SMILES C1(C(N(CCCCN(C(=O)CCn2cccn2)C)C)=O)CC12CCOC2 N1(C(C(C)CN2CCOCC2)=O)CCN(C(=O)C(C)(F)F)C(c2cn[nH]c2)C1 N1(C(C(C)OCC#C)=O)CCN(C(=O)CCc2cscn2)CC(O)C1 N1(CC)CC(C(=O)NC2CC2NC(=O)CCn2ccc(C)n2)CCC1=O c1(N(C23CC(N)(C2)C3)C(c2ccccc2-n2ccnc2)=O)nc(OC)ncc1F CN1CC=C(CC(=O)NC2CC3CCC(C2)N3C(c2c[nH]cc(F)c2=O)=O)CC1 N1(C(C(CCC)O)=O)CCC(CNC(=O)CC2NC(=O)NC2=O)C(C2CC2)C1 C1(N(C(=O)C=Cc2cscn2)C)CCCC(NC(C2CCSCC2)=O)C1 C1(CCC=C)CCN(C(=O)NCC2(Cl)CC2(F)F)CC1 N1(C(C(C)CN(C)C)=O)CCOC2(CCCN(C(C3CC34CC(C)(C)C4)=O)C2)C1 Cc1cn2c(n1)C(C)CC(C(=O)NCCCNC(c1ccc(Cl)cc1Cl)=O)C2 c1(SC)ccccc1C(C)C.c1oncc1C(=O)NC1CC(C)C1.C(=O)C C1(NC(CC(C)N(C)C(C2CC(CF)C2)=O)=O)CCCCCC1C C1(C(=O)NCC(C(C)C)(F)F)CN2CCC1(C)C2 n1(CC(N2CC3CN(C(c4ccn(C(C)C)n4)=O)C3C2)=O)cnc2ccccc12 c1(OC)ccc(C(=O)N)cn1.C1C(C)CCN1C(=O)CC12COCC(C1)C2.C C(=O)(C(F)C(C)CC(C)(C)C)N1CC(C)N(C(c2cccc(C#C)c2)=O)C(C)C1 c1(C(N2CCN(C(CCS(C)=O)=O)C3C2C3)=O)ccc2c(c1)CCC2(C)C C1(C(=O)NCC2N(C(C=NOC)=O)CCCCC2)CN2CCN1C(C)C2 c1(C(=O)NCC23C(CN(C(C(CC(=C)C)C)=O)C2)C3)nsc2c(Cl)cccc12 C12(C(N3CCC(NC(c4cc(C)[nH]n4)=O)C(O)C3)=O)CC1COC21CCC1 c1(C(=O)NCC=CCC(=O)NCc2ncc(C)[nH]2)ncccc1Cl C(=O)(C(C(C)CC1CCC1)N1CCC(C(F)(F)F)(OC)CC1)NCCCC c1(N2C(C(N3CCCC3)=O)CC(F)C2)cc2sc(Cl)nc2cn1 C(CN=c1[nH]c(=NCC2CCCS2)c2sccc2[nH]1)c1cccc(C)n1 N1(C(c2ccn(C)c2)=O)CC2CCOCC2(NC(c2cc(N)c(F)cn2)=O)C1 C1(NC(C2CC(CNC(=O)COCCF)C2)=O)CC1C1CCCC1 C1(NC(CNC(C)=O)=O)COC2(CCCN(C(c3cc(Br)cs3)=O)C2)C1 N1(C(C(C=CC)O)=O)CCC2CN(C(c3cc(OC)c(Br)c(=O)o3)=O)CC2C1 C1CN(C(c2nccc(N)c2Cl)=O)CC(C)(C)O1.C1(C(=O)NC)(OC)CCSC1 CC(O)CCCC(=O)N1CCC(NC(=O)CNc2cnn(-c3ccncc3)c2)C1 Cc1ccc2[nH]c3c(c2c1)CCCC3NCc1ccnc(F)c1 C1(NC(C2(SC)CCC2)=O)CN(C(=O)C=CCn2cncn2)CC1F c1(C(=O)NCC(=O)N(C)C)cc(-c2ccc(C3(C#N)CC3)cc2)c2cc[nH]c2c1 C1(C(=O)NCC2CN(C(COCCC=C)=O)C2)CCC(SCC)CC1 CCCCCC(O)CNC(=O)CCC1CCCN(C(C2CC(C)(O)C2)=O)C1 C1(NC(=O)NC(C(=O)NCC)CC)CNc2ccccc2C1 C1(CNC(C2C(C=C)C2)=O)CCCCN1C(=O)CSc1ccccc1Cl c1(OCC#C)ccc(C(=O)NC2(C)CCC2)cc1.N1(CC=O)CCCC1C.N c1(OCCC)ccc(C(N2CCC(CO)CC2)C(=O)NCc2cccs2)cc1 C1(CNC(c2nncc(OC)c2)=O)CN(C(c2ccn(CCF)n2)=O)CCC1C C(c1ccccc1C)=CC(=O)N(C1CCN(C(C(C)=C(CC)C)=O)C1)C C1(c2nc(-c3ccc(OCC)nc3)nn2Cc2cccnc2)OCCCC1(C)C CCC(CC(=O)NCC(Cc1ccccc1)NC(c1csnc1Cl)=O)C(F)F Cc1c(F)ccc(N)c1C(N1CCC1CNC(C1CCN(C)C1=O)=O)=O c1(CCC(=O)N(C)C)ccc(O)c(F)c1.C1(C(N2CCCC2)=O)CCC(=O)NC1 N1(C(C2N(CC)CC2)=O)C(C(=O)NOCCC(C)O)C2CC(O)C1C2 c1(C(C(N2C(Cn3cc(CNC(CC)=O)nn3)CCC2)=O)=O)ccc(Cl)cc1C C(=O)(C#CC1CCOC1)NCC1(O)CN(C(C2(C#C)CC2)=O)C1 C1(CC=C)(NC(=O)CC2CCC=CCC2)CCN(C(=O)Cn2ccnn2)C1 C(CN=c1[nH]c2cccc(Br)c2o1)(C1CCCCC1)NC(c1cc(C)c(C)s1)=O C(=O)(C#CC1CCOC1)NCC(C(=O)NC(C(=O)N(C)C)CO)CC1CC1 c1(C2C(CN3CCN(C(c4ccccc4)=O)C4C3C4)C2)nc2ccccc2[nH]1 c1(C(=O)NCCC2(OC)CN(C(=O)C(O)C(C)C)C2)ccc(Br)cc1C CC(C)CCCC(=O)NCC1C2CCC(C2)N1C(=O)C(=O)N.c1ccc(F)cc1 C(=O)(C(C)N(OC)C(=O)CSCCNC(=O)CCc1cnccn1)OC c1(COCCN(CC)Cc2c[nH]nc2OC(F)(F)F)ncccc1O C1(NC(c2cc(OCC)n[nH]2)=O)CN(c2nc(Cl)nc(C)c2F)C2CCCCC12 N1(C(c2nc(C)sc2)=O)CC(NC(=O)Cn2cnnc2O)CCC1C c1(C(=O)NCCC2COCCO2)ccc(-n2cc(CO)nn2)cc1 c1(COC)nc(C)ncc1C=O.C1(C(N2CC(C)C2)=O)CC(N(C)C)CCO1 c1(C(=O)NC2CN(C(C3COCCOC3)=O)CC23CC3)ccc2c(c1)OCC2 Nc1ccc(C(=O)NC2CCCC(NC(c3cncc(F)c3)=O)C2)cc1O c1(C(=O)NC(CCC)CCCNC(=O)CC2C=CCC2)cnc2c(Cl)cccn12 c1(OC)cc(C(N2C(C)CC3CC23)=O)cc([N+](=O)[O-])c1.c1(C=O)cnc(Cl)s1 c1(C(=O)Nc2n(C(C)C)ncc2)ncn2cc(-c3ccc(S(C)=O)cc3)sc12 c1(OC)ccc2nc(C(=O)N(C)CC)ccc2c1.C(=O)CC1CC1C(F)(F)F c1(CCC)onc(C)c1C(=O)NCC1CCCCC1.C1(O)(CC=O)CCOC1 N1(C(CC(=C)Br)=O)CCC(CNC(=O)CCN2CCCC2=O)CC1 C1(CNC(c2c(SC)ccs2)=O)CCC(NC(c2ccn(C)c2)=O)CC1 c1(NC(C2C(C=C(C)C)C2)=O)ccc2c(c1)CCCCC2 c1(C(=O)OCc2nccs2)cc2c(Cl)c(Cl)ccc2[nH]1 N1(C(CCc2onc(CC)n2)=O)CCCC2(CNC(c3cccc(C)c3C)=O)CC12 c1(C(=O)NCC=C2CCN(C(c3ccn(C)n3)=O)CC2)cncc2cccnc12 c1(C(=O)NC(CN(C)C(C2CCN3CCC2C3)=O)(C)C)ccc(N)c(Cl)c1O S(=O)(=O)(c1ccc(N2CCCC2)cc1)N1CCN(Cc2c(C)nn(C)c2C)CC1 Cc1nccc(C(=O)NCc2cc(C(N3CCOCC3CCO)=O)co2)c1N Cc1c(C(=O)NCC(F)CNC(C2C=CCC2)=O)n[nH]c1-c1ccc(Cl)cc1 Cc1ccc2[nH]c(C(N3CC(NC(c4cnoc4C4CC4)=O)C3)=O)cc(=O)c2c1 c1(CNC(=O)C(=O)NCC(F)F)cn(CC2CCCOC2)nn1 c1(C(N2C3C(NC(c4nc(Cl)cs4)=O)C(C3)C2)=O)cc(Cl)c2c(c1)OCCCO2 c1(C(N2CCC(NC(C(C)n3cccn3)=O)(CO)C2)=O)ccn2c1CSCC2 C1(C(N2CCC(n3cc(CCC(C)O)nn3)C2)=O)Cc2cscc2C1 N1(C(=O)Cc2ccco2)CC(CN=c2[nH]nc(-c3ccccc3)o2)C2(COC2)C1 CC1CC2CN(C(c3[nH]nc4ncccc34)=O)CC2N1C(C1C=CCC1)=O c1(CC(=O)NCCC(C)N(C(=O)CC23CC(C2)C3)C)csc2nccn12 c1(C(C)=O)cnc(Cl)[nH]c1=NC1CCCCC1CNC(C1(C)CC1Br)=O C1(CNC(c2cnncc2O)=O)CCC2(CN(C(=O)CC3CCC3)C2)O1 C(c1ccc2c(c1)OCCO2)=CC(=O)N(C(CNC(C(CC)COC)=O)C)C N1(Cc2n(C)c(Cl)cn2)CCC(NC(=O)C(F)Cc2ccccc2)CC(C)(C)C1 CCCCC(O)CC(=O)N1CCN(C(=O)C=C(C)C)CC1c1cn[nH]c1 N1(C(c2ccc(C3CC3)cc2)=O)CCCCC1CCn1cc(C2(O)CSC2)nn1 C1(NC(c2cn3ccccc3n2)=O)CN(C(=O)Cn2cncn2)C2CCCCC12 C(=O)(C(C#N)C(C)(C)C)NC1CCN(C(c2n[nH]c(C3CC3)c2Cl)=O)CC1.CC N1(C(C2C(OCC)C2)=O)CCN(C(=O)Cc2ccnn2C)CC(O)C1 Cc1c(C(N2CCC(C)(NC(C3CSCN3C)=O)C2)=O)cnn1CC(C)(C)O c1(OC)ccc(CC(=O)NC)cc1F.C1(O)(CC(N2CCC2)=O)CCCN(C)C1 O=C1NCC2(CCNCC2)C1NC(C1(CC(F)F)CC1)=O c1(C(=O)NCC(=C)CCNC(=O)CC)ccc2[nH]c3ccccc3c(=O)c2c1 C1(C=O)CC(C)(C)OC1(C)C.C1(CNC(C(C)=C(CC)C)=O)CCC(O)C1 C(=O)(CS(=O)(=O)C(C)(C)C)N(C1CCN(C(=O)CC)C1)C.C1(C=O)CCC1 Cc1cnc(NCC2(C)CCOC2)c(S(=O)(=O)NCC(n2ccnn2)C)c1 c1(CCC(=O)N)cc(C)cc(C)c1.C1(CN(C(C=CCCC)=O)C)CCCCC1 c1(N(C2CCOCC2)CC)nnc(C(C)C)n1CC1CCCOC1C(C)(C)C CCC(C)(C)C(C)CC(=O)NC1CCCN(C(c2cc(Cl)c(Cl)[nH]2)=O)C1 CC(CC(=O)NCCC1(C)CCN(C(=O)C=Cc2ccnn2C)C1)C(C)(C)C N1(C(=O)OC(C)(C)C)C2CCC1C(CNC(C13CC4CC1C3C4)=O)NC2 C1(C)(c2ccc(OC)cc2)NC(=O)N(CCCC(C)C)C1=O Cn1cc(NCc2ccc(CO)cc2)nc1C(=O)NCC(c1ccc(O)cc1)O CC(C)C1CC(NC(C2CC(P(C)(C)=O)C2)=O)c2ccccc21 C(=O)(C1=CCN(C(=O)CCCn2ccnc2)C1)N(CCCCOC)C N=c1[nH]c(=NCC2CCC=CCCC2)[nH]c(=NCCC2COCCO2)[nH]1 Cc1cccn2c(CN3CCCOC(c4ccccc4Cl)C3)cnc12 N1(C(=O)Cc2cncs2)CCN(C(C2C=CCS2)=O)C2(CC2)C1 N1(C(C#CC(=O)O)=O)CC2CN(C(=O)Nc3ccc(Cl)cc3F)CC12 N1(C(c2nc(OCC)sn2)=O)CC(NC(c2ccc(Cl)[nH]2)=O)CC1CO C(C(C(C)(C)C)NC(=O)Cc1ccsc1)NC(C(C)Oc1cccnc1)=O C1(C(N2CCC(C)(OC)C2)=O)CN(C(c2ccc(Br)s2)=O)CCC1O C#Cc1ccc(NC(C2CCN(C(=O)C(CC)C(F)(F)F)CCO2)=O)c(C)c1 C(C)(C(=O)N1CCC(CCO)C1)(C1CCC1)NC(C1C(CC(C)C)C1)=O N1(C(C(C=C)(C)O)=O)CCC2(C=C(C(=O)NCCC(C3CC3)C3CC3)C2)C1 C1(c2n(C(CC)C)nnn2)(Nc2cccc(C(N)=O)c2)CC2CC2C1 c1(C(=O)NCC2CCN2C(=O)CC2CCCOCC2)scc2c1CCCC2 C#Cc1ccc(Br)c(C(=O)NC2CN(C(=O)CC(C)(F)F)CCC2CO)c1 C#CC1(C(=O)NC2C(C)C2(C)C)CN(C(C2C3COCC23)=O)C1 N1(C(CCC=C=C)=O)CC(CNC(c2cc(CCC)n(C)n2)=O)OC(C)(C)C1 Cc1cc(C(C)C(=O)N(CC(C)NC(=O)CSc2cn[nH]c2)C)cc(C)c1 O=c1ccc(Cl)cn1Cc1nnc(C(F)(F)Cl)o1 c1(C(N2CC(NCc3ncco3)C3(CC3)C2)=O)cc(Br)c(F)cc1F c1(CC)conc1CC(=O)NC(CO)C(C)NC(=O)CCc1ccccc1 C(N=c1cc(C)[nH]c(=NCCc2ccc([N+](=O)[O-])cc2)[nH]1)c1c(OC)cncc1 N1(C(C2C(NC(c3c(C)ccc(Br)c3F)=O)C2)=O)CCc2ccccc2C1C c1(OC(C)C)cccc(C(=O)NC2CC(C)C2)c1F.C(=O)(C(C)N(C)C)N C1(CC)(CC)CC(NC(c2nscc2C)=O)CN1C(c1ncc(C)cc1F)=O C(CC(=O)N1CCC(CCNC(=O)Cc2ncn(C)c2C)C1)(C(F)(F)F)OC CN1CCC(C2(C(=O)NC3(C4CCN(C(=O)Cc5cc[nH]c5)C4)CC3)CC2)CC1 N1(C(CS(=O)(=O)NCC)=O)CCCN(C(=O)C=CC2(C)CCOCC2)CC1C C1(C(N(C2CCN(C(c3conc3C3CC3)=O)C2)CC)=O)CCc2cncn2C1 N1(C(c2c[nH]c(=NC)s2)=O)CCC(C2(NC(=O)CN3CCC3C)CC2)C1 C(C(O)COC)N(C(CN(C(=O)COCC)CCC)=O)C C1(C(=O)NCC(=O)OCC(=O)CCC2CCCCO2)CCCC(F)C1 C1(CN(C)CC)CCN(C(=O)C(c2ccco2)NC(=O)COC)C1 c1(C(=O)NC2(C(=O)NCC(CC)CO)CCC2)ccn2ccnc2c1 c1(C=O)cc2ccc(Cl)c(F)c2o1.C1(C(N)=O)CCC(C(=O)NC2CCC2)O1.N C12(CNC(c3ccc(SC)s3)c3nnnn3C(C)C)CC(C)(CO1)C2 c1(CC)cc(C(=O)N)c(C)o1.c1(C(N2C(C(C)C)CCC2)=O)cnc(C#N)s1 N1(C(CC(CSC)NC(c2cc(COC)no2)=O)=O)CCCC(C2CCC2)C1 Cc1ncc(C(=O)NCC2CC(C(=O)N)C2)c(C)n1.C1(CC)CCOC(C)C1 c1(NC(C2C(CC)CCCC2)=O)nc2cccc(-c3nn[nH]n3)c2[nH]1 C1(NC(C)=O)CN(C(=O)C(C)CC(=O)c2cccc(F)c2)C2(CCOCC2)C1 N1(C(Cn2ncc(C#C)c2)=O)CCOC2(C1)CN(C(C1CC3(CCCCC3)C1)=O)C2 C(=O)(CCC(C)C#N)NC(CN(C(c1ncccc1OC)=O)CC)C c1(CCC(=O)NC2CCN(C(c3ccnc(OC)n3)=O)C2C)ccc(F)cc1Cl C1(C=O)OC(C)(C)OC1(C)C.c1ncoc1.C(C(=O)NCC1CC1)OC.C CC1(C)CC(NC(=O)CCCCC2CC2)CN1C(c1ccnc(C(F)(F)F)c1)=O N1(C(c2cc(CCOC)on2)=O)CCC(C)(NC(c2c(C)cnn2C)=O)C1 c1(CCC(=O)NC(CC)CN(C)C(C2(C)C=CCC2)=O)cccc(F)c1 Clc1cccc(-c2nnn(-c3noc(=O)n3-c3ccccc3)n2)c1 CCC(C)CCCCC(=O)NC(COC)CNC(=O)C(C)NC(=O)OC C1(NC(c2c(Cl)ccc(C)c2)=O)CC1C1CCN(C(=O)C(C)C(F)(F)F)CC1 Cc1cccc(Cl)c1CC(=O)NCC1(O)CC(NC(C2CC3CC3C2)=O)C1 c1(NC(=O)NCCCC)ccc(-c2noc(C(C)C(C)CC)n2)cn1 c1(NC(C(c2ccccc2Cl)OC)=O)cc(NC(N)=O)ccc1Cl C1(N(C)C)CCCN(C(=O)CCCNC(=O)C(C(C)(C)C)N(C)C)CC1 c1(CCC(=O)NC2CCC(NC(C3C4COCC34)=O)C2)ccc(Br)c(F)c1 C=CCC(CNC(=O)COc1cnn(C)c1)C(=O)NC1C=CC(CO)C1 c1(NC(CF)C(F)(F)F)nccc(Br)c1I CCC(C)CCCC(=O)NC1CCC(N(C(=O)C(C)SCCOC)C)CC1 c1(NC(C2CCN2C(c2cnnc(O)c2)=O)=O)ccc([N+](=O)[O-])c(F)c1 c1(C(C(=O)NC)N(CCn2cccn2)C(C)C)cc(F)c(F)c(OC)c1F C1(COC)CCCCN1C(=O)NC(c1nc(-c2ccccc2)no1)C Cc1cc(C(F)(F)C(=O)NCC2CC2)cnc1Cl.C1(C)(C=O)COC(=O)OC1 C1(C(=O)NC2C(NC(c3c(OC)c(C)cs3)=O)CCC2)CCCCC1(F)F c1(CC(C)C)ccc(C#N)c(N2CCC(C)(NC(C3CNC(=O)CC3C)=O)C2)n1 CC1CC2(CCO1)CCN(C(=O)C(=O)NC1CC1c1ccc(F)c(F)c1)C2 C1(NC(C2N(CC)C(=O)CC2)=O)CC2CC1CN(C(=O)C1=COCCC1)C2 N1(CC(=O)N(CC(CNC(CSCCC)=O)C)C)CCCCCC1=O c1(CC)ccc(F)c(C=O)c1.C(C)C(C)C.c1(C=O)cc(C(C)(C)O)on1.N N1(c2ccnc(OC)n2)CCCC(C2CN(C(c3cc[n+]([O-])cc3)=O)C2)C1 NC(=O)CCC(=O)N1CC(c2ocnc2CN(C(=O)Cc2cncnc2)CC)C1 c1(C(=O)NC2CN(C(c3c(NC)c(F)ccc3)=O)CC2O)ncnc2c1CCC2 c1(C(=O)NC2CCC(C)N(C(=O)CCCC(F)F)C2)c(F)ccc(N)c1F c1(C(=O)NCC(CN(C(c2ncn(C(C)C)n2)=O)C)(C)C)ccc(Cl)c(F)c1 C1(NC(Cn2c(C)ncc2)=O)CN(C(C2CCC(C)(C)C2)=O)C(C)(C)C1 c1(CNC(C(=O)OC)c2ccsc2)ccc(C(C)(C)C#N)cc1 c1(NCCC)c(C(=O)NCC(CC2CCOCC2)OC)cccc1C c1(OCC)ccc(Cl)cc1NC(c1cccc(Cl)c1C)c1nnnn1C Cc1nc(O)nc(C)c1C(=O)NC1CC1NC(c1cccc2[nH]ncc12)=O c1(CN2CCC(C(N3CCC(C(=O)OC)CC3)=O)C(O)C2)c(F)ccc(Cl)c1Cl Cc1cc(CN(C(=O)CCC(C)NC(C2CCCOCC2)=O)C)nn1C CC(C)(C)C(C)C=O.C1(C(=O)N)CC(=C2CCC2)C1.N(S(N)(=O)=O)CC N1(C(C(C(=C)C)(C)C)=O)CCC(NC(=O)Cc2ccns2)C2(CCC2)C1 c1(C(N2CC(N(C(C3CCN(CC)CC3)=O)C)C2)=O)cnn2cccc2c1 CCC(CC)(CO)C(=O)NCC(F)CNC(c1ncc2ccccn12)=O CCCC(C(=O)OC)C(=O)NC(CC(=O)NCc1cc(OC)ncn1)C(C)OC N1(C(C(C2CC2)OCC)=O)CCC2(CCN(C(=O)COC3CCCOC3)C2)C1 CCCCC(O)C(=O)N1CCN(C(C2CCN(CCC)CC2)=O)CC1CC C1(CNC(CSCC)=O)CN(C(c2cc(C(F)F)[nH]n2)=O)C2CCCCC12 N1(C(CN(C(C)=O)C)=O)CC(NC(C2CCc3ncsc3C2)=O)CC12CCCC2 c1(OC)cc(C#N)ccc1C(N1CCC(=CC)CC1)=O.C(=O)(CC(C)C(F)F)N C1(C(C)NC(c2cnc(CC(C)C)s2)=O)CN(C(c2ccnc(F)c2)=O)CCO1 c1(C(=O)NCC(=C)CCNC(C2(CF)CC2)=O)cc(C)c(CC)o1 c1(N(C)Cc2ccccc2CNC(C2(C)CC(F)C2)=O)snc(Cl)c1C#N c1(C(=O)NC(C)C(c2ccccc2)O)cc2c(nc1O)CC(C)(C)CC2=O c1(C(=O)NC2CC3(C(NC(C(CCCC)CC)=O)C3)C2)nccn2cc(C)nc12 CC12CCN(CC1)CC2C(N1CCCC(C(F)F)C1)=O C1(NC(C2CC(C)(C)OCC2)=O)CCSC12CN(C(C1(CO)COC1)=O)C2 Cc1cc(C(N2CCCC2CCNC(c2occc2F)=O)=O)nnc1C N1(C(CCc2cn(C)nn2)=O)CC(NC(=O)CN2CCOCC2)CC12CCOC2 CC(C)CC(C(=O)NC1CCCCCC1O)NC(=O)CC1CCCC2CC12 c1(C(=O)NCC(C)NC(=O)CC(c2cccc(F)c2)O)cccc2cnccc12 C12(NC(C3C(CNC(C4(C)COC4)=O)CCCC3)=O)CCC(CC1)C2(C)C C#Cc1ccc(F)c(C(=O)N(C)CCNC(c2ccc(-c3ccsc3)cc2)=O)c1 n1(CC(N2CC(C(C)NC(C(CC)OCC)=O)C2)=O)c([N+](=O)[O-])cnc1C N1(C(c2cc(CN(C)C)on2)C(=O)NCC)CCCC2C(=O)N(C)CC12 C(=O)(CCCC(=O)c1ccc(F)cc1)N.C1(C(N(C)CCOCC)=O)CCC1F C1(C2CC2)(CNC(C(C)c2cncs2)=O)CCN(C(=O)CCC2CCC2)C1 n1(CC)c(C(=O)N(CCNC(c2cn(C)c(C)n2)=O)C2CC2)cnc1O CCC(C)C(C(=O)N1CC(O)(CC)C1)NC(C)=O.C(=O)CC(C)C1CCCC1.N N1(C(C2CCN(CC)C2)=O)CC(C)C(O)C1.C(=O)C(F)(F)F.C(=O)(C)N C=CCC(CC(C)C)C(=O)N(CCC(C)NC(C1CCC([N+](=O)[O-])CC1)=O)C C1(NC(c2cccc(SC)n2)=O)CN(c2ncc(C)cn2)CCC12CCC2 N1(C(C2N(C)C(=O)CC2)=O)CC2(CCC2)CC1C(=O)NC1(C)CCSC1 C(=O)(C1=NOC2COCC12)N(C(C)(C(N1CC2(CC(O)C2)C1)=O)C1CC1)C C=C1COc2c(C(=O)NC(CO)C(C)NC(c3cc(C)c(C)s3)=O)cnn2C1 CC1CC(NC(C2CC23CC(NC(=O)CCCC(F)(F)F)C3)=O)C(C)CN1C c1(OC)oc(C)nc1C(=O)NC(c1ccccc1)C1CCOCC1 c1(CCC(=O)NC(CNC(c2ncccc2O)=O)CO)ccc([N+](=O)[O-])cc1Cl N1(C(C(CC)CC)=O)CC(C(=O)NCC2CC2CO)CC(C)(C)C1 N1(C(c2c(NC(C)=O)cc(Cl)cc2)=O)CC2CN(C(=O)CCC(N)=O)CC2C1 C1(NC(c2c(C)nc(C3CC3)s2)=O)CCN(C(c2cnns2)=O)CCC1CO c1(C(N2CCC(CNC(C(c3ccc(Cl)cc3)C)=O)C2)=O)cc(Cl)ccc1F c1(C=O)oc(C2CC2)nc1C(F)F.C1CCCC1.C1(CCOC)CC1C=O C1(C)(COC)CCN(C(=O)CC=CCNC(=O)Cc2cccc(C)c2)C1 c1(C(N(C)CC2N(C(c3c(C)nc(CC)o3)=O)CCC2)=O)cnc(F)c(Cl)c1 N1(C(c2c(C)nsc2N)=O)CC2(CCC2)CC1CNC(c1cccc(Cl)n1)=O c1(C(=O)NC2CC3CN(C(CCC=C=C)=O)C2C3)cnn2c(C)c(C)ccc12 C(C)(C(=O)NCCOc1ccc(C)cc1C)C(C)C.C(=O)(CC)N.CC=O CN=c1nc(N2CCc3ccccc3C2)[nH]c(=NC(C)c2cnc(Cl)c(Cl)c2)[nH]1 C1(NC(c2c(C)ccc(Cl)c2)=O)CCCCN(C(=O)C(F)(F)C2(O)CCC2)CC1 N1(C(CC(CCC)C)=O)CC(C2CCN(C(C3(O)CCCC(C)(C)C3)=O)CC2)C1 C#CCC(CC(=O)NCCCOC(=O)NC)NC(=O)C(=C1CCCCC1)F C1(NC(C2(NC(C3C(C)(C)C(=O)C3)=O)CCCC2)=O)CC2(CCC2)C1O C1(SCC)CCC(C(=O)N(C2CCCCC2NC(c2cccc(N)c2)=O)C)CC1 c1(C(=O)NCC(CC)NC(=O)C(C)C(=O)OC)cc2c(s1)CCCCCC2 N1(C(C(c2ccc([N+](=O)[O-])cc2)(C)C)=O)CCCC2(CCS(=O)(=O)C2)C1 C1(CNC(CCSCC(C)C)=O)C(C2CC2)CCN1C(c1c[nH]c(=N)o1)=O c1(C(=O)NC(CN(C)C(c2cccc3nn[nH]c23)=O)(C)C)cc2nnn(C)c2s1 c1(OC)ccc(C(CO)N(C)C(C2CC3CC2C3)=O)cc1 c1(OCC)ccc(NC2(c3nnnn3CCCSC)COCC2C)c(C)c1 C(=O)(C1c2ccccc2OCC1C)NC1CC(NC(c2ccc(C)nc2O)=O)C1 CCC(CC)C(=O)NC(C)C(C1CCCCC1)NC(c1nc(Br)c[nH]1)=O CC1CN(C(=O)CCCCCC2CC2)CCN(C(=O)C(C)O)C1 C1(CC(=O)NCC2(F)CCCC2)CCCCC12CC2.c1(C(=O)N)cncc(F)c1 c1(OC)ccc(C(=O)NCC2CN(C(c3ccn(C)c(=O)c3)=O)C2)cc1F C1(CNC(CSCC=C)=O)(OC)CCN(C(=O)CCC(C)(C)C)CC1 C1(SC)CN(C(C2CCOC2)=O)CC1NC(C1(c2ccnn2C)CC1)=O N1(C(C2(C)COCC2(F)F)=O)CCOC2(CCc3ccccc32)C1 c1(CC(=O)NC2C(C)N(C(c3cn(C)c(O)n3)=O)CCC2)ccc2[nH]ccc2c1 c1(CC)sc(C(=O)N(C2CCN(c3ncccc3C(C)=O)C2)C)cc1C C(=O)(C1=CCCN(C(C2CN3CCC2CC3)=O)C1)NCCC(C)CO Cc1ccc(C(N2CCC(N(C(=O)CCn3ccnn3)C)C2)=O)c(C)c1Br c1(NC(CCCCCn2cc(CNC(C)=O)nn2)=O)ccc2c(c1)CCN(C)C2=O Cc1ccc(CC(=O)NC2CC(C(=O)NC3(c4ccn(C)n4)CC3)C2)cc1 C1(CCC(=O)NC(C(=O)NCC)CC)CCCN(C(c2cnnn2C)=O)C1 CCCCCC(=O)NCC(=O)NCC1CCC(NC(c2cc(Br)n[nH]2)=O)C1 CC1CC(NC(C2CC(C#N)C2)=O)CN1C(c1ccc(C(F)F)cn1)=O C1(O)CCCN(C(C2CCNC2)=O)C1.O=CN1CCCC1CCN.c1ccccc1 N1(C(C=CC)=O)CC(C2(NC(C3CCCC(C)C3)=O)CC2)C1 CC(C)(C)C(O)CNC(=O)C(C1CC=CCC1)NC(=O)Cn1ccnn1 N1(C(c2cc(C)no2)=O)CC(C)CN(C(=O)C(C)(C)C(N)=O)CC1C CC1CC=C(C(=O)NC2CCN(C(c3ocnc3C3CC3)=O)C23CCC3)CC1 C1(C(N2CC3C(CNC(=O)Cn4ccccc4=O)C3C2)=O)OCCOC12CCC2 c1(C(N(CC(=O)NC2(CC#C)CCOCC2)CC(C)C)=O)cc2ccccc2[nH]1 C1(CCNC(c2cn(CC)nc2)=O)CCOCC1.c1(CCC=O)nnc(C)o1.N C1(CC)CN(C(C2CCCC2)=O)CC1NC(c1c[nH]nc1-c1ccc(Cl)cc1)=O c1(CN(C)C)ccccc1C(N1CCN(C(C2CC23CCCC3)=O)CC1)=O N1(C(c2cc(OC)n[nH]2)=O)CC(NC(c2cccc[n+]2[O-])=O)C2(CCCC2)C1 c1(CC(N2CC(C(C)NC(C3CN(C(C)=O)C3)=O)C2)=O)cc(C)cs1 C1(NC(c2ccc3c(c2)CC3)=O)CC2CCC(C1)N2C(c1cn[nH]c1)=O CC1Cc2cccc(C(=O)NC3(C)CN(C(c4cc([N+](=O)[O-])nn4C)=O)C3)c2O1 CC1C2CCCCC2CN1C(=O)CCN(C(c1cccc(O)c1)=O)C1CC1 C#CC1(C)CCN(C(C2(NC(=O)COCc3nc[nH]n3)CCCCC2)=O)CC1 c1(CC)ncc(C(=O)NC(C)C(=O)N(C(C)CO)C)s1 C=CC(O)(C(=O)NCC1CN(C(c2cccc(F)c2C)=O)CCO1)C(F)(F)F C1(C(N(C2CCC2)CC)=O)C2C(CN1c1ccncn1)C2(C)C C(=O)(C(O)CC(C)(C)C)N1CCN(C(CNC(C2(CC)CCCCO2)=O)C)CC1 C(C(CNC(C1CC12CC2)=O)S(C)(=O)=O)NC(COC(C)=O)=O N1(C(c2c(C)c(C(C)C)[nH]n2)=O)CC(CNC(=O)C(C)(C)O)C(C)(C)C1 CC1CCC=C1C(=O)NC1CN(C(=O)Cc2nccn2C)CC1(C)C c1(OC)nc(NC(=O)CSCc2cc(O)ns2)cc(C)n1 c1(C(N2CCCC(N(C(=O)Cc3ccns3)CC)C2)=O)sc2ccccc2c1C C1(NC(C2(CC)CCC2)=O)CN(C(=O)CCc2ccc(C(F)F)cc2)C2CC12 CCC(C)(C(=O)NCC1CC1CC(=O)C=CC(C)(C)C)C(N)=O C12(C=O)CCCN1S(=O)(=O)CC2.Cn1cnnc1CCC(=O)NCC=CC.N N1(C(c2c(CCC)nns2)=O)CCCC(NC(=O)C(C(C)C)SC)CC1 C(=O)(C#CC1CCOCC1)NC(C=CC(=O)NC1(C(=O)NC)CC1)C Cc1cccc(F)c1CC(=O)NC1CCCCC1.C1(C=O)(CCN(C)C)CC1.N c1(Nc2c(C(=O)NC(CC)C)cc(OC)nc2)ncc(Cl)cc1[N+](=O)[O-] c1(C=O)cc(O)cc(C#N)c1.C(C(C)(C)C(=O)NC1CCC(C)CC1)N(C)C.N N1(C(CN(CCOC)C)=O)CCCC(C(=O)NCCn2cnc(CO)c2)C1 N1(C(C2C(C(C)C)(CC)C2)=O)CCC(CO)(C)C1.c1(C=O)cncc(Cl)c1 c1(CNC(c2nnnn2C2CCOC2)(COC)C)ccc(SC2CCC2)cc1 c1(C(C2C(C(=O)NC3(CC)CC3)CC2)=O)ccccc1.C1(C=O)CC1.N C1(CCCNC(CC2C(C)(C)C2)=O)CCCCN1C(=O)COC.c1cscn1 C1(C(=O)NC(C)CN(C)C(C23CCC(CC2)CC3)=O)CC2CCCC(C1)C2 c1(COC)nn[nH]c1C(=O)N.C(=O)(CCCn1ccnn1)N(CC)C1CC1 c1(C(N2CCC(CC(=O)Nc3c(OC)nccc3)C2)=O)cc(Br)cc(I)c1 C(CCN=c1[nH]c(=NCC(=O)N2CCCO2)c2[nH]ccc2[nH]1)=CCCC c1(CN2CCCC(C(=O)NCC3(CO)COC3)CC2)cncc2ccccc12 CN=c1nc(N(CC(C)(C)OC)C)[nH]c(=NCCc2ccc3ncccc3c2)[nH]1 c1(NC(=O)NC)ccc(Cl)c(C(=O)N(C)C(c2cc(F)ccc2F)C)c1 N1(C(C2CN3CCN2CC3)=O)CC(CNC(C2(CO)CCCO2)=O)CC12CCC2 CC1CN(C(C2CC2c2cccnc2)=O)CCC1CNC(c1c[nH]c(CN)c1)=O c1(OCC(C)NC(C)C(=O)Nc2cc(C3CCC3)n[nH]2)ccccc1 N1(CS(CC)(=O)=O)CCCC1CN(CC(C)NC(C1CCCCO1)=O)C CCCC(C(=O)OC)C(=O)NCCC1CCCCN1C(c1csc(C)n1)=O C1CC(F)(F)CN1C(c1ccn(C2CC2)n1)=O.n1(C(C)C)cc(C(=O)N)nn1 N1(C(C2=CCCC2C)=O)CCC2(CCCN2C(C2CC3(CCO2)CC3)=O)C1 C12(C(=O)NCC3(NC(CC(C)c4ccncc4)=O)CCCC3)CCC(CC1)CO2 CCC(CC(=O)NCCCCCCN(C)C(c1nn(C)cc1C)=O)SC N1(C(CCC(C)(C)F)=O)CC(NC(=O)CN=S(C)(C)=O)CC2(CCC2)C1 c1(CCC)cc(C(=O)NC2CN(C(C3CC3C3CCC3)=O)CC2O)ccn1 c1(C=O)cc(N)c(F)cc1F.C1(C2CCC2)(C(N(C(C)C2CC2)C)=O)CC1.N c1(N(C)CCN(C)C2CC2)nc2ccsc2c(=NC2CCN(C3CC3)C2)[nH]1 c1(OC)ccc(CN2C(=O)CN(CCS(=O)Cc3ccccc3)C2=O)c(O)c1 Cc1ccc2c(C(=O)NCCc3nnc4n3CCC4)ccnc2c1Cl c1(C(=O)OCC)ccc(NC(=O)COc2ccc(CC)cn2)cc1 C(C1CCCN1C(=O)C=CC(F)F)=CC(=O)NC(C1(O)CCC1)C c1(C(C(C)C)NC(C(N2CCC(COC(C)=O)C2)=O)=O)ccc(F)cc1 N(C1CCOc2ccc(F)cc21)C(=O)NC(c1ccnn1C)C C1(CC)(NC(c2c[nH]cc(Cl)c2=O)=O)CCCN(C(c2ccc(N)c(F)n2)=O)C1 c1(C(=O)NC(CCC)CNC(C2CCN(C(=O)NC)C2)=O)cc2cccn2cn1 c1(CNC(C(CC)NC(N)=O)=O)n[nH]c2c1CN(C(=O)CCC(C)OC)CC2 N1(C(C2CC=CC(NC(=O)CC=C(Cl)Cl)C2)=O)CC2CCC(CO)(C2)C1 C12(C(=O)NCCCC(=O)NCCN(CCCC)C)CCC(C1)C2(C)C c1c[nH]c2ccccc12.C1(C(N(CCN(C(=O)C)C)C)=O)(C(N)=O)CC1.C C(=O)(CCC1=CCCCC1)N1CCCC(C(=O)Nc2c(CC)nccc2)(CC)C1 N1(C(C2C(C)(C)C2CNC(c2coc3c2COC3)=O)=O)CCCCC12CC2 c1(N(C(C2(C=C)CCOCC2)=O)C)cnn(C)c(=O)c1Cl C(=O)(C1=CCOCC1)NC(C)C(C)NC(=O)CCc1cccc(O)c1 c1(C(N(C)CC2CN(C(=O)C(F)(F)C(F)F)CCO2)=O)cc2nc[nH]c2cc1F CC(C)C(C)C(C)CC(=O)N(C1CCCN(C(C2CC(F)(CO)C2)=O)C1)CCF C1(C(=O)NCC2CCC3(CC3)CO2)CC12CCN(C(c1ncncc1Cl)=O)CC2 Cc1cccc2[nH]c(C(N3CCC(CCN=c4ncc(Br)c[nH]4)C3)=O)cc12 C1CN(C(=O)CC2(C)CCS(=O)(=O)N2)CCC12CCC2.N1(CC)CCC1C=O c1(C(N2CCCC2)=O)cccnc1SC(F)F.CC(C)(C(=O)NCC)C1CC1.O c1ncsc1C(F)(F)F.C(C)(C=O)SCCCC.CC(=O)NCCO.CC c1(CN2CC(CCNC(c3ncn(C)c3)=O)C2)c(F)cccc1Cl c1(-c2c(C)occ2)nc(CCc2cn(C)nn2)n(CC2CCCOC2)n1 c1(CC)cccc(OCC(=O)NC23CC(C)(C2)C3)c1.C(=O)CC(C)C.N N1(C(C=CC(C)=O)=O)CCC2C(CCCN2C(=O)CCc2ccc(C)s2)C1 C12(CNC(CCc3ncc(C)[nH]3)=O)CCC1CN(C(C1CC1c1cnc[nH]1)=O)C2 C1(CC)CN(C(=O)C(C)(C)c2cscn2)CC1C(=O)N.c1nocc1C(C)C c1(C(=O)NCC(=O)NC2CC(NC(C3C4COCC34)=O)C2)ncccc1O Cc1cc(Br)c(F)cc1C(=O)NC(CNC(C1(F)CCCC1)=O)CO c1(C(=O)NC2C(NC(CC(C)C3CC3)=O)CCC2)cccnc1C1CC1 Cc1cc(-n2ccc(C(F)(F)F)n2)ccc1CNCCCC1(C#N)CNC1 N(C(=NCCc1cccc(NC)c1)N1CCC(N2CCCS2(=O)=O)CC1)C(C)C c1(C(C)C)nnsc1C(=O)N(CCCN(C)C(C1SCCC1C)=O)C C#CCC(C)(C(=O)NC(CC)CCO)NC(c1ccsc1)=O c1(COC)nc(C)ncc1C(=O)NCC#CC.c1(CCC=O)ccn(C)n1.N C1(NC(COC(C)=O)=O)CCC(NC(=O)C(=O)c2ccco2)C1 c1(C(=O)NC2CN(C(c3c(CC)occ3C)=O)C2)cc2cc(Cl)cnc2o1 c1(C(=O)NC(C(C)NC(c2cscc2Cl)=O)(C)C)cc(C2CC2)nc(O)c1 S(=O)(=O)(c1ccc(OC(F)(F)F)cc1)Nc1cc(CN(C)C)c(F)cc1 C1(C(N(C2CCCN(C(=O)C(COC)COC)C2)CC)=O)CCC=CCC1 C12(Cn3c(N(C)Cc4ccc(Cl)s4)nnn3)COCCN1C(=O)COC2 N1(CC(=C)Br)CCC(NC(=O)CC2(C)CCCC2)C(O)C1 C1(NC(C(C)(CO)OC)=O)CCCN(C(c2cnn(CCF)c2)=O)CC1 N1(C(C2(C(=O)OCC)CC23CC3)=O)CCC2C(C1)CN2C(=O)C#CC1CC1 N1(C(c2ccc(Cl)c(Br)c2)=O)CCC2CN(C(c3cnc(Cl)s3)=O)CC2C1 C(=O)(CCCC(=O)N1CC(C)(OCC(=O)NCCC2OCCC2(C)C)C1)N(C)C C1(C(N(C2CCCN(C(=O)CCS(C)=O)C2)C)=O)C2CC(=O)CC12 c1(C(=O)NC2C(NC(C=NOC)=O)CCC2)cc([N+](=O)[O-])c(C)cc1Cl N1(C(C(=O)N(C2CC(C)(C)OC2=O)C)=O)CCSC2CCCC12 C1(C(=O)NC(C)CN(C)C)(Cc2cccnc2)CCOC1 C(=O)(CC1OCc2ccccc21)NC1CN(C(C2C(CC)C2)=O)C1 C(CCCN=c1[nH]c(N2CCCC3(CCN(C)C3=O)C2)nc2cc[nH]c12)N(C)C N1(C(C2(C#C)CCCC2)=O)CC(S(=O)(=O)c2cccc(F)c2)C1 C1(O)(C(C)NC(Cc2nc(C)sc2Cl)=O)CCN(C(C2CC2C#N)=O)CC1 C(C(=O)NOCCCCCC1CC1)(C1CN(C(=O)CC(C)SC)C1)OC CCC(C(=O)NCC1(F)CN(C(=O)CCn2ccnc2C(C)C)C1)OC N1(C(C=CC=CC)=O)C2CCC1C(F)C(NC(c1ccnc3c1ncn3C)=O)C2 CCC(C(=O)NC(CNC(c1nc(C)ccc1C)=O)C1CC1)C(C)(F)F Cc1c(C(=O)NCC2CC2CNC(=O)CN(C2CCCC2)C)ccn1C CCCCC(CNC(=O)C(O)Cc1cnn(C)c1)NC(=O)CCCCSC c1(NC(C2CC(C)SC2)=O)cnccc1N1CCN(C)CC1 CCC(CC)(CO)C(=O)NC1CCCC(N(C(=O)CCNc2ccccn2)C)C1 C1(COC(=O)CC2CCCC3(CC3)C2)CCC2(CCOCC2)O1 c1(CCC)ccc(NC(c2oc(C(F)(F)F)nc2C)=O)c(C)n1 N1(CCC)C(=O)CCC(C(N2CC(c3ccccc3)C2)=O)C1c1ccccc1 Cc1cnc(NCCCC(C)(C)NC(c2cc(F)ccc2C)=O)c([N+](=O)[O-])c1 c1(C(=O)NC(C)C(=O)NCCc2cn(C)cn2)cccn2nccc12 C(=O)(CC(C)C(F)F)NC(CCSC)C(=O)NCc1ccccc1CO C1(NC(c2c(C(C)(C)C)con2)=O)CCN(C(C2CCC3(CC2)CC3)=O)CC1O C(=O)CS(=O)(=O)Cc1ccc(Cl)s1.CCC(=O)NCC=O.C(C)C1CC1.N c1(CNCc2c(OCC(=O)NC)cccc2)ccc2c(c1)CCS2 C1(N(C)C(=O)NC2CC2C(F)F)CCNC1=O O=C(C1=CCOC1)NC1CCC1NC(C1(O)CCSCC1)=O c1(C(N2CCC(F)(C(N3CC(C)C(O)CC3)=O)C2)=O)ccc2[nH]nc(O)c2c1 C(=O)(C#CC1CCOCC1)N1CCC(CCNC(c2ccc(CSC)o2)=O)CC1 S(=O)(=O)(c1cc(C)cc(C)c1)NC1C2CN(S(CCC)(=O)=O)CC21 N1(C(C(C(F)(F)F)OC(C)=O)=O)CC2CCCN(C(=O)CC3CC3)C2C1 CC(C)(C)CC(O)CC(=O)N1C2CCC1CC(C(=O)NCC1CCC(O)CC1)C2 O=S(=O)(c1ccc2[nH]c(=NCCNS(=O)(=O)C3CC3)ccc2c1)N1CCC2CC12 C=C(CNC(=O)C=CC(C)(C)NC(=O)Cc1csnn1)c1ccccc1 C(CC(CC)C(=O)N1CC(C(=O)N(C2CCOC2)C)C2(CC2)C1)=CC C=CC1COCC1NC(C1CCCN(C(=O)C(C)(C)C2CCOC2)C1)=O C(=O)(CCP(C)(C)=O)N1C(C)(CC(=O)NC2CC(C)(C(N)=O)C2)CC1 c1(C(=O)NCC2CCC(CCC)CC2)cc2ccc(O)cc2oc1=O C(C)(C)(CC(C)(c1nnnn1CC1CCOC1)NS(=O)(=O)C(F)(F)F)OC C1(NC(c2cccn3nnnc23)=O)CCN(c2cnc(F)cn2)C12CCC2 N1(C(CCCC(=O)NCC)=O)CC2(CCCN(C(c3c(C)nn(C)c3N)=O)C2)C1 N1(C(CCN(CCC)C)=O)CCCC(F)(CNC(C2COCCO2)=O)C1 CC1(C)CC(C)(CNC(c2csc3cncn23)=O)CN1C(=O)CCS(C)(=O)=O c1(CC)cc(C(=O)NCC=CCNC(C2CC(C)C2(C)C)=O)c(C)o1 N1(C(=O)CC2=CCCC2)CCC2OCCN(C(C3CS(=O)(=O)CC34CC4)=O)C2C1 c1(CSc2cccc(Br)c2)cc2ccc(Br)cc2o1 Cc1cccn2ncc(C(=O)NCC3C=CCN3C(=O)C(O)CN(C)C)c12 c1(C(N(CC(C)NC(c2c(Cl)nsc2Cl)=O)C)C)ccccc1Cl c1(C=O)coc(C=CC=O)c1.c1(C(N(C)CC)=O)cccnn1.C(C)(C)C n1(CC(=O)NCCSCC(=O)N(C2CCC2)CCO)cnnn1.CCCC C1(NC(CCC=C)=O)CC2CC(NC(=O)C=CCCC(C)C)C2C1 c1(C(N2CC3(CC)CC2(CNC(=O)CCSC)C3)=O)ccnc2c1CCO2 O=C(N=c1ccnc(Br)[nH]1)C1CCC(NS(=O)(=O)C2CCOCC2)CO1 O=C(C#CC1CCC1)NC1CCC(NC(c2cc(O)ncc2Br)=O)C1 C1(NC(C2CCC(CNC(C#CC(C)C)=O)CC2)=O)CC2(CCCCO2)C1 Cc1cc(C(=O)NCCCC(O)C(=O)N(CCC(F)(F)F)C)cc(F)c1 Oc1noc2c1CCN(c1cc(-c3cccs3)ncn1)C2 C=CCCCCC(=O)N1CCCCC1CNC(c1ccc(-c2cnc[nH]2)cc1)=O C1CC2CCCC2C1.C1(C(=O)NC)(CNC(c2nsnc2O)=O)CC12CCC2 Cc1nc(C)c(C(N2CCN(C(=O)CCc3ccc(F)nc3)C3CC23)=O)nc1C c1(C(=O)NC(c2ccc(F)cc2F)COC)ccc(Br)c(OC)c1 c1(CNC(c2n(C)ncc2Cl)=O)cccc2c1CCN(C(C1(C)CCOC1)=O)C2 N1(CCF)CCC(N=c2[nH]c3c(c(=NCC4CC4c4ccccc4)[nH]2)CSC3)C1 N1(C(CSCC)=O)CC2(COC(CNC(C3COC(=O)N3)=O)C2)C1 CC(=Cn1ccnn1)C(=O)N1CCCC(CN(C)C(c2cc(=O)c(C)c[nH]2)=O)C1 n1(C(C(C)C)C#N)c(COC2COC2)n[nH]c1=O N1(C(CC2CNC(=O)O2)=O)CCOC(CNC(=O)CC2CCCNC2=O)C1 c1(C(N(CC(CC)NC(=O)CC(F)(F)CC)C)=O)cc(C)cc2ccoc12 C1(n2c(N3CC(COC)SCC3)nnc2SCCSCCO)CCC2(CC1)CC2 c1(OC)ccc(C(N2CCC(C)C(NC(c3cccnc3Cl)=O)C2)=O)c(Cl)n1 S(=O)(=O)(c1ccc2c(c1)CCO2)N1C2CN(C(=O)C)CC1C2.N1C(=O)C=CC1=O C(=O)(C(C)(C)C(C)C)N(C1CCN(C(=O)C(C)=CC=C)C1)CC#C C(N=c1[nH]cnc(NCCCNc2ccccn2)c1C)C1(OC)CCC(C)C1 CC(C)CC(C)CC(C)C(=O)N1CCC2C(NC(=O)CC3CCSC3)C2C1 N1(C(C)C)N=C(C(=O)N2CC(C)CN(C(=O)COCC(F)F)CC2C)CCC1=O C1CN(C(C2(C3CCCO3)CCC2)=O)CCC1(F)F.C1(CC(=O)N)(CC)CC1.C c1(C(=O)NC(CN(C(=O)C(C)NC(=O)NC)CC)C)ccnn2ccnc12 CCC(CC)C(F)C(=O)NC(C)(C)C=CC(=O)N(CC1CCCCC1)OC C1(NC(c2cc(C)ncn2)=O)CCC2(CC1)CC2NC(=O)C1=CCC(C)CC1 c1(CNC(C2C(C(C)C)CCO2)=O)ccc(OCC(F)(F)F)nc1 C1(C(=O)N)CCCCC1(C)C.Cn1ncc(C2CC2)c1C(=O)NCCC(C)(C)C CCC(C)(C)CC(=O)NC1(C(=O)NCC2(Cl)CC2(F)F)CCN(C)C1 C(=O)(CC(C)Cc1ccc(Cl)cc1)NCC(CO)NC(c1c(CC)scc1)=O c1(NC(CCC2(C)CCCN2C(c2cccc(O)n2)=O)=O)ccc2c(c1)COC2 C1(NC(c2c(SCC)non2)=O)CCC2CCN(c3cc(C)nc(OC)n3)C1C2 c1(OC)nc(C(=O)NC(C)CCN(C)C(c2ccc(OC)s2)=O)ncc1F c1(C(=O)NCCC2CC(NC(=O)C(F)F)C2)c[nH]cc1-c1ccccc1 C(c1cnccn1)=CC(=O)NCC(C1CC1)NC(Cc1nnc(C)o1)=O C1(NC(C(C2CCC(=O)N2)C)=O)CN(C(C2CCC(=O)N2C)=O)CC2(CC2)C1 C1(C=O)CC12CCOCC2.C1(C(=O)NCC(C)OCC#C)COC(C)C1.N C(=O)(C(=O)N=c1cc(C)o[nH]1)N1C(CCN(C(CN(C)CC)=O)C)CCCC1 Cc1ccc(C#N)cc1OC1(COC(C2CCCC2C(C)C)=O)CC1 C1(C(=O)NC2CC(NCc3ccsc3Br)C2)CCC(F)(F)C1 C1(CNC(C(C(C)C)F)=O)CN(C(=O)COc2ccccc2Cl)CCC1(C)C C1(C(N(CCCC)CC)=O)CC(C)=NO1.c1(C=O)cc(SC(F)(F)F)c[nH]1.N C=CC(CC)C(=O)NCc1cccc(NC(c2ccnc(OC)c2)=O)c1 C1(C(=O)O)Cc2ccsc2CN1C(C1CCNC12CCCC2)=O CC12CCC(C1)N(C(c1ccc(-c3ccccc3)nc1)C(=O)NCCC#N)C2 N1(C(C(C(CCC)NC(c2ccc(C)cn2)=O)O)=O)CCN2C(=O)CCC2C1 N1(C(c2c(OC)cccn2)=O)CC2CCC1CN2C(c1nc(C)n(C)c1C)=O C1(CNC(C(C2CCCO2)NC(C2CS(=O)C2)=O)=O)CCCCC1 Cc1cc(CC(=O)NCC2(F)CC(C)C2)on1.c1(C=O)cn(C2CC2)cn1 c1(COC)nc(-c2cccnc2Cl)n(-c2ccnc(O)c2)n1 C1(C(N(CCCCC(=O)NCC(O)CF)C)=O)CN2CCN1CC2 C=C(Br)CCC(=O)NCC1COCCN1C(c1ccc(C(C)=O)cc1)=O C=C1c2ccccc2C(=O)N1CC(=O)NC1CC1CNC(=O)C(C)(C)CF C1(C(=O)Nc2c3ccc(OC)cc3[nH]c2)Cn2nc(-c3ccccc3)cc2NC1=O C1(CNC(CC(C)(F)F)=O)CCC(C)(C)CN1C(=O)Cc1c(F)cccc1F N1(C(C(C)C)=O)CCN(C(C2CCC(=O)N2CCC(F)(F)F)=O)C(C)C1 C1(NC(Cc2cccc(C)c2)=O)C2CC3C1C3C2C(=O)NCC1CC12CCC2 N1(C(CN(C)C(N)=O)=O)CC(NC(c2ccc(-c3ncc[nH]3)cc2)=O)C2CC12 C12(C(=O)NCC(CC)NC(=O)C(C)OC)CC3CC1C2C3 c1(C(N2CC(C(C)NC(c3n(CC)c(O)nc3)=O)C2)=O)cn(C)c2ccccc12 C1(C(=O)OC)C2CN(C(=O)CO)CC12.C(=O)C(O)CN(C)C.C1CCC1 CC1=NS(=O)(=O)NC=C1C(=O)N1CCCC2(CCCN2C(=O)C2=CCOC2)C1 N1(C(c2n(C=C)ncc2)=O)CC2CC(NC(c3snnc3CCC)=O)C2C1 n1(CCC)nc(C)cc1C(=O)NC(C)(C)C(C)C.C1(C=O)CC(C)(C)CO1 c1(CSC)cccnc1C(=O)NCC=CCNC(c1occc1C)=O.S C(=O)C(O)CC(F)(F)F.c1(N(C)C)cc(CNC2(CF)CC2)ncn1 C1(OC(c2csc(C(F)F)n2)=O)CCCCC1OCCC(F)(F)F N1(C2(C)CC2)CCN(C(=O)C(O)CNC(C2(C)CC2(C)C)=O)CC1 c1(CN(C(c2c(C)cnn2C)C(=O)NCCC)C)cc(C)ccc1Br C1(NC(C2CN(C(C)=O)C2)=O)CCCC1.C1(C=O)CCN(CC)C1.C(C)=O CC(O)(CC(F)(F)F)C(=O)NC1CCCCC1NC(=O)CS(=O)(=O)C1CC1 C(C)(c1ccccc1F)=CC(=O)NCC(CNC(CCC#CC)=O)OC c1(C(=O)OC)cc(Br)c(Cl)cc1NC(c1cccn1C1CCNCC1)=O C#Cc1ccc(C(N2CC(NC(=O)C(c3ccc(C)cc3)C)C(C=C)C2)=O)cc1 C(=O)(C(C)(C#N)CC(=O)NC1CCCCC1)OC.c1(O)cccc(C(F)(F)F)n1 C12CC3CC(C1)CC(O)(C3)C2.N1(C(c2cnc(NC)o2)=O)C(C=O)CC2CC12 c1(NCCC(CC)C)nc(=NCc2nc(=N)n(C)[nH]2)[nH]c2c(C)nn(C)c12 Cc1ccc(CCC(=O)N)s1.C1(C(N(CC)CC)=O)CCC(C(N)=O)O1.CC Cc1cnccc1C=CC(N1CC(O)(C2CCCN2C(=O)C)C1)=O.C(C)(C)C.O c1(C(=O)N)cccc2c1CCN2.S(=O)(=O)(CC(=O)N(C1CCCCC1)C)NCC C1(Cn2cc(C3C(C)C3)nn2)CCCN(C(=O)C(C(C)(C)C)C2CCCC2)CC1 C(=O)(CCCC(F)(F)F)NC1C(SC)CN(C(c2n[nH]c3c2CC2CC32)=O)C1 C#CC1(NC(=O)C(C)C(C)NC(c2occc2COC)=O)CCCOC1 C1(F)(C(=O)NC)CC=CCC1.C1(ONC(c2conc2C)=O)CCOCC1 C1(CC(=O)NCC2C(NC(C(C)(C)CO)=O)C2)C2CC3CC(C2)CC1C3 C1(C(=O)NCCC(C)(C)NC(CCCc2cc(C)no2)=O)CC(C2CC2)=NO1 C1(C=O)CC(=O)CCO1.C1(C(=O)NCC2(SCC)CC2)CC(CC)C1 N1(C(c2ccc(CC)o2)=O)CC2(C(=O)N(C(C)CC(C)CC)C)CC1CO2 O=CN1CCCC1C(N1CCC(N(CCO)C(C2CNC(=O)N2)=O)CC1)=O CCC(CCC(=O)NCC=CBr)NC(=O)C=C(C)c1ccccc1 Cc1ccc(C(N2CC(CNC(c3cn(C)ccc3=O)=O)C(O)C2)=O)c(=O)n1C CCC(C)CC(C(=O)NCCCC(=O)N(C)C)NC(c1cc(OC)cs1)=O C12(C(=O)N)CC(C#N)(C1)C2.Cc1csc(C(=O)NC2CC(C(F)F)C2)c1 C1(C(N2CC(CC(C)NC(C3(C)CCCCC3)=O)C2)=O)CC2(CCCC2)CO1 C(=O)(CCC1CCc2ccccc21)N1CC=CC(NC(COCC(C)(C)C)=O)C1 C1(CC(=O)NC2(C)CN(C(c3c[nH]c(C(F)(F)F)c3)=O)C2)CCCCCC1 c1(NC(CN(C(=O)C(C)OC(C)=O)CC)=O)ccc(C)nn1.C1CO1 c1(C(N2CC(C)(NC(C(CC)OC)=O)C2)=O)cc(C#N)c(SC)nc1O CC1(C)C(C#N)C1(C#N)C(=O)NC1CC(NC(c2ccc3ncccn23)=O)C1 C1(N(C(=O)Cc2cnsc2)C)CN(C(=O)C=CC2(C)CCOCC2)CC1(C)C Cc1nccc(C(=O)N(C2CCN(CC(F)F)CC2)C)c1O N1(C2CN(C(CCc3[nH]c(=N)sc3)=O)C2)CC(NC(c2cnc(O)o2)=O)CC1=O c1(C(N2CC(NC(=O)CSC3CC3)(CO)C2)=O)ccnc2cc[nH]c12 Cc1cnn(C)c1C(=O)NCC1(O)CC(CNC(c2ccccc2)=O)C1 O=C(CCCCc1ccccc1)NCC1CCN(C(C2CC3(C2)CC3F)=O)C1 N1(Cc2n(-c3ccc(C(=O)O)cc3)ncc2C(=O)O)CC2(C1)CC2(F)F c1(CC(N2CCN(C)CC2CNC(C2C=CCC2)=O)=O)c[nH]c2cc(F)ccc12 C1(CC(=O)NCC2CC(NC(C3(CCO)CC3)=O)C2)CC1(Cl)Cl C1(C(=O)N)CN(C)CCO1.C(C(F)C(=O)N1CCCC1C(C)C)N(CC)CC c1(C(N2CC(NC(c3n(CC)nnc3C)=O)C(C)C2)=O)cn2c(n1)COCC2 c1(COC)ccccc1CC(N1CC2CC2(NC(C2CCN(C)C2)=O)C1)=O c1(NC(CC2(C)CN(Cc3cnccc3Cl)C2)=O)ccc(F)cc1Cl c1(NC)cnc(Cl)cc1C(N1CC2(CCC2NC(=O)CCc2cccnc2)C1)=O c1cc(=NCCC2CCOC2)[nH]c(CC2CC2)n1 N1(C(CP(C)(C)=O)=O)CCCN(C(C2CN3CCCN2CC3)=O)C(CO)C1 c1(CC(=O)NCC(C(C)C)NC(Cc2scc(C)c2)=O)coc2ccccc12 C=C=CC(C)C(=O)N(C1CCCN(C(C2(CC=C)CC2)=O)C1)CCF c1(CC(=O)NCCCN(c2ncc(Br)cn2)C2CC2)ncncc1Cl c1(C(=O)NC2C(NC(=O)C=Cc3cc[nH]n3)COC2)ccc2ccnc(Cl)c2n1 C1(C=O)CCC(S(N)(=O)=O)CC1.Cc1cc(C(=O)NC(C)CC(C)C)oc1C.N c1(C(=O)NCC(C)(C2CC2)NC(=O)CC2CCOCC2)ccn2nnnc2c1 Cc1c(C(N2CCC(C)(CC(=O)NC(C)Cc3cnc[nH]3)C2)=O)c[nH]c1C#N n1(C(C)C)cnc2c(N3CCC(CF)(NC(=O)COC4CC4)C3)nc(Cl)nc12 c1(C(=O)NCC2(OC)CCN(C(C(C=C)O)=O)C2)c(F)cccc1[N+](=O)[O-] N1(Cc2cccc(C)c2)CCC(NC(c2cccs2)=O)C(C)(C)C1 c1(C(N(C2C3CN(C(c4nn(CC)c(C)c4)=O)CC32)C)=O)cnn2ccn(C)c12 C1(C(=O)NCC2(C)CCN(C(c3cn(C)nn3)=O)CC2)CCc2nc(O)[nH]c2C1 CC1CCc2nc(C(N3CCC4CN(C(=O)CCC(N)=O)CC34)=O)ccc2C1 C(CC(C(C)(C)C)NC(=O)COc1cccnc1Cl)N(C)C(c1ccns1)=O CCCCC(C)(F)C(=O)NC1CC(NC(c2noc(CC)c2C)=O)C1 C1(CC#N)C2CN(C(=O)CNC(=O)NCC3CC3)CC12 N1(C(CS(=O)(=O)NC(C)(C)C)=O)CCN(C(=O)C(C)(C)C2CCOC2)CC1.C N1(C(c2n(CCC)ncc2)=O)CCOCC(F)(CNC(C2(CC)CCOC2)=O)C1 C1(C(=O)NC2CC(C)(CNC(c3c(C)cccc3)=O)C2)CC(C2CC2)=NO1 c1(-c2cc(C)c(F)cc2C)ccc2nc(C(=O)Nc3cc(Cl)nc(Cl)c3)oc2c1 c1(C(N2CC(NC(c3c(OC)n(C)nc3C)=O)C2)=O)ccnc2c1CCO2 c1(C(=O)NC2C(NC(C3(F)C(C)C3)=O)CCCC2)ccn2c1CCCC2 N1(C(CC=CC=C)=O)CCC2CCC(C1)N2C(=O)C(C)S(N)(=O)=O C1(C(N)=O)(CNC(C(C)OC)=O)CN(C(=O)COC)C1.C1CCC1 C(CC(F)(F)C(F)(F)Br)NC(c1cc(C)n(C)c1C)=O.c1cn(CC(C)C)nn1 C1(C(N(CCC)C2CC2)=O)CC(NC(C2(CCN(C)C)CC2)=O)C1 C1(C(N2CCC(OCC=C)C2)=O)CCN(C(c2cc(C)ns2)=O)C(C)(C)C1 c1(C(N2C(C(=O)Nc3cc(OC)cc(Cl)n3)CC(=C)C2)=O)c(C)ccc(C)c1O N1(C(c2cnc(CC)nc2C)=O)CC2CC(NC(=O)C(C)(CO)OC)CC(C2)C1 N1(CC=CC(=O)N(CC(C)CNC(C2CC2(F)F)=O)C)CCOCC1 C1(=CC(=O)NC(CNC(C2N(C(C)=O)CCC2)=O)CO)CCCCCC1(F)F C=CCCCCCC(=O)NC12CCN(C(c3ccc(Br)o3)=O)CCC1C2 C(=O)(CCC(F)(F)C(F)(F)F)N.C#CCC(C(=O)NCC1CCCCC1)C1CC1 c1(NC)ccc(C(=O)N)cc1[N+](=O)[O-].C(C1CC1)=CC=O.CC.CC.CC C1(NC(N(c2cc(C)cc(C)c2)CC)=O)CCc2c(Br)cccc2C1 c1(C(=O)NCC(C(C)(C)C)NC(C2CCC(C)(O)CC2)=O)ccc2n[nH]cc2n1 N1(C(COCC)=O)CCN2CCOCC2(CNC(=O)C(C)c2ccco2)C1 C(=O)(CCC(C)(F)F)NCc1ccc(-c2cn(CCOC)nn2)cc1 CC(CNC(=O)CC1CC=CC1)C(=O)N(C)CC1CCOCC1 N1(C(C2N(C(Cn3ncc(C#C)c3)=O)CC3CC32)=O)CCC2(CC1)CC2C#N c1(OC)cc(CN2CCCC(C)(C(=O)NCC(=O)N)C2)cc(C)c1.CC(C)C C1(CNC(CC=C=C)=O)COC(C)(C)CN1C(c1cn(C)c(C)n1)=O c1(C(N2CC(NC(c3c(C)nn(CCO)c3)=O)C2)=O)cc(O)c2ccccc2c1 Cc1cccc(Cl)c1CC(=O)N(C)CC1COCCN1C(=O)CC(O)C1CC1 CS(=O)(=O)c1ncc(C(=O)NC2CCn3nccc3C2)s1 CN1CCN(CC(=O)NC2(CF)CCN(C(=O)Cc3ccccc3Br)C2)CC1 c1(C(=O)NCC(CN(C(C2CCCS2)=O)CC)(C)C)cc(C(F)F)ncn1 c1(OC)ccc(CC(C)C(=O)NCCC(C)NC(=O)C=CC(C)(C)S)cc1 c1(C(N2CCN(C(CCC(=O)OC)=O)C(CF)C2)=O)cnn2c1OCC(O)C2 CCCC(C)(CC)C(=O)NCC1CC1NC(c1ccccc1)=O.C(=O)CC#N CC1(C)CC(C(N2CC3CC(NC(=O)C(F)=CC4CC4)C2C3)=O)CC(C)(C)C1 C(C1CCCN1C)=CC(=O)NC(COC)C(=O)NCC(N1CCCC1)C c1(OC)cc(NC(C2CN(C(=O)C(OC)OC)CC2C)=O)cc2c1OC(C)C2 c1(C(N2CC(C)C(CC(=O)NC34CC3COC4(C)C)C2)=O)ccnc(O)c1F c1(C=O)ccc(OC(F)(F)F)cc1C.n1(CC(=O)N(CC)CC)ccnc1C.N C(c1ccncc1C)=C(C)CNC(=O)CNC(=O)C(C)Oc1ccccc1F c1(C(=O)NC(CC)(CC)CCNC(=O)C=CCO)cc(C)cn2ccnc12 N1(C(CCCNC)=O)CCCN(C(c2cccc(Cl)c2Cl)=O)CC1 c1(NC(C(C)C)=O)ccc(CCOC(C2C3CCC(F)(F)C23)=O)cc1Cl CCC(CC)CC(=O)N(C1CCCCC1NC(c1cc(C(F)(F)F)n[nH]1)=O)C C1(CNC(c2ncc(C)cc2C)=O)C2CCCC1N(C(c1cc(CO)[nH]n1)=O)C2 N1(C(C(C)C2CC2)=O)CCC(NC(c2ccncc2)=O)C1.C1CCC1.C1CC1.O c1(CNC(C2(C)CC(=C)C2)=O)cccc(F)c1.c1(C=O)cc(C(C)C)on1 C1(NC(C2N(C(=O)NC)CCC2)=O)CCC(NC(=O)CC#N)CC1 O=C(C1=CCSC1)NCC1CC1CNC(c1cc(-c2ccccc2Cl)[nH]n1)=O N1(C(CCCOC)=O)CCC2(NC(=O)Cc3c(C)noc3Cl)CCCCC12 n1(CC#C)c(C)cc(C(=O)NCCC2(C)CC2)c1C.C(=O)CNC=O.N CC1CCC(CN(C2CCC2)C(=O)NCc2cnn(C)c2)C1 C1(CC)CN(C(c2cscc2C)=O)CCC1NC(c1cc(C2(C)CC2)n[nH]1)=O c1(C(=O)Nc2c(C(N(CC(F)(F)F)CC)=O)cccc2)c(C)nc2sccn12 N1(C(C(C)O)=O)CC(NC(c2csc(Cl)c2Cl)=O)C2(CCOCC2)C1 N1(C(C)=O)CCN(CCN(C)C(c2c(C(F)(F)F)ncn2O)=O)CC1.C#CCO c1(C(N2CCC(F)C2)=O)cc2nn[nH]c2cc1F.C(C)(C)(C(=O)NC)OC(C)C C#CCCCCCC(=O)NC12CCN(C(c3ccc(C(N)=O)o3)=O)CC1C2 c1(C(N2CC(NC(C(C)OCC=C)=O)C(C)C2)=O)cccc(C(F)(F)F)c1C C1(C(N(C2CCCN(C(C(CSC)C)=O)CC2)C)=O)CCC([N+](=O)[O-])CC1 N1(CCCC=O)C(=O)CN(C)C1=O.C(CC1CC1)(C(=O)NCC(C)C)OC N1(C(C(C2CCCC2)NC(C)=O)=O)CCC(N(CC(=O)NC(C)(C)C)C)CC1 c1(NC(=O)NCC2(CCO)CN(C)C2)ccc(N(C)C)c(C#N)c1 c1(OC(CC2CC(OCCC)C2(C)C)=O)ccnc2c(OCC)cnn12 O=C(C1=CCN(C(C2CCCCCCC2)=O)C1)N1CC=C(CO)CC1 C1(C2CC2)(C(N(C(CCCC)C)C)=O)CN(C(=O)C=CC(F)(F)F)C1 c1(C(=O)NCC(C)NC(Cc2ccc(C(C)=O)s2)=O)coc2c(F)cccc12 C=CC(C)(CC)C(=O)N1CCC(O)(CNC(=O)CCN(C)CCO)C1 C1(C(=O)NCc2c(C)cncc2)CCN(C(=O)Cc2cnn(C)c2)O1 N1(C(CN(C)CC)=O)CCCC1C(c1ccccc1)NC(=O)C(C)OC C#CC12CC(CN1C(c1nnc(-c3ccc(Br)cc3F)s1)=O)C2 C(CCC(C)CCC(C)NCCN(C)CCc1ccccc1)=C(C)C C12(CNC3C(C)CN(C(=O)C[SH](=O)=O)C3)CCCCC1NC(=O)C2.C(C)(C)C C1(NC(c2cc(CC)ncc2)=O)CCC2(CC1)CC2.c1(C(=O)N)cnn(C)c1N CCC(C)C(C(=O)N1CC(OCCOc2ccco2)C1)N(C)C c1(C(=O)N)c(F)cc(F)c(F)c1F.C1CC2(C1)CN(C(C1C3COCC13)=O)C2 CC1(C)CCC(C(=O)NCC(C)(O)CNC(=O)C=CC(F)(F)F)CC1 C(N=c1ccnc(N2CCC(C#N)CC2)[nH]1)C1C(C)COCC1 CS(=O)(=O)C1CC(C(N2CCC(NC(C3CN4CCC3CC4)=O)C(CO)C2)=O)C1 C(C)(C)(CCCNC(=O)CCCC1CC1C)NC(C(C)=C1CC1)=O C(=O)(C1Cc2c(Cl)cccc21)N1CC(NC(c2cnn3c2CC(C)CC3)=O)C1 S(=O)(=O)(c1cccc2c1OC(C)C2)Nc1nc(CC)c(C(=O)OC)s1 c1(NC(C2CCCC(OC)C2)=O)cc(=O)n(CCO)c(O)n1.c1ccc(F)cc1 CCC(C)CCCCC(=O)N1CCCCC1C(=O)NOCCOCCO c1(C(=O)NCCN2CCC(NC(C(CCC)(C)O)=O)CC2)ccnc2ncnn12 c1(C(=O)NCC23C(CN(C(C4(OC)CC4)=O)C2)C3)cc(C)c(C)cc1C c1(C(=O)OCC)cc(Nc2cccc(C(F)(F)F)c2)c(C)cc1[N+](=O)[O-] C1(NC(c2nc(CC(C)C)sc2)=O)CCC12CN(C(=O)CC1CCCC1(F)F)C2 c1(C2C(NC(C(c3ccc(Cl)cc3)OC)=O)C2)cc(F)cc(F)c1 N1(C(C2C(CNC(Cc3cn(C)nc3)=O)C2)=O)CCCOCC1 C1(C(N(CCC(C)NC(c2cc(O)cs2)=O)C)=O)CCC(Nc2cnccn2)C1 C(C(=O)NC1CC2CCC1C2)(C(C)(C)C)NC(=O)OC.c1(C=O)ccsc1 N1(C(c2ccn(CC(C)C)n2)=O)CCN(C(C2CC(=O)C2C)=O)C(C2CC2)C1 CCC(C)(C)CNC(=O)CC1CCCC1NC(=O)CC.C(=O)C1CC1.N CCCC(C(=O)OC)C(=O)NC1(CCC(=O)N(C2CCC(C)(C)C2)C)CCCC1 c1(CCC(=O)NCC=CCNC(=O)C(F)(F)C(F)F)ccc(F)cc1F c1(C(=O)NCCCN(C(=O)CCC(N)=O)C)ccc(Oc2ccccc2Cl)nc1 N1(C(C=Cc2ccc(C)cc2)=O)CC(C)CC(C)(C)C1.C(=O)C(C)CC1CC1 C1(NC(c2nc(-c3ccc(C)o3)sc2)=O)CCN(C(C2CC(F)C2)=O)CC1 C1(N(C(=O)C2=CCCCO2)C)CC2CC(C1)N(C(=O)C(=O)Cc1cccs1)C2 c1(CC(=O)Nc2c(C)nc(C(F)(F)F)s2)c(C)nc2c(c(C)nn2C)c1C CCC1=NOC(CC(N2CC=CC(NC(=O)CCCOC)C2)=O)C1 C1(NC(c2cccc(C)n2)=O)COCCN(C(c2cnc(C(C)(F)F)s2)=O)C1 N1(C(=O)CCC2CC2)CCN(C(c2csc(-c3ccccn3)n2)=O)C(C(F)F)C1 Cc1noc(C(N2CCCC2CCCNC(=O)CC2CCCCN2C)=O)c1C c1(NCCN(CCC)CCC)nc2c(C(=O)O)cccc2s1 N1(C(CSC(C)=O)=O)CCC2(CC1)CC(NC(C1CCCCCCC1)=O)CO2 C1(CNC(C2OCC(C)C2)=O)(NC(=O)CS)CC(F)(F)C1.c1nc[nH]n1 NS(=O)(=O)c1csc(C(=O)NC2CN(C(=O)Cc3nc[nH]n3)CC3(CC3)C2)c1 C1(CC)CN(C(=O)CNS(C)(=O)=O)CCN1C(c1cc(O)nc(Cl)c1)=O N1(C(C2CC(C)CN2C(=O)C(C)(C)F)=O)CCN2CCCC2C1 C1(OC(C)C)CCN(C(C2(C)CCCN2C(=O)CC2CCOC2=O)=O)CC1 C(=O)(C(CC(C)C)NC(=O)C(N1CC2CCC2C1)c1csc(Br)n1)OC N1(C(C=C(C)C)=O)CCC2CCC(C1)N2C(C1C2CC3C(C2)C13)=O C1(CNC(C=CC)=O)(NC(=O)CC2(C)CC(F)(F)C2)CCCCC1C C1(CC)(NC(c2nccc(OC)c2C)=O)CCCN(C(C2OCCOC2C)=O)C1 C=CC1(CNC(C2C3CN(C(=O)CCCCC#N)CC23)=O)CCOCC1 N1(C(CC(C)(C)OC)=O)CCCC2(CNC(C3CCCCN3C)=O)CCCC12 C1(NC(C2C(OC)CCCC2)=O)CCC2CC1CN2C(=O)Cc1cnnn1C c1(C(=O)NCCC(CNC(=O)CCc2cscn2)O)cc2cccnc2s1 C1(CNC(C(c2cscn2)N(C)C)=O)CCCCC1NC(C1(C)CCCO1)=O c1(C(C(=O)NCCC2(C)CC2)N(CC(C)(F)F)C)cccc(Br)c1F N1(C(C(OCC)OCC)=O)C2CCC1CC2.C1(C=O)CC2(C1)CC(O)C2.C c1(N2CCN(C)C3(C2)CC3)cccc(S(=O)(=O)NCCCOCC2CCOC2)n1 CCCC(C(=O)O)NC(=O)OC(C)(C)C.CC(=O)N(C1CCC1)C1CC1 C1(O)(CNC(Cc2ccc(C)nc2)=O)CCCN(C(c2cnc(C(C)C)[nH]2)=O)C1 c1(C(N2CCC(CC=C)(NC(C3CC(F)C3)=O)C2)=O)cc2n(n1)CCCO2.C CC1(C(N2CCCC(CC(=O)NCCc3ccccn3)C2)=O)C=CCCC1 Cc1cccc(NC(=O)C(=O)N(C2CCN(C(C3CC(C)(F)C3)=O)C2)C)c1 c1(C(C(=O)OCC)C2CN(C(=O)C(CC)OCOC)C2)ccccc1 N1(C(CC(CCC)O)=O)CCC(N(C)C(c2cc(OC)ccc2Cl)=O)C2(CC2)C1 C(=O)(C(F)(F)C(F)F)N.n1(COCC)nnc(C(N2CCCC(CC)C2)=O)c1N c1cc(F)cc(Cl)c1.C(C(F)(F)F)=CC(=O)NC(CN(C1CCSC1)C)=O C(CC1CCC1)(C(=O)NC1(CO)CC1)NC(C1N(CC)CC1)=O C(=O)(CC(C(F)(F)F)NC(c1ccc2cc[nH]c2n1)=O)N1CC(O)(C(N)=O)C1 C1(CC)CCCC1C(=O)NC1(C(C)C)COC1 c1(C(=O)NC2C(NC(C(C)(c3ccccc3)OC)=O)C2)ccc(Cl)c(N)c1 C1(CC#C)(C(N2CCC(C(=O)NC3(C(N)=O)CC3)C2)=O)CCCO1 C1(CNC(CC2(OC)CCC2)=O)CC2CCC(C1)N2c1cc(Cl)ncn1 N1(C(c2c(CC)non2)=O)CC2CCCN(C(C34CC(CO3)C4)=O)C2C1 n1(CC(=O)N(CCNC(=O)CCc2cnc[nH]2)C2CC2)cnccc1=O N1(C(C(C)NC(N)=O)=O)CCCC(CCNC(C23CSCC2C3)=O)C1 C1(C(=O)NC2CCN(C(c3cnc(C)s3)=O)C2C)CCCN(C(C)(C)C)C1=O CCCCCC(O)CC(=O)NC1CCN(C(c2nccc3occc23)=O)CC1O C1(NC(Cc2cc(C)[nH]n2)=O)CCC12CCN(C(c1coc3c1COC3)=O)CC2 Cc1nc(CSCCC2CNCCS2(=O)=O)c(CO)c(C)c1C Cc1nc(C(=O)NCC2(C)CC(NC(C3CCOC3)=O)C2)c2ccnc-2[nH]1 CCCCCCCCCn1cc(C2CCN2C(C23CCCN(CCC2)C3)=O)nn1 Fc1ccc(F)c(CNCC2CC(F)(F)CO2)c1.C12CCCCC1C2 Cc1ccc(C)c(N(C)C(c2occc2CNC(=O)CSC(F)F)=O)c1 C1(C(=O)N)CCN(S(N)(=O)=O)CC1.N1(C(C=C(CC)C)=O)CCCC1C(C)C C1(C(C)C)N(C(c2ccc(Cc3nn[nH]n3)cc2)=O)CC12CCSCC2 O=C1COCC2(CN(C(=O)CC3CC4(CC4)CN3C(c3cccc(O)c3)=O)C2)N1 C1(C(=O)NCC(CC(=O)NCCCCN2CCC2)O)CCCC12CCC2 O=C(CCCCC1CC1)N1CCN(c2ccc(C(N3CC=CC3)=O)cn2)CC1 C1(CC)CN(C(=O)Cc2cccs2)CCC1NC(=O)C=CCO c1(C(=O)OC)ccc(F)c(OC)c1C(=O)OC.c12cccc(c1)NCCC2 C(=O)(C1=CCCCC1)NCCC1CC(NC(c2c(C)sc(Br)n2)=O)C1 CC1CCC(NC(c2ccc(=N)[nH]n2)=O)CN1C(c1csnc1Cl)=O c1(C(=O)NCCCCCNC(CSCCOC)=O)nc(C2CC2)ncc1Br Cc1cc(C(=O)NC2(CNC(C3CCCCC3O)=O)CCC2)nc2[nH]nc(O)c12 C(=O)(C1=C(C)OCCC1)N1C(C)CCC(C(=O)NCC(C(=O)OC)C)C1 c1(CC)cc(C)ccc1C(=O)NCC1(NC(c2ccnc(C)c2)=O)CCC1 C(CCC(=O)N1CCCC1C(C)CCC)NC(CC=CCC)=O c1(OC)ccc(CC(=O)NCCC(C)CCNC(=O)CN2CCCC2)cc1Cl Cc1c(C(=O)N(CCN(C(=O)CC2CCC2C2CC2)C)C(C)C)cnn1C CCC(CCC(=O)NC(c1cccnc1O)C)NC(c1coc(CO)c1)=O Cc1cc(C(=O)NC)cc(N)c1Cl.C1CN(C)CCN1C(=O)CN(C)C(N)=O N1(C(C2(OCC)CCC2)=O)CC2CN(C(=O)Cc3nc(F)c(F)cc3F)CC2C1 CC(C)CC(O)C(=O)NCC1CC1CNC(=O)CCc1ccc(F)cc1F N1(C(C(CC)CCOC)=O)CC2CCCC(C1)N2C(C1CCCCCN1C)=O N1(C(CC2(OC)CCC2)=O)C2CCC1CN(C(c1csc(C(C)C)n1)=O)C2 c1(NC(=O)NC2(C(=O)OCC)CCCC2)ccc(C(=O)OC)c(Cl)c1 C1(C(=O)NCC(C)CNC(=O)CC2CSC2)CCC(C)CC1 Cc1nc(Cl)c(C)c(=NCC(C)(C2CC2)NC(=O)C2=Cc3cc(F)ccc3OC2)[nH]1 CC(C)C(O)C(C)(C)C(=O)NCc1ocnc1C(N1C(CO)CC1C)=O C(=O)(CC(O)CCSC)NCCCN(C(c1nn(CC)nc1Br)=O)CC Cc1[nH]nc(CN2CC(O)C2)c1C(F)(F)F.C1(CC=O)C=CS(=O)(=O)C1 CCCCCCC(=O)NC(CC(F)F)C(=O)NCCCCCC1CC1 CCC(CC(=O)NC1CC1CNC(c1ccncc1C)=O)C(C)C C12(NC(c3ccc(CC(N)=O)cc3)=O)CCCC(CN(C(c3ccco3)=O)C1)C2 C(=O)(C#CC(C)(C)C)NCC(CNC(c1c[nH]nc1C1CCOC1)=O)OC C1(O)(CNC(c2ccccc2C2CC2)=O)CCCN(C(c2cnc(Cl)s2)=O)C1 Cc1cc(N2CC(NC(c3ccc(C4CC4)c(F)c3)=O)CC(C)C2)nc(C)n1 c1(CC(C(=O)NC(C)CN(C)C(c2cccnc2)=O)C)ccc(F)cc1F C1(NC(COC(C)(C)C)=O)CC2CCC1(NC(=O)CCc1ncco1)C2 c1(NCC(N2CC(C#C)(C(=O)OCC)C2)=O)cc(OC)c(O)cc1[N+](=O)[O-] CC1(C)C(NC(c2cccc(F)c2Cl)=O)CCN1C(=O)COc1cccnc1 C1(NC(C2(C)CCCCC2)=O)CC2CC(C1)CN(C(C1CC3CCC(C1)O3)=O)C2 C1(NC(=O)NCc2nccs2)COC2(CCOCC2)C1O c1(NC(C2CCCC(S(C)=O)C2)=O)c[nH]c2c(Cl)cccc12 CCCC(CCCO)C(=O)NC1(C)CN(C(c2ccn(CC(F)F)n2)=O)C1 N1(C(C)=O)CCC(NC(=O)NCC(C)S(C)=O)c2ccccc21 C(=O)(CCCN=[N+]=[N-])NC(CCSC)C(=O)NC(c1nc(C)oc1C)C Cc1nc(C(N)=O)ccc1NC(c1nc(Cl)sc1Cl)=O c1(OC)cccc(C(C(=O)NC2CCCCC2)C(C)C)c1.C1(C)(C(=O)N)CCC1 CCC(C(=O)N(C)CC1CCCN1C(=O)Cn1cc(N)cn1)C(C)O c1(CC(N2CC3C(CNC(=O)CC4CC45CC5)C3C2)=O)cccc2c1OCCO2 N1(C(C2(CC#C)CCOC2)=O)Cc2ccc(-c3nn[nH]n3)cc2C1 c1(OC)c(C(=O)NC2(CF)CCN(C(=O)C(C)C)C2)cccc1[N+](=O)[O-] c1(C(N(C2CCC2)C)=O)ccc(N)c(Cl)c1.c1cc(F)cc(F)c1.C(=O)(C)N c1(OC)ccc(O)cc1C(=O)N(C(C)CNC(=O)Cc1ccon1)C C1(C(=O)NCC(C(=O)NC)C)CCCN1NC(=O)C1(O)CCSCC1 N1(C(C=Cc2n(C)ccc2)=O)CCC12CN(C(=O)CCC1CCC(=O)N1)C2 c1(C(N2CC(CNC(C(CC)=CC)=O)N(C)CC2)=O)ccc(C#N)c(F)c1 c1(C(=O)NC2(CO)CN(Cc3c(OC)cccc3Cl)C2)ccc2c(ccn2C)c1 N1(C(C)=O)CCC(C)(C(=O)N(C)CCNC(=O)CC(C)C2CCCCC2)C1 Cc1c(CN(CC(C)NC(C2(C(F)F)CC2)=O)C)cccc1Br c1(C(=O)NC2CCN(C(c3ccc(C#N)cc3F)=O)C2)ccc2c(c1)COCC2 c1oc(C)nc1C=O.C1CN(C(=O)CC2CC2(C)C)CC1.C1CC1.CCO c1(C(=O)NC(C)CNC(=O)COC2CCCCC2C)cccn2nnnc12 CC1CCCn2c(C(=O)NCC3(O)CN(C(=O)CCn4cccn4)C3)cnc21 C1(CC)CN(C(=O)CCc2cnn(C)c2C)CCC1NC(c1ccc(OC)s1)=O N1(C(=O)Nc2c(C3CC3)cccc2Cl)CCCC2(CCOC2)C1 C1(NC(=O)Cn2cncn2)C2CC3CN(C(=O)CCCc4ccccc4)C1C3C2 c1(-n2c(C)nnn2)cc(C(=O)NCC2CCC2)ccc1Cl.C1(C=O)CC(O)C1.N N1(C(CC=C=C)=O)CC2CCCC2(NC(c2ccc(Br)c(O)c2)=O)C1 C#CC1(CC(=O)OC)COC1 Cc1nc(CCC(=O)NCC2(O)CN(C(C3CCN(C)C3)=O)C2)oc1C C1(CNC(CN(CC(C)(C)C)C)=O)C=CC(NC(C2CCC3CC23)=O)C1 C1(CNC(c2ccnn2C2CCOCC2)=O)CCN(c2nncs2)CC1(F)F c1(CNC(C(N2CCC(O)(CC)C2)=O)=O)cc(C(F)(F)F)ccc1Br C(=O)(C(C)(C)CNC(c1ccc(OC)s1)=O)Nc1cn(CC#C)nc1 N1(C(c2cc(C(C)(F)F)n[nH]2)=O)CCCCC1CNC(C12CC(F)C1C2)=O c1(C=O)cc(C(F)(F)F)cc(O)n1.C1(NC(CCCSC)=O)CC2(C1)CC2.N C(=O)(C1CC(O)c2ccccc21)OCC(=O)Cc1ccccc1Br C1(CNC(C(CCOC)C)=O)CCCCN(C(=O)CCOCCOC)C1 c1(C(CC)CC)cc(C(N2CCC(CCNC(c3coc(SC)c3)=O)C2)=O)on1 C1(NC(C2(CCC=C)CN(C(C3CCCCO3)=O)C2)=O)CCCCC1N(C)C C(=O)(CS(=O)(=O)c1ccccc1)N1C(C(=O)N=c2cc[nH]cc2Cl)CC2CC21 N1(C(CC)C)CCC(NC(C)=O)CC1.C123CC(CN1C(=O)Cn1cc2nn1)C3 C1(CCNC(c2cc(COC)no2)=O)CN(C(C2CCCN2C)=O)CCCO1 c1(C(=O)NC(CNC(c2c(CC)cno2)=O)(C)CO)cc(C)ccc1O C(=O)(C#CC1(C(F)(F)F)CC1)N(C(C)C)C.Cc1cc(COCC=O)on1.N N(C(=NCc1nc(C)c(C)s1)NCC1(C(C)C)CCCC1)C(C=C)C c1(C(N(C(CNC(c2c(SC)snn2)=O)C)C)=O)ccc(O)nc1Cl C1(C(N2CCCN(C(C(C)C3CCCC3)=O)CC2)=O)CCn2cncc2C1 CCC(CC)(CC)C(=O)NCC1CC1C(=O)NC1CCCC1CF C(C)(C)(CC(=O)NCCC1(C)CCCO1)N(C(=O)CC1C=CCCC1)C c1(C(=O)NC2C(C)(CNC(C(C(C)O)(C)C)=O)CCC2)ccc2ncncc2c1 CC1CCCN(C(C2OCCC2NC(=O)C=CC(=O)N(C)C)=O)CC1 Cc1cccc(-c2ccc(C(=O)NCCN(C(=O)CN3CCCCC3)C)n2C)c1 N1(C(=O)CC2CSCCS2)CCCN(C(c2cc3cccnc3s2)=O)CCC1 C1(C(=O)NC2CCC(CCNC(c3c(OC)nsc3)=O)C2)CN2CCCN1CC2 C1(NC(c2cnccn2)=O)CN(c2ncnc3ccsc23)CC2(CCC2)C1 Fc1cc(C(c2nnnn2C2CCOC2)NCCCc2ccccc2Br)ccn1 O=C1NCCCCC1C(=O)NCCNC(=O)CCNC(c1ccoc1)=O N1(C(CC=CCNC(=O)Cc2cccnc2O)=O)CCc2c[nH]nc2C1 C=CC(C)(C)CC(=O)NC1CC(NC(=O)CCOCC2CCCO2)CC1O CCCC(O)CC(=O)N(C1CN(C(c2ccc(C3CC3)cc2)=O)CC1O)C N1(C(=O)CSCC(F)F)Cc2ccc(CNC(C3(CO)CCC3)=O)cc2C1 c1(CC(N2CC(NC(CN(CC=C)C=O)=O)C2)=O)csc(Cl)n1.C=O c1(CC(C(=O)OC)NC(=O)C(C2CCOCC2)C)c[nH]c2cc(F)ccc12 C(=O)(C1=CCCSC1)N1C(C=CC(=O)N(CC(C)(C)C)CCC)CCC1 C(=O)(CCC(=O)C(C)(C)C)NC(CC(=C)C)C(=O)N1CCCC(C)CC1 N1(C(CN2CCN(CC)CC2)=O)CCN(C(=O)C(C)C)CC1C1CCCC1 c1(CC(=O)NCCCNC(=O)C(C2CCCCCCC2)O)ccc(Cl)c(F)c1 C(CC(C)C)(C(=O)N(C)OCC(F)(F)F)NC(C=C=C(C)C)=O c1(C=O)ccc2nc(C(F)(F)F)cn2c1.C1(NC(CSC(C)C)=O)CCC1C CCC(C)CC(C)C(=O)NCC1CN(C)CCN1C(=O)Cn1ccc(=N)[nH]1 C(C(C)(CC(C)C)NC(=O)CC1CC2(CC2)CO1)NC(COCCCC)=O C(CS(=O)(=O)C1CCCC1)N1CC(C(=O)O)C(O)CC1 c1(C(=O)NC(C(C)NC(c2c(C)n(C)nn2)=O)C)cc(Cl)c(Cl)n1C c1(C(N(C)CCN(C)C(C2CCC([N+](=O)[O-])CC2)=O)=O)cc2ccc(O)nc2s1 C1(C(N2CCOCC(NC(CN(C(C(C)C)=O)C)=O)C2)=O)CCn2cncc2C1 Cn1cccc1C(=O)NC1CC(C)C1.c1ccccc1.C1(C=O)CC1.C=O.N N1(C(C(C)=C2CCC2)=O)CCN(C(C2C3COCC23)=O)C(C)C1C C(=O)(C1=CCCN(C(=O)Cc2csc(C)c2)C1)NCCc1nc(C)on1 N1(Cc2ccc(C(=O)OCC)s2)CCCC2(CCc3cnc(C)nc32)C1 Cc1ccc2cc(Oc3cc(-c4ccc(N(C)C)c(F)c4)cc(F)c3)ccc2n1 CC1CC(NC(=O)CN(C)Cc2ccccc2)CN1C(c1cccnc1)=O c1(N2CCC(CC=C)(NC(C(CC=C)C)=O)C2)nc2ccc(N)cc2s1 O=C(CCCC(=O)N1CCCC1C1(NC(c2cccc(Cl)c2F)=O)CC1)C1CC1 c1(CCC(=O)NCc2n(CC)ncn2)cncc(Br)c1 c1(C2CCC(C)O2)nc(Cc2cnn(C)c2)nn1-c1cccc(C(N)=O)c1 c1(OCC)c(NC(c2nnc(C)s2)c2nnnn2C(C)CC)cccc1Cl N1(C(C2C(C(=O)OC)CCO2)=O)CC2CCC2C1.c1(CC(=O)N)cnn(C)c1 C1(NCCCc2c(OC)cccc2)CCN(C(c2ccc(Cl)o2)=O)CC1C C1(NC(C(c2ccccc2)C)=O)CC2CC(NC(C3CN(C)C3)=O)CC2C1 C1(N(C(C(C)(C)n2cc(CCCCO)nn2)=O)C(CO)C(=O)O)Cc2nccn2C1 C1(CC)CCN(C(c2csc(C(C)C)n2)=O)CC1.N1(C(C)=O)CCC(C(=O)N)C1 C12(NC(c3nnsc3-c3ccccc3)=O)CCOCC1CN(C(C1CCC1)=O)C2 c1(C(=O)N)ccc(O)nc1C.C1(NC(C2N(C(=O)NC)CCC2)=O)CCCCC1 C12(NC(C(CCC)NC(c3cc(CC)n(C)n3)=O)=O)CCC(CC1)C2(C)C c1(C(=O)NCC2CN(C(C(C(C=C)C)C)=O)C2)ccc2cc(C)cn2c1 