1)OCC C1(CCC)CN(C(=O)OC(C)(C)C)CCN1C(c1cc(I)c[nH]1)=O C(=O)(C1CCc2nccn21)N1C(C)(C(=O)NCC(C(=O)OC)C)C=CC1 CC(CO)CCCNC(=O)C(C(C)O)NC(c1cc(Cl)cn1C)=O c1(C(=O)NC2CC(C)(NC(COC(CC)C)=O)C2)ccnc(P(C)(C)=O)c1 N1(C(c2ccon2)=O)CCN(C(C2(c3cc[nH]n3)CC2)=O)C(C2CC2)C1.CO.C C1CCN(C(c2cccc(C(N)=O)c2)=O)C12CC2.C(C)(C)(CC(=O)NC)OC C1(C(=O)NC2(CN(C(C(C)(C)OC(C)C)=O)C)CC2)CC(C)N(C)C1 C1(C(=O)NC2C(C(=O)NC(C)Cc3ccco3)CC2)CC(=O)OC1(C)C CCCC(CC(=O)N(C1CC2CC2C1)C)NC(c1ccccc1CC#N)=O CCC(CC(C)C)C(=O)NC(CNC(c1ocnc1C1CC1)=O)CC(F)(F)F O=C(N=c1cc(C2CC3CCC2C3)[nH][nH]1)C1CCN1Cc1cccc([N+](=O)[O-])c1 CC1CN(C(=O)C(F)C2CC2)CCN(C(C2C(CN=[N+]=[N-])C2(C)C)=O)C1 CCC(C)C(C)C(=O)NC(C(=O)NC1CCN(CC)C1)C(C)(C)C C12(NC(C3CCC(C)CC3)=O)CCOCC1CN(C(=O)CN1CCSCC1)C2 N1(C(C2CC(NC(c3n(CC)ncc3C)=O)C(O)C2)=O)CCc2ncn(C)c2C1 c1(CNC(C2(C#C)CC2)=O)ccc(C(=O)NCc2ccc(C)o2)s1 c1(C(N2CCCC(NC(c3c(C)cc(C)[nH]3)=O)CC2)=O)cc2cccnn2c1 N1(C(c2c(C)nsc2)=O)CCCN(C(=O)C(C)n2cnnn2)CC1C(C)C C1(NC(c2cc(COC)on2)=O)CC2CC1CN(C(c1n[nH]cc1[N+](=O)[O-])=O)C2 c1(CCC)nccn1CC(=O)N(S(=O)(=O)CCn1ccnn1)CCC#N CC(C)(C)C(C)(C(N)=O)NCC1(O)CCCCC1 C1(F)(C(N(C2(CC(=O)NCCS(CC)(=O)=O)CC2)C)=O)CCC(C)CC1 N1(C(CCNC(CCCOCCOC)=O)=O)CC2C3C=CC(O3)C2C1 C1(CNC(c2ccc(C)c(Cl)c2Cl)=O)CCCC2(CN(C(=O)C3=CCCC3)C2)O1 C1(NC(c2cc[nH]c2)=O)CN(C(C2(c3ccccc3)CC2)=O)CC12CCCC2 CCCCC(CC(=O)NC(c1ncc(F)cn1)C)NC(C12CCC(OC)C1C2)=O C(CCC)(C(=O)NCC(c1ccccc1)CNC(=O)C(C)O)=CCC C1(C)(OC)CC(NC(=O)CC(C(C)C)NC(C2(C3CC3)CC2)=O)C1(C)C c1(C(=O)NCCCN(C(C2CCC(CC)C2)=O)CCO)ncc(F)cc1C c1(C(N2CCC(N(C(C=CCC)=O)C)C2)=O)cc(C)cc2c1NCCC2C C1(OC)(CO)CCN(C(=O)CNC(=O)CC2OCCO2)C1 c1(C=O)cc(Cl)cc(F)c1F.C1(NC(C(C)(O)C2CCC2)=O)CC2(C1)CCC2.N C12(C(=O)NCCCCNC(CN(C)Cc3ccccc3Cl)=O)CCCC(C1)OC2 CCC1=NOC(C(=O)OCCNC(N2CCCC2)=O)C1 C(=O)(C(CCC)OCC)NC(C(=O)NC(CCC)c1ccco1)C C(C1CCOC1)=CCNC(C(c1cccnc1)NC(C(C)C1CCC1)=O)=O C1(CNC(c2ccc(O)nc2)=O)CCN(C(c2cnn(CC(F)F)n2)=O)CC1 CC1(c2ccccc2)CN(C(=O)Cn2cc(COc3ccccc3)nn2)C1 c1(CC(=O)NCC2CCCN(C(CCC3(C)CC3)=O)CC2)ccc2nc(O)[nH]c2c1 C(=O)(N=c1ccn(-c2ncccn2)[nH]1)N1CCC(C(C)(C)C)OCC1 N1(C(C(C)CCN(C)C)=O)C2CCC1(CNC(C1CCCC1(F)F)=O)CC2 CN1CCN(C(C2CC2C(N)=O)=O)CC1C(N1CC(O)(CO)C1)=O CCC(CCCC(=O)NC(C1(O)CCCC1)(C)C)NC(=O)CC(Cl)Cl CC1CN(c2cc(N3CCN(C4CCCC4)CC3)ncn2)CCC1(F)F Cc1occc1C(=O)N(CC(C)NC(=O)C(Cc1ccccc1)n1cnnn1)C C(C(=O)N1CC(O)CCO1)C1(C(N(C)C(c2cnc(=N)[nH]c2)=O)=O)CC1 N1(C(=O)NCCOC)CC(C#N)C2(CCC2)C1 Cc1ccc(C=CC(=O)NCCNC(c2ccccc2-c2ccccc2C)=O)o1 C(C(C)(C)C(=O)NC1CCOC(C(C)C)C1)N(C(Cn1ccc(C)c1)=O)C Cc1cc(O)cc(O)c1C(N1CCCC(CN(C(=O)C(C)n2cccn2)C)C1)=O c1(OC)cccc2cc(C(C(=O)NC3CCOCC3)N(C)CC3CCSC3)oc12 C12C3CN(CC13)C(=O)c1ccnc(c1)C2.n1(CC)nnnc1C1CCCC1 c1(C2C(NC(=O)C=Cc3ccco3)C2)cccc(Cl)c1 C(=O)(C1=NNC(=O)CC1)N1CCC(CC=C)(NC(c2conc2C2CC2)=O)C1 CCCC(C)(CC)C(=O)NCc1ncoc1CCNC(C1CCC(=O)N1)=O C1(C(N)=O)CCN(C(c2csc(Br)n2)C(=O)NC2CCN(C3CCCC3)C2)CC1 CN1CCC(C)(C(=O)N(CC(CO)(CO)NC(=O)Cn2cccnc2=O)C)CC1 c1(C(=O)NC2CCC(NC(=O)CCCC3CC3)CC2)cc(Cl)ncc1O C(C(C(=O)NCCCCOC)NC(c1ncccn1)=O)OCC C#CC1CCCC(CNC(=O)C(c2ccco2)NC(=O)CC(=O)OCC)C1 c1(OCC)nccc(C(=O)N(CCCCNC(=O)CO)C)c1F.C1CCCOC1 c1(C(=O)NC(C(=O)Nc2c(C)ccnc2)CCF)c[nH]c2cnccc12 Cc1nc(O)nc(O)c1CC(N1CCCCCC1CNC(C1CC1F)=O)=O ClC1=CCCc2nc(CNc3cnn4c(C(C)(C)C)ccnc34)ccc21 c1(CC(N2CC(C(C)NC(c3ccc(=O)oc3)=O)OCC2)=O)c(Cl)cccc1Cl CCC(CC)(CCNC(=O)C(C)Sc1ccc(OC)cc1)NC(c1ccsc1)=O c1(NC(CNC(CCCCCNC(C)=O)=O)C2CC2)ncc2scc(Br)c2n1 c1(C(=O)NCC(CO)NC(C(CC)C2CCOCC2)=O)sccc1S(N)(=O)=O Cc1ccc(C(c2nnnn2-c2ccccc2Br)NCc2ncco2)cc1 c1(C(N2CCC(CN(C)C)C2)C(=O)NCC=C)cnc(C)nc1 O=C1CCC(C(=O)NCc2cc(C(=O)NCCCC3CC3)no2)N1 c1(COC(c2cc(OCC)ccc2)=O)ccc(C)n(C)c1=O.c1ccccc1.O c1(CNCC(C)(C)C)ccc2ccccc2n1 c1(C(=O)NC2(CO)CN(C(C3C4CCCC34)=O)C2)cccc(SC(F)(F)F)c1 n1(CC2N(C(c3ncc(I)s3)=O)CC2)cc(CCC2CCCCO2)nn1 c1(C(N(CCC2CCN(C(CS(CC)=O)=O)CC2)C)=O)cc(C)c(CO)cn1 C12(C(=O)OC)CC1CN(C(=O)CCC1CC1)C2.C1(C(=O)N)CCS(=O)CC1 c1(CCCC(=O)Nc2cc(Cl)ccc2I)ccc2c(c1)OCO2 N1(C(C(=O)NC2CC2)=O)C2CCC1C1CC1(NC(c1cccc(CO)c1)=O)C2 CCC(C)(CO)C(=O)NCC1(O)CCN(C(=O)CC2(C(F)(F)F)CC2)C1 N=c1[nH]c2cc(C(N3CCC(NC(=O)CCN4CCC4)C(O)C3)=O)ccc2s1 C1(NC(CCn2ncc(C)c2)=O)CC(C)CN(C(=O)CC2COCC2(C)C)C1 C(=O)(C(O)c1cnc[nH]1)N(CC(C)O)CCNC(=O)C=CCO c1(C(=O)NCC2(C)CN(Cc3ccccc3C#N)C2)cc(I)c(O)c(I)c1 CCC(C)C(O)C(C)C(=O)NC1CCCCC1CC(=O)NC1(C)CC(O)(CO)C1 CCC(C)(C(=O)NCc1ccc(CCNC(=O)CCC(C)OC)cc1)C(N)=O C(COC(C1CCN(C(=O)CN2CC(=O)NC2=O)CC1)=O)(c1ccccc1)OC CC(C)CC(C(=O)N(C)CC1CN(C)CCO1)N(C)C(C1CC(=O)C1)=O C12(C(=O)NCc3ccc(C)cc3)COC(C1)C(NC(=O)C(C#N)C(C)C)C2 Cc1cc(C(N2CCOC(C(C)NC(=O)CCC(C)(C)O)C2)=O)c(N)c(C)c1 C1CCCN(CC(F)F)C1.c1(COC(C)C(=O)N)cn(C2(C(N)=O)CC2)nn1 c1c(F)cccc1F.C(=O)(CC(C)C)N.c1(C(=O)OC)cnc(CN2CCC2)o1 C1(C(=O)NCCNC(=O)OC)CC2(CC(NC(=O)CCF)C2)C1 CCCC(C)(C)CC(=O)N1CCC(C(=O)NC(c2c[nH]ccc2=O)C)C1(C)C c1(OCC)nc(C)ccc1C(=O)NC1CCN(C(C2CC(O)C2)=O)C12CC2 N1(C(C)C)C(=O)COCC1C(=O)NC1CC1C.C(=O)C.C(=O)C1CC1 C(C(CO)C(C)C)NC(CNC(c1cc(C)[nH]c1)=O)=O c1(OCC(=O)NC(CNC(COCCOC)=O)CO)ccccc1[N+](=O)[O-] CCCCC(CC)C(=O)NCC(CO)NC(C1CC(NS(C)(=O)=O)C1)=O C=CCCCCC(=O)NC(CCC=C)C(=O)NC(C)CC=C N1(C(c2c(C)coc2C)=O)CCC(C)C(NC(=O)Cc2sc(O)nc2O)C1C C1(NC(C(CC)O)=O)COC2CN(C(=O)COc3cccc(C)c3)CC12 CCCCCCC(F)C(=O)NC1CC2CC(C1)N(C(c1cncc(OC)c1)=O)C2 c1(C2C(C)C2)nnc2ccc(N3CCCN(C(c4ccco4)=O)CC3)nn12 CC1CC(=O)NC1C(=O)NCc1csc(C(=O)NC)c1.c1nccc(O)n1 C1(NC(C(NOC)=O)=O)CCCC12CN(C(c1sncc1C)=O)C2 c1(NC(CC)COCC(F)(F)F)nc(C)cc(=NCc2cc(Cl)ncc2Cl)[nH]1 Nc1cnc(C(F)(F)F)cc1C(=O)NCCCCCNC(=O)C.C(N)(=O)N c1(COC)ncc(C(=O)NC2COCC2NC(=O)CS)s1.c1ccccn1 S(=O)(=O)(c1cnccc1C)N(CCC(C)Nc1ccc(Cl)cc1)CC.C(C)=O.N C1(C(COC(C(Cc2cn(C(C)(C)C)nn2)C2CC2)=O)=O)CC(=O)NC(=O)C1 c1(C(=O)NCC2CCN(C(C3N(CC)CC3)=O)C2)cc(C)c(O)c(C)c1 N1(C(CC(=O)NCC)=O)CCN(C(=O)CC23COC(C2)C3)CC1CCO c1(CN2CCC(C(N3CCC(O)(C(F)(F)F)C3)=O)C2)cc2cc(Cl)ccc2[nH]1 c1(CC)cc(C(N2CCC(C)C(N(C(=O)C(C)OC)C)C2)=O)cc2c[nH]nc12 C1(NC(c2cncc(SC)c2)=O)CN(C(c2ccc(Cl)c(F)c2)=O)CCC1C c1(CC(N2CC(C)(NC(C3CC3c3cccs3)=O)C2)=O)c[nH]c2ccc(F)cc12 c1(CC)ncsc1C(=O)NCC1CC(NC(C2(C#N)CC2)=O)C1 Cc1cccc([N+](=O)[O-])c1NCCC1CC(NC(=O)C2CC2)C1 c1(CC)ccc(F)cc1C(=O)N(C1CN(C(=O)CNC(C)=O)CCC1O)C C1(C(C(C)C)NC(c2cccc(-n3cccc3)n2)=O)CCN(C(=O)CCF)CC1 CC(C)C(O)C(C)(C)C(=O)N(CC(C)N(C)C(c1cnc2ccoc2c1)=O)C N1(C(C=Cc2cn(C)nc2)=O)CC2CCCC(CNC(=O)Cc3cnsc3)C2C1 c1(C(N2CCCC(CCCC)C2)=O)n[nH]c2c1CN(C(=O)C1=CCCC1)C2 C1(C2CCN(C(=O)CCc3ccc(OC)nc3)C2)(NC(CCC(=C)C)=O)CC1 c1(C(N2C(C(=O)NC(C)Cc3cn[nH]c3)CC3CC32)=O)cncc(C#N)c1 C1(n2cccn2)(CNC(CCC)=O)CCN(C(c2ccc(OC)c(N)c2)=O)CC1 C(=O)(C1=NN(CCO)C(=O)CC1)N1CCC(NC(c2cc(Cl)ns2)=O)C(O)C1 N1(C(CCC)=O)CCCC(C(=O)NCC2(COC)CC=CC2)C1 N1(C(C(c2ccc(C)cc2)=O)=O)CCN(C(c2ccccc2C)=O)C2CCC12 CC1(C)CN(C(=O)CCCF)CC(CNC(c2n[nH]c3c2COCC3)=O)O1 C1(C(N2CC(C)C(NC(=O)C(C)(C)CCC#N)C2)=O)CCc2cncn2C1 Cc1cncc(CCNC(C2CCN(CC(C)CO)CC2)=O)c1 C(c1cnc(O)nc1O)=CC(=O)N.c1(OCC)ncccc1CC(N1CCC1)=O c1(C(N2CCC(C)(CNC(C3CCCC(=O)O3)=O)CC2)=O)ccc2c[nH]nc2n1 C1(CNC(CNC(=O)NC)=O)C=CCN1C(=O)C(F)OC O(N=C1CCCCCC1)CC(N1CC(C)C(NC(=O)C#CC2(C)CC2)CC1)=O N1(C(C=CCC)=O)CCN(C(=O)C2=CCCSC2)CCC1C n1(CC(=O)NC(CN(C(CCC)=O)C)C)cc(Br)c(O)nc1=O C=C1CCC1(C(=O)OC)C(N1CC(NC(c2cc(C)ns2)=O)C1)=O C1(NC(C(C)(C)C)=O)CC2CC(NC(c3ncc(Br)cc3F)=O)C2C1 C1(NC(c2nnnn2CC(F)F)(CSCCC)C)CCCOC12CCOCC2 Cc1ccc(=O)n(CC(=O)NCCC(O)C)n1.C1(CC(=O)N)CCCC(C)(C)C1 S(=O)(=O)(c1cccs1)N(CC(C)C)CC(N1CCCCC1CC1CCC1)=O c1(C(=O)NCCNC(C(C)N(CC(F)(F)F)C)=O)cnc(C(C)(C)C)o1 C1(C(=O)NCCSCCOC)CCCCN(C(C2CCC(=O)O2)=O)C1 CC1CN(C(C2CCC(=O)N2C)=O)CC1CCNC(c1n[nH]cc1F)=O Cc1ccc2c(c1)CCN2C(c1coc(CNC(=O)CC2COC(=O)C2)c1)=O CC1CN(C(C2CC(=O)N(C3CC3)C2)=O)CCN1C(=O)Cc1cncs1 N1(CC(N2C3(CN(C(CSCCCC)=O)C3)CC2)=O)Cc2ccccc2C1=O C1(c2n(-c3c(C)cccc3)nnn2)(NC2CC2)CCN(CC2CCCC2O)CC1 Cn1cc(C(=O)NC2COCC2C(=O)NC2CC(CC3CC3)C2)cn1 C(=O)(CCC(=O)CC)N1CC(CC=C)(C(N2CCOC3CC23)=O)C1 c1ccc(C#N)cc1.N1(CCC)CC(C(=O)NCCN(C(=O)CS)C)CC1=O c1(CC)nc(C)n(C)c1C(=O)N.C1(CC=O)CC(F)(F)C1.CC=CC CN1CC(C)(C)CC1C(=O)NCCC1CCCN(C(c2n[nH]cc2Cl)=O)C1 CC1CCC=C1C(=O)N1CC(C(=O)NCC(C)(C)CC2CC2)C(C)(C)C1 Cn1c(C(=O)NCCC2CC2)cc2ccc(O)cc12.C(=O)C.C(=O)C1CC1 c1(CC)nc2n(n1)CC(Nc1ncnc(NC(C)C(C)C)c1C)CC2 N#Cc1ccc(C(=O)NCCCO)c(O)c1.C1(CO)C(=O)N1 C1(C2CCN(C(c3ccn(C4CC4)n3)=O)C2)CC1.CN(S(N)(=O)=O)CC(=O)N C1(O)(CNC(=O)CC2C=CCC2)CCN(C(=O)C=CC2CCOCC2)CC1 C(C(C(=O)N)C(C)(C)C)NC(Cc1cn(CC)nn1)=O.C1CC2(C1)CN(C)C2 CC(=O)CCCC(C)C(=O)N1CCC2CCCC12C(=O)N(C1CCCCC1O)C c1(C=O)ncn(-c2ccccc2)n1.C1(O)(CC)CN(C(c2c[nH]c(=N)o2)=O)C1.N C=C(C)CC(C)C(=O)NC1(C)CC(NC(C2(S(N)(=O)=O)CCC2)=O)C1 Cc1nc(C(=O)NC(C2CN(C(=O)Cc3nncn3C)CCO2)C)nn1C C(C)(C)(C(F)(F)F)NC(CCN(C(c1cc(C)sc1)=O)CCO)=O Cc1c(C(=O)OCC2CCC3(CC2)CC3)oc(=O)c2ccccc12 C(=O)(C(CO)C(F)(F)F)NC(C1CN(C(c2ccc([N+](=O)[O-])cc2)=O)C1)C c1(OC)cc(N)c(C(=O)NCC2CN(C(=O)C(C(C)O)N(C)C)C2)cc1Br CCC(C)CC(C)C(=O)N1CCCC(CCC(=O)N(C)Cc2nc[nH]n2)C1 C(=O)(C(C)(C)CNC(=O)CCNC(C1CN(C(C)=O)C1)=O)OC Cc1noc2ncnc(NC3CC(C)N(C(=O)C(F)C(C)(C)O)C3)c12 C1(C(=O)NCc2n(C(C)C)ccn2)CCCC2(CCCC2)O1 C(=O)(C(C)(C)CO)NCCN(C(c1cc(OC)n[nH]1)=O)CCOCCO c1(OC)ccsc1.C(C)(CCC)N(CC(C)NC(C)C)C.CC.CC.N CC(C)CC(C(=O)NCCN1CC(CF)C1)N(C)C(c1c[nH][nH]c1=N)=O N1(C(C(C)=O)=O)CCCCC(CNC(=O)CCC2CCCOC2)C1 CC1(CNC(=O)C=CSc2ccccc2)CN(C(c2cnns2)=O)CCO1 N1(C(c2ccc(C)n2C)=O)CC2(CCCN(C(c3cc(Cl)c(F)cc3Cl)=O)C2)C1 c1(C=O)ccc2cnsc2c1.C(C(=O)NC1CCC1)(C(C)C)N(CC)CC.C CC1CN(C(C2(C)SCCCS2)=O)CCCN1C(=O)CCCc1cnccn1 C1(C(=O)NCC(CNC(c2cncc(NC)c2)=O)(C)O)CCC2(CCC2)C1 c1(CCCC)oc2ccccc2c1C=CC(=O)NCC1CCC(C(N)=O)CC1 c1(C(=O)NC2CC(NC(=O)C(O)(C3CC3)C3CC3)C2)ccnc2[nH]nnc12 N1(C(COCCC#C)=O)CCCC(C2CN(C(c3cccc(N)c3C)=O)C2)C1 CC#CCC(C(=O)Nc1cc(O)ccc1OC)NC(=O)C(C)OCC1CC1 C1(CNC(c2cc(Cl)c[nH]2)=O)CCCN(C(=O)C(O)Cn2cncn2)C1 C(=O)(CC(C)(C)C(F)F)N1C(C)(COC)CCC1.c1(C(=O)N)ccc(F)cn1 C1(NC(c2cnc(CC)[nH]2)=O)CCC(NC(c2c[nH]nc2OC)=O)CC1 C(=O)CCC=O.C(=O)(CC(=O)NC1CCCC1C)N(CC)CC.C1CCC1 C1(CNC(c2[nH]nc3cnccc23)=O)CC2CCC(C1)N2C(=O)C(F)F Cc1nc(CO)oc1-c1nc(-c2cnccn2)nn1CCOCC(F)(F)F c1(C(=O)NC(C2(O)CN(C(c3ns[nH]c3=O)=O)C2)C)cc(=O)n2ccsc2n1 c1(NC(CC)=O)ccccc1C(=O)NCC1(NC(C2CCC2)=O)CCC1 c1(CC(N2CCC(N(C(=O)C(C)(F)F)C)C2)=O)cn2cc(Cl)cc(Cl)c2n1 N1(C(c2cccc(C)c2)=O)CCCC(CCNC(c2ccc(C)[nH]2)=O)CC1 Nc1c(C(=O)NCC2CCCCN(C(=O)CC(F)(F)Cl)C2)ccc(F)c1F CCC(C(=O)NC1CC(NC(=O)Cc2nnc(O)s2)C1)c1cccnc1 CON(CCC(=O)NCC1(C)CCCC1O)C(=O)c1ncn(C)n1 c1(CC)oc(C)cc1C(=O)NCCC(O)CNC(c1cc(C)ns1)=O N1(C(CN(C)CC)=O)CC2CCC1C1CN(C(c3cnc4[nH]cnc4c3)=O)CC21 CC1CCN(C(=O)CNC(=O)C(C2CCOCC2)F)C1CC1CC1 C1(C(=O)NCCC(C)(C)C)CC2CC2N1C(=O)CSCc1ccccc1 c1(CC)cc(C(=O)NC2CN(C(=O)CN3CC(CC)C3)CC2C)c(C)nn1 C1(NC(CC#N)=O)CCC12CCN(C(=O)CCc1cnccn1)CC2 C1(CC)CN(C(=O)C(N2CCCC2c2cn(Cc3nccs3)nn2)=O)CCCO1 Cc1cc(C)n(CCC(N2CC=CC2C(=O)NCC(=O)NC2CC2)=O)n1 c1(C(=O)NC2CC(CCNC(=O)C=C(Cl)Cl)C2)ccnnc1NC1CC1 Cc1nc2ccccc2n(CCNC(c2sc3nccc(Cl)c3c2C)=O)c1=O c1(CC(=O)NC(CC)(C)CNC(c2cnc(OC)cn2)=O)ccc(Cl)cc1.O Cc1cc(C)c([N+](=O)[O-])cc1C(=O)NC1CN(Cc2cc(O)ccc2Br)CC1O c1(C(=O)NC(CN(C(=O)C=Cc2ccccc2)CC)C)cccc(F)c1O C=CCC(C)(C)CC(=O)NCC(C1CCN(C(=O)C(C)C(CC)CC)CC1)O c1(OC)ccnc(CC(=O)NC(C)CNC(C2(C)CCNC2=O)=O)n1 CC1(C(=O)NCC2(O)CCN(C(=O)CCCc3ccccc3)C2)CC=CCO1 c1(C(N2C(CNC(C(CC=C)C)=O)CC3(CCC3)C2)=O)cc2c(cn1)OCCC2 N1(C(C2N(CC)CCOC2)=O)CC2CC3CC2C1C3NC(=O)COCCCF c1(OC)cccc(NC(C)C(=O)NC2CC(CC)C2)c1.C(=O)C1=NOCC1.N N1(C(C(CSC)(C)C)=O)C2CCC1CC(NC(c1cc(C)[n+]([O-])cn1)=O)C2 C1(C(=O)NC2CC(OCC(N3CC=C(C)CC3)=O)C2)CCC=CCCC1 N1(C(C2C(C)C2C)=O)CCC2(CCOCC2)C(NC(c2ccnn2CCF)=O)C1 CC1CCCCC1CC(=O)N(CC1CCC1)CC1CCOCC1 C1(C(=O)NCCC2N(C(CC=CC)=O)CCOC2)CC(c2cccc(F)c2)=NO1 c1(OC)cc(Cl)ccc1C(=O)NC1CC2C1CCN2C(=O)CCN1CCCC1=O C1(CNC(CSc2cn(C)nc2)=O)CCCCN1C(=O)C(O)Cc1cnc[nH]1 c1(OC)cc(C(=O)NC2CCCN(C(=O)C3=COCC3)C2)cc2nc(O)[nH]c12 O=C(NNc1ccncn1)c1cnc2[nH]nc(O)c2c1 C(=O)(C1CCc2c[nH]nc21)NCC(CO)NC(c1[nH]ccc1C1CC1)=O c1(OCCOC)ccccc1.C1CCN(C(=O)N)C1.n1(CC)ccc(C(F)F)n1 c1(C(C)NCc2ccco2)ccccc1C(F)(F)F.c1nnnn1C1(C)CC1 N1(C(C(C2(O)CN(C(C(C)O)=O)C2)F)=O)CC(C)CCCC1C C1(C=O)CC(=O)N(OC)C1.O(N(C)C(=O)C=CCC1CCC1)CC=O.C C1(CNC(C(C2CCC2)OC)=O)CC2CC2N1C(=O)C(c1ccccc1)=O C1(NC(=O)CCCc2ccccc2)CC(F)CN(C(c2ocnc2C(F)F)=O)C1 c1(N2CCC(CCNC(C3CC(C)OC3C)=O)CC2)ncnc2[nH]cc(CN)c12 c1cccc([N+](=O)[O-])c1.c1(OCC)cc(Cl)cc(C)n1.C1(C=O)CC1C=O C1(C(F)(F)F)(OC)CC(C(=O)NCCC2CC2)C1.c1(C=O)ccns1.N CN1CCC(CC(=O)NCCC2CCCN(C(=O)CCc3nc(O)n[nH]3)C2)C1=O C12(C(=O)NCC(C)CO)CC3CC1(CO)CC3C2.C(=O)(CCCc1ccsc1)N CC1(C(N2CCCC(CN3CCCCC3)C2)=O)CCCN(c2ccc(Cl)nn2)C1 N1(C(=O)NCC(C)(O)c2ccco2)CCOC(C(F)(F)F)C1 c1(NC(CCC=C)(CC)c2nnnn2C)ccc2c(c1)oc(=O)n2C1CC1 C1(NC(=O)CCOCC2CC2)CCN(C(C2CC=CCC2)=O)CC12CCC2 C1(NC(Cc2cc(C)[nH]n2)=O)CCC2(CC1)CN(C(=O)C(c1cnn(C)c1)=O)C2 c1(C(=O)OC)ccc(OC)c(NC(=O)NC2CCCC2(C)CO)c1F CCCC(F)(F)F.c1(C(C)OCC)nc(C)c(C(=O)N)s1.c1(C=O)cnn[nH]1 N1(C(C(n2c(C)ccn2)C)=O)CC2CC1(C(=O)NCC(O)CCC1CC1)C2 Cc1ccc2nc(C(=O)NC3CC(CNC(C4CCC4)=O)C3(C)C)ccc2c1 N1(C(C(C=C)(C)C)=O)CCC2CCC(C1)N2C(c1cn(C(C)C)nc1Br)=O N1(C(c2c[nH]c(=NCC)s2)=O)CCCC1C1CCCN1C(c1cn(C)cc1C)=O C1(NC(c2cc(C(=O)OC)no2)=O)CCOCC1.C1(CC=O)CCN(C)C1.C n1(CC)nc(C)c([N+](=O)[O-])c1N1CC(C)C1.C(=O)(C(C)(C)n1cnnn1)N c1(C(=O)NC2C=CC(CNC(C(CCCC)(C)F)=O)C2)ccc2n[nH]cc2c1Cl CC1CC(NC(=O)Cc2cscn2)CCN1C(=O)CCCCC1CC1 N1(C(C(F)=CCC)=O)CCN(C(c2sccc2C#N)=O)CC1CC(F)F Cc1cc(C=CC(=O)NCC2CC2)c[nH]c1=N.C1(C(N(C)C)=O)CCC1C C1(CNC(CC2CCC(C)(C)C2)=O)CCCC2CN(C(=O)CCS(C)(=O)=O)CC12 c1(C(CCO)NC(c2n(CCOC)nnn2)c2ncnn2C)ccccc1Br N1(C(c2ccc(C(=O)OC)o2)=O)CCC2CC1CN(C(c1cnsc1)=O)C2 C1(CCNC(C2CC(OC)C2)=O)CCCN1C(C1CCCCN1C(C)=O)=O N1(C(c2cccc(C(=O)NC)c2)=O)CC2C3CCC(C2C1)N(C(=O)C=CSC)C3 CCCCC(O)C(C)C(=O)NC1CC(C)(NC(c2cnn3ccccc23)=O)C1 C12(NC(C(C)=CC)=O)CCCC1N(C(c1ncsc1C1CC1)=O)CC2 C1(C=O)CCC2(CCOCC2)O1.c1(C(=O)NCCC)ccc(CSC(F)F)o1.N C1(NC(c2cn(CC)nn2)=O)CCCC(NC(c2ccccc2CO)=O)CC1 c1(C(N(CC(C)(C)NC(CCSCC(C)C)=O)C)=O)cn(C)c(O)n1 c1(C(N2CCC(CNC(C=C3C(C)(C)CCCC3)=O)C2)=O)ccn2nccc2c1 Cc1ccc(C(=O)C(N2CC(NC(=O)C(N3CCCC(C)C3)=O)C(C)C2)=O)cc1 C1(C=O)CCC(C)(C)OC1.c1(C=O)cnn(CC)c1.CCCOCC1CC1 N1(C(=O)NCC(C2(O)CCOC2)(C)C)CCCC(O)(C(F)(F)F)CC1 c1(C(c2nnnn2C2CC2)NC(C(C)C)c2cncs2)ccnc(Cl)c1 C(=O)(C1=CS(=O)(=O)CCC1)N.CC1(NC(=O)CN2CC(F)(F)C2)CCC1 C(=O)(C1=CCCOCC1)NC1CN(C(C(C)Cc2ccnn2C)=O)CC1C C1(C(=O)NCC23CCN(CC2)C3)CC2CC2N1C(=O)C(O)CC1CCCC1 Cc1cccc(CC(=O)NCC2CCCCN2C(C2CCS2(=O)=O)=O)c1Cl CC(C)C(O)C(=O)NCC(O)CN(C)C(c1sccc1CN(C)C)=O S(=O)(=O)(c1ccc(NC(COC)CC)c(C#N)c1)NC(CC)(CC)c1ccccc1 N1(C(C(=O)NCC)C2CC=CC2)CCCCC1COC(C)(C)C c1(CCCNC(c2nn[nH]n2)C)c[nH]c2ccccc12 c1(CCC(=O)NCCNC(=O)CCNC(N2CCCCC2)=O)nncnc1O N1(C(Cc2cccc(C)c2)=O)CC2CN(C(c3cnc(C)[nH]3)=O)CC12 C1(C(=O)NCCC(C)(C)O)CCCN(Cc2ccc(Br)cc2I)CC1 c1(C(C)(C)NC(=O)CC2C=CCCC2)cc(Cl)ccc1F c1(C(=O)NCCN(C(C(C)OCC=C)=O)CC(C)O)cc(Cl)ccn1 C1(NC(c2c(C)csc2)=O)CCN(CC2CC3CCC2O3)C(C)C1 C1(C(CNC(c2c(CC)cc[nH]2)=O)O)CCN(C(c2coc(C)c2)=O)CC1 C1(C(=O)NCCOC(CC)CC)CCN(C(=O)CN2C(=O)CCC2=O)C12CC2 C1(C(N2CCC(CCC#C)CC2)=O)CC(CC)CCN1C(c1cc(OC)ns1)=O C1(CNC(C2N(S(C)(=O)=O)CCC2)=O)CCC(NC(c2cnoc2)=O)CC1 N1(C(C(C)OC(C)(C)C)=O)CCC(c2ccccc2)(NC(C2CCC2)=O)CC1 CCCC(C(=O)N1CCCC1Cc1cccc(C(F)(F)F)n1)OCC C1(O)(C(C)NC(C2CC(N(CCC)C)C2)=O)CCN(C(=O)CC2CC2)C1 C12(C(=O)NCC(C)(C3CCC3)NC(CCC(=O)NC)=O)COC(CCO1)C2 N1(C(C(CNC(C2(C)C(C)OCC2)=O)N(C)C)=O)CCC2C(C(N)=O)C2C1 CC12CCCC1NC(=O)CN(C(=O)NC1CCOCC1F)C2 CC(C)(C)C(C(=O)NCc1cc(=O)c(O)co1)n1cc(-c2cnsc2)nn1 S(=O)(=O)(c1ccc(Br)cc1NCC1CCc2nccn21)NCCCOC(C)(C)C C1(CC=O)CCC(C)(C)CC1.c1(C(C)C)nnsc1C(=O)NC1CC1C.N C(=O)(CCCC(=O)NC(C(=O)NCc1ccccc1)C1CCCO1)OCC.C c1(C(N2CC3(CN(c4c(CC)cnc(Cl)n4)C3)C2)=O)ccc2c(n1)CCCC2 c1(CNC2C=CC(C(=O)Nc3ncccc3I)C2)ccc(Br)cc1I CC(C)CC(O)CC(=O)NCC1(NC(=O)C(C)C2CC2)CC(F)(F)C1 c1(C(=O)NC(CC)(CNC(=O)C(C)NC=O)CC)oc2ccccc2c1CO C1(N(C(=O)Cn2cc(C#N)cn2)C)CN(C(c2cc(C)n(C)n2)=O)CC12CC2 c1(C(N2CCN(C(CNC(C3(CC)CCCC3)=O)=O)CC2)=O)ccnc(C)c1Cl Cc1oc(C#N)cc1C(=O)NC1CCOC1C(=O)NC12CCN(CC1)C2 C1(C(=O)NCC2N(C(CCC#C)=O)CCCC2)CCCC(C)CC1 c1(C(=O)NCCOCCC(=O)N(C2CCOCC2)CC#C)ccnc(C)c1 C(=O)(CS(=O)C(F)(F)F)NCC1(CO)CCN(C(CC(C)SC)=O)C1 c1(NC(C2C(NC(c3ccc(Cl)c(F)c3F)=O)C2)=O)cccc2c(Br)ccnc12 N1(C(C(C)c2cccs2)=O)CCCC1C(C)(C)C(=O)NC1CC(C)C1 Cc1cc(N(C(=O)CC(C(F)F)NC(C2CCOC2(C)C)=O)C)cc(F)c1 C1(CN)CC(C(=O)N2CC3CC4CC3C2C4)=CC1O C1(N(C(CC2(OC)CCOCC2)=O)C)CN(C(C2C=CCS2)=O)CC12CC2 c1(OCCC)ccc(C(=O)NCC(n2cc(C3(C)CSC3)nn2)C)cc1 c1(C(N2CC(C(N3CC(CC)C(F)C3)=O)C(C)C2)=O)c(O)cccc1F Cc1[nH]c2ccccc2c1C(=O)NC(CNC(=O)C(C)c1ccco1)CO c1(CC)cccnc1C(=O)NCCc1ccc(CNC(C2CC2C)=O)cc1 N1(C(C(C)N2CCC2)=O)CCC(CN(C)C(c2ccc(C3CC3)nc2)=O)CC1 c1(CN2CCC(C(C)C(=O)NC3(C)CC3)CC2)ccc(Br)cc1I Cc1scc(C(=O)NC2(CNC(=O)CCc3nccn3C)CCOC2)c1N C1(C(=O)NC(C(C)NC(c2ccn(C3CCCC3)n2)=O)C)CCC(C)CC1 C1(C(C)C)N(C(=O)CC2COCCO2)CC12CCN(C(=O)C)CC2.CCN(C)C.S Cc1nn2c(c1C(N1CCCC(NC(C3CC3(C)C(C)C)=O)C1C)=O)NCCC2 C1CN(C(c2ccc(N)c(Cl)n2)=O)C2CCN1C2.n1(CC)cc(C(=O)NC)cn1 N1(C(C=CCOCCOC)=O)CC(C)C2CC12.c1(C=O)ccn(C)n1.N c1(C(=O)NC(CNC(CC2CC(=C)C2)=O)C(C)C)ccc(NC(C)C)cn1 C1(NC(CCC(N)=O)=O)CN(C(C23CC(C2)S(=O)(=O)C3)=O)CC2(CC2)C1 c1(C(N(CCC)CCNC(C2CC2Cl)=O)=O)cc(O)cc(F)c1 CCCC(CNC(C1CCSC1)=O)NC(=O)C(C)C c1(C(N(C(CNC(c2ccc(CCCCC)o2)=O)C2CC2)C)=O)cnn(C)c1N C1(NC(C(CC)N(C)C)=O)C2CC3C(C2)C13C(=O)NC C1(C(=O)NCC#CC(=O)N(CC)CC2CC2)CCN(OC)CC1 c1(C(N2CC3C(CNC(c4c(CC)csc4)=O)(C3)C2)=O)ccc(F)c(C)c1 N1(C(C=CCCC=C(C)C)=O)CC(CNC(=O)C(C2CCCCC2)O)C(C)C1 C1(CC(=O)N(C)Cc2ccc(O)c(I)c2)CCc2ccccc2C1=O c1ccc(S(=O)(=O)N2CCN(C(c3cc(C)c(S(N)(=O)=O)s3)=O)CC2)cc1.CO CC1C(NC(C2CCN(C)CC2)=O)CC2CCC1N2C(=O)C#CC1CC1 c1(C(N(C2CCC(NC(CN(C)C(N)=O)=O)CC2)C)=O)csc2c(O)ccnc12 c1(C(=O)NC(C(C)NC(C=CC=CC)=O)C)cc2ccc(OC)cc2nn1 c1(OC)ccc(OC)cc1-c1cn(C2CCOCC2C(C)(C)C)nn1 C(C(=O)NCCC1CCN(C(=O)Cn2ncnn2)CC1)(C(C)C)n1cc(C)nc1 CC(CC(C)(C)C)N1CCC(C(N2CCCCC2CO)=O)CC1 c1(NCC2OCCN(C(c3cc(Br)co3)=O)C2)ncc(Cl)cc1[N+](=O)[O-] C1(NC(CN(C(=O)C(c2cnn(C)c2)=O)CC)=O)CCCC1(C)COC c1(C(N2CC(Cn3cc(COCC)nn3)OCC2)=O)oc2ccccc2c1C c1(CC(=O)NC2CC(NC(=O)CN3CC=CC3)C2)cc(O)ccc1Br C1(CC#C)(C(=O)NCC(C)CC2CCC2)CCN(C(c2csc(CO)n2)=O)C1 c1(NCCNS(C)(=O)=O)ccc(S(=O)(=O)N2CCC(n3cncn3)C2)cc1Br CC12CCC(C(=O)NCCC3CCC3)(CC1)CO2.N1(CC=O)CC2CC2C1.N C1(CCC(=O)OC)CCC(C)N(C(=O)CC(N)C(F)F)C1 Nc1c(C(N2CCC(CNC(=O)C(O)P(C)(C)=O)C2)=O)nc(O)nc1O c1(CN2CCC(NC(c3c(O)cccc3Br)=O)C(F)C2)c(Br)ccc2c1OCO2 C1(OC)(C)CCN(C(c2ccc(C(F)F)cn2)=O)C1.c1(CC=O)c[nH]nc1C.N O=C(CC=C(Cl)Cl)NC1CCOC(C(=O)NCc2cc(C3CC3)on2)C1 C1(NC(C2C(=C)C2)=O)CC(F)(CNC(c2c[nH]nc2C2CCCO2)=O)C1 C1(CNC(C)=O)CCCCN1C(C1COC(C)(C)O1)C(=O)NC1CCC1 c1(CCCNC(C(=O)OCC)C)ccc(OC)nc1 CCC(C)CCCCC(=O)NCC(=O)NCC(=O)N(C)CC1CCCC1(C)C CC(=O)C(C)(C)CC(=O)NCC1CN(C(=O)Cc2nocc2C)CC1C O=C(C1=CCCN(C(C2(F)C(C)(C)C2(C)C)=O)C1)NCCCn1nccn1 CC1=C(C(=O)NCC(C)N(C(=O)C(O)CC2CC2)C)CCO1 C(=O)(C(F)(CNC(c1cc(C)sn1)=O)C(C)C)NCCCOCC=C c1(CC)cccc(C)c1NC(=O)CCC(F)F.C1(C(=O)N)COCC1C(N)=O N1(C(C(C=C)OC)=O)CC(C2CCCN(C(=O)C(O)C(C)(C)C)C2)C1 c1(C(N2CCCC(NC(CCC(C)OC)=O)C2C)=O)ccc2oc(=O)oc2c1 c1(C2(C(=O)OC)CC(OC(c3c[nH]nc3C3(CN)CC3)=O)C2)ccccc1F C1(NC(COCCCCCC)=O)CCCN(C(c2cccc(F)c2F)=O)C1C C1(C(=O)NCC(CNC(C2(CC=C)CCC2)=O)F)CCN(C(=O)OC)C1 Cc1ccc(Br)c(C(N2CCN(CC(=O)Nc3ccnc(Cl)c3C)CC2)=O)c1 C=CCC(C)C(=O)NC1(C(=O)NCc2nnn(C)c2C)CCCC1 N1(C(CC(=O)NCC#C)=O)CCN(C(=O)CCN2CCOCC2=O)CC(C)(F)C1 c1(NC(CNC(C2C(OCC)C2)=O)=O)ccc(F)cc1 N1(c2ccnc(C(CC)C)n2)CC2(CCN(C(c3cc(C(F)(F)F)no3)=O)C2)C1 c1(C(N2C(CN(C(=O)CCC(F)F)C)COCC2)=O)cc(F)cc(N)c1N C1(C(N2CCC(OC3CN(C(CC(C)C)=O)C3)CC2)=O)C2CCC(C2)S1(=O)=O c1(C(N(C)CC2(O)CCN(C(=O)CCC#N)C2)=O)ncnc(O)c1F N1(C(Cn2c(C)ccn2)=O)CC(CCNC(c2cc(Cl)cnc2O)=O)OC(C)C1 C(=O)(C1=CCCCCC1)NC(C1CCCN(C(C2CC3(CSC3)C2)=O)C1)C c1(OC)ccc(CN(C(=O)C(=O)NCC2C=CCOC2)C)cc1F C1(CC(=O)N(CCCCNC(=O)CN2CCCC2=O)C)CCCC1(F)F c1(C(=O)NCC2CCC(NC(=O)C=CC=C(Cl)Cl)C2)c[nH]cc(F)c1=O C(=O)(C(C)S(N)(=O)=O)NC(CN(C(c1c(C)sc(-c2ccccc2)n1)=O)C)C N#CC1(C(=O)NC2CC(CNC(c3ccc(Cl)cc3)=O)C2)CC2CCC1CC2 N1(C(Cn2ncc(C)c2)=O)CC2CCCC2(NC(c2cccc(Br)c2N)=O)C1 C1(CC(=O)NC2C(CNC(CC=CC)=O)CCC2)CCC2(CC1)CCC2O Cc1nc(=O)c2c(C)c(C(=O)NC3CC3)sc2[nH]1.C(=O)(C1=CCCOC1)NC.C Cn1cc(C(=O)NC2CC3CC(NC(=O)CCC(C)(C)C#N)C2C3)c(O)nc1=O CC1CN(C(c2ccn(C)c2)=O)CCN(C(c2ccc(=O)n(C)n2)=O)C1 c1(C(N2CCCC(NC(C3(CCCC)CC3)=O)CC2)=O)ccc2ccncc2n1 C=CCC(F)(F)C(=O)NC(C)C(C)NC(=O)Cc1cccc(Cl)c1 Cc1cc(C(=O)N(C(C(=O)NC(C(N)=O)C2CC2)C2CC2)C)c(C)cn1 CC1(C(=O)NCCCN(C(=O)CCCC2CC2)CCO)CCCC1(F)F C(=O)(CCC(=O)NC1CC(C)N(C(c2ccc(C)cc2)=O)C1)Nc1nnc(C)s1 C1(OCC(=O)NC(C2CCCCN2C(c2ccsc2)=O)C)CCCCCC1 c1(C(=O)NCC(CNC(c2c(C)cc(C)o2)=O)C)nc(C)n(C)c1C C(=O)(C1CCCc2n[nH]cc21)N1C(CNC(C2CCCCCCC2)=O)CCC1 C1(C(=O)NC(C(N)=O)C2CC2)(CC)CCN(C(c2cnn(C)c2Cl)=O)CC1 c1(N2CC(O)(CCNC(C(C)OC)=O)C2)ncncc1I Cc1cc(=O)c(C(N2CCC(CC(N)=O)(NC(C3CC(C)C3)=O)CC2)=O)cn1C c1(CNC2CC(C(N3C(C(N)=O)CCCC3)=O)C2)c(Cl)cccc1[N+](=O)[O-] c1(CN(C(CC)C(=O)O)C)ccc(OC)cc1CO N1(C(CCOCC)=O)CC2CC(NC(C3(OC)CCCSC3)=O)C1C2 c1(C(=O)NCCCN(C(C(C)OC(C)(C)C)=O)C)c(F)ccc(Br)c1F N1(c2cccc(C(=O)OC)n2)CCCC12CCCS(=O)(=O)C2 C#Cc1c[nH]nc1C(=O)NCCC(O)CNC(=O)C(O)Cc1ccccc1Cl C(=O)(C(C)CC(N)=O)N1CC(NC(c2c(Br)cn(CC)n2)=O)(CO)C1 c1(C(N2CC(C)C(CNC(c3sncc3Br)=O)C2)=O)cncc2[nH]ccc12 C(=O)(C1=NOC2COCC12)NCC1CC(C)N(C(c2cnnc(O)c2)=O)CC1 CC(C)(CC(=O)NCC(O)CCO)NC(=O)C=CCF C1(CNC(CCCN(C(C)=O)C)=O)CCN(C(C2C(C)C2C)=O)C(C)C1 Cc1ccnc(O)c1C(N1CCC(C)(CNC(=O)C(C)Cc2cnco2)CC1)=O N1(C(C(CCC)NC(CCCOCC=C)=O)=O)CCC2(CNC(=O)O2)C1 Cc1cc(-c2nnc(CC3(C4CC4)CCCN3C(c3ccccc3)=O)o2)nn1C c1(CC)ccc(C(N2CC3CC(C)C3C2)=O)c(C)n1.C(=O)CCC=C(C)C.N C(=O)(C1CCCn2nccc21)NC1CCCN(C2C(=O)NCC2)CC1 N1(C(=O)Cc2cc[nH]c2)CCN(C(c2cc(Cl)ccc2F)=O)CC(CO)C1 C(Cc1ccccc1)(CCNC(c1cocn1)=O)NC(C=CC=CCC)=O C1(NC(CCC2N(C)CCCC2)=O)CC2CC(NC(c3ccncc3Cl)=O)CC12 C1(NC(c2cnn(-c3ccncc3)c2)=O)CN(C(=O)C(F)CC2CCC2)CC1O C=Cn1nccc1C(=O)NCCCN(C(=O)C(C)CSc1ccccc1)C C1(CCNC(C=CCOC)=O)CCN(C(=O)C(C2CCCC2)O)CC1(F)F CC1=C(C)CC(C(=O)NC2CCN(C(=O)CO)C2(C)C)CC1.c1ccc(Cl)cc1 N1(C(Cc2cc(C)on2)=O)CCC(NC(c2cn(CCO)nc2C)=O)C1(C)C c1(C(=O)NCCC2(CNC(C(CCCC)O)=O)CC2)ccc(Br)c(F)c1C C1(CNC(c2cnc(CC)o2)=O)CC12CCC2.C(=O)C(C)CC1CCC1.C c1(C(N(CCN(C(C2(C=C)CCC2)=O)C)C)=O)cnn2ccn(C)c12 C(=O)(C1=NN2CCCN=C2N1)NCC1CCN(C(C2(C)CCN(C)CC2)=O)C1 C1(C)(C(N(C)CC2CC(=C)C2)=O)CCN(C(c2cnc(Cl)s2)=O)C1 C(=O)(CC(C(F)F)n1ccnc1)NC(CCNC(c1cc(CC)oc1C)=O)C C1(C(N2C(C)(C)C(NC(C3CC34CCCC4)=O)CC2)=O)CCc2n[nH]cc2C1 c1(C(N2CCCCCC2)C(=O)NC2(C)CC2)cn2cc(Cl)ccc2n1 C1(CN(C(c2ccn(CC(F)F)n2)C(=O)NC2CCOC2)C(C)C)CC=CCC1 c1(COC(C2(Br)CCC2)=O)ccc(C(F)(F)F)c(Cl)c1 N1(C(c2ncc(CC)o2)C(=O)NC2COC2)CCCC2OCCC2C1 N1(C(CCC(CCC)CC)=O)CC2(C=C(C(=O)N(C)CC3(C)CCCO3)CO2)C1 C1(C(=O)NC2C=CCN(C(C3(F)CC=CC3)=O)C2)CN2CCN1CC2 C#Cc1cc(C(=O)NC2CC(NC(c3ccc(O)nc3)=O)C23CCC3)cc(F)c1 S(=O)(=O)(c1cnc(N2CCCC(C(F)F)C2)c(Cl)c1)N1C(C)CCCC1 c1(C(=O)OCC(=O)Nc2ccccc2Br)c[nH]c2c(F)cc(F)cc2c1=O CC1(C)CCN(C(C2CC2(Cl)Cl)=O)CC1C.C1(C(=O)N)CCCCN1CC(F)F c1(CC)ccc(C(=O)NC2CC(NC(c3cc(-c4ccncc4)no3)=O)C2)o1 NS(=O)(=O)c1ccc(CCC(=O)NC2C=CCN(C(=O)CNC=O)C2)cc1 Cc1nn(C)c(C)c1CC(N1CCC(C)C(C)C1)=O.C1(C)(CC=O)CCCC1.N N1(C(Cc2ccccn2)=O)CCCC(F)C1.C(C)(C(C)(C)C)=CC=O.CCO Cc1ncn(O)c1C(N1CCC(Cn2cc(CO)nn2)CC1)=O n1(CC)ncc(C(N2CCC(c3nncs3)C2)C(=O)NC(C)C)c1C CCC(C)C(O)C(=O)NCCC1CCCCN1C(=O)Cc1ccc(C(N)=O)cn1 N1(C(C(C2CCOC2)NC(C=C(C)c2ccco2)=O)=O)CCCC2C(O)CC12 N1(C(C(=O)NC2CCC(C(=O)OC)C2)CCc2ccco2)CCOC(C)(C)C1C CCCC(C(=O)NC(c1cccc(-n2cc(CN(C)CCOC)nn2)c1)C)OC N(C1CCCS(=O)(=O)c2ccccc21)C(=O)NC1(c2cn(C)nc2)CCCO1 c1(OC)cc(C)c(C(=O)NC2CCN(C(c3ncccc3Cl)=O)C(C)C2)c(C)c1 c1(C(=O)NCC2C(C)CCN(C(C(C(C)C)O)=O)C2)ccn2nccc2n1 c1(N2CCC(C)C2CNC(c2cccn(O)c2=O)=O)nc2cccc(F)c2o1 c1(C(N2CC3C(C(=O)NCC(CC#C)(C)C)(C3)C2)=O)cc[nH]c(=NC)c1 N1(C(CC(CCCCC)C)=O)CCCC(C2CN(C(=O)CC3(C4CC4)CC3)C2)C1 CC1CCN(C(c2cc(Cl)c(Cl)s2)=O)C1CNC(C1CNC(=O)N1)=O CN1CCOc2ccc(C(=O)NCCNC(=O)CS(F)(F)(F)(F)F)cc21 c1(C(=O)NC(C2OCCN(C(C=CCC)=O)C2)C)cncc(C(=O)OC)c1C c1(CN2CCC(C(N3CC(O)C3)=O)C(c3ccccc3)C2)cc(Cl)c(Br)c(Cl)c1 C(C)(C)(C#CC(C)(C)O)NC(CONC(c1ccn(CC)c1C)=O)=O c1(C(=O)NC2CCCCN(C(C3CC(C)(F)C3)=O)C2)c(O)cnc2ccccc12 C1(NC(c2ccc3nc[nH]c3c2)=O)CN(C(c2cnc[nH]2)=O)CC(F)(F)C1 c1(C(N2CC(CNC(c3cnc(CCCC)s3)=O)(OC)C2)=O)ccc(C#N)s1 c1(CC)cc(F)ccc1C(=O)NC1CCCC(NC(=O)CCSC)CC1 c1(-c2ccc(NCc3ccc(C)c(F)c3O)c(F)c2)ccc(S(=O)(=O)F)cc1 N1(C(Cn2nnc(C)n2)=O)CCC(NC(=O)C(C)S(C)(=O)=O)CC1C Cc1ccc(O)cc1C(N1CCOCC1CC(=O)Nc1ccc(Br)nc1)=O C1(ONC(C2CCNC2C(=O)O)=O)CCc2ccccc2C1 C1(NC(C(C)OC)=O)CCN(C(=O)CCc2c(F)cccc2F)C12CCC2 n1(C(CC)C)nnnc1C(CCC1OCCO1)N1CCCC1 CC1CC(NC(=O)Cc2cnccc2Cl)CCN1C(c1ccc(C(F)F)cc1)=O c1(CCC)cccc(C(=O)NC2CC(O)(CNC(=O)C(C)OCC)C2)c1 CCCCCC(O)C(=O)N1CCN(C(c2nn(C)c(C)c2Cl)=O)CC1 c1(C(N2CC(F)CC(NS(CCOCC)(=O)=O)C2)=O)cc(O)c(O)cc1O CCC(CC(=O)NCCC(C)F)NC(=O)C(C)(CO)OC CC1CN(C(=O)C=C2CCCCC2)CCCN1C(=O)C=Cc1cnc[nH]1 C1(OC)CCC(C(N2CC(C(N)=O)(C)C2)=O)CC1.c1(C=O)cncc(F)n1.N CCC(CCC(=O)N1CC(O)CO1)NC(=O)C(O)Cn1cncn1 C(=O)(CCCC(=O)NCCC(C)CC)OCC.C1(S(N)(=O)=O)(C=O)CC1.N c1(C=O)cc(Cl)c(Cl)n1C.Cc1cc(C(=O)NCC2CCC(C)CC2)cnn1.N C1(CCNC(C=CC(C)C)=O)CN(C(C2CC2C2CCC2)=O)CCS1(=O)=O c1(CN(C=O)C(C2CCCO2)C2CCC2)cccc(F)c1C(F)(F)F C1(CCNC(CCSC)=O)CC(F)(F)CN1C(c1ncn(-c2ccccc2)n1)=O O=C(O)C(CCNC(c1cc(O)nc(-c2ccc([N+](=O)[O-])cc2)n1)=O)C(=O)O c1(NC(C2CN(Cc3cccc4c3OCCO4)C2)=O)nnc2ccc(Cl)nn12 CC(C)(C(=O)NCCN1CCN(c2nc(Cl)ncc2C(N)=O)CC1)C(N)=O CCC1=C(C(=O)NC(C2(CNC(=O)CCC(C)(C)F)CC2)C)SCCO1 C1(C=O)(NC(C=CCOCCOC)=O)CC(F)(F)C1.CC(C)(C)CO c1(C(N2CC=C(CNC(C3(CC#C)CCCO3)=O)CC2)=O)ccc2nonc2c1 N1(C(C2(C)CC(=O)C2)=O)CC2(COC(C)C2)C1.C1(C=O)CCCCS1(=O)=O.N Cc1cnn2ccc(C(=O)N(C3CCCCC3NC(C3(CO)COC3)=O)C)nc12 C1(C(=O)NCc2nc(COC)on2)CCC2CCC1N2C(c1cscn1)=O c1(C(C)C)ncc(NC(=O)CCOCCCNC(C2CCN(C)C2)=O)cn1 c1(C=O)cc2c(s1)CCCC2.C1(CNC(C=C(COC)C)=O)CC(F)C1.C S(=O)(=O)(c1csc2ccccc12)N1CCCC(C(C)NC(c2ccnnc2)=O)C1 c1(C(=O)NCCn2cc(-c3cccnc3)nn2)ccccc1C(F)F C12(NC(C(CC)CC3CCCC3)=O)CCC(C1)OC2.C(=O)C(F)=C1CCC1.C C1(NC(c2cccc(OC)n2)=O)CN(C(=O)CC2CCCOC2)CC12CCC2 Cn1nc(Br)c2c(NCC3(C)CCN(C(=O)C(F)CC4CC4)C3)ncnc12 C(=O)(C1=CCCN(C(c2[nH]cc3c2CCC3)=O)C1)NCc1cncc(C)c1 C(=O)(C1=C(C)CCOC1)NCCCCCCN(C(C(C1CCC1)OCC)=O)C CC1(C)C2CCC(C2)C1C(N1CCC(C)C12CC2)=O.c1(CC=O)csc(Cl)c1 C1(C(=O)NC2C(NC(=O)Cc3cc(Cl)ccc3Cl)CCC2)CCn2nccc2C1 c1(C(=O)N)ccc([N+](=O)[O-])c(C)n1.C=C(C)CCCC(=O)NCC1CC1C N1(C(CN(CCOC)C(c2nc(CC)oc2C)=O)=O)CC2(CCNC(=O)O2)C1 Nc1cc(F)c(F)cc1C(=O)NC1CCCN(C(c2ccc3c(c2)CCC3)=O)C1 N1(C(COC2CCN(C(C(CCC)(C)C)=O)C2)=O)Cc2ccc(O)cc2C1 C=CC(O)C(=O)N(CC(CC)NC(=O)Cc1cn[nH]c1)CC C(=O)(C(CCN(C)C)NC(C1CC=CCO1)=O)NC1C(C)C1C