N1(C(C2C(C)C2(F)F)=O)CC(CNC(c2ccnn2CC#N)=O)C(C)(C)C1 C1(CNC(c2onc(C)c2C)=O)CCC(C)CN1C(=O)Cc1ccn(C)n1 c1(CC=O)nc2ccc(N(C)C)nc2[nH]1.C1(C(N(CC)CC)=O)CC2CC1C2 c1(CC(N2CCC(O)C2)=O)ccc(Cl)nc1C.C1(C=O)(COC)CC1(F)F.N C1(C(=O)NC2(CC3CCC3)CC2)CCCN1C(c1ncc[nH]1)=O C1(C(=O)NC2C(C)(CNC(Cc3n(C)ccn3)=O)CCC2)CCC(C#N)CC1 c1(C(=O)NC2(CCOC)CCN(C(=O)C=NOC)CC2)cc(C)c(OC)c(C)c1 c1(CC(=O)N(CCCN(C)C(c2cnc(S)nc2)=O)C)c(Cl)ccc(O)c1Cl c1(CC(=O)NC2CCCN(C(c3ncncc3F)=O)C2)ccccc1Cl N1(C(c2nc(C(C)C)oc2)=O)CCN(C(=O)C(C)NS(C)(=O)=O)CC1 C1(CCCC)CN(C(C23COCC(C2)C3)=O)CCN1C(c1cc(CO)oc1C)=O N1(C(C=NOC)=O)CC2CCC(N(C)C(c3cc[nH]n3)=O)C2C1 CCCC(CCCNC(C)=O)NC(=O)C(c1cc(F)ccc1OC)(F)F C(CO)(C(C)NC(c1oncc1C)=O)NC(C(C)NC(=O)NC)=O c1cccc(C#N)c1.n1(CC)ncc(C(=O)NCC2CC2)c1Cl.C(=O)(C)N c1(C(=O)NCC(CC)NC(C2CC(C(F)F)C2)=O)cc(C)c(N)cc1Cl C=C(Cl)CC(C(=O)NC1CCC(C)(C)C1)NC(=O)CCCCNC(C)=O CCC(CC#N)N=c1nc(N(C)Cc2ncc(Br)cn2)c2c([nH]1)CSC2 C1(NC(CCCCOC)=O)CCN(C(=O)CCC2CCOC2)CC1(C)C Cc1cc(C)c(C(N2CC(NC(c3cnn(C(C)C)c3Cl)=O)CC2C)=O)s1 C(=O)CCCCCc1cccs1.C1(C(=O)NC(C2(C)CC2)C)CC2CCC1O2.N C(=O)(C1=NN(C)C(=O)CC1)N1CC(CN(C(=O)CC2(O)CCOC2)C)OCC1 c1(CC)nc2ccccn2c1C(=O)NCCCc1ccc(N)cc1 N1(C(c2c(NC)cccc2)=O)CCC(NC(c2ncc(F)cc2F)=O)CC1C Nc1cnc(C(=O)N(C2CCN(C(c3cc(C4CC4)[nH]n3)=O)CC2)CCO)cn1 c1(CC)cc(NC(=O)CC(C)(C)N(C)C(C2(F)CC2)=O)cc(F)c1 CC1CC(C(=O)NC2CCC(CNC(=O)C(C)(C)c3cccnc3)C2)CCS1 c1ccc2c(CN=C(NCC3CCCO3)NCC3COCCOC3)coc2c1 C1(CNC(c2ccc(SC)s2)=O)CC2(CCN(C(=O)C(C)(O)CC)CC2)C1 N1(C(C(C(C)O)NC(C)=O)=O)CC2(C1)CN(C(=O)CC(C)CN(C)C)CCO2 C1(C(N(C)CC2CCCCC2)=O)COC2(C1)CN(C(=O)C(C)(C)c1ccno1)C2 C1(C(=O)NC(CC)C(=O)OC)CCN(C(C2CN3CCC2C3)=O)C(CC)C1 N1(C(CCC(C)OC)=O)CC(C)C(C)(C(=O)NCC2CCC3(CC3)CO2)C1 CC1=NOC(C)(C(=O)NCC(C)(F)CNC(C2CSCCS2)=O)C1 n1(CC(=O)NCCCCCC)c(C)c(C)sc1=O.c1(C=O)[nH]ccc1C1CC1.N C1(CCC)CN(C(c2csc(C(C)=O)n2)=O)CCN1C(=O)COC(C)=O c1(C(=O)N)cc2c(C#N)cccc2[nH]1.N1(C(C2N(CC)CC2)=O)CCC(C)(C)C1 CCCC(CCCNC(c1cc(C(C)(C)C)on1)=O)NC(c1cc(C)cs1)=O C1(C(=O)NC2C3CN(C(CCC(C)(C)OC)=O)CC32)Cc2cccnc2C1 N1(C(C(CC)SC)=O)CCC2C(NC(c3ccn(C(F)F)n3)=O)C12 O=S(=O)(c1cnc(NC2CCOCC23CCCC3)c(Cl)c1)NCC(F)CO c1(CNC(C2(OC)CCOC2)=O)nc(C)c(C=O)o1.CC(C)(O)C(C)C.N CN1C(=O)CC(C(=O)NCCC2(NC(c3cc(Cl)c[nH]3)=O)CC2)NC1=O CC1(C)CN(C(=O)C=Cc2cn[nH]c2)CCC1NC(=O)C1=COCCC1 C(=O)(C(CC)(CC)CC)NC1C(NC(C(C)=C(CC)C)=O)COCC1 CCCCN=c1[nH]c(=NC2CCCC(CC)C2)[nH]c2cccnc12 C1(NC(c2c(CC)ocn2)=O)CN(C(=O)C(C)Sc2nncn2C)CC12CC2 c1(NC(C(CC)N2CCC(CC(=O)N)C2)=O)ccc(C(=O)OC)cc1.C1(C)CC1 c1(CC)ccc(C)nc1C(N1CCCC1C)=O.c1(C(=O)N)nc[nH]c1C(F)(F)F C1(CN(C(c2c(C)nn[nH]2)=O)C)CC(F)CN1C(C1CC1(F)F)=O C(c1ccc(Cl)c(Cl)c1)=CC(=O)NCC1C(C)CN(C(=O)CNC=O)CC1 c1(C(c2n(CCCOC)nnn2)NCC=CCl)cnc2ncccn12 C12(C=O)CCCCN1CCC2.C(CC(=O)NC)SCC(C)C.C1CC1.CC(F)F C(=O)(C(O)CCNC(=O)C(F)(F)CO)NC(c1n(CC)ccn1)C CC(C)(C)CCCCCC(=O)N1CCOCC1CNC(C1CC2CCC2C1)=O C1(C(=O)NC2(C)CCNCC2)CC2(CCCCO2)C1 c1(N)cncc(Cl)n1.N12CCCC(C1)C2=O.C1(COCC=O)CCC1.C1CC1 c1(NC(C2CN(C(C(C)NC(C)=O)=O)CC(F)C2)=O)cccc2c1C(=O)NC2 C1(C(=O)NC2C=CCN(C(c3cc(F)c(F)cc3F)=O)C2)CN2CCCN1CC2 c1(C(=O)NCC2C(C)CCN2C(=O)C=Cc2ccoc2)cccc2c1OCCN2 Cc1ccncc1OC1CN(C(=O)C(=O)CCc2ccccc2)C1 c1(N(CCCC)C)nc(N2CCC(Cc3ccncc3)C2)c2ccsc2n1 CCC(C)(C)C(C(=O)NCC1CC(NC(c2ccc(N)c(Cl)c2)=O)C1)OC C1(NC(Cc2cc(CC)no2)=O)CC(C)CN(C(c2c[nH]ccc2=N)=O)C1 CC1CCC(CCC(=O)NCC(C)(C)CC2CN(C(c3cc(Cl)c[nH]3)=O)C2)O1 CC1CC=C(c2cc(C(=O)NCCc3cccc(O)c3)ccn2)CC1 C1(CNC(C(COC)O)=O)CCCCC1NC(c1cc(C(F)(F)F)n[nH]1)=O c1(OCCC)cc(OC)ccc1NC(c1c(C)cnn1CCN)=O c1(C(=O)NC2CCC(Cc3nc(C)on3)C2)cccc(C(C)(C)C)c1 c1(C(N2C(C(=O)OC)CCC2)=O)ccnc(CNC(=O)CC)c1.C(C)C.O C1(NC(C(C)SCc2ccccn2)=O)CCCC(NC(c2cccs2)=O)C1 c1(CNC(=O)NC(C2CCOC2)CC)cnc(O)s1 Cc1cccc(C2=CCN(C(c3csc(Br)n3)C(=O)NC3CCCC3)CC2)c1C Cc1cccc(C2CCN(c3nnc(C(C4CCCSC4)(C)O)n3CC(C)C)C2)c1 c1(OCC)cccc2[nH]c(C(N3CC(C)CN(C(=O)C4=CCC4)C(C)C3)=O)cc12 N(C1CCC(NC(C2(C)CC=CC2)=O)c2ccccc21)C(C1(C)CC(C#N)C1)=O c1(C(N2CCC(NC(c3ccoc3)=O)C(F)C2)=O)cc2scc(Cl)c2[nH]1 C(=O)C(C)CC(N)=O.c1(C(=O)NCCC(C)C)ccc(C=O)cc1.C1CC1.N C12(CNC(CC(C)C)=O)CC1CN(C(c1ccc(-c3ccsc3Cl)s1)=O)C2 C12(C(=O)NC3CCC(C)(C)C3)CCCC1CN(C(C1CC(F)(CF)C1)=O)C2 Cc1nc(C2CC2)ccc1C(=O)N(C1CCN(C(C2C3(CC3)C23CC3)=O)C1)C N1(C(C2C(C)CC2)=O)CCCC(C(=O)OC(C)(C)C)C1 c1(C(N2C(CC)(CC)CC(NC(c3cscn3)=O)C2)=O)cccn2nnnc12 CC(C)(CNC(c1n[nH]cc1[N+](=O)[O-])=O)CC(=O)NC1COCCOC1 C1(NC(CCCCCC#C)=O)CCN(C(=O)CN2CSCC2=O)C12CCCC2 N1(C(CCCCC=C)=O)CC(NC(C2CC2C2CC2)=O)C(C2CC2)C1 CN1CC(NC(=O)C(O)C2CN(C(=O)CC3CCSC3)C2)C(F)(F)C1 C1(C(N2CCC(C3OCCC(OC)C3)CC2)=O)CC2CC(=O)C1O2 C(c1ccc(C=O)cc1)=CC(=O)NC(CCNC(CCCCOCC)=O)C.O c1(C(=O)NC(C(C)NC(c2c(CCC)[nH]cc2)=O)C)sccc1S(N)(=O)=O N1(C(c2nc(C#C)sc2)=O)CC(NC(c2c(C)noc2C)=O)C(C2CC2)C1 C1(O)(C(C)NC(=O)CC(=O)N(C)C)CCN(C(=O)CCC(=O)C2CC2)C1 n1(CCCC(=O)OCC2CCC(F)(F)C(=O)N2)c(O)nc2ccccc12 Cc1cc(O)ccc1CN1CC(C(C)NC(=O)CNC(=O)C(C)(C)C)C1 O(S(=O)(=O)c1ccc(C2(C)OCCO2)cc1)c1c(C(C(C)C)O)cccc1 C(CC1CCC1)(C(=O)NC1CC(N(C(=O)CC2CCC(=O)N2)C)C1)OC c1(CC(=O)NCCN(C(C2C(C)CC(=O)NC2)=O)C)cc2ccccc2oc1=O O=C1COC(CNC(C2CC(C)(NC(c3ccnnc3O)=O)C2)=O)CN1 C1(C(=O)NC(C)(C)CC(=O)NCC(=O)OCC2CC2)CC2(CCO1)CC2 C1(OC)(CNC(=O)CN(C(=O)CC=C(Cl)Cl)C)CCC(C)C1.C1CC1 CCCCC(C(=O)N1CCCC(C(N)=O)C1)NC(C1CCOC1C1CC1)=O N1(C(C2(CC)CC2)=O)CCCC2(CCO2)C1.C12CCCC1C(=O)N2 C1(NC(Cn2c(C)ncc2)=O)CCCC(NC(=O)C2=CCCS2)CC1 Cc1ccc(C(N2CC(C(C)NC(c3n[nH]cc3C)=O)C2)=O)nc1 c1(NC(C2(C)COC2)=O)ccc(F)c(F)c1 c1(NC(c2n(CC=C)nnn2)CCC2(C)CC2)cc(C(=O)OC)cnc1OC C=C(Br)CCC(=O)NC1(C)CCN(C(=O)C(C)(Cl)Cl)C1 O=S1(=O)CC(CNc2nnnn2CCSc2ccccc2)C(O)C1 C(=O)(C(CC)C(C)(C)CC)NCC(CC=C)NC(=O)C(CC)=CCCC c1(C(N(C(CC(F)F)C(=O)N)C)=O)cc(O)ccc1F.C1(C(C)(C)O)CC1.C N1(C(CN2CCCC(CC)C2)=O)CCN(C(=O)Cc2cc(C)on2)C(C(C)C)C1 C1(CC#C)(C(=O)NCCCCN(C)C)CCN(C(=O)CC2(O)CCCCC2)C1 c1(CC)sc(C(=O)NC2CCC(N(C(=O)C(C)N(C)C(C)=O)C)CC2)cc1C C1(C(Cn2cc(-c3cc(CC)no3)nn2)F)CCN(C(c2occc2Br)=O)CC1 C1(CCOC)CN(C(c2nnc(C)s2)=O)CCN1C(c1c[nH]c(Br)c1)=O c1(C(N(CCCNC(C2(C)CC=CC2)=O)C)=O)cn(C)cc(Br)c1=O CCCC(C)(C)CC(=O)NCCCC(CO)NC(c1cc(F)c(F)c(F)c1)=O C12(NC(c3cc(CC)ncn3)=O)CCN(C(c3cnc(CC)s3)=O)CC1C2 C12(NC(CC3N(C(c4cc(COC)no4)=O)CCOC3)=O)CCC(C1)OC2C c1(C(N2CC(OC)C(NC(c3ccc(F)c(F)c3)=O)C2)=O)cc(Cl)cc(C)c1C C1(NC(C(C(C)C)C#N)=O)CN(C(=O)CCN2CCCC2)C2(CCC2)C1 C=CC1(CC(N2CC(O)(C(N)=O)C2)=O)CN(C(=O)C=Cc2cnccn2)C1 C1(C(N2CC(CCC)C2)=O)(OC)CS(=O)(=O)C1.c1(C(=O)N)nc(C)oc1C C(C(C(=O)NOC(COC)COC)C(C)(C)C)NC(C=CC)=O N1(C(c2ccc(CC)nc2C)=O)CCN2CCN(C(=O)CC3CN(C)C3)CC2C1 c1(C(=O)NCC2N(C(c3c(C(C)C)nn(C)c3)=O)CC2)cc2sccc2s1 N1(C(=O)OC(C)(C)C)CCC2CC(NC3COC4OCCC34)CCC2C1 N1(C(C=C(C)Cl)=O)CCN(C(=O)CCN2CCN(C(C)C)CC2)C(C(C)C)C1 C#Cc1cc(C(=O)N(C(C)CNC(C2CCC=CCC2)=O)CC)cc(N)c1 S(=O)(=O)(c1cnc2ccc(Cl)cc2c1)NC1CCCC(N)C1 C1(CNC(C(N)=O)=O)CCCC1NC(=O)CC1CCC(=O)O1 CCC(C)CCCC(=O)NC1(C(N2CCCCC2CC)=O)CCN(C)C1 Cc1cc(C(=O)NCC(O)CN(C(=O)CC2CC23CC3)C)c(O)cc1F C(=O)(C=CS(C)(=O)=O)N1CC(C(C)NC(=O)C=CC2CCOCC2)OCC1 c1(C(N2C3CC(C3)C2)=O)cnn2c1OCCC2.CC(C=O)NC(C1CCC1)=O.N CC1(NC(=O)CCc2cnccn2)CN(C(C2CCCCS2)=O)C1 C1(NC(C2CN(C(C(OCC)OC)=O)C2)=O)CCNC1=O C(=O)(C1=C2CCN=C2NC=C1)N1CC2CC(CC(NC(C(CC#C)C)=O)C2)C1 N1(CC(C)NC(=O)Cc2cnoc2)CCN(C(c2ncc(Br)cn2)=O)CC1 C#CC1(C(=O)NC(CNC(c2cn[nH]c2)=O)CC)CCC1 N1(C(c2c(C)sc(O)n2)=O)C2CCC1CC(C)C2.C1(CC=O)CCC(F)(F)C1.N N(C(=NCCCC1(C)N=N1)NCc1cc(C)n(C)n1)C1C(C)C1.c1ccccc1 N1(C(c2ncccn2)=O)CCC2CCN(C(c3cc(C(F)(F)F)ccn3)=O)C2C1 C1(C(N2C(CCC)CSC2)=O)CCC2(COC)CC12 N1(C(C(C(CC)C)N(C)C)=O)CC(CO)C2(C1)CN(C(C1CCCC(=O)N1)=O)C2 c1(C(N(CC(C)NC(=O)C)CC)=O)ccccc1F.c1(C(=O)N)cccs1 c1ccc(O)cc1C.c1(C(c2cc(C)no2)NCC(=O)N)ccccc1C(F)(F)F c1(C(C(=O)NC(CC)(C)C)N(CC(CSC)OC)C)csc2ccccc2c1=O N1(C(C(C2N(C(c3cnc(CC)s3)=O)CCC2)(C)C)=O)CCC2(CCO2)C1 CC(C)CC(CCO)NC(c1cc(CNC(=O)CC(C)F)on1)=O c1(C(=O)NCCCC=C)ccc(CC)c(N)c1.C1(C)(C=O)CS(=O)(=O)C1.N N1(C(CCn2c(C)csc2=O)=O)C2CCC1C(C)C2.C(=O)(C(C)SC(F)(F)F)N C1(C(=O)NC2C(C)CC=CC2)CC2CC1CN(C(C1(C)CCC1)=O)C2 N1(C(C2(C)CC2)=O)CCN(C(c2cc(N)ccc2Cl)=O)C(CCO)C1 C1(CC(=O)N)CCCCC1.C(CCCC)N(C(=O)CNC=O)C.C(=O)C1CC1 C1(C(=O)NCC2C(NC(CCC=CCC=C)=O)CCC2)CC(C(C)C)=NO1 C(C(C(=O)NC(c1cccnc1)CO)NC(C1OCCC1C)=O)OC c1(C(C)O)cnc(CNC2(C(=O)O)CC2C)s1 c1(CNC(C(C)NC(CCCOCCC)C)=O)ccc(CSC)cc1 C1(NC(=O)NC2(c3cccc(C(F)(F)F)c3)CCC2)CCC2(CCOCC2)CC1 N1(C(c2c(C(C)C)cccc2)=O)CCCC2(CCCN2C(=O)C=CCBr)CC1 C12(NC(C(=O)NCC)=O)CC(C1)OC21CN(C(=O)C(C)(C#N)CC)C1.C N1(CCC=O)C(=O)CCC1=O.C1(O)(CC)CCN(C(=O)CN2CC3CC3C2)C1.N c1(C(=O)NC(CCNC(CC2CC(=C)C2)=O)C)cccc2nncn12 c1(OC)cnc(F)cc1C(=O)NC1CN(C(=O)CC2(O)CCCC2)CCC1C c1(N2CCC(CC)(NC(C=CC=CCC)=O)C2)nc(C(C)C)cc(C)n1.O C=C(C)c1cccc(NC(=O)CC(C)C(C)(C)NC(=O)CC(=O)N)c1.C1CC1 c1(C(=O)NCCCOC(=O)NC)nc2ncc(Br)cn2n1 C1(NC(CCC2CCN(C(CN(C(C)=O)C)=O)C2)=O)CC(=O)NC1=O N(C(=NCCc1cccc(F)c1)NCc1ccoc1)C1C(C)(C(F)F)C1 C(=O)(C(CCN(C)C)NC(=O)CCc1cccnc1)NC(c1ncccn1)CC C(=O)(CCC(C)c1ccccc1)NC(C)CCNC(C1CC1C)=O Cc1c(-n2nnnc2SC(C)CCS(C)(=O)=O)cccc1Cl C1(CNC(CC2CCN(C)C2)=O)CCC(F)(CNC(c2ccncc2)=O)CC1 C(=O)(C#CC1(C)CCCO1)N1CCCC(O)(CNC(c2cc(C)c(F)cc2)=O)C1 C1(CC=C)(NC(=O)C(c2ccnn2C)C)CCN(C(=O)Cc2cccc(C)c2)C1 c1(CCCC)nc(C2CC(=O)N(c3ccc(Br)cc3)C2)n(-c2ccnnc2)n1 c1(-c2cc(C)cc(F)c2)c[nH]c2ncc(C(=O)Nc3nc(Cl)cnc3Cl)cc12 N1(C(c2c(SC)nccn2)=O)CCC2(CCCN2C(C2(C)CCN(C)C2=O)=O)C1 N1(C(CC(C=C)CC)=O)CCN(C(c2ccc(=N)[nH]c2Cl)=O)C2(CC2)C1 C1(NC(=O)COC2CC(F)(F)C2)CN(C(c2cnsn2)=O)CC2(CC2)C1 CC1=CC(C)=NS(=O)(=O)N1CC=O.C1(O)CN(C(=O)CC2(O)CC2)C1.C C(=O)(CS(N)(=O)=O)NC1(CC=C)CN(C(=O)CCCc2ccc(Br)s2)C1 C1(OC)CCN(C(C2(C#N)CC(C)C2)=O)CC1.C(=O)C(F)(F)CC1CC1.C c1(C(=O)NCC(CNC(C(CN(C)C)O)=O)O)cc2c(F)ccc(F)c2[nH]1 C(=O)(CCCCC1CC1)N1CC(N(C(CC)=O)C)C1 CC1(C(=O)NCCNC(c2snc3ccccc23)=O)CCCCCCC1 C1(C(=O)NC2(c3cccs3)CC2)(NC(c2cc(Cl)ns2)=O)CC(F)(F)C1 C1(C#N)(C(N(CC(CN(C(=O)Cc2cnn(C)c2)C)O)C)=O)CCCO1 C1(C(N2C(CNC(c3cn(C(F)F)cn3)=O)CC2)=O)CN2CCCC2CO1 CCCC(CCC)C(=O)N1CC2CC2(CNC(c2cc(Cl)ncc2O)=O)C1 Cc1ccc(Cl)c(C(N2CC3CC(NC(c4cc(C)n(C)c4)=O)C2C3)=O)c1N CCC(C)(C)C(O)C(=O)N1CC(O)(C(C)NC(c2cccnc2N(C)C)=O)C1 c1(C(=O)OC(C)(C)C)ccc(C(N2CCOCC2C(F)F)=O)cc1F Cc1ccc(C(=O)NC2CCCN(C(C3CCC4(CC4)C3)=O)C2)nc1C C(=O)(C(C)CC(C)(C)C)NCCN(CCC)C(c1cccc(F)c1OC)=O c1(C(C)NC(C2CCCC(c3ccccc3)O2)=O)csc2ccccc12 C1(CC)(NC(c2nc(CN)ncc2Cl)=O)CCCN(C(=O)C(C)=C2CC2)C1 C1(NC(CC(COC)COC)=O)CC2CCC(C1)N2C(=O)CCC(C)OC c1(C(=O)NCC(CC)NC(=O)CCC2CCCOC2)ccccc1C(F)F C1(C=O)C2(CC2)C12CC2.C1(CC(=O)N)CCCC1.O=CC.C1(CC)CC1 c1(C(C)NC(N(CCOC)C)=O)ccc(-c2cccc(OC)c2)cc1 C1(NC(C=CSC)=O)CC(C)CC1O.c1(C(=O)N)cc(C=O)n[nH]1.C(C)(C)C c1(C(N2CC(CCC)C2)=O)cc(C(N)=O)cs1.C(=O)(C(C)(C)N1CCCC1)N C1(CC)(NC(=O)C=CC2CCCCCC2)CCCN(C(=O)CN2CCCCC2)C1 c1(C(=O)NCC(CNC(C(C(C)C)C)=O)O)c[nH]c2nccc(Br)c12 N1(C(Cc2ncc(C)o2)=O)CCC(C)C(CNC(c2ocnc2C)=O)C1 c1(C(N(C(C)C)CCNC(=O)C(C)C(C)O)=O)cc(OC(F)F)ccc1F N1(CC2C(CC)CCC2)CCN(CC(=O)Nc2cnn(C)c2)CC1 c1(C(=O)NCCCN(C(C2(C)CC2(F)Cl)=O)CC)cnc(N(C)C)nc1 C1(NC(c2c(CC)cccc2)=O)CCN(C(=O)Cc2c[nH]nc2O)CC1F Cc1cnc(NCC2CCOCC2(C)C)c(S(=O)(=O)NC(c2csnn2)C)c1 C(CN=[N+]=[N-])(C(=O)NC(C)CC=O)NC(C1(C(CC)=O)CC1)=O.C(C)C.N n1(CCCCC)nc(-c2ccc(OCCOC)cc2)nc1C1COC(=O)C1 N1(C(C2N(C)C(=O)OC2)=O)CC2(CCCC(CNC(C3CCOC3)=O)O2)C1 C(=O)(C1CCCc2nc(C)[nH]c21)NC1CCC(F)(CNC(C(OC)OC)=O)C1 c1(C(=O)NC(CN(C(c2cc(C)sn2)=O)C)C)cccc(Cl)c1 C(=O)(C1=NOC(C)C1C)NC(C(C)C)(C)CNC(c1cnc(C(F)F)s1)=O C1(C(=O)NCC(C)(C)C)(OC)CCOCC1.c1(C=O)cc(CC(C)C)nn1C.N Cc1nc(Cl)nc(N2CCCC(CNC(C3CCCC4CC34)=O)CC2)c1F C1(OC(C)(C)C)CC(NC(=O)NCC(Cl)C(F)(F)F)C12CCC2 Cc1cc(Cl)ncc1CC(=O)NC1CC(C)C1.C1(CC(=O)N)CN2CCN1CC2 C1(C=O)C2CCC1CN(C(c1cc(C)oc1C(F)(F)F)=O)C2.C(=O)(CC)NC C=CCCCCC(=O)N1CCC1CC(=O)N(C)CC1(C#N)CC1 c1(OC)cscc1C(=O)NC1CC1NC(C1CC1C(=O)OC)=O C1(C(N(CCF)CC)=O)CC2C=CC1N(C(=O)CC1CCC=CCC1)C2 CCCCCCNC(c1ncoc1C(C)(C)C)=O.C1(C=O)(C(F)F)CCCC1.N C(=O)(C(C)S(C)(=O)=O)NCCN(C1CCCCC1)C(C=C(C)Cl)=O C1(C(N(CC(C)(CO)CO)C)=O)CN2CCC1CC2 c1(CCC)cc(O)cc(O)c1C(=O)N=c1ccn(-c2nccs2)[nH]1 N1(C(Cc2ccc(C)s2)=O)CCC(C2CCN(C(=O)C3=CSCCO3)C2)CC1 Cc1nc(-c2ccc(-c3c(C)n[nH]c3C)s2)n(CCS(N)(=O)=O)n1 c1(C(N(CC(CNC(c2c(CC)nc[nH]2)=O)O)C)=O)cccc2nc(CO)[nH]c12 c1(NC(C2CN(Cc3cc(Cl)ccc3C(F)(F)F)CCS2)=O)nc(Br)ccc1Cl C1(CN(C)C(c2c[nH]nc2C2CCC2)=O)CCCN(C(c2nn(C)cc2Cl)=O)C1 c1(C(=O)NCCNC(c2cncc(C(C)C)c2)=O)cnc2nccnc2c1 c1(CC(=O)NC2CC(CCC(=O)NC(CO)CCF)C2)ccnc(O)c1 N1(C(C2N(C)CSC2)=O)CCOCC(CNC(=O)CCCn2ccnc2)C1 c1(C(C(=O)NCC2CCCO2)N(CCN(C)C)C2CC2)cccc(Br)c1 C(=O)(C(O)C(F)F)NCCC1CCC(NC(C2CC(F)(F)C2)=O)C1 CCCC(CC)CC(=O)N1CCCC(NC(C23CCC(C(F)F)(CC2)C3)=O)CC1 C1(CCC)CC(C(=O)NC2C3CC2N(C(c2coc(C(F)F)c2)=O)C3)CCO1 Cc1cc(C)c(CNC(C2CCC(CNC(c3c(C)noc3C)=O)O2)=O)s1 C1(C(N(CCCC(=O)OC)C)=O)CC(C)CN(C(C2CCCC(OC)C2)=O)C1 c1(C(N(C2CCCC2)C)=O)cc2nc(C)cc(C)n2n1.C(C=O)N(CC)CC.N c1(C(=O)NC2CCC(C)N(c3ccc(C#N)cn3)C2)cnn2c1C(=O)NCC2 C1(CCCNC(C2CC(OC)C2)=O)CCN(C(C2CC2)=O)CC1.N(C)(C)C C1(CN(C)C)CCCCC1NC(=O)NCc1ccccc1-n1cccn1 C1(C(=O)NC2CCN(C(c3cc(OCC)no3)=O)C2C)CCOC2(CCC2)C1 N1(C(C(C)(C)CCF)=O)CC2(NC(=O)CN3C(=O)CCCC3=O)CCCC2(F)C1 c1(CC)[nH]nc(C(=O)NC)c1C.C1C2CC1N(C(C1(C(N)=O)CCC1)=O)C2 CC1(CNC(=O)CCC(=O)c2ccc[nH]2)CCN(C(=O)CS)C1.CC(F)(F)F N1(C(CC2(OC)CCCC2)=O)CCN(C(=O)CCCC(C)=O)CC1CC(F)F C1(C(=O)NCCCC(C)(C)NC(=O)C2=CCCCO2)CCC2CCC(=O)N12 Cc1ccc2c(C(N3CCCCC(NC(=O)CCS(C)=O)C3)=O)onc2c1 N(C(=NCCC1COc2ccccc2O1)N1CCN(Cc2ccon2)CC1)C(C)C c1(C=O)cc(C)c(C)cc1Cl.c1(OCC)cc(C(=O)NCCC2CC2)[nH]n1 Cc1n[nH]c(C)c1S(=O)(=O)N1CCC2CN(c3ncnc4sc(Br)cc34)CCC12 C1(O)(CN(C(C(C)N(C)C)=O)C)CCN(C(C23CC(C#N)(C2)C3)=O)CC1 N1(C(CN(C(C)=O)C)=O)CC(NC(=O)CC2CCC(C)(C)C2)CC12CCOCC2 N1(CC)CCCCC1C(=O)NCCCNC(C1CC1C(C)O)=O Cn1cc(C(F)(F)C(=O)NCCN(C(=O)CC2CCCCO2)C2CC2)cn1 C1(NC(CC(C)NC(C2(C)CCC(=O)N2)=O)=O)C2CCCOC12 S(=O)(=O)(c1ccc(NCc2ncoc2C(F)F)c(Cl)c1)NCC(CCCCC)O c1(C(=O)NC2CN(C(C=C(C)C3CC3)=O)CC2F)nccc(C)c1F C1(N(C(CSCC(=O)OC)=O)CCO)CCN(C(c2cnnn2C)=O)C1 N1(C(C(COC)(F)F)=O)C2CCC1C(CNC(=O)CC1CCCCO1)C2 c1(-n2cc(CNC3C(N)COC3)nn2)ccc(S(=O)(=O)C(F)(F)F)cc1 c1(C(N(C2CN(C(C(CC(C)C)OC)=O)C2)C)=O)cc(C)cc2c1OCC2 N1(C(CCC(C)(C)F)=O)CC2CCC1CN2C(C1CC(C)(C)C1C(F)(F)F)=O Cc1cccc(NC(=O)C(C)OC(=O)C(c2ccc(-c3nn[nH]n3)cc2)C)n1 C1(C(=O)NC2CC3(C2)CN(C(c2cn[nH]c2)=O)C3)CC12CCC1(CC2)OCCO1 C1(C=O)CCN(C2CC2)CC1.CCC(C)CNC(=O)C=CCN1CCCCC1 Cc1ccc(C(=O)NCC2CC(C)CCN2C(C2CC3CCC3C2)=O)c(F)c1F S(=O)(=O)(c1cccc(OC(F)F)c1)Nc1c(CN2C(C)(C)CCC2)ccc(Cl)n1 C12(C(N(CC=C)CCOC)=O)CCCC1CCN2C(=O)CCc1ccncc1 Cc1ccc(OCCNC(C2CC2c2ccco2)=O)c(F)c1 N1(C(c2c(Br)ccc(C)n2)=O)CC2CCOCC2(NC(=O)CO)C1 c1(C(N2CCC(NC(c3cc(C)on3)=O)CC2C)=O)coc2cc(O)ccc12 C(=O)(CC(C(C)CC)NC(c1nnc(S)n1C)=O)NC(C#C)C1CCC1 C(=O)(C(O)C(C)(C)C)N1CCC(N(C(c2cc(C)sc2Br)=O)CC)C1 Cn1[nH]c(=Nc2ccc3c(c2)OCO3)cc1C1(O)CCC1 n1(CCC)nccc1C(=O)NCCNC(=O)COC1CCCOC1 C(C(C)(C)C(=O)NCCNC(=O)C=CS)SC.c1ccco1.C1CCCC1.C Cc1cc(N)c(F)c(C=O)c1F.CC(C1CC1)N(C)C(C1CC1)=O.C(N)=O C12CCCC(C1)C(=O)N2.n1(CC2C=CCC2)ccnc1CCCC1(CO)CC1 C1(NC(CCn2cc(C3CCC(C(N)=O)CC3)nn2)=O)CCC2COC1O2 CC1(C(N2CCC(CNC(c3n[nH]cc3C3CC3)=O)CC2)=O)CCNC(=O)C1 CC1(C)C(CNC(=O)C(O)CF)CCN1C(c1cnc2sccn12)=O c1(CNC(CN(C(=O)C(C)C2CCCC2)CC)=O)ccon1 C(=O)(C(C)C(F)(F)C(F)F)NC(CN(C(=O)C(=C1CCCCC1)F)CC)C Cn1cc(C=CCO)cn1.C12CCC(C1)n1cc(nn1)CCCNC2=O Cc1[nH]c2ccccc2c1C(N1CCC(C(C)(C)C)(C)C1)=O.C(=O)C(C)(C)F.N c1(CC)ccc(C(=O)NC(C)CC2CCN(C(=O)C(O)C(C)CC)CC2)c(C)n1 C1(NC(c2csc(Cl)n2)=O)CCC12CCN(C(=O)CCc1ncco1)CC2 C(C(C)(C)CS(C)(=O)=O)NC(c1nnnn1CCC1(C)CC1)C(C)C1CC1 C12(NC(CN(c3ccccc3)C)=O)CCCN(C(=O)CC3(CO)CC3)CC1C2 C1(C(=O)NC2(C(=O)OCC)CCC2)CN(C(C2CCCSC2)=O)CC12CCC2 c1(C(=O)NC(c2c(C)cccc2)C(=O)O)ccc2ncn(C)c(=O)c2c1 N1(C(CN(C)CCc2ccccc2)=O)CCCC2(NC(=O)C3=C(Cl)CC3)CC2C1 c1(CCCNC(C2CCC(NC(C3C4COCC34)=O)C2)=O)cccnc1 c1(CN2CCC(N(C(CC(=O)NC)C)C)C2)ccc2c(c1)OCCCO2 C1(N(C)C(C2(CCNC(=O)CC3CNC(=O)O3)CC2)=O)CCCCC1(C)C C(=O)C1=C(C)CC(C)(C)CC1.N1(C(COCC)=O)CC(C(F)(F)F)OCC1.C CCC(C)C(C#N)c1nc(C(=O)NCCSSC)cs1.C(=O)COC N1(C(CN(CCC#C)C)=O)CCC(N(C)C(c2cn(CCOC)cn2)=O)C1 c1(CNC(c2n(CCOC)nnn2)C2CC2)cc(F)ccc1OC(F)F C1(CC(=O)N(C2CN(C(=O)C(C)(C)c3cnco3)C2)C)CC(O)C1(C)C Cc1cnc(CNC(=O)CONC(C2CCCC2F)=O)[nH]1 C12(C(=O)NCCCCCC#C)C(NC(=O)CC3CCCC(=O)N3)C3CC1C2C3 c1(C(=O)N)n[nH]c2cc(C)ccc12.c1(SC)ccc(C(=O)NC2CC(C)C2)o1 N1(C(C(C)(F)F)=O)CCN2CCN(C(c3ccnc4c3CCO4)=O)CC2C1 Cc1ccc(O)c(C)n1.c1(CC(N2CC(C)(CC(=O)N)C2)=O)ccc(F)cn1 C1(CNC(CCCCC=C)=O)CC2CCC(C1)N2C(c1cccc2oncc12)=O Cc1ccncc1-n1cc(CN(C)C(C2CCC2(F)F)=O)nn1 c1(C(=O)NC(C(=O)NC(CCC=C)CO)CCC)cc(C)c(C)cn1 c1(C(CNC(c2cc(-c3cccc(C#C)c3)[nH]n2)=O)O)cccc([N+](=O)[O-])c1 N1(C(C2(C)C(CC)CCC2)=O)CCC(C2CC(NC(c3cc(C)cs3)=O)C2)CC1 CCCC(C)C(=O)N1CC(NC(=O)COCC2(F)CC2)C(O)C1 c1c(C)cccc1C.Cc1ccnc(C(=O)NCC(C2CC2)N(C(=O)C)C)n1.O N1(C(Cc2c(C)occ2)=O)CC2CN(C(=O)C(C)Oc3ccc(F)cc3)CC2C1 Cc1c(NC(C2CC(F)CN2C(=O)CCc2cccnc2)=O)cccc1CO CCC(CCCC(=O)NC(CO)CCO)NC(=O)CN1CCCC1 N1(C(c2ncn(C)c(=O)c2)=O)CCC2C(C1)CN2C(C1C(Cl)(Cl)C12CC2)=O N1(C(C(C)OCCOC)=O)CCOCC(C)(CNC(c2ccnn2C)=O)C1 C(=O)(CC(O)CC(C)C)NC(CC)CN(C)C(c1coc(C(C)C)n1)=O Cc1ccccc1OCCN(C(c1ccc(Br)nc1)C(=O)NCc1ccco1)C c1(OC)cccc(C(=O)N(CCC(C)NC(=O)CN2CCC(C)C2)C)c1[N+](=O)[O-] C1(N(C(C=C(C)Cl)=O)C)CCN(C(=O)Cn2cnc(C(N)=O)n2)CC1C C(=O)(C1=NOC(C)C1)NC(C(C)C)CCNC(=O)Cn1nnc(C2CC2)n1 c1(C=O)cnc([N+](=O)[O-])n1C.C=CC(C(=O)NCC1CC(F)(C)C1)OC.N c1(CC=O)cc(F)ccc1C.c1(CC)nocc1C(=O)NCCCOCC.N C1(C(=O)NC2C(OCC)CCC2)CNC(=O)CN1C(C1CC(C)(O)C1)=O c1(NC(CC)CCCO)cc(NCC(c2nncn2C)C)nc(C)n1 C(=O)(C(Cc1ccccc1)CC(C)C)N(C(C)COC)CC=C c1(C=O)ccc(O)c([N+](=O)[O-])c1.N1(C(C(C2CCC2)OC)=O)CC(O)CC1C c1(C=O)cc(Cl)cc(Cl)c1O.C1(CNC(C=CCCC=C(C)C)=O)CCCC1 N1(C(C2(CC=C)CC2)=O)CCC2CC2(NC(C2CC=CC2)=O)CC1 C(=O)(C(CNC(=O)CCN(C)C)C(C)C)NC(C#C)C1CC1 c1(C(=O)NC2(CNC(c3cn[nH]c3)=O)C(C)CCCC2)cncc2nc[nH]c12 C(=O)(C(CCC(C)C)NC(c1coc(SC)c1)=O)N(CC(CCC)C)C C(=O)(C(C)(C)C(F)F)NCC(C)N(C(=O)CCC1CC1(Cl)Cl)CC N1(C(COc2ccc(SC)cc2)=O)C2CCC1C(NC(=O)Cc1cnccn1)C2 c1(NC(C(CSCC)NC(c2nnn(C)c2C)=O)=O)cccc2c1OCO2 C1(C(N2C(C(C)NC(c3c(C)snc3)=O)CCC2)=O)CCC2CC2CC1 c1(C=O)c([N+](=O)[O-])c(C)nn1C.c1(CC)cc(C(=O)NC(C)CC)ccc1C.N c1(-c2c(OC)nccc2)ccc2nc(C(=O)N(CCC#N)C3CC3)oc2c1 C=CC(C)C(C)C(=O)N(C)CCN(C)C(c1ccc(-c2ccco2)nc1)=O N1(C(C2C(CNC(C(C(=O)OC)C)=O)C2(C)C)=O)CCN(C)C(C)C1 C1(C(=O)NCCCN(CCC)C(C2CCOC(C)C2)=O)CCC2(CCC2)CC1 Cc1cc(=NC(C)C2CCOC2)[nH]c(N(C)Cc2cc(Cl)ccc2C)n1 C#CCCCC(C(=O)NCSc1ccccc1)N1CCC(c2cn[nH]c2)CC1.O C(=O)(CC(C)(C)N(C(=O)Cn1cccn1)C)NC(c1ncc[nH]1)CC c1(C(=O)NCCC2(NC(CCCOC(C)(C)C)=O)CCC2)cccn2cncc12 Cc1oc(C#N)cc1C(N1CC(N2CCN(C(C3(C)CSC3)=O)CC2)C1)=O Cc1cccc(CCC(=O)NCC(N2CCN(CCCS(C)(=O)=O)CC2)=O)c1 C(CCN=c1cc(C)c(S(=O)(=O)NCCCn2ccnc2)c[nH]1)c1nnc(C)s1 CN1CCCC(CC(N2CC(O)CC2C(N2CCOCC2C(N)=O)=O)=O)C1 CCCS(=O)(=O)C(C)C(=O)NC1CCCCC1NC(=O)CCc1nc(CC)no1 N1(C(C(COC)C)=O)CC2C(NC(c3c(OC)cccc3Cl)=O)CS(=O)(=O)C2C1 N1(C(Cn2nnc(C)n2)=O)CC2(C1)CN(C(=O)Cc1ccc(F)cc1C)CCO2 c1(C(C)C)ncc(Cl)c(C(=O)NC2CC(NC(C3(C)CCOCC3)=O)C2)n1 C1(CNC(C2CCCC(CF)C2)=O)CCC12CCN(C(c1ccccc1)=O)CC2 c1(OC)ccc2c(c1)cc(C(=O)NC1CCCC1NC(=O)CC(C)C(C)C)n2C c1(C(N2C(C)C(NC(=O)CSc3cn[nH]c3)CC2)=O)ccc2scnc2c1 c1(CN2CCC(O)(C(=O)Nc3cc(C)c(Cl)cc3)C2)cc2ccncc2[nH]1 C1(NC(c2nccc(N)c2Cl)=O)CN(C(=O)CCc2nccs2)C2(CCOC2)C1 C1(CNC(C2C(C)C2)=O)CC2CCC(C1)N2C(C1(C)CC(=O)C1)=O c1(C(N2C3C(NC(C4C(OC)CCC4)=O)C(C3)C2)=O)cnc2sccc2c1 O=C1CCCC(CC(=O)NCc2ccc(C(=O)NC3CCCCCC3)nc2)C1 CC(C)(F)C(C)(F)CNC(=O)CCC1CCN(C(=O)C=CC(F)(F)F)C1 c1(C(=O)Nc2cccc(C)c2)cnn2cc(-c3cnn(CCO)c3)ccc12 N1(C(=O)CN2CCOCC2)CCC2(CCCN(Cc3c(F)cc(Cl)cc3Br)C2)C1 c1(C(=O)NC2CC(N(C(=O)Cc3cn[nH]c3)C)C2)nc(C2CC2)cs1 C1(C)(CC(N2CCCCC2)=O)CCS(=O)(=O)N1.[nH]1cnc(C(=O)NC)n1.CC N1(c2nnc(C(C)(C)C)o2)CCOC(C)(CNC(=O)CCc2ccccc2F)C1 N1(C(c2c(C)cc(F)cc2)=O)CCCC(O)(CNC(=O)C2CC2)CC1 N1(C(c2c(COC)cco2)=O)CCN(C(c2cn(C3CCC3)nn2)=O)C2CC12 c1(C(=O)NCCC2CCN(C(c3nc(COC)oc3)=O)C2)cnc(S)nc1 CCC(CC)C(C(=O)NC1(CO)CN(C(C2CC(=O)N(C)C(=O)N2)=O)C1)OC C1(NC(C(CC)C2CCOCC2)=O)CC2CCC1N2C(=O)CN(C)C1CC1 C1(C(=O)NCC(CO)NC(C(n2ccc(C)n2)C)=O)CCN(C)CC1 C(C)(C)(CC(C)C)NC(c1oc(CC)c(C)c1)=O.c1(CC(=O)N)ncccc1C C(=O)(C(C)(C)CCS(C)(=O)=O)N1CCN(C(CCC(=C)C)=O)C(CO)C1 c1(C(N(C2CCN(Cc3nnnn3C)CC2)C(C)=O)=O)c(C)nn(C)c1C N1(C(COCCC)=O)CCN(C(C2CC(F)C(=O)N2)=O)C(c2ccccc2Cl)C1 N1(C(c2c(OC)n[nH]c2)=O)CCC(CO)(NC(c2ccnc(OC)c2F)=O)CC1 C1(NC(c2cc(COC)sc2)=O)CN(C(C23CC(C)(C2)C3)=O)CC1C c1(C(=O)NCCN2CCN(C(C3(O)C(C)(C)C3)=O)CC2)cn2ccccc2n1 C=CC1(NC(c2cccc(CNC(c3sccc3C)=O)n2)=O)CCCC1 C(=O)(CCCC1CCCO1)NCC(C)(C)OCC(=O)N(CC(C)C)C N1(C(c2cc(COC)no2)=O)CCN(C(C2CCS(=O)CC2)=O)C2CCCCC12 C(=O)(CC(C)C(=O)NCC(C(=O)NC12CCN(CC1)C2)N(C)C)OCC N1(C(C2(C#N)CCCC2)=O)CCCCC(CNC(c2cccnn2)=O)C1 N1(CC(=O)NC(CC=C)CNC(=O)C(C)N(CC(F)(F)F)C)CCCNC1=O Cc1nonc1CC(=O)NCCCOCCN(C)C(c1scnc1C(C)C)=O C=CC1(C(=O)NC)CCN(C(=O)CSc2nc[nH]n2)C1.c12ccc(c(F)c1)[nH]2 C1(CC(C)(C)C)CN(C(c2csc(CO)n2)=O)CCN1C(=O)C(F)=CC1CC1 n1(CC(COCC)O)cc(C(C)NC(=O)C(CSC)NC)nn1 N1(C(C(C)(F)F)=O)CCC2(CCN(C(=O)COc3ccc(Br)cc3)C2)C1 N1(C(c2cnc(C(C)C)s2)=O)CCOCC(CNC(=O)C)C1.c1cnn(C)c1.S Cc1ccc(NC(C2CCCN(C(c3ccnc(C(C)C)c3)=O)CC2)=O)c(C)c1 c1(C(N2CCCC(CCNC(C(C)(C)C(F)F)=O)C2)=O)cc2cc(F)ccc2o1 c1(N(C(=O)CN2CSCC2=O)CC)ccc2c(c1)OCO2 C(CC(O)C(=O)NC1CCC2(CC2)C1)NC(C(C)NC(CC)(C)C)=O C(=O)(C1COc2c(C)cccc21)NC1(C)CC(NC(C(CC)OCC)=O)C1 C(=O)(C(C)CC(N)=O)N1C(CNC(c2ccc(NC(C)=O)cn2)=O)C=CC1 C1(NC(C(C)N(C(=O)CCCCN=[N+]=[N-])C)=O)CCn2ccnc2C1 c1ccc(S(N)(=O)=O)cc1.Cc1cc(C(=O)NC2CCC2NC(=O)C)cs1 N1(CC(=O)NC(C(=O)NC(c2cnc[nH]2)C)C2(O)CCC2)CCCC1C CC(C(=O)NCC1CC(C(N2CC(C)(C)C2C2CC2)=O)C1)C(F)F C(=O)(C1CCOc2ccc(Cl)cc21)NC(C)CNC(=O)CCCN1CCCCC1 c1(C(N2CCC(N3CCOCC3)C2)C(=O)NC(CC)C)cc(C(F)F)on1 Cc1noc(N)c1NC(=O)NCC(=O)NC(C)C(C)F N1(C(c2nn(C)c(=O)cc2)=O)CCC2(CC1)CN(C(=O)COc1cn[nH]c1)C2 CC(C)CC(O)CC(=O)NC1(C(N2CCNC(=O)C2CCO)=O)CCSC1 N1(C(C2(CC#C)CCN(C(=O)CN3CCC(C)CC3)C2)=O)CCCN(C)C(=O)C1 c1(CC(=O)N(CCC)C)cc(Cl)n(C)n1.c1(C(=O)N)ccc(-c2nc[nH]n2)nc1 C(C)(CCN=c1ncc(Br)c[nH]1)NC(c1n[nH]c(C)c1[N+](=O)[O-])=O C(CC(C(=O)N)NC(=O)C(C)COC(C)=O)SC.C1(CC)CCCC2CC12 N1(CC(=O)NC2CC2)CCN(C2CC2C2CCNCC2)CC1 CC1CN(C(=O)C(=O)NCC2CC2)CC1.C(=O)CC.c1(C=O)ccco1.N c1(C(=O)NC2CN(C(CC(=O)OC)=O)CC(F)C2)cc(OC)c(F)c(OC)c1F Cc1ccc(=O)n(CCOC2CCN(C(=O)CNC3CCN(C)C3(C)C)CC2)c1 Cc1cccc2cc(C(=O)NC3CCC(CNC(c4cnn(C)c4Cl)=O)C3)nn12 CC1CCN(C(=O)CC2CCCC2)CC1CNC(=O)CCc1cnco1 c1(OC)ccc(CNCc2cccc(CN3CCN(C)CC3)c2)cc1O Cn1nc(-c2ccc(N(S(C)(=O)=O)CCC3CCNC3)cc2)nc1C(F)F C1(C(C)C)CN(C(C2N(C(C3COCC(C)O3)=O)CCC2(C)C)=O)CCN1C C(=O)(CN=S(C)(C)=O)NC1C(CNC(C(CC=C)c2ccccc2)=O)CCCC1 c1(CN2CC3(C(C(=O)NCc4n(C)ccc4)C3)C2)ccc(F)c(Br)c1F Cc1ccc(C(c2nnnn2C2CC(F)(F)C2)NC(c2ccco2)C)n1C C(CCC(C)NC(=O)C(C)(C)C1CCCCO1)NC(CN(C(C)C)C)=O CCC(C(=O)NCC1CCC(C)(C)CC1)C(C)C c1(C(=O)NCc2scc(C(C)(C)C)n2)c(Br)cc(F)cc1Br Cc1cccn(CC(=O)NCCOCCN(C)C(C2CCCCC2O)=O)c1=O CC(C)C(O)(C(=O)N(CC(C)C)C)C(F)(F)F.c1(CC=O)nc([N+](=O)[O-])n[nH]1 C1(C(=O)NC2(CNC(C(C)(C)c3cc[nH]n3)=O)CCCC2)CCN2CCC1C2 C(CCCCCN=c1ncc(Br)c[nH]1)NC(C1C=CCCC1)=O c1(C(N2C(CCNC(c3cnc(O)o3)=O)CSCC2)=O)ccc2nc(S)oc2c1 c1(C(N2CCN(C(C3(CC)CC3)=O)CC2C)=O)cc(I)c(F)cc1F CC(N=[N+]=[N-])C(=O)NCc1cc(C(=O)NCCCS(C)=O)cs1 C=C(F)CN=c1[nH]c(=NC(CF)c2ccc(C#N)cc2)c2cc(Cl)ccc2[nH]1 C1(NC(C(Cn2ccc(C)n2)C)=O)CCCN(C(c2cnc(C#N)s2)=O)CCC1 CCC(C)C(C(=O)N1CC(O)(CN(C(=O)CO)C)C1)NC(c1ccco1)=O C1(NC(C2CC3OC2C2CC32)=O)CCCOC12CCN(C(C1CC(O)C1)=O)CC2 C1(NC(c2c(C)cc(C)s2)=O)CCN(C(=O)C(c2ccccc2Cl)O)CC1F c1(N(C)C)ccc(C(=O)NCC2(NC(C3(O)COC3)=O)CC2)nc1 c1(C(=O)OCC(C(C)(C)C#N)=O)cccc2[nH]c(=O)c(=O)[nH]c12 C(C)C(C)(C)C.c1ccccc1.C(C=O)N(C1CC1)CC.C1(C=O)CC1.N c1(C(N2CC(CC)C2)=O)cc(C2CC2)nc2cc(C)c(C)cc12.C(C(=O)N)OC C1(C(=O)NCc2c(C)ocn2)CCCN(C(C2(C)CCCCO2)=O)CC1 C1(O)(C=O)CCOCC1.c1(-c2cc(C(=O)NC3CC3C)on2)ccc(Cl)cc1 CC(CC#N)N=c1[nH]c(N2CCNC(=O)C(F)(F)C2)nc2c1SCC2 C1(NC(C(F)=CC)=O)CC2CC(NC(c3cc(C)c(F)cn3)=O)CC2C1 Cc1cc(C)c(C(=O)NCC(F)CNC(C2(C)CCOCC2)=O)cc1N C(=O)(C(CC)(CC)C(=O)O)N1CCC(NC(c2c(CC)cccc2)=O)CC1 N1(CC2(CC)CCC2)CCCC(O)(CC(=O)OC)C1 CCC(CC(F)(F)F)C(=O)NC(C)CC1CN(C(=O)C(C)Sc2nncn2C)C1 C1(C)(CC)CCCN(C(C23CC(NC(c4n[nH]c(C)c4C)=O)(C2)C3)=O)CC1 CCCCCC(O)CC(=O)N1CCC(CNC(=O)C(O)c2ccsc2)CC1 Cc1nc(C(C)NC(=O)CCCN(C)C)c(C)o1.C12(C(=O)N)CC(C1)C2 C(=O)(C(CCCC=C)NC(=O)C(C)C1(O)CCC1)N1CCCC(C#C)C1 C1(NC(CSC(C)(C)C)=O)CC(F)CN(C(c2nc(=N)cc[nH]2)=O)C1 c1(C(=O)NCC2CCCCN(C(C(COC)(C)O)=O)C2)ccc2nc[nH]c2n1 C(=O)(CC(O)CNC(C1CN(C(c2cccc(O)n2)=O)CC1OC)=O)OC c1(N2CC3CN(C(c4ccccc4C4CC4)=O)CC32)ncnn2cccc12 C(CCCCC(=O)NCC(CC(=O)NCc1ncc(C)cn1)OC)=CC C1(CC)CN(C(c2cccc(F)c2Cl)=O)CCC1NC(C1(C)CCC(=O)NC1)=O c1(OC)cc(F)c(F)cc1-c1ccc(C2(C(=O)N)CC2)cc1.c1ccc(Br)s1.C C1(N(C(=O)CCc2cscn2)C)CCN(C(=O)Cn2nnnc2-c2ccsc2)C1 c1(CC(=O)NCC2CC3(CC3)CN2c2ncncc2Br)ccc([N+](=O)[O-])cc1 c1(C(=O)NC2CCC(CNC(=O)C3=CCOC3)CC2)cnc2cc[nH]c2c1 Cc1cc(C)c(C(=O)N)[nH]1.C1(C)CCN(C(=O)C(c2ccc(Cl)cc2)(F)F)C1.C C1(NC(CC2CCCC(NC(C(C)OCCCC)=O)C2)=O)CC(F)(F)C1(C)C C1(OCC(=O)N(CCC)CCNC(=O)CC2CCCC2)C#CCCCCC1 Cc1nnn2cc(C(=O)NC3(Cc4ccccc4F)CCCC3)ccc12 C1(NC(C(C)NC(C)=O)=O)CC2CC(NC(c3ccc(N)c(F)n3)=O)C2C1 c1(C(N2CC(CC(C)NC(C3(C#N)CC3(C)C)=O)C2)=O)ccnc2ncccc12 C1(C(=O)NCCNC(C(C(C)C)n2ccnc2)=O)CC2(C1)CC2(F)F CCC(C)(C#N)C(=O)N1CC(NC(=O)CCC(C)C)C(CO)C1 Cc1ccc(CC(c2ccc(C(C)(C)C)cc2)NCCCNC(=O)C(C)C)cc1 C12(OC)CCC1CN(C(=O)C(C1CCOC1)NC(=O)CCc1nncs1)C2 N1CCS(=O)(=O)CC1.c1(OC)ccc(C(=O)NCC2CC2)s1.[nH]1ccnn1 c1(N2C(=O)CCC2)ccc(S(=O)(=O)N2CC=C(F)C2)cc1 C(=O)(C(CCF)NC(c1cc(C)nn1C)=O)NC(c1ccnn1C)CC c1(C(=O)NC2CC(NC(c3c(C)cc(C)cc3N)=O)C2)cnc2c(Cl)cccn12 c1(OC)ccc(C(C)C(N2CC(CC(=O)O)C2)=O)cc1.C(=O)(CN(C)C)N c1(OC)cc(C(=O)NC(CCNC(c2c(C)ncn2OC)=O)C(C)C)ccc1Cl S(=O)(=O)(CC(=O)N1CC2CC1C2)N(C)C.c1(C=O)cccc(C2CC2(F)F)c1.N N1(C(c2cc(C(C)=O)on2)=O)CC2(CCCC2)C1C(=O)NC.c1nnc(O)o1 CCC(C(=O)N1CCCC(C)(C(=O)NC(CC2CC2)CO)C1)C(F)(F)F Cc1cc(N)n2ncc(C(N3CC4CC4(NC(c4oncc4C)=O)C3)=O)c2n1 c1(CC2N(C3CN(C(C4CCCCCC4)=O)C3)CCC2)cccc(Cl)c1 N1(C(C(CC2CCC2)OC)=O)CCCC(C)(C)C1C(=O)NCC1=NOC(C)C1 N1(C(C(C)SC)=O)CCC(F)C(NC(C2(c3ccccc3)CC(F)C2)=O)C1 c1(C(=O)NC(C2CCCCN2C(=O)C2=C(Cl)CCC2)C)cccc(N)c1O Cc1ccc(C=C(C#N)C(=O)NCC2CCCC2)cc1.n1(CC=O)ncnn1 CCCCCS(=O)(=O)CC(=O)N1CCN(C(c2snnc2CCC)=O)C2CCC12 C(=O)(C(CC(C)C)C(N)=O)NC(C(=O)NCC(CCC)CCC)CC N1(C(C2(C=C)CCC2)=O)CC(CNC(c2c(C)ncnc2C)=O)C(F)(F)C1 N(C(=NCCc1ccncc1C)N1CCC(F)(C(=O)OC)C1)C(CC)C c1(CC)cccc(C(=O)NC)c1C.C(=O)(C(CN(C)C)C(C)C)N1CCCCC1 c1(NCC(C(CC)C)O)cc(Br)ccc1S(=O)(=O)NCc1cc(C)c(Br)cn1 C1CC2CCC(C1)N2C(=O)C=Cc1cncs1.C(C=O)N(S(C)(=O)=O)C.C C(C)(CC1CCC1)C(=O)N1CCOCC1.C1(C(F)(F)F)(C(NC)=O)CC1.C Cc1cc(C(N2CC(N(C)C(C3CC4C=CC3C4)=O)C2)=O)c(C)nc1C c1(C(N2CCC(CN(C)C(c3ccns3)=O)C2)=O)ncccc1.CC(F)(F)F.O CC1CC(O)CN1C(=O)CCC1CCN(C(C2COCOC2)=O)C1 c1(C(N2C3(C(N4CC(CN=[N+]=[N-])C4)=O)CC(C2)C3)=O)ccc2ccoc2c1 C12(NC(CCc3n(C)ncc3)=O)CCN(C(=O)Cn3cncn3)CC1C2 C1(F)(CNC(=O)CC2CCCCC2(F)F)COCCN(C(c2ccncc2)=O)C1 c1(C(C)NC2CCCN(C(CNC(C)C)=O)C2)nc2cccc(Br)c2[nH]1 Cn1nc2c(c1NC(C1C3CN(C(c4cc(Cl)cnc4F)=O)CC13)=O)CCC2 c1(C=O)cnc([N+](=O)[O-])n1C.C1COCC1.C1(CC(=O)NC)(OCC)CC1 c1(OC)cc(N)c(F)cc1C(=O)N(C)CCN(C)C(c1cc(C)sn1)=O C1(C(N2CCC(C(C)NC(Cc3c(C)cnn3C)=O)CC2)=O)CCS(=O)(=O)CC1 CC1CN(C(c2cn(CCNC(c3cc(O)nc(O)n3)=O)nn2)=O)C(C)C1C c1(-c2cn(CC)nc2)ccc2ccnc(NC(c3sccc3Br)=O)c2c1 N1(C(C(=O)Nc2cc(C(=O)OC)c(F)cc2F)=O)CCCC(C2CCC2)CC1 N(C(=NCCCCC(F)(F)F)NCc1cnns1)CC1CC(=O)NC1 C12(CC)CCC(C(=O)NCCC)(CC1)CO2.c1(C=O)ccc(N(C)C)cc1F.N C1(CNC(c2ccc3c(c2)CC3)=O)CCCN(C(=O)CSC2CC2)CC1 c1(OC)nc(C)sc1C(=O)N(CCCNC(C1(C)CCCS1)=O)C1CC1 C12(C(=O)NC(C(C)NC(c3c(N)cccc3F)=O)C)CCC(C)(CC1)CO2 c1(CC(=O)N(C)Cc2c[nH]nc2-c2ccccc2)ccc(Cl)cn1 C1(CN(C(c2ccsc2Br)C(=O)NCCC)C)CC(OC)C12CCC2 C1(CC(=O)NC(CN(C(C)C(=O)NC2CC2)C)C)CCCN1C(C)=O N1(C(C(=O)NC(C)CCNC(c2ncccc2O)=O)C)Cc2ccccc2C1=O N1(C(COCCN(C)C)=O)CC2CCC(C1)N2C(C1CCC=CCCC1)=O C=CCCCC(=O)N1CCCCC1CCCNC(=O)C(C)Sc1ccc(C)cc1 CC1CCn2c(C(N3CCN(C(=O)C=CCO)C(CC(F)(F)F)C3)=O)cnc2C1 C1(C)(NC(Cn2ccc(C)n2)=O)CCN(C(C2(Br)CC23CCC3)=O)C1 c1(C(N2CCN(CCCNC(C(C)CF)=O)CC2)=O)coc2c1NC(=O)CCC2 N1(C(COc2cccc(CC)c2)=O)CCC2(NC(=O)CN(C)CCO)CCCC12 Cc1csc(=O)n1CCC(N1CC2CC1(CNC(c1cccnc1CO)=O)C2)=O CC1CN(C(C2CN(C(c3ccc(Cl)cc3)=O)C(C)(C)C2)=O)CCC1O CC(CCCCNC(=O)CN1CCC(F)(F)C1)NC(=O)CCC1CCCO1 C1CC2CC(C1)N(C(=O)C1=CC(C)(C)C1)C2.Cn1nccc1C1(C(=O)N)CC1 Cc1ccnnc1C(=O)N(CC(Cc1ccccc1)NC(c1cncn1C)=O)C O=C1C(NCc2cccc3cncn23)CCN1C1CCCc2ccccc21 N1(C(CCC(C)OC)=O)CCCC(NC(=O)C(C)CSc2ccccn2)CC1 CCCC(O)CC(=O)N1CC2(CNC(c3cn(C)c(=O)n3C)=O)CCC1C2 N(C1c2ccccc2CCC1C(=O)O)C(Cn1cc(C2C(C)(C)OCCO2)nn1)=O Cn1nc(C(=O)NCC(F)CNC(c2ncnn2C(C)C)=O)ccc1=O C1(C(=O)OC)CC(C=O)C12CCC2.C12COC(C1)C2.CC=CC.CCO.N N1(c2ccnc(C(C)C)n2)CC(NC(=O)Cc2ccc(F)cc2)CC(F)(F)C1 C1(C(=O)NC(CCCC)CO)CC12CCN(C(=O)C(=O)Cc1ccc(O)cc1)C2 N1(C(C2(C)ON=C(C)C2)=O)CCN(C(c2cnns2)=O)C(c2cccnc2)C1 C1(C(=O)NCCC(C)C)(OC)CCS(=O)(=O)C1.c1(C(=O)N)ccc(F)cn1 C(CN=C(NCC(O)CF)N1CC(C)CC(C)(C)C1)OC CC1CN(C(=O)CN(C)C2CC2)CC(C(N2CCC(c3ccon3)C2)=O)O1 C(CC(C)C)(C(=O)N)NC(C)=O.c1(C=O)ccnn1CC(F)(F)F.CC(C)C C(c1ccc(Br)cc1F)=CC(N1C(C(=O)N(C)CCN(C)C)CC(OC)C1)=O Cc1[nH]c2ccccc2c1C(=O)NCCC1(NC(=O)CN2CC(C)C2)CCC1 C(=O)(C#CC1(C)CC1)N1C(CCNC(C2CC(OCC)C2)=O)CSCC1 CCC(C)(C(=O)N(CCCCCCNC(=O)C(C(C)C)n1cncn1)C)C(N)=O C1(C=O)COCC1C(N1CC(O)(CC)C1)=O.c1(C=O)coc(C2CC2)n1.C C(N=c1[nH]cnc(Cl)c1C(C)=O)C1(F)CC(NC(C(C(COC)C)C)=O)C1 c1(C(N(c2cc(O)c(Cl)cc2Cl)CCCC)=O)nccc2c(C)cccc12 c1(N2CC(CNC(C3(C)ON=C(C)C3)=O)OCC2)nc2cc(Cl)ccc2s1 c1(OC)cc(C(C(=O)NC(C)C)N(C2CCCC2(C)C)C)ccc1Br CC1(C)C(C(=O)NC2COCC2n2cc(-c3ccc(Cl)s3)nn2)C1C(F)F N1(C(C2CC(OC)C2)=O)CC(NC(=O)CC2CCCCCCC2)CC12CCC2 Cc1ccc(=O)n(CC(=O)NCC2(F)CN(C(=O)CN=S(C)(C)=O)C2)c1 C=C(C)C(CC(=O)N1CCN(C(c2cc(CC(C)C)[nH]n2)=O)CC1CC)OCC N1(C(C2C(CC)N(C)CC2)=O)CCN(C(c2cnc(O)n2C)=O)CC1C Cc1cc(C(=O)NCC2CCOC2CNC(=O)C)cc(C#N)c1.CCF.O CCC(CC)CCCC(=O)NC(CC(N1C(CO)CCC12CCC2)=O)C(F)F CC1(C(=O)NC23CC2CN(C(c2noc4c2CCCC4)=O)C3)CCCCNC1=O N(C)(C1CN(C(C2C(C)C2C)=O)CCc2ccccc21)C(c1nc(C)sc1C)=O c1(OC)ncccc1-n1ncnc1C1CC(=O)N(C)C1 Cc1cc(C)c(C(=O)NCC(O)C(=O)NC2CCC(N(C)C)C2)cn1 c1(OC)ccc(C)c(C(=O)N)c1.c1(C(N2CCC2)=O)ccnc(C(N)=O)c1.C c1(OC)ccc(C(N2CCC(C(=O)NCCCc3ccccc3)C2)=O)s1 C(=O)CC(C)O.Cc1ccoc1C(=O)NC1CC1C.c1(C=O)ccccc1.N c1(OC)ccccc1C(=O)NC1CCC(NC(C2CC2C(=O)OC)=O)CC1 CC(C)C(=O)N(CCCN(C)C)C(C)C.C1CC(C#N)C1.CC=O.CC=O.O c1(OC)ccc(C(C)CC(=O)NC(C)C(C)NC(c2c(C)noc2N)=O)cc1 Cc1cccc(CN2CCC(F)(C(=O)Nc3ccnc(F)c3Br)C2)c1Cl C=CC(C)C(C)C(=O)N1CCC(NC(c2[nH]c(C)c(C(N)=O)c2CC)=O)CC1 N1(CCC(=O)NCCN(C(=O)COC2CC2)CCCCCF)CCCCCC1 CC1CN(C(C23CCC2CC3)=O)CC1NC(=O)CSCc1cccs1 N1(C(C(C)c2cc[nH]n2)=O)CC2(CCCC2)C1C(=O)NOCC(F)F c1(C(N2CCC(F)(CO)C2)=O)ccc2ncc(-c3ccc4ncsc4c3)n2c1 N1(C(c2cc(Cl)ncn2)=O)CC2CCC1CN2Cc1scc2c1OCCO2 C=CCCCC(C(=O)NCC1(N(C)C)CCC1)NC(=O)CCC(=O)CC Cc1nc(CC(=O)NCC2CC(NC(=O)C=CC=O)C2)[nH]c1C.C1CC1 c1(C=O)ccc(C)c(C)c1.N1(C(CCOCCOCC)=O)CCCCC1C.N Cc1cc(CCC(N2CCC(NC(=O)CCOC3CCOC3)C2C)=O)nn1C Cc1nc(NCc2ccccc2Cn2cccn2)c2ccsc2n1 c1(C(N2CC(F)(CNC(Cn3ncc(C#C)c3)=O)C2)=O)sccc1[SH](=O)=O.N C1(NC(CCC(C)O)=O)CN(C(c2cn(CC3CC3)nn2)=O)CC2(CCC2)C1 c1(C(=O)NCC2(C)N(C(CC(CC)OC)=O)CCC2)ccn2[nH]c(=N)nc2c1 C(CCC)(CCCNC(c1csc2nnsc12)=O)NC(COCCCC)=O C1(NC(C2OCCO2)=O)CS(=O)(=O)C2CN(C(C3CCCNS3(=O)=O)=O)CC12 C1(C(N(C2(C(=O)NC(C(C)F)C)CCC2)C2CC2)=O)CCC(C)CC1 N1(C(C2CSC2)=O)CCCCC2(CCN(C(=O)Cc3cnn(C(F)F)c3)C2)C1 CC1Cc2cccc(S(=O)(=O)NC3CC=CCC3C(F)(F)F)c2O1 C1(NC(c2ccc(Cl)s2)c2nnnn2CCC2CC2)CCCOC12CCC2 CC1CN(C(=O)CC2CCOCC2)CCC1CNC(c1ccc(N)c(Cl)c1)=O C1(Nc2cccc(-n3ccnc3)c2)C2C3CCC(C3)C12 c1(OC(C(N2CC(O)(CNC(CC(C)C3CC3)=O)C2)=O)C)ccccc1F C12(NC(=O)OC(C)(C)C)CCC1(C(=O)O)CN(Cc1nc3ccccc3[nH]1)C2 C1(NC(C(=Cc2ccco2)C)=O)CN(C(=O)C(F)Cc2ccccc2)CC12CC2 Cc1nc2ccc(NC(C3CCCN(Cc4ccc5c(c4)OCO5)C3)=O)cc2s1 N(C(=NCc1ccc(F)cc1)NC(C)C)CC(CC)(C)O c1(NC(C)CO)cc(Br)ccc1S(=O)(=O)NCc1ccc(C(C)(C)C)nc1 c1(CNC(c2nnc(C)s2)=O)nc2c(s1)CCN(C(=O)C(C1CCOCC1)F)C2 c1(C(=O)NC(CC2CN(C(C(CC)(F)F)=O)C2)C)nc2n(c1Cl)CCCC2 C(=O)(CC=C(Cl)Cl)NCCN(CCOC)C(c1cc(C(F)(F)F)ns1)=O C(=O)(C(CC(C)SC)N(C)Cc1ccccc1OC(F)F)NCC(=C)C c1(C(N(CCCOCCNC(CCCCC=C)=O)C)=O)cc2c[nH]nc2cc1C Cc1cc(C)c([N+](=O)[O-])c(C)c1C(=O)NC1CCN(C(C23CC(C2)C3)=O)C1 c1(C(=O)NC2CCCN(C(c3cnc(C)nc3)=O)C2)cnc2n1CCC(C)C2 C(=O)(C1(C)CCCc2ccccc21)NCCNC(CCc1scc(C)n1)=O c1(C(N2CC(N(C(c3ccc(COC)o3)=O)C)C2)=O)c(C)cccc1[N+](=O)[O-] CCC(CN=C(NCC(C)(C)C)NCC1(O)CCCC1)C(=O)OC(C)(C)C C1(C(=O)NC(CN(C(C(C)(C)OCCC)=O)C)CC)CCN(C)C1C c1(C(=O)NC2CC(CNC(CC=C)=O)C2)ccc(N(C)C)cc1 Cc1c(NC(C2COCCN2C(c2ccc(F)cc2F)=O)=O)ccc(C#N)c1F N1(C(c2ncc(C)cc2F)=O)CC2(CCN(C(C3CCOC3C)=O)CC2)C1 N1(C(CC(C)C)=O)CCCC2(CCC2NC(=O)CC2CC=CCC2)C1 N1(C(C(CC)CC)=O)CC(NC(C2(C)CCOC2)=O)CC2(CC2)C1 CC1=CC(C(=O)NC(C)(C)C=CC(=O)NCC(c2cccs2)O)SC1 N#Cc1ccc(C(=O)NCC(C2CC2)NC(C2CCOC2)=O)s1 N1(C(CCC2CC2)=O)CCC(C(N)=O)C(C)(C)C1.C(=O)(CC=O)OCC N1(C(c2n(C)ccc(=O)c2)=O)CC2CCN(C(c3cccnc3O)=O)C2C1 c1(C(N2CC3(CCN3C(c3cccc(Br)n3)=O)C2)=O)cc(F)cc(F)c1F C1(NC(C(C2CCCC2)NC(=O)CC2CC2)=O)C2CCCOC12 C1(C(=O)NCc2nc(CCOC)no2)CCCCN1C(=O)Cc1cccs1 C1(NC(C=CSC)=O)CN(C(C2(c3ccc(C)nc3)CC2)=O)CCC1O C1(C(N2CC(N3CC(NC(=O)C)CC3=O)C2)=O)(CC)CCNC1=O.C(C)=O CCC(CCC(=O)NC1(C(=O)NC2CCN(CCO)CC2)CSC1)OC c1(CC(=O)NC2CC23CC(NC(C2C=CCC2)=O)C3)ccc2c[nH]nc2c1 Cc1cn2cccc(NC(C3CC34CCN(Cc3csc([N+](=O)[O-])c3)C4)=O)c2n1 N#Cc1cccc(-n2ccc(C(N3CCC(CF)(NC(=O)CNC=O)C3)=O)n2)c1 [SH](=O)(=O)c1c[nH]c(C=O)c1.C(C)(C)CO.N1(CC=O)CCCC1=O.CCN C=C(F)C1(C(=O)NCC2CC2NC(=O)CN(CC)CC)CCC1 CC1CCCCC1(c1nnnn1C1CCCC1)NCCn1cncn1 c1(CC)cc(C(N2CC(C)(C)C2C2CCN(C(=O)C#CC3CC3)CC2)=O)ccn1 N(C1CCCc2n[nH]cc21)C(C1(CC=C)CCCN1C(C1CC12CC2)=O)=O N1(C(c2c(C)ncnc2)=O)CC2CCCC2(CNC(=O)CCc2cc[nH]n2)C1 C(=O)(CCC(C)(C)c1ccccc1)NCC(CC)NC(C1CC(C)=NO1)=O C(N=c1[nH]c(Cl)ncc1C(N)=O)C1C(C)CCCN1C(C1CCCC(O)C1)=O CC(C)(C#N)CC(C(=O)NCCC1(C)CC1)N1CCCC1c1cccc(F)c1F C#CCCC(=O)NC(c1ccccc1)CNC(C1(CCOCC)CCC1)=O C(C(C)(C)CC(=O)N(C)CC1(NC(C2CCCC2C)=O)CC1)OC(C)=O c1(C(=O)NCC=CC(=O)N(CCCCO)C)n[nH]c2ccccc12 N1(Cc2c(OC)n(C)nc2)CCS(=O)(=O)C(Cc2ccccc2)C1 N1(C(C=CC)=O)CCCN(C(=O)COCC2CCCCO2)CC1C c1(C(=O)N)cnn2ncccc12.C(C1CCCN1C)=CC(=O)N(CC(C)O)CC C1(C(=O)N)(OC)CCC(C)C1.CC(C)(F)C.n1(C2(CC=O)CC2)cncn1 CCCCCC(C)CC(=O)NC(C(=O)N(CC(C)N(C)C(C)=O)C)C(C)(C)O CC1(C)CC(NC(c2ncccn2)=O)CN(C(C2CCOC2)=O)C1.CC(F)(F)F.O c1(CC)cc(NC(=O)CC23CCC2CN(C(=O)C(=O)NC)C3)ccc1F C(=O)(CCN=c1[nH]ccs1)N1CC(NC(C2CSCCS2)=O)C1 C(N=c1cc(C)c(S(=O)(=O)NC(CC2CC2)CO)c[nH]1)c1c(OC)cccc1Cl C1(C(=O)NCCc2c(C)cccc2)CC12CCN(C(C1CC3CCC1CC3)=O)C2 C1(NC(C2CN(C(CC3(OC)CCC3)=O)CC2C)=O)CCC(C2CC2)CC1 C(C(C)(C)CN=c1[nH]c(=NCC2CC3C=CC2CC3)[nH]c2cc[nH]c12)OC c1(C(=O)OC(c2c(F)cccc2Br)C)c(O)cc(Br)cc1F C1(NC(CCC(=O)NCCC)=O)CCCCN(C(=O)C(O)C=CCCC)C1 C(=O)(CCCCC(=O)NCC(N1CCN(C(c2oc(C)cc2C)=O)CC1)=O)NC C(=O)(C(CNC(=O)C(c1ccccc1)O)C(C)C)NCC(=C)C CCC(C)CC(C)CNc1nccc(C(F)F)n1 CC(C)(CC(=O)NCC(c1cccc(Cl)c1)NC(c1cc(Cl)no1)=O)C(F)F N1(C(C(C=C)(C)C)=O)CC2CCCC2(C(=O)NC2COC(C(C)C)C2)C1 N1(C(c2cc(Cl)on2)=O)CC2CCN(C(c3cccc4cnsc34)=O)CCC2C1 c1(CNC(NC(c2ccnn2C)COC)=NCC2CC2)cc(F)c(F)c(F)c1F c1(C(=O)NCC(CC)NC(C2(F)CCCCC2)=O)ccc(Br)c([N+](=O)[O-])c1 c1(OC)ccc(C(C(=O)NCC(C)C)N(CCC(O)C(C)(C)C)C)c(C)c1 C(CC(N)=O)(C(=O)NCC(CO)N(C)C)NC(C(C1CC1)SC)=O C1(CN2CC(C(=O)NC)(Cc3ccccc3)C2)CC(=O)N(C)C1 C(C(C)(C)C(=O)NC1C=CCC(C(N2CCC2C)=O)C1)SC O=S(=O)(c1c[nH]ccc1=NC1CC1C(F)(F)F)NCC1(CO)CCC1 C=CC(C)(C)CC(=O)NC(CO)C(C)NC(C1CCC(=O)N1CCC)=O Cc1cc(C(=O)NC2(C)CCOC2)cc(C)c1.c1(C(=O)N)cc([N+](=O)[O-])n[nH]1 C1(NC(=O)C(O)c2cnc[nH]2)CCCN(C(=O)C(F)=C2CCCC2)C1 CCC(C)(CNC(=O)CCC(C)=O)C(=O)N(C(C)C(=O)NC)C c1(COC(c2c(Br)cncc2Br)=O)cc(I)cc([N+](=O)[O-])c1 C1(C=O)CC2(C1)CC(F)(F)C2.C1CCCC1O.CC(C(=O)NC)=C1CCCC1 N1(C(C(C)OCC)=O)CCCC1CN(C)C(c1snnc1C1CCC1)=O Cc1ccccc1CCC(N1CC(N(C(=O)COc2cnn(C)c2)C)C(F)C1)=O CC1(C)CC(NC(=O)CSc2ccccc2)CN1C(=O)CC1CCOC1=O N1(C(c2c(SC)n(C)nc2)=O)CCC(NC(=O)C(=Cc2ccccc2)N)C(O)C1 c1(C(N2C(C)C(C)N(C(=O)C(=O)N=S(C)(C)=O)CC2)=O)cnc2nccnc2c1 C=CCC(C)(CC)C(=O)NC1CCN(C(=O)Cc2cc(C)ns2)CC1F N1(CCNC(C2CC3CCC2C3)=O)CCN(C(C2(C(F)F)CCCCC2)=O)CC1 c1(CCC(=O)NC2CN(C(c3nc[nH]n3)=O)CC23CC3)cccc(Br)c1F CCCCCC(O)CC(=O)N1CC2CC1CN(C(c1nnc(C(F)(F)F)s1)=O)C2 N1(C(c2c(SC)scc2)=O)CCCCC(CNC(=O)C(C)S(C)(=O)=O)CC1 C12(C(=O)NCC3(CNC(c4onc(C)n4)=O)CCCC3)CCCCN1CCC2 C1(NC(C=C(C)Cl)=O)COC2(CNC(=O)CCCNC(N)=O)CC1C2 C(=O)(CCCCCS(N)(=O)=O)NCCCCNC(c1cccc(CCC#N)c1)=O N1(C(c2cccc(CC)c2OC)C(=O)NC(C)C)CC(C)OC2(CCCC2)C1 c1(NC(C)=O)cccc(F)c1C(N1CC(c2[nH]nnc2C)C1)=O N1(C(c2cc(C)on2)=O)CCC(C(=O)NC2(c3cccnc3)CC2)C(O)C1 Cc1cc(C(=O)N(C2CCN(C(c3ccc(C4CC4)cc3)=O)CC2)C)c(C)s1 C1(C(=O)NC2CC3(CCN(c4snc(COC)n4)C3)C2)CCn2c(O)nnc2C1 C1(NC(C2(O)CCN(C(C)C(C)(C)O)CC2)=O)COC2(CCCC2)C1 c1(C(N(C)C)=O)sc(-c2ccc(OC(F)F)cc2)nc1N C(=O)(C(C)(C)C(F)F)N1CC(CN(C(=O)Cn2nnc(=O)[nH]2)C)OCC1 C1(C(N(CCCN(CC)CC)C)=O)CCN(C(=O)C(C2CCOCC2)=O)C1.C C1(OC)C2CC3CN(C(c4cc(F)cc(F)c4)C(=O)NC4CCOC4)C1C3C2 c1(C(=O)NC2CCC(N(C(C=CC=CC)=O)C)C2)ccc2cccc(O)c2c1 Cc1cccc(F)c1C(=O)NC1CN(C(c2cnc(C(C)(C)C)o2)=O)CC12CC2 c1(C(N2CC(C)C(CNC(c3cnc(Cl)s3)=O)CC2)=O)cccc2nccnc12 c1(OC)ccccc1-n1nnnc1C(C)(CCC1CC1)NC1CCC(CO)C1 C1(NC(CS(=O)(=O)NCC)=O)CC(O)CN(C(=O)CC(O)CCSC)C1 c1(C(=O)NC(c2n(C)ncc2)C(F)F)cc2cc(F)c(F)cc2[nH]1 N=c1ccc(C(=O)NCC2CCC2)c[nH]1.c1(C2C(CC=O)C2)ccccc1.N N1(C(CC2CCC(C)C2)=O)CCC(O)(C(C)NC(c2ccn(C)n2)=O)CC1 c1(CN2CC(NC(=O)NC(C(=O)OC)C)C(F)C2)ccc(C#N)c(F)c1 C(=O)(CC1=CCCCC1)NCCOCCNC(C(C)(C)Cc1cnn[nH]1)=O N1(C(c2cc(SC)c(F)cc2)=O)CCCC12CCN(C(=O)C=Cc1cn[nH]c1)C2 CCC(C)C(O)CC(=O)NC1C=CCCC1C(=O)Nc1cn(C)nc1C#N Cc1ccc(F)c(C(=O)NCCCCCC2CCN(C(C3CC3Cl)=O)CC2)c1F N1(C(c2c(CC)nccn2)=O)CCC(NC(c2scnc2C)=O)C(C)(C)C1.O C(=O)(C(CC)C(C)O)NCC1CCC(NC(CCCC#C)=O)CC1 CCCCC(C(=O)NCC1(F)COCCN(C(C2(C(C)C)COC2)=O)C1)C(C)C CCN1C(=O)COc2cc(NC(C3CCCC3C(F)F)=O)ccc21 Cn1cc(NC(=O)C(N2CCCC(CC(F)(F)F)C2)=O)c(C2CC3CCC2C3)n1 c1(CN(CCNC(c2c(CC)[nH]nc2Cl)=O)CC)ccc2c(c1)CCO2 C(CCN(C)C(C1CC2(C1)CC(O)C2)=O)C(C)(C)C.C1CCC1C=O.CO c1(CC(=O)N)c[nH]c2ccc(F)cc12.C1(CC)CCCC1(C)C(=O)NCC(O)C CCC(C)(Cc1cn(-c2ccc(CC3CCC3)cc2)nn1)C(=O)O CS(=O)C1CCCC(NC(N2CC(c3ccc(F)c(F)c3)C2)=O)C1 n1(CC)c(C(=O)NC(C(=O)NCC(F)C(C)(C)O)C(C)C)cnc1O N1(C(CC(CCC)C)=O)C2CCC1CC(CCNC(C1CC(C(F)(F)F)C1)=O)C2 C1(OC)(OC)CCSCC1NC(C1CCC2CC12)=O C1(NC(CN(C)CC)=O)CC=C(C(=O)OC)C1 N1(C(C(CC=C)(C)C)=O)CCN(C(=O)Cn2nnnc2C)CC(C)(C)C1 c1(C(=O)NCCOCCN(C)C(c2nsnc2O)=O)cc2cccn2c(O)n1 CC(CC(F)F)C(=O)N1CCN(C(=O)COCCF)C(c2cn[nH]c2)C1 N1(C(c2c(Cl)cnc(C)n2)=O)CCC2(CC1)CC(NC(C1CCCCC1C)=O)C2 c1(N2CCC(C(C)NC(COC3CCOC3=O)=O)C2)ccc(OCCO)cc1 C1(C(=O)NC2C(C(=O)NCC(C)(C)O)COCC2)Cc2ccccc2C1 C(=O)(C(C)C(F)(F)C(F)F)NCCCN(C(C12CC1COC2(C)C)=O)CC C1(C=O)CN(CP(C)(C)=O)C1.C(CC(C)(C)C)NC(CNC(=O)OC)=O c1(C(N2C(C)CCC(NC(c3ccncc3)=O)C2)=O)cccc2cnnn12 C1(CCC)CCCN(C(C2(NC(=O)CCOCCOC)CCSC2)=O)C1 O=C(CC1=CCCCC1)NC1CN(C(C2(CC(F)F)CCC2)=O)CCC1CO C1(CNC(=O)CCc2nccs2)CCC(O)C1.c1(C=O)ccc(C2CC2)cc1.N Cc1ccc(C(C)C(=O)NC2CC2CNC(c2coc(C3CCC3)n2)=O)o1 c1(C(N(CCCNC(=O)CSCCOC)CC)=O)ccc(Cl)o1 N1(C(COCC)=O)CCCC12CCCN(C(c1c(C)nn(C)c1C(F)(F)F)=O)C2 c1(C(=O)OC)cccc(NC(C2(F)CN(C(=O)C(O)C(C)C)C2)=O)n1 c1(OC)cc(C(=O)NCC2CC(NC(=O)C(C)C(C)(C)C)C2)cc(Cl)c1 CC1(C)COC(CC(=O)NC(C)(C(=O)NCCCC2CCOCC2)C2CCC2)C1 C(C(C)(C)CCNC(=O)C(C)C1CCCO1)NC(c1c(C)occ1)=O C(=O)(CC(F)(F)Cl)NCCC1(NC(c2cn(CC)nn2)=O)CC1 N1(C(c2scc(CC)c2)C(=O)NCC(F)F)CCC2(CC1)CC(=O)NC(=O)C2 N1(CC)C(=O)CCC1CC(=O)N.C1CN(C(C23CC(C#N)(C2)C3)=O)CCO1 c1(C(=O)N)cnc2ccoc2c1.C(C)(CCC)NC(COCCOCC#C)=O CC(O)(C(=O)NC1CC(NC(=O)CC2CC=CCC2)C1)C1CCC1 N1(C(CCS(C)=O)=O)CCN(C(=O)Cc2cccnc2)CC1C(F)F c1(C(N2C3C(NC(CCC(CC)OC)=O)C(C3)C2)=O)cc(C)[nH]c(=NC)n1 Cc1cccc(OCC(N2CCN(C(c3csc(CO)n3)=O)CC2CO)=O)c1F c1(OC)cccc(CC(=O)NC2CC(CCNC(C3(C)CSC3)=O)C2)c1 C1(NC(C2CCCCN2C(c2ncccn2)=O)=O)CCCCCC1O c1(C(=O)NC2C(C)(C)N(C(=O)C#CC3CC3)CC2)cc2cccc(F)c2s1 N1(C(COC(CNC(CC2CC(=C)C2)=O)(C)C)=O)CC(C)CCC12CC2 C(=O)(C1=CC2C=CC(C1)C2)N(CCCC(C)(C)C)C.c1(C(=O)N)cc(N)ccn1 c1(C=O)c(C(F)F)nc2ccccn12.C1(CC)(OC)CN(C(=O)C(C)C#N)C1.N C1(CNC(CCN(C)CC)=O)CC2(CC2)CN1C(C1CCCC12CCC2)=O C1(COC)CN(C(C23CC(OC)(C2)C3)=O)CCN1C(c1nc(C)ccc1C)=O c1(N(C)CC2CCCN2C(c2cccc(N(C)C)c2)=O)ccc([N+](=O)[O-])c(O)n1 c1(CCCC(=O)NCC2(NC(C3C4CC4C4CC34)=O)CCCC2)ccccc1Cl c1(-c2cn(CC3CCN(C(c4c(CC)noc4)=O)C3)nn2)ccccc1C(=O)O C1(NC(C(c2ccncc2)C)=O)CCN(C(C2CCS(=O)(=O)N2)=O)C(C)C1 c1(C(=O)NCC2(F)CCN(C(C3(C)CCC3)=O)C2)c(C(F)(F)F)cccc1F Cc1nccn1CCC(=O)NC1C(C(=O)NCCCC(C)C)C1(C)C Cc1ccnc(O)c1C(N1CCN(C(=O)CC2(C)CC2)C(c2ccccn2)C1)=O C1(C)(CNC(CN(C(C)=O)C)=O)CN(C(=O)CC2CC2(C)C)CCO1 Cc1snnc1C(=O)NOCC(=O)NCC1CCOC1=O N1(C(CCCn2ncc(C)c2)=O)CC(O)CC1CNC(=O)Cc1cncnc1 C1(C(C(=O)N(C(CNC(c2ccns2)=O)C2CC2)C)O)CCOCC1 N1(CC2N(C(C)C)CCC2)CCC2C(C(F)(F)F)C12 C1(C(=O)Nc2c(C(N)=O)cccc2)CC12CCN(C(c1cnc(O)c(Cl)c1)=O)C2 c1(CCC(=O)N(C2CCCC2)CCNC(C2CC2F)=O)cnc(O)[nH]1 c1(CNC(C2CC3(CC(NC(C=CC)=O)C3)C2)=O)oc2ccccc2c1C C1(CN(C(=O)CCNC(=O)Cc2cn[nH]c2)C)CCC(=O)N1 c1(C(N2CC(F)CC(NC(=O)CCC3CC3)C2)=O)cccn2cnnc12 CCCCCCC(C)CC(=O)NCC(C)(C)CNC(=O)CCOCC C1(CCC(N2CC(O)(c3cc[nH]n3)C2)=O)CCCN(C(c2csc(Cl)n2)=O)C1 c1(C=O)cnn(CCN)c1.C(=O)(C(O)CN1CCCC1)N(CC(C)O)CC c1(NC(C23CC(NC(c4c(C)nc(Br)s4)=O)(C2)C3)=O)ccc2ccoc2c1 CCCC(C(=O)NCc1ncccc1C)NC(N)=O.c1(C=O)nccnc1N.N N1(C(C(C)(C)SC(F)(F)F)=O)CCN(C(=O)CC2CCOC2)CC12CCC2 c1(OCC)ccc(S(=O)(=O)N(C)CCc2ccccc2OC)c(C#N)c1 N1(C(CC)=O)CCC(C(C)C(=O)NCC2(C)CC(C)=NO2)CC1 c1(C(=O)NCC(=O)NC(c2cccc(Cl)c2)CC)cccc(Cl)c1 c1(CC)ccc(N)c(C(=O)NC(C)CCNC(C2OCCC2C)=O)c1 C1(COC)CCCC2(CC2)C1.C12CN(CC1)C(=O)N2.C(C)(C)C.C=O.C N1(C(c2c(CC(=O)OC)cccc2)=O)C2CCC1CN(C(=O)C(N)=O)CC2 O=C(C1Cc2ccccc21)NC1CCN(C(=O)C(c2ccc(Br)s2)=O)C1 CC1CCC(NC(=O)Cc2cccs2)CN1C(c1csc(C(F)F)c1)=O N1(CC(=O)NC2CN(C(CCC)=O)CC2N=[N+]=[N-])CCc2ccccc2C1=O N1(C(C2CCC(CC)N2C(c2cc(C)c(C)s2)=O)=O)CCCNC(=O)CC1 N1(C(C2(COC)CC=CC2)=O)CCCC(C2CCN(C(=O)C3=NOCC3)C2)C1 CCC(CNC(C1(C)CCCC1)=O)(CC)NC(C1CC2CCC1O2)=O c1(C(CC)C)ccccc1N(CC(C)(C)CN(C(=O)C(C)CC)C)C(=O)CCF CCC(CC)(CC)C(=O)N1CCC(OCC=CBr)C1 N1(C(c2nn(C(CC)C)c(C)c2)=O)CCOCC(CNC(=O)CCCF)C1 C(=O)(CC(C(C)C)NC(C1C2CCC(C2)C1C)=O)N1CCC(N(C)C)(CC)C1 C1(NC(C2(CNC(=O)Cc3cnoc3)CC(=C)C2)=O)CN2CCC1CC2 C1(C(=O)NC2CN(C(c3ccc(C(C)C)o3)=O)CC2C)CCC2CC2CC1 c1(C(N2CC(COC)(CNC(C3CC(C)CO3)=O)C2)=O)cnc(O)cc1 N1(C(C2OCCN(Cc3ccc(OC(C)C)c(Cl)c3)C2)=O)CCC2(CCCO2)C1 c1(OC)ccccc1CN=C(NCc1ccco1)NC1CCCC1(F)F c1(C(=O)NCC(C2CCCC2)NC(C2(C)CCOCC2)=O)ncnc2c1CCC2 C1(NC(C(CC2CC2)OC)=O)CCCC1(C)C.c1(C=O)cnc(C2CC2)[nH]1 CC12CCC(C(N3CCCC3CNC(C3COCCC3(F)F)=O)=O)(C1)OC2 N1(C(C2NC(=O)OC2)=O)CCC2(CC(C(N3CC(CO)C3)=O)C2)C1 N1(C(c2c(C)oc(Cl)n2)=O)CCCCC(CNC(=O)CN2CCC(O)CC2)C1 C1(C(=O)NC2(CF)CCN(C(c3ccncc3F)=O)C2)CCCC1C1CC1 Cc1cccc(F)c1CC(=O)NC(C)CN(C)C(c1ccc(-c2cc[nH]n2)s1)=O N1(C(c2cc(OCC)ncc2)=O)CCCC(C)(NC(c2cnc(CC)cn2)=O)C1 C1(CC(=O)NC2CCN(C(C)C)C2)CCC(NC(C2(F)CCOC2)=O)CC1 C1(NC(C2(OCC)CCCCC2)=O)Cc2ccccc2C1NC(c1cnco1)=O C(=O)(C(C)(C)CCCNC(c1nc(=N)cc[nH]1)=O)NC(C1CCOC1)C c1(C(=O)NC2(CF)CCN(C(C3(C#N)CCCO3)=O)C2)c[nH]c2cccnc12 C#CC(C)(C)C(=O)N(CC(C)(C)NC(c1cc(CO)ccn1)=O)C C1(COC)(NC(=O)CCc2cnn(C)c2)CCN(C(C2CCSC2)=O)CC1 C1(CNC(c2cc(C)nc(O)n2)=O)CC2(CCOCC2)CN1C(C1CC12CC2)=O C1(NC(CC(C)CF)=O)CN(C(c2ccc(F)c(O)c2)=O)CC2(CC2)C1 c1(C(N(CCCNC(C(C=C)(F)F)=O)CCO)=O)cc(OC)ccc1C C(=O)(CCCCCC(C)(C)C)NCC1(NC(C(=COCC)C#N)=O)CC1 CC(=O)CCCC(=O)NC1CN(C(c2cc(Cl)c(Br)[nH]2)=O)CC1(C)C C1(NC(CSCC=C)=O)CC2CCC1CN(C(=O)C(CC)SC)C2 N1(C(c2c(OC)ncc(C)c2)=O)CCC2(CCC2)C1.C(=O)(C(F)(F)C1CC1)N c1(NC(C2C=CCN2C(=O)Cc2ccc(O)cn2)=O)cnn2ccccc12 C1(C(C(=O)NCCC#N)NCCCNS(C)(=O)=O)CC12CCOC2 C1(NC(C(=O)Nc2c(C(=O)OC)sc(Br)c2)=O)C(C)CCCC1C Brc1ccsc1CNC(c1ncc(C(F)F)s1)c1nnnn1CC1CCOCC1 C1(CN2C(COC)C=CC2)C(F)(F)C12CC2 c1(OC)cc(C)cc(C(=O)NCC(C)(C)NC(=O)C(c2ccc(Cl)s2)C)c1O c1(C(CNC(C(CO)OC)=O)NC(=O)Cc2cnn(C)c2)ccccc1F C(=O)(C1=CC(C)(C)C1)N(CCC(C(C)C)NC(=O)CC(C(F)F)n1cccn1)C