N1(C(C=C(CC)C)=O)CC2(CC(NC(=O)C(C)C(C)(F)F)c3nccn32)C1 c1(N2CCC(C)CC2)c(Cl)cc(Cl)cc1Br.c12nc(ccc1C#N)N2 C(CCCCN=C(NC1CCCCC1)NC1CCOC(C(C)C)C1)SC CCC(CCCC(=O)NCC1CN2CCC1C2)NC(C1(C)COC(=O)N1)=O CC1(NC(c2ncn(C(C)(C)C)n2)=O)CCN(C(C2C3CC3C3CC23)=O)CC1 C1(CCNC(c2c(C)ncs2)=O)CN(C(=O)CCC2CCC(C)O2)CCCO1 N1(C(Cc2ccc(C)nc2)=O)CCCC(NC(=O)Cc2nncs2)C1C C1(CNC(C(CSCC)NC(C)=O)=O)(CO)CCN(C)C1 C1(C(N2CC(NC(C(C)OCC#C)=O)C2)=O)CSCC(=O)N1 C1(OC)CN(C(=O)C(C)(C2(C)CC2)OC)CC1C(=O)N.C(C)CC1CC1 c1(CC(=O)N(CC(C)NC(C(C2CCOCC2)OC)=O)C)cn(C)nc1C Cc1cc(CCNC(=O)C(F)CC2CN(C(c3cncnc3)=O)C2)on1 C#Cc1c[nH]nc1C(N1CCC(C(C)(C)NC(c2cccnn2)=O)CC1)=O C1(CNC(c2cnc(C)nc2O)=O)C(C2CC2)CCN1C(=O)Cc1nccn1C N1(C(CC(C)CSC)=O)CCC2C1CCCN2C(=O)CCN(CCC(C)(C)C)C c1(C(C)C)ccc(C#N)c(N2CC3(CCCC3NC(C3C4COCC34)=O)C2)n1 Cc1ccc(C(N2CCOCC(CNC(c3ccc[n+]([O-])c3)=O)C2)=O)c(=O)n1C C1(C(=O)NC(COC)CNC(c2sccc2C#N)=O)CCCCCN1C C1(C(N2CCCC2CO)=O)CCN(CC2CCOCC2)C1 Cc1nc(C)c(F)c(=NCCC(C)(C)NC(c2cc(=O)c3ccccc3[nH]2)=O)[nH]1 C1(CC=C)(C(N2CCC(OC)C2)=O)CCCN1C(c1c[nH]c(C)c1)=O c1(C(NC2CCCN(C(=O)CCC3(C)CC3)C2)=O)cnn(C(C)CC)c1C.CC c1(C(N2CC(NC(=O)Cc3ccsc3Cl)C2)=O)cc2cnccc2[nH]1 c1(C(=O)Nc2c(C(=O)Nc3cncc(C#N)n3)nccc2)cccc2scnc12 N1(C(CC)=O)CC(CNC(C2(CC3CC3)CC2)=O)C(CCC)C1 C1(NC(c2ccncn2)=O)CN(C(c2ccc(Br)s2)=O)CCC1CO CC1(C)CCCC2(CCN2C(C(=O)NCC2CCOC2)c2cc[nH]n2)C1 Cc1ccc(Cl)c(NC(=O)C(n2cc(CN3CCS(=O)CC3)nn2)C)c1 c1(C(N2CC3C(NC(CCOC)=O)(C3)C2)=O)nc(Br)n2c1CCCCC2 c1(NCC(C(CC)(F)F)(C)C)ccc(S(=O)(=O)NC2CC=CCC2)cn1 N1(C(C2C(OCC)C2)=O)CCCC2(CCN(c3ccnc(S(C)(=O)=O)n3)C2)C1 CS(=O)c1ccc(Br)cc1NC(=O)NCCC(c1cnc2ncccn12)=O N1(C(c2c(C)cns2)=O)CCCC2(C1)CN(C(=O)C=CC(F)(F)F)C2 N1(c2ncc(C(=O)OCC)cn2)CCC=C(C(=O)NC2CCCCC2)C1 c1(SC)cc(NC(C2(CNC(=O)C(N3CCCCC3)C)CC2)=O)co1 N1(C(c2ccc(CC)[nH]2)=O)CCC2(CC1)CC2NC(C1CC2C=CC1CC2)=O Cc1cc(C(=O)NC2CC(F)(CNC(=O)COc3ccccc3)C2)oc1Br c1(CC(=O)N(CC(CNC(CC(C=C)CC)=O)(C)C)C)cc(Cl)c2c(c1)OCO2 c1(-c2occ(CC=O)n2)ccc(F)cc1.CC(CN(C)C)C(=O)N.C1CC1.C c1(NC(c2nccn2C)CC)ccc(S(=O)(=O)NC)cc1Cl.c1ccc(C)c(Cl)c1 N1(C(CCc2cc(C)no2)=O)CCCCC1C=O.C(=O)(CC=O)NC.C(C)(C)C C(CC(F)F)(C(=O)N1CC(C#N)C1)N(C(c1cc(CC)ncn1)=O)C Cc1cc(O)nc(C)c1C(N1CCCC(N(C(=O)C=C(Cl)Cl)C)CC1)=O C1(C(C)C)CN(C(=O)CCSCC(N)=O)CCCN1C(=O)CC1C=CCC1 C(=O)(CCS(=O)(=O)c1ccccc1)NC1CC(NC(C(CCCC)C)=O)C1 C1(CNC(=O)CSCC(F)F)CCN(C(=O)Cn2cnccc2=O)CC1 Cc1cc(C(N2CCC(C(F)CNC(=O)CCn3cncn3)CC2)=O)ccc1O N1(C(CN(C)C(N)=O)=O)CC2CC1CN2C(c1ccc(-c2ccncc2)s1)=O C1(NC(C2(C)CCCCCCC2)=O)CC(C2CCN(C(=O)Cc3ccoc3)C2)C1 c1(C(=O)NC2CCN(C(C(c3ccc(C)cc3)C)=O)C2)c(C)ccc(Cl)c1O N1(C(CCCC(=O)NCC)=O)CC2CCCC1CN(C(=O)CN1CCNC1=O)C2 c1(NC(C)=O)cncc(C(=O)Nc2ncc(C(N3CC4CCC3C4)=O)s2)c1 C1(NC(CC2CN(C)C2)=O)CCCC12CCN(C(C1COC(=O)N1)=O)CC2 N1(C(CC(n2ccc(C)n2)C)=O)CCC(C2CN(C(=O)C=CC(F)(F)F)C2)CC1 c1ccc2c(O)cc(S(=O)(=O)O)cc2c1.C1(C(=O)NCC#N)CC1C(=O)N Cc1c[nH]cc(-c2nc(COC(C)C)nn2-c2cnn(C)c2)c1=O CCC1=C(C(=O)N2CC(NC(c3nn(C)cc3C)=O)C(N=[N+]=[N-])C2)SCCO1 C1(C(=O)NC(C)CCC2CC2)CCCCN1C(c1ccns1)=O CC1(C)CC(F)(F)C1.C1(CC=O)C2CN(C(=O)CC3CCCNC3=O)CC12.N S(=O)(=O)(c1cccc(C=O)c1)NC.c1(OC)ccc(C(N)=O)cc1.C1CC1.C N1(C(C(CSC)O)=O)CC2CCCC2C1C(=O)NC(c1ccco1)CO c1(CC)nc(CCc2csc(Br)c2)n(-c2ncnn2C)n1 CC1(C(=O)NC2CCC2NC(=O)C(=O)NC2CC2)CC=CC1 C(=O)(CC(C(F)F)N1CCOCC1)NCCCN(C(=O)CC(C)C(C)C)CC c1(OC)ccc(C(=O)NC2(CO)CCN(C(=O)C3=CCOC3)CC2)cc1C1CC1 C1(C)(NC(C2C(C)C2C)=O)CCCN(C(c2nc(-c3cnccn3)no2)=O)C1 Cc1ccc(C(=O)NCc2cc(O)ncc2Br)c([N+](=O)[O-])c1 Cn1cnc(N2CCCC(CCNC(=O)C3=COCCC3)CC2)c(Br)c1=O c1(NC(=O)Nc2cc(Cl)nnc2Cl)ccc2c(c1)CC(=O)N2 C1(CNC(C(CC)OC)=O)CCN(C(=O)CCOc2cccc(Cl)c2)CC1(F)F c1(C(N2CCC(N(C(=O)CCF)CC#C)C2)=O)cnncc1C C1(C(=O)NCCCC2CCC2)(CC)CCCN(C(=O)C(O)CSC)C1 c1(OC)ccc(F)c(Br)c1C(N1CC(C)(NC(C2NC(=O)CC2C)=O)C1)=O c1(C(=O)NCCN2CCN(C(C3C(SC)CCC3)=O)CC2)ccc2c(n1)NCC2 c1(SC)ncc(N)c(C=O)n1.c1(C(N(CCC)C)=O)c(C)nn(C(C)C)c1C CCC(C(C)C)S(=O)(=O)NC(c1ccc(C)cc1OC)=O C1(NC(CCOCC)=O)CN(C(C2CCCOC2)=O)Cc2ccnn2C1 N1(C(C(C=C)O)=O)CC(C2CCCN(C(=O)CNS(=O)(=O)C3CC3)C2)C1 CC(CC(=O)N1CC(C(N)=O)(CNC(=O)CC2CN(C)C2)C1)C(F)F C=CC(O)(C(=O)N1CCCC(NC(=O)CCn2cccnc2=O)CC1)C(F)(F)F N1(C(c2nc(CC)[nH]n2)C(=O)NCC2CCCO2)CC(C)CC1C C1(C)(CNC(C=CC(C)NC(C(CSC)OC)=O)=O)CCN(C)CC1 Cc1cc(OCC(=O)NC(C)(C)CC)cc(C)c1Cl.c1(C(=O)N)cc(N)ccn1 C(=O)(C1=CCN(C)CC1)N1CC(C(C(=O)NC2(C(N)=O)CCOC2)OC)C1 C#CCCC(C(=O)NC1CC1c1ccccc1)NC(=O)CC(C)F C(=O)(CC(O)C(C)(C)C)N1CC(CNC(C(C)OCC=C)=O)OCC1 N1(C(CC)C(=O)NC2CC2CNC(c2ncccc2N)=O)CCc2ccccc21 CC1CC(N=c2nc(N3CC(F)(F)C(F)(F)C3)c3[nH]ccc3[nH]2)c2ncnn21 Nc1cc(Br)cc(Cl)c1C(=O)NCC1(C)CC1.c1(CC(=O)N)nc[nH]n1 C1(NC(c2ccco2)=O)CCN(C(C2COC2)=O)CC1F N1(C(C)=O)CC(CNC(=O)CS(=O)(=O)CC2CCCO2)OC2COCC12 c1(C(N2C(C)CC(C)C2)=O)ccc(C(C)(F)F)nc1O.C1(C(=O)N)CCN(C)C1 C1(NC(c2cn(C3CC3)cn2)=O)CCOC2(CCN(C(c3ccsn3)=O)CC2)C1 N1(C(c2cocc2Br)C(=O)NC(CC)C)CCOC(c2ccc(C)o2)C1 C1(C(N2C(C)CCC(Nc3ccncn3)C2)=O)Cc2ccccc2CO1 c1(CONC(C2CCCN2c2cnccn2)=O)ncc(Cl)cn1 C1(C(=O)NC2CCN(CC)C2)(OC)CCN(C(C2CCCO2)=O)C1 C#CCCC(O)C(=O)N(CC(C)NC(=O)Cc1cc(C(C)C)no1)CC CCCC(CNC(c1cc[nH]c1)=O)NC(=O)Cn1cnc(C(N)=O)n1 N(C(=NCCC1CCC(F)(F)C1)NCC(C)(C)C1CCCO1)Cc1cc(C)on1 C(=O)(C1=CCCOC1)NCCCC1CCN(C(C2(CC)CCCC2O)=O)CC1 c1(C(N(C2CCN(C(C3C(CN(C)C)C3)=O)C2)C)=O)ccc2cnnc(O)c2c1 C1(CNC(CC(=O)NCC)=O)CN(C(c2cnc3c[nH]nc3c2)=O)CC12CCC2 C(=O)(C(C)(C)CS(C)(=O)=O)NC(C(C)NC(c1c(C)n2c(s1)ncc2)=O)C N1(C(C=C(C)C)=O)CCC2(CCN(C(c3cccc(F)c3N)=O)CC2)C(C)C1 CC1CC(CNC(=O)CCCC2CC2)CN1C(c1ccc(CO)o1)=O n1(CC)ncc2cc(C(N3CCCC(C)C3)=O)c(C)nc12.C(=O)C=C1CCC1.N N1(C(=O)OC(C)(C)C)CCCC1C1CCCN1Cc1c(OC(F)F)cccc1Cl c1(CCC)cccc(C(N2CC(O)(C(C)NC(=O)C)C2)=O)c1.[SH](C)(=O)=O c1(C(=O)NC2CC(CCNC(C3C(C)C3)=O)C2)cnn2ccsc12 N1(C(Cc2ncc(CC)[nH]2)=O)CCC2(CCOC2)C(CNC(=O)C(C)CCO)C1 C1(=O)C(C)(C)CN2S(=O)(=O)C(C)C1=CC=CC=CC(CC)C2=O.CC.O c1(C(=O)NCC(CN(C(CCNS(CC)(=O)=O)=O)C)O)sc(F)cc1Cl C1(F)(C(N2C(C(=O)Nc3nc(OC)nc(O)c3)C=CC2)=O)CCCCC1(F)F C(=O)(CCCCC(C)C)N(CCN(C(C(COCc1ccccc1)OC)=O)C)C C1(CCOC)(CNC(=O)CSCC(=O)O)CCC1 C1(CNC(c2n(CC)ncn2)=O)CCCC(NC(=O)C(=O)N(C)C)C1 CN1CCCC12CCCN(C(=O)NCCCCCC1CCCC1)C2 c1(C(N2CC(NC(C3CCc4nncn4C3)=O)(CO)C2)=O)cnc2nccn2c1 Cc1ncc(=NC(=O)c2ccc(NCc3ccc(C(=O)O)cc3Br)nc2)[nH]c1C C(C)(C)(CCCCC(=O)NC1CCC(NC(=O)CCCCCF)C1)OC N1(C(C(CC)(F)F)=O)CC(NC(c2ccc(C(O)CF)cc2)=O)CC2(CCC2)C1 CCC1=C(C(=O)NC2CC3CCC2N3C(c2ccc3c(c2)COC3)=O)CCCO1 C1(C(C)C)CCCN1C(C1CSCN1C(C1(CF)CC1)=O)=O c1(C(N2CCC3(C(CNC(CCC=CC)=O)C3)CC2)=O)cc2n(n1)CCNC2=O C(=O)(CCCS(=O)(=O)N1CCCC1)NCCN(CCC)C(=O)Cn1cnnn1 C(=O)(N1CCCCCO1)C1COCCN(C(C2(OCC)CCC2)=O)C1 c1(OCC)ccc(C)cc1C(N1CCN(C(c2nc(C)ccc2C)=O)C2CC12)=O N1(C(C2CC(C)C2)=O)CCC2(CC1)C(NC(C1CC(F)C1)=O)CS2(=O)=O C#CCC(C(=O)N1CCC(CC)C1)NC(=O)C=CCCC C1(N(C)C)CCN(CC(N2CCCCC2Cc2cn(C3CCC3)nn2)=O)CC1 C1(NC(C2(CC=C)CCC2)=O)CN(C(=O)Cc2cncn2C)C2(CCOC2)C1 c1(C(=O)NC2C(C)N(C(c3cc4ncccn4n3)=O)CCC2)ccc(F)c(C#N)c1 c1(OC)n[nH]cc1C(=O)NC(C)C(CO)NC(c1csc(-c2ccoc2)n1)=O c1(C(N2C(C(N(CCN(CC=C)C)CC)=O)C(C)C2)=O)cnn(C)c1N c1(CC)cnoc1C(=O)NC1CCC(NC(=O)C(CC)c2ccccc2)C1 c1(C(N2CC(NC(CCSC)=O)C(O)CC2)=O)cc2cc(Cl)cc(C)c2[nH]1 C1(NC(c2c(C)nn(C3CC3)c2)=O)Cc2ccccc2C1NC(C1(O)CCC1)=O Cc1cc(C(=O)NCCc2cccnc2Cl)cc(-c2ccc(CO)cc2)c1 c1(C(N(C)CC2CCN(C(=O)CC3NC(=O)NC3=O)CC2)=O)cc(Br)ncc1Cl Cc1ncc(Cl)c(C(=O)NC2CN(C(c3cc(F)ccc3C(F)F)=O)CC2C)n1 CCCCC(CC)CCCNC(c1cc(F)c(Br)cc1OC)c1nnnn1CC C1(O)(C(C)NC(Cc2c(C)ccs2)=O)CCN(C(C2(C#N)CC23CCC3)=O)CC1 c1(COCCN(C)C)cn(CCC(=O)NC2CCN(C(N)=O)C2)nn1 c1(NC(C23C(CN(C(=O)Cc4cccc(F)c4)C2)C3)=O)cc(Cl)ncc1I CC(C)CC(C)CC(=O)N(CC(O)CNC(c1occc1-c1cnn(C)c1)=O)C C1(CNC(CCC2CC(OC)C2)=O)CN(C(=O)C=CSC)CCC12CCOC2 C1(O)(C(N2CCC(CNC(c3ccc(OC)s3)=O)C2)=O)CCCC(C)(C)CC1 c12cc(on1)COC2.CCCCC1(C(=O)N(C)CCN(C)C)CC1 C(=O)(C1=C(C)CCCC1)N1CCC(CNC(COCC(=C)C)=O)C(C)C1 C1(C(=O)NCCCC(=C)C)CCN(C(=O)CN2CCCCCC2)C1CC CCC(CC(=O)N(C1(C=O)CCC1)C1CC1)C1CCC1.C1CN(C(C)=O)C1.N N1(C(C)=O)CCCC(O)C1.C1(C=O)CCS(=O)(=O)C1.CC(C)(C)OC=O.N C(=O)(C(C)(C)CCC(=O)N1CCC(C)C1)OC.n1(CC(=O)N)nc(C)ccc1=O c1(C(=O)NC(C(C)O)C(=O)NCC2(C)CCCC2O)ccccc1C#N N1(C(Cc2c(C#C)cccc2)=O)CCC2(CCCN(C(c3ncc[nH]3)=O)C2)CC1 c1(CNC(c2c(C(=O)OC)n[nH]c2)=O)cnccc1-c1nn[nH]n1 n1(C(C)C)ncc2cc(NC(N3CC(CCO)OC(C)(C)C3)=O)ccc12 c1(CC)ccc(OCCN(C(C)(C)CN2CCCC(C)C2)C)cc1.C1C(C)N1 N1(C(CCCC)=O)CCN(C)CC1CNC(=O)CC(C)C1CCCC1 CCC(F)(C(=O)OC)C(=O)NC1CN(C(c2cc(C)cc(C)c2)=O)CC(C)(C)C1 c1(C(N2CCOCC(C(=O)N(C3CC3)CC3CCOC3)C2)=O)n[nH]c2c1CCC2 c1(CNC(N2CC(C)NCC2)=O)ccc2c(c1F)CCC2 c1(C(N2CC(NC(CC=C)=O)C(OC)C2)=O)ccc(N=S(C)(C)=O)cc1 N1(C(c2cc(CC)n(C)n2)=O)C2CC=C(C(=O)NOC3CCCCC3)C1CC2 N1(C(COc2ccc(C(C)=O)cc2)=O)CCCC12CCN(C(=O)Cc1ccco1)C2 Cc1cc(CNC(C2CC(NC(=O)CC(C)(C)C)C2(C)C)=O)ccn1 Cc1ncc(NC(C2CC(O)CN2Cc2cccc(Oc3ccccc3)c2)=O)n1C N1(CC(=C)C)CCN(C(c2ccc(OCC(C)C)nc2)=O)CC1=O c1(C(N(CC(C)C)C)=O)cnn2c1N(C)CC2.c1(C=O)ccc(C=O)[nH]1.CO c1(C(=O)NC2(C)CC(NC(C3(C)CC=CCC3)=O)C2)cn2ccccc2n1 CC1CN(C(C2(C(C)(F)F)CCOCC2)=O)CC(C)N(C(=O)Cc2cscn2)C1 n1(CC(N2CCCC23CC3)=O)nc(C)c([N+](=O)[O-])c1C.CCC(C(=O)NC)OC C(=O)(CC(C(F)(F)F)NC(=O)C(C)C(C)(C)C)Nc1c(C)ccc(C)c1 C1(CCCNC(C=CCC)=O)CCN(C(C2CCN(C(=O)CC)C2)=O)CC1 C1(NC(c2cnc(C(C)=O)s2)=O)CC(F)CN(C(=O)C(F)(F)C(C)O)C1 C(=O)(C(C)CN=c1[nH]c(=NCCC2CC3C=CC2C3)c2ccccc2[nH]1)NC c1(CNC(c2ccc(CNC(c3ncn(CC)n3)=O)o2)=O)cccnc1Cl Cc1oc(C2CC2)nc1C(=O)NCC.c1ccncc1.C(=O)(C)N.C(N)=O C(=O)(CCC(C)C)NCC(C)(C1CC1)OC.C1(C=O)CC2CC(=O)C1O2.N c1(OCOC)cc(-c2ccc(NC(=O)NC3(C)CCOCC3)cn2)ccc1C C(=O)(C(F)(F)C(F)(F)C(F)F)N.C1(C(=O)NCC(C)C)Cc2ccccc2CO1 c1(OC)ccc(-c2cc(C)cs2)c(CN(C)Cc2ccc(Cl)c(C)c2)c1 c1(C(N2CC(NC(=O)CC3CC4(CC4)C3)C(O)C2)=O)ccc(F)cc1Cl N1(C(c2cc(CCC)c(C)s2)=O)CCCC(NC(=O)C(C)C2CC2)C1C c1(CC)cc(C(=O)N(C)C)ccc1F.C1CC(F)CN1C(=O)C=CC1CCOC1 c1(N2CC3C(C(NCC)=O)C3C2)ncc2c(n1)NC(=O)C2.c1cccc(O)c1.C c1(N2CC(C)Oc3c(cccc3)C2)nc(=NCC2=COCCO2)[nH]c2cc[nH]c12 c1(OCC(=O)NCCC2CN(C(CC(CC)O)=O)C2)cc(C)ccc1Cl CCC(CC)CC(=O)NCCC1(O)CN(C(=O)C(O)C2CCCC2)C1 c1(CC(=O)N)nn(C)cc1[N+](=O)[O-].Cc1nc(C(=O)NC(CC)C(C)C)nn1C C1(C2CCCO2)(C(=O)NCCC2(NC(CCC=C(C)C)=O)CC2)CCOCC1 C1(NC(CCCC)=O)CN(C(=O)Cc2ccc(OC(C)C)cc2)CC1OC Cc1nccc(C(N2CCC(NC(c3ccsc3C(F)(F)F)=O)CC2C)=O)c1N c1(C(=O)NC(C)C(C)NC(=O)C(F)OC(F)(F)F)cc(F)cnc1O n1(CC)ncc(C(=O)NC(CNC(=O)C2CC2)CO)c1C C(C)(CC(=O)NCCCOCCOCCNC(c1cnsc1C)=O)SC N1(C(C(F)=CC)=O)CCN(C)C(C)C1.c1(CC(=O)N)ccccc1.C(C)C C1(NC(c2c(C)ncnc2)=O)CN(C(=O)Cc2ccnc(F)c2F)C(C)(C)C1 C12(NC(CC(C=C)C)=O)CC(CNC(=O)CN3CCC(C)CC3)(C1)OC2C c1(CCC(=O)NCC)cnc(C2CCC2)o1.N#CC1CC1C(=O)N.C1CC1 c1(N2CCC(NC(CC3CC(OC)C3(C)C)=O)C2)ncc(Br)c(C)n1 C(=O)(CC1=Cc2ccccc2C1)N1CC(C)N(C(C2C(C)(C)C2(F)F)=O)CCC1 c1(C(C)=O)ccc(O)cc1NC(C1CC(F)CN1C(C1CNC(=O)C1)=O)=O Cc1ccc(CNC(=O)C(C)C(C)NC(C2CC(=O)CCO2)=O)cc1C c1(C=O)ccc([N+](=O)[O-])cc1F.Cc1oc(C#N)cc1C(=O)NCC(C)(C)C.N C1(CNC(=O)C(N2CCN(Cc3csc(Br)c3)CC2)=O)CCOCC12CCC2 Cc1ccc(C(=O)NCCCNC(C2CC2c2ccc(Cl)s2)=O)c(C)c1 Cc1ncc(Br)c(C(N2CCC(C)(CNC(C3COC(=O)N3C)=O)C2)=O)n1 c1(OC)cnc(Cl)nc1N(C)CC1CCCN1C(C1CCC(C)=C(C)C1)=O Cc1cc([N+](=O)[O-])ncc1C(=O)NC12CCC1CN(C(=O)C(C)S(N)(=O)=O)C2 Cn1ncc(=NC(=O)C2CCCC23CN(C(C2CCCCO2)=O)C3)[nH]1 C(=O)(C1=C(C)CCOC1)NCCC1(NC(C(CC)N(C)C)=O)CCCC1 c1(C(N2CCOC(C)(CCO)C2)C(=O)NCCSC)cc(=O)c2ccccc2o1 C1(NC(C(C=C)(C)C)=O)CC2CCC1CN2C(c1cccc(F)c1F)=O c1(CC)cc(C(N2CCCCC2CN(C(=O)CC2CCCC2O)C)=O)oc1CC C1C(C)(C)C1(C)C.c1(CCC)ncoc1C(=O)N.C(C(=O)NC)C1(C)CC1 N1(C(C=C(CC)CC)=O)CCC2CN(C(=O)COCCCN(C)C)C(C)C12 C(Cc1ccccc1)(C(=O)N1CC(CC(C)NC(=O)C)C1)OC.C1(C)CCC1 C1(C(N(CC(C)NC(=O)Cn2ccc(C3CC3)n2)C)=O)CCOC(=O)N1 C1(CCOC)(NC(C2(C3CCCO3)CC2)=O)CCN(C(c2csnn2)=O)CC1 c1(CCN(C)C(=O)NCC2C(F)(F)C23CC3)ccc(F)cc1 N1(Cc2c(C)ccc(OC)c2)CC2(CN(C(c3c(Br)cnn3C)=O)CCO2)C1 N1(C(C2CC(CNC(C(COC)C)=O)OC2)=O)CC(C(N)=O)C2(CC2)C1 C1(CNC(c2c(C)cco2)=O)CN(C(=O)Cc2cccc(O)c2)CC(C)(C)O1 CC(C)(C(=O)NC1C2CCC3C(C2)CC13)C1=CCN(C(=O)CC2CC=CCC2)C1 C1(C(C)CN(C)C)CCCCN1C(CCC1CC1)C(=O)Nc1ccc(F)cc1 C1(CNC(C(CC(C)C)C)=O)CN(C(=O)CN2CC(C)C2)CCC1(F)F c1ccc(CCC(c2nnnn2Cc2cccs2)NCC(C2CC2)C2CC2)cc1 c1(C(=O)NC2CCN(C(c3ccc(C)nc3)=O)CC2C)cc2cncc(C)c2s1 C=CCC(C(=O)N1CCN(C(=O)C(O)CC2CCCC2)C(C)C1)C(C)C c1ccc(C)cc1.N1(C(C(C2CC2)OCC)=O)CC=CC1C.C(=O)CCC.N CN1C(=O)c2ccccc2C1C(=O)NC(CNC(c1cccnc1)=O)CO c1(C(=O)NC2C(NC(c3c(CC)occ3)=O)C2)ccnc(Cl)c1O C=CCCC(CC(C)C)C(=O)NCC(C)CNC(=O)CN1CCNC(=O)C1 Cc1nn(C)c(C(N2CC(F)CC2C(=O)NC(c2ccccn2)CO)=O)c1F c1(CNC(c2cccc(OC)n2)=O)n[nH]c2c1CN(C(c1cc(C)cs1)=O)CC2 c1(COC)cc(C(=O)NCC2CN(C(C34CCC3C4)=O)C2)n[nH]1 N1(C(CCC(=O)N(C)C)=O)CCCCC(C(=O)NOCc2ccc(F)cc2)C1 c1(OC)cc(C)sc1C(=O)NCC1CC(NC(=O)C(N2CCOCC2)C)C1 C1(CNC(=NCCOC)NCc2csc(C)c2C)COc2ccccc2C1 Cc1cccc(OCC(N2CCC(OCCNC(=O)CC)C2)=O)c1.C1CC1.O C1(C)(CNC(C(N(C(=O)CC2OCCO2)C)C2CC2)=O)CC=CCC1 N1(c2snc(SC)n2)CC23CCCC2(CN(C(=O)C(C)(C)C(F)F)C3)C1 c1(C(=O)N)cc2c(F)c(C)ccc2[nH]1.C1(NC(C2C(CC)CCO2)=O)COCC1 C(C)(C)(CC(C)=O)NC(C(=O)NCC(c1ccccc1)OC)=O N1(c2ncc(CC)cn2)CC2CN(S(=O)(=O)Cc3ccc(C)cc3)C2C1 c1(OC)ccc(F)c(C(=O)N(CCCNC(C)=O)C)c1Cl C1(C(=O)NC2(c3cccnc3)C(C)C2)CCCSC1 N1(C(Cc2cnc(C)s2)=O)CC(O)CC1(C)C(=O)N(C1CSC1)C N1(C(c2cc(C)c(Cl)cc2)=O)CC2CN(C(=O)C(C)(F)F)CC2(C)C1 C(=O)(C(C)=Cn1ccnn1)NC(C1N(C(C(CC)O)=O)CCC1)(C)C CCC(O)(CC)C(C)(C)CNC(C1CC1C1CC(N=[N+]=[N-])C1)=O C=CC1(CO)CCN(C(=O)C(CC(C)C)NC(C2CCCN(C)C2)=O)CC1 CC(C)S(=O)(=O)C(C)C=O.c1(C=O)cc(S(N)(=O)=O)c[nH]1.C(C)(C)CO.N CCC(CC(F)(F)F)N=c1nc2scnc2c(NC(c2cnccc2C)C)[nH]1 Nc1cc(F)c(O)cc1C(N1CCC(CCNC(C2CC3(CCCO3)C2)=O)C1)=O c1(C(N2C(C3CCN(C(C4CC(C)OC4)=O)C3)CCC2)=O)ccc(=O)n(C)n1 O=C1CC(NC(=O)CC2COCCN2C(=O)COC2CC=CC2)C(=O)N1 CC1c2cc(C(=O)NCCNC(c3ccc4nc(O)[nH]c4n3)=O)ccc2OC1C Cc1c(C(=O)NCC2CCCCN2c2cncc(Cl)n2)cnn1C1CCCC1 c1(CC(=O)NC2C3CCN(C(C(C)NC(CC)=O)=O)C32)cnn2c1CCCC2 C(CC(=O)NOCC(=O)N(C(C)CCO)C)=CC.C1CC1 N1(C(CCN(CC)CC)=O)CCC2(CC1)CC(C)N(C(=O)C=C1CCOCC1)C2 C1(NC(c2cc[nH]c2C2CC2)=O)CCCCCCC1NC(C1CC1(Cl)Cl)=O C1(C(=O)NC(CCNC(c2c(C)oc(C(C)C)n2)=O)C)COc2ccccc2O1 N1(C(C)=O)CCCC(O)(CC(=O)NC2CCC2CNC(=O)CCCCC#N)C1 c1(N(CC(CC)O)C)ccncc1S(=O)(=O)N1CCCC(CC(F)F)C1 c1(C(NOCc2cn(Cc3scc(C(=O)OC)n3)nn2)=O)noc2ncccc12 c1(CCC(=O)N(CCNCC)CC)ccccc1F.c1cc(CC(C)C)on1.C C(CSC)(C(=O)NCCCN(C)C(C1(F)CCOC1)=O)OC N1(C(C(CCOC)(C)C)=O)CCC=C(C(=O)NCC2(C(C)C)CCCC2)C1 c1(C(=O)NCC2(C)CN(C(CS(CC)=O)=O)C(C)(C)C2)cc([N+](=O)[O-])cnc1C C(=O)(CC(C)(C)C(=O)N1CCCOC(C)C1)OC.c1(C=O)cc(C(F)F)cs1.N C1(C(=O)NCC2N(C(CCCCCC)=O)CCC2C)CCc2cnn(C)c2C1 c1ccc(O)cc1F.c1(CNC(C2CCCN(C)C2)=O)cc(Cl)ccc1OC(F)F C1(C(=O)NC(CC=CC(=O)NCc2nnc(C)o2)(C)C)CCOC(C)C1 CCCC(C(=O)OC)C(=O)NC1(CO)CCN(C(=O)C(CC)NC(C)=O)CC1 Nc1c(Cl)c(C(N2CCC(NC(C3CCC(F)(F)CC3)=O)C2)=O)cc(F)c1Cl c1(CCC)cc(C(=O)N(C(CC)C(=O)N(CCC(F)(F)F)CC)C)n[nH]1 C1(C(C)C#N)CCN(C(C2COC(C)C2)C(=O)NCc2ccccc2)CC1 C(CC(C(=O)NCCOCCCO)NC(C1CC(O)C(F)C1)=O)SC CC(C(=O)NCC(C(C)(C)C)NC(=O)C=CC1CCCCC1)C(C)(C)O c1ccc(Cl)cc1.c1(C(C)NC(C2(CNC(=O)CC)CC2)=O)ccncn1 C(=O)(CC1COCc2ccccc21)NCC1C(NC(C2C(=C)CC2)=O)CCCC1 Cn1c(=O)c2cc(NC(=O)C(F)(F)CC3CNC3)cnc2n(C)c1=O c1(C(=O)NC(CNC(CCCCC#C)=O)CCC)ccc2[nH]nc(Cl)c2c1 N1(C(c2c(OC)ccs2)=O)CCC(NC(=O)C(C)SC)C(C)(C)C1 CC1(C)CCC(C)(NC(C2CCOCCN2C(c2ccc(C#N)s2)=O)=O)CC1 c1(-c2ccc(OC)c(C)c2)ccc2occ(CC(=O)N3CC(O)CCO3)c2c1 C1(C(=O)NCCC(CNC(C(N)=O)=O)O)CCCC12CCC2 Cc1ccc2cccnc2c1C(=O)NC12CC1CN(C(=O)C(C)SC(F)(F)F)C2 c1(C(=O)N)cc2cnccc2o1.N1(C(C(C)NC(=O)C(C)(C)C)=O)CCC(O)C1 CCCC(C(=O)NC1CN(C(=O)C2CC2)C1)NC(C1(C)CCSCC1)=O C1(CNC(NC(c2cccs2)C)=NCC2CC2)C2CC3CC(C2)CC1C3 C(C(C)(C)CN=C(NC(C)C)NCC(C)(O)Cn1cc(Br)cn1)OC C1(C(N2CC(C#C)(N(C)C)C2)=O)CCN(C(=O)C(C)n2cncn2)CC1O c1(C(C)NC(C(n2cc(CCN(C(C)(C)C)C)nn2)C)=O)ccc(Br)c(F)c1 c1(CC(=O)NC2CCC2CNC(C2CCC(O)CC2)=O)ccc2[nH]ccc2c1 N1(C(c2cc(C)cc(Cl)n2)=O)CCOC2CN(C(=O)C=Cc3cccs3)CC12 C(=O)(CCCCCF)N1CC(CC(N2C(CC)CCCC2)=O)C(C)C1 c1(C(=O)NC2C(C)CN(C(c3cncc(CO)c3)=O)C2)c[nH]cc(Br)c1=N C1(C(=O)NC2CCN(C(c3c(C)nco3)=O)CC2O)CC2(C1)CC(C)(C)C2 C#Cc1cc(C(=O)N(C(CC(F)F)C(=O)NCc2nc(C)sc2C)C)ccc1C c1(C(=O)NC2CN(C(c3c(OC)n[nH]c3)=O)CC23CC3)c2c(nn1C)CCC2 C1(CNC(c2cnc(=N)[nH]c2)=O)CC(C(F)F)CCN1C(=O)Cc1cccnc1 C(CN=C(NC1CC1C(F)(F)F)N1CCC(CON2CCOCC2)C1)SC N1(C(CC2C(C)CCN(C(c3ncn(CC)c3)=O)C2)=O)CCc2c[nH]nc2C1 C(C(C)C(=O)NC1CC(CCNC(=O)C(O)Cc2cnn(C)c2)C1)SC N1(C(C(n2c(C)ccn2)C)=O)CCC(NC(=O)CSC(C)(C)C)CC1 C(C)(C(C)(C)C(=O)NC)NC(c1c(CC)n(C)nn1)=O.C1CCC1C=O C(=O)(C(CC(F)F)NC(=O)C(F)OC(F)(F)F)NCC(NOCC)=O C1(F)(CSC)CN(C(C2(CC)CC2)=O)C1.C1(C=O)CCOC1C1CC1.N C1(C(=O)NC2CCC(NC(c3c(C)cccc3Cl)=O)CC2)CCC2C(C1)C2(F)F C1(C(=O)NCCCC(C)NC(=O)CC(C)(F)F)CC1C1CCOCC1 N1(C(c2c(OC)ccc(C(F)F)c2)=O)CCCC2C1CCN2C(C1CCOC1)=O C#Cc1cccc(CC(=O)NCC(C)=CC(=O)NCc2ccc(C#N)cc2)c1 C1(Nc2cc(NCC(COCC)(F)F)nc(C)n2)CCn2ncnc2C1 CC(Cc1cnn(C)c1)C(=O)N(C)C.C1CCN(C(c2coc(C(F)F)c2)=O)C1 Cc1ncc(C(=O)NC2CCC(CNC(C3CCC(C(N)=O)C3)=O)CC2)n1C Cc1ccc(CNC(=O)N(C2CCOC2C)C)c(Br)c1 Cc1oc(C(C)C)nc1C(N1CCOC(CC)C1)=O.C(c1nccs1)=CC(=O)N C1(O)(CNC(c2ccn(CC)c2)=O)CCCC1.C1(C=O)CCOC1C1CC1 C1(NC(COCCOC)=O)CN(C(=O)Cc2cc[nH]n2)CC2(CC2)C1 C(=O)(N=c1cc[nH]cc1Cl)c1scc(-c2c(C)c(F)ccc2)c1 Cc1nc(C)c(C(=O)NCC(=C2CN(C(=O)C(C)C(C)O)C2)F)o1 c1(C(=O)NCCOCCN(C(c2scc(C)c2C)=O)C)ccc(O)cc1F CC1CCC(=CC(=O)NC(C2(O)CN(C(C3COCCO3)=O)C2)C)C1 C1(NC(C=Cc2nc(C)sc2)=O)CC12CCN(C(=O)C(C(C)C)N(C)C)CC2 C(=O)(C(CO)C(C)(C)C)NC12CN(C(CN(C(C(C)C)=O)C)=O)C(CC1)C2 C1(CNC(C=CSC)=O)N(C(c2cc(Br)c[nH]2)=O)CCCC1(C)C c1(C(=O)NCC(CNC(c2ccc(C)c(F)c2N)=O)C)cncc2ncn(C)c12 Cc1nn(C)c(NC(C2CC(O)CN2C(c2ccc(O)nc2Cl)=O)=O)c1Cl c1(C(N2C(C)CC(NC(c3cc4cnccc4o3)=O)C2)=O)cc(F)c(F)cc1Cl Cc1cc(C(=O)NCC2CC2CNC(=O)Cn2cnnc2O)cc(C)c1N c1(C(=O)NC2CC(NC(COCCCOC)=O)C2)scc(C)c1C c1(C(=O)NC(CC2CCC2)C(N2Cc3ncsc3C2)=O)ccc2[nH]nc(Cl)c2c1 C1(c2n(C(C)C)nnn2)(NCC23CCC(CC2)O3)CNC(=O)C(C)(C)C1 c12ccc(cc1)C=CCc1cn-2nn1.c1(NC)nc(CNC=O)cs1 c1(N2CC(CNC(c3c(C)cno3)=O)C(F)(F)CC2)ccc([N+](=O)[O-])c(C#N)c1 N1(C(CCc2cn(C)nn2)=O)CC2CCCC2(CNC(=O)C(C)(C)C)C1 c1(N(C2CCN(C(C3COc4cscc43)=O)C2)C)nccc(-n2ccnc2)n1 C1(NC(=O)CC(O)C2CC2)(CF)CCN(C(=O)C(=O)Nc2ncc[nH]2)C1 C(=O)(C(CO)C(F)(F)F)N(C)CC1CCCN1C(=O)C(F)CC1CCOC1 C(=O)(C(C)(C)CO)NC(C(C)NC(=O)CCNC(C1CCCO1)=O)CO N1(C(c2cccc(C)c2)=O)CCC(O)(c2nc(-c3ccc(F)c(F)c3)no2)CC1 N1(C(c2cc(C)nnc2O)=O)CC2CC1CN(C(=O)CCC1CCCOC1)C2 N1(C(c2cc(CC)no2)=O)CCC(NC(c2sccc2C(F)F)=O)C12CCCC2 c1(OC)ccc(Cl)cc1C=CC(=O)NC1CCN(C(=O)Cc2nc[nH]n2)CC1C C1(O)(CNC(C(Cc2cn(C)nc2)O)=O)CCN(C(c2ccncc2N)=O)C1 CC1CCC(CNC(c2ccc(N(C)C)cc2F)=O)CN1C(=O)Cc1cn[nH]c1 O=C(N=c1[nH][nH]c2cccnc12)C1CCCN1Cc1cc(C(F)(F)F)ccc1Br C1(C(N2CC(SC)CC2)=O)CC2(CCOCC2)C1.C(=O)(CC=CC(C)(C)C)N C1(CC#C)(C(N2CCC(NC(C3(CC)CCCCC3)=O)C2)=O)CCCCO1 CCC(CCCC(=O)NOCCCC(F)(F)F)NC(=O)CC1CCC(=O)C1 c1(C(=O)NC)cccc(NC(c2ncsc2Br)c2nnnn2C2CCCC2)c1 c1(C(=O)NC(C(=O)OC)Cc2cn(CCCCO)nn2)cc(C)nc2cc(C)nn12 C1(CC)Cc2ccccc2C1N=c1[nH]c(N2CCC(F)(CO)C2)nc(=N)[nH]1 Cc1nc(CC(=O)NCC(C)N(C(=O)CCC2CCCN(C)C2)C)sc1C CC(C(=O)N1CCC(CCN(C(=O)C(c2ccnn2C)C)C)CC1)C(C)(F)F c1(C(=O)NCC(CNC(c2ccc(=NC)[nH]c2)=O)OC)cnc2c(c1)ncn2C Cc1ccc(CNC(=O)NC2CCN(S(C)(=O)=O)C2)cc1O CCCCCC(F)C(=O)NCC(O)CNC(C1CCS(=O)(=O)N1)=O N1(C(C=CCCC)=O)CCN2CCN(C(=O)C=CSc3nc[nH]n3)CC2C1 N1(C(C(CC)CC)=O)CCCCCC(NC(=O)Cc2cc(F)c(N)cc2F)C1 C(=O)(C(C)(C)C(=O)N1CCC(NC(=O)C2=CCCCC2)C(O)C1)OC(C)(C)C c1(OC)ccc(COCC(N2CCN(CC(C)C)CC2)=O)cc1C C=C(C)C(O)CC(=O)NC1(C)CC(NC(c2ccc(Cl)cn2)=O)C1 Cc1cc(C(=O)NCCC2CCCCN2C(C2CCCCN2C)=O)n(C)n1 N1(c2nc(OC)cc(OC)n2)CC(C)(C)CCC1CNC(C1CCCC1O)=O S(=O)(=O)(c1c(F)ccc(Br)c1F)N(C(=O)COc1cncc(Cl)n1)CCO c1(C(c2nnnn2C)Nc2ccc(-c3c(C)nco3)cc2)cccc(F)c1Br C(=O)(C(O)C(F)(F)F)NC1CC(C(NOC(C(=O)OC)(C)C)=O)CC1O C12(C=O)CC(CCO1)N(C(=O)CC1(C)CCC1)C2.C(C)(C(F)(F)F)OC.N CC1(C)CN(C(c2cc(Cl)ns2)=O)CC(CNC(=O)CC2CC3CC3C2)O1 c1(CC)ccccc1CC(=O)NCCC(C)(C)C.c1(CCC(=O)N)ccn(C)c1 N1(C(C)C)CCCCC1CNC(C1CN(C(=O)CCc2ccccc2Cl)C1)=O c1(C(=O)Nc2ccnn2CCCO)ccc(=NCc2cccc(O)c2F)[nH]c1 c1(C(=O)NCC(C)(C)NC(=O)CCCC2CC2)cc(-c2ccccc2)ccn1 CCC(F)(F)CC(=O)N1CCN(C(=O)CCC2CCCCN2C)CC1C N1(C(c2c(C)noc2)=O)CC2CCC(C1)N(C(=O)CCCC1CCCO1)C2 N1(C(C(=O)Nc2ccccc2)COCC2CCOC2)CCCC2(CCC2)C1 C(CC(C)C(=O)N(C)CCN(C(c1ncoc1C1CC1)=O)C(C)C)OC C1(NC(C2(NC(c3c(C)nccc3)=O)CCCCC2)=O)CCC(C)(C)C(C)C1 Cc1nc(SCC(=O)NCC2CC2CNC(=O)CC2COCC2O)n[nH]1 N1(C(c2cccc(C#C)c2)=O)CC2(CCC(CNC(=O)C(C)c3ccsc3)O2)C1 N1(C(c2cc3cnccc3o2)C(=O)NCCCOC)CCOCC12CCOC2 N(C1c2ccccc2C2CCC1C2)C(C1CC1c1cc(Cl)cc(Br)c1)=O c1(C(=O)NCCN(C(C(C(CC)C)OC)=O)C2CC2)ccc2oc(=O)oc2c1 N1(C(c2ccc(C)s2)=O)CCCC(CCNC(C2NC(=O)C3CC23)=O)CC1 c1(OC)c(CN2CCN(C(c3cc(C)cs3)=O)C3CC23)cc(Cl)cc1Cl CN1C(=O)NCC1C(=O)NCCCNC(c1ncoc1C1CCCO1)=O c1(SC)nc(NCCN(C)CCc2ccc(Cl)s2)cc(=NCC(C2CC2)S)[nH]1 N1(C(C2N(Cc3ccc(C)c(C)c3)CC(O)C2)=O)CCN2C(=O)OCC2C1 N1(C(CN2CC(CC)C2)=O)CCCC(CCNC(c2cc(OC)cnn2)=O)CC1 CCCC(C#N)C(=O)N1CCC=CC1C(=O)NC1(c2ncccn2)CC1 c1(CC(C=O)NC=O)cccc(Cl)c1.Cc1n[nH]cc1C(=O)NC(C)(C)CC.N C(=O)(C(CC1CC(C(=O)OC)C1)N(C)Cc1nc(=O)o[nH]1)NCCCC N1(C(CCCc2nc(C)sc2)=O)CCCN(C(c2cc(C(F)F)n(C)n2)=O)CC1 Cc1cc(C(O)CNC(c2ccc(Br)c(Cl)c2)=O)cc(C)c1 CC1(C)COC(C(=O)NC2CC(C)(NC(c3c[nH]ccc3=O)=O)C2)CO1 c1(OC)ccc2cc(C(N3CC(N(C)C(c4nncs4)=O)C3)=O)nnc2c1 C1(NC(C2CCCN(C(CC)=O)C2)=O)CN(C(=O)COCCO)CC1(C)C c1(CC(N2CC(NC(=O)COC3CCOC3)CC(C)C2)=O)cnc2n1CCOC2 C(CC(C)C)(C(=O)N(C1C2CN(C(=O)CS(N)(=O)=O)CC12)C)OC CN1CCCC(N=c2nc(N3Cc4ccc(Cl)nc4C3)c3ccccc3[nH]2)C1 c1(Cc2c(C(=O)OC)scc2)cccc(C(=O)NCCN2CCOCC2C)n1 c1(OC)cc(F)c(Cl)cc1C(=O)NCC1CCN(C(=O)Cn2nccn2)CC1 C(=O)(CCCCNC(=O)Cc1nc(=N)[nH][nH]1)NCCC1CC(C)(C)C1 c1(C(=O)NCCOC2CCN(C(C3(C)CCOC3)=O)C2)cnc2c[nH]nc2c1 c1(-c2nc(C(C)OC)n(Cc3cccc(C)n3)n2)ccc(C)c(F)c1 N1(C(COCCC=C)=O)CCC2CCN(C(=O)C(C(C)C)N3CCCCC3)C2C1 C1(C(N(CCNC(c2snc(C)c2N)=O)C)=O)CC2(C1)C(F)(F)C21CC1 c1(C(C)(C)C(=O)NC2CCC2C)c(F)cccc1F.C1(C=O)CCC(=O)NC1.N C(Cc1cnc[nH]1)(C(=O)N(C(C)C(F)F)C)NC(CSCCCC)=O c1(C(N(CCC(C(C)C)NC(C2C(C)C2C)=O)C)=O)cc(=O)n(C)cn1 c1(CC)nc(O)c(C(N2CC3CC(NC(=O)C(C)(O)C(C)C)CC2C3)=O)cc1C c1(CN(C)CCN(C)C(c2coc(C3CC3)n2)=O)nnn(C)n1 C1(C(N2C(C)CC2C(=O)NC(CO)C2(O)CC2)=O)C(C#N)C1(C)C N1(C(C(CC=C)CC)=O)CCOC2CN(C(c3sc(C)c(C)c3C)=O)CC12 Cc1ncc(CC(=O)NCC2(NC(C3CCC3c3ccccc3)=O)CCC2)o1 c1(CC)cc(C(=O)NC2CN(C(c3cnc(Cl)[nH]3)=O)CC2(C)C)cc(Cl)c1 c1(C(N(C)CC2CCCN2C(c2ccn(C)n2)=O)=O)[nH]nc([N+](=O)[O-])c1Cl.C C(C(=O)NC(CC1CC1)C1CC1)(N(C(C=CC=CC)=O)C)C1CC1 C#CCCCCCCC(=O)N(CCC(=O)Nc1ccc(COC)cc1)C CCCCCC(O)C(=O)NC(C)(C)C(C)NC(=O)CCCSC(C)(C)C c1(-c2cnc(CNC(C(CCC)C)=O)nc2)ccc(OC)cc1OC CCCC(O)CC(=O)N1CCC(O)(CNC(c2ccc(C)c(CC)c2)=O)C1 N1(C(=O)Cn2cc(Cl)cn2)CCCN(C(=O)C2CC2)C(CO)C1 C(C1CN(C(=O)C(C)CC2CC2)CC1C(=O)N(CCC)C)=CC.C(C)C.O N1(C(C2C(C)C2)=O)CC(c2ccccc2)(NC(=O)C(C)n2ccnc2)C1 C1(C)(CC)C=C(C(=O)NCC2CCC2C(=O)Nc2cnccc2CO)C1 c1(CC=O)ccc(C)c([N+](=O)[O-])c1.c1(CC)nnc(N(CC)C)s1.C1CC1 CCCCC(CC(=O)NCc1scnc1C)NC(=O)C(c1cnn(C)c1)O N1(C(COCC(=C)C)=O)CCC(F)CC1C(=O)NC(c1noc(C)n1)CC c1(C(N2CCC(N(C(=O)CN3CCC3)CC#C)C2)=O)ccc(O)c(Cl)c1.C N1(C(c2c(CNC(CCOC)=O)nnn2C)=O)CCC2(CCOCC2)C1 c1(C(N2C(C)CC(NC(C3(C)CC4CC4C3)=O)CC2)=O)cnc2nccnc2c1 C(=O)(C1=C(CCl)N(C2CC2)C(=O)NC1c1cccc2c1CCOC2)OC(C)(C)C N1(C(c2cc(CCC)ncc2)=O)CCN(C(=O)C(C2CCOCC2)C)CC1CC CN1CCN(c2nccnc2F)CC1CNC(=O)CCF c1(C(N2CC(N(C(c3c(C)nc(CC)s3)=O)C)C2)=O)cnc2snc(C)c2c1 CS(=O)(=NC(=O)CCN1C(=O)NC(c2cc3ccccc3o2)C1=O)C1CCC(N)C1 C=C(C)CCC(=O)NCC1CCCC(NC(=O)CC(C)(C)SC)C1 CC1CN(C(C2C=CCN(C(c3cc4cccnn4c3)=O)C2)=O)c2ccccc21 CCC(CC)C(=O)N1CC(c2cn(-c3ccccc3Br)nn2)C1 C(C(C)CC(C)(C)C)NC(C1N(C(C(N2CC3CC3C2)C)=O)C2C(C1)C2)=O C1(NC(C2CCCCCC2)=O)COCCN(C(=O)CC2CCCS2(=O)=O)C1 N1(C(CC2CCN(C)CC2)=O)CCCC(NC(c2nc(C3CC3)cs2)=O)CCC1 c1(C(=O)NCC2C(C(=O)NCC3(C)CCCC3)CCO2)ccc(O)c(F)c1 C1(NC(Cn2c(C)ncc2)=O)CC2CC1CN(C(=O)C(C)(C)C)C2 CCC(C(=O)NCC(C)CNC(c1cccn1C1CCCC1)=O)C1CCOCC1 c1(C(=O)NC(C(=O)OC)CC2CCCCN2C)cnc2c(Br)c[nH]c2c1 CC1(C)CC(C(=O)O)CC(C)(C)S1.c12c(cccc1F)NC(=O)NCC2 C(CCCC(=O)NCC(C)(C1CCC1)NC(=O)Cc1cccn1C)N(C)C c1(C(N2C(CNC(=O)CCF)CC(OC)C2)=O)ccc(Br)cc1F C(CN=c1[nH]nc(C(F)F)o1)(c1ccccc1F)NC(COCCOC)=O c1(CC(N2CCOCC2)=O)ccc(S(N)(=O)=O)s1.Cc1ccccc1C(=O)N.C c1(C(=O)NC2CC(NC(C3CCC4CCC34)=O)C2)ccc2c(n1)CCCN2 c1(C(=O)NCC(C(=O)NC2CC2c2ccsc2)N(C)C)cc(O)ncc1F c1(C(=O)NCC23CC2CN(C(C2CCC(O)CC2)=O)C3)cccc2nsnc12 c1(C=O)ccnnc1.c1(CC(N)=O)occc1C(=O)N.C1CCC1.C(C)(C)C CP1(=O)CCN(CCC(=O)NC2CCOCC2NC(C2CC2C(F)F)=O)CC1 C1(CCCC=O)CCCC(=O)N1.C(CC(C)C)NC(C1(COC)COC1)=O.N C(C(CC(C)(C)C)NC(c1cccnc1Br)=O)OC c1(CC)ccccc1C(N1CCC(O)(C)C1)=O.c1(C=O)ccoc1.C(=O)C.N c1(C(N2CC(O)CCC(NC(=O)C(F)C3CCC3)C2)=O)n[nH]c2ccc(F)cc12 Cc1cc([N+](=O)[O-])ccc1C(N1CCC2CN(Cc3cnc(C4CC4)s3)CC12)=O C(C(=O)NC(CC)C(N)=O)(C(C)OC)NC(C(CC)C)=O Cn1cc([N+](=O)[O-])c(C(N2CCC(NC(=O)CCC[N+](=O)[O-])C(F)C2)=O)n1 C1(COC)CN(C(=O)CCc2cnoc2)C1.c1(C=O)ccn(C2CCC2)n1.C N1(C(=O)CN2CCOCC2)CCC2(CCN(C(C3COCC4(CCC4)O3)=O)C2)C1 Cc1cc(C(=O)NC2C3CC2N(C(c2cc(=N)[nH]c(Cl)n2)=O)C3C)c(F)cc1Cl C(=O)(CC1=CCOCC1)N1CC(C)CC(CNC(c2nnc(C)s2)=O)C1 c1(C(=O)NC2CN(C(C(CO)N(C)C)=O)CC2O)cc2ncc(Br)cc2o1 CC1CN(C(C2CCC23CCC3)=O)CCN1C(=O)CC12CC(C1)C2 Cc1ccc2nc(C3CCCN(C(C4CC(C)OC4C)=O)C3)[nH]c2c1 c1(NC(c2n(C(CC)(C)C)nnn2)c2ncsc2Br)cc(Cl)c2c(c1)OCCO2 c1(NC(=O)CNC(c2ccc(Cl)cc2)CCO)ccc([N+](=O)[O-])cc1 Cc1ccc(OCCC(=O)NCC2CCN2C(C2(O)CCOC2)=O)cc1 c1(C(N2CC(N3CCN(C)CC3)C2)=O)c(Cl)ccc2cc(CO)cnc12 c1cc2n(n1)CCN(C(C1(C(F)F)CCCO1)=O)C2.CC(CC(N)=O)C(=O)NC CC1CN(C(=O)C=CC2CC2)CC1NC(C1(CC2CC2)CCC1)=O c1(SC)ccc(C(=O)NCC(C)N(C)C(c2[nH]ccc2-c2ccccc2)=O)cc1 c1(N(C)C)n[nH]c(=NC(=O)C(=O)N2CCC3(CC2)CN(C(=O)C(F)(F)F)C3)s1 C12(NC(c3c(CCC)n[nH]c3)=O)CCCN(C(=O)C=Cc3cc[nH]n3)CC1C2 C#CCC(O)C(=O)NCc1ccc(C(=O)NC(C)Cc2cccs2)cn1 N1(C(C2C(OC(C)(C)C)C2)=O)CCC(C(=O)N)CC1.N1(CC)CC2CCC1C2 C(=O)(CCS(=O)(=O)COC(F)(F)F)NCC(C)N(C(CCC=C)=O)C c1(C(N2CC(NC(CC(COC)(C)O)=O)C(C)CC2)=O)cccc2c1NCC2 c1(C(=O)NCC(C)N(C(=O)Cc2csc(S)n2)C)ccc(C2CCOCC2)cc1 CC1CNc2c(C(=O)NC3CCC3)cccc2C1.C1(C)(C(=O)N)CS(=O)(=O)C1 c1(C(N2CCN(C3CN(C(C(CC)C)=O)C3)CC2)=O)ccc(OC)c(C(C)C)c1 N1(C(Cn2ncc(C#N)c2)=O)CC(NC(C2CCCOC2)=O)CC12CCC2 c1(C=O)cnc(C2CC2)nc1.C(C(C)(C)C)N(C(=O)CC)CC.C(C)C.N N1(C(C(C)C2CCCO2)=O)C2CCC1CN(C(c1cc(C3CC3)cs1)=O)CC2 C12(C(=O)NCC(N3CCN(C(CC(C)O)=O)CC3)C)CCC(C1)C2(C)C Cc1cc(C)c(C(N2CCC3(NC(=O)C(C)NC(N)=O)CCCC23)=O)c(N)c1 N1(C(c2c(C)oc(C(C)C)n2)=O)CC2CN(C(=O)CCC3CCCCC3)CC2(C)C1 c1(NC(=O)NC(C)CS(C)=O)c(Br)cnn1C1CC1 S(=O)(=O)(c1ccc(Cl)c2cccnc12)NC1C(=O)N2C(C1)CCCC2 N1(C(C(C(C)C)O)=O)CCN(C(C2CCN(C(N)=O)CC2)=O)C(CS(C)(=O)=O)C1 C1(CCC(=O)NCC2CC(NC(C3(c4ccno4)CC3)=O)C2)CCCCO1 c1(COC)cc(C(=O)NCC2CCCC2NC(c2csc(C)n2)=O)no1 C(=O)(C(CO)C(C)(C)C)NC(CC)(CC)CCNC(=O)CCc1ccccc1Cl N1(C(C(CSC)OC)=O)CCCC(CC(=O)NCCN2CC3CC3C2)C1 