N1(C(C(CO)NC(N)=O)=O)CCC(NC(=O)CNC=O)C2(CCC2)C1 C(C(C)C(=O)N1CCCC1C(=O)NCCCC1CC1C)OC(C)=O C1(CNC(C2CCC(=C)CC2)=O)CCCCN(C(c2cc(C)cc(C)n2)=O)CC1 CC1CC(NC(=O)C(C)(Cl)Cl)CN1C(=O)C(F)=CC1CC1 Cc1csc2c(C(N3CCC(F)C(NC(=O)CS(C)(=O)=O)C3)=O)ncnc12 c1(C(=O)NC(C(C)NC(=O)CCOCC2CCC2)C)cncc2nc[nH]c12 N1(C(C=CCOC)=O)CC2CCCN(C(C3CCc4[nH]nc(O)c4C3)=O)C2C1 c1(OC)cccc(CN2CCSC(C(=O)NCc3csc(C)n3)C2)c1F C(=O)C(C)C(F)(F)F.Cc1cc(C(=O)NCC(=O)NC)n(C)n1.C1CC1 c1(C(N2C(CNC(CC(C=C)(C)C)=O)CCC2)=O)cc(F)c(Cl)cc1F Cc1cc(C(F)F)n(CC(=O)NC)n1.C1(C=O)CCCC(O)C1.C1(CC)CC1 C1(C2(NC(C3CCOC3)(C)C)CC2)CCOC1 C1(C(N2CCC(N(C(=O)CCOC3CCOC3)C)CC2)=O)(SC)CCOCC1 C1(O)(C(=O)NCC2(NC(C3CCN(C)CC3)=O)CCCC2)Cc2ccccc2C1 C1(C=O)CCC(F)(F)C1.C1CN(C(C2CC(N3CC(O)C3)C2)=O)C1.CCO C=CC(F)(F)C(=O)NCC1C=CC(NC(=O)CCc2nc(C)cs2)C1 N1(C(c2c[nH]c(=N)s2)=O)CCCC2(NC(c3ccsc3Cl)=O)CCCC12 Cc1ccc(CC(=O)NCC(CO)NC(=O)C(C)Sc2ncccn2)cc1 C1(CNC(CC=C(C)C)=O)CCCN(C(c2csnc2-c2ccccc2)=O)C1 c1(C(=O)NCC2N(C(C=C(C)C)=O)CC=C2)ccc2c(O)n[nH]c2c1 C(=O)(CCN=[N+]=[N-])NCC1C(C(=O)NCc2n(C)ncc2)CCC1 C(C)(CCC(=O)N1CCC(OCCNC(c2c[nH]cc2C2CC2)=O)CC1)OC C1(OC)CCCCN(CC(=O)N(C2CCN(C(c3[nH]c(C)cc3C)=O)C2)C)C1=O c1(C(=O)NC(CCCC)CNC(C2(C(C)(C)O)CC2)=O)ccc(SC)cc1Cl N#Cc1ccc(C2=CCN(C(=O)NC3CCn4nnnc4C3)CC2)cc1 C#CC1CCCCN1C(C1CC(C)(NC(=O)C(O)C(C)C)C1)=O c1(C(=O)NCC(CC=C)NC(c2coc(Br)c2)=O)nn(C)c(Cl)c1Cl C1(C(N2CC(C)(C(=O)OC)C2)=O)CC(O)C(O)CC1C.C(=O)(C(C)O)N C(=O)(CCCC)OC.C(=O)C(C1CC1)N(C(=O)CC1(N(C)C)CC1)C.N Cn1ncc2c1CCC(C(=O)NC1CN(C(c3ccc(F)cc3)=O)CC3CC13)C2 Cc1cccc(C(=O)N(C)CC2(NC(C3CCC(=O)O3)=O)CC2)n1 C1(C#N)(CC(=O)NC2CN(C(c3cc(C)n(C)n3)=O)CC2C)CCCCC1 Cc1cc(C#N)ccc1-c1cccnc1C(=O)NCC(c1cccc(O)c1)O N1(C(C(C(C)C)C2CCC2)=O)CCC2(CC1)CC2NC(C1(Cl)CC1(F)F)=O Cc1sc(C(N2CCC(C(F)F)(C)C2)=O)nc1O.C1(CC(=O)N)CCN(C)CC1 Cc1c(CNCC[Si](C)(C)C)ccc(F)c1F CCC(CC(=O)N1CC(OC)CC1C)C(C)(C)C.C(=O)(C(C)(C)C)N.C(C)C C12(NC(=O)C=C3CCCC3)CCN(C(c3[nH]nnc3C3CC3)=O)CCC1C2 C1(C(N2CC(C#C)(F)C2)=O)CC2CCCC2N1C(=O)Cn1nnc(C)n1 Cc1cc(=NCC(CNC(c2coc(C(F)F)c2)=O)C(F)(F)F)[nH]c(CO)n1 C1(C(=O)NCC(CSC)OC)CCOC1CNC(c1nnsc1C)=O C(=O)(C1=NOC(C)C1)N1CC(CC(C(=O)Nc2cnc(CCC)nc2)F)C1 C12(CNC(=O)C(F)n3ccnc3)CC1CN(C(=O)Cc1ccc(Br)cc1)C2 CC(=O)CCCC(=O)N1CC(CCCCNC(c2ccccc2OC2CC2)=O)C1 N1(C(CCC=C)=O)CCCC1C1CCCCN1C(c1cnc(O)n(C)c1=O)=O CC(CC(=O)NC(C1CCCN1C(=O)Cc1ccc(O)c(F)c1)C)CC(F)(F)F N1(C(C2CCN(C(c3nc(C)sc3C)=O)C2)=O)CCC(CC2CC2)C12CCC2 Cc1occc1C(=O)NCCC(C)(C)NC(c1cn(CCCC#N)nn1)=O c1(C(=O)NCC2(NC(C(CC)N(C)C)=O)CCC2)ccc(CCF)cc1 CC1OCCC1(C)C(N1CCCCC1c1ccc(-n2cc(CO)nn2)cc1)=O C1(CNC(C2CCCCC2(F)F)=O)CC2(CC2)CN1C(C1(CCF)CC1)=O C#Cc1cc(NC(C2(F)CN(C(=O)Cc3cn(CC)nn3)C2)=O)cc(F)c1 c1(C(C)=O)cccc(C(N2CC3(NC(C4CCOCC4(C)C)=O)CC2C3)=O)c1O CC1(C)CN(C(=O)CCc2ccncc2)CC1NC(c1cc(C(F)F)cs1)=O C1CCN(C(=O)CN(C)C=O)C12CCC2.c1(CC)occ(C)c1C(=O)N.C C1(OC)CCCCC1n1cc(C(C)N(C(=O)Cc2cnn(C(C)(C)C)c2)C)nn1 C(=O)(CC(C)C(C)C(C)C)N1C2CN(C(CS(=O)(=O)N(CC)C)=O)C(CC2)C1 CCCC(C)(O)CNC(=O)C(CSCC)NC(c1cc(Cl)no1)=O c1(-c2cn(CC(CNC(=O)Cc3ccc(O)nc3)OC)nn2)cnn(C)c1.S c1(OC)nc(-c2cn(CC(=O)NCC3CC(c4cccc(F)c4)C3)nn2)sc1C Cc1cccnc1C(C(C)C)NCc1cnc(N2CCCC2)s1 c1(N2CCCC(C(F)(F)F)CC2)nc(=NCc2cnn[nH]2)[nH]c2c1COCC2 c1(CC(=O)NCC2(O)CN(C(c3ccc(F)cc3)=O)C2)c(F)cncc1Cl N1(C(c2cc(C#N)no2)=O)CC2CCC1CN2C(=O)C=CCO c1(C(=O)NC(C2CCN(C(CCc3ccc(C)o3)=O)C2)C)ccnc(S)c1 CC(C)CCCN(C)C(C1CC(C(C)O)C1)=O.C(=O)(C(C)CC1CCCCC1)N C(=O)(C(C)C(F)F)NCC(CNC(CN(C)CC)=O)(C)O C(=O)(C#CC(C)(C)C)N1CCCC(C=O)C1.C1(CC=C)(C(=O)NCC)CC1 C1(CN(C(=O)CC2CCC(=O)NC2)C)CCCCN1C(=O)CCc1cscn1 C=CC(C)(C)CC(=O)N(C)CCN(C(=O)Cn1nc(C)cc1N)C C(C(C)(C(=O)NC(C1CCN(C(=O)CC)CC1)C)OC)OC.C1(C=O)CCC1 N1(C(CCCC)=O)CCC2(C1)CN(C(=O)C(c1ccccc1Br)O)C2 c1(C(=O)NCCCN(C(C2CCC(C)O2)=O)C)cc([N+](=O)[O-])ccc1Br c1(C2(C(=O)NC3(CNC(C=CC(C)C)=O)CCC3)CC2)ccccn1 C(C(=O)NC(C)CC1CCCCC1)(C(C)(C)O)NC(c1c(C)cco1)=O c1(C(N(CC)CCC)=O)cc(Cl)ccc1Cl.c1(OCC#C)cccc(C=O)c1.N N1(CCC(C)C(F)F)CCc2nc(O)[nH]c2C1 Cc1cncc(=NC(=O)C(=O)NCC2CCN3CCCC3C2)[nH]1 c1(C(N2CCC(CN(C(=O)CC3CC3)C)C2)=O)cc2c(o1)CCCNC2=O.C CC(C)CC(O)CC(=O)NCC(F)(C(=O)NCc1cncc(O)c1)C(C)C C1(F)(C(=O)OCC)CN(Cc2nnc3c(=O)n(C)ccn23)CC12CNC2 N1(C(C(CCN(C)C)NC(C(=O)NC(C)C)=O)=O)CCCC2OCCC12 CC(CC(=O)N(CCC(C)O)C)C(C)(C)NC(=O)C=Cc1nccs1 n1(CCOCC)c(NC(C2(C(=O)OC)CC3CCC23)=O)cc2ccccc12 CCCCCCC(C)(CCC)C(=O)NC1CCN(C(=O)CCCN(C)N=O)CC1 C1CC(C(=O)N)C12CCC2.Cc1onc(Cl)c1.C(=O)C=CC(=O)N(C)C.C N1(C(C2CCCC(C)C2)=O)CCC2(NC(c3cnc4occc4c3)=O)CCCC12 CCC(c1cccc(Cl)c1)=CC(N1CCCC(CNC(c2ccc[nH]2)=O)C1)=O c1(C(=O)NC2CC(N(C(Cc3cc(C)[nH]n3)=O)C)C2)cc(C2CC2)nnc1O n1(CC(=O)NC2CC(CNC(C(CC=C)(C)C)=O)C2)nnc2ccccc2c1=O c1(C(=O)NC2C(SC)CN(C(c3ccc[nH]3)=O)C2)cc(C)cc(C)c1.CCO.O C(=O)(CC1=NN(C)C(=O)C1)N1C(C(=O)NC2(C#C)CC2)CCC(O)C1 C1(c2n(CCCOC)nnn2)(NC2C=CCCCC2)CCC2(CN(C(C)C)C2)C1 C1(CNC(=O)NC(CS(C)=O)c2nc(-c3nc[nH]n3)no2)CCSC1(C)C C1(C(=O)NC2C(NC(=O)Cc3sc(O)nc3O)CCC2)CCn2ccnc2C1 c1(CC)sccc1C(=O)NCCOCCOCCN C12(NC(CCn3nc(C)c(Br)c3)=O)CCN(C(c3ccncc3N)=O)CC1C2 c1(C(=O)NCC2CN(C(C3CCCC(C)(C)CC3)=O)C2)ccc2ccncc2n1 C(=O)(CCCCCCCCCO)N(CCCCCC)CCNC(=O)C(C)(C)F Cc1cc(C)c(C(N2CCCCC(NC(C3(F)CCCC3)=O)CC2)=O)c(O)n1 C1(NC(N2CCCC(C(c3n(C)ccn3)O)C2)=O)CCc2c[nH]nc2C1 c1(C(=O)NCCCc2n(C)cnn2)c(CNC(C2CCC(F)C2)=O)cnn1C C(=O)(C1=C(CCl)N(c2ccc(F)cc2)C(=S)NC1c1cccc(SC)c1)OCC c1(C(N2CC(OCCC(=O)NC3CN(C(C)=O)C3)C2)=O)snnc1C O=C(C(O)CCNC(C1C2CCCCC12)=O)NCCC1(O)CCCC1 N1(C(C2CC(C)C2)=O)CCC2(CCCN2C(=O)C=Cc2ccccc2)C1 C1(CNC(C2C(c3ccc(F)cc3)(C)C2)=O)CCCCC12CC2(F)F N1(C(C)C)CC(NC(=O)CC(CNC(c2c(Cl)cnn2C)=O)C2CCC2)CC1=O C1(NC(C(C)(C)NC(C)=O)=O)CN(Cc2cc(Br)ncc2Br)CC1C#N CC1CCN(C(C2CCCC2)=O)C1CNC(c1c[nH]nc1-c1cccnc1)=O Cc1c(C=CC(=O)N(CC(O)CNC(C2CC23CCC3)=O)C)cnn1C N1(C(N)=O)CCC(N(C(=O)C)C)C1.C12(CC1)C(=O)N2.C1(C=O)CCC1 c1(CCC(C)NC(c2cc(OCc3ccccc3)ccn2)=O)cccc(Br)c1 N1(C(C(c2n(C)ncc2)O)=O)CCCC(C)(NC(=O)C=Cc2cccs2)C1 c1(C(N2C(CNC(c3c(C)cco3)=O)CC3(CC3)C2)=O)cnn2c1OCCC2 Cc1ccc(C(=O)NCC2(NC(=O)CSC3CCCCC3)CC2)cc1C O=C(CCC1(NC(=O)CSC(F)(F)F)CCC1)NCCc1nncs1 CCCCC(C)(F)C(=O)N(CCNC(c1c[nH]nc1C(F)(F)F)=O)C1CC1 N1(C(Cc2nnc(C)s2)=O)CCCC(C(C)NC(c2cc(C)n(C(C)C)n2)=O)C1 c1(CC)ccc(=NCCN=C(NCC(CC)(CC)C(F)(F)F)NC2CC2C)[nH]c1 C1(C)(CCC)CCN(C(=O)COC2CCN(C(C3(C)CCC(=O)C3)=O)C2)C1 C1(NC(c2cc(C)nn2C)=O)CC2CCC(C1)N2Cc1cc(C)on1 c1(C(=O)NCC(CC=C)NC(C2(F)CC=CCC2)=O)cccc2c1cnn2C c1(OC)ccc([N+](=O)[O-])c(NCC(C)NC(c2ncnc3ccsc23)=O)c1F CCC1=NOC(CC(=O)NC2CC(C(C)NC(=O)CP(C)(C)=O)C2)C1 CC(CCC(=O)NC1CC(C(F)(F)F)C1)NC(c1nonc1N)=O c1(NCC2(O)CC(C(=O)OC)C2)ccc2c(c1)OCC(F)(F)C(F)(F)CO2 c1(NC(C(CCCC)NC(c2sc(O)nc2C)=O)=O)cc(C)cc(C#N)c1 C1(NC(CC(CC)(F)F)=O)COC2C(NC(=O)C(Cl)=CCl)COC12 Cc1sc(C)c(C(=O)NCCNC(=O)CC)c1C.C1CC1.C(=O)C1CC1 c1(NC(C(CCC(N)=O)Nc2c(OC)nccc2)=O)ccc(F)c2ccccc12 Cc1cc2n[nH]cc2cc1-c1ccc(NC(c2csnn2)=O)cc1F c1(C(=O)NCC2(O)CN(C(Cc3c(C)n[nH]c3C)=O)C2)cnc2c(ccn2C)c1 C1(C(=O)NC(COC)C(C)C)C2CN(C(=O)Cc3ccsc3)CC12 C1(CC)C(=O)NCCCN1C(C1C(C)C1(C)C)=O.C1(CC=O)COCCOC1.N Cc1c(C(N2CC(CCNC(=O)Cn3cccn3)C(C)C2)=O)[nH]c2ccccc12 C1(CCOC)CN(C(=O)C(O)CN2CCCC2)CCN1C(c1cncc(N)n1)=O c1(C(=O)NC(CC)C)cnc2ncc(-c3ccc(C#N)cc3OC)cn12 c1(CCC(=O)N(CC(C)(C)NC(C(C)C2CC2)=O)C)ccc(Cl)nc1 c1(C(=O)OC)ccncc1NC(=O)C(c1ccc(Br)cc1)N C12(C(N3CC(C)(C)C(CN)C3)=O)CCCCN1S(=O)(=O)CC2 c1(C(N2CCCC(C)(NC(C3CCCS3)=O)C2)=O)ccnc(S(N)(=O)=O)c1 c1(C(=O)NCC(CCCC)NC(=O)CC=C(C)C)ccc(C(C)=O)nc1O N1(C(C(CC)(C)OC)=O)CC2(C)CC1(C(=O)NCc1nc(C3CC3)n[nH]1)C2 C1(C(N(C(C)C(N2CC(F)C2)=O)CCC)=O)CCCOC1 S(=O)(=O)(c1ccc(Br)cn1)NC1CCCN(C(c2scc(C)n2)=O)C1 c1(-c2n(CCNC)ccn2)ccnc(-c2ccc(F)cn2)c1 c1(C(=O)NC2CCC(CNC(CC3CC(N(C)C)C3)=O)C2)ccc(Cl)cc1Cl C1(COC(C23CCCN(CCC2)C3)=O)CCC2(CCCCCCC2)O1 C#Cc1ccc(F)c(C(=O)NCC(CC(C)C)NC(=O)C(Cl)=CCl)c1 O=C(CC1CCOc2ccccc21)NCC#CCNC(C1C2CCCC12)=O C(=O)(C1=C(Cl)CCOC1)N(CC(=O)NCCn1cccnc1=O)C1CC1 n1(C(C)C)cnc(C=O)c1.c1(CC(=O)N(C2CCC2)C)cc(C(F)(F)F)co1 C1(C(=O)NCC(C2CC2)NC(Cc2c(C)cccc2)=O)CCn2c(O)nnc2C1 C(CCSC)(C=O)OC.C1(C)(CC=O)CCN(C(N2CCCC2)=O)C1.CC.N C(=O)(C1=CCCC1(C)C)N1CC(CNC(CC(C=C)C)=O)OCCC1 N1(C(C=CC)=O)CCCC(C2CC2NC(c2cnn3ccncc23)=O)C1 c1(C(N2CCC(C(C)(C)NC(c3cccnc3)=O)C2)=O)cnc2c(n1)CCCC2 N1(C(CN(CC)CC)=O)CCC(N(C)C)CC1.c1(CCC(=O)N)ccn(C)c1 N1(C(c2c[nH]c(=NC)s2)=O)CCCC2(CNC(=O)CCC(C)(F)F)CCCC12 C=CCC(F)(F)C(=O)NC1CN(C(=O)C(C)CCCC)CC1n1cccn1 S(=O)(=O)(c1ccc2c(c1)OCO2)Nc1scc(C(=O)Nc2cncnc2Br)n1 c1(N2C(CN=c3nc(C(C)C)[nH]s3)CCCC2)ccnc2cc(C(=O)O)ccc12 C1(C(N(CCC(=O)OC)C)=O)CC(C)CN(C(c2cc(=O)n(C)cn2)=O)C1 C1(CNC(C2CCCN(C)C2)=O)CCN(C(C2CCSC2)=O)CC1C1CC1 N1(Cc2ccc(C)nc2)CCN(CC(=O)N(C)C)C(=O)C1 C12(C(=O)NC(CC(C)NC(=O)Cn3ccc(Br)n3)C)CCC(CC1)O2 N1(C(CC(CC)C)=O)CCCN(Cc2ccc(F)c(C)c2Cl)CC1C Cc1ccc(C=CC(=O)NCC2CCOC2)s1.c1ccc(Cl)nc1.C(=O)C.N CC1CSCC1N=c1ccnc(N2CCCc3c(cnn3C)C2)[nH]1 C(c1ccc(=N)[nH]c1C)=CC(N1CC(NC(c2c(CC)scn2)=O)C(O)C1)=O c1(NC(=O)NCC(=O)Nc2ccc3nc(O)oc3c2)nccc2cccnc12 C1(OC)C(NC(C2CC2CNC(C2C3COCC23)=O)=O)CC12CCC2 c1(C(=O)NCC2C(NC(=O)CC3CCCCCC3)CCC2)ccn2cccc2c1 c1(CC(=O)Nc2cncc(C(N3C(C)C(O)CCC3)=O)c2)c[nH]c2ccccc12 C1(CNC(CCCc2onc(CC)n2)=O)CN(C(c2ccsc2Cl)=O)CC1C c1(OC)ccc2c(N3CC=CC3)nc(=NCC(C)C(F)F)[nH]c2c1 C(CC(C(=O)NCCCC(=O)NC)NC(c1cccnc1OC)=O)=CC n1(CCCSCC)nnnc1C(c1ccccn1)NC(C)CC(N)=O N1(C(C2CC(C)(O)C2)=O)CCC(CO)C(NC(c2cc(C3CC3)ncn2)=O)C1 C(=O)(C(C)(C)CC(F)F)NCCOCCCNC(C(C(C)C)n1cnnn1)=O c1(-c2ccc(C(=O)NCc3cc(OC)nc(OC)c3)nc2)ccc2ocnc2c1 C(=O)C(S(C)(=O)=O)C1CC1.c1(OC)ccccc1C(=O)C(=O)N.CC(O)C C1(NC(C2CCCOCC2)=O)CN(C(C2(c3ccc(F)cn3)CC2)=O)CC1F C(=O)(C(F)(F)C(O)C(C)C)N1CCCC(O)(CCNC(C(C=C)(C)C)=O)C1 N1(C(c2ccn(C)n2)=O)Cc2occ(C(N3CCC(O)CC3C3CC3)=O)c2C1 C1(C(N2CC(C(=O)NC(C)CCCO)(CC)C2)=O)CCCC12CCC2 c1(C(N(CCC)CCNC(C2(F)CC2(F)F)=O)=O)ccc(Cl)cc1OC c1(C(N(C(C#C)C)C)=O)cc(C)n(-c2cccc(C)c2)c1C CC1=C(C(=O)NC(c2ccc(C)cc2)CNC(C2CC3(CC3)C2)=O)CCO1 c1(C(N2CC3(CCC3)C2)=O)cc(N2CCOCC2)cc(F)c1.C(C(=O)NC)SC N1(C(C(C)c2ccco2)=O)CCOC(CN(C)C(C2CS(=O)C2)=O)C1 C(=O)CC(C)CC(F)(F)F.N1(C(c2c(CC)non2)=O)CCCC(C)(C)C1C.N c1(C(N2CCC(CNC(C(C(CC)O)(C)C)=O)CC2)=O)ccc2nc(=N)[nH]n2c1 CCCCCCCC(=O)N1CC(C(N)=O)(CNC(C2(C)CCC(F)(F)CC2)=O)C1 CC(C)(C)C(O)C(=O)NC1CCN(C(c2cc(Br)cnc2F)=O)CC1 c1(SC)cccc(C(=O)NCC2CC3CC3N2C(=O)CC(C)C(C)C)c1Cl Cc1cc2[nH]c(=O)c(C(=O)NCC34CC3CN(C(=O)C(C)O)C4)cn2n1 c1(OCC)c(CNCC2CCC(C)(C)O2)cccc1Cl c1(Nc2c(-c3cn(C(C)C)nc3)cncc2)c(Oc2ccccc2)cccc1F C1(C(C)C)C(=O)N2CC=CC2(C)C(=O)N(C)C(C)C(=O)N1.CCO N1(CCC(C(F)(F)F)c2nc[nH]n2)CC2C3CCC(C3)C2C1 Cc1cc(NC(N2CC3(O)CC2C3)=O)c(C)cc1F c1(N2CCN(C)CC2)ncnc2c1ncn2C1CN(c2ccc(O)c(Br)c2)C1 C1CN(C(=O)C[SH](=O)=O)CCC12CCC2.C(C)(C(=O)N)=CC.C(C)(C)C.C N1(C(C(CC(C)C)O)=O)CC2CC(C1)CN(C(=O)C#CC1CCOCC1)C2 Cc1cc(C)n(CC(C)CNC(N2CCN(C(c3cnn(C)c3)=O)CC2)=O)n1 C1(O)CCC(C)(C)C1.c1(CC)oc(C(=O)NC2CCCC2CC(=O)N)cc1C C(CC1=CCOCC1)NC(=O)Nc1cnc2sccn12 N1(C(c2c(Cl)nc(OC)s2)=O)CC(CNC(c2cscn2)=O)C2(CC2)C1 c1(C(=O)NCC2CN(C(c3c(C)[nH]nc3C(C)C)=O)C2)ccc(N)c(F)c1F Clc1ccccc1-c1nc(CC2COC3CC2C3)n(Cc2ccsc2)n1 C1(C2CCCC2)(C(N(C2CCN(c3nnc(CCOC)s3)C2)C)=O)CCNC1=O c1(C(=O)NC2CC3CC2CN3C(c2csc(O)n2)=O)ccc(F)c2cccnc12 C1(NC(C2C(C)(C)C2)=O)CCCN(C(C2CC2F)=O)CC1 N1(CC(CC)(C)C)CCCC(C(F)(F)F)C1 C(=O)(C1=CCCOC1)NCC(C)(C)NC(C(C)Cc1cnco1)=O C1(NC(c2cn(CC)nc2)=O)CCC(C)N(C(C23CC(C#N)(C2)C3)=O)C1 Cc1nnc2ccc(C(N3CCC(CC(C)NC(=O)C(O)C4CC4)CC3)=O)cn12 c1(C(=O)Nc2cccc(CN)c2)ccc(-n2ccnc2)c([N+](=O)[O-])c1 Cc1ccc(F)c(C(N2CCOCC2CNC(c2sncc2Br)=O)=O)n1 c1(N(CCOCCOCC)C)nc2c(F)cccc2c(=NCCC(C)C(C)C)[nH]1 C1(NC(c2cc(OC)cc(OC)c2)=O)CN(C(C2CCCSC2)=O)C2(CCC2)C1 c1(CC(=O)NC2CCC(NC(c3coc(O)n3)=O)C2)coc2ccc(F)cc12 N1(C(C(C2CC(F)(F)C2)OC)=O)CC(Nc2nc(C)nc(C)c2F)CC(C)(C)C1 c1(C(=O)NCC2N(C(C=C(C)C)=O)CCCC2(C)C)nnc2ccccc2n1 c1(COC)cccc(C(=O)NCCCCN(C(=O)C(N2CCCCC2=O)C)C)n1 c1(C(N2CCCC(C3N(C(C=CC)=O)CCCC3)C2)=O)cnc2snc(C)c2c1 c1(C(=O)NC)c(F)ccc(CC)c1F.c1(OCC#C)ccc(C(=O)O)cc1C N1(C(C(CC)SC)=O)CC2CC(NC(c3ccc(OC)cc3Br)=O)C1C2 N1(C(CNC(C)=O)=O)CCC(CC(C)(C)C)C1.C(=O)(CC)N.[SH](C)(=O)=O C1(C(N2CC(N3CCN(C(C=CC(C)C)=O)CC3)C2)=O)CC1C1CCOCC1 C1(CC)(CC)CC(NC(c2nncs2)=O)CN1C(=O)CCC1CCCO1 C(C(CC)(CC)C(=O)N1CC(=O)N(C)C(=O)C1)NC(C(CCC)OC)=O C1(NC(Cc2c(C#C)cccc2)=O)COC2CN(C(=O)CC3C=CCCC3)CC12 C(=O)(C(O)CC(F)(F)F)N(CC(=O)NCC1CC2COCC2C1)CC#C Cc1cn2nc(C(=O)NC3CC3NC(C3CN4CCCN3CC4)=O)cc2c(=O)[nH]1 C(CCCCN=c1cccc(S(=O)(=O)N2CCC(N3CCN(C)CC3)C2)[nH]1)SC C1(CNC(=O)Cc2cnccc2Cl)CC2CN(C(=O)Cc3c(F)cccc3F)CC12 O=C(C1=Cc2ccccc2C1)NC1CCN(C(C2C=CCCC2)=O)CC1O C(=O)(CCCN(C)N=O)NCc1ccc(CNC(C(CC#C)O)=O)cc1F S(=O)(=O)(c1nc(N(C)CCN(C)CCO)ccc1Br)N1CC(CO)CC(C)C1 c1(C(N2C(C)CC(NC(c3cccc(F)n3)=O)CC2)=O)cc2c(F)cccc2s1 CC1(CNC(c2ccsc2C#N)=O)CCCN(C(=O)CC2(O)CCCCCC2)C1 c1(NC(COC(C2(C)COC2)=O)=O)nc2cc(C(F)(F)F)ccc2s1 c1(SCC)cccnc1C(=O)NC(CNC(c1ccc(CO)cc1)=O)CC C1(CNC(CCC(=C)C)=O)CCN(C(c2ncc(Br)cc2N)=O)CC1C CC(C)CC(C)CC(=O)NC1(CNC(=O)CC2(O)CCC2)CC1 N1(C(C2ON=C(CC)C2)=O)CC(C)CN(C(=O)C(C)CC2CCCCC2)C(C)C1 C(=O)(CCC(=O)c1ccc[nH]1)N1CC(C(C)NC(C2CC2)=O)C1.N(C)(C)C N1(C(C2N(C)CCOC2)=O)CCCN(C(=O)C(O)c2cnc[nH]2)CC1 C1(NS(CC)(=O)=O)CN(Cc2ccnc(-c3ccccc3)c2)CC1F C1(NC(c2cc(C)on2)=O)CC2CC1CC2C(=O)Nc1ccc(F)cc1F O=S(=O)(c1ccc(NCc2cccc(Cl)c2Cl)c(F)c1)NC1CCC2CC12 C1(CNC(c2c(CC)noc2)=O)CCN(C(=O)CCN2CCOCC2)C12CCC2 C1(NC(C2CC(CC)(CC)C2)=O)CCN(C(=O)CC(C)(C)C#N)CCC1CO N1(C(c2c(C)[nH]cc2)=O)CCN(C(C2CCC(C)(C)CO2)=O)C(C)C1 Cn1cc2cc(-c3cnccc3C(=O)NCc3ccncc3F)ccc2n1 N1(C(C(CCOC)OC)=O)CCC2(CC1)CCN(C(=O)C(C)C(F)F)CC2 c1(NC(c2cc(-c3c(F)ccc(OC)c3)ncc2)=O)cnc2cccnc2c1 N1(C(C(=O)NCC)=O)CCN(C(=O)C(C)CC(F)F)C(CS(C)(=O)=O)C1 c1(C=O)ccc2c(c1)OCCO2.C(=O)(C(C)C(=O)OC(C)(C)C)NCCCC N1(C(CC)=O)CC2CCOC2(CNC(C2CCC2(F)F)=O)C1 C12(NC(C(=O)NCC)=O)CCOCC1CN(C(=O)COc1cccnc1Cl)C2 O=C1NCc2cc(Br)cc(N3CCC4C3CC4(O)C(F)(F)F)c21 C1(C2CCN(C(CCC)=O)C2)CCCCN1C(c1cnn(C2CCCC2)c1)=O C1(OC)CCn2cc(C(=O)NCC3(NC(c4nonc4N)=O)CC3)nc2C1 N1(C(CC(C(C)(C)NC(CS(CC)=O)=O)C)=O)CC=C(C(C)(C)C)CC1 N1(C(C#C)=O)CCOCC1CNC(c1cccnc1-c1ccco1)=O c1(C(N2C(CC(=O)NCC(C(C)C)OC)CC2)=O)cncc(CO)c1 C1(CC(=O)N(C(C)C(=O)NCC(=O)N)CC)CC(C)=NO1.C1CCCC1 C(=O)(C1=CCN(C(=O)C2=C(Cl)CCC2)CC1)NC(CCC=C)C c1(OC)ccc(C(C)C(=O)N)c(C)c1.C1(C)CN(C(=O)C=CC=C(Cl)Cl)C1 N1(C(CCOCCC)=O)CCN(C(c2ccnnc2C)=O)CCC1C C12(C(N(CC(C)NC(c3ncnc(C)c3C)=O)C)=O)CCC(=O)N1CCS2 Cc1nc(C(N2C(C(=O)N(C)CC#N)CCC2C)=O)c(=O)[nH]c1C N1(C(c2c(C)nc(O)[nH]2)=O)CCCC(C2CC2NC(=O)C=Cc2ccco2)C1 C1(C(=O)NC2CCCN(Cc3ccccn3)C2)CCC2(CCC2)O1 C#CCCCCC(=O)NC1CCC(NC(C2CC23CCCC3)=O)C1 C1(NC(c2c(C)n[nH]c2)=O)CC2(C(=O)N(C(C)CC(C)C)C)COC1C2 C1(N(C)C(C2CC23CCC3)=O)CCCCN(C(=O)C=Cc2ccccc2)C1 N1(C(CCOCCCOC)=O)CC2(CC2)CC1C.c1(C=O)cc(C)cnc1F.N O=C1COc2cc(NC(N3CCc4c(ccc(Br)c4)C3)=O)ccc2N1 CC1CN(C(=O)C(c2cccn2C)=O)CC1(C)CNC(c1ncccc1Cl)=O C(C(C)(C)CS(=O)(=O)NCCC(CO)C(C)C)OC c1(NC)cnc(Cl)cc1C(=O)N.C1(F)CCCN(C(=O)C=C(C)C(C)C)C1 N1(C(C(C)C2CC2)C(=O)NCc2ccccc2)CCOC2(CCCS(=O)(=O)C2)C1 N1(C(C2C(C)C2C)=O)CCCCC12CC(NC(C1CCCCC13CCC3)=O)C2 c1(NC(C2CC(=C)CN2C(=O)CCc2ccnc(C)c2)=O)cc(C)c(C)c(Br)c1 CC1CN(C(c2ccc(F)cc2)=O)CCC1NC(=O)Cc1sccc1Br Cc1cccc(C(F)(F)C(=O)NC2CCC2NC(c2cncc(F)c2)=O)c1 c1(C(N2C(C)(CNC(=O)C(O)C(F)(F)F)CCC2)=O)cnc2ccc(F)cc2c1 N1(C(CCC2CCN(C(C3N(C)CC(O)CC3)=O)C2)=O)CCCC2OCCC2C1 N1(C(c2sccc2Cl)C(=O)NC2CCN(C)CC2)CCCCCCCC1 c1(OC)cc(N2CCC(OCC(=O)OC=O)C2)c(I)cc1Cl.c1ccccc1 c1(Cn2cc(CNC=O)nn2)[nH]nc2ncccc12 CCCCCC(CC)C(=O)N1CCCCC1CCC(C)(C)NC(c1cnsc1)=O CCCCCCOCC(=O)N(C1CCCC1)CCCNC(=O)CC12CCCC1C2 N1(c2nc(C)cc(N3CCC(CC(=O)NC)CC3)n2)CCCC2(CC=CCC2)C1 n1(CC)nc(C2CC2)cc1C(=O)N.CCC(C)C.c1(C=O)ncoc1C(C)C c1(NC(c2cn(CCNC(C3C(C)=CCS3)=O)nn2)=O)cccc(NC=O)c1 N1(C(c2c(CC)n[nH]c2)C(=O)NCCOC)CCSC(C(F)(F)F)C1 N1(C(c2c(OC)scc2)=O)CC2CN(C(C3CCCC(=O)C3)=O)CC2C1 c1cnc(Cl)cc1C=O.c1cc(C2CC2)ncn1.C1(C(=O)OC)(C=O)CC1.N C(=O)(CC(CC)C(C)C)N(C1C(C)CCN(C(C=CC)=O)C1)C N1(C(CCOc2cc(NC(C3C(C)C3)=O)ncc2)=O)CCC(O)CC1C(=O)N c1(C(=O)NCC2CN(C(COC3CCCC(C)C3)=O)C2)c(O)ncc2c1CCC2 C1(C(N2CC(N(C(=O)CP(C)(C)=O)C)C2)=O)CC2(CCOCC2)CO1 CCC(C)(C)CCCC(=O)NC(C(=O)NCC(O)C(C)(C)O)C(C)C C1(C(N2CCCC(N(C)C(C3CCCOC3)=O)CC2)=O)CC(F)(F)CCC1(C)C N1(C(C(CN(C)C)O)=O)CCC2(C1)CN(C(C1CCN(S(C)(=O)=O)C1)=O)C2 c1(C(=O)NC(C(=O)NC(CC#C)C(=O)OC)c2ccco2)cc(C)nc(O)c1 Cc1cc(C#N)ccc1C(N1CCC(CC(=O)NCCCN(C)C)C1)=O c1(CC=O)ccc(F)cc1F.C1(C(N(CCOC)CC)=O)CC2(C)CC1CO2 c1(C(c2n(CCCSC)nnn2)NCc2cnn(C)c2C)ccc2scnc2c1 c1(C(=O)NCCC2CCCN(C(C3CC(=C)C3)=O)CC2)cccc2ncccc12 C(=O)(C1CCCc2scnc21)NCCN(CCC)C(C12CCC(C)(C1)OC2)=O C#Cc1cccc(C(=O)NC2CCC(CNC(=O)CC3C=CCCC3)C2)c1 C12(OC)CCCCC(C(=O)NCC3COCCN(C(c4cc[nH]n4)=O)C3)(C1)C2 Cc1cccc(C)c1C1CCN1c1sc(C2CCC2)nc1C C(C(N=[N+]=[N-])C(=O)NCC=CCC(=O)NC(CO)CCC1CC1)OCC CCC(C(=O)NCC(C)(C)CNC(=O)C=Cc1cncc(O)c1)C(C)O C1(CNC(C2C=CCCC2)=O)CN(C(=O)CCn2cnnn2)C2(CCC2)C1 c1(C(N2C3CCN(C(c4c(C)noc4C)=O)C3CC2)=O)cc(Br)cc2[nH]ccc12 c1(C(N2CCC(NC(=O)Cc3ccsn3)C(F)C2)=O)cncc2c[nH]nc12 N1(C(COCC(=C)C)=O)CCC(O)(CCNC(=O)C(O)CCC)C1 C12(NC(C3CC3c3ccccc3)=O)CCCN(C(c3cc(O)no3)=O)CC1C2 N1(C(C)=O)CCN(C(C2CC2CC(C)C)=O)C(c2ccncc2)C1.C(=O)(OC)N Cc1cc(NC(C2CSCC(=O)N2)=O)ccc1NC(C1CCCN1C(C)C)=O CC(=Cn1ccnn1)C(=O)N1CCC(CCNC(C2(C)CC(C)C2)=O)C1 N1(C(c2ccc(F)c(OC)c2F)=O)CCOC2CCN(C(=O)CC(C)C)CC12 N1(c2n(CC)c(C(C3CC(F)(F)C3)O)nn2)CCN(c2cccnc2)C(=O)C1 C1(O)(CC(=O)N(C(C(CC)C)C)CC)CCCCC1.C(c1ccco1)=CC=O c1(CN2CCC(C(N3CCC(c4ccccc4)CC3)=O)C2)ccc(O)cc1F c1(C(=O)NCCC(C)NC(C=CC=CC)=O)ccccn1.CC(F)F.O c1(CC(=O)OCC2C(C(C)C)C2)ccc2c(c1)OCCCO2 c1(C(=O)NC2CCN(C(c3ccoc3C(F)(F)F)=O)C2)c(Cl)nc2ccccn12 N1(CC)C2CCC(C2)C1C(F)(F)F.N1(C(=O)OC(C)(C)C)CCOC(C)C1 CCC(CC)C(C(=O)N1CCC=C(C(=O)NCC2(C)CCOC2)C1)OC Cc1nncc(CNC(=O)CC2(C)CCN(C(=O)CCC3CC3(C)C)C2)c1C C(=O)(CC(C)(O)C(F)(F)F)NC1(CCOC)CCN(C(=O)C(C)O)CC1 c1(Cn2c(C(=O)NC(C#CC(OCC)O)C)ncc2)ccc(C)c(F)c1.C N1(C(Cc2n(C)ccn2)=O)CCCN(C(=O)CC2COC(=O)C2)C(CO)C1 n1(CCOC)cc(C(=O)NC(C)C(CO)NC(=O)CC)cn1.C(C)=O.O C1(CC)CCOCCN1C(=O)C(C)N(C(C1CS(=O)C1)=O)C1CC1 C1(NC(c2ccc(OC)nc2)=O)CC2CCC(C1C)N2C(c1cnc(C)cn1)=O C1(c2n(CC)nnn2)(NC2COC(C3CC3)C2)CCN(Cc2ccccc2)CC1 c1(SC)cc2c(cc1CNCc1csnn1)OCCO2 Cn1cnc2sc(C(N3CC(NC(=O)CCCn4ccnc4)CC3CO)=O)cc12 c1(C(N2CCC(Cc3cn(CCCCCO)nn3)CC2)=O)ccc(F)cc1 c1(C(N(CC(C)O)CC)=O)ccc2cncn2c1.C1(CC(F)F)(C=O)CCC1.N N1(C(C2(CC)CC2)=O)CCOC(CNC(=O)COCC2(F)CC2)C1 c1(NC(CN(C(C)C)C(C2CC3CCC2C3)=O)=O)cn(C)c(=O)nc1O c1(C(C)OC)nc(-c2nc(O)sc2C)n(-c2cnc(C)s2)n1 N1(C(CCC(=O)NCC)=O)CCC(NC(c2cn(C)cn2)=O)CC(O)C1 c1(N2CC(CCOC)(C(N3CC(C(=O)OC)C3)=O)C2)ccnc(CO)n1 c1(C(=O)NC(C)CN(C(=O)C2=C(Cl)CCCC2)C)cccc(S(N)(=O)=O)c1 c1(C(=O)NCC(CC)NC(c2[nH]nnc2C)=O)ccnc(C(F)(F)F)c1[N+](=O)[O-] CCCCC(O)CC(=O)NC(C)(C)CC=CC(N1CCOC(C)CC1)=O C1(CC)CCCCC1C(=O)N(CC(C)(C)Nc1cc(C(F)F)ncn1)C c1(CNC(=O)NC(C2(C)CC2(F)F)C)nc(-c2ccsc2)no1 N1(C(C(C(C)C)SCC)=O)CCCN(C(c2ccc(C)nc2C2CC2)=O)CC1 c1(OCC)ccc(Cl)c(C(=O)NC(C)(C)CC(C)C)n1.c1(C=O)c[nH]nc1C C1(C(N2CC(N(C)CC)C2)=O)CC2CC1CN(C(c1cc(C)nnc1O)=O)C2 c1(CC(=O)NC2CC(C)N(C(=O)COCC3CCC3)C2)ccc(F)cc1Cl C1(CC(=O)NCCC2CCN2C(=O)CC2CC2)CCCSC1 c1(COC)nc(-c2ccccc2COC)n(CCc2ccccc2)n1 c1(CC(=O)OCC(c2cc(C(=O)OC)no2)=O)ncn2c1COCC2 c1(OC)ccn2ncc(C(=O)NCC3(NC(c4coc(Cl)c4)=O)CC3)c2c1 C1(NS(CC2(S(C)(=O)=O)CC2)(=O)=O)CCCS(=O)(=O)C1 N1(C(C(CC(C)C)ONC(c2ccn(C)c2)=O)=O)CCC(C2(C)CC2)CC1 c1(OC)cc(CCNC(=O)N(C2CCCC2)C)ccc1O.C(C)(C)C.C=O.N C1(CCOC)CN(c2cc(NCCOC(=N)O)ncn2)CCO1 C1(CNC(C2(CC#C)CC2)=O)(CO)CCN(C(C2CSCCS2)=O)CC1 CC1CCC(CC(=O)N(C)CC2(O)CN(C(=O)Cc3ccsn3)C2)O1 N1(C(c2c(OC)c(Br)ccc2)=O)CCCCC(NC(=O)C(O)C2CC2)CC1 C(=O)(C1CCCc2nccn21)NCC(C)CNC(c1cncc2n[nH]cc12)=O CC1=C(C)CC(C)(C(=O)N(CC(O)CN(C)C(c2snnc2C)=O)C)CC1 C(=O)(CCS(C)(=O)=O)NC(CC(=O)NC(CC=CC)CO)(C)C N1(C(C2(C(=O)OCC)CC23CC3)=O)CC2(CCN(C(C3CC3)=O)CC2)C1 c1(C(N2CC(OC)C(NC(=O)C3=CCSC3)C2)=O)ccc([N+](=O)[O-])cc1F N1(C(c2cnc(CC)o2)=O)CCCC(N(C(=O)CCc2cc(C)n(C)n2)C)CC1 c1(OC)ccc(C(N2CC(N(C)C(c3cnc(O)n3C)=O)C2)=O)c(OC(F)F)c1 C(=O)(C(C)=Cn1ccnn1)N(C1CCC(NC(C(C(CC)CC)OC)=O)CC1)C C1(C(=O)NCC2CC(C)N(C(c3cnsc3)=O)C2)CC2CCC1CC2(F)F C(=O)(C1=CCC(C)(C)CC1)NC(C1CCCCC1)CNC(c1c(C)nccn1)=O N1(C(C(c2ccccc2)C)=O)CCOCC(C)(CNC(=O)CCC(C)N(C)C)C1 c1(C(N2CCC(C)CC2)=O)ccc2[nH]c(=N)oc2c1.C(CC)(C(=O)N)OCC.C CCCCC(=O)C(=O)NC1C2CN(C(C3CCC(CC)CC3)=O)CC12 N1(C(c2c(C)nc(Br)o2)=O)CCC2CCN(C(=O)C=CC(F)(F)F)C2C1 n1(CCC#N)ccc(=NC(=O)C(=O)N2CCN(c3ccccc3)C(CCO)C2)[nH]1 N1(C(c2c(CC)ncs2)=O)CCC(C(=O)Nc2cnn(CCO)c2)(CC)C1 Cc1c(CCNC(C2(C)CCCO2)=O)cnn1C.C(=O)(C(C)C1(O)CCC1)N C=CCC(CC(=O)NCCc1ncc[nH]1)NC(C1(O)CC1)=O c1(C(N2CC(NC(C3CC4(CCC4)CO3)=O)C(O)C2)=O)n[nH]c2ccc(F)cc12 c1(C(N(CC(CC)NC(=O)Cc2noc(C)c2C#N)C)=O)cnc2c(c1)COC2 CCC(O)C(C)C(=O)NCC1(NC(c2cc3scnc3[nH]2)=O)CC(F)(F)C1 CCC(C)CCCC(=O)N1CCN(C)C(CNC(=O)C(C)(C)c2cnn(C)c2)C1 C(=O)(C1=CCN(C(=O)C2=CCCOCC2)CC1)NCC(C)(C)n1ccnc1 c1(C(N2CCN(C(CCN(C(C)=O)C)=O)CC2CCO)=O)cncc2ccsc12 N1(C(C(C)(CO)NC(C(COC)OC)=O)=O)CCNC(=O)C1CCO C1(C(C)=O)CC(CC(N2CCC(C(C(F)F)Nc3ccncn3)CC2)=O)C1(C)C C(=O)(C(C)(F)CCCC)NCCCC(C)NC(CCCC(=C)C)=O CCCC(C(=O)N(C)CC1COCCN1c1nnc(C)s1)NC(N)=O c1(NC(=O)NCC2COCCC2(F)F)cc(Cl)c(Br)cn1 Cc1nocc1NC(c1ccc(I)s1)c1nnnn1CCN1CCOCC1 CN1CCN(C(c2ccc(C(N)=O)o2)=O)C(C(=O)NCCC(C)(C)F)C1 C(Cn1cccn1)(C(=O)N(C)OCC(F)(F)F)NC(c1c(C)cc(C)o1)=O C(=O)(N=c1cc(Cl)c(C#N)c[nH]1)C1(C)CN(Cc2ccc(-n3cccc3)cc2)C1 C(C(C(C)(C)C)NC(c1occc1C)=O)NC(C(C)SC)=O Cc1nc(=N)[nH]cc1C(N1CC(NC(=O)C(=O)NCC(F)(F)F)C2CC12)=O N1(C(C(C)=C(CC)C)=O)CC(C)(C)CC1C(N1CCC2(CCC2)C1)=O C12(C=O)C3CC(CC13)C2(F)F.Cc1cnccc1C(C)C(=O)NCC1CC1 c1(CNC(NCCOCC)=NCC)cccc2c1OCC2 C(=O)(C1=CCC(C)CC1)N(CCC(=O)NOC1CC2CCC1C2)C1CC1 c1(NC(C2C(CCC)CCC2)=O)ccc(NC(c2occ3c2CCC3)=O)cc1C C1(CC(N2CCC(c3nc[nH]n3)C2)=O)C2CCC(C2)N1C(C1CSC1)=O CC1(CNC(C2(N(C)C)CC2)=O)CCCC1NC(C1(O)CCSC1)=O C(=O)(C(C)(C)CCC#N)N(C(CNC(c1cc(CC)c(CC)o1)=O)C)C c1(OC)cccc2c1C(CNC(=O)NC1CCc3ncncc3C1)CC2 C1(OC)CN(C(=O)CCc2cc(C)no2)CCC1NC(=O)C1=CCOCC1 C1(C(=O)NCCC(=C)CNC(=O)C(F)=C(C)C2CC2)CCC(=O)NC1 c1(OC)ccc(CN2CC(O)(CNC(=O)C)C2)cn1.N1(C=O)CCOCC1 N1(C(C2OCCN(C(c3cccc(O)c3Cl)=O)C2)=O)CCc2cc(O)ccc2C1 Cc1cc(-n2cncn2)ccc1C(=O)NC1CCC(n2cc(C3CC3)nn2)C1 C(C(=O)NCCN1CCCCC1C)(C(C)(C)C)NC(C(CCC)N(C)C)=O N1(C(CC2C(C)(C)CC2)=O)C2CCC1CC(C)C2.c1(C(=O)N)ccc([N+](=O)[O-])o1 Cc1ccccc1S(=O)(=O)CC(=O)NCC1(O)CCC1.C(=O)C(C)N(C)C.C c1(C(=O)NC2CCN(C(c3c(CC)nn(C)c3)=O)C2C)cnc2ncnn2c1C c1(CC=O)cc(C)nn1C.c1(CC(=O)NCCCC)ccccc1.C(C)(=O)N N#CC1(CN2CCC(CCC3CCCNC3)CC2)CCS(=O)(=O)CC1 C1(C(N(CCCC)C)=O)CN(C(=O)C(C)c2cc[nH]n2)CC(C)O1 c1(C(=O)NC(C2CCCC2)C)cc(O)cc(=O)o1.C1(C2CC2)(C=O)CC1.N O=C(C1Cc2ccccc21)NCCN(CC(=O)NC1COCC1(F)F)CCF C1(NC(C(CCF)NC(CC(CC)CC)=O)=O)CCc2nn[nH]c2C1 c1(CN2CCN(C(CC(OC)OCC)=O)C3C2C3)cc(Br)c([N+](=O)[O-])s1 CC(C)C(CNC(C1(C)CC1(Cl)Cl)=O)NC(=O)Cn1cncn1 CC1(C)CCC(C(=O)N2CC(F)(CNC(=O)CCCC(N)=O)C2)c2ccccc21 C1(C)CCN(C(c2cn(C3CCCCC3)nn2)=O)C1.N1(CC)CCC1C(=O)N.C C(CCCC(C)NC(c1ccc(C(C)(C)CC)cc1)=O)NC(COCC)=O C(=O)(C(CC)CC(F)(F)F)NC(CCN(c1c(C(=O)OC)cccn1)C)C C1(C(N2C3CCCC2CC3)=O)CC2(CO1)CC(F)(F)C2.C(F)(C=O)=C(C)C.N C1(CNC(CC=CCC)=O)CCN(C(=O)C(C)C2CCC2)CC1C1CC1 c1(C(=O)NC(C2CCN(C(=O)CC3C=CCC3)C2)C)ccc2c(c1)CCCCN2 c1(C(=O)NC2CN(C(C34CCC(F)(CC3)CC4)=O)CC2F)cc2ccncc2[nH]1 N1(C(C(C(C)C)C)=O)CC2CCC(C1)N2C(c1cc2c(ccn2C)[nH]1)=O N1(C(C2CC(=O)OC2)=O)CCC2(CC1)CC(NC(=O)C1=CS(=O)(=O)CCC1)CO2 N1(CCC)CCC(CNC(=O)C(F)CC2CN(C(c3nccn3C)=O)C2)C1 c1(C(=O)NC2C(NC(C=CC(CC)C)=O)C2)cnn2c(C)c(C)ccc12 C(C(N=c1[nH]nc(C(C)C)o1)C(C)C)NC(C1(CC#C)CC=CCC1)=O n1(CC(CC)NC(=O)C(C(C)C)c2cnn(C)c2)cccc(C(=O)O)c1=O O=C(C(F)C1=CCCCC1)NC.C1C2CN(C(c3ccsc3C(F)(F)F)=O)CC12 C1(NC(CCC=CCC=C)=O)CCN(C(=O)C)C1(C)C.c1nccn1C(C)C.S C(C(C)(CO)NC(c1ccsc1SC)=O)NC(CC=CC=C)=O C(C(O)CC(F)(F)F)NC(COC1CN(C(C(C=C)(F)F)=O)C1)=O CC(C)(C)C(CC(=O)NCCC1CC(NC(c2ccns2)=O)C1)C(F)F c1ccc(C(=O)O)cc1Br.C1(C(=O)OC)CC(F)CN1C(C1CC12CNC2)=O.C c1(C(=O)NC2(c3c(C)cccc3)CC2)ccc(SC(F)F)c(F)c1 C1(CNC(=O)Cc2csc(S)n2)CCCC2(CN(C(C3CCC(F)C3)=O)C2)O1 CCC(O)C(F)(F)C(=O)N1CC2C(CNC(=O)C(F)(F)C3CC3)C2C1 N1(C(C2CCCN(CCC)C2)=O)CCCN(C(C2CC(F)C2)=O)CCC1 C(C(C)CC(=O)NC1CCCC1F)NC(CNC(CC(C)C)=O)=O C1(NC(C(CC)OC)=O)CCCN(C(=O)C(Cc2ccsc2)NC=O)C1C c1(C(=O)NCC(C)(C)OCCNC(C2CCOC2)=O)cc(Cl)ccc1O Cc1c(C(=O)N(CC(O)CN(C(=O)CSc2cnn(C)c2)C)C)ncn1C Cc1cc(C(=O)NC2(C(C)C)CC2)cc(Br)c1 C1(NC(C(=Cc2ccncc2)C)=O)CC12CCN(C(C1CC(O)C(F)C1)=O)CC2 C(CN=c1nc(O)c(Br)c[nH]1)C1N(N2CCCC2)CCC1.C(C(F)C=O)SCC=O C(=O)(C(C(C)NC(=O)CC(C)N(C)C)C(C)C)NCC=CCCOC CC1COCCCN1C(=O)C(C)(C)C(C)NC(=O)CCCN(C)C(C)C C1(C)(C(=O)NC(CC)C(N)=O)C=CCN1C(=O)CCn1cccn1 C(CO)(CN=c1[nH]c(N2CCC(F)(F)C(C)C2)nc2ccccc12)OC C(C)(CCC(=O)N1CCC(CCC(=O)NC2COC(=O)C2)C1)OC c1(OC)ccc(C)c(CN2CC(NC(=O)C(C)(CO)CO)C(F)C2)c1 c1(OC)ccc(F)c(C(N2CCC(O)C(N(C(=O)C=Cc3cnc[nH]3)C)C2)=O)n1 CS(C)(=O)=NC(=O)C(=O)NCC1C2CN(C(=O)CCNC3CC3)CC12 C(CC1=CCN(C(C2CC=CCO2)=O)CC1)NC(c1scc(OC)c1)=O c1(C(=O)NC)ccc(CC(=O)NCCNC2CCCC2C(=O)O)cc1 CCCC(C(=O)OC)C(=O)N1CC(O)CC1C(=O)NC(C)(C)C(F)(F)F C(=O)(C1=C(Cl)CCC(C)C1)N1CCN(C(COCCCCCC)=O)CC1CF c1(C(=O)NC2(C)CC(NC(c3n(CC)ccc3)=O)C2)cc(F)cc2c1CCC2 C(C(CO)(CO)NC(C1CCCCC1)=O)N(C(=O)CC(=O)NCC(F)(F)F)C c1(NC(C(CCC)CNC(=O)CCC(C)(C)F)=O)ccc2c(c1)CCC2 Cc1cccc2oc(C(=O)NCC3C4CN(C(c5ccc[nH]5)=O)CC34)cc12 c1(CC(=O)N)ccccc1[N+](=O)[O-].CC(O)C(C(=O)NC1CCC1C)N(C)C O=C1CC(C(=O)NCCCC2CCCN2C(c2c[nH]ccc2=O)=O)CCN1 c1(C(=O)NCc2cn(CC(=O)N(CCC)CC)nn2)cc(O)n(C)n1 C(=O)C(C)S(N)(=O)=O.Cc1nc(C2CCCC2)sc1C=O.C(C)(C)C(C)C.N C(CS(=O)(=O)c1ccccc1)NC(C1C(c2ccccc2Cl)(C)C1)=O CC1CCN(C(=O)C2=CCCCO2)CC1CNC(c1c(Cl)nsc1Cl)=O N1(CC(=O)N(C(CC(CC)C)C)C)CCCC(C(C)(C)C)CC1 c1(C(C(=O)NCC(=C)C)N(C2CCCCC2)C)nccc2ccccc12.C1CC1 CCC(C)(CO)C(=O)NC(CO)C(C)NC(=O)C=Cc1ccc(Cl)s1 C1(C(=O)NC23CN(C(CCC(=C)C)=O)C(C2)C3)CCc2nc[nH]c2C1 C1(CNC(c2scc(C)c2C)=O)C(O)C(O)CN1C(=O)C=Cc1cn[nH]c1 C#Cc1ccnc(C(=O)NC2CCC2CNC(=O)C(F)CC2CCOC2)c1 c1(OC)cncc(C(=O)NCC2CC2CNC(=O)CC(C)(C)SC)c1C c1(C(N(CC(C)NC(C(C(C)C)NC(N)=O)=O)C)=O)sc(C#N)cc1Cl c1(C(=O)NC(CNC(=O)CCC2CCCCC2)C2CCC2)ccc(C(F)F)nc1 c1(C(=O)NC(CCCNC(c2coc(Cl)n2)=O)c2ccccc2)c(Cl)nsc1Cl Cc1c(F)cccc1S(=O)(=O)NCC1(NC(c2cccc(Cl)c2)=O)CCC1 Cc1cc(N)c(C(N2CC(CNC(C3CC3C)=O)C3(CC3)C2)=O)c(F)c1 C(C(CO)(CO)NC(C1C2CCCOC12)=O)N(C(=O)C)C.[SH](=O)(=O)C1CC1 Cc1cc(C(=O)NC(c2ccccc2)C)sc1Cl.c1(C(=O)N)coc(C(N)=O)c1 Cc1cc(C(=O)NCC2(O)CC(C)C2)cnc1O.C(=O)(C(C)(C)C(C)C)N c1(CC)cc(C(=O)N(CCCC)CC)ccn1.C1(C(=O)N)CCN(C(C)=O)C1 C(=O)(CC(C)C(C)(C)NC(=O)CC(O)CC(C)C)NCC(C(=O)OC)(C)C C1(C(=O)NC2CC(NC(Cc3scc(C(N)=O)c3)=O)C2)CCn2cncc2C1 CCCC(C(=O)OC)C(=O)NCCC(C)CCNC(C1Cc2cccnc2C1)=O C1(CCCN(C)C)CN(C(=O)CCCC2CCOCC2)CCO1 CCC(C)C(C)C(=O)NCCC1(O)CN(C(=O)C(F)CC2CCOCC2)C1 CC1CCCC(C(=O)NCC(C)(C)CN(C(=O)CCCc2cncs2)C)C1 C(=O)(CCN=C(NCc1nc(C(F)(F)F)n[nH]1)NC1CC1C)NCC N1(C(c2cc(C(=O)OC)cc(F)c2)C(=O)NCCCC)CCCC2C(O)CC12 c1(C(=O)NC2C(C)N(C(=O)CC(C)(C)O)CC2)c(Cl)c([N+](=O)[O-])nn1C c1(C(=O)NCCS(=O)(=O)N(C)C)noc2c1CN(C(=O)Cc1cnccn1)CC2 CCC(C)C(O)C(C)C(=O)NCCN(C(=O)CCC1OCCO1)C1CC1 C12(NC(CC=C=C)=O)CC(C)(C1)OC21CCN(C(C2C3CC4C(C3)C24)=O)CC1 c1(C(N(CCC(N2CC3CC2CS3=O)=O)CC#C)=O)c[nH]c2ccccc12 Cc1c[nH]c2ccc(C(=O)N(C3CCS(=O)(=O)C3)C(C)CO)cc12 Cc1cnc(Cl)c(C(=O)N(c2nccc(Br)n2)C2CCC(N)C2)c1.C1CCCOC1.N CS(=O)(=O)CCNC12CC(C(=O)NC3C4CNC3C4)(C1)C2 c1(C(C)C)ccccc1NC(=O)C(C)N1CCC1C.C1(CC(=O)N)CCCC1 Cc1cc(CNC(C2(NC(=O)CC(C)F)CC(F)C2)=O)cc(F)c1 C12(C(=O)NC3(C(=O)N(C)Cc4cncnc4)C(C)C3)CC(C#N)(C1)C2 O=C(CS(=O)CCC(F)(F)F)NC1CC(NC(=O)C2CCCc3nccn32)C1 C1(NC(c2ccc(C)nc2)=O)CCN(C(=O)CC2CC2C2CC2)C12CCC2 C1(C(N2CC(N3CCCCC3)C2)=O)(NC(c2ccsn2)=O)CCCC1 N1(C(CC2(OC)CCC2)=O)CC(O)(CCNC(=O)CCCN2CCOCC2)C1 C12(CC)CCC1CN(C(c1nnn(C)c1C(F)F)=O)C2.Cc1cc(C(=O)N)no1 C1(NC(CC2(C=C)CC2)=O)CCN(C(c2nccn2C(C)C)=O)CC1C c1(OC)cccn2ncc(C(=O)NC3CC3C)c12.C(=O)C(C)Cc1cnc[nH]1 C1(NC(CCCc2n(C)cnn2)=O)COCCN(C(=O)CC2(C)CCCC2)C1 c1(C(=O)NC2CCN(C(C(C)SCC)=O)CC2(C)C)c(C)nc2cccnn12 Cc1ccc(-c2cnc(C(=O)NC(=O)NCCCl)nc2)cc1CO C=C=C(C)CC(=O)NCC(C1CCCC1)NC(c1ccnn1C1CCC1)=O C(=O)(C1c2ccccc2C2CC1C2)NCC1C(NC(c2c(C)cno2)=O)C1 CCC(CC)CCC(=O)NCC1C(C)CCCN1C(c1cnn2ccncc12)=O C=C1CCN(C(=O)C(C)C(C)NC(c2ccc(C3CC3)o2)=O)CC1 N1(C(C(CSC)O)=O)CCC2(CC1)CC2C(N1CCCCC1)=O C1(CC(=O)OC)CC2(CCC2)CN1C(=O)C(C)Cc1ccccn1 C1(CN(CCN(C(COC2CCCC(C)C2)=O)C)C)Cc2ccccc2CO1 c1(C(=O)NC(C(C)NC(=O)CNC(N)=O)CO)ccc(O)c(F)c1F C1(C(=O)NCC(CC)(C)NC(=O)CC2CC=CCC2)CCC(=O)N1C C(C)(C)(CC(=O)Nn1cccc1)N(C)C(C1(C)CCCCC1)=O N1(C(c2cncc(CNC(C3CC=CCC3)=O)c2)=O)CCc2ncsc2C1 CCC(C)C(C)CNC(=O)CC(C1CC1)NC(=O)C(CO)OC C1(C(NOCCNC(=O)OC(C)(C)C)=O)CCCCC1.C1(S(C)(=O)=O)CC1.C c1(C(N2CC(OC)C(NC(C3(C)CCN(C)C3)=O)C2)=O)ccc(N)c(N)n1 Cc1coc(C(=O)N(C(C)CNC(C2CCCC3CC23)=O)C)c1C c1(Nc2ccc(CN3CCCC(C)(O)C3)nc2)nc2ccc(N)cc2s1 C(CC(C)C(=O)NC1(C(=O)NCC(C)(C)C(C)O)CC(F)C1)=CCC c1(OC)cn(-c2ccccc2)nc1C(=O)NC(C)CN(C)C(C1CCCO1)=O C=CCC(CNC(=O)CC(C(F)(F)F)NC(C1CN(C)C(=O)N1)=O)CC(C)C C(=O)(C(C)S(C)(=O)=O)NCCN(C(=O)C(C(C)O)N(C)C)C(C)C N1(C(Cn2nc(C)oc2=O)=O)CC2(CCC(NC(C3CCCNC3=O)=O)CC2)C1 C1(NC(C2(NC(c3cnn(C(F)F)c3)=O)C(C)(C)C2)=O)CCN2CCCCC12 C1(C(=O)NC(CC)CC(C)CO)CCCN1NC(=O)C=C(C)C N1(C(CCC)=O)CCN(C(=O)C(O)CC(C)C)CC1c1ccc(F)cc1 N1(C(c2cnc(C)[nH]2)=O)CCC2(C1)CN(C(c1cncc3ccsc13)=O)CCO2 Cc1ccc(CCC(=O)N)c(C)c1.C1C(O)C(O)CN1C(C12CC(C)C1C2)=O.C C1(C(C)O)CCN(C(=O)CCC2CCCN2C(=O)Cc2ccccn2)C1 Cc1cc(=NCCC2CC(NC(c3cnc4ncccn34)=O)C2)[nH]c(C2CC2)n1 N1(C(c2cnnc(O)c2)=O)CC2(C(=O)NCc3ccc(F)cc3)CCC1CC2 c1(C(N2C(CNC(C(CCC)C)=O)CC(F)(F)C2)=O)cc2sccc2n1C c1(OCCOC)ccc(C(=O)NCC(C)C)cc1.C1(CC=O)(C=O)CC1 Cc1cccc(F)c1C(N1CC(CC(C)NC(c2ccc(=O)n(C)c2)=O)C1)=O c1(C(c2n(C(C(=O)OC)C)nnn2)NCc2csnn2)cn(C(C)C)nc1Br c1(C(=O)NCCCC(C)NC(c2cnc(COC)s2)=O)ccnc(Cl)c1N c1(C(C2C(C=O)CC2)=O)ccccc1.C(C)(CC)OC.C(=O)(CC1CC1)N c1(C(=O)NCC2(C)CCN(C(C(C)=C(CC)C)=O)C2)c(C)ccc2n[nH]cc12 C1(CC=C)(NC(=O)CC(=C)C)CCN(C(c2ccc(C)cc2)=O)CC1 C(=O)CCP(C)(C)=O.C(C)(C)(C(=O)NC1CCC1)NC(=O)NCC.C C1(C)(CC)CCCN(c2nnc(C3CC3)n2CCC2(O)CCOC2)C1.C1CC1 c1(C(N(C2CN(C(c3ccc(CO)cc3F)=O)CC2F)C)=O)cccc(=S)n1O Cc1ccc2nc(N3CC4C(NC(=O)CC(C)(C)C(C)(F)F)C4C3)sc2n1 C(CCOC)(C(=O)N=c1cc(C)n(CCOCCO)[nH]1)NC(CCCC)=O c1(C(=O)NC(C)CCN(C)C(C2(CO)CCOCC2)=O)ccc2ncncc2c1 C1(NC(C=CSC)=O)CC2CN(C(C3(S(C)(=O)=O)CC3)=O)CC2C1 c1(N(C)Cc2cc(OC)cc(OC)c2)nc2ccsc2c(=NCCOC2CC2)[nH]1 c1(OC)ccc(C(C(=O)NC(C)C)N(C2CC3CCC2O3)C)cc1C#N n1(CC(=O)NCC2CC(NC(C(C=CC)O)=O)C2)ncc(O)nc1=O N1(C(c2ccc(C)c(O)c2)=O)CCC2C(CCCN2C(=O)CCS(C)=O)C1 c1(OC)cccc2c1OC(C(=O)NCCC1CCCN(C(=O)CC(F)F)C1)C2 C1(CN(C)C(C2(CF)CCC2)=O)COCCN1C(=O)CCC1CC1 Cc1cc(C)c(C(=O)N(CCC)C2CC2)c(=O)o1.C1(C=O)CC2OC1C1CC21 Cc1cc(C#N)c(O)nc1C(=O)N(CC(C)CNC(=O)C(C)N1CCC1)C C(=O)(C(C)(C)CC(=O)NC(C)(C)CO)OC.c1(C(=O)N)ccc(CCO)cc1 CC1=CC(C)CN(C(C2CC(O)CN2C(c2cnc(C)s2)=O)=O)C1 CC(CC(C)(F)F)C(=O)NC1CC(C)C(O)C1.c1(C(=O)N)c[nH]c2nccc-2c1 O=C(N=c1[nH][nH]c2c(Cl)cccc12)C12CC1CN(Cc1cnc(Cl)nc1Cl)C2 N1(C(CNC(CCC(C)C)=O)=O)CCN(C(C2CC(O)CN2C)=O)CC(C)(F)C1 C1(C(=O)NCC(C)(C)NC(c2cn(C)[nH]c2=N)=O)CCc2nn[nH]c2C1 C(=O)(CCCC(=O)ON)N1CCN(CCCNC(=O)CCOCC(F)F)CC1 C1(OC)CC(NC(=O)CCC2CCCC2)CN(C(C2CC(C(=O)OC)C2)=O)C1 N1(C(CCn2c(C)nc(C)n2)=O)CCCN(C(=O)CC2OCCC2(C)C)CCC1 c1(SC)ccnc(C(N2CCC(C)C2CNC(=O)CC(C)SC)=O)n1 Cc1sncc1C(=O)NC1CC(OCC(=O)NCCCC2C=NNC2=O)C1 c1(CC(N2CC(NC(CCN3C(C)CCCC3)=O)(CO)C2)=O)cc(F)cc(F)c1 C1(CC=C)(NC(c2csnc2OC)=O)CCCN(C(c2ccc(O)c(Cl)c2)=O)C1 C(=O)(C1CCC(=O)c2cccn21)N1CC=CC(NC(c2c(C)[nH]nc2Cl)=O)C1 c1(NS(CC2ON=C(CC)C2)(=O)=O)nc2c(s1)CCN(Cc1ccccc1)C2 Cc1c(C(N2CCOC(CNC(C3OCCC3C)=O)C2)=O)ccc2ccccc12 C1(C(=O)OCC)OCCN(C(=O)CCc2cc(F)ccc2Br)CC1N(C)CCO c1(CC)ccccc1C(=O)N.C1CC2CC2N1C(=O)Cn1ccc(C(F)F)n1 C=CCC(C(=O)NOCC(=O)OC)NC(C12CSCC1C2)=O Cc1ccc(C(=O)NCC2(C(=O)NCCC3CCCCO3)CCCC2)nc1C C1(OC)CN(C(=O)CC(C)c2cnn(C)c2)CCC1NC(=O)CCC(C)N(C)C N1(C(CN(CCC#C)C)=O)CCC(C2CCN(C(C3CC3(C)C(F)F)=O)C2)CC1 CCC(CC)CCC(=O)N1CC(NC(=O)C(C)C(C)(F)F)CC(C)C1 C1(CC)(NC(c2cccc(N)n2)=O)CCCN(C(=O)CN2C(=O)CCC2=O)C1 N1(C(CCCCOCC)=O)CCC(C)CC1CNC(=O)CCn1cnccc1=O N1(C(c2c(OC)cccn2)=O)CCOC2(CCN(C(=O)CC3CCC3)C2)C1 C(CN=c1[nH]cc(C(F)F)s1)c1c(C(C)C)con1 c1(C(=O)NC2CN(C(CCCC(C)=O)=O)CC(C)(C)C2)cc(=O)n2ccsc2n1 Cc1c(C(=O)NC(C)(C)CCCNC(=O)C(C)(C)N2CCCC2)sc2cncn12 N1(CC)CCCC1C(=O)NC1CC(NC(c2csc(-c3ncccn3)n2)=O)C1 Cc1c(C(=O)NC(C)CO)cnc2ncnn12.C1(C)(CCC(=O)N)CCC(=O)N1 Cc1n[nH]c(C)c1CC(=O)NC1CCC(C)(CNC(c2cocn2)=O)C1 c1(CC)cc(CCNC(C2(NC(=O)C(F)=C(C)C)CSC2)=O)on1 C1(C(N2CCCC(N(C(C3CC(C)(C)C3)=O)CC)C2)=O)CC2C=CC1C21CC1 c1(C(=O)NC2CCN(C(c3cc(C(C)=O)[nH]n3)=O)C2(C)C)cnn2cccnc12 N1(CC(=O)NCC(COC)NC(=O)CCCc2cc[nH]n2)CCCCC1=O CCCC(CCNC(=O)C(CC1CC1)NC(=O)CC(C)OC)C1CC1 C=CC1CN(C(=O)C=Cc2sccc2C)CC1NC(=O)C(c1cccc(F)c1)O N1(CCOC(C)C)CCOC2(CCN(C(C3CCCC(=O)N3)=O)CC2)C1 Cc1cnc(C(=O)NC2CCN(C(c3[nH]nnc3C)=O)C2)s1 N1(C(C(C)c2ccsc2)=O)CCC(C)(CC(=O)NCCC#CCO)C1 CCC(C(=O)NCCC1CN(C(c2cnc(O)c(OC)c2)=O)C1)C(C)C c1(CC)ccc(OC2CCN(CC(N3CCOC(c4n[nH]c(C)n4)C3)=O)C2)cc1 N1(C(c2c(C)ccc(N)c2)=O)CCCC2CN(C(=O)CC(F)(F)F)CCC12 C1(OCC=C)CCN(C(c2ccsc2Cl)C(=O)NCC2CCCO2)C1 Cc1cc(C)c(CC(=O)NC(C(C)NC(=O)CCc2c(C)n[nH]c2C)C(C)C)s1 N1(C(c2c(C)nsc2C)=O)CCC=C(CNC(=O)C=CCO)C1 CC1CCOCCN1C(C1(NC(=O)CC(C)(C)CN(C)C)CSC1)=O Cc1ccccc1C(C)CC(=O)NC1CN(C(=O)CC(C)C)CC1O CC(CN=c1cc(-c2cccc(Cl)c2)nc[nH]1)NC(c1ccnn1CCF)=O c1(NC)nc(C)ccc1C(=O)NC1(C)CCN(C(C2(O)CC2(C)C)=O)CC1 c1(CC(=O)NCCCNC(C2C(C(C)(F)F)C2)=O)cnoc1.C1CCOC1 c1(C(N2CCC(CCNC(c3ccc(F)cc3F)=O)CC2)=O)c[nH]cc(F)c1=O Cc1nnccc1C(N1CCOC(C(C)NC(=O)CCn2ccccc2=O)C1)=O C(=O)(CCC(CC)NC(=O)Cn1nnc(C)n1)N(CC(=C)C)CC N1(C(C(C)N2CCC2)=O)CC(NC(=O)C(F)(F)C2(O)CCCC2)C(C)(C)C1 c1(C(=O)NCC2CCN(c3ncc(Cl)c(O)n3)CC2)cccc2nc(O)ccc12 N1(C(c2ncc(NC)nc2)=O)CC(C2CCCN(C(=O)CSC3CC3)C2)C1 N1(C(C(C)SC)=O)CCN(C(c2cncs2)=O)CC2(CC2)C1 c1(C(CCC)C)nc(C2CCN(C(=O)OC(C)(C)C)C2)n(-c2cnn(C)c2)n1 Cc1cc(=NC2CCN(c3ccc(=N)[nH]c3)CC2)[nH]c(=NCC2CC2(Cl)Cl)[nH]1 C12(CNC(CCn3cc(-c4cccc(COC)c4)nn3)=O)CCC(F)(CC1)C2 O(P(C)(=O)CCCN=C(NCCCc1ccc(C(F)(F)F)cc1)NC(C)C)CC C1(C(N2CC(CC(C(N3C(C)(CC)CC3)=O)F)C2)=O)(CF)CC2(CCC2)C1 c1(C(N2CCC(F)(CNC(c3c(CC)onc3)=O)C2)=O)cccc(F)c1O c1(OC)c(C(=O)NC2(C)CCN(C(C34CCC(CC3)C4)=O)CC2)ccnc1Cl.C N1(C(c2c[nH]c(=NC)o2)=O)CCCC(CNC(=O)C)CC1.N1(C=O)CCCC1.N c1(C(N(CCn2cc(Cc3cc(C)on3)nn2)CC)=O)ccccc1Cl N(C1CN(C(=O)CN(C)C(C)=O)Cc2ccccc21)C(C(C1CC1)SC)=O c1(C(=O)NCCC2CCN(C(=O)C=C(Cl)Cl)C2)cnc2sccn12 N1(C(c2cnn(C(C)C)n2)=O)CCC(O)(CNC(C2(C)CC2(F)F)=O)CC1 Cc1c(C(=O)NCC2(C)CCN(C(C3(C)CC3(C)C)=O)C2)cnn1C N1(C(COCCOC)=O)CCC2(CCC2NC(C2CC(=O)N(O)C2)=O)CC1 Cc1cccnc1CC(N1CCCC1CCNC(c1cc(C(C)C)nn1C)=O)=O CC(C)CC(C)(O)CNC(=O)CC1C(NC(=O)CCc2cscn2)CC1O c1(CCNCCNC(C(Cc2ccc(C#N)cc2)C#N)=O)cc(Br)c(F)cc1O CCCCC(C(=O)NCC1CC1)C(C)C.c1(C(NC)=O)cc(C2CCC2)c[nH]1.C c1(C(N(C)CC2OCCN(C(C(CC)C)=O)C2)=O)cnc2sc(C)cn12 c1(C(N2CC(NC(c3cc(C)cc(F)c3)=O)C(F)CC2)=O)ccc2ccnn2c1 C1(C(=O)O)COC2(CCN(CCCc3ccc(C(F)(F)F)cc3)CC2)C1 c1(OC)ccc(C(=O)NC2CC(NC(=O)CCC(N)=O)C2)nc1OC CC1(F)CN(C(c2cc(Cl)cc(Cl)n2)=O)CCN(C(c2cc(C(F)F)[nH]n2)=O)C1 C1(CC(=O)N(C)CC2CC2)CC2(CCO1)CC2.C1(C)CCC1.C(=O)C.C N1(C(C2C(C)(C)COC2)=O)CCCC(C)(CNC(=O)Cc2cscn2)C1 c1(C(N(CC(C)NC(CC(C)CN(C)C)=O)C)=O)ccc2c(c1O)CCCC2 C1C2CCC1CN(C(c1ccc(Cl)c(Br)c1)=O)C2.c1(C(=O)OC)cc(NC)cs1 C1(CNC(C2(F)C(C)OCC2)=O)CC2CCC(C1)N2C(=O)C(C)(C)C(N)=O CC1C(NC(=O)C(C)CC2CC2)CC2CCC1N2C(=O)C=Cc1ccccn1 N1(C(CS(CC)=O)=O)CC(F)(F)CC1CCNC(c1ccn(CCF)n1)=O N#Cc1ccc(NC(=O)C(CCC2CCC2)NC(C2C=CCS2)=O)c(O)c1 c1(NC(C2C(C(=O)NCC(O)CO)C2)=O)cc(F)c(Cl)cc1[N+](=O)[O-] CC1CCCN(C(C2CCOC2)=O)C1CNC(=O)C=CC=C(Cl)Cl CC(C)(C)C(O)C(=O)N1CCN(C(=O)CSC(F)(F)F)C(C2CC2)C1 c1(C(=O)NCC(C)N(C(C(C)OCCCC)=O)C)cc(C)nn1C N1(C(c2ccccc2C)C(=O)NCCCC(=O)OCC)CCN(C)CC(O)C1 C1(c2cccnc2)(C(=O)NCC(CNC(C(CC)(C)C)=O)O)CC2(CCC2)C1 c1(C(=O)NC2(C)CC(NC(C3CCC34CCC4)=O)C2)ccnc(N2CCCC2)c1 CCCC(C)CC(=O)NC1CC(CCNC(=O)C=Cc2ncc(C)[nH]2)C1 C#CCCN=C(NC1CC(OCc2ccccc2)C1)N1CCCC(CC(N)=O)C1 CCCCC(CNC(=O)CCCn1ccnn1)NC(=O)C=CCF c1(C(=O)NCC2C(NC(c3c(C)[nH]nc3Cl)=O)CCC2)c(N)cc(F)cc1F CC(F)(F)C(F)C(=O)NCc1cn(CC(=O)NC(C2CCCO2)CO)nn1 c1(CCCCC)nc(-c2cn(C)cn2)n(C2CCCC(C)C2)n1 c1(C(=O)NC)ccc(-c2ccc(OC(F)(F)F)nc2)nc1.c12cccc(c1)NC2 Cc1cc(C)c(CC(N2CC(CNC(=O)C3=CCOCC3)CC2(C)C)=O)c(C)c1 C1(C(=O)Nc2cc(SC)n[nH]2)CC2(CCN(C(=O)C3=COCCC3)CC2)C1 N1(C(c2ccc(Br)o2)=O)CC2(CCCCN2C(C2CCOCC2)=O)C1 c1ccc(S(=O)(=O)C(F)(F)F)cc1.NS(=O)(=O)c1ccsc1CNC=O.N N(C(=NCCC=C)NCC(c1ccc(Cl)c(Cl)c1)O)C(C#C)COC c1(OC)cc(NC(=S)N2CC(c3nnc(S)n3C)C2)cc(C#N)c1 C1(NC(CCc2nc(C)sc2)=O)CC2CN(C(c3ccccc3C(C)O)=O)CC12 C1(C)(NC(c2c(OC)cncc2)=O)CCN(C(=O)CC2(C)CC2(F)F)CC1 c1(CC)cnc(C(=O)N(CCC(=O)NC(C2CCCOC2)CC)CC)nc1 Cc1ccc(N)c(C)c1C(=O)N(C(=O)CCC(=O)N)CC(C)C.CC(N)=O CC1CCCC1(C(=O)N(C)Cc1nnc(O)o1)NC(=O)CCc1cscn1 N1(C(C2C(C=C)CC2)=O)CCC(CN(C(=O)CC23CCC(CC2)C3)C)CC1 C1(CC(=O)NCc2nocc2C(N2CCC(CCO)C2)=O)CC2CC2C1 C=C1CC(C(N2CCN(C(c3ccc(C)cc3)=O)CC2)=O)N(C(=O)CN(C)C)C1 Cc1c(NC(=O)C(O)CCCNC(C2(C)C=CCCC2)=O)cccc1F C(=O)(C(C)CC(=O)NCC1CCN(c2cccnn2)CC1)OC c1(C(=O)NCC2N(C(CCC(=C)C)=O)C3C(C2)C3)ccc2c(c1F)CCC2 N1(C(C2C(C)OCCC2)=O)CCC2(CC1)CC2NC(c1nccn2ccnc12)=O c1(OC)cnncc1C(N1CC=CC1C(=O)Nc1cncc(F)c1)=O C1(CC(C)N(C)C(=O)NCc2ccccc2)Cc2ccccc2O1.C(C)(C)(C)O C1(CC(=O)N(C(CC)C)C)C2CCCC2N1C(=O)C(C1CC1)C1CC1.CS N1(C(C(c2cccnc2)C)=O)CCn2c(nc(C(=O)N(C3COC3)C)c2Cl)C1 C(=O)(n1[nH]c(=NC(=O)c2cccc3c2NC(=O)C3)c2c1CN(C(C)=O)C2)OCC Cc1c(C(=O)OCC(=O)O)sc2c(Cl)cccc12 n1(CC)cc(C(=O)NC2COCCC2C=O)c(C)n1.C1(CC)COC(C)(C)C1 CCCC(O)CC(=O)N1CCN(C(=O)Cc2ccsn2)CC1C1CC1 c1(C(N(CC(C)CNC(c2ccc(Cl)nc2)=O)C)=O)ccc(Cl)c(F)c1N C12(C(N(C)Cc3ncc(C)o3)=O)CCCC1CCN2C(c1csnc1Cl)=O c1(C(=O)NC(CNC(C(CC)(C)CC)=O)(C)C2CCC2)cc2cccnc2[nH]1 CCCCC(O)CC(=O)N1CCCCCC1C(=O)NCC1CCC(F)(F)C1 C1(C(N(C(CN(C(C)=O)C)C)C)=O)CCN(C(=O)C(F)OC(F)(F)F)C12CCC2 Cc1ccc2n[nH]cc2c1C(N1CCN(C(=O)CC2CCC(=O)N2)CC1C)=O C(CC(=O)NCC(C)(O)CSC)(C(C)(C)C)NC(c1c(OC)n(C)nc1)=O c1(CC)ccc(NC(N2CCC(N3CCN(C(=O)CC(O)CC)CC3)C2)=O)cc1 CC(CF)CC(=O)N1CCN(C(CNC(=O)CCN2CCOCC2)C(F)F)CC1 CN1CCN(C(C2CCC=CCC2)=O)C(C(=O)NOC2CCOCC2)C1 S(=O)(=O)(c1ccc(C(N2CCCC2)=O)cc1)N1C(CC(C)=O)CCCC1 Cn1ncc2c1CCC(C(N1CCC1CNC(c1csnn1)=O)=O)C2 C(=O)(C(O)CCCNC(C1CCOC1C1CC1)=O)NC1C(C)COCC1 c1(CCC(=O)N)ccccc1C.C(CCC(=O)N(C1(COCCC)CC1)C)SC c1(C2(C)CC2)ccccc1C(=O)NCC(CO)NC(C1CC(CCO)C1)=O N1(C(CSCC)=O)CC2CC(C(N3CCCC3CN=[N+]=[N-])=O)C(C2)C1 c1(OC)ncc(NC(=O)CCCOC(=O)CC2OCCC2C)cn1 C=CCCCCCC(=O)N1CCCC1(CC=C)C(N1CCC(N(C)C)CC1)=O Cc1cn(C)nc1C(N1CC(C)(NC(=O)CC2(C)CC2)C1)=O c1(NC2CC(CNC(C3C(=C)CC3)=O)C2)ncnc(Cl)c1F CC(C)(C)C#CC(=O)N1CCC(c2ccccc2)(NC(=O)CC2CC3(CC3)C2)C1 N1(C(c2cn(CCOC)nn2)=O)CCCC2(C1)CN(C(=O)C)CCO2.C(N)=O.N C1(NC(=O)CC2CCS(=O)(=O)CC2)C2CC1CN(C(=O)C(F)F)C2 N1(C(C2(C#C)CC2)=O)CCC(O)(CNC(C2CC(C)(CC)C2)=O)C1 CC1(C(=O)NC2CCCCC2NC(c2scnc2Cl)=O)C=CCCC1 n1(CC(=O)NCC2C3N(C(CCOC)=O)C(CC3)C2)cc(Cl)c(O)nc1=O N1(C(c2ncn(CC)c2)=O)CCCCC1CCNC(c1n[nH]cc1OC)=O C1(CN(C(c2occc2C)=O)CC)CCCCN1C(=O)CCc1cnoc1 C=CC(CC)CC(=O)NCCCC(C)NC(=O)CC1COCC1(C)C CC1c2ccc(O)cc2CCN1Cc1cc(OC(F)(F)F)ccc1Cl c1(CC)ccc(C(=O)NCC(CC2CCCC2)C(=O)N)cc1.C1(C)CCCC1.C Cc1cccc(CC(=O)NC2(CC(=O)NCC3CN4CCC3C4)CCC2)c1 C(CCCOC)(C(=O)N(C)Cc1ccc(C)cc1)NC(C1C(=C)C1)=O C1(Cn2c(N(CC(CC)C)C)nnn2)CC2CCOC12 c1(NC)snc(C)c1C(=O)NCC(c1ccccc1F)OC n1(C(C)C)ncc(C(=O)NC(C)(CNC(=O)C(C)(C)N2CCOCC2)CO)n1 c1(C(N(C(CNC(CC2C(C)C2)=O)C2CC2)C)=O)cc(C(C)(C)C)n[nH]1 c1(CC(=O)NCC#CCNC(C(=Cc2ccccc2)CC)=O)c(C)cccc1C n1(C(C)(C)C)cc(NC(c2ccoc2)=O)cn1.C1(CC=O)CC2(CC2)C1.C CCCC(CNC(=O)C(Cl)Cl)NC(c1cc(CC)no1)=O C=CC(C)CN=C(NCc1ccccn1)NCC1CCCC(OC)C1 c1(C(N(CC(C)N(C(CN(CCCCCC)C)=O)C)C)=O)nc(=N)cc[nH]1 c1(C(=O)OC(C)(C)C)c(F)ccc(NC(C23CCCC2OCC3)=O)c1Cl c1(C(N2C(CO)CC(NC(=O)CCc3nc[nH]n3)C2)=O)cccc2oc(O)nc12 c1(C(N(C2CN(C(CCOCC(C)C)=O)CC2(C)C)C)=O)ncnc2ccsc12 Cc1ccccc1C(C)CC(=O)NC1CCC(NC(C2(C)CCCC2)=O)C1 C1(CC(=O)NC2C(NC(Cc3c(C)cccc3)=O)COC2)CCCCCC1(F)F N1(C(CCC2N(C(=O)CO)CCC2)=O)CCC12CCCOCC2.S(C(F)(F)F)CC=O c1(CC(=O)N(CCC)C2CC2)ccc([N+](=O)[O-])cc1Cl.CC1CC(C=O)CO1.N C1(CCNC(CC2N(CC)CCC2)=O)CCCN(C(c2scc(C)c2C)=O)CC1 N1(C(c2nc(C)n(C)n2)=O)CCC(NC(=O)Cc2ccnn2C)C(C)C1 C(CC(C)(C)C(=O)NCCCC(C)C)NC(CCC=C=C)=O c1(C(=O)NCC2(NC(C(CC)C)=O)CCCC2)cncc(C(F)F)c1 c1(C(N(C2CCN(C(c3ccc(Br)s3)=O)C2)C)=O)n[nH]cc1F O=C(CCC(F)(F)C(F)(F)F)NCC(C1CC1)NC(c1cc2cnccc2[nH]1)=O c1(C(=O)NCC2(F)CC(CNC(CS(CC)=O)=O)C2)cccc2c1NCC2 C1(C)(COC)CCN(C(C2CCC(n3cc(C4(C)CCCC4)nn3)CC2)=O)C1 C1(COC)(C)CCCN1C(=O)C.c1ccc(F)cn1.C1(C=O)CC1(C)C.N n1(CC(N2C3CN(C(c4c(C)cc(Cl)cn4)=O)CC32)=O)nnc2ccccc12 N1(C(CCSCC)=O)CCC(C2CCN(C(c3cnc4[nH]cncc3-4)=O)C2)CC1 c1(COC)nc(NCc2nccn2CC(C)C)cc(N(C)CC2CCOC2)n1 c1(C(=O)NC2(CCCNC(C(C=CC)O)=O)CC2)ncccc1N=[N+]=[N-] Cc1ccc(C(=O)NC(CO)C(C)NC(=O)C(C)N(CC(F)(F)F)C)cc1C C1CCN(C(=O)Cn2nc(C(F)F)cc2C(F)F)CC1.C=C1CC1C(=O)N c1(N2CCCC(NC(c3occ(C)c3)=O)C2)cc(O)nc(O)n1 C1(NC(c2c(C)n(C)nc2)=O)CC(F)CN(C(=O)C=Cc2ccccn2)C1 Cc1cc([N+](=O)[O-])c(Cl)cc1NC(C1CC(C)CN1Cc1cccc(CO)c1)=O N1(C(C2(OC)CC2)=O)C(CC(N2CC(F)(F)CC2C(N)=O)=O)C2CCCC12 c1(C(C)=O)nc(C(=O)NC(C)CCNC(=O)Cc2cscn2)cs1 c1(C(c2n(CCCSC)nnn2)NCC2CCCOC2)c(Cl)cccc1[N+](=O)[O-] CCCCC(C)CCC(=O)N1C2CCCC1CN(C(=O)C(C)S(C)(=O)=O)C2 N1(C(c2cc(C)c(Br)o2)=O)CCN(C(c2cnncc2O)=O)CC1CCO N1(C(C)C(=O)NCC2CCN2C(C2CC=CC2)=O)Cc2ccccc2C1=O Cc1[nH]nc(C(=O)NC(CN(C)C)C(=O)NC(c2ccoc2)C)c1Cl C1(C(=O)NC2C(NC(C(c3ccccc3)NC(C)=O)=O)C2)CCCCC1 C1(C(=O)OC(c2cccc(F)c2F)C)COc2ccc(F)cc2C1 C(=O)(C(C)(C)C(=O)N1CC(C)(CCC(=O)NC2CCC(C)C2)C1)OC c1(C(=O)NC2C(C)CN(C(C3CC34CC4)=O)C2)cc2c(Cl)nccc2o1 Cc1ccc(CS(=O)(=O)NCC2CC(F)(F)CN2)cc1C c1(C(=O)NCCNCCn2c(C)nnc2)ccc(Nc2ccccc2)cc1 C1(NC(c2cc3cnccc3[nH]2)=O)C2CCC1CN(Cc1c(Cl)ccnc1Br)C2 c1(CC)ccc(C(N2CCCC(N(C(=O)C=Cc3cnc[nH]3)C)CC2)=O)cc1Cl C1(NC(C2(COC)CCOC2)=O)CC(F)CN(C(c2ccoc2Cl)=O)C1 c1(C(N2C(CNC(C3CC3(Cl)Cl)=O)C=CC2)=O)cc(O)ccn1 N1(C(C(CCC)OC)=O)CCC2CN(C(=O)CCCn3ccnc3)CC12 N1(Cc2c(C)nccn2)CCCC(NC(c2coc(C(C)(C)C)n2)=O)CC1 C(=O)(C(C)CCN1CCOC(Cn2nc(C)nc2C)C1)OC c1(CCC=O)cn(C)nn1.C(C)(C(=O)NCCOCCC)OCCC#C.N C12(C(=O)NCC3CC3F)CCCCC1CS(=O)(=O)C2 c1(C=O)ccc2c(c1)CNC(=O)N2.N1(C(C(C)OCCC#C)=O)CCC(C)C1.N c1(C(=O)NCCCN(C(=O)C=CC2CCCN2C)C)cnn2c1N(C)CC2 c1(C(N2CC3(CCN(C(CC(C)(C)C)=O)CC3)C2)=O)ccc2c(c1)C(=O)NC2=O C1CCN(C(=O)CC)CC1.c1(C(NCC)=O)cnn(C(C)C)c1Cl.C(N)=O.C C(=O)(C(C)S(=O)(=O)C1CCOCC1)N1C(CNC(c2c(C)cncc2)=O)CC1 Cc1ccc(CC(=O)NC2CC(C)N(C(c3cnc(C)c(C)c3)=O)C2)cc1C c1(C(=O)NCCN(C(Cn2ccc(C)n2)=O)C2CC2)ccc(C2CCOC2)cc1 C1(c2scc(C)n2)CCCCN1C(CC1(C)CC1)C(=O)NCc1cccc(Cl)c1 C1(CN(C(C(CC)N(C)C)=O)C)C2CN(C(c3c(OC)nsc3OC)=O)CC12 C1(NC(CC)=O)CCC2CCN(C(=O)CCOc3cc(C)cc(C)c3)C12 c1(C(N2C3(CN(C(CCCCC)=O)C3)CC2)=O)cnc2c([N+](=O)[O-])cnn2c1 C(=O)(C(C)C(C)(F)F)N1C(CNC(=O)C=Cc2cccs2)CC(OC)C1 c1(CNC(C(C)OCCOC)=O)c[nH]nc1C1CCN(C(=O)C(C)C)C1 N1(C(C2(C(C)C)C(C=O)C2)=O)CCC(c2ccncc2)S(=O)(=O)CC1.CC.O C(c1cc(C)cc(C)c1)=CC=O.c1(CC)cc(C(N2CCC(O)C2)=O)n(C)n1 N1(C(Cc2n(C)cnc2)=O)CCCC2CN(C(c3cccc(F)c3O)=O)CC12 N1(C(C2CCN(C)C2=O)=O)CC2CCC1C(CNC(C1CCCC(F)(F)C1)=O)C2 N1(C(C(C)Cc2cnc[nH]2)=O)CCC(CNC(C2(Br)CC2)=O)C(C)C1 c1(OC)cc(CNC(C)(C)CO)cc(S(=O)(=O)NC2CC2)c1 C(C(C)CC(=O)N1CCC(c2n[nH]cc2CNC(c2ncn(C)n2)=O)C1)OC N1(C(Cc2c(C)nsc2)=O)CC(F)CC1CN(C(=O)CCOC1CCCOC1)C CC1(CNC(C2CC(O)C2)=O)CCC(NC(=O)CC(=O)NC2CC2)C1 Cc1cc(CN2CC3CC2CN3Cc2ccccc2)cc(C)c1Br C(=O)(CCCCCOC)NCC1CCC(C(=O)NC2(C#C)CCOC2)CC1 N1(C(CN(C2CC2)CC)=O)CCCC(F)(C)CC1.C1(C)(C=O)C=CCCC1.N CCCC(C)C(=O)N1CCC2CC12C(=O)Nc1cccc(O)c1 C12(C(=O)NC(C)CN(C)C(c3cncn3C)=O)CCC(CF)(CC1)CC2 c1(CN2CCC(C(N3C(CN(C)C)COCC3)=O)CC2)cccc(O)c1F c1cccc(C=O)c1.C(C)(C)CO.C1(C)(C=O)CC1C(F)(F)F.CN(C)C C1(C(=O)NCc2ccc(C(=O)NC(CC#C)C(N)=O)cc2)CCCCC(=O)C1 c1(OCC)cc(C(=O)OCC=O)ccc1[N+](=O)[O-].C(C)C=O.C(C)(C)C.N C(=O)(C(CCC)NC(c1ccn(CCOC)n1)=O)N(CCCC)CCCC N1(C(COCCSC)=O)CCN(C(c2ccccc2O)=O)CC1c1ccnn1C c1(OCC)nc(C)ccc1C(=O)OCc1ccc(C)cc1 c1(C(=O)NCCOC2CN(C(c3sccc3F)=O)C2)cc(Cl)cc(Cl)c1O CCC(CC)C(CN=c1cccc(S(=O)(=O)NCCOC)[nH]1)OCC1CC1 N1(C(C2C(OC)CCCC2)=O)CCC2CC(C1)CN(C(=O)CCCNC(C)=O)C2 C1(NC(N(CCCC)Cc2nnc[nH]2)=O)CCC(C)N(C=O)C1.C(C)(C)C CC1(C)CCCN(C(=O)C=CC2CCCCCC2)C1CNC(=O)COCCO C(c1ccc(Cl)cc1Cl)=CC(N1CCCC(CCNC(C2COC2)=O)C1)=O N(C1CCOc2ccncc21)C(c1cc(C2CC(F)(F)C2)[nH]n1)=O c1(C(=O)NC(CNC(c2cc(OC)c(F)cc2)=O)C)c(F)ccc(Cl)c1N C(c1cccc([N+](=O)[O-])c1)=CC=O.NS(=O)(=O)C1(C(=O)N)CC1.C1CC1 Cc1ccc(C(C)(C)C(=O)NC2CC2CNC(=O)CCc2scnc2C)cc1 C(=O)(CCCCCF)NC(C)CC1CN(C(c2cccc(C(=O)N(C)C)c2)=O)C1 CCC(CC)C(F)C(=O)N1CCN(C(C2COCC2C(N)=O)=O)C(C2CC2)C1 N1(C(C2C3CN(C)CC32)=O)CCC2CCN(C(=O)C(F)C(F)(F)F)CC12 C1(C(=O)OC)CN(c2cc(NC3CC=C(C)CC3)nc(C)n2)CCC1O C1(NC(CCSCCC)=O)CCC(CNC(=O)C(CC)NC(C)=O)C1 CCC(CCCC(=O)NCC1CCCCO1)NC(=O)CC1=CCCC1 c1(C(=O)NCCC(CNC(c2ncc(C)c(C)c2)=O)O)ccc2nn[nH]c2n1 C1(CNC(c2ccc(OC)s2)=O)CCCCC1.C1(C(N(C)C)=O)CC(C)C1 c1(NC(C(COC(Cc2c(OC)cccc2)=O)C)=O)ccc(F)c(CO)c1 Cc1cc2ncc(C(N3CC(NC(=O)COCC(F)F)CC(C)C3)=O)cn2n1 c1(OC)c(Br)ccc(C(N2CC3CC2CN3C(c2cnc(C)[nH]2)=O)=O)c1F N1(C(c2nc(C)sc2)=O)CC2COCCC2(NC(c2n[nH]c(C(C)(C)C)n2)=O)C1 CCC(C)CCC(O)CC(=O)NCCC1(OC)CN(C(c2cc(CO)[nH]n2)=O)C1 c1(C(=O)NCC(C)CNC(=O)CCc2ccnn2C)cccn(C)c1=O Nc1c(F)c(F)cc(C(N2CC(NC(=O)C#CC3CC3)CCC(O)C2)=O)c1Cl C1(N(C(=O)CCC2CC2)C)CN(C(C2(C#N)CC2)=O)CC1O N1(C(C2ON=C(C(C)C)C2)=O)CCC=C(C(=O)N(C)CCc2ccccc2)C1 c1(C(CC)C)nc(N2CC3CC2CN3C(C23CC(CN2C2CC2)C3)=O)cc(C)n1 C1(C(C(=O)NC2CCC2)N(CCC#C)CC)C2CCOCC12 c1(OC)ccnc(C(=O)NC(C)C(=O)NCC(C)(C)C(C)O)c1 C1(C(=O)NCC2CCN(C(C3(C4CC4)CCC3)=O)C2)CC(O)c2ccccc2O1 C1(CNC(c2ccn(C)n2)=O)CCC12CCC2.c1(C=O)ccn(C(C)(C)C)n1 N1(C(c2c(OC)cccc2Br)=O)CCN(C(=O)Cc2ccc(Br)cc2)C2(CC2)C1 Cc1cc(NC(C2(C)CCCN(C(c3c(C)cccc3Br)=O)C2)=O)cc(Br)n1 c1(C(N2C(CNC(=O)Cn3cccnc3=O)CC2)=O)cnc2[nH]nc(O)c2c1 C1(CNC(c2c(CC)con2)=O)CCC(C)N(C(=O)CC(C)(C)O)C1 C(=O)CC(F)(F)C(F)(F)F.N1(C(C2N(C)CCC2)=O)CC(C(F)(F)F)C(C)C1 CC1CC2(CC2)CN1C(C1(NC(=O)CCCCCF)CC1)=O C=CC1(C(=O)NCc2cc(C(=O)NCc3ncoc3C)on2)CCC1 C1(c2n(C)nnc2)CCCN(C(N2CCCC2(C)Cc2nccs2)=O)C1 C1(CNC(CSC(C)C)=O)CCN(C(=O)CCC2CCN(C)C2)CC1(F)F [N-]=[N+]=NCC(F)(F)CCC(=O)N1CC2CC1CCC2NC(C1CNC(=O)N1)=O C(=O)(C(C)CC(C)(C)C)N1CC(NC(c2ncc(OC)nc2)=O)C(C)(C)C1 C1(CC=O)CCCC1(F)F.C1(CNC(C(C)NC(=O)NC)=O)CCCC1 C1(NC(c2cc(COC)[nH]n2)=O)CCN(C(c2cccs2)=O)C(C2CC2)C1 CC1(c2ccccc2)CCCN1N1CCC(N2CCCCS2(=O)=O)C1 C(CC(C)(C)C(=O)N1CCC(O)(CNC(=O)CC2CCOCC2O)CC1)OC C1(NC(c2cnc(OC)cn2)c2n(CCSC)nnn2)C=C(C)CCC1 N1(C(CC(C)(C)O)=O)CC2=C(C1)CN(C(C1CCC(C)(C)OC1)=O)C2 N1(C(C2CN(C(CCN(CC)CC)=O)CC2C)=O)Cc2cnn(C)c2C1 C1(C(=O)NCC(C)N(C(=O)C=Cc2nc[nH]n2)C)CCc2nc[nH]c2C1 N1(C(c2nccc(CC)c2)=O)CC(C)N(C(C2CC3(CCC3O)C2)=O)CC1C C(=O)(CCNC(=O)C(C1CCOC1)N(CCC)C)OCC.[SH](C)(=O)=O c1(CN(C(=O)CC2(O)CN(C(=O)CSc3nc[nH]n3)C2)C)ccccc1F CC(CCCOc1cccnc1)NC(c1conc1-c1ccccc1)=O C(=O)(CS(=O)(=O)C12CC(C1)C2)N1C(C)CN(C(=O)CS(N)(=O)=O)CC1 c1(C(N2CC(CC)(NC(c3cc(O)nc(C)n3)=O)C2)=O)cc2nc(Cl)ccc2s1 c1(C(C)N)csc(NC(c2ccn(C(C)(C)C)n2)=O)n1 CCCCC(C(=O)NC1CCCC12CN(C(c1ccc(C#N)o1)=O)C2)C(C)C c1(CC)onc(C)c1C(=O)NCC(CC)N(C)C(C1CC1(F)Cl)=O C1(C(N2CC(c3cn(CCC(=O)NC)nn3)C2)=O)CCn2c(C)nnc2C1 C1(NC(c2cn(C(C)C)nc2)=O)COc2cc(Cl)ccc2C1 c1(CN2CCC(F)(C(=O)NCC3(F)CCC3)CC2)cccc2[nH]ccc12 Cc1c(C(=O)NCC2CCN(C(=O)CC3CC4C=CC3C4)CC2)cncc1F Cc1nc2c(s1)CCCC2C(=O)NCc1cccc(-n2cc(CNC=O)nn2)c1 C1(CCNC(C2CCS(=O)(=O)N2)=O)(NC(=O)Cc2csnn2)CCOCC1 c1(C=O)sccc1C#N.c1(OCC)n[nH]cc1C(=O)N(C1CCCCC1)CC.N c1(N2CC3CN(C(c4n(C)c(=O)ccc4)=O)C3C2)ncc2c(ccn2C)n1 N1(C(CN(C2CC2)CC)=O)CC(NC(c2cccc(N)c2C)=O)CC12CCC2 C1(CC)C(=O)NCCCN1C(=O)CC(C)(C)n1cc(C(C)(C)OC)nn1 C(C(=O)NNc1ccc(Cl)c(Cl)c1)(c1cccc(Cl)c1)NC C(=O)(CCCC(CC)NC(c1cnc(C)nc1C)=O)NCCOCCCC#C C(N=c1[nH]c(C2CC2)nc2ccccc12)C1CCC(NC(C(C(C)(C)O)F)=O)C1 C(CC1=CCN(C(C2CS(=O)(=O)C2)=O)CC1)NC(c1ccc(OC)cc1)=O.O C(=O)(C(CCF)NC(c1cc[nH]c(=N)n1)=O)NCCc1n(C)cnc1 c1(C(=O)NCCNC(CC2CCCC(C)C2)=O)ccc(C(C)C)cc1O Cc1cc(N2CCCCC2CNC(c2sccc2F)=O)ccc1[N+](=O)[O-] CC(C)(C)C(C(F)F)NC(=O)CCCNC(c1occ2c1CCC2)=O C(C(C)(C(=O)NCC(C)CO)NC(=O)CCC(N)=O)SC C=C1COc2c(C(=O)NC3CC3CNC(=O)CC3COCC3O)cnn2C1 CC1CCN(C(C2CN3CCN2CC3)=O)CC1NC(c1ncccn1)=O C(=O)(C(C)(C)C(C)C)N.N1(C(C)=O)CCCC(NC(=O)CCC2CCOCC2)C1 N1(C(Cc2cn(CC)nn2)=O)CCC(C(N2CCC2COC)=O)(COC)C1 CCCCC(CC)CC(=O)N1CC2(C(=O)NCCN3CCC(C)C3)CCC1CC2 C(=O)(C1CCCc2nnn(C)c21)NC12C(NC(CC(=C)C)=O)CC(CC1)C2 c1(NC(CCC)CCO)ncnc(N(CC(C)(C)S(C)(=O)=O)C)c1C c1(C(N2CCC2)=O)cnn2cc(C)cnc12.c1(OC)ccc(C(=O)NC)c(C)c1 Cc1ccn2cc(C(N3CCCC4(C3)CN(C(=O)C(C)C(C)(C)C)C4)=O)nc2c1 S(=O)(=O)(c1cnc(N2CC(OCC)C3(CC3)C2)c(Cl)c1)N1C(CCC)SCC1 Cc1cn(C)nc1C(=O)NCC(CC1CC1)C(=O)NCCC(C)(C)O C1(CCC)C(=O)NCCN1C(=O)C(CC(F)F)NC(c1cnn[nH]1)=O C1(OC)CC2(C1)CC2NC(c1c[nH]nc1CNC(C1CCCCO1)=O)=O C(=O)(CCC(C)(F)F)N(CC(CC)NC(=O)CCc1ccc(N)cn1)C c1(Cc2nn(-c3n(C)nnc3)c(CCc3cc[nH]n3)n2)ccc(F)cc1F c1(C(N(C)CC2CCCN(c3ccnc(C4CC4)n3)C2)=O)ccc2n[nH]cc2c1 Cc1ccncc1C(C)NC(C1(C)CCCN1C)=O c1(C(N(CCCNC(c2cnn(C)c2F)=O)C(C)C)=O)ccc2c(n1)CCOC2 C1(NC(C2C(C(=O)OC)CCC2)=O)CCCN(C(c2cc(Cl)nn2C)=O)C1 Cc1c(C(=O)NCC2CN(C(C3CCC(=O)N3)=O)CC2C)nn(C)c1N c1(C(N(CCC(=O)NCC(c2ncc[nH]2)C)C(C)C)=O)cncc(F)c1 C(c1ccc(NC(C)=O)cc1)=CC(=O)NC(C1CCCCC1)C(=O)NC C(CCCC(=O)NC1CCC(C(=O)Nc2ccccc2C2CC2)CC1)NC(N)=O C(=O)(C(C)(C)C(=O)COC(c1coc(C(F)F)n1)=O)OCC N1(CC)CC(C(=O)NCc2ccccc2)CC1=O.c1(C=O)c[nH]c(=NC)o1.C C(CCC(=O)NCC(O)CNC(=O)CCc1ccccc1)NC(=O)OC Nc1cc(C(=O)NC2CCC2)ccc1-n1cncn1.C1(C(=O)N)CC2(CC2)CO1 C1(C(C)NC(C2N(CC#C)CCC2)=O)CN(C(=O)CCC2CC(O)C2)CCO1 N#Cc1cccc2[nH]cc(CN3CCC(NC(c4ccc(=O)oc4)=O)C3)c12 c1(C(N2C(CN(C(C(CC)C#N)=O)C)CCCC2)=O)cc2c(OC)cccc2s1 C1(NC(c2c(NC)nccc2)=O)CN(C(C2CC(O)CN2C)=O)C2(CCC2)C1 c1(N2CC(CNC(C3(CCOC)CC3)=O)N(C)CC2)ncccc1[N+](=O)[O-] C1(CNC(C(CCSC)O)=O)CN(C(c2c(C)cccc2O)=O)CC(C)(C)O1 C(=O)(C(C)=Cn1ccnn1)NCC1CCN(C(C(n2cnc(C#N)n2)CC)=O)C1 c1(CC(=O)NC2CCN(C(c3sccc3Cl)=O)CC2O)ccnc(Cl)c1F C1(C(N2C(C)CC(CNC(C3(C4CC4)CCC3)=O)C2)=O)CCCCC1(C)C Cc1cc(=NCc2nnc(C)n2C2CC2)[nH]c(=NCC(C)(C)NS(C)(=O)=O)[nH]1 C1(CC(N2CC(C)C(NC(=O)C(C3(O)CCCC3)F)C2)=O)CCCNC(=O)C1 C#CCC(CC(=O)N=c1ccn(C)[nH]1)NC(=O)Cn1cccn1 Cc1cccc2c1OC(C(=O)NCC1CCCN1C(=O)C(N1CCOCC1)C)C2 CN1C(=O)Cc2c(C(N3CCCC(NC(=O)C=C4CCCC4)CC3)=O)cccc21 N1(C(CC(C)OC)=O)C2CCC1CC(CC(C)NC(c1cc(C)c(C)o1)=O)C2 N1(C(C(C)C(F)F)=O)CCC2(CCN(C(C3(Br)CC3(C)C)=O)CC2)C1 C1(NC(c2cc3ccncc3[nH]2)=O)CCOC12CCN(C(=O)C(F)C1CC1)CC2 N1(C(c2c(C)ocn2)=O)CCN(C(=O)Cn2cnnc2)C2CCCCC12 C=CCCCCCCC(=O)NCc1ccc(CNC(=O)C)cc1.C(=O)C(C)C.N c1(OC)ccc(C(C)(C)C(=O)N(C)CCNC(C23COCC(C2)C3)=O)cc1 c1(C2C(C(N(CC(C)N(C(CSCC)=O)C)C)=O)C2)ccccc1Cl C=CCC(C(=O)NCC12CCC(NC(=O)CC(C)(O)CCC)(CC1)CO2)C(C)C C1(C(N(C(CNC(=O)CSC(F)F)C2CC2)C)=O)CC(C)(F)C1 c1(CC)ncc(C(=O)NC2CCCN(C(=O)C(O)CCSC)C2C)c(O)n1 C1(CC(N2CC(CNC(CC(=C)C)=O)(OC)C2)=O)C(=O)N(C)N=C1C C1(CN(C(C2N(CC(C)C)CCC2)=O)C)CCCN(C(=O)CCC(N)=O)C1 C(c1cccs1)=CC(=O)NCC(CNC(c1cnco1)=O)OC N1(C(CC(COC)C)=O)CCN(C(=O)CC2CCC(C)CC2)CC(C)(C)C1 N1(C(CSCCOC)=O)CCC(C(=O)NCc2cccc(O)c2F)C(O)C1 C(=O)(C1=CC(O)C(NC(C2COCC(C)O2)=O)C1)NC(C)C(F)(F)F c1(C(C(=O)N)O)ccccc1.c1(C(=O)NC2CCC2)cc(-c2ccc(Cl)s2)[nH]n1 C1(C(N2CCC(CC=C)(NC(c3ncccn3)=O)C2)=O)CC2C(C1)C2(C)C.O C#Cc1cccc(C(=O)NC2CN(C(=O)C(F)(F)C(F)F)CC2OC)c1F c1(NC(C(CN(C)C)NC(CCCCOCC)=O)=O)c(C)ccc(O)c1C C#CC1CCC(C(N2CCCC(CNC(=O)C(C)CN3CCOCC3)C2)=O)CC1 S(=O)(=O)(c1cccnc1NC12CCCCC1C2)NCc1ccc(CCCCC)o1 C1(CNC(C2C(CC)C2)=O)(NC(c2c[nH]c(=N)s2)=O)CC(F)(F)C1 c1(C(=O)NC(C)CN(C(=O)CC2COC(=O)C2)C)cc(Br)c2ccccc2c1 c1(C(=O)N)cc(F)c(F)c(F)c1.CC1CN(C(C2CC(C(C)(C)C)C2)=O)CC1 C1(Cn2cc(CCN(C)C)nn2)(CNC(=O)Cn2cnnc2O)CC12CCC2 C(c1ccccc1)=CCC(=O)NCC(C)(CO)NC(CC1(C)CCCO1)=O C#Cc1cc(C(N2CCCC2CNC(=O)CN2CCCCC2)=O)cc(N)c1 c1(C(N(C)CC2(C)CC2)=O)cccc2c1CCC(=O)N2.C1(C=O)CC1(Cl)Cl c1(C(N2CCCC(NC(c3nc(C)oc3)=O)C(F)C2)=O)cccc2[nH]cc(Cl)c12 C(CCCCC(=O)N1CC(C#N)(NC(CCC2(OC)CCC2)=O)C1)OCC C1CN(C(c2coc(Cl)n2)=O)C(C)(C)C1.C1(C(C)C)CC(CC(=O)NC)CCO1 CC1(C)CCC(CC(=O)Oc2cccc(C(=O)Oc3ccccc3)c2F)OC1 Cc1nc(C(N2CCCC(CCNC(c3cnco3)=O)CC2)=O)ccc1C#N N1(C(c2c(C)nncc2)=O)CCC(C)N(C(=O)Cn2cc(F)ccc2=O)CC1 C(=O)(C(C)(C1CC1)N(C(=O)CCc1ccn(C)c1)C)N(C1CCSCC1)C CC(CC(F)F)C(=O)NCC1CC(O)CN1C(c1ncc(Br)cn1)=O C1(NC(C2CCN2C2CCCC2)=O)CC2CCC(C1)N2C(c1ccnc(F)c1)=O C(=O)(C1=NOC(C)C1)N1CC(C)(NC(C(CCOC)C)=O)C1 Cc1ccc(C=CC(=O)NC(CCF)C(=O)NC(c2nccc(C)n2)C)cc1 c1(C(=O)NCc2nc(CC)on2)c(Cl)noc1C C1(C(N(C)CC2CCCC(NC(c3cc(C)ncc3)=O)C2)=O)COCCN1C=O c1(NC2C(CCC)C2)nc2c(c(=NCC(C)CN3CCOCC3)[nH]1)CCC2 c1(OC)ncc(Cl)cc1C(=O)NC(C)CCCNC(=O)CCc1nc(C)cs1 Cc1cccnc1C(C)NC(C1(CNC(C2COCC(C)O2)=O)CC1)=O CCCCC(C)CCC(=O)NC(C)C(=O)Nc1cn(C)nc1OC c1(OC)cc(N2CCOC(C(C)NC(C3(CO)CCOCC3)=O)C2)nc(OC)n1 Cc1cc(N2CCCC(c3n[nH]c(C)n3)C2)c2cnn(C)c2n1 c1(C(=O)NC2(C)CC(NC(Cc3c(C)cco3)=O)C2)csc2ncnc(O)c12 C(N=c1nc(N2CCC3(CCCO3)CC2)c2c([nH]1)COC2)c1n(C)ncc1 C1(NCCc2c(OC)cccc2)C2CCC1(C)C2(C)C C(CC(CO)C(C)C)NC(CCCC1(NC(C(C)NC(CC)=O)=O)CCC1)=O C1(C(N2CC(CNC(CCCC#C)=O)(OCC)C2)=O)CC(C)(C)OC1(C)C N1(C(c2cc(CC)c(F)cc2)=O)CC2(CNC(C3C=CCC3)=O)CCC1CC2 C1(NC(C(=O)Nc2ccc(Cl)c(-c3nn[nH]n3)c2)=O)CCCC12CCCO2 CCCC(C)CC(=O)NC(C1CCCC1)CNC(=O)C(C1CCOCC1)F Cc1cccn2c(CC(=O)NC(C)(C)C(C)C)cnc12.C12(C=O)CC(F)C1C2.N N1(C(C2C(NC(c3c(F)cncc3F)=O)COC2)=O)CC2(CCC2)CC1CO C1(O)(CNC(CC(CC)C2CC2)=O)CCCN(C(C2C3(CC3)C23CC3)=O)CC1 C(=O)(C1(C)CCCc2ccccc21)NC1CN(CCOC)CC1(C)C C=CC1(C(=O)NC2CCCN(C)CC2)CCN(C(=O)C(C)n2cnnn2)CC1 C1(CCNC(=O)CN2CCCC2)CCN(Cc2ccc(C(=O)O)s2)CC1O C1(C(=O)N)C2CCC(C2)N1C(C1CCCC2(CC2)C1)=O.C(CCO)OC(C)=O C1CC2(C1)CCC2.c1(CC=O)c(C)cnn1C.C(C=O)OCCOCC.N Cc1coc(C2CC2)c1C(=O)NCC(C)(O)CNC(C1CC(C)C1)=O C1(C(N2CCCC(NC(C34CC(CO)(C3)C4)=O)CC2)=O)CCCN2CCCC12 Cn1cc(C(=O)NC2CN(C(C3CC34CCOC4)=O)C2)c(C(F)F)n1 c1(C(=O)NC2CCN(C(C(CC)CC)=O)C2C)cc(C(F)(F)F)cc([N+](=O)[O-])c1 N1(C(C(COCC)C)=O)CC(CNC(c2[nH]ccc2CO)=O)CC1(C)C C1(O)(CNC(C2CC2C(F)(F)F)=O)CCC1.C1(C=O)CS(=O)C1.C C=CC(C)CC(=O)NC12CC(C)(C1)C2.c1(C=O)c(Br)cnn1C1CCC1.N N(C1CCOc2ccccc21)C(C(C)NCc1ncc2c(n1)CCOC2)=O c1(C(=O)NCCCN(CCCNC(C(c2ccnn2C)C)=O)C)c[nH]c(=N)s1 CC(C)(CCCNC(=O)Cn1cc(C2CC2)cn1)NC(C1CC=CC1)=O c1(CC)ccn2ncc(C(N3CCC(n4cc(C(C)O)nn4)(CC)CC3)=O)c2c1 c1(OC)ccc2[nH]cc(CC(=O)NC3CCN(C(=O)C(C)N(C)C)C3(C)C)c2c1 C#CCCCC(=O)NCC1CCN1C(=O)C(c1ccccc1O)NC(C)=O CCCC(C)(O)CC(=O)NCC(C)N(C)C(C1CCc2nncn2C1)=O c1(-c2ccc(C(N(CCNC(CS(CC)=O)=O)CC)=O)cc2)ccccc1C#N C(=O)(C1=C(Cl)CCCC1)NC1CCN(C(c2c(C)ncn2O)=O)CC1C CC1(C)CN(C(C2(C)CCCCO2)=O)CC1c1ccccc1 Cc1cn2c(n1)C(C)N(N1CCN(c3cccc4[nH]ccc34)CC1)CC2 c1(OC)cccc2c(C(N3CCN(C(=O)CCn4cccn4)CC3C)=O)n[nH]c12 c1(CCC(N2CCC(=CC)CC2)=O)ccc(O)c(Cl)c1.C1(CC)CC1C=O.N CONS(=O)(=O)c1ccc(C(=O)NCC2CCN(C(=O)C=C(C)C)C2)cc1 N1(C(c2ccc(C)cc2C)=O)CCC2(CCCN2C(=O)C(c2ccc(C)s2)C)C1 CCC(CC(=O)NCC1(NC(=O)CCC2CCCC2)CC1)SC c1(C(N2C(C(=O)O)CSC2c2ccc(Cl)cc2Cl)=O)cnc2c(F)cccc2c1 N1(C(C(C)=C2CCCC2)=O)CCN(C(c2cc(CO)n(C)n2)=O)C2CCCCC12 N1(C(c2cscc2Cl)=O)CCCCCC(NC(C2(N3CCNC3=O)CC2)=O)C1 c1(-c2nc(C)sc2)ccc(C(N2CCC(CNC(C3(O)CCOC3)=O)C2)=O)cc1 c1(NC(COC)C)nc(=NCCC2(OC)CCC2)[nH]c2c(C)nn(C)c12 c1(C(=O)NC2C(C)CN(C(=O)CN(CC(C)(C)C)C)CC2)nnc2n1CCCC2 C(=O)(C(F)C(C)CNC(C12CCC(C1)C2)=O)NC1CN(CC)C(=O)C1 CCC(C)(CNC(=O)CC1CC2CC2C1)NC(C1(c2ncco2)CC1)=O C1(NC(=O)CC2CC3CC3C2)Cc2ccccc2N(C(C2CC(F)(CO)C2)=O)C1 C(CCCCC(=O)NCC1CCN(C(c2cccc(CC#N)c2)=O)C(C)C1)OC N1(C(C2(CO)CC2)=O)CC2(CCCCN(C(C3(F)CC4(CCC4)C3)=O)C2)C1 C1(CNC(CCCNC(C)=O)=O)CCN(C(c2cc(=O)c(O)c[nH]2)=O)C12CC2 c1(CC)ccccc1OCCC(N1CC(C)C2CC12)=O.c1(C=O)cnc(O)o1.N C1(N)(C)CCC(C)(C)CC1.c12nc(C)ccc1c2=O.c1(CC)nnnn1CCCF Cc1cc(C(=O)NCCN2CC(C(=O)O)C(C(F)(F)F)C2)nn1C C#Cc1cncc(C(=O)NCC2CC3CCC2N3C(c2nn[nH]c2Cl)=O)c1 c1(C(=O)N(C2CC2)CC2CCCN2C(c2cncs2)=O)cnc2[nH]ncc2c1 C=CCCC(C(=O)N1CC2CSCC2C1)NC(=O)CN1CC=CC1 C1(OCC)CCC(C(=O)NCCC2(O)CN(C(c3cc(C)ns3)=O)C2)CC1 c1(CN2CCC(c3ccc(NC(CCSC)=O)cc3)CC2)ccc(F)c(C#N)c1 c1(C(=O)OCC)[nH]c(C)c(C(=O)CN2CCC(CO)C(C)C2)c1C C1(C(C)CNC(=O)C=Cc2ccoc2)CCN(C(C2COC(=O)O2)=O)CC1 C1(C(=O)NCC(CNC(C(C)OCC#C)=O)C)CCCC1F N1(C(C(CSC)OC)=O)CCCC(CCNC(=O)C2=NOCC2)CC1 C(=O)(C1=CCCC1(C)C)N1CCC(O)(CN(C)C(c2cnc(N)c(N)c2)=O)CC1 CN1C(=O)CCCC1C(N1CC(C)(NC(C23CC2CCC3(F)F)=O)C1)=O C1(N(C(CCC(C)SC)=O)C)CN(C(c2c(O)cccc2F)=O)CC12CC2 c1(NCCCOCCNC(C2CC3CCC2C3)=O)ncnc(O)c1Br C(=O)(C(O)CC(F)(F)F)N(C(CNC(c1c(CC)ccc(OC)c1)=O)C)C CCCCC(F)C(=O)NCC1(O)CC(NC(=O)CC2CCOC(C)(C)C2)C1 C(CC(C)C)(C(=O)N1CCCC1C(C)NC(C1CC1F)=O)NC(C)=O c1(CN(C(C)=O)C2CC2)cn(CCCC)nn1.c1ccc(C)s1.C(=O)(CC)N c1(C(N(C2CCN(c3nc(C)cc(OC)n3)C2)C)=O)ccc2ncncc2c1 c1(C(C(N2CCC(NC(Cn3nnc(=N)[nH]3)=O)C2)=O)(F)F)ccc(F)c(F)c1 N1(C(CSc2cn(C)nc2)=O)CC(NC(=O)C(=O)NC)CC1(C)C.C1CC1 C1(NC(C2(C(=O)OC)CC2C)=O)CCCN(C(c2cc(CO)c(C)o2)=O)CC1 c1(OC)c(Cl)cc(N2CCN(CCC3(C)CC3)CC2)cc1Cl N1(C(C)=O)CC2CCN(S(C)(=O)=O)CC2C1.c1(OC(C)C)ccccc1C(=O)O C1(C(=O)NC2(C(=O)NCC(=C)C)CSC2)CCCCC1F C1(NC(c2ncc(F)cc2F)=O)CC2CCC1N2C(=O)COc1ccc(O)cc1 C#CC1CC2CCC1N(C(C1(O)CCCCC1)=O)C2.C1(=O)C(CC(C)C)CN1CC C1CC2CN(C(=O)Cc3cc(C(F)(F)F)co3)CC12.Cc1cn(C)nc1C=O.N c1(C=O)ccc(C#N)cc1C.C1(CC)CCC(O)(C(=O)NCCCOCC)C1 C1(NC(=O)Cc2c[nH]ccc2=O)CCN(C(=O)CCCn2ccnc2)CC1O c1(OC)ccc(C(=O)NC)nc1N.c1(C(C(N2CCC2)=O)O)ccc(F)c(F)c1 Cn1ccc(C(c2nnnn2C2CC2)NC=O)c1.C1CCOC1c1ccnn1C.N c1(C(=O)NCC2CC(CNC(CNC=O)=O)OC2)cccc2cnsc12 N12CCCC(C1=O)C2=O.N=c1ccnc(N2CCNC(=O)C2)[nH]1 N1(C(C(CCC)F)=O)CC(C(=O)NCC(CC)C(C)C)OC(C)C1 Cc1cccc(C(=O)NCCC2CCN(Cc3nc(CC4CC4)no3)CC2)c1C c1(N(C)Cc2cc(OC)c(C)cc2OC)cccc(S(C)(=O)=O)c1 N1(C(CC(C)(C)C#N)=O)CCCC2(CCCN2C(C2CCC(C)(C)C2)=O)C1 Nc1ccc(Cl)cc1C(N1CCOCC1CCNC(C1CCC2(CCC2)O1)=O)=O CC1(C)C(NC(c2csc(Cl)c2)=O)C2CCCN(C(=O)CSC(F)(F)F)C12 CC1C=C(C(=O)NC2C3CN(C(=O)COc4ccc(C#N)cc4)CC23)CC1 Cc1coc2ccc(C(=O)NCCCCN(C(=O)COC3CCCC3)C)cc12 Cn1cccc1CC(=O)NC(CO)C(=O)NCC1CC1(C)C c1(CNC(c2c[nH]cc(F)c2=O)=O)nnc2n1CCN(C(=O)C1=NOCC1)C2 c1(C(=O)NC(CNC(CCC(=O)NC)=O)(C)CO)cc(C)c(Cl)c(C)c1 c1(C(N2C(CC)CCC2)=O)cc(S(N)(=O)=O)c[nH]1.CN1CC(O)CC1C(=O)N C1(C2CCN(C(C3CCCC(F)(F)C3)=O)C2)(NC(c2cc(C)nn2C)=O)CC1 N1(C(=O)CCCn2cccn2)CCC2CC12C(=O)NCc1cnco1 CCCCS(=O)(=O)c1ccc(-c2cc(=NCc3cc4sccc4s3)cc[nH]2)cc1 C1(CC(=O)N2CCC2)CC2(C1)CN(C(=O)COC1CCCCC1)C2 Cc1ccc2c(c1)CN(C(C1(F)CCCN(C(=O)CCCCC(C)C)C1)=O)C2 CC1(C)C(NC(=O)CNC(N)=O)CCN1C(C1C2COCC12)=O C=C1CC2(C1)CC(C(=O)NC1CCN(C(=O)C(CC)n3cncn3)C1)C2 C1(C=O)CC(O)CN1C(C1CC1CC)=O.c1(C=O)nccn1C(C)C.CN N1(C(C(C)Cn2cccn2)=O)CC2(CCC(NC(c3cccc(Br)n3)=O)CC2)C1 C=CC(C)(C)CCCN=c1[nH]c2c(c(=NCC(C(C)(C)C)OCCO)[nH]1)COC2 c1(CCC)ccc(C(=O)NCCCN(C(=O)CCc2csc(C)n2)CCO)s1 N1(C(C(CC=C)(C)N(C)C)=O)CCC2(COC(CNC(C3(C)CCC3)=O)C2)C1 Cc1cc(F)c(N)cc1C(=O)NC1CS(=O)(=O)CC1.C(=O)CCCC1CCC1 C(=O)(C#CC1(C)CCCO1)N1C(C)CC(NC(=O)CCCc2csc(=N)[nH]2)C1 c1(C(N2C(CNC(C3OCCC(C)C3)=O)COCC2)=O)ncc(F)cc1N C(=O)(CC(F)(F)C(F)F)N1CCC(C(N2CCCC(OCC)C2)=O)C1(C)C N1(C(C2CCN(C(C3C(C)OC(=O)N3)=O)CC2)=O)CC2CC(C(N)=O)(C2)C1 c1(C(N2C(C(=O)Nc3nc(C)nc(O)c3)CSCC2)=O)nc(C)c(C)[nH]c1=O c1(CN2CC(C(=O)Nc3ncc(C(C)=O)s3)SCC2)c(F)cc(C#N)cc1F Cc1cc(=N)[nH]cc1C(N1CC(CC(C)NC(=O)CC(O)c2ccccc2)C1)=O Cc1ccccc1CC(N1CCC(CF)(NC(=O)CC2CC(F)C2)C1)=O c1(N(CC(=O)N(CC(=O)O)CC2CCCCO2)CC)ccccc1C#N.CO N1(C(c2c(C)nc(C)o2)=O)CCC2CC(C1)CN(C(C1(C(C)C)CCCO1)=O)C2 C1(N(C(C2(C)CCN(C)C2)=O)CC)CCN(C(=O)OC(C)(C)C)C12CC2 C12(C(=O)NCC(C)OCCO)CCC(CN(C(=O)CCS(C)(=O)=O)C1)C2 c1(C(=O)NCC(C2CCN(C(C3C4CCCC34)=O)CC2)C)ccc([N+](=O)[O-])o1 C1(SC)CN(N(CC2CCCO2)Cc2cccs2)CC(F)(F)C1 c1(-c2cn(CCCCCNC(C(C)NC(CC)=O)=O)nn2)cc(Cl)nc(=N)[nH]1 C(=O)(C1=CS(=O)(=O)CCC1)N(C1CN(C(=O)CCO)CC12CC2)C.C1COC1 c1(C(N2CC(CNC(c3cccc(C)c3)=O)OCC2)=O)nnc2ccccn12 C1(C(=O)NC(CNC(C(C(C)C)O)=O)(C)Cn2cccn2)CC1C1(C)COC1 C(C)(C(=O)NCCOC1CCN(C(C2CC(=O)CCO2)=O)C1)(C(C)C)OC C(=O)(C(C)C(CC)CC)NCCC(C)N(C(Cc1c(CC)noc1CC)=O)C C1(CCNC(c2coc(CC3CC3)n2)=O)CCCN1C(c1coc(Br)n1)=O N(C(=NCCC(O)(C(F)(F)F)c1nccn1C)NC1CCCOC1)CC(C)C Cc1cccc(O)c1C(=O)NC1CCN(C(=O)C=CC2CCCO2)CC1 C1(C(=O)NCCc2ccc(F)nc2)C(C2CC2)CCN1C(c1ccccc1O)=O Cn1nc([N+](=O)[O-])cc1C(N1CCC(CO)C(NC(C2(C)CCCC2)=O)C1)=O c1(C(C(=O)NCC(n2cc(C3CCCC3O)nn2)C)O)ccccc1C(F)(F)F C1CN(C(=O)CC2(O)CCCN(C)C2)CCC1(F)F.C=CC1(C(=O)NC)CCC1 c1(C(N2C(C)(C(N3CC4CC4C3C#N)=O)CCC2)=O)cc(F)c(F)cc1F N1(C(C(N2CCNC2=O)C)=O)CC2(C1)SCCC2NC(=O)OC(C)(C)C c1(NCc2cn(-c3c(OC)ccc(N)c3)nn2)ccc(Br)c2cccnc12 N1(C(c2c(C)coc2)=O)CCC(C2CC2)C1CNC(c1ncc(C(F)F)s1)=O n1(CC(=O)NCCN(C(=O)C(C)C(CC)CC)CCC)cc(Cl)c(O)nc1=O C1(C(N(C(CC)C(=O)NC2C=CCCCC2)C)=O)CC12CCCCC2 C1(CNC(=O)C=CBr)(NC(=O)CCNc2ccccn2)CCOC1 C1(CNC(c2ccc3c(n2)OCCO3)=O)CC(N=c2[nH]c3ccccc3s2)C1 C1CN(C(=O)CCNc2cc(F)ccc2F)CC1(C)C.CC(F)(F)C1(C=O)CC1 C(=O)(CC(CNC(C1(F)CCOC1)=O)C1CCC1)NCCSC c1(NC2C(C)CCN(C(c3cc(Cl)nnc3O)=O)C2)ncnc2ccsc12 c1(C(N2C(CNC(C3(CC=C)CC3)=O)CCC2)=O)cnn(C2CC2)c1Br C(CC(=O)N1CCC(c2ccncc2)C1)(C(F)(F)F)NC(COC)=O C(N=c1[nH]c(=NCCc2cnco2)[nH]c2c1SCC2)C1C(C)(C)CCCO1 N(C1CCCc2c1[nH]c1ccc(Br)cc21)C(C1C2CCNC12)=O Cc1conc1CC(N1CCC(CCNC(=O)CCC#N)C1)=O Nc1cccc(CC(=O)NCCC2CCCC2)c1.C(=O)C=CC=O.C1CC1.N C1(NC(C(CN(C)C)O)=O)CC12CCN(C(=O)C1=CCC1)CC2 c1(NC(C2CCN2Cc2cnc(Cl)cn2)=O)ccc(Cl)cc1Br C1(C(=O)NCc2cccc(F)c2)CC2(CC(NCc3ccc(Br)[nH]3)C2)C1 Cc1cccnc1CCC(=O)NCC(CO)NC(=O)C(C)C=Cc1ccccc1 N1(C(CC2N(C(c3c(C)cc(F)cc3)=O)CCC2)=O)CCC2(CC1)CCN(C)CC2 C1(C(=O)NC2C(C(=O)NCCC(C)CO)COC2)COCCC1C C1(C(N2C(C(=O)NC3CCCC(OC)C3)CCC2)=O)CN2CCN1CC2C c1(NC(C(N2CCC(OCC=C)C2)C2CCSC2)=O)ccccc1OC C1(SCC)OCCC1C.[nH]1ccnc1-c1ccccc1.c12nnnn1C1(CC1)C2N Cc1c(Cl)cnc(N2CC3C(NC(=O)CC4=NNC(=O)C4)C3C2)c1C#N N1(CC)CCOC(C(N2CCC(CO)(NC(=O)CCOCC(C)C)C2)=O)C1 O=C(NNC(=O)c1cnn(C2COC2)c1)N(c1ccccc1)CCO C1(CCCNC(=O)CCc2nc(C3CC3)no2)CN(C(C2CCCO2)=O)CCO1 N1(C(CC(C(F)(F)F)NC(c2cc(C)nnc2O)=O)=O)CCC2(CNC(=O)C2)C1 N(C(=S)N1CCC(CCC(=O)OC(C)(C)C)CC1)CCC C1(N(C(C(=Cc2ccccc2)CC)=O)C)CCCCN(C(C2(F)CCOC2)=O)C1 c1(C(N2CC3C(C(=O)NC(c4cccc(O)c4)C)(C3)C2)=O)cnn2cccc2c1 C1(CC(=O)NC2(CC=C)CCOC2)C2CCC(C2)N1C(=O)C(C)CC=C C1(CNC(C2CCC(CC)O2)=O)C(C2CC2)CCN1C(=O)C1=NNC(=O)C1 N1(C(C=C(C)C2CC2)=O)CCC2C(C1)CN2C(c1csnc1Cl)=O N1(C(CC#C)=O)CCN(C(c2cc(F)cnc2OC)=O)CC1C#N c1(CNC(N(C)Cc2cc3ccccc3o2)=O)csc2cccc(Cl)c12 N1(C(c2ocnc2CC)C(=O)NCCCCCC)CC2CC3CC2C1C3OC C1(CNC(C(C)(C)CCF)=O)C2CCCC1N(C(=O)CCC(N)=O)C2 C1(C2CN(C(c3cc(C4CCCCC4)[nH]n3)=O)C2)(NC(C=COCC)=O)CC1 C(=O)(C1=CCS(=O)(=O)C1)N1CC(CN(C)C)CC1(C)C c1(C(=O)NCC(CC)NC(=O)Cc2ccccn2)c(Cl)n[nH]c1C c1(C(N2CC3C(C(=O)NC(c4cccnc4)CC)(C3)C2)=O)cc(F)c(C)cc1F C1(NC(C2CC(C)SCC2)=O)CC2(C1)CN(C(C1(C(N)=O)CC1)=O)C2 C(=O)(C#Cc1cccc(N)c1)N1CCN(CC(C)(C)OCC(=O)OC)CC1 c1(C(=O)NC2C(n3cc(C(CC)(C)C)nn3)CCC2)cc(C#N)oc1C c1(CNC(C2CC23CC3C(=O)NC)=O)cccc2c1SCCC2.c1cccs1 C(=O)(CC(COC)NC(c1ocnc1C)=O)NCC#CC Cc1nn(C)c(N)c1C(N1CC2CC2(CNC(c2ncn(C)n2)=O)C1)=O c1(CC)ccc(Cl)c(C(C(=O)NCc2ccco2)N(C(C)CC#N)C)c1 C1(C=O)COc2ccccc2O1.C(=O)(C(C1CCC1)C1CCC1)N(CC)CC.N O=CN1CCOCC1C(N1CCC(NC(=O)CCCn2cccn2)C(CO)C1)=O CON(CCC(=O)Nc1cc(O)cc(F)c1)C(=O)c1cccc2c1CCC2 c1(C(=O)NCC2(C)CN(C(C=CCC)=O)C(C)(C)C2)cnc2c(F)cccc2c1 Cc1ccc(F)c(C(=O)NCCC2CCCC2)n1.C1(C(=O)N)CC1.C1CCC1 N(C1CCOc2c(Br)cccc21)C(CCCC#C)c1nnnn1CCC CCC(O)C(F)(F)C(=O)NC1CCN(C(=O)CCOCCOC)C1 c1(CC)cc(C)c(C(=O)NCCN2CCCCC2)o1.C(=O)(CC)N.C(C)=O c1(C(N(C(C)CNC(=O)Cc2cccs2)C)=O)cc(-n2cccc2)ccn1 N1(C(C2CCC(CC)O2)=O)C2CCCC1CN(C(=O)Cn1cccn1)C2 c1(N(C)Cc2ccc(Cl)c(F)c2)nc(N2CC(F)C(F)C2)nc2ccc(Cl)cc12 C=C(CN=C(NCC(F)F)NC1CCOCC1F)c1ccccc1 C1(CNC(C2(SC)CCC2)=O)CN(C(C2CCSC2)=O)CC1(C)C N1(CCC#C)CCN(C(=O)CCCOCC)CC1.C1(=O)C(C(C)C)OC2CN1C2 c1(CCC(=O)N(C)CC2(NC(Cc3nnc(C)o3)=O)CC2)cccnc1Br C(=O)(CC(C)(C)C#N)N(CC(=O)NCCC(O)C1CC1)C O=C1CN(C(C2CC(F)C(=O)N2)=O)C(C(=O)NCC2CC2C2CCC2)CN1 C1(C)(C(N(C)CCOCCNC(=O)Cn2cnnc2O)=O)CCSCC1 CC1(F)CCCCN(C(C2CC(NC(c3cc(C4CC4)no3)=O)C2)=O)C1 N1(C(c2c(CCC)[nH]cc2)=O)CCCC(NC(=O)COC(F)(F)F)C1 C1(c2n(CCC)nnn2)(NC(c2nc3c(s2)CCC3)C)CC(C2CCOCC2)C1 C1(NC(C(C)c2ccsc2)=O)CCC(CNC(=O)Cc2cccc(F)c2)CC1 c1(CC(N2CCC(O)(CNC(=O)CCc3cnoc3)C2)=O)ccc2ocnc2c1 Cc1ccc2c(C(=O)NCC(O)COCCOCC3CC3)cnn2c1C CCCCC(CC)CC(=O)NC(Cc1cc[nH]n1)C(=O)NCC(C)(O)CC(C)C C(=O)(CCCCC(C)C)N1CC(OC)(CNC(=O)C(C)CO)C1.c1ccccc1 C1(NC(C(CC)C)=O)CCCCCC1C(N1CC2(CCC2)C1)=O c1(C(N(C(CC)C)C)=O)n[nH]c(C)c1F.C12CCN(CC1)C2 c1(CC)nc(C)c(C(=O)NCc2ncoc2CC)s1.c1(C=O)ccno1.N CC(C)C(N=[N+]=[N-])C(=O)NC1CC(CC(N2CCC(C)(C)CC2)=O)C1(C)C c1(C(N2C3CN(C(C(=O)NCC)=O)C(CC3)C2)=O)cccc2c1OC(C)C(=O)N2 Cc1cc(O)ncc1C(=O)NCCCCCNC(C1CC1(Cl)Cl)=O C1(CCNC(C2CC2C(F)(F)F)=O)CN(C(=O)CN2CCCC2=O)CCO1 C#CCCC(C(=O)NC(c1ccc(C)cc1)C)NC(=O)C(C)=CC=C c1(C(=O)NC2CC(CNC(c3cc(C)c(C)[nH]3)=O)C2(C)C)n[nH]c2c1CCSC2 C1(CC=C)(NC(=O)C=O)CCN(C(C2CCOCC2)=O)C1.C1CC(F)C(=O)N1 N(C1CCOc2c(F)cccc21)C(c1ccc2c(c1)COCCN2)=O c1(C(C)C(=O)NCCNC(=O)CC2CCCC23CC3)c[nH]c2ccccc12 Cc1[nH]nc2c1CC(C(N1CCCC1CNC(c1cnc(Cl)c(Cl)c1)=O)=O)CC2 C1(C(=O)NC(c2nn[nH]n2)CC)CCN(C(C2CCC(C)O2)=O)C(C)C1 O=C(CCCCc1cnn[nH]1)NCCNC(=O)CCCCN1CCCCC1 n1(CC)nnc2cc(C(=O)N)ccc12.C1(C(N2CCC2)=O)CC2(CCOCC2)C1.C c1(C(N2CCC(Cn3cc(-c4cncc(C)c4)nn3)CC2)=O)nc(C)ccc1F C1(NC(N(CC=C)Cc2cccc(SC(F)(F)F)c2)=O)CCC(O)C1(C)C c1(C(=O)NC(C2CN(c3nnc(CC)c(CC)n3)C2)C)ccc2nc(O)[nH]c2c1 CC1N(C(C2N(C(C3CSC3)=O)CC23CCCC3)=O)CCCC12CCC2 c1(C(=O)NC2CC(OC)CN(C(=O)C(O)CSC)C2)cc2c(C)ccc(F)c2[nH]1 CC(CCCCN=c1[nH]c2ccc([N+](=O)[O-])cc2s1)NC(C1CCOC1C)=O c1(C(=O)NCC2CCCC2)ccc(=O)n2c1COCC2.C(=O)(C(O)C1CC1)N CC1CCC(C)(C=CC(=O)NC)C1(C)C.C1CCN(C(C2(F)CC2)=O)CC1 N1(C(c2c(C)cccn2)=O)CCN(C(C23CC(C)(CO2)C3)=O)CC1CO C1(CC=C)(NC(C2CCCC(F)C2)=O)CCN(C(c2ccc(N)c(O)c2)=O)CC1 C12(C(=O)NCCNC(C(C(C)C)OC)=O)CCC(C(C)=O)(CC1)CC2 c1(SCCNC(c2n(CC=C)nnn2)CCOCC)cccc(F)c1 C=CC(C)CC(=O)N(CCCNC(C1CCCC1c1nc(S)n[nH]1)=O)C c1(C(N2C(CNC(Cc3cc(C)no3)=O)C=CC2)=O)oc(C)cc1C Cc1nc(NCCCc2nc(C3CC3)n[nH]2)cc(N2CCC3CC3C2)n1 N1(C(c2ccc(SC)s2)=O)CCOC2(CCC(NC(=O)CCCC(C)=O)CC2)C1 C(=O)(C(O)C(C)C)NCCC1(NC(C(C)NS(CC)(=O)=O)=O)CCC1 C1(NC(CC=CC=C)=O)C=CCN(C(=O)CCC(C)C)C1 c1(NC(C(CO)SC)C)ccc(S(=O)(=O)NC2CC(C)(C)OC2(C)C)cn1 c1(NC(CN(C(=O)C2=CCCC2)C(CC)C)=O)ccc(-c2ccsc2)nc1C c1(NC(=O)CN2CCCCC2C(F)F)ccc(C(F)(F)F)cc1 CC1CCC(C(=O)NC)N1C(C12CC(C#N)(C1)C2)=O.C1CC1.C1CCC1 c1(NCCOCCN(CC(c2ccccc2)OC)C)cn2cccnc2n1 n1(CC(CN(CC)Cc2cc(Br)ccc2F)=O)cc(C#N)ccc1=O c1(C(=O)NC2(CO)CN(C(=O)Cc3cc[nH]c3)C2)cnc2[nH]c(O)nc2c1 c1(NC2CCN(C)C2)ccc(S(=O)(=O)NCC(=O)Nc2ccc(F)cc2)cc1Cl N1(C(C2C(COC)(COC)C2)=O)CCCC1.c1(C=O)sc(C)nc1C.C C1(CNC(C=C(C)C(F)F)=O)CCC2(CN(C(c3ccsc3Cl)=O)C2)O1 CCC(CC(F)F)C(=O)N(C1CCN(C(=O)C(O)C(F)(F)F)C1)CC c1(COC(C(C2CCC2)OCC)=O)cc(C(F)(F)F)no1 c1(-c2n(CCC)nc(C)c2)[nH]nc2ncc(C(=O)NCc3cc[nH]n3)cc12 C(=O)(C(C)CS(C)=O)N1CC(O)(CNC(c2c(OCC)nccc2)=O)C1 NC(=O)CN=c1[nH]c(=NCc2ccccc2Br)c2ncccc2[nH]1 CC(CCCO)CN=c1[nH]c2c(c(=NCCCc3cccc(Br)c3)[nH]1)CCC2 c1(NC(=O)C(c2ncccc2F)(F)F)ccccc1OCCOc1ccc(I)cc1 N1(C(CCCOC(C)=O)=O)CC2C(C)C2C1.c1(C=O)c[nH]cc1C(C)(C)C.N CC1(CNC(C2CCCCS2(=O)=O)=O)CN(C(=O)Cc2cccc(F)c2)CCO1 Cc1cc(NC(C23CC(NC(C4CCC(F)(F)C4)=O)(C2)C3)=O)cc(O)c1 c1(C(N(CCC(C)(C)O)C)=O)n[nH]c2c1CN(C(c1ccc(=N)[nH]c1)=O)C2 CCC(O)C(F)(F)C(=O)NC(C1(O)CCN(C(c2cccc(S(C)=O)c2)=O)C1)C CCCC(C)C(=O)N1CCCC(N(C(=O)Cc2sc(C)cc2C)CC)C1 C1(NC(c2c(C)nsc2)=O)CC(NC(c2coc(Cl)c2)=O)C12CCOCC2 CCCC(CNC(=O)C(C)C(=O)OC)C(=O)NC(C)(C)CCO c1(C(N2CCC(C(C(=O)O)F)C2)=O)cnn2c1S(=O)(=O)CC2 C1(C(=O)NC(c2cnn[nH]2)C)C2CCCC2CN1C(=O)CSC(F)(F)F N1(C(C=CC=CC)=O)CCCC(O)(CNC(=O)CCS)C1.C1CCCC1 CCC(C(=O)N1CCC(N(C(=O)CC2(N3CCCC3)COC2)C)C1)NC(N)=O c1(C(=O)NCCNC(c2n(C(CC)C)ncc2)=O)ccc(C#N)cc1O CC1CC(N=c2[nH]c(-c3ccccc3)nc(=NCC(C)CCO)[nH]2)C1 C1(C)CCC1.c1(C2C(F)(C=O)C2)ccccc1.C(CC(=O)N)NC(=O)NC C1(NC(C(C)OCC)=O)C2CCC1N(C(=O)C(F)(F)c1ccncc1)C2 C1(OC)CCC2(C(=O)NC3(C(=O)NCCCCF)CSC3)CC12 N1(C(CCC2C(C)C2)=O)CCC(C2CCCN(C(=O)C=Cc3cccnc3)C2)C1 C1(NC(CN2C(C)CC2)=O)CN(C(=O)CCc2ccncn2)CC1n1ccnn1 N1(C(c2c(OC)nsc2)=O)CCC(NC(=O)Cc2cnsc2)C1C c1(C(=O)OC)cnccc1C(=O)N.c1(C(N2CCCC2)=O)cnnc(C2CC2)c1 C1(C(N2CC(C)CC2)=O)C2CCC(CC2)C1C(F)(F)F.C(=O)C(F)=C1CCC1 C1(C(=O)NC(c2ccccc2)COC)CC(O)CN1Cc1ccc(F)nc1 c1(C(=O)NCC(C)(CC)NC(COCCOCC)=O)cc(Br)oc1C c1(C(=O)NC2CN(C(C3(C)CC(C)C3)=O)CC2C)cc(Br)n2ccccc12 Cc1cc(OC2CCN(C3CC3)C2)cc(NC(n2ccnc2)=O)c1.CC(F)(F)F C1(CNC(C=C(CC)C)=O)C(C2CC2)CCN1C(c1cccc(CC)n1)=O N1(C(CCN(C)CC)=O)CCC2C1CCCN2C(c1cnc(O)[nH]1)=O C1(CCC)CN(C(c2nc(C)ccc2F)=O)CCN1C(=O)CCC1(C)CC1(F)F CC(=O)CCCC(=O)NCc1ccc(C(=O)NCC(C)CC(F)(F)F)s1 C1(CN(C(c2c(C)[nH]cc2)=O)C)CCCCN1C(C1CC(C2CC2)C1)=O CCCCCCC(C)C(=O)NC(C1CCN(C(=O)C=C(C)C(C)(C)C)CC1)CO c1(-c2cccc(C)c2C)cnc2ncc(C(=O)NCC(N)=O)n2c1 C(c1cccnc1)=CCNC(C1CC(O)CN1C(=O)CC1CCC(O)C1)=O Cc1cc(C)c(C)c(C(=O)NCC2CC2)c1C.c1(C2C(C=O)C2)cccnc1 C#CC1SCCN1C(=O)C(=O)N(C)C.c12ccccc1N(CCN(C)C)C2 c1(Oc2c(CN(CC(C)CC(F)F)C)cccc2)cc(Cl)cc(Cl)c1 C1(NCc2ccc(OCC=C)c(OC)c2)CC2CCC1N(C)C2 CC1(C)CCC=C(C(=O)N2C3CCCC2CN(C(=O)C(C)(O)C2CCOC2)C3)C1 N1(c2ncc(C)c(C)n2)CCN(Cc2cnc(Br)c(F)c2)CC1C#N CC1OCCCC1C(=O)NC.C1CCN(C(=O)Cn2ccc(C(F)(F)F)n2)CC1 N1(C(c2nc(C)c(C)[nH]c2=O)=O)CC2CCCC(C1)N2Cc1cccc(Br)c1F C1(NC(CCCOC(C)C)=O)CN(C(=O)C(C)C2CCCO2)CC2(CC2)C1 c1(C(N2C3CC(NC(=O)Cc4cnsc4)(C3)C2)=O)nnc(O)cc1O c1(C(=O)NC(CC)CN(C(=O)C=CC(C)(C)C)C)ccnnc1.C(C)C.N C1(c2nnnn2C2CC2)(NCCC2CCC(C)(C)C2)CCCOCC1 C1(NC(c2c(C)c[nH]n2)=O)CN(C(C2CC3C(C2)C3(C)C)=O)Cc2ccnn2C1 Cc1cc(CNC(=O)C(Cc2cc[nH]n2)NC(=O)CO)c(C)s1.CC=O C(=O)(CC1=CCN(C(=O)CCn2ccnn2)CC1)NC(CCOC)CO C1(NC(C(CCC#C)O)=O)CCSC12CN(C(c1ccc(Cl)cc1)=O)C2 CS(=O)(=O)c1coc(C(N2CCC3CN(C(=O)CC4(O)CCC4)CC23)=O)c1 c1(N2CCC(N(CC#C)C(C3CCC(C)(C)O3)=O)CC2)ccnc2ncnn12 c1(C(=O)NCC(n2cc(C(CC)N(C)C)nn2)C)cccc(C(F)F)n1 c1(OC)cccc(NC(=O)CC(CC2CC2)NC(C2CCCCC2)=O)c1 N1(C(C23CCC(OC)C2C3)=O)CCC(N=[N+]=[N-])(C(=O)N(CC(C)C#N)C)C1 C=CCCCCCC(=O)N1CCN(C(=O)C(C2CCCC2)OC)CC1CO CCCC(O)CC(=O)N(CC(C)N(C)C(c1cnc(O)s1)=O)C C1(C)(C(N2CCC(NC(C34C(C)(C)OCC3C4)=O)C2)=O)CCC2(CC1)OCCO2 CC(C)CC(C(=O)NCC1CC(CF)C1)ONC(=O)Cn1ccnn1 C1(C(N(C(C(=O)OC)C)C)=O)(NC(c2nccs2)=O)CC(F)C1 C(C#Cc1ccc(C(F)(F)F)cc1)N(CC(c1ccccc1)C)C N1(CC)CCC(c2nnnn2Cc2cccs2)(NCCCP(C)(C)=O)CC1C N1(C(C2CCC(C)(C)CO2)=O)CC2CCN(C(c3csc([N+](=O)[O-])c3)=O)C2C1 c1(NC(Cc2nc(C(C)C)on2)=O)cc(Br)cnc1Cl.C12COCCN1C2=O c1(NCC(C)(C2CC2)NC(C=C(C)c2ccco2)=O)cc2nncn2cn1 CC1(C2CCN(C(C3CCCC(NC(=O)Cc4cnns4)CC3)=O)C2)CC1 CC1=C(C(=O)NC(C)C(C)(C)C(=O)N2CCC2(C)C)CCCO1 C1(CC(=O)NCCC2(NC(C(C)c3ccco3)=O)CC2)CC2(CCC2)CO1 N1(CC(N2CCC(NC(c3c(CC)scc3)=O)C(O)C2)=O)CCn2ccnc2C1 C(=O)(CS(=O)(=O)CCOC)NC(CNC(C(CCC)(C)O)=O)CO C1(CN(C(c2c(CC)nc[nH]2)=O)C)CCN(C(C2CCC3(CC3)C2)=O)CC1 c1(CCC(=O)NC23CC(CNC(CC=C(C)C)=O)(C2)C3)cccnc1Cl CC1CC(C(=O)NCCCCNC(C2(C(F)(F)F)CC2)=O)Cc2nn[nH]c21 C=CC1CCCC(NC(C2CN(C(c3cn(C(C)C)nn3)=O)CC2F)=O)C1 C1(C(=O)NCCC(C)N(C)C(c2cc(C#N)ccc2O)=O)CN2CCN1CC2C CCCC(C(O)C(=O)NCc1cncs1)NC(=O)C(C)(C)CCF c1(N2CCC(O)(C(C)NC(=O)C(C)(C)CF)CC2)nc(C#N)ncc1Cl c1(OC)ccc(F)cc1C(=O)NCC1CN(C(=O)C(F)C2CCC2)CCO1 N1(C(COCCCC)=O)CCN(C(=O)C(C)(C)C(F)(F)F)CC2CCCCC12 C1(CNC(CC2CCCC(NC(c3n(C)c(Cl)nc3)=O)C2)=O)CCOC(C)(C)C1 n1(CC(=O)NC(CC2CN(C(c3c(OC)n[nH]c3)=O)C2)C)ncc(Cl)c1C Cc1cccc(CCC(=O)NCC(C)N(C(=O)CC2CC=CCC2)C)c1Br N1(C(CC2CC(C)(C)N(C(=O)Cc3cnsc3)C2)=O)CCn2cncc2C1 CCC(CC(=O)NCCCCC1CN(C(C2CCN(CCOC)CC2)=O)C1)SC C1(C(NOCC2(C)CC2)=O)C(C2CC2)CCN1C(C1CCCOC1)=O C1(NC(C(CC)NC(N)=O)=O)CCN(C(=O)CCn2ncn(C)c2=O)CC1O Cc1c(C(=O)N(CC(O)CN(C)C(c2nc(=O)n(C)[nH]2)=O)C)nnn1CC c1(C2C(C)C2)cc(=NC(=O)C2CC2C2CC3CC3C2)[nH][nH]1 C1(C)(C=O)CCC(=O)N(C)C1.Cc1nc(C(N2CC3CC3(C)C2)=O)n(C)n1.N N1(CC(=O)N(C)Cc2ccccc2F)CCC(CCn2cc(C3CC3)nn2)CC1 N1(C(CC=C)=O)CC2OCC(C(=O)NC(c3ccc(F)c(F)c3)C)C2C1 C(=O)(C1(C)CCCc2ccccc21)N1C2CN(C(C3C(C)(C)C3)=O)CC1CCC2 c1(C(=O)NC2CN(C(C3CC(F)C3)=O)CCC2F)[nH]nc([N+](=O)[O-])c1Cl CC(C)CC(C(=O)N(CC(C)NC(=O)CN1CCCNC1=O)C)C(N)=O c1(OC)ncc(Br)c(C)c1NC(C1CN(C(=O)C=CC2CC2)CCC1O)=O c1(CC(=O)N)ccc(F)cc1.c1(CC(=O)NCC2CC2C)csc(Br)c1 CC1CN(CC2CCS(=O)(=O)C2)CC1N=[N+]=[N-] c1(COCCCNC(=O)C(=O)NCC2CCC(F)C2)ccc(F)cc1 N1(C(C23CCC(C)(CC2)OC3)=O)CCc2ccc(C(=O)O)nc2C1 C12(C(N3CCCC(C(=O)NCc4n(CC)nnc4C)C3)=O)CCCN(CC1)C2 C(=O)(C(C)CCC(C)(C)C)NCCC1N(C(C2C(CC)OCC2)=O)CCSC1 c1(C(=O)NC2CC(NC(c3c(C)ncs3)=O)C2)cc2c(s1)CCC(C)C2 C1(CNC(CC2(SC)CN(C(c3c(NC)cccc3)=O)C2)=O)CCC=CCCC1 C1(NC(=O)COc2ccccc2)CC2CC1N(C(c1ccnn1CC(F)F)=O)C2 C1(CNC(C2(COC)CCN(C(CCCC)=O)C2)=O)CC(C2CC2)=NO1 C(=O)(C1=Cc2ccccc2OC1)N(C1CC2N(C(CC(=C=C)C)=O)C(CC2)C1)C C1(C(N2CC(O)(COC)C2)=O)CC2CN(C(=O)C(C)(C)COC)CC12 Cc1cccc2c(C(=O)NCC3CCN3C(C3CC4(CCC4)CO3)=O)csc12 c1(CC(=O)NCC(CCNC(C=CCC)=O)O)ccc(F)cc1C CCS(=O)CC(=O)N1CC=CC1CNC(=O)Cc1cccnc1OC N1(C(C(C(C)C)SC)=O)CC(C)OC2(CCN(C(=O)Cc3cncnc3)C2)C1 C1(CC(=O)NCCN(C(=O)C(=O)Nc2ccccc2)CCC)CCNC1=O c1(C(N(CCC)CCNC(C2(F)CCCOC2)=O)=O)cc2ccccc2n1C C1(CC(=O)N(CCC(N2CCC(OC)C2)=O)C)CCCN(C)C1 C(CCOCCO)(C(=O)N(C)CC1CCCN(C)C1)NC(C(CC)SC)=O c1(C(=O)NCCCC(C)NC(COC(C)C)=O)ccc(Cl)c(Br)c1F n1(CC)ccnc1C(=O)NC(C(=O)NC(CCO)C1CC1)c1cccs1 C1(CNC(c2cc(SC)oc2)=O)CCN(C(C2CCCC2(F)F)=O)C1(C)C c1(OC2(C(N(CCC)CCc3nnc(-c4ccco4)o3)=O)CC2)ccccc1 n1(CC(=O)OC)cc(C)nn1.C1(O)CC(C=O)C1.C(C)(C)C.C(=O)N c1(C(=O)NC(CCNC(c2c(CC)csc2)=O)(C)C)cc2c(cc1O)CCCC2 c1(CC(N2CCCC(NC(c3c(C)occ3)=O)C2)=O)ncn2c1CCCC2 CCCC(CCC)CCCC(=O)N1CCC23CCCCC2(C1)C3(F)F Cc1ncc(C(N2CCN(C(=O)COCC(C)(C)C)CC2CO)=O)c(C)n1 c1(C(=O)OC(CC=C)CC=C)cc2c(C)nn(CC)c2s1 CC1(C(=O)NC2CCC2)CCC(F)(F)C1.c1(C(=O)N)ccc(C2CCCC2)cc1 C(=O)(C(C1CN(C(=O)C(C2CCCC2)O)C1)OC)NCCSCC=C c1(C(C(=O)N(C2CCN(C(CSCC=C)=O)C2)CCC)C)c(F)cccc1F c1(C(N(CCCNC(CC=CCC)=O)C)=O)cn(CCCC)nn1 CC1CCN(C(C2(C)CC3CC3C2)=O)CCN1C(c1ccnc(CN(C)C)c1)=O c1(NC(=O)COC(c2n[nH]c(-c3cccnc3)n2)=O)ccc(C(F)(F)F)cc1 c1(C(N(CC(=O)N(CCN(CCCN(C)C)C)C)C)C)ccc2ccccc2c1 C(CC(C)(C)NC(=O)CSCc1cscn1)NC(C1(CC)CC1)=O C1(C(CNC(CNC=O)=O)F)CCN(C(c2ccc(-n3cccn3)nc2)=O)CC1 C1(C)(NC(c2cn(C)nn2)=O)CCCCC1C(N1CC2CCC2(C)C1)=O N1(C(CC2CC(=C)C2)=O)CC2(CC(C(N3CCOC(CCO)C3)=O)CO2)C1 CCCCCCC(C)C(=O)NCC1(NC(=O)CN2CCCNS2(=O)=O)CCC1 C12(C(=O)NCC3C(C)CCN3C(=O)CCCn3cncn3)CC1COC2(C)C C1(NC(c2ccc3ccoc3c2)=O)CCSC12CN(C(c1cc[nH]c1)=O)C2 C(=O)(C#CC1CC(=O)C1)NC1(C)CCC(NS(=O)(=O)c2cccs2)CC1 C1(O)CN(C(=O)C(O)CC2CCCC2)C1.c1(C(=O)NC)cc(C2CC2)on1 C1(CNC(c2nc(C)[nH]n2)=O)CN(C(c2cc(C(F)F)nn2C)=O)CC1C C1(CC(=O)O)CC(NC(=O)Cn2cc(-c3cc(Cl)ccc3Cl)nn2)C12CCC2 c1(NC(C)=O)cc(F)ccc1NC(c1nn(C)cc1)=O.c1(C=O)ccco1.C c1ccc2c(c1)CCC2N1CCCC(OCc2ccsc2)C1 c1(C(=O)NCC2C(NC(=O)CCCCC3CC3)C2)c(Cl)ccc2cccnc12 c1(OC)cccc(C(N2CCC(CN(C(C3CCOC3C)=O)C3CC3)CC2)=O)c1 c1(C(=O)NCCN(C(c2c(OC)cc(C)s2)=O)C)[nH]cc2c1CCS2(=O)=O C(CC(C)(C)C)(C(=O)NC(C)(C)CCNC(C1COCCO1)=O)OC c1(C(=O)NCC(C)N(C(=O)Cc2ccno2)C)ccn(C2CCCC2)n1 C1(NC(C(CCC)OCC)=O)CC12CCN(C(c1cc(OC)n(C)n1)=O)C2 c1(C(=O)NC2(CCC(=O)N)CCC2)ncnc(O)c1F.n1(C2CC2)ccnn1.C N1(C(C2CC(=C)C2)=O)CCN(C(c2cnsc2)=O)C(C)C1C c1(NC)cnc(C(=O)NC(C)(C)CNC(=O)C=CBr)cn1 c1(OC)ccc(CO)cc1C(N1CC2CC2C1)=O.c1(C=O)ccc([N+](=O)[O-])o1.N C(c1ccncn1)=CC(=O)NCC1CC(NC(=O)CCCc2cccnc2)C1 N1(c2cc(NCC(C)C)ncn2)CCC2(CC1)CC2(C)C(N1CCCC1)=O C12(CC(=O)OC)CCCCC1N(C(=O)CC1(OC)CCCCC1)CCC2 c1(NC(C(CC)N(C(=O)CC(=O)N(C)C)C)=O)cnc(OC)nc1 c1(C(N(CC(O)CN(C)C(C2CC3C=CC2O3)=O)C)=O)c2c(nn1C)CCCC2 N1(C(C(CC)c2cccnc2)=O)CC2(CCN2C(=O)CC(C)(C)O)C1 Cc1ccc(CCNC(=O)NC(CNC2CCCCC2)CC(C)C)cc1 C(=O)(C(O)C1=CCCCC1)NCC1N(C(c2c(C)nncc2)=O)CC1 c1(C(=O)NC2C(C)N(C(=O)CC3CC3(C)C)CC2)csc2ccc(F)cc12 O=C(C1=CCCCO1)NCC12CCC1CCN2C(c1cc(C2CCCC2)[nH]n1)=O CCCC(O)C(=O)NCCCN(CCCNC(C1CC(C)C1)=O)C C1(CNC(c2csc(O)n2)=O)CCCCN1C(C1(c2ccsc2)CC1)=O c1(C(N2C(CCNC(C(C)OCC)=O)CSCC2)=O)cccc2c1NCC2 C1(OC)CC(NC(=O)CN(C)C)CN(C(=O)C(N2CCOCC2)C)C1 c1(C(N2CCC(n3cnnn3)C2)C(=O)NCC=C)ccc(I)c(C)c1 C(=O)(C1CCCc2c[nH]nc21)NC1(COC)CN(C(=O)OC(C)(C)C)C1 C1(C(N(C(C)CN(C)C)C)=O)CCCN1NC(=O)CC1CCC1 CC1(C)CCc2cc(C(N3CCC4CC3CN(C(=O)C(O)C3CC3)C4)=O)ccc21 N#Cc1cnn2c1CN(C(c1cc(O)cc(Cl)c1Cl)=O)CC2 C1(N(C(=O)CCC2CCC2)C)CCN(C(=O)C(C2CCCO2)C2CC2)CC1 C1(NC(CC=CCC)=O)C2CCN(C(C3CCOC3c3ccnn3C)=O)C12 N=c1ncn(CC(=O)NC(CC2CCC2)C(=O)NCCCCC2CC2)[nH]1 C(C(=O)N1CCCC(NC(c2cc(C(N)=O)cs2)=O)CC1)(C(C)(C)C)SC Cc1cccc2[nH]c(C(=O)N(C)CCN(C)C(C3COCC(C)(C)O3)=O)cc12 CC(C)C(C(=O)NCCCCCO)NC(C1(C)C=CCCC1)=O c1(C(C)(C)NS(C)(=O)=O)cn(CCCNC(C2COCCO2)=O)nn1 c1(C(=O)NCC(CNC(C2CCC(C)C2)=O)S(C)(=O)=O)ccn2nnnc2c1 c1(C(=O)NCC=CCNC(c2ccc(Cl)c(Cl)c2)=O)ccc2ncncc2c1 C1(SCC(c2cccc(F)n2)C)CN(C(=O)OC(C)(C)C)CCN1C N1(C(C2C(C)C2c2ccccc2)=O)CC(C)C(N=c2c(Cl)c[nH]cc2[N+](=O)[O-])C1 C#CCCCC(C)C(=O)NCCCCC(=O)N(C)Cc1nnc(C)s1 CC(C(=O)N1CCCC(F)(CO)C1)S(=O)(=O)Cc1cccc(Br)c1 C1(C(N(C2CCN(C(CC3(C=C)CC3)=O)CC2)CC)=O)CCc2cncn2C1 C1(CC)C(C(=O)NOC)CCN1C(c1cc(C(=O)OC)on1)=O C1(C(=O)NC(C2CC2)C)C2CC3C(C2NC(C2CCCN(C)C2)=O)C13 c1(N2CCCC(C(C)C)CC2)ccc(S(=O)(=O)N(C2(CO)CCCC2)C)cc1Cl c1(OC)ccc([N+](=O)[O-])cc1-c1ccc(C(=O)NC2CN(C)C2)c(OC)n1 Cc1c(Cl)cc(CNC(=O)CN2CCC(=O)NC2=O)c(Cl)c1C N(C(=NCCCCOC)NC1CCCCC1C)CC(=C)Cl Cc1ccccc1C(c1nnnn1Cc1ccccc1)NCC1=CCSC1 c1(C(=O)OC)c(C(N2CC(O)(CNC(=O)CCCF)C2)=O)cnn1C c1(NC(C2CCCN(C(=O)C(F)(F)Cl)CC2)=O)cccc([N+](=O)[O-])c1Br c1(C(=O)NCCCC=C)cnn(C2CC2)c1C.C1(CC(C)C)(C(=O)N)CCCC1 C(=O)(CCC(=O)NC1CC(CCC(=O)N(C(C)CCO)C)C1)NCC N1(C(C(=O)N(CC(F)(F)CO)CCOC)=O)Cc2ccccc2OC(C)(C)C1 C1(C(N2CC(CCC)C(C(=O)NCc3nonc3C)C2)=O)CCN(OC)CC1 C1(C(=O)NC2C(C)C(C)CCC2)CS(=O)(=O)c2ccccc2O1 C(C(F)(F)C(=O)N1CCCCC1C1CCCN(C(c2cc(=O)cc[nH]2)=O)C1)OC C1(C(=O)NCCn2ccnn2)CC2C=CC1N(C(c1cc(Cl)ns1)=O)C2 c1(C(=O)NCC2N(C(C(CC=C)NC(C)=O)=O)CCC2)c(C)cccc1N.O N1(C(c2ccc(C)s2)=O)CC(CCNC(=O)Cn2ncccc2=O)OC(C)C1 C1(C(=O)NCC2(O)CCN(C(c3n(CC)ccc3)=O)C2)CC(=O)NC1(C)C O=C(C(O)CN1CCCC1)NCC#CC(=O)N1CCC(N2CCC2)C1 c1(CNC(C2CCCN(CCCC3CCC3)C2)=O)ccc2ccccc2c1O C12(CNC(c3c(C)nc(C(C)C)s3)=O)CCCCC1N(C(c1cscn1)=O)CC2 C(=O)(CCC(C)(C)[N+](=O)[O-])NC1C(C(F)(F)F)CCN(C(c2cc(C)sc2)=O)C1 c1(CC)ccc(OCC(=O)NCCCCNC(C2CC(F)C(=O)N2)=O)cc1 c1(C(N(CCC)C)=O)ccc(F)c(C)c1C#N.c1(OC)cc(C=CC=O)sn1 C=CC1(O)CCN(C(C2(NC(=O)CC(C)c3ccco3)CCSC2)=O)C1 c1(OC)cc(CC(=O)NCCN(C(=O)C(OC)OC)C(C)C)on1 C(CN=c1ccnc(C2CC2)[nH]1)(N(C)C(C1CCCC2CCCCC12)=O)C1CC1 Cc1ccccc1C(C(C)NC(=O)C(C1(O)CCOCC1)O)N(C)C C1(NC(C(c2c(C)cncc2)C)=O)CC2(C1)CN(C(=O)C(C)CF)C2 c1(C(=O)NC2CC(Cn3cc(-c4ccnn4C4CC4)nn3)C2)ccc(C)cc1 c1(C=O)cn2cccnc2n1.C1(NC(c2c(OC)ccs2)=O)CCC(F)(C)C1.N CCCC(C(=O)OC)C(=O)NC(C)(C)CC=CC(=O)NC1CCC1(C)C N1(C(COC)=O)CCC(C2CC2)C1C.c1(-c2ccc(C(=O)N)o2)ccc(F)cc1 c1(C(=O)NC(CNC(CCc2c(C)cccn2)=O)(C)C)cc(C)c(N)c(C)c1 C1(N(C(c2cc(CC)[nH]n2)=O)C)CN(C(c2cc(C)ncc2C)=O)CC12CC2 C(=O)(C(F)CC(C)(C)NC(c1coc(COC)n1)=O)NCC(C#C)C(C)C Cc1ccc(C(=O)NC2CCN(c3nnc(C(F)F)s3)C(C)C2)cc1Cl CCC(C(=O)NCC1CC(NC(c2c(Cl)cccc2Cl)=O)C1)C(C)O N1(S(CC(C)C2CCCC2)(=O)=O)CCn2cc(C(=O)O)cc2C12CCC2 N1(C(Cc2cnc(C)s2)=O)CC2CN(C(=O)CCCC(C)C)CC2C1 Cc1cc(O)cc(C)c1CC(=O)NC1CCN(C(C2CC(C)C2)=O)CC1(C)C C#CC1(C(=O)NCCCC2CCOCC2)CCN(C(=O)C2=CCCC2)CC1 CC(C(=O)N1CC(F)CC1C(N1CCOC(C(N)=O)C1)=O)C(C)(C)C C1(NC(C2(CC)CCCN2C(c2cc3n(n2)CCC3)=O)=O)CCOC2(CCC2)C1 CC12CN(C(=O)C(N)Cc3ccc(O)c(O)c3)CC1(C)CS(=N)(=O)C2 c1(CC)ccc(F)c(C(=O)NCCC2CCCN(C(=O)C)C2)c1.c1cn[nH]c1.O c1(C(=O)N)scc2c1CCCC2.C(C)(C(C)C(C)C)NC(CS(=O)(=O)NC)=O c1(OS(CC2(N(C)C)CC2)(=O)=O)ccnc2cc(F)ccc12 C1(CNC(=O)COC2CC=CC2)CCCCN1C(C1CC(F)C1)=O c1(CCC)ccc(C(N2CCC(c3cn(CCOC)nn3)C2)=O)cc1[N+](=O)[O-] c1(C(N2CCC(CN(C(C(CN(C)C)O)=O)C)C2)=O)cn2cnnc2cn1 C1(OC)CCC2(C=O)CCC12.C(=O)(CP(C)(C)=O)N(C1CCC1)C.C(=O)C CC1(C)CCCC1C(=O)NCC1CN(C(C2(CO)CCC2)=O)CCO1 c1(C(=O)NCCCN(C(=O)CCCC(=O)OC)CC)cccc2c1ncn2C c1(C(N(CC(C)(C)C)C)=O)cc2cccnc2[nH]1.C1(C=O)CC2(C1)CC21CC1.N N1(C(C(C)NC(C)=O)=O)CC=CC(NC(=O)C(n2cc(C)cn2)C)C1 n1(CC(=O)NC(C(CO)NC(CC(C)O)=O)C)[nH]cc2c(=O)ncnc1-2 C1(C(N2CC(C)(NC(C(C)C3CCC3)=O)C2)=O)COCCN1CC1CCC1 c1(C(N(CC(CC)NC(C(CC=C)C)=O)C)=O)c(C)ccnc1OCC c1(NC(C2C(=C)C2)=O)ccc(-n2cc(-c3nccn3C)nn2)cc1 Cc1nccnc1C(C)NC(=O)CCN(CCCO)C(=O)CC1CCCC(C)C1 N1(C(C(CCC)c2ccccc2)=O)CCc2[nH]nc(CNC(C3CC3C)=O)c2C1 c1(CC)c(NC(C2CCC(C(F)(F)F)CC2)=O)cnn1-c1ccccc1OC N1(C(C2N(C(c3c(CC)noc3C)=O)CCC2)=O)CCCC(C)(C)CC1 C[n+]1ccn(CC(=O)NCC(Cc2ccccc2)NC(C2CCC(=O)N2)=O)c1 Cc1nn2ccccc2c1C(N1CC(NC(C23CCCC2C3)=O)C(C)C1)=O Cc1cccc(C)c1C(=O)NC1CCC(CNC(=O)C(C)S(N)(=O)=O)C1 C(=O)(C(F)(F)C(O)C(C)C)NCC1(NC(Cc2ccc(C)c(Br)c2)=O)CC1 c1(N2CCC(NC(Cc3c(OC)cccc3)=O)C(C)C2)cc(S(C)(=O)=O)ncn1 C1(NC(C(CCCC)ON=C(C)C)=O)CC2CC(C1)N(C(=O)CCCCSC)C2 O=C1CC(NC(=O)N(CCCO)Cc2cccc(Cl)c2)C(=O)N1 C(CC(=O)NC(C)CCNC(c1oc(C2CC2)nc1C)=O)(C(C)C)OCC Cc1cc(Cl)c(Cl)cc1C(N1CCC(O)C(C(=O)NCc2cncs2)C1)=O c1(-c2c(C=O)ncn2C)ccccc1F.C12(C(=O)OC)CC1CN(C(C)=O)C2.N c1(C(N2CCC(C)(NC(C3CCC3(F)F)=O)CC2)=O)cc2ccc(F)cc2o1 C1CC2COCC(C1)C2.N1(C(CCOCCOC)=O)CCC(C=O)(C(C)C)C1.N C1(N(c2cncc(OC)c2)C(=O)CN2CCN(C)CC2)COC2(CCNCC2)C1 CCC(C)CNC(=O)COCC(C)(C)C.c1(C(=O)N)cc(C(F)F)cs1 C(=O)(C1=CCCSC1)N1CC2C(C(=O)NC(C#C)(C)C3CC3)C2C1 C1(C(=O)NC2CC(C)(NC(C3C(C)(C)OCC3)=O)C2)CCCCCS1(=O)=O C1(NC(c2cc(Cl)cs2)=O)C2CC(O)C1N(C(=O)C(F)=C1CCCC1)C2 c1(C2C(C(NC)=O)C2)ccc(F)cc1C.c1(CC)ccc(C(=O)N)o1.C1CC1 C(=O)CCC(F)(F)F.c1(C=O)cc(C)c(O)nn1.C(C)(C)(C1(C)CC1)OC Cc1cc(O)n2ncc(C(N3CCC(NC(C45CC(C)(CCO4)C5)=O)C3)=O)c2n1 Cc1ccc2cc(C(=O)NC3CCCC(C)C3)cn2c1.C1(C(=O)N)CC(C)(O)C1 c1(C(=O)NCC(F)CNC(c2cn(C3CCC3O)nn2)=O)ccc2[nH]ccc2n1 c1(C(=O)NCC(C)CNC(C2C(C)C2(F)F)=O)ccc2c(c1)CC2 N1(C(C2CCN(C(C=NOC)=O)CC2C)=O)CC2CCC1C(O)C2O CN1CCOC(C(=O)NCC#CCNC(C2CCCC2n2cccc2)=O)C1 c1(C(COC)NC(=O)NC2CN3CCCC2C3)cc(F)c(F)c(F)c1 C(C(=O)NCC1CCC1C(=O)NOCC1CC1)(C1CC1)OC C(CC(C)(C)C(=O)NC1CC2C(NC(c3oncc3C)=O)C2C1)SC C(=O)(C#CC(C)C)NC1(CC=C)CN(C(C2CCN(CC(F)(F)F)CC2)=O)C1 C(=O)(C(C)CS(C)(=O)=O)N1CCC(NC(COCCOCC)=O)CC1C CCC(CC)C(C)C(=O)N1CC(C2(NC(=O)C(C)Cc3ccnn3C)CC2)C1 C1(C(=O)NC2CC(CC(=O)NC3CCN(CC)C3=O)C2)CCCC(=O)N1C C(CC(=O)N1CCCC(CNC(=O)CCc2cncs2)C1)(C(F)(F)F)OC C(=O)(CS(=O)(=O)C(C)(C)C)NC1C(C)CCN(C(CCN(CC)CC)=O)C1 C1(C(=O)NC(CNC(CC2(C=C)CC2)=O)C2CCC2)CN(C(C)=O)CCO1 C1(C)(C=O)CCNC(=O)C1.c1(C(=O)OC)c(NC(CC)C(C)C)ncnc1Cl.N C1(C(N2CCC(C#C)C2)=O)C2CC3C(C2NC(c2cscn2)=O)C13 CCCCCCCCS(=O)(=O)N1CC2CCN(C(C3CCCO3)=O)C2C1 c1(CN(C)CC2CN(C(c3ccc(Br)c(Cl)n3)=O)C2)ccc(Br)cc1F [N-]=[N+]=NCCCC(=O)NCC1CC(NC(C2CC3(CC3)CO2)=O)C1 c1(NC(N2C(C(N(CCOC)C(C)C)=O)CCC2)=O)cncc(Br)c1C C(=O)(C(O)CC(C)(C)C)NC(C1(O)CCN(C(C=C(C)C(F)F)=O)C1)C C1(C(=O)NCCCCN(C(=O)C=CC2CCOCC2)C)CCCCN(C)C1=O CN1CCCC(O)(CC(N2CCCC(F)(CNC(C3CNC(=O)N3)=O)C2)=O)C1 N1(C(C2N(C=O)CCC2)=O)C2CCC1CC(CNC(=O)COC1CC1)C2 C(=O)(CCCC(F)F)N1CCC(C(C)(C)C)(CNC(=O)CO)C1 c1(COC)ncc(C(=O)NC2CCC2NC(=O)CO)s1.C1CCCCO1 C(=O)(CC(CN(C)C)C(F)F)N1CCCCC1.C1(CCOC)CC1C(=O)NC c1(C(=O)NCC2C3CN(C(C=CCC)=O)CC32)cc(Br)cc(C)c1C CCCCCCC(F)c1nc(-c2ncccc2C(F)(F)F)nn1Cc1cnn(C)c1 N1(C(c2nc(C3CC3)no2)C)CCC(C2CC2)CC1.C1(C=O)CC(=O)N(C)C1.N c1(C(=O)OC)cc(NC(=O)CC2CCN(Cc3ccc(NC)cc3)C2)ccc1I c1(C(=O)NCC2(NC(C(C)OCCC=C)=O)CC2)c(F)cccc1F.O Cc1cc(C)n(-c2ccccc2C(=O)NC2CCC2)n1.C(=O)(C(O)C1CCC1)N C1(NC(=O)NCC(C)(C)C)CCCN(Cc2cn(CCF)nn2)C1 C1(O)(CC(N2C(CC)CCC2)=O)COC(C)(C)C1.c1(C(=O)N)scc(C)c1Cl C1(NC(c2ccn(CC)c2C)=O)CN(C(C2(F)CC2)=O)CCC12CCC2 Cc1ccc(F)c(C(=O)NC2CCCC(NC(=O)CN3CCOCC3)C2)c1O CCC(C)C(C(=O)NC(C1CC2(CCC2)C1)C)N(C)C(C1CC2(CSC2)C1)=O C1(CC(N2CCCC2)=O)CCC2(CCC2)O1.C=CCCOCC(=O)NCC.O c1(C(=O)NC2CCC(NC(c3n(C)ccc3)=O)CC2)nc(C2CC2)ncc1Cl Cc1ccc(F)cc1CNC(=O)C=CC1CCN(C(C2CCC(=O)N2)=O)CC1 C#Cc1cncc(C(=O)NCCC(C)(C)NC(=O)C)c1.c1ccc(F)c(C)c1.O Cc1ccc(CNCc2cc(C3(F)COC3)no2)nn1 CC1C(C(=O)N2CCC(CNC(C3C(C#N)C3(C)C)=O)C2(C)C)=NOC1C O=C1NCC2(CCN(C(C3CC(O)CN3C(c3nc[nH]n3)=O)=O)C2)N1 Cc1ccc(C)c(CC(=O)NCC2(NC(c3ccc(Cl)nc3C)=O)CC2)c1 N1(C(C(CC)F)=O)CCC(NC(c2oc(S(N)(=O)=O)cc2C)=O)CC(C)(C)C1 [N-]=[N+]=NCC(C(=O)N1CC(OCC(F)F)C1)NC(c1ccc(Cl)cn1)=O n1(CC)nc(C)c(C(N2CC(Cn3cc(COCC)nn3)C(O)C2)=O)c1C c1(N2CCC(CNC(=NC)NCC(c3ccsc3)C)C2)ccc(Cl)cc1Cl C1(CNC(c2n(CC)nnc2)=O)CC(F)(F)CN1C(=O)CCS(=O)(=O)N C1(NC(C=CCN(C)CC)=O)CC2CCC1(NC(=O)C)C2.CC(C)C.O C1(CN(C(=O)CNC(c2ccoc2)=O)C)CCCN1C(C1CCC1)=O C(=O)(C(C)CC)N(CC#C)CCO.C1CCCO1.C(C)(C(F)F)=CC=O c1(C(=O)NC2(CNC(C3(C)CS(=O)(=O)C3)=O)CCC2)coc2c1CSC2 c1(C(N2C(CNC(c3nccc(CC)c3)=O)CCC2)=O)ncnc2cc[nH]c12 n1(CC)nc(C)c2cc(C(=O)NC3CN(C(=O)CC(C)C)CCC34CCC4)sc12 C1(C(N(C2CC(OC(C)(C)C)C2)C)=O)CCOC1c1nc[nH]n1 C1(C(N2CCC(NC(c3nncn3C)=O)C2)=O)(COC)C=CCC1 c1(OC)cnc(F)cc1C(=O)NC1CN(C(c2cc(N)cc(O)c2)=O)CC1C C(CCC(=O)NC(C)(C)CC)OC(C)C.c1(C=O)ccc(-c2cnn(C)c2)o1.N N1(C(CN2CC(=O)NC2=O)=O)CCC(C)C(O)C1.C12(C=O)CCC(CC1)CC2.N c1(NC(=O)NC(C2CC=CCC2)C(=O)O)cccn(C(F)F)c1=O c1(OC)cc(C(F)(F)F)ccc1N(C1CCNCCC1C)C(=O)C(N)CN N1(C(C(C)N(C(C)=O)C)=O)CCCC2(CCN(C(C3(C(F)F)CC3)=O)C2)C1 N1(C(C2(CC=C)CC2)=O)CC2CC(C1)CN(C(=O)Cc1cccc(C=O)n1)C2 c1(N(C(C)C(C)C)C=O)c(C)nn(C)c1C.c1(C(CC)OC)ccc(Cl)cc1.N N1(C(C(C2CCCN(C(C3CCS(=O)CC3)=O)C2)C)=O)CCCC(O)(CO)C1 c1(C(=O)NC(CNC(=O)CC2CCOC2)C2CC2)ccco1.c1cnn[nH]1.C CC(C)(C)C(CNC(=O)Cn1cnc(Br)c1)NC(=O)C(F)=CCCF c1(C(=O)NC(CN(C(Cc2ccc(C)nc2)=O)C)C)cnc(F)cc1C C1(CC(=O)N(CCCO)C)CC(O)C12CCC2.C1(O)(CC=O)CCC1.CC c1(CC=C)ccccc1C(=O)NC1COCC1C.C(=O)(C(C)C)N.C(C)C CC(C)(CC(F)C(=O)NC1(CCF)CCC1)NC(=O)Cn1ccnn1 Cc1cn2c(C(=O)NC3CC3CNC(=O)Cc3cccc(F)c3F)cnc2s1 c1(NC)cc(Cl)ccc1C(=O)NC1CN(C(=O)Cc2ccc(F)cn2)CCC1F O=C(C1CCCn2cnnc21)NC1C=CCN(C(c2ncoc2C2CCC2)=O)C1 C(=O)(C1CCCc2nc[nH]c21)N1CCC(CN(C(CC(C)CC(C)(C)C)=O)C)C1 N1(C(C=C2CCC(C)C2)=O)CC2CC2(NC(c2sccc2Cl)=O)C1 C1(NC(C2(COC)CCC2)=O)COCCN(C(=O)CO)C1.c1ccc(Cl)cc1 Cc1ccc(C)c(CNC(C2CCN(C(=O)OC(C)(C)C)C23CC3)=O)n1 c1ccccc1.CCS(=O)(=O)N(CC(=O)NCC1CC1C)C.C(=O)C.N CCC(CC(=O)N1CCCC1CC(C)C)NC(=O)Cc1ccoc1 C1(CC)CCC(C(=O)NCC2CC(C(=O)N(CCS(N)(=O)=O)C)CO2)CC1 c1(CC)nn[nH]c1C(=O)NCCC1(OC)CN(C(=O)CC2CCC(C)C2)C1 CC1CN(C)CC(C=O)O1.C1(C)(CC(=O)N(C2CCCC2)CC)CC1(Cl)Cl.N C(=O)C(C)(C)C(F)(F)F.CCC(C(C)CN(C)C)NC(c1ccc(C)s1)=O N1(C(c2c(C)ncs2)=O)CCCCC(NC(=O)C(C)Oc2ccc(F)cc2)C1 N1(C(c2cn(C)nc2)=O)CCC2(CCCN2C(=O)CCc2cnn[nH]2)C1 c1(OC)cc(F)cc(C(N2CCC3(NC(=O)C#CC(C)(C)C)CC3C2)=O)c1N Cc1cc(F)ccc1C(N1CC2CC2(C(=O)Nc2ccns2)C1)=O CCC(CC(=O)N1CC2(C(=O)O)CC1(C)C2)CC(F)(F)F C1(C(=O)NCC2CCN2C(=O)C(=Cc2cccnc2)F)CCC2(CCC2)OC1 Cn1cc(C(=O)NCC2CCC2NC(c2ccn(C3CC3)n2)=O)cn1 C(=O)(C1=CCS(=O)(=O)C1)NC1CN(C(C(C(C)C)n2cccc2)=O)CC1O C1(N(C(C(CC)OC)=O)C)C2CN(C(=O)C=Cc3ccnn3CC)CC12 N1(C(CSC(C)C)=O)CCCCC(NC(C2CC(CC(F)(F)F)C2)=O)CC1 n1(CCC(=O)NC(CNC(c2nccnc2O)=O)CO)cc(Br)ccc1=O N1(C(C(CC=C)C)=O)CC2CCC(C1)N2C(=O)CC(OCC)OCC N1(C(c2cc(OC)ns2)=O)CC(OC)CC1CNC(=O)C(F)=C1CCC1 CC(C)C(C(=O)NCCC(=O)NC(C)(C)C)NC(c1ccoc1Cl)=O O=C1Cc2cc(-c3cscc3CN3CC4CCCC34)ccc2N1 C1(CC(N2CCN(C(CNC(C3CCC4(CC4)C3)=O)=O)CC2)=O)CCC=CCC1 S(=O)(=O)(CCCCC#N)NC(c1ccc(CSCCOC)cc1)C C1(CC=O)CCCNC1=O.c1(CC)conc1CNC(=O)CCC1CCC1.N C=CCC(CC)C(=O)NCC1CN(C(c2cc(C(C)C)nc(O)c2)=O)C1 c1(C(=O)NC2CCC(NC(C3(C4CC4)CC3)=O)C2)cnc2ccccn12 C1(NC(CSC)=O)(CNC(c2cnc(C(F)(F)F)s2)=O)CCCCC1C c1(NC(N(C(C)CC2CC2)C(C)(C)C)=O)c(S(N)(=O)=O)cnn1C c1(C(=O)NC(C(C)NC(c2cc(C)sc2C)=O)C)cc2n(c1)CCCNC2=O C(C(C(=O)NCC(C)C)N(CCCC(C)(F)F)C)(C1CC1)OC C1(C(N2CCC(NC(c3n[nH]cc3Br)=O)C2)=O)CC2CC1CC2(F)F c1(NCC2(C)CCCN(C(=O)CC3(O)CCCCCC3)C2)ncc(C#N)cc1Cl CC1(CCNC(C2CCCCC2n2ccnc2)=O)CCN(C(c2cc[nH]n2)=O)C1 c1(C(N2C(CN(C(C(C(C)C)C)=O)C)COCC2)=O)cc(F)ccc1Br N1(C(C)=O)CCCN(C(CC2CCCCC23CC3)C(=O)NCC2CC2)CC1 C1(C(N2CC3C(C(N(C)C(C4CC4)C)=O)(C3)C2)=O)CC2C(C1)C2(F)F O=C(C(F)C1=CCCCC1)NC1CCCCCN(C(c2ccccc2)=O)C1 CCC(C#N)C(=O)NCC(C)CNC(c1cc(N(CC(F)(F)F)C)ccn1)=O c1(C(N(C(CC)CC(=O)NC2CCC(OC)C2)C)=O)c[nH]c2ncccc12 c1(C(=O)Nc2ccc(C(N3CCC(O)(C(F)(F)F)C3)=O)nc2)cc2ncsc2[nH]1 C1(C(=O)NC(CC(C)NC(c2ncoc2C2CC2)=O)C)CN=C2N=CNN2C1 N1(C(CC(CC2CC2)NC(CSCCCC(C)C)=O)=O)CC(C)OC(C)(C)C1 C1(C=O)(NC(=O)OC)CCCC1.C1(C=O)COCC1C(F)(F)F.CCC.N C1(c2nnnn2C2CC2)(NC(c2cccc(C)c2)CSC)CCN(C2CC2)CC1 C(=O)(C(O)C(F)(F)F)N1CCC(CN(C)C(c2cc(-n3cnnc3)ccn2)=O)C1 Cc1ccc(CC(=O)NCCN(CC(C)O)C(c2sccc2Cl)=O)s1 C=C1CC2CCC(C1)N2C(=O)C(c1ccco1)NC(=O)C(CC)SC c1(OC)cnccc1C(N1CC(OC)CC1C)=O.N1(CC=O)CCN(C)CC1.N CCC(C)C(O)C(=O)N1CCCC(N(C(=O)Cc2cn(C)nn2)CCOC)C1 CS(=O)c1ccc(CNC(=O)Cc2nocc2C(C)(C)C)cc1 