C1(C(=O)NCCC2(C(N(C3CCCCCC3)C)=O)CCCC2)CCC(=O)NC1 C(C(C(=O)N1CC(OC)CC(C)C1)C(C)C)NC(c1c(CC)cc[nH]1)=O c1(CC)cccc(F)c1C(=O)N(C)CC1(NC(=O)C(CC)N(C)C)CC1 C1CN(C(c2c[nH]nc2C2CCC2)=O)CC12CC2.N1(CC)CCCC1C(=O)N.C C1(CNC(=O)CN2C(=O)C=CC2=O)CCN(Cc2ccc(Cl)nc2Cl)CC1(F)F c1(CC(N2CCC(CC(=O)N)C2)=O)cc(C(F)(F)F)ccn1.C1CCOC1.CC CC1(C)C(NC(=O)CCCn2ccccc2=O)CCN1C(C1CCS(=O)(=O)C1)=O N1(C(C2CC(SC)C2)=O)CCC(O)CC1C(=O)N(C(C(N)=O)C1CC1)C c1(SC)cccc(C(=O)NCC2CCC(NC(C3(C)CCOCC3)=O)C2)c1Cl CC(C(F)C(=O)N1CC2CN(C(c3cc(F)c(F)cc3F)=O)CC2C1)C(F)(F)F C1(CNC(CCCC)=O)(NC(c2cc(Cl)no2)=O)CC(C(F)(F)F)(OC)C1 N1(C(C(CSC)C)=O)CCN(C(=O)CSc2nnc(-c3ccco3)o2)CC(O)C1 Cc1cccc(C)c1CC(N1CCN(C(C2CCN(C)C2C)=O)CC1C)=O c1(C(=O)OC)nn(C)cc1C(=O)NC(C)CN(C)C(c1cnoc1C)=O N1(C(c2cccnc2O)=O)CCOC2CCN(C(C34CCCC3C4(F)F)=O)CC12 C1(CC)(NC(=O)C(C)S(N)(=O)=O)CCN(C(c2c(Br)noc2C)=O)CC1 Cc1nn(CC(=O)N(C)CCOCCC(N2CCC(C(F)F)C2)=O)c(=O)o1 C(=O)(C1=C(Cl)CC1)NC(C)C(C)NC(c1cnccc1N1CCOCC1)=O CCC(C)C(C(=O)NC(c1ncc[nH]1)C)NC(C1C(C)(C)C1(C)C)=O N1(C(=O)Cc2cccc(Cl)c2)CCC2CCN(C(C3CC4C=CC3C4)=O)CC2C1 N1(C(CN2CC(CC)C2)=O)CCC(CCNC(=O)C=CC(C)(C)C)C1 C=CCC(CC(F)F)C(=O)NCC1(C)CN(C(c2cnc(C)nc2)=O)CCO1 C1(CC)CN(C(=O)C=CS(C)(=O)=O)CCC1NC(c1cncc(NC)c1)=O C1(C(N2CCC(CCC)C2)=O)C2CCC(C2)C1NC(=O)C(C)(C)CCOC Cc1ccc(C(=O)C(=O)COC(=O)CSc2n[nH]cc2C(N)=O)cc1 N1(C(C2CC(=O)NCC2)=O)CCC(NC(C2CC3CCC2CC3)=O)C(CO)C1 c1(CC)cc(C(N2CCOCC(NC(C3CC(=O)N(CC)C3)=O)C2)=O)cc(O)n1 C=C1CC2(C1)CC(C(=O)N(CC(O)CN(C(=O)CC1CCCN1C)C)C)C2 C=CCC(CC=C)C(=O)N1C2CCC(C2)C1CNC(=O)C(F)(F)CO C(c1ccc(C)c(C)c1)=CC(=O)NC1(CC=C)CN(C(c2nccn2C)=O)C1 C1(C(N(C)CCc2ccccc2)=O)CC2CC2N1C(c1ccncn1)=O CC1(C)C(NC(c2n[nH]cc2Cl)=O)CC1N=c1nc(C2CC2)[nH]s1 N1(C(c2c(COC)scc2)=O)CCOCC1.c1(CC(=O)NC)c(C)noc1Cl.C N1(C(c2c(CC)cccc2)=O)CC2CCC(CNC(=O)CCc3cn[nH]c3)C2C1 N1(C(C2(C)CCN(C)C2=O)=O)CCC(C)(C)C(C)C1.C1(C=O)(CCF)CCC1.N c1(C(=O)NC2C(NC(C(C)OCC#C)=O)CC2)noc2c1COCC2 c1(C(N(CCN2CCN(C(C(CC)OC)=O)CC2)C)=O)cc2cccn2c(O)n1 C1(C(=O)NCC=C=C)CC(F)(F)CN1C(c1[nH]nnc1CC)=O c1(C(=O)NC(CCNC(CCN(C(C)=O)C)=O)C(C)C)ncc2cc(Cl)ccn12 C1CCCC1.CCS(=O)(=O)NCC=O.C1(C=O)(C(=O)N(C)C(C)C)CC1 c1(C(=O)NC2CCC(NC(c3c(C)cc(SC)s3)=O)C2)cc(N)c(Cl)cn1 c1(C(=O)NC(CC(C)NC(C=C(CC)C)=O)C)cccc2cccc(O)c12 c1(-c2cccc(OC)c2O)cc(C(=O)Nc2sccc2C#N)cc2c[nH]nc12 S(=O)(=O)(c1cccc(C#N)c1)NCCCOCC.CC(C(C)C)N1CCCC1.N C(=O)(C1CCc2ccccc21)NC(CCOC)CNC(c1cc(Cl)c(Cl)n1C)=O N1(C(C2COCC(C)(C)O2)=O)CCC2(CC1)CC(NC(=O)CN1CCOCC1)C2 N1(C(c2cccc(OC(F)F)c2)C(=O)NCCCOC)CCC(O)C(F)(F)CC1 C=C(C)CCCC(=O)N1CCN(C(C2(CCC)CC2)=O)CC1C1CC1 c12c(-c3ccccc3)csc1CCOC2=O.Cc1ccc(C(C2CCCC2)=O)s1 N1(C(CCN(C(CCC#C)=O)CCCO)=O)CCC(F)(CF)C1 Cn1c([N+](=O)[O-])cnc1CN1CC2COC(=O)C2C1 c1(C(=O)NCC(CCOC)NC(=O)CCn2c(C)ccc2C)ccnn(C)c1=O n1(CC)nc(C(N2CCCN(C(C3CCCCO3)=O)CC2C)=O)c2ccccc12 N#CCCCC(=O)NC1CCCN(C(=O)CC2(O)CCCCC2)C1 CC1CN(C(=O)C2=CCCS2)CC(C)C1NC(c1cncc(-n2cccc2)c1)=O Cc1cccc(C(c2cccc(Br)c2)NCC2C3COCC23)c1 c1(CCNC(c2c(CNC(CCCSC)=O)ocn2)=O)cc(O)ncn1 c1(C(=O)OC)nccc2c1CCN(N1CC(CN3CCN(C)CC3)C3(CC3)C1)C2 c1(NC2(C(N(CCNC(COCCC)=O)CC)=O)CC2)ccccc1 C(=O)(C(CC#CC)NC(=O)COC(C)C)NC(CC=C)C c1(NC(C23CC(CNC(C4CCCCN4O)=O)(C2)C3)=O)cccc(F)c1O c1(CC(N2CC(CCC)C2)=O)cccc(Cl)c1F.c1(SC)ccc(C(=O)N)cc1 c1(C(=O)NCCC2CCCN(C(c3c(C)noc3C)=O)C2)cccc(=O)n1O c1(C(N2C(C(C)NC(=O)C(C)(C)n3ccnn3)CCC2)=O)cc(Cl)nn1C C(CC(C(=O)N1CC(CC(=O)NC(c2ncccc2C)C)(OC)C1)OC)OC c1ccc(S(C)(=O)=O)cc1.C1(N(C(C=CCC)=O)C)CCCCC1.C(=O)(C)N c1(C=O)nn(C)c(Cl)c1C(F)(F)F.C12CC(C1)C2.CC1CC1C(=O)N C1(NC(CCOC)=O)CN(C(c2cnc(-c3cnn(C)c3)s2)=O)CCC1C c1(CNS(CC)(=O)=O)cn(CCCC(=O)N)nn1.C1CCCC1C(F)(F)F.C c1(C(=O)NC2CCN(C(C(C3CCC3)OC)=O)C2)cncc(N)c1 c1(OCCC)ccnc(NCC(C)(C)NC(c2cn(C3CC3)nc2C)=O)n1 N1(C(=O)CC2(N(C)C)CCC2)CCOC(C(=O)NC(c2cnnn2C)C)C1 C1(C(N(CC(CC)NC(=O)CCN2CCCC2=O)C)=O)CC12CC(O)C2 C(=O)(C(F)(F)CC1CCN(C)CC1)OC.C12(CCOC1)C(=O)N2.c1ccccc1 N1(C(C2C(C(N)=O)C2)=O)CC2(CCC(C)O2)C1.C1(C=O)CC2C=CC1CC2.N C1(c2nc(C(C3CC3)OC)nn2C2CCC(F)(F)CC2)CCn2ccnc2C1 C#CC1(NC(C2CCC2NC(=O)C(C)(C)CCOC)=O)CCCOC1 CCC(CC(C)C)C(=O)NCC1(CO)CCCN(C(=O)CS(=O)(=O)CCO)C1 C1(CN(C(C(C)n2cccc2)=O)C)CCN(C(=O)Cn2ccnn2)CC1 CC(C)(F)CCC(=O)NCCC1(NC(C2CCCC2(F)F)=O)CCC1 N1(C(c2ccn(CC)n2)=O)CC(NC(=O)CCc2cocn2)CC(F)(F)C1 C=CCC(CC(F)F)NC(=O)CC(C1CC1)NC(=O)C=Cc1cccnc1 N1(C(c2cnn[nH]2)=O)CCC(O)(CCNC(C2(C(F)F)CCOCC2)=O)C1 CN(CCCC(=O)NCC1CC1C)N=O.C1(CC=O)CCCC(C(F)(F)F)C1 C1(C(=O)NC(CNC(C2CCC(=C)CC2)=O)CCCC)COc2ccccc2C1 c1(COC)nc(NCC2CC3CCC3C2)cc(=NC2COC3(CCCC3)C2)[nH]1 CC1OCCC12CN(C(=O)N=c1nc(C3CCCN3)[nH]n1C)CCO2 C(CC(=O)N1CC2(C1)CC2(F)F)(CC(C)C)NC(c1c(OC)cccc1)=O C(=O)(CC(COC)CO)NCCCN(C(C1CCN(CC)C1)=O)C1CC1 C1(CC(=O)NCCCOCC=C)CCN(C(c2cnc(S)nc2)=O)C1(C)C C1(CNC(C(=O)N(C)C)=O)CN(C(C23CCC(C2)C3(C)C)=O)CC1(F)F c1(C(N(CC(=O)NCC(C)(C)n2ccnc2)C)=O)cnn2ccccc12 C1(C(=O)NC2(CNC(C(C)CO)=O)CCCC2)C(F)(F)C12CC2 C1(C(N(CCOC)CCNC(c2cccnn2)=O)=O)CC12CC(O)C2 C1(NC(COC)=O)CC2CC(NC(c3cccc(-n4ccnc4)c3)=O)CC12 CCC(C(=O)N1CSCC1C(=O)NC(C)(CC)CC)OC Cc1[nH]nc2ncc(NC(C3CCCN(C(=O)CC4CC4)CC3)=O)cc12 N1(C(CCC#C)=O)CC2CCN(C(c3cnn(CC)c3C(F)(F)F)=O)CCC2C1 C1(N(C(N(CCCO)CC#C)=O)C)CCC2(CC1)CC2(F)F N1(Cc2scc(C(=O)OC)n2)CC2CC2C1C#N.c12cc(cc(Br)c1)NC2=O N1(C(C(SC)SC)=O)CCC2CCN(C(c3cc(C4(C)CC4)n[nH]3)=O)CC12 c1(OC)cccc(CC(=O)NCC2(NC(=O)Cc3cnoc3)CCOC2)n1 C(C)(CC(=O)NCC1CCN1C(c1cnn(C)n1)=O)OC C1(c2c(F)cccc2)CCCCCN1N1CCOCC1Cc1ccco1 CCCCC(C)CCC(=O)NCCCNC(C1CCc2c(ncn2C)C1)=O N1(C(CCCCCC=C)=O)CC2COCC(C1)C2NC(=O)C(C)c1cc[nH]n1 Cc1ccnc(C)c1C(N1CC2(C)CC1(C(=O)N(C)Cc1ccncc1F)C2)=O c1(C(C)NC(CC2N(C(c3c(C)nc(C)o3)=O)CCC2)=O)cccc(C#N)c1 c1(C(=O)NC2CC(NC(CC3CC(C)(C)C3)=O)C2)nc(C(F)(F)F)ccc1F N1(C(C(C)C(C)(F)F)=O)CCC(NC(C2CCS(=O)(=O)N2)=O)C2(CCC2)C1 c1(C(C)OC)nc(C)c(C(=O)N)s1.c1(C(N2CCC2)=O)cccc(N(C)C)n1 C1(C(C)C)CN(C(C2(C)CCCS2)=O)CCCN1C(c1cc2cccnc2s1)=O C1(NC(C2(SC)CC2)=O)CCC(C)CC1.C(=O)C(N1CCCC1)C1CC1.C C1(OCC)(CNC(=O)C)CCN(C(C2(O)CCOC2)=O)C1.c1ccccc1 C1(C(=O)OC)N(C(c2ccc(NS(=O)(=O)C(C)C)cc2)=O)CCCC1(C)C C1(C(=O)NCC2(NC(c3coc4c3COC4)=O)CCC2)CCc2ccccc2C1 N1(C(C(C)CC2CCCCC2)=O)CC2(CCN2C(C2CCC(F)(F)CC2)=O)C1 N1(C(CC2(OC)CC2)=O)CCC2(CC1)CN(C(=O)C(c1ccc(F)cc1)(C)F)C2 Cc1cc(Cl)c(C(=O)NCCCNC(=O)C(C(C)C)N2CCC(C)CC2)cc1F c1(C=O)cn(C(C)C)nc1C.n1(CC)cc(C(=O)NC(C)C2CC2)nn1.N CC1=C(C(=O)N(CCCCCNC(C2C(C)(C)C2(F)F)=O)C)CC1 C1(C=O)CC2(C1)CC1(CC1)C2.Cc1cc(Cl)ccc1C(=O)NC1COCCC1.N C(=O)(CN=S(C)(C)=O)NCCCC(c1ccccc1)NC(c1onc(C)n1)=O N1(C(C(CC)NC(C)=O)=O)CCC(CC)(NC(=O)C(C)Cc2cnco2)CC1 C1(C)(C(=O)NCC(C(C)(C)C)NC(c2csc(CO)n2)=O)CC2CCC1O2 C1(C(=O)NC(CC(CC)C)C)CCC(C)CN1C(=O)CN(C)CCOC N1(CC(=O)NC2C(CNC(C(C)OCCCC)=O)C2)CCC(C)CC1 Cc1c(C(=O)NC)cc(C(C)C)n1C.C1(C=O)CC2CCC2C1.C1(CC)CC1 N1(C(c2c(C)oc(C)c2C)=O)CCC(C)C(NC(=O)C2=CCCOCC2)C1C S(=O)(=O)(CC(=O)NC1CCCC(NC(=O)CC2CC2)C1)NC c1(C=O)cc(N(C)C)ccc1C.c1(OC)ccccc1CCNC(=O)C(C)O.N c1(OC)ccc(Cl)c(C(N2CCC(C)(NC(C3COCCOC3)=O)C2)=O)c1F c1(OC)ccc(C(=O)NCC2CC(OC)C23CCC3)c(OC)c1C CC(C(=O)N1CC(NC(=O)CNC(=O)C(F)(F)F)CC(F)C1)C(C)(F)F c1(-n2cc(C(N(C(c3c(C)n(C(C)C)nc3)=O)C)C)nn2)ccc(F)c(Cl)c1F N1(C(CC(c2c(C)cccc2)C)=O)CCC12CN(C(=O)C(F)C1CCC1)C2 N12CCC3CN(CCC13)C2=O.c1(OC(C)=O)ccc2c(cnn2C)c1 CCCCS(=O)(=O)CC(=O)NC1CC1C.c1(C=O)cn(CCO)c(=O)nc1O.N C=CC(C)(C)CC(=O)NCC1CN(C(c2cccc(C(C)=O)c2)=O)CCN1C C1(C(=O)NC2CCOC2)(COC)CCN(C(=O)Cc2c[nH]c(C=O)c2)CC1 Cc1cccc2c1C(NC(=O)NC1CCCN(Cc3ccccc3)C1)C(=O)N2 CS(=O)(=O)c1cccnc1N1CC2(CCN(C(=O)CCCCc3cnn[nH]3)C2)C1 CC1CCCC(C(N2CCOCC2CN(C(=O)C(O)C2CCCC2)C)=O)CC1 C1(NC(C(n2c(C)ccn2)C)=O)C2CC1N(C(=O)CC(C)n1ccnc1)C2 CCC(CC(=O)NCC1CC(C(N2CC(CO)OC(C)C2)=O)C1)CC(C)C Cn1ncc2c(O)c(C(=O)NCCNC(C3CC4(CCOC4)C3)=O)cnc12 N1(C(C)=O)CCCC(C(=O)NC(CNC(=O)CS(N)(=O)=O)C2CC2)C1 N1(C(C2C(C)OCCC2)=O)CC2CC(C(=O)NOCC(C)(C)C)(C2)C1 c1(OC)cc(C(N2CCC(O)C(C(N3CCC(O)C3)=O)C2)=O)ccc1I CC1(C)CCC(C(=O)NC2CC2C(F)(F)F)(NC(=O)CCP(C)(C)=O)C1 N1(C(C2CC(C#C)(O)C2)=O)CCC(NC(=O)CCc2nc(C)cs2)CC1C C1(C(N2CCC(CC=C)(C(=O)NCCCC(=O)N(C)C)C2)=O)C2CCCCCC12 c1(CC)cccc(C(N2CC(F)CC2C)=O)c1F.C1(CC(=O)N)CC(C)=NO1 N1(C(CC)C(=O)NC)CCN(Cc2ccccc2)CCC1(C)C C1(NC(C2CCCN2c2ccncn2)=O)CCN(C(=O)C=Cc2ncc[nH]2)CC1 CC(C)CCCCCNC(=O)C(CC1CC1)NC(=O)C(C)OCC1CC1 N1(C(Cn2c(C)cc(=O)cc2)=O)CCC2CN(C(=O)C(F)n3ccnc3)C2C1 c1(C(N2C3CCC2CN(C(C2(O)CCSCC2)=O)C3)=O)cc2cc(Cl)ccc2[nH]1 Cc1cc(C(C)NC(=O)CCNc2ccccn2)cc(Br)c1 c1(OC)ccc2[nH]c(=NCC3(CCO)CC3)[nH]c(=NC(C)C(C)CO)c2c1 c1(OC)ccc(F)c(C(N2CCCC(C(N3CCC(C(C)O)C3)=O)CC2)=O)c1 c1(C(N2CC(N(C(C(c3c(C)n[nH]c3C)C)=O)C)C2)=O)cc(N(C)C)ccc1F CC1(C)C(O)C2CCN(C(=O)CCCn3cc(-c4ccccc4)nn3)C12 c1(C(=O)OC)ccc(C(F)(F)F)nc1N.C1CN(C(=O)COC(F)F)CCO1 C#CCC(O)C(=O)NC(CNC(c1ncoc1-c1cnn(C)c1)=O)CC=C C1(C(=O)NCCN(C(C)C)CC)N(C(=O)CCCCC#N)CC12CCCC2 Cc1ccc(C(N2CC(C(=O)NC3COCC3N(C)C)C(C)C2)=O)nc1O Cc1ccc(C2(C(=O)NCC(C(C)C)NC(c3ncccc3C)=O)CC2)cn1 C1(C(N2CCC(NC(c3ccc(C(N)=O)s3)=O)(C)C2)=O)CC2C=CCC(C1)C2 N1(C(c2cnc(C)[nH]2)=O)CC2(CCC2)CC1CNC(c1cccnc1CO)=O c1(N(C(=O)CCOCC(F)F)C)cccnn1.C1(C2CC2)CCCN1C(N)=O CCC(Cc1cccc(C)c1)C(=O)N(C)CCOCC.C(=O)CS(C)(=O)=O.N c1(CCC(=O)NCC(CNC(C=C(C)Cl)=O)(C)C)ccc2ccccc2c1O N1(C(C(N2C(=O)CCC2=O)C)=O)CCC(CCNc2ncc(C(F)F)cn2)CC1 n1(CC)cnc2c(NCC(C)CO)[nH]c(=NC(CCO)c3ccco3)nc12 C1(NC(=O)Cn2cnnc2)CCC2CN(C(c3cc(F)c(Cl)cc3F)=O)CC2C1 c1(C(c2n(C(C)(C)C)nnn2)NC2CCOC2)csc2cccc(F)c12 N1(C(CC2(C(=O)OCC)CC2)=O)CCCC(C)C1.C(=O)CCCCN(C)C.N CC1CN(C(=O)C2=CCC(NC(C3CCCC3)=O)C2)CCN1C1CC1 c1(NC)c(C(=O)N(CCC(C)NC(C2CCN2C)=O)C)cccc1N N1(C(c2c(CC)nc(C)nc2)=O)CCC2CCN(C(C3CC(C)(CC)C3)=O)C2C1 CC1CCN(C(=O)C=Cc2ccncn2)C1C(=O)NCCc1cnccn1 c1(CCC)nnc(S)n1CC(N1CCC(OCC)C1)=O.C1(=CC=O)CCCC1 CC(O)C(C(=O)NOCCN(C)C)NC(=O)CC1COCCO1 CCCCC(O)C(C)C(=O)N1CCC(C2CCCCN2C(=O)CCSCCC)C1 C(CCCCCNC(=O)C1=CSCS1)NC(=O)CCOC1CCC1 CC1(C)CCOC1C(=O)NCC(=O)NC1CC(O)C(O)C1 c1(CC)ccc(CNC(=O)CCN(C(=O)C(O)C2CC2)CCO)s1 c1(C(N2C(C(C)NC(C(CC)n3cccn3)=O)CCC2)=O)cccc(C(N)=O)n1 CC(C)C(C(=O)NCC1(O)CNC1)n1cccc1 C(=O)(C#CC1CCOCC1)N1CCC(CC(=O)NC(C)CSC(F)F)CC1 N1(C(c2ccc(CSCC)cc2)=O)CCC(NC(c2nccs2)=O)CC1C C=C(C)C(C)(C)C(=O)NC1CCC1.c1(CC(=O)N)c(C)nn(C(C)C)c1C C1(NC(C(c2ccn(C)n2)C)=O)C2CC3C(C2)C13C(=O)N.C1CCC(C)C1 c1(SCC)cncc(C(=O)NC2CC(CCNC(c3c[nH]nc3F)=O)C2)n1 C1(C(=O)O)CCCCC1.C1(CC#C)CCC1.C(=O)CNC.C(=O)(C1CC1)N N1(C(C(OCC)OC)=O)CC2(CC(C(=O)NCCOC(F)(F)F)CO2)C1 C1(C(=O)OCC)CC2(CCC(NC(c3cc(C)n(C)c3C)C)CC2)C1 Cc1cnn(C)c1C(=O)NCC(C)(C1CC1)NC(=O)CCc1ccc(Cl)s1 C#Cc1cn(C)nc1C(=O)NC1CCCC(CNC(c2ccc(N)cc2F)=O)C1 N(C(=NCCC(C)N1CCCCC1)NCC1CCOC1)CC(CC=C)(C)C c1(NC(C(=O)NC2CN(C)C(=O)C2)=O)cncc2c1CCCC2 CCCCC(CNC(=O)CC1CCCN1C)NC(=O)C(F)CN(CC)CC N1(C(C2CN(C(c3c(CC)non3)=O)CC2F)=O)Cc2ccc(C)cc2C1 C(CN=C(NCCC1CCCCO1)NC1CCCC1)SC(C)(C)C c1(N(CCC#N)C(CN2C(C)C(C)(C)CCC2)=O)cccc2ncccc12 N1(C(COCC)=O)CCCCCCC1C(=O)N(CC)CC1CCCO1 CC1=C(C(=O)NC2CC(CNC(C3CCC(C)C(C)C3)=O)C2)CCC1 N1(C(C2CCC(C(C)C)CC2)=O)CCN(C(c2ccnc(Cl)c2O)=O)C(CF)C1 N1(C(COCCSC)=O)CC(C(=O)NC(C)CC(C)C(F)F)C2(CCC2)C1 N1(C(CCn2c(C)ncc2)=O)CC2CC2C1C(=O)NOCCOC(C)C C1CN(C(c2cc(C)cc(Cl)c2)=O)C2CCCC12.C1(C(=O)OC)CC1C(=O)N C(C(C)(C)C(=O)NC1CC(O)C(O)C1)N(C)C(c1ccnnc1O)=O n1(CC)[nH]c(C)nc1=NC(=O)N1CCC(c2ncccc2C(F)(F)F)CC1 c1(C(=O)NCC2N(C(C(C=C=C)C)=O)CCCCC2)cccc2c1COCC2 C=CCCCCCCCC(=O)NCCCNC(=O)C(C)(C)CC(C)C C(=O)(C#CC1CCCCO1)N1CC2C(NC(c3c(C)oc(C#N)c3)=O)C2C1 c1(C(=O)NC2CN(C(c3c(C)[nH]nc3Br)=O)CC2C)cc(=O)n(C)cn1 N1(C(C(C)(C)C2CCCCC2)=O)CCC2CCCC(C1)N2C(c1cnsc1)=O Cc1nc2cccnn2c1C(=O)NC1CCSC12CN(C(=O)C)C2.CCN(C)C.O Cc1nc2ccc(C(=O)NC3CN(C(=O)CCCCC(C)C)CCC3O)cn2n1 Nc1nc(Cl)ccc1C(=O)NCCOCCNC(c1ccon1)=O O=C(Nn1ccnn1)C(O)CNC(=O)C(O)C1CCC1 C(=O)(C1SCc2cccnc21)NC1(CCOC)CCN(C(=O)CCCCC#N)C1 Cc1nc(O)c2c(n1)CCN(C(C1CC(c3cccc(Cl)c3)(O)C1)=O)CC2 S(=O)(=O)(c1c[nH]ccc1=NCCCN1CCC(CO)CC1)NC1C(C2C(C)C2)C1 c1(N2CCC(O)(COC)C2)ncnc2c1ncn2C1CC(CCO)C1 C(=O)(CC(C)CCC)NCC(C(=O)N(C)CC1CC(=C)C1)CN(C)C c1(-n2cc(CNC(c3c(C)ccc(C)c3)=O)nn2)ccc([N+](=O)[O-])cc1F C1(CC)CN(C(=O)C(C(C)C)SC)CCN1C(=O)Cc1cscc1Br CC1CCOCC1C(=O)NC12CC1CN(C(C1CCC(C(N)=O)N1C)=O)C2 O=S(=O)(c1ccc(NCC(C2CCC2)C2CCC2)cc1Cl)NC1CCOCC1F c1(C(=O)NCCOC2CN(C(C3(C)C=CCC3)=O)C2)ccc(C(F)F)cc1F N1(C(CC2(C#N)CCOCC2)=O)CC2CC(NC(=O)CSCCNC=O)CC1C2 N1(C(C2CC(OC)C2)=O)CCC2(C)CCCC12.C(=O)(CCCc1ncc(C)o1)N Cc1[nH]nc(CO)c1C(=O)NC1C=CC(C(=O)NC(CO)C2(C)CC2)C1 N1(C(CCC#C)=O)CC(C)(C)CC1CC(=O)Nc1cccc(CC)c1C Cc1cc(=NC(=O)c2ccc3ncc(-c4cnc(F)c(F)c4)n3c2)[nH]c(Cl)n1 N1(C(C(C2CN(C(=O)CC3CCCC4CC34)C2)O)=O)CCC12CCCSC2 C1(O)(CNC(CCNC(COC)=O)=O)CCCN(C(c2cncn2C)=O)C1 C(=O)(CC(C)(C)C(F)F)NCC12N(C(c3c(F)ccc(C)c3)=O)CCC1CC2 N1(C(C)=O)CCCCC1C(N1CC2CC1(CNC(C13CC1C3)=O)C2)=O CCCC(C)CCCC(=O)N1CC(NC(c2cc(C(N)=O)[nH]n2)=O)CC2(CC2)C1 Cc1ncncc1C(N1CC(O)(CN(C)C(C2CC2Cl)=O)C1)=O N1(CCc2cn(CC(C)NC(C3CC(C)(O)C3)=O)nn2)CCC(C)(C)CC1 N1(C(C(CC)(C)O)=O)CCCC(CO)(NC(=O)C(O)Cc2ccccc2)C1 C1(C(=O)N)CC(C)(C)CCN1C(=O)Cn1c(O)nnc1O.C1(CC=C)CCOC1 c1(CC)cc(F)ccc1C(=O)NC1COCCC1.C1(CC=O)CCCC(=O)N1.N C(=O)(CCCCC(C)C)N1CCC(CC=C)(NC(=O)CN2CCCC2C)C1 CC1CCc2nc(C(=O)NCC(C3CCC3)NC(C3(C)CCCC3)=O)cn2C1 N1(C(c2c(C)cc(Br)cc2)=O)C(C)CC2CN(C(=O)CC3CCC(=O)N3)CC12 N#Cc1c(F)cccc1S(=O)(=O)N(CCO)Cc1ccoc1 C1(COC(=O)C(c2ccc(F)c(Cl)c2F)O)CCC2(CC1)OCCO2 c1(C(C(=O)NCCCSC)N(C2CC2)Cc2cn(C)nn2)sccc1Cl C1(CC(N2C(CN(C)C)CCC2)=O)CCC1(C)C.N1(C(C(=O)N)C)CCCCC1 c1(C(=O)NC(C)CCCNC(C2(F)CC2)=O)ccc(-c2ccccc2Cl)nc1O C1(O)(C(N2CCCC2C2(O)CN(C(C3(N4CCCC4)CC3)=O)C2)=O)CCCCC1 CCC(C)(CNC(=O)Cc1ccc(O)cn1)C(=O)NC(C)Cc1ccco1 C1CN(C(=O)C)CC(F)(F)C1.c1(CC)ccccc1.C(C)(C(=O)N)OCC=C C1(NC(c2c[nH]c(Br)c2)=O)CN(C(C2C3CCCOC23)=O)CCC1F C1(NC(c2csc(C)c2N)=O)CCN(C(c2cn(CC(N)=O)nn2)=O)CC1(C)C N1(C(C2CC2)=O)CC2CCC1C1CN(C(C3CC(C)OC3C)=O)CC21.CCOC CC1(C)CN(CC2CC3(CCNC3)C(=O)O2)Cc2c(Br)cccc21 C(C)(C(O)C(=O)NC1(CNC(c2ccc(SC(F)F)cc2)=O)CC1)OC N1(C(CC=CC)=O)CC2CCN(C(=O)CN(CCCCCC)C)CC12 Cc1ccc(C(O)CNC(C2CC(O)C2)=O)c(C)c1 C(CC1=CCN(C(=O)C(C)(C)C(F)F)CC1)NC(c1nc(CCC)sc1)=O c1(NC(C(CC=CC)NC(=O)CSCC(N)=O)=O)ccc(OC)c(C)c1 N1(C(=O)NCC2CCS(=O)(=O)N2)CCc2sc(Cl)cc2C1 CCC(C)C(CNC(=O)C(CC(F)F)N(C)C(c1ncccc1F)=O)CO CCS(=O)(=O)c1cccc(CNC(=NCCCF)NCC2CCC(=O)NC2C)c1 Cc1nnc(COCCOC(C2(c3ccc(C)s3)CC2)=O)o1 C1(NC(c2ccc(F)s2)=O)CN(C(C2C=CCC2)=O)CCC1F Cc1c(CC(N2CCC(CCNC(c3ccco3)=O)CC2)=O)sc2ccccc12 c1(NC2(c3n(CCOC)nnn3)CCN(C)C2)ccc(C)cc1C c1(C(=O)NC(CNC(CC(CC)C2CC2)=O)(C)CC)cc(O)ncn1.C(C)C.O CCC(C)(C)C(=O)C(=O)NC1(CO)CN(C(C23CCCC(C)(C2)OC3)=O)C1 N1(C(c2c(C)cno2)=O)CC(C2CCCN(C(C3CC(O)CN3C(N)=O)=O)C2)C1 C1(C)(C(=O)NC2C(C(=O)NCC(COC)C)CCOC2)C(C)(C)C1(C)C S(=O)(=O)(c1c[nH]ccc1=NCCN1CCC(C)C1)N1CC(C)N(C(C)=O)C(C)C1 c1(C(N(CC(CC)NC(c2nn[nH]c2C2CC2)=O)CC)=O)ccc2c[nH]nc2c1 C=C(C)CCCC(=O)NC(C)C(C(C)C)NC(C1CN(CC(C)C)C1)=O Cc1nc(=N)[nH]cc1C(=O)NC1CC2(C1)CC(NC(C1CCC1CF)=O)C2 N(C1CCCc2nc(C)sc21)CCc1cc(-c2ccc(OC)cc2)c(OC)cc1 N1(C(c2n(C(C)C)ccn2)=O)CC2CC(NC(C3CCCOC3C)=O)C2C1 N1(C(c2ccc(SC)o2)=O)C(CNC(=O)CC)CC2CC12.c1ccc(F)cc1 Cc1cc(N)c(C(N2CCCC2CCNC(C2(C)CCC(=O)N2)=O)=O)cc1C C1(N(c2c(C)cccc2)C(C2CCc3nc[nH]c3C2)=O)CCCC12CCNCC2 O=C1CCCc2sc(NC(C3CCC(NC(C4CC5C=CC4C5)=O)CC3)=O)nc21 N#Cc1ccnc(N2CC3CC3(C(=O)N(CC(O)CO)C(C)C)C2)n1 c1(OC)ncc(F)c(N2CC(C)(CC(=O)NCCc3ccc(C)c(C)c3)C2)n1 CCCC(C1CCCC1)NC(=O)CN(C(=O)C(C)SCC)CCOC c1(C(N2CC(O)(CN(C(CCC(C)N(C)C)=O)C)C2)=O)cccc([N+](=O)[O-])c1Cl Cc1nnc2n1CCC(C(=O)NCC1CN(C(=O)CCCC3CC3)C1)C2 N1(C(C)=O)CCCN(C(C2(C)C=CCN2C(=O)C=Cc2ccsc2)=O)CC1 C1(NC(C(C(CC)C)O)=O)C2CC3CN(C(=O)C=CC4CCCCCC4)C1C3C2 CC1CCN(C(=O)CCCCN(C)C)CC1N(C(=O)C(C)C1CC1)C C1(CNC(CN(C(C)C)CC)=O)CC(C)C1.C(=O)CNC1CC1 c1(NC(CC(C)O)=O)ccc(C(N2CCN3CCC2CC3)=O)cc1[N+](=O)[O-] C1(NC(CNC(=O)NC)=O)CCOC(C)C1.C(c1cc(C)no1)=CC=O C12(NC(C=C(CC)CC)=O)CC3CCC(C1C2)N3C(=O)CCCc1ncc(C)o1 c1(C(=O)NCCC2CN(C(CCCOC)=O)CC(C)O2)cnc2[nH]c(C)nc2c1 c1(OC)ccc2c(c1)cc(C(=O)NC1CC3CC1C(O)C3O)n2C CC(C)C(O)C(C)(C)C(=O)NC1CC(CC(N2CC(O)C(C)(C)C2)=O)C1 CC#CCC(C(=O)NC1CC(O)C1O)NC(=O)C=CCN1CCCC1 C1(C(N2CC(N(C(=O)CSc3nncs3)C)C2)=O)CCN(c2ccccc2)C1 c1(CN(C2CC3CCCCCC23)C=O)nc2ncc(C(=O)O)cn2n1 c1(OC)cc(C)cc(C(N2CC(C)N(C(c3cnccc3C)=O)CC2C)=O)c1N C(CCC1CC1)(C(=O)NC(C1CCOCC1)(C)C)NC(C(C1CCCCC1)C)=O N1(C(CC(=O)OC)=O)CCN(C(=O)CC2CCC3(CC2)CC3)C(C(C)C)C1 Cn1ncc2c(NC(=O)CNC(=O)C(c3ccc(F)cc3F)(F)F)ncnc12 CN1CCC(CC(=O)NCC2CC2(F)F)C1=O.C1(C)(C=O)CNC(=O)N1.C C1(CN(C)C(C2CC(CF)C2)=O)CCCN1C(=O)CCc1ncc[nH]1 C(C)(CC(=O)NCC1(CNC(=O)C(O)Cc2ccccc2)CC1)OC N1(C(c2cccc(CNC(=O)Cc3ccco3)c2)=O)CCCCCC1CCO N1(C(CC2(C=C)CC2)=O)CCC2(CCCN2C(=O)C=Cc2ccc(OC)cn2)C1 Cc1ccc(C(C)(C)C(=O)NCC2(C)CC23CCC3)cc1.C(=O)C1=NOCC1 c1(C(N2CC(NC(CCC#CC)=O)C(C)CC2)=O)cc2cccc(Cl)c2[nH]1 CCC(CC)C(C)C(=O)NCCCN(C(=O)Cc1cc(C)nn1C)CCO Cc1c(CC(N2CCCC2CC(=O)NCCCc2cn[nH]c2)=O)cnn1C C1CCCC(F)(F)C1.c1(C(=O)NCC2CC(C(=O)N)C2)ccccc1CCO C(C)(CN=c1ccc([N+](=O)[O-])c(O)[nH]1)C1CC1.C1(OC)CN(C)C(C)(C=O)C1.N C1(C(=O)NC2(C(=O)OC)CCC2)CCC(C(=O)NC2CC2)CC1 C1CC(OC)C(=O)N1.C1(C)(C(=O)OC)CCN(C)C1.C12(CC1)CC(=O)N2 c1(SC)n[nH]c(NC(=O)CN2CCN(C(c3cccc(C)c3Br)=O)CC2)c1C#N c1(SC)nc(N2CCC(C)C2CNC(=O)CCN2CCOCC2)cc(C)n1 C1(NC(c2cc(C(C)=O)[nH]n2)=O)COCCN(C(=O)CC2(C)CCOCC2)C1 c1(OCC(=O)N(CCn2cc(CCC(C)=O)nn2)C)cc(F)cc(Cl)c1 N1(C(C(=O)NCC)C)C(=O)CCC1=O.C(C)(C=O)SCCCC.C1CC1.N C(=O)(CCCN=[N+]=[N-])N1CCC(C)(C(=O)NC(CO)CCO)C1 Cc1cc(CN2CCCC(O)(C(N3CCC(F)CC3)=O)C2)cc(F)c1F C(CC(=O)NC(CNC(C1CC(C(F)(F)F)C1)=O)C1CCC1)=CC=C c1(CCC(=O)NCC(CNC(c2c(CC)nns2)=O)(C)C)ccc(F)cc1 C1(CC(=O)N(C2CC2)C)CC(C)(C)OC1=O.N1(C(CCOC)=O)CCCCC1 c1(OC)c[nH]c(C(=O)NC2CCN(C(=O)Cc3nn(C)cc3Cl)C(C)C2)cc1=O C1(C=O)CC2CC1CC2(F)F.N1(C(C2(C(=O)NC)CC2)=O)CCC(C)CC1.C C1(C(N2C(C)CC2CO)=O)CCN(C(=O)C(C2CC2)N(C)C)O1 N1(C(c2c(C)snc2)=O)CCC(NC(c2c(C(F)(F)F)cc[nH]c2=N)=O)C(C)C1 C1(C(=O)NC2CN(CC)C(=O)C2)CCN(C(=O)CCn2cc(C)cn2)C1(C)C N1(C(C)=O)CCCC(NC(c2ccc(C(=O)Nc3[nH]ccc3C)cc2)=O)C1 c1(C(=O)NCC(CC)NC(c2c[nH]nc2-n2cnnn2)=O)cc2cccn2cn1 c1(OC)ccc(F)c(C(=O)NC2CN(C(C3CCC4(CC4)C3)=O)CCC2C)c1 c1(CNC(C(CC=CC)NC(c2cncnc2)=O)=O)cc(C)c(C)nn1 CCCC(CC(=O)NCc1ccnc(F)c1F)NC(=O)Cc1cc(C)[nH]n1 C12(C(=O)NC(C)CCNC(c3ncc(Cl)s3)=O)CCC(C(F)F)(CC1)CC2 c1(C(=O)NC(c2ccc(Cl)c(Cl)c2)C)cc2nc(Cl)ccc2s1 C(N(O)C(=O)C(C)C#N)c1cn(C(C(=O)OC(C)C)C)nn1 CCCC(C)CC(=O)NCCN(C)C(c1ccccn1)=O S(=O)(=O)(c1cccnc1NCCCCCSC)NCC(C1CCCC1)OC c1(C(N2CC(N(C)Cc3cc(Br)cc(I)c3)C2)=O)cc(Cl)cnc1Br C(C)(CNC(=O)C(Cn1cncn1)NC(=O)CCC1CCC1)(CO)OC CCCCS(=O)(=O)NCC(=O)NC1CN(C(c2cnc(C)s2)=O)CC1C C1(CC(N2CCCC(CN(C)C(c3cc(O)n(C)n3)=O)C2)=O)CN2CCC1CC2 c1(NC(c2nnnn2C2CCCC2)(COC)C)cccc(C(C)SC)c1 c1(C(=O)N)ccc2c(c1)CCCS2.CC(C)CCNC(C1(n2cccn2)CC1)=O CC(C)C(O)C(C)C(=O)NC1CCN(C(=O)COC2CCCC2)CC1(C)C c1(C(N2CCC(N(C(c3c(C)csc3)=O)C)C(C)C2)=O)ccc2c(c1O)CCC2 C(=O)(CCS(=O)(=O)C(F)(F)F)NC(C)CC1CN(C(c2sccc2C#N)=O)C1 C1(CC(=O)NCCC)CC2C=CC1CC2.c1(CC(=O)N)ccc(C(F)F)cc1 S(=O)(=O)(CC(=O)N1CCCCC1CCN(C)C(c1c(C)ncn1O)=O)NCC c1(NCc2ccc(C)cc2)ccc(Cl)cc1C(=O)NC(=O)C(C)CO Nc1c(F)cc(C(=O)NCC2(CNC(C3C4CCCOC34)=O)CC2)cc1F c1(-c2cc(C(=O)N)n[nH]2)cccc(Cl)c1.C1(C(C)NC(CNC=O)=O)CCCC1 N1(C(c2c(NC)cncc2)=O)CC2CCCC1CN(C(=O)CCCCC1CC1)C2 C(c1cc(F)c(F)c(F)c1)=CC(N1CCC(N(C(CC=C)=O)C)C1)=O C(CCCCCNC(C1(C)CCOCC1)=O)NC(c1c(CC)[nH]cc1)=O c1(C(N2CC(NC(C(CCC)O)=O)C(OC)C2)=O)cc(Cl)c2ccccc2c1O CCC(CC)(CCNC(C1(C)COC(=O)OC1)=O)NC(c1cccc(OC)c1)=O c1(C(=O)NC(C(C)C)CNC(C2(CO)CCCO2)=O)ccc(F)cc1Cl c1(CC)c(C(N2CCC(N(C(=O)C(Br)=C(C)C)CCO)CC2)=O)cnn1C c1(C(CC)=O)ccc(C(N2CCCC2CN(C)C(c2cocn2)=O)=O)cc1 C1(C=O)CC2CCC1N2C(C1CCC1)=O.C1(SCC)(C)CC1.C1CC1.N c1(OC)ccnc(C(=O)N(CC(O)CN(C)C(c2cnn[nH]2)=O)C)c1 c1(OCCOC)cc(C(N2CC3C(NC(C4CCC4)=O)C3C2)=O)ccn1.C N1(CC(=O)N(CC(C)CNC(=O)CC2CCN(C)C2)C)C(=O)CNC1=O N1(C(C(CC(C)C)=O)=O)CCCC(C2(NC(=O)CC3CCCC(=O)N3)CC2)C1 C1(C(N2CC(C)(COC)C2)=O)CCC=CC1NC(=O)CO.C1CCCO1 CCCC(O)CC(=O)N1CCOCC1CN(C(=O)CCSCc1ccccn1)C c1(C(N2CCC(N(C(C3CCN(C)C3=O)=O)C)C2)=O)cc2sccc2n1C C(CC(C)C)(CC(C)C)(c1nnnn1C1CCOCC1)NCCn1c(C)ncc1 C(=O)(C(CC)C(C)(F)F)NC1(CC=C)CCN(C(c2ccncn2)=O)C1 c1(OC)ccn2ccnc2c1C(=O)NC(C)CCC.c1(C(=O)N)nc(C)n(C)n1 c1(N(C)Cc2nccn2-c2ccccc2)cccc([SH](=O)=O)n1.C12CC(C1)C2.N c1(C(N2CCCC(N(C(C=CCOC)=O)C)CC2)=O)c(N)cc(Cl)cc1F Cc1cc(C(=O)NCCC(O)CNC(=O)C2=CCOC2)n(-c2ccccc2)n1 C(C1CCCN1C(c1cnn[nH]1)=O)=CC(=O)NC1CCCCCC1 CC1CCC(NC(c2cccc(Cl)c2)=O)CN1C(c1cc(O)n(C)n1)=O O=C(C1=CC2(CCOCC2)C1)NC1CCCCCN(C(=O)CCOCC(F)F)C1 C1(C)(CNC(c2c(C)ccs2)=O)CCC(NC(=O)CCN2CCCC2)C1 N(C(=NCCCF)NCC(C)(C)C)CCOCC.c1(C)cn(C2COC2)nn1 c1(NC(=O)CC2CSCCO2)ccccc1-n1cc(-c2ncoc2C2CC2)nn1 C1(N(C(C)=O)Cc2ccnn2C)CCCC(NC(=O)CCc2ccc(O)nn2)C1 N1(C(C(CC2CC2)OC)=O)CCC(NC(=O)C(=Cc2cccnc2)C)C12CC2 c1(C(=O)NCC(C2CCC2)NC(=O)Cc2cnc[nH]2)csnc1C1CC1 c1(C[SH](=O)=O)ccccc1.C(=O)(C(C)(C)C)N1CC(N(C)C(=O)CO)C1.N Cc1cc(C(N2CC(NC(=O)CCCF)CC2CO)=O)c(C)n1-c1cnccn1 N1(C(CCN(C(c2c(CC)ocn2)=O)C)=O)CCC(O)C1(C)C CC(C)C(C)(C)CNC(C1CCCOC1c1ncc[nH]1)=O Cc1nn(C(C)C)c(C)c1CC(=O)NCCn1cc(C(F)F)cn1 C1(NC(c2c(CCNC(CCCOC(C)=O)=O)n[nH]c2)=O)CC2CCCCCC12 c1(C(N2CC(CNC(C3SCCS3)=O)OCCC2)=O)cc2ccccc2o1 c1(OC)ccc(C)c(C(N2CC(O)(C3CCCN3C(=O)C(OC)OC)C2)=O)c1 CC1(NC(c2occc2CNC(=O)C(c2ccccc2)F)=O)CCCC1O N1(C(C2N(CC)CC2)=O)CCN(C(=O)CCCc2ccc(O)c(F)c2)CC(O)C1 c1(C(N2CCC(NC(c3c(OCC)ccs3)=O)C2)=O)cc(C(C)C)ccc1C N1(C(CC2C=CC(NC(CC(=O)N)=O)C2)=O)CC2(C1)NC(=O)NC2=O.C1CC1 C12(NC(CC(C=C)(C)O)=O)CCC(CC1)N(C(C1CC(=O)N(C)C1)=O)C2 C1(NC(CNC(C(CC)C)=O)=O)CN(C(c2cccc(NC)n2)=O)CC1OC Cc1c(F)ccc(C(=O)NC(CNC(C2CC2)=O)C(C)C)c1O.N(C)C.C C=CCC(C(=O)NCc1nc(CNC(=O)C(C)CC)cs1)C(C)(C)C Cc1ccc(C=CC(=O)NCC2CCN2C(c2csc(=N)[nH]2)=O)cn1 c1(SCC)ncc(F)c(OC)n1.C12(CCCOC1)c1cn(nn1)C(C)C(=O)N2 C1(COC)(CNC(=O)CCC2CCOCC2)CCN(C(C2CC=CCC2)=O)C1 C1(NC(C(CC)(C)C)=O)CC2CC1N(C(c1ccc(OC)c(OC(F)F)c1)=O)C2 CCCCCC(C(=O)N1CCC(O)(CNC(c2csc(O)n2)=O)C1)C(C)C N(C1c2ccccc2CC1NC(=O)C(O)C1CC1)C(C1(C)C=CCCC1)=O CCC(C)CC(C(=O)N(CC(C)(C)C#N)C)NC(c1coc2ccccc12)=O N1(C(c2cnnn2C)=O)CC2CC(C(=O)O)C(C2)C1.C(=O)(C(=O)N)N(C)C N1(C(CC=C)=O)CC2CC(NC(=O)Cc3cccc(OC)c3Cl)C(C2)C1 C1(NC(C(N(C)C(c2cc(CCO)on2)=O)C2CC2)=O)CCC(C(N)=O)CC1 C1(C(N(C2CCCC2)CC(=O)OC)=O)CCC1(C)C.c1(C=O)ccccn1.N c1(C(=O)NCC#CCNC(=O)COc2ccsn2)cc(Cl)cc(Cl)c1F C1(CNC(c2c(COC)ncs2)=O)CN(C(C2C(C)C2C)=O)CCN1C CC1(C)CC1(Cl)C(=O)NC1CCC1CNC(=O)Cn1ccnn1 N1(C(C2(C)CC(O)CN2C(c2cccnc2O)=O)=O)CCCC2(CC1)CC2 c1(C=O)cc(F)c(F)cc1F.C(=O)CCN(C(=O)C(F)=CC1CC1)C C1(CNC(C=CCCC)=O)CN(C(=O)C(C)OCC)CCC1(F)F C(C1CCN(C(=O)C(C)OCC2CC2)CC1)=CC(=O)NCCC=C C1(C(N2CCC(O)(CNC(=O)CN3CCOCC3)C2)=O)(OC)CCCSC1 Cc1nc(Br)sc1C(c1nnnn1C1(C)CC1)NCCC1(C)CC1(F)F COn1cnc(C)c1C(=O)NCC(O)CNC(=O)C(c1ccc(F)cc1F)C N1(C(C(CC#C)(C)C)=O)CC2CC(C1)N(C(c1cnc3[nH]ncc3c1)=O)C2 c1(C(=O)N)cc2n(n1)CCCC2.c1(OC)ncc(C(N2CC3C(C)C3C2)=O)cn1 CC1(C)CCCC(O)(C(=O)NCC2CCN(C(C3CCCC3O)=O)C2)C1 CC1CCc2ncc(C(=O)NCCN(C)C(c3cc4sccc4s3)=O)n2C1 c1(C(C)(C)C)ccc(C(N2CC(NC(c3coc(Cl)n3)=O)C(O)C2)=O)cn1 C1(CC(=O)NC2C(CCOC)C2)CCN(C(C2C=C(C)CS2)=O)CC1 c1(C(N(c2ncc(OC)cn2)C2CCNCC2)=O)cnc2c(F)c(F)ccc2c1 Cc1ccncc1CC(=O)NCc1c[nH]nc1C(=O)NCC(O)C(C)O N1(C(CCC(=O)N(CCC)CC)=O)CC2(CCC2)C1.C1(=CC=O)CCOCC1 N1(C(C2(COC)CCC2)=O)C2CCC(C2)C1C(=O)NCc1ccccc1 C(=O)(C1=COCC1)NCC1C(CNC(Cn2c(C)cnc2)=O)C1 C=CCC(C)(C)C(=O)N1CC2CC2(NC(=O)C=Cc2cccnc2)C1 c1(C(N2CCN(C3CCCN(C)C3)CC2)C(=O)NCCC)cc(C)nn1C C1(C(=O)NC(c2ccccc2F)CC)CC2CC2N1C(c1nn(C)cc1Br)=O C12(OC)CCC(C(N3CC4CC4C3)=O)(CC1)C2.c1(C(NC)=O)csc(S)n1.C N1(C(C2N(CC)CC2)=O)CC(NC(C2CCS(=O)CC2)=O)CC(C)(C)C1 C(C(O)C(F)(F)F)N(C(CN(C(C1(CC#C)CCC1)=O)C(C)C)=O)C C(=O)(C(C(C)C1CCCCC1)N(C)Cc1ccc(OC)cc1)NC(C(=O)OC)C C(=O)(C(Cn1cccn1)NC(=O)Cc1cnoc1)NCCC(C)c1cn[nH]c1 c1(C(=O)OCc2cccc(F)c2OC(F)F)c[nH]c2ccc(Br)cc12 C1(CCCNC(CCCOCC)=O)CN(C(c2ccnn2CCOC)=O)CCO1 C1(OCCOC)CCCN(C(=O)C(C)CNC(=O)C(C)(C)N2CCCC2)C1 Cc1nncc(C(N2CCCC(CN(C(=O)COC3CCCC3)C)C2)=O)c1C c12ccnc(c1)CNC2=O.N1(CC)CC2C(C1)N2C(c1cc(C)ccn1)=O c1(OCC(C)C)ncc(-c2nnc(N3CC4CC3C(=O)O4)n2CC2CC2)cc1Cl c1(C(N2CCC(C(=O)NCC3(OC)CCCC3)C23CC3)=O)ccc2nccn2c1 N1(C(C2(C(N)=O)CC2)=O)CCC2(C1)CN(C(=O)C=Cc1cc[nH]n1)CCO2 N1(C(CCC=C)=O)CCC(C)C1CNC(c1ncc(F)cn1)=O C(=O)(CCS(=O)(=O)Cc1cccs1)NC1CC(CNC(C(C(C)O)C)=O)C1 Fc1ncc(Cl)c(CNC(C2CCCCO2)C2CC2)c1Cl C(c1nc2ccccc2o1)=CC(N1CC(C)(NC(C2CCC3CCC2O3)=O)C1)=O N1(C=O)CC2CCCC1C2c1cn(C2CC(=O)N(c3cn[nH]c3)C2)nn1 N1(C(CC)=O)CCN(C(=O)COC2CCN(C(=O)CCC=CC(C)C)C2)CC1 C1(CCC)(NC(=O)C(C)(C)NC(=O)C(O)C2CC2)CCNC1=O c1(C(=O)NC(CC)CNC(=O)C(c2cncn2C)=O)cnc(F)c(C)c1 C(CCCCC(=O)N1CCCC(N(CCO)C(c2ccc(C)nn2)=O)C1)OC Cc1ccc2c(c1)CC(C(N1CC(NC(=O)C#CC3CCCCO3)CC1C)=O)S2 N1(C(C2C(C)SCCC2)=O)CCC(O)(CNC(c2ncnc(O)c2Cl)=O)CC1 C1(O)CCN(C(c2ccnc(-n3ccnc3)c2)=O)C1.CC1(C)CC1CC(=O)NC C(=O)(CCCC(N)=O)N1CC=CCC1.Cc1cc(NC(=O)C2CC2)sc1C=O.N c1(OC)ccc(C(=O)N(C2CN(C(=O)CCC3(O)CCC3)C2)C)c(N)c1F C(=O)(C1=Cc2ccccc2C1)N1CC(C(=O)NC(CCCC)C)C(OC)C1 C1(C(=O)NC(Cc2cncs2)CO)C2CCCC12 c1(C(C(=O)NCC2CCCO2)N(CCOC)C)cc(C(F)(F)F)ccc1C c1(C(C(C)NC(=O)NCCC(C(C)C)C)O)c(F)cccc1F C(=O)(CCCCC(F)F)N1C(C2(NC(CCCCN(C)C)=O)CC2)CCC1 CC1(C)C(CC(=O)NC2CCC(NC(=O)C=CCF)C2)C1(C)C C=C1CC(C(=O)OC(COC)CC)N(C(COC(C)(C)C)COC)C1 N1(C(CS(=O)(=O)N)=O)CC2=C(C1)CN(C(c1cc(C)cc(F)c1)=O)C2.CC C(CCCCC(=O)N1CC(O)CCC1C(=O)NCC(O)CCO)SC C1(NC(=O)CNc2ccccc2Cl)CN2CCC1CC2 C1(NC(C(C=CC)O)=O)CN(C(c2ccn(-c3ccncc3)n2)=O)CC1N=[N+]=[N-] N1(CC)CCCC(C(=O)N(CC(C)(C)NC(c2ccccn2)=O)C)C1.C(C)=O C(=O)(CCC(=O)NC(Cc1ccoc1)C(=O)NC(c1ncc(C)cn1)C)NC C1(C(=O)NCC(CCCC)NC(=O)CN2CCSCC2)NC(=O)OC1(C)C N1(C(C2CCCC(C)C2)=O)CCC(C2(NC(c3cnc4n3CCS4)=O)CC2)CC1 N1(C(c2scc(COC)c2)=O)CCCCC1C.c1(C(C=O)C)ccc(C)cc1.N CC(C)(O)C#CC(=O)NC1CC(CNC(C2CCCO2)=O)C1 c1(C(=O)OC(C)(C)C)cc(NC(c2cc(-c3cn(C)nn3)on2)=O)ncc1F c1(C(=O)NCCNC(=O)CSC(F)F)cccc2[nH]ccc12 c1cnc(C)c(C(=O)O)c1.C1(C(=O)N)(SC)CN(C(=O)CCc2ccsc2)C1 N1(C(C(C)(C)C)=O)CC23CCCC2(C1)CN(C(c1cnc2c(c1)CCCC2)=O)C3 N1(C(C(C)NC(CC)=O)=O)CC2CCC(N(C(=O)CC(CC)C(C)C)C)C2C1 c1(C(N2C(CN(C(=O)C(C)(C)C#N)C)CCC2)=O)cnnc(-c2ccccc2)c1 C1(CC(NOCC(CC)C)=O)CC2(C1)CN(C(C1CCC(=O)CC1C)=O)C2 N1(C(CN(C)CC)=O)CC2CCCC2(NC(=O)CC2(CC(=O)OC)CC2)C1 C1(C(N(C2CCN(C(=O)CCC(C)SC)CC2)CC)=O)CC(OC)C(OC)C1 C1(C(=O)NC(Cc2ccco2)CO)CCN(C(=O)CN2CCCCC2=O)O1 CCCCCC(O)CC(=O)N(CC(C)O)CCNC(=O)Cc1ccco1 N1(CC)CC(C(N2CCN(C(=O)CSc3cccc(F)c3)CC2)=O)CC1=O CCC(CC)CCNC(=O)C(=Cc1ccccn1)C.C(=O)CCN(C)C(C)=O.N c1(OC)ccc(C(N2CC(N(C)C(c3cnc(Cl)cc3OC)=O)C2)=O)c(C)c1 C12(NC(c3c(Cl)cn(CC)n3)=O)CCC(C1)N(C(c1c(O)ccnc1F)=O)C2 Cc1ccc2[nH]cc(CCN(C(c3ccccc3)=O)CC3CCCC3CF)c2c1 C(=O)(C1=CC2(CCOC2)C1)N(C)CC1CN(C(c2cnncc2O)=O)C1 c1(OC)ccc(S(N)(=O)=O)c(C(=O)N(C)C(c2ncccc2Cl)C)c1 C(=O)(C1=NOC2(CCOC2)C1)NCC(CO)NC(CCCN(C(C)C)C)=O C=C1Cn2c(C(N3CCN(C(c4cc(OC)cnn4)=O)C(C)C3)=O)nnc2S1 c1(C=O)cnc2c(c1)CCC2.c1(NCC)ccc(C(=O)NCC2CC2)cc1 c1(C(N(C2CC3CC2CN3)Cc2ccc(C)c(Cl)c2)=O)cn2ncccc2n1 C1(NC(Cn2ccc(C)n2)=O)CC2CN(C(=O)CC3(C)CC3(F)Cl)CC12 N1(C(CC(CC)C(C)C)=O)CC2(C=C(C(=O)N3CCC3CO)CO2)C1 CCS(=O)c1ccccc1C(=O)NC1CC(F)(CNC(=O)C2=COCCO2)C1 c1(CC(=O)N)ccc(C#N)cc1.c1(-c2cn(CC(C)OC)nn2)ccc(F)cc1Cl C=CCC(C)N=c1[nH]c(N2CCCC(OC3CCC3)C2)nc2cc(OC)ccc12 CC1(C)CN(C(C2CCC2CNC(=O)COCC2CCC2)=O)CCS1 C(C(C)(CNC(C1CCCN(c2cnccn2)C1)=O)C(=O)O)OC C1(S(N)(=O)=O)(C(=O)OCc2cc(OC)c(Cl)cc2)CCCC1 Cc1cc(C(=O)NC2CC(CNC(=O)CN3CCC(O)CC3)C2)ccc1F C(=O)(C1CCc2cc(Cl)ccc21)NCCCC(C)NC(c1c(C)c(O)ccc1)=O c1(C(N2C(C(=O)NC3CCCN(C)C3)CC(O)C2)=O)ccnc(F)c1F c1(C(N(CCCN(C)C(c2ccc(Cl)nc2N)=O)C)=O)cc([N+](=O)[O-])nn1C N1(C(c2cncc(OCC)c2)=O)CCC(O)C(NC(=O)C(C)n2cncn2)C1 c1(C(=O)OCC)c[nH]c(C)cc1=NCC(C)NC(=O)C(C)c1cccs1 O=C(C1=NN(C2CC2)C(=O)CC1)NC1CC1C.C1(O)(C(=O)N)CCCCC1 CCCCC(CNC(=O)C=CCNC(c1ccn(C2CC2)n1)=O)CC C1(C(N2CCC(CCCNC(C(C)CC(F)F)=O)CC2)=O)CC(C)(C)OC1(C)C c1(OC)cc(C(N2CC(NC(c3ccnnc3)=O)CCC2C)=O)cc(N)c1OC N1(C(c2nc(C)sc2C)=O)CCN(C(=O)C2=CC(C)C2)C(C2CC2)C1 CCCCC(O)CC(=O)NC1CC(=O)N(C2CN(C(c3ns[nH]c3=O)=O)C2)C1 c1c(Cl)c[nH]c2nccc1-2.Cc1[nH]nc(O)c1CCNC(C1CCCC1NC)=O Cc1cc(C(=O)NCC2COCC2)c(O)nn1.c1(C=O)ccc(C(C)(C)C)s1 C(c1sccc1C)=CC(=O)NC(CCCNC(c1c(SC)ccs1)=O)C c1(CC)cccc(C(N2CCC(C)C(NC(=O)CC34CCC(CC3)C4)C2)=O)c1N CCCCC(F)C(=O)N1CCCCC1CC(N1CCC(CC(N)=O)C1)=O C1(C)(C(N(C(CNC(c2c(C)nc(CC)s2)=O)C)C)=O)CCN(C)C1=O C1(NC(C2(OC)CCOC2)=O)CCCCN(C(=O)C(=Cc2cccc(F)c2)F)C1 c1(C(=O)NCC2OCCC(NC(=O)C3=COCCC3)C2)ccccc1[N+](=O)[O-] Cc1ccc(C(N2CCC(c3cc(CNC(=O)C(C)O)on3)CC2)=O)c(O)n1 c1(C(N2CCC(C)(NC(=O)COC(F)F)C2)=O)csc2c1CCCC2 Cc1[nH]c2ncccc2c1C(=O)NCCCCNC(=O)Cc1cnns1 Cc1nonc1CC(=O)NC(c1ccnn1C)C(=O)NCc1ncnn1C(C)C C12(NC(c3ccc(Cl)nc3Cl)=O)CCCC1N(C(C1CCC1)=O)CCC2 c1(CC(=O)OC)cc(C(=O)NCC)cs1.CC(C)C.C(=O)CC.C(C)C C1(CNC(COCCOC)=O)CCCC2CN(C(=O)CCC3OCCO3)CC12 c1(C(=O)NCC(C)(C)NC(C(CCC)F)=O)nnc(O)nc1O CCC(N=c1ccnc(C2CCCC2)[nH]1)c1cccnc1 c1(C(C)C)ccc(CNC(c2cc(-c3cnn(CCF)c3)ccn2)=O)cc1 CC1=NS(=O)(=O)NC=C1C(=O)NC1CCOC(C)C1.c1(C(=O)N)csc(Cl)n1 C1(NC(c2ncn3c2COCC3)=O)CCCC12CN(C(C1CCCCC1O)=O)C2 C1(CNC(Cc2cccc(OC)c2)=O)CC2CCC1N2C(c1cc(C)[nH]n1)=O C1(CC)CN(C(=O)Cc2cnn(C(F)F)c2)CCC1NC(=O)C#CC1CC1.C c1(OC)ccc([N+](=O)[O-])c(N2CCOC(CNC(=O)CC3CCC4CC34)C2)c1F C1(C(=O)NC2CC(NC(c3sc(F)cc3Br)=O)C2)CCCCC1F C(CN=c1[nH]c(=NCCN2CCCC2)[nH]c2c1CC(C)CC2)N(S(CC)(=O)=O)C N1(C(C2(NC(C(OCC)OCC)=O)CCOC2)=O)CCCC(C#N)C1 C1(C(N2CCN(CCCNC)CC2)=O)COCCN(c2ccc(C(=O)O)nn2)C1 c1(C(N2CCC(NC(c3cc(C(N)=O)[nH]c3)=O)C2)=O)cc(F)c(F)c(F)c1F C=CCC(CNC(C1CC(CF)C1)=O)C(=O)NC(CO)C(C)C Cc1c(C(N2CCCC(NC(=O)Cc3nc(=N)[nH][nH]3)C2C)=O)cncc1Br C(=O)(CCCC(F)(F)F)N1C(C(=O)N(C(CF)CF)C)CCC(C)C1 N1(C(C)C)CCC(C2CCN(C(c3cc(=O)c4ccccc4[nH]3)=O)CC2)C1 c1(CNC2C(C3(C)CC3)(C)C2)ccc([N+](=O)[O-])cc1[N+](=O)[O-] C1(C(=O)NCC(C)NC(=O)Cc2cocn2)CN(C)CCN(C)C1 C(=O)(C1=CCCCCC1)N1C(C(N2CC(F)(CC)C2)=O)C2CCC1C2 c1(C(N2CCC3(CN(C(=O)C4=CCSC4)C3)C2)=O)cnn2ccc(O)nc12 c1(C(=O)NC(CN(C(CCC(=C)Cl)=O)C)CC)cc(F)ccc1CC FC1(F)C2CCC(N=c3[nH]ccn4c(Br)cnc34)CCC12.C(C)OCC1CC1 c1(C(=O)NCCc2c(CNC(=O)C=CBr)nco2)ccc2c(c1)C(=O)NC2 N1(C(c2c(C)nccc2)=O)CCCC(F)(CNC(=O)CC2(C)CCOCC2)C1 N1(C(C(C2CCOCC2)C)=O)CCC(CC(N2CCNC(=O)C2)=O)C(O)C1 C1(C(=O)NC(C2CCCN2C(=O)CCOC2COC2)C)CC(Cl)(Cl)C1 C(CN=c1nc(N2CCC(N3CCC3)C2)c2c([nH]1)CCCC2)c1cc(=N)[nH]cc1 Cc1ccc(N2CCOC2=O)cc1NC(N1CCCNC(=O)C1)=O CC(C)CN=C(NCC1CCCC1(C)C)NCC1(C#N)CC1 Nc1ccc(C(=O)Nc2nc(CC(N)=O)cs2)cc1C(F)(F)F Cc1ccc(-c2nc(C)c(-c3nc(C4CCC(C(C)(C)C)CC4)no3)s2)cc1 N1(C(Cc2c(CC)n[nH]c2CC)=O)CCOCC(CNC(=O)CO)C1 Cc1occc(=O)c1OCC(N1CCC(CC(N2CCCC2)=O)CC1)=O C1(C)(C(=O)NCCC(C)(C)NC(=O)Cc2nc[nH]n2)CCCCNC1=O c1(CNCCCn2c(C)ncc2)cc(Cl)c(Br)cc1F C12(CNC(CCC)=O)CCC1CCN2C(=O)Cc1cccc(F)c1F CCC(C(=O)NC1CC(C)(NC(c2ccns2)=O)C1)N(C)C C1CCN(C(c2cn(C3CC3)cn2)=O)CC1.N1(CC(=O)N(C)C)CCC(O)CC1 N1(C(C(c2ccco2)NC(C(C=C)OC)=O)=O)Cc2n[nH]cc2C1CO CC1CCC(C(=O)NCc2nnn(C)n2)N(C(C2CC(C)(C)C2)=O)C1 Cc1ccc(C(N2CCN(C(=O)C(C)N(C)C)CC(O)C2)=O)c2ccccc12 c1(C=O)cccc(C(=O)N(C)C)c1.N1(C(CSCC(C)C)=O)CCC1C.N c1(N(C)C)ncnc(N2CC3CN(C(=O)CC4CC5(CC5)C4)CC3C2)c1[N+](=O)[O-] C(=O)(CC1=CCOCC1)NCC(CC)N(C(=O)COc1ccon1)C C12(C(=O)NC(C)CNC(=O)CC3CCCO3)CCCCC(=O)N1CCC2 N1(C(=O)Cc2cnccn2)CC2CCC(C1)N2C(=O)CC1C=CCC1 c1(C2(NC(=O)NCC3CCCN3CCCO)CCCC2)ccc(F)cc1Cl C(=O)(CCC(=O)C(C)(C)C)N1C2CC(NC(Cn3ccc(C)n3)=O)CC1CC2 C(CC(CNC(c1cc(Br)co1)=O)NC(C1COCCO1)=O)OC C1(CC(=O)N(C(C(=O)NCCOCCC=C)C)C)CC2(CC2)C1 c1(CNC(Cc2c(OCc3ccc(C)cc3)cccc2)=O)cnc2n1CCC2 c1(C(=O)NC2C3(CC(NC(C(c4scc(C)n4)C)=O)C3)C2)cnn2ccncc12 Cc1c(F)ccc(C(=O)NC2CC(NC(C3CC(F)C3)=O)C2)c1Cl Cc1cc(=NCC2CCC(NC(=O)CCCCc3ccccc3)C2)c(C#N)c[nH]1 C1(C)(CC=O)CCN(C(=O)CC2CC(=O)NC2=O)CC1.c1(CC)nnco1.C c1(NC(C2N(c3cc(C)ncn3)C(C)CC2)=O)cnn2cccnc12 c1(CC)cccc(F)c1C(=O)NCC(C)(C)NC(C1CCCNS1(=O)=O)=O C1(CNC(C23N(C(Cc4cc(C)no4)=O)CC(C2)C3)=O)CC(O)C12CCC2 Cc1cc(NC(C2CCCC2(C)C)=O)ccc1NC(=O)CC(C)(C)CN(C)C C1(OC)CC(CNC(=O)CCCc2cccnc2)N(C(C2CCN(C)C2)=O)C1 CC1CCC(CNC(=O)COCCCF)CN1C(=O)CO.C1CCOCC1.C Cc1cnc(C(=O)NC(CNC(C2Cc3nncn3C2)=O)CO)c(F)c1 N1(C(C=CC=CCC)=O)CCC2OCCN(C(c3oc(Br)nc3C)=O)C2C1 CC1CN(C(=O)C(c2ccc(Cl)s2)=O)CCC1NC(C1CC2(CC(=O)N2)C1)=O c1(C(=O)NC2CCCCN(C(c3ccc[nH]3)=O)CC2)ccc2cccc(F)c2n1 c1(C(=O)NC2CC(NC(CCc3ccn(C)n3)=O)C2)cccc(NC=O)c1.C C1(C(N(C23CC(C2)C3)C)=O)CCC(CNC(C2CC(C)(C)C2)=O)O1 CCC(C)C(O)C(C)C(=O)N1CCCCC1C(N1CCCC1(C)CO)=O C(=O)(CC(C)CC(C)C)N1CCOCC(C(=O)NCC2(CC)CCCO2)C1 CS(=O)(=O)CC(=O)NCCOCCCNC(=O)CCCc1cccc(Cl)c1 c1(C(=O)NCCC(C)CO)ccc(F)c(-c2c(COC(C)(C)C)cccc2F)n1 N1(C(C)C)CCC2CCN(N3CCC(C(=O)Nc4ccc(F)cc4)C3)CC12 C1(NC(c2nc(CCC)oc2)=O)CN(C(c2ccnn2CC2CCC2)=O)CC1C C1(C(N2CC(C(C)Nc3cccc(F)c3C#N)OCC2)=O)CC(C(C)(C)C)=NO1 C=CC1(C(=O)NCC(C)N(C)C2CC2)CCN(C(=O)CC(C)(C)N(C)C)CC1 Cc1ccc(O)c(NC(=O)CCc2cc(C)on2)n1 C1(N(CCCC(=O)OC)C(=O)C(C)(C)C)CC2(CNC2)C1 N(C1CC2(CN(C(c3cnn[nH]3)=O)C2)n2ccnc21)C(c1n[nH]c(C)c1C)=O c1(C(N2CC(F)(CNC(c3oc(CC)c(C)c3)=O)C2)=O)c(N)sc(C)c1C C(=O)(C1=NOC(C(C)(C)C)C1)NCCN(C(C(C)(C1CC1)OC)=O)C C1(C(N(CCOCCOC)C)=O)CCN1C(C1(n2nccn2)CC1)=O Cc1cn(C)cc1C(=O)NC1(C)CCC1.c1(CC=O)cccc(C(C)C)c1.N C(C)(CCC(=O)NCC(C)N(C(=O)CC1(O)CCC1)C)OCC c1(C(NC2CCN(C(=O)C(C)Cc3ccncc3)C2)=O)csc(C(C)C)n1.CC c1(C(=O)NCC(C)(C)NC(C(C)OCCCC)=O)ccc(C)nc1O N1(C(C2C(NC(C(CCC)N(C)C)=O)CCO2)=O)C2CCCC1CC2 c1(C(=O)Nc2nccc(I)n2)ccc(Cl)nc1NCc1ccc[nH]1 N1(CC(=O)Nc2c(C(=O)OC)cc(CC)s2)CC(C)(C)c2ccccc21 N1(C(C(C)=NOCC#N)=O)CCN(C)C(C(N2CC(O)(C(F)(F)F)C2)=O)C1 C12(CNC(c3c(N)ccc(OC)c3)=O)CCCC(CN1C(c1ccon1)=O)C2 CCCC(N)C(=O)NCC1(C)CCCO1 CC(C)(C)C(C(=O)NC)NS(C)(=O)=O.c1(CC=O)cnco1.C1CC1 N1(C(CC=C(C)C)=O)CC(NCc2cc(Nc3cccs3)cs2)C(F)C1 c1(C(=O)NCC2N(C(c3cccc(C)c3F)=O)CCCC2)ccc2cnoc2c1 C1(NC(c2n(CC)ncc2Cl)=O)CC(O)CN(C(c2ccnc(S)c2)=O)C1 c1(OC)nscc1C(=O)NCC(O)C(=O)NCC1CCSC1 c1(C(=O)NC(C(C)C)CCNC(C2(C(N)=O)CCC2)=O)cc2nc[nH]c2cc1F C1(NC(c2c(CNC(CS(CC)=O)=O)noc2)=O)CCCCC1(F)F C1(C(=O)NC2(CC=C)CN(C(C3(C#N)CC3)=O)C2)OCCN(C)C1=O c1(OCC)ncc(C(=O)N)cn1.C12CC(C1)C2.C1(CC=O)CCC(=O)C1 Cn1nc(C(N2CCC(CCNC(=O)CCC3CCCOC3)C2)=O)cc1Cl C(=O)(C1=CC2C=CC1C2)N(C1CCN(C(=O)Cn2cccc(N)c2=O)C1)CC C1(CNC(CC=C)=O)CCC2(CCC2)CN1C(=O)CC(C)c1cccnc1 C12(C(=O)NCC3C(C(N4CC(CC)(CO)C4)=O)C3)CCC(OC)C1C2 C1(NC(c2cc(OC)ncc2)=O)CCC2CN(c3ncccn3)CC2C1 C=CCC(C(=O)N1CC2(CCC2)CC1CNC(=O)Cc1cnn(C)c1)C(C)C N1(C(CCc2nnc(C)o2)=O)CCN(C(=O)C(C)c2ccsc2)CC1C(C)C N1(C(=O)NC2(C(F)(F)F)CC2)CCOCC1CC(c1ccccc1)O Cc1nn(CC(=O)NCC(C)NC(C2CCCC2(F)F)=O)c(C)c1C=NO c1(C(=O)NCCN(C(CC(c2cccc(Br)c2)C)=O)C)cnc(S)n1C c1(OC)cc(CNC2CN(C(c3cc(Br)ccc3Cl)=O)CC2C)cc(O)c1 c1(C(=O)NC2CN(C(C3(C)CCN(C(C)=O)C3)=O)C(C)C2)cnc(C)nc1O N1(C(C2CC(=C)C2)=O)CC(NC(=O)C=Cc2cccc(OC)c2)CCC(O)C1 C1(NC(CN(C2CC2)CC)=O)CCC12CN(C(=O)C(c1ccccc1)F)C2 c1(COC)nc(N2CCN(C(=O)CCCc3cc(C)sc3C)CC2C)cc(Cl)n1 CCCC(C)(C)C(=O)N1CC2(C)CC1(C(=O)NCCc1cncc(C)n1)C2 C1(F)(C(=O)NC2C(C#N)CCC2)CCCN(C(=O)C(c2cccnc2)O)C1 CC1(CNC(c2ccc(F)cc2F)=O)CCCN(CC(O)Cc2ccccc2)C1 c1(COC)cccc(NCc2csc(C)c2C)c1C N1(C(c2c(N)c(Cl)ncc2)=O)CCC2(C1)CN(C(C1(O)CC1)=O)CCO2 Cc1cccc2[nH]c(=NC(C)CCNC(C3(O)CCSC3)=O)sc12 N1(C(c2occc2Br)C(=O)NCCCSCC)CCc2c(nn(C)c2C)C1 C12(NC(=O)CCCCN3CCOCC3)COC(C1)C(NC(C1(Br)CC1)=O)C2 Cc1nc(CC(C)C)c(C(=O)NC(C)CNC(c2cscn2)=O)s1 CS(=O)(=NS(=O)(=O)N1CCC(NC(N)=O)C1)c1ccccc1F c1(CCCC(=O)N(C2CN(C(C3(C(C)(C)C)CCCC3)=O)C2)C)ccccc1Cl C1(COC)CCCN1C(=O)C=Cc1cnn(C)c1.C1(C=O)CC2CC2C1.C C1(C(=O)NCCCC)CN(C(=O)C(C(CC)CC)OC)CC12CCC2 CCCCC(C(=O)NC(C)(CNC(=O)COCCF)CC)N1CCCS1(=O)=O Cc1cc(C(=O)NCCCCC2CCN(C(=O)CCC(C)(F)F)CC2)nnc1O CC1=CCSC1C(=O)NCCC1CCN(C(=O)CCC2CCCN2C)C1 CC1=CCN(C(C2COC(CNC(=O)C=Cc3cscn3)C2)=O)CC1 C(=O)(C1CCCc2cccnc21)NC(CC=C)CNC(c1ccco1)=O c1(CC(=O)N(C)C)ccc2occc2c1.C12(C(N3CCCC3)=O)CC(F)(C1)C2 C1(C(=O)NC2CCC(NC(CC(COC)COC)=O)CC2)Cc2ccncc2C1 c1(C(N2CC(CC=C)(NC(=O)Cc3ccoc3)C2)=O)ccc(NC)c(F)c1 N1(C(CSC(C)C)=O)CC2CCCCC2(CNC(c2cn(C)[nH]c2=N)=O)C1 C1(NC(=O)CCC2CCC2)CC2CC(Nc3ccc(SCC(F)F)cn3)C1C2 C(C(C)(C)CNC(=O)CCC1CC1(Cl)Cl)N(C(=O)CO)C.C1CC1.C C(=O)(C1=NOC(C)(C)C1)N(C(CC(F)F)C(=O)NCC1C2CCCC12)C Cc1ccc(CC(C)C(=O)NC2(C)CN(C(=O)CSc3nccn3C)C2)cc1 c1(C(N2CCC(CNC(C(CCCOC)C)=O)C2(C)C)=O)nc[nH]c2nccc1-2 c1(CNC(C(N2CC(C(=O)OC)C(C(F)F)C2)=O)=O)ccn2nnnc2c1 C1(OC)CC(CNC(C2CCCC2)=O)N(C(=O)CCCCc2cnc[nH]2)C1 C1(NC(C=Cc2ccc(C)s2)=O)CN(C(=O)CP(C)(C)=O)Cc2ccnn2C1 C1CC2(C1)CN(C(c1nn[nH]c1C(F)(F)F)=O)C2.C1(C)CCC(C=O)O1.CC C#Cc1ccc(C(=O)N(CC(C)N(C(=O)CCc2ccc(F)nc2)C)C)cc1C Cc1nn(C)c(C(F)(F)F)c1C(N1CCC(C)C1)=O.C1(C=O)CC2(CC2)C1 N1(C(CC2(CC)CCC2)=O)CCN(C(c2cc(F)c[nH]2)=O)CC2CCCCC12 CC1OC2(C(=O)NC3C4CN(C(c5cncc(Cl)c5Cl)=O)CC34)CCC1CC2 C1(NC(C2C(=C)C2C(=O)OC)=O)CCOC(C(=O)N)C1.c1ncc(Cl)cn1 CC1=C(C)CCC1.C(=O)(C=CC(=O)N(C)C)NC(C1(C=O)CC1)C.N c1(C(N2CC(CNC(CNS(NC)(=O)=O)=O)(OC)C2)=O)sc(F)cc1C n1(CCC(=O)NC(CN(C(C(C)SC)=O)C)C)ccc(C)n1 C(C1CCOc2ccc(Br)cc21)NC(=NCCCOCC)NCC(C)(F)F C12(C=O)CCC(CC1)C2.c1(C(C)NC(c2c(OC)csc2)=O)cccc(C)c1 C1(C(N(CC(O)COCc2ccccc2)C)=O)CCC2(CCCN2)CC1 C1(Nc2ccc(N(C)CCn3ccnc3)cc2)CCCCC1c1nc[nH]n1 C1(CNC(c2ccc(SC)s2)=O)CC(NC(=O)C)C1(C)C.CC(C)C.S C(CCCCCC(=O)NC1COCCOC1)NC(c1ccn(C)c1)=O O=C(CCCCCCn1cc(C2CCCC2)nn1)NC(CC1CCOCC1)CO c1(CC)ccc(C=CC(=O)NC)cc1.C(=O)C(C)(C)C(N)=O.C1COCC1 Cc1ccc(C(=O)NC(C)CN(C)C(c2ncncc2F)=O)cc1Br CCCCC(CNC(=O)C(F)(F)c1ccsc1Cl)NC(=O)C(C)C(C)C c1(CCC(=O)NC2(COC)CCCN(C(=O)C(C)S)C2)c(C)nc(O)nc1O N1(C(C(C)(CO)OC)=O)CCCN(C(=O)CCCCc2ccc(Cl)cc2)CC1 CCCCCCCCC(=O)NC1CCCC1(C)NC(C1CCC(C)C1)=O C1(N(C(C2C(C)C2C)=O)CCNC(c2ccc(C(N)=O)o2)=O)CCCCCC1 C1(NC(CC(=O)NCC)=O)CCCC12CCN(C(C1(O)CCCCCC1)=O)C2 c1(NC(c2ccc(C3CCC3)nc2)=O)ccc2c(c1)CC(F)C2 CCC(C#N)C(=O)NC12CC(C(=O)NCCN=S(C)(C)=O)(C1)C2 Cc1cc(F)c(CN2CC(F)(F)CC2C(N2CCn3nccc3C2)=O)cc1Br Nc1cc(C(=O)NC(CC(F)F)C(=O)N2CCC(OCCO)CC2)cc(F)c1 C=CCC(CC(=O)N(C(CO)C1CC1)C)NC(C1CNC(=O)N1)=O N1(C(CCc2scc(C)n2)=O)CCN(C(=O)CC2(CO)CCC2)CCC1C C1(C(N2CC(C3(NC(C(CC)F)=O)CC3)C2)=O)OC(C)(C)OC1(C)C C1(F)(C=O)CCS(=O)(=O)C1.C(c1cncnc1O)=CC(N1C(C)(C)CCC1)=O N1(C(C2(C)CC(O)CN2C(=O)CCNC(=O)CO)=O)CC2CCC(C1)C(=O)N2 CCC(CC(=O)N(CC(=O)Nc1cccc(OC)c1)C)C1CC1 CCCCC(C(=O)NCC1COCC1NC(=O)CCN1CCOCC1)C(C)C CC1CN(C)CC1N=c1cc[nH]cc1S(=O)(=O)NCc1nc(C(C)(C)C)ns1 C1(CCNC(CC=CCNC(CC=C(C)C)=O)=O)CCCN1C N1(C(c2cnc(CC)[nH]2)=O)CC(O)CC1CNC(=O)CN1CCCC1CO Cc1nccn1CCCC(=O)NCCn1cc(C2C3COCC23)nn1 C(CC(=O)N(C)CCn1cc(C)cn1)(C(F)(F)F)NC(C(CC)(C)O)=O c1(C(N2CC=CC(NC(c3c(C)nc(O)cc3)=O)C2)=O)coc2c1CCCC2 N1(C(c2c(Cl)cnc(CC)n2)=O)CC2CCC(C2)C1.C1(C)CCC1.C(=O)(C)N N1(CCC(c2ccccc2)C)CC(C(=O)O)C(c2ccc(Cl)cc2)C1 N1(C(CC2CC(OC)C2)=O)CC2CCC1CN2C(c1cc(F)c(F)cc1OC)=O C1(C(N2CCN(C(c3cc(CC)nn3C)=O)C(CC)C2)=O)CCCCC(F)(F)C1 c1(C(=O)NC2C(C)CN(C(c3cc[nH]n3)=O)CC2C)ccc2c(ccn2C)c1 c1(SC)ccc2oc(=NC3CCC(O)C(N)C3)[nH]c2c1 C(CCN=[N+]=[N-])N(C(C1(N(C(CC=CC)=O)C2CC2)CCC1)=O)C C1(NC(C(C2CN(C(c3ccncc3Cl)=O)C2)OC)=O)CCCC(N(C)C)C1 c1(C(=O)NCC2CCN2C(c2cn(CC(F)F)cn2)=O)ncccc1Cl n1(CC)c(O)nc(NCC(O)CNC(c2ccc(C)nn2)=O)cc1=O c1(C(=O)NC2CCN(C(Cc3nc(C)oc3)=O)CC2CO)coc(S(N)(=O)=O)c1 N1(CC)CCOCC1C(=O)NC1(CC=CC(=O)N)CCC1.c1ccccn1.C C1(NC(CCN(CCCCC)C)=O)CN(C(=O)CC(C)C)CC2(CC2)C1 c1(NC(C2C3CCC(C3)N2C(C2CC2(Cl)Cl)=O)=O)cccn2ccnc12 C1(CNC(Cc2c(C)c(-c3ccccc3)on2)=O)CCC(C)(C)CN1CCNO N1(C(CNS(CCCOC)(=O)=O)=O)CCC(NC(=O)CC)C12CC2.C=O.N C12(C(N3C(CC(=O)NC)CC3)=O)CCC(CN(C(=O)C(C)SC)C1)C2 C1(CNC(C(CC)(C)O)=O)CCN(C(=O)CCc2ccc(SC)cc2)CC1(F)F S(=O)(=O)(c1[nH]c(=NCc2c[nH]ccc2=N)ccc1Br)N1C(C(C)(C)C)CCCC1 C1(C)(C(=O)NCc2c(C)noc2C)CN(C(C2CCOCC2(C)C)=O)CC1C N1(C(C2CC(=C)C2)=O)CCN(C(=O)Cc2n[nH]cc2Br)CC1C(F)F CS(=O)(=O)c1cnc(NC2CC3CC(C2)N(C(=O)COC(F)(F)F)C3)c(Cl)c1 C1(C(=O)NC2CCCN(C(CCC=C)=O)C2)CN2CCC1CC2 C#Cc1cc(C)nc(N2CC(c3nc(-c4ccccn4)no3)CC(C)C2)n1 O(S(=O)(=O)c1ccc(S(=O)(=O)C(C)C)nc1)c1c([N+](=O)[O-])ccc(C)c1 C1(NC(CC2CCN(C)C2=O)=O)CCN(C(C2CC(F)(F)C2)=O)C12CC2 Cn1c(C(N2CC(NC(C3(F)CCC(=O)CC3)=O)CC2(C)C)=O)cc2occc12 C1(CNC(C=COCC)=O)CC(C)CCN1C(C1CCCCC1F)=O CC(O)(CNC(=O)CCOC1CCOCC1)CNC(C1C=CCCC1)=O N#CC1CCN(C(=O)CCC2CCCCN2C(=O)CCn2cccn2)C2(CC2)C1 C1(Cc2cn(CC(C)C)nn2)CCCCN1C(c1cn(-c2ccccc2)cn1)=O C(CC(C)C)(C(=O)NCC#CCNC(c1ccc(C2CC2)o1)=O)OC c1(OC)cccc2c(C(=O)N(CC(C)CNC(=O)C(C)(C(C)C)O)C)cnn12 C1(C(=O)NCc2c(CNC(CCCC)=O)cccc2)CC2C=CC1CCC2 C1(CSC)CC(O)CN1C(=O)C.c1ccc(-n2cnnn2)cc1.C1(C)C(=O)N1 Cc1nn2cnnc2c(C)c1CCC(N1CC(CO)C1(C)C)=O C1(NC(C2(CCNC(=O)COc3ccccn3)CC2)=O)CCC2CC2CC1 C1(NC(C=CCCC)=O)CN(C(c2ccc(CCN(C)C)cc2)=O)CCC1CO c1(CC)cc(C(N2CCN(C(=O)C=CC(C)(C)C)C(CO)C2)=O)cc2c[nH]nc12 CCCC(C)(C)CNC(C1CC12CC(NC(C1(CC)CCCCO1)=O)C2)=O CCC(C)C(C(=O)NCCC(=O)N1CCCC1)NC(=O)CCc1ccco1 Cc1cccc2c(C(=O)NC(C)C)cccc12.c1(C=O)ccc(S(C)(=O)=O)o1.N c1(OCCC(=O)NCC(CC)NC(=O)CC)ccc2c(c1)CCC2.C=O.N C1(C(=O)NC2CC(CC(=O)NCCc3ccncc3)C2)CC2C=CC1C2 c1(C=O)ncccc1O.c1(SC)cscc1C(=O)NCC1CCN(C(=O)C)C1 c1(C=O)cn2c(n1)CN(C(=O)CS(C)(=O)=O)CC2.c1(C(=O)OC)n[nH]cc1.N c1(OCCNC(=O)Cn2ncc3ncccc23)cccc(N(C)C)c1[N+](=O)[O-] C1(C(=O)NCC(C)N(C)C(c2cc(CF)on2)=O)CC12CC(O)C2 C1(CC=C)(C(=O)NCCC2(O)CCCC2)CCCN1C(C1CCCCO1)=O c1(C(N(CCN(C(C2CCN(C(C)C)C2)=O)C(C)C)C)=O)cccc(F)c1N Cc1cc(C(=O)NCC2(NC(c3ccncc3Br)=O)CCCC2)cc(O)n1 C1(C(=O)NC2CN(C(=O)COCc3ccccc3)C2)CCCS1(=O)=O CCC(C)(CO)C(=O)N1CCC(O)C(NC(=O)C(=Cc2ccccc2)OC)C1 Cc1nn(CC(=O)NCC(C)N(C(=O)C(=O)N)C)cn1.C1CC1.C1CC1.C c1(C(N2CCC(F)(C(N(C3CCC3)CC)=O)CC2)=O)cc(F)c(Cl)c(F)c1 CN1CCN(C(=O)Cc2cc[nH]n2)C(CNC(C23CC(F)C2C3)=O)C1 C1(CC#C)(C(=O)NC2CN(C(C3CCSCC3)=O)C3CC23)CCCCC1 Nc1c(C(=O)NCC(O)CNC(=O)CCCC2CC2)cc(Cl)cc1Cl c1(OC)cccc(Cn2nc(-c3occc3C)nc2Cc2ccoc2)c1 C(CC(C)C(=O)N1CCCCC1)=CCC.CC(C)(C)C.C(=O)(C)NC1CC1.C C1(CCNC(C2(COC)CCCCO2)=O)CN(C(c2[nH]cnc2C)=O)CC(C)O1 c1(OCC)cc(N(C2CCCN(C(=O)C(C)=CC3CC3)C2)CCO)nc(C)n1 c1(C(=O)N)cnc(C(F)F)nc1.C(c1ccsc1)=CC(=O)NCCC1CCC1 C(=O)(C1=NOC2(CCOC2)C1)NCC1(O)CCN(C(c2ccc(OC)o2)=O)C1 c1(CC=O)ncccc1F.C1(C(=O)NCCCNC(=O)NC)CC(C)C1.N C=CCCC(C)(C)C(=O)NCC(C1CCN(C(c2cc3n(n2)CCO3)=O)CC1)O C=C1CCN(C(=O)C(=O)NC2CC3(C2)CC3(F)F)C(CN)C1 CC1=CC(C(=O)NCC2(C(=O)N(CCCCO)C)CCC2)SC1 NS(=O)(=O)c1cc(C(=O)NC2CC(NC(c3ccccc3F)=O)C2)c(Cl)cc1F C1(C(=O)NCC(n2cc(-c3ccnc(CO)c3)nn2)C)Cc2ccccc2C1 O(NC(=O)C(c1ccoc1)NC(=O)Cn1ncccc1=O)CCC c1(OC)cc(C(=O)NC2CC3CC(NC(=O)C(C)(C)F)CC3C2)cc(O)c1O CC1=NNC(=O)C1CC(=O)NC(C)C(=O)NC(C)(C)C(C)O Cc1ccc(C(=O)NC2CC(C)N(c3cc(Cl)ncn3)C2)nc1C c1(CN2CC3CCN(C(C(C)(C)Br)=O)C3C2)cn2cc(Br)ccc2n1 N1(C(C(CC)=CCCC)=O)CC(NC(c2cncc(CC)c2)=O)CC1(C)COC C1(CNC(c2c(C(C)C)n[nH]c2)=O)CC(C)CN(C(C2CC23CCCC3)=O)C1 CC(CC(=O)N1CCCC(O)(CN(C(=O)C2=CC3C=CC2C3)C)C1)CC(F)(F)F c1(OC)cc(NCc2cc3ccccc3nc2OC)cc2ccccc12 C1CN(C(=O)CC2CC2)CC1(C)C.CCC(C(=O)N)NC(C)=O.C(C)=O Cc1cc(C)c(C(=O)N(CCCCNC(C2(n3cnnn3)CCOCC2)=O)C)s1 c1(C(N2CC3CN(C(c4occc4Br)=O)C3C2)=O)cccc2c1OCO2 C1(C(=O)NC2C(CC=C)CCC2)N(C(=O)C=C(C)C(C)C)CCC1(C)C c1(CC(=O)NCC(CC)NC(C2(C)CCCCO2)=O)n[nH]c(=NC)s1 CC1CN(C(C2CC(O)(c3cccnc3)C2)=O)CCC1NC(=O)Cc1ccns1 N1(C(c2ccc(CC)c(Cl)c2)=O)CCCC2(CCN(C(=O)COC(C)CC)C2)C1 N1(C(CN(C)CC)=O)CCC(C)C(CC(=O)NC(C(O)CO)C2CC2)C1 C1(NC(CCSCC)=O)CN(C(c2cc[nH]c2CC)=O)CC(F)(F)C1 Cc1nc(C)c(C(=O)N(C)CC2CN(C(c3cc(C(N)=O)cs3)=O)CCO2)o1 C1(NC(=O)Cn2cnnn2)CN(C(=O)C=Cc2ccc(Br)o2)CC1O N1(C(C(C(=O)OCC)(C)C)=O)CC2CC(C)N(C(=O)C(C)NC=O)C2C1 C1(C(=O)NC(C=CC(=O)NCc2c(C)n[nH]c2)(C)C)CCCC(C)C1 N1(C(C(CN(C)C)O)=O)CC2C=CC1C(C(=O)Nc1cccnc1C(N)=O)C2 C1(C(=O)NC(CNC(c2c(OC)c(Cl)sc2)=O)(C)CO)CCCC(C)(C)O1 C(=O)(C#CC1CCC1)NC1CC(C)(C(N2CCCC(CCC)C2)=O)C1 C12(NC(C)(C(C)COC)c3n(CC)nnn3)CCC(C(N)=O)(CC1)CC2 O=C1CC(C(=O)NC2CC(c3cccc(C(=O)O)c3)C2)c2ccccc21 Cc1cncc(CCNC(=O)CCOCCNC(=O)C(C)O)n1.C1COC1 C#CC1(C(=O)NC(CO)C(C)(C)C)CCN(C(c2ncncc2OC)=O)C1 C(C(C)(C)CC(=O)NC1CC12CC(NC(c1nc(Cl)c(Cl)s1)=O)C2)N(C)C C(C(C)(C(C)C)NC(=O)C(C)Cn1cccn1)NC(Cc1ccn(CC)n1)=O c1(C(=O)NC2CCC(NC(CC(C)(C)O)=O)CC2)cc2n(n1)CCCC2O c1(NC(=O)CC2COCCN2c2ncncc2Br)cccc(Br)c1O N1(C(=O)OC(C)(C)C)CCCC2(CCC2)C1.C1(CC(=O)N)COCC(C)(C)O1 c1(C(N2CCC(NC(C(C=CCCC)O)=O)C(C)C2)=O)cccc2c1ccn2C c1(NC(CCNC(C(C)=C(CC)C)=O)C)cc(C)c([N+](=O)[O-])cc1C(C)=O c1(C(=O)Nc2cccc(NC(CN3CCC(C)C3)=O)c2)nnn2c1CCC2 CCCCCCN(CCNC(c1scnc1C)=O)C(c1c[nH]nc1Br)=O Cc1nc(C(C)C)sc1CC(=O)NC1COCC1.C1(O)(C(C(=O)N)F)CCCC1 c1(C(N2CC(CC(C)NC(C3CCOC3=O)=O)C2)=O)ccc(C2(C)CC2)cc1 c1(C(=O)OC)c(C)nsc1NC1CN(C(c2ccc(C(=O)OC)[nH]2)=O)C1 N1(CC(C)NC(C2CCCC2)=O)CCN(C(c2ccn(C)n2)=O)CC1 CN=c1[nH]c(=NCc2cscc2C(F)(F)F)[nH]c(=NCC=CCl)[nH]1 C1(C)(NC(CCSCCCC)=O)CC(NC(=O)C(O)C2CCCC2)C1 N1(C(C2(O)CC(C)(C)C2)=O)C2CCC1CCC2.C(=O)C1=NNC(C(F)(F)F)C1.N C1(C(=O)NCC2(F)CCN(C(C(CC=C)C)=O)CC2)CC2OC(C)(C)OC2C1 CCC(C)CCCC(=O)N1CCOC(CCNC(=O)Cn2ncc(O)nc2=O)C1 C1(C(=O)NCCC(=C)CNC(c2c(Cl)cn[nH]2)=O)(N(C)C)CCCOC1.C c1(C(=O)NC(c2cn(CCC(=O)OC)nn2)C)cccc(C2(C)CC2)c1 N1(C(C2CC3(CSC3)C2)=O)CCC2(CCCN(C(C3CCCC3)=O)C2)C1 N1(C(c2cnc(COC)[nH]2)=O)CC2CCCC2C1.c1(CC(=O)N)ccc(F)cn1 c1(C(N(C(CNC(COC(CC)C)=O)C)C)=O)c(F)cc(OC)cc1F N1(C(C2(F)C(C)OCC2)=O)CC2(CCCCN2C(c2cc(S(N)(=O)=O)co2)=O)C1 c1(CC)sc(=N)[nH]c1C(=O)NCC1CCCCC1NC(=O)C(CC)CC C(c1csc2ccccc12)=CC(N1CCCC(NC(C(CCC)C(C)C)=O)C1)=O C=CCCC(CC(C)C)C(=O)NC1CN(C(=O)C(C)(C)C(F)(F)F)CC1O C(=O)(C1c2c[nH]nc2CCC1C)N1CCCC(C)(NC(c2c(C)n(C)nn2)=O)C1 C(=O)(CC(C)(C)CNC(=O)Cc1ccc(C)o1)NCC(C(=O)NC)O Cc1cc(CCC(=O)NCCCN(C2CCCC2)C(=O)CSCC(N)=O)no1 Cc1nc(C=CC(N2CCCCC2CN(C)C(c2ccccc2O)=O)=O)cs1 c1(C(=O)NC)ccc(OC)c(N(C2CC3CNC2C3)C(=O)C(F)Br)c1 c1(C(N2CC(CNC(c3c[nH]cc3C3CC3)=O)C(O)C2)=O)cccc2ncnn12 C1(CNC(C2C(SC)CCC2)=O)CC(C)CN(C(=O)CC2OCCO2)C1 c1(C2C(C(=O)NC)C2)ccccc1C(=O)O.c1nccn1CNC(=O)C Cc1ccc2oc(=NC3CC(CCNC(C4(CO)CCC4)=O)C3)[nH]c2c1 Cc1sc2ccc(F)cc2c1C(=O)NCCC1CCN(C(=O)C(C)N(C)C)C1 C1(NC(C2OCCN(C(C3N(C)CC(F)C3)=O)C2)=O)CNC(=O)C12CC2 c1(C(=O)NC2C(NC(C(COC)(C)O)=O)CC2)cccc2c1CCC2 N1(C(COC(C)(C)C)=O)CC2(CCC(C(=O)NC(C)(C)CC(C)(C)C)O2)C1 C1(C(=O)N)CC2C=CC1CCC2.CC(C(=O)N(CCC)CCO)OCC1CC1 C12(NC(CCCCC#N)=O)CCC(CC1)N(C(c1ccnnc1)=O)C2 C1(OC)CCC1C(=O)N(CCNC(=O)C(C)SC(F)(F)F)C1CC1 c1(C(N2C(CN(C(=O)C=CCO)C)CCC2)=O)[nH]c2ccccc2c1Br N1(C(c2c(C)c(Br)ccc2)=O)CCC2C(CCN2Cc2cc(F)c(O)c(F)c2)C1 O=S1CCC(N=c2cc(NCCSC(F)F)nc(C(F)(F)F)[nH]2)C1 C1(CC(=O)O)CC2(CCN(C(C34CC(CN3)C4)=O)C2)CO1.c1ccccc1.C=O C1(C(=O)NC2CN(C(C3CCCSC3)=O)C2)C2CC3C(C2)C13 c1(COC)cc[nH]c1C(=O)NC(C)CN(C)C(c1cc(C2CC2)no1)=O N1(C(C23OCC(COC)(C2)C3)=O)CC2CC(NC(C3CCCCC3)=O)C1C2 C=CCCCCC(=O)NC(C)(CNC(=O)C1=CSCCO1)C(C)C CC(CNC(c1c(F)cc(F)cc1F)=O)N=c1ccnc(C(C)(C)C)[nH]1 N1(C(c2c(CC)n(C)nn2)=O)CC2(C1)CN(C(=O)C=Cc1ccccc1)C2 C12(C(N3CC(NC(=O)C(O)P(C)(C)=O)CC(C)C3)=O)CCC(CO)(CC1)CC2 S(=O)(=O)(c1cccc(=NC(Cc2nccs2)CO)[nH]1)N1CC(CC)OCC1 Cc1cc(C(N2CC(NC(=O)CC(C)c3ccco3)C(F)C2)=O)c2n[nH]cc2c1 C1(NC(C=NOC)=O)CCC2(CC1)CCN(C(=O)C(c1cccs1)SC)CC2 CCC(CNC(=O)Cc1ccc(C(C)=O)s1)CC.c1ccncc1.C(=O)(C)N CC(F)(F)CC(=O)NCC1CC1C.c1(-c2cc(C(=O)N)no2)ccccc1Cl C1(C2CCC2)(CNC(C(C#C)(C)C)=O)CCN(C(=O)CCc2cnn(C)c2)CC1 N1(C(C=CC=CCC)=O)CC(NC(=O)CCC(=O)NCC)C(CC)C1 C(=O)(CC(C)(C)C(F)F)N1C(C)C(C(=O)NC2(C)CCCC2(C)C)CCC1 CC1CN(C(=O)C2=CC(O)C(NC(=O)CP(C)(C)=O)C2)c2cccnc21 CC1(C)CC(C(=O)NCCC[Si](C)(C)C)CCN1C(=O)Cc1cnns1 C=C1CCN(C(c2nccnc2C)=O)C(C(=O)NCCCCC(C)(C)C)C1 C=CCCC(C(=O)Nc1cccc(F)c1C)NC(=O)CCCOCCOC C(CCN(C)C)(C(=O)N(C)CCc1cccnc1)NC(CSCCOC)=O CC(C)CC(CC(C)C)C(=O)NCC(O)CN(C)C(c1cnc(C(N)=O)cn1)=O N1(C(c2cc(OC)no2)=O)CC2(CCN(C(=O)CC3CCCC(C)(C)O3)CC2)C1 C1(NC(=O)C(F)C(F)(F)F)CC2CCC1N(C(C1(CO)CCOCC1)=O)C2 C(=O)(CCC(F)(F)F)N1C(CCC(=O)NCC2CC2Cl)CCCC1 C1(NC(CCC#C)=O)CC(C)CN(C(c2cc(C(N)=O)ccc2OC)=O)C1 CCC(CC)(CC)C(=O)N1CC(NC(C2(F)CCS(=O)(=O)C2)=O)CC2(CC2)C1 c12ccccc1NCC2.c1(NC(CSC)=O)cccc(C(F)(F)F)c1 c1(C(N2CCC(N(C(C3C(C)CCOC3)=O)C)CC2)=O)csc(N=S(C)(C)=O)n1 c1(CN2C(CO)C=CC2)ccc(-c2ccc(OCC(F)(F)F)cc2)cc1F C1(CNC(CC(C)OC)=O)CCC2(CN(C(c3occc3C(C)C)=O)C2)O1 c1(C(=O)NCCCNC(c2c(OC)n[nH]c2)=O)cnn(C)c1N.c1ccccc1 c1(C(N2CC(COC)C2)=O)n[nH]c2c1CN(C)CC2.C1(C(=O)N)CCOC(C)C1 c1(C(N2CC(C)(NC(C(C)CC3CC3)=O)C2)=O)cc(F)ccc1C(F)(F)F C1(CCNC(Cc2cn(CC)nc2)=O)CC(OC)CN1C(c1csc(C)c1N)=O [SH](=O)(=O)c1c[nH]c2ncccc12.N1(C(C(F)=CC)=O)CCC(NC(=O)C)CC1 C1(C(N(CCC)C)=O)COC(C)(C)CO1.c1(C(=O)OC)sccc1C(=O)N C1CCCCC1O.c1(C(=O)N)ccn[nH]1.C1(C(=O)OC)CC(C(=O)NCC)C1 C(=O)(C#CC(C)(C)CNC(=O)C(C)CC#N)N1CC(C=C)OCC1 c1(C(=O)NCCC2CN(C(c3c(C)scn3)=O)CC(C)O2)cc2ncccc2[nH]1 C1(C(N2CCC2)=O)CC(C)(C)C1.c1(CC)ncsc1C(=O)NC.CC=O Cc1nccn1CC(=O)NC1(C)CC(C(=O)NCC(O)C(C)O)C1 c1(C(=O)NCCc2n(C)cnn2)c(C)nnn1C.C(=O)C=CCN1CCC1 CC1(C)OCC(CCC(=O)NCC2(NC(C3CC(CF)C3)=O)CCOCC2)O1 c1(C(=O)NCCCN(C(c2[nH]c(=NC)sc2)=O)C(C)C)ccc(C)c(C)n1 c1(NC(=O)N=c2[nH]occ2-c2ccc(F)cc2F)nc(Cl)cc2ccccc12 N1(C(CC2CCC(OC)CC2)=O)CC(NC(=O)Cc2nc[nH]n2)CC(C)C1 C1(NC(c2c(Br)cn(CC)n2)=O)CN(C(c2[nH]ccc2C)=O)C2(CCC2)C1 Cc1ncc(C(=O)NC2CC2CNC(=O)CC2CC2C(F)(F)F)[nH]1 N1(C(c2c(OC)cccc2)=O)CCC(C2CCC2)(C(N2CC3CCNC3C2)=O)C1 N1(C(=O)CNc2cccnc2)CCC2(CCCCN(C(c3cccnc3)=O)C2)C1 c1(CN2CC(CNC(c3cccc(OCC)c3F)=O)C2)cccn2ccnc12 c1(CC)ccccc1.c1(CC=O)nnc(C)o1.C(C=CC(=O)N)(CC)=CC N1(C(=O)C(O)C2CC2)CCN(C(c2cocn2)=O)C2(CCC2)C1 c1(CN(C2CCCC(CC(=O)O)C2)C)cc(C(F)(F)F)cc(F)c1 N1(C(C(CC)CO)=O)CCC(CNC(C2CC(O)C2)=O)C1(C)C Cc1snnc1C(=O)NCC1(NC(=O)CNc2cccnc2)CCCC1 c1(OC)cc(Cl)c(C)cc1NC(=O)C.c1(C=O)cccc(C)c1.C(C)=O.O N1(C(c2cc(Br)c(F)cc2Cn2cc(CO)nn2)=O)CCC(C2CCOCC2)C1 c1(C(=O)OC)nc(N2CCC(CNC(=O)C(C)NC(=O)NC)C2)ncc1Cl C12CC(CO1)N(C(c1ncn(C)n1)=O)C2.C1(C)(CC)CCC(C(=O)NC)O1 c1(C(=O)NCCSc2scc(C)n2)ccc2c(=O)n3c(nc2c1)CCCCC3 N1(Cc2c(C)n[nH]c2C)CCC=C(C(=O)Nc2c[nH]nc2-c2ccccn2)C1 CCCCCCC(C)C(=O)N1C2CC1CN(C(c1cc(O)cc(F)c1)=O)C2 c1(C(N(C2CCCCC2)C)=O)cc(S(N)(=O)=O)c[nH]1.C(CC(=O)N)N(CCC)C C(=O)(C(O)CCNC(c1ccn(CCF)n1)=O)N1CC(CC(C#C)C)C1 N1(C(C(C(C)O)C)=O)CC2(C1)OC1(C)CC2(NC(=O)COCCF)C1 CC1C(C)CCN1C1CCN(C(C2C3CCN2CC3)=O)CC1 C1(NC(C2(c3ccccc3)C(C)C2)=O)CCN(C(=O)C(O)C(F)(F)F)CC1(C)C CCC(CC)C(F)C(=O)NC1COCCC1NC(c1cnccc1Cl)=O CC(=O)CCC(=O)NCC1CC(NC(C2(C3CC3)CC2)=O)C1 N1(C(CCc2c(C)nn(C)c2C)=O)CCC(C2CCN(C(=O)C=CCF)C2)CC1 c1(NC(C2OCCC(NC(=O)CC3CCC=CCC3)C2)=O)ccc2nc[nH]c2c1 Cc1c(F)ccc2[nH]c(C(=O)NCC)cc12.C12(CC=O)CCC(CC1)C2(C)C.N C1(NC(C(N2C(C(=O)OC)CCCC2)CC2CCCC2)=O)CCC(F)(F)CC1 c1(COC)ccc(C(=O)NC(CN(C)C)C(=O)N(C2(C)CC2)C)o1 Cc1nn(C)c(Cl)c1CC(=O)NC1CC1.C1(CC=O)CCCN(C(C)C)C1.N N1(C(CC(CC)C)=O)CCCN(C(c2c(C(F)F)cccc2F)=O)CC1CO CC1CCNC(C)C1CNCCCOCc1ccccc1 CC(C)=C=CC(=O)N1CCC2CC12C(=O)NCCN1CCC(C)(C)C1 c1(C(N(C(C)C)CCNC(C2CSC2)=O)=O)ccc2nc(N(C)C)sc2c1 c1(CC(=O)NC(CC(C)NC(c2ncnc(C)c2C)=O)C)n[nH]c2ccccc12 CC1=CC(C)CN(C(C23CC2CN(C(=O)CCc2ccncc2)C3)=O)C1 S(=O)(=O)(c1nc(N2CCC(C)(C)C(CO)C2)ccc1Br)N(CC(C)(C)C)C Cn1nc(C(=O)NC2CC2C(F)F)c(Cl)c1Cl CC(C)C(CN(C)C)C(=O)N(C)CC1(NC(=O)CCc2cn[nH]c2)CC1 CCC(C(=O)N1CCCC1CN(C(=O)COc1ccc(C)c(Cl)c1)C)C(C)C CC(C)CC(O)CC(=O)NCC(C)(C)OCCNC(=O)C(C)S(N)(=O)=O C1(COC)(NC(c2cc(C(F)(F)F)ncn2)=O)CCCN(C(=O)C(O)CF)C1 C=CC(C)(O)CC(=O)N(CCCNC(c1nnn(C)c1C)=O)CC O=S(=O)(c1cnc(NCCn2cccn2)c(Cl)c1)NCC(Cc1ccco1)CO N1(CC2(C)CCN2C(c2ccc(O)c(CO)c2)=O)CCc2ccccc2C1 CC(C)C(F)(CNC(C12C=CC(CC1)C2)=O)C(=O)NCC(O)C1(Cl)CC1 C(=O)(C(CC)CC(C)C)NCC(CNC(Cc1c(CC)cccc1)=O)OC C1(n2nnc(CCCCc3cc(F)cc(F)c3)n2)(C(=O)O)CCC2CCC12 N1(C(C(c2cnnn2C)NC(C(N2CCOCC2)C)=O)=O)CCC(C)(CO)C1 C1(C)(CC(=O)NC(C)CNC(=O)CCC2CCCCN2C)CCCCCC1 Cc1cc(C)c(C(N2CCC(C)(NC(=O)Cc3ccnnc3O)C2)=O)cc1C C(=O)(C1CCc2nccn21)NC(C(=O)NCCN(C)C)C1CCCO1 O=C(CCC(=O)c1cccs1)NCCCC1CCCCN1C(C12COCC1C2)=O C1(C(N2CCC(C)(CNC(C3CC3C(N)=O)=O)C2)=O)(CC)CCCOC1 CC1CN(c2nnc(C3COCCO3)n2Cc2cccs2)Cc2ccccc2O1 C1(C(=O)NCCN(C(C2CCC(C)(C)C2)=O)C2CC2)CCCCC(F)(F)C1 N1(C(C(C(C)(C)C)OC)=O)CC2CCN(C(c3cc(C)on3)=O)C2C1 C(=O)(C(C#N)CC)N1CC(C)(CCC(=O)N(CCN(CC=C)C)CC)C1 C1(C)(C(=O)N)CCCN(C)C1.C1(C(=O)NC(COC(C)=O)CO)CC=CCC1 c1(C(=O)OCC2(C=C)CCC2)cc(N)nc(F)c1 C1(C(N(CCCCNC(C(C)CSC(F)(F)F)=O)C)=O)CCc2cn(C)nc2C1 c1cc(F)ccc1F.C1(CC)C(NC(=O)CC)CCN1C(=O)CC1CCOCC1.O S(=O)(=O)(c1cccc(Br)c1F)N1CC(NC(C(CCC)C)=O)C(C#N)C1 N1(C(COC2C(CC)CCCC2)=O)CCOc2ccccc2C1CO C(C(F)(F)C(=O)NC(CO)C(C)NC(=O)CCc1cnc[nH]1)OC C1(CNC(Cc2c(C)nc(SCC(C)C)s2)=O)OCCOC12CCC2 c1(C(=O)N)cnc2sccn2c1=O.C1(N(C)C)CC(C(=O)NCCC2CCC2)C1 c1(C(N2CC(C)(NC(C(CC(=O)OC)C)=O)C2)=O)cccc2oc(O)nc12 C12(C(N3CCC(C)(O)C3)=O)CCCC1CCN2C(c1cc(C(N)=O)co1)=O C(=O)(C(O)CC(F)(F)F)NC1C(NC(c2c(OC)n[nH]c2)=O)CCC1 C1(NC(C2CC(O)(CC#C)C2)=O)COCCN(C(=O)C=CC2CCCC2)C1 c1(NC)ncc(C=O)cc1Br.c1(NC(C2C(C(=O)OC)C2)=O)ccnn1C c1(OC)ccc(CCC(N2CCCC2CN(C)C(C2CC2(Cl)Cl)=O)=O)cc1O c1(C(N2CC(CNC(C(C3CCC3)OCC)=O)OCC2)=O)c[nH]c2ccncc12 CCC(CNC(=O)CC(C)n1ccc(C)n1)(CC)NC(c1cc(=O)n(C)o1)=O c1(CC(=O)N(C(CNC(C=CC(C)C)=O)C)C)ccc2ncccc2c1 N1(c2ncc(C#N)nc2)CCC(C2CC2)C1CNC(C1CCCN(C(N)=O)C1)=O CC1(NC(C2CC(n3cnnc3)C2)=O)CN(C(=O)C(C#N)C2CC2)C1 CCC(CC(=O)NCC1CSCCO1)N(C)C(c1nocc1Cl)=O Cc1ncnc(C)c1OCC(=O)NC(C1CSC(C(F)(F)F)C1)=O N1(C(c2cc(OCC)ns2)=O)CC2(CCN(C(=O)Cn3cc(C)cn3)C2)C1 CC1(C(N2CCN(C(=O)CC3(O)CCCCC3)C(CCO)C2)=O)CCCCCC1 C(N=c1[nH]nc(CO)s1)C1OCCN(C(C(C)(C)OCC(F)(F)F)=O)C1 C1(CNC(C2CCCC(C)(C)C2)=O)CCN(C(C2CC(F)(C)C2)=O)C12CCC2 c1(CNC(C(C)C)=O)cnc(C(C)O)s1 N#Cc1cccc(Br)c1NC(C1CCC(NC(c2ccn(C(F)F)n2)=O)C1)=O C1(NC(c2c(C)coc2C)=O)CN(C(=O)Cc2csc(Br)n2)CC1(C)C Cc1cc(C(=O)N(C(CNC(C2CCN(C)C(=O)C2)=O)C2CC2)C)nnc1O c1(C(N2CCC(N(C(CCC#C)=O)CCOC)CC2)=O)ccc([N+](=O)[O-])[nH]1 c1(C(N(C(C)CNC(c2n[nH]c3c2CCC3)=O)C)=O)nccc2ccncc12 CCCCC(CNC(=O)C=C(C)C(F)F)NC(=O)C(c1ccccc1Cl)O N1(C(c2ccc(SCC)cc2)=O)CCCC(NC(=O)C(C)(C)C2CCCC2)C1C c1(-n2cc(CNC=O)nn2)cccc(C)c1.c1(C2(C=O)CC2)cccc(Cl)c1.N c1(C(=O)N)cc(F)ccc1Cl.C1(F)(CNC(C(F)=CCC)=O)CC(C)C1 