N1(C(C(C(C)C)NCC)=O)CC2(C1)CN(C(c1ccc(=O)n(C)n1)=O)C2.C N1(C(=O)NC(c2cc(C)no2)Cc2ccc(F)cc2)CC(C2=NOC(C)C2)C1 c1(CC=O)cc(Cl)cc2ccccc12.C(C)(C(=O)N(C(C)C)C)OCCC#C.N C(=O)(C1=C(Cl)CCC(C)C1)N1CCN(C(CN(CC)CC)=O)C(COC)C1 Cc1cc(Br)cnc1C(=O)NCC#CCNC(=O)C(C)Cc1cccnc1 Cc1nccc(C(=O)NCC2(C(=O)NC(c3ccccn3)CO)CCCC2)n1 C12(NC(C(CC)SC)=O)CC1CN(C(=O)Cc1cc(OC)no1)C2 C1(NC(CCC(CC)OC)=O)CCCC12CN(C(=O)C(=Cc1cccnc1)F)C2 C1(C(=O)NCc2c(C(C)C)ocn2)CC1C1CN(C(=O)CC2CCCC2O)C1 CCCC(O)CC(=O)N1CCN(C(=O)C(C)(C)C2CCC2)CC1C c1(C(=O)OC)cnc(N2CCC(NC(c3ccc(C4CCC4)cc3)=O)C2C)nc1 c1(C(C(=O)N(CC=C)C)O)cccc(OC)c1 Cc1cc(CNC(=O)CC2(C)CCC2)oc1C(=O)NCC(c1ccsc1)O c1(C(N2CC(OCCNC(C(C)CC3CCC3)=O)C2)=O)cncc(F)c1 Cc1nc(C(C)C)oc1C(=O)NCC1CN(C(=O)CCCn2ccnn2)CC1C c1(C(=O)NC2CCC(NC(C3(F)C(C)OCC3)=O)CC2)ccc2occc2c1 Cc1ccc(Cl)cc1C(=O)NCC1CC(C)N(C(c2cccnc2)=O)C1 CC(C)(C(=O)NCCS(=O)(=O)Cc1cn(Cc2ccncc2F)nn1)C(F)F C1(NC(C#C)=O)CCCN(c2nccc(-c3ccccc3)n2)CC1 C1(CC)(NC(c2cnccc2OC)=O)CCN(C(C2(C)CC2(F)F)=O)CC1 c1(C(N(C)C)=O)ccccc1C(=O)NC1(CC)CC1.C1(C=O)CC(F)C1.N CN1CCOC(C(N2CC(O)CC2CC(=O)NCC(F)Br)=O)C1 O=C(C1=CC2(CCOC2)C1)NCCNC(C1CC(=C(F)F)C1)=O N1(C(C(C#C)(C)C)=O)CCC2(CC1)CCN(C(=O)C(C)OC1CCOC1)C2 C1(CC=O)CCC(N(C)C)C1.C(=O)(CC)NCC(C1CCC1)OCC.N CCCC(C(O)C(=O)N1CC(F)CC1C)NC(c1cc(C)nc(C)c1)=O N1(C(Cc2c(C)scc2)=O)CCN(C(=O)CSC(F)F)C2CCCC12 N1(C(C(=O)NC(c2ncccn2)CCC)=O)CCC2C(C1)NC(=O)CCN2C c1(C(=O)NCC(CNC(C(c2c(OC)cccc2)O)=O)O)cnc2ccccn12 c1(CCC(N2CCC(O)(CCNC(C3C(C)C3)=O)C2)=O)ccc(F)cc1F c1(C(=O)NCC2(NC(Cc3ccc(C)nc3)=O)CCC2)cc2ccccn2c1 c1(C(=O)NCCC(CC)(CC)NC(C2CCC(C)S2)=O)cnc2c(c1)nnn2C C(=O)(C(C)(C)C(F)F)NC1C(CNC(CC2(CSC)CC2)=O)CC1 C1(CN(C(=O)CC(C)(F)F)CC)CCCN(C(=O)CC2(C)CCCCC2)C1 N1(C(c2cc(C)n(C)c2)=O)CC(C2CC2C(=O)NCc2ncnn2C(C)C)C1 N1(C(C2CCC(=C)CC2)=O)CCN(C(c2cnc(C)s2)=O)CC(C)C1 CCC(C)(C)C(O)C(=O)N1CCCC1CCNC(=O)Cc1cccc(SC)c1 N1(C(C2CN(C)C2)=O)CCN(C(c2cn(-c3cccnc3)nn2)=O)CC1C(F)F C(=O)(N=c1nc2cc(Cl)ccn2[nH]1)N(C)Cc1onc(C)n1 N1(C(CN(C(COC)=O)C)=O)CC2CC2C1C(=O)N(CCCO)CCO c1(NC(C2C(NC(c3cc4nccn4cn3)=O)CCC2)=O)nc2ccccc2s1 N1(C(CCC=CC)=O)CC2CC3CC2C1C3NC(c1ccc2c(n1)CCCC2)=O c1(C(=O)NC(C(C(C)C)NC(COC)=O)C2CCCCC2)cccc2cnsc12 Cc1cc(C(=O)OCC2(C)CC3CC3C2)n(-c2ccncn2)n1 Cc1nc(NC2(CNC(=O)C(C)SC(F)(F)F)CCOCC2)c(C)c(C)n1 N1(C(C(C2CCOCC2)C)=O)CC(C(=O)Nc2ccc(O)c(CO)c2)C(C)(C)C1 c1(C(=O)N)cc2ncn(C)c2cn1.CC(CC)NC(=O)COCC1CCCC1 C=CC(CC)CC(=O)N1CC(N2CCN(C(=O)COc3cccc(F)n3)CC2)C1 N1(C(C(CCC)OC)=O)CC(=O)NCC1C(=O)NC(C12CCC(CO1)C2)C N1(C(C(C)NC(C)=O)=O)CC(O)C1.N1(C(C2(C=O)CC2)=O)CCCC1.C c1(N(C(=O)CC2CCN(Cc3ccc(C#N)nc3)C2)CC)c(F)ccc(C)c1F C1CC2CC(O)C1C2.C(CCC=O)NC(CNC(=O)OCC=C)=O.C1CC1 C(=O)(C(C(C)(C)C)NC(C)=O)NCCCC=C.C1(C)(C(=O)N)CCSCC1 N1(C(C=CCC)=O)CC2(C1)SCCC2NC(=O)C(n1ccnc1C)C Cc1cscc1NC(=O)C(Cc1cnc[nH]1)NC(C1C(C)C1C)=O c1(C2(C(N(CCC)C)=O)CC2)ccc(C(N)=O)cc1.c1(OC)cc(C=O)[nH]n1 C1(NC(C2C(C=C)C2)=O)(CNC(c2ccnn2C(F)F)=O)CCOC1 c1(C(N2C(C)(CNC(CC=CCC)=O)CCC2)=O)cccc(F)c1C C(C)(c1ccccc1)=CC(=O)NC1C(CC)N(C(=O)CCC2CC2)CC1.O N1(C(C2C=CCCN2C(C2CCC3(CCC3)O2)=O)=O)CCCCC(F)(F)C1 N1(C(C(n2ncc(C)c2)C)=O)CC(N(C)C(C2CC(N(C)C)C2)=O)C(C)(C)C1 c1(OCC=C)ccc(Cl)c(C(=O)NC(C)CC)n1.c1(C=O)cnnc(C)c1.N N1(C(c2c(CC)ocn2)=O)CCCN(C(c2cc(C(N)=O)cn2C)=O)C(CO)C1 C1(CCC)CCN(C(C)=O)CC1.c1(C(=O)NC(=O)CC)ccc(C2CCCO2)[nH]1 C1(CC(=O)NCCCN(C(=O)C(C2CCCO2)C2CC2)CC)CCCO1 C1(C(=O)NCCCCN(C(c2ccc(C#C)o2)=O)C)CC2(CCCC2)C1 N1(C(C2(C(C)C)CCCO2)=O)CCCCC(NC(=O)C=Cc2cccnc2)C1 c1(NCCNC(CC)=O)ncccc1S(=O)(=O)NC(c1ncnn1C)C CC1CN(C(c2cccc(F)c2N)=O)C(C)CN1C(c1cnc(C(F)F)nc1)=O C1(NC(C2OCCCO2)=O)CCN(C(C2COC(Cn3cccn3)C2)=O)CC1 C1(C(=O)NC(c2ccccn2)CO)CN(C(C2CC(O)C2)=O)CCC1(F)F CC(C)C(C)CC(=O)NC1CC(C)(CNC(c2n[nH]cc2C2CCC2)=O)C1 c1(SC(C(=O)NCCN(CCOC)C(c2c[nH]nc2F)=O)C)ccccn1 N1(C(C2CC(=C)C2)=O)CCCC2(CC(C(=O)NC3CCCOC3)=NO2)C1 C(N=c1[nH]c(=NCCN2CCCC2)[nH]c2c1SCC2)c1cn(CCC)nn1 N1(C(c2ccc(C)n2C)=O)CCCC(O)(CNC(C2CC3CCC3C2)=O)CC1 Cc1cccc(C(=O)NC(C)(C)CNC(C2CCCC(O)C2)=O)n1 c1(CC(=O)NCC2(O)CN(C(CCCCC)=O)C2)ccc(C)c(F)c1F C1(C(C)NC(CN(CC)CC)=O)CN(C(C2CC3C=CC2C3)=O)CCO1 C(CCCC(=O)N1CC(F)CC1CNC(c1ccccc1CC(F)(F)F)=O)SC Cc1cc(C(N2CC(CNC(c3ccc(C#N)s3)=O)C(C)C2)=O)cc(Cl)c1 C1(NC(=O)CC2OCCO2)CCN(C(c2nnc3n2CCCC3)=O)CCC1CO CCC(CC(=O)NCC(=O)NC(C)CCC1CCCC1)C1CC1 CC1CCN(CCNC(=O)CCN(C(=O)CCn2ccnc2)C2CC2)C1 C(=O)(C(C)(C)CCC#N)N1CC(C)C(N(C(=O)CSCC(F)(F)F)C)CC1 C=CC(C)(C)C(=O)NCC(C)(C(C)C)NC(=O)COCC1CCCCO1 CCCCCCCCC(C(=O)NCC)N(CCOC1(C)CC1)CC N1(CC(C)C)CCC(CNC(c2nc(C3CCCOC3)cs2)=O)C1 Cc1cc(C)n(CC(=O)NC2(C)CN(C(C3CC(O)(c4cccnc4)C3)=O)C2)n1 C1(C(N(C)Cc2cn(Cc3ccccn3)nn2)=O)CCc2nn(C)cc2C1 C#Cc1c[nH]nc1C(=O)NCC1CN(C(=O)C(c2cnn(C)c2)C)CCO1 N1(C(C2(N(C(CC(C=C)C)=O)C)CC2)=O)CCC12CCCCC2 C(=O)(C1=CC2(CN(C(C3CCCC3)=O)C2)OC1)N.C(=O)(C(C)C1CC1)OC C1(NC(c2ncn(CCNC(C3C(C)(C)C3)=O)c2)=O)CCCCC1CO C(C1CCOCC1)=CC(=O)NCC(CC)NC(=O)CC(C)SC N1(C(CC(CNC(c2ccc(C)s2)=O)(C)C)=O)CCC2(CCC(O)C2)C1 Cc1ccc(C(=O)NCCC2CCC2)cc1Cl.C1(C(=O)N)CCC1.C(C)(C)C C1(NC(C(c2cccs2)SC)=O)Cc2ccccc2C1NC(=O)CCC(C)(C)F O=C(C1=CCCN(Cc2scnc2-c2cccs2)C1)N1CCOC2CC12 C=C1CCC(C(c2ccccc2)NC(=O)NCCCCNC(N)=O)CC1 C1(NC(C(CCO)N(C)C)=O)CCCN(C(c2cnc(C3CC3)nc2)=O)CC1 CC1CN(C(C23C=CC(CC2)C3)=O)CC1CNC(c1ccoc1)=O C1(CNC(c2c(OC)cc(C)cn2)=O)C2CCCC1N(C(=O)CN(C)C)C2 c1(NC(C(CC)O)=O)ccc(N(C(=O)C(=O)NC2CCN(CC)CC2)C)cc1C CC(C)(C)C(C#N)C(=O)N1CCC1CNC(c1ccc2nn[nH]c2n1)=O c1(OCC)cccc(-c2nc(CC3CCCO3)n(CCCO)n2)c1 n1(COC)ncc(=NC(=O)NC2C3CCC2(c2ccc(Br)cc2)C3)[nH]1 Cc1cccc(-n2cc(O)c(C(=O)N(CC(C)C)Cc3cc(O)nc(O)n3)n2)c1C c1(C(N2C(C)CCC(NC(=O)CC3=CCCCC3)C2)=O)csc2cccc(F)c12 C(=O)C(C)C(C)S(C)(=O)=O.c1cc(C=O)c(C)o1.C(C)(C)C1CC1.CO c1(OCC)ccccc1NC(=O)CC1C2CN(C(c3sccc3Cl)=O)CC12 N1(C(CCC(=C)C)=O)CCC2(CCCN2C(C2CNC(=O)O2)=O)C1 Cc1ccc2c(c1)CC(C(=O)NC1CC(C)C1)O2.c1(C(=O)N)cc(Cl)ccc1C C1(C#N)(C(=O)NC(CN(C(C2(CC=C)CCC2)=O)C)C)CC1(C)C C1(CC(=O)NCCC(C)NC(c2occc2C2CC2)=O)CC(C)(C)OC1=O C1(C(NC)=O)CCN(C(C2C(C#N)C2(C)C)=O)C1C(C)C.C1CCCC1.CO C1(CC=O)CC2CCC1CC2.c1(C(=O)NCC(C)(C)O)ccc(CO)s1.CC c1(NC(CC2CCN(C(c3n[nH]c(C)c3Cl)=O)C2)=O)nc2ccc(O)cc2[nH]1 O=C1Cc2c(N3CC4CC3CN4C(c3ccnc(Br)c3Cl)=O)ncnc2N1 c1(SC)cccc(NCC2CCCC2)c1[N+](=O)[O-].c1(C(=O)N)cc2c([nH]1)CCC2 Cn1cncc(C(=O)NCCOCC(=O)NCCOCC2CCC2)c1=O CC1(CCCO)CCCN1C(=O)C(C1CCN(C(=O)CCn2cncn2)C1)F Cc1ccn2ncc(C(=O)NCC(O)CNC(C3CCC(C(C)C)CC3)=O)c2c1 c1(OC)cc(Cl)c(I)cc1C(=O)NC1CCC(C(=O)NC2CC2(F)F)C1 C1(COC)CN(C(C2CC(c3ccc(O)cc3)C2)=O)CCN1C(=O)C(C)O C1(C(N2C(C(=O)NC(C)(C)CCCF)CC2)=O)CCC(C2CC2)C1 C1(NC(=O)CC2CCCC(F)(F)C2)CC2CN(C(c3cc(Br)co3)=O)CC2C1 C(=O)(C(C)C(O)CC)N(CCCNC(=O)Cc1c(C)noc1C)CCC N1(C(C(CC(=C)C)OC)=O)C2CCC(C(=O)NOCC(C)O)C1CC2 c1(N2CCN(CC)C(C)C2)ccc(S(=O)(=O)N2Cc3cncnc3C2)cc1Br CC(C)C(O)C(=O)N1CCC(CCNC(=O)CCCc2cccnc2)C1 c1ccc(F)cc1[N+](=O)[O-].C1(NCc2ncc(C)s2)C2CN(C(=O)C(=O)N)CC12 N1(C(C(Cc2c(C)noc2C)C)=O)CCC(NC(=O)C(F)C(C)C)CC1C C(=O)(CCCS(C)(=O)=O)N1CCC(F)(F)C1.C1(C(=O)N)(COC)CCCO1.C c1(C(=O)NC(C2CCOC2)CNC(C(CCC)(C)C)=O)cc(N)c(F)c(F)c1F CC1(C)CCCCC1NC(C1CCC1NC(=O)CCCC#N)=O C1(OC)CC2(C1)CC(C(N1CCCC(CCCCNC(=O)C)C1)=O)C2.C(C)C N1(C(=O)Nc2ccc(C)c(C)n2)CCC2(CC1)COC(CO)C2.C(C)(C)C CC(C)C(O)C(C)C(=O)NCC1(F)CCCN(C(c2cccc(N)c2)=O)CC1 C1(C)(C(=O)NCC(CNC(CCNC(CC(C)C)=O)=O)F)CCC(O)CC1 C1(C(=O)NC2(C)CCC2)CC(=O)N(C2CCCCCC2)C1.C1(C=O)CC12CC2.N Cc1nn(CCO)c(C)c1C(N1CCC(C)(CNC(C2CCOC2)=O)C1)=O C(C1=CCN(C(c2cc(C(C)C)sn2)=O)CC1)NC(c1nn(CC)c(O)c1)=O C1(F)(C(N2CC3C=CC3C2)=O)CCN(C(C2(CO)CCCCO2)=O)C1 c1(C=O)cc(N)c(C)c(N)c1.c1(OC)ccccc1SCC(=O)NCC(O)C c1(N2CCN(C(=O)CC3CCCCC3)CC2)ccc2ncc(=O)[nH]c2n1 C(=O)(CCC(C)NC(=O)CN(C)C(C)C)N(CC=C)CC1CC1 C(=O)(C(CC)(CC)c1ccc(Cl)cc1)NCC1(O)CN(C(C(C=C=C)C)=O)C1 C1(F)(C(=O)O)CCN(C(=O)CCC2CCN(C(=O)C(F)(F)C3CC3)C2)C1 CC1CCN(C(=O)CN(CCC#N)C)CC1CC(=O)NCCOCC(C)(C)C c1(N(C(c2cc(-c3ccccc3)co2)C(=O)NC(C)(C)C)C)ccc(CO)cc1 N1(C(CC=C)=O)CC(NC(c2cc3c(s2)CCCC3)=O)C2CCCCC12 Cc1csc(=NCC(=O)NCC2(F)CCCC2)[nH]1.C1(C=O)(C(N)=O)CC1.C Cc1cc(C(=O)NCC(CNC(C2CCCCS2)=O)C(F)(F)F)c2n[nH]cc2c1 C1(NC(C2(OC)CCOC2)=O)CCCCN(C(c2c[nH]nc2C2CC2)=O)CC1 CCC1=NOC(CC(=O)NC2(CC(=O)NCc3cccc(CO)n3)CC2)C1 CCCC#CC(C)(C)NC(c1cccc(CNC(C2(C)CCOC(C)C2)=O)c1)=O N1(C(C(C)CN(C)C)=O)CC(O)CC1C.c1(C(=O)N)sc(N2CCCC2)nc1Cl Cc1cc(F)c(C(=O)NC2CCN(C(C3CCC3)=O)C2C)cc1F.C(C)(C)(C)O N1(C(c2cc(C)c(F)cc2)=O)CCCC(C)(C)C1C(=O)NCc1ccc(O)cc1 C#CC1CC2CCC1N(C(C1(NC(c3cc(CC)nn3C)=O)CC1)=O)C2 N1(CCC=O)C(C)CCCC1C.CC(C)CCCNC(=O)CSCCN(C)C C1(CNC(CCNC(C)=O)=O)CC(C)(C)CN1C(=O)CCc1cccn1C N1(C(c2nc(C)oc2)=O)CCC(C)(CNC(C2CCC23CCCO3)=O)CC1 N1(C(CC)=O)CCC2(CCCC2NC(=O)C(C)Cc2cccc(F)c2)CC1 c1(C(N(CCNC(=O)C(C)(C)C(C)(C)C)CC)=O)n[nH]c2cc(Cl)ccc12 N1(C(C2C(NC(=O)NCCCCCCCC)C2)=O)CCCC2CCCCC12 c1(NC(C2CC(C)CN2C(c2cnc(Cl)nc2)=O)=O)cnc(O)c(C(F)(F)F)c1 c1(C(=O)NC2CCC(F)(CNC(CCC#CC)=O)C2)cc(O)nc(C2CC2)n1 c1(C(=O)NCC(CNC(C(CCC=C)(C)C)=O)F)cc(S(C)(=O)=O)ccc1C c1(CC)[nH]nc2c1CN(C(C1CC1c1ccc(OC)c(OC)c1)=O)CC2 C1(C)CCC1.C1(C=O)CCC(F)C1.CC(C)(C)OC=O.CC=O.C1CC1.N c1(C(=O)NCC2N(C(C(C)O)=O)CC(O)C2O)cc2cc[nH]c(=O)c2s1 C=CC1(NC(c2ccc(CNC(=O)C(CC)CCOC)o2)=O)CCOCC1 c1(N2CCC(C(=O)O)(C(F)F)CC2)nccc2c(Br)cncc12 N1(C(c2ccc(SC)s2)=O)CCCC(NC(=O)C(c2ccc(O)cc2)C)CC1 Cc1cccc(Cl)c1CC(=O)NCCC(C)NC(=O)Cc1coc(C(F)F)n1 C1(C(=O)NCc2cccs2)CCC2(CC2)N1C(=O)CC1CCCOC1 C1(NC(CCNC(NC)=S)=O)CCC2CN(C(c3ccc(O)nn3)=O)CC12 C1(CC(=O)NC2CCN(C(COC(C)C)=O)CC2)COC(C)(C)CO1.C1CC1 N1(C(c2cc3c(s2)CCOC3)=O)CCN(C(C2CC3C=CC2O3)=O)C2COCC12 c1(OC)ccc(C(=O)NC(C)C(C)NC(=O)COC(F)F)c(Cl)c1OC c1(C(C)(C)C)ccc(C(=O)NCCNC(=O)COCC(F)(F)F)o1 c1(C(=O)NC(CCCNC(C2ON=C(CC)C2)=O)(C)C)ncc(C)cc1C C(c1cccn1C)=CC(=O)N(C1CCN(C(=O)CCc2ccc(CO)cc2)C1)C c1(C2C(C(N3CC(NC(=O)CCC4CCOC4)C3)=O)C2)occc1Br O=S(=O)(c1cnc(C2CC2)nc1)NC(C(F)(F)F)C1CC1(Br)Br C(c1cccc(Cl)c1)=C(C(=O)N)C.C1(NC(CC2CC(SC)C2)=O)CCCCC1 C(=O)(C(O)CC(N)=O)N(CC(CC)NC(c1cn(C2CC2)nc1C)=O)C C1(C(=O)NC2(CNC(Cc3ccc(OC)cc3)=O)CCC2)CCC=CCCC1 C1(O)(C(C)(C)C)CN(C(C2CC2(C)C(F)(F)F)=O)C1.C(C=O)N(C)CCC CC1(C)C(C)(C(=O)N)C1(C)C.C1(C=O)CCN(c2ncccn2)C1.C1CC1.C N1(C(C(c2ccn(C)c2)C)=O)CCC(F)(CNC(c2cc(C(F)F)[nH]n2)=O)C1 C(CC(C)C)(C(=O)NCC1CCCN1C(C12CC(C)C1C2)=O)NC(C)=O c1(C(=O)NC2CCC(NC(C(CC#C)O)=O)C2)ccc(C(C)=O)cc1F c1(C(C(=O)NCCn2cc(CNC)nn2)O)cc(F)cc(F)c1.c1ccccn1 C(C1c2ccsc2CCN1C(c1cnncc1O)=O)NC(C1ON=C(C)C1)=O CCC(C(=O)N1CC(CF)(NC(c2cnn(C(C)(C)C)c2)=O)C1)C(C)(C)CC c1(C(=O)NC2C3CC2CN(C(C2CC4CCC2O4)=O)C3)cc2sc(Cl)cc2[nH]1 C1(NC(C=COc2ccc(OC)cc2)=O)CN(Cc2nccn2C)CC1(C)C Cc1nn(C)c(C)c1C(=O)NC1CC(C)CN(C(=O)Cc2csnn2)C1 CCCC(C(=O)NCC1CCC(NC(C2CCc3n[nH]cc3C2)=O)C1)C(C)C n1(CCC(=O)NCC23C(CN(C(CCN(C)CC)=O)C2)C3)ncc2c1CCCC2 Cc1oc2cc(C(=O)N(CCCNC(=O)Cc3ncoc3C)C(C)C)[nH]c2c1C CS(=O)c1ccc(CN(C=O)CCCn2cnnn2)cc1 c1(N(C)C)cc(C(N2CCCCC2C)=O)ccc1[N+](=O)[O-].C1(C(=O)N)CC2CC2C1 N1(CC(=O)NC)CCC2(CC1)OCCc1sc(C(N3CC(=O)NC(C)C3)=O)cc12 c1(C(=O)NC2CCCC(C(=O)Nc3ccnc(F)c3F)C2)cc(Cl)c(Br)c(Cl)c1 c1(OC)csc(C(=O)N(C2CCC(NC(c3nnsc3N)=O)C2)C)c1 N1(C(C(=Cc2ccco2)C)=O)CCC2CC2(C(=O)NC(C)(C)CCCF)CC1 n1(CC)nc(C(=O)NCC2CN(C(c3cc(C)n(C)c3)=O)CC2C)c(Br)n1 N1(C(C(c2nc(C)[nH]n2)C(C)C)=O)CCN(C(=O)OC(C)(C)C)CC(O)C1 CC(CC1CCC1)C(=O)NCc1cn(CCNC(=O)CO)nn1 CCCCC(C(=O)NC1CC2CC(NC(=O)Cc3c(Cl)cnn3C)C1C2)C(C)C c1(C(=O)Nc2c(C(=O)Nc3scc(C)n3)scc2)cc(=O)ccn1C C(=O)C1=CC2(CN(C(C3CNC(=O)C3)=O)C2)OC1.C(C)(C1CCC1)OCC N1(C(COCc2cc(C)on2)=O)CCC2CN(C(=O)C#CC3CCOC3)CCC12 c1(CCCOCCOc2c(C(=O)O)c[nH]n2)ccc(Cl)cc1 c1(CNCC2(C=C)CCC2)ccc2o[nH]c(=N)c2c1 C(=O)(C1CCCn2cc(C)nc21)N(CC(C)(C)NC(C(CCCC)CC)=O)C N1(C(C(C)=CC)=O)CCN(C(=O)C=Cc2ccc(Br)s2)CC1CCC C(=O)(C1=CSCCO1)N1CC(NC(CCC(C)OC)=O)C(OC)C1 C(=O)(C1CCc2nccn21)N(C1CCN(C(c2c(CC)cccn2)=O)CC1)CC C1(C)(C(N2C(C(=O)NCC(C)C#N)CSC2)=O)CC2C=CC1C2 C=C1CC2CCCC(C1)N2c1nc(NCc2nc(C(C)C)cs2)c2ncsc2n1 N1(C(C(CCC)F)=O)CC(NC(c2[nH]cc(C(C)=O)c2C)=O)CC12CCOC2 CC1CN(C(=O)NC2COC(c3ccccc3)C2)CC1(F)F C(=O)(C1=CC2(CCOC2)C1)N.Cc1oc([N+](=O)[O-])cc1C(=O)NC1CCCCC1 C1(COC)(NC(C2CC3CC(OC)C3C2)=O)CCN(C(=O)CCSC)CC1 n1(CC(=O)N(C)CC2CCCC(NC(C(CC)(C)C)=O)C2)c(C)c(C)sc1=O Cc1cn2c(n1)C(C(=O)N1CC(O)(CC)C1)CCC2.C12(C(=O)N)CCN(CC1)C2 c1(C(N2C(CNC(C(CC)n3ccnc3)=O)CC(C)(C)C2)=O)ncn2ccccc12 CCC(C)(CO)C(=O)NCC1CCCCCN1C(C1CC(n2ccnn2)C1)=O c1(C(C(=O)N)O)ccc(Cl)c(F)c1.N1(C(CC2(C=C)CCC2)=O)C(C)CC2CC12 C1(C)(CC(N2CC(C)C(NC(=O)CCc3cccs3)C2)=O)CCS(=O)(=O)N1 C1(NC(c2cnc(OCC)s2)=O)CCN(C(C2(F)CCCCC2)=O)CC1O C1(NC(C2(CCOC)CCC2)=O)CCC(NC(=O)CCCCN2CCCC2)CC1 C(=O)(C1=Cc2ccccc2C1)NCCNC(C1CN(C(C(NOC)=O)=O)C1)=O c1(C(=O)NC2(CC=C)CN(C(c3nccnc3N)=O)C2)nc2sccn2c1C CC1(C)CN(C(c2ccnn2CCF)=O)CC1CNC(=O)CNC(N)=O N1(C(C(c2c(C)cccc2)C)=O)CCCN(C(=O)C(C)N(C)C)CCC1 C(=O)(CCCC(F)(F)C(F)(F)F)N1CCC(NC(C(CCC#C)O)=O)CC1 Cc1c(C(=O)NC23CC2CN(C(C2(F)CC2C)=O)C3)cccc1C(F)(F)F Cc1cccc2c1CCOC2C(=O)N(CCC(C)NC(=O)C=CC(C)C)C CC1CCC(CNC(c2ccc(Cl)cc2Cl)=O)N(C(=O)CS(C)(=O)=O)C1 N1(C(c2scc(C)c2)=O)CC2(CCC2)CC1C(=O)NCC1(C)CCOC1 Cc1ccc(C(C)CC(=O)NCC2(C)CC2)cc1.c1(C(C=O)F)ccccc1.N C(=O)(C1=C(C)CCN(C(=O)C(=O)Nc2ccc(C#N)cc2C)C1)OC CCCCC(CC)CC(=O)NC1CC(F)(CNC(=O)C(COC)CC(C)C)C1 C(=O)(NNC(=O)Cc1ccccc1)NCc1cccc(OC(C)C)c1.N(C)C.C CCC(C(=O)NC(C1(C)CC1)C)OC1CCCC1.C(=O)C=CSC1CC1.N N1(C(C(C2CCC2)OC)=O)CCCC(F)(CO)Cc2ccccc21 C12(C(N3CCC(CC(=O)NCc4cnc(CC)s4)C3)=O)CCC(CC1=O)C2 C1(C(C(=O)N(C(C)CNC(=O)CC)CC)F)CCOCC1.CC(F)(F)F.O Cc1nc2cccc(C(N3CCC(CN(C)C(C4CCO4)=O)C3)=O)c2[nH]1 N1(C(c2c(CC)[nH]cc2)=O)CC2CCC(C1)N2C(=O)CCCc1ccccc1 C(=O)(C1Cc2ccc(Cl)cc21)NCC12CC(NC(CC(C)F)=O)(C1)C2 C1(NC(C(N)=O)=O)CCCN(C(=O)C=Cc2ccc(Br)o2)C1 C(C(C)(C)C(=O)NCC1(O)CCN(C(C2(C(C)(C)O)CC2)=O)C1)OC c1(CC)cccc(C(N2CC(F)CC2C(=O)NCCN2CCC2)=O)n1 C#CC1(NC(=O)C(O)Cc2[nH]cnc2C)CC2(CCOCC2)C1 CC1(C)COC(CC(=O)NC2(C)CCN(C(=O)C(C)(C)c3cnsc3)C2)C1 C1(CNC(Cc2nc(C)[nH]n2)=O)CC2CCC1N2C(=O)C(O)c1ccco1 CC1(C(=O)NC2CCCN(c3ccccc3)C2=O)CC2(C1)CC2(F)F N1(C(CCC(C)OCC)=O)CCC(CC)(NC(=O)CCc2cncc(C)c2)CC1 CN=c1cc(C(=O)Nc2cc(C(F)(F)F)ccn2)c2ccccc2[nH]1 Cc1ncccc1-c1cn(CC(=O)NCc2ccc(C(=O)NC(C)C)o2)nn1 c1(C(N2CC(CC(N3CCN(CC)C(C)C3)=O)(OC)C2)=O)cccn2cncc12 C1(C(=O)NCC2C(C(=O)NCC(C#C)OC)C2(C)C)C=CC=CC=C1 C(C(C)(C)CN(C(=O)C=C1CCSCC1)C)NC(C1C(C)(CC)C1)=O c1(C(=O)NCCOCC(=O)N(C(CCCC)C)C)cccc(C)c1C#N N1(C(C2=C(C)OCCS2)=O)CCC(NC(C2CC2(C)C)=O)C12CCCC2 C=CCCC(C(=O)NCCCS(N)(=O)=O)NC(=O)C(C(C)CC)N(C)C S(=O)(=O)(c1ccc(-c2csnn2)s1)N(C1CCSCC1)C(C)CO C#CC1CN(C(C2(CC)CN(C(=O)C(C)S(N)(=O)=O)C2)=O)CC1OC N1(C(C(C)=CC)=O)CCC(CCNC(C2CCC2c2ccccc2)=O)CC1 c1(C(=O)NCCN(C(c2nn(CCC)nc2)=O)CC)ccc2occc2c1 C1(CCC)(NC(c2ncc(Cl)cc2F)=O)CCN(C(=O)CC2CCOC2C)CC1 N#CC1CCC1C(N1CCC(CCNC(c2cncs2)=O)C1)=O S(=O)(=O)(c1c[nH]ccc1=NC1CCc2c(C)cccc21)NCCCC(CC)O N1(C(CNS(CC)(=O)=O)=O)CC2CC(NC(C3C4CCC(=O)C34)=O)C2C1 c1(CC)cccc(CNC(=NCCc2ccc(OCC)cc2)NC(C)C)c1CC c1(CC)ccnc(C(=O)NC(C)CNC(=O)C(C)(F)c2ccon2)c1 C(=O)(CCC(F)(F)F)N1CCCCC(N(C(C(OC)OC)=O)C)C1.C(=O)C1CC1 C1(C(N(CCCF)CC)=O)CN(C(C2CCCSC2C)=O)CC12CCC2 C1(C(=O)NCCC)CC12CCN(C(C1(C)CCC(C)CC1)=O)CC2 C=CC1CN(C(C2(NC(c3oc(CC)cc3C)=O)CCCC2C)=O)CC1O C(=O)(N1CC=CCO1)C1(C(C#CC)(C)C)CCOC1 c1(C(=O)NC2(C)CCN(c3c(OC)cnc(Cl)n3)CC2)ccc2nc(O)sc2c1 c1(C(=O)NC(CCCNC(C2(C(=O)NC)CC2)=O)C)ncccc1Cl c1(C(N2C3CN(C(C(C)(C)OC(C)=O)=O)CC2CC3)=O)cc(F)c2cn[nH]c2c1 c1(CNC(c2c(CC)ccs2)=O)ccc(I)cn1 c1(CC)oncc1C(=O)N(C1CC(NC(C2(CC)COC2)=O)C1)C c1(C(=O)NCC2CN(C(c3nc(CC)oc3C)=O)C2)cc(C)c(C)cc1C N1(c2n3nc(c2)CC3)CC(C(=O)O)C2(COC2)C1.C(c1ccc([N+](=O)[O-])o1)=CC c1(-c2nnc(C(C3CCN(Cc4ccccc4)C3)C)o2)ccc2nccnc2c1 N1(C(C(CCC(C)C)F)=O)CC2(C=C(C(=O)NC3C4CCC3CC4)CO2)C1 C(C1=CCN(C(=O)CN(C)S(N)(=O)=O)CC1)NC(C1CN(CC)C(=O)C1)=O C(=O)C1=C(C)CCOC1.N1(CC)CCCC1=O.C1(CC=O)CCC1.C(=O)CC.N c1(C(=O)N)cc2sccc2[nH]1.CC(CC)NC(=O)C=CC(F)(F)F.C1CC1 c1(C(=O)NC2CC3(C(NC(c4cc(SC)oc4)=O)C3)C2)cc2c(s1)CCOC2 N1(C(=O)C=Cc2ccc[nH]2)CCCC(F)(C(N2CCC(F)C(F)C2)=O)C1 C1(C#N)(C(=O)NC(C2OCCN(C(C(CSC)(C)C)=O)C2)C)CC12CCOCC2 c1(CN(C(=O)Nc2cnn(-c3cnn(C)c3)n2)CC)cccc(C)c1C CC(C)CCC(C(=O)N1CC2COCC(C2)C1)NC(=O)Cc1cccnc1 N1(C(C(CC=C)C)=O)CC(CNC(c2ccc(F)c(F)c2)=O)C2(CC2)C1 c1(C(=O)NC2(CO)CCN(C(c3cccc(OCC)c3)=O)C2)nc(C)ccc1F C1(C(N(CCN(C(=O)CCc2cnco2)CC)C)=O)CCS(=O)(=O)N1 Cc1cc(C(=O)NCCCCNC(=O)C(C)CS(C)=O)cnc1C N1(C(C=CCCC(C)C)=O)CCCCC1CN(C(=O)CC(C)(C)C)C c1(C(=O)NCC(CCNC(C2(CC#C)CCCO2)=O)OC)cc(Cl)ccn1 CC(C)(O)CC(C)C.c1(CC)ccccc1C(=O)NC1CC(CC(=O)N)C1(C)C c1(C(=O)NCC2C3CN(C(c4n(CC#N)ncc4)=O)CC32)ccc2cnnn2c1 N1(C(c2c(C)noc2C(C)C)=O)CCCC(F)(F)CC1.C1(CC=O)CC12CC2.N C(=O)(C1=C(C)CCC1)N1C(CC)C(NC(=O)CSCc2ccncc2)CC1 c1(C(=O)NCC2N(C(CNS(C)(=O)=O)=O)CC2)n[nH]cc1Cl C1(C(N2C(C)(C)C(CN)C2)=O)Cc2c(F)cccc2C(=O)O1 c1(CN2CCC(NC(c3ccc(OC)s3)=O)C(C)(C)C2)ccc([N+](=O)[O-])c(F)c1 N1(Cc2cncc(OC)c2)CC2(CN(C(C)=O)CC2c2ccccc2)C1 c1(C(=O)NCC(CNC(c2ccc(CC)[nH]2)=O)C)cn2c(n1)CCCC2C Cc1cccc(CCC(=O)NCCC2COCCN2C(=O)C(=O)NC(C)C)c1 C(=O)(C1=NOC(C)C1C)NC1CCC(NC(c2ncc(C)cc2Br)=O)CC1 C1(C(=O)NC(CN(C(C2CCC2)=O)CC)C)CCC=CCC1.c1(C)cnn[nH]1 C=CC(C)(CC)C(=O)NC1CCN(C(C2(F)CC2)=O)CC1.C(C)=O.C1CC1 Cc1[nH]cc(C(=O)NC)c(=O)c1Cl.C(=O)CS(=O)(=O)N(C)C.C1(F)CCC1 C12(CC(=O)NC3(CC)CCCCC3)CCC1CN(C(=O)Cc1nccn1C)C2 C12(C(=O)NCCC(C(=O)OC)C)CC(CCO1)N(C(C1CCC3CC13)=O)C2 C1(C(=O)NCC2(F)CC(NC(C(CC)C(C)C)=O)C2)CCc2c(n[nH]c2C)C1 N1(C(C(C2CC2)SC)=O)CCN(C(=O)CNC(c2c(Cl)cnn2C)=O)CC1 c1(C(=O)NC2CCN(C(C(CCC#C)O)=O)C(C)C2)cnc2ccnn2c1C CC1CN(C(=O)Cn2cccc2)CC1CNC(c1cc(Br)n(C)c1)=O c1(C(=O)NC(CCCNC(Cn2c(C)cnc2)=O)C)cccc(S(N)(=O)=O)c1 O=C(C1=CCCN(C(=O)Cc2c(F)cccc2Cl)C1)Nc1ccc(Cl)c(F)c1F C(CCO)(C(F)(F)F)NC(C1CCN(C(=O)CN2C(=O)CCCC2=O)CC1O)=O N1(Cc2ccn(CC)n2)CC(NC(c2ccnc(F)c2OC)=O)C(C)(C)C1 C#CCCCC(C)C(=O)N1CCC(O)C(NC(c2csc(Cl)c2)=O)C1 c1(CC(=O)N(C(C(=O)OC)C(C)C)C)c(C)nc(-c2ccccc2)nc1O c1(NCCCCC(C)NC(C(C2CCC2)OC)=O)nc(C)ccc1C#N CCC(CCCc1ccccc1)N=c1[nH]c(=NCC=CC2CC2)c2sccc2[nH]1 C1(C=O)CC(C2CCC2)C1.c1(COC)ccc(C(=O)NCCC2CCC2)s1 Cc1c(F)cc(C(=O)O)cc1S(=O)(=O)N(CC(c1ccc(Br)cc1)O)C C1(CNC(C2N(C)CCOC2)=O)CN(C(=O)C=Cc2ccoc2)C2CCCC2O1 CC(C)CC(C)CC(=O)NCC(C)(C)C(=O)NC1(CO)CC1 c1(OC(C)C(N2C3CCC2C(C)C3)=O)ccc(C#N)cc1.C(=O)C1=C(Cl)CC1.N c1(OCC)ccc(C=CC(N2CCN(C(=O)C(C)O)C(CCO)C2)=O)cc1C N1(C(C2(F)CCN(C(C3CC(=O)N3)=O)C2)=O)CCNCC(F)(F)C1 Cc1cccc(C(=O)NCCC2CN(C(=O)C(c3cncn3C)O)CCO2)n1 c1(C(N2CC(CC)OCC2)C(=O)NC2(C)CC2)cc(S(C)(=O)=O)co1 C(=O)(C1=CC2(CCN(C(=O)C(C)N=[N+]=[N-])C2)C1)N(C(CCCC)C)C C(=O)(CC1CCc2ccccc21)N1CC(N(C(C(C(C)(C)C)NC(C)=O)=O)C)C1 C(=O)(C1=CC2C=CC1C2)NCCN(C(c1sccc1CC#N)=O)CC CCC(C)(CCNC(=O)CCc1ccco1)NC(=O)CNC(C)=O N1(C(C2C(COC)CC2)=O)CCC(C)CC1.N(C)(S(N)(=O)=O)CC=O.C O=C(C#CC1CCCO1)NC1CCCN(C(c2cc3c[nH]nc3s2)=O)CC1 C1(N(C(C2CCOC2C)=O)CC)CCCN(C(c2nn(C)nc2Br)=O)C1 C(c1ccncn1)=CC(=O)NCC(C)=CC(=O)NC1(c2cccs2)CC1 c1(C2C(C=C)C2)nc(-c2ncccn2)nn1CCC(F)(F)CC N1(C(C(=O)NCc2cccs2)C2COC2)CCN(C2CC2)CC1 CC1(C(=O)NCCNC(=O)C2CC2)CCCN1C(C1(O)CCCCC1)=O c1(CN2CCC(NC(=O)CCc3ccoc3)C2)c(Br)ccc(Cl)c1F Cc1cn(C)cc1C(=O)NC1(CO)CN(C(C2CCOCC2C)=O)C1 CC1C(C(=O)NC2CCN(C)CC2C)CCCN1C(c1cnc2n1CCC2)=O c1(C(=O)NCC(CC)NC(c2cc(OC)no2)=O)csc(Cl)c1OC C#CC(CO)(CO)NC(C1CCCCC1NC(C1OCCOC1C)=O)=O C1(CNC(CC=CC)=O)CCCC1C(=O)Nc1csnc1 C1CN(C(=O)CCc2ccco2)CC1C(F)(F)F.C1(C(=O)N)CC12CC(O)C2 N1(C(C(C)=C2CCC2)=O)CCC(C(F)CNC(=O)CCS)CC1.c1ccccc1 C1(CC(=O)N(CCCCN(C(C(c2cnccn2)C)=O)C)C)CCOC1C Cc1c(CN2CCCC(NC(C3(CCF)CC3)=O)C2)cccc1Br NS(=O)(=O)c1cnn(CCC(N2CC(NC(=O)CCC3CC3)CC23CCC3)=O)c1 C(C)(CO)(C(F)F)NC(C=C(CNC(c1n(CC)nnc1)=O)C)=O CCCCC(CNC(=O)C(C)OCc1ccccc1)NC(=O)CCO.C(N)=O Cc1[nH]nc(Cl)c1C(=O)NC(c1cn(CC2CC=CC2)nn1)C N1(CC(=O)N)C(=O)CCC1=O.C1CCN(C(C2CC(=C3CCC3)C2)=O)CC1.C C=CCCCCCCCC(=O)NCCN(C)C(c1cccc(C(=O)NCC)n1)=O n1(CC=O)ccc2c(N)cccc12.C1(CC(=O)NCCC)C=CS(=O)(=O)C1 C1(C(=O)NCc2n(C)cnc2)CCN(C(=O)CCCC(F)(F)F)CC1(C)C c1(OC)cncc(C(=O)NCCC(O)CNC(c2ccoc2)=O)c1 c1(C(N2CC(NC(CC)=O)C(F)C2)=O)cccc2cc(C)ccc12 N1(C(c2cc(Cl)nc(Br)c2)=O)CCCc2c(F)cc(F)cc21 C1(C(F)(F)F)(CNC(=O)NCC2(CC(F)F)CC2)CC2CCC1C2 c1(C(=O)NCC2(F)CCCN(C(C3CCC(=O)O3)=O)C2)cc2nccn2c(O)n1 Cc1oc(C(=O)NC(C)C(CO)NC(C2CCCN2N=O)=O)cc1Br Nc1cc(C(N2CCCCC(NC(=O)CSc3ccccc3)C2)=O)cc(Cl)n1 C1(NC(c2cn[nH]c2)=O)CCCC(NC(C2CC2(F)F)=O)C1 c1(-c2ccc(NC(c3ncc(Cl)nc3Cl)=O)cn2)ccc2cc(O)ccc2c1 c1(CNc2c(C(=O)Nc3cc(C(=O)OC)no3)n[nH]c2)ccnc(F)c1 CCC(C)(C#N)C(=O)NC(CCN(C(=O)CCc1ncccn1)C)c1cccs1 Cc1nn(C)cc1C(=O)NC1C2CC1N(C(C1CC1(c1ccccc1)F)=O)C2 CN1CC(CC(=O)NCCC2CN(C(=O)CC(O)c3ccccc3)C2)C(O)C1 O=S(=O)(c1c[nH]ccc1=NC1CCC(NC)C1)NCCC(C(F)(F)F)NC1CC1 C(=O)(C#CC1CCOC1)N(CCC(N1CCC(O)(CCC)CC1)=O)CC c1(C(=O)NCCCCNC(C(CCOC)C)=O)cc(F)cc(F)c1OC N1(C(Cc2c(C)cco2)=O)CC(CNC(=O)C(C)(C)S(C)(=O)=O)N2CCC1C2 Cc1nc(C(=O)NCCC(C)NC(=O)CCc2ccsc2Br)c(C)s1 C#CC12C3C4C1C1C2C3C41C(=O)NCCCCCNC(=O)C(C)O.CCCC c1(NC(CN2CCN(Cc3c(OC)ccc(C)c3)CC2)=O)cccc2c1CCN2 c1(NC)ccc(F)cc1C(N1CCC(C)C(C)C1)=O.C(=O)(C1=NNC(=O)C1)N C1(C(N2CCC(COC)C2)=O)CCCN(C(c2c(C)noc2C)=O)CC1 C(=O)(C#CC1CCOC1)N(CCCNC(c1cnn(CCCC)c1C)=O)C(C)C C1(NC(C2C(C)C2C)=O)CCN(C(C2C3C4CCC(C4)C23)=O)C12CCC2 Cc1ccc(Br)c(C(=O)NC2(C3CCCN3C(c3cnn(C)n3)=O)CC2)n1 N(C1CCCc2c(F)cc(F)cc21)C(N1CCC(=O)NCCC1)=O c1(C(CC)NC(CC2CCCN(CC(CC)O)C2)=O)c(F)cccc1F CC1CC(CO)CN1C(=O)CNC(=O)Cc1nc(O)n[nH]1 CCC(F)(F)C(C)(C)C(=O)NC1CCCC(NC(c2cc3c(ncn3C)[nH]2)=O)C1 c1(C(C)(F)F)cc(C(=O)NCC2(O)CCC2)[nH]n1.C(=O)CCC1CC1.C C1(C)(C(=O)NCC(C)OC)CN(C(=O)CN2CCCC2)C1 CC(=O)CCCC(=O)N1CCC(C)(CNC(c2ccccc2SCC#N)=O)CC1 C1(NC(c2ccc(Cl)[nH]2)=O)CCN(C(c2cncs2)=O)C1 c1(C(=O)NCC2N(C(CCCOC(C)(C)C)=O)CCC2)cccc2ncccc12 C(CN=[N+]=[N-])(C(=O)NCC1(F)CCN(C)C1)NC(c1c(NC)scn1)=O Cc1oc2cc(C(=O)NC3CC(NC(=O)C(F)C4CCC4)C3)[nH]c2c1C c1(C(=O)NC2CN(Cc3ccc([N+](=O)[O-])cc3)CC2O)cccc2ncccc12 N1(C(C2(COC)CCCCO2)=O)CCC(O)(C)CC1.C(=O)CC1(C)CC1.N c1(C(=O)OC)cc(C)cnc1NCC(C)C1CC1.C1(C=O)CC2CCC(C1)C2 N1(C(C(C(CC)C)=O)=O)CC2CCC(C1)N2C(C1CCC1OCC1CC1)=O C(=O)(C1=Cc2ccccc2C1)N1CCC(O)(CCNC(=O)C2=CCC2)C1 C1(CC)(CC)CC(NC(c2cnc(O)n2C)=O)CN1C(=O)CNC=O.N c1(C(N2CCCC2)=O)ccc([N+](=O)[O-])c(N)n1.c1(OC)cc(CC(=O)N)on1.C C=CCC(C)(C)C(=O)N1CC(NC(c2cc(C)[nH]c2C)=O)CC(C)C1 CC1OC2(C(=O)NC3CCC(NC(=O)CCc4ccc(Cl)nc4)CC3)CC1C2 C(C(C=O)NC(=O)CC(c1cccs1)NC(=O)COCCCOC)OC c1(N2CC3CCC(O)CC3C2)[nH]c(=NCc2ncc[nH]2)nc2scnc12 CC(CC(=O)NC1CCCNC1=O)C(C)(C)NC(c1occ2c1CCC2)=O C1(C)(C(N(CC(O)CNC(c2occc2Br)=O)C)=O)CS(=O)(=O)C1 N1(C(CCn2ncn(C)c2=O)=O)CCC2CC(NC(C3CC3F)=O)CCC2C1 C(C(C)(C)CC(=O)N1CCN(C(=O)C(F)C2CCC2)C(CO)C1)OC(C)=O C=CC1(C(=O)NCCC2CCCN(C(C3(O)CC(CF)C3)=O)C2)CCCCC1 C1CCN(C(C2CCCN2C(C)C)=O)CC1.C1(C(N)=O)CN(C(N)=O)C1.C Cc1cc(Br)ccc1SCC(=O)NCC(C)NC(c1ccc(C#N)cc1)=O Cc1ccc(C(N2CCC3(NC(c4c[nH]c(Br)c4)=O)CCCC23)=O)cc1C#N c1(CNC(c2n(CCSC)nnn2)c2nnn(C)n2)cc(Cl)c(F)cc1F c1(C(N(C(C)CC)C)=O)nn(C)c2c(=O)[nH]cnc12.C(=O)CS(=O)(=O)C1CC1.N C(C(=O)NCCCCCC)(C(C)(C)C)NC(C)=O.C1(C=O)CC2(CCC2)CO1.N c1(CCC(N2CCC(NC(C3(COC)COC3)=O)C2C)=O)nc2ncccn2n1 CCC(F)(F)CC(=O)N1CCCC(NC(=O)C(C)NC(=O)C(C)(C)C)C1C c1ncc(-c2ccccc2)n1C.CC(CNC(=O)CC1(O)CC1)N(C(=O)C)C Cc1cccc(OCC(C)NC(N2CCN(CC3CCCOC3)CC2)=O)c1 c1(C(=O)NC2CC(N(C)C(C3CCCCC(=O)N3)=O)C2)cc2n(n1)CCCO2 CCCCCCCNC(=O)CC1CCS(=O)(=O)CC1.C1(C(=O)N)COC(=O)N1C c1(CNC2CC(NC(c3ncccc3F)=O)C2)cc(B(O)O)co1 c1(C(=O)NCCC(=C)C)sc(CC(F)(F)F)nc1C.c1(CC=O)cc(C)on1 C=CC1CCCCN1C(=O)CC1C(NC(=O)C=Cc2ccn(C)c2)CC1O c1(CCCC)ccc(C(C(=O)NCCC)N(c2ccccc2N(C)C)CC)cc1 C1(C(=O)NCCCCNC(C23CCCC2CCC3)=O)CC2(CCC2)CCO1 c1(C(N2CCC(CNC(C3C(C)(C)CC3)=O)C2)=O)cc2c(F)cc(F)cc2o1 C1(NC(CCCOCC)=O)CCCCN(C(C2CC(=O)NC(=O)N2)=O)C1 C1(C)(OC)CCN(C(C2(CCNC(=O)C=CCCC(C)C)CC2)=O)C1 c1(CC(=O)N(C)CC2CCN(C(C3(C)CCOC3)=O)CC2)cc(F)ccc1Br C(=O)(C(F)C(C)CNC(=O)CCc1cccn1C)NC(CC)(CC)CC c1(C(N2CC(C)(C)C2C2CC2)C(=O)NC2(C)CC2)ccc(OC(F)F)c(Br)c1 C1(C(=O)OC)(SC)CN(C(=O)CCC2CCNCC2)C1 c1(C=O)cccc2nonc12.c1(C(=O)NC2(CC)CCC2)cn(C(F)F)cn1.N CN=c1[nH]cc(C(=O)NC(c2ccccc2)C(=O)NC2CN(C)CC2C)o1 n1(C(C)C(=O)N(C)CCc2cc[nH]n2)cnc2c(N)ncnc12 Cc1ccc(NNC(=O)C(N)CCCNS(=O)(=O)C2CC2)c(C)c1 Cc1ccncc1C(N1CC(CNC(C2CC2c2ccncc2Cl)=O)C(C)C1)=O C1(CC(N2CCN(C(CSC(C)C)=O)C(C(C)C)C2)=O)Cc2ccccc2C1=O CC(C)(C)CCCC(=O)NC1CC1NC(c1conc1C1CCCO1)=O C1(C(=O)NCCc2n(C)ncn2)CCN(C(C2CCCCC2)=O)C1C(C)C C1(NC(Cc2scc(C)c2)=O)CN(C(c2c(C)noc2N)=O)CC1C c1(CC(=O)N(C(C)CNC(=O)C(N)=O)C)c(Br)ccc(Cl)c1F c1(OC)cccc(C(=O)NCC2CCCC2NC(=O)CC2CC2)c1O C(c1ccc(C)nc1)=CC(=O)NC(CNC(c1nc(CCCCC)sc1)=O)C N1(C(COCCCC(C)C)=O)CCCC2(NC(=O)C3=CCCS3)CC2C1 C1(CC(=O)NCCCCN(C(=O)Cc2cncc(O)c2)C)CCOC1(C)C C1(C(=O)NCc2cc(F)ccc2F)(OC)CCN(C(C)CCC(=O)O)CC1 c1(COC)ncsc1C(=O)NC(C)C(C)(C)NC(c1snnc1C)=O CC(CC(=O)N1CCOCC1CNC(c1cccc2ccoc12)=O)C(C)(C)C CC1(C)CCc2cc(C(=O)NCC(C)(CO)NC(c3c[nH]nc3F)=O)ccc2O1 N1(C(C2NCC2)=O)CC2CC(C1)CN(C(C1CC(C)(C)OC(C)(C)C1)=O)C2.CC c1(CC)c[nH]c2ncnc(NC3CCCC(NC(c4cc(Cl)nnc4O)=O)C3)c12 C1(C(C)C)OCCCC1C(=O)Nc1cn(C)nc1C1CC1 C1(CNC(c2cc(OC)no2)=O)CC(C)(C)CCC1.C(=O)CC=O.C1CC1 C(=O)(CC(C)C(F)F)NC(CNC(Cn1ncc(C#C)c1)=O)C(C)C C=CC(C)(O)C(=O)N1CCC(C)(NC(=O)CN2CCCC2=O)C1 C(C(C(=O)N(CCCN(C(=O)COC1CC1)C)C)c1ccccc1)C1C(C)C1 C1(NC(C=Cc2scc(C)n2)=O)CC12CCC(NC(=O)C#CC(C)C)CC2 c1(COC)cccnc1C(N1CC(CC(C)NC(c2c[nH]c(Br)c2)=O)C1)=O c1(C(=O)Nc2ccc(C(=O)N(CCCO)C3CCC3)cc2)cn2c(n1)CCC2 n1(C(CC)C)nc(C)cc1C(=O)OCc1ccc(C(F)(F)F)s1 C1(C(N(CC#C)CCOC)=O)CCCCN1C(c1cnn(C)c1C)=O N1(C(c2c(C(C)(C)C)[nH]cn2)=O)CCCC2(CCN(C(=O)COCC(F)F)C2)C1 C1(N(C2COCC2F)C(C(C)n2ccnn2)=O)CC2CC1CN2 CC1CC2(CC(NC(=O)CC34CCC3CN(C(c3ccnnc3O)=O)C4)C2)C1 C#CC1(C(=O)NOCC(=O)OC)CN(C(=O)C(CO)N(C)C)C1 N1(C(c2c(C(C)(C)C)[nH]cn2)=O)CC(F)CC1C.C1(C=O)CCS(=O)(=O)N1 c1(NC(C2CNCCN2Cc2ccc(Cl)cc2Cl)=O)ccc2nnsc2c1 C(CCCCCN=C(NCc1cnn(C)c1C)N(C)CC1CCCS1(=O)=O)SC C(=O)(C(F)C(C)(F)F)N(C(C)C(=O)NC(c1cnn[nH]1)C)CCC N1(CC(=O)N)CCNC(=O)C1.C1(C(N(CCC)CC)=O)CCC(N(C)C)C1 C12(C(=O)Nc3cnc(NC(C)C)nc3)CC3CC(C(=O)N1)C2C3 C=C1CC(C(=O)NOCCF)(CNC(=O)C(C2CCCO2)OCCC)C1 N1(CC=C)CCC(N2CCC(N(C(=O)C(C)SC)C)C2)C1=O N1(C(CNC(CSC)=O)=O)CCC(O)(CO)CC1.C12CC(C1)N2 N1(C(c2n(C)cnc2)=O)CC2CCN(C(c3ccc(OCC(F)(F)F)o3)=O)CC2C1 N1(C(CCCCC)=O)CCC2(CC1)CN(C(C1(S(C)(=O)=O)CC1)=O)CC2CO C(CC(C)C)(C(=O)N(C1CCCC1C)C)NC(Cc1c(C)n[nH]c1)=O C(=O)(CCC(=O)OC)N1CCC(N(C(C2C3CCC23)=O)CC)C1 C(=O)(C(O)CCCNC(C1(C)SCCCS1)=O)N1C(CC)COCC1 C12(NC(c3cc(CC)on3)=O)CCCCC1N(C(c1cnns1)=O)CC2 C1(C(N)=O)CCCCN1C(C1CCC(NC(C2CCCSC2)=O)C1)=O Cc1csc2cc(C(=O)NCCCCCCNC(C3(C(F)F)CCCC3)=O)[nH]c12 N(C(=NCCc1ccc(F)cc1)NCc1ccsc1C)C(C#C)C CC1CC(C)CN(CCCNC(=O)Cc2cccc(CC(=O)O)c2)C1 N1(C(C(C(C)C)C)=O)CCCN(C(c2ncn3c2COCC3)=O)C(CO)C1 Cc1ccc(F)c(-c2cn(C(C)CNC(=O)C(=O)N(C)C)nn2)n1 c1(C(=O)NC(CC(C)NC(c2c(C)ccc(C)c2)=O)C)cccc2c1NCCC2 Cc1cc(CC(N2CCC(C)C(NC(=O)CSc3nc[nH]n3)C2)=O)cc(C)c1 C12(CNC(C(CCOC)(C)C)=O)CCCCC1CN(C(c1cc(OC)no1)=O)C2 C1(CC(C)NC(CCN(CC#C)C(c2cncs2)=O)=O)CCCCC1 C1(CNC(C(CSC)O)=O)COC(C)(C)CN1C(c1occ2c1CCCC2)=O c1(C(N2CC=CCC23CCC3)C(=O)NCCCOC)ccc2cnccc2c1 C1(CC(=O)NC(C2CCOC2)C#C)CN(C(=O)CN(CC)C)CC12CC2 C1(CCC(=O)N(CCC(=O)NCCC)CC=C)CCN(C(=O)C(C)(C)C)C1 C1(CC)CC2CCC(C1)N2C(=O)C(F)(F)c1nccs1.CC1(F)CC(C=O)C1.N C(=O)(CC(C)(C)O)NCC1C(NC(C=COCC)=O)C1 Cc1cc(C(=O)NC(C)CN(C(=O)CCC(C)O)C)ncc1C#N CCC(COC)C(=O)NCC=C1CCN(C(c2nc(O)sc2C)=O)CC1 N1(C(C(c2ccc(Cl)cc2)N(C)C)=O)C2CCC(C2)C1C(=O)Nc1nn[nH]n1 c1(C(=O)NC2CCC(C)(CNC(c3c(C)cns3)=O)C2)c(F)ccc(C)c1O c1(C=O)c(C)nc2sccn12.c1(SC)cn(C)nc1C(=O)NCC1CC1.C C1(C(C)C(=O)N(CC(O)C(=O)N2CC(c3ccncn3)C2)C2CC2)CCN(C)CC1 C12(CC(=O)NC3COCCN(C(C4(Cl)CC4)=O)C3)CCC(CC1)OC2 C1(CC)C(C(=O)NCCC(CNC(c2cnns2)=O)OC)CCN1C N1(C(c2cccc(CNC(C)=O)c2)=O)CC2CC1CN(C(=O)CC(C)(C)CC)C2 c1(NC(=O)NC2(C(=O)OC)CCSC2)c(C#N)cnn1C Cc1cnc2cc(C(N3CC(O)(CNC(=O)Cc4ccc(F)cc4)C3)=O)ccn12 N1(C(C(C)CN)=O)CCc2cc(-c3ccccc3OC(F)(F)F)ccc2C1 C(=O)(C1CC=Cc2ccccc21)NCCCCCN(C)C(C1CC(O)CN1C)=O c1(OC)ccc2[nH]cc(C(=O)NCCNC(c3ccc(CC(C)C)cc3)=O)c2c1 CC(C)CC(C(=O)NC1COC2CN(C(=O)Cn3cnnn3)CC12)C(N)=O c1(C(=O)NCCCC(C)NC(c2c(OC)cccc2)=O)c(F)ccc(OC)c1F C1(C(=O)NCC(CC)NC(=O)C=Cc2ccc(C)o2)CCCCC1(C)C CCCCC(CC)C(=O)N(C(C)C(=O)NC(C)C(C)(C)C)CCC c1(NC(=O)C=C2CCN(C(=O)Cc3ccc(O)cc3)CC2)cc(Cl)c(Br)cc1Cl CC1(C(=O)NC2CCN(C(=O)Cc3cc[nH]c3)CC2F)CCC(O)CC1 CC1CCC(CNC(C2(F)CCCC2)=O)N(C(=O)C=CC=C(Cl)Cl)C1 C12(NC(COCC)=O)CC(C)(C1)OC2(C)C.c1nccc(C)c1C=O.N N1(C(CC(=O)N(C)C)=O)C(CC(N2CC3CC2CC3CF)=O)C2CCCC12 c1(CC)sc(C(N2CC(CNC(=O)Cn3cc(C)cn3)C(O)C2)=O)cc1C c1(NC(C2SCCN(C(c3cnc(SC)nc3)=O)C2)=O)cc(Br)cc2[nH]ccc12 N1(C(=O)NCC2(C#N)CCCC2)CCc2c(Br)ccc(F)c2C1 c1(C(N(CC(C)NC(C(c2cccc(F)c2)C)=O)C)=O)ccc[n+]([O-])c1 C1(NC(CCc2onc(CC)n2)=O)COCCC1NC(C1CCC=CCC1)=O C(=O)(C1=CCCCCC1)N1CCC(=CCNC(c2cc(SC)c(C)o2)=O)CC1 c1(CCF)ccccc1Cn1cc(CN2CCCCC2CCCl)nn1 C(=O)(CCN(OC)C(=O)C(CC)(CC)OC)NC(CC(CC)C)CO N1(C(c2cncc(OC)c2)=O)CCC(C)C(C)C1.C(=O)(C(C)(C)n1cnnn1)N N1(C(c2c(C)n(C)nn2)=O)CC2CCCC1CN(C(=O)CN1CCN(C)CC1)C2 c1(NCC(=O)NCC2(O)CN(C(CC(C)(F)F)=O)C2)nc2ccccc2s1 c1(C(=O)NCC(CNC(C2ON=C(C)C2)=O)(C)C)ccc2[nH]ccc(=O)c2c1 c1(CC)cccc(-c2cn(CCCCNC(c3cc(C)nn3CC)=O)nn2)c1 C1(CC)CC(O)CN1C(=O)CCCN(C(=O)CCOCC(F)F)C c1(C(N2C3C(C(N(CCC)CCN(C)C)=O)C(C3)C2)=O)ncc(F)cc1F N1(C(C2(CC#C)CC2)=O)CC(C)CN(C(c2ccccc2)=O)C(C)C1.C(C)C.S c1(C(=O)NCC2CCC(CNC(c3nccc(C)c3)=O)CC2)ccc(Cl)cc1C CN1CC(O)CCC1C(=O)NC1C2CCC(C2)C1C(=O)NCCCN1CCC1 CC1(C#CC(=O)N2C(CNC(c3cc4n(c3)CCOC4)=O)CC3CC23)CCCO1 c1(C(=O)NCC(CNC(CCOCCCOC)=O)(C)F)cnc(N)c(Cl)c1 c1(N2CCC(NC(c3c(CC)scc3)=O)C(F)C2)cc(O)nc(=O)n1C N1(C(CCN(C(=O)C=CC2CCCN2C)CC#C)=O)CCC2C(C(N)=O)C2C1 N1(C(CC(COC)COC)=O)Cc2occ(C(=O)NCCc3cc(C)on3)c2C1 c1(CC(=O)NC(C(C(C)C)NC(=O)C2=CCCCC2)C)ccc2c(c1)CCOC2 N1(C(C2CC(OC)C2)=O)CCCC2CN(C(c3cc(C)c(C)nc3O)=O)CC12 CN1CCC(C(N2CCCC(N(C(=O)Cn3nccn3)CCF)C2)=O)S1(=O)=O c1(CC)ccc(C(=O)NC2CCC2NC(=O)Cc2cc(CC)no2)c(N)c1 c1(CC(C(=O)NC2CC(N3CCC3)C2)NC(CC(C=C)C)=O)ccc(Cl)cc1Cl C1(C(=O)N(C)C)CCC(=C2CCC2)CC1.C1(=O)C(C)CCCN1C(C)C Cc1nc(NC2CCCCC2NC(=O)C(F)C(C)C)ccc1[N+](=O)[O-] c1(C(N(CCCCN(C(c2nncc(C)c2)=O)C)C)=O)cc(C#N)ccc1F C1(CC(C)C)CN(C(=O)C(c2ccco2)NC(c2cc(C#N)c[nH]2)=O)CCO1 C(=O)(C(=NOC)c1ccco1)N1CCN(C(c2c(C)cc(OC)nc2)=O)CC1C c1(C(=O)NCC2C=CCN2C(=O)CCO)ccc([N+](=O)[O-])cc1.CC(F)F C1CC(C)(C)C12CCC2.c1(NC(C(N2CCC(CC)C2)=O)=O)ccc(F)cc1.C C1(CNC(CCOCCC)=O)CC(C)N(C(=O)Cc2ccc(OC)cc2)C1 C1(NC(C(c2ccccc2)C)=O)CCCCC1NC(=O)CCC(C)N(C)C c1(C(=O)NCC(C)NC(c2c(C)ccnc2)=O)c[nH]c(=N)nc1O c1(C(N(C(=O)C(Cc2ccccc2)NC)CC)C)cc(C2CCCO2)n(C)n1 N1(C(C2C(=C)C2)=O)CCCN(C(=O)COc2c(C)cccc2C)CC1 c1(C(=O)NCC(CCNC(c2c(C)nc(CCC)s2)=O)O)cc(OC)ccc1F C1(O)(CN)CCN(C(C2(O)CCOCC2)=O)CC1 CN1C(=O)NCC1C(=O)NC1CC(F)(CNC(=O)CC2CCSCC2)C1 C(CC(O)C(=O)N1CCN(C(C)CNC(=O)CSC(C)C)CC1)SC c1(C(=O)NCCC(C)N(C(=O)CC2CCC=CCC2)C)ccn2ccsc12 C(=O)(C(CN(C)C)NC(=O)CCC1CCCOC1)N(C(CN(C(C)=O)C)C)C c1(C(=O)N)ccc2c(c1)NC(=O)NC2.C=CCC(C(=O)NC(C)C(C)C)C(C)C C1(C(=O)NC2CN(C(=O)OC)C2)CCN(C)C1.C1(CC(=O)N)CCCOC1 C(CCCCC(=O)NCC=Cc1cnn(C)c1)n1cc(COC)nn1 C1COCCN(C(=O)CC2CN(C)C2)C1.C1(C(=O)OCC)(C(=O)N)CCC1 CC(C)C(C)CC(=O)NC1CCN(C(c2ccc(F)c(Cl)c2)=O)C12CC2 c1(OCCC)ccc(C(=O)NCc2cn(C3CCNC3)nn2)cc1OCC C=CC(O)C(=O)NC(C)CNC(c1csc(C)n1)=O Cc1cccc2c(=O)c(C(=O)NC(C)C(C)NC(c3csc(C#N)c3)=O)c[nH]c12 c1(C(=O)NCC2(O)CN(CC(C3CCC3)OC)C2)ccc2nnc(O)n2c1 Cc1nc(-c2ccccn2)sc1C(=O)NC1CN(C(=O)CCc2scnc2C)C1 C1(C(=O)NC2CCCCN(C(Cc3c(C)nc(C)s3)=O)C2)CCC(C2CC2)CC1 C1(C(N2CC(N(C(CCCOC(C)C)=O)C)C3(C2)CC3)=O)CCCC(F)(F)CC1 C1(CC=C)(C(=O)NCc2ncnn2C)CCCN1C(=O)CC(C)(F)F C#CC1(C(=O)N)CCN(C(C2CC3(C2)CC32CC2)=O)C1.C1(C#N)CCOCC1.C N1(C(c2cc(C)oc2)=O)CCC(F)(F)C(CNC(c2cc(=O)n(C)o2)=O)C1 C(=O)C(F)(F)C(O)C1CC1.C1(NC(Cn2c(C(C)C)ncc2)=O)CCCCC1.C c1(C(=O)OC)oc(C(=O)NC(C)CN(C(=O)CN2CCCCC2)C)cc1C N1(C(C2=C(C)OCCS2)=O)CCC2(C=C(C(=O)NC3CCCCC3F)C2)C1 C(CC1c2ccccc2CCN1C(c1cocn1)=O)NC(CSCC)=O O=C(CCC1=CCCCC1)NCC1CC(C(=O)NC2CC(n3ccnc3)C2)CO1 c1(NC(=O)CC2CCN(Cc3cc[nH]n3)C2)nc2cccc(Br)c2s1 N1(C(C(C(CC)C)O)=O)CC(C)(C)OCC1CNC(c1ccc(F)s1)=O N1(C(CC(C=C)C)=O)CCCCC(N(C)C(c2ccc(OCC)c(OC)c2)=O)C1 Cc1cc2c(C(=O)NC3CCC34CN(C(=O)Cc3ccnn3C)C4)cccc2o1 N1(C(C(C2CC2)OCC)=O)CCC(NC(=O)C)C(O)C1.CCN(C)C.S c1(OC)ccnc(C(=O)N(CC(C)C(=O)N(C(C)C(F)F)C)C)c1 c1(C(N2CC(CC(C)NC(=O)CCNC(N)=O)C2)=O)cccc2ccsc12 C1(CN(C(C(CC)O)=O)C)CN(C(=O)CCCn2cccc2)CCO1 c1(C(N(CCn2cc(CNS(N)(=O)=O)nn2)CC)=O)cn2cccnc2n1 Cc1cc(Cl)cc(C)c1OCC(=O)N.C1C=CCN1C(=O)C(C)c1cccs1.C Cc1ccc2c(c1)C(=O)NCCN2C(=O)NC(c1ccccc1-n1cccn1)C CP(C)(=O)CCC(=O)N1CC2CC1C2CNC(c1cc(Cl)ccn1)=O C(C(=O)N)(C(C)(C)C)SC.c1(C=O)cc(C)n(C)c1.c1(CC)ccc(C)cc1 C1(CNC(C(C=C)(C)CC)=O)CCN(C(=O)Cc2cc(Cl)ccc2O)CC1(F)F c1(CNC(N2CCC(C)(C(=O)NC)C2)=O)cc(C(C)C)ccc1C(C)C N1(C(c2ncc(NC)nc2)=O)CC2CN(C(C3(O)CCC(C)(C)CC3)=O)CC2C1 O=C(CCCCCCn1cc(CN2CCOCC2)nn1)Nc1cnccn1 C1(NC(C2C(c3cn(C)nc3)C2)=O)CCCCC1NC(c1ncccc1Cl)=O c1(NC(c2nc(C)sc2)=O)ccc(C(=O)NCCc2ccccc2C)cn1 CCC(C)C(C(=O)NCc1cc(OC)no1)NC(=O)CC1CCOCC1 CC(CN=c1ccc([N+](=O)[O-])c(-c2ccccc2)[nH]1)NC(=O)C(CO)NC(N)=O C=C(C)C(CC(=O)N1CC2(CC(NC(=O)CC3CCCN3CC)C2)C1)OC CC(C)C(C)C(C)CC(=O)N1CC2CCC(NC(=O)CC(F)(F)C(F)F)CC2C1 c1(C(=O)NCCC(C)NC(C2CC3CCC2C3)=O)cnn2cnnc2c1 C=CC(C)(O)CC(=O)NC1CC(C)(NC(=O)C)C1.C(=O)C.C(C)=O.N c1(C(N(CCC)C2CC2)=O)ncccc1C(F)(F)F.C1(C=O)CCCCC1O.N CC(C(=O)NC(c1ccc(F)cc1)CNC(=O)CC1=CCCC1)S(C)(=O)=O CCCC(C#N)C(=O)NCC1(O)CCN(C(=O)Cn2cc(Cl)c(C)n2)C1 Cc1nn(C)c2nc(C(N3CCN(CCn4cncn4)CC3)=O)ccc12 C1(NC(c2nc(C)sc2)=O)CCCN(C(C2CC(N(C)C)C2)=O)CC1 C(=O)(CC(C)CC(C)(C)C)NCC12CN(C(C(C3CC3)SC)=O)C(C1)CO2 c1(OC)cc(C(=O)NC2CCCC2C)ccn1.c1(CC(=O)N)cc(C)cs1 CC1(C)Cc2cccc(S(=O)(=O)N3CC(OCCn4ccnc4)C3)c2O1 c1(C(=O)Oc2ccc(C)nc2)cccc2nc(O)ccc12 C1(C=O)CCN(C)C(=O)C1.S(=O)(=O)(CC(=O)NC1C=CC(C)C1)NC.N S(=O)(=O)(c1ccccc1N(C=O)Cc1cccc(F)c1)NC1(C#N)CCOCC1 N1(C(c2cc(C(F)F)on2)C(=O)NCCC)CCCCC1CN(C)C(C)C c1(CC(=O)Nc2cc(O)ncn2)ccc(-c2ccc(I)cc2)cc1 c1(NCC)ccc(CNC(=O)CCCCNC(=O)CC(C)COC)cc1 c1(C=O)ccc(N)c(C(F)(F)F)n1.C(C(O)C)N(C(C1(OC)CC1)=O)C.N c1(CCC(=O)NCC(C)N(C(=O)CC2CCOC2)CC)cncc(C)c1 C(=O)(C(C(=O)N1CCC(N(C(c2sccc2C)=O)CC)C1)C(C)C)OCC N1(C(CCc2ccnc(C)n2)=O)CCC(NC(=O)C(C2CC2)C2CC2)C(CO)C1 C(=O)(C(C)CC(=O)OCC)NC(CNC(C1CC(C#C)(O)C1)=O)C(C)C N1(C(C2CC(=O)NC2)=O)CCN(C(=O)CCF)CC1c1ncc[nH]1 C(=O)(C(C)CCCOC)NC(C(=O)N(CCC(=O)OC)CC)CO Cc1cc(C)c(NC(C2OCCC2NC(c2coc(C3CC3)n2)=O)=O)c(C)c1 C(=O)(C1CC=Cc2ccccc21)NC1CC(NC(c2c(C)cc(F)c(N)c2)=O)C1 C1CCC(C)CN1C(=O)C(F)C(C)C.Cc1nc(C(F)(F)F)c(C(=O)NC)o1 C1(NC(C2CC2(F)F)=O)CCC2CC1CN2C(=O)C(=CC1CCCCC1)F O=C(C1CCCc2nncn21)NC1(CO)CN(C(=O)C(F)(F)C2(O)CCCC2)C1 N1(C(=O)C=CC(F)(F)F)CCC2CN(C(=O)COCC(F)F)CCC2C1 CCCC(C)CC(=O)N1CC(C)(NC(C2CC2(c2ccccc2F)C)=O)C1 C=Cc1cnn(C)c1C(=O)NCC1CCC1NC(c1ccc(Cl)cc1O)=O c1(C(C)(F)F)ccccc1C(=O)NCC1CCCC1.C1(C=O)CC1[N+](=O)[O-].N c1(CNC(C(C2CCCN(C(=O)C=CCF)C2)C)=O)cnc(C2CC2)nc1 c1(C(=O)N)cnn(C)c1C.C1(C(C)NC(CN(C(COC)=O)C)=O)CCOC1 c1(OCC)cnc(C(C(=O)NCc2nnn(C)n2)N(C)C)nc1.C1CCOC1 C(=O)(CCCCCN=[N+]=[N-])N(CCCC(N1CCCC(C)(C)C1)=O)C c1(SC)c(C(=O)NCCN(CC(C)O)C(=O)CN2CCCC2C)cccc1F C1(CNC(COCC(=C)C)=O)(CO)CC12CCN(C(=O)CSC)CC2 O=C(C1=NNC(C(F)(F)F)C1)NC1CN(C(c2nccc(Cl)c2F)=O)CC1F CCC(C)C(C(=O)Nc1ccc(O)cc1OC)c1ccccc1 N1(C(c2c(CC)ccs2)C(=O)NC(C)CC)CCN(CC)CC1.CC(C)C c1(C=O)cnc(N)c([N+](=O)[O-])c1.CC1(C(=O)N)CS(=O)(=O)C1.C1CCCCC1 C=CC(CC)CC(=O)NC1CC12CCN(C(c1ncc(OC)cc1F)=O)C2 N1(C(CCN(CCC)C)=O)CCCC(C)(C)C1C(=O)NC(c1ccc(C)s1)C N1(C(c2[nH]cc(C)c2)=O)Cc2ccc(CNC(c3sc(Cl)nc3C)=O)cc2C1 N(C(=NCCC1(O)CCCOC1)NCC1CN(C)CCO1)C(C)C c1(C(=O)NCCC(C)C)ccc(OCC(N)=O)cc1.C1(C(=O)N)CCOC1=O CC(CC(N)=O)C(=O)NCC(C)(C)NC(c1ccn(C2CCCCC2)n1)=O CC(C)CC(C)(O)C(=O)N1CC2CCC(C(=O)NC3CN4CCC3(F)CC4)(C2)C1 Cc1ccc(C(=O)NC2CCN(C(C3(c4cccnc4)CCC3)=O)C2)cc1C Cc1nc(C(C)C)[nH]c(=NCC2(NC(c3ccc(=O)oc3)=O)CCOCC2)c1Br CS(=O)CCC(O)C(=O)N(CCNC(c1cc(CO)[nH]n1)=O)C1CC1 C1(NC(C(C)c2cccs2)=O)CN(C(=O)CCC(=O)C2CC2)CC12CCCC2 C(=O)(CC(=O)NCC1(CC(=O)NC2CC(CCC(=O)OC)C2)CC1)OC c1(C(N2CC(C(=O)Nc3c(C(C)=O)csc3)C(O)CC2)=O)cccc2ccoc12 C(c1cccc(Cl)c1)=CC(=O)NC1C2CN(c3nc(Cl)ncc3Br)CC12 Cc1cc(C(=O)NC2CN(C(c3cc(CO)oc3C)=O)C3CC23)c(C)o1 n1(C(CC)C)ncc2c(C(=O)NCCC(C)NC(c3cnns3)=O)cc(C)nc12 c1(C(=O)NC2C(NC(C(C(C)(C)C)SC)=O)CCC2)cccc2cnccc12 C1(NC(C2(C)CC2(Cl)Cl)=O)CN(C(c2ccc(CO)s2)=O)CCC1O C(CN=c1cc(Cl)nc[nH]1)C1CCN(C(c2ccc(CCC)s2)=O)CC1 c1(C(N2CC(C(=O)NCc3cnc(C)nc3)SCC2)=O)cc(Cl)cc(Cl)c1O c1(-n2ncc(NC(C(=O)N(C)Cc3cccc(F)c3)=O)c2)nccnc1C#N C1(C)(CNC(CCC)=O)CC(OC)CN1C(=O)CCc1cc(F)ccc1F O=C1CCCCC(C(N2C3CCC2C(CNC(c2cc4n(n2)CCC4)=O)C3)=O)C1 C1(NC(c2cc(C)[nH]c2C)=O)CCN(C(=O)C=CC(C)(C)C)CC1(C)C CCC(C)CC(C)C(=O)NC1CCC1CNC(c1cccc(N(C)C)c1)=O N1(CCC)CCN(C(=O)CC(O)CNC(=O)CCc2ccoc2)CC1 N1(c2nc(Cl)nc(Cl)c2)CCn2ncc(-c3ccnn3C3COC3)c2C1 c1(NC(C)=O)cccc(C(=O)NC2(C)CN(C(C3CCC(C)S3)=O)C2)n1 C1(C(N2CC(O)(C(C(=O)Nc3cn(C)nn3)F)C2)=O)CCCCC1OC(F)F N1(C(Cc2cn(CC)nn2)=O)CC(C(=O)NC2(CO)CC=CC2)C(F)(F)C1 c1(C(N2CCN(C(C(CC(=O)OC)(C)C)=O)CC2)=O)ccc2c(c1)NC(=O)CS2 C1(NC(=O)COC)(CF)CCN(C(C2(COC(C)(C)C)CC2)=O)C1 c1ccc2c(=NCCCC3CC3)[nH]c(=NC3CCCSCC3)[nH]c2c1 C1(NC(CSCCC)=O)COC2(CCN(C(c3nc4cc(O)ccc4[nH]3)=O)C2)C1 C1(C(=O)NC(CC#C)CC(F)F)CN(C(c2c[nH]nc2[N+](=O)[O-])=O)CCC1(C)C N1(C(C2C(CCC)C2)=O)CC2CC2(CNC(=O)Cc2nc[nH]n2)C1 CC1CC(CNC(C2CC(F)C2)=O)CN1C(=O)C(=O)NC1CC1 C1(NC(C(C)n2cccn2)=O)C=CCN(C(=O)CCc2cccc(F)c2)C1 C(CCCCC(=O)NC(C(=O)Nc1cnn(C(C)C)c1)C(C)C)OCC CCCCC(CNC(C1CCCN1C(=O)C1CC1)=O)NC(=O)C.C(CC)=C.O C(=O)(CS(=O)(=O)NCc1n[nH]cc1Cl)NCC(C)NC(C1CCCO1)=O Fc1cccc(C2CC(N3CCC(OCC4CCCCC4)CC3)CCO2)c1 C(CC(C)C(=O)N(C(C)(C(=O)N(C1CCCOC1)C)C1CC1)C)=CC N1(C(C2(CCOCC)CCCC2)=O)CCCN(C(C2CCOC2C(C)C)=O)CC1 N1(C(COC(CC)C)=O)CC2(NC(=O)CC(C)c3cccnc3)CCC1CC2 c1(C(C)C)c(C(=O)N(C)CCn2cccn2)cnn1-c1ccccc1Cl C(C(=O)NC(c1ccccc1)C(=O)NCCc1nc(C)cs1)(C(C)C)OC c1(OC)cc(COC(N2CCOC(C3CC3)C2)=O)ccc1N1CCCCC1 c1(C(N(CCC(C)NC(C=Cc2cncc(C)c2)=O)C)=O)ccc2nn[nH]c2c1 C(=O)(C1=CCC(C)CC1)N(C)CC1CN(C(Cc2cc(C)nn2C)=O)CC12CC2 CCC(C)CCC(O)CC(=O)NCCCN(CCC)C.C(C)(C(F)F)=CC(=O)N C1(C(=O)NC(CCC(=O)Nc2ccc(C)c(Cl)c2)C)Cc2ccccc2C1 c1(C(C)C)ncncc1NC(=O)C(C1CCN(C(C2CNC(=O)N2)=O)C1)C CCCC(C(=O)NCC1CCOC1(C)C)NC(=O)C(N)=O c1(C(=O)NC2C(C)CCN(c3cc(OCC)nc(C)n3)C2)ccnc2ccnn12 C(=O)(CCCC(F)(F)F)N1CC(C(C)NC(=O)CCC2CCCCCC2)OCC1 N1(CC)CCN(Cc2cn(-c3ccccc3)nn2)CC1CC(F)(F)F c1(OC)ccc(-n2cc(C3CCCN3C(C3CC4CCCC4C3)=O)nn2)cc1Cl C(=O)(CC1COc2ccccc21)NC(C)(CNC(C1(Br)CC1)=O)C1CCC1 C1(NC(c2c(C)csc2)=O)CCC2(CCN(C(=O)CCCC(F)(F)F)C2)C1 C(CCCCCC(=O)NC1CCCCC1NC(C12CCCC1C2)=O)SC C1(C(=O)NC2CC2c2cccs2)CCCCCCN1C(=O)CCc1nc(O)n[nH]1 N1(C(=O)NCCCn2nccn2)CCC(O)(c2cccc(Br)c2)C1 N1(C(C(C)OCCOC)=O)CCCC(C(N2CC(N=[N+]=[N-])C2)=O)C1 c1(CC)cccc2[nH]c(C(=O)NC3CC(C)N(C(=O)CC(C)(O)C4CC4)C3)cc12 c1(C(N(C2CCN(C(C(C=C)O)=O)CC2)CC(C)C)=O)cnc2[nH]cnc2c1 C(CCCCC(=O)N(C1CCN(C2CC2)C1)C)N(C(CC1N(C)CCC1)=O)C C1(CC)CCC(C(=O)NCC(CC(=O)N(C(CC)CO)C)OC)CC1 N1(C(CCCOCC=C)=O)CCCC(C(=O)NC(c2nc(C)no2)C)C1 C1(C(NCC)=O)CSCC(=O)N1.C1(CC(=O)NCC=O)CCCC1.C1CC1 N1(C(CCC(CC)CC)=O)CC(C)OC2(CCN(C(c3ocnc3C)=O)CC2)C1 c1(C(=O)NC(C2CCN(C(c3nc(C)oc3)=O)C2)C)cccc2c(C)[nH]nc12 c1(OCC#C)ncccc1C(N1CCC1CNC(=O)CCc1cc[nH]n1)=O c1(N(c2c(Cl)ccc(OC)c2)C2CCNCC23CC3)cc(Br)c(C)c([N+](=O)[O-])c1 N1(C(=O)NC(C(=O)OC)C(C)C)CCC2(CC1)CN(Cc1ccc(Cl)cc1C)C2 Cc1cc(C(N2CCC(O)(CNC(=O)CCc3cccc(O)c3)C2)=O)[nH]c1C c1(C(=O)NCCC2(O)CCN(C(C=CC(CC)C)=O)C2)cc(F)ccc1OC C1(NC(C(C)C2CCC2)=O)(CNC(C2CN(C3COC3)C2)=O)CCOC1 C1(C(N2CCOCC2CC2CCC2)C(=O)NC)CCCOCC1 N1(C(c2cnc(Cl)s2)=O)CCC(N(CCO)C(C2CCC23CCC3)=O)CC1 C1(CNC(=O)OC(C)(C)C)C2CCC(C2)C1C.C1CC1(F)F.C=O C(=O)(C(CC(C)C)Nc1cccc(-c2cc(C3CC3)no2)c1)OC N1(C(C(C)SC)=O)CCOCC1CC(=O)NCC(F)Cl c1(N2CC(CC)C(O)C2)cccc(S(=O)(=O)NC2(c3ccc(Br)cc3)CCC2)n1 N1(CC)CC(NC(c2nn(CC)cc2Cl)c2nnnn2C2CCC2)CC1=O C1(CC)(CNC(=O)CC=CC)CCOCC1.N1(CC(=O)N)CC2CC2C1 N1(C(CSCCOC)=O)CCCC(CNC(=O)CC2CCCOC2)(OC)C1 N1(C(C=C(CCC)CCC)=O)CCCC(CNC(c2ccc(=O)n(C)c2)=O)CC1 C(=O)(C(O)C1=CCCCC1)N1C(C)CC(CC(=O)NCc2c(C)noc2)C1 C(=O)C(C#N)C(C)(C)C.C(C(F)(F)F)N(C)CC=CC(=O)N(CCC)C.N c1cc2c([nH]1)CCN(C=O)C2.c1(COC)nocc1C.C(C)(C)C.C=O.N C(CN=C(NCC1C2COCC12)NCC1CC1)n1ncc(Br)c1 N1(C(C(CSC)C)=O)CCC(C2CCCN(C(=O)CCCCC(C)(C)C)C2)CC1 S(=O)(=O)(c1ccsc1C(=O)NC1CN(C(C2CC3CCC2O3)=O)C1)N(C)C CCCCCC(C)(CC)C(=O)N1CCC(CNC(=O)C(OCC)OCC)CC1 N1(C(C2N(C(CCn3ccc(C)n3)=O)C(C)C2)=O)CC2CC1(CO)C2 C(=O)(C1c2ccnn2CCN1C(c1scnc1C)C(=O)NC(C)C)OC c1(C(N2Cc3[nH]nc(I)c3C2)=O)nn(-c2cccc(Br)c2)c2c1CCC2 C1(NCCCN(C2CCN(CCC)CC2)Cc2ccccc2)CCOC(C)(C)C1 N1(C(C2CCCC(C)C2)=O)CCn2nc(CNC(c3cc(O)n(C)n3)=O)cc2C1 c1(OC)cccc(N(C(=O)C(CNC(=O)C(C)(C)C2CCOC2)N(C)C)C)c1 CC(C)C(F)(F)CC(=O)NCC1(C)CCCN(C(=O)Cc2ccsn2)C1 C(CC(C)C)(C(=O)NC1CC2C=CC1CC2)NC(C(C)OC)=O n1(CCCC)ncc(C(N2CC(CNC(c3[nH]c(C)cc3C)=O)C(C)C2)=O)c1C C(CCC)(C(=O)N1CCC2C(NC(c3cc(C4(C)CC4)n[nH]3)=O)C12)=CCC c1(CC(=O)N(CCn2cc(CCCC(C)O)nn2)C(C)C)cccc2c1SCCC2 C(=O)(CC(F)(F)C(F)(F)Br)N1C(C)C(NC(C2(O)COC2)=O)CCC1 Cc1ncc2ccc(C(N3CC(NC(=O)C(CC(C)C)N(C)C)C3)=O)cn12 C(=O)(N=c1c(Br)c[nH]c(C)c1Br)NC1CC(CC)C1 CC(C)(C)C(O)C(=O)N1CCC(OC(C2CN(C(=O)C3=CCCCC3)C2)=O)CC1 n1(C(C(=O)N(C(C)CNC(=O)CCOC(C)=O)CC)C)nccc1C C1(O)(C(=O)NCC(CNC(C2(C)CCNC(=O)C2)=O)CO)Cc2ccccc2C1 CN1CCC(C(=O)N(CCCCC(=O)NCC2CC(F)(F)C2)C)CC1=O C(=O)(C(C)(C)CC(F)(F)F)NCC(CN(C(C(C)n1ccnc1)=O)C)C O=S1(=O)CCC(c2nnc(C3CC3)o2)(NCc2cc3ccsc3s2)C1 C(CC(C(=O)NCC1(n2nccn2)CC1)NC(=O)CCOC1CC1)SC c1(C(=O)NC2C3(CN(C(C(C)(C)C(N)=O)=O)C3)SCC2)cc2ccoc2cc1F c1(C(N2C(CN(C(C(C3CCC(=O)N3)C)=O)C)CCC2)=O)cncc2sccc12 C(=O)(C(F)CCCC)NC(C(N1CC2C(CC)(C2)C1)=O)Cn1cccn1 C(=O)C(C)C(F)F.c1ccncc1.C(CCNCCC)N1CCC1.C(=O)C.N Cc1ccc(NC(C2CN(C(=O)CCC3CCC(=O)C3)CC2F)=O)cc1O C12(NC(=O)CCc3ccncc3)CCCC1N(C(=O)C(C1CC1)C1CC1)CC2 c1(C=O)cc(Cl)ncc1N.c1(SCC)cccc(CC(=O)NCC(C)(O)C)c1.N Cc1ccc(C#N)c(C(=O)C(N2CCNC(CC(F)F)C2)C)n1 C(c1cnccn1)=CC(=O)N.c1(CC)cnc(CC(N2CCCC2C2CC2)=O)[nH]1 N1(C(C(c2ccc(Cl)s2)C)=O)CCCC2(CCN(c3nnnn3C)C2)C1 CCCCCC(O)CC(=O)NCC1CN(C(=O)CC2CCCN(C(C)C)C2)CCO1 C(=O)(C1=NOC(c2ccc(OC)cc2)C1)N1C(C(N(OC)C)=O)C=CCC1 C1(NC(COCc2ncc(C)o2)=O)CC2CCC1C2.C(=O)CC=O.C1CC1.N C=CCC(C(=O)NCC1CN(C(c2ccc(C#N)cc2)=O)CCC1(F)F)C(C)C c1(CCC)cc(C(=O)NC2CC(NC(C3CC(C(F)(F)F)C3)=O)C2)sc1C CCCCCCOC(C)C(=O)N(CCC)C.c1(C=O)cccs1.C(=O)C1CC1.N Cc1ccnc2c(C(=O)NC(C)CNC(C3CN(C4CCC4)C3)=O)cnn12 C1(NC(C(C)C2CCC2)=O)CCCC1NC(C1(c2ccccc2)CCC1)=O C1(C(=O)NC2CC(CO)N(C(=O)C=CC(F)(F)F)C2)CCC2(CCC2)C1 c1(C=O)ccnc(P(C)(C)=O)c1.n1(CCC)nccc1C(=O)NC1CCCC1.N c1(C(N2C(CNC(c3c(C)occ3)=O)CCC2)=O)cc2ccc(Cl)cc2[nH]1 C12(NC(=O)CC3CC=CC3)CC1CN(C(=O)CC1(c3ccccc3)CCCO1)C2 c1(C(=O)NCCC(=C)C)sccc1S(=O)(=O)C(F)F.C1(C(=O)N)CC1(F)F C1(S(=O)(=O)NC(C)(C)C)(COC(c2cc(C)on2)=O)CCC1 C1(C)(NC(C23N(C(C(=Cc4ccco4)C)=O)CCC2C3)=O)CCCC1(C)C c1(CC)ccc(NC(c2ccnc(C)c2)=O)c(C)n1.C(=O)CCc1ccsc1.N CCCC(CC)C(=O)N1CC(O)(CCNC(=O)CC(C)(C)CC)C1 C1(N(c2nc[nH]n2)C(C2CC2F)=O)CC2(CCNCC2)C1 CCC(C)(C)CC(=O)NCCNC(=O)C(c1ccc(Cl)cc1F)(C)C N1(C(C(C(C)C)F)=O)CCC(CNC(=O)CNC(c2ccoc2)=O)C1(C)C Cc1cc(C)c(C(N2CC(CO)(NC(c3ccc4n[nH]cc4c3)=O)C2)=O)cc1C Cc1cn2c(n1)CC(C(=O)N)CC2.C(=O)(CC(C)N(C)C)N(C1CCCC1)CC c1(C(=O)NC(C(CO)NC(C(CC)n2ccnc2)=O)C)cc(C)ccc1F S(=O)(=O)(CCC(=O)NCC1(C)CCN(C(=O)Cc2ccccc2)CC1)NC Cc1cccc(OCCCC(=O)NCCC(C)(C)NC(=O)CC2(O)CCC2)c1 N1(C(C(CCC)S(N)(=O)=O)=O)CCC2CC(C1)CN(C(C1CCCC1)=O)C2 C1(NC(c2c(Cl)cn(C)n2)=O)CCN(CC2CCC2)CC1O CC1(CNC(C2C3C4CCC(C4)C23)=O)COCCN(C(=O)CCCCC2CC2)C1 C(=O)(CN=c1[nH]c2ccccc2s1)N(C1CCN(C(c2n[nH]c(C)c2C)=O)C1)C C1(NC(c2scc(C(N)=O)c2)=O)CN(C(=O)CC2CCC(=O)N2)C2CCCC12 CCCC(CCCNC(=O)Cc1csc(N(CC)CC)n1)NC(=O)C(C)C N1(C(C2CCOC2)=O)CCC(NC(c2cnc(O)s2)=O)CC1.C1CC1.COC CC(C)CC(F)C(=O)NC1CCC(CNC(=O)C(N2CCCC(O)C2)C)CC1 C(=O)(C(F)(F)C(F)(F)F)N1CC(C)CC(NC(c2c(C)ccnc2)=O)C1 O=S(=O)(c1c[nH]ccc1=NCC1CC1(F)F)NCC1(F)CCOC1 C=C1CCC(NC(C2(CNC(=O)C(C)=C3CC3)CCC2)=O)CC1 C(=O)(CCC(C)(C)F)NC1(CNC(C(C)NC(CC)=O)=O)CCC1 N1(C(CC(C)C2CCCC2)=O)CCC(CNC(c2ccno2)=O)C1(C)C N1(C(c2cnc(C3CC3)[nH]2)=O)CCCC2C1CCCN2C(c1cccnc1S)=O CC(C)CC(C(=O)N1CC2CC2(C)C1)C1CCC1.C(=O)CC(C)(C)CN(C)C.N Cc1cc(C(=O)N)c(S(N)(=O)=O)s1.C1(CC=O)CCCS(=O)(=O)C1.CCC Cc1cccc(C)c1CC(=O)NC1C=CCN(C(C2CC3(CCC3)CO2)=O)C1 