c1(C(N2C(CNC(c3c(CC)[nH]cc3)=O)CCC2)=O)nn(C)c2c1CSCC2 C1(C(=O)NC2C(CN=[N+]=[N-])CCC2)CCN(C(=O)Cn2ccnc2)CC1O c1(C(N2CCC(CNC(CCCSC)=O)(CO)CC2)=O)coc2ccc(Cl)cc12 C1(C(N(CCN(C(CC)=O)C(C)C)C)=O)CCC2(C1)CC2(F)F.C=CCC C1(CC(=O)NC(C)C2CC2)CCCC2(CC2)C1 C1(C(N(C2CC(OCC)C2)C)=O)CCN(C(C2CN3CCC2C3)=O)C12CC2 N1(C(C(C)(C2CC2)OC)=O)CCC2(CCCCC2NC(c2nc(C)oc2C)=O)C1 N1(C(C=CSC)=O)CC2CC2(CNC(=O)Cc2cc(C)ns2)C1 CONC(=O)CNC(=O)COC1(C)CN(C(c2ncc[nH]2)=O)C1 c1(C=O)cccc(SC(F)(F)F)c1.CC(C)CSCC(=O)N.C(C)C1CCC1 NS(=O)(=O)c1sccc1C(N1C2CCC1CN(C(=O)CCc1ccsc1)C2)=O CCC(C)(C)CCNC(=O)C(CNC(=O)CC1CCOC1=O)CC1CCCC1 N1(C(c2c(OC)ccs2)=O)CC2CCCC(NC(C3CCC(C)(C)O3)=O)C2C1 c1(CC(=O)NC2CCC(N(C(C(C=C)O)=O)C)CC2)cn2c(n1)CCCC2 c1(C(=O)NC2C(C)(C)CN(C(=O)C(O)C(F)F)CC2)ccc(N)c2ncccc12 N1(C(c2c(CC)onc2)=O)CCC2CCC(NC(c3ccc(F)cc3Cl)=O)C1C2 N1(C(C(CC)n2cccn2)=O)CC(C2CN(C(=O)Cc3csc(C)n3)C2)C1 c1(N2C(C)C(NC(=O)CC3CC(F)(F)C3)CCC2)nc2cc(F)ccc2o1 C1(NC(C#C)=O)CN(c2ncc(F)c(C)n2)CC1(F)F CCCC(C)(CC)C(=O)N1CCN(C(c2cnc(C)nc2CC)=O)C(CCO)C1 N1(C(CCCOC(C)=O)=O)CCC12CN(C(c1cn(C)nc1C(C)C)=O)C2 C1(CNC(C2CC(C)(C)O2)=O)CCC(CO)CC1 C1(C)(COC(c2snc(C)c2Br)=O)CC(c2cc(Cl)cc(Cl)c2)=NO1 C1(C(=O)NCC2(Nc3ncnc(CC)c3F)CCCC2)CCCC(F)(F)CC1 N1(C(C2(CC=C)CCCN2C(=O)CC2C=CCC2)=O)CC2(COCC(=O)N2)C1 Cc1c(O)ccc(C(=O)NCC2(F)CCC2)c1C.C1(=CC=O)CCOCC1.C c1(OC)ccnc(OC)c1C(=O)N(CCCCCCNC(c1cnc(C)o1)=O)C N1(C(C=CC)=O)CCCCC1.C1(C#N)(C(NC2CC2)=O)CC1C.CC.CO N1(C(C(C=C=C)C)=O)CCCC(C(=O)N(CC(=O)OCC)C)CC1 c1(C(N2CCC(=CCNC(C3CCCC3O)=O)CC2)=O)ccc(C2CC2)nc1O C1(CN=C(NCC2(C(C(C)C)O)CC2)NC2CCOCC2)OCCOC1(C)C CC(O)C(C(=O)N1CCC1C(=O)Nc1ccc(OCF)cc1)NC1CCCC1 C1(CNC(c2cc(C)sn2)=O)(NC(c2cnn(CC(F)F)c2)=O)CCCCC1C C1(CC)COCCN1C(=O)CC1CSC1.C1(C(=O)OC)C(C(=O)N)C1(F)F c1(C(=O)NCC2(NC(C(C)(O)C3CCOC3)=O)CCOCC2)cc(Cl)ccc1N c1(C(N2CCC3(C(NC(C(C)CF)=O)C3)CC2)=O)ccc(F)c2c1CCC2 c1(C(=O)NC2CC(CNC(CCCCCOC)=O)C2)cc([N+](=O)[O-])c(C)s1 c1(C(=O)NC(C)CCN(C)C(c2cnccc2Br)=O)cnc2ncccn12 C(=O)(CC(C)CC(C)C)N1C(CNC(c2cc(OC)cc(C)c2)=O)CC(F)C1 CCC(CO)(C(=O)NCC1(C)CC12CCC2)OC.c1(C=O)ccc(C)cc1N.N O=S(=O)(c1c(F)cc(Br)cc1F)NCc1ccc(F)c(CO)c1 c1(C(N2CCC(CN3CCCCC3CO)C2)=O)cccc(Cl)c1Cl c1(COC(C(CCC)NC(N)=O)=O)ncc(Br)cc1C CC1(C)OCC(C(=O)N(C2CCN(C(=O)CNS(N)(=O)=O)C2)CCO)O1 C=C(C)CN=C(NCC(C)(O)c1ccsc1)NCC1(C2CC2)CCC1 C1(NC(CCc2cncc(OC)c2)=O)CC(O)CN(C(c2coc(Cl)c2)=O)C1 C(CCC(C)CC(=O)N1CCC(N2CCN(Cc3cnc(Cl)s3)CC2)C1)=C(C)C CCC(C(C)(C)C(=O)OC)NC(c1ccc(-c2cncnc2)cc1)=O Cc1ccc(C(N2CCOC(CCNC(=O)CC3CCCC34CC4)C2)=O)nc1 c1(CC)c[nH]nc1CNC(c1cc(CC)on1)=O.c1(CC=O)cn(C)cn1 c1(CCCC)nc(C)c(CC(=O)N(CCNC(=O)C(C)C(F)F)C(C)C)s1 Nc1c(F)cc(C(=O)NCC2CC(F)CN2C(C2CC3(CCCO3)C2)=O)cc1F C1(C(=O)NCCC2CCSC2)(NC(C2N(C(C)(C)C)CC2)=O)CCSC1 c1(OC)cccc2c(CC(N3CC(NC(C4(O)COC4)=O)CCC3C)=O)coc12 N1(C(CCC(N)=O)=O)CCC(C2CCCN(C(c3cc(Cl)c([N+](=O)[O-])[nH]3)=O)C2)C1 c1(OC)cccc(CCNC(=O)C(C)N(C)Cc2ccccc2)c1 C(=O)(C1=CNC2=NCCC2=C1)NC(C)CN(C)C(C1CCc2cn(C)nc2C1)=O C1(C=O)C2CCCCCC12.C1(C(N(C2CC2)CC)=O)CCCCC1.N1CCCC1.N c1(OC)cccc(CCC(=O)NC(CNC(=O)CC(O)C2CC2)C(C)C)c1F c1(C(N2CC(OCCNC(C(C)n3cncn3)=O)C2)=O)cn2ccccc2n1 CCCCC(O)C(=O)N1CCC(C(=O)NCc2cc(F)cc(F)c2)O1 N1(C(Cc2onc(CSC)n2)=O)CCOC(CNC(C2CCOC(C)C2)=O)C1 C1(CNC(C(C2(O)CN(C(=O)CNc3ncccn3)C2)F)=O)CCC=CCCC1 c1(C=O)ccc(S(N)(=O)=O)cn1.n1(CC(N2CC(C)C2)=O)ccc([N+](=O)[O-])n1 Cc1ccc(-c2ccc(NC(c3c(C)cccc3Br)=O)s2)c(C#N)c1 c1(N2CC3CC(NC(C(C=CC)O)=O)C3C2)cc(C)c([N+](=O)[O-])cn1 c1(C(=O)NCCC2CN(C(=O)CCC3CC3(F)F)C2)ncoc1C1CC1 Cc1ncc(C(N2CCN(C(c3nc[nH]n3)C)CC2)C(=O)N(C)C)cn1 c1(C(=O)NCC2(SC)CC2)cc(CNC(C2CC2[N+](=O)[O-])=O)cs1 C(=O)(C1c2ccccc2CN1Cc1sc(Cl)nc1Cl)Nc1nnc(C(C)(C)C)o1 N1(C(C(CC)C#N)=O)CCC(S(C)(=O)=O)C1.c1(C=O)cc(C)n(C(C)(C)C)n1 CC1CN(C(C2(S(C)(=O)=O)CCC2)=O)CC(C)C1.C(=O)(CC1=NNC(=O)C1)N CCCCCCC(=O)N(CCOCCO)CCOCC.c1(C=O)ncn(C)n1.N C=C1CC2CCC(C1)N2C(C1CCCN(C(=O)C(C)C(F)F)C1C)=O c1(C(N2C(C(N(C(C)CO)C)=O)CCC2C2CC2)=O)cccc2nccn12 c1(C(N(C(C)CNC(=O)Cc2[nH]cnc2C)CC)=O)nccc(C)c1Br n1(CCOC)nccc1C(=O)N.C1(C)CN(C(C2SCCN2C(C)=O)=O)C1 c1(OCCOC)ncccc1C(=O)N(C1CN(C(c2cc(C)co2)=O)CC1F)C Cc1n[nH]c(C)c1C(C)NC(=O)C(F)CC1CN(C(=O)C)C1.c1cn[nH]c1.S C1(NC(C(C2(O)CCC2)NC(c2c(N)snn2)=O)=O)CC2CC1C(O)C2O C1(OC)CC(CC)N(C(C2CCCC2(F)F)=O)C1.C1(=C(C(=O)N)F)CCCCC1 C1(C)CN2CCC1CC2.n1(CC)nc(C(=O)NC2(CCC(=O)N)CCC2)c(C)n1 c1(Cn2cc(-c3c(C(=O)OC)nsc3)nn2)c(Cl)n[nH]c1C1CC1 C1(CNC(=O)C(c2cccnc2)O)CCCN(C(C2(C3CCCCO3)CC2)=O)C1 CN=C(NCC1CCCC1)N1CCc2cc(OC)cc(Br)c2C1 c1(OC)cc(C#N)ccc1C(N1CCCN(C(=O)C=C(C)C)CC1CO)=O N1(C(CN(C(=O)OCC)C)=O)CCN(C(c2sc(N(C)C)nc2Cl)=O)CCC1C C1(CC(=O)N(C(C)C)C(c2cnc(Cl)s2)=O)CCCC(C(F)(F)F)C1 C1(C(=O)N(C2CC2C)C)(OC)CCN(C(c2cc(C)oc2C)=O)C1 C(C1C(C(=O)N(C(C)C(N2CCN(C(=O)CC)CC2)=O)C)C1(C)C)=C(C)C Cc1ncc(Cl)c(C(N2CCC(CNC(=O)C=CBr)C(C)C2)=O)n1 C=CCC(C)C(=O)NCCN1CCN(C(C2CCS(=O)(=O)C2)=O)CC1 C1(C(C)NC(=O)CCCC2CCCC2)CN(C(=O)CC2CSCCO2)CCO1 C(=O)(C(C(C)NC(=O)CCc1nncn1C)C(C)C)N(CCSC)CC Cc1cccc(C(N)C(=O)NCCC2CCCCC2)c1.C(CS(C)(=O)=O)C(=O)N N1(C(CSCC(=O)OC)=O)CCCC1(C)C.c1(CCC(=O)N)nc(C)no1 Cc1ccccc1C=CC(=O)N(CC(C)NC(=O)CC1(C)CC1(Cl)Cl)C C1(NC(c2nncc(OC)c2)=O)COC2(C1)CN(c1cnc(F)cn1)C2 C1(O)(C(=O)NC(c2nc(C)on2)(C)C2CC2)CC(C)(C)C1 C12(C(N3CCC(C)N(C(=O)CC(C)(C)C#N)CC3)=O)CC(C)(C1)OC21CCC1 c1(C(=O)NC2CN(C(CCCC=C)=O)C(C)C2)n[nH]c2c(C)cccc12 C(N=c1cc(Cl)nc(C(F)(F)F)[nH]1)C1C2CN(C(=O)CCn3cc(Cl)cn3)CC21 C1(CNS(=O)(=O)c2c[nH]nc2Br)CCC2(CCC3(CC2)OCCO3)O1 CCCC(C(=O)NCC1(CNC(=O)C(CC)SC)CC1)N(C)C C(=O)(CC(C)(C)C(F)F)N1C(C(=O)NC(c2cscn2)C)CC1C C(CCCCC(=O)NC1CCN(C(C2C3CCC2CC3)=O)CC1)NC(C)=O Cc1nsc(C(N2CCC(NC(=O)C(C)(C)Cc3cnn[nH]3)C2C)=O)c1N O=C(C1=Cc2ccccc2C1)NCCCCC(CO)NC(c1csnn1)=O c1(NCC(C)NC(=O)C(C)Sc2nncn2C)ncc2ccsc2n1 Cc1ccc(C(=O)NC(C2(O)CCN(C(C3(C(C)C)COC3)=O)CC2)C)cc1F c1(C(=O)NCCCN(CCCCNC(C(COCC)C)=O)C)snc(O)c1Cl c1(NC(c2n(C)ncc2)=O)ncccc1C(N1CCN(CCF)CC1)=O c1(OCC)cnnc(C(=O)NCCOC(C)(C)C)c1 C1(NC(C2CC=CCO2)=O)CCCCCN(C(c2cc([N+](=O)[O-])c[nH]2)=O)C1 c1(C(=O)OC)c(F)cc(OCC(O)CN2CC(C)OC(C)C2)cc1Br c1(C(=O)NCC(C)(CO)NC(C2CCCO2)=O)ccc2n[nH]cc2c1 C1(C(C)NC(c2cn(CC(N)=O)nn2)=O)CCN(C(c2ccccc2Cl)=O)CC1 c1(C(=O)NC2(c3noc(C4CC4)n3)CC2)cc(C(F)(F)F)ccc1O C(CCCCCCC(=O)N1CCCC1C(C)(C)CNC(C1CCCCO1)=O)SC CCC(c1ccccc1)=CC(=O)NCCC(C)NC(c1c(C)nsc1NC)=O C(=O)(C1CCCc2c(O)cccc21)NC1C2CN(C(C=C(C)C)=O)CC21 c1(C(N(CCCNC(CSCC)=O)CC2CCCC2)=O)ccncc1CC N1(C(CSCC=C)=O)CCC(O)(C(C)NC(=O)CCCC2CCCC2)CC1 Cc1cccc(CC(N2CCN(C(=O)C(C)C(F)(F)F)CC2C(C)(C)C)=O)c1F C1(OC(C)C)CN(C(c2cccc(NC(=O)CCS(C)=O)c2)=O)CC1C(=O)O c1(CCCN(CCC(=O)OC)C(C(=O)N(CCOC)CCO)=O)ccccc1 C(=O)(C1CN(C)c2ccccc21)N1CCN(c2nc(C)cc(C)n2)CC1 CCC(O)C(C)C(=O)NCC1C(C)CCN1C(C1CCOC(C)C1)=O CC1CN(CCC(=O)Nc2cc(F)cc(F)c2)c2ccccc2NC1=O C1(n2cc(-c3c(C)c[nH]n3)nn2)CCC(C(=O)NCCN2CCC(CO)CC2)CC1 c1(NC(C(CC)NC(=O)C(F)n2ccnc2)=O)cnc(F)nc1 C#CCC(CC(F)F)C(=O)N1CCC1C(=O)NC1CCCC1N=[N+]=[N-] N1(C(c2nccc(C)c2)=O)CCC(C)N(C(c2cc(C(C)C)no2)=O)CC1 C=C=CC(C)C(=O)N1CCC(NC(c2[nH]ccc2CC)=O)C1 Cc1c(-c2cncc(C(F)(F)F)c2CC)cncc1F C1(C(NOCC(C)C)=O)(NC(=O)COC2(C)CCC2)CC(F)(F)C1 C(=O)(CCCC(=O)N1CC(OCCNC=O)C1)OCC.c1c(C)cccc1Cl C(C(=O)NCc1ncc(-c2ccc(C)cc2)o1)(C(C)C)NC(=O)OC c1(CN2CCCC(C(N(C)C)=O)C2)c(F)cc(C#N)cc1Br c1(NC(C(C2CCN(C(C3CC(C)(C)C3)=O)C2)F)=O)cnc2ccccc2c1 C12(CC(=O)N(CC(C)NC(=O)CO)C)CCC(CC1)OC2.c1ccccc1Cl N1(C(C(n2cnc(-c3cccs3)n2)C)=O)CCN(C(=O)CCCC(N)=O)C2CC12 n1(CC(=O)NCC2CC3CCC2N3C(=O)CCC2CCC2)ccc(O)nc1=O N1(C(c2nc(CC)oc2)=O)CCC(NC(=O)C(C)NC(=O)NC)C(C)C1 CC1=NOC(CC(=O)NCC(C)(C2CC2)NC(=O)Cc2cncnc2)C1 C(=O)(C=C1SCC(=O)N1C)NCC1(F)CCN(C(Cc2cccc(OC)c2)=O)C1 C1(CNC(C(n2cc(CCC#N)nn2)C)=O)CN(C)CCN1C(C1(C)COC1)=O c1(OC)cccc(C2=NOC(C(=O)NCCCCC)C2)c1.C1(C#N)(C(=O)N)CC1 N1(C(CSCC=C)=O)CC2(CCOCC2NC(=O)Cc2cc(F)ccc2)C1.O C(CCCCCC(=O)N1CC2(CCCC2)C1)NC(C(C)OC)=O Cn1ncc(CC(C(=O)NCC23CCC(CC2)C3)NC(=O)CN=[N+]=[N-])c1O N1(CC(=O)NCC(C)C)CCC2(CCCCN(C(=O)CCc3ccsc3)C2)C1 C(=O)(C1=NN(C)C(=O)CC1)N(CC(C)C)CC(=O)N(C(CO)C1CC1)C CC1CCN(C(=O)CC(C)(C)C)C(C(=O)NCc2c(F)cncc2F)C1 c1(C=O)ccc(P(C)(C)=O)cc1.C=CC(C)(CC)C(=O)NCCC1CCCC1.N C1(CCNC(c2cn(CC=C)nc2)=O)CCCN(C(=O)C(C)n2cccn2)CC1 Cc1cc(N)c(C(N2CC(NC(C3CCC4CC3CO4)=O)CC(F)C2)=O)cc1F c1(C(N2CCC(F)(CNC(C(CCCC)C)=O)CC2)=O)cn2cccnc2n1 C(C(=O)N=c1cnn(-c2ccccc2)[nH]1)Oc1ccc(NC(N)=O)cc1 c1ccc(C(c2ncc[nH]2)NCc2cn(Cc3cnc[nH]3)nn2)cc1 CCC(CC)CCCC(=O)NCC1CCC(NC(c2csc(F)c2)=O)CC1 c1(CNC(c2n[nH]cc2I)=O)n[nH]c2c1CN(C(c1cnon1)=O)CC2 c1(C(N2CCCC(C(C)C(=O)N(CC(F)F)CCO)C2)=O)c[nH]c2cccnc12 N1(C(c2cc(COC)[nH]n2)=O)CC2(C(=O)NCC(c3cccs3)O)CC1CCO2 c1(CC)ccc(NC(c2cc(N(C)C)cnn2)c2nnnn2CCCF)cc1Cl C1(NC(c2ncc(C)cn2)=O)CN(C(=O)CC2(C)CCCO2)C2(CCCCC2)C1 Cc1nn(C(C)C)cc1C(=O)N(C1CN(C(=O)COC(C)(C)C)CC1F)C c1(C(N2CCN(C(C(CSC)OC)=O)C(C(C)C)C2)=O)ccc2nnn(O)c2c1 c1(C(N2CC(CNC(C(CC)Sc3ccccc3)=O)C2)=O)cc2n(c1)CCCC2 c1(NC(=O)NCC2(OC)CCOC2)ccc(Br)cc1C(C)(C)C C1CC12CCN(C(C13CCC(O)(CC1)CC3)=O)CC2.C(C)(C(=O)N)OCCC#C N1(C(COC(CC)C)=O)CCC2CN(C(=O)CC(C)(C)F)C2C1 c1(N(CCC(N)=O)C(c2ccccc2F)CO)ncccc1S(=O)(=O)NCCF C1(c2n(C)ncc2)CN(C(c2cc(F)c[nH]2)=O)CCN1C(C1CC(N(C)C)C1)=O C1(C(N2CC=C(CNC(c3nc(Cl)sc3Cl)=O)CC2)=O)CCCC2(CCC2)O1 C1(C(N(CCCNC(=O)CC2CC(SC)C2)CC)=O)CCC(=O)NC1 c1(CCC(=O)NCC(C)NC(C2CC(SC)C2)=O)cnc(O)[nH]1 C1(C(=O)NC2CN(C(COC(C)C)=O)C(C)(C)C2)CCn2cnnc2C1 C1(CC(C)NC(CCCc2nc(C)sc2)=O)CCN(C(=O)CS)CC1.C(C)(C)C O=C(C1=CS(=O)CCC1)NCC1C2CN(C(=O)CN3CCOC3=O)CC12 c1(C(N(C2CCCN(C(C3CCN(C(CC)=O)C3)=O)C2)C)=O)cc(O)cc(F)c1 C1(CNC(CC2(CSC)CC2)=O)CN(C(=O)CC(C)c2ccco2)CC1O C1(CNC(c2ccc(O)nn2)=O)CCCN(C(=O)C=C2CCOCC2)CC1 N1(C(c2cc(CC)on2)=O)CCN(C(=O)CC2CC3CC3C2)C(c2cn[nH]c2)C1 O=C(N=c1ccc(-c2ccc(Cl)s2)n[nH]1)N1CC(NS(=O)(=O)C2CC2)C1 CCC(C)C(O)C(=O)NCc1cn(C2CN(C(c3cnc(SC)n3C)=O)C2)nn1 C1(NC(C(C)NC2CCCC2)=O)(CNC(C2COCCOC2)=O)CCOCC1 c1(C(=O)NC2CN(C(c3cc(C)n(C)c3)=O)CC2O)nn(C)c2ccc(Br)cc12 CN1CC=C(CC(=O)N2CCC(NC(c3cc(=O)cc[nH]3)=O)C2(C)C)CC1 C1(O)(CN(C(CN(C(C)=O)C)=O)C)CCCN(C(C2C3COCC23)=O)C1 c1(CCCC(=O)NC2COCCN(C(C3(Cl)CC3(F)F)=O)C2)c(F)cccc1F N1(C(CCN(CC)CC)=O)CC(NC(C2(c3cc[nH]n3)CCC2)=O)CC1C N1(C(c2c(OC)ccs2)=O)CCC2CC2(C(=O)NCc2cc(C)on2)CC1 Cc1nn(C)cc1C1=NOC(C(=O)NC2(Cc3ccccc3)COC2)C1 CCC(CCOC)C(=O)NC(C(=O)NC1CC(n2cncn2)C1)C(C)O C1(NC(CCNS(CC)(=O)=O)=O)CCCC(NC(C2CCCCN2C)=O)C1 c1(C(N2CC(NC(c3c(NCC)scn3)=O)C(C)C2)=O)ccnc(F)c1Cl C1(C(=O)NC(CC)COC)N(C(=O)COCC(=O)N(C)C)CCC1(C)C.O CC1(C)C(CNC(=O)C=Cc2ccccc2F)CCN1C(C1COCCOC1)=O N1(C(C(CC)C(F)(F)F)=O)CCC2(C=C(C(=O)NCCC(=O)NO)C2)C1 N1(C(C2CCC(=O)N2)=O)CC2CCN(C(c3ccnn3CC3CC3)=O)CC2C1 Nc1c(C(=O)NCC(CC2CC2)C(=O)NC2CCC(CCO)CC2)cccc1F C(=O)(CCC(C)CN(C)C)NC1CC(C)(NC(c2c(C)cc(F)s2)=O)C1 c1(CN2CCN(C(c3c(OC)ccs3)=O)C3C2C3)cccc2c1OC(F)(F)O2 C1(CNC(=O)C(=O)N)(NC(C2CCC23CCC3)=O)CCCCC1.C1CC1.C c1(CC(=O)N(C2CCCN(C(=O)CSC3CC3)C2)C)ccccc1OC(F)F C(=O)(C#CC1CCCOC1)NCC1(O)CN(C(Cc2cc(C(C)C)no2)=O)C1 c1(C(N(C2CN(C(=O)C=C3CCCCC3(C)C)C2)C)=O)cccc2cccnc12 N(C(=NCCC1=CCOCC1)NCc1ccccc1)CC1C(C)CCC1 C1(CN=[N+]=[N-])CCCN(C(=O)C(O)C2CN(C(=O)Cc3ccc(O)nc3)C2)C1 N1(C(c2c(C)ocn2)=O)Cc2nccn2CC(NC(=O)Cc2cccs2)C1 c1(CC)cc(OC)cc(C(=O)NCC2CCN2C(=O)C=Cc2cocn2)c1 CC1=C(C(=O)N2CCC(NC(c3cscc3Cl)=O)C(O)C2)CCCO1 c1(C(N(CCC#N)C)=O)ccccc1N1CCOCC1.c1ccccn1 Cc1[nH]c(C#N)cc1C(=O)NCCN(C(C1CC1(C)Br)=O)C(C)C C(N=c1nc2c(cnn2C(C)C)c(NC(c2cn(C)cn2)C)[nH]1)C1(OC)CCC1 CC1ON=C(C(=O)NC2(CNC(c3cccc4ccoc34)=O)CCOC2)C1C Cc1cc(C(=O)N(C(C)C(=O)NCC(O)Cn2cccn2)C)no1 C(=O)C1=NN2CCCN=C2N1.C1(C(N(CCOC)CC)=O)CN2CCN1C(C)C2 C1(C(N2CC(COC)(CNC(=O)CCC)C2)=O)C2CCCCC12.C(N)=O CCCCC(CC)C(=O)NCC1(CNC(c2nc(O)nc(O)c2N)=O)CCC1 C1(NC(COC2CC(NC(C(CC)n3cncn3)=O)C2)=O)CCC(F)(F)C1 C(N=c1[nH]c(=N)[nH]c(Cl)c1[N+](=O)[O-])C1CCCCN(C(CC(CC)C(C)C)=O)C1 C1(NC(CSCC)=O)CCCCC1NC(c1cnc(Cl)cn1)=O c1(C(=O)NC23C(CN(C(CSC(C)(C)C)=O)C2)C3)c(N)cc(F)cc1F N1(C(C(C)(O)C2CC2)=O)CCN(C(c2cccc(C(F)F)c2)=O)C(CF)C1 C1(C)(C(=O)OC)C=CCN1C(C1CC2CC2C1)=O C1(NC(c2c(SC)ccs2)=O)CCN(C(=O)C#CC2(C)COC2)CC12CCC2 C1(NC(CNC(CC)=O)=O)(CNC(=O)C(N2CCOCC2)C)CCCCC1C C#CC1CCCCN1C(=O)CCN(CC=C)C(c1cnccn1)=O O=C(C#CC12CC3CC(CC(C3)C1)C2)NC1CCN(C(C2OCCO2)=O)CC1O c1(C(=O)NC(C)CCNC(c2ccn(C(F)F)n2)=O)sc(Br)cc1F c1(C(=O)NCCN(C(=O)C(c2ccc(O)cc2)=O)CC)ccc(OC)nn1 C(N=c1[nH]c(=NCc2cnns2)[nH]c2cc[nH]c12)c1nc(O)c(Br)cc1 c1(CCCC(=O)NCC2(CNC(c3cnn[nH]3)=O)CC2)nc2ccccc2o1 N(C1CCCN(C)c2ccccc21)C(c1c(OC)ccs1)=O c1(OC)ncc(C)cc1NC(C1(F)CN(C(C2C=CCCC2)=O)C1)=O C1CC2(CCN(C(C34CCC3C4)=O)C2)C1.c1(C(=O)N)cccc(C(F)(F)F)n1 c1(C(=O)NC2C(CNC(C(C)Cn3cccn3)=O)CC2)cc(N)ccc1Br c1(CCC(=O)NC2C(NC(C=CSC)=O)C2)ccc(C(=O)OC)nc1 C1(NC(=O)COC2CC=CC2)CC2CC(NC(=O)C3=CCOC3)CC2C1 N1(CC(=O)NCCC2CCCN2C(c2csnc2Cl)=O)CCCCC1=O C1(C(=O)NC2C(NC(C3(C)CC(=C)C3)=O)CCC2)CC(C2CC2)C1 C1(CCN(C(=O)CCC)C)CCN(C(=O)CC2CC2)CC1.C(C)(C)C.C=O C(=O)(C(O)C(O)c1ccc(O)cc1)NCCC(C)(O)C1CC1 C1CC2(CCN(C(C3C(C(F)(F)F)C3[N+](=O)[O-])=O)CC2)C1.O=CC.C1CC1.S c1(C(N2C3CN(C(C(C)SC)=O)CC2CC3)=O)cccc2cc(F)ccc12 C1(C)(C(=O)NCC2CCC(C)CC2)CCCN(C(c2cc(O)nn2C)=O)C1 C(=O)(C(O)C(C)(C)C)N(CC)CC1CCCCN1C(=O)Cc1nncs1 C(=O)(C(C)C(O)C(C)C)NC(C(C)C)CNC(=O)C(c1ccccc1F)C N1(C(c2cn(C)nc2)=O)CC2CCC1CN2C(c1ccc(C#N)s1)=O O=C(CC(F)F)NC1CC1N(c1ccccn1)C(=O)CCN1CCCC1 C1(C)(NC(C(c2ccoc2)NC(CCCC(=O)OC)=O)=O)CCC(=O)N(C)C1 C(=O)(CC1OCc2ncccc21)NCC(CNC(c1c(C)c(Cl)cnc1)=O)(C)C C(=O)(CC(C)P(C)(C)=O)NC(CC)(CNC(=O)CN(C)CCOC)CC N1(c2ncnc(NCc3cnnc(C)c3C)c2C)CCCC2CC1C2(C)C c1(C(=O)NC2C(F)CCN(C(CN(CCC)C)=O)C2)ncc([N+](=O)[O-])n1C CC(C)(C)C(=O)CCC(=O)N1CCC(CCC(N2CCCN(CCO)CC2)=O)C1 c1(C(c2nnnn2C)NC(C(=O)OCC)C2CC2)oc2ccccc2c1CO N1(C(C(CSC)OC)=O)CCCC(O)(CNC(=O)CCc2cc(C)on2)CC1 c1(C(N2CCC(N(C(=O)CC(=O)N(C)C)CC)C2)=O)ccc(N=[N+]=[N-])cc1 C1(C)CCN(C(=O)C(C2CCCCC2)C)CC1.c1(CC)nc(C)c(C(=O)NC)s1 N1(C(C(C)=C2CCCC2)=O)CCCC(O)(CNC(=O)C(C)(O)c2ccccc2)C1 CCCCCCC(C)CC(=O)N(C)CC1CCN(C(=O)COCC2CCCC2)C1 C(=O)(C(CNC(=O)Cn1cnc(=N)[nH]1)C(C)C)NCc1ncc(C)cn1 C(c1cc(F)cc(F)c1)=CC(N1C2CC(NC(C(C)n3cnnn3)=O)C2CC1)=O C1CCC2(CC1)CN(C(=O)C(C)C#N)CCO2.C1(COC)(CO)CC1C=O c1(C(N(CCCN(C(=O)CC2CCCCO2)C)C)=O)cccc([N+](=O)[O-])c1 c1(C(N2CC3CN(C(C4(O)CCSC4)=O)CCC23)=O)cc2c(s1)CCOC2 N1(C(c2cn(CC=C)nn2)=O)CC(C)(C)CC1(C)C.C1(C)(CC=O)OCCO1 c1(C(N(C2CCN(C)C2)CCC)=O)cc(Cl)cc(C)c1C.C1CC1C(F)(F)F C1(NC(C(OC)OC)=O)C=CC(C(=O)NCCCn2ccnn2)C1 C(CCC(F)(F)F)NC(CC)CN1CCCC1 N1(C(c2c(C)ccc(C#N)c2)=O)CC(NC(C23CC(C)C2C3)=O)CC2(CCC2)C1 N1(C(CC2(C=C)CN(C(=O)CC3CC(SC)C3)C2)=O)CC2(CO)CC2(CO)C1 C1(NC(C=CC(CC)=CC)=O)CCC12CN(C(C1(CC=O)CCC1)=O)C2 CC1CCN(C(C2SCCS2)=O)C1CNC(c1ccc(-c2ccncc2)nc1)=O C1(C(=O)NC23CC2CN(C(c2cscc2Br)=O)C3)Cc2ccccc2C1 c1(CNC(CNC(CC)C)=O)cc(C(=O)NC(C)C(C)SC)cs1 c1(C(=O)NC2(CO)CCN(C(=O)C(O)CN3CCCC3)C2)cnc2n1CCOC2 CCCN=C(NCCCc1ccccc1F)NCC(C)(O)c1ccco1 S(=O)(=O)(c1cccc(C(OC)OC)n1)N1CCC(NS(CCC)(=O)=O)C1 CCC(C)(CC(=O)N1CC2CC(NC(=O)CCCC(F)(F)F)C1C2)C(=O)OC CCC(O)C(C)(C)C(=O)NCCC(C)(C)CNC(=O)C(C)(C)OC(C)=O C1(CC(=O)NCCC(CC)O)N(C(=O)CCc2nc(=N)[nH][nH]2)CCC1(C)C C1(NC(Cc2cccc(OCC)c2)=O)CCN(C(C2SCCCS2)=O)CC1F N1(C(C(CCC=C)(C)C)=O)CCCC2(C1)CN(C(=O)CS(=O)CC)CCO2 C1(c2n(C(CC)C)nnn2)(NCc2nc(Br)sc2C)CC2(CCC(F)(F)CC2)C1 c1(CC(=O)NC2CC(N(C(=O)C(C)(C)CN(C)C)C)C2)c(O)ncnc1O C#CCC(O)C(=O)NCC1CCCN1C(C1C(CN=[N+]=[N-])C1(C)C)=O Cn1ncc2c(NCCC3CC(F)C3)[nH]c(=NCCSCCc3cccs3)nc12 c1(C(N2CC(NC(CC(C)SC)=O)(CO)C2)=O)[nH]c2ccc(C)cc2c1Cl NC(=O)CCC(N)C(=O)NC1CC(n2cnnc2)C1 C1(CNC(c2cncc(C)c2C)=O)CC2(CCOCC2)CN1C(=O)C(C)N(C)C N1(C(C(CC=CC)CC)=O)CCC2CN(C(c3cnc(C4CC4)[nH]3)=O)C2C1 CS(=O)c1ccc(C(=O)NCC2(F)CCCC2)cc1.C1(F)(C(=O)N)CCCC1 N1(C(c2cnc(C)c(N)c2)=O)CCC2CCN(C(=O)CCCN=[N+]=[N-])C2C1 Clc1cc(NC(=S)NC2(Cc3ccccc3)CCC2)cc2c1OCCO2 c1(OC)cncc(-c2cn(CC3CCN(C(C4OCC4(C)C)=O)C3)nn2)c1 N1(CCNC(C(C)(C)NC(C(F)=CCC)=O)=O)CCCCCC1 N1(C(c2c(CCC)onc2C)=O)CC2CN(C(c3coc(CC)n3)=O)CC12 C1(C(C)(C)O)CN(C(=O)C)C1.C(C)(C(=O)NC)SC.C1(C=O)CCC1 N1(C(C2(C)C(C)C2)=O)CCC(NC(c2cccc(N3CCOCC3)n2)=O)C(O)C1 Cc1csc(C(N2CC(CNC(c3cn(C)nc3-c3nccs3)=O)C2)=O)c1Cl C1(Nc2cc(NCC3CN(S(CC)(=O)=O)C3)ncn2)C(=O)N(C)CCC1C c1(C(N2CC(C(C)NC(c3c(CC)nns3)=O)OCC2)=O)cc(Cl)ccc1N c1(CNCc2cccc(C(=O)NCCC(=O)NC)c2)cc(Br)ccc1C C12(CC)CCC(CC1)C2.c1(CC)nc(CC=O)cs1.C(C)(C)CC=CC=O.N C1CCN(C(C)=O)CC1.C=C1C(C=O)C1C(=O)N(CCC(C)C)C1CC1.O C1(NC(c2ccn(CCC)n2)=O)CC2(C(=O)NC3CC(C)C3)COC1C2 N1(C(C2CN(CP(C)(C)=O)C2)=O)CC(=O)N2CCOCC2C1 N1(C(c2c(C)nc(CC)o2)=O)CC2CCN(C(c3cnc4n3CCCC4)=O)C2C1 c1(C(=O)NCCC2N(C(CC(C(C)C)C)=O)CCC2)cccc2[nH]nc(O)c12 c1(C=O)c(F)ccc(F)c1F.CN1C(=O)CCC1C(=O)NC(C)C(C)(C)C.N N1(C(COCCCC)=O)CCCC(CO)(NC(C2CC(C)CO2)=O)C1 c1(C(C)NC(=O)N)cnc(C(F)(F)F)s1.C1CCN(CCc2ccccc2)C1 C(=O)(C(O)C1=CCCCC1)NC1CCN(CCNC(C(CC=C)C(C)C)=O)CC1 C(CC(C)C(=O)NCC1CCC(C(=O)NCc2ccnc(O)c2)CC1)OC c1(C=O)c(C)nn(C2CC2)c1Cl.C1(C(=O)N)(COC)C=CCC1.C1CCC1 C1(NC(=O)CCc2cncs2)CCC2CN(C(C34CCCC3C4(F)F)=O)CC2C1 CC(C)(F)C(C)(F)C(=O)N1CC(CO)(NC(C2CCC3CCCCN23)=O)C1 c1(C(N2C3CC(NC(C(=O)N(C)C)=O)(C3)C2)=O)cc(Br)cc([N+](=O)[O-])c1N c1(N2CCCC(CNC(C(C)=C3CC3)=O)CC2)ncnc2c1nnn2C N1(C(c2nnc(C(C)C)s2)=O)CCC2(CC1)CC(NC(=O)C(C)(C)F)CCO2 c1(C(c2n(C(CC)C)nnn2)NCc2ncc(C)s2)ccnc(F)c1C Cc1ncnc(C)c1NC(C1CCN(C(C2CCC(=O)C(C)C2)=O)CC1)=O CN1CCOC(C(=O)N(C(CNC(C2(CF)CC2)=O)C2CC2)C)C1 c1(C(N2CCC(C(C(NOC(CC)CC)=O)F)C2)=O)ccccc1N=[N+]=[N-] C12(C(N3CCC(CNC(=O)C(C4CCC4)C4CCC4)C3)=O)CCC(CC1)C2 C1(CC(=O)N)CCOC1(C)C.c1(C(N(CCC)CC)=O)ccccc1.C1CC1 N1(C(C=C(C)c2ccsc2)=O)CC(CNC(=O)CC)C2(CC2)C1.C(N)=O.N c1(C(=O)NCC(C)(C)NC(Cc2n(C)ncc2Br)=O)cn(C)c2ncccc12 Cc1cc(Br)c(C(N2CC(CCc3cn(CCC(F)(F)Cl)nn3)C2)=O)s1 N1(C(c2cccc(CC)n2)=O)CCC2CC2(C(=O)NC(C(=O)O)C2CC2)CC1 c1(OC)cccc2c1CC(NCC1CCC1C(F)(F)F)C2 c1(C(C)(C)NC(=O)CC2(O)CCC2)c(F)cccc1Cl C1(C)CN(C(=O)C2=NOC(C)C2C)C(C)(C)C1.CC(CSC(F)(F)F)C(=O)N C1(N(C(c2cc(C)oc2)=O)C)CC2CC1N(C(=O)C(C)Cc1ccccn1)C2 C(CC1=CCN(C(c2ncoc2C2CCOCC2)=O)CC1)NC(C1C(CC)C1)=O c1(C(N2CC(O)(CCNC(=O)CC3CCCSC3)C2)=O)ncc(Cl)cc1O S(=O)(=O)(c1c[nH]ccc1=NC(C)c1sc(C)nc1C)NCC(=C)Cl c1(OC)ccnc(C(N2CC(NC(=O)CCn3ccnn3)C(SC)C2)=O)c1O c1(C(=O)NCC(CN(C(C(CC)n2ccnc2)=O)C)O)ccc(C#N)cc1OC C(=O)(CC(O)(c1ccccc1)C1CC1)NCC(C)N(C(CN(CCC)C)=O)C N1(C(c2cnc(CC)s2)=O)CCC(C(=O)NC(c2ccoc2)C)C12CC2 Cc1c(C(=O)NCC(O)C)nnn1C(C)C.C1(C(F)(F)F)(C=O)CCC1.N N1(C(C2C(=C)CC2)=O)CCCC(N(C(=O)Cc2ccccc2COC)C)CC1 N1(C(C=CC=CC)=O)CC2CCN(C(=O)CCCCNC(N)=O)C(C2)C1 C1(C)(OC)CCN(C(c2sccc2)=O)CC1.C1(C(=O)NC)CCC1.C(C)=O C1(C(N2CCCC(C)C2CO)=O)CN(C(=O)OC(C)(C)C)CC1C1CC1 c1(C(=O)NC2(CC=C)CN(C(=O)C(C)(COC)OC)C2)cc(Cl)c(Cl)s1 C1(C(=O)NCc2c(C)noc2)C2CCCC2CN1C(C1C(C)C1C)=O CCC(C)(C)C(C)CC(=O)NC1(CO)CN(C(c2ccc(F)c(SC)c2)=O)C1 CCC(C)(C(=O)NCC(C1CCCC1)NC(=O)CC1CCOC1)C(N)=O Cc1cn2nc(C(N3CCC(CCN(C(=O)C(C)C#N)C)CC3)=O)cc2c(=O)[nH]1 c1(C(N2CC(CC)C2)=O)cncc(C(C)(C)C)c1.C1(CC)CC1CC(=O)N C=C=C(C)CC(=O)NCC(C1CCN(C(C2CCN(C3COC3)C2)=O)CC1)C c1(OC)ccc(C)cc1C=CC(=O)NC(C)CC(C)C.C(=O)(C=CCO)N C1(NC(c2c(C)cc(C)s2)=O)CC2CCC1N(C(C1CC1F)=O)C2 C1(C(=O)NCCNC(Cc2nc(C)oc2)=O)CC(F)C(=O)N1 c1(C(=O)OC)ccc(CC(C(=O)OC)NCc2ccc(CN)cc2)c(Br)c1 CC(F)(F)CCC(=O)NCC1(NC(C2CC(F)C(=O)N2)=O)CCCC1 Cc1nc(C(N2CCC(NC(=O)CN3CCC(C)(C)C3)CC2C)=O)cc(O)n1 C#CCC(CC(=O)NCCC(C)F)NC(=O)C(Cl)Cl Cc1ccc(C)c(NC(=O)CNCC2CN(Cc3cccc(Cl)c3)CCCO2)c1 Cc1cccc(CNC(C2CCCC(NC(=O)COCCCF)CC2)=O)c1C C1(CNC(CC(=O)NCC)=O)CCN(C(C2CN(C)C(=O)N2)=O)C12CC2 N1(C(CSCCC)=O)CCC(NC(c2ccc(N)c(F)n2)=O)C(C)C1 Cc1nn(C)c(C(=O)NC2CCCCCN(C(c3c[nH]nc3F)=O)C2)c1[N+](=O)[O-] N1(CCC(=O)NC(CC)CN(C(c2cc(Cl)cs2)=O)CC)C(C)CCCC1C Cc1sccc1NC(=O)CC1(C)CCN1C(C1(C)CCCC1)=O c1(CC)ccc(C(=O)NC2CCN(C(c3ccc(O)nc3)=O)CC2)c(F)c1 C(CC1CC1)(C(=O)N(C)Cc1c[nH]nc1C)NC(CN(C(C)=O)C)=O C(CC(C)(C)C(=O)N(C)CC1CCN(C(c2coc(C(F)F)n2)=O)C1)OC n1(CCNC(C2(C)C(C)C2)=O)cnc(C(=O)NCCc2ncc[nH]2)c1 N1(C(c2nccc(CC)c2)=O)CC2CC(NC(c3occ4c3CCC4)=O)CC2C1 C(=O)(CC(C)C(C)C)N(CCN(C(c1cn(CC)nc1C(C)C)=O)C)C C(CC(C)C)(C(=O)N1CCC(C)(C)C1C(N1C(CO)CC1C)=O)OC c1(C(N)C(N2CC(O)(CCC(F)F)C2)=O)c(F)cccc1F.C12=CC=C(C=C1)C2 CN1CCN(C(=O)C=Cc2nccs2)C(C(N2CCC(C#N)C2)=O)C1 N1(C(CN(c2ccccc2)CC)=O)CCC(C)C1(C)C.C1(C=O)CC(=O)N1.N C1(NC(C2(OC)CCCC2)=O)CN(C(=O)Cc2cnc(C)[nH]2)CC(F)(F)C1 NC1(C(=O)NC2(CO)CCOC2)CS(=O)(=O)C1 C1(C(N2CC(C(C)C)OCC2)=O)CNC(=O)CN1C(=O)CC1COCCO1 C(=O)(C1CCc2c[nH]nc21)NCC(C1CCCN1c1ncncc1Br)(C)C Cc1cc(CC(=O)NC2CC3(C2)CC3NC(c2[nH]nnc2C)=O)ccc1F Cc1nc(C(C)C)sc1C(N1CC(N(C(=O)CN(C)C2CC2)C)C(F)C1)=O C(C(=O)N(CCCNC(c1cccc(S)c1)=O)C(C)C)(C(C)C)OCC C1(OCC(N)=O)CCN(C(c2sccc2CNC(c2cnccn2)=O)=O)C1 C1(NC(C(C=CCCC)O)=O)CC2CCCC(C1)N2C(c1ccccc1O)=O C1(C)(c2cn(CC(C)(C)C)nn2)CCCN(C(C2OCCO2)=O)C1 CCC(CC(=O)NC1C=CCC(C(=O)NCC2CSCCO2)C1)C(C)C N1(C(C2SCCCS2)=O)CC2CCN(C(=O)C(C3CCOCC3)F)CC2C1 CCC(C)(C)CC(=O)N1CCCC1(C)C(=O)N(CC(C(C)C)OC)C c1(CCOC)nc(=NCC2(O)CN(C(=O)C(C3(O)CCCC3)F)C2)s[nH]1 C1OCCOC12CCC2.C1(NC(C)=O)CCCCC1NC(=O)CC1(C)CN(C)C1 N1(C(c2ccc(CC(C)C)s2)=O)CC(CO)C2(C1)CN(C(=O)C(C)C1CCC1)C2 c1(C(N2CC(C)C(NC(C34CC3COC4(C)C)=O)CC2)=O)c[nH]nc1S(N)(=O)=O CCCC(C)(C)CN=c1cc[nH]c(=NCCCC2CCCC2)[nH]1 c1(OC)cc(CC(N2CC(NC(C3C4CC4C4CC34)=O)C2)=O)ccc1F N1(c2[nH]c(=NCc3n(C)ncn3)[nH]c(=N)n2)CCC(C2CCCCC2)CC1 C(N=c1nc2sccc2c[nH]1)C1C(NC(CC2CCCC(=O)N2)=O)CCC1 N12CCCC(C1)C(=O)NC1C=CCCC1C2=O.C(C(O)CC(=O)OC)OC c1(C(N2CC(N(C(COCCC=C)=O)C)C(F)C2)=O)c[nH]c(=N)nc1C C(C)(CCC(=O)NCc1cc(C(=O)NCCC2CCC2)no1)OCC.O CC1OC2(C)CC1(C(=O)NC1CCC(CNC(c3cccc[n+]3[O-])=O)CC1)C2 c1(NC(CC2(C)CCN(Cc3n(C)ccc3)C2)=O)ncc([N+](=O)[O-])cc1Br c1(C(=O)NC2CN(C(C(COC)(C)C)=O)CC2C)[nH]c2ccccc2c1Br c1(NC(C)CS(C)(=O)=O)ncccc1S(=O)(=O)N1CCCC1CN1CCCCC1 N1(C(c2c(C)noc2)=O)CC(F)(F)CC1(C)CNC(=O)CC1OCCCC1(C)C Cc1cc(C(=O)NC2CCOC2C(=O)NCCC2(C)N=N2)ncc1F CCC(CN(C)C)CC(=O)N(C1CN(C(c2cc(CCCO)on2)=O)CC1O)C c1(NCC(CC(C)C)NC(=O)COCC2CC2)nc(Cl)nc2c1ncn2C c1(CC)ccccc1C(=O)NCC1CCCC(NC(=O)C(F)=C(C)C)C1 C(CC(C)CCNC(=O)CCCc1cccnc1)NC(C(CSC)C)=O Cc1n[nH]c(C)c1C(=O)NC(C1CCCN1C(c1c[nH]c(=N)s1)=O)C C1(C)(CNC(c2ncn(C)n2)=O)CCCN1C(=O)CSCc1cscn1 C#Cc1ccnc(C(N2CCOC(CNC(C3(C)CCN(C)C3)=O)C2)=O)c1 N1(C(CCCOCC)=O)CCCC(n2cc(-c3cccc(CO)n3)nn2)C1 c1(C(C(=O)NCCOCC2CC2)N(CCOC)C)scc(C)c1C c1(C(N2CCC(C)(NC(COCc3cc(C)no3)=O)C2)=O)nc[nH]c2nccc1-2 C(=O)(C(C)c1ccco1)N(C(C)C(=O)N(C1(COC)CC1)C)CC N1(C(c2cc(C(N)=O)[nH]n2)=O)CC2(C(=O)NC3C(O)CC3O)CC1CO2 C1(C(=O)NCC(C(F)(F)F)OC)CCCCCCN1C(c1ccnc(O)c1)=O C1(CC(=O)NCCCN(c2nc(C(C)(C)C)ns2)C)CCCCN1C C1(C(=O)NCCCNC(CSC)=O)CCCCN1C(=O)C1CC1 C(=O)(C(C)CN1CCOCC1)NCCCN(C(CC1CC(CC)C1)=O)C C1CC(C)(C)CN1C(=O)Cn1cc(C(F)F)cn1.C(CC(C)C(=O)N)=CC CN1CCC(CC(N2CC3C(CN(C)C(c4cc(Br)co4)=O)C3C2)=O)CC1 C1(C(=O)NCC(CC)C(C)C)CCN(C(c2cc(COC)[nH]n2)=O)C12CCC2 c1(C(=O)NCC2N(C(C=Cc3c(C)ncs3)=O)CC2)nnc(O)c2ccccc12 Cc1nn(CC(=O)NC2CCN(C(c3c(Cl)nn(C)c3Cl)=O)C2)c(C)c1[N+](=O)[O-] N1(C(C(N2CC(NC(C(C)N(C)Cc3cccs3)=O)C2)=O)C)CCOCC1 CC1CC(CNC(c2ccc(CS(C)(=O)=O)o2)=O)CN1C(c1ccccc1)=O c1(C(C(=O)NC(C)CNC(C2(CO)CCCO2)=O)(F)F)cccc(Br)n1 N1(C(CN2CC(C)(OC)C2)=O)CCN(C(C2(c3cccc(Cl)n3)CC2)=O)CC1C Cc1ccc2c(C(N3CCC(O)C(C(=O)NC4CS(=O)(=O)C4)C3)=O)cccc2c1 N1(C(=O)CCCCC2CC2)CCC2(CCCN2C(C2CCOC2C2CC2)=O)C1 c1(C(=O)NC2CCC(C)N(C(=O)CS(=O)(=O)C3CC3)C2)cn2cc[nH]c(=O)c2n1 CC1c2cc(F)cc(F)c2CCN1C(=O)C(C1CS(=O)(=O)C1)N c1(OC)ccc(C(C)=O)cc1CC(N1CCC(CO)CC1C)=O Cc1cnc(NCCCCF)c(S(=O)(=O)NC(c2cnn(C3CC3)c2)C)c1 N1(c2ccc(C)nc2N2CCCC2)CCn2c(nc3ccccc23)C1 c1(C(=O)NC2CN(C(c3scc(OC)c3)=O)C3C2C3)csc(S(C)(=O)=O)c1 Cc1ncc(Br)cc1CNC(=O)NC1CC(F)C1 c1(CC)n[nH]c(=NC2CCN(C(C3CCc4nn[nH]c4C3)=O)CC2C)s1 N1(C(C2CCCN(C(c3n(C)c(=O)ccc3)=O)CC2)=O)CCOCC(C)(C)C1 C1(NC(C=Cc2c(C)nccc2)=O)CC2CN(C(=O)COCC3CC3)CC2C1 CC(C)(F)CCC(=O)NCCC1CN(C(=O)CNC(C2CCC2)=O)CCO1 C(c1cn(C)c2ccccc12)=CC=O.C(=O)(CSCC=O)OC.C1CC1.N c1(C(=O)NC2CN(Cc3ccc(OC(F)(F)F)cc3)CC2F)ccc([N+](=O)[O-])s1 N1(C(C2C(C(=O)OC(C)(C)C)C2(C)C)=O)CCC(N)C(F)(F)CC1 N1(C(CC(=O)NCC#C)=O)CCN(C(c2ccccc2COC)=O)C2CC12 Cc1cccc(O)c1NC(c1csc(NC(c2ccc(O)nc2)=O)n1)=O C(=O)(CCC(F)(F)Cn1cc(CCc2nn[nH]n2)nn1)N1CCC(C(C)(C)F)CC1 c1(C(N2CC(CN(C(CCC(C)=O)=O)C)C2)=O)c(C(C)C)cccc1C c1(C2(F)CCN(CC(=O)NC(c3cc(C)oc3C)C)CC2)cccc([N+](=O)[O-])c1 N1(C(CN(C(C)=O)C)=O)CC2CC(NC(=O)CSc3cccs3)C1C2 CC1(C(=O)NCC(O)CCNC(=O)C(c2ccccc2Cl)(F)F)CCC(=O)N1 C(C)(N=c1[nH]c(N(C)CCOC(F)F)nc2c1CSC2)c1c(C)nn(C)c1 C1(C(=O)NC2C(NC(CC(C)C)=O)CCOC2)CCc2ccc(F)cc2O1 C1(C(=O)NC2(C)CCSC2)C2CC3C(C2NC(c2ccc(F)cn2)=O)C13 C(CCC(C)CC(=O)NC1CCC(C)N(C(c2nnnn2C2CC2)C)C1)=C(C)C c1(OC)cc(C)c(C(=O)NC2CCC(C(=O)NC)OC2)cc1C.C1(C)CCC1 c1(N2CCC(N(C(CC(C(F)(F)F)OC)=O)C)C2)ncc(S(C)(=O)=O)cc1Cl c1(OC)cc(=NC(=O)C(=O)NC2CC(C)(C)C2c2ccc(Br)cc2)[nH]n1C CC1C(C(=O)NCCC2CCN(C(c3occc3-c3ccccc3)=O)C2)C1(F)F c1(OC)cc(C(N2CCN(C(c3csnc3Cl)=O)CC2CO)=O)cc(C)n1 N1(C(C2C(C)C2)=O)C2CCC1CC(CC(C)NC(c1cccc(F)c1)=O)C2 c1(C(C(=O)NC(CC)CNC(c2nn[nH]c2Cl)=O)(F)F)ccc(=O)n(C)c1 CC1(C)COC2(CC3CC(NC(N4CCC(CS(N)(=O)=O)CC4)=O)CC3C2)OC1 C1(NC(C2C(C)C2)=O)CCOC12CCN(C(=O)CC1CCCN1C)CC2 C(=O)(CC1CCCc2c1[nH]c1ccccc21)NC(CNC(COCC)=O)C(C)C Cc1nc(C)c(C(=O)NCCC2CCCCN2C(c2csc(C#N)c2)=O)c(C)n1 N1(C(CCN(CC)CC)=O)CCCC(C2CCCN(C(=O)C(C)(C)C(N)=O)C2)C1 c1(C(N2CCC(CCOC)C2)C(=O)NC(CC)C)cc2cc(OC)ccc2o1 c1(CCOC)nc(-c2ccc(C(F)(F)CF)cc2)n(C23CC(C2)C3)n1 N1(C(C2C(C(=O)OC)C2)=O)CCC(NC(c2cc(C)ncn2)=O)C(C)(C)C1 C1(CNC(CN2CC(CC)C2)=O)(NC(=O)CC(C)C(C)C)CC2CCC1CC2 C1(C(C)NC(=O)CCCn2cncn2)CCC(CNC(=O)CC(C)F)CC1 C12(C(=O)NCCC3CC(C)C3)COCC1CN(C(=O)C(O)C1CCC1)C2 CC1(C)CCCCC1=CC(N1CCC2CCC12CNC(=O)CC1CC1)=O c1(OC)ccc(Cl)c(C(=O)NC2CCC(C)N(C(C3CCOCC3(C)C)=O)C2)n1 c1(CNC(C2CCC(NCc3ccc(CO)o3)C2)=O)cnc(Br)s1 Cc1cc(F)ccc1C(O)C(N1CC(CNC(=O)Cc2nncn2C)C(C)C1)=O C(=O)(CCCC(=O)N1CC2CC1(C(N1CCCC1(CO)CO)=O)C2)OC C1(C(=O)NCC)(CC)C=CCN1C(C1CCCN1C(C)C)=O.c1ccccc1 c1(OC)ccc2c(c1)C(CO)(NC(c1ccc(OC)c(Br)n1)=O)CC2 CC12CN(C(c3ccccn3)=O)CC1(C)CN(C(C1(CO)CCC1)=O)C2 c1(C(=O)NC2C(CNC(c3ccc(C(C)=O)[nH]3)=O)CC2)cc(C)oc1C c1(NC(c2ncc(Br)s2)=O)cc(-c2cnc(N3CCNCC3)s2)ccn1 C=CC1(CC(=O)NC2CN(C(c3coc(OCC)n3)=O)CC23CC3)CCOCC1 c1(CC(N2CCC(NC(c3c(CC)noc3)=O)(CF)C2)=O)nsc2ccccc12 C1(OCC(=O)NC2(CC=C)CCN(C(c3ccc[nH]3)=O)C2)C#CCCCCC1 N(C1Cc2ccccc21)C(=O)Nc1n(C)cc(Cl)c1 c1(NS(=O)(=O)c2cscn2)ccc(Cl)c2nsnc12 C1(CNC(C(C2CCC(=O)N2)C)=O)CC(F)(C)C1.c1(C=O)c[nH]c(=N)s1 N1(C(c2cc(C)cc(Cl)c2)=O)CC(C2CN(C(=O)Cc3sc(C)nc3C)C2)C1 c1(C(=O)OCC)cc(NC(=O)CC2CCC(C)(C)O2)ccc1N1CCCCC1 Cc1cccnc1CNCC1CCCCN1C(c1ccc(-c2ccccc2)o1)=O N1(CC(N2CC3CC2CN3C(C2CC3CCC2O3)=O)=O)CCn2nccc21 CC1C(NC(C2CCCC(F)C2)=O)CCCN1C(=O)CCC1CC(C)(C)CO1 c1(C(=O)NCCN(C(CC=C)=O)CC(C)O)cc[nH]c1-c1ccccc1 c1(C(=O)NC(CNC(C(C)SCCCC)=O)CC(C)C)cnc2scnc2c1 c1(OC)c(Cl)cc(C(=O)NC(C)CNC(C23CC=CC(C2)OC3)=O)nc1Cl c1(NC(C(CC#C)(C)NC(C2CC2C2CCCC2)=O)=O)cc(C)c(C)c(C)c1 