c1ccc(Cl)cc1Cl.C(CCCNC(=O)CS)NC(CN(C1CC1(C)C)C)=O c1(N2C(C(=O)Nc3cccc(C(C)O)c3)CCCC2)ncnc2cccnc12 N1(C(CCOCCC)=O)CC(CC(=O)NCc2nc(C)c(C)s2)CC1C N1(C(c2cccc(F)c2Br)C(=O)NCCOC)CCCC12CCS(=O)(=O)CC2 Cc1ccnn1C(C)C(=O)NCCN(C(=O)C(=O)NCC(C)C)C C(c1c(C)noc1C)=CC(=O)N(CCCN(C(c1c(CC)c[nH]c1)=O)C)C C(C)(CCC(=O)N1CC(C)(C)C1C1CCN(C(=O)C(=O)N(C)C)CC1)OC N1(C(c2c(C)occ2)=O)CCN(C(c2cnc(O)c3ccsc23)=O)C(C)CC1C C1(NC(c2n(C)ncc2C(N)=O)=O)CC2CN(C(=O)CS(N)(=O)=O)CC12 c1(C(=O)N)ccc2c(c1)CCS2(=O)=O.C=CCCCNC(=O)CCc1nncs1 CCC(C)C(C)(O)CNC(=O)CCCNC(=O)CNC(N)=O c1(OCC(=O)NC(C(=O)NC)C(C)C)ccc(F)c(F)c1 N1(C(c2cnn(C)c2N)=O)CCC(C(=O)NCC2(C)CNC(=O)O2)C12CCC2 Cc1cn2cc(C(=O)NCC(F)CNC(=O)CC3CCN(C)C3=O)sc2n1 c1(N2CCN(C(C(CC)=O)=O)CC2CC#N)ncc2cc(Br)cc(F)c2n1 CC(C)C(F)(F)CC(=O)NC(C1CCCCN1C(=O)CCN1CCN(C)CC1)C N1(C(C2CC(C)(NC(CCC(C)OCC)=O)C2)=O)Cc2c[nH]nc2C(C)C1 C1(F)(CNC(CSC)=O)CCC(NC(=O)CS)C1.c1c(C)noc1C.C C(CN=c1cc[nH]cc1S(=O)(=O)NCC(C)O)Nc1ccc(CN(OC)C)cc1 N1(C(C2(C(=O)OCC)CC23CC3)=O)CC2CC(C1)CN(C(=O)C(C)OC)C2 C1(CN)CCC12CCN(Cc1ccc(CSC(F)(F)F)o1)CC2 C1(C)(CNC(c2c(CC)c[nH]n2)=O)CCN(C(=O)C(C)(C)n2cncn2)C1 C(=O)(C(F)n1ccnc1)NC(C1(CNC(C=C(COC)C)=O)CC1)C c1(C(N(C(CCNC(C2(COC)CCOC2)=O)C)C)=O)ccc2ncccc2n1 c1(C(=O)NC2(C)CCN(C(C3ON=C(CC)C3)=O)CC2)nc2ccccc2[nH]1 N1(C(C2(CC=C)CC2)=O)CC(C)CN(C(c2ccc(Cl)o2)=O)C(C)C1 N1(CCC)CCC(C(=O)NCCC(C)(C)C)CC1.c1(CC(=O)N)ccc(F)cc1 C1(n2cc(CC(CC)(C)O)nn2)CON(C(=O)c2ccc(Br)c(C(F)(F)F)n2)C1 N1(C(c2cc(COC)no2)=O)CCN(C(C2(F)CCOC2)=O)CC(C)C1 C(=O)(C1CCc2nccn21)N1CCC(C(=O)NCCc2cn(C)nn2)C1 Cc1cc(C(N2CC(NC(=O)Cc3cnc[nH]3)C3CC23)=O)cc(N)c1 CC1=CCC(C(=O)NCC2CCOC2C(=O)NCCC2OCCC2C)CC1 CC1(NC(=O)NC2CC(CCF)C2)CCCC(F)(F)C1 c1(C(=O)NC2CCN(C(c3c(CC)noc3)=O)C(C)C2)ccc2c(c1)C(=O)NC2 C1(CNC(CCS(N)(=O)=O)=O)C(C2CC2)CCN1C(=O)Cn1ncccc1=O CN1CC2CCN(C(=O)CNC(=O)CC3COCCO3)C2C1 N1(C(C(CC)=CCCC)=O)CCCCC1CCC(C)(C)NC(=O)Cn1cnnc1 CCCCC(CNC(=O)CC1CSCCS1)NC(=O)CC1(O)CCOCC1 c1(CC)nn(C)cc1C(=O)NC1CC(CCC(=O)N)C1.c1(CC)cnc(C)o1 C1(NC(CC(C=C)C)=O)CN(C(c2oc(C)nc2CC)=O)C(C)(C)C1 C1(NC(C2N(C(C(C)=CCC)=O)CCC=C2)=O)COCC(C)(C)C1 c1(OC)ccc(C(=O)N(C)C)cc1NC(=O)CCCc1ccc(Cl)cc1 C1(C(N2C(CN(C(C(CC)CC)=O)C)CCC2)=O)Cc2nccn2C1 N1(C(C)=O)CCC2(CCC2)CC1.C(=O)C(Br)Cc1ccccc1.C(=O)(C(=O)O)N N1(C(C(C(C)C)SCC)=O)CCn2nc(CNC(C3CC(C)C3)=O)cc2C1 Cc1nc(C(C)C)oc1C(=O)NCC(C)NC(C1CCCC(C)C1)=O CCCCC(C)(F)C(=O)N1CCN(C(=O)Cc2nncn2C(C)C)CC(CO)C1 CC(CF)CC(=O)NCCCCN(C(=O)C(O)CCc1ccccc1)C CC(C)CC(O)C(=O)NCC1(NC(=O)CC2CSCCO2)CC1 C1(C(=O)NCc2cn(CC(=O)NCc3nnc(C)s3)nn2)CC2CCC1O2 c1(C(N(CCCC)C)=O)cc(C(F)F)ccn1.C(C(C)(C)C)N(CC(=O)N)C C1(CNC(C2(CC=C)CCC2)=O)C2CN(C(c3ccc(CF)cc3)=O)CC12 c1(C(=O)OC)ccc(C(N2CC(F)(F)C23CCC3)=O)c(C(F)(F)F)c1 C1(OC)CCCC1NC(=O)C(C)N(C(=O)COC1CCCC1)C1CC1 c1(C(=O)NCCC2CCN(C(C3C(OC)CC3)=O)C2)ccc(Cl)cc1 CC1OC(C)C(C(=O)NCCCNC(=O)Cc2cnoc2)C1C.C1CCCC1.C c1(C(N2CC(NC(C(CC)C)=O)C2)=O)c[nH]c2cc(OC(F)(F)F)ccc2c1=O c1(C(=O)NCC(CCCC)NC(c2cn(CC)cn2)=O)nc(OC)ccc1F N1(C(=O)CN2CCC(O)CC2)CCCC2C(CCCN2C(=O)Cc2ccno2)C1 c1(C(C(N2CC(C(C)NC(C(COC)C)=O)C2)=O)C)ccccc1C N1(C(=O)OC(C)(C)C)CCCOC(CCNC2CC3OCCC3O2)C1 N1(CCCC#C)CCC(C(N2CCN(c3nc(O)n[nH]3)CC2)=O)CC1 S(=O)(=O)(c1[nH]c(=NCC2CC(CO)CO2)ccc1Br)NC(CC=C)C c1(C2N(CC(=O)NC3CCOCC3)CCC2)ccc2c(c1)OCCO2 c1(OC)ccnc(CNC(=O)C(C2CCN(C(=O)C(C)=C3CC3)C2)C)c1 Cn1nc(CN)cc1C(=O)NC1CCN(c2cc(Br)ccn2)CC1 C(CC(=O)NOCC(=O)N(C(CO)C(C)C)C)(OCC)OC c1(CNc2cn(C)c(C(N3CCC(O)C3)=O)c2)ccc2c(c1)CCCO2 C=CC1(CC(=O)NCC2CC3(CC3)C2)CN(C(C2(OC)CCCC2)=O)C1 Cc1cc(C(=O)NC2(CC)CC2)cc(N)c1.c1(C(=O)N)csc(C(N)=O)n1 Cc1cccc(C)c1.C(=O)CC(C)C(C)C.N1(CC(=O)NC(C)C)CCCC1.C C1CN(C(c2ocnc2C(F)F)=O)C2CC12.CC=O.C(COCCO)OC c1(OC)ncc(CN2CC(F)(C(=O)Nc3cccnc3-c3ccccc3)C2)cn1 c1(NC(=O)CN(C(=O)CCCC2CCC2)CC2CC2)cnccc1CO c1(C(C(=O)N(C(CNC(CC=CCC)=O)CC)C)C)ccnn1C C(C)(CC(=O)NC1CCCCN(C(=O)CCC(F)(F)F)C1)(C(F)F)N(C)C c1(C(N2CCCC2Cc2cn(-c3nccs3)nn2)=O)cc2ncccc2s1 C1(NC(=O)CC2CCCC(O)C2)CCCC(C(=O)NCc2ccccn2)CC1 N1(C(CCCCOCC)=O)CCC(NC(=O)C=CCCc2ccccc2)C12CC2 C1(NC(C2CCC(=O)CC2)=O)CCCC(O)CC1 CCC(C)CC(=O)C(=O)N1CC(C(N2CCC(O)C(C)C2)=O)CC(C)(C)C1 C#Cc1cccc(CCC(=O)NC(C)CCN(C)C(C2CC=CCC2)=O)c1 C1(C(=O)NC(CC2CN(C(CSCC(C)C)=O)C2)C)CCCC(C)(C)C1 Cc1nc(CNC(C2(NC(C3CC4CCC4C3)=O)CC2(C)C)=O)sc1C C1(NC(C(C(C)C)C(C)C)=O)CCC2(CC1)CN(C(=O)C(F)=C1CCC1)CCO2 C1(OCC(=O)N(C2CCC2(C)C)CC)CCN(C(c2cccs2)=O)C1 N1(C(COc2c(Cl)ccc(C)c2)=O)CC2(CCN(C(c3ccccc3C)C)C2)C1 Cc1cccc2nc(C(=O)NCC3CC(C)(C)CN3C(=O)C(C)(C)F)cn12 C(=O)(N=c1[nH]n(CC(F)(F)F)cc1C#N)Nc1c(C)c(Cl)ccc1F N1(C(C2N(C(C(N3CCOC3=O)C)=O)C(C3CC3)CC2)=O)CCC(F)(C#N)C1 C(CC(C)(C)C)(C(=O)NC1CCC(O)CC1)NC(c1ccn(COC)n1)=O N1(C(C(C)CC2CCCC2)=O)CC2(CC(NC(C3CC4(C3)CC(O)C4)=O)C2)C1 C1(NC(C2(C)CSC2)=O)CC1C1CCOCC1.C12(CC1)C(=O)NC2 N1(C(c2c(C)n(C)c(C(C)C)c2)=O)C(C)CC2CN(C(c3ccnnc3)=O)CC12 C(=O)(C1CCCn2nccc21)N1CC(C(C)NC(c2c(NC)ccc(F)c2)=O)C1 C(=O)(CCCCCCCCCO)N1C(CNC(=O)C(O)Cc2cnc[nH]2)C=CC1 C(CCC(C)(C)NC(=O)C(CN(C)C)c1ccccc1)NC(C)=O c1(C(N2C(CNC(=O)C(O)c3ccsc3)CCCC2)=O)cccc([N+](=O)[O-])c1Cl C1(NC(c2n(C=C)ncc2)=O)CC2CCC1(C(=O)NC)C2 C(N=c1cc(C)nc(C)[nH]1)C1CC2N(C(CN(C)CC)=O)C(CC2)C1 C12(NC(C(C)C)=O)CC(C)(C1)OC21CCN(C(=O)C=Cc2cc[nH]c2)CC1 C#CC1(NC(C2CC3CCC(C2)N3C(C2(C#C)CC2)=O)=O)CC2CCCC12 N1(CC(=O)NC(C)CC#N)CCN(Cc2cc(C(F)(F)F)cc(F)c2)CC1=O C1(NC(CCOCC#C)=O)CCN(c2nc3ccc(Br)cc3s2)CC12CCC2 CC1(C(=O)O)CC(F)CN1Cc1ccc(CS(C)(=O)=O)cc1 C(=O)(CC(C)CCC=C(C)C)N(CC)C(C)C.c1(SC)cc(C=O)co1.N CCCCC(C)CCC(=O)N1CC2(CC(NC(c3cnn(CC)c3)=O)C2)C1 N1(C(=O)CC2CCCN(C(C3(CO)CCOC3)=O)C2)CCc2nc[nH]c2C1 C=CCCCCCCC(=O)N1CCCC(C(=O)N(C(C)CC(F)(F)F)C)(CC)C1 C(CC(C)C(=O)NCC(C)CC(=O)NC1CCCC1O)OC C(C#Cc1cnn(C)c1)NC(C(c1ccoc1)NC(Cc1cc(CC)no1)=O)=O C12(OC)CCC(C(=O)NC(C)CN(C(=O)C(F)C(C)C)C)(CC1)C(=O)C2 N1(C(CC(CC)C2CC2)=O)CCCC(CCNC(=O)C(C)(C)n2cccn2)CC1 C1(C(N2CCN(C(C3C(C)(CC)C3)=O)C(COC)C2)=O)CCC2CC1C2(C)C Cc1[nH]nc(C(=O)NCCCCC(C)NC(=O)CSC(C)C)c1C c1(CN(C2CCC(O)CC2)C)cccc(C(N)=O)c1F c1(C(C)(C)C)ccc(CCC(=O)NC2CC2NC(=O)CC2COCCO2)cc1 CC(C)CC(C(=O)NCCCCC1CCN(C(C2CCCSC2)=O)CC1)C(N)=O c1(CCCC(=O)NCC2CCCN(C(c3nc(C)sc3)=O)C2)cc(F)ccc1F c1(C(=O)NCC2N(C(c3c(CC)cc[nH]3)=O)CC(O)C2)cnn2ccsc12 C(CC(CC)C(=O)N1CCCC(C)(C(=O)Nc2cn(C3CC3)nc2C)C1)=CC N1(C(C=C(C)C(C)(C)C)=O)CC(C(F)(F)F)OCC1C.C(=O)C.CC(C)C N1(C(c2cc(C)n(C)c2C)=O)CCC(C2CC(NC(=O)CS)C2)C1.C(C)(C)C CCC(C)C(=O)C(=O)NC12CC(C(=O)NC3CCCC(O)CC3)(C1)C2 c1(C(C(=O)NCCC2CCN(C(=O)C3CC3)C2)F)ccccc1.O=C1CS1 c1(C(CC)NC2CCC(Oc3ccccc3)CC2)c(C)cc(C)cc1C Cc1nnc(O)c(C(=O)NCCC2CC3CCC(C2)N3C(=O)C2=NOCC2)c1C C1(C(N(C(C)C)C)=O)CN(C(C)C)CCO1.C(C=O)=CCOCCOC.N c1(CC2CCC(COC)N2C(=O)C(CO)C(C)(C)C)ccccc1N=[N+]=[N-] C(=O)(C1CCCn2nccc21)NC1(CC=C)CCCN(C(C2CC(C)(F)C2)=O)C1 C1(NC(COCC#C)=O)CCN(C(c2cn(C(C)C)nn2)=O)CC1CC Cc1cc(CNCC2CC(C(=O)Nc3[nH]cnc3C#N)C2)n(C)n1 N1(C(c2c(N)sc(-c3ccccc3)n2)=O)CC2CCC1CN2C(=O)CO.CC(=O)O c1(SCC(=O)NCC(CC)NC(=O)CCS)ccc(C#N)cc1.CC(C)C C(=O)(CC(C)(C)CC(F)F)NC1(CC=C)CCCN(C(=O)CCC(C)(C)O)C1 Cc1ncc(C(=O)NCC2CCCCC2NC(C2CCC(=O)N2)=O)cc1C#N c1(C(=O)NC2CN(C(C(CCC)O)=O)CC2C)cc(C)c(OC)c(C)c1 C=CCC(CC(=O)N1CCS(=O)C(C)C1)NC(=O)Cc1cccs1 S(=O)(=O)(c1ccccc1Cl)N1CC(NC(c2ccc(CC=C)cc2)=O)C(C)C1 C1(C(N2CCC(Oc3cccnc3)C2)C(=O)NCCC2CC2)CC12CCOCC2 C1(NC(COC2CN(C(C)=O)C2)=O)CCC2CCN(C(C3CCOCC3)=O)C1C2 CC1CC(NC(c2ccc(-n3cnnn3)cc2)=O)CN(S(=O)(=O)CC2CCC2)C1 C1(C(N(CC(N2CCCC2)=O)C)=O)CCN(C(C23CCC(CC2)C3)=O)CC1(C)C N1(C(C2CC(S(C)(=O)=O)C2)=O)CC2CCC1C1CN(C(c3ccns3)=O)CC21 C#CC1(NC(=O)CCCN(C)C(C2CCCO2)=O)CC(F)(F)C1 C1(F)(CNC(C(c2ccccc2)OC)=O)CCN(C(C2(C)CC2C)=O)CC1 N1(C(C2(CC#C)CCC2)=O)CC(CNC(=O)CC2CC2C)(OC)C1 C(C)(CNC(=O)Cc1cnn(C)c1)(CO)NC(CN(CCOC)C)=O c1(CC)ccsc1C(=O)NCCCCN(C)C(C12COCC1C2)=O c1(NC(C2CC2C(=O)Nc2cnnc(Cl)c2Cl)=O)cc(CO)ccc1F c1(CCC(=O)NC2C3CC2N(C(=O)CCc2ccon2)C3)cccc([N+](=O)[O-])c1 Cc1cc(C(N2CCC(C)C(NC(=O)CSCC(C)C)C2)=O)c2c(n1)CCCC2 N1(C(C2(C)COC2)=O)CCN(C(=O)Cn2nc3n(c2=O)CCCC3)C2COCC12 S(=O)(=O)(CC(=O)NC(C1CN(C(=O)C(C)(C)F)CCO1)C)N(CC)CC N1(CC(N2C(c3ccccc3)CN(C)C(=O)C2)=O)CCCN2CCCC2C1 C(=O)(C(O)C(C(C)C)OC)N1C(C=O)(C(C)C)CCC1.C=C(C)COCC c1(C(N2CCC(NC(C3CCN(C)C3)=O)C23CC3)=O)cn2c(Br)cnc2s1 C1(C(=O)NC2C(CCC)C2)CCn2ccnc2C1 c1(NCc2cn(C3C(CNC(C(C)CO)=O)COC3)nn2)ccc(C#N)nc1O CCC(C(=O)NC(Cn1cccn1)C(=O)NC)NC(C)=O.c1nnc(C)s1.C S(=O)(=O)(c1cc(C)cnc1N(CCCOCC1CC1)C)N1C(CC)CCCC1 c1(C(=O)NC(C)(CO)C2CCCC2)cc(C)on1.c1(C=O)cc(C(N)=O)c[nH]1 CCCCC(C(=O)NCCc1nc[nH]n1)NC(C1CC(N=[N+]=[N-])C1)=O c1(C(=O)NCC2(F)CCCN(Cc3cc(Br)co3)C2)cc2c[nH]nc2cc1F O=C(C1=C(Cl)CCCC1)NC1CCN(C(=O)CC2CCCOC2)C1C1CC1 N1(C(Cc2nc(C)sc2C)=O)CCCC2C(NC(=O)C(C)C(C)(C)C)C(C)(C)C12 N1(CCC)CCCCC1C(=O)NCC1CCCC1.c1(CC(=O)N)ccc(C)s1 c1(OCCCNCC)cc(Cl)ncc1C(N1CCCCC1)=O.c1(N)nnc(C)s1 C(CCN=C(NCCSc1cnc(C2CC2)o1)NC1CCS(=O)(=O)C1)=C(C)C N1(C(C(CC)(C#N)CC)=O)CCCC2(CCCN2C(c2cnc(C3CC3)[nH]2)=O)C1 n1(CC(N2CCCC2)C)c(N2CCC(CC#N)C2)nnc1CCN(C)C Cc1cncc(C(=O)NC2COCC2NC(C2CC2Br)=O)c1 c1(CCC(=O)NCC2C(C)CN(C(C3CCCOC3)=O)C2)ccc2ocnc2c1 c1(NCc2cc(OC)no2)ncc(S(=O)(=O)NCCC(C)CCO)cc1Cl c1(C(=O)NC2CN(C(C3CC3(F)Br)=O)C2)cc2ccc(Cl)cn2c1 CN(CCCC(=O)NCC1CC(NC(C2CCCO2)=O)CC1O)N=O c1(NC(CC=CCNC(c2ccc(C)c(O)c2)=O)=O)ccc(C)c(C#N)c1 c1(C(=O)OC)cc(Cl)cc(S(=O)(=O)NCCn2cnnc2C(C)C)c1F N1(C(C=C(C)C2CC2)=O)CCC2(CCCCN(C(=O)CN3CC=CC3)C2)C1 CN=c1nc(N2CC3(C)CCC3(C)C2)[nH]c(=NCc2cccc(N)c2C)[nH]1 C1(C(=O)NC2C(NC(C(CCC=C)(F)F)=O)CCC2)CCc2ccccc2C1 C1(NC(c2ccc(CCCC)cc2)=O)CCCCCN(C(C2(C)CC2)=O)C1 c1(NCC2CCC(NC(c3ccn(C)n3)=O)CC2)cc(F)ccc1OC(F)(F)F N#Cc1cc(C(=O)NC2CC2CNC(C2CCCC(=O)N2)=O)ccc1F C(=O)(CC(C)(C)C#N)NC(CCC)CNC(c1ccnc(CO)c1)=O CCC(C)C(C)CNC(=O)C(C1CN(C(C2(C(=O)CC)CC2)=O)C1)OC CC(CCNC(c1cccc(N)c1)=O)CCNC(C1(C)CCCN1C)=O c1(C(C(=O)NCCCn2nccn2)NC(C=CC(C)C)=O)cn(C)nn1 c1(NC(CC(COC)NC(C2CCC2)=O)=O)cccc(F)c1OC.C1CC1.C CC(C)CC(O)CC(=O)N1CC(O)(CCNC(C2CN3CCC2CC3)=O)C1 Cc1cc2c(cc1O)CCN(C(=O)CC1CCC3(CCOCC3)CO1)C2 CC(C)C(C(=O)NCCC1CC(F)(F)CN1C(=O)Cc1c[nH]ccc1=O)C(C)C N1(C(C2CCN(C(C3CC34CCCC4)=O)CC2)=O)CCCC12CCCOC2 c1(CCC)ccc(C(=O)NC(CO)C(C)NC(=O)C=Cc2cnc[nH]2)cc1 c1(C(=O)OC)ccc(C(=O)N(CCC)C)c(C)c1.c1(C=O)ccnn1C(C)C c1(NC)cncc(C(=O)NC(C2CN(C(=O)C(C)OC3CCCC3)C2)C)n1 C1(CN(C(c2cccc(CCC)c2)C(=O)NC2CC2)C)CC12CCOCC2 c1(CC(=O)NCC2C(NC(c3nc(CCC)sc3)=O)C2)c(C)noc1Cl C=CC1(C(=O)NC(C2CSC2)C)CCN(C(c2cccn3nccc23)=O)CC1 N(C1CCc2ccccc21)(CCC)Cc1cscc1Br Cc1csc(C(N2CC=CC2CNC(C2CCCN2C(N)=O)=O)=O)c1Br C1(C(=O)NC2(CNC(C34CC(CO3)C4)=O)CCCC2)CCn2ncnc2C1 N1(Cc2c(OC)nccc2)CCc2c(-c3ccc(O)c(F)c3F)cccc2C1 C(=O)(C1CCCc2ncnn21)NCC1CCCC2CN(C(C(C)C#N)=O)CC21 C1(CCOC)(C(=O)NC(C)C2CC2)CCCC1.C1CCOC1=O.C(=O)C.N c1(CNC2C(C(=O)Nc3n(C(C)(C)C)ncc3)CCC2)csc([N+](=O)[O-])c1 N1(C(c2cn(C)[nH]c2=N)=O)CCC2CCN(C(C3CC34CCCC4)=O)CC12 c1(C(=O)N(C2CCN(C(C3CC(O)C3)=O)C2)CCO)cc2n(n1)CCCO2 CCCC(CC)CC(=O)NCC(CCOC)NC(=O)CNC(c1ccccc1)=O c1(C(=O)NC(CC=C)CNC(c2cn(CC)cn2)=O)cn(CCCC)nc1C N1(C(C2(CNc3cc(CC)ncn3)CC2)=O)CCC(O)C(C)(CO)C1 c1(C(=O)NCCC)cncc(Cl)c1.C1(C#N)(C=O)CCOC1.C(C(F)(F)F)O C(=O)(C(C)=Cn1ccnn1)NCC(CC)NC(=O)Cc1csc(C(C)C)n1 C(CCC(C(=O)NCC(C)(C)C#N)NC(c1coc(SC)c1)=O)OC C1(C(N2CCC(CC)(CC)CC2)=O)CC(C)(C)CCN1C(c1cc(C)c(C)s1)=O c1(C(=O)NCC(CCNC(c2ccc(C)nc2)=O)O)oc2c(C)cccc2c1C CCC(C)C(C(=O)NCc1ccc(C(=O)NCC(C)(C)N(C)C)cn1)OC C1(C(N2CCC(C3CCCN3C(=O)COC3CC3)CC2)=O)CC(C2CC2)=NO1 C(=O)(C(CC)C(C)C)NCC(CC=C)NC(C1(P(C)(C)=O)CC1)=O C1(O)(C(C(=O)OCC)(F)F)CCN(C(c2cc(C)c(O)nn2)=O)CC1 c1(C(N2CC3C(NC(c4nc(O)nc(O)c4F)=O)C3C2)=O)ccc(O)c(F)c1F C(=O)(CCS(C)=O)N(C)CC1CCCN1C(c1ccc(F)s1)=O Cc1cc(C(=O)NC2CCCN(C(=O)CSC(C)C)CC2)cc(C)c1O c1(C(N2CC3C(CO)C3C2)=O)ccc(C)nc1Nc1cc(OCC)ncn1 c1(C(N2CC(N(C(CCCN(C)C)=O)C)C2)=O)ccc(Nc2ccccc2)cn1 C12(C(=O)OC)CCNCC1CN(C(c1nccc(C3CNC3)n1)=O)C2 CCCCCCCCC(=O)N1CCC(C)(C)CC1C(=O)NCC1CC(OCC)C1 C(=O)(C1CCOc2ccc(Cl)cc21)NCCCCNC(CC(CCSC)O)=O C#CC1CCC(NC(=O)CCc2ccccc2COC)CC1 N1(C(CC(C)C(F)F)=O)CC2(CCN(C(=O)CNS(=O)(=O)c3cccs3)CC2)C1 N1(C(CCCOCC)=O)CCC(NC(c2nonc2N)=O)C(C)C1 C1(C(=O)NC2CN(C(c3nc(C)sc3C)=O)CC(C)C2)CNC(=O)C(C)(C)C1 C1(C(N2CC(C)(NC(CC3(CC=C)CCCC3)=O)C2)=O)CCCC(=O)O1 C1(C=O)C2CC3C(C2)C13.C12(CCNC(C(C)N3CCC3)=O)CCC(CC1)C2 N1(C(Cc2c(C)cco2)=O)CC(NC(C2CCCN2C2CCCC2)=O)C(C)(C)C1 C(=O)CC1CCc2ccccc21.C(CS(N)(=O)=O)C1(C(N(CC)CC)=O)CCC1 C(=O)(C1=CC2C=CC(C1)C2)N1C(CC(=O)NC23CCC(CC2)C3)CC1 C(C)(C=O)(C(C)C)NC(C)=O.c1(N2C(C)CCC2)nc(C(F)F)nc(=N)[nH]1.N CCC(CN(C)C)C(=O)N1CCCC(C(=O)NC2CCOC2=O)C1 N1(C(CN(C(=O)Cc2ncccn2)C(C)C)=O)CCC(F)(F)CC1 Cc1cnc(C(N2CCC(N(C)C(c3ccc(CN(C)C)nc3)=O)C2)=O)nc1 C1(NC(C(C)(C)C)=O)CCCC(CC(=O)NC2CCN(C3CC3)C2)C1 C1(CC=C)(C(=O)NCC(CNC(c2conc2C2CCC2)=O)CO)CCOC1 c1(OCC)ccnc2sc(C(=O)N(CCC(C(C(=O)N)O)C)C3CC3)cc12 C(=O)(C(CC)CCOC)NC(C1CCCN(c2nnc(CC)o2)C1)C CC(CCCN=c1cc(C(N)=O)nc(Cl)[nH]1)NC(c1cc2n(n1)CCO2)=O N1(C(c2coc3c2CN(C(CC(CCCC)O)=O)C3)=O)CCc2cccc(C)c21 Cc1ccc(C(=O)NCCNC(=O)Cn2nnnc2C)c(F)c1Cl C1(C(N2CCC(COC)C2)=O)C2CCC3(COC(=O)C13)O2.c1(C=O)csnn1 c1(C(=O)NCCC(C)N(c2cc(-c3cccs3)ncn2)C)c(F)ccc(F)c1F N1(C(C2N(C)C(=O)OC2)=O)CC2(C1)CN(C(=O)Cc1coc(-c3cccs3)n1)C2 C(C(C)C(=O)NC(C)(C)CC1CCC1)NC(C=CC=CC)=O C=CC1(C(=O)NCC2CCN(C(c3cc(CCC)[nH]n3)=O)C2(C)C)CCCCC1 C1(N(C)C)CCCN(C(=O)C=CCNC(c2cnc(Cl)s2)=O)C1 N1(C(C=COCC)=O)CCC(NC(c2cc(C(F)F)cc(F)c2)=O)C(CO)CC1 C1(OC)CCOCC1NC(=O)CC1(CNC(c2cc(C)on2)=O)CC1 c1(C(=O)NC2C(NC(C(CC)SCc3ccccc3)=O)C2)ccc2n[nH]cc2n1 C(CC1CCCC1)(C(=O)N1CCC(C(=O)OC)O1)NC(CC(CC)OC)=O C1(C(C)NC(C=CCN(C)CC)=O)CCCCN1C(=O)CC(F)(F)F C12(NC(=O)COC3C=CC(C=O)C3)CC3CC(CC1C3)C2.c1ncc(Cl)cn1 N1(C(c2ccc[n+]([O-])c2)=O)CCC2(CC1)CC2NC(C12CCC(CO1)C2)=O C(=O)(CC(N)CC(=O)NCC1CCNCC1C1CC1)OC Cc1cc(CCCNC(C2(NC(=O)CC3C=CCCC3)CCSC2)=O)on1 Cc1nn(C)cc1CC(N1CCC(CCNC(C2(n3cncn3)CC2)=O)CC1)=O C1(CC)CN(C(=O)Cc2cccnc2)CCC1NC(=O)C(C)CN(C)C N1(C(C2(SC)CCC2)=O)CCCN(CCNC(C23CCCC2OCC3)=O)CC1 N1(C(Cc2ncc(C)[nH]2)=O)CCC2CN(C(C3CC(=O)N(C)C3)=O)CC12 n1(CC)ncc2cc(C(=O)NCCN(C)C(C3CC4(CCCCC4)C3)=O)cnc12 C1(C(N2CC(C#N)C2)=O)CCCCCCN1C(=O)Cc1ccc2c(c1)CC2 C(=O)(C1SCc2cccnc21)N1CCC2(N(C(c3c(CC)ncs3)=O)CCC2)C1 C1(N(C(C(c2c(C)cncc2)C)=O)C)CN(C(C2C=CCC2)=O)CCC1C CCCCC(F)C(=O)N(CC(=O)NC(CC)C(N)=O)C C12(C(N3CCCC(N(C(CCCOC(C)C)=O)CCO)C3)=O)CC=CC(C1)OC2 N1(C(C(C)=NOCC#N)=O)CC2(C(N3CC(CO)C(CO)C3)=O)CCC1CC2 Cc1cccc(CCC(=O)NC2CC2CNC(C2(n3cccn3)CC2)=O)c1 C12(CNC(CN(C)CCO)=O)CC(CN1C(=O)CC1CC3(CCC3)C1)C2 S(=O)(=O)(c1cccs1)NC(C)C(=O)N.c1(CC(=O)NC)cnco1.C1CC1 Cc1[nH]c(C(=O)N)c(C)c1C(N1CCC(C(F)(F)F)C1)=O.c1nccc(C#N)n1 CC1(CNC(=O)Cn2ccsc2=N)CCCN1C(=O)Cn1cc(Cl)cn1 C1(C(N(CC(=O)NC)C)=O)CCN(Cc2ccccc2Oc2ccccc2)CC1 O=C(CONC(=O)C1CC(NC(c2cccnc2)=O)C1)NOC1CCOC1 C1(C(=O)NCCCCN(C)C2CC2)CCC2CCCCN12 N1(C(C(C)(C)OC(C)C)=O)CC(CC=O)C(C)C1.C1(CC)CC2(CCC2)C1.N N1(CCNC(C(C)Sc2nnnn2C2CC2)=O)Cc2ccnc(Cl)c2C1 c1(CC)nocc1C(=O)NCc1ccsc1C(=O)NC.c1nc(C)no1 N1(C(CCOC)=O)CC(C)(C)C1C1CCN(C(=O)CC2CCCC2O)CC1 Cc1cccc(C(N2CCCCC2C(=O)NCC2CN(C3CC3)C2)=O)c1C c1(C(=O)NCCCCOC)sc(C)nc1C.C(c1cccs1)=CC=O.C1CC1 Cc1sc(C(N2CCOCC2CNC(c2cc(Cl)cn2C)=O)=O)nc1O C1(C(C(N2CC(CCCCC)C2)=O)F)CCN(C(=O)Cc2nocc2C)C1 c1(OC)ccccc1C(N1CC(CF)(NC(=O)C=CCCC(C)C)C1)=O C1(N(C(C(C)Oc2ccc(O)cc2)=O)C2CC2)CCC(O)(C(F)(F)F)CC1 C1(F)(C(=O)NC2CCN(C(C(CC)(F)F)=O)C2)CCCN(C)C1 c1(C(=O)NC2CN(C(C(CSC)C)=O)CC2O)cnc(C)c(Br)c1Cl C(=O)(C1CCCn2cnnc21)NC1C(C)N(C(=O)COc2ccc(F)nc2)CC1 C(=O)(CCCCCn1cc(C2CCN(C)C2=O)nn1)NC(CC(C)O)C C(=O)(CCS(=O)(=O)CC(C)C)N.Cc1cc(Cl)cc(C)c1C(=O)NC(CO)CC C(=O)(CCS(C)(=O)=O)N1CC(C)C(NC(=O)CC2CCS(=O)(=O)C2)C1 N1(C(CCN(C)CC)=O)CCC(O)(CN(C(=O)CC2CC3(CC3)C2)C)C1 C=CC1(C(=O)NC(CO)CCC2CC2)CCN(C(=O)COC2CCCOC2)CC1 C1(NC(CSCCOC)=O)CCCC12CCN(C(c1cc(CCO)on1)=O)C2 OC1(C(F)F)CC(NCCCCn2cc(Br)cn2)C1 N1(C(C(COC)(F)F)=O)CC(NC(c2cc(Cl)nnc2O)=O)C(C)(C)C1 N1(C(c2c(CC)[nH]c(=N)s2)=O)CCC2(NC(c3cc4sccc4[nH]3)=O)CCCC12 CS(=O)CCC(O)C(=O)NC1CCN(c2ccc(C(C)(C)C)cc2)CC1 Cc1nc(C(c2nnnn2C)NCC(c2nccs2)C)nn1C Cc1cnc(C(=O)NC2CC(NC(C3CCCCC3N3CCCC3=O)=O)C2)cn1 c1(C(N(C2CCCN(C(C(C)OCC=C)=O)C2)C)=O)ccc(F)c(F)c1F C(=O)(C1=C(C)OCC1)N(C)CC1C2CN(C(C3N(CCC)CCC3)=O)CC21 C=CCC(F)(F)C(=O)N1CCCC(N(C)C(C2CCOC2C(C)C)=O)C1 Cc1ccc(NC(=O)CC2(NC(C3NC(=O)CC3C)=O)CC2)cc1Cl CCCCCC(CC)C(=O)NC(CC(=O)NCC(O)C(C)(C)C)C(F)(F)F c1(CC)cccc(C(N2CCCC2CN(C)C(C2CC2CC(C)C)=O)=O)c1 N1(C(c2c(C)ccnc2)=O)CCC2C(C1)CN2C(C1CCc2ncsc2C1)=O C1(C(N(C)CC2C(C)OCC2)=O)CC(=O)CN1C(=O)C(N1CCNC1=O)C c1(NC(CC2(N)CC3CCC2C3)=O)ccc2oc(C(N)=O)nc2c1 Cc1cc(CNC(=O)C(=O)NC2CCOCC2(C)C)ccc1N(C)C c1(C(CC(C)C)NC(=O)C(N2CCN(C)CC2)c2ccccc2)ccc(Cl)cc1 c1(OC)ccnc(C(N2CCC(NC(=O)CC3(O)CCCCC3)C(C)C2)=O)c1F N1(C(c2cc(C)c(F)cc2Br)C(=O)NCC2CC2)CC2CCCCC2(CO)C1 C1(CC=C)(NC(c2cc(C(C)C)n(C)n2)=O)CCCN(C(=O)C(C#N)CC)C1 C1(NC(c2ccc(C3CC3)s2)=O)CC2(C1)CN(C(=O)C=CCF)C2 C1(C2CCCN(C(=O)CC3CC3)C2)(NC(C(C)(O)CCc2ccccc2)=O)CC1 C1(CNC(C(C)CC2CC2)=O)CC2(CC2)CN1C(=O)CO.c1ccsc1Cl CCCCC(=O)C(=O)N1CCC(COC2(C(O)C(F)(F)F)CCC2)CC1 N1(C(C(C)CSc2ccccc2)=O)CCC(CNC(C2(F)CC=CC2)=O)CC1 N1(C(CSCC=C)=O)CC2(CCN(C(=O)C(=O)NC(C)C)CC2)C2COCC12 Cc1cc(OCC(N2CCN(C(c3cnc(O)s3)=O)CCC2C)=O)cc(C)c1Cl C(C(C)(O)CC(=O)NC1(C(=O)NC(C)CSC(F)F)CSC1)OC N#CC1(F)CN(C(=O)C=CCNC(c2cscn2)=O)C1 N1(C(c2cncc(C)c2)=O)CCC2CN(C(c3ccc4ccoc4c3)=O)CC2C1 c1(OCC(N2CC(N(C(=O)CC3CSCCS3)C)C2)=O)ccccc1F N1(C(C(C)CC2CC2)C(=O)NC2CCC2)CC23CCC2(COC3)C1 CCC(CC)CCCC(=O)N1CC=CC(C(=O)NCCC2(C)CCOC2)C1 c1(OC)nccc(C(=O)NC(C)CC(C)NC(c2csc(-c3cnc[nH]3)n2)=O)n1 C(C1CCCCC1)=CC(=O)N(CC(=O)NCC1COC(=O)N1)CCC c12ccc-1cc2.N1(C(=O)C(F)(F)c2cccnc2)CCCC(CF)C1 N1(C(C2CCN(C)C2=O)=O)CC(NC(=O)C(F)OC(F)(F)F)Cc2ccccc21 O=C(CN=c1[nH]c(=NC2CC(=C3CC3)C2)[nH]c2c1CCC2)NCc1ccccn1 S(=O)(=O)(c1cncc(Br)c1)NC(=O)Cc1ccc(F)cc1Br c1(C(N2CCC(N(C(=O)CSC)CCC)C2)=O)cc([N+](=O)[O-])sn1 N1(C(C23CC(CN(C(c4n(C)nnc4)=O)C2)C3)=O)CCOCC2(CCC2)C1 c1(C(=O)NCCCNC(C2C(C(C)C)OCC2)=O)ccccc1.n1(C)ccnc1 C(C(C)C(C)C(=O)NC1CCC1)OC.c1(C(=O)N)cc(C)ccc1-n1ccnc1 c1(CC)ccc(C(C2CC2)COC(=O)CC2CCC(c3n[nH]cn3)O2)cc1 Cc1ccccc1OCCCC(=O)NCC(C)N(C)C(c1c[nH]cc1C1CC1)=O Cc1cc(F)c(C(=O)NCc2c[nH]c(=N)s2)c(Br)c1 C12(C(=O)NC3C4CN(C(C5(C)N(C)CCC5)=O)C3C4)CCCC(=O)N1CCC2 c1(C(=O)NCC(CNC(c2c(Cl)c(C)n(C)n2)=O)(C)O)cnn2c1OCC(C)C2 c1(CC)cc(C)c(C(=O)NCC(CC)NC(c2ccc(C(N)=O)[nH]2)=O)o1 c1(C(=O)NC(CN(C(C2(COC)CCC2)=O)C)C)cccc(OC)c1O C1(NC(C(C)CC2CCCO2)=O)CC2CCC1N(C(c1cccc(O)n1)=O)C2 Cc1cc(C)c(C#N)c(SCC(=O)NC2CC(N3CCC3)C2)n1 CCCCN=C(NCCC1CC(C(F)(F)F)C1)NCc1nnc(C)s1 c1(C(=O)NC(C2(C)CC2)C)cn(C)c(O)n1.c1(C(=O)N)ncc(F)cn1 c1(C(=O)NC(C)C(=O)NCC(=O)NC2CC(n3ccnn3)C2)ccccc1C#N CCC(CC)(CC)C(=O)NCC(CNC(c1c(C)ccc(Cl)c1N)=O)OC n1(CCC=C)cc(C=O)nn1.c1(C(N(CCC)CCO)=O)ncc(C(F)F)s1.N C(C(C)C(C)C(=O)NCC(O)CNC(c1ncc(Cl)s1)=O)OC c1(C(N(C)CC2N(C(COC(CC)C)=O)CCOC2)=O)ccc(P(C)(C)=O)o1 C12(NC(CSCCNC(C3CC(SC)C3)=O)=O)CCC(CC1)C2(C)C C(C(=O)NCC(C)(O)CNC(c1ccc[nH]1)=O)(C(C)C)n1ncc(C)c1 N1(CCN(c2ccccc2)C(=O)C(N2CCCNCC2)=O)CC2CC(O)C(O)CC2C1 N1(C(C(C=C)C)=O)CCC(NC(C23CC=CC(C2)OC3)=O)CC1C c1(C(=O)NCC2N(C(C)(C)C)CC2)cncc(C)c1.C1(O)(C=O)CCSC1 C1(C)(NC(C(C=CCCC)O)=O)CCCN(C(c2cc(C)oc2C)=O)C1 c1(-n2cc(C3(C)CN(C(C4CC=C(C)CC4)=O)C3)nn2)cc(C)c(Cl)cc1F C1(NC(c2c(C)onc2CO)=O)CN(C(c2ncc(Cl)cc2Cl)=O)C(C)(C)C1 C1(NC(CN(C)CC)=O)CCCC(CNC(=O)C(C2CCC2)OC)C1 C1(C(N2CCCC(N(C(c3nc(C#C)sc3)=O)C)C2)=O)CN2CCN1CC2C CC(C)C(C(=O)NC1(CCNC(=O)CSCC(N)=O)CCC1)C1CCC1 c1(C(=O)NCC(C(=O)OC)CC2CCOC2)ccn2ccsc12 CCC(C)C(C)C(=O)NCC1=CCN(C(C2(c3cccc(C)c3)CC2)=O)CC1 C(Cc1ccccc1)(CS(=O)(=O)N1CCN(CC(C)(C)N)CC1)OC Cn1nnc2c1C(C(=O)N1CCCCC1CNC(c1cnc(S)[nH]1)=O)CCC2 N1(C(C2CC(C)N(C)CC2)=O)CCC(C2CCN(C(C3CSC3)=O)C2)CC1 CCCC(C(=O)NC1(CO)CN(C(=O)CN2CCCNC2=O)C1)OC c1(C(=O)NC(C)CC(C)NC(c2cc(F)cnc2Cl)=O)cc2c(s1)CCCC2 c1(C(N(CC(CNC(c2c(C)n[nH]c2)=O)O)C)=O)sc(-c2ncccn2)nc1C C(CC(C)C)(C(=O)NCCC(C)(C)NC(C1CCCOC1)=O)NC(C)=O C=CC(C)(O)CC(=O)NC1C2CN(C(c3nc(C(F)(F)F)oc3C)=O)CC12 C(=O)(C1OCCn2ccnc21)NC1CN(C(C(S(C(C)C)(=O)=O)C)=O)C1 C1(c2cn(C(c3ccccc3)C)nn2)CCCCN1C(c1ns[nH]c1=O)=O C1(OC)CC(NC(c2c(C)cnnc2O)=O)CN(C(=O)CC2CC3(CCC3)C2)C1 CC1(C)CC(NC(C2CN3CCCC3CO2)=O)CCN(C(=O)CCC2(C)CC2)C1 Cc1ccc(C(N)=O)cc1C(N1CCCCC(NC(c2c(O)noc2C)=O)C1)=O CCCC(O)(CCC)CC(=O)N(C1CCCN(C(=O)C=CCN(C)CC)C1)CC C1(C(=O)NCC(CC)NC(=O)COC)CC2CC1CC2(F)F.c1ccnn1C n1(CC(=O)NC2CCN(c3ncnc4c3CCO4)CC2F)ccc2ccccc12 N1(C(C2(C)CCOC2)=O)C2CCC1CC(NC(=O)CCc1ccc(CO)cc1)C2 C1(NC(C=C(C)C(F)F)=O)COC2(CCN(C(=O)CC3(O)CCCC3)C2)C1 C12(NC(c3cc([N+](=O)[O-])c[nH]3)=O)CCCN(C(=O)C(F)=CC3CC3)CC1C2 N1(C(CC2CC(=O)C2)=O)CCC2(NC(c3ccc(F)c(Cl)c3)=O)CCCCC12 N1(C(C(CC)OCC)=O)CC(C2CN(C(c3cc(N)c(O)c(F)c3)=O)C2)C1 c1(C=O)ccc(C2COC2)cc1.c1(OCC)cc(C(=O)NC2CCC2)[nH]n1.C C(C(CC1CCCC1)C(=O)NCCCS(N)(=O)=O)NC(C(CO)OC)=O C1(C(N2C(C(N3C(C(C)C)CC3)=O)CC(O)C2)=O)CC2COCC2C1 O=C(C1=NOC(c2ccc(F)cc2)C1)NC1CC1NC(c1nnc(O)cc1O)=O C=CC1(O)CN(C(c2cc(CNC(C3(SC)CC3)=O)no2)=O)C1 N1(C(c2ccc(CC)o2)=O)CC(CC=O)C2(CC2)C1.C(C)CCN(C)CCC.N C(CC(O)CCc1ccccc1)NC(c1n(CCOC)nnn1)C1C2COCC12 c1(OC)ccc2cc(C(=O)NC3CCCCC3NC(C3CCCCS3)=O)sc2c1 N1(CCCCN2CCOC3(C2)CCSC3)CCC(C2CCCCC2)CC1 N1(C(C2CC(=O)NCC2)=O)CC2CN(C(=O)CNC(=O)NC3CC3)CC2C1 CCC(C)C(C(=O)NC(C1CN(C(=O)CN(C2CCCC2O)C)C1)C)OC CCC(C)C(O)C(C)C(=O)N1CC(F)(F)CC1C(=O)NC1CON(CC)C1=O CCCCCC(C)CC(=O)NC1CCCCC1CNC(=O)Cc1cnnn1C C1(C(N(C)CC2C3CN(C(CSCC)=O)CC32)=O)CC2(CC(OC)C2)C1 Cc1occc1CC(=O)NC1CC(CCNC(=O)CC2CCC2C)C1 Cc1cc(C(=O)NC(C)CCNC(=O)C(C2CCOCC2)C)cc(Cl)n1 C1(NC(CN2CC(CC)C2)=O)CCCC(CNC(C2CC(C)(F)C2)=O)C1 C1(CC(N2CC(N(C(=O)CCSCC(N)=O)C)C2)=O)(COC)CCCC1 c1(NC(=O)Nc2c(C)nc(CC)s2)cc(C(F)(F)F)cc2c1OCC(=O)N2 c1(CC)nc(C(C)C)ccc1C(=O)NCC1CN(C(C2CCCN2C)=O)C1 C1(CC(=O)NCC)(OC)CN(C(=O)Cc2ccon2)C1.C(=O)C(F)(F)F Cc1nc(C(=O)N(CCCCCCNC(C2CC(C)(C)O2)=O)C)cn1C c1(N2CCC(n3ncc(NC(c4ccccn4)=O)c3)CC2)ncnc(Cl)c1F Cc1c(Br)ccc(C(=O)NC2CN(C(C3(C)CCCN3)=O)CC2C)c1C Cc1cn2c(n1)CC(C(N1CCCC1CNC(C1CCC(C)(C)CC1)=O)=O)CC2 C(CC(CC)C(=O)NCCC(C)CCNC(c1cccc(=O)o1)=O)=CC N1(CC=O)CCCNC1=O.Cc1csc(C(F)(F)C(=O)NCC2CCCC2)n1.N C1(O)(CNC(=O)CCC(=O)c2cccs2)CCN(C(=O)COC2CCOC2)CC1 C1(C(=O)NCC2(NC(C(C)OCCC#C)=O)CCCC2)CCc2nccn2C1 CC(CC(C)(C)C)C(=O)NC1CC2(NC(c3cn4cccnc4n3)=O)COC1C2 N1(C(C2C(C)OC(C)C2)=O)CCC2CN(C(C3(C#N)CCCOC3)=O)CC2CC1 c12cc(cc(OC)n1)c(=O)[nH]c1cc(ncn1)[nH]2.n1(CC)cnccc1=O C1(C=O)CC2(C1)CC1(CCC1)C2.CC(CS(C)=O)C(=O)NCC1(F)CCC1 CCC(CCC(=O)Nc1ccc(C)c(Cl)c1)NC(C1(C#N)CCOC1)=O Cc1nc(O)nc(C)c1C(=O)NC1CC1NC(c1nnn(C)n1)=O c1(C(=O)NCCN(C)C(c2cc(-c3cccnc3)[nH]n2)=O)cccc2c1OCC2 c1(C(N2CCOCC(NC(CC(CCC)C)=O)C2)=O)cnc2c(Cl)cccn12 C1(C(=O)NC(CN(C(Cc2c(C)non2)=O)C)C)CC12CCSCC2 c1(-c2cn(C3CC(N(C(=O)C(C)C4CCOC4)C(C)=O)C3)nn2)cccc(N)n1 c1(OC)ccc(CN(C(=O)C(=O)Nc2c[nH]nc2C(C)C)C2CC2)cc1 C(=O)(C(C)C(CC)CC)N1CCCCC(N(C(c2cnc(CC)nc2O)=O)C)C1 CC1c2ccccc2NC(=O)CN1C(=O)CCc1ccc(Cl)c(F)c1 C1(F)(CNC(c2c(CC)cno2)=O)CCCN(C(C2CCC(F)(F)C2)=O)C1 c1(C(C(=O)NCC(CC(C)C)NC(C2CC3CC3C2)=O)O)ccc(F)c(Cl)c1 CC(C)(C)C(=O)C(=O)NCCC1CN(C(c2cc(-c3ccco3)c[nH]2)=O)CCO1 c1(CC2N(CC(CC)=O)CC2C(C)C)cccc2c1OCCCO2 c1(OC)ccccc1C(N)CNCC(c1nc(-c2ccccc2)no1)C c1(-n2cnc(C(=O)O)n2)cccc2c1CCCC2 C(=O)(CC(O)C(C)C)NC(CC)CNC(c1cccnc1C(C)=O)=O C#CC1(O)CC(C(=O)N(C2CCN(C(C3(F)CCOC3)=O)C2)C)C1 C1(NC(C)C(C)(C)c2ccccc2)CCN(c2nnnn2C)CC1 CN(C(=NCC1CCOC1)NCC(C)(C)C(C)(C)O)Cc1nc2c(s1)CCC2 N1(C(C(C2CCN(C3COC3)CC2)C)=O)CCN(C(C2CC3(CCC3)C2)=O)CC1 C(CCNC(=O)CCCn1ccccc1=O)(C(C)C)NC(CCOC(C)=O)=O C(C(=O)NCC(C)N(C(=O)CC1CCCO1)C)(C1CCC1)OCC CC(C)C(CO)CCNC(=O)CC1(C)CC1.C12(C=O)CCC(C1)C2(C)C.N C12(C(N(C3CCN(C(CCCc4onc(C)n4)=O)C3)C)=O)C3C4C1C1C2C3C41C C(CCS(C)=O)N(CC(C)NCC(F)(F)F)C(=O)OC(C)(C)C c1(CCC(=O)NC2CCN(C(=O)Cn3cccc3)CC2)ccc(Cl)nc1 C(=O)(C1Cc2ccccc21)NC1(C(N(C)CCN(C)C2CC2)=O)CCN(C)C1 C1(C(C(=O)OCC)F)CC2CCC(C1)N2C(=O)C(Cc1ccccc1C)CC c1(C(=O)NC(CNC(C(COCC)C)=O)C(C)C)c(N)sc(C)c1C n1(CC)ncc2cc(C(=O)NCC(O)CNC(C3CC(F)C3)=O)c(C)nc12 c1(OC(C)(C)C)ccc2c(Nc3cccc(-c4ccccc4F)c3)ncnc2c1 N1(C(CCCCC)=O)CCC2(CNC(=O)CCc3cc(C)sc3C)CCCCC12 CCCC(C(=O)NCCCOC(F)(F)F)NC(=O)C(C1CCCCC1)=O n1(CCC)ncc(C(=O)NC2(CO)CN(C(c3c(C)noc3C)=O)C2)c1Cl c1(CC(=O)NC2CC2NC(C2CCOCC2)=O)coc2cc(O)ccc12 CC1(C)C(NC(c2csc(-c3ccsc3)n2)=O)CC1CNC(C1CCC1)=O C1(C(C)C)CC(n2cc(C(C3CC3)N(CC(C)(C)C)C)nn2)C(=O)N1 O=S(=O)(c1ccn(C2CC2(F)F)n1)N1CCNCC1c1ccc(Br)cc1 CC1CCCCC1(C)C(=O)NC1CC2(C1)CC(CNC(c1nccnc1N)=O)C2 Cc1cc2cccnc2nc1C(=O)NCC(C)CN(C(=O)CC1CCC(=O)O1)C C1(C(N2CCN(C(c3ccc(NC)cc3Cl)=O)CC2)=O)CCC2(CC1)CC2(F)F C12(CC(=O)NC3(CC=C)CC(C)(C)C3)CCC1CN(C(=O)C(C#N)CC)C2 n1(CC(=O)NC2CCC(NC(CCC(C)OC)=O)CC2)ccc2ccccc12 C1(CNC(c2cncc(CO)c2)=O)CCC(C(=O)NCC2CCCO2)CC1 N1(C(C(COC)CC(C)C)=O)CC2(CCN(C(=O)C=Cc3cc[nH]c3)CC2)C1 N1(C(c2cc(C#C)cc(F)c2)=O)CCCC12CCN(C(C1CC1F)=O)C2 C1(NC(CC2C(OCC)COCC2)=O)CCN(CCOC)CC1O C(=O)(C1CCCc2ncnn21)NC1C(NC(COCCN(C)C)=O)CCC1 N1(C(C2(C(C)C)CCC2)=O)CC2CC(C(N3CCC34CCSCC4)=O)C(C2)C1 C1(c2cn(C3C(Cc4n[nH]c(C)c4C(N)=O)CCCC3)nn2)CC2CCC1CC2 C(C)(C(=O)N1CC(CC(C)NC(c2snnc2C)=O)C1)(C1(C)CC1)OC N1(C(C(C)(C2CC2)OC)=O)CCC2(CCN(C(=O)CCC(=O)c3cccs3)C2)C1 C(=O)(C(CNC(=O)C(n1ccc(C)n1)C)N(C)C)NC1CN(CC)C1 C1(C(N2CCCC2)=O)CCC(=O)N1C1CC1.CC(C)CCOCC(=O)NC c1(CN(C)C(=O)N)ccc(F)c(F)c1.C1CC(C=O)C1(C)C.C(C)(C)C C1(C(=O)NCC(CC=C)NC(C2CCCN(C(N)=O)C2)=O)CCCCC1O Cc1nn[nH]c1C(=O)N(C(C(=O)NCC(F)(F)F)C1CC1)C C=CCCC(C)(C)C(=O)NCC1(O)CCCN(C(C2COC3COCC3O2)=O)C1 c1(C(=O)NC2(COC)CN(C(C3CCSCC3)=O)C2)ccc2c(n1)CCC2 C#Cc1cccc(C(=O)N(C2CN(C(C3(C)CC=CCC3)=O)CCC2C)C)c1F c1(C(CN(C(C2C(C)OCCO2)=O)C2CC2)=O)ccc2c(c1)OCCO2 N#Cc1cc(C(=O)NCC2CN(C(C3CC4CCC3O4)=O)CCO2)ccc1Br C(=O)(CC1=NNC(=O)C1)NC(C1(O)CCN(C(C(CCC)N(C)C)=O)C1)C C1(NC(C2CC(CC)C2)=O)CCN(C(=O)Cc2cc(C)sc2C)C1(C)C C1(CN2CCC(c3nc(C)on3)C2)CN(S(C)(=O)=O)CCO1 C(=O)(C(C)(O)COC)NCC#CCNC(c1cnc(COC)s1)=O c1(C(=O)NC(CC(CC)=O)C(=O)O)cc(C2CC2)nc2onc(C)c12 CCC(COC)C(=O)NCc1cccc(C(=O)NC(CC)C(C)(F)F)n1 C1(CC=O)CCCC2(CC2)C1.CCS(=O)CC(=O)NCC1CC(F)(F)C1.C C#CCCC(C(=O)Nc1cnc(F)nc1)NC(=O)C1=C(C)CC1 Cc1ccc(NC(=O)N)cc1.C1CC(O)CCN1C(c1cc(C(C)(C)C)n[nH]1)=O C(=O)(C(O)CC(F)(F)F)N1CCC(CCCNC(c2c(C)n[nH]c2C)=O)CC1 N1(C(CC(c2ccncc2)C2CCC2)=O)CCC(F)(F)C(O)C1.CC(C)(C)OC=O C(C(CC(C)C)C(=O)NCC(C)NC(C1CN(C(N)=O)C1)=O)OC C1(CNC(C(CCC)C)=O)CCCCN(C(=O)CCCCN2CCCCC2)C1 C(=O)(C(C)(C)CC(F)(F)F)NCC1N(C(CN2C(C)CCC2)=O)C2C(C1)CCC2 C1(C(=O)NOCCCCC2CC2)C=CCN(C(C2CC3(CC3)CO2)=O)C1 C(c1ccc[nH]1)=CC(=O)NC1(C(N2CCC2CF)=O)CSC1 C(=O)(C1=C(Cl)CCCC1)N(CC(=O)NC1CN2CCC1C2)CCC C1(NC(c2ccc(CC)s2)=O)CCC12CN(C(=O)C(C)(O)c1ccccc1)C2 c1(C(=O)NC2(C3N(C(CSc4nc(C)[nH]n4)=O)CCC3)CC2)cccc(CF)c1 c1(C(=O)NC(CNC(c2cc(Cl)cs2)=O)C2CC2)ncc[nH]c1=O Cn1nnc(CNC(=O)CCC2CCOC2)c1C1CC1.C(C)(C)C.C=O.N O=C(CS(=O)(=O)CCO)NCCCC1CCCCN1C(=O)C(C1CCCCC1)F CCC(CN(C)C)CC(=O)NCC1(NC(=O)C(C)=CC2CC2)CCOC1 CC1(C(N2CCC(NC(=O)C(=Cc3cccnc3)F)C2)=O)CC2(CCC2)C1 N1(C(CCNC(=O)OC)=O)CCOCC1CC(=O)Nc1cccc(OCF)c1 C1(OC(F)(F)F)CCN(C(=NCCN2CC3CC3C2)NCC2CCC2)CC1 C1(C(N2CCCC(C(C)(C)O)C2)=O)CN(C(=O)C(F)F)CC1C1CC1 c1(NC(CCC=C)C)nc(=NCC2CCCN2C2CC2)[nH]c2c(C)nn(C)c12 C1(N(C(C2CN(C(C)=O)C2)=O)C)CCCN(C(C23CC(C)(C2)C3)=O)C1 C=CCC(C)(CC)C(=O)N(CC(C)C(N1CCC2(CC(CO)C2)C1)=O)C c1(CC(N2C(CNC(C3CCC4(CC3)CC4)=O)CCC2)=O)c[nH]c2cccnc12 C(c1ccccc1)=CCC(=O)NCC(CNC(CCc1n(C)cnn1)=O)CO C1(C(=O)NCC2N(C)CCN(C(c3nc(C)sc3C)=O)C2)CCn2ncnc2C1 Cc1sc(S(N)(=O)=O)cc1C(=O)N.C1C(C)CCN1C(=O)C(F)=C1CCC1 N1(C(C2N(C(C)=O)CCC2)=O)CCC(NC(=O)CC(c2c(C)n[nH]c2C)C)C1C Cc1cccc(C(N2CCC(C(=O)NCc3ccoc3C)(CO)C2)=O)c1F c1(CNC(CC)(CNC(=O)Cc2ccc(Cl)nc2C)CC)nccc2ccsc12 c1(CNC(C2COCCO2)C)nc(-c2ccccc2C)nn1Cc1ccccc1 C1(NC(CCC(=C)Cl)=O)CCCCCCC1NC(C1NC(=O)OC1C)=O N1(c2nccc(C(=O)NC3CC3)n2)CC(c2cc[nH]n2)C2(CCC2)C1 C(=O)(C(C)(CSC)NC(C1CCN(C)CC1)=O)NCC(CSC)(C)O C1(CC(N2C(CCCNC(C3CSCCS3)=O)CCC2)=O)CC2(COC2)C1 c1(C(=O)NCC(F)C2CCC2)cncc(CNC(=O)C(O)C2CCC2)c1 C12(COC)CC(CN1C(c1ccn(C)c1)=O)C2.c1(CC=O)ccnc(C)c1 CN1CCC2CN(C(c3nc(Cl)cs3)C(=O)Nc3ccccc3)CC2C1 N1(C(CC(CC)OC)=O)CC2(CC2)CC1CNC(=O)CC(O)C1CC1 c1(NC(C)CNC(c2c[nH]cc2Br)=O)ncccc1[N+](=O)[O-] N1(C(C2(C(=O)NC)CCC2)=O)CC2CC1C2NC(c1cnc(C)cn1)=O c1(C(N2CC(CNC(C(C=C=C)C)=O)C3(C2)CCC3)=O)ccc2oc(C)nc2c1 c1(C(N2CC(CC)C2)=O)cc2cccc(F)c2o1.c1(C=O)ncc(C(N)=O)s1.N c1(C(N2CCCC(NC(CSCCCC)=O)C2)=O)cc2ccc(CC)cc2[nH]1 N1(C(C2C(C)(C)C2)=O)CCOCCC1C(=O)NCc1cnns1 C1(C)(NC(C2C(C(C)C)C2)=O)CCN(C(c2cc(C(F)(F)F)ncn2)=O)C1 c1(C(N2CCC(CNC(C3CC3(F)F)=O)C23CC3)=O)ccc2[nH]ccc2c1 C(=O)(C#CC1CCC1)N1CC(C(C(N2CC(F)(C#N)C2)=O)OC)C1 C(=O)(CC1=CCN(Cc2ccc(N3CCCC3)nc2)CC1)NC1CCN(C)C1=O C1(CC)CN(Cc2ccn(C)n2)CCN1C(=O)NC(c1ccccc1)C C(=O)(C(C)C#N)N(CC(=O)N(C1CC1C)C)CCC c1(C(n2cc(C(CC)(O)CC)nn2)CCc2ccccc2)ccc(F)c(F)c1 N1(C(CCc2ccc(C)nc2)=O)CC2(CCN2C(c2n[nH]c3c2COC3)=O)C1 C(=O)(CC1OCc2ncccc21)N1CCOC2CN(C(CCCC)=O)CC21 Cc1c(CCNC(C2COC(=O)N2C)=O)ccc(F)c1F CC(C)CC(C)CC(=O)NCc1ccc(-n2ccnc2)nc1 c1(C(=O)N)cc(F)cc(Cl)c1.c1(N2C(C3CC3)CCC2)ccnc(C(F)(F)F)n1 C1(c2n(C(C)C)nnn2)(NCC2(C)CCCCCCC2)CC2CCC(C2)C1 c1(C(N(CC(C)NC(=O)CCOC(C)C)CC)=O)cc2cc(F)ccc2o1 c1(C(=O)NCCC(C)NC(c2sncc2Br)=O)c[nH]cc1Br C=CC1(c2cn(-c3cc(C)nn3C)nn2)COCCN1C(=O)C(C)(O)COC C(=O)(C(C)CCCC(C)=O)NC1CC2CC(NC(CCC(C)OCC)=O)C1C2 N1(C(CCCCSC)=O)CC(NC(c2cc([N+](=O)[O-])c[nH]2)=O)C2(CCOCC2)C1 N1(C(COCC)=O)CCN(C(c2cc(SC)c(C)o2)=O)C(C)C1C C=CC1(C(N2CC(CCC)C2)=O)CCN(C(C)=O)C1 C1(OC)CN(C(=O)C(F)(F)c2cncs2)CC1NC(=O)C(F)OC(F)(F)F N1(C(c2c(N)cccn2)=O)CCC2(CCN(C(C3OC4CCC3CC4)=O)C2)C1 C(=O)(C1=CNS(=O)(=O)N=C1C)N1CCC2(CC2)CC1.C(C)(C(=O)N)NC(C)=O C1(C(=O)NC(C2(O)CCC2)C)C(C)C1(C)C.C(=O)(CCC1OCCO1)N C1(C(N2CCC(N(C(c3ccc(C4CC4)o3)=O)CC)C2)=O)CCCC(C)(C)C1 CC(C(=O)N(C(c1ccccc1)CNC(=O)CCCN1CCOC1=O)C)C(F)F N1(C(C(CCC)C)=O)CC2(NC(=O)CCSCc3ccccn3)CC1(C)C2.O N1(C(C(C)OCCC(C)C)=O)CCC(c2nccn2C)C1.C1(O)(C(=O)N)CCC1 Cc1cc(C(N2CCC(C(N3CC(F)(CO)C3)=O)C(C)(C)C2)=O)ccc1C#N c1(C2(NC(CC3C(CNC(CSCC#C)=O)C3)=O)CC2)cccs1 c1(C(=O)NCC2(C)CCCN(C(C(CCCC)O)=O)C2)c(N)ccc(F)c1F c1(CNCC(CCC)CC)cnc2c(c1)c(C)nn2C CC1CC(=O)NCC1C(=O)NCCn1cc(C(=O)N)cn1.C1CC1(F)F.C C12(NC(CC=C=C)=O)CCN(C(=O)CCC(=O)c3cccc(F)c3)CCC1C2 N1(C(c2n(C(C)C)ncc2)=O)CC(C(F)(F)F)OCC1CO N1(C(C(F)=CCC)=O)CCC2(C1)CN(C(=O)CCCc1ncc(Br)cn1)C2 c1(OC)cc(C(=O)Nc2ncoc2-c2ccccc2-c2nn[nH]n2)ccc1O c1(C(N(CCCN(C)C(C2OC3CCC2C3)=O)C)=O)ccc2c[nH]nc2c1 c1(CC)cc(=NC(=O)c2cnn(CCNC(=O)C=Cc3ccncn3)c2)[nH]n1C C12(C(=O)NC3CCN(C(C4(CC#C)CCOC4)=O)C3)CCC(C)(CC1)OC2.O Cc1cc(C(=O)NCC2C3CC2N(C(C2CC(C(C)C)C2)=O)C3)nc(C)c1 C1(NC(C(=O)NCC)=O)CC2(C1)CN(C(C1(OC)CCSCC1)=O)C2 c1(C2CC2)cc(Cl)ccc1[N+](=O)[O-].N12CC3CC3(C1)C(=O)N(C1CC1)C2=O N1(C(C(C)CC(F)F)=O)C(CNC(c2nc[nH]c3nccc2-3)=O)CC2CCCC12 c1(C(N(CCN(C(c2ccc(CC)o2)=O)C)C(C)C)=O)ccc(CO)cn1 N1(C(C2N(CC)CCCC2)=O)CCOCC(NC(=O)CSC2CC2)C1 c1(N(C)C)ccc(C=CC(=O)NCC2C(O)C(O)CN2C(=O)CO)cc1 C1(C(N(CCCCNC(C2C(C)OCC2)=O)C)=O)CCC2(CCC2)CC1 C(=O)(CC(C(F)F)NC(C12CCC(O)C1C2)=O)NC(CC(=O)NCC)C Cc1ccn2ncc(C(=O)NCC(O)CCNC(=O)C(C)(C)C(O)C(C)C)c2c1 C12(C(=O)O)CCCC1N(C(C1C3Cc4ccccc4C13)=O)CCC2 c1(C(N2CC(NC(COC(C)=O)=O)C(CO)CC2)=O)ccc2sccc2c1 CC1CCC(C)(C(=O)N(C)CC2CCCN2C(C2(O)CC2)=O)C1 c1(CNC2C(C(=O)NCc3c(OC)nccc3)C2)cc2cc(C)ccc2[nH]1 C1(C(C)=O)CC(C(=O)N2CCCCC(OC)C2)=NN1c1ccccc1.C(C)(C)(C)O C1(C)CCCC1.C1(CC=O)CC(C)(C)C1.C(C=CC(=O)N)(CC)=CC C12(NC(c3c(C)nc(CCC)s3)=O)CCCN(C(c3ccccc3F)=O)C1C2 c1(C2(OC)CCC2)cccc(NC)c1.C12CC1CN2 C(=O)(C(F)(F)C(F)(F)F)N1CC2C(NC(COc3ccc(C#N)cc3)=O)C(C2)C1 CCCC(CC)CC(=O)NCC1CCN1C(c1cn(C2CCC2)nn1)=O Cc1ccc2sc(C(=O)NC3CC3NC(c3cc(C)n(C)c3)=O)cc2c1 C1(CNC(c2ccccc2-c2cnc[nH]2)=O)CCCC2(CCC2)O1 C1(C(=O)NC2CN(C(c3c(OC)c(C)sc3)=O)CC2O)CC2(CCC2)CO1 c1(C(=O)N)cnc2n1CCCCC2.N1(C(C(=O)NCC(C)C)C)CC2C(C)C2C1 c1(NC)ccc(F)cc1CN1CCCC(C)(C(N2CCC(C(=O)O)C2)=O)C1 c1(C(=O)NCC2OCCN(C(c3csc(COC)n3)=O)C2)nc(C)ncc1Br C1(NC(c2c(C)scc2)=O)C2CC1CN(C(C1(F)CCOC1C)=O)C2 c1(CCC)onc(C)c1C(=O)NCCC1(C)CC1.C1(C=O)CCCC(C)O1 c1(C(N2CCCC(NC(C(C)OCC#C)=O)C2C)=O)cc2c(nc1O)CCOC2 C1(C)(CC)CC(NC(c2ncccc2C)=O)CN1C(=O)Cc1ccsc1C.S c1(C(N2C(C)CC(NC(c3ccoc3)=O)CC2)=O)cc2c(F)cccc2s1 N1(C(C(C)(CO)OC)=O)CCCC(C)(C)C1.c1(CC(=O)N)cc(C)cc(F)c1 C(=O)(C(C)(O)CC(F)(F)F)N1CC(C)N(C(c2cscc2F)=O)CC1 CC1CCCN(C(=O)CCC2CC(F)(F)C2)C1CNC(c1cnco1)=O CCCC(C)(C)CC(=O)N1CC(C)(CNC(c2sccc2OC)=O)CC1(C)C c1(C=O)c2c(nn1C)CCCC2.C(C)(C(=O)N(CC)C(C)C)N(C(C)=O)C.N CC(O)C(C)CN=c1nc2scnc2c(NCC2(C)CS(=O)(=O)C2)[nH]1 Cc1nn(C)cc1C(O)C(=O)N1CCC1CNC(c1nnsc1C)=O Cc1sc2ncc(C(=O)N(CC(O)CN(C)C(C3CC34CC(O)C4)=O)C)n2c1C C1(C=O)CCOC(=O)CC1.C1(C(C)(C)C)(C)CCN(C(=O)CSC(=N)N)C1.N CC(O)(CNC(C1(NC(C2CS(=O)(=O)C2)=O)CCC1)=O)CCO c1(C(=O)NC(CC)C)coc(C(C)NC(c2nnsc2C)=O)n1 C1(C)(C(=O)NCCCCC2CCN(C(CC(=C)C)=O)CC2)CCCC1(F)F N1(C(C2(C)CC2)=O)CCOC(Cc2cn(CC3CCC3)nn2)C1 N1(C(c2ccc(C(=O)OC)s2)=O)CC(NC(c2ccncc2Cl)=O)C(F)C1 Cc1ccc(C)c(C(=O)NC(c2ccncc2-c2ccc(C3CCC3)cc2)C)c1 Cc1cc(Cl)ncc1CC(=O)NCC(O)CN(C)C(C1(F)CC=CCC1)=O N1(C(C(=COCC)C#N)=O)CCC(C)C(F)(F)CC1.C1(C(=O)N)CNC(=O)N1C c1(CN(c2cc(OCC)ncn2)C2CC2)ccc2n[nH]cc2c1.C1CCC(N)CC1 C#CCCCC(C)C(=O)NC1(CCC(N2CCCCN(C)CC2)=O)CCC1 C(=O)(NNC(=O)C1CCCC1N)C1C(N)COC1 CCC(C)C(C)CNC(C1CC(NC(C2CC(=O)CCO2)=O)C1(C)C)=O C(C)(C)(CC(F)C(=O)NCC1CN2CCC1CC2)NC(Cn1c(C)cc(C)n1)=O N(S(=O)(=O)N1CCCC(CC(=O)O)C1)CC(C)Cc1cn[nH]c1 N1(C(CC(C)C(F)F)=O)CCCC(O)(CNC(c2c[nH]c(C(N)=O)c2)=O)CC1 C(=O)(CC(O)CNC(c1ccnnc1)=O)N1CC(CS(C)=O)C1 N1(C(C2(c3ccccc3)CC2)=O)CCCC(N2CCCC2)CC1.N1CC2CC2C1 N1(C(=O)CC(c2ccccc2)Sc2cncc(O)c2)CCCCC1C1CCC1 c1(C(=O)NC23CCN(C(c4ccc(CC)cn4)=O)CC2C3)cc(C)c(C)cc1Cl Cc1cc(C)c(CC(N2CCCC2C(C)(C)CNC(c2cnco2)=O)=O)s1 Cc1n[nH]cc1CC(=O)N(CC(O)CN(C)C(C1CC(Cl)(Cl)C1)=O)C N1(C(C2(C(N)=O)CCC2)=O)CCCC(CCCCNC(c2ccc[n+]([O-])c2)=O)C1 c1(C(=O)NCC2(C)CCC(NC(=O)C(N)=O)C2)[nH]nc2ncnc(O)c12 C1(NC(C(C)CCc2ccccc2F)=O)CC2CCC1N(C(c1ccoc1)=O)C2 C1(CC(C)NC(C(C)N(C(C)=O)C)=O)CCN(C(=O)OC(C)(C)C)CC1 N1(C(CC(n2ccc(C)n2)C)=O)CC2CC(NC(C3CC4CC4C3)=O)CC1C2 N1(C(CCC=CC)=O)CC=C(CCNC(C2CCC2n2cccn2)=O)CC1 c1(C(N2C(CNC(C3C(C)(C)OCC3)=O)CCC2)=O)cc(S(C)(=O)=O)co1 c1(C(N2C(C)(CC(N3CCC(C)(N(C)C)C3)=O)CC2)=O)cccc(F)c1F C1(C(=O)OC)CCC(C2CCCCC2)CN1C(=O)CN(c1ccnc(Cl)n1)C C=CCC(CC=C)C(=O)NC1CC(F)CN(C(c2ccc(C(F)F)cc2Cl)=O)C1 CC#CCC(C(=O)Nc1cnn(CCC)c1)NC(c1cncn1C)=O c1(C(=O)NCC2CC2C(=O)NCCC2CCC2)ccn2ccnc2c1 c1(C(C(=O)NC(CC)C)N(C(C)(C)C(=O)NC)C)ccc2c(c1)CCC2 Cc1cc([N+](=O)[O-])ncc1C(=O)NCC1CCN1C(c1sccc1C)=O c1(CC)conc1C(=O)NC1CCC1NC(=O)C(O)c1ccsc1 C12(CNC(C3(C)CCOCC3)=O)CCC1CCN2C(=O)C(c1ccc(Cl)cc1)=O Cc1nc(CCC(=O)NC2CC(NC(=O)CC3CCC(=O)NC3)C2)oc1C CCC(CC)CC(F)C(=O)NCc1c[nH]nc1C(=O)NCC(C)(C)O.C(C)C N1(C(CCC2CCC(C)O2)=O)CCCC(CNC(=O)CCOC2CCOCC2)C1 C1(C(N2CCC(CCC(=O)NCC(CC)N3CCCC3)C2)=O)CC2(CC2)CO1 c1(C(N2C(CNC(c3c(Cl)sc(C)c3C)=O)CCC2)=O)cccn2c(C)cnc12 c1(C(=O)O)cc(S(=O)(=O)NCC(CN2CCCC2)C2CC2)ccc1Br c1(C(N2CC(CC=C)(C(N3CC(C(C)CC)C3)=O)C2)=O)cc[nH]c(=NC)c1 c1(OC)ccc(C(C)(C)C=O)cc1.C(C)C(C)(C)C.C1(C=O)CC1C(C)O c1(C=O)ccc(N(C)C)nc1.c1(COCC)nc(C=O)cs1.CCC(C)C.N N1(CCC(=O)N2CC(n3cc(C4CC4)nn3)CO2)C(=O)c2ccccc2C1=O c1(C(N2C(CNC(C=C(C)C(=O)O)=O)COCC2)=O)cc(C)ccc1I C1(CNC(C=CCC)=O)CN(C(=O)CCNC(=O)CC(C)C)CCO1 C1(CNC(C2CSCCS2)=O)CCC2(CN(C(c3cccs3)=O)C2)O1 c1(C(N(C)CCOCCCNC(=O)CCC2CCCCO2)=O)nccnc1N C1(C(N(CC(=O)N(CC(C)OC)C)CCC)=O)CCCS1 c1(C(=O)NCCC(C)(C)NC(c2cn(C)nn2)=O)ccc[n+]([O-])c1 C=CCCCCCCC(=O)NC(CCOCC)C(=O)NC(CN(C)C)CC C1(NC(C(C)(C)c2cscn2)=O)CC(C2CCN(C(=O)Cc3ccsc3)C2)C1 C1(C(=O)N)CCCC2(CC2)C1.C(=O)(CCc1ccccc1)NC(c1cccs1)C c1(OC)cccc(CCC(=O)N(C2CCC(NC(C3CCC3CF)=O)CC2)C)n1 C1(CN(C(c2cn(CCCF)nn2)=O)CC)CCN(C(c2ccoc2C)=O)CC1 c1(C(N2CCC(F)(C(=O)Nc3cc(C(N)=O)ncc3)C2)=O)c(F)cc(Cl)cc1F C12(COCCO1)CC(=O)NC2.c1(CC(=O)O)n[nH]cc1C(=O)O N1(C(CCCC)=O)CC2(NC(C3Cc4nncn4C3)=O)CCC1CC2 N1(C(c2cc(Br)ccc2F)C(=O)NCC(=C)C)CCn2c(CN(C)C)nnc2C1 CCCCS(=O)(=O)CC(=O)N(CC(C)NC(c1cnc(OCC(F)F)cn1)=O)C C(=O)(C1CSc2ccccc21)NC(C1N(C(C2CCN(C)CC2)=O)CCC1)(C)C N1(C(C23CCC(OC)C2C3)=O)CC2CCC2(CC(=O)NCC2=CCCCC2)C1 c1(CNC2(c3nnnn3C3COC3)CC(C)OC2)ccc2ccn(C)c2c1 CC(O)C(C)(C)C(=O)NCCC(C)N(C(=O)CCOC1CC1)C C(=O)(C1=C2CCN=C2NC=C1)N1C(CCNC(c2c(C)ccnn2)=O)CCCC1 C(CCC(=O)NNC(=O)C(N)=O)N1CCC(S(=O)(=O)N(C)C)C1 C1(CCCNC(C=C(CCC)C)=O)CCN(CC2CCCN2C(=O)CC)CC1 c1(CN2CCN(C3CCN(C(=O)CC(F)F)CC3)CC2)cc(Cl)ncc1Br CCCCC(C)(F)C(=O)N1CC(OC)C(NC(C2(C)CSC2)=O)C1 c1(C(=O)NCCC2CN(C(c3n(C(C)C)ncc3)=O)C2)ccnc2ccncc12 C(=O)(C1=NN(C)C(=O)CC1)N1CCCCC1C1CC1.C(CC=O)NC(=O)NC c1(NC(C(=O)NC)Cc2ccccc2)ncc2c(Br)cccc2n1 c1(C(=O)OC)cnc(SC2CCC(C(N)=O)O2)[nH]1.C12CCCN1C(=O)CC2 C1(C(=O)NC)(COC)CCCCO1.C1CCCCC1.c1(CC=O)csc(C)n1 N1(C(c2c(C)cc(F)cc2)=O)CCC2(CNC(c3cscc3Cl)=O)CCCCC12 N1(C(CC)=O)CCC(NC(=O)CCC2CCCN(C(=O)C(C#N)N)C2)CC1 c1(C(N(CC(CNC(CCCC#C)=O)C)C)=O)cc([N+](=O)[O-])ccc1C(F)(F)F c1(OC)cc(OC)c(F)c(C(N2CCC(C(N3CCC(Br)CC3)=O)C2)=O)c1 N1(C(CC(CC)CN(C)C)=O)CCC2CC1CN(C(c1cc(C)on1)=O)C2 Cc1ccc(CCC(=O)NC2CCC(NC(=O)C(C)n3cncn3)C2)o1 c1(CC)oc(C(=O)NC(C)CN(C(=O)CCC2CCCCN2C)CC)cc1C c1(OC)cc(C(=O)N(c2ccc(F)cc2)CCC(C)(C)O)cnc1Br C1(C(=O)NC2CCCN(C(C3(C)CC(F)(F)C3)=O)C2)CCCCC1(F)F c1(C(=O)NC(CC)CNC(c2cc(Br)sn2)=O)cc(OC)nn1C c1(C(N2CC(O)(C(CNC(c3cn(C)nc3)=O)(C)C)C2)=O)cc2cscc2s1 c1(SCC(=O)N(C2CCCC(NC(=O)CO)C2)C)ccc([N+](=O)[O-])cc1 c1(C(N2CCN(C(C(C)OC)=O)C(C)CC2)=O)cc2c(Br)cc(C)cc2[nH]1 C1CCCC2(CN(C(c3ccnn3C(F)F)=O)C2)O1.C1(CC(=O)N)(OC)CC1 Cc1c(F)ccc(CN2CC3CC(NC(=O)Nc4ccc(Cl)cc4)CC3C2)c1F Cc1ccc(CC2CCCO2)cc1.C(=O)(C(O)C1CN(C(=O)CC2CCC2)C1)N c1(C(=O)NC(Cc2cc[nH]n2)C(=O)N)ccc2c(c1)CC2.C12CCC(CC1)C2 c1(OC)ncnc(C)c1C(=O)NCC1CCN1C(=O)C=Cc1cnc[nH]1 c1(OC)cc(CNC2CN(C(c3cc(C#N)c[nH]3)=O)CC2C)cnc1Cl CC1=C(C(=O)N2CCC2CNC(c2cccs2)=O)CCCC1 c1ccc(Cl)nc1.c1(C(C(=O)N)NC(C2C(OCC)CC2)=O)cnn(C)c1 C#CC1(O)CC(C(=O)NC(C)C(=O)NCC(CO)OC)C1 O=C1NCCn2nnc(C(N3CCC(NC(C4CC5CCC4O5)=O)CC3)=O)c21 C1(CC(=O)N(CC(COC)C)C)CC(O)CN1C(=O)C=CC(F)(F)F C1(N(C(C(C2CCCCC2)OC)=O)C)CCCCN(C(=O)Cn2nccc2C)C1 C(=O)(C1=CCSC1)NCCOC1CCN(C(C2(C)CC2Br)=O)C1 c1(OC)cc(Br)ccc1CC(N1CC(NC(=O)CS(N)(=O)=O)C1)=O N1(C(C(CC)OC)=O)CCCN(C(=O)CN2CCN(C)C(=O)C2)CCC1 C1(C(=O)NCC(C)(C)NC(c2ccsc2Cl)=O)CC2CC1C1OC(C)(C)OC21 N1(C(C2(C=O)COC2)=O)CCCC1.N(S(N)(=O)=O)CC=O.C1CC1.CO CCCC(CCC)C(=O)N1C(CNC(=O)CCNC(=O)CO)CC2COCC12 c1(C(=O)NCC2CCCN2Cc2cc(I)c[nH]2)ccc(O)c(O)c1O N1(C(Cc2cccc(OCC)c2)=O)CCC2(CC1)CC2C.C(=O)C(C#N)CC.N C(=O)(C(CCOCC(=O)O)C=O)OC(c1nnc(O)o1)C.C(C)(C)C.N c1(NCCc2scc(C)n2)ccc(S(=O)(=O)NC(c2ccccc2C)C)c(Br)c1 N1(C(C(C)SCCCC)=O)CC2C(CC(=O)N(C)Cc3ccsc3)C2C1 C(=O)(CC(C)(O)CC(=O)O)N1CC(F)(C=O)C1.c1(C(=O)O)ccccc1.CC C(=O)(CCCCC(F)F)N(C1CCN(C(C2(C)CC2(Cl)Cl)=O)C1)C Cc1cnc(C(N2CCC2C(=O)NC2CCCCC2(C)C)=O)cc1C C=CCC(C(=O)NC1CCCC1CC(=O)NC(C1(CO)CC1)C)C(C)C CC(C(=O)NCCC1CN(C(c2cccc(C3CC3)n2)=O)CCO1)S(C)(=O)=O C1(CN(C)C(c2ccc(N3CCCC3=O)cc2)=O)CCCCN1C(=O)CC#N c1ccc(Cl)c(C)c1.Cc1cncc(C(=O)N(C)CC2CCN(C(=O)CO)C2)n1 C(=O)(C1=CC(C)C1)N.N1(C(CSCCN(CC)CC)=O)CC(CC)C1 C=CCN=C(NCC1CCCC(C)(C)C1)NC1CCC12CCC2 N1(C(C(CC)OC)=O)CC2(NC(=O)CCc3cc(C)cc(C)c3)CCCC2(F)C1 C1(CNC(c2nc(C)c(C)s2)=O)CN(C(=O)C(C)c2cc[nH]n2)CCCO1 c1(C(=O)NC2CCCN(C(CC3COCC(C)(C)O3)=O)C2)cc2sccc2cn1 C1(C(=O)NCc2nc(C)cs2)CC2(C1)CCC2.C1(C=O)CC2CC2C1.N Cc1cccc(C=CC(=O)N(C)CCN(C)C(C2CCC(O)CC2)=O)c1 Cc1cc(S(N)(=O)=O)oc1C(=O)NC(CO)CCCC.C1(C=O)CC(F)(F)C1 N1(C(c2n[nH]c3ccc(Br)cc23)=O)CCC2(CCCN(C(c3cnco3)=O)C2)C1 c1(C2CCN(C(C3N(Cc4c(OC)cccn4)CC3)=O)CC2)ccc(C#N)cc1 c1(C(N2CCC(c3cc(CN=[N+]=[N-])on3)CC2)=O)ncn2cccnc12 c1(OC)cc(C(=O)NC23CCCC(NC(=O)C(C)O)(C2)C3)nc(Br)c1 C(C(CC(C)C)C(=O)NCc1ccccc1-n1cc(CCOC(=N)O)nn1)OC C12(NC(C(C)OCCCC)=O)CCCC1N(C(C1CCC(=O)CC1C)=O)CCC2 c1(CO)cc(NC2CC3(CCOCC3)C2)cc2cccnc12 CC(C)S(=O)(=O)C(C)C(=O)NCCCCC(CO)NC(c1cccc(CO)c1)=O c1(CC)cc(F)c(C(=O)NCC2(C)CCCN2C(=O)COC)cc1F C1(NC(C=CC)=O)CCC12CCC2.C1(C=O)CCC(C=O)CC1.C(C)(C)C C(=O)(C(C(C)(C)C)c1cccc(C)c1)NCCCCCCN(C(CCSC)=O)C N1(C(c2cnn(CCCC)c2C)=O)CC(CO)C2(C1)CN(C(C1CC1C#N)=O)C2 C1(c2ccccc2)(C(=O)OC(C)C(=O)NCC(F)(F)F)CC(=O)C1 C(=O)(C#CC(C)(C)CNC(=O)CO)NC1(CSC)CCC1.CC(C)C c1(C(N(CC(C)NC(CCCOCC)=O)C)=O)cc(C)nc2ccnn12 C1(CNC(c2ccc(NC)cc2)=O)CC2CCC1N2C(c1cncs1)=O C1(C(=O)NC(C(=O)NC2C3(CC(OC)C3)C2)C)CC(=O)OC1(C)C C12(C(=O)NCC3CCCC(C)(C)C3)CCN(C(=O)CN3CCOC3=O)CCC1C2 c1(NC(COC(C(C)Oc2ccccc2Cl)=O)=O)ccc(F)cc1 CC1COCC(C(=O)NCC2(O)CC(C(=O)N)C2)O1.c1(C(C)C)ccccc1 c1(C(N(C(COC)C)C)=O)ccoc1CNC(C1(F)CC=CC1)=O CCCC(C(=O)N(C(C)(C(=O)NCCCCN(CC)CC)C1CC1)C)OC C1(NC(CCc2scc(C)c2)=O)CCCCC1N(C)C N1(C(C(COC)OC)=O)CC2(CC(NC(C3CC4C=CC3O4)=O)C2)C1 c1(C(=O)NC2C(CC)N(C(C3C=CCC3)=O)CC2)cnc(C)nc1C(C)C n1(CC(=O)NC)[nH]nnc1=NCCCN1CCN(C(=O)CC2CC(F)C2)CC1 c1(C(=O)OCC2CCN2Cc2ccccc2)cc(Br)co1 CCCCCCC(=O)NCCC(O)CNC(c1ccc(-c2cnn(C)c2)cn1)=O n1(CC#C)cnnc1C(=O)N(C(C)C(=O)N(CC(O)CO)C)C1CC1 c1(C(=O)NC(c2cccnc2)C(=O)N(CCN(C)CCO)C)cnc(=N)[nH]c1 N1(C(CCCC=C)=O)CCCC2(CCC(NC(=O)Cc3conc3C)C2)C1 N1(C(Cc2cc(C)ns2)=O)CCC(C)C(N(C(=O)C(C(C)C)n2cncn2)C)C1 Cc1ccnc(NC(C2CC(NC(=O)C(C)Cn3cccn3)C2)=O)c1Br c1nc2c(s1)CN(C(c1csc(C#N)c1)=O)CC2.c1(CC)ccc(C(=O)N)s1.C c1(-c2cn(CC(F)(F)F)nc2)nc(C2CCC2)nn1CCn1cccn1 C1(NC(c2c(C)cno2)=O)CN(C(=O)CSc2nccn2C)Cc2ccnn2C1 C=CC1(C(N2CC3(CNC(c4ccn(C)c4)=O)CCC2C3)=O)CCCCC1 c1(C(=O)OC)ccc(C(=O)N)n1C.C1(O)(CC)CN(C(C2CC2(Cl)Cl)=O)C1 CC1C(=O)N(C)CN1C(c1nc(N2CCOCC2)ncc1Br)=O n1(CC(N2CC(CC(C)NC(=O)CN3CCSCC3)C2)=O)nnc(=O)[nH]1 C1(C)(C(N(CCN(C(C(CC)Sc2ccccc2)=O)C)C)=O)CCNC(=O)C1 c1(CCC(=O)N(CCC)C)cccc2ccccc12.C(=O)(C(C)(C)S(C)(=O)=O)N C1(CNC(Cc2n(C)ncc2)=O)CC2CC(C1)N(C(c1nc(Cl)cs1)=O)C2 N1(C(C(C2CCC2)NC(c2cnn(C)c2C(F)F)=O)=O)CCCCC(CO)C1 c1(NC(C2CC(F)CN(C(c3cn[nH]c3)=O)C2)=O)ncnc2sc(Br)cc12 C1(C(=O)NCC(CNC(CCC(=C)C)=O)(C)O)CCCCC12OCCO2 c1(C(=O)NCC2(F)CC(NC(=O)CCn3cccc3)C2)nccc2ncccc12 CCCC(CC)C(=O)N1CCN(C(=O)CN(C)CC)C(C2CC2)C1 c1(C(=O)N)cc(O)cc([N+](=O)[O-])c1.C(C(C)(C)C(=O)NCC(C)(C)C)OC C(C(C)(C)CC(C)O)NC(C1C2(CC(NC(C3C=C(C)CS3)=O)C2)C1)=O C(=O)(C(CCC1CC1)NC(=O)CC(C)C)NCC(COC)C.C(C)=O.N C1(CNC(c2n(C)nc(O)c2)=O)CN(C(=O)C(CO)c2ccccc2)CC1(C)C O=C(C1Cc2ccc(F)cc21)NCC1C2CCCC1N(C(=O)Cc1csnn1)C2 C1(C(N(CCC(C(C)C)Nc2cc(CC)ncn2)C)=O)CCN(OC)CC1 C1(NC(=O)COC2CCCCCC2)CN(C(c2csc(S)n2)=O)CCC12CCC2 N1(C(=O)NC(CCOC)C)CCCCC(NS(C)(=O)=O)C1 CC(C)(CNC(c1ccc(C2CCOC2)s1)=O)CNC(c1csc(C)n1)=O C=CC(CCC)CC(=O)NCCCN(C(=O)C=Cc1cn(C)nn1)CCO C1(C)(C(=O)OC)CCCN1CC1C=CCC1 CCS(=O)CC(=O)NCC(C)(C)CN(C(=O)C(C)Cc1ccccc1Cl)C N1(CC=O)C(=O)NC(C)(C)C1=O.CC1CC(C)C1C(=O)NC1CCC1.C Cc1ccc(C(N2CCC(N(C)C(c3ccc[nH]3)=O)C(C)C2)=O)cc1S(C)(=O)=O CC(C)C(C(=O)N(C)CCNC(=O)C(F)(F)CC1CCCO1)n1ccnc1 c1(C(=O)NCC2CC(C)N(C(=O)C(=O)C3CCCC3)C2)cnc2sccn12 Cc1cc(C(=O)NC(C)CC(C)NC(=O)C(C)O)nc(C)c1.c1ccc(F)nc1 N1(C(C(CC)(C)OC)=O)CCCC2(C1)CN(C(c1cc([N+](=O)[O-])ccc1C)=O)C2 C1(CCCOC(C2C(OC)CC2)=O)CCCN1C(C)=O c1(-c2ccc(OC)c(F)c2F)cc(C(=O)Nc2cncs2)c2ccccc2n1 c1(NC(=O)NCC#C)cccc(C(=O)NCCn2ncnn2)c1 N1(C(CCN(C(=O)C(=CC2CCCC2)C)CC#C)=O)CCC2CCC(C1)N2C C1(n2cc(C(CC)(C)O)nn2)CN(C(c2nonc2C)=O)CC1C C(c1cncn1C)=CC(=O)NC(C)C(C)(C)NC(C1CC1(Cl)Cl)=O C1(C)(C(N(C)CC2N(C(CCOC)=O)CCC2)=O)CCC(OC)CC1 O=C1COc2cc(F)c(C(=O)NC3CC3)cc2N1.c1(C(=O)N)cc2c(s1)CCC2 N1(C(CC(C)C)=O)CCN(C(=O)C2=CCSC2)C2CCCC12 c1(C(N2CCC(N(C(C3CCN(C)C3)=O)CC)C2)=O)cncc(-n2ccnc2)n1 CCCCC(CC)CC(=O)NCC(C(N1CCSC(C)CC1)=O)N(C)C C(=O)(C(C(=O)N)C(C)C)OCC.C(c1cncn1C)=CC=O.C1CCC1.C C1(NC(Cc2nc(C(C)OCC)sc2)=O)CCCCC1NC(C1SCCS1)=O C(=O)(C1=C(Cl)CC1)N(CCNC(=O)COC(F)(F)F)Cc1ccccc1 c1(C(=O)NC2C(NC(c3ccc(Cl)c(F)c3)=O)COC2)c[nH]c2cccnc12 c1(CNC(C2(C(C)C)N(C(C(C=C)CC)=O)CCC2)=O)cc(C)cc(C)c1 C1(CC=O)COC2(CCC2)CO1.C1(C(=O)OCC)CC1CC(=O)NCC CC1CC(NCc2nccc(-n3ccnc3)n2)CCS1 CC(CC(F)F)C(=O)NCCC1CN(C(=O)C2=CCC2)CCO1 C1(C(=O)NCCCCC2(NC(C3CC(=O)NCC3)=O)CC2)CC12CCSCC2 C1(C(=O)Nc2c(C)n(C3CC3)nc2)CNC(=O)CN1C(=O)C(C)c1cc[nH]n1 C#CCCCC(C)C(=O)NC(CC(=C)Cl)C(=O)N1CCC(C2CC2)C1 C1(NC(N2C(C(=O)OC)CC(C(F)(F)F)C2)=O)COc2c(OC)cccc2C1 C(c1cccc(O)c1)=CC=O.c1(CC)nn[nH]c1C(=O)NCCC1CCOC1 c1(C(=O)NCC(CN(C(=O)CCCC(N)=O)C)(C)C)ccc(Cl)c(F)c1N C1(C(=O)NCCC(CCNC(c2c(C)ccs2)=O)C)CCC12CCOCC2 c1(C(=O)NCC(CC)(CC)NC(=O)C(C)N(C)C(C)=O)coc2c1CCCC2 