N1(C(C2N=C(C)SC2)=O)CCC(NC(c2ccc(Cl)nc2C)=O)C12CCCC2 c1(C=O)ccccc1S(C)(=O)=O.CC(O)(C(=O)NC12CC(C1)C2)C1CC1.C CCC(C)C(=O)N1CCC(n2cc(CNC(c3csc(SC)n3)=O)nn2)C1 c1(CC(N2CC(NC(C3(SC)CCC3)=O)C(F)C2)=O)noc(C)c1C#N Cc1[nH]nc(Br)c1C(=O)NCC1CN(C(=O)C(C)N(C)C)C1 C(=O)(CC(O)C(C)C)N1C(C)(CNC(CCc2c(C)n[nH]c2C)=O)CCC1 C(=O)(CCCS(C)(=O)=O)N.c1(OCCOC)ccc(CC(=O)N(C)CC)cc1 c1(OC)ccc(C(N2CC(C)(C(=O)Nc3ccc(C#N)s3)C2)=O)cc1Br CC1(C)CN(Cc2c(O)cccc2Cl)CCC1C(F)(F)F CC(CC(=O)NCCN(c1ccc(F)cc1)C)C(F)(F)F N1(C(=O)C(N2CCCC2c2cccnc2)=O)CCSC2(CCC2)C1 C=CC(CCC)CC(=O)NC1CN(C(c2cc3cccn3cn2)=O)C2CCCC12 C(C(C(C)(C)C)Nc1cccnc1-n1cncn1)NC(N(CC=C)CC)=O c1(OC)ccc(C(N2CCOCC2)CC(Cc2ccc(Cl)cc2)CN)c2ccccc12 C12(C(=O)NCC(C)C3CC3)CC(CN(C(C3(C#N)CC4CC4C3)=O)C1)C2 C1(N2CCC(OCC#C)CC2)CCCC(N=c2ccnc(C(C)(C)C)[nH]2)C1 C1(CC(=O)NCC2CC(F)C2)NC(=O)NC1=O.N1(CC=O)CCC(O)CC1 N1(C(c2cc(CC)[nH]n2)=O)CCN(C(c2ccc(C)nc2O)=O)C(C2CCC2)C1 Cc1cc(C#N)ccc1C(=O)NCC(C1CCCC1)NC(=O)C(C)c1ccsc1 N1(C(C(COC)C)=O)CC2CC1C2C.c1(C(N(CC(=O)N)C)=O)ccoc1 c1(C=O)ccccc1.c1(OCC)cc(C(=O)NC2(C)CCC2)[nH]n1.N(C)C n1(CC)ccc2cc(CN3CCC(CC(=O)Nc4cn[nH]c4)C3)ccc12 O=S(=O)(c1cccc(C2CC2)c1)NCC(c1ccco1)CO C1(CC(N2C(C(=O)NCC3C(C)OCC3)CCC2)=O)CCC(C)(C)O1 C1(NC(C(C)N(C(=O)Cn2ccnc2C)CC)=O)C2C=CC(C2)C1CO N1(C(C2C(C=C)OCC2)=O)CCC2(CCCC2NC(=O)COC2CCC2)CC1 C1CC(C(F)F)C1.C(C(C)(C)OCC(=O)N)NC(C1(SC)CC1)=O.C Nc1c(C(N2CCN(C(C3CCCNS3(=O)=O)=O)CC2)=O)ccc(F)c1Cl Cn1nc(CNC(CC(C)(C)C)C(F)(F)F)c2c1CCC(F)(F)C2 C1(C(=O)NC2C(NC(c3cnc[nH]3)=O)CCC2)CCc2nncn2CC1 N1(C(CCC#C)=O)CCN2C(=O)C(NC(c3cnn4c(N)ccnc34)=O)CC2C1 CC(C)CC(C)CNC(=O)CO.C1CCCCC1.c1(C=O)cc(C(N)=O)co1 c1(C(=O)NC2CC2NC(C2CC(F)(F)C2)=O)ccc2ccc3ccccc3c2n1 C1(CC=C)(C(=O)NC(CNC(=O)C=CC)CC)CCOCC1 Cc1c(C(N2CCCCC2C(C)NC(=O)C2CC2)=O)sc2cccc(F)c12 Cc1oc(C)c(C(N2CC3C(CNC(c4cn(C)nc4O)=O)C3C2)=O)c1C c1(-c2scc(NC(C(CCC)O)=O)n2)ccc(OC)cc1O C(=O)(CC(C)O)NCCC.C1(C=O)CC2(CC2)CO1.C(C)(C)C.C(=O)N C1(C(=O)NCc2c(OC)cccn2)CCN(C(=O)C2(OC)CCCOC2)O1 C#Cc1cccc(C(=O)N(CCC(C)NC(=O)CC2CCSC2)C)c1F C1(C(=O)NC(c2ccoc2C)=O)CN2CCC1C2.C1(N(C)C)COCC1C=O C(CC(=O)N1CCCC(C)(NC(=O)C(C)n2cncn2)C1)(C(F)(F)F)OC C(=O)(C1=CCN(C(=O)C(C)C2CCCO2)CC1)N(CC(COC)O)C c1(C(=O)NC2(CC=C)CCN(C(=O)CC(C)(C)C)C2)cc([N+](=O)[O-])cn1C Cc1cccc(C(=O)NCC2CN(C(=O)C3=CCOC3)C(C)(C)C2)c1Br C(=O)(C(F)(F)c1cncs1)NCC(C)CN(C(=O)CCC1CCCN1C)C c1(C(N2CC3C(CNC(c4n(C)cnc4)=O)C3C2)=O)cnn2cccnc12 C(C1CCOCC1)=CC(=O)NCC1(F)CCN(C(=O)C(F)F)C1 c1(COC)nc(N2CCCC2(CNC(c2cccnc2C)=O)C)cc(Cl)n1.O C=CC(C)CC(=O)NC(C)CNC(=O)CSc1cccc(Br)c1 Cc1ccc(CNCCCCNC(=O)C(=O)Nc2cc(F)ccc2F)c(C)n1 c1(CC)nc(C)ncc1C(=O)N(C)CC1CCCCN1C(=O)C(O)CF N1(C(C2CCS(=O)(=O)C2)=O)CCC(C2CN(C(C3(C)CCCC3)=O)C2)CC1.CO C1(NC(C2CCN(C(CC)=O)C2)=O)CC2CCCC(C1)N2C(=O)CCCN(C)C Cc1ncc(Br)cc1C(=O)NC(C)(C)CNC(=O)C(C)c1ncco1 c1(CC(=O)NC(C)C=Cc2ccco2)cccnc1Cl C1N(C(c2ccc(Cl)o2)=O)CCCC1(C)C.c1(SCC)ccc(C(=O)N)cc1.C C1(C(=O)Nc2cn(CC(C)C)nc2)CCCCN(C(=O)C(CO)NC(N)=O)C1 C1CN(C(c2cccc(=O)o2)=O)CCCO1.C(C(=O)NC)(C1CCOC1)OCC C(=O)(C(O)C1CCCC1)N(C1CCCC1)CCCNC(COCCC)=O N(C1CCOc2ncccc21)C(CCc1ccc(C(=O)OCC)cc1)=O C=CCC(CNC(=O)C(C)n1cncn1)NC(c1cn(-c2ncccn2)cn1)=O Cc1nc(C)n(CC(N2CCC(CCNC(C3CC3CC(C)(C)C)=O)C2)=O)n1 C1(C(=O)NCC2C(NC(c3c(C)con3)=O)CC2)C2CCCCC12 c1(C(=O)NCC2CC(NC(C(C=CCCC)O)=O)C2)cncc2ccccc12 C1(CC(=O)NCCN(C(c2cc(C)sc2)=O)C(C)C)Cc2ccccc2NC1=O c1(C(=O)NCC2CCN(C(CN(C(=O)OC)C)=O)C2)cc2cccc(Cl)c2[nH]1 c1(C(=O)NCC(CCNC(C(CC=C)(C)O)=O)OC)cnc2cccnn12 c1(OC(C(=O)NCCNC(C2CC(CC)C2)=O)CC)cc(Cl)cc(Cl)c1 c1(CN(C2CCCN(c3cnn(C)c3)C2)C)cc(F)c(C(F)(F)F)cc1F C1(NC(C2CC(C)CN(C(C3(C)CNC(=O)N3)=O)C2)=O)C2CCN(CC2)C1C Cc1n[nH]c(=NCC(C2CCCCC2)NC(C2CC2c2ccco2)=O)o1 C1(C)(CNC(C(C)OC)=O)CN(C(=O)CCCCc2ccc(Cl)cc2)CC1C C(c1ccc(C)cc1)=C(C(N1C2C(NC(CCC#CC)=O)C(C2)C1)=O)C C1(C(C(=O)NCC2CC(NC(CN(CCC)C)=O)C2)OC)CCCCC1 Brc1ccc2[nH]c(-c3nc(C4CCCCCC4)nn3CC3CCCCO3)cc2c1 C1(CNC(c2cc(C)n(C)n2)=O)CC2CCC1N2C(=O)C(C1CCOCC1)O N1(C(CCC)=O)CCC2(CC1)CCS(=O)(=O)N2C.C(=O)(CC1CC1)N.C(N)=O CC#CCCCC(=O)NC1CCN(C(=O)CSCC(N)=O)CC1F Cc1nc(C(F)(F)F)c(C(=O)NCC2CCCCN2C(c2ncccc2Cl)=O)o1 c1(C2(C(=O)NC3C(C)N(C(C4CC45CC5)=O)CC3)CCC2)c(F)cccc1F O=C(C(Cc1ccccc1)C1CCCCC1)NC1CC(O)(c2ccccc2)C1 N1(C(C=COCC)=O)CCC2(CCCC2N2CCc3c(C(=O)OC)csc3C2)CC1 c1(OC)ccc(C(N2CC(O)(C(C)NC(=O)C(C)SC(F)(F)F)C2)=O)nc1Cl Cc1cnsc1C(=O)N.CC(C)(C)CC1CN(C(C2CN(C3CCOC3)C2)=O)C1 CC1OC(C)C(NC(C2CCCN(Cc3coc(-c4cccs4)n3)C2)=O)C1C c1(CC)nn[nH]c1C(N1CC(F)(CNC(=O)Cn2nccc2C)C1)=O C1(CNC(c2ccnc(C3CCC3)c2)=O)CN(C(C2CCCO2)=O)CCO1 c1(C(N2C(CNC(c3cccnc3)=O)CCC2)=O)ccc2cc(O)ccc2n1 c1(OC)cncc(C(=O)NC2CCOCC2NC(=O)COCC(=O)O)c1C c1(C(NCC)=O)sc(S(N)(=O)=O)cc1C.c1(C=O)ccoc1.C(=O)C.C CC1CCCN(c2nc(Br)co2)C1C c1(C=O)cc(C(C)(C)C)ccn1.C1(C(=O)OC)CC(CC(=O)NCCCO)C1 c1(C(=O)NCC2CC(C)N(C(c3c(Cl)cccc3Cl)=O)C2)c(Cl)nn(C)c1Cl C1(CNC(=O)CCc2ccccn2)COCCN(C(=O)C2=CCCS2)C1 c1(C(=O)NC23C(CN(C(C4(C)CCC(=O)NC4)=O)C2)C3)cc2cc(F)ccc2[nH]1 N1(CCOCC=C)CCC(n2cc(C(C)(C)C)nn2)CC1 c12cc(cnc1Cl)NC2=O.C1(NC(C=COCC)=O)CCCCC1C(=O)OC Cc1ccc(C(N2CCC(CCC(=O)N(C3CC(C)(CO)C3)C)CC2)=O)cc1F C(CC(CO)C(C)C)NC(C(=O)NCc1c(OCCOC)cccc1)=O C1(CNC(c2ccc(NC)c(F)c2)=O)CN(C(=O)CCC(C)SC)CC12CCC2 C1(O)(CNC(C2(CC#C)CCCO2)=O)CCN(C(=O)C)CC1.C(N)(=O)N N1(C(C(COC(C)C)N)=O)CCC(O)(C(F)(F)F)C(O)C1 N1(C(Cn2c(C)csc2=O)=O)CC(NC(=O)CCOCC(F)F)CC(C)C1 N1(C(C2C(C(C)C)C2)=O)CCC(C(C)C(=O)NCCCN2CCCCC2C)CC1 CN1CCN(C(C2CC3CC2C2CC32)=O)C(CNC(C2(O)CCCCCC2)=O)C1 c1(NCc2cc(C)oc2)nc(N2CCC(C3CC(F)(F)C3)C2)nc2c1ncn2C Cc1cc(C)c(-n2nc(Cn3cncn3)nc2-c2ccsc2)c(C)c1 c1(NC(C2CC(N(C(C(C3CCCC3)OC)=O)C)C2)=O)cn(C)nc1C C1(CC)CCN(C(C2CC2)=O)CC1.CC(COc1ccccc1)C=O.C1CC1.N c1(C(N2CCC(O)(C(=O)NCC(C)(C)O)C2)=O)cc2c(Cl)cccc2s1 C(c1cnc(C(C)(C)C)o1)=CC(=O)N.n1(CC(=O)N(C(C)C)C)cccn1 Cc1nn(C)c(=O)c(C(=O)NC(C)(C)CO)c1C.c1ncccc1C(F)(F)F C(C1CCCn2cc(C)nc21)NCc1c(F)c(OCC)c(F)c(F)c1 C1(C)(C(=O)OC)CCC(NC(c2cccnc2)C(=O)NCc2nccn2C)CC1 c1(NC(=O)NC(c2c(C)nc(COC)s2)C)ccccc1[N+](=O)[O-] N1(C(C)=O)CC(N=c2nc(N(CC(C)(C)CO)C)c3c([nH]2)CCS3)C1 C(=O)C(C)(C)S(C)(=O)=O.C1(N(C(C2C(CC)OCC2)=O)C)CCC(C)CC1 C1(C2CCC2)(C(N(CC(C)C)C)=O)CC1(F)F.C12(CC)COC(C=O)(C1)C2 CC1CC(C)(C(N2CC3CC2(CNC(C2(O)CCCCC2)=O)C3)=O)CC(C)O1 c1(C(=O)Nc2ccc(C(F)(F)F)n(CCC)c2=O)ccc2c(n1)CCNC2 N1(C(c2ccc3c(c2)C=CCCC3)=O)CCn2c(nc3c2CCCC3)C1 C1(C(=O)NC2CCCN(C(c3c(C)oc(Cl)n3)=O)CC2)OCC2CCCCC12 C(CN=C(NCC1COC(=O)N1)NCCN1CCOCC1)c1c(C)cn(C)n1 c1(C=O)cc(F)c(Cl)cc1Cl.c1(CC(=O)N(CCC)C)ccc(C(N)=O)cc1.N C1(CC)CCN(C(c2ccc(O)cc2)=O)C1C(=O)NCc1nc[nH]n1 N1(C(c2cc(C3CC3)[nH]n2)C(=O)NC2(C)CC2)CCC(O)(C2CCC2)CC1 C(C(C)(C)C(=O)N(CC(C)CNC(=O)C(O)Cc1ccccn1)C)OCC n1(CCC(=O)NCCCC2(NC(COC(CC)C)=O)CC2)ncn(C)c1=O c1(-c2c(OC)c(C)ccc2F)c[nH]c2cc(C(=O)Nc3c[nH]nc3Cl)ccc12 C(=O)(CC(O)C(C)C)NCC1(C)CC(NC(c2[nH]cc(C)c2)=O)C1 C12(C(=O)N)C(=O)C3CC1C2C3.N1(C(C2(N3CCCC3)CCC2)=O)CCCCC1 c1(C(=O)NC(CC)CNC(=O)CCC2CCC2)c[nH]c2nccc-2c1C C1CC2(CCN(C(=O)C)CC2)CO1.c1cc(C)on1.C(F)(C(=O)NC)=C(C)C c1(C(=O)NCCCC(CCC)NC(=O)C(C)(C)F)oc2ccccc2c1Cl CC(CC(C)(C)C)C(=O)NC1CC(CNC(=O)CN2CCCCCC2)CC1O Cc1ccc2c(=NCC(C)S(C)=O)[nH]c(=NCc3nc(C)c(C)o3)[nH]c2c1 c1(SC)ccsc1C(=O)N.C12CC(C1)C2.C1(C=O)CC(C(F)(F)F)CO1 c1(C(=O)NCC(CC)NC(c2cccc(C)c2F)=O)c(F)cc(O)cc1F Cc1ccc(NNC(=O)NCC2CC3(CCOC3)CO2)c(Cl)c1 C1(CCOC)(NC(C(CC=CC)C)=O)CCN(C(c2csc(=NCC)[nH]2)=O)CC1 C(=O)(C1=CC(O)CC1)NCc1n(CC)nnc1C.C1(C=O)CCCCCN1C.N c1(NCC(C)O)cc(S(=O)(=O)NC2(C)CC=CC2)ccc1C#N CC(C)(C#N)CC(=O)N1CCCC1C(C)(C)NC(=O)CC(=O)NC.C1CC1 C1CC2(CO1)CN(C(C1COC(=O)C1)=O)C2.C1(CC)CC(CC(=O)N)CCO1.C CC(CC(=O)OCCOCCOc1cn(-c2ccccc2)nn1)c1ccncc1 Cc1sc(C(=O)NCC(F)CNC(c2cc(N)cnc2Cl)=O)cc1[N+](=O)[O-] CCN=c1ccc(C(N2CC(C)N(C(=O)C=C3CCN(C)CC3)CC2C)=O)c[nH]1 C1(C(=O)NC2C(CN(C(c3nn(CC)c(O)c3)=O)C)CCC2)CN2CCC1CC2 C1(COC2C(NCC)CCCC2)CN2CCC1CC2 C(=O)(CCCN(C)N=O)NCC(c1cccc(C)c1)NC(c1c[nH]c(=N)o1)=O c1(C=O)cnc2n1CC(C)CC2.c1(COC)cc(C(=O)NCCC(O)C)no1.N CC1OC2(C)CC1(C(=O)NCCc1c(F)cncc1F)C2 c12cn(nn1)CC(C)NC(=O)CN(C)CC2.C1(SCC)CCOC1=O C(=O)(C(C#N)CCC)N(C1CC(NC(c2c(C)nc(CCC)s2)=O)C1)C C1(C)(CC)CCN(C(=O)C(C2CCN(C(C34CCC(C3)C4)=O)CC2)C)C1 C1(S(C)(=O)=O)(CN(C(c2ccccc2OC(C)C)C)CC)CC1 c1(CC)nc[nH]c1C(=O)N(C)CC1CC1.C1(C2(C(=O)N)CC2)CCCCO1 CC1(C)CC(C(=O)NCC2CCCCO2)c2ccccc2O1 c1(C(=O)NC2CC(n3cc(Cn4ncc(C)c4)nn3)C2)ccc2c(c1)CNC2=O Cc1nc2cc(C(=O)NCC34CC(C3)C4)cnc2[nH]1.C(=O)CCC1CC1C.N C1(CCC(=O)NC2CC(CC(C)(C)C)C2)CCCN1CC(C1CC=CCC1)=O c1(C(N2C(C)CCC2)=O)cc(S(N)(=O)=O)c[nH]1.C1(C=O)(N(C)C)CC1.C Cn1nnc(CNC(C2CCC3(CC3)C2)=O)c1C(N1CC2CC2C1)=O Cc1n[nH]cc1C(=O)NCC1CC1NC(C1(C(C)C)CC1)=O c1(C(=O)NC2CCN(C(CC3CC(C)C3)=O)CC2O)ccc2c(c1)CC(C)(C)O2 O=C1CC(C(N2CCC(CCNC(c3cc(O)ncn3)=O)CC2)=O)C2(CCC2)C1 Cc1cc(C(=O)NCC2CN(C(c3cccnc3F)=O)C2)n(C(F)F)n1 CC(C)(C#N)CCCC(=O)N1CC(CC(C)(C)CNC(C2(C)CC(F)C2)=O)C1 c1(C(=O)NC(C)C(C)NC(C2CCC(=O)N2C)=O)cccc(-n2nnnc2O)c1 Nc1c(C(=O)NCc2ccccc2CNC(=O)C(O)C2CCC2)cccc1F C1CC2CCCC(C1)C2.C(C)(C(=O)NC(C)C=CC(=O)N)OCCOC N1(S(c2ccc(C)cc2)(=O)=O)CCc2nc(Cl)ccc2C1 C1(C(=O)N)CCc2nncn2CC1.N1(C(C2CC(OC)C2)=O)CC2(CC2)CC1C O=C1CCCC(CC(=O)NCC#CC(N2CC=CC(O)C2)=O)C1 Cc1oc(C)c(C(=O)NCCCCCNC(=O)CCC2CC(C)(C)CO2)c1C C1(C(=O)NCc2nc(CC)sc2)CCCCC1(C)NC(c1cccc(C)c1C)=O c1(CC(=O)NCC2(CCOC)CC2)cc(OC(=O)C=NOC)ccc1Br CC(C)CC(O)C(=O)N1CCC(C(C)NC(C2C(F)(F)C23CC3)=O)CC1 C(C1=NOC2CN(C(C3(c4ccnn4C)CC3)=O)CC12)NC(c1c(C)noc1)=O c1(C(N(C2CC(C#N)C2)CC=O)=O)cncc(F)c1C.N1(CC)CCCCC1.N c1ccc(C(C)=CC(N2CC(=C(F)C)C2)=O)cc1.C1(CC=O)CCOC1.CO c1(C=O)cnn2c1N(C)CC2.C(C(=O)NC(C)CC(F)(F)F)(C(C)(C)C)SC C(=O)(C1CCCc2nc[nH]c21)NC(C(C)NC(=O)CCc1ccc(F)nc1)CO N1(C(CCSC)=O)CCC(C2CCN(C(c3cc4cc(C)ccc4s3)=O)CC2)C1 Cc1nc(CO)ncc1C(=O)NC1(CF)CCN(C(=O)CC2CSCCS2)C1 N1(C(CC(C=C)(C)O)=O)CC2(CCCC2NC(c2ccccc2)=O)C1.C(N)=O.N c1(C=O)c[nH]c(C#N)c1.C1(C#N)(CN(C(=O)CCc2ccco2)C)CCC1.N Cc1cccc(C(C#N)C(C2CCN(c3cc(C)[nH]n3)CC2)=O)n1 C1(C(=O)N)(COC)CC(F)(F)C1.c1(C(C=O)(C)C)cccnc1F.C1CC1 c1(C(N2CCC(N(C(c3sccc3)=O)C)C2)=O)cccc(F)c1C(F)(F)F.CO C1(O)(CNC(C(CC=C)(C)C)=O)CC2CCC(C1)N2C(c1csc2nnsc12)=O CC(C(F)C(=O)N1CCCC(NC(=O)CC2C=CS(=O)(=O)C2)C1)C(F)(F)F C1(C(C)NC(C=NOC)=O)CCCN(C(c2ccc(OC(C)(C)C)cc2)=O)C1 CCS(=O)(=O)CC=CCNC(=O)C(=O)NC1COC(C(C)C)C1 C#CCC(CC(F)F)C(=O)NC1CC(C(=O)NCCOCC(C)C)C1(C)C N1(C(C2(CC(C)C)CCC2)=O)CCCC(C(C)C(=O)NCc2cccnn2)C1 C1(C=O)CC(=O)NC1(C)C.CC(C)C(C=O)NC(c1ccco1)=O.C1CC1.N C12CC3CCC(C1C2)N3C(C1CCS1(=O)=O)=O.c1(CC(=O)N)c(F)cccc1Cl CC(F)(CNC(=O)COCCC1CCCC1)CNC(C1CC=CCC1)=O c1(C(=O)NCC(C)CN(C)C(c2ccccc2C(F)F)=O)ccc2ccnn2c1 C1(=C(C=O)F)CCN(S(=O)(=O)C(F)(F)F)CC1.CCCN(C)CC.CC.O N1(C(CS(CC)=O)=O)CCCN(C(=O)C(C(C)(C)C)C2CCC2)C(C)C1 C1(NC(C(n2c(C)ccn2)C)=O)CCCC12CN(C(=O)CCC=O)C2.C(C)(C)C.O c1(C(N2CC(CC)C(C(N3CC=CC3COC)=O)C2)=O)c[nH]c(C)cc1=O N1(C(CC(c2c(C)cccc2)C)=O)CCC(O)C(C)(O)C1 C=CC1(NC(C2CCC(C)N2C(=O)CC2CCCNC2=O)=O)CCOCC1 C1(NC(=O)Cn2cccc2)CCN(C(c2ccc(CC3CC3)s2)=O)C1 C1(NC(c2cnnc(O)c2)=O)CN(C(c2cc(O)cc(O)c2)=O)CC1(F)F C1(NC(=O)NC2(CC=C)CC=CC2)CCCC(N(C)C)C1 C(CC(=O)NNc1cccc(Br)c1)N1CCC(C(=O)OCC)CC1 N1(C(c2cc(C(=O)OC)sc2)=O)CCCC2(CCCNC2=O)C1 c1(C(N2CC(CC)C(NC(=O)COCCC)C2)=O)ccc2c(c1)CCOC2.O N1(C(C(C)OCC#C)=O)CC2CC1CN(C(c1c(C)cc[nH]c1=N)=O)C2 C#Cc1cnc(C(=O)NC2COC3(C2)CN(C(=O)CSC(F)(F)F)C3)c(C)c1 Cc1ccc2c(c1C(=O)NCC1CC(NC(C3SCCC3C)=O)C1)CCCN2 C=C1CC2CC1CN2C(c1ccoc1CNC(=O)C(c1ccc(C)o1)C)=O C1(OC)CC2(C1)CC(C(=O)N)C2.C(C)(C)CCC.C12(C=O)CC(F)(C1)C2 C(=O)(C1=C(C#N)CCC1)NC(CNC(C=Cc1c(C)coc1C)=O)C1CC1 c1(CC)cccc(C(=O)NC2CC3(C2)CC3NC(c2cnc(Cl)s2)=O)c1F C1(CNC(CC)=O)CN(C(c2ccc(C(C)(F)F)cn2)=O)C2(CCC2)C1 C1(NC(=O)CC2COCCN2C(C2CC2(F)F)=O)CCCC2(CC1)CC2 N1(C(c2c(C)coc2C)=O)C2CCC(C2)C1CNC(c1nnc(O)cc1O)=O N1(C(c2c(C)n(C)nn2)=O)CC(NC(=O)C=CCF)CC(O)C1 N1(C(CC(=O)OC)=O)CC2CCC(C1)C2NC(=O)CCN1CCCC1 C1(C(N2CCC(N(C(=O)Cn3nccn3)C)C2)=O)C(C2CC2)C1(F)F C#Cc1ccc(C(=O)NCCO)nc1.C1(N(CC(=O)N(CC)C)C)CCSC1 CN1CCN(c2nc(C3CC3)nc(=N)[nH]2)CC1CNC(=O)CN=S(C)(C)=O N1(C(Cc2ncn(C)c2)=O)CC2CC(NC(C3CCC(=O)NC3)=O)C(C2)C1 c1(C(N2CC(C(C)NC(=O)C3=CCCOC3)C2)=O)cc(Cl)c([N+](=O)[O-])[nH]1 CC(C)CCC(C(=O)N1CC(CC(F)(F)F)C1)NC(=O)CC(=O)NC.C1CC1 c1(CC(=O)NCC(CN(C(C(COCC)C)=O)C)(C)C)ccc(OC)nc1 c1(C(=O)NCC2CCCN2C(c2ccc(C3CC3)s2)=O)ccnc(Cl)c1 C1(C(N(CCC(=O)NC(C23CC(CO2)C3)C)C(C)C)=O)CCC=CCCC1 N1(C(C2CCN(C(C(N3CC(C)C3)C)=O)CC2)=O)CCS(=O)(=O)CC1 c1(CCC(=O)NCC2(CC)CC2)ccc(F)cc1Cl.C1(C=O)CC2(CSC2)C1 C1(C(=O)NCCSCCC=C)CCN(C(=O)c2cccc(F)c2)O1 C1(NC(c2cc(OCC)n[nH]2)=O)(C)CCCCC1C.C1(C=O)CC(F)(F)C1 N1(C(C(C(C)C)F)=O)CCN(C(C2CC3C=CCC(C2)C3)=O)CCC1C C1(C(=O)NCCCC=CC)CCCCN(C(c2[nH]ccc2C2CC2)=O)C1 C1(C=O)CC(CC)=NO1.C1(C(=O)OCC)(C(=O)NCC(O)C)CC1C.N N(C1CCCc2cn(C3CCCC3)nc21)C(N1CC(O)CC2(CCCC2)C1)=O Cc1ncc(C(N2CC(OCC(=O)NCC3COCC3O)C2)=O)o1 N1(C(C2C(C)C2)=O)CCC2(CC1)CC(NC(=O)C(c1ccc(Cl)cc1F)O)C2 c1(N2CC(O)(C(C)NC(C(C3CCCC3)OC)=O)C2)ncnc2[nH]cnc12 N1(C(c2cc(CNC(C(C)S(N)(=O)=O)=O)sc2)=O)CCc2nn(C)cc2C1 C1(C#N)(SC)CN(C(=O)C(Cc2ccoc2)NC(=O)C(C)CC2CCC2)C1 N1(C(C2CC(C)(C)OC2(C)C)=O)CCN(C(C2CC23CC3)=O)C2(CCCC2)C1=O c1(OC)ccn2cc(C(=O)NCCC3CN(C(=O)CCc4nccs4)C3)nc2c1 c1(OC)cc(NC(C)(C)CNC(c2cc(CN(C)C)c[nH]2)=O)ncn1 Cc1cc(C(N2CCC(NC(=O)CC3CCC3)C(C)C2)=O)c(F)c(Br)c1 N1(C(c2cn(CC=C)nn2)=O)CCOC(C(C)NC(=O)Cc2conc2C)C1 N1(C(C(CC#C)C)=O)C2CCC1CC(O)(CNC(c1cnn3c1CCC3)=O)C2 C(CN(C)C)(CC(C)C)NC(CCN(CCC)C(c1sc(O)nc1C)=O)=O c1(C(=O)NCC(CN(C(C(CCC)C)=O)CC)(C)C)cccc([N+](=O)[O-])c1.O C1(CNC(C(C(COC)C)C)=O)CC2CCC(C1)N2C(c1[nH]ccc1C)=O N(C(=NCCCOCC)NCc1cccc(Cl)n1)C(C=C)C C1(C(N(CCN(C(C)C)C(C2CN(C)CCO2)=O)C)=O)CCc2cn(C)nc2C1 C(=O)(CCCN(C)N=O)N1CCCC(CN(C)C(C23CC(C)(C2)C3)=O)C1 C1(C2CN(C(=O)C(O)C3CCC3)C2)(NC(=O)CSc2nnc(S)s2)CC1 N1(C(CCOC)=O)CCOC2(CCCN(C(c3ccc(C)c(C(C)=O)c3)=O)C2)C1 N1(C(c2nc(CCC)oc2)=O)CC=CC(C(=O)NCCN(C)OC)C1 Cc1ccc(C)c(C(=O)NC(C)CNC(c2sc(-c3ccccn3)nc2C)=O)n1 C1(N(C(C2CCN2)=O)CC23N(C)CC(C2)C3)CCCN(Cc2ccccc2)CC1 c1(OC)ccccc1CC(C)(C)CNC(N1CCC(c2cc(=N)[nH][nH]2)CC1)=O c1(OCC#C)ccc(C(=O)NC2CN(C(=O)CP(C)(C)=O)CC2O)cc1 c1(SC(C)C)ccc(C(N2CCC(O)C2)=O)cc1.c1(C=O)cscc1C1CC1.N c1(C(C)OC)nc(C)cs1.C1(CC=O)CCN(C(=O)CN(C)C(C)=O)C1 CCC(C)(C)CC(=O)N1CCC(C(C)(C)C)(CN(C(=O)C(C)c2ccsc2)C)C1 C1(OC)(CNC(=O)C(c2ccnn2C)O)CCN(C(=O)C(F)=C(C)C)C1 CC1(C)CC(CNC(=O)Cn2cncn2)CN1C(c1csc(Br)c1)=O C(=O)(CCCOCCO)NCCCOC(C)C.c1(C(=O)N)cc(F)n(C)n1 N1(C(c2c(C)cc(C)[nH]2)=O)CCC2(CCC2NC(=O)CN2CC3CC3C2)CC1 C12(NC(C3C(=C)C3)=O)CCC(C)(CC1)OC2.C1(C=O)CCNCC1.C1CC1 C1(C)(C(N2CCC2)=O)CCC(=O)NC1.C(=O)(CC(C)N(C(=O)CO)C)OC N1(C(C2N(CC)CCC2)=O)CCCC(O)(CN(C(=O)C(=O)N(C)C)C)C1 C(=O)C1CCCc2scnc21.c1(C2(c3cn(C(C)N)nn3)CC2)cc(Br)ccc1F c1(C(=O)OC)ccc(Cl)c(C(N2CCC(NC(c3cnn(C)n3)=O)CC2C)=O)c1 C1(F)(C(=O)NC(C)CCN(C)C(c2cn(CCO)nn2)=O)CCCCC1 O=C(CC(O)C(Cl)(Cl)Cl)NCC#CCNC(c1c[nH]nc1C(F)F)=O C1(C(N(CCCNC(CC=C=C)=O)Cc2ccccc2)=O)CC2CCC(C1)C2O Cc1ccc2cc(C(=O)NC3CN(C(=O)COC(C)(C)C)CC3C)cnc2c1 c1(NC(c2n(CC)nnn2)c2cnc(C(C)(C)C)[nH]2)cc(Br)cnc1C c1(OC)c(C(=O)NCC2CCCC2NC(=O)CC2=CCCC2)cccc1Cl CC(CC(=O)NCCC1CCCN(C(=O)Cc2cnsc2)CC1)C(F)(F)F CCCCCCCCC(F)C(=O)NC1(c2nn[nH]n2)CC12CCC2 C1(NC(=O)CCc2ccncc2Br)CCN(C(C2(CO)CCC2)=O)CC1F C1(C=O)CCC2(CC1)CC(N(C)C)C2.C(C)(C(C)C(C)C)NC(COC)=O.N N#Cc1cc(S(=O)(=O)NC2CCCn3ccnc32)ccc1NCC1CCCC1 c1(C(N(C2CCCN(C(c3ccnc(C4CC4)n3)=O)C2)C)=O)cn2ccsc2n1 c1(CCOC)n[nH]c(=NC(C)CCNC(C2(C)CNC(=O)C2)=O)s1 C12(C(=O)OC)CC(CNC(=O)Nc3ccc(C#N)cc3Cl)(C1)OC2(C)C C1(NC(C(CC)SC)=O)CCN(C(=O)COCc2ccccc2)C1C C1(NC(=O)C2=C(Cl)CCC2)CCCN(C(c2cc3n(n2)CCCC3)=O)CC1F c1(OC)ccc(N)c(C(=O)NC)c1.C1CCN(C(c2nc(C)c(C)s2)=O)CC1O Cc1csc(C(=O)NC2CCCC2C(N2CCOC3CC23)=O)c1Cl c1(CCCCC)nc(C(=O)NC(C2(O)CN(C(c3n[nH]cc3Cl)=O)C2)C)cs1 N1(C(CS(CC)(=O)=O)=O)CC2CC(NC(c3c[nH]cc(F)c3=O)=O)CC1C2 C1(NC(C2CN(C(C)C)C(=O)C2)=O)CCCCN(C(c2cnc(S)n2C)=O)C1 C1(NC(C(=Cc2cnc[nH]2)C)=O)CCCC12CN(c1cc(Cl)nc(C(C)C)n1)C2 CCCC(C)(C)CC(=O)NC1C2CCN(C(=O)CC(C)C3CCCC3)CC12 C1(NC(c2nccc(OC)c2)=O)C2CCC(C2)C1C(=O)NC(C)CC(C)C c1(NC(C2N(C(c3cc(C)[nH]c3)=O)CCC2)=O)ccc2nn[nH]c2c1 c1(C(N2C3CN(Cc4ccc(O)cc4)CC23)=O)cc(Cl)cc(Cl)c1O C12(C(NC)=O)C3CC(CC13)C2(F)F.N1(C(CNC(CCC)=O)=O)CCOCC1.C CCCC(O)CC(=O)NCCCCC(CO)NC(c1n[nH]c2c1COC2)=O N1(C(=O)Cc2cncc(F)c2)CC2CCC1CN2C(c1coc2ccccc12)=O C=C(C)CCCC(=O)NCCC1CCCN1C(C1CCCN(C)C1)=O c1(OCC)ccc([N+](=O)[O-])cc1NC(=O)CC1CCC(O)C1 c1(C(=O)NCC23C(CN(C(c4cccc(C)c4)=O)C2)C3)occ2c1CCOC2 c1(-c2nc(C3(O)CCCNC3)on2)cccc2cnccc12 N1(C(c2[nH]cc(C)c2)=O)CCC2(CCC(CNC(=O)CCCC(F)(F)F)O2)CC1 C12(CNC(c3cnc(C)s3)=O)CCC1CN(C(=O)CC(F)(F)c1ccccc1)C2 N1(C(CC(C(C)C)C)=O)CC2CC(C1)N(C(C1CC(C)(C)CCO1)=O)C2 N1(C(C2(C)CC(C#N)C2)=O)CCC(NC(c2cc(F)cs2)=O)C(O)C1 c1(C(=O)NCC=O)ccccc1-c1ccccc1.C(CCOCCN)N(C)C C1(CCNC(c2ccc(F)o2)=O)COCCN1C(c1ccc(C2CC2)o1)=O c1(CC)nncn1NC(=O)C1C=CCN(C(C2CC23CCCC3)=O)C1 CN1CC2(C)CN(c3nnnn3C3CCSC3)CC2(C)C1 C1(C(F)(F)F)(C=O)CCCC1.c1(C(=O)NC2CCC2)cc(C2CC2)cs1.N C1(NC(C(C2CCCC2)OC)=O)C(C)CCN(C(c2ncsc2C)=O)C1C c1(C(N(C2CCCCC2)CCC(=O)OC)=O)cccnc1C(=O)NC1CNC1 C1(NC(c2c(C)noc2)=O)CCC2CCN(C(c3csc(F)c3)=O)C1C2 CC(C)C(C)(CNC(=O)COc1cccc(Br)c1)NC(c1cocn1)=O C1(CC(=O)NC(COCC)C)CN(C(=O)Cc2cncnc2O)CCO1 N1(C(c2cnc(CC)s2)=O)CC2(CCC2)CC1CNC(c1cnc(C)[nH]1)=O c1(NC(=O)NCC(C(=O)OC)(F)C(C)C)ncc([N+](=O)[O-])cc1F Cc1cccc(C2(C(=O)NCC3CCC3N)CC2(F)F)c1 C1(C(N2CCC(N(C(c3cnccc3C)=O)CC)C2)=O)Cc2ccccc2N1C C1(c2nnnn2CC)(NC2(CSC)CC2)CCCC(OCC)C1 CC(C)CC(F)C(=O)N1CC(O)(CNC(c2ccccc2)=O)C1.N1(C)CCCC1 Cc1cc(C)c(C(=O)CN2CCCC(C(=O)O)C[N+](=O)C2)c(C)c1C Cc1nnc2n1CC(C(N1CCC(NC(c3cnc(O)n3C)=O)CC1C)=O)CC2 c1(C(N2C(C)CC(NC(CCC=C)=O)C2)=O)cc(S(N)(=O)=O)ccc1C N1(C(C(c2ccc(Cl)s2)C)=O)CC2(CC2)CC1CNC(c1ncc(F)cc1F)=O N1(C(C(c2c(OC)cccc2)O)=O)CC2CCN(C(c3coc(C)c3)=O)CC2C1 n1(CC)ccc(C(N2CCC2CNC(C2(C)CCCC2C)=O)=O)cc1=O c1(OC)c(Cl)nc[nH]c1=NCCCC(C)NC(C1(C)CCCOC1)=O N1(C(=O)OC(C)(C)C)CC(C)(C)C1c1cn(C2CCCC2(C)O)nn1 c1(C(N(CC(CNC(C=C2CCC(C)C2)=O)O)C)=O)cc(P(C)(C)=O)cs1 c1(C(=O)NC2CN(C(CCS(C)=O)=O)CC2C(F)F)ccc(Br)c(N)n1 N1(C(C(C)OCCCC)=O)CC(CNC(=O)CNC(=O)CCC)C(O)C1 C(c1ccc2ncccc2c1)=CC(N1CC(C(C)NC(c2ccncc2)=O)C1)=O Cc1cn2c(C(N3CCC(=CCNC(=O)CCC4CCCC4)CC3)=O)cnc2s1 n1(C(C)C)ccnc1C(=O)NCC.c1(C=O)cnc(C(F)F)s1.C(C)(C)C C(CN=c1cc(NCc2ccnc(Cl)c2)nc[nH]1)c1ccc(Cl)nc1 S(=O)(=O)(c1cnc(N(C)CCC2CCCCC2)c(Cl)c1)N1C(C)CC(F)(F)CC1 C1(C(=O)NCCOCC(N2CCC(CCO)C2)=O)CCN(C2COC2)C1 C1(CNC(CCC(C)OCC)=O)CCN(C(c2c[nH]nc2C2CC2)=O)CC1C C(=O)(C1CCOc2ccc(F)cc21)N1CC2(CN(C(C(C)(C)F)=O)C2)C1 C(=O)(C=CS(C)=O)NCC1(CNC(c2ncn(C)c2)=O)CCCC1 CC#CCCC(=O)NC(C1CC(NC(c2ncn(C)c2C)=O)C1)C C1(NC(C2(CC)CCCO2)=O)CC2CN(C(c3cccc(O)c3)=O)CC12 C12(NC(CCS(C)(=O)=O)=O)CCCCC1N(C(c1cc(F)cc(F)c1N)=O)CC2 N1(C(CC(CCC)(C)O)=O)CC2OCCN(C(=O)CNC(=O)CN(C)C)C2C1 c1(C(N2CC3C(C3)C2)=O)cnc(C)c(CC(C)C)c1.CCC(C(=O)NC)N(C)C C1(C(N2CC(NC(c3c(OC)csc3)=O)C2)=O)CCN(C(N)=O)CC1 N1(C(Cn2ccc(C)c2)=O)CC2(CC(C(=O)NC(c3cnn(C)c3)C)CO2)C1 c1(C(N2CCCC(N(C(CC)=O)C)C2)=O)c(P(C)(C)=O)cnn1Cc1ccccc1 n1(COC)nccc1C(=O)N(CC(O)CNC(=O)CCC1CCCO1)C CC1C(NC(c2ccc(C(F)(F)CF)cc2)=O)CCCN1C(c1cnsn1)=O N1(C(CC2CC(=O)OC2)=O)CCCC2(NC(C3CC34CCCC4)=O)CC2C1 C1(NC(C(c2cccnc2)NC(CC=C=C)=O)=O)CCC(C)(C)C1 O=C(C(O)C(F)F)NCCC1CCN(C(=O)C(c2ccc(Cl)cc2)O)CC1 C1(C(C)O)COCCN1C(c1cccc(C(C)(C)NC(=O)O)c1)=O.C(C)(C)C N1(C(=O)Cc2ccns2)CC2CCC(CNC(C3(C4CC4)CC3)=O)C2C1 C1(C(=O)N)CC(C)(C)CC(C)(C)C1.N1(C(CN(CCC#C)C)=O)CCCC(F)C1 N1(CC(=O)NC(C2N(C(c3n[nH]c(C)c3F)=O)CCC2)C)C(=O)CN(C)C1=O C1(C(C(N)=O)O)CCN(C(=O)CN2CCCOCC2)CC1 CC1CCCC(N(C(=O)CCn2cc(-c3ccsc3)nn2)C)C1C c1(NC(c2cnc(Cl)s2)C)ncc(C(=O)N(C)C)s1 N1(C(CNC(CC(C)C)=O)=O)CCC2(CC1)CC2NC(c1cnn(C)c1)=O Cc1nc(C)n(CCC(=O)NC2CCCC(NC(=O)C)C2)n1.C(=O)C(C)(C)C Cn1ncc(NC(C2CCNC(=O)C2)=O)c1-c1cn(C2CCCCC2)nn1 CCCCCC(O)CC(=O)N1CCN(C(=O)C(CO)OC)CC1C(C)C c1(C(=O)NC(C)CCN(C(=O)CN2CCSCC2)C)ncccc1F c1(CC(N2C(C)CN(C(C3(C)CC3(F)Cl)=O)CC2)=O)c(F)c(F)c(F)c(F)c1F c1(C(=O)NC2CC3CN(C(c4c(F)ccc(N)c4)=O)C2C3)ccc2ccnn2c1 C=CC(CCC)CC(=O)NC1CCC1CNC(C1(N(C)C)CCCSC1)=O CCC1=NOC(C(=O)NC2CC(NC(c3sccc3C3CC3)=O)C(O)C2)C1 C(CCCC(=O)NC(C)(C)CC)OCC.c1(CC=O)scnc1-c1cccs1.N CC1(C)CCCC(Cc2nnc(N3CC[Si](C)(C)CC3)n2CC2CC2)C1 C(=O)(C(C(C)O)Nc1ccc(C(C)C)nc1)NC(CC)C N1(C(c2cc(C(C)C)n(C)n2)=O)CCN(C(C2CCCC23CCC3)=O)C(CF)C1 c1(N(C)Cc2nnc(CO)s2)nc(N2CCC(C3CCC3)C2)nc2sccc12 C(=O)(CCC(F)(F)F)NC1C=CCC(C(N(CCCOC)C)=O)C1 C1(C(N(CCOC)CCNC(=O)CC(C)O)=O)CCC(C)NC1=O N1(C(c2cccc(C#C)c2)=O)CCC2(CCCC2NC(c2cc(O)no2)=O)C1 CN1CC=C(CC(=O)NCCC2CCC(NC(c3ccncc3Cl)=O)C2)CC1 N1(C(c2nc(=NC)[nH]c(C)c2)=O)CC2(CCCCN(C(C3C4COCC34)=O)C2)C1 c1(SC)ccccc1CC(N1CCN(C(c2cc(Cl)no2)=O)CC1)=O C1(NC(C(CCCCC)O)=O)CCOC12CCN(C(c1nnn(C)c1C)=O)CC2 CC(CC(N)=O)C(=O)NCC1CC(C)(C)CN1C(=O)Cc1ccncc1Cl C1(NC(=O)NCCC(C)OC)CN(C)CC1C CCC(CC(=O)N1CCCC2(NC(C3CC(=O)N(C)C3)=O)CC2C1)C(C)C c1(CCN(C(C)C2CC2)C(c2ccc(COCC(C)N)o2)=O)ccccc1 c1(C(N2CCC(NC(C(CC(C)C)OC)=O)CC2C)=O)cc2n(c1)CCCC2 C12(NC(Cc3n[nH]c(=NC)s3)=O)CCCC1CN(C(=O)Cc1nocc1C)C2 c1(OC)ncc(Cl)cc1C(=O)NC1CCN(C(=O)C(C)Cc2cnn(C)c2)C1C C1(O)(CC(N2CCC(CC(=O)N(C3CC3)CC)C2)=O)CCNCC1 c1(C(C2CCC2)NC(C(C)OC)C)ccc(Br)cc1 C1(c2cc(CC=C)no2)CCN(S(=O)(=O)Cc2cnn(C)c2F)CC1 c1cnn2cccc2c1Cl.C(CCCCCC1CCC1)CC(N)=O N1(C(C(=O)NCC2N(C(CN(C(C)C)C)=O)CC2)C)CCOC1=O N1(C2CN(Cc3cn(C(C)C)nn3)C2)CC(NC(c2ncn(C)n2)=O)CC1=O C#CCCCC(C)C(=O)NC1CCOCC1C(=O)N(CC(C)C)C(C)C C=CCC(C)(C)C(=O)NC1CCN(C(C2(C)CC2)=O)CC1 C=C=CCCC(=O)NCCCN(C(C1CCOC1C1CC1)=O)CC C12(C(=O)N)CCN(CC1)S(=O)(=O)C2.N1(C(C(C)O)=O)CCC(c2ccccc2)C1 CC1=NOC2(C1)CC(C(=O)N(CC(C)O)CC)C2.c1(C=O)cncc(C)c1C.N C1(F)CC2CCC(C1)N2C(=O)CCc1cnco1.C(CCC)(C(=O)N)=CCC.C C=CC(CCC)CC(=O)NCCN(C(=O)C(O)C(C)CC)C1CCCCCC1 c1(CC=O)cc2ccccc2s1.C1(CC)CCC(C(=O)NC(C)(C)C2CC2)O1 c1(C(N(CC)CC2CCN(C)C2)=O)ccncc1I C(=O)(C(C)CC(C)CC(C)C)NC(C1CC(NC(CN(CC)CC)=O)C1)C c1(CC)ncccc1C(N1CCCC(CNC(c2cc(OC)cs2)=O)C1)=O N1(C(c2ccc(C(C)(F)F)nc2)=O)CC(C2CN(C(C3CCC4(CC4)C3)=O)C2)C1 N1(C(c2c(C)cccc2)=O)C2CCC1CC(N(C(=O)CCc1c[nH]c(=N)[nH]1)C)C2 Cc1ccc(C(=O)NC2CCCCC2)c(C)c1.C1(C=O)C2CS(=O)(=O)CC12.C N1(C(C2CCCC(=O)N2)=O)CCCC(CNC(c2nccnc2Cl)=O)CC1 Clc1cccc(Cl)c1-c1nc(N(C2CCCC23CCC3)c2ccccc2)n[nH]1 c1(OC)nc(C(=O)NCC(C)CNC(=O)CCCn2c(C)csc2=O)ncc1F Cc1ccc(C(=O)NCc2ccccc2)cc1Cl.C(=O)CC1(C(F)F)CC1.C C1(CNC(=O)C(O)Cn2cncn2)CCC(C(N2CC3(CCC3)C2)=O)CC1 N1(C(CC(=C)C)=O)CC(NC(=O)CCC(=O)N2CCN(CCOC)CC2)C(F)C1 N1(C(CC(CC(C)C)O)=O)CC(C)CN(C(C2CC2CC(C)(C)C)=O)CC1C N1(C(c2cncc(C(C)=O)c2)=O)C2CCC1C(CNC(C1C=CCC1)=O)C2 CC(O)CCC(=O)N1CCCC(c2cn(Cc3ccc(Cl)nc3)nn2)C1 C(=O)(C1=CC(O)CCC1)N1CC(c2ccccc2)(NC(C2CCN(C)CC2)=O)C1 c1(CN(C(C(C2CN(C(=O)C(C)OC3CCCC3)C2)OC)=O)C)nccn1C C(c1ccc(F)cn1)=Cc1cn(CC=C)nc1.C12(CCC(=O)NC1)CN2 CC1(CS(C)(=O)=O)CCN(C(=O)OC2(C)CCOC2C2CC2)CC1 N1(C(C(C)SCC)=O)CCC2CCN(C(=O)C=C3CN4CCC3CC4)C2C1 N1(C(C(C)OC2CCCC2)=O)CC2CCN(C(c3cnc(N)c(N)c3)=O)CC12 Cc1noc(Cl)c1CCC(=O)NCC1CN(C(=O)CC2CCC2)C2CC12 N1(C(C2CCC(C(F)F)C2)=O)CCC2(CCCN2C(=O)Cc2ccccc2Cl)C1 c1(NC(CC(C)NC(c2cc(C)cc(F)c2)=O)=O)cnc(C)c(C#N)c1 N1(C(CCOCC#C)=O)CCC2CN(C(C3CC3C3CC3)=O)CC12 N1(C(CC(C)(C)CNC(C2CCNC(=O)C2)=O)=O)CC2CCC1C(O)C2O C1(C(N2CCC(=CC)CC2)=O)CCCCC(C)(C)C1.C1(CC#C)(C(=O)N)CC1 C1(C2CC2)CC12CCC(O)CC2.CN1CCCCC1c1cnn(C)c1.C(=O)NCC C1(NC(c2n(CCC)ncc2)=O)CN(C(=O)C(C)CCOC)CC12CCCC2 c1(CN(C(C(C)n2cncn2)=O)C2CN(CC#N)C2)ccc(C2CC2)cc1 c1(C(=O)N)c[nH]c2cc(Br)ccc12.C#Cc1cn(C)nc1C(=O)NC1(C)CC1 Cc1cnc(C(=O)NC2C3CC4C(C3)C24C(=O)NC2CCN(C)C2)c[n+]1[O-] CCCCCC(C)CC(=O)NC1CC=C(C(=O)N2CC([N+](=O)[O-])C2)C1 c1(CCC)cc(C(=O)NC2(C(N3CC(COC)(SC)C3)=O)CC2C)ccn1 c1ccc(C#N)cc1.CN=C(NCCNC(=O)OC(C)(C)C)NC1CCC1 C1(CNC(C2C(C(C)C)OCC2)=O)CCC(C)CC1.c1(C=O)ccc(C#N)o1 c1(C(N2CCC(O)(CNC(C(C)(CO)OC)=O)CC2)=O)cc2c([nH]1)CCCC2 c1(NC(CNC(CNC(CN2CCN(C)CC2)=O)=O)=O)cnc2ccccc2c1 c1(C(=O)NCCCC(C)NC(C2(C#N)CCSCC2)=O)ccc(CO)c(Cl)c1 C(=O)(C1CCCc2ncnn21)N1C2C(NC(c3cccc4[nH]ncc34)=O)C(C2)C1 C1(NC(C(c2c(Cl)cccc2Cl)C)=O)CCN(C(C23CC(CCO2)C3)=O)CC1O CC(F)C.O=C(CNC(=O)NC1CC1)N.C1(C(F)(F)F)(C=O)CC1 C1(C(N2CC(N(C(=O)Cc3cccnc3)C)C2)=O)C2CCC1(C)C2(C)C Cc1cc2c(C(=O)NCC3COCC3NC(=O)C(Cl)=CCl)cccc2o1 C1(O)(CNC(c2ccoc2)=O)CCCN(C(=O)Cn2ncnn2)CC1 C1(C)CC(F)(F)CN1C(c1cccc(C)n1)=O.C#CCCCOCC(=O)NC C1(CNC(CSC)=O)CCN(C(c2cccc(C(F)(F)F)c2O)=O)C12CC2 c1(C(=O)NCC(CC(C)C)NC(c2ccc(C)cc2C)=O)cc2ncccc2s1 C(CC(C)(C)C)(C(=O)NC(c1cn(C)nn1)C=O)OC.N1(CC)CCCC1=O.N Cc1cc(NC(C2CC2)=O)sc1C(=O)N(C1CCO1)C(C)C.C(C)C.O c1(OC(C)C)cnccc1C(=O)NC1CC(F)(C)C1.c1(C=O)cscc1F.N CC(C)(CCCC(=O)NC1CC(CO)(CO)C1)NC(c1cc(O)cc(F)c1)=O Nc1ccc([N+](=O)[O-])c(C(=O)NC2CC(O)(C)C2)c1.C1(CC=O)CCCC1O C1(C)(C(N(CC(O)CNC(C2(c3ncco3)CC2)=O)C)=O)CCCN1C CCS(=O)(=O)c1cccc(C)c1.C1(CC=O)CC2CC1CN2C(=O)CC1CC1 N1(C(=O)CCCN2CCCC2)CC2CCN(C(c3cccnn3)=O)C2C1 Cc1c[nH]c(C#N)nc1=NCCCNC(c1csc(Cl)c1Cl)=O C1(CNC(c2c(CC)scn2)=O)CCCCN1C(c1cccnc1N)=O N1(C(C(c2ccccc2)SC)=O)CCC(CNC(C2CCCCC2)=O)C1 N1(C(C(COC)OC)=O)CC(N(C(=O)Cn2cnc(Br)c2)C)C(C)(C)C1 c1ccc(C)cc1.C(C(F)C(=O)N(CC(C)NC(=O)CS)C)N(CC)CC c1(OC)ccc(CC(=O)NC2CN(C(=O)Cc3csc(C)n3)CC2F)nc1 C1(C(=O)NC2C(C(=O)NC(CC=C)C(=O)OC)OCC2)CC2(C1)CC(C)C2 c1(NC(C2N(c3nc(C)nc4c3scc4)CCC2)=O)cccc2c1CN(C)C2=O C(=O)(CCCCCNC(=O)C(c1cnn(C)c1)O)N(C(C)CC(F)(F)F)C Cn1cc2c(n1)CC(C(=O)NCC1(C)CC1)CC2.C1(C=O)CC2COCC2C1 c1(C(=O)OC)cc(C#N)cnc1N(CC(C)NC(c1scnc1Cl)=O)C Cc1cc(C(=O)N(C)CC2CCCN2C(c2cnn(C)c2F)=O)nc(N(C)C)n1 c1(NC(C2CC3CC3N2C(c2cnc3ncccn23)=O)=O)ccc2ncnn2c1 N1(C(C2C(C)C2C)=O)CC(NC(=O)CCCn2ccccc2=O)CC(C)(C)C1 N1(C(C(CC)C2CCOCC2)=O)CCCCCC(NC(=O)C=NOC)C1 Cc1nc2ccccc2c(C)c1C(=O)NCCN1C(C)CCCC1C C1(C(=O)N(C2CCCCC2)CCO)CN(Cc2ccc(O)cn2)CCC1O O=[N+]([O-])c1ccc(CN2CC(Nc3ncnc4c(Br)cccc34)C2)c([N+](=O)[O-])c1 N1(C(c2csc(CCc3ccccc3)n2)C(=O)NCCCC)CCCC(CO)C1 N1(CC)CCC(C(=O)NC2CCCC(C(N3CC(F)(F)C3C3CC3)=O)C2)CC1 CCC(F)C(=O)N(C1CCN(C(=O)CC2(CO)CC2)C1)C c1(C(CSC(C(=O)OCCC)C)(C)NC(N)=O)ccccc1 N1(C(c2c(C)cn(C(C)C)n2)=O)CCC2(C)C(C1)C2(Br)Br CCCC(C#N)C(=O)NC1CN(C(=O)CCP(C)(C)=O)C(CC)(CC)C1 C1(C(N2CC(CC=C)(C(=O)N(CCCO)CC)C2)=O)CC12CCOC2 C(=O)(C(O)CNC(=O)CN1CSCC1=O)NCC1CC(CN=[N+]=[N-])C1 CC1CC(=O)NC(CNC(C2CCCC2)=O)C1.C1(C)(CC=O)CCOCC1.C O=C(CCCCBr)NC1CCC(C(=O)NCc2cccc(OC(F)(F)F)c2)CC1 c1(OCC)cccc(CNC(C2CCCCO2)c2ccccc2)c1OCC N1(C(C(C)OCC)=O)CCN(C)C(C(=O)NC2(C)CS(=O)(=O)C2)C1 c1(C(CC)NC(=O)NC)cccc(OCC(N2CC(F)C2)=O)c1 c1(N(CC(=O)NC)C)nc2c(c(=NC(C)c3ccc(Br)cc3)[nH]1)COC2 CC1CC(NC(=O)CSc2n[nH]c(O)n2)CN(C(C2(C)CCN(C)CC2)=O)C1 C1(C(N(C)CC2N(C(CCSC)=O)CCC2)=O)CC2CCCCCCC12 N1(C(CC2(C)CCOCC2)=O)CCC2(CCN(C(=O)C(C)(O)CCN(C)C)C2)C1 c1(SC)ncc(C(=O)NC2CC(NC(c3cc(C)c[nH]3)=O)C2)s1 N1(C(CC(C)(C)O)=O)CCC2(COC(CNC(C3(C)COC3)=O)C2)C1 C1(F)CCCN(C(C2(C(N)=O)CCC2)=O)C1.c1(CC)nonc1C(=O)NC N1(C=O)CCC(O)C1.C(c1ccncc1)=CC(C)C.C(C(F)(F)F)=CC=O CC1=C(C(=O)N2CCC(F)(C(=O)NCc3cc(O)cc(F)c3)C2)CCC1 CCC(C)CCCC(=O)NCC(C(=O)N1CCCC1C1CC1)C(C)(C)C C(CCS(C)(=O)=O)(C(=O)NCC1CN(C(c2cccc(F)c2O)=O)C1)OC Cc1cc(-n2cncn2)ccc1C(=O)NC(CO)C(C)NC(=O)C(C)(C)C Cn1nnc(=NC2(CO)CCCN(C(C3CCNC3=O)=O)C2)[nH]1 C12(NC(C(=O)NCC3CC3)=O)CCN(C(=O)CCCCCF)CC1C2 N1(CC)CCCC1C(=O)N(C(CNC(=O)CC(=O)N(C)C)C1CC1)C C1(C(N(OC)Cc2ccc(C)o2)=O)C2CC3C(C2)C13.C12(C)CC(C#N)(C1)C2 C(CS(=O)(=O)C(F)F)NC(c1n(CC)nnn1)C1(CC)CC1 c1(CN2CC3C(C(=O)Nc4cc(C)cc(Br)n4)(C3)C2)cc2ccccc2cc1O C1(NC(C(=O)NCCCCCCCC)=O)CC(OC)C12CCCCC2 C1(NC(c2cnc(C(C)C)[nH]2)=O)CCCN(C(C2CCSCC2)=O)CCC1 c1(COCc2c(C)cc[nH]2)nc(-c2cn(CC3CCCCC3)nn2)nn1CCF N1(C(=O)NCC(c2ccc(C)cc2)OC)CCN(C)CC1C C1(C(=O)NCCN(CC(C)O)C(c2[nH]cc(CC)c2)=O)CCn2ccnc2C1 Cc1ccc(C(=O)NCC2(C)CCC(NC(=O)CC3(O)CC3)C2)c(O)c1 CC(C1=CCN(C)CC1)NC(C1CCN(C(=O)C(C)(C)C)CCO1)=O c1(C=O)cc2c(nc1O)CCCCC2.C1(CC)CCCC1C(=O)NC1(C)CC1.N Cc1ccc(O)cc1C(=O)NC1CC(NC(c2ccc(I)c(F)c2)=O)C1 Cc1cnc(O)c(NC(=O)C2=CCC(NC(=O)C(C)(C)C3CC3)C2)c1 CN=c1[nH]c(C(=O)NC2CN(C(C3CC(C)C3)=O)CC2c2ccc(F)cc2)cs1 N1(C(CCCN(C(C)C)C)=O)CCOCC1C(=O)NCCN1CCCCC1C c1(C(=O)NC2C(NC(CC3(OC)CCCC3)=O)COCC2)cn2c(n1)CCC2 c1(CC)ncoc1C(=O)NC1CCC(N(C)C(c2cn(C(C)C)cn2)=O)C1 C1(NC(CN(S(CC)(=O)=O)C)=O)CCCN(C(C2CCOC2)=O)C1C c1(C(=O)NC(CCC)CCCNC(C2(OC)CC2)=O)ncc(F)c2ccccc12 N1(C(CCC(C)(C)C)=O)CC2CCC1C(NC(=O)C=CC1CCC1)C2 CC(C)C(Cc1ccccc1)CN=C(NC(C)C)N1CCN(c2nncs2)CC1 C1(CC)(NC(C2CCC(C)(C)O2)=O)CCN(C(c2ccc(O)cc2C)=O)CC1 C(C(=O)N1CCN(C(c2ccc(Cl)c(N)c2)=O)C(C2CC2)C1)(C(C)(C)C)SC S(=O)(=O)(c1cccc(=NCc2scnc2C)[nH]1)N1CC(OC)OCC1 C1(CNC(C2C(OCC)C2)=O)CCCC2(CN(C(c3ccccn3)=O)C2)O1 Cn1cccc1CCC(=O)NCCCOCC(C)C.C(=O)CCC1CC1(C)C.N CC1CCC(C)(C(=O)N(C)CC2COCCN2c2cc(C(N)=O)ncn2)C1(C)C c1(N(C)CC2(OC)CCC2)cc(Cl)c(Cl)cc1[N+](=O)[O-] Cc1ccc(C=CC(N2CC=CC2C(N2CCCC(C)CC2)=O)=O)cc1 N1(C(C(CC)SC)=O)CC(NC(c2cnns2)=O)CC(C)(C)C1 CC(CCCCCO)NC(=O)CN(C1CCC1)C(C1CC(C)(F)C1)=O C1(OCC)CN(C(c2ncoc2C)=O)CC1.c1(C2C(C=O)C2)cnn(C)c1.C Cn1[nH]c(=NC(=O)NC2CNCC23CCCCC3)c2ccncc12 C1(NC(COC(C)=O)=O)CCC2CCN(C(C3CCC4(CCC4)CC3)=O)C12 c1(CN2C(C)(C(=O)NCC3(C)CC3)CC2)cc(Cl)c(F)c(Cl)c1 C(CCSC)(C(=O)NCCC1CCN(C(C2(C(F)(F)CC)CC2)=O)C1)OC c1(N(C)C)nccc(NNC(=O)C2CNCCC23CCOC3)n1 C=C(C)CC(C(=O)NCc1ccsc1C(=O)NCc1nc(C)ccc1C)OC c1(C(=O)NCC2(C=O)CC(=C)C2)cnn(C)c1N.c1(C(C)O)cnn(C)c1.N c1(C(N2CC(CNC(c3cncc(O)c3)=O)C2)=O)cc(F)cc(Br)c1F Cc1c(C(N2CCC(F)(F)CC2)=O)[nH]c2ccc(C(N3CCOC4CC34)=O)cc12 N1(C(c2ccn(C)c2)=O)CCC2C(NC(=O)C(c3ccc(Cl)c(Cl)c3)(F)F)CC12 c1(C(N2CC(NC(C3C(C)(C)OCC3)=O)C(CO)C2)=O)cnc2[nH]ccnc1-2 c1(C(=O)N)cccc(C(F)F)c1Cl.CCC(CNC(=O)C(F)CC1CCC1)CC c1(OC)cc(NC(=O)NC(CC#N)C(F)(F)F)cc(Cl)c1OCC(C)C C1(CC(=O)NC)CN(C(=O)CCc2cccnc2Cl)CCN1C(=O)CCF N1(CC)CCC(C(N2CCC(CCC(=O)NC3CCOC3)C2)=O)CC1 C1(n2cc(CNCc3sccc3)nn2)CCC(CC2CC3(CCC3)C2)CC1 c1(C(C)C)c(C(=O)N(C2CCCC(NC(=O)C(Cl)=CCl)C2)C)cnn1CCO C1(C(N2C(CNC(c3nnc(O)cc3O)=O)CCCC2)=O)CC2(C1)CC21CCC1 C12CCCN1CCC2.c1(C(=O)NCc2ccsc2C(=O)N)cc([N+](=O)[O-])c[nH]1 N1(C(c2c(C)ncc(N)c2)=O)CC(NC(=O)CN2CC(C)(C)C2)C2CCCC12 c1(C(N2C(CCNC(c3ccccc3)=O)CC(OC)C2)=O)cccc2nncn12 C1(=CC(=O)NCC(C)CNC(=O)CC2(C)CCCCC2)CCCCC1(C)C CCCCC(O)C(=O)NC1C2CC1N(C(c1cccc(C(C)(F)F)n1)=O)C2 Cc1ccc2cc(C(N3CC4CC4(C(=O)NCc4cccc(Cl)c4)C3)=O)sc2c1 CCC(CC)(C(=O)NC(c1ccccc1)C(=O)NC1COCC1CO)OC c1(CC)cc(NC(C2CCCN2C(C2(SC)CC(=O)C2)=O)=O)cc(O)c1 C#CCCCCC(=O)N1CCCCC1c1n[nH]cc1C(=O)N(C)CC1CC(O)C1 O=C1NC2CCN(c3ccnc(NC4CCCNC4)n3)CC2O1 N1(C(CC2C(C)(C)CCO2)=O)CC(NC(C2CC=CC(O)C2)=O)CC(O)C1 c1(C(=O)NC(CNC(CCc2c(C)cccc2)=O)C(C)C)ccc(Cl)c(F)c1F N1(C(C2CCN(CC)CC2)=O)CCCCC(CCC(=O)NC2CCCSCC2)C1 N1(CC)CC(C(=O)NCC(O)CNC(=O)CCCC(C)=O)c2ccccc21 C1(NC(C(CCC)CC)=O)CC2(CCN(C(=O)C=Cc3c(F)cccc3F)C2)C1 C1(C(=O)OCC)CC2(CCNCC2)CN1C(=O)C(c1ncccc1OC)(F)F N1(c2nnc(CC)o2)CCN(C(=O)C(c2c(C)nn(C)c2C)C)CC1C c1(C(N2C(CNC(c3cc(C)[nH]n3)=O)CC(F)(F)C2)=O)cccc2nc(O)oc12 Cc1cccc(CN2CCCC(NS(=O)(=O)CC#N)C2)c1C c1(CC(N2CC(OC)C(OCO)C2)=O)ccc2c(c1)CC2 C1(N(C(=O)CN2CC(C)(C)C2)CC)CCCN(C(=O)Cn2cc(C)cn2)C1 c1(C=O)cccc(Cl)c1.CCCCNC(=O)CC1CN(C=O)C1.C(C)(C)C c1(C(C)NC(c2n(CC(=C)C)nnn2)(COC)CC)ccc(Cl)c(Cl)c1 CON=Cc1ccc(C(N2CCCC(N(C(=O)C3=COCCO3)C)CC2)=O)cc1 O=C1CC(C(=O)NCCn2cc(-c3nc(C4CC4)cs3)nn2)C2(CCC2)C1 c1(C(=O)Nc2cc(OC)nnc2)ncn2cc(-c3ccc(C#N)c(C)c3)sc12 c1(CC(C(=O)OCC)NCc2cnc(C)cn2)cc(Br)cc(Br)c1 C(=O)(CC(O)CN(C)C)NC(CC1CN(C(CC(C)C)=O)C1)C N1(C(C2C(C=C)C2)=O)CCC(O)C(NC(=O)C=Cc2cncc(C)c2)C1 Cn1cc(C(C)(C)C(=O)NC(CNC(c2cn(C3CC3)nn2)=O)CO)cn1 c1(C(N2CCCC(NC(c3cc(C)c(Cl)s3)=O)C2C)=O)cc2cccnc2o1 Cc1ccc(-c2nc(-c3ccc(Cl)c(F)c3)n(CC(N)=O)n2)cc1Br c1(-c2c(C(N3C4CC(CC(OC)C4)C3)=O)csc2)ccc(S(C)(=O)=O)cc1Cl C12(C(N3CC(CC=C)(NC(=O)CCc4ccco4)C3)=O)CCCC1C2(F)F CCCCCC(O)CC(=O)NCC(n1cc(CCC2CCCC2)nn1)C c1(NC(C2CCN(CCn3cc(CO)nn3)C2)=O)cc(O)nc(O)n1 C(c1cn[nH]c1)=C(C=O)C.N1(C(CNCC=O)=O)CCC1.C(=O)C1CC1 N1(C(Cc2ccn(C)n2)=O)CCC(CNC(C2(C3CCCCO3)CC2)=O)C12CC2 C(c1ccc(F)cc1)=CCC(N1C(C(CNC(C=CC)=O)(C)C)CCC1)=O CCCCC(CC)CN=c1cc(C2CCC2)o[nH]1.N(C)C C1(CC(=O)NC(c2ccccc2)C(=O)N(CC)CC)CC2(CC2)CO1 Cc1ncnc2c1CC(C(=O)NC1CCc3nc(C(C)C)[nH]c3C1)CC2 c1(-c2ccn(C)n2)c(C(=O)NCCc2nc3ccccc3[nH]2)nn2c1CCCC2 C1(CC(=O)NC)CN(C(c2cscn2)=O)CCN1C(C1CSCCS1)=O C(c1cccc(F)c1F)=CC=O.n1(CC)cnc(C(=O)NCC2CC2)n1.N N1(C(C2OCCN(C(C=C(CC)CC)=O)CC2)=O)CCCNC(=O)C1CC n1(C2CN(C(CN(CCOCC)C3CC3)=O)C2)cc(C(C)(C)C)nn1 c1(C(N2CC3CCC2CC3)C(=O)Nc2ccc(OC)cc2)c2c(nn1C)CCOC2 c1(SCC)ccc(Cl)cc1C(N1CCCCC1CNC(=O)CC(F)F)=O c1(CC(=O)N(CC)C2CC2)c[nH]c2cccc(C)c12.C(C)(C(O)C=O)OC.N C(=O)(CC(F)(F)F)OC(C)C(=O)NC1CCN(C)CC1.c12ocnc1C2 C#CC1(CNC(C2(CNC(c3cc(C)sn3)=O)CCCCC2)=O)CCOCC1 C1(CNC(c2ccc(F)s2)=O)CCC2(CC1)CCN(C(=O)Cc1ccco1)CC2 CC1CCN(C(=O)CN(CCCN(C)C(C2CCC(F)C2)=O)C)CC1 Cc1cc(C(=O)N(CCCCNC(=O)CCc2ccsc2Cl)C)cnc1C CC1CCC(NC(=O)CCc2ccc[nH]2)CN1C(=O)CSc1ccncc1 C=Cc1ccc(C(=O)NC(C(=O)NCC2CC3(CCC3O)C2)C2CCC2)cc1 N(C1COc2ccccc21)C(C=Cc1ccc(SC)cc1)=O C1(C(N(c2cccc(O)c2)CC)=O)CCN(C(C2CCC(=O)NC2)=O)CC1O Cc1cc(CNC(C2CCCCN(C(=O)CC3CCCCO3)C2)=O)cnc1F CCC(O)C(C)C(=O)NC1CCN(C(=O)C(C)(C)CN(C)C)CC1CO c1(C(=O)NC(C(C)NC(CC(CC)CC)=O)C(C)C)ccc(C)c(C)c1O C1(C(=O)NC(CN(C(Cc2ccc(C)c(F)c2)=O)C)C)CN2CCN1C(C)C2 N1(C(c2cnc(OC)s2)=O)CCC(NC(=O)CC2CC(=O)NC2=O)C(F)C1 c1(C(=O)OC)cc(C)cnc1N1CC2CC(NC(=O)C=Cc3nccs3)C2C1 Cc1cc(C(=O)NC(C)(Cc2ccccc2)CO)n(C2CCC2)n1 Cc1c(C(c2nnnn2C)Nc2ccc(C(N3CCOCC3)C)cc2)nnn1C n1(CCC)ncnc1C(c1nnnn1CC)NCC(C)(C1CC1)OC CC1(NC(c2cnn(-c3ccccn3)c2)=O)CCCN(C(c2cnc(Cl)s2)=O)C1 c1(C(N2C(C)CC(NC(c3c(OCCC)cccn3)=O)C2)=O)cc[nH]c(=N)c1N N1(C(Cc2cc(C)no2)=O)CCC2CCCN(C(=O)CN(C)C)C2C1 C(=O)C1=CCC(F)(F)CC1.c1(CNC(CCOCC#C)=O)ccc(CC)cc1 C=C(Br)CC(C)(C)C(=O)NC(C1CN(C(=O)CN(C)C2CC2)CCO1)C N1(Cc2c(C)noc2C)CCC(CNC(=O)CCN2CCCCC2)C(F)(F)C1 Cn1cc(CCC(N2CCN(C(=O)CCC#N)C3COCC23)=O)c2ccccc12 Cc1nc(Cl)nc(N2C3CCC2CC(NC(C2C4CCCC24)=O)C3)c1Cl C#Cc1ccc(C(=O)NC(CC(=C)Cl)C(=O)N2CC3C(C(N)=O)C3C2)c(C)c1 C=CC1(CC(=O)NC2CC(=O)N(C)C2)CN(C(C2CCCN2C(C)=O)=O)C1 c1(CNC(C)(CCCO)c2n(CCC)nnn2)ccc(C)nc1NCC CC1CN(C(C2CC2C)=O)CCC1C(N1CCN(c2ccc(Br)cc2)CC1)=O c1(C(=O)NCC(C2CCOC2)NC(c2cnc(O)s2)=O)cccc(CCO)c1 C(=O)(CCCS(N)(=O)=O)N1C(CNC(CC(CC)C2CC2)=O)CC1 N1(C(C(C)OC(C)(C)C)=O)CC2(C(=O)NCC3(O)CCCC3)CC1CO2 N1(C(c2cncc(C)c2)C(=O)NCc2ccccc2)CC(CC(F)(F)F)OC(C)C1 N1(CCCCNC(CN(CCOC)C)=O)CCCN(C(=O)CCC(C)(C)F)CC1 Cc1cscc1C(=O)NC1CCC1NC(=O)C(C)Cn1cccn1 Cc1noc(N)c1C(=O)N(CC(O)CN(C(=O)Cc1ccc(Br)cc1)C)C c1(OC(N2CCN(C(C)=O)CC2Cc2ccccc2)=O)ccccc1S(C)=O N1(c2n(CCC#C)c(-c3ccncc3C)nn2)CCN(C)C(COC)C1 C1(c2nnc(N(C)CC3(OC)CCCC3)n2CC2CC2)CCc2ncc(C)n2C1 C1(O)(CC)CCN(C(C2(NC(c3ccc(OC)o3)=O)CC2(C)C)=O)C1 c1(C(=O)NC(COCC)C)ccn2c(-c3ccc(OC)c(OCC)c3)cnc2c1 C1(NC(C(C)(C)O)=O)CC2CC(NC(C3CNC(=O)C3)=O)C1C2 C1(NC(C(C)N(C)C)=O)CN(C(c2ccc(F)cc2Br)=O)CC12CC2 c1(C(=O)N(C2CC2)CCO)ccc(S(=O)(=O)N2CCc3sccc3C2)cc1 c1(N(C(=O)NCC2CCC(CC)O2)C)ccc(C)nc1Cl CC(CC(=O)N(C)CC1(NC(C2CCC2)=O)CC1)n1cccn1.N(C)(C)C O=C(CCCC(F)F)NCC12CC1CN(C(c1ccccc1Cl)=O)C2 C(=O)(CCCCN=[N+]=[N-])NC(CC(C)C)C(N1CC2COCC2(CO)C1)=O N1(C(C(C(CNC(CCCCCCC)=O)C)F)=O)CCC2CCCC2CC1 C1(C(=O)N)CCN(CC(F)(F)F)CC1.C1(O)(CC)CN(C(C2CSCCS2)=O)C1 n1(CC)cc(C(=O)NCC(C)CN(C)C(C2(C#N)CC2)=O)c(C2CC2)n1 C1(CNC(c2n[nH]c(C)c2O)=O)CC2(CCN(C(=O)C(F)C(F)(F)F)CC2)C1 N1(C(C(c2ccccc2)OC(C)C)=O)CCC(n2cc(C(C)(C)C)nn2)C1 n1(C)cnc2cc(F)c(Br)cc2c1=O.C1(CN)CCOCC1 C#CC1(C(N2CC(=O)NC(CC)C2)=O)CCN(C(=O)CCNC(N)=O)CC1 c1(C(N2CCC(CCNC(C(C=CC)O)=O)C2)=O)ccc(-c2nc[nH]n2)cc1 C1(CNC(c2nc(OC)c(C)s2)=O)CC2(CCN(C(C3(C)CC3)=O)CC2)C1 C1(CNC(C2C(=C)CC2)=O)CC2(CO1)CN(C(=O)Cc1ccc(Cl)cc1C)C2 Cn1cnc2c(c1=O)CCN(S(=O)(=O)CC(C#N)C1CCNCC1)C2 c1(-c2cnc(C)s2)cccc2[nH]c(C(=O)Nc3c(C(=O)ON)cnn3C)cc12 C12(C(=O)N)C3C4C1C1C2C3C41C.C1(CC)CN(C(C2(C)CCCS2)=O)CCC1 C1(NC(CNC=O)=O)CCCCN(C(c2ccc(-c3nc(=O)o[nH]3)cc2)=O)C1 CCC(CCC(=O)N1CCCO1)NC(=O)CC(C)C1CC1 C12(C(N3C4C(CNC(COC)=O)CC(CC4)C3)=O)CCCCC(=O)N1CCC2 N1(C(C(CC#C)C2CC2)=O)CCC(CNC(=O)C(C(C)(C)C)OC)C(F)(F)C1 N1(C(=O)NCC2(OC)CCC2)CCCC(C)(C(=O)N(CC(F)(F)F)C)C1 C12(NC(C(C)Cn3ccnc3)=O)CC(C1)N(C(C1CCN(C3CC3)C1=O)=O)C2 N1(C(C(CC=C)C)=O)CCCCC(NC(=O)C(C)(C)c2ccccn2)CC1 C1(NC(=O)Cc2ccc(F)cc2Cl)CCOC2(C1)CC(C(=O)O)C2 N1(C(CCC(N)=O)=O)CC2(CCC2)CC1CNC(c1n[nH]c2ccccc12)=O N1(C(C(CC)NC(C)=O)=O)CCC(C(C)C(=O)NC(C)(CO)CO)CC1 Cc1cc(C(=O)NC(C)CC2CCN(C(C3OCCCO3)=O)CC2)ncc1Cl N1(C(CC(=C)C)=O)CCC(C)C(CNC(c2cnoc2-c2ccccc2)=O)C1 C1(C=O)C2CC3C(C2)C13.c1(C=O)cc(-c2ccccn2)[nH]n1.C(C)C1CC1.N C=CC1(C(=O)NC(C)Cc2nccn2C)CCN(C(=O)C#CC2CC2)C1 C(=O)(CC(C)C(=O)NC1CCCCC1C(N1CC(OC)C1)=O)OC c1(C(=O)NCC(CC)(C)NC(=O)CCOC2CC2)cc2c(s1)CCC2 C(=O)(C1Cc2ccccc21)NC(C(N1CC2(CN(CC)C2)C1)=O)CC1CCC1 c1(C(C(=O)NC2CCC2)N(C(C(C)SC)C)C)nnsc1SC CCCCCCCCCC(=O)NC1CN(C(=O)C(F)C(C)CC(C)(C)C)CC1O c1(C(=O)NCC(CNC(CS(CC)(=O)=O)=O)C(F)(F)F)ccc2[nH]ccc2n1 C(C1=NOC2CN(C(=O)CCSCC(C)C)CC12)NC(C=CCOC)=O N1(C(COCCC)=O)CC2CCCC(N(C)C(c3sc(C)cc3Cl)=O)C2C1 c1(C(N2CCC(NC(c3c(C)nco3)=O)C2)=O)cn2c(n1)CCC(C)C2 C=CCCCC(=O)N(C1CCC(NC(=O)CCc2ccc(=N)[nH]c2)C1)C c1(CC(C(=O)OC)NC(=O)CC)ccnc(F)c1OC.c1ccccc1.C(C)C N1(C(C(CCC)NC(COC2(C#C)COC2)=O)=O)CCS(=O)(=O)CC1 C1(NC(c2ccc(O)c(Br)c2)=O)CN(C(=O)CS)CC12CC2.c1n[nH]c(O)n1 c1(C(C)C)ccc(Cl)cc1C(=O)NC.C1CCCCN1C(c1cn(C)c(C)n1)=O N1(C(CC2(C=C)CC2)=O)CCC(NC(c2cncs2)=O)CC1 N1(C(Cc2cnc(C)o2)=O)CCOC2(CCCN(C(c3ccc(O)nc3)=O)C2)C1 Cc1nc(C)c(CN2CCNCC2C2CCC2)o1 N1(CC(=O)NCC(CO)NC(C(CCC(C)C)O)=O)C(=O)c2cccnc2C1=O C1(NC(C(C)=CC)=O)CC(C)CN(C(c2ccc(OCCF)cc2F)=O)C1 C(=O)(C(C(C)(C)C)N1CCCC1=O)NCCN(C(CCC(C)OCC)=O)C Cc1ncc(C(N2CCC2C(=O)NC2CC(C#N)C2)=O)cn1 c1(C2(CN3CC(NC(C(C)(O)c4ccccc4)=O)C3)CCCC2)ccccc1F Cc1c(C(N2CCCC2CCNC(=O)C(=O)N(C)C)=O)cc(O)cc1N Cc1cc(Br)cnc1C(=O)NC(C)CCC.C1(C=O)CCN(C(=O)C2CC2)CC1 Cc1cc2c(cc1NC(=O)NNC(=O)c1cn(C3CCCCC3)nn1)sc(=O)n2C Cc1nn(C)cc1CCNC(C1C(C)CCN1C(C1CC2(CC2)C1)=O)=O C12(CNC(CCCOC(C)=O)=O)CCC(CC1)OC2.c1(CC=O)ccoc1.C C1(c2cn(C)nc2)CNCCN1C(C1(C)CC1(Br)Br)=O c1(C(=O)NCC2(O)CN(C(C(CC)(C)OC)=O)C2)ccc(Cl)c(Cl)c1N C(=O)(CC1OCc2ccccc21)N(CC(CC)NC(CC1CC(=C)C1)=O)CC N1(C(c2c(Cl)cn(C(C)(C)C)n2)=O)CCCC(O)C1.c1(C(=O)N)c[nH]c(=O)cn1 C1(C=O)CC2CC(=O)C1C2.c1(C(=O)NCC2CCCCC2)cccc(Cl)c1F.N C(=O)(C#CC1CCCC1)N1CCCCC(CCC(=O)N(C)Cc2scc(C)c2)C1 N1(C(C23N(C(C4N(C)CC(C)(C)C4)=O)CC(C)(C2)C3)=O)CCCC(C)(O)CC1 c1(N(C)C)nccc(=NC(=O)CC2CN(Cc3ccc(F)c(C(F)(F)F)c3)C2)[nH]1 N1(C(C=C(CCC)C)=O)CCN(C(C2COCCOC2)=O)CC1CCOC C1(NC(c2conc2C(F)(F)F)=O)COCCC1NC(C1C=CCC1)=O C(C)(c1cnn(C)c1)=CC(N1CCC(C(F)(F)F)C1)=O.CCCCS.CC=O C1(CNC(c2nnc(C)s2)=O)CN(C(C2CCC(C)CC2)=O)CC1(C)C C1(NC(C(C)CO)=O)CCN(C(=O)CC2(CS(C)(=O)=O)CC2)C12CCC2 C12(NC(C(CCC)C)=O)C3CC(CC13)N(C(c1cc(Cn3cccn3)on1)=O)C2 N1(C(CCOC)=O)CC(CNC(=O)C(F)C2CCC2)C(C)C1 CN1CCCCCC1C(N1CCCC1C(=O)NCc1cocn1)=O c1(C(=O)NCC(C)N(C)C(c2cc(CO)n(C)n2)=O)cncc2[nH]ccc12 CC1CCN(C(=O)NC2CCN(C(=O)C(c3ccccc3)F)C2)C1 C12(CNC(C(C)C3CC3)=O)CCCCC1N(C(=O)C=Cc1cccc(O)c1)CC2 c1(CC(C)OC)nc(-c2ccc(CN3CCCCC3)cc2)n(C(C2CCC2)C)n1 C(=O)(C1Cc2c(Cl)cccc21)NCCC(C)NC(C(C)NC(C)=O)=O C12(CC(N3C(C=C)CCC3)=O)CCC1CN(C(=O)COC)C2 CC1CN(C(C2CCN(C(N)=O)CC2)=O)CCC1NC(c1sccc1Cl)=O C(=O)(CC(C)C(C)C)N1CCC(CC(=O)NC)C1.N1(CCC(=O)N)CCCCC1 N1(C(C23CC(NC(=O)Cc4cnns4)(C2)C3)=O)CCCCC1CCO N1(C(c2c(CC)noc2)=O)CC(NC(=O)Cc2cc(C)n(C)n2)CCC1C C1(CNC(c2cnn(CC)n2)=O)CN(C(=O)Cc2cscn2)CC1(C)C C1(OCC)CN(C(c2ccc(OC)cc2)=O)CC1c1cn(-c2ccccc2)nn1 N1(C(C(C)C#N)=O)CC2C(CN(C(=O)CSc3ccc(Cl)cc3)C)C2C1 C1(C(N(CCC(=O)NCC(Cl)Cl)CC)=O)CC2CCC1O2 Cc1ccc(S(C)(=O)=O)cc1S(=O)(=O)Oc1ccccc1OCC(C)(C)C N#CC1CCN(C(=O)C(CNC(c2ccsc2C#N)=O)CC2CCCC2)CC1 CC(CC(N)=O)C=O.c1(NCC(=O)NCCNC(=O)C)ccccc1Br.N CCC(O)C(C)C(=O)N(CCCC(=O)N1CC2(CC2)C1)C N1(C(C(CC)CC(F)F)=O)CCC2(C1)c1[nH]cnc1CCN2C(=O)C(C)OC c1(C(=O)NCC(CNC(c2c(C)[nH][nH]c2=N)=O)OC)nc(C)c(C)nc1O Cn1ncc(C(F)F)c1C(=O)NCCC1CN(C(C2(F)CC2)=O)C1 C(C(C)(COC)C(=O)N1CCN(CC(=O)NCc2ccncc2C)CC1)OC C1C2CCC1N(C(=O)CN1CC3CCC1C3)C2.c1(OCC)ncccc1C(=O)N c1(C(N2CCC(C)(N(C)C)C2)C(=O)NCC(F)F)cccc2nc[nH]c12 O=C(CC1=CCCC1)NC1CN(C(C23CC(C2)C(C(F)(F)F)O3)=O)CCC1C c1(CNC(=O)Nc2c(OC)ccc(C)n2)cc(F)c(O)c(F)c1 C1(CC=C)(C(N2CCSC(CC)C2)=O)CCN(C(=O)CNC(=O)OC)C1 c1(CC)noc(C)c1.C(=O)(C(C)CC1CCCC1)N.C(=O)CC(O)CN(C)C N1(C(C2C(=C)CC2)=O)CCC(CO)(NC(=O)Cc2csc(C)c2)C1 C(=O)(CCCS(N)(=O)=O)NC1CN(C(C(C)CC2CC2)=O)CC1c1nccn1C CC#CCCC(=O)NCC(C)(C)CNC(C1CCS1(=O)=O)=O C1(C(N(CC(=O)NCCCc2cc(C)no2)CC#C)=O)CC(C)(C)CO1 CC1(C)OC(=O)C(CC(=O)NCc2ccc(CNC(=O)C=CBr)cc2)O1 c1(OC)cc(OC)c(C(=O)NCC(CO)NC(=O)CO)cc1N.c1cccnc1 C1(C(CC)C)CCN(CC(=O)N(c2ccccc2)C)CC1.C1(OC)CCCO1 CN=c1[nH]cc(C(=O)NC2CCOCC2C(=O)NCCc2cnc(C)o2)s1 c1(NCC2(OCC)CCCSC2)nc(C)cc(=NC2CCCN3CCCC23)[nH]1 C1(C)(CNC(c2c(C)cc(CC)o2)=O)CCCN1C(c1ccc(C)cn1)=O CC(CC(=O)NCC1(O)CN(C(=O)Cc2cccn2C)C1)c1cccnc1 c1(SC)ccc(O)c(C(N2CCC2C)=O)c1.c1(C=O)cnoc1C.C(=O)C.N N1(C(CC2C(C)(C)C2)=O)CC(NC(C2CC23CCOC3)=O)C2CCCCC12 Cc1nc2c(o1)CCCC2CC(=O)NC1CCN(C(=O)CCCCCF)CC1F O=S1(=O)NCC2CN(c3cc(NC4CCCc5ccoc54)ncn3)CCN12 C1(C(N2CCC(CCCNC(C(C=C)O)=O)CC2)=O)CCC2(CC1)CC2 c1(OC)ccc(C)c2c1CC(C(N1CCC(c3cc[nH]n3)CC1)=O)N2 N1(C(C2(C)CCC2)=O)CCN(C(=O)CC2(C)CCCO2)C(C(F)F)C1 c1(C(=O)OC(C)(C)C)ccc2nc(NCC(C3CC3)C3CC3)cn2c1 C1(OCC)(CO)CCCN(C(c2cn(C(C)C)cn2)C(=O)NCC)C1 CC1CN(C(=O)C=CC(F)(F)F)CCN1C(=O)CCC(N)=O c1(CCOC(C)C(=O)NCC(C)C)ccccc1.C(C1CCCO1)=CC(=O)N c1(C(N2CCC(C3(NC(=O)Cn4ccnn4)CC3)C2)=O)cc2c(nn1)CCCO2 c1(OCC)ccc(CC(C)CNC(=NC)NC2CC23CCC3)cc1 c1(C(=O)NCC(C)C2CC2)n[nH]c2c1CN(C(=O)CC#N)C2 CCS(=O)(=O)CC(=O)NC(CN(C(=O)C(c1ccccc1)OC)C)(CO)CO C(C(=O)N)(C1CC1)OCC.C(=O)(CC)NC.c1(C=O)cccs1.C1CC1 CC1=CCC(C(=O)NCCC2CCN(C(C3(N(C)C)CCCCC3)=O)C2)CC1 C(C)(C(C)(C)C)NC(COCCCOC)=O.C(c1ccncn1)=CC=O.N C1(C(N2CC(O)(CCNC(=O)C(O)c3cnc[nH]3)C2)=O)CCC(C2CCC2)CC1 C(C(=O)NCC1CC1C(=O)N)(C(C)(C)C)OC.c1ccc(C#N)cc1.C c1(CC(=O)N(CCN(C(C2CC2)=O)C)C(C)C)sc2ccccc2c1C.CO c1(SC)cncc(C(=O)NCCN2CCN(C(=O)CC(O)C3CCCC3)CC2)c1 c1(NC(C)(CNC(C2CC(O)C2)=O)C2CC2)ccnc(C2CC2)n1 C1(NC(C=CC)=O)CC2(CCNCC2)C1.c1cc(C(F)(F)F)cc([N+](=O)[O-])c1 C1(OC)CN(C(=O)C(C)(C)CO)CC1NC(c1csc(C(C)(F)F)n1)=O CC1(C)CC=C(C(=O)NC2CC(CNC(C3CCCSC3)=O)CC2O)CC1 C1(C(=O)NCC(CNC(c2c(C)n(C)cc2)=O)F)CCc2c(nnn2C)C1 C(C(=O)NOC(C)(C)C)=CCN(C(=O)COCC1CC1)C C(=O)(CCCC(=O)N1CC(NC(=O)C(c2cncnc2)C)CC1(C)C)NC(C)C CC(C)(C#CC(=O)Nc1ccn2nccc2c1)CNC(=O)OC(C)(C)C Cc1noc(C)c1C=O.c1(CC(N2CC(c3cnco3)C2)=O)cc(Cl)n(C)n1.N C#CCC(C(=O)NCC(C1CCN(C(c2cc(F)n(C)n2)=O)CC1)C)C1CC1 C(=O)(C(O)CC(F)F)NC(CCCCNC(c1n(CC)cnn1)=O)C C=CC1CN(C(C2CCC=CCCC2)=O)CC1NC(C1(F)CCCCCC1)=O c1(C(N2CCC(C)C2CNC(=O)CC2CC=CC2)=O)cc(Cl)cc2c1CCC2 CCCS(=O)(=O)C(C)C(=O)N1CC2CC2(CNC(c2ccnnc2)=O)C1 c1(C(=O)NCC(C)CNC(=O)C(C)(C)C)nccc2cc[nH]c12.CC(F)F.O c1(NC(C2C3CC2N(C(c2ccccc2S)=O)C3)=O)cc(Br)nc(Br)c1 c1(C(=O)NCCNCc2c(C)nn(-c3ccc(F)cc3)c2)[nH]nc2ccncc12 C1(CC)CCCC(N=c2[nH]c(=NC)[nH]c(=NCc3cn4cccnc4n3)[nH]2)C1 N1(C(C(C2CCN(C(c3ncc(C)nc3)=O)CC2)C)=O)CC2CC1CN2C CC(C)(C)C(CO)C(=O)NCC1CCC1.c1(C(=O)N)cccc(C2CCCC2)c1 c1(C(=O)NC2C(CNC(C(CC=C)CC)=O)C2)ccc(OC)c(OC)c1O c1(C(=O)NC2(CN(C)C(c3cn(C)[nH]c3=N)=O)CC2)cc(Br)nn1C C1(NC(C2CCN(CC#C)CC2)=O)CCCN(C(c2noc(C)n2)C)C1C c1(NC(C)Cn2cnnc2)cc(N2CCCOC(C)C2)nc(C(F)(F)F)n1 N1(CC)CC(C(N2CC(NC(c3nccn3C)=O)C(O)C2)=O)NC1=O c1(CC(=O)N(CCNC(CCC#CC)=O)CC2CCCC2)cc(F)cc(Cl)c1 c1(C(=O)OC)ccc(CNC(C2CCCCC2C#N)=O)c(Cl)c1 c1(C(=O)NC(CC#C)C(=O)NC(CN(C)C)C(C)C)cc2n(n1)CCC2 N1(C(CCOCCOC)=O)CCOCC(C(=O)N(C)CCc2ncccn2)C1 c1(CNC(C2C(C)(CC)C2)=O)ccc(F)cc1NC.c1cccc(C)c1C c1(C(=O)NC2CCCN(C(c3cnc(C)s3)=O)CC2)cnc2sc(C)nc2c1 Cc1ccnc2nc(C(=O)NC3CC4CN(C(=O)CCNC(N)=O)CC4C3)nn12 Cc1cc(C(=O)NC2CC3CCC2C3)c(C)n1NC(N)=O.C(=O)(C(C)C1CC1)N CC(CC(F)(F)F)C(=O)NCCC1=CCN(C(=O)COCCCN(C)C)CC1 CCS(=O)(=O)c1ccc(C(NC(=NCCCCl)NCC(C)CSC)C)cc1 C1(C(C)C)OCCC1C(N1CC(CO)(NC(=O)CN(C2CCC2)C)C1)=O N1(C(C2(C=C)CC2)=O)CCC2CCC(C1)N2C(c1cnn(C(C)C)c1Cl)=O c1(CN(C(c2ccccn2)CC)C)ccc(OCCSc2ccc(OC)cc2)cc1 N1(C(C(C)Sc2ncccn2)=O)CC(C)C(C)C1.n1(CC(=O)N)c(C)ccc1C c1(C(=O)NCCCCNC(=O)CC2CCC2C2CC2)csc([N+](=O)[O-])c1 c1(C(=O)NCC(C2CC2)NC(=O)OCC)cc(Br)ccc1C1=NCCO1 C1(C(N(CCOCC)CCNC(C2CC2C)=O)=O)CCC(=N)N1 c1(C(=O)OC)cc(C(=O)NC2CCC(N(C)C(c3cc(Cl)no3)=O)C2)c[nH]1 C(CC(=O)NCc1cn(C)nn1)(CC(C)C)NC(CCCC#CC)=O Nc1cc(Cl)cc(F)c1C(=O)NCC1(O)CCCN(C(=O)C(O)CC(F)F)C1 Cc1cc(O)cc(C)c1C(N1CCCCC(C)(F)C1)=O.N12C3CCC(C3)C1C2 C1(C(N(CC)Cc2ccccc2)=O)CN(C(c2ncn(C)c2C)=O)CCN1C c1(C(N2C(C)C(C)N(C(=O)C3=CCCCCC3)CC2)=O)noc2c(F)cccc12 N1(C(C(C)NC(C2CCCCC2)=O)=O)CC2CC(C1)N2C(c1ccncc1Br)=O N1(C(C(C)CO)=O)CCC2(C1)CN(C(c1ncc([N+](=O)[O-])n1C)=O)CCO2 C(=O)(C(C)C(C)S(C)(=O)=O)N(CC)CC.c1nc(C)no1.C(=O)C.CO C1(C(=O)NC2C(NC(c3nc(CCC)oc3)=O)C2)CCNC(=O)C1 c1(N2CCC(COC)C2)nc2cc[nH]c2c(=NC2CCCCC2)[nH]1 C=CCC(C)(CC)C(=O)N1CCC(N(C(=O)CCCC(OC)OC)CCO)C1 c1(C=O)cc2cc[nH]c2cn1.n1(CC)nc(C)c(C)n1.C(=O)CC1(C)CC1.N Cc1ccc(S(=O)(=O)NCCC(=O)NC(C)C(C)C)cc1.C(=O)C.C(C)C C1(CNC(c2cnc(N)s2)=O)CCC(NC(c2n[nH]cc2Br)=O)C1.C1CC1 c1(N(C)C)ccc(C2CC2C(=O)NCCN2CCCC2C2CCOCC2)cc1 Cc1ccc2c(ccn2CC(N2CCNC3(COC3)C2)=O)c1 C1(NC(C2(N(C(C(C(C)C)C3CCC3)=O)C)CC2)=O)CCCCCC1C N1(S(c2c(C)onc2)(=O)=O)Cc2[nH][nH]c(=NC(=O)c3ccc(C(C)C)cc3)c2C1 c1(C(=O)NCC(C2(O)CN(C(C(C)O)=O)C2)(C)C)cc2ccc(Br)cc2o1 N1(C(COc2cc(C)on2)=O)CC2CCC1C1CN(C(=O)Cc3ccco3)CC21 c1(C(=O)NCC2OCCCN(C(C(F)OC)=O)C2)ccc2snnc2c1 N1(C(c2c(CC)onc2)=O)CCC2CCN(C(=O)Cc3csc(Cl)n3)C2C1 C1(C(N(CC(=O)NCc2cc(F)ccc2F)C(C)C)=O)CC(=O)C12CCC2 c1(CNC(C(n2cc(C(C)(C)O)nn2)C)=O)cnc(O)[nH]1 C1(C(=O)NCc2n(C)ncc2)CCC(C)(C)N(C(=O)C(O)C2CCC2)C1 c1(C(C(=O)NCCCC)N(C)Cc2cnc(C)s2)ccc(OC(F)F)cn1 c1(C(C(=O)NCCCN(C(=O)CNC(N)=O)CC)C)nc(F)ccc1Cl C1(CNC(C2CCN(C(CCc3cc(C)[nH]n3)=O)CC2)=O)CC(C)(C)C(=O)O1 N1(C(C(CC(C)C)OC)=O)CC2CC(C(=O)NOCC(C)C)C(C2)C1 c1(CC)nnc(C)cc1C(N1CCC(C(C)(C)F)C1)=O C(C(=O)NC1C=CC(C(=O)N(c2cccc(F)c2)C)C1)(C(C)C)SCC C1(C2CN(C(c3cccc(C(N)=O)c3F)=O)C2)(NC(C2N(C)CCCC2)=O)CC1 CC1CN(C(=O)CC2CC(C)(C)CN2C(=O)CP(C)(C)=O)CCC1O c1(CN(C(c2cn(CC)nc2)C(=O)NCC2CCOC2)C)ccc(SC)cc1 N1(C(C2CC3CCC2C3)C(=O)NC2CC2)Cc2ccccc2CC1CCO C(CC(O)C(=O)NCCn1cnc(C(=O)NC2CCC(COC)CC2)c1)SC C1(CNC(C(CC)(F)F)=O)CC2(CCOCC2)CN1C(=O)CCC1CCC(C)O1 CC(F)(F)C(C)(C)C(=O)N.C12CC1CN(C(=O)Cc1ccc(C3CC3)cc1)C2 C(=O)(CCC1=NNC(=O)CC1)NC1C2CN(C(C3C(=O)NCC3)=O)CC1CC2 C1(C(=O)NC(CC#C)(C)C)(COC)C=CCN1C(c1ccoc1)=O C1(OC)CCC12CCN(C(C1CN(C(C)=O)C1)=O)CC2.c1(CC=O)ccsc1.N N1(C(c2c(C)nc(C3CC3)[nH]2)=O)CCC=C(CNC(=O)C(C)SC(C)C)C1 C(=O)(C(C)(C)C(O)C(C)C)N1CCC(C(=O)NCCC(C)OC)C1 Cc1oc(CNC(=O)CC2CCC2)nc1C(=O)NCCCc1cncnc1 c1(C(N2CCC(NC(C3C(=C)C3)=O)(CF)C2)=O)c(Cl)ccc(C)c1N CC(CF)C(=O)NCC(C)CNC(=O)CSC.c1coc(-c2ccccc2)n1 c1(CNC(C23CC(NC(C(NOC)=O)=O)(C2)C3)=O)cc(C)ccc1O c1(C(N2CC(C)(NC(C(C3CC3)SC)=O)C2)=O)cc(C)cc(Br)c1O N1(C(C2C(=C)C2)=O)CCCC(O)(CCNC(c2cccnc2N)=O)C1 C1(C(=O)NCC(C2CCC2)NC(=O)COc2ccccc2Cl)OC2CCC1CC2 C(C)(CCC(=O)NCC(CNC(=O)C(C)(C)O)OC)SC.c1ccc(Cl)cc1 N1(C(c2cc(F)ccc2Cl)C(=O)NC(CC)C)CCOc2c(Cl)cc(Cl)cc2C1 c1(NC(c2n(CCCC)nnn2)(C)C(C)OC)cc(Br)cc2c1OCCO2 N1(C(C(CCC)C)=O)CC(C)CN(C(=O)C(=O)NCCOC)CC1C C(CC1CC1)(CC(=O)NC1(C)CCCOC1)NC(c1c(OC)n[nH]c1)=O c1(C(=O)NC2CC(N(C(CN(C3CC3)CC)=O)C)C2)cccc2c1OCCC2 CC1c2nncn2CCN1C(=O)CCNC(=O)CC(C)O CC1(C)C(NC(C2CC(O)C2)=O)CCN1C(=O)CCn1ccnn1 C1C2CC1N(C(=O)Cc1ccnc(C(F)F)c1)C2.c1(SCC(=O)N)ccccc1 c1(C(C)(C(=O)NCCCCN(C(=O)C(C)O)C)OC)ccccc1Cl C1(C2CC2)(C(N2CCC(O)(CNC(C3(C)CC(F)C3)=O)C2)=O)CC=CC1 c1(C(N(C2CCCN(C(=O)C=C3CCOCC3)C2)C)=O)cccc2c1CCO2 C1(C(=O)NCc2c(C)n[nH]c2)CCCCCC1NC(=O)C(c1cnn(C)c1)O c1(N(CCC)C(C2CNC3CC23)=O)ccc(C)cc1 c1(C(=O)NCC2(OC)CCN(C(=O)CC(C)CF)C2)cc(Br)cnc1O N1(Cc2ccn(C)c(=O)c2)CCOC2(CCCN(C(C3CC34CC4)=O)C2)C1 C1(C#N)(CNC(CCN(C(C2CCC(CC)C2)=O)CCO)=O)CCCC1 C1(O)(C(C(=O)NC(c2cc(C(=O)N(C)C)no2)C)F)CCCC1.C1CCCS1 CP(C)(=O)COCC(=O)NCC1(C)CC1.C(c1cncs1)=CC(=O)N c1(OC)cc(C(=O)OCC(c2cc(C)n(Cc3ccccc3)c2C)=O)cnc1O N1(C(c2cn(CC)nn2)=O)CCC(C(N2CC3CC3C2)=O)C1C C(=O)(C(F)(F)C(C)O)N(C1CN(C(c2ccc(-c3ccccc3F)[nH]2)=O)C1)C Cc1cncc(NC(c2cc(-c3ccc(F)s3)ccn2)=O)c1 N1(C(Cn2cc(C(C)=O)nn2)=O)CCCC(NC(C2(O)CCCC2)=O)CC1 n1(CC(N2C(CNC(C(CC#C)C)=O)CCCC2)=O)cc(Cl)c(O)nc1=O N1(C(C(C)(C)O)=O)CCC(F)(CNC(=O)C)CC1.C1(CC=O)CCCC1.N C1(Nc2nc(C)nc(C(C)C)c2)CCN(C(c2cccnc2F)=O)CC12CCC2 C(=O)(CC(C)(C)C(C)(F)F)N1C(C)CN(C(c2ccc(C)cn2)=O)C(C)C1 c1(C(N(CCNC(=O)C(F)CC2CC2)CC)=O)cc2ccc(F)cc2o1 CS(=N)(=O)N1CCN(C(=O)CC2CCN(c3ccc(OCC(F)F)nn3)C2)CC1 N1(C(=O)Nc2ccnn(C)c2=O)CCC2C(C1)NC(=O)CN2C=O.C(C)(C)C.O CCCCCC(C)CC(=O)NC12CCCC1CN(C(=O)C=Cc1ccccn1)C2 C1(C(=O)NC(CCOC)C(=O)NC2CCCC2F)CCC(C)(O)CC1 C=C1CC2(C1)CC(C(=O)NC1(C)CCN(C(=O)CCc3csc(C)n3)CC1)C2 c1(N(CCN(C(c2c(C)noc2C)=O)C(C)C)C)cnc(C#N)c(C#N)n1 C1(C(N(CCOC)C)=O)CCN(C(=O)C)C1.C1(C(=O)N)CC1C(N)=O C(C(C(C)(C)C)NC(C1CCN(C2CCSC2)CC1)=O)NC(C(C)C)=O C(=O)(C(C)CC(C)C)N(CC#C)CC1CC1.C1(C=O)(C(N)=O)CC1.N c1(NC(c2ccc(CNC(C(C3CCC3)OC)=O)cn2)=O)cn(C)nc1C#N C(=O)CC(C)CC.C1(CC=C)(C=O)CCCC1.CCC1CC1.[SH](C)(=O)=O.N C(=O)(CC(Cc1ccc(OC)cc1)NC(=O)CC1CCCC12CC2)OC C(=O)(CCCCCF)N1CC(OC)C(NC(C2(c3ccc(F)cc3Cl)CC2)=O)C1 N1(C(C2CCC(CC)O2)=O)CC2(CCCC2NC(=O)Cc2[nH]cnc2C)C1 C1(OC)CCC2(CCN(C(C3CCN(C(C4CC5(CCO4)CC5)=O)C3C)=O)C2)C1 c1(C(N2C(CNC(C(CC)NC(N)=O)=O)CCC2)=O)cc(F)cc(Br)c1 Cc1ncc(C(=O)NCC2(C)CCN(C(=O)CC3CC3(C)C)C2)c(O)n1 c1(C(=O)NCCC(C)NC(C(C)OCC(C)C)=O)ncc([N+](=O)[O-])n1C C(=O)(C1CCCc2c[nH]nc21)NC(CN(C(=O)C(N1CCCC1)C1CC1)C)(C)C c1(OC)cc(C(N2CCCC2C(N2CCCCC2CO)=O)=O)ccn1 C(CCCC(C)C)N(C(CCN(C(=O)C(C1CCCCC1)F)CC#C)=O)C CCCCC(O)C(C)C(=O)N1CCC(C)(CNC(=O)C(CCC)OC)CC1 CC(C)CC(CNC(=O)C=Cc1cccnc1)C(=O)NC1Cc2ccccc2C1 c1(NCCCC(CCCC)CC)ccc(S(=O)(=O)NCC(C)O)c2ccncc12 C1(C(=O)NCC(=O)NCC(=O)NCc2ccco2)CCCC(F)C1 C1(CNC(C2CC(CCO)C2)=O)CCN1C(=O)CSC1CC1 c1(C(C(=O)NCCOCC)N(C)C)cc(C(C)C)[nH]n1.c1cnc(C)s1 CC1(C)CC(c2nc(-c3sc(F)cc3Br)no2)N(CC(=O)O)C1 c1(CCNC(CCN(C(=O)CC2CC3(CC3)CO2)C)=O)nccc(O)n1 C1(=CC(N2CCN(CC)CC2)=O)C2CC3CC(C2)CC1C3.C(CC)(C=O)=CC c1(CC(=O)NCc2ccc(CNC(C(C=C)O)=O)cc2)ccc(C)cc1C C12(C(N3CCC(F)(CNC(c4cc[nH]c4)=O)CC3)=O)CCCC1CC(F)(F)CC2 Cc1cc(C(=O)NC2CC(C(=O)Nc3cn(C)cn3)C2)ccc1[N+](=O)[O-] c1(CNCCCCOCC)c(OC(F)(F)F)ccc(Br)c1F c1(C(N2C(CO)CC(NC(C3CC34CC(O)C4)=O)C2)=O)cccc2sncc12 N1(C(CN(CCC)C)=O)CC2OCCN(C(=O)C3=NNC(=O)C3)C2C1 C1(NC(c2cc(C)c(Cl)cn2)=O)CN(C(=O)C(C)NC(N)=O)C2(CCC2)C1 C1(NC(=NCCC=C)NCCN2CCCC2(C)C)CCn2c(C)cnc2C1 N1(C(CCc2onc(C)n2)=O)CCN(C(C2CN3CCN2CC3)=O)CC1C(C)C CC1CC(C(N2CC(CC(C)(C)CNC(=O)C3=CCCSC3)C2)=O)CCS1(=O)=O c1(C(c2nnnn2C2COC2)NC2C3(CC(OC)C3)C2)ncc(Br)cc1F C1(N(C)C(c2cc(CNC(=O)CN=[N+]=[N-])[nH]n2)=O)CC(=O)NC1=O C1(N(C)C)CC(CC(=O)NCC(O)CNC(=O)Cc2ccns2)C1 c1(CC)nc(O)c(C(=O)N(CC)CC2CCCN2C(=O)CC(C)O)cc1C.C N1(C(CC2CCCC(NC(C3(OCC)CCC3)=O)C2)=O)CCN(C)CC1CCO N1(C(C(C2CCN(C(C3COCCC3C)=O)CC2)C)=O)CCOC(CC2CC2)C1 C1(CC(=O)Nc2ccc(-c3nccs3)s2)CCCNC1=O C1(NC(C2(OCC)CCC2)=O)CN(C(c2cnsc2)=O)CC(F)(F)C1 C1(NCc2cccc(OC(F)F)n2)CCC(C2CC2)C1 N1(C(c2cc(C(C)C)[nH]n2)=O)CCOCCC1C(=O)NC1CNC(=O)C1(C)C c1(C(=O)N)cc2c([nH]1)CCOC2.c1(OC)ccc(C(=O)NCC(C)(O)C)cc1F c1(C(=O)NC2(C)C(C(=O)NC(C3(O)CCC3)C)CCCC2)ccc2[nH]ccc2c1 c1(C(N2C(CN(C(C(CCC)O)=O)C)CC(F)C2)=O)cc(Cl)c(F)c(Cl)c1 C1(NC(C2CCC(C)(C)C2)=O)CC12CCN(C(=O)CCCCc1cnc[nH]1)CC2 N1(C(c2nc(OC)c(C)s2)=O)CCC2CCN(C(C3C4CCCCC34)=O)CC12 N1(C(c2cc(CC)no2)=O)CC(NC(=O)CCc2cccc(F)c2)CC(O)C1 c1(CC(C(=O)NCc2cccc(COC(C)C)c2)C)ccc(F)cc1F c1(OC(C)C(=O)NC)ccc(C#N)cc1.C1CCCN1C(C1CS(=O)(=O)C1)=O N(C1CCc2c(O)cccc21)C(N1CCC(CC(=O)NC)C1)=O C1(CC#C)(C(=O)NCCn2cc(CC)cn2)CCN(C(=O)C(F)C(C)C)C1 C(C(CNC(C1(c2cccnc2)CC1)=O)CO)NC(CCN(CCC)C)=O Cc1ccc(C(N2CCOC(C(C)NC(c3cccc(Cl)c3N)=O)C2)=O)c(C)n1 CC1(C)OCCC1C(=O)N.C1C2CC1N(C(c1ccc(C(F)(F)F)s1)=O)C2.C N(C1CCCc2ccoc21)C(C1(C(C)C)CCCN1C(=O)C1=CCCCO1)=O Cc1c(F)ccc(O)c1C(N1CCC=C(CNC(=O)CC2=CCOCC2)C1)=O c1(N2CCC(OCCNC(=O)C3=C(Cl)CCOC3)C2)ncnc2[nH]c(Cl)cc12 Cn1cc2cc(C(N3CC(NC(C4CC(C)(C)CO4)=O)C4(CC4)C3)=O)ccc2n1 C=CCCCCC(=O)N1CC(CNC(c2ncccc2NCC)=O)C(O)C1 Cc1ccc(C(C)C)cc1C(=O)NCCC(O)CNC(C1CN(C)C1)=O c1(C(N2CCC(NC(CN(C3CCC3)C)=O)C(O)C2)=O)ccc(C#N)c(O)c1 C(CCCC)(C(=O)NC(C)CCN(C)C)NC(C=CC=CCC)=O C(=O)(C(C)C(O)C(C)CC)N1C(C)(C(=O)NC2CCCC(C=C)C2)CCC1 C(=O)(C1COc2ccccc21)NCC=C1CCN(C(CC(C=C)(C)O)=O)CC1 C1(C(=O)NCCOC2CCOC2)CCC2(CC2)N1C(c1ccncc1O)=O c1(OC)ccc(CNC(=O)CN2CCN(c3ncc(F)cn3)CC2)c(Cl)c1O CCC(C(=O)OC)C(=O)NC(C)(C)CCNC(=O)C(C)OCC(F)(F)F c1(C(N(C(c2n(CC)nnc2)C(=O)NC2CCC2)C)C)ccc(Cl)c(Cl)c1 O=C(C1=COCC1)NC1C2CC(NC(c3cc(C4CCC4)on3)=O)CC12 Cc1nc(C)c(C(=O)NC2CCC(CC)C2)[nH]1.c1(C=O)scnc1C(C)(C)C Cc1nc(C)c(C(=O)NC(CNC(=O)C(c2cncn2C)O)C(C)C)s1 C(=O)(C1CCc2cccc(O)c21)N(CC(CNC(CC(CC=C)(C)C)=O)C)C CCC(C)CC(C)C(=O)N1CCC(CC(N2CC(C(N)=O)C2)=O)CC1 C1(NC(Cn2c(C)nnn2)=O)COC2(C1)CN(C(=O)CCCSC(C)(C)C)C2 c1(CC(=O)NCCNC(C2C3CCC23)=O)ccccc1O C1(C(=O)NCCOCCCNC(Cc2cc(C)[nH]n2)=O)CCCC(C)(C)C1 C(N=c1[nH]c(=NC(C)CC(N)=O)c2c(ncn2C)[nH]1)c1scc(CC)n1 C1(CN(C(CCC2CC(OC)C2)=O)C)CCCCN1C(c1ccsn1)=O C(C(C(=O)NCCc1ccccc1C)C(C)(C)C)NC(CCCCCSC)=O c1(NCC2S(=O)(=O)CCC2)cc(=NCC23CC=CCN2CCC3)[nH]cn1 C1(c2cn(C(C)C)nc2)NC(=O)N(CC(=O)NOCCCCCC2CC2)C1=O Cc1c(C(N2CCC(C)(CNC(=O)CCc3cnn(C)n3)C2)=O)nnn1C CN1CCN(C(C2CCNC2=O)=O)C(CNC(c2cccnc2N)=O)C1 c1(C(N2CCC(NC(C(CC)n3ccnc3)=O)C2)=O)cc(C)c(N)c(C)c1 C1(C(=O)NCC(CC)NC(=O)CC(C)COC)CCc2ncccc2C1 C1(O)(C(C=O)(F)F)CCOCC1.C(CCC=CC(=O)N)=C(C)C.C1CCC1.C c1(NC(C2(F)CCN(Cc3c(C)cc(Br)cn3)C2)=O)nccn2c(Br)cnc12 C1(COC(=O)NC2CCCOC2)CCCCN1C(=O)C(F)(F)F C(=O)(CC(F)(F)CC)NC1CCC(CNC(C2C(CCC)C2)=O)C1 c1(C(=O)NC2C3CN(C(C4(C(C)C)CCCO4)=O)C2C3)cc2cccc(F)c2o1 C1(C(=O)NCC2(C(=O)OC)CCC2)CCC2CCC1N2C(c1ccoc1)=O c1(OC)ccc(CO)cc1-c1nc(C(=O)NCc2ccnc(Cl)c2)ccc1F