C(C(=O)NOCCCC1CC1)C1(NC(=O)CC2C=CCC2)CCC1 c1(OC)ccc(C(=O)NCC2CC(OC)CN2C(=O)CC(F)(F)Cl)c(C)n1 c1(NCC(C)(C2CC2)NC(=O)CCc2ccc(F)cc2)nc[nH]c2nccc1-2 CC(C)C(C)(C)C(=O)NCc1cn(CC)nn1.C(=O)(C=O)N.CCC(N)=O CC1CCC(NC(C23CC(CN2C(C2CCC2C)=O)C3)=O)CC1 C1(NC(CS(CC)=O)=O)CCN(C(C2C3CCCC23)=O)CCC1CO C=CC1OCCCC1C(N1CCOCC(NC(=O)COC2CCOCC2)C1)=O Cc1cn2cc(CC(=O)NC3CN(C(=O)C(C)P(C)(C)=O)CC4(CC4)C3)nc2s1 N1(C(c2c(C)nncc2)=O)CC(C2(NC(=O)C(C3CCC(=O)CC3)F)CC2)C1 C1(CNC(C2(C)C(C)C2)=O)CCN(C(=O)CN(c2ccncc2)C)C1 C1(NC(C(CC)(CC)CC)=O)CN(C(=O)C(Br)=C(C)C)C2CCCCC12 c1(OC)cc(C)c(C(=O)NC(C)C2CC2)cc1Cl.c1(C=O)cc(C)nc(C)n1 N1(C(c2ccc(SC)s2)=O)CCC(C)C(CNC(c2cc(C)nn2C)=O)C1 C1(c2cn(CCN3CCOCC3)nn2)(NC(c2ncoc2Br)=O)CC(F)(F)C1 c1(C(N(CC(O)CNC(=O)COc2ccccc2O)C)=O)ccc2cccnn12 C1(C(N2CCCCCC(NC(=O)Cc3cnc[nH]3)C2)=O)CCS(=O)(=O)C12CCC2 C#CCCCC(C(=O)NC1(C(=O)OC)CCCC1)N1CCCC(CF)C1 C1(OCCCC)CC(N(C(C2CCN(CC(C)C)CC2)C(=O)NCC)C)C1(C)C N1(C(c2c(C)nc(C)s2)=O)CCC(C(F)(F)F)C(NC(C2CCC(F)CC2)=O)C1 C12CC(CO1)N(C(C1CCN(C)C(=O)C1)=O)C2.C(C(=O)NC)(C(C)C)OC Cc1ccc(CC(=O)NCCC(C)N(C)C(c2coc(C(N)=O)c2)=O)c(Cl)c1 CC1CCN(C(c2cnc3[nH]ccc3n2)=O)CCN1C(=O)C(F)C(C)(C)O Cn1cc2c(n1)CCC(NC(c1cc(C3CC3)sn1)=O)C2 N1(C(C(F)=C(C)C)=O)CCCC2(CCC2)C1.C1(C)(C=O)CC(C(C)(C)C)=NO1 C1(C(=O)NCC(C(CC)C)(C)O)CC2C=CC1N(C(=O)C(C1CCCCC1)C)C2 C1(O)(CN(C(C2ON=C(CC)C2)=O)C)CCCN(C(c2c(Cl)ccnc2C)=O)C1 N1(C(CC2CN(C(c3cc(C)cc(F)c3)=O)C(C)(C)C2)=O)CCC(C)C(C)(C)C1 C1(C(=O)NCCN2CCC(OC)C2)CN(C(=O)C(C)CC(N)=O)CC12CCC2 c1(CC)ccc(Cl)nc1.C(=O)C(O)CC1CC1.C(C)(C)C1(C=O)CC1.CO C(CNC(C1(CCOC)CCC1)=O)(CC)(CC)NC(CC1CC(=C)C1)=O Nc1ncccc1C(N1CCN(CCCNC(c2ccncc2F)=O)CC1)=O N1(C(c2nc(C)[nH]n2)=O)C2CCC1CC(N(C(=O)C(C)Oc1ccccc1)C)C2 CN1CCCC1CC(=O)NCC(C)(CO)NC(c1ccn(C)n1)=O C1(NC(C2CC3(CCC3O)C2)=O)CCN(C(=O)C=CC(F)(F)F)CC1F N1(CCC(=O)N(C)CC2(NC(C(n3cc(Br)cn3)C)=O)CC2)CCCC1=O N1(C(C2CCN(C)C2)=O)CC2CCC(C1)C2NC(=O)CCSCC(N)=O C=CCC(C(=O)NC1CC(NC(c2cc(C3CC3)ccn2)=O)C(O)C1)C(C)C c1(C(N(C2CCN(C(c3c(C)csc3Cl)=O)CC2)CCO)=O)cnn(C)c1C#N c1(OCC)cc(Cl)ccc1C(=O)NCc1ccc(Cl)nc1 CCC(O)CCc1cn(C2CCCC2C(=O)O)nn1.C1(=O)CC(=O)N1 C1CN(C(C2(C)CC2(F)F)=O)CC12CC2.c1(NC(C)=O)cccc(C(=O)N)c1 C1(NC(C(n2cc(Cl)cn2)C)=O)CN(C(=O)C(=O)N)C2(CCCCC2)C1.C1CC1 c1(CCC(=O)NCCC2CCN(C(C3CC34CC4)=O)C2)n[nH]c2ccccc12 CC(C)(F)CC(=O)N1CCCC(NC(C2CCCN2C(=O)C(C)(C)C)=O)C1 c1(C(=O)NC2CC(C#C)C2)cncc(CNC(=O)COCCC=C)c1 CC(C(=O)NC1CN(C(C2CC(C)(CO)C2)=O)C1)C(C)C(C)(C)C.C(=O)O C(CCC(=O)NC(c1ccnn1C)COC)N(C(COCCC=C)=O)C c1(C(=O)NCC(CCNC(CC(CC)C2CCC2)=O)O)c(C)nc(C)n1O N1(C(C2CCN(CC)C2)=O)CCC(C(N2CCCC2C(=O)NC)=O)C1C(C)C N1(C(C2CC(=O)NCC2)=O)CCC2(CCCN(C(=O)CC3CC3C3CC3)C2)CC1 CC(CC(=O)NCC1CC1NC(c1cc(F)c(N)c(F)c1)=O)C(C)(C)C N#Cc1ccc(NC(C2CCCN(Cc3ccc(F)c(O)c3)C2)=O)c(C#N)c1 C1(C(N2CCC(NC(CC(C)c3ccncc3)=O)C2C)=O)CN2CCN1CC2 C1(CNC(c2ncn(C)c2)=O)(C)CC2CCCC2C1.c1cccs1.C(=O)(C)N Cc1cccc(C(=O)NC(C(=O)NCC(c2ccccc2)C)C2CCCC2)c1O CCCCCCCCNC(C1CSCCN1C(=O)CCN1CCCC1=O)=O N1(C(c2cc(CNC(C3(C)C(C)CCC3)=O)ncc2)=O)Cc2ncsc2C1 C(=O)(C(C)=Cn1ccnn1)NC(CCCC)CNC(c1cnccn1)=O CCC(CC)C(C)C(=O)NCC1CCN1C(=O)Cc1ccccc1.C(C)(=O)N C1(CC(=O)NC(c2c[nH]nn2)C)CCC(C(C)C)CC1.c1occc1C(N)=O C(=O)(CCC(C)CCCC)NC1(C(=O)NC(CC=C)CC=C)CCSC1 C1(NC(C=CC(=O)N(C)C)=O)COC2(C1)CN(C(=O)C1=CCCO1)C2 c1(CC(=O)NC(C2CCN(C(C3C=CCC3)=O)C2)(C)C)cc(F)ccc1F C1(CC(=O)NC)CN(C(c2cccc(N)n2)=O)CCN1C(C1CC(C)(F)C1)=O n1(CC)ccc(CC(=O)NCCC2CCN(C(C3CC3(Cl)C(=O)O)=O)C2)n1 CCCC(C)(C)CC(=O)NCC(=O)NCC(=O)NC(C)CCOC N1(C(c2csc(CC(F)(F)F)n2)=O)CC2CC1CN2C(=O)C(O)(C1CC1)CC C1(C(N(CC(C)NC(C2(S(C)(=O)=O)CC2)=O)C)=O)CCn2ncnc2C1 C12(C(N3CC(=CC)C3)=O)CC(CO1)N(C(=O)CC1C3CCCCC13)C2 N1(C(c2cc(C)oc2)=O)CCOC(CN(C)C(C2CC3(C2)CC3F)=O)C1 N1(C(C(C)SC)=O)CCCC2(CCCN2C(=O)OC(C)(C)C)CC1 C=C(C)c1ccccc1NC(C1CCCCCCN1C(c1ccnnc1O)=O)=O C1CN(C(c2cc(Cl)ccn2)=O)CC1C.C1(CC(=O)NC)(C(=O)OC)CCCC1 C1(C)(C(=O)NC(CNC(C(C2CC2)OC)=O)C)Cc2ccccc2N1 N1(C(c2nc(CCC)sc2)=O)CC=CC(NC(=O)Cc2ccsc2C)C1 Cc1nc2cncc(C(N3CCC(C)N(C(=O)CC4(C5CC5)CC4)CC3)=O)c2[nH]1 N1(C(c2cnoc2)=O)CCN(C(C2CCCCO2)=O)C2(CCC2)C1 c1(CNC(Cc2nc(C)sc2)=O)ccc2c(c1)CN(C(c1cn(C)nc1Cl)=O)C2 C(CCF)(C(=O)NCCCc1cncnc1)NC(c1ccccc1O)=O c1(C(N2CC(C)N(C(=O)Cc3cc[nH]n3)CC2C)=O)cc2c(F)c(Cl)ccc2[nH]1 N1(C(c2nccc(Cl)c2Cl)C(=O)NCCC2(C)CC2)CCC2(CC1)C(O)CC2O C12(CNC(C(CSC)O)=O)CCC1CN(C(C1CC3(C1)CC3(F)F)=O)C2 C1(NC(C(C)C(F)F)=O)CC2(NC(C3CCC3)=O)COC1C2 CC(C)C(C)(C)C(=O)NC1CN(C(C2COCCN2C)=O)CC1F Cc1nnc(CC(=O)NCCCCCN(C(=O)C(C)(C)c2ccc(Cl)s2)C)o1 N1(C(C(C(CC)O)(F)F)=O)CCOC2(CCN(C(c3nnsc3SC)=O)CC2)C1 C(C)(CC(=O)NC(C)(C)C1CC1)OC.c1(CC=O)cnn(C(C)(C)C)c1 N1(C(C2(OCC)CC2)=O)CCC(CC(=O)NCCC(O)C2CC2)C1 C(CC(=O)N(C)CC1(O)CCC1)N(C(=O)C)CC=C.C1(C=O)CC1C.N N1(C(=O)COC2CN(C(C3CC4(CCCO4)C3)=O)C2)CCC12CCCOCC2 N1(C(C(C)(C)c2cncnc2)=O)CCN(C(=O)C=Cc2cncs2)CC12CCC2 S(=O)(=O)(c1nc(N2CCC(CCCO)C2)ccc1Br)NCC=CCCOC S(=O)(=O)(c1cc(C(N2CCCC(O)C2)=O)c(C)o1)NC.C1(C(=O)N)CCOC1 C(=O)(CCC(=O)NC1CC1)OC(C)(C)C.C(=O)C(F)(F)CC1CCCO1.C c1(C(=O)O)cc(N2CCCCC2CNCc2cccc(C(F)(F)F)c2)ncn1 Fc1ccc(-n2nnnc2C(c2ccc(CO)o2)NCCC2CCCCO2)cc1 C(C(C)C(C)OCC)OC(C)C.C1(=O)CCOC(=O)C=CCN1 c1(OC)cc(C(N2CCN(C(c3cc(F)cc(Br)c3)=O)CC2)=O)cc(C)c1 C1(C(N(CCOC)C2CC2)=O)CCCC(NC(=O)C(O)C(F)(F)F)CC1 c1(CNC(N2CCCC(C(=O)NCCC)C2)=O)cccc2cc(C)oc12 c1(C(=O)NC(CC(=O)N(c2ccccc2O)CC)C)cnc(C)nc1C CC1CN(C(=O)CCc2ccccc2Cl)CC1NC(C1CC(=O)N(C2CC2)C1)=O C1(NC(=O)Cc2coc(-c3ccccc3)n2)C2CC1N(C(=O)COC1CC1)C2 CC1CCN(C(=O)COC(F)(F)C(F)(F)F)CC1C.c1(C=O)cncn1C.N CC(C)(CCNC(=O)C(C)(C)c1cscn1)NC(=O)CCc1nc(O)n[nH]1 c1(C(=O)NCC2(OCC)CN(C(C3CCOC3C)=O)C2)cn(C)[nH]c1=N c1(C(=O)NCCCCC(C)NC(c2ccn(C)c2)=O)ccc2nnc(O)n2c1 N1(C(CCc2c(C)c[nH]c2C)=O)CCC2(NC(c3ccc(Cl)cc3O)=O)CC2C1 CC(O)(CCC1CC1)CN=C(NC1CCC1)NC1CC(=O)N(C2CC2)C1 c1(OC)cc(CN2CCOC(C(=O)NCc3cnccc3C)C2)c(F)cc1F C1(C(C)C)CCN(C(=O)CC(C)n2ccc(C)n2)C1.C(CCOCC=O)OC.N c1(C(=O)NCC(C2CC2)NC(CCCC)=O)cc(F)cc(N)c1F c1(C(=O)NC(CNC(c2sccc2-n2cnnn2)=O)CO)scc2c1OCCO2 C1(C(=O)NCc2ccn(C)n2)CC2(CCC2)CN1C(=O)C(=O)NC1CC1 C(=O)(C1=NOC(c2ccc(F)cc2)C1)N1C(CC(N2CCCS2(=O)=O)=O)CCC1 c1(C(=O)NCC2CCN(c3cc(C)ncn3)C2)ccc2nn[nH]c2c1 CC1CCC(SC(C)C(=O)N(C23CC(CCN2)C3)C)CC1 CC1SCCCC1C(=O)NC1(CN2CCCCC2)CCC1 S(=O)(=O)(c1ccc(N2CCSc3ccccc3C2)c(F)c1)NC(C(CCC)C)C n1(C(C)CC(=O)NCCNC(=O)C(C)(C)c2ccnn2C)cnc2ccccc12 C(C)(C)(CCCNC(c1csc(C)c1C1CC1)=O)NC(c1[nH]cc(C)c1)=O c1(C(=O)NCC(CC)NC(c2cnccn2)=O)cnc2c(c1)CCCC2 CCC(CNC(=O)CN(CCO)C(C1CC(C#N)(OC)C1)=O)(CC)CC CCC(C)C(=O)C(=O)N1CC2C(C(=O)NC(C)C(=O)NC)C2C1 N1(C(C(C)N2CCC2)=O)CCC(CNC(=O)C=Cc2cc[nH]n2)C(O)C1 N1(C(c2c(-c3cc(C)no3)ocn2)=O)CC(NC(=O)CCc2nncs2)C(O)C1 n1(CC(=O)NC2C(CNC(c3c(C(C)C)con3)=O)CC2)ncccc1=O N1(C(Cc2cccc(CC=O)c2)=O)CCN(C(=O)C(C)=C(C)C)C2CCC12.CO Cc1ccnc(C(=O)NCCCN(C(=O)CC2CC(F)C2)CCO)c1N C(=O)(C#CC1CCCOC1)NC1CN(C(C(COC)COC)=O)CC(O)C1 N1(C(CN)=O)CCCC1C1CC1.C1(CC)CCCCO1.C=C1CC1C(=O)NC C1(C(N(CC(C)NC(=O)CCCC(N)=O)C)=O)CC(=O)c2cc(Cl)ccc2O1 C(C)(C)(CC(=O)NC1CCCC1NC(=O)C=Cc1ncc[nH]1)OC C(=O)(CC1=NN(C)C(=O)C1)NCCCCC(=O)NC(CCC#C)C(=O)NC C1CN2CCCCC2CN1C(=O)C=C1CCC1.C(CC(Cl)=CC(=O)NC)N(C)C n1(C(C(=O)N(C(CC)(C)C)CCC#N)C)cc(CCS(N)(=O)=O)nn1 Cc1cccc2c1CCOC2C(=O)N1CC(NC(c2ccc(S(N)(=O)=O)[nH]2)=O)C1 N1(C(c2c(C)onc2)=O)CC(NC(c2sccc2S(N)(=O)=O)=O)CC2(CC2)C1 N1(C(c2nc(C)c([N+](=O)[O-])cc2)=O)CCCC2C1CCCN2C(c1cnco1)=O CS(=N)(=O)C1CN(C(C23CC(CN2C(C2CCCS2)=O)C3)=O)C1 c1(C=O)ccc2c(c1)OCC(=O)N2.c1(COC)cc(C(=O)NC(C)C)no1 O=C1CC(C(=O)NCc2ccoc2)N(C(=O)C(O)c2ccsc2)C1 N1(C(C2N(C(C(C=C)CC)=O)CCC=C2)=O)CC2CC(OC)C(C2)C1 C#Cc1ccccc1CC(N1CCCC1CN(C(=O)C(O)C1CCCC1)CC)=O c1(C(=O)NC2CC(NC(CC(C(C)C)(F)F)=O)C2)ccc2nnn(O)c2c1 C12(C(NC)=O)CC3CC(F)(C1)CC(F)(C3)C2.N1(C(C)=O)CCOCC1.CCO C1(C(N(CC(CCC)C)C)=O)CCN(C(=O)C2(COC)CC2)O1 C(=O)(C(CC1CCCOC1)NC(=O)NCCCSCC(=O)OC)NC C1(OCC(CC)N)C2CC1N(C(=O)OC(C)(C)C)C2 c1(OC)ccc(O)c(C(=O)NC(CNC(=O)C(Cl)=CCl)C2CCC2)c1 Cc1nc(O)c2cc(C(N3CCC(N=[N+]=[N-])CC3)=O)ccc2n1 C1(C(N(C(CNC(C2(C(=O)OC)CC2)=O)C)C)=O)COC2(CCC2)C1 S(=O)(=O)(CCS(=O)(=O)c1ccc(C)cc1)NCC(c1c(OC)cccc1)O C#CCCCCC(=O)N1CC(CNC(c2ccc(SC(F)(F)F)cc2)=O)(OC)C1 C(=O)(C(C(C)C)C(C)C)N1CCN(C(c2ccc(COC)cc2)=O)CC1C(F)F c1(C(=O)NC2C=CCN(C(C34CC3C4)=O)C2)ccc(F)cc1F N1(C(C2CC(C#C)(O)C2)=O)CC(NC(=O)CCO)CC(C)(C)C1.C1CCCO1 C=C1CC(CN(CC(F)(F)F)CC(F)(F)F)C1 c1(CNC(C2N(C(c3c(C(C)C)c[nH]c3)=O)CC(=O)C2)=O)cccc(F)c1F N1(C(CCC=C)=O)CC2CCCC(C1)N2C(c1cccc2nncn12)=O Cc1ccc(F)c(Cn2cc(CNC(=O)CNC(=O)CC(C)C)nn2)n1 C=CCCC(C(=O)NCCC1CC(C)=NO1)NC(C1CN(C(C)C)C1)=O C1(C(N2CCCCC2CNC(C23CC(F)(C2)C3)=O)=O)Cc2ccncc2C1 c1(C(C)C)c(C(=O)N(C)CC)cnn1C.C(=O)CN(C)C=O.C(C)(C)C.N C1(NC(C2(CCNC(C3CCCC3F)=O)CCC2)=O)CC12CC(O)C2 c1(CC)cc(C(=O)NCC2CC2)nn1CCO.C1(CC=O)CCC1C1CC1 c1(CC)ccc(C(N2CCCC(O)(C)C2)=O)c(F)c1.c1(C(=O)N)c(C)nsc1C c1(C(N2C(C(=O)Nc3c(C)ccc(Cl)c3)CC3CC32)=O)cc(C)c([N+](=O)[O-])cn1 Cc1cn2c(n1)CCC(NC(=O)CCCn1cc(C3CC(F)(F)C3)nn1)C2 Cc1cncc(C(=O)NC2CN(C(=O)COc3ccc(Cl)nc3)CC2F)n1 N1(C(C(C(CC)C)O)=O)CC2(CCCN(C(=O)CC3CC34CC4)C2)C1 C1(N(C(c2cnn(CCOC)c2)=O)CC)CCCN(C(c2c(Cl)cnn2C)=O)C1 C(CC1CCOCC1)(C(=O)N)NC(C(C)n1cccn1)=O.C12(CC)CC(CO1)C2 c1(C(=O)NCCNC(C(COCC=C)c2ccccc2)=O)oc(CCC)nc1C Cc1ccc(C(N2CC(NC(c3c(C)nc(O)nc3C)=O)C(O)C2)=O)c(N)c1C C(CCCCCNC(c1cccs1)=O)NC(=O)C=Cc1cccs1 Cc1csc(C(=O)NC2CCCC(CNC(=O)C(C)c3ccco3)C2)c1Cl c1(SC)ccc(CC(=O)NCC2CCN2C(=O)CCCN2CCOCC2)cc1 CC1=C(C)CN(C(c2coc(CNC(c3nn(C)cc3Cl)=O)n2)=O)CC1 C1(CC=C)(NC(=O)CCc2cncnc2)CCN(C(C2CC2)=O)CC1.C(N)=O N1(C(=O)CC2CCCN2C(C2CCCO2)=O)CCC(CO)C(F)(F)C1 n1(CC(C)O)cc(C(=O)NC2CN(C(c3nncs3)=O)CCC2C)ccc1=O N1(C(C(CC)N(C)C)=O)CCOC2CN(C(C3(Cl)CC3(F)F)=O)CC12 c1(OC)cc(C(N2CC(C3CCC3)C2)=O)ccc1OC1CCCC1 CC1(C)C(C(=O)O)CCN1CC=CC(F)F.c1(C=O)ccc(Cl)cc1 N1(C(C2(C)CCN(C(c3cnn4c3OCC4)=O)C2)=O)CC2(CCCO2)C1 C1(NC(c2c(CC)occ2)=O)CCC2CN(C(C3C4COCC34)=O)CC2C1 N1(C(C2(C)N(C)CC(OC)C2)=O)CC2CC(C1)N(C(=O)CC1CC1(C)C)C2 c1(C(=O)NCC(C)NC(C2CCCC3(CC3)C2)=O)ccc(=O)n2c1CCCC2 c1(C(N2CCCCC(NC(C3CC(OC)C3)=O)C2)=O)cc(C)c(C)cc1Cl N1(C(C(C)N(C)C)=O)CCC(F)(C)C1.c1cccc(C(F)(F)F)c1.C(=O)C.N c1(OC)cc(C(N2CCC(O)(CN(C(=O)C(C)O)C)C2)=O)cc(Cl)c1 C(C(=O)N1CCCC1CNC(C)=O)(C(C)CC)NC(CC(CC)SC)=O c1(C(N2CC3(CN(C(c4c(C)ccnc4Cl)=O)C3)C2)=O)c(O)nnc2c1CCC2 c1(C(C(=O)NCC2(O)CCN(C(=O)CCc3cnc[nH]3)C2)O)ccc(F)cc1F c1(CC)ccccc1CC.c1(CC=O)ccc(C)s1.C(=O)CN(C)C(N)=O CS(=O)(=O)C(CCc1ccc(F)cc1)C(=O)NCCc1ncco1 C1(NC(C2C(OC)C2)=O)CCCCCC1O.C12CCC(CC1)c1cn(nn1)CC2 c1(C(=O)NCCC2CC(NC(c3ccc(C)cn3)=O)C2)cc(=O)cc(Cl)[nH]1 Cc1ncnc(O)c1CCC(N1CCC2C(NC(=O)CCCN=[N+]=[N-])C12)=O N1(C(C(n2ncc(C)c2)C)=O)C(C(N2CC(OC(=O)N(C)C)C2)=O)CCC1C CC1(O)CCN(C(C2C3CC4C(C3NC(=O)CC3CCCO3)C24)=O)CC1O C#CCC(C)(C)C(=O)NC1CCCCC1NC(C1CNC(=O)N1)=O C1(C(=O)NCC(CCC)NC(c2ccccc2SC)=O)CCc2ccccc2C1 C1(C(N2CC(C#C)C2)=O)(OC)CCN(C(c2cnn(C)n2)=O)C1 c1(C(=O)OC(C)(C)C)cc(=NC(=O)c2sc(NC(C)=O)nc2C)[nH]c(Cl)n1 Cc1ccc(C(=O)NCC23CC2CN(C(=O)C(C)(C)c2sccc2Cl)C3)c(O)n1 c1(OC)cc(NCC2CCCC(C(=O)OC)C2)cc(F)c1 CC1NC(=O)C2=C1N(c1ccccc1)C(=S)NC2c1cc(F)c(Br)cc1F c1(CCNC(=O)NC2C(CC(C)C)C2)nc(-c2cnco2)cs1 C(C(C)C(=O)NC(C1CC(NC(=O)Cc2cccs2)C1)C)SC n1(CC)ncnc1C(N1CC(CNC(=O)CCC2(C#N)CCC2)C1)=O c1(CC(N2CC3CC2C3CNC(C2(CF)CC2)=O)=O)ccc(Br)c(F)c1 CC1CCN(C(C2CCS(=O)(=O)N2)=O)C1C.C1(N(CC(=O)N)C)CCSC1 C1(NC(c2cc(COC)[nH]n2)=O)CC2COC1C2.C(=O)(C(C)c1ccco1)N c1(OC)ccc(C(C)C(N2CCC(CCNC(c3csnc3OC)=O)C2)=O)cc1 Cc1ccccc1CNC(c1ccc(CNC(c2ccsn2)=O)s1)=O Cc1ccc(S(=O)(=O)CC(C)NC(c2ccsc2Br)=O)cc1 N1(C(C2N(C(c3c(C)nn[nH]3)=O)CCC2(C)C)=O)CC(C)OC2(CCC2)C1 c1(C(=O)N)cncnc1-c1ccccc1.CC(F)(F)C(=O)NC(C)(C)C1CCC1 C1(C(=O)NC2CCC(C(C)O)CC2)CC2CCC1N2C(=O)C(C)(C)C(C)O c1(C(c2nnnn2CCCF)NC(C2(C)COC2)C)nc2c(s1)CC(C)CC2 C1(CC(=O)NC(C(=O)N(C)CC)C)(NC(c2ccncn2)=O)CCCCC1 CC1(C)CCC(C(=O)NC2(C(=O)NC3CC(CC(N)=O)C3)CCC2)C1 C(=O)(CC(=O)OC)NCCC1(C(=O)NCC(COCC)C)CC1 C1(C(=O)NCC(CC)NC(CCCN(C(=O)OCC)C)=O)CCCC(F)C1 C(CCC(=O)NCC1CCOC1)N(C)C(C1CC1(F)F)=O CN1CCOC(C(=O)NC23CC(NC(=O)CP(C)(C)=O)(C2)C3)C1=O Cc1cc(C(N2CCCC(C)C2CNC(=O)C)=O)ccc1C1CC1.C(N)=O C1(NCc2cnc(CC)o2)CC2CCC1N2 C(=O)(CC(C)(C)N(C)C(c1c[nH][nH]c1=N)=O)N(CC(F)(F)CO)C C#Cc1cccc(OCC(=O)NCC(C(C)(C)C)NC(c2c[nH]nc2F)=O)c1 Fc1cnc(Br)cc1-c1nc(C2CCOC2)nn1-c1ccc(Cl)cc1 c1(C(=O)NCCN(CCOC)C(c2ccncc2F)=O)ccc(F)c2occc12 C1(C(C)C)(C(=O)NC2CC(C(F)F)C2)CCN(C(C2CCC2C#N)=O)C1 n1(CC(=O)OC(CCCC)C)cnc2ccc(F)cc2c1=O c1(OC)cnc(C(=O)N)cn1.C1(C)CCCN1C(C1CCN(C2CC2)CC1)=O.C N1(C(=O)C(C2CCCCC2)NC)CC(C2CCN(C(c3ccns3)=O)CC2)C1 C#CCC(C(=O)NCC1CC(C)C1)NC(c1cnc(OCC)nc1)=O C1(NC(C(=C(C)C2CC2)F)=O)CN(C(c2csc([N+](=O)[O-])c2)=O)CC1(C)C c1(CN2CCCC(C(=O)NC(c3ccc(Cl)cc3)C(C)C)C2)cccc(O)c1O c1(NCC2(COC)CCC2)ccc(S(=O)(=O)NC2CCCC2C#N)cc1Cl n1(CC(=O)NC2CC(O)CN(C(c3ccc(CO)s3)=O)C2)cnc2ccccc12 N1(C(C2CCC2)=O)CCCC(C)C1CCO.C(C)(C)(C(=O)N)NC(=O)OC C(CCC(=O)NCC1CCC(NC(=O)CC(=O)N)C1)OC(C)C.c1nccs1 Cc1cc(C(N2CC3CC(NC(=O)C(F)(F)CC(C)C)C2C3)=O)c(N)c(F)c1 N1(C(CNC(CC)=O)=O)CCN(C(=O)Cn2nc(C(F)(F)F)cc2C)CC1CO CN1CCOC(CNC(=O)C(Cn2cncn2)NC(C2CC3(CC3)C2)=O)C1 C1(NC(C2(C3CC3)CN(C(c3ccsc3)=O)C2)=O)CC12CCCCCC2 c1(OCCCOC)ccc(C(=O)NCCC2(N)CCC(C)CC2)cc1OC C1(C(N2CC(C=O)C2)=O)CCC(C)(C)N(C(=O)CCc2cn(C)cn2)C1.CC C1(C(=O)NC(CC)CNC(c2cc[nH]n2)=O)CCC2(CC1)NC(=O)NC2=O CN=c1ccc(C(=O)NC2CCCCN(C(=O)C=Cc3ccccc3Cl)C2)c[nH]1 c1(CC(=O)NC2CC(C)N(C(c3c[nH]nc3C3CC3)=O)C2)cnc2n1CCOC2 N1(C(C(C)C(F)F)=O)CCN(C(c2cc(-c3cccnc3)on2)=O)CC1C(F)F C(c1ccc([N+](=O)[O-])s1)=CC(=O)N(CC(C)(C)NC(=O)COC(F)F)C c1(CC)ccc(C(=O)NC2CN(C(=O)C(F)(F)C(F)F)CC2C)cc1[N+](=O)[O-] Cc1nc2cc(C(N3CC(CNC(=O)CCCO)C(C)C3)=O)cnc2s1.C(C)C C1(CN(CC(CCO)C(=O)O)C)CCCCCN1C(=O)OC(C)(C)C CN1CC(C2CCN(C(C3(c4cccs4)CCCC3)=O)CC2)CC1=O CC1CN(C(=O)Cc2ccccc2Cl)CCCN1C(=O)C=Cc1cccc(O)c1 c1(C(=O)NCc2ccc(CN(C(C(C=C)C)=O)C)cc2)cc(C)c(C)nn1 N1(C(CCCCN(C)C)=O)C2CCC1C(C(=O)NC1CC3C=CC1C3)C2 c1(C(=O)NC(C)C2CC2)csc(C2CCCN2C(C2CCN(C)C2)=O)n1 c1(C(=O)OC(c2ccccc2)C#C)ccc2ncn(C)c(=O)c2c1 Cc1cc(C(N2CCC(C(=O)N(C3CC4CCC3O4)C)C2C(C)C)=O)c[nH]c1=N CC(CCC(=O)NC(C)CC1CC1)NC(=O)CC1(N(C)C)CCC1 C1(NC(C2C(=C)C2)=O)(COC)CCCN(C(c2c(C(F)F)cccc2N)=O)C1 c1(CC(=O)NC(C)C(C)(C)NC(=O)CC2OCCO2)c(Br)ccc(F)c1F C(CC(N)=O)(C(=O)NCc1ncccc1O)NC(c1cnc(C)o1)=O C(=O)(C(C)C(O)CC(C)C)N1CC(CC(=O)NCC(CC)C)CC1(C)C Cc1cc(C(=O)NC2(CO)CC(O)C23CCC3)c(Br)c(C)c1 c1(OCC(CNCC=CC(=O)OC)O)ccc(C#N)cc1 CCC(C)(C)C(C)CC(=O)N1CCC(NC(c2scc(C)c2C)=O)C(CO)C1 N1(C(C)C(=O)OCC(C)(C)CC(F)F)CCc2ccccc2C1 c1(C(N(CC(C)N(C(=O)Cc2cccs2)C)C)=O)ccccc1 Cc1c(C(N2CC(NC(=O)C(N3CCOCC3)C)CC2C)=O)cccc1O C1(NC(C(CCC)C(C)C)=O)CN(C(c2cncnc2)=O)C2(CCOCC2)C1 Cn1c(C(=O)NCC2CCCC2)cnc1O.c1(CC(C(=O)N)O)ccc(F)cc1 c1nc(C)c(C(=O)N(CC(=O)N(C)C)C)o1.C(C(=O)NC)(C1CC1)SC c1(C(N2CC3COCC(C2)C3NC(=O)C(F)(F)F)=O)cnc2c(c1)COCC2 C(c1c(Cl)nc2sccn12)=CC(=O)NCC(C)C.C(=O)CC.C(C)(C)C.N c1(C(N2CCC(C)(CNC(c3ncc(OC)cn3)=O)C2)=O)cccc(Br)c1F CCCCC(O)C(=O)N1CCC(O)(CN(C(=O)Cn2ccc(C(F)F)n2)C)C1 c1(N2C(C3CCN(C(C(C)(C)c4cncnc4)=O)C3)CCC2)ncc(O)cn1 O=C(C1=CCOCC1)N1CCC(O)(CCNC(C2(N3CCCC3)CC2)=O)C1 C(CC(C)C(=O)NCc1ccc(C(=O)N(CC)CC2CCOC2)s1)=CC c1(OC)cccnc1C(F)(F)C(=O)NC1CCCC1C.c1(C=O)cc(C)[nH]n1 NC(=O)CCC(=O)NCC1CC1NC(=O)CCc1cccs1 C12(C(N3CCC(C)(CCS(C)(=O)=O)CC3)=O)CCC(C)(CC1)OC2(C)C C1(CNC(CN(C(=O)CCNC(C)=O)CC)=O)CC=CC1 c1(OC)ccc(F)c(C(N2CCC(C)(NC(c3ccc(N)c(Cl)c3)=O)C2)=O)c1F n1(CC(=C)C)nnnc1C(c1ccc(CSC2CCC2)o1)Nc1ccccc1 C1(CC)CN(C(c2cccc(C(F)F)c2)=O)CCC1NC(=O)C(O)CCSC C(CCC(=O)NCC(O)CCNC(c1csnc1Br)=O)=CCC=C C1(CC=O)CCCC2(CC2)C1.C1CCC1.C(=O)(COCC(=O)N)NC.C c1(C(=O)NCCC(=C)CNC(=O)C(N)=O)c(OC)cc(OC)cc1N O=C1NC2(CCN(C(c3cc4n(n3)CCCCO4)C(=O)NCC3CC3)C2)CO1 C1(NC(c2nc(Cl)cs2)=O)CN(C(=O)CCS)CC1c1ccccc1.C1CC1 C(c1c(F)cccc1F)=CC(=O)NCC1CC(C)CO1.c1(C(=O)N)csnn1 c1(NCC#C)cccc(C(=O)NC(CNC(C2CCCSS2)=O)C(C)C)c1 C1(NC(C2C(=C)CC2)=O)CCC2CC1CN2C(=O)CSCCCc1ccccc1 C1COCCN1C(=O)C.C(=O)CC(C)(C)C.CCS(=O)(=O)NC(C)C(=O)N C1(C(=O)NCCC(=O)NCC(=O)N(C)C)CCN(C)C1=O C1(NC(COCCC(C)C)=O)CCN(C(=O)CP(C)(C)=O)C1C(C)C C(=O)(C(CC)CC(C)C)NC1CN(Cc2ccc(OC)cc2Cl)CC1(C)C C1(C2CC2)(OC)CCC1.C1(C=O)CN(C(=O)CC2CCCCN2C)C(C)(C)C1.N C1(CC(=O)NC(C2(C)CC2)C)CCCC1(F)F.C(=O)(C=O)N.C1CC1 C(=O)(C(C)CC(C)C(C)=O)N1CCN(C(C(CCC)OC)=O)C(c2ncc[nH]2)C1 c1(CC(=O)N(C2CCCN(C(C(C(C)C)SC)=O)C2)C)ccc(F)cc1[N+](=O)[O-] C1(C)(C(N(CCCNC(c2cccnn2)=O)CC)=O)CC2C=CC1C2 C12(C(N(C)CC3CCCN3C(=O)CCn3cccn3)=O)CCC(F)C1CC2 C1CCC2(CN(C(=O)CN3C(=O)NC(C)(C)C3=O)C2)O1.C(C=O)=CC.CO C(=O)(CC(C)P(C)(C)=O)NC(CNC(CCCC(=O)OC)=O)(C)C c1(C(N2CCC(C)C2)=O)c(C)ccc(Cl)c1O.c1(CC)cccnc1C(=O)NC C1(C)(C(=O)NCC(CCC)C)CC(O)CN1C(c1snc(C)c1N)=O C1(CC)CCCN1C(=O)Cc1cncnc1.c1(C(=O)N)conc1C1(C)COC1 C1(CNC(C2CSCC(=O)N2)=O)CCC2CN(C(c3cc(O)ccc3Cl)=O)CC12 C(=O)(C#CC1(C)CC1)NC1(c2ccccc2)CC(NC(C2OCC(C)C2)=O)C1 N1(C(C(c2ccc(C)cc2)(F)F)=O)CCC(C)(C)C(CNC(=O)C(C)O)C1 C1(N(CCC)C(C2(CC(F)(F)F)CC2)=O)CCN(C(C2CCCN2C)=O)C1 C1(C(=O)NC2CC(C)C2)(COC)C=CCN1C(C1CCC1)=O C1(NC(c2cnc(CC)o2)=O)CN(C(c2sccc2CC)=O)C2CCCC12 C1(C(=O)NCC(COCC)O)CC2(CCN(C(=O)CC3OCCCO3)C2)C1 c1(N2CC3C(CNC(CN4CCC(C)C4)=O)C3C2)nc(Cl)nc2ccc(Cl)cc12 N1(C(c2cc(C)c(C)s2)=O)C2CCC(C(=O)Nc3ccc(F)cc3F)C1CC2 C1(F)(CNC(CCN2CCN(CC)CC2)=O)CCCN(C(C2CCCS2)=O)C1 C(=O)(C1SCCc2sccc21)NCC1C(NC(=O)Cc2cccnc2Cl)CC1 Cc1cc(F)ncc1NC(=O)CCCOCCO.c1(C=O)ccn(C(C)C)n1.N N1(C(c2c(C)cccn2)=O)CCC(NC(=O)C(C)Sc2ccc(F)cc2)C12CC2 C1(C(N(CCCC)Cc2ccc(C)cc2)=O)C2CN(Cc3cc(O)no3)CC12 C1(C(N2CC(C(=O)NCCOCCC#C)OCC2)=O)CC(=O)N(OC)C1 c1(OC)cncc(C(N2CC(NC(=O)Cc3nnc(S)n3C)CC2C)=O)n1 C1(C(NOCC(C(C)C)O)=O)C2CCC(C2)N1C(C1(O)CCCCCC1)=O c1(C(N2C(C(C)C)CN(C(C3CCO3)=O)CC2)=O)cnn2c1CCCC2 C(C(O)C(=O)NCCCC1CCCCO1)NC(COCC(C)(C)C)=O C1(COC)CN(C(=O)CC2(O)CCC2)CCO1.C(c1ccco1)=C(C=O)C.N Cc1[nH]nc2c1CCC(C(=O)NCCNC(c1ccncc1N)=O)C2 Cc1cncc(C)c1C(N1CC(C(=O)NCCC(C)C(F)F)C(C)(C)C1)=O CCC(C)(CNC(=O)C=Cc1cnccn1)C(=O)NCc1ccc(SC)o1 C12(CC(=O)NC3CC(NC(C4CN(C)C(=O)N4)=O)C(O)C3)CCCN1CCC2 c1(CNC(C2(C(C)(C)OC)CC2)=O)ccoc1C(N1CC2CC2C1)=O C=CC(C)(CC)C(=O)NCC1CCC(NC(=O)CCCN(C)C(=O)O)CC1 c1(C(C)C(N2CCC(CN(C)C(c3n[nH]cc3F)=O)C2)=O)ccc(F)c(F)c1 Cc1cc(Br)ccc1CC(=O)NC1(CNC(c2ccc(N)cn2)=O)CCC1 C1(CCNC(C(C2CCC(=O)N2)C)=O)CCCN(C(=O)Cn2cnnc2)CC1 c1(C(N(CC(CC)NC(C2(n3nccn3)CC2)=O)C)=O)cc(Br)cs1 C1(NC(C2N(C(C(CC=C)CC)=O)CC3CC32)=O)CCCOC12CCC2 C(CN=C(NCC1CCC1)NC1CCC(C(N)=O)C1)C1C(C)C1 c1(C(=O)NCCNC(c2ccn(C)c(=O)c2)=O)cc2cccc(Br)c2o1 C1(C2CN(C(c3cc(Br)cnc3O)=O)C2)(NC(CC(C)CF)=O)CC1 c1(OC)c(C(=O)N(C)CC2CCCN(C(=O)Cc3cocn3)C2)ccnc1F C12(C(N3CC(CNC(COCCCOC)=O)C3)=O)OCCCC1C2(F)F Cc1cc(OCc2scc(Br)c2Br)nc2cc(Cl)ccc12 N1(C(Cc2c(C)cccc2)=O)CCC(CNC(=O)C(C)(C)N2CCCC2)C1(C)C C=CCCC(C(=O)OCCOC1CCCCC1C)c1ccccc1 N1(C(C=C(CC)CC)=O)CCC(C)C(C)C1.c1(C(=O)N)c(C(F)(F)F)noc1C N=c1[nH]c2c(C(=O)NC3CCCC(NC(C4C=CCCC4)=O)C3)cccc2o1 c1(C(=O)NC(C2CCN(C(c3cccnc3)=O)CC2)C)ccc(N2CCC2)nc1 c1(NCC(C(C(C)C)O)(C)C)ccc(S(=O)(=O)N2CCc3nn(C)cc3C2)cc1Cl c1(C(N2C3C(N(C(=O)CCC4(C)CC4)C)CC(C3)C2)=O)cccc2[nH]c(=N)oc12 CCCC(C(=O)NCC12CC1CN(C(c1ccc3cnoc3c1)=O)C2)S(N)(=O)=O N1(C(C(C)OCCCC)=O)CC2CCN(C(c3coc(C(F)(F)F)n3)=O)CC2C1 Cc1cncc(C(N2CCOCC2CNC(=O)CCC(N)=O)=O)n1 N1(C(CCCC=C)=O)CCC(C)C(NC(=O)Cc2c(CC)nn(C)c2CC)C1 Cc1sc(C)c(C(=O)NCC2CCCC2)c1C#N.C1(C=O)CC12CC(C)(C)C2 C1(C(N2CC(CO)C(C(F)(F)F)C2)=O)CC2CCC1N(C(c1csnn1)=O)C2 C1(NC(c2c(N)cncc2)=O)CC2CCC1N(C(C1CN(CC(F)(F)F)C1)=O)C2 c1(NC2CC(CC)(CC)NC2)cc(Cl)cc(C)c1OC N1(C(C)=O)CCN(C(C2C=CCN(C(C3CCC(=O)N3C)=O)C2)=O)CC1 N1(C(C2C=CCN(C(=O)CCC3CCOC3)C2)=O)CCn2nccc21 c1(CC(=O)NCCC(O)C(=O)NC(c2cscn2)CO)ccc(O)cc1 N1(C(c2cnc(C)n2C)=O)CC(NC(C2CCC(=O)N2)=O)C(S(C)(=O)=O)C1 Cc1cccc(C(=O)N(CC(O)CNC(=O)CCC(N)=O)C)c1Br Cc1c(C(=O)NCC(C2CC2)NC(c2[nH]cnc2C#N)=O)ccc(F)c1F C1(NC(Nc2cccc(Cl)c2)=S)CCCOC12CCC2 C1(C(=O)NCC2CCN(C(C3CC(C#C)(O)C3)=O)C2)CC2(CCOC2)C1 CCCCC(CC)C(=O)NCCCC(C)NC(c1nnn(COCC)c1N)=O c1(CC)ccc(C(N2CCC(NC(c3ccc(Cl)c(O)c3)=O)C(F)C2)=O)cc1Br C1(C(=O)NCC2COC2)COC2(CCN(C(C3CCSCC3)=O)CC2)C1 N1(C(C2(C(N)=O)CC2)=O)CCCCC(C2CN(c3ncc([N+](=O)[O-])cn3)C2)C1 CC1(C)CCC(CO)N(C(C2CN(C(c3cc(C(N)=O)co3)=O)CC2(F)F)=O)C1 c1(OC)ccnc(C(=O)NC(CNC(=O)CCC(C)(F)F)C(C)(C)C)c1F C(N=c1cccc(S(=O)(=O)N2CCC(CS(C)(=O)=O)C2)[nH]1)c1cnc(C)s1 c1(C(=O)N)cc(F)cc2c1CCC2.N1(CC)CCCC1C(N1CC(O)(CC)C1)=O C1(O)(CN(C(=O)CC(F)(F)Cl)C)CCN(C(C2CC2C2CC2)=O)CC1 c1(C(N(CCCC(=O)N2CCOCC2)C(C(=O)NCC)=O)C)ccccc1OC CCCC(CCC)CC(=O)N1CCN(c2ccc(C(=O)OC)cn2)CC(C)(F)C1 CCC(C)(COC)C(=O)NCCC1CN(C(C2CCCC2)=O)CC1C.N(C)C.C c1nnc(S)n1C.N1(C(C)C(=O)N2CCC2CNC(=O)CO)CCNC1=O.C c1(CC(=O)NC2CCN(C(C(CC(=C)C)C)=O)C2C2CC2)cn2c(C)csc2n1 CC1(C(=O)NCC2CC(NC(=O)CCOC3CCOC3)C2)C=CCC1 N1(C(CNC(NCC)=S)=O)CCCC2(CCN(C(c3ccc(F)cc3)=O)CC2)C1 C1(CC)COCCN1C(c1c[nH]nc1C1CC1)=O.C1(C=O)C2CC3C(C2)C13.N C1(C(=O)NCCCCC2CN(C(c3c(C)occ3)=O)C2)CC1C1CCCCC1 N1(C(CCc2c(OC)cccc2)=O)CC2(CC(NC(c3cc(C#N)on3)=O)C2)C1 c1(CSCC(=O)NCCCC)nccn1C.c1(C=O)cc(C(C)(F)F)on1 c1(C(N2CCCC(C(=O)OCC)C2)C(=O)NCC2CCOC2)cc(C)ccc1C N1(C(CCCOC)=O)CCC(=CCNC(=O)COc2ccsn2)CC1 N1(C(C(C)SCC)=O)CC2C(C)C2C1.c1(C=O)nc(C)[nH]c1C(F)(F)F c1(C(N(C(C)CC)C)=O)cc(C(N)=O)c[nH]1.C1(C=O)CC1C(F)(F)F Cc1cc(CC(=O)NCC2(NC(C3CCCOCC3)=O)CCOCC2)ccc1F c1(C(=O)NC2C(OC)(OC)CCCC2)ccccc1S(C)=O CC1(F)CCCN(C(C23CC(CN(C(=O)C(O)C(F)(F)F)C2)C3)=O)C1 C1(c2scc(C(=O)OC)n2)CCCN(C(=O)N(c2ccccc2)CC(N)=O)C1 c1(CNC(C2CCOC2)=O)nc2ncnc(N3CCCC3C3CCC3)c2s1 C1(C(N2CC(C#C)C(O)C2)=O)CN(C(C2CCN(CC)CC2)=O)CCC1(C)C CS(=O)(=O)C1CC(NC(=O)Cc2csc(NC(=O)Cc3cc[nH]n3)n2)C1 CC1CCN(C(=O)CNC(=O)O)CC1CC=O.c1cccc(Cl)c1.C(C)(C)C C(=O)(C(CC(C)C)N(C)C)N1CC(O)(C(C)NC(CCSCC)=O)C1 Cc1cc(Cl)cc(C(=O)NC23CC2CN(C(=O)CC2(C)CCCO2)C3)c1O N1(C(C=CCCC(C)C)=O)CCn2ncc(CNC(=O)CCc3ccoc3)c2C1 N(C(=NCC=C)NCC(c1ccncc1)O)C(C#C)CC1CC1 C(CC(C)C)(C(=O)NCCCC(O)C(=O)NC1(CC(C)(C)C)CC1)OC n1(CC=C)nnnc1C.C1(C)(CC)CCOC1.CC(C(=O)N1CCC1)=C1CCOC1.N CCCC(C)CCCC(=O)NCCC1(OC)CN(C(=O)COCCF)C1 c1(OC)cccc(C(N2CCC(CNC(=O)C(C)Sc3ccccc3)C2)=O)c1C N1(C(CCOC(C)C)=O)CCC(NC(C2(O)CCOC2)=O)C(CO)C1 C(=O)(C1=Cc2ccccc2C1)N1CCOCC1.C1(C(N(C)C)=O)(C(=O)NC)CC1 C(=O)(CC(F)(F)C(F)F)N1CC(C)C(NC(=O)Cc2ccccc2[N+](=O)[O-])CC1 N1(C(COC2(C)CCCC2)=O)CCCC12CCN(C(=O)CCc1csc(=N)[nH]1)C2 C(CC)(C(=O)Nc1ccccc1)N(C(CONC(CCOC)=O)=O)C N1(C(c2cc(CC)on2)=O)CCCC1(C)CNC(C1(O)CCOCC1)=O C1(C(=O)OCCCCC)(CNC(c2cc(OCC(C)C)cs2)=O)CCOCC1 CCC(CC)C(=O)N1CCOCC1CNC(=O)Cc1cccc(C(F)(F)F)n1.C C(c1cccc(O)c1)=CC(N1CCC(C(C)NC(c2c(C)occ2)=O)CC1)=O C(C(C)(C(=O)N1CCC(C(C)C)CC1)NC(=O)CCc1ccccc1)SC c1(CNC(c2c(CCC)[nH]cc2)=O)ccc(C(N2C(CO)CC2C)=O)nc1 C1(NC(=O)CC2CC3CC3C2)CN(C(=O)CSc2cccs2)C2(CCCCC2)C1 c1(NCC2(C)CCCOC2)nc2ccc(O)cc2s1 CN=c1[nH]cc(C(N2CCC(CCC(=O)NC3CC=CCC3)CC2)=O)o1 C12(NC(CC3N(C)CCC3)=O)CC1CN(C(=O)CC1CCCCO1)C2 c1(CC(=O)NC2CCC(CNC(c3cn[nH]c3)=O)C2)cccc(Br)c1F c1(C(N2CCOCC(NC(Cc3c(C)nn(C)c3)=O)C2)=O)ncnc2ccsc12 C1(C(N2CC3C(N(C)C(C4CC(C)(C)C4)=O)C3C2)=O)CCc2nnc(O)n2C1 C1(NC(CCN(C(C)=O)C)=O)CC2CCC1CC2NC(C1(F)C2CCCCC12)=O c1(OC)nc(N2CCC(C#N)(NC(=O)CC(C)c3ccccc3)C2)ncc1Br N1(C(c2n(C(C)C)ncc2)=O)CC2CC(NC(C3CC(N=[N+]=[N-])C3)=O)CC2C1 Cc1cccc(Cl)c1NC(=O)C(c1ccc(Cl)c(Cl)c1)(C)C C1(O)(CC)CCN(Cc2cc(C(F)(F)F)ccn2)C1.C(=O)CN(C)C1CC1 C1(O)(CC#C)CC(C(=O)N(C2CCC(NC(=O)CCc3cc[nH]n3)C2)C)C1 c1(C(COC)=O)c(C)[nH]c(C(C)OC)c1C.C12CN(CCO1)C(=O)C=CC2 C1(C)(NC(C(OC)OC)=O)CC(C(=O)N(CC(=O)NC(C)C)C)C1 C1(C(=O)NCCN(C(=O)Cn2ncnn2)CC)CCCCN1C1CCCC1 C1(CC(=O)NCC(c2ncc[nH]2)C)(NC(C2CCCS2)=O)CCCC1 N1(Cc2c(C)nc[nH]2)CCC(NC(=O)C(=O)NC(C)CC2CCCO2)CC1 C1(OCC)CN(C(c2cccc(OC(c3ccc(C#N)cc3)=O)c2)=O)CCC1=O C=CC(C)C(C)C(=O)NCCN(C(c1ccc(NC(=O)CC)cc1)=O)CC O=C(CC(CNC(=O)C(c1cccnc1)O)C1CCC1)NCC(F)Cl C1(NC(c2c(C)ccs2)=O)CCC2CCN(C(c3cnc(S)n3C)=O)C1C2 c1(C(N2C3CC(C3)C2)=O)cc2c(s1)CCCC2.CCC(C)C(C(=O)N)NC(N)=O N1(C(C(=O)Nc2cnn(COc3ccc(Cl)cc3)c2)=O)CCNCCC12CC2 c1(C(N(C(C)Cc2nn[nH]n2)C)=O)cc(Br)ccc1O C1(NC(c2nc(C(C)C)n(-c3ccccc3F)n2)=O)CC12CCc1ccccc12 C1(CC(=O)NCCC(COC)OC)CN(C(=O)Cc2cc(C)no2)CCO1 N1(C(CC(CNC(COc2ccn(C)n2)=O)O)=O)CCC2CCCC2CC1 Cc1cc(C)c(NC(=S)NC(c2ccco2)C)c(C)c1 C(CC(C)C(=O)N1CC(O)(CNC(C2CC(F)(F)C2)=O)C1)=CC c1(N2CC(CF)OCC2)nc(N2CCC(c3ccccc3Br)C2)c2[nH]ccc2n1 C(=O)C(O)(CN(C)C)C(F)(F)F.C(=O)(CC(=O)NC1CC1)NCC#C C1(C(=O)NCC(C)CC2CCCC2)CCN(C(C2(CO)CCOC2)=O)CC1 C1(NC(C(C2CCOC2)NC(CCCC2C(C)C2)=O)=O)CC2(CCCCC2)C1 C1(C(=O)NC2CC(C(=O)Nc3c(C)scc3)C2)COCCN1C C1(OC)CCC(C(N2CC(O)CC2C(=O)Nc2cnn(C)c2C)=O)CC1 c1(CCC)ccccc1C(N1CC(N(C(=O)C(C2CC2)SC)C)C1)=O C(=O)(CCS(C)(=O)=O)NC1CN(C(c2c(SC)nn[nH]2)=O)CC1C(F)F C(=O)(C1=COCCC1)NCCC(C)(CC)NC(c1c(CC)n(C)nc1)=O CCCC(CCC)C(=O)N1CC2C(CNC(C34CCOC3CCOC4)=O)C2C1 c1(OC)ccc(CNc2ncnc(N3CC4CCC4(C)C3)c2C)c(C#N)c1 C1(NC(CN(CCC#C)C)=O)CN(C(=O)C(C)(C)F)CCC1c1cccc(F)c1 c1(C(N(C)CC2CN(C(=O)CC3COCCO3)C2)=O)cnccc1Cl C1(C(CNC(CCSCC)=O)F)CCN(C(C2CCCC23CC3)=O)CC1 C1(O)(CC(=O)NCC(CNC(c2c(C(C)C)con2)=O)C)CCCN(C)C1 C(=O)(C(C)(C)C(=O)NCc1cc[nH]c1C=O)NC.C1(O)CCCC1(C)C.N C1(NC(C2(C(C)C)CC2)=O)CCC2(CC1)CN(C(C1C(C)OC(C)C1C)=O)C2 C1(C)(C(N(CCCCN(C(=O)C(C)(C)CO)C)C)=O)CCC(=O)C1 c1(CCN=C(NC2C(C)CCCC2)NCC2(Cl)CCCC2)ccc2c(c1)OCO2 N1(C(CN(C2CCCC2)C)=O)CC2(CC(C(=O)NCc3cnn(C)c3)CO2)C1 CCC(C)CNC(=O)CSc1ncc[nH]1.c1(C(=O)N)cnc(C2CCCO2)s1 c1(C(=O)NC2C(NC(C3OCC(C)(C)C3)=O)COC2)cccc2c1OCC(=O)N2 C(C(C)(CNC(=O)C(=O)NCC(F)F)OC)NC(CC1C(CC)C1)=O c1(OC)ccc2c(C(=O)O)cnn2c1.c12ccccc1-c1nc(no1)C(=O)N2 C(=O)(CC(C)CC(C)C)N.Cc1c(CNC(=O)Cn2cc(C)nn2)cccc1F N1(C(C)C(=O)Nc2cc(F)c(Cl)cc2I)c2ccccc2CC1C N1(C(C(CSC)OC)=O)CCC2(CC1)CCN(C(=O)CN(c1ccccc1)C)C2 c1(C(=O)NCC2C(NC(c3cccc(C#C)c3)=O)C2)ccc(F)c(Cl)c1F c1(N(C)Cc2ccc(Br)cc2)nc(NCc2nccc(=N)[nH]2)c2ccsc2n1 N1(C(c2c(C)n(CC(F)F)nc2)=O)CCCC(NC(C2(C)CCCS2)=O)CC1 c1(C(c2n(CC)nnn2)NC2CC(C)(OCC)C2(C)C)ccc(F)cc1F.O CN1CCC(C(=O)NCC2CCN2C(C2CN(S(N)(=O)=O)C2)=O)CC1=O N1(C(C(C(C)C)O)=O)CC(CN(C(=O)CC2CN(C)C2)C)C2(CC2)C1 N1(C(C=CCC)=O)CCCC12CCOC2.C1(C(=O)N)CCCN1C(=O)C(C)(C)C c1(C(=O)NC2C3CN(C(C(C=C)(C)CC)=O)C2CC3)cc(C#N)ccc1F C(=O)(C(CCF)NC(=O)CC1CCCC1O)NCC(C)(F)F c1(NC(C2CC(F)(F)CN2C(c2cc(Cl)ccc2I)=O)=O)cc(F)cc(F)c1F CC(C(=O)N1CCCC(F)(C(=O)Nc2cncc(C3CC3)c2)C1)S(N)(=O)=O C1(NC(C(CNC(C2C(C)OCCO2)=O)CC2CCCC2)=O)CC2CC(O)C1C2 c1(COCCOCC)nc(-c2ncccc2)nn1-c1cnc(C)s1.C1CC1.O C1(C(=O)NCCOC(CNC(C2ON=C(C)C2C)=O)(C)C)CCCCCCC1 C1(SC(C)(C)C)CCCN(c2nnc(C(C)(C)C)s2)C1 N1(C(c2c(C)sc(O)n2)=O)CCCC2CCN(C(=O)CC3CCC(=O)N3)CC12 Cc1c(C(N2CCC(F)(C(=O)NCC3CC(C#N)C3)CC2)=O)c[nH]c1C#N c1(CC(=O)NC2CCCN(C(=O)C(O)C3CC3)CC2)ccc2nsnc2c1 c1(N2CCC(COc3ccc(C)cn3)CC2)ncc(F)c(=N)[nH]1 c1(C(C)C(N2CC(F)CC2CNC(C2(O)CCCCC2)=O)=O)c(F)cccc1F O=C1CN(C(=O)C=Cc2cc[nH]n2)C(C(=O)NCCOCC(F)(F)F)CN1 Cc1ccc(C=CC(=O)NCc2nc(CNC(=O)CNC=O)cs2)o1 C1(C(=O)NC(CC=C)CC(F)F)CCN(C(c2cc(CCC)on2)=O)C(C)(C)C1 Cc1ccc2cc(C(=O)NCC(C)NC(c3cccc(Cl)c3)=O)[nH]c2c1 c1(C(=O)NC2CN(Cc3c(OC)cc(F)cc3)CC2C#N)ccc(F)c(Cl)c1F Cc1cccc2sc(C(=O)NCC(C)NC(=O)Cn3cc(C#N)cn3)c(Cl)c12 N1(C(C2CC3CCC2N3C(=O)C(C2CCCCC2)O)=O)CCN2CCCCC2C1 C(=O)(CC(C)C(F)(F)C(F)(F)F)N1CC(CNC(CC2CC(=C)C2)=O)OCCC1 C12(NC(Cc3nc(C)[nH]n3)=O)CCOCC1CN(C(=O)C(C)(O)C(C)C)C2 N#Cc1ccc(C(N2CC(C(=O)Nc3csc(Br)c3)C2)=O)c(Br)c1 C1(CNC(c2cc(C)ns2)=O)CC12CCN(C(c1nnsc1C)=O)CC2 c1(CC(N2CCC(NC(C3N(C(C)=O)CCC3)=O)CC2)=O)ncnc2sccc12 c1(-c2cn(C(CC(=O)C(CCN3C(C)CCC3)=O)(C)C)nn2)cn2cccnc2n1 CS(=O)(=NC(=O)C1CCS1(=O)=O)c1cnn2c1CN(C(=O)CN1CCC1)CC2 c1(C(=O)NCCCN(C(C2CCCO2)=O)CC)cnc2cc(OC)ccn12 c1(C(=O)NC2(C(=O)NC3CC(CSC)C3)CCSC2)ccc(C)nc1 N1(C(CCC)=O)CCCCC1C(=O)NC1(C)CN(C(c2n[nH]c(C3CC3)n2)=O)C1 CC(C(=O)N1CCC1CNC(C1CC1(c1ccccc1)C)=O)C(C)(C)C c1(CC(N2CC3(CN(C(C(C(C)(C)O)F)=O)C3)C2)=O)c[nH]c2ncccc12 C1(N(C(CCCN(C(C)C)C)=O)C)CCCN(C(c2cnc(S)nc2)=O)C1 C1(NC(C(CC)NC(N)=O)=O)C=CCN(C(=O)COc2ccccc2C)C1 CC1CN(C(=O)CCc2cc(Br)sc2Br)CCCO1 c1(C(=O)NCC2C(C)CCN2C(C2CCCC(C)(C)C2)=O)cn2cnnc2cn1 C1(NC(C(CC)NC(C)=O)=O)COC2(C1)CN(Cc1nnc(C(F)F)s1)C2 N1(C(C2(CC#C)CCCC2)=O)CCCC(C)(CNC(=O)CC2CSCCS2)C1 C1(C(=O)NC2CC(NC(CC=C=C)=O)C2)C2CC3CC(C2)CC1C3 Cc1c(C(=O)NC2CCN(C(=O)CC(C)P(C)(C)=O)C2(C)C)ccc2cncn12 c1(-n2c(C(N3CC(C(Cn4cc(C(C)O)nn4)F)C3)=O)ccn2)ccc(Br)cc1 CC1c2ccccc2OC1C(=O)NC(C)(C)CNC(c1c[nH]c(=O)cn1)=O N1(C(C2(C)CCCO2)=O)CC2CCCC(C1)N2C(c1ccc(Cl)nc1Cl)=O C(CCCCCNC(=O)C(O)Cc1ccccn1)NC(C(C)C1CCCC1)=O C1(CC(=O)N(CC(C)O)CC)CCCC(F)(F)C1.C1(CC=O)CC1.CS.C CCCC(CCC)CC(=O)N(CCC(=O)NOCCCCCC1CC1)C N1(C(c2c(C)onc2)=O)CC2(CCCC2NC(c2cc3scnc3[nH]2)=O)C1 c1(C(=O)NC2(C3CC3)CCN(C(c3nc(C)[nH]n3)=O)C2)cc([N+](=O)[O-])ccc1C c1(OC(C)C(=O)NCCCC2CCCN2C(=O)C=CCF)ccccc1Br C1(C(=O)NC2CC(F)(CNC(c3c(C)csc3)=O)C2)CC12CCOCC2 c1(C(=O)NCC(C)C)cccn(CC(F)(F)F)c1=O.C1(C(=O)N)CCC1(C)C CCCCCCCCC(=O)NC(CNC(=O)Cc1ccc(O)cn1)CO C(=O)(C(CCC=C)NC(=O)C(C)SC(C)C)NCC(C#C)(C)C Cc1oncc1C(=O)NC(C)C(=O)NC1CC1.C1(CC=O)C=CCCC1.C C1(CC=O)CCCCC1.C1(C=O)CC1(C)C(F)F.C(=O)(COCC)NC CCCC(C)(O)C(=O)NCC1(NC(=O)Cc2ccno2)CC1 N1(C(C(C)(O)c2ccccc2)=O)CC2(NC(c3snc(O)c3Cl)=O)CC1C2 N1(C(C(C)SCC)=O)CCOC2(C1)CN(C(c1ncc(Br)cc1N)=O)C2 c1(NC(C2CCCC(NCc3cc(Br)ccc3I)C2)=O)cccc([N+](=O)[O-])c1Br C1(NC(C2C(C(C)(F)F)C2)=O)CCCCN(C(=O)CCC2CCC(O)CC2)C1 C1(C(N2CCC(=C)CC2)=O)CCN(C(c2cnc(Cl)n2C)=O)C1(C)C C1(C(=O)NC(CC)CNC(=O)CCc2ccc(N)c(F)c2)CCc2cncn2C1 N1(Cc2c(CC)cccc2C)CCC(NC(=O)OC(C)(C)C)CC12CCC2 C(=O)(CCCC(C)(C)CC)N1CC(CC)C(C(=O)Nc2c(COC)cccc2F)C1 C1(NC(C2(COC(C)C)CC2)=O)CCCCC1.c1(C=O)nc(=N)cc[nH]1.N c1(-c2n(C(C)Cc3cc(=O)cc(CO)[nH]3)ccn2)c(-c2ccns2)ccnc1O c1(C(N2CCCC(NC(=O)C(F)(F)C3CC3)C2)=O)ccc(-c2cc[nH]n2)cc1 N1(C(C(C)Sc2cccs2)=O)CCC(OCCNC(=O)C)CC1.C(N)=O.N C(C(=O)Nc1c(C)cccc1C)(C1=CCCCC1)N1CCN(CC)CC1 C1(NC(C=CCCC)=O)CCC12CCN(C(C1(C)CCNC1=O)=O)CC2 N1(C(COCc2cc(C)on2)=O)CCC2CCN(C(c3occc3C)=O)CC2C1 Cc1cc(Cl)ccc1CC(N1CCC(O)(C)C1)=O.c1(C(=O)N)cnoc1C1CC1 n1(CC(N2CC(OC)CC2)=O)nc2n(c1=O)CCOC2.C(=O)C(F)(F)C(F)F.N C1(NC(CCCC)=O)CN(C(=O)CCCCC2CC2)CC(C)(C)C1 c1(N2C(c3scc(C)n3)CCC2)nnc(C2CCC(=O)N2)n1CCC(=O)N(C)C Cc1nn(C)c(Cl)c1C=CC(=O)N(C)CC1CCN(C(C2CCC(O)CC2)=O)C1 C(=O)(C#CC(C)(C)C)N1CCC(C(C(=O)NCCCCCCC)C)CC1 C1(CNC(CSCC(C)=O)=O)CC2CCC1N(C(C1CCCCC1(F)F)=O)C2 C1(NC(N(C2CCC(SC)C2)C)=O)CCC(c2ccc(F)cc2)CC1 C(C(CC(C)C)NC(=O)Cn1cnnc1)NC(C1N=C(C)SC1)=O Cc1cnc(C(=O)NC2CN(C(=O)C(C)Cc3ccccc3C)C2)cc1Cl C(=O)(CCCCCN=[N+]=[N-])NC(C(=O)NCC(CCOC)O)CCSC c1(C(C(=O)NC)N(C2CC2)C(c2ccccc2Cl)C)ccnc(S(C)(=O)=O)c1 C1(O)(CC(=O)NCCOCCCC)CN(C(C2CCO2)=O)C1 CCC(C(=O)OC)C(=O)N1CCN(CCCNC(C2CCCS2)=O)CC1 CC1CCCN(C(=O)CC23CCC(CC2)CC3)C1CNC(=O)CCC1CCOC1 N1(C(C(C)NC(=O)NC)=O)CCC2(C1)CN(C(=O)C(N1CCC(O)CC1)C)C2 c1(NC(=O)NC2CCC(C#C)C2)cc(OCC(C)C)c(Br)cn1 C1(NC(c2c(C)nco2)=O)(C)CCCCC1.c1(C=O)ccnc(C(C)(C)C)c1.N CC1(C)CCC(C)(C(N2C3CCC(C3)C2C)=O)CC1.n1(CC(=O)N)cnnc1 Cc1ccc(C(=O)NC(C)(CNC(c2cnn[nH]2)=O)CC(C)C)cc1Br Cc1cnc(NC2CN(C)NC2=O)c2ccc([N+](=O)[O-])cc12 C1(C(=O)NCc2c(C(=O)NC(c3cnc[nH]3)C)scc2)CC2(CCC2)C1 C1(C(N2CCC(c3ccon3)C2)=O)(SC)CN(C(=O)CCC2CC2(C)C)C1 c1(NC2(CNC(C(CCC)C)=O)CCCCC2C)ncnc2sccc12 c1(OC)ccc2c(c1)CCC2C(=O)N1CC2=C(C1)CN(C(C1CCC(O)C1)=O)C2 CCCCCCC(=O)N1CCCC(C(N2CC3CCC2(CO)C3)=O)CC1 C1(C(=O)NC(C(C)(F)F)c2ccccc2)CC=CC(N)C1 c1(C=O)ccc(O)c([N+](=O)[O-])c1.C1(NC(=O)OC(C)(C)C)CC12CCC2.N CCCCCC(CC)C(=O)N1CCN(C(c2cnoc2C)=O)C2(CC2)C1 c1(-c2cn(CC(C)C)nc2)cccc2cc(C(=O)Nc3cc(Cl)ccc3F)sc12 Cc1ccc(CN2CCC(CNC(=O)CO)C2)c(O)c1.c1ccc(Cl)c(C)c1 c1(C2CC2)ccc(C)cc1.N12CCC(CC1)N(C)C(=O)CC2.C(=O)(CO)OC c1(C(N2C(C(=O)NCC(c3ccsc3)C)CC3(CC3)C2)=O)cn2ccccc2n1 N1(C(c2[nH]ccc(=N)n2)=O)CCCCCCC1C(=O)N(C1CCC1)C1CCC1 Cc1cc(NC(C2CC(NC(=O)Cn3nnnc3C)CCO2)=O)c(O)cc1F N1(C(C(COC(C)=O)C)=O)CCC(O)(C)CC1.C1(C(=O)N)(N(C)C)CCC1 C(=O)(C#CC(OCC)OC)N1CCC(N(C(c2c(CCC)nco2)=O)C)C1 Cn1[nH]c(=N)cc1NC(C1(CCC)CCCC1)=O.C1(CC=O)CC(=O)NC1=O CCCCCC(O)CC(=O)N1CC(OC)CC(NC(c2cnc(C(C)C)s2)=O)C1 CCCC(CCC)CC(=O)N(C)CCOCCCN(C(=O)CN1CCOC1=O)C CCCS(=O)(=O)C(C)C(=O)NC1CC1NC(C1(C(=O)O)COC1)=O.C N1(C(C2CC2(Cl)Cl)=O)CC2(C1)CN(CCn1cc(C(c3ccccc3)O)nn1)C2 C(=O)(C(F)C(C)(C)O)N1CCC(N2CCC(Nc3ccnc(C)n3)CC2)C1 c1(CN(C2CC2)CC)nnc(Sc2ccc(Cl)cc2)n1CC1CCCO1 c1(OC)ncc(Cl)c(C(N2CC(CNC(=O)CCCN=[N+]=[N-])(OC)C2)=O)c1Cl CCC(CC(=O)NCC1(C(N)=O)CCCC1)N(C(=O)COC)C CC1(C)C2CCC1(C(N1CCC(C)C1)=O)CC2.c1(C(=O)N)cc(C(N)=O)c[nH]1 C(=O)(CC(C)(C)CC=C)NC(C(=O)NC(C#C)CC1CCC1)C(C)C N1(CC(=O)N(C2CN(C(c3cocn3)=O)CC2O)C)C(=O)c2ccccc2C1=O c1(C(CC(=O)NCCN(C(C2CC3CCC2C3)=O)CC)C)c(C)noc1C c1(CCC(=O)NC(C2CCN(C(=O)Cc3cn[nH]c3)C2)C)nncn1C CC1(C)CCC=C(C(=O)NC2CCN(C(c3cc(F)c(F)c(N)c3Cl)=O)C2)C1 C(C(=O)NCCS(N)(=O)=O)(C(C)(C)C)NC(CCSCC)=O C1(CNC(CCn2cc(CCC(C)=O)nn2)=O)CC2CCCC2N1C c1(NC(CCOC)=O)cccc(NC2CCCN(CCC(=O)NCC)C2)c1 C(CC(C)C)(C(=O)N1CC(CO)C2(CC2)C1)NC(C(C1CC1)SC)=O N1(C(C(COCC)C)=O)CCC2CCCC12C(=O)NCCC1(C)CCOC1 C1(O)(CNC(C(C)OCCC#C)=O)CN(C(=O)Cc2cccs2)C1 c1(C(=O)N(C2CCC2)Cc2ccccn2)cc2c(Br)cccc2o1 N(C1CCCCc2ccccc21)C(C1CCN(C(c2ccc(Cl)cc2)=O)CC1)=O Cc1cc(N(C(C)CNC(c2c[nH]nc2-c2ccsc2)=O)C)c(C#N)cn1 c1(C(=O)NC2(C)CN(C(CS(CC)=O)=O)C2)cn(C)c2ccc(Cl)cc12 c1(C(=O)NC(C(=O)O)C2CCCO2)cc[nH]c2nccc1-2 C(=O)(C1=CCCOC1)NC1C(C)(C)C(CC(=O)NCCCP(C)(C)=O)C1 c1(OCC)ccc(C(N2CCC(CNC(=O)CCOCC)C2)=O)cn1.O Cn1ccc(=O)c(C(=O)NCC2CN(C(C3CC3c3cnc[nH]3)=O)CCO2)c1 C(=O)(CCC(F)(F)F)NCC1CCCN(CCC)C1 c1(C(N(C(C)C)CC)=O)cccc(C2CCCOC2)c1.C(=O)(CC1CCC1)N c1(C(N2CCOCC2(C)C(=O)OC)C(=O)NC(C(=O)OC)C)ccc(F)cc1Br c1(C(N2CCCC(NC(c3[nH]nc(OC)c3Cl)=O)CC2)=O)n[nH]c2c1CCOC2 N1(C(CCCC(C)NC(C(CCCCC)F)=O)=O)CC2C3C=CC(C3)C2C1 CC1(C(=O)NCc2ccnc(O)c2)CCN(C(=O)CC2CSC2)C1 N(C1CSc2ccccc21)C(N(CCCF)C)=O N1(C(C2CCC3CC23)=O)CC2CCC(NC(C3(c4cccs4)CCCC3)=O)CC2C1 C(=O)(CCN=C(NCC(Cc1ccoc1)CO)N1CCC(C)(C(N)=O)C1)NC C1(O)CCN(C(C23CSCC2C3(F)F)=O)CC1.CC12CC(CC(=O)N)(CO1)C2.C C1(CC(=O)N(C(C)CNC(c2c(Br)nnn2C)=O)CC)CCC(=O)C1C CC1CC(N=c2ccnc(N(CCCNC(=O)OC(C)(C)C)C)[nH]2)c2ncnn21 C12(NC(=O)C3=CCOC3)CCCCCC1N(C(=O)Cc1cc(Cl)ccc1O)CC2 Cc1ncc(NC(=O)CC(C(C)C)NC(C2(C)CC3C=CC2C3)=O)cc1C#N C1(CC(C)(C)C)CN(C(c2cccnn2)=O)CC1NC(c1cccc(F)c1)=O c1(C(=O)NCCCCC)cccc(C(F)(F)F)c1F.C1(C=O)C2CCC(=O)C12.N C(CC(N=c1[nH]c(C(=O)OC)c(C)s1)c1ccc(C)o1)OC C1(CSCc2n(-c3ccc(C)cc3)nnn2)CC2OC1C1CC21 N1(C(C2N(C(C3CC(SC)C3)=O)CC=C2)=O)CC2COCC2(CO)C1 C(=O)(C(C)CC(C)(F)F)NCCC(C)(C)NC(c1cc(CC)cc(F)c1)=O C(CCCCCCNC(=O)COCCCC(C)C)NC(C=CCOC)=O CC1C=C(C(=O)NC2CN(C(c3cnsn3)=O)CC2c2ccccc2F)CC1 Cc1nocc1C(=O)NCC=CCNC(=O)CNC(C1CCC1)=O c1(OC)cnc(NC2C=CCN2C(c2ccccc2)=O)nc1.C(=O)(N(C)C)O C1(C(N2CC3C(NC(CCC=CC)=O)CC(C3)C2)=O)Cc2cc(C)c(C)cc2O1 Cc1cc(CC(=O)NC(C)CCCNC(c2nc(O)c(C)s2)=O)cc(O)n1 Cc1cc2[nH]c(C(=O)NCC(O)CN(C)C(C3CCC3(C)C)=O)cc2s1 c1(C=O)cnccc1C(C)(C)C.C1(C(N(CC)CC)=O)CN(C)CCO1.CO Cc1cncc(CC(=O)NCC2CCN2C(=O)CCc2cc(C)nn2C)c1 C(=O)(C1=NOC(CNC(=O)C(C)(C)C2CCCO2)C1)N(C1CCCC(O)C1)C CC(O)(CNC(c1cnn(CCO)c1)=O)CNC(C1SCCS1)=O CC1C(C(=O)N(CCCCNC(C2COCC2(C)C)=O)C)OC2CCCCC12 c1(C(=O)NC23C(CN(C(C4ON=C(CC)C4)=O)C2)C3)ccc2c(c1)nc(C)n2C c1(CCN(C)Cc2c(C)cc(Oc3ccc(F)cc3)cc2)c[nH]c2ccncc12 c1(C(N2CCN(C3CCN(C(C45CC(C4)C5)=O)CC3)CC2)=O)cc(O)cc(Cl)c1 C1(CCN(C(C2(CC=C)COC2)=O)C)CCN(C(=O)CCN2CCCCC2)CC1 c1(C(=O)Nc2c(NC(=O)Cc3cccc(Cl)n3)ccs2)cc2n(n1)CCCC2 N1(C(c2n(C)ccn2)=O)CCOCC(NC(=O)C(c2ccccc2F)O)C1 C(=O)(CC(CC)C(C)(C)C)NC1(C(N2C(CC)CC2)=O)CCSC1 N1(C(CCOC(C)C)=O)CCC(O)CC1C(=O)NCCCC1CCCCC1 C1(NC(c2cccc(OC)c2)=O)C2COCC1CN(C(=O)C(C)n1ccnc1)C2 Cc1c(Cl)ccc(C(N2CC3(C2)CN(C(=O)CN2CCC(C)(O)C2)C3)=O)c1O c1(CC)ccc(C(=O)NC2CC3(C2)CC3NC(=O)C(C#N)C(C)C)cc1C CC12CN(C(=O)CC(O)C3CC3)CC1(C)CN(C(C1(C(F)F)CCOCC1)=O)C2 C(CC(C)(C)NC(C1CC1F)=O)N(C)C(C12CC(c3ccccc3)(C1)C2)=O CCC(C)CC(C(=O)NCCC1CCN(C)C1=O)NC(=O)C(C)C(F)F c1(CC(=O)NC(CC(C)NC(C2(SC)CC2)=O)C)cnc2n1CCCC2C C1(NC(c2cn(C(C)(C)C)nn2)=O)CCN(C(c2cncc(Cl)c2Cl)=O)CC1F c1(NC(C2CC23CN(C(C2CCCS2)=O)C3)=O)ccc(Br)c(F)c1F C12(C(N(CC3N(C(C=C(CC)CC)=O)CCCC3)CC)=O)CCCC(C1)OC2 C#CC(C(C)(C)C)NC(=O)C(C1CCCO1)NC(=O)CCOCCO c1(C(=O)NC2(C)CCN(C(c3ccc(N)cc3F)=O)C2)cc2n(n1)CCNC2=O c1(C(c2n(CCSC)nnn2)NCCC(O)c2cccs2)cc2ncccc2o1 C(=O)(N=c1[nH][nH]cc1-c1cccnc1)N1C(C(=O)OCC)CSC1C C(C(F)(F)C(=O)N(C)CCN(C)C(c1ccc(C(N)=O)cn1)=O)N(C)C c1(C(=O)N)cnc([N+](=O)[O-])n1C.C(CCCC(=O)NCC1CC(C)CO1)N(C)C CC(C)(C)CC(O)CC(=O)NC1C=CC(C(=O)NCC2COCCO2)C1 CC1(C)COC(C(=O)NC2CN(C(c3ccc(CO)c(F)c3)=O)CC2O)CO1 C=CCC(CNC(C)(C(C)C)c1nnnn1CC1CC1)CC(C)C CC1(C)CCC12CN(C(C1C3CCC(C3)C1NC(C1CCCCC1(C)C)=O)=O)C2 C1(n2cc(CS(CC)(=O)=O)nn2)CCCN(C(c2cocc2Br)=O)C1 c1(C=O)cnc(O)c2c1NCCC2.CSC=CC(=O)NCCOCCOCC.N c1(C2(C(=O)NCCCNC(=O)C(O)Cc3cnc[nH]3)CCC2)c(F)cccc1Cl c1(C(=O)NC(CC(C)NC(c2cnccn2)=O)C)cnc(OCC(F)F)cn1 C1(CNC(CCOCC)=O)OCC2CCN(C(c3cc4sccc4s3)=O)CC12 C(CSCC)(C(=O)NC(CN(C)C)C(=O)NC)OC.C1CCN(C)C1.C CCCCCCC(=O)NCC(c1ccccc1)NC(c1cc(CC)cc(C)c1)=O C1CN(C(=O)CCC2CCOC2)C2(CCC2)C1.c1(C(=O)N)cc(F)cc(Cl)c1.C c1(CC)cccc(C(=O)NC2CC23CC(NC(=O)C(=O)N(C)C)C3)c1N N1(C(C2CCN(CC)C2)=O)CCC(N(C(=O)Cc2ccc(C)s2)CC)CC1 Cc1coc(C=CC(=O)NCC2CCCCN2C(=O)Cc2ncn(C)c2C)n1 C12(C)CCCN1S(=O)(=O)CC2.N(C)(S(N)(=O)=O)C(C)C=O.C12CC(C1)C2 Cc1cc(O)c(Cl)cc1C(=O)NCCCN(C(=O)CCC1CCC(=O)N1)C C#CCCCCC(=O)N(CCC)CCNC(=O)CC(c1ccc(O)cc1)C1CC1 C1(O)(NC(=O)NCCOC2CCS(=O)(=O)CC2)CC2CCC(C2)C1 C1(CNC(c2c(C)cnn2C)=O)CC2CCC1N(C(C1CC3CCC1CC3)=O)C2 N1(C(C23OC(C)(C)C(CO)(C2)C3)=O)CCC(N=c2[nH]c3cc(Br)ccc3o2)C1 C1(NC(CC(C)(C)OC)=O)CN(C(c2c[nH]nc2C2CCC2)=O)CCC1CO N1(C(c2cc(CC)on2)=O)CC(NC(c2ccsc2)=O)C2CC12 C12(C(=O)NC(C3CCOC3)C)CC1CN(C(c1cccc(CO)c1)=O)C2 CC1CCN(C(=O)C(C)NC(c2cccs2)=O)CCN1C(C1CC(C#N)C1)=O N1(c2cc(C(=O)OC)ncn2)CCC(NC(c2ccc(C)c(Cl)c2)=O)C12CCC2 O=C1NC(=O)C(CCNC(C2(NC(C3CC=CCC3)=O)CC2)=O)N1 C#CCCCC(C)C(=O)NCCCN1CCC(NC(=O)C(CC=C)N(C)C)C1 CCCC(O)(CCC)CC(=O)NCC(C)NC(=O)CC1(O)CCC1 C(=O)(C1=CC2(CCOC2)C1)NC1CC(C)(C(NOC(C(C)C)CO)=O)C1 CC(CC(=O)Nc1cccc(NC(=O)C(=CC2CCCCC2)F)c1)CC(F)(F)F N1(C(C(C)OCC)=O)CCC2CC12C(=O)N(CC)CC1CCCCC1 c1(C(NCC)=O)c(F)cc(OC(F)F)cc1F.C1(CCOC)(C=O)CC1.N c1(CNC(C(C2(C)CC2)NC(COC(CC)C)=O)=O)ncc(C)[nH]1 C(=O)(CCC(C)(F)F)N1C(CCC(=O)NCC(CCC)C)CCCC1 c1(-n2c(-c3c(C)cno3)nc(C(F)F)n2)cc(O)nc2ncccc12 O=C(CC1CN(C(c2ncccn2)=O)C1)N=c1cc[nH]cc1O Cc1csc(C(=O)NC2CC(F)(C)C2)c1C.C(=O)(CC)N.C1(C=O)CCC1 c1(C(C)C)cc(C(=O)NC)c(C(C)C)[nH]1.C1CCC1(C)C.c1(C=O)ccco1 C1(C(=O)NCCCCNC(c2nc(CCC)sc2)=O)CCCCC1OC C12(C(N(CC(CC)NC(C3(c4cccc(F)c4)CC3)=O)C)=O)CC1CNC2=O c1(C(CC(=O)N(C(C)C)C)C2CC2)ccc(C#N)cc1.C1(C=O)C2CCCC12.N C1(C(=O)NC2CC(O)(Cn3cc(C(CC)(C)C)nn3)C2)CCCN1N=O C12(C(=O)NCC(C)(C)N(C)C)COC(C1)C(NC(C1(C)COC1)=O)C2 C1(CC2CN(C(=O)NCCc3cn(CC)nc3)C2)CCCC(C)(C)C1 C(=O)(C(C)C(C)(C)C)NCC(C)NC(C(C)(c1ccccc1)OC)=O C1(CNC(=O)CCCC2CCOCC2)CCCN(C(C2C3CC4C(C3)C24)=O)CC1 Cc1nn(-c2ccccc2)[nH]c1=NC(=O)N1CC(F)CC1C#N Cc1cc(C(=O)NCC2CC(C)N(C(c3cnccn3)=O)C2)ccc1O C#Cc1cnc(C(=O)NC(C2CCCN(C(=O)C#CC3(CC)CC3)C2)C)c(C)c1 C(=O)(C(C(C)(C)C)NC(=O)C(C)N=[N+]=[N-])NCC1CCN(C(C)=O)CC1 C(=O)(CC(CC)CC(C)C)NC(CCC)CC(=O)NCCOCCN(C)C CCCC(C(=O)O)N1CCN(C(c2cccn2C)=O)CC1 c1(NC(C(=Cc2ccc(OC)c(F)c2)C)=O)cc(Br)c2c(c1)CCO2 C1(CNC(c2ccc(C3CCCN3)s2)=O)CCCN(CC(F)F)C1 N1(C(C=C(C)C(F)F)=O)CCC(C(C)C(=O)N(C)Cc2ccncc2)C1 CC1=NOC(C)(CNC(C2CCCCN2C(=O)C(n2ccnc2C)C)=O)C1 CCC(C)(COC)C(=O)NC1CCCCC1NC(c1cc(C)c(Cl)s1)=O c1(C(N(CC(C)CNC(C2(CCN(C)C)CC2)=O)C)=O)cc(Cl)ccc1F C(=O)(C(CNC(=O)CC1CSC1)C(C)(C)C)NCc1c(C)cccc1F CCCCC(F)C(=O)N1CCCC(NC(=O)C(C)C2CCCC2)C1CC C1(C(N2CC(N(C)C(c3cscc3F)=O)C2)=O)CCCCNC1=O C1(C(=O)NCC2CC(=O)NCC2)CCN(C(=O)c2ncncc2Cl)O1 c1(CN2CCN(CC(N3CCC(C#N)CC3)=O)C(=O)C2)cc(Cl)c(Cl)cc1F C1(C(=O)NC(C2CCN(C(=O)C3=CCSC3)CC2)C(C)C)C2C3CCC(C3)C12 N1(C(c2nc(C(C)NC(C(SC)SC)=O)oc2)=O)CCCCC1C1(O)CC1 C(=O)(C1=CS(=O)CCC1)Nc1cccc(NC(Cc2c(C)cc(C)s2)=O)c1 N#Cc1n[nH]c(=NCCC2CCCCN2C(=O)CCn2cnccc2=O)s1 C12(NC(CC3CCCN(C)C3)=O)CCCCC1CN(C(=O)CSS(C)(=O)=O)C2 CC1C(NC(=O)C(F)OC(F)(F)F)CC2CCC1N2c1nccc(CO)n1 c1(C(=O)NCCCC2N(C(C3=C(C)CCC3)=O)CCC2)nc2ncccn2n1 C1(NC(N(C2CCN(c3cccnn3)C2)CC)=O)CCP(C)(=O)CC1 c1(C(N2CCC(N(C(=O)Cc3cocn3)C)C2)=O)ccc(S(N)(=O)=O)cc1Cl C(c1ccc(Cl)c([N+](=O)[O-])c1)=CC(=O)N.C1(C=O)CCC(C)(C)OC1.CCC Cc1c(Cl)ccc2[nH]c(C(N3CCC(NC(=O)C=CC4CCOC4)CC3)=O)cc12 N1(C(C(c2cccnc2)C)=O)CCC(NC(c2cc3n(n2)CCO3)=O)C12CCC2 c1(CC(C)C)cccc(C(N2CCC(N(CCO)C(C3CCCO3)=O)C2)=O)c1 N(C(=NCCCN1CCCS1(=O)=O)NC1CC1)C(c1ccc(F)c(F)c1)C CC(F)(F)CC(=O)NCC1(NC(=O)CCC2CCCC2)CCOCC1 N1(C(c2nc(C)oc2C)=O)CC2CCN(C(=O)C(O)CF)CC2C1 c1(NC2CCC(=O)NCC2)ccc2ncccc2c1[N+](=O)[O-] C1(NC(C(n2cc(Cl)cn2)C)=O)CCN(C(C23CCCC(CO2)C3)=O)CC1F C(CC1CC1)(CC(=O)NCC(C)(Cl)CC)NC(CCCOCCC)=O CCCCCCC(C)C(=O)NCC1CCCC1NC(C1(C2CC2)CC1)=O CC(CNC(=O)CCC1CCCCO1)C(=O)N(C(C)CN(C)C)C C(c1cncc(O)c1)=CC(=O)NC1COCCC1NC(C1(C2CCC2)CC1)=O CC1OCCCC1C(=O)NCCn1cnc(C(=O)NC2CCC2)c1 C12(CNC(=O)C(O)CC3CCCCC3)COCCN1CCN(C(C1CC1F)=O)C2 c1(N(CCCCC(C)C)C)nc2c(c(=NC(C)CCC(F)(F)F)[nH]1)CC(C)CC2 C1(NC(C(C)=C2CCCC2)=O)(CF)CCN(C(C2(n3cncn3)CC2)=O)C1 N1(C(C(C)(C)NC(C)=O)=O)CCN(C(c2ccns2)=O)C(C(F)(F)F)C1 Cn1cncc1CC(=O)NCC(C)(C)OCC(=O)N(CC(F)F)CCO Cn1c(C(=O)NC2CC(C(=O)NOC3CCCCC3)C2)ccc1C#N C1(F)(C=O)CCS(=O)(=O)C1.CC1CCC1.c1(C=O)csc(C(F)(F)F)n1.N N1(C(COCC(C)C)=O)CC(NC(=O)CC2CCCC23CC3)CC2(CCC2)C1 c1(C(=O)Nc2ccc(O)cc2Cl)ccc2c(c1)CN(C(c1cnon1)=O)C2 C1(C(=O)NCCC2N(C(C=C(CCC)CCC)=O)CCSC2)CNC(=O)CC1C C1(C(=O)NCC=CCNC(C(CC(C)(C)C)O)=O)CC2(CCOCC2)CO1 C1(C(N2CC(C)(NC(CCc3onc(CC)n3)=O)C2)=O)CCC2(CCCC2)CC1 N1(C(C=C(C)C2CC2)=O)CC(NC(=O)C(C)Cc2ccco2)CC12CCC2 C1(C2CCCN(c3ncc4c(n3)CCC4)C2)(N(C)C)CC1.C1(=O)C(=O)NCCN1 N1(C(C(C)CC2CC2)=O)C2CCC1CN(C(c1cc(C(F)F)on1)=O)CC2 CCCCCCCCC(=O)N1CC(CNC(C2NC(=O)CC2C)=O)C(C)C1 CC(O)CC(C)(C)CNC(=O)C.c1(C=O)cncc(C2CC2)c1.C1CCC1.O N1(C(Cc2c(C)nsc2)=O)CCC2(CCCN(C(=O)C3=COCCC3)C2)C1 CC(CCCCNC(c1cccnc1N1CCCC1)=O)NC(=O)CC(C)F N1(C(CC=CCCCCC)=O)CCC2CC12C(=O)NC1(C)CCOC1=O C(CC(C)C(=O)NCCC1(O)CN(C(c2n[nH]c(C3CC3)c2Br)=O)C1)OC CC1CC2(CCN(C(=O)NCCC34CC5CC(CC(C5)C3)C4)CC2)CO1 CCC(O)C(C)C(=O)NCCC1CCC1.c1(C=O)cccc(CCN(C)C)c1.N c1(C(=O)NC2(CC(=O)NC(CC#C)C)CC2)cccc(CC#N)c1 c1(C(=O)NC2CN(C(c3cc(C)n(C)c3)=O)CC(C)C2)ccc2c(n1)OCCO2 C(=O)(CC(F)(F)CC(=O)NC1CCN(CCNC(=O)C(F)C(C)C)CC1)OC N1(C(C(=O)NC)=O)CC2CC1CN2C(=O)C=Cc1ccc(OC(C)C)cc1 Cc1cccc2cc(C(=O)NCC3C4CN(C(c5ccc(C#N)[nH]5)=O)CC34)nn12 c1(N(C(C2C(c3cccc(C)n3)C2)=O)C)ccc(Br)cc1Cl CCC(C)CNC(=O)C=Cc1cnc[nH]1.c1(C(=O)N)cc(C(C)(C)C)on1 c1(C(=O)NCCCN(C(C(C)C2CCCO2)=O)C)ccc(Cl)c(Cl)c1N C1(NC(CCC)=O)CCCCCN(C(c2cc3sc(Br)cc3s2)=O)C1 C=CC(CCC)CC(=O)NCC=CCNC(=O)CCc1cc(Br)cs1 c1(C(=O)NCC(CNC(CC2(C)CC2)=O)O)cccc(-c2ccoc2)c1 C12(CNC(CCCN(C)C)=O)CCCN(C(c3csnn3)=O)C1C2 c1(OC)ncc(C(N2CC(NC(=O)CCNC3CCCCC3)CC2C)=O)cc1Cl C1(N(CC(=O)NC2(CO)CCC2)C)CC(F)CN(C(c2ccc(Cl)cc2)=O)C1 c1(OC)cccc(C(N2CC(Nc3nccc(C)n3)C(C)C2)=O)c1C c1(C(=O)NCC(CC(C)C)NC(C2CCCC(C)(C)C2)=O)ccc2c[nH]nc2n1 N1(C(c2n(C=C)ncc2)=O)CCCN(C(c2ccc(F)s2)=O)C(C)C1 C1(C(=O)NC2CN(C(CC)C)C(=O)C2)CCN(Cc2cc(OC)ccn2)CC1O CC1CCC(NC(=O)C=Cc2ccn(C)c2)CN1C(=O)CCc1nnc(S)n1C N1(C(CSCC)=O)CC2CC(NC(c3cccnc3NCC)=O)C2C1 N1(C(CNC(C)=O)=O)CCC(NC(c2csnn2)=O)C1C(C)(C)C C1(C)(NC(CCC(=O)OCC)=O)CCCCC1.c1(C2C(C=O)C2)cccs1.N C(=O)(C(C)(C)C(C)(F)F)N1CC(CC(CNC(c2c(C)cns2)=O)(C)C)C1 C(=O)(C1=COc2ccccc2O1)NCCCN(C(C1=C(C)OCC1)=O)C C12(NC(CS(C)(=O)=O)=O)CCCC1N(C(=O)CCc1nc3ncccn3n1)CC2 N1(C(C(COC(C)=O)C)=O)CCC=C(C(=O)NC2CCCCC23CCC3)C1 C=CCCCCCC(=O)NC(C)(CNC(C1CC1c1ccc(C)cc1)=O)C1CC1 C1(NC(c2c(C)nc(O)s2)=O)CN(C(c2cc(C(N)=O)co2)=O)C2CCCC12 C(C(C)(C)CC(=O)NC1CCCCCC1F)NC(CCCN(C)C)=O c1(C(C(=O)O)N(C)Cc2ccccc2)ccc(OC(F)(F)F)cc1 CC(O)CCCNC(C1(N(C(c2ccsc2Cl)=O)C2CC2)CCC1)=O c1cc(C(=O)NC(CO)CO)cs1.C(C(=O)NC)=CCOCCOC c1(C(N2C(COC)CN(C(C3CC4CC4C3)=O)CC2)=O)cnn2ccc(C)cc12 C#CCC(O)C(=O)NC(CNC(=O)C=Cc1csc(C)n1)CC N1(C(=O)Nc2c(C(=O)OC)occ2)CC=C(c2ccccc2)C1 c1(OC)ccc(C(=O)NCC(C)(C(C)C)NC(C2CCCSC2)=O)cn1 c1(SC)nc(N2CCCC(C(=O)Nc3cncnc3Br)CC2)cc(C)n1 Cc1cc(Cl)cc2[nH]c(C(N3CCC4CN(C(=O)C(C)CF)CC34)=O)cc12 C(C(C(=O)NCCOCCCF)C(C)(C)C)NC(C(C1CCOC1)OC)=O C(=O)(C(CCC(C)C)NC(C1CNC(=O)N1)=O)N(CCOCC=C)C N1(C(c2c(C)[nH]nc2Cl)=O)CCC(C2(NC(=O)CCCS(N)(=O)=O)CCC2)CC1 c1(-c2n(CCC)nc(C)c2)cnc2ncc(C(=O)Nc3cc(Cl)c(Br)cn3)n2c1 c1(OCC)ccc(CN2CCSC(C(=O)NCc3ccc(O)nc3)C2)cc1 