CN1CC(CNC(=O)CCC2CCN(C(=O)CCCC3CCCC3)CC2)CC1=O Cc1ccsc1C(=O)NC(C)C(CO)NC(C1(C#N)CC1)=O Cc1nc(C(C)C)oc1C(=O)NCC1CCCC1NC(=O)CS(N)(=O)=O c1(C(CNc2nccc(C(C)(F)F)c2)O)ccc(C#N)cc1 CCC(C)CCC(=O)N1CCCCC1CNC(c1ccc(OC(C)C)cn1)=O c1(-c2cc(C(N(CCCN(C)C(c3cc(F)n[nH]3)=O)C)=O)on2)ccc(Cl)cc1 Cc1nccc(Cl)c1C(=O)NCC1CC(NC(=O)CCn2ccnn2)C1 CC(C)CC(C)(O)C(=O)NCC1(O)CN(C(=O)C(C)(C)C(C)O)C1 C1(NC(C(c2ccccc2)NC(=O)C=CC2CCCC2)=O)CC12CCOC2 C(C(C)(C)C(=O)NCC1(F)CCN(C(c2ccn(COC)n2)=O)C1)OCC c1(C=O)ccnc(C2CCC2)c1.c1(C(C(N)=O)N(CC)CC)cccc(Br)c1.N C(CCC=O)NC(C)=O.CCCN(C(=O)CN(C)C(=O)C1CC1)CCO.N C12(NC(C=CCCC(C)C)=O)CCN(C(=O)Cc3cccc(F)c3F)CC1C2 C1(C(=O)NCC(CNC(C(C2CCOCC2)C)=O)O)(CF)CCOCC1 CC(C)C(CC(=O)NC(C)CCCCCO)NC(=O)C(C)C#N Cc1cc(C(=O)NC)nc(C)c1.C12CC(C1)CCO2.C1(C=O)CC2(CC2)CO1 C1(F)(c2cn(CCCOC)nn2)CCN(C(c2ccc(C(N)=O)[nH]2)=O)C1 N1(C(C2(C)CNC(=O)C2)=O)CC2CC(C1)N(C(=O)Cc1nc(C3CC3)cs1)C2 c1(NC(C2N(C(C(C)(F)F)=O)CC2)=O)ccc(N(CCO)C2CC2)cc1 CC(C)C(C(=O)NCC(CO)NC(=O)Cn1cc(F)ccc1=O)C(C)C N1(C(COCCOCC)=O)CCC2(CCCN2C(=O)Cc2cc(C)[nH]n2)C1 N1(C(C2CC3(CC3)CO2)=O)CCC2CC12C(N1CC(OCC(F)F)C1)=O C1(N2CC(C(C)NC(c3n(CC)nnc3)=O)C2)CCCN(CC(C)(C)C)C1=O Cc1oc(C(C)C)nc1C(=O)NCCNC(=O)CN1CC=CC1.C1CC1 N1(C(C2CC(C)(C)OC2)=O)CCCC(CNC(=O)CC2CCCC(F)(F)C2)CC1 C(=O)(C(C)C(=O)NC(CNC(c1cc[n+]([O-])cc1)=O)C1CCC1)OC C(=O)(CCCC(C)(C)C)NC(CC(C)C)C(=O)NCC(C)OC(F)F C1(N(C(C2CCN(C(CC)=O)C2)=O)CC)CCCN(C(c2ccnc(O)c2)=O)C1 c1(C(=O)NCC2N(C(C(CC)NC(C)=O)=O)CC2)cc2n(n1)CCN(C)C2 C(=O)(CC(C(C)OC)NC(c1cc(=N)[nH][nH]1)=O)N1C(COCC#C)CCC1 CC1Nc2c(C(=O)Nc3cc(Br)c(Cl)cc3Cl)cccc2NC1=O c1(NC(N(Cc2cc(C)c(C)o2)CC2CCC2)=O)nc(N2CCCC2)ncc1Cl c1(C(=O)NC2(CO)CN(C(C(c3cccnc3)OC)=O)C2)ccc(O)c(Br)c1 C(=O)(C(F)CC(C)C)NCCCC(C)NC(CSc1cccc(OC)c1)=O c1(CC(=O)NCC2CC(F)(CNC(c3cnccn3)=O)C2)ccc(Br)cc1 C1(CNC(=O)C2=COCCC2)CCCC2CN(C(=O)C(F)(F)Cl)CC12 N1(C(c2ncc(C)cn2)=O)CCCC2(CCN(C(C34CC(C)(C3)C4)=O)C2)C1 C1(C(=O)Nc2cc(C)ccc2)CC2(CO1)CC(F)(F)C2.C(=O)(CCC(C)(C)F)N c1(CN2CCC(NC(=O)CC(F)(F)F)C2)cc(Cl)ccc1Cl C1(NC(=O)NC(CN(C)C)Cc2ccccc2)CN2CCC1(C)CC2 C1(C)CC=CCC1.Cn1cc(OCC(=O)NC2(CCC(=O)NC)CCCC2)cn1 N1(C(CC(CC)C2CCC2)=O)CCC(CC)(NC(c2ncc[nH]c2=O)=O)CC1 C1(NC(C(Br)=C(C)C)=O)(CNC(=O)C(O)C2CCCC2)CCOCC1 N1(CC)CCN(C(=O)C(C(C)C)NC(C2(F)CC=CC2)=O)CC1C C(=O)(C(O)C(C)C)NC1(CC(=O)Nc2c(OC)nsc2)CCC1 c1(C(=O)OCC)cccc(CN2CCC(N(C)Cc3ccccc3Br)C2)c1 C1(NC(C(CNC(C)=O)C)=O)CCCCN(C(=O)COCCC(C)C)C1 c1(CC)c(C(=O)NC)nn[nH]1.C12CC1CN(C(C1(C(N)=O)CCC1)=O)C2 C1(c2nc(-c3ccc(C)o3)nn2-c2ccnnc2)CCC2CCC(=O)N12 c1(NC(N2CC(CC#C)C2)=O)c(F)c(F)c(Br)c(F)c1F c1(C(=O)OC)ccc(Br)c(S(=O)(=O)N2CCCC2C(=O)O)c1 c1(C(=O)NC2C(CNC(c3ncc(F)cn3)=O)CC2)ncccc1O C1(C(=O)NCC2(COC)CCN(C(c3scnc3C)=O)C2)CCc2c[nH]nc2C1 N1(C(C2N(C(C=CC=CCC)=O)CCC(F)C2)=O)CCC2(CC1)CSC2 N1(C(c2ccc(C)o2)=O)CCC(O)C(C(=O)Nc2c(C)nn(C)c2C)C1 C1(C(=O)NC(c2nc(C)sc2)C)CC(C)CN1C(C12CC(CO)(C1)C2)=O C1(CCC(N2CC(O)CC(NC(C(CC)=CC)=O)C2)=O)CCc2cnn(C)c2C1 c1(C(N2CCC(N(C(=O)CC3CCCC3)CC)C2)=O)cc(F)c(N)cc1F C1(N(C(=O)C(C)n2ccnc2)CC)CCN(C(=O)CC=Cc2ccccc2)CC1 c1(NC(CSC(C(C)OC)C)=O)cc2c(nn1)CCOC2 c1(C=O)cccc(C)c1N.Cc1nc(OC(F)F)c(C(=O)N(C)CC2CC2)s1.N N1(C(C(c2cccc(OC)c2)C)=O)CC(C)CN(C(=O)C(C)(C)OC)C(C)C1 C(c1ccc2[nH]ccc2c1)=CC(N1CC(N(c2ncnc(Cl)c2CO)C)C1)=O C1(NC(c2ccc(CO)c(F)c2)=O)CCN(C(=O)CN2CCOCC2)CCC1CO C(CCCCCNC(c1cccn1CC)=O)NC(C(CC)N(CC)CC)=O C1(N(C(C=O)C)C(=O)C(=O)O)COC2(CCN(C=O)C2)C1.C(C)(C)C.C Nc1ccc(C(=O)NC2CCN(C(=O)CC34COCC(C3)C4)C2)c2c1CCCC2 c1(C(N2CC(C)C(CNC(=O)CO)CC2)=O)cccc([N+](=O)[O-])c1O CSC1=C(C(=O)NCCC(C)N(C(=O)CCCc2cncs2)C)CCCC1 N1(C(CN(C2CCC2)C)=O)CC(C)(C)CC1CC(N1CCCC(C#N)C1)=O c1(C(N2C(CNC(CCc3cnc(C)s3)=O)CC2)=O)cc(C)n(CCO)n1 C1(COC)(NC(=O)CCc2nccs2)CCN(C(=O)C(F)CC2CC2)C1 CC1(C(=O)NCCC(Cc2ccccc2)NC(C2CCCC2O)=O)CCOCC1 S(=O)(=O)(c1ccsc1C(N1CCCCC1C)=O)N(C)C.c1(C(=O)N)cccnc1 C1CCCC1.C(=O)C(=O)Cc1ccccc1.CC(C(=O)NC)OCC1CC1 c1(C(=O)NCC(CNC(c2csnn2)=O)OC)cnc(O)c2cnccc12 N(C(=NCCNC(=O)OC(C)(C)C)N1CC2CCN(C)C2C1)CC(=C)CC N1(C(Cc2c(C)ccs2)=O)CCC(CO)C(NC(C2CCC3(CCC3)O2)=O)C1 c1(C(C(=O)NC)N(C2CC2)C)cccc(OC2CC2)c1.c1ccc(O)cc1 Cc1cnc(Cl)c(C(=O)NC2CC3(C2)CC(C(=O)N)C3)c1.c1cc(Br)cs1.C C1(C(=O)NCc2n(CCC)cnc2)CCN(C(=O)Cn2cc(CO)nn2)O1 N(C(=NCCF)NCc1cnc(-c2ccccc2)o1)C1C(C)CCCC1 CC1CN(C(=O)CCCN2C(=O)CCC2=O)CC1NC(=O)C=Cc1cnccn1 CCC(CC(=O)N1C(C(=O)N(C2CCCC2C)C)CC2CCCC12)C(C)C C(=O)(CCCN=[N+]=[N-])NCC(CC)NC(C1(C#C)CC1)=O c1(C(N(CCN(C(C2(C(=O)O)CC2C)=O)CC)CC)=O)ccccc1F c1(CN(C(C)C(=O)N(CC(O)CN(C(=O)C(F)F)C)C)C)ccccc1 C1(C)(C(=O)NCC(C)(C)NC(CN(CC)CC)=O)CC(=O)N(C)C1 C1(C)CC(F)(F)CN1C(C1CNC(=O)N1)=O.C1(C(=O)N)(OC)CCCCCC1 C(=O)(CCC(C)(C)C)N(CCCNC(CC1CC(CC)C1)=O)CCO N(C(=NCC(C)S)NC1CCC1)C1C(C)(OCC)C1.c1ccc(Cl)c(F)c1 Cc1cc(C(N2CC3CCC2CN(C(=O)C2CC2)C3)=O)nc2ccccc12 c1(C=O)cnn2ccc(Cl)c(F)c12.CC(F)(F)C1(NC(C2CC2)=O)CC1.C CCCCC(C(=O)N1C2CCC(C2)C1CNC(c1cnc(O)o1)=O)C(C)C c1(C(=O)NC(C(C)C)C(C)NC(C2(CF)CCC2)=O)cc(O)ccc1[N+](=O)[O-] Cc1[nH]c(=N)sc1C(=O)NC(C)CNC(C1C2COCC12)=O C(C(C)(C)C(=O)N1CCC(O)C1)NC(C)=O.C1(C2CCCO2)(C=O)CCC1.C Cc1ncn(O)c1C=O.C1(O)(C(C)C)CCN(C(=O)C)C1.C(=O)C(C)(C)C.N N(S(=O)(=O)N(C(C)CC#N)Cc1ccccc1Cl)(CC(C)C)CC(C)C c1(CCN(C)C)ccc(C(=O)NC)cc1F.C1(O)CCN(C=O)C1.C(C)(C)C CC1(NC(=O)CCOC2CCC2)CCCN(C(=O)CC(F)(F)F)C1 N1(C(C2(OC)CCCC2)=O)CCCC(C(C)(O)CNC(c2cc(Cl)c[nH]2)=O)C1 c1(NCc2nccc(NC)c2)ncnc(Nc2cc(C3CC3)cc(C)c2)c1C c1(C(=O)NC2CCC2)cc(O)c2cc(F)cc(F)c2n1.C1(C=O)CC(F)C1.C c1(C(=O)NC2CC(N(C(=O)C=CC3CCOC3)C)C2)c[nH]c(=O)cn1 N1(C(C2(C(CC)(F)F)CC2)=O)CCC2(CC1)CN(C(=O)C(O)C(C)(C)C)C2 CC1(C)C(CNC(=O)CC2=CCCC2)CCN1C(c1cccc(=O)o1)=O N1(C(c2nc(Cl)ccc2Cl)C(=O)NC)CCOC2(CCC2)CC1 N1(C(COC(C)(C)C)=O)CC(=O)NCC1C(=O)NC1CCNC(=O)C1 N1(C(CC(n2ccc(C)n2)C)=O)CCN(c2cc(F)ncn2)C(CCO)C1 Cc1cc(C(F)(F)F)nc(NC2CCN(C(=O)Cc3ccc(F)cc3F)C2)n1 C1(NC(C2(C)CC(O)CN2C(=O)CCC2CCOCC2)=O)CC2C(O)C(O)CC12 c1(NC(=O)NC(c2cc(OC)c(F)cc2)C)cc(S(N)(=O)=O)c(C)cc1C c1(CN2CCN(CCCNC(c3cccc(I)c3)=O)CC2)ccc(Cl)cc1Br N1(C2CCCN(C(CCC(=O)NC)=O)C2)CCN(C(C)C(=O)N)CC1=O.C1CC1.C N1(C(c2c(CC)oc(C)c2)=O)CCCN(C(C2CC(F)C2)=O)CC1C C(=O)(CS(=O)(=O)C1CC1)NC12CC(NC(CC(C)c3cccnc3)=O)(C1)C2 c1(C(=O)NCC2(C(N3CCCC(CCF)C3)=O)CC23CCC3)cc(O)ncc1F O=C(N=c1ccc(C2CCCCC2)n[nH]1)c1ccccc1C1CCOC1 S(=O)(=O)(c1cccc(N2CCCC(CNn3ccnn3)C2)n1)N(C(C)CC#N)C CC(C)(C#N)CCC(=O)N1CCCC(C(N2CC3(CSC3)C2)=O)CC1 c1(CN=C(NCC2CC(=O)c3c(cccc3)O2)NCCl)cnc2c(F)cccc2c1 N(C)(C1CN(C(c2cc(F)ccc2C)=O)CCc2ccccc21)C(C(CC)O)=O c1(CNC(CC2(N(C(C3(SC)CC3)=O)C)CC2)=O)cccc(O)n1 c1(OC)ccc(CN2CC3C(CN=[N+]=[N-])C3C2)c(C)c1 C(CC(C)C(=O)N(C1(C)CC(NC(=O)CC)C1)CC)OC.c1ccc(C)cc1 c1(C(=O)OCC)nccc(N2CCCC(CCNC(C3CSCCS3)=O)C2)n1 Cc1ccc(C(=O)NCC2C(C)CCCN2C(=O)C=C2CC2)c(=O)n1C C1(NC(C(C)CO)=O)CCCC2CN(c3ccc([N+](=O)[O-])cc3)CC12 c1(C(COC)(C)O)cn(CCNC(c2ncsc2-c2ccccc2)=O)nn1 C1(CNC(Cn2c(C)nc(C)n2)=O)N(C(=O)CC(C)C(C)C)CCC1(C)C c1(C(=O)NC2(CNC(c3ccc(CO)o3)=O)CCOC2)cc(F)ccc1O C1(C(=O)NCC2CC(NC(C3CC(n4cccn4)C3)=O)C2)CCNC1=O Cc1cc(NC(=O)CC2CCN(C(c3cc(Cl)c(O)cc3F)=O)C2)c(I)cc1F C(CCCC(C)NC(=O)Cc1csc(C)n1)NC(C1(c2cc(C)no2)CC1)=O c1(C(N2CCCC(CC(N)=O)C2)C(=O)NCCC)ccc(Br)cc1C c1(C(N2CCN(C(=O)CCn3cncn3)C(C(F)F)C2)=O)ncn2ccccc12 c1(C(=O)NCC2CC(NC(=O)C3=NOCC3)CC2O)csc2ncnc(O)c12 C(CC(C)(C)CO)CNC(C(N1CCC(c2nc(C)on2)C1)=O)=O C1(CC(C)(C)C)CN(C(=O)CNC(C2CCC2(C)C)=O)CCO1 c1(NC(C(C)C)C(C)NC(=O)C2=C(Cl)CCOC2)cnc(C#N)c(C#N)n1 CS(=O)C=CC(=O)N(C1CCN(C(c2ccccc2CC2CCC2)=O)C1)CCO C1(C(=O)NC(CCC)C(F)F)CC2(C1)CC(N)CCS2 C1(C=O)CCc2nccn2CC1.CC1(C)NC(=O)CC1C(=O)NCC1CCC1.N n1(CCC)nnc(=NC(=O)c2cc(OC)cc(Cl)c2)[nH]1 c1(OC)ccc(C(N2CC3CC2C3NC(=O)Cc2csc3nccn23)=O)c(F)c1 C1(NC(C(c2cscn2)N(C)C)=O)CCCCCN(C(=O)Cc2ccoc2)C1 c12cnc(s1)Cc1ncoc1COC2=O.C(=O)CCN.COC C1(N(C(C)=O)CCN(C(C2(c3ccno3)CC2)=O)C(C)C)CCCCC1.C c1(C(=O)NC(CC(C)NC(COC)=O)C)ccc(Cl)cc1 N1(C(c2cc3scc(Br)c3[nH]2)=O)CCC2(C1)OCc1ccccc12 C1(NC(c2cc(=O)cc(Cl)[nH]2)=O)CN(C(c2ns[nH]c2=O)=O)C2(CCC2)C1 c1(OC)ccc(NC(C2CN(C(c3ccc(O)cn3)=O)CCS2)=O)c(C#N)c1 C(=O)(CCN(OC)C(=O)CC1CCCC2CC12)NCc1cn(CC)nn1 c1(C(=O)NC2CC3(C2)CN(C(c2cnnc(O)c2)=O)C3)c(F)cccc1[N+](=O)[O-] c1(N2CC(=C(CNC(C3=C(C)CCCC3)=O)F)C2)ncnc2c1ncn2C C1(C(N2CC(NC(COCC)=O)C(C)(C)C2)=O)CCCC(C)(C)CC1 N1(C(=O)CC2C=CCCC2)CCC2(CC1)CN(C(C1(O)CCOCC1)=O)CCO2 N1(C(C(N2CC(F)(CNC(CCCC)=O)C2)=O)C)CCP(C)(=O)CC1 c1(CC(=O)OC2CCC(COC)C2)cnc2ccc(Br)cn12 C1(C2(NC(CC(=O)NC3CC3)=O)CC2)CCCCN1C(c1cncc(Cl)c1)=O Cc1cc2c(C(=O)NCC(C)NC(C34CCC(CC3)CC4)=O)cccc2o1 C(CN(C)CC1(N)CC1)(CO)OC C(C(C(=O)N(C)C)C(C)C)NC(CN1CCC(n2cc(CCCC)nn2)CC1)=O C1(c2nc(OC)c(C)s2)CCCCN1N(CCCO)C1CC1 C(CS(=O)(=O)CC(=O)NC1CCCCCN(C(C2CCC3(CC3)C2)=O)C1)OC CCC(CC(C)C)C(=O)NCCN1CCN(C(=O)C(C)(C)c2cnn(C)c2)CC1 C1(CNC(c2ncc[nH]2)=O)(Cn2cc(C3CCOC3)nn2)CC12CCC2 N1(C(C(COC(C)=O)C)=O)CCC(C)(C)C(C(=O)NC(C)(CO)C(C)C)C1 c1(OC)ccc(Cl)c(C(=O)NC(CNC(=O)CCc2ccon2)C(C)C)n1 N(C1CCc2ccccc21)C(CCN(C(C(C)(C)OCC)=O)C)=O N1(C(CC2(OCC)CC2)=O)CCC(CC)CC1C(=O)NC(C)CC(C)C C1(C)(C(N2CCC(CNC(C=COCC)=O)C2)=O)CC(=O)N(C)C1 C12(CCNC(=O)COC3CC=CC3)CCC(CC1)C2.C1(O)(C=O)CCSC1 c1(C(=O)NCCCCCCNC(CC(=C=C)C)=O)ccc2cncc(Br)c2c1 Cc1cc(C(N2CC(C)(NC(c3ccccc3Cl)=O)C2)=O)ncc1C(N)=O CC1COCC1N=c1[nH]c(NC2CCOc3c(Cl)cccc32)nc2ccsc12 C(CCCC(=O)NC1CN(C(c2cc(C(F)(F)F)on2)=O)CC1C)NC(C)=O Cc1c[nH]c(=NCCC2CCN(C(C3CCOC(C(C)C)C3)=O)C2)nc1SCCO C1(NC(C(C)CF)=O)CC2CCC(C1)N2C(c1ccc(O)cn1)=O C1(C)(C(N(CC(CNC(c2c(C)nc(CO)o2)=O)O)C)=O)CCC(F)(F)CC1 C1(NC(C2(CC)CCC2)=O)CN(C(c2ccnc(C)c2N)=O)C2(CCOCC2)C1 C1(C(N2CCC(CC)CC2)=O)CC2CN(C(=O)CCCC#N)CC2C1 N#CC1CN(C(c2ccc(F)cc2F)=O)CCN1C(=O)CC1CC1 c1(C(=O)NC2C(OC)CN(C(C3CCCCS3)=O)C2)cnc2ccnn2c1 c1(CCC(=O)NCC(C)N(C)C(c2nnn(C)n2)=O)c[nH]c2ccccc12 c1(CN(C(c2cnn(-c3ccc(Br)cc3)c2)C(=O)NCCC)C)cccc(Cl)c1 C1(CS(=O)(=O)NC2(C)CCCCC2O)CCC(F)(F)C(=O)N1 CC(CC(=O)N1CCC(NC(=O)CC2CSCCO2)C(O)C1)CC(C)(C)C c1(C(N2CCCC2)=O)oc2ccccc2c1CN(C1CCCCCC1)c1cccs1 C(CC(=O)NC)(C(C)C)OCC.C1(C)CCN(C(=O)Cc2csc(C)c2)C1 C1(NC(CCSCC(N)=O)=O)CCCCC12CCN(C(c1ccnnc1)=O)C2 C(=O)(C1=C(C#N)CCC1)N1CC(C)C(NC(c2nn(C)nc2Br)=O)C1 Cc1ncc(CC(=O)NC(C2CCCC2)CNC(=O)Cc2ccon2)[nH]1 C1(C2CCC2)(C(N2CCC(c3n(C)c(S)nn3)CC2)=O)CCC1 C1(CNC(c2cnc(C)n2C)=O)CC12CCN(C(=O)C(C)OC1CCOC1)CC2 N1(C(C2(C)ON=C(C)C2)=O)CCC(N(C(=O)CCC2(C)CC2)C)C2(CC2)C1 c1(CN(c2nnc(C3CC3)n2CC(C)(C)CN(C)C)CCC)ccc(F)cc1 N1(CC(N2C(CNC(=O)C(F)C3CCCC3)CC2)=O)CCC(=O)NC1=O c1(C(=O)NCC(C)C)cccc(S(=O)(=O)N(C(CO)C(C)C)C)c1 N1(C(CCCCCC)=O)CCC2(CC1)COC(CNC(c1csc(C)c1N)=O)C2 C12(OC)CCN(C(c3cc4occc4n3C)=O)CCC1C2 Cc1cc(C)c2c(c1)C(N(C)C(=O)NCC13COCC1C3)CCO2 c1(-c2cn(C3C(NC(c4c(C)noc4C)=O)CCC3)nn2)ccc(C#N)c(Cl)c1 N1(C(C2C(=C)CC2)=O)CCC(NC(c2ccc(-c3cccs3)s2)=O)C2(CCC2)C1 C1(CC(=O)NCC2N(C(COC(C)C)=O)CC2)OCCOC1(C)C CCC(C)C(O)C(C)C(=O)N1CCC(C(=O)NCC2(C(N)=O)CC2)C12CC2 N1(C(C(C)O)=O)CCC(C)C(CNC(=O)C=C2CCCCC2(C)C)C1 C1(NC(c2c(C)cns2)=O)CN(C(c2cc(CO)on2)=O)CC1c1ccccc1 Cc1ncc(C(=O)NC2CN(C(c3ncoc3C3CC3)=O)CCC2F)cc1C#N N1(C(C(C)=CC)=O)CCC(C)C(NC(c2cc3ccncc3s2)=O)C1C c1(C(=O)NC2(C(N3CC(CC)C3)=O)CC(O)C2)cccc(O)c1C c1(CC(N2C3C(NC(C(CC)OC)=O)C(C3)C2)=O)nnc(O)c2ccccc12 c1(N2CCN(C(C(=O)NC(c3ccc(F)c(F)c3)C)=O)CC2)ccc(F)c(F)c1 CC1=CCC(C(N2CCOC(CNC(=O)Cc3cccnc3C)C2)=O)CC1 CC12CSCC1CN(C(=O)CCC1CCCCN(C(c3ccsc3Cl)=O)C1)C2 C(c1c(Cl)cccc1Cl)=C(C)C(=O)N(C)CCNC(=O)CC1COC(=O)N1 C1(NC(c2cnns2)=O)CCN(C(=O)C2CC2)C12CC2 Cc1nonc1CC(N1CCCC1C(C)(C)C(=O)NC1CC(N2CCCC2)C1)=O C1(NC(c2ccc3c(c2)CCC3)=O)CC(C(=O)NC2COC3(CCC3)C2)=CC1O c1(C(=O)NC(CCC)C(N2CCOCC(C)C2)=O)cnn2ccoc12 c1(C(=O)NCc2c(C)cc(Br)cc2)cncc(C2=CCOCC2)n1 Cc1cc(O)ncc1C(=O)NC.C1(CC=O)CCC2(CCC2)O1.C1(F)CCC1 c1(SC)cccc(N2CC(NC(c3ccc(CO)o3)=O)CC(C)(C)C2)c1[N+](=O)[O-] c1(C(N(C2C(C)CCC2)C)=O)ccc(CO)cn1.C1(=O)CC=CCN1 CCCC(C(=O)NC1CN(C(=O)CCOCC(F)(F)C(F)F)C1)OCC c1(C(=O)NCC2(F)CN(C(c3nc(C)oc3)=O)C2)ccccc1S(C)=O N1(C(c2cccc(CC)c2)=O)CC(C)CN(C(=O)CCS(C)(=O)=O)CC1C C(C(COC)CC(=O)N1CCOC(C)(C)C1)OC.c1(C(C(=O)N)C)ccc(Cl)s1 c1(C(=O)NC(CC)CNC(=O)CC2CC(F)C2)ccc(CC(N)=O)cc1 c1(C(=O)NCCCNC(C(=Cc2cccc(Cl)c2)C)=O)cnn2c1NCC(C)C2 c1(C(=O)Nc2cc(C)cc(Cl)n2)ccn2cncc2c1 Cc1onc(O)c1C(N1CCC(N2CCN(C(C3CCC(C)O3)=O)CC2)CC1)=O c1(C(N(CC(C)NC(C2CCC2(F)F)=O)CC)=O)ccnc(S)c1 N1(C(c2nc(CCC)sc2)=O)CCCC(CNC(c2cccc(O)n2)=O)C1 C=C1COc2c(C(=O)N(C(CNC(=O)Cc3ccccc3)C3CC3)C)cnn2C1 N1(C(C2CC(=O)NC2)=O)CCCC(CCCCNC(=O)C)C1.[SH](=O)(=O)C1CC1 C(CC(O)CNC(=O)Cc1ccns1)NC(=O)Cn1cncn1 C(C(=O)NCC1(C)CCN(C(c2cc(O)cs2)=O)C1)(C(C)(C)C)OC.O C1(C(=O)OCC)CCCN(C(=O)Cc2ccccc2)C1.c1(C(=O)N)nn[nH]c1Cl c1(N(C)C)ccc(CN2CCN(C(=O)Cc3cccc(I)c3)C3CC23)c(O)c1 n1(C(C(=O)OC)C)cc(CSCCNC2CCOC2=O)nn1 CCC(C)CCCCC(=O)N1CC(NC(=O)CN2CCCCC2=O)CC(F)C1 C(=O)(CCC(C)(C)C)NC(C)C(=O)NC(c1cnn[nH]1)C c1(-c2cn(CCCCNC(c3c(C(=O)OC)coc3)=O)nn2)ccc(F)c(F)c1 N1(C(C(C)NC(Cc2nc(C)oc2)=O)=O)CCn2nncc2C1 C1(C(=O)NCC(C(C)C)NC(=O)C2=C(Cl)CCC(C)C2)CCc2c(cnn2C)C1 C1(CNc2cc(N(CC(C3CCCCC3)C)C)ncn2)Cc2cc(Br)ccc2O1 c1(C(=O)NC(CNC(C=C(CCC)C)=O)CO)c(COC)nn(C)c1Cl N1(C(C2(C(C)C)CC2)=O)CCC(C)C1.c1(C=O)cnccc1C(F)(F)F.C N1(C(C(N2CCC(C3N(C(C4CC(C)C4)=O)CCC3)C2)=O)C)C(C)CCC1C C1(CNC(c2c(C)n[nH]c2)=O)CCCCN(C(C23CCC(CC2)O3)=O)C1 N1(C(c2scc(C)c2)=O)CC(CNC(C2CC(C3CCC3)C2)=O)C2(CC2)C1 N1(C(c2[nH]n(C)c(=O)n2)=O)CCC2(NC(c3cc(N)ccc3Br)=O)CC2C1 C(CNC(c1nn[nH]c1Cl)=O)(CC(F)(F)F)NC(C1CCN(C)C1=O)=O N1(C(c2nc(OC)oc2)=O)CC2CC1C2NC(C1CCN(C)C1=O)=O CCC(C#N)C(=O)N1CC(=C(F)CNC(=O)CSSC)C1 C(=O)(C#CC1CC1)NC(C(=O)NCC1CC(N(C)C)C1)C1CCCO1 C1(CC(=O)N(CCNC(=O)C(C)(C)c2cnc[nH]2)CC)CCCCCCC1 CC1(C(=O)NCCC2CC2)CCS(=O)(=O)CC1.c1(C=O)cc(C#N)ccc1F C1(CC)CSCCN1C(c1ccnn1C1CCCC1)=O.C(C)(C(=O)N)NC(C)=O C(=O)(C(F)(F)C(O)C(C)C)NC(CC=C)CNC(c1cncc(C(F)F)c1)=O N1(C(CC(C)C2CCCCC2)=O)CCC(O)(CCNC(=O)C=Cc2ccco2)C1 c1(NC(CC2OCCN(Cc3c(C)cccc3)C2)=O)scc(O)c1C#N c1(C(=O)NC2CC(C)(CNC(=O)CN3CC=CC3)C2)cc2cn[nH]c2cn1 CN1CCC(N2CCCCC2)(CNC(=O)CCCC(N)c2ccccc2)CC1 N1(C(CSC2C(=O)OCC2)=O)CC2CCC1CN2C(=O)CC1CC2CCC1CC2 O=C(C1SCCc2ccccc21)N1CC(Nc2ncnc3ccccc23)C1 c1(C(C(=O)Nc2ccccc2)N(CCC2CC2)CC)ccc(C)c(OC)n1 C(=O)(CCC(=O)NN(C)C)NC(CC(=O)NC(C#C)CC(C)(C)C)C(C)C N1(C(C2OCCN(C(C(C)C)=O)C2)=O)CCn2nccc2C1 C(C(C)(O)C(F)(F)F)NC(CCC1N(C(C2C3CN(C)CC32)=O)CCCC1)=O C1(NC(c2cnn(CCC)c2C)=O)CC2CC1CN(C(=O)C=CCOC)C2 c1(OC)cc(Cl)ncc1C(=O)NC1CN(Cc2c[nH]nc2C)C1 c1(C(=O)NCC(C)C)oc2ccccc2c1CO.C1(C(C)(F)F)(C=O)CCC1 N1(C(C(C)SC)=O)CC(NC(c2cc3ccccc3cn2)=O)C(S(C)(=O)=O)C1 c1c[nH]c2ccccc12.c1(N(C)C)cc(NCCC2CC2C2CC2)ncn1 C(=O)(CCC(C)(C)N1CCOCC1)NC(C)CN(C(=O)C(C)C1CC1)C C(C)(CCCCNC(=O)CSCc1cccs1)NC(C(c1ccccn1)C)=O C=C(C)CC(C(=O)NCc1coc(C)n1)NC(=O)CC(O)C(C)C C(=O)(C(C)CC(C)(F)F)N1CCC(N(C(c2cc(OC)nc(C)c2)=O)CCO)C1 C1(NC(C2CCN(CC(F)F)CC2)=O)(C)CCOCC1.C1(C=O)CC2CC2C1.N c1(C(C)C)c(C(=O)NC(C)CCNC(=O)C(C)(C)c2ccsc2)cnn1C c1(-c2n(CCC)nc(-c3ccc(Cl)nc3)n2)cccc(C#N)c1Br N1(C(C2N(C)CCCC2)=O)CCCN(CCNC(C2CSCC(=O)N2)=O)CC1 N1(C(c2ccc(OC)s2)=O)CCC(NC(C2CC(C)(C)C2)=O)C(C)(C)C1.C N1(C(C2CC(C(N)=O)C2)=O)CCCCC1CC(N)C(F)(F)F c1(C(N2C(CNC(=O)C#CC3CCCO3)COCC2)=O)cc2c(nc1O)CCC2 c1(CNC(=O)NC(C)C(=O)N2CCCC2)nc(Br)n(C)n1 Cc1nc(C2CCCO2)sc1C(=O)NC(C)C(C)NC(=O)C(O)C(C)C C(CCCC(C)(C)C)NC(CCCN(C(=O)CS(C)(=O)=O)C)=O CCC(C)(C)C(=O)C(=O)NC1(CC(=O)NCC(C)(C)C)CC1 c1(NCc2c(C)n(C)nc2)[nH]c(=NC(C)C2CCCO2)nc2c1ncn2C(C)C C1(NC(c2c(CC)nccc2)=O)CN(C(C2OCCC2(C)C)=O)CCC1C C(=O)(C1=CNC2=NCCC2=C1)N1CCC(O)(CNC(CCCCC(C)(C)C)=O)C1 C1(NC(C2CC(=C)C2)=O)C(C)CCN(C(=O)C=Cc2cccc(C)c2)C1C C#CC(CC)(CC)NC(C1CC(O)CN1C(c1ccc(C(C)=O)o1)=O)=O Nc1c(C(=O)NCC2(F)CCC(NC(c3ccnc(CO)c3)=O)C2)cccc1F N1(C(c2ccc(C#C)nc2)=O)CC2CCOC2(CNC(c2cc(OC)no2)=O)C1 CC1(C)C(NC(C2CCCCC2)=O)CCN1C(C1CCCC1C1CC1)=O c1(SC)cc(C(=O)NCC2CC(Nc3cc(C(F)(F)F)ncn3)C2)ccn1 CCC(CN(C)C)N=c1[nH]c(=NCCCN2CC=CC2)c2ncccc2[nH]1 C12(C(=O)NCC3CC(NC(CC(CN(C)C)O)=O)C3)CCCC1CCC2 N1(C(COCCOC)=O)CCC(C2CCCN(C(c3cnc(C)nc3C)=O)C2)C1 Cc1nn(C)c(C(N2CC3CC(NC(=O)CCC4CC4(Cl)Cl)C3C2)=O)c1[N+](=O)[O-] C1(C(=O)NCC(CNC(C=C(c2cn(C)nc2)F)=O)F)CCc2nc[nH]c2C1 c1(OC)cc(N2CC(CCCCNC(=O)CC3(C)CCCO3)C2)ncn1 c1(C(=O)NC2C(NC(=O)C=CCO)COC2)c(F)ccc(Cl)c1F c1(C(=O)NCC2CC(NC(C=CCCC)=O)C23CCC3)ncc2n1CCCC2 c1(CC)nc(NC2CC(C)N(C(c3ccnn3C)=O)C2)c2ccsc2n1 C=CC(CC)CC(=O)NCCC(C)(C)CNC(c1cnccc1C(F)F)=O C1(CCC)(NC(C2CC3(C2)CC3F)=O)CCCN(C(=O)CCCn2cccn2)C1 C1(CNC(=O)Cc2ccc(Br)c(Br)c2)CCNCC1C1CC1 CCC(CC)(CCNC(=O)CN1CC(C)(C)C1)NC(c1n[nH]cc1Cl)=O C1(CNC(c2n(C)ncc2)=O)N(C(c2ccc(CF)cc2)=O)CCCC1(C)C c1(OC)n[nH]c(C(=O)NCCN(C)C(C2CCCSC2)=O)c1Cl Cc1c(CC(N2CCC(CF)(NC(=O)C3=NOC(C)C3)C2)=O)oc2ccccc12 CC(C)C(C)C(CNC(c1cn(C)cn1)=O)N=c1[nH]nc(C2CC2)s1 N1(C(Cc2c(C)cccc2)=O)CCCC(C)(CNC(c2ccoc2C(C)C)=O)C1 c1(C(=O)NC(CN(C(=O)C(=Cc2cn[nH]c2)C)CC)C)cc(C)n(C)n1 N1(C(c2c(C)sc(Br)n2)C(=O)NCCCF)CCOCC(O)C1 C1(C(=O)NCC(CNC(C(CC=CCC)C)=O)C)CC2COCC(C1)C2 c1(C(N(CC)CCOC)=O)cnc(C2CC2)cc1C.CCC(C)OCC(=O)N C(=O)(C#CC1CC(F)(F)C1)N1C(CNC(C=Cc2c(C)cncc2)=O)CCCC1 C1(OC)(CNC(c2nonc2N)=O)CCN(C(c2cnnc(C)c2)=O)C1 C1(C(CC)O)CCCN1CCC(C)OC(C)(C)C C12(CO)COCCN1C(=O)OC2.C(C)(C)(CC(=O)OC(C)(C)C)N(C)C CC1OCCC1(C)C(=O)NCC#CC(=O)NCCCn1cccn1 c1(C(=O)NCC(C2(O)CCN(C(=O)CN(C)CCO)C2)C)cccc(CO)n1 C1(CC#C)CCCCN1C(=O)Cc1scnc1C(=O)O c1(NC(c2noc(C)n2)C(=O)OCC)ncnc2cccc(F)c12 Cc1ccccc1Cn1nc(-c2ccco2)nc1C(C)CCCc1ccccc1 c1(C(=O)NC2CC2C(=O)NC2CC2(F)F)cc2cccnc2s1 Cc1[nH]nc2c(C(=O)NCC(C)S(C)(=O)=O)cccc12.C1(C=O)CS(=O)C1.N CC(C)C(F)(CNC(C1CCC1C(C)(C)C)=O)C(=O)NCc1ccsc1 c1cc2n(n1)CCCO2.n1(CCC(=O)OCC)nnnc1CC1(C)CCCS1.N c1(C(N2C(CC)CN(C(=O)CC3CCOC3=O)CC2)=O)cc2ncccc2s1 C1(NC(C2C(C=C)CC2)=O)CC2CCCC(C1)N2C(c1ccc(C)c(Cl)c1Cl)=O c1(C(N(C2CCC(NC(CSCCCC)=O)C2)C)=O)cc2cn[nH]c2cn1 N1(C(c2cncc(C)c2)=O)CCC(C2CC2)(NC(=O)Cc2ncoc2C)C1 N1(C(CCC2CCCN(C(c3cc(C)sc3C)=O)C2)=O)CCC2(CCOC2)CC1 CC1(C)OCCOC1CC(=O)NC1CCCCC1NC(=O)CCc1cn[nH]c1 CCCC(CCC)=CC(=O)NC1CCCC(CN(C)C(C2(O)CCCC2)=O)C1 c1(CN2CC(C(N3CCC(CN(C)C)CC3)=O)OCC2)ccc(Br)c(C#N)c1 N1(C(c2ccc(OC)nn2)=O)CC(NC(c2cnc(C)[nH]2)=O)CC12CCOC2 c1(C=O)cn(C)nc1-c1nccs1.C1(CC)(OC)CN(C(c2cc[nH]c2)=O)C1.N N1(C(C2CC=CCC2)=O)CCC2(CCCN2C(C2CC3CCC3C2)=O)C1 N1(CC2CN(C(C)=O)C2)CC(C)(C)OC2(C1)CN(C(=O)C(C)(C)C1CCC1)C2 C(=O)(CC(C(F)(F)F)NC(=O)C1=C(Cl)CCOC1)NCCC(CC)(C)C C1(NC(C(CCC)CC)=O)CC2CCC1CN2C(c1cc(CC)sn1)=O c1(C(N2CC(COC)C2)=O)ccc2ccc(Cl)cc2n1.C(=O)C.C(C)(C)C.N N1(C(Cn2c(C)ncc2)=O)CC2CCCC(NC(c3cc(=N)[nH]c(=N)[nH]3)=O)C2C1 c1(C(N(CC(C)C)C)=O)ccc(CC(N)=O)cc1.C(c1cc[nH]c1)=CC(=O)N c1(C(N(CC(C)O)CC)=O)cnnc(O)c1.c1(C2C(C(=O)N)C2)cncn1C C1(C(C)C)CN(C(C2CC23CCCCC3)=O)CCN1C(c1cnnn1C(C)C)=O c1(C(N2CCC(N(C(=O)C(=O)N(C)C)CC)C2)=O)ncc(Cl)c(N)c1Cl C(CC(C)C(=O)N1CCC(C(C)NC(=O)CNc2nccc(OC)n2)C1)OC c1(SCC(N2C(C(N3C(CCN(C)C)CCC3)=O)CCC2)=O)ccc(F)cc1 c1(C(=O)NC(C)(C)CNC(=O)CCCC2CCOCC2)cncc2c1CCC2 N1(C(CCc2cc(C)on2)=O)CCN(C(=O)C(C)Cc2ccco2)C2CCCC12 c1(C(N2CC(SC)C(NC(c3c(Cl)nn(C)c3Cl)=O)C2)=O)cc(C)c(F)cc1N C1(NC(=O)C(=O)NC2C=CCCC2)CCC(O)(c2cccc(F)c2)CC1 c1(C(=O)NC2CN(C(C3CSC3)=O)C2)cccc(C(=O)C2CC2)c1 c1(OC)ccc(CC2CC2)cc1.C(c1nnc(-c2ccc(Br)cc2)o1)=CC=O.N C1(CCCCN(C(=O)CC2CCOC2)C)CCN(C(=O)OC(C)(C)C)CC1 C1(CNC(c2cc(C)c(O)nn2)=O)CCC2(CCC2)CN1C(C1CCCOC1)=O c1(C(=O)NC(C)CC(C)NC(=O)CCCCCN(C)C)coc2c(Cl)cccc12 c1(C(=O)OC)cc(C(=O)NC2CC2NC(c2cnsc2)=O)c(C)s1 c1(C(NNC(=O)NC(c2ccc(C)o2)C(F)(F)F)=O)cc(S(C)(=O)=O)ccc1F N1(C(COCC#C)=O)CCN(C)C(C)C1.c1(CC)cc(C)ccc1OC(F)F c1(CNC(=O)NC(c2nc(C)on2)(C)C)sc(C)cc1Br N1(C(C(C)=CCC)=O)CC(C)(C)CC1C(=O)NCc1cccc(F)c1C c1cc2c(s1)CCC2.C(C)(C)CC.C(C)(C(=O)N)NC(=O)NC.C(=O)C CC#CCCCCN=c1ccnc(NCCC2OCCCC2(C)C)[nH]1 CC(C)CCC(O)C(=O)NCC(CC(=O)NCCc1cccc(F)n1)C1CCC1 O=C(N=c1[nH][nH]c2cccnc12)C1COCCN1 C1(O)(CCNC(c2cnc(Cl)[nH]2)=O)CCCN(C(=O)Cc2ccc(F)cc2F)C1 CCCCCC(C)(C)C(=O)N1CC=C(CNC(=O)CCCCCN(C)C)CC1 C1(C(=O)NCc2ccc(C)cc2)CCC(C)CN1C(=O)CCc1cnc(C)o1 c1(N2C(CNC(c3cccc(F)c3F)=O)CC3(CC3)C2)nc2ccc(F)cc2s1 N1(C(c2c(C)coc2)=O)CC2N(C(=O)CC3CCCC(C)(C)C3)CCC2(C)C1 c1(C(=O)NCCN(C(c2ncoc2-c2cnn(C)c2)=O)CC)n[nH]c(C)n1 N1(C(C(CC)N(C)C)=O)CCCC(NC(C2CC(=C3CC3)C2)=O)CC1 C(=O)(CC(C)(C)CC(=O)N1CC(NC(=O)CCc2ccncn2)CC(O)C1)OC C1(CC(=O)NC)CN(C(c2cnc(OC)nc2)=O)CCN1C(=O)Cn1nccn1 C(=O)(C1CCCc2nn[nH]c21)NC(CNC(Cc1ccc(OC)cn1)=O)C1CC1 C1(S(=O)(=O)c2ccccc2)(C(N2CC(CNC(CSCC)=O)C2)=O)CC1 CC1(C)CC(NC(c2cccc(N)c2O)=O)CN1C(c1ccco1)=O C12(NC(CCNC(=O)NC)=O)CCCC1N(C(c1ccncc1N)=O)CCC2 c1(SCC#N)ccc(NC(=O)CCCn2cc(CCN3CCCC3)nn2)cc1 C1(C(=O)NC23C(CN(C(c4n(CC)ncc4Cl)=O)C2)C3)(CC)CCCCCC1 c1(OC)ccc2[nH]c(C(N3CC(NC(c4cccn4C)=O)C(C)(C)C3)=O)cc2c1 N1(c2nccc(C#N)n2)CCOCC12COCCN(C(c1cccc(F)c1)=O)C2 C1(C(=O)NC(C)Cc2cn[nH]c2)CC12CCN(C(=O)CC1(C#N)CC1)C2 c1(CN2CC(CC(N3Cc4cncnc4C3)=O)OCC2)cccc2ccoc12 N1(C(Cc2scc(C)c2)=O)CCC2(NC(c3cc([N+](=O)[O-])cn3C)=O)CCCC12 CCCCC(C)CCC(=O)NC(CCF)C(N1CCN(C)CC1CCO)=O C(C1=CCN(C(=O)COC(F)F)CC1)NC(CN(C)C(=O)C1CC1)=O CN1CCC(CCNCC2(c3cccc(C(F)(F)F)c3)CCC2)OC1=O c1(N(C)CC2CCN(C(COC(CC)(C)C)=O)C2)c(C)cncc1[N+](=O)[O-] N1(C(C(CC(F)F)OCC(=C)C)=O)C2CCC(NC(=O)NC)C1CC2 N1(C(C2(OC)CCCOC2)=O)CCC(CNC(C2(C#N)CCSCC2)=O)C(C)C1 c1(C2(CNC(=O)NCC3CCN3C3CCCC3)CC2)ccc(Br)s1 CC(CNC(C1(F)CC=CC1)=O)C(F)C(=O)NCC1CCC(=O)O1 CN1CCCCCC1C(N1CC(C)(C)CC1CC(=O)NC1C2CCCCCC12)=O C1(O)(CC(=O)NC2C(CNC(C(CN(C)C)O)=O)C2)CCOCC1 c1(OC)ncccc1C(=O)NC1(CCNC(=O)Cc2ccoc2)CCCC1 CC1CC(NC(C2CCC=CO2)=O)CCN1C(=O)COCc1nccn1C CC12CC(C(=O)NC3CN(C(=O)CC(C4CC4)C4CC4)CC3F)C(CO1)C2 C12(NC(CCOc3ccc(C)cc3C)=O)CCCCCC1N(C(=O)C1CC1)CC2 C1(C=O)C(F)(F)C12CC2.C(=O)(CC(=O)N1CCC(C)C1)OCCC(C)C.N c1(-c2n(C(CC)CC)nc(COC(C)C)n2)ccnc2[nH]c(O)nc12 CCCCC(C(=O)NCc1cc(C)cc(C)n1)NC(=O)C(C)OCCOC C#CC1C(C=O)C1(C)C.N1(CCCC(=O)N(CCC)C2CC2)C(=O)CCC1=O CCC(COC)(CC)C(=O)NCc1ccoc1C(N1CC(C(N)=O)C1)=O N1(C(=O)NCc2c(C)c(Cl)ccn2)CC2(CCOCC2)CC1C c1(C(=O)NC(c2c(C(=O)NC(CC#CC)C)con2)C)cncc(CC)c1 CC(C)C(CCN(C(=O)CC1CC1C)C)NC(=O)CC(C)c1ccco1 c1(OC)ccc(Br)c(C(=O)N)c1.c1(C2(C(N3CCCC3)=O)CC2)ccnc(Cl)c1 c1(C(=O)NCC(C(C)C)NC(C2C(CCC)C2)=O)cc(CC)cnc1O N1(C(CC(C)NS(C)(=O)=O)=O)CCCC2(CCN(c3cc(C)ncc3C#N)C2)C1 C(CCC(C)CC(=O)N1CCC(NC(c2c(F)cccc2F)=O)C(F)C1)=C(C)C c1(C(N2CC(CCC)N(C(=O)C(C)C(O)CC)CC2)=O)nccc2ncncc12 N1(c2snc(C(=O)OC)n2)CCCC2(NC(=O)CN(CC(C)(C)C)C)CC2C1 c1(C2(C(N(CC(CC)NC(=O)C=Cc3ccsc3)C)=O)CC2)ccncc1 c1(C=O)ccc2sc(C)nc2c1.CC(C1CC1)=C(F)C(=O)N.C1(CC)CC1.C C(CCCCCNC(c1ccnc(C2CC2)n1)=O)NC(=O)COCC1CC1 c1(C(=O)OCC)ccc(NC(=O)Cc2cccc(OCC(C)C)c2)cc1Cl N1(C(c2n(CC#C)ccc2)=O)CCCC(C)(NC(=O)CC=CC(C)(C)C)C1 c1(CC(=O)NC2CCCC(NC(C(C(C)C)C3CCC3)=O)C2)ccc(F)c(F)c1 CC1CN(C)C(C)CC1NC(C1CC(C)CN(C(=O)CCC(C)(C)N(C)C)C1)=O CC1C(NC(c2cn(C)cc2C(F)(F)F)=O)CCCN1C(c1ccc(Cl)nc1)=O C1(N(C(CCCOC(C)C)=O)C)CCCCN(C(c2cnn(C3CCC3)c2)=O)C1 CC(C)C(C(=O)NC1CCN(c2ccncn2)C1)N1CCCC1=O CC(CCNC(=O)CC1(C)OCCO1)CCNC(C1CCS1(=O)=O)=O Cc1cc(C#N)cnc1C(=O)NC(C)(C)CCCC(=O)NC1CC(=O)NC1=O C(=O)(C(C)C(C)C)N(CCC)CCNC(c1ccc(F)cc1)=O.C(C)=O C(=O)(CCC(=O)N(C)Cc1cccc(NC(=O)CSC)c1)NCCC Fc1ccc2[nH]c3c(c2c1)CCCC3NCCN1CC2C3C=CC(O3)C2C1 N1(C(CN(C(=O)OC)C)=O)CCN(C)C(C)C1.c1(C=O)cnc(C2CC2)nc1 C1(C(=O)NC2C(NC(C3(COC)CC3)=O)C2)OCC1(C)C c1(C(N2CCC(NC(c3c(N)c(Cl)ccc3F)=O)C2)=O)cnc2c(c1)CNC2=O Cc1oc(C)c(C(=O)NCC(C)(CO)NC(c2cc(N)ccn2)=O)c1Br c1ccsc1[N+](=O)[O-].c1(C(N(C)CC2CCCN2C(=O)C)=O)ccc(O)nc1.S c1(C(C)C(=O)N(C)CCN(C(=O)C(C)(C)N2CCCCC2)C)c(F)cccc1F CC(C)(C)C(=O)C(=O)N1CC2(NC(C3CC=CC3)=O)CC1C2 C1(NC(c2cc(OC)n(C)n2)=O)CC2CN(C(c3cn(CCF)nn3)=O)CC2C1 Cn1c(C(=O)NC23CC(NC(=O)C4=NNC(=O)C4)(C2)C3)cccc1=O C1(C2CC2)(NC(C=CCCC)=O)CCN(C(=O)CC(=O)NCC2CC2)C1 Cc1cccc(NC(=O)C(=O)NC2CC(C(N3CCC(C)CC3)=O)CC2O)c1 C1(N(C)C(c2cncnc2)=O)CCCN(C(C2(CF)CCOCC2)=O)C1 C#Cc1cncc(NC(C2CN(C(=O)Cc3ccon3)CC2(F)F)=O)c1 C1(C=O)CCOCC12CCC2.C1(C(N2C(C3CC3)CCC2)=O)C2CC3C(C2)C13.N Cc1cc(C(=O)NC(C)(C)CNC(C2(C(=O)N(C)C)CC2)=O)ncc1Cl c1(C(N(C)Cc2cc[nH]n2)=O)cc(CNC(C2COCCO2)=O)ccn1 c1(CNC(CCc2cc(C)on2)=O)ccc(C(=O)NCCC(=O)N(C)C)cc1 N1(C(c2c(OCCC)cccc2)=O)CCN(C(C2CCCN(C)C2)=O)CC12CC2 c1(NCC(C)(C)CC2CC2)ncccc1S(=O)(=O)NC1(C)CCOC1 CC1CC(NC(=O)CCS(C)(=O)=O)CCN1C(=O)OC(C)(C)C CC1(C)CN(C(C2CC3C=CCC(C2)C3)=O)CCC1NC(C1CNC(=O)N1)=O c1(OC)ccnc(C(N2CC3(C2)CN(C(=O)C(C)(O)C2CC2)C3)=O)c1C c1(CC)oc2ccccc2c1C(N1CCCC(C)(NC(C2CC3CC3C2)=O)C1)=O C#Cc1ccc(C=O)cc1.C(=O)(C#CC(C)C)N(CCN(C(C(C)CC)=O)C)C C1(C(=O)NC(C)CCCNC(C23COCC2C3)=O)(NC(C)=O)CCCC1 C1(C(CO)NC(c2cnc(OC)s2)=O)CCN(C(=O)CO)CC1.c1ccnn1C C1(C(=O)N)CC2(C)CCCN2S1(=O)=O.CC(C)CC(C)(C)C(=O)NCCC(C)C C1(NC(C2(OC)CCSC2)=O)C2CN(C(c3ccc(N)cn3)=O)CC12 c1(C(N(C2CCCN(C(=O)Cc3cncn3C)C2)C)=O)cc(C2CC2)ccc1Cl C1(NC(C2N(CC)CC2)=O)COCCN(c2nccc(-n3ccnc3)n2)C1 C(=O)C(F)C(F)(F)F.c1(OC)ccccc1CCNC(=O)CSC1CC1 C1(CNC(=O)Nc2c(-c3nc(C)[nH]n3)cccc2)CCCCS1(=O)=O c1(C(=O)NC2(CNC(c3ccc(OC)s3)=O)CCOC2)cc2scnc2[nH]1 C1(F)(CC)CN(C(c2c[nH]nc2CC)=O)C1.C(=O)C(C)(C)N(C)C(C)C.N Cc1ccnc(Cl)c1C(N1CCCC1C(=O)Nc1ccccc1OCF)=O Cc1nc(-c2ccccc2)[nH]c1C(=O)NCCC1CN(C(C2(CO)CCC2)=O)C1 CCCC(CC)CC(=O)NC1CC(N(C)C(c2cn3c(n2)SCC3)=O)C1 c1(C(=O)NCCC(C)CCNC(C23CCCC2C3)=O)ccc(O)c(F)c1F N1(C(C2C(C(=O)OC)CC2)=O)CC(C(=O)NC)(C(N)=O)C1.[nH]1ccnc1 C1(NC(c2nc(C)c(C)s2)=O)CN(c2nnc(C(F)F)s2)CC1(C)C c1(C(=O)NCc2scc(NC(C(CC)SC)=O)n2)c(NC(C)=O)c[nH]c1C c1(C(N2CC(C3CN(C(=O)CO)C3)C2)C2C(C)C2)nc2ccccc2[nH]1 C1(C)(CNC(c2c(C)cccn2)=O)COCCN(C(=O)CCCC(C)(C)C)C1 c1(NC(C)CC2CN(C(=O)C(C)CO)C2)ncc([N+](=O)[O-])cc1CO C(=O)(CC(C)C(F)(F)F)N1C(CN(C(CCCCOC)=O)C)COCC1 c1(C(N(C(CCC)CO)C(C2CC(=O)N2)=O)=O)cc(C)c(C)c(C)c1 Cc1cccc(Cl)c1CC(=O)N(CC(=O)O)Cc1ncc(-c2ccccc2)[nH]1 C1(C(N2CCC(N(C(=O)Cc3csc(S)n3)C)CC2)=O)CCn2nncc2C1 Cc1oc(C(N2CCC(O)(CNC(C34CCC3C4)=O)C2)=O)cc1S(N)(=O)=O C1(C=O)CC2(C1)CC2.C(C(C)C)OCC(C)C.C(=O)C.C=O.C1CC1 N1(C(CS(=O)(=O)N(C)C)=O)CCC2(C1)CN(C(=O)Cc1noc3ccccc13)C2 CC(C)(C)C(C(=O)NC1CCN(C(C2(C(F)F)CCOCC2)=O)C1)C1CCCC1 c1(C(=O)OCC(=O)Nc2c(C(C)=O)cccc2)c(C)nn(C2CCOCC2)c1C C(C)(CCC(=O)NC1CCC(CC(=O)NCC2(C)CC2)C1)OC.C1CCC1 C1(CN2C(c3c(F)ccc(C)c3F)CCC2)CCC2(CC1)CC2(F)F Cc1ccc(C(=O)NC2CC2NC(=O)CC(c2ccc(F)cc2)C)c(C)c1 N1(C(c2occ(C)n2)C(=O)NCC2CCOC2)CC2(CCCC2)CC1C N1(C(c2c(CC)n[nH]c2)=O)CCC(CNC(=O)C(c2c(C)noc2C)C)C1.O c1(-c2cn(CC(=O)NC(C(N)=O)C3CCOC3)nn2)cccc(F)c1 c1(C(=O)NC(C)CNC(=O)C(C)NC(c2ccoc2)=O)cccn2nncc12 N1(S(c2cccc(N3CCCN(C)CC3)n2)(=O)=O)CC23CCCC2(C1)CN(C)C3 C=CCC(CC(C)C)C(=O)N1CCN(C(=O)CC2CC2(C)C)C(CO)C1 Cn1cc(CCC(=O)N(CCNC(C2CN(c3nnnn3C)C2)=O)C2CC2)cn1 N1(C(CCCOCCC)=O)CCCC2(NC(=O)CCc3cccnc3F)CC2C1 CCC(C(=O)NCc1cc(C(=O)N(c2ccccc2)CC)co1)N(C)C C(F)(F)(C(=O)NNc1cc(-n2cc(Cl)cn2)ncn1)NC1C(C)Oc2ccccc21 N1(C(CC(C)F)=O)CCC(C(=O)NCCOC2CC2(F)F)C(C)(C)C1 Cc1cc(C(=O)NCC2CCC2)cc(C)c1O.c1(CC(=O)N)cc(F)ccc1Cl Cc1c(C(=O)NCC2(O)CCN(C(c3cnc(O)o3)=O)C2)cnc2ccccc12 C12(CNC(=O)C=CC3CCOC3)CC(CN1C(c1occc1Br)=O)C2