C12(CNC(=O)Cn3cc(C4CC4)nn3)CC(CN1C(C1CCOCC1)=O)C2 c1(NC(CCCC=C)C)cc(C)c(S(=O)(=O)N(C2CCCN(C)C2)C)cn1 Cc1cc(C)c(C(=O)NCCCNC(=O)CCc2nncs2)s1.C1CCCC1.C N1(C(CC=C(C)C)=O)CCN(C(C2COC3(CCC3)C2)=O)CC1CC(F)(F)F C12(CNC(C(C=C)C)=O)CCCC1CN(C(c1cc(C)c(F)c(C)c1)=O)C2 N1(C(c2c(C)nncc2)=O)CCC2CCC(NC(C3(C)CCC(F)(F)C3)=O)C1C2 C1(C2CCCC2)(C(=O)NCC2(O)CC(NC(c3cccnc3Cl)=O)C2)CCC1 c1(C(=O)N)cc(C)c(F)c(S(C)(=O)=O)c1.CCCC(O)CC(=O)NC(CO)CC Cn1ncc(C(=O)NC2(CC(=O)NC3(C4CCCCO4)CC3)CCCCC2)c1N CC1CN(C(c2cc(CCNC(=O)CCn3ccnn3)on2)=O)CCC1CO CC1(C)C(C)CCN1C(c1csc(C(N)=O)n1)=O.c1(C=O)cnn2c1CCC2.N CCC(CC(=O)NC12CC(C(=O)NC3CCOC3(C)C)(C1)C2)C1CC1 c1(C(=O)NC2CCC(NC(C3Cc4nccn4C3)=O)C2)cn2ccnc2s1 Cc1cc(C)c(C(=O)NCC2CCN2C(=O)C(C)COc2ccccc2)s1 C1(NC(C2(C(=O)NC)CC2)=O)CN(C(c2cc(Br)no2)=O)CC2(CCC2)C1 C1(NC(c2c(OC)cccn2)=O)CC2COC1C2.C1(C(=O)N)CCC(C)(C)OC1 c1(C=O)cnn2c(Cl)cccc12.C1(NC(CN(C)CCO)=O)CCC(C)(C)C1.N C1(C(=O)NCC2(C)CC2(F)F)CCC2(CC2)N1C(C1CC(=O)C1)=O C(=O)(C1CCCn2nccc21)NC1(C)CC(NC(c2[nH]cc(C(C)=O)c2)=O)C1 CC(C(=O)N1CCC(NC(C2(n3cccn3)CCCC2)=O)C1)C(F)(F)F C(N=c1[nH]c2c(c(=NC3CCCC3CF)[nH]1)SCC2)C1(OC(C)C)CCC1 CC1(C)CC(CNC(c2cc(CO)on2)=O)N(C(=O)C=CC2CCOC2)C1 c1(C(N2CCC(CCNC(CCNC(C)=O)=O)C2)=O)cnc2ccccn2c1=O N1(C(c2ccc(SC)o2)=O)CC2CC2(NC(=O)C=C2CCN(C)CC2)C1 C1(C(N2CC(CC(=O)N(C(C)C(C)C)CCO)C2)=O)CC(C(C)C)=NO1.CO C=CCC(C)(CC=C)NC(=O)C(c1cc(F)cc(F)c1)C N1(C(CN(C(=O)OC)C)=O)CC2CC(NC(c3nnc(O)nc3O)=O)CC(C2)C1 C1(CC=O)CCCCC1N(C(=O)CNc1ccccn1)C1CC1.CC(O)CF.N Cc1cc(N)c(C(=O)NCC2CC2)cc1C.C(=O)C(C)(C)C.C(=O)CC.C c1(C(=O)NCC(c2cc(F)cc(F)c2)O)cc2cc(Br)cc(Br)c2o1 CC(C=O)C(C)(C)C.n1(CC(N2CCC2)=O)ccc(=O)n(C)c1=O.C=CCO C#CC1(O)CCCN(C(=O)C(C2CCC2)NC(=O)Cc2cccc(O)c2)C1 C1(C(N2C(C(=O)NC3CC(=O)NCC3)C3CC3C2)=O)CCC2(CCC2)C1 N1(C(C2(C)ON=C(C(C)C)C2)=O)CCC2(CC1)CN(C(C1C(C)C1C)=O)CCO2 Cc1cc(Br)cnc1CC(=O)OC(C)(C)C.C12CN(C13CCC3)C(=O)C2 C(C(C)S(C)(=O)=O)NC(C(Cn1ccnn1)NC(c1c(C)ncs1)=O)=O N1(C(Cc2c(C)nccc2)=O)CC2CCCC2(NC(c2sccc2Br)=O)C1 Cc1cc(C(=O)NCC(C)(C)NC(C2CC(N(C)C)CCO2)=O)c(F)cc1Cl c1(C(N2CCC(NC(C(c3ccc(F)cc3)(C)O)=O)C2)=O)cc(F)c(F)cc1F c1(C=O)n[nH]c2cccnc12.C1(CNC(CCNC(=O)NC)=O)CCCCC1.N c1(C(C)=O)cc(C(=O)NC2CC(C)C2)c(C)o1.C1(CC=O)OCCC1(C)C c12ccc(SC)c(c1)S(=O)(=O)N1CCC3CN2CCC13.CS CCCC(CNC(c1cc(C(C)=O)c[nH]1)=O)C(=O)NCC12CCCC1OCC2 N1(C(C2CC(C)(CC)C2)=O)CCC(NC(C2(F)CCS(=O)(=O)C2)=O)CC1C C=CCCCCC(=O)N1CCC(C(C)NC(c2cscc2C(=O)OC)=O)C1 C(=O)(CCC(N)=O)N(C1CC(C#N)C1)CC(=O)NCC1COCCO1 C(CC(C)C)(C(=O)N1CCC(c2nn[nH]n2)C1)ONC(CC=C(C)C)=O CC(C)CC(CC(=O)NCCOCCCNC(=O)C#CC1CCCC1)CC(N)=O C1(NC(C(CC)CC)=O)CN(C(c2ccn(C(C)C)n2)=O)C2(CCOC2)C1 c1(C=O)ccc(F)c(C#N)c1.c1(SC)ccc(NC(=O)CN2CCCC2)cc1.N c1(C(=O)NC2CCCN(C(C(C3CC3)SC)=O)C2)[nH]c2c(F)cc(F)cc2c1C C12COCCN(C1)C(=O)N2.c1(OC)ncc(COCCO)s1.C(C)(C)C C1(NC(c2n(C)ncc2C(F)F)=O)CCC2(CC1)CC2Nc1ncccn1 CCCC(CCO)CN=c1[nH]c2c(c(=NCc3cc(O)ncn3)[nH]1)CSC2 CCCC(CCC)CC(=O)N1CCSCC1CCNC(c1ccn(CCF)n1)=O N1(C(CCNC(=O)NC)=O)CCCC(C2CCN(C(=O)CC3CC(F)C3)C2)C1 CC(C)CC(CNC(=O)C=CC1CCOC1)C(=O)NCC(C)(C)CCO N(C(=NCC1(S(C)(=O)=O)CC1)NCC1CCCCC1)C(C)(C)CF n1(CC)nc(C)c(C(N2CCC(CCNC(c3nonc3N)=O)C2)=O)c1Cl c1(C(N(C(C)C)CC)=O)cnc(CC(C)C)s1.C(=O)C(C)Cc1ccccn1 C1(NC(COC2CN(C(C(C)CC3CCC3)=O)C2)=O)CN2CCC1CC2 Cc1ccc(C(=O)NC2CC(CNC(c3c[nH]ccc3=O)=O)C2)c(O)c1 O(N1CCC(c2nnnn2C2CCCCCC2)(NCCC2CC2(Cl)Cl)CC1)CC c1(CC(N2C(CCNC(CCOCCC)=O)CCC2)=O)ccc(C#N)cc1 N1(C(C=O)=O)CC2CCC1C2.C1(C=O)C2CNC(=O)C12.CC(=O)NCC.N C(C)(CCC#N)(c1nnnn1C(C)C(=O)OC)Nc1cnc(CC)nc1 C1(OC)CC(NC(=O)CC2CCC2)CN(C(c2cc(C)n(C(C)C)n2)=O)C1 C#CCCCCC(=O)N1CCCC(CCNC(C2(F)CCCCCC2)=O)C1 N1(C(C(C)O)=O)CC(NC(c2cnc(Cl)s2)=O)C(F)C1 c1(C(=O)NCC2COC(C)C2)sc(Cl)cc1Cl.C12(C(=O)N)CCC(C1)C2 C1(N(C)C(c2ccc(Cl)s2)=O)CN(C(c2nnn3c2CCC3)=O)CCC1O C1(CN(C(C(C)NS(CCC)(=O)=O)=O)C)COCCN1C(c1cc(C)c[nH]1)=O C1CN(C(=O)C(O)Cc2ccccn2)CC1(C)C.CC(C(=O)N)OCCN(C)C c1(OC)ccc([N+](=O)[O-])cc1NC(C1CCCN1Cc1[nH]cnc1C)=O c1(CCC)n[nH]c(=NC2CCCN(C(c3cc(CC(C)C)on3)=O)C2)s1 CCC(CC(=O)N(CC(=O)NCC(C)(C)C(=O)NC)C1CC1)C(C)C C#CCCCC(C)C(=O)NCC1CC2CCC1N2C(=O)C(C)(C)CCOC CC(C)CC(CC(=O)NC(c1ccccn1)CO)NC(C12CCC(CC1F)C2)=O c1(NCCC(C)N(CCC)C)ncc(S(=O)(=O)NCc2ncccc2N)cc1Cl C(C)(C(C(=O)N1CCc2nn[nH]c2C1)C(C)C)NC(C=C(C)C(C)(C)C)=O C1(CC(=O)N(CCN(C(CC2CC(F)(F)C2)=O)C)C)CCN(C)C1.CC.O Cc1cc(C(=O)N(C(C)CNC(=O)C(C)OCCOCC)C)sc1C.O c1(-c2nnc(C)o2)cccc(NC(=O)NCC2(CO)CCCC2)c1 c1(CNC(C(=O)N(CCN(C)C)CCC2CC2)=O)cccc(F)c1Cl C(=O)(C(C)(C)CN(C(=O)CNC=O)C)NC(C)Cc1ccccn1 C1(CNC(C2CC2F)=O)CCN1C(=O)C(C1CCC1)C1CCC1 N(C1CN(C(=O)CN2C(=O)CCC2=O)Cc2ccccc21)C(=O)CC1(O)CCC1 C(C(C)(C)C(C)(C)O)NC(CCC(=O)OC(C)(C)C)c1n(C(CC)C)nnn1 C1(CNC(C2(CCO)CC2)=O)CCC(C(N2CCC2c2ccccc2)=O)C1 N1(CC(C)C)CCC(C(=O)NC2(CNC(C3CC(=O)N3)=O)CCC2)C1 c1(N2C(CNC(c3cn(CC=C)nn3)=O)CC(C)(C)C2)ncnc2c(C)csc12 c1(CC(=O)NCC2C(NC(C=CC)=O)COC2)ccc(Br)cc1 CP(C)(=O)CCC(=O)NC(CN=[N+]=[N-])C(=O)N1CCN(CC2CC2)CC1 C(=O)(C(CC)(CC)CO)NCC1(C)CCC(NC(C2CC(=C)C2)=O)C1 C1(OC(C)(C)C)COCCC1NC(=O)CCc1ccccc1OC(C)(C)C [SH](=O)(=O)CCC(=O)N1CCCC1C(C)(C)C.C1(F)(C=O)CC2(CCC2)C1.C c1(C(=O)NCC(CC(F)(F)F)NC(C2C(C=C)C2)=O)c(C)nc(C)nc1C C(CCC(=O)NC1CC(N(C(=O)C(O)C2CC2)C)C1)OC(C)C N1(C(C(CCC)=CCC)=O)CC2CN(C(c3cc(C(F)F)cs3)=O)CC2(C)C1 C1(CNC(=O)NCc2ccco2)(C)CCCO1.c1nnc(-c2ccccc2)o1 c1(N2CC(COC)N(C(C3(Br)CCC3)=O)CC2)ncnc2[nH]cc(C#N)c12 N1(C(C(c2cnn(C)c2)C)=O)CCOCC(C(=O)N(CCCCO)C)C1 c1(C(=O)NCC2N(C(C3C(C)C3)=O)CC(C)(C)C2)noc2c1CCCCC2 CC1CC=C(C(=O)NC2CC3CN(C(=O)CCN(CCC(C)(C)C)C)CC23)CC1 n1(CCCC)nnnc1C(C(C)(C)C1CCCO1)NCC(C)(C)CC C1(C(C)C)CC(O)CN1C(C1CC(NC(=O)C=CC2CCCN2C)C1)=O C1(NC(c2ccn(CC)n2)=O)(CC)CCN(C(=O)CC2(C#N)CCCCC2)CC1 c1(C(=O)NC2C3CN(Cc4c(C)nn(C)c4)CC32)c(Cl)oc2ccccc12 c1(C(N2C(C)(C(=O)OC)CCC2)C(=O)NC2CCC2)nc2ccc(Br)cc2s1 c1(OC)cc(C(=O)NOCC(N)=O)ccc1N1CCSCC1 c1(COCC)nc(N2CC(C)CC2C)cc(C)n1.C1(CC=O)CCC2CC12.N C1(N(C(COC(C)(C)C)=O)Cc2cnn3ccccc23)CCCC12CCNCC2 C1(CCC)CN(C(=O)CCS(C)(=O)=O)CCN1C(C1CC(C)=NO1)=O c1(NC2CC(CNC(C3(O)CCC(C)(C)CC3)=O)C2)cc(=O)n2ccccc2n1 C(CC(C(=O)Nc1cncc(Cl)c1)NC(c1ccc(F)s1)=O)=CC C=CC1CN(C(C2(COC)CCCO2)=O)CC1NC(=O)C(C)=C(C)C N#Cc1ccc2c(c1)CN(C(C1CC(O)CN1C(c1cnon1)=O)=O)C2 CC1(C)CCN(C(c2cc(C3CC3)nc(O)c2)=O)CC1C.c1(C(=O)N)cnco1 N1(C(C2CCC(C)O2)=O)CC(CNC(=O)CC23COCC(C2)C3)C(C)(C)C1 CC1CN(C(=O)C(c2ccccc2F)C)CCN1C(C1CCS(=O)(=O)C1)=O N1(C(=O)Cc2csc(S)n2)CCC2(CCCN2C(C2CCN3CCOCC23)=O)C1 c1(CC)cccnc1C(N1CCC(N(C)C(c2cc(Br)ccn2)=O)CC1)=O c1(C(=O)NCC2(C(=O)NCC(C)C(F)F)CC2)csc(C#N)c1 c1(CC(=O)NC(CC(C)NC(CC2(OC)CC2)=O)C)sc2ccccc2c1C C1(C(N)=O)(NC)CCN(C(=O)C(C(=O)OC)OC)C1 C(CC(C)C)(C(=O)NCCCN(C(c1cc(C)sc1N)=O)C1CC1)OC CCCCS(=O)(=O)CC(=O)NCC1CN(C(c2cc3cn[nH]c3cn2)=O)CC1C C1(C=O)CC(=O)NC(C)C1.Cc1nc(O)[nH]c1C(=O)NCC1(C)CC1.N C1(NC(C(C)Oc2ccccc2)=O)CC2CC1CN(C(C1CCC(=O)N1C)=O)C2 C1(C(=O)NC(CCNC(c2c(CC)nccc2)=O)C)CCCC(C)(C)CC1 CN1C2CCC1CC(C(N1CC(CNC(c3ccc[nH]3)=O)C3(CC3)C1)=O)C2 c1(CC)ncncc1C(=O)NCc1cc(C(=O)N(C)OCC(F)(F)F)on1 c1(N2CCC(OC)CC2)nc(N2CCSC(C)C2)c2ccsc2n1 CCCC(CC(C)C)C(=O)NCC(CO)NC(c1cn(-c2ccn(C)n2)cn1)=O c1(C(=O)NC(CNC(c2csnc2Cl)=O)CO)cc(-c2cccs2)[nH]n1 C(=O)(C(C)(C)CCC(=O)N1CCN(CCNC(=O)C(C)N(C)C)CC1)OC CC1CN(C(C2CC2(C)Br)=O)CCN1C(c1cn[nH]c1)=O N1(C(c2sccc2OC)C(=O)NC(CC)C)CCN(C)C(C(C)(C)C)C1 C=CC(CCC)CC(=O)NC1CCN(C(c2cccc(C#N)c2C)=O)C(C)C1 S(=O)(=O)(c1cccc(CNC(=O)N)c1)NCCOC.CC(=O)N(C)C N1(C(Cc2n(C)cnn2)=O)CCC2CN(C(=O)C#CC(C)(C)C)CC2C1 Cc1cc(CNC(=O)C(C2CC=CCC2)NC(c2cnns2)=O)co1 c1(C(N2CC(N(c3ncnc4c3cnn4C)C)C2)=O)ccc2c(c1)OCCO2 C1(C)(CNC(c2nc(C)oc2)c2nnnn2CCC2CC2)CC(F)(F)C1 C#Cc1ccccc1.C1(N(CC=O)C(C2CC2)=O)CC(C#N)C1.C(C)=O.C N1(C(C(n2c(C)ncc2)C)=O)CCC(O)CC1C(=O)N(C)CCn1cnnc1 Cc1cc(-c2cnc(NCC#N)s2)cc(C)c1NS(=O)(=O)CCBr Cc1ncc(C(=O)NC2CCCC(CNC(C3CNC(=O)N3)=O)C2)cn1 CC(CC(=O)NC1(CO)CC(F)C1)N(C(=O)CCOC1COC1)C C1(C(=O)NCCCCCN(C(=O)C(C)SC(F)(F)F)C)(OC)CCC12CCC2 c1(C(=O)NCCC(C)NC(=O)C(C)(O)C2CCC2)cncc(C(F)F)c1 C1(NC(CC2(C)CC2(Cl)Cl)=O)CN(C(=O)COC2CCOC2)CC1C(F)F C1(C(=O)NC2CCC2NC(=O)C(C)O)(OC)CCOCC1 c1(-c2cn(C3CCN(C(=O)CCc4ccc(Cl)cc4)CC3)nn2)ccc(Cl)nc1 C(=O)(C1CCOc2c(F)cccc21)NCC1CC(NC(CCC#C)=O)C1(C)C c1(C(N2CC(CN(C)C(C3Cc4cscc4C3)=O)C2)=O)cn2cnnc2cn1 CCC(CNC(=O)C(C)(C)NC(C)=O)(CC)N=c1[nH]nc(C(=O)OC)s1 C1(CC)CN(C(C2(C)CC2(F)F)=O)CCN1C(c1cnn2ccsc12)=O c1(OC)c(C)csc1C(=O)NC1(CO)CCN(C(C2CC3CC3C2)=O)C1 N1(C(c2n(CCC)ncn2)C(=O)NC2CCCCC2)CCN(C)C(C)C1 c1(CC(N2CCC(NC(C(CC)(F)F)=O)(CC)CC2)=O)ccn2cncc2c1 N1(C(c2oc(C)c(Br)c2)=O)CC(CNC(=O)CCC2(C)CC2)OC(C)(C)C1 N1(C(C(=Cc2ccncc2)C)=O)CCN(C(C2CC(C)(F)C2)=O)C(C)C1 C1(C2CC2)OCCO1.C1(c2ccccc2)(C(=O)OCC2CC2)CC1(Cl)Cl c1(CC)nn(C)c(CC)c1CC(N1CC(CO)(NC(=O)C(O)CC)C1)=O C(=O)(CC(C)CCC=C(C)C)N1CCC(CNC(CC(=O)NC)=O)CC1.C C1(C)(CC(=O)N)Oc2ccccc2O1.C(C)(C)(CC(=O)NC1(C)CCC1)OC C#CC1(NC(C2CN(C(C3C=CC=CC=C3)=O)CC2OC)=O)CCOC1 C#CCCCCCC(=O)NC1CCC(CNC(c2ocnc2C2CC2)=O)C1 CC1CCCCC1CNC(c1ccnn1C(C)(C)C)=O.c1(CC=O)nc[nH]n1 c1(C(=O)NC(C)(C)CNC(c2cc(C(F)F)no2)=O)cnc2nccn2c1 n1(C(C)C(F)(F)F)nc(-c2nc(C(F)(F)F)cs2)nc1CCC=CBr C1(C)(NC(=O)Nc2ncc(C(=O)NC(C)C)s2)CCC(C)(C)CC1 c1(C(=O)NC(C(CO)NC(CCCSC)=O)C)ccc([N+](=O)[O-])cc1Cl c1(C(=O)NC2C(NC(C3(C)CCOC3)=O)COCC2)ccc2ncncc2c1 N1(Cc2n(CC)cnc2)CC(O)CC1C(=O)Nc1csc(-c2ccccc2)c1 c1(CCCC(=O)N2CC(CNC(C(COC)N(C)C)=O)C2)ccc(C)cc1 C#CC1(CNC(c2cc(CNC(c3cnc(C)o3)=O)no2)=O)CCCC1 c1(OC)ccc(I)c(CCNC(=O)NCC(C2CCOCC2)(C)OC)c1 CCCCC(O)CC(=O)NC1CN(C(c2ccc(=O)n(CCF)n2)=O)C(C)(C)C1 C1(SC)CN(C(c2cnc[nH]2)=O)CC1NC(c1ccnn1CC1CC1)=O N1(C(COCP(C)(C)=O)=O)CCN(C(C2C(Cl)(Cl)C23CC3)=O)C(CO)C1 N1(C(c2cnn(-c3ncc(Cl)cn3)c2)=O)CCC2C(CCN2C(C2CC2F)=O)C1 c1(C(N2C(C(C)NC(c3cnccc3Br)=O)CCC2)=O)ccc2nc[nH]c2c1 N1(C(CCn2nc(C)c(C)c2C)=O)CC2CCN(C(=O)Cn3cc(Cl)cn3)C2C1 C1(CC)CCN(C(c2noc(C3CC3)c2C)=O)C1.C1(C=O)CC(=O)N(C)C1.C C1(C(N2CC(C(F)(F)CO)(C(=O)OC)C2)=O)CCCNC1C Cc1nc(C(N2CCN(C(=O)C(O)C(F)F)CC2c2nccn2C)=O)cc(O)n1 C1(NC(C2CCC3(CC2)CC3)=O)CN(C(=O)C)CC2CC12.C(=O)C(F)(F)F c1(CC(=O)NCC2(OC)CN(C(=O)C3=CC(C)CC3)C2)cc(C)ccc1C Cc1ccc(C(F)C(N2CCC(N(C(=O)CCOC3CC3)C)C2)=O)cc1 C1(CC)COC(C)(C)CN1C(=O)C(C)(C)CN(C(=O)CCc1cscn1)C c1(C(=O)NCC(C)(C)NC(c2cc(C)ns2)=O)ccc2c(c1)CCCC2 CCCC(C(=O)OC)C(=O)NC1CC1CNC(C12CCC(F)(CC1)CC2)=O N1(C(C(C(C)C)n2cnnn2)=O)CCC(C)(C)C(NC(=O)Cc2ccsc2)C1 Cc1cc(Cl)c(C(=O)NC2CC2C)cn1.c1(C=O)cc(C2CCCCC2)on1.N C1(C=O)CCCC12OCCO2.CC1(C(=O)NCC2CC(F)C2)CC(F)(F)C1.C Cc1nc(C#N)ccc1NC(C1COCCN1Cc1c[nH]c2cccnc12)=O c12ccc(C#N)c(n1)S2.Brc1ccc(OCC(F)F)nc1 N1(C(C2C(C)(C)CC(F)(F)CC2)=O)CCC2(CCCN(C(=O)CCF)C2)C1 S(=O)(=O)(c1ccc(Br)c(C(=O)OC)c1)NC(C#C)(C)C1CCOC1 CC1CCCC(N=c2cc(NCCc3cn4c(n3)SCC4)nc(C(F)(F)F)[nH]2)C1 N1(Cc2nccnc2)CCC2(CC1)CC2.C12CCN(CC1)c1ccnc(n1)OC2 C(=O)(CCCCCCCCC1CC1)NCC#CCNC(C1(C)CCC(C)CC1)=O C1(C)CC2(CCC2)C1.C(C)(CC(=O)NCC(C)(C)OCC(=O)NC)SC C(=O)(C1=NOC(C)C1C)N1C(C(N(CC#C)C)=O)CNC(=O)C1 Cc1nnc2n1CC(C(=O)NC1CC(NC(=O)Cc3cncc(O)c3)C1)C2 c1(-n2cc(C(N(C(c3c(C)cc(C)o3)=O)C)C)nn2)ccc(F)cc1F N1(C(c2c(C)c[nH]n2)=O)CCC(C(=O)N(C)Cc2c(C)cnn2C)C1C n1(CC(=O)N(CCC)CCNC(=O)C(F)OC(F)(F)F)cnc2c1CCCC2 C(C(C)(C)CC(=O)NC1(C)CCOC1)NC(c1occ(C)c1)=O CC(CCNC(C1CCC(N=[N+]=[N-])C1)=O)N=c1ccn2nccc2[nH]1 C1(C(=O)NCCNC(C(n2c(C)ccn2)C)=O)CCN(C)C(=O)C1 C(=O)(C(F)(F)c1cccnc1)N(CC(C)NC(=O)CC1OCCC1C)C c1(C(=O)NC2CCCC(N(C(COCCCC#C)=O)C)C2)ccc(OC)cc1C C(=O)(CCC(CF)CF)N1CCC(OCC(=O)NC(C)(C)CC(F)(F)F)C1 c1(C(N(C(C)CNC(=O)C=Cc2cnccn2)C)=O)cc2cn[nH]c2cn1 N1(C(C2(C)CC(C)(C)C2)=O)CCCOC(CCNC(C2CCS2(=O)=O)=O)C1 N1(CC)CC(C(N2CC(O)(c3cn(C(c4ccccc4F)C)nn3)C2)=O)CC1=O C12(CNC(C3CCN(C)CC3)=O)CCCN(C(=O)COC3CCC3)C1C2 c1(C(N2CCCC(C(=O)N(CC(F)F)C)(CC)C2)=O)cc[nH]c2nccc1-2 c1(C(N2C(C)CN(C(c3ccc(C(C)(C)C)[nH]3)=O)CC2)=O)ccc2ccnn2c1 c1(CC)nc2cccc(C(N3CC(NC(c4ncnn4CC)=O)C(C)C3)=O)c2[nH]1 CCCCC(CC)C(=O)NC(C)C(=O)NS(C)(=O)=O C1(CNC(C(c2ccn(C)n2)C)=O)N(C(=O)C=C2CCCCC2)CCC1(C)C c1(OC)ccc2nc(COC(=O)Cc3csc(C)c3C)[nH]c2c1 N1(C(C2C(C)(C)CCO2)=O)C2CCC1C(C(=O)NCc1ccc(CO)cc1)C2 N1(C(CC2CC(SC)C2)=O)C(C(=O)NCC(F)(F)C(F)F)CCC1C c1(C(N2C(CNC(c3sccc3C3CC3)=O)COCC2)=O)cc2ccccc2s1 N1(C(C(C)CCN(C)C)=O)CC2CCC(Nc3nc4ccccc4o3)C2C1 C1(C(C)NC(C(C)O)=O)CN(C(c2coc(-c3cnn(C)c3)n2)=O)CCO1 c1(C(C)C)ccc(C=CC(=O)NCC2C=CCN2C(C2CCSC2)=O)cc1 c1(CCCC)ccc(C(=O)NCCN(C(c2snc(O)c2Cl)=O)CC)cc1 S(=O)(=O)(c1cc(C)cnc1NC(c1ncnn1C)C)NCCC=CCCC N1(C(c2n(C)c(O)nc2)=O)CCN(C(c2cc([N+](=O)[O-])n[nH]2)=O)C2CCCCC12 CC1(C)CC(C(=O)NCC(C)(CO)NC(=O)CC2CC(=O)C2)C(C)(C)O1 C1(NC(CCCCSC)=O)CCCC12CN(C(=O)C1=COCC1)C2 CCCCCC(O)C(=O)N1CC=CC(NC(=O)C=CCN(C)C)C1 N1(C(c2ccccc2)=O)CCCC2(CC(C(=O)N3CCOC(CO)C3)=NO2)C1 CC(C)(O)C(F)C(=O)NC1COCCC1NC(=O)C=Cc1ccccc1 c1(NC(C2C=CC(NC(c3ccncc3)=O)C2)=O)nccc(I)n1 Cc1ccccc1CC(=O)NCC1CCCC1.c1(C=O)ccnn1C(C)(C)C.N c1(C=O)cc(=O)c2ccncc2o1.C1(C)(CC)CC1C(=O)NCCO.CC Cc1ccc2c(=NCC3(Br)CC3)[nH]c(=NC(C)c3cccnc3)[nH]c2c1 N1(C(C2CCCN2c2cccnn2)C(=O)NCCCSC)CCS(=O)CC(C)C1 N1(C(C(C)(C)C)=O)CC(N(C)C(c2ccccc2)=O)C(F)C1.C(CCO)S.C1CC1 C1(CC(=O)NC(CCCCNC(CCn2c(C)ncc2)=O)C)CCC(F)(F)CC1 c1(CC)cc(C(=O)OC)ccc1NCc1cnc(-c2ccccn2)s1 C1(CC(N2CCCC2)=O)C(=O)N(C)N=C1C.C1(OC)(OC)CCC1C(=O)N C1(CN(C)C(C2CCN(C3CCCC3)CC2)=O)CCN(Cc2ccccc2)CC1 c1(C2(C)CC2)cc(C(N2CC(CCCCNC(=O)CCCF)C2)=O)[nH]n1 Cc1nsc(N)c1C(=O)N(C1CCCN(C)C1)CCO CP(C)(=O)c1ccnc(C(=O)NCCOCC)c1.c1(C(=O)N)ncc[nH]c1=O C1(NC(c2c(F)ccc(CC)c2)=O)CCN(C(=O)C(C)C(C)(F)F)C12CCC2 c1(OC)cccc(C(=O)NC2CC(NC(C3(C)C=CCC3)=O)C2)c1 Cc1cncc(-n2nc(C(C)C3CC3)nc2CC2CC3CCC2O3)c1 Cc1c(C(N2CC(NC(C3(O)CCC3)=O)C(O)C2)=O)ccn1CCO.C(C)C C(=O)(C1=C(C2CC2C)N(C2CCOCC2)C(=S)NC1c1cncc(C)c1)OC N1(C(CC2CC(OCC)C2)=O)CCCC2(NC(=O)C(C)=C(C)C)CC2C1 c1(NC(=O)OCC)cccc(C(=O)N(CCCCNC(=O)C(C)O)C)c1 N1(C(COCCOC)=O)CC(C)N(C(C2COCCC2(F)F)=O)CC1C N1(C(C2(CC)CCCC2)=O)CC2CCC2(CCNC(=O)C)C1.c1ccccc1.O N1(C(=O)CCOCC(F)F)CCC(NC(C2(N3CCCC3)CCC2)=O)C(F)C1 c1(N2CCC3(CC3)C2)cnc(C#N)c(C#N)n1.C(C(=O)N)(C(C)C)OCC.C N1(C(Cc2cnc(C)s2)=O)CCC(C(N2CC(O)C(O)C2)=O)C1C C(CC(C(=O)N(C)CC1CCN(C)C1)NC(C1CC(C)C1)=O)=CC N1(C(C(CCC)NC(N)=O)=O)CCC(C)C(NC(C2CC(C)C2)=O)C1 c1(C(N2CC(NC(c3c(C)nns3)=O)C(C)C2)=O)cc(Br)c(O)nc1C Cc1cc2cc(c1)CN2.n1(CC(=O)OCc2ccccc2)ncc(C#N)c1N N1(C(CNC(=O)NC)=O)CCN(C(C23CC(C(F)(F)F)(C2)C3)=O)CC1 c1(CN(C(=O)CCC2CC2)C)cccc(C)c1.C(=O)CC=CC(C)(C)C C1(CC(=O)NCCC(CNC(CN(C)C(N)=O)=O)O)CCC(=O)NC1 CC(C)CC(O)C(=O)N1CC2CCC2(CNC(c2cnc(CC3CC3)s2)=O)C1 CC1(CNC(C2(F)CC=CCC2)=O)CN(C(c2cnn[nH]2)=O)CCO1 C(=O)(C(C(=O)OC)OC)N(CC(=O)NCC(C)CC)CCC C1(NC(=O)CCc2cncnc2)CC(NC(c2nscc2Br)=O)C(O)C1 C(=O)(CCCS(=O)(=O)N1CCCC1)N1CC(N(C(=O)COC(F)F)C)C(F)C1 C(=O)(CCCC(=O)N1CCC(C)C(NC(=O)C)C1)NCC.C1(C=O)CCCC1 N1(C(CC(=O)NC2CC2)=O)CC(NC(=O)C2=COCC2)CC(O)C1 C1(C(=O)NC2CC(CNC(=O)C=Cc3cnc[nH]3)C2)CC2(CCCCC2)CO1 CCCS(=O)(=O)CC(=O)NC1CN(C(=O)C(O)(C(F)(F)F)C2CC2)CCC1O C(CCC(=O)NC(c1ccccc1)CNC(=O)Cn1nccn1)=C(C)C c1(CC)ccc(CN2CCCC2CCC(N2CCC(OC)C2)=O)c(O)c1 CC1(C)CC(C(=O)NC2COC(C3CC3)C2)CN(C(C2(C)CSC2)=O)C1 Cc1ccc(C)c(C(=O)NCCCNC(=O)Cc2cccc(Br)c2)c1 C12(NC(C3CCN(C)C3=O)=O)CCC(CN(C(=O)CCc3ccncn3)C1)C2 c1(N2CC(CC(C)NC(c3c(OC)ccc(F)c3)=O)C2)cc(C)ncc1C#N n1(CCC=CC)c(-c2cccc(Cl)c2C)csc1=Nc1cccc(F)n1 C#CC(O)CC(=O)Nc1cccc(C(C)(C)C)c1 O=C(NN1CCCC1C(=O)NCCN1CCC(CO)C1)C1(CO)CCOCC1 c1(C(N2CCCCC2)=O)ccc(C(F)(F)F)c(O)n1.n1(CC)cccc1C(=O)N C1(NC(C=CC=CC)=O)CC(C)CN(C(c2cccc(CF)c2)=O)C1 c1(C=O)ccc(S(=O)(=O)N(C)C)o1.C1(F)(C=O)CC=CCC1.CC(C)CC.N Cc1c(Cl)ccnc1CC(N1CC(O)CC1c1ccc(Br)cc1)=O C1COC2(C1)CN(C(c1ccnn1CCF)=O)C2.c1(CC)cc(C(=O)N)n(C)n1 Cc1cc(C(=O)C(=O)NCc2ncccc2C(=O)O)ccc1F CCCC(C)(C)C(=O)NCCN(C1CCCC1)C(c1ncccc1)=O.C(C)C.O N1(C(C=COCC)=O)CCN(C(C23CC4CC2C3C4)=O)CC1c1ccc(F)cc1 c1(N(CCOCCN(C(C2(CC#C)CCCC2)=O)C)C)nc(C#N)c(Cl)s1 C1(C(N(C)CCNC(=O)CC2CC(F)(F)C2)=O)CCCCC12CC2(F)F c1(C=O)cc[n+]([O-])cc1.C1(C(C)(C)O)(C)CN(C(c2ccc(C(F)F)s2)=O)C1 N1(C(C2(C(C)(C)C)CCCC2)=O)CC2CCC2(CNC(=O)Cc2cncs2)C1 c1(C(=O)NCCC2(CNC(CSC)=O)CC2)cc2n[nH]cc2cc1C N1(C(CCC(c2cc(C)sc2C)=O)=O)CCC2(C1)CN(C(=O)C=C(Cl)Cl)CCO2 CN1CCN(C(C2CSCCS2)=O)C(CNC(c2ncc(Cl)cc2O)=O)C1 CN1CCC(=CC(N2CC(N(C(=O)CC3(C)CC3(Cl)Cl)C)C(O)C2)=O)CC1 c1(OC)ccc(Cl)c(C(=O)NCC(C)N(C(=O)CCc2cn[nH]c2)C)n1 C(=O)(C1=C(NC(=O)C(C)CCC)CCC1)OCC.C12CC(C(=O)N)(C1)C2 C(=O)(CCCCC(N)=O)N1CCC(C2N(C(c3c(C)ncs3)=O)CC2(C)C)CC1 c1(C(C)NC(CC2(NC(COCCCCC)=O)CCC2)=O)cccnc1C C(=O)(CC(C)CF)N(C1CCCC1)CC.c1(C(C=O)NC(C)=O)ccccc1O.N c1(OCC)ccc(NC(=O)NC(c2ccc(C(=O)OC)cc2)CO)cc1F C(CC(C)C)(C(=O)N(CC(C)CNC(=O)CC(C)(C)N(C)C)C)OC c1(C(=O)NCCCc2cn(-c3ccc(CO)cc3)nn2)ccccc1[N+](=O)[O-] C1(C(N2C(CC(N3CCCC(O)C3)=O)CCC2)=O)CCc2nnc(O)n2C1 c1(C(=O)NCCCCCNC(C(C(C)O)N(C)C)=O)ccn2cncc2c1 C1(CC)Oc2ccc(Cl)cc2C1NC(C1(C(C)(F)F)CCOCC1)=O c1(OC)cc(C)c(C(N2CCCCC2C(=O)NCCn2ccnc2)=O)cc1OC Cc1cccc(C)c1OCCC(=O)NC(C1CCCC1)C.C(=O)CP(C)(C)=O.N C1(C(=O)Nc2cnc(C(F)(F)F)nc2)CC(F)CN(C)C1.c1ccc(Br)c(Cl)n1 C(CC(=O)NC(C1(O)CCN(C(=O)Cc2cccnc2N)C1)C)(C(F)(F)F)OC Cc1csc2ccc(C(=O)NCC(C)N(C)C(c3ccc4[nH]ccc4n3)=O)cc12 c1(N(CC(CC)(C)OC)C)ncccc1S(=O)(=O)NCc1ccncc1C(C)C C(=O)(C1=CC(O)CCC1)N.Cn1cccc1-c1cc(C(=O)NCC=CC)n[nH]1 N1(C(CC)=O)CCc2c(c(CNC(c3sc(C)c(Br)c3C)=O)nn2C)C1 C1(C(N(C(CC)CC)CCO)=O)CCN(C(c2n[nH]c3c2CCC3)=O)C(C)(C)C1 C(=O)(C(CC=C)C(C)C)N(C1CCN(C(C2CCC3(CCC3)O2)=O)CC1)CC#C C(C(=O)N1CCN(CC2CC2)CC1)(C(C)C)SCC.C1(C=O)CC12CC2.N N1(C(C(C(CC)C)N(C)C(c2cnn(CCO)c2)=O)=O)CCCCCCCCC1 c1(C(N2CC(C(C)NC(C(CC)O)=O)C2)=O)nc(C)nn1C C1(NC(c2c[nH]nc2C2CCC2)=O)CC(O)CN(C(=O)Cn2cnnc2)C1 C1(C(N(CCC(=O)OC)CC=C)=O)CCC(C)N(C(=O)CN(C)C2CC2)C1 N1(C(=O)Nc2c(C)cc(C#N)s2)CCCC(C)(C)C1c1nc(C(C)C)no1 C(C)(CCC(=O)NC1CCCC1CN=[N+]=[N-])NC(C1C(C)CC1)=O Cc1cccc([N+](=O)[O-])c1C(=O)N.C1(C(N2CCCC2)=O)CC(=O)NC(C)C1.C c1(C(=O)NC(C)C(=O)NC(C)(Cc2ccc(Cl)cc2)CO)ccc2c[nH]nc2c1 CCCCC(C)(F)C(=O)N1CCC(C(C)CNC(=O)CS(=O)(=O)CCO)CC1 N1(C(=O)CC2CCS(=O)(=O)C2)CC2CC1CCN2C(c1ccnn1CCF)=O N1(C(C(=O)N(CC(c2ccc(Cl)cc2)O)CCO)=O)CCCC2(CCC2)C1 CC1CCC(NC(=O)CCOC2CC2)CN1C(c1sccc1OC(F)F)=O C1(O)(C(N2CC(C(=O)NCC3N(C(C)(C)C)CC3)C(F)C2)=O)CCOC1(C)C Cc1ccc(C(O)C(=O)NCCC(C)N(C(=O)C(=Cc2cn(C)cn2)F)C)cc1 CC(CS(=O)(=O)N(C)C)N=c1ccnc(NCCC2CC3C=CC2C3)[nH]1 C1(c2cn(CCN)nn2)C2CCCC1N(C(C13CCC(CC1)C3)=O)C2.C[SH](=O)=O N1(C(c2c(OC)ccs2)=O)CCCCC(N(C)C(C2CCCN(C)C2)=O)C1 C1(OCC)CC2(C1)CC2C(=O)N(CC)C(C)C.C1(O)(C=O)CCOC1 C1(CCNC(=O)NCC(=O)N(C)CC2CCCO2)COC(C)(C)C1 CON1CCC(CC(=O)NC2CCCC(NC(=O)CCS(C)=O)C2)CC1 c1(CCNC(=O)NC(CCCOC)C(=O)O)c(C)nc2ccccn12 N1(C(=O)OC(C)(C)C)CC2CCN(C=O)C2C1.c1(CC(C=O)O)ccccc1Cl C(C(CC(C)C)C(=O)NCCC1CC(=O)N(C)C1)NC(C1(C#C)CC1)=O Cc1cc(C)n(CC(N2CC(C3(NC(=O)CCc4ccon4)CC3)C2)=O)c(=O)n1 c1(C(N2CC(C(N3CCC(C(N)=O)C3)=O)OCC2)=O)cc(C#N)ccc1N C1(CNC(CC(CC)C2CC2)=O)CCN(C(=O)C=Cc2cccc(F)c2)C1(C)C C12(CNC(c3cnn(-c4ccc([N+](=O)[O-])cc4)c3)=O)CCCCN1CCC2 C(C(C)C)(C(O)C(=O)NCC1(NC(c2cscc2C)=O)CC1)OC C(=O)(CS(=O)(=O)CCO)NCCC1OCCN(C(CCc2cc(C)[nH]n2)=O)C1 c1ccc(C)cc1.C(F)(C(=O)N(C)CCOCCN(C(=O)C)C)=CC.S c1(N2CCCCC(NC(C3CCS(=O)(=O)N3)=O)C2)nc(Cl)ncc1[N+](=O)[O-] N(C1CC2(CN(C(c3cc(Cl)cs3)=O)C2)n2ccnc21)C(C1=CCC(C)CC1)=O c1(CN(CC(COC)C)C)nccc(OC)c1C Cc1ccc(C=CCC(=O)NC2CN(C(=O)C(C)OC3COC3)CC2(C)C)cc1 C1(NC(C=Cc2ncc(C)[nH]2)=O)C2CC1CN(C(C1CCN1C1CCCC1)=O)C2 N1(C(CC(C)SC)=O)CC2(CCNC(=O)C=CC3CCOC3)CCC1CC2 C(CN=C(NCC1C2COCC12)N(C)Cc1cn(C)nc1C(F)(F)F)OC N1(C(C2ON=C(C(C)C)C2)=O)CC2CCCC1C2CNC(=O)Cc1ccco1 C(=O)(C1=CCCCC1)N1CCC(c2cccc(F)c2)(NC(=O)CC(F)(F)Cl)C1 N1(C(C2=CCC(NC(c3c(OC)nsc3)=O)C2)=O)CCC(O)C(C)(O)C1 N1(C(CCc2ccc(C)o2)=O)CCN(C(C2CCS2(=O)=O)=O)C(CC2CC2)C1 N1(C(C2N(C(C(CCOC)OC)=O)CCC2O)=O)CCC(O)CC1C1CC1 C1(F)(C=O)CCCOC1.c1(C(N2CCC(OCC)C2)=O)ccnc(C2CC2)c1.N C1(CNC(c2nc(C)sc2)=O)CCN(C(C2CC2[N+](=O)[O-])=O)CC1O c1(C(=O)NC2CC(N(C(C3C(=C)C3)=O)CC)C2)cccc2ccnn12 C(=O)C1=C(CC)OCCC1.C1(OCC)(CO)CN(C(=O)CC2CSCCO2)C1 CS(=O)(=O)c1ccc(OCC(=O)NCCC2(NC(=O)C=CBr)CC2)cc1 C1(C(=O)NC(CNC(=O)CCC(F)F)CO)C2C3CCC(C3)C12 CC(C)(CN(C(CO)CCOCc1ccccc1)CCCCO)CCC#N C1(C(N2CC3(CN(C(CCC4C(C)=NOC4=O)=O)C3)C2)=O)Cc2ccccc2O1 C(c1nnc(C(C)C)o1)=CC=O.C1(C(=O)NC2CC2)(OC)CCSC1.C CC1CN(C(c2ccc(Cl)nc2N)=O)CCN1C(=O)C(c1cncc(F)c1)C C=CCC(C(=O)NOCC1(C)CCC1)NC(=O)CC1CCCC(=O)N1 O=C1OC2CC(C(=O)N(CCCNC(C3CC(F)C3)=O)C3CC3)CC2O1.C c1(Cc2nc(C(C)(Cc3ccccc3)C(F)(F)F)on2)ccc([N+](=O)[O-])cc1F CC1(C)CCC=C(C(=O)NCCCCCCNC(C2Cc3nncn3C2)=O)C1 c1(C(=O)NCc2cccc(CNC(C3CCCC3O)=O)c2)cc2ccccc2[nH]1 N1(C(c2scc(C(=O)Nc3onc(C)c3C)n2)=O)CCCNC(=O)C1 C12CC=CCC1C(=O)NC1CC1C(=O)N2.C(C)(CO)(C(=O)OC)OC C(CN=c1[nH]ncs1)NC(Cn1c(C(C)C)nnn1)=O CC(CCC(=O)NC1C(CNC(c2cccnn2)=O)CCC12CCC2)S(C)(=O)=O c1(CNC(c2nccc(C)c2)C2CC2)ccc(F)cc1F Nc1cncnc1C(=O)NC1C=CC(CC(=O)NCC=CC2CC2)C1 c1(C2C(N(CCCC)C(c3ccc(OC)cc3)=O)C2)ccccc1Cl C1(c2nnnn2C2CCOCC2)(NCC2ON=C(C)C2)CC(C)(C)CC(C)(C)C1 N1(C(C(CCC)C)=O)CC2CCCC(C1)N2C(c1ccc2oc(S)nc2c1)=O CC(C)(C)C(=O)NCC(=O)NC1CCC1.C1(C(=O)N)CCN(CC(F)F)C1 C1(NC(C(C)C(C)O)=O)CCN(C(C2CCCC(C(F)(F)F)C2)=O)CC12CCC2 CP(C)(=O)C1CCC(NC(=O)CSc2cc(F)ccc2F)C1 S(=O)(=O)(c1ccc(NC2CCS(=O)C2)cc1Cl)NCc1c(C)ccs1 C(=O)(C1=CCC(NC(C2CC2C(F)(F)F)=O)C1)NCc1ccc(C#N)s1 CC1C(NC(C2(F)CC2c2ccccc2)=O)CCN1C(=O)C(c1ccccc1)=O N1(C(c2ccc(OC)s2)=O)CCC(C2CC2NC(=O)COCCSC)CC1 C(=O)(C1=CC2C=CC1C2)N(CCCCNC(C(N1CCC(C)CC1)=O)=O)C C=CCCCCC(=O)NCC(CC)(CC)NC(=O)CCOc1ccccc1OC C1(C(=O)NC(C(=O)N2C(C(=O)NC)CC2)C)OCCCC1(C)C C(c1ccc(O)cc1)=CC(=O)NCC=CC.c1(C(C=O)O)ccc(Cl)cc1.N N1(C(COc2cn(C)nc2)=O)CCC(F)(CNC(c2n[nH]c3c2CCC3)=O)CC1 CC(C)(O)C(C)(CO)NC(C1CC12CC(NC(=O)C1=CCCCC1)C2)=O c1(Cn2cc(NC(N(C)Cc3nncs3)=O)nn2)ccccc1 N1(C(C(c2nc(F)ccc2Cl)C)=O)CC(C)(C)OCC1CNC(C1(F)CC1)=O Cc1sc(C(N2CCCC(O)(CNC(C3(CCF)CCC3)=O)C2)=O)c(C)c1C Cc1c(NCCc2nc(C(C)C)n[nH]2)ncnc1N1CCN(CCC#N)CC1 c1(C(=O)NC2CCCN(C(c3nc(CCOCC)oc3)=O)C2)nccc(Cl)c1O Cc1[nH]nc2sc(C(=O)N(CC(C)NC(c3ccccc3F)=O)C)cc12 c1(N(C2C3CNCC23)C(c2cc(Cl)c(O)cc2O)=O)ccnc2cc(Br)nn12 c1(-c2c(C(=O)NCCCOCCOC)cccn2)cnc(OC)c(C)c1 c1(C(N2CCN(C)CC2c2nn[nH]n2)=O)coc2cc(Br)ccc12 Cc1cc(F)ccc1CC(=O)NC1CN(C(C2CCOCC2(C)C)=O)CC1O C1(NC(c2ccnc(F)c2)=O)CCCN(C(C2CC3CCC(C2)C3)=O)CC1 N1(C(c2ccc(C#N)s2)=O)CC2(CCC(NC(c3ccc(Br)cc3Cl)=O)CC2)C1 c1(C(=O)NC2CC(O)CN(C(c3cc(C(F)F)cs3)=O)C2)cc2ccncc2[nH]1 c1(OCC=C)ccc(C(=O)NCCNC(C2(C3CCCCO3)CC2)=O)cc1 c1(C(N2CC(CN(C(=O)CN3C(=O)CNC3=O)C)C2)=O)cc(O)ccc1O c1(C=O)nn(C)c(N)c1C.Cc1nc(C)c(C(=O)NCc2ncoc2CC)s1 n1(CCC)nc(C)c(C(=O)NC2C3CN(C(=O)CC(C)n4cccc4)CC23)c1C c1(OC)cccc2[nH]c(C(=O)N)cc12.N1(CCC(=O)N(CCC)C)CCC(F)C1 CCCCC(CCCC)C(=O)NCC1(COC)CN(C(=O)CCn2cccn2)C1 C1(CNC(C(C#C)(C)C)=O)(NC(=O)Cc2ncccc2C)CC2CCC1CC2 Cc1ccc(-n2cc(C3COCCN3C(c3n[nH]c(O)n3)=O)nn2)c(Cl)c1 C(=O)(C(CCNC(c1ccsn1)=O)OC)N1CCC(CC#C)C1 CC1CCC(F)(C(=O)NC2C3CCC(C3)C2C=O)CC1.C1CCC1.N(C)C.N C1(C(=O)OCCc2n(C)cnc2)CCN(Cc2ccccc2)CC1 Cc1c(C(N2CCC(F)(C(=O)Nc3ccnc(OC(F)F)c3)C2)=O)cccc1F C1(C(C)C)CN(C(C2CC(=O)NC2(C)C)=O)CCN1C(=O)C(C)CC#N C=C(C)CCC(C(=O)NCCSC)N(C(C)C)Cc1ccc(C)s1 C=CCC(CNC(=O)OC(C)(C)C)C(=O)N.CCCC(C)C.C(=O)C=CSC N1(C(CC(CCC)C)=O)CC(=O)N2CCOCC2(CNC(=O)C(N)=O)C1 C(=O)(C#CC1CCOC1)NCC1(CNC(CCc2ccc(C)cc2)=O)CC1 C1(C(N2CCC(CC)C2)=O)CC1C1CCCC1.c1(C(=O)N)csc(C(C)(C)C)n1 C(=O)C=C1SCC(=O)N1C.C1(O)(CC#C)CC(C(=O)NC(C)C2CC2)C1.N CC(CC(=O)N1CCSC(C)CC1)C(C)(C)NC(C1CCCC(=O)C1)=O C1(CCOC)CCN(C(C2CC23CCCC3)=O)CC1.c1(CC(=O)N)nnc(O)s1 C=CC(CCC)CC(=O)NC(c1cn(C)nn1)C(=O)NC1CCN(C)C1 c1(C(=O)NCCCN(C(C)C)C(C2(F)CCOC2)=O)ccc2nc(CO)[nH]c2c1 C1(C)(CC)CC(NC(c2cn[nH]c2)=O)CN1C(c1ccnc(O)c1)=O CC1OC2CCC1(NC(C1COCCN(C(C3(C)CCCN3C)=O)C1)=O)C2 C1(CNC(C(CCC=C)(C)C)=O)CCC2(CO1)CC(NC(C1CC1F)=O)C2 Cc1ccc2nonc2c1NCC(N1CCc2nc(-c3ccccc3)sc2C1)=O c1(N2C(CCCNC(C(C3CCCCC3)OC)=O)CCC2)ccc([N+](=O)[O-])cn1 c1(OCC(=O)N(CCCCN(C(C=C(C)C(C)C)=O)C)C)cc(C)ccc1C Cc1ncc(Br)c(C(=O)NC2(c3nc(-c4ccccn4)no3)CCN(C)CC2)n1 C(=O)(C(=O)N=S(C)(C)=O)N1CCCC(N(c2cc(N(C)C)ncn2)CCO)C1 N1(C(c2nc(OCC)oc2)=O)CCC(NC(C2OC(C)CC2C)=O)C(F)C1 Cc1cnn(C)c1CNC(C1CC(C)(NC(=O)CC2CCCC2O)C1)=O CCCCC(C)C(=O)NC1CC1(c1ccccc1F)C(=O)O C1(C(N2C(CNC(=O)CC3C=CCC3)CCC2)=O)CC2CC(O)CC(C1)C2 C1(N(C(C=CCCC(C)C)=O)CCO)CCCN(C(=O)CS(=O)(=O)N(C)C)C1 c1(C=O)ccc(F)c(O)c1.Cc1nc(C(C)C)oc1C(=O)NC1CC(CC)C1 C1(NC(C(CCC)C)=O)CCC2CN(CC(=O)N(C)C)CC2C1.C1CCO1 C1(C(=O)NCCC=C=C)C=CCN1C(c1ccon1)=O C=CC(CCC)CC(=O)NC1CC2CC(NC(=O)C(C)(C)n3cnc(C)c3)CC12 C12(NC(c3ccc(O)cc3)=O)CCC(CC1)C2.c1(C=O)cc([N+](=O)[O-])n[nH]1.N N1(C(CC=CC)=O)CCC2CN(C(c3cc(C(F)(F)C(F)(F)F)on3)=O)CC2C1 C12(C=O)CCCCC1CS(=O)(=O)C2.N1(C(C(=O)NCC2CC2)=O)CCCCC1 C1(C(N2C(CCOC)CN(C(=O)C(O)C(F)F)CC2)=O)CN2CCN1C(C)C2 Cc1csc(C(C)NC(=O)CNC(=O)CCCF)n1 CC(C)C(C)(F)CNC(C1(NC(C2CC2C(N)=O)=O)CCN(C)C1)=O c1(C(=O)NC(CCNC(c2cc3nc(C)sc3[nH]2)=O)C)nccc2cccnc12 CCC(C)C(CC(=O)NC(C)CCCO)NC(C1Cc2ccccc2C1)=O Cc1cc(Cl)ccc1OC(C)C(=O)NC(C(N)=O)C1CCCO1 N1(C(C#CC)=O)CCOC2CN(C(c3cc(F)c(F)c(Cl)c3)=O)CC12 C1(CN(C)C(C2CCC3(CC3)C2)=O)COCCN1C(c1ccncc1Cl)=O N1(C(CC(=O)NCC)=O)CCC(CNC(C2CCCN2C)=O)(OC)C1 N1(C(C(C(=O)OC)OC)=O)CC2(CC2)CC1CNC(=O)C.CC(F)F.S c1(CNC2(CC=C)CNC2)cn(C)c(=O)c2cnccc12 C1(NC(C(Cc2c(C)nc[nH]2)O)=O)CC2CCC(C1)N2C(=O)CC(F)(F)C(C)C c1(CC)n[nH]c(=NC(C)CN(C(=O)C=Cc2ccc(F)cc2F)C)o1 S(=O)(=O)(C(C)C(=O)OC)NC1CCN(CC(=C)C)CC1 N1(C(C2C(C)CC2)=O)CC2(CCC2)CC1C(=O)N(C)CC1CCOCC1 c1(NC(C2CCN(S(CCC=C)(=O)=O)CC2)=O)c(C#N)oc2ccccc12 CC(C(=O)N(C1CC(C(=O)NC2(CCO)CCC2)C1)C)S(C)(=O)=O c1(N(C)Cc2ccccn2)nccc(=NCCCN=c2cc[nH]cc2)[nH]1 N1(C(C)=O)CCC2CCC(C1)S2.C1(CC(=O)NCC)(OCC)CC1.C(C)=O C1(NC(c2nn(C)c(Cl)c2)=O)CCC12CN(C(c1c(C3CC3)cccc1F)=O)C2 c1(CC)cc(NC(C2C=CCN(C(=O)CN3CCC(C)C3)C2)=O)cc(O)c1 C1(C)(C(=O)NC(CCC)CNC(=O)C=CCCC(C)C)CCCCNC1=O C1(C(N(CC(C)SC)C)=O)(CNC(=O)C(C2CCOCC2)F)CCCCC1 Cc1csc(C(=O)NCCCOCCOCC)c1Cl.c1(C(=O)N)cccn1C C1(C(=O)NC2(C3N(C(CCN(C)CC)=O)CCC3)CC2)CCc2cnc(C)n2C1 N1(C(C2C(OC(C)(C)C)C2)=O)CCCC2(C1)CN(C(c1cnncc1O)=O)C2 C1(NC(C2C(C)(C)C2)=O)CCN(C2CN(C(=O)C=C3CCOCC3)C2)CC1 n1(CC)nncc1C(N1CC=CC1C(=O)NCC(C)SC)=O C1(CNC(C2CCCN(C)C2)=O)CCCCCN1C(C1CC(F)C(=O)N1)=O C(c1ccc(F)c(C)c1)=CC=O.C(=O)(C(F)(F)c1csc(Cl)c1)NCCCC N1(C(CC(C)O)=O)CC2CN(Cc3ccccc3N3CCCC3)C2C1 n1(CCC(=O)NCC(CC)NC(c2cnc(S)[nH]2)=O)ccc(O)nc1=O Cc1cnc2cc(C(=O)NCC3(CC)CC3)nn2c1.C1(C)(C(=O)N)CCCC1 c1(C(=O)NC2(OC(C)C)CCC2)coc2ccc(F)cc12 C1(NC(C(C)OCC#C)=O)CCOC12CCN(C(c1cc(C)c(C)nn1)=O)CC2 c1(C(=O)NC(CNC(CCSCC(C)C)=O)C)cc(C(C)(C)C)n(C)c1C CCC(CCCC(=O)NOCC(O)CO)NC(=O)C=C(C)COC c1(C(N2CCCCC2)=O)ccc(=O)n(C2CC2)c1.CC(C(=O)NC)=C1CCC1 N1(C(C2C(CC)CCN2C(=O)Cn2cc(CO)nn2)=O)C2CCCC1CC2 C1(CNC(CCCC)=O)CN(C(C2(CO)CC(C)(C)C2)=O)CCO1 c1(C(CCC)NC(C2CC2NC(=O)CO)=O)cccc([N+](=O)[O-])c1.CC C1(CS(=O)(=O)NC)NC(=O)N(C)C2=C1C(=O)N(c1ccc(Br)cc1)C2=O Cn1cc(C=CC(=O)NCC2CCCC2)cn1.C12(C(=O)N)CCN(CC1)C2 CC(C)CC(C)CN=C(NCc1n[nH]c2c1CCCC2)NC(C1CC1)C1CC1 Cc1nnc2n1CC(C(=O)NC1CC(O)CN(C(=O)CNC(N)=O)C1)CC2 c1(CNC(C(C)NC(=O)C(C)(C)C2CCCO2)=O)ccc(O)cc1 c1(C(N2CC(C)C(CCNC(=O)COc3ccon3)C2)=O)cc[nH]c2nccc1-2 C(=O)(C1CCCc2nc[nH]c21)NCCCC1(NC(CCCCCC#N)=O)CC1 C1(NC(c2c(OC(C)C)n[nH]c2)=O)CN(C(=O)CS(N)(=O)=O)CC(C)(C)C1 C(N=c1[nH]ccn2nc3c(c12)CCCC3)C1CCC(C)CO1 C1(C(=O)NCC(C2CC2)NC(=O)C2CC2)CC(C2CCOCC2)=NO1 c1(C(N(CCCC(=O)NC(C#CCC)(C)C)C)=O)cc(C)ccc1O N1(C(CC(=C)C)=O)CC(CCNC(C2(OC)CC(C)C2)=O)C(C)C1 CCCCCCCCNC(=O)C(=O)NCC(C(C)C(C)C)NC(c1cnn[nH]1)=O CCC(O)C(C)C(=O)NC(C1CCCC1)CNC(c1cnn(C2CCC2)c1C)=O N(C(=NCC(C)(C)C)NCC(c1ccco1)N(C)C)C(COC)C C1(C(N2C(C(=O)NC(CCC=C(C)C)C)CC3CC32)=O)CC(=O)NC(C)C1 N1(C(C2(C)CCC(C)C2)=O)CC2CC(C1)N(c1ncnc(-c3ccccc3)n1)C2 C12(C(=O)NCCC3(CNC(=O)C4=CCSC4)CC3)CCCCC(=O)N1CCC2 C1(CNC(C(C(C)C)CO)=O)CCCC2(CN(C(=O)C(C)N(C)C)C2)O1 C1(CCN(C)C)(C(N2CCC(SC(F)F)C2)=O)CCCCC1 C1(NC(C(C)C)=O)CCOC12CCN(C(c1ccn3ccnc3c1)=O)CC2 c1(CCC(=O)NCC(CN(C)C(C2(C)CC2F)=O)(C)C)ccc(F)c(F)c1 C1(C#N)(OC)CC(C(=O)NCC(C)N(C(=O)C(F)Cc2ccccc2)C)C1 N1(C(CC(C)SC)=O)CCC2(CNC(=O)Cc3ccc4c(c3)CCC4)CCCC12 c1(C(c2nnnn2CC=C)NCC=C=C)coc(C)n1 C1(CC)NC(=O)NC1=O.C(CSC)(C(=O)N)NC(C)=O.C1CC(CC=O)C1 C(=O)(C1=NOC2COCC12)NC1CN(C(CCNC(N)=O)=O)CC12CCC2 c1(C(N(C2CN(C(C3CCN(C4CC4)C3=O)=O)C2)C)=O)nnc(O)nc1O N(C(=NCCCN1CCc2ccccc21)NC1CCC1)CC(C=C)C c1(C(=O)NC2CC(NC(c3cnc(-c4ccoc4)s3)=O)C2)cccc2cnsc12 Cn1cc2c(n1)CC(C(N1CC3CC3C1)=O)CC2.c1(C(=O)N)cc(C(N)=O)cs1 c1(CCC(=O)NCC(C(CC)CC)N(C)C)ccc2c(n1)NCCC2 C1(CC(=O)NCCN(CCC)CC)CN(C(=O)COCC)CCC1C N1(C(CCN(C(c2c(C)ccs2)=O)C)=O)CCOC(C2(C)N=N2)C1 N(C(=NCCCCl)NCC1CC12CCSCC2)CC(C)(C)C C1(NC(CCOC(C)C)=O)CN(C(C2CC2c2ccsc2)=O)CC1N=[N+]=[N-] c1(C=O)cnc(C)c(C#N)c1.C12(C(N3CC(CC)(CO)C3)=O)CC3CC1C2C3 Cc1cc(Cl)c(C(=O)N(C)CC2(O)CCN(C(C3CCCS3)=O)C2)cc1[N+](=O)[O-] c1(C=O)cc(F)n(C)n1.c1(C(C)OCC)nc(C(=O)N(C(C)CC)C)cs1 n1(C(C)(C)C)ccc(C(=O)NCC(O)C)n1.C1(C)(CCC(=O)N)CC1(F)F CC(C)C(C(C)NC(c1ccc(O)nc1)=O)NC(c1cccc(C(N)=O)c1)=O c1(C(=O)N)c(F)ccc2ccoc12.Cn1ncc(C(=O)NCC(F)C)c1C(F)F C(=O)(C1CNc2ccccc21)N1C(C)CC(NC(C2(C)CCCO2)=O)CC1 C(=O)(C(C)C(C)(C)C)NCC1N(c2cc(C)ncn2)CCCC1 CC1CN2CCN1C(C(=O)NCC(O)CN(C(=O)C=Cc1cnc[nH]1)C)C2 c1(C(N2C(CCNC(C(C3CC3)OC)=O)CCCC2)=O)cc(F)c2[nH]nnc2c1 c1(N(C2CCN(C(c3cnc(C(C)(C)C)[nH]3)=O)CC2)C)nc2ccccc2s1 CC(C)C(C(=O)NC(C)CNC(=O)Cc1nc[nH]n1)N(C)C c1(C(N2CCC(N(c3ncc(C#C)cn3)CCO)CC2)=O)ccnc2ccsc12 c1(NCCC2(COC)CC2)ccc(S(=O)(=O)N(C(C)CS(C)=O)C)cn1 CC1CCCC(S(=O)(=O)NC(C2CCCCC2)(C)CO)C1 CC1(NC(c2cccnc2C(N)=O)c2nnnn2C2COC2)CCSCC1 N1(CCCOC)C2CCC1CN(C(c1ccc3nn[nH]c3c1)=O)C2 C1(NC(c2ccc(OCC(F)F)cc2)=O)CCCCN(C(c2ccsc2Cl)=O)C1 c1(C(N2CCC(NC(Cc3c(C)cco3)=O)(CO)C2)=O)cnc2c(ccn2C)c1 Cc1cc(C(=O)NC(Cc2cc[nH]n2)C(N2CCN(C3CC3)CC2)=O)n(C)n1 C1(C=O)CCCC(C(F)(F)F)C1.C1(NC(C(C)=C(C)C)=O)CC(O)(C)C1 C1(CNC(C2(CC)CC2(F)F)=O)CC2CCC1N2c1ncc(C)c(O)n1 c1(C(=O)NC2CC(CCC(=O)NC(c3cn(C)cn3)C)C2)ccc(F)cn1 N1(C(C(C)C#N)=O)CCOC(NC(=O)CCCc2nc(CC3CC3)no2)C1 C1(O)(CNC(CC2C(C)=NOC2=O)=O)CCN(C(=O)CCc2nc[nH]n2)CC1 C(=O)(C1CCCn2cc(C)nc21)N1CC(NC(c2c(CC)nco2)=O)C(F)CC1 C1(C(N(CC(C)(C)CNC(=O)COCCF)CC)=O)CN2CCN1CC2C C(CC1=CCN(C(=O)CSC(F)F)CC1)NC(C(Cc1c(C)cccc1)C)=O c1(CNCCC(c2cnn(C)c2)C)cn(C)nc1C1CCC1 c1(CC)ncccc1C(=O)NCC(C)(F)CNC(=O)C(C)=CC(C)(C)C C12(C(=O)OC)CN(C(=O)NC(c3c(O)cccc3F)C)CC1CCCO2 Cc1cc(C(N2CC3CC3(NC(=O)CC3CC3c3ccccc3)C2)=O)ccc1O C1(c2n(C(CC)(C)C)nnn2)(NCc2sncc2Br)CCN(C2CC2)CC1C C(c1coc(-c2ccccc2)n1)=CC(c1csc(-c2ccc(F)cn2)n1)=O N1(C(CN(C(C(CCSC)(C)C)=O)C)=O)CCC2CN(C)CC2C1 N1(C(CCOC(C)=O)=O)CCN(C(=O)CN(C(=O)CS(N)(=O)=O)C)CC1 C=CC(C)C(C)C(=O)N1CCN(CCCNC(=O)C(C)(C)CN(C)C)CC1 N1(C(c2cc(-c3cn(C4CC5CC5C4)nn3)no2)=O)CCOCC12CC2.CCO.C C(=O)(CCC1CCCC1)NCCCNC(CSC(C)(C)C)=O C(CCC(=O)N1CCC1CNC(c1sccc1CN(C)C)=O)=CC c1(OC)ccc(C(=O)NNC(=O)NC2COCCC2O)c(OC)c1 Cc1ccc(NC(=O)C(N2CCC(C(F)F)C2)=O)c(C)c1.C(=O)COC(F)F c1(C(=O)Nc2ccc(Oc3ccc(C)cc3)nc2)cccc(O)c1F c1(C(=O)NC2(CNC(CSCC(N)=O)=O)CC2)coc2cccc(O)c12 C1(C(N2CC(C(C)C)N(C(=O)C3=CCCS3)CC2)=O)CC2C=CCC(C1)C2 c1(C(N)=O)cc(=NCC2CCCC(NC(c3cc[nH]n3)=O)C2)[nH]cn1 C1(N(C(C(CO)NC(c2c(C)coc2)=O)=O)C)CC2CCC1CC2 n1(CC)cnc2[nH]c(=NCCCCF)nc(OC)c12 CCCC(C)(O)CC(=O)N(C(C)C(=O)NOC1CCCCC1)C N(C1CN(C(c2nccc(Cl)c2F)=O)CCc2ccccc21)C(CC(=O)OC)=O CC1CCN(C(c2ccc(C3CC3)o2)=O)CC1N(C)C(c1cnc2n1CCS2)=O CC1C(NC(c2cnn3cc[nH]c23)=O)CC2CCC1N2c1ncnc2c1CCC2 Cc1[nH]nc(C(N2CC(CNC(=O)CN(C3CCC3)C)C(C)C2)=O)c1C C(=O)(NNc1cccc(C#N)n1)Nc1ccc(C(C)(C)N)cc1 c1(-c2ccc(C)cn2)nc(S(=O)(=O)CC2CCCS2)sc1C CC(C)C(C)CC(=O)N1CCC(NC(c2ccc(O)nc2Cl)=O)CC1C c1(-c2cn(C(C)C(=O)NC3CCC(C(N)=O)C3)nn2)ccc(S(N)(=O)=O)s1 Nc1cc(C(=O)NCC2CC(NC(=O)CC3CC34CC4)C2)nc2ccccc12 C1(CC(=O)NC)CN(C(=O)CCCC(N)=O)CCN1C(C1CCCCN1C)=O c1(C(=O)NC(C(C)NC(c2cc(C(CC)CC)no2)=O)C)c(C(C)C)n[nH]c1C C(=O)(C#CC1CCCC1)NCC(C)N(C(=O)CCCc1ncco1)C Cc1cc(C)n2nc(CC(=O)NCc3cc(C(F)(F)F)cnc3C)nc2n1 C1(NC(C(COC)(F)F)=O)CN(C(C2(C)CCC(=O)N(C)C2)=O)CC1N=[N+]=[N-] C1(NC(C(CC)O)=O)CCN(C(c2nnn(C)c2C(F)F)=O)CC12CCC2 N1(C(C2(N(C)C)CCCSC2)=O)CC(C2CN(C(=O)Cc3ccsc3Cl)C2)C1 C(CC(O)C(=O)NCCC1(C)CCN(C(C2(C(C)C)CCOCC2)=O)C1)SC c1(NC(C2(F)CCN(C(CCc3cc(OC)ncc3)=O)C2)=O)c(O)cccc1F C1(C(=O)NCC(CCC)OCC)CCN(C(=O)CC2OCCCO2)C(C)C1 CS(=O)(=O)CCCNC=O.N1(C(C)=O)CCN(c2ccc(C(=O)O)cc2)CC1.N Cc1cc(C(=O)NC2CN(C(c3ccccc3F)=O)CCC2CO)nc(C)c1 N1(Cc2cccc(SC(=O)N(C)C)c2)CCC2(CC1)Cc1ccccc1NC2=O C(=O)(C(O)C1=CCCCC1)NC1(CNC(c2ccc(Cl)s2)=O)CCOC1 N1(C(=O)CC2CCOC2)CC2CC(C1)N2C(=O)Cc1ccnc(Br)c1 Cc1cc(C)c(C(=O)NC2CC23CC(NC(=O)CCCc2ccncc2)C3)s1 C1(NC(c2c(C)n(C)nc2)=O)CN(C(c2n[nH]c(=N)s2)=O)Cc2nccn2C1 C1(C=O)C2CC(CC2F)N1C(=O)CN1C(=O)CSC1=S.c1(CC)ccccc1.N C(=O)(C1CCNc2cc(F)ccc21)N(C)CCn1cc(-c2ccsc2)nn1 N1(CC)CC(C(=O)N2CC3NC(=O)c4ccccc4C3C2)c2ccccc21 C1(C(=O)NCC=CCNC(C2(O)CCSC2)=O)CCS(=O)CC1 n1(C(CC)CC)ncc(C(=O)NCC(C2CC2)NC(=O)CC2CCCSC2)c1C Cc1ocnc1CNC(=O)COC1CN(C(=O)C(F)=CC2CC2)C1 C1(COC(c2nc(C(C)OC)oc2)=O)CC(Cc2ccccc2)CCO1 N1(C(C2CCC(OC)CC2)=O)CC2(CCCC2N=c2nc(C(F)(F)F)[nH]s2)C1 c1(N2CC(COC)OC(C)C2)nc2c(c(=NCc3cnc(C)[nH]3)[nH]1)SCC2 CCC(CC(=O)N1CC(C)(C(N2Cc3ccnn3CC2C)=O)C1)C(C)(C)C Cc1cc(C)n(CC(=O)NC(C)CCCNC(c2ccn(C3CC3)n2)=O)n1 CCCCCC(C)CC(=O)N1CCC(NC(c2ccc[nH]2)=O)C12CCC2 N1(C(C(C)OC2CCCC2)=O)CC2C3CCC(C2C1)N(c1ccc(C#N)nc1)C3 c1(C(N2C(CNC(c3c[nH]nc3[N+](=O)[O-])=O)CC2)=O)ccc2cnsc2c1 Cc1noc(Cl)c1CCC(=O)NCC1CC(F)(C)C1.c1(CC=O)nccn1C N(C1CCc2cccnc21)C(CC=CCNC(COCCOCC)=O)=O N1(C(C2(C=C)CC2)=O)CCC(O)(C(C)CNC(c2sc(Br)nc2C)=O)C1 C12(NC(CCN(CCCCC)C)=O)CCC1CN(C(=O)CCCSC)C2 C1(NC(COCC)=O)CC2CN(C(c3ccc(C)cc3)=O)CC12.C(N)=O.N c1(C(N2CC(O)(C(C)NC(C(CC)NC(N)=O)=O)C2)=O)cccc2ccoc12 c1(CN=C(NC(C)C2CC2)NCC23CCCC2CCC3)cn(CCO)c(=O)nc1O CCCC(C(=O)NCC(C)(F)CNC(c1cc(CO)on1)=O)OC C1(C(=O)NCCN(CCO)CC)CN(C(=O)CCC(C)(C)C#N)CC12CCC2 C1(C)(CNC(C(C)(C)F)=O)CCCC1.c1(C(=O)N)cnncc1C(F)(F)F C1(O)(CC(C)C)CCN(C(=O)C(=O)Nc2cnn(CC3CCOC3)c2)CC1 c1(C(=O)N)c(C)nc(C2CC2)nc1C.C1(C(=O)NCCCC)(CC)CCNC1=O c1(-c2c(C(C)(C)C)noc2)cccc(N)c1[N+](=O)[O-] CC(O)(C(=O)NCCc1ccc(C(=O)NC2CCC(C)CC2)cc1)C(F)(F)F c1(C(N(CC(C)(C)CNC(=O)COC(F)F)C)=O)ccccn1.c1cn[nH]c1 CC1CC(C(=O)NCc2ncoc2C2CC2)CCN1C(c1cc(C#N)cs1)=O N1(C(CN(C2CCS(=O)(=O)C2)C)=O)CC2CC(C1)C2.C1(C=O)CCCCCC1.N c1(C(=O)NCC(N(C(CC2N(C)CCCC2)=O)C)C2CC2)cc2ncccn2n1 CN1CCC(C2(C(=O)NCC3CCN3C(c3c(F)cncc3Br)=O)CC2)CC1 c1(CCn2cc(CN3CCC(c4c(OC)cccc4)C3)nn2)ccc(O)cc1O CCCC(C(=O)N1CC(CC)C1)OC.c1(C(=O)N)ccccn1.CC(F)F.C(C)=O C1(NC(c2cc(CC)oc2C)=O)CC(O)CN(C(c2cncc(C)c2)=O)C1 N1(C(CC(C(C)C)C)=O)CC2(C(=O)NCc3ncccn3)CCC1CC2 C(=O)(CC1CS(=O)(=O)c2ccccc21)N1CCCN(C(C2CC(=C)C2)=O)CC1 C(CC(C(C)(C)C)NC(C1CC(C#N)C1)=O)N(C(c1c(C)ocn1)=O)C C(=O)CC(C(F)(F)F)N(C)C1CC1.C1CC1C(=O)N(C(C)C1CC1)C.C Cc1ccc(CNC(C2CC2CNC(=O)C(C)CO)=O)nc1C n1(CC(C)C)ccc(CC(=O)N(CCC(C)NC(C2(c3cncs3)CC2)=O)C)n1 N1(C(C(C)OC)=O)CC(NC(=O)Cc2ccc(C)nc2)CC(F)(F)C1 N#CC1CN(C(c2ccc(F)cc2)=O)CC1NC(=O)CCNc1ccccn1 C12(C(=O)NCc3cccnc3N3CCCCC3)CCCCC1OCC2 CC1CC=CCC1CN1CCOC(c2ccc(C(F)(F)F)cc2)C1 C=CC(C)(O)C(=O)N.C1(=CC(N2CC(CC)C2)=O)CCC(C(C)(C)C)CC1 c1(C(=O)NC2CCC(CNC(c3ccc(CCCCC)o3)=O)C2)c(C)n[nH]c1C c1(C(C(=O)N(C(CNC(C(CCC)O)=O)C)CC)OC)c(F)cccc1F C1(C(N2CC(C)(C)C(NC(C3(CO)CCCC3)=O)C2)=O)CCC2C(CC1)C2(F)F N1(C(c2ccc(C(C)O)cc2)=O)CC2CC(C1)N(C(C1CC(CF)C1)=O)C2 C1(NC(c2ccc(C)cc2)=O)CCC(C)N(C(c2cc(C)n(C)c2C)=O)C1 c1(C(N(C2C(C)CCN(C(C(SC)SC)=O)C2)C)=O)cc2ccccn2n1 c1(CC)c[nH]c(C(=O)NCCCC(C)NC(=O)CCc2cnc[nH]2)c1.C(C)=O C1(NC(=O)NC(CC=C)C)(CO)CC2(CCC2)C1 N1(C(C2N(C(=O)OC)CCC2)=O)CC(F)CC1.C1(C(N(C)C)=O)CC(O)C1 N1(C(c2nc(C(C)OC)sc2)=O)CCN(C(=O)CNC=O)C(CC(C)(C)C)C1 c1(C(=O)NCC(C)N(C(c2c(C)cc(CO)o2)=O)C)cc(C)c(=O)n(C)c1 C(=O)(C1=CCCCC1C)N1CCCC(C(N2CC(F)(CO)C2)=O)(CC)C1 C1(NC(C(C(CC)C)O)=O)CCC2(CC1)CN(C(c1nc(C)c(C)s1)=O)CCO2 C1CCS(=O)(=O)C1.c1(C(NC(=O)C)C)ccccc1.CC(C(=O)N(C)C)N c1(CC(=O)NCCCCC(C)NC(=O)C2=COCCC2)ccc2c(c1)COC2 C1(COC)CN(C(C23CC(C=O)(C2)C3)=O)CC1.C1(C=O)CCOC(C)C1 C1(O)(C(=O)NC(c2cn(CC3CCOC3)nn2)C)CCCC(C)(C)C1 C1(NC(c2c(C)n(C)nc2)=O)CC2(CCN(C(=O)C(F)Cc3ccccc3)C2)C1 C1(NC(CS(CC)=O)=O)CCC2(CC1)CC2NC(c1cc(OC)ccc1Cl)=O S(=O)(=O)(c1ccc(Br)cc1C(F)(F)F)N1CC2(CCC2)C1.N1CCC(F)(F)C1 c1(OCC)ccc(C(=O)NC2C3CC2N(C(c2cc(C=O)no2)=O)C3)cn1 Nc1cc(C(N2CCCC(CCNC(C34CCN(CC3)C4)=O)C2)=O)c(F)cc1F c1(CC(=O)N(C)CC2C3CN(C(=O)CC4OCCO4)CC23)c[nH]c2cnccc12 C(=O)(C(C(C)NC(c1cc(C#N)[nH]c1C)=O)C(C)C)NC1CC(OC)C1 Cc1cccnc1CC(=O)NCC(O)CNC(c1coc(C(N)=O)n1)=O c1(CNC(C2(C)CCN(C(c3n(C)ncc3)=O)C2)=O)ccc(Cl)cc1F Cc1c(-n2cc(CCCNC(c3cc(Cl)c(Cl)[nH]3)=O)nn2)cccc1[N+](=O)[O-] C1(C(=O)NCC(CC=C)NC(c2ccnnc2O)=O)CCCC12CC2 c1(OCC)ncc[nH]c1=NC(=O)c1scnc1-c1ccc2nncn2c1 c1(CNC(C=CCC)=O)ccnc(C(=O)NCC2CC(C)CO2)c1 C1(C(=O)NC(C(C)NC(CNC(=O)NC)=O)C)(C(F)F)CCCCC1 c1(NC2c3[nH]c(=N)sc3CCC2)nc2ccsc2c(=NCC(CO)C(F)(F)F)[nH]1 c1(OC)cc(NC(C2CC(F)(F)CN2C(C2CNC(=O)C2)=O)=O)c(F)cn1 CC1CCc2nc(NC(=O)COC(=O)C(C)OC(c3ccccc3)C)sc2C1 C1(C(=O)OC)CN(C(CC2CC(F)(F)C2)C(=O)NCC(F)F)CCO1 N1(C(c2n(CC)nc(C)c2)=O)CCC2(CCCC2)C1.C1(=CC=O)CCCCC1.N Cc1cccc(C)c1CNC(=O)C(C1CCN(C(c2nonc2N)=O)C1)C C1(NC(c2ccc(-c3ccco3)[nH]2)=O)CCCN(C(=O)Cc2cncs2)C1 c1(C(=O)NC2C(NC(c3ccc(CC)s3)=O)CCCC2)cccc2c1SCCC2 c1(NC)c(C(N2CCC(CN(C(=O)CO)C)C2)=O)cccc1F.C1(F)CC1 c1(C(c2cccnc2)NCC2(SC)CC2)nnnn1C1CCOCC1 c1(C(=O)N)c[nH]c2cc(Cl)ccc12.C#CC1(OCC(=O)N(CCC)CC)COC1 N1(C(C2OCCN(C(C3(CC#C)CCOC3)=O)C2)=O)CC2(CNC(=O)C2)C1 N1(c2ccnc(C)n2)CC(NC(c2ccc(F)c(C)c2)=O)C(C#N)C1 c1(C(=O)NC2(CO)CN(C(C(n3ncc(C)c3)C)=O)C2)ccc2occc2c1 C(=O)(CCCC(C)c1ccccc1)OCCS(=O)(=O)NCC(=O)OC C1(CNC(C(CC)C#N)=O)CC2(CCN(C(=O)C=Cc3cncs3)CC2)CO1 C1(C(=O)NC2CC(CC)C2)CCC(O)CN1C(c1ccc(NC)cc1)=O C1(NC(c2nc(C(=O)OCC)sc2)=O)CCN(C(c2ocnc2C)=O)C1C.C C(C(O)CC(=O)N1CC(N(C)C)C1)NC(C(C)N1CCCC1)=O C1(C(N2CCCCC(NC(c3c(C)c(Cl)ccn3)=O)C2)=O)CNC(=O)CC1(C)C C(N=c1[nH]c2ccc(N)cc2s1)C1(O)CCN(C(CC2C(C)OC(C)C2)=O)CC1 c1(C2CCN(C(C(=O)N(C(c3cnc(Cl)s3)C)C)=O)C2)ccc(F)c(F)c1 c1(C(N(CC(CC)NC(=O)CCCOc2ccc(Cl)cc2)C)=O)cnnc(O)c1 C1C2CCCC1N(C(c1cc(C(F)F)no1)=O)C2.n1(CC)nccc1C(=O)N.C c1(OCC)cc(CN2CCC(O)C(CO)C2)c(Br)cn1.N12CC(N)C(C1)C2=O N1(C(c2c(Cl)cc(C)s2)=O)CC=C(CNC(c2ccccc2)=O)CC1.N(C)C.C Cc1ccc(Cl)cc1OCC(=O)N(CCC(C)NC(=O)CC1CSCCS1)C C1(C(=O)NCC2(C)CCCN(S(C(CC)C)(=O)=O)C2)Cc2nnc(C)n2C1 c1(N2CCC(CNC(=O)C(C3CCOCC3)F)C2)ncc([N+](=O)[O-])cc1Br C(CCCOC)(C(=O)NC1CN(C2CCC2)C1)NC(c1n(CC)cnc1)=O c1(C(N2CC(CC(=O)Nc3cncc(Cl)c3Br)C2)=O)ccc(F)cc1I N1(C(c2ccc(S(C)(=O)=O)cc2)=O)CCC2CCN(C(C3CC(O)C3)=O)CC2C1 C1(NC(c2nc(C)oc2C)=O)CN(C(c2cc(C)n(C)c2)=O)C2(CCCOC2)C1 Cn1cc(C(F)=CC(=O)NC(C)(C)C)cn1.C1(C=O)CCOC1C(F)(F)F Cc1cc([N+](=O)[O-])cnc1C(=O)NCCC(C)(C)C.C(=O)(CCN1CCCC1)N c1(C(=O)NCCOCCNC(c2c(C)nns2)=O)cc(Br)cnc1N c1(NC(N2CCN(C(=O)OC(C)(C)C)C(C#N)C2)=O)ccc2c(c1)CCOC2 C1(CCC)(NC(=O)C(C)S)CCCN(C(C2C3(CC3)C23CC3)=O)C1.C(C)C Cc1nc(Cl)c(NC(C2CCCC2NCc2cc(Cl)c(Cl)cc2O)=O)nc1C CC1(C(=O)NC2CCN(C(c3ncccn3)=O)C(C3CC3)C2)CCCCCCC1 C1(C(N2CC(O)(CNC(CN(S(CC)(=O)=O)C)=O)C2)=O)CCc2nccn2C1 CS(=O)(=O)c1ccc(C(=O)NC(C(=O)O)C(O)c2ccncc2)c(F)c1 N1(C(COCCOC)=O)CC2(CCC2)CC1C.c1(C=O)n[nH]c2c1CSCC2.N C=CC1(C(=O)NC2CCC(NC(c3ccc(CC(C)C)cc3)=O)C2)CCOCC1 c1(C(=O)OCC)nc(-c2cccn2CCN2CCOCC2)c2ccccn12 CC1(C(=O)NCC(O)CNC(c2ccc(C(F)(F)F)cn2)=O)CCC(=O)N1 C1(NC(C2(C)CC2)=O)CCC2(CCCN(C(c3cnc4ncc(Cl)cn34)=O)C2)C1 Cc1ccc2c(=NCCCC3CCCC3O)[nH]c(=NCc3ccoc3C)[nH]c2c1 CC(O)(CC(=O)N1CC2CCCC(C1)C2C(=O)NCC1(C#N)CC1)CC(=O)O c1(C=O)ccc(C=CC=O)o1.C1CN(C(=O)Cc2cc(C)cs2)C2CC12.C N1(C(C2N(CC)CC2)=O)CC(C)(CNC(c2ccc(Cl)cc2Cl)=O)CC1(C)C C1(C(N2C(C)(CNC(CC(COC)COC)=O)CCC2)=O)CCc2c[nH]nc2C1 c1(NC(c2ccccc2)CF)nc(Cl)[nH]c2ncnc1-2 S(=O)(=O)(c1ccccc1-c1cccc(NCc2cnc(Br)s2)n1)N(C)C N1(C(c2ccc(N(C)C)nc2)=O)CCN(C(c2cc(C(N)=O)cs2)=O)CC(O)C1 C=CC1(C(N2CCC2(C)C(C)C)=O)CCN(C(=O)CCc2cnn[nH]2)CC1 c1(CN(C(Cc2onc(C)n2)=O)C)cc(C(F)(F)F)cc(F)c1 C1(CNC(C(CC)OCC)=O)CN(C(=O)CN(C)C)CCN1C Cc1cc(C(=O)NC2CCN(C(=O)C(C)(C)C3CC3)CC2O)nc(C)c1 C1(CN(C(CCCSC)=O)C)C2CN(C(=O)CCc3cc(Br)cs3)CC12 C#CC(C)(C)CNC(=O)C(CNC(=O)CCc1ccco1)OC C1(C(N2CCC(CC)C2)=O)CCC(=O)N1C.c1(C(=O)OC)csc(C(=O)N)c1 c1(OC)cc(OC)nc(C(N2CCOCC2)=O)n1.C1(C(NC)=O)(C(N)=O)CC1 C1(C(N(C)CCn2cc(CC)nn2)=O)C2Cc3ccc(Br)cc3C12.[SH](C)(=O)=O C(=O)CC(C)(C)C(C)(F)F.CC(F)(F)F.CCCN(C(=O)C=CCN)C CCCC(C)(O)C(=O)N1CC(OC)CC(NC(C2(c3ccc(C)cc3)CC2)=O)C1 c1(CC)cc(C(N2CCC(NC(=O)CCP(C)(C)=O)C(CO)C2)=O)c(C)nn1 c1(COC)cc(NC(=O)C(CC)Oc2ccccc2)ccc1OC(F)(F)F C1(CC(=O)NCCC(C)NC(CCCN(C(C)C)C)=O)CC=CCN1C c1(OCC)cccc(C=CC(=O)N)c1.c1(C(C=O)C)nc(C)cs1.C1CC1 N12CCC3(CC(C3)C(=O)NCCC1=O)C2.C(C=CCl)NC(=O)NC c1(C(N(CCC2N(C(C=CSC)=O)CCCC2)C)=O)cnc2sccn2c1=O c1(C(=O)NCC(CN(C(C=Cc2scc(C)n2)=O)C)C)cc(C)c(CO)cn1 Cc1ccc2[nH]cc(C(=O)NCC3COC(CN=c4[nH]cnc(Cl)c4Br)C3)c2c1 c1(CC)cc(NC(C2C3CN(C(=O)CCCN(C)C(C)C)CC23)=O)cc(O)n1 C(C(CC(C)C)C(=O)N(CCCC)CCOC)NC(CC(C=C)C)=O C1(C2CCCCO2)(C(=O)NC(c2ccccc2)C(C)C)CCCO1 c1(CCC)cc(C(=O)NC2CCN(C(=O)CCCCCOC)CC2O)cc(O)n1 C1(NC(C(CO)N(C)C)=O)CC2(C1)CC(C(N1CC3CC1CN3C)=O)C2 C1(COC(=O)Cc2cccc(F)c2I)OCCOC12CCC2 Cc1[nH]nc(Cl)c1C(=O)NCC1C=CC(NC(c2cc(CO)oc2C)=O)C1 c1(C(=O)NCC(C(C)(C)C)NC(=O)C2=COCCC2)cccc([N+](=O)[O-])c1 Cc1cc(C(N2CCCCC2CNC(=O)CO)=O)c2cnccc2c1 C(=O)(CCCCC(=O)N1CCC(C(C)(C)C)(CNC(=O)C(C)C(C)O)C1)NC C(=O)(C(C)(C)CCCF)NC1C(C(C)C)N(C(=O)CCc2ccccn2)CC1 C1(CC)CN(C(=O)C(C)=C2CCC2)CC1C(=O)N(C)C(C)C1CC1 C1(C(CNC(=O)C=C2CCC2)F)CCN(C(c2csc(-c3cn[nH]c3)c2)=O)CC1 C1(NC(c2ccc(C(F)(F)F)s2)=O)(CO)CCCC2CC12 c1ccc(Cl)cc1Cl.C1(C(=O)O)CCC(C=O)C1.C1(O)(C=O)CN(CC)C1.N c1(C(N(C)CCNC(c2ccc(Cl)nc2O)=O)=O)ccnc2c1cnn2C Cc1oc(CNC(CC2=NOC(C)C2)=O)nc1C(=O)O C12(NC(=O)CCCF)CCCC1(F)CN(C(C13CCCC1C3(F)F)=O)C2 C1(C(N)=O)CCN(C(C2CN(C(c3ccns3)=O)CCN2)=O)CC1 C1(CC(N2CC(CC#C)C(O)C2)=O)CCC(N)CC1 c1cnn(C)c1.C(CC(=O)NCC1CC1C(=O)N)NC(=O)OCC N1(C(Cc2c(C)ccnc2)=O)CCCC(NC(=O)CN2CCCNS2(=O)=O)C1C c1(C(=O)NCCCCNC(CN(CCCCCC)C)=O)ccc2[nH]ccc2c1F C=C1CC2(C1)CC(C(=O)NC1CCC1NC(c1c(Cl)cncc1Br)=O)C2 N1(C(C2CC(C)=C(C)CC2)=O)CCCC(C2CN(C(C3(C(C)C)CCC3)=O)C2)C1 Cc1ccc(OCC(=O)N(C)CCn2cc(C3CCCC(O)C3)nn2)c(F)c1 c1(C(NC)=O)ccc(C)cc1C.C1(C)(CC)CC1C(=O)NCC1CC1.C C(=O)(C1CCC(=O)c2cccn21)NC1C(NC(=O)CC2C=CCCC2)CCCC1 N1(C(c2cn(C)c(=O)cn2)=O)CCC2(CCCN2C(c2cc(=O)n(C)cn2)=O)C1 N1(C(C2C(C#N)C2)=O)CC2(CCC(NC(c3nc(Cl)ccc3F)=O)CC2)C1 N1(C(CC(=O)NCC)=O)CCC2(CCCC2)C1.c1(C=O)sc(C2CC2)nc1C.N CC1(C(=O)NCC2CSCCO2)CCCN(C(c2ccc(O)c(F)c2)=O)C1 c1(N2CC3(CN(C(C(C(CC)O)C)=O)C3)C2)nc(Cl)nc2sccc12 c1(CN(CCc2nnco2)Cc2ccccc2)ccnc(C2CCC2)n1 C1(C(=O)NC(CNC(CCCCCOC)=O)C2CC2)CC2(C1)CC1(CC1)C2 C1(CN(C)C(C2(C(C)(F)F)CC2)=O)COCCN1C(=O)CCN1CCOCC1 C1(C(N(CCN(C(=O)CS(=O)CC)CC)CC)=O)CC2(C1)CC21CCC1 C1(CNC(c2ncnn2C2CCOCC2)=O)C=CC(NC(C2CCC2)=O)C1 c1(C(N2CC=CC(NC(C(C)OCc3ccncc3)=O)C2)=O)coc2c1COC2 CC1OC2CCC1(NC(=O)CC1CC1CNC(C1CCCN1C=O)=O)C2 CC1CN(C(=O)CNS(C)(=O)=O)CCCN1C(c1cc(O)cc(O)c1)=O Cc1cc(C(N2CC(C(=O)N(C3CC(F)(F)C3)C)CC2(C)C)=O)nc(O)c1 C12(CC)CC(C1)C(Oc1ccc(C(=O)Oc3ccc(OCC)cc3)cn1)CO2 C1(CNC(C(CC)F)=O)CC2(CCN(C(=O)CSc3ccc(C)cc3C)CC2)C1 Cc1cnc(O)cc1NC(=O)Cc1cccc(-c2cc(O)cc(F)c2)n1 c1(OC)cc(C(N2CCC3(NC(c4cc(Cl)ccc4Cl)=O)CC3C2)=O)ccc1C c1(C2(C(N3CCC(O)C3)=O)CCC2)c(F)cccc1F.C=C1CC1C(=O)NC N1(C(C2=NOC(C)C2)=O)CCOC2CCN(C(c3cn(C4CC4)cn3)=O)CC12 N1(C(COCCC)=O)CCN(C)C(CNC(=O)C(OC)OC)C1 C(=O)(C(CN=[N+]=[N-])NC(=O)Cc1cccnc1)NCC(CCC)O CCC(F)(F)C(C)(C)C(=O)NC1CN(C(C2CCCC(C)(C)C2)=O)C1 c1(OC)c(NCC2(F)CCCN(C(c3cnn(CC(F)F)c3)=O)C2)ncnc1Cl c1(-c2cn(C(C(=O)N(C3(CC)CC3)C)C)nn2)ccc(C)c(Cl)c1 c1(C(N(CCN(C(c2c(C)cccc2C)=O)C)C)=O)ccc2cccnc2c1N c1nn(C)c(Cl)c1C(=O)N(C)CC.c1(C(N(CC)C)=O)cn(C)nn1.CO N1(C(c2c(OC)nsc2)=O)C2CCC(C2)C1C.c1(C=O)cccc(N(C)C)c1 N1(C(C(C=C)(C)O)=O)CCC(NC(=O)CC2CC=CC2)C(C)(C)C1 C(C)(CNC(C1CC1(C)C)=O)(CC(C)C)NC(c1cncc(OC)c1)=O Cc1ccc(C(=O)NCC2CCCCN2C(c2cncc(N(C)C)c2)=O)cc1F N1(C(C2N(C(Cc3cn(CC)nc3)=O)CCC2C)=O)CCCC(F)(CO)C1 C1(CCNC(Cc2c(C)nsc2)=O)CCCCN1C(=O)CCC(N)=O C1(C(=O)NCC#CCNC(C(CC)C)=O)COCC2(CCC2)O1 N#Cc1cccc(-c2n[nH]cc2C(N2CC(NC(C3CC4CC4C3)=O)C2)=O)c1 C(=O)(C#CC1CCCCO1)N1C2C(NC(c3c[nH]c4cccnc34)=O)CC(C2)C1 C(=O)(C1=CCCN(C(=O)CCN(C)C)C1)Nc1c(OCC)n[nH]c1 N1(C(C(CC=C)C)=O)Cc2ccnn2CC(NC(=O)CC2(O)CCCCC2)C1 N1(C(Cn2cc(C(=O)NC)nn2)=O)CCC(C)N(C(=O)CNC(=O)O)CC1 N1(C(c2c(CC)cco2)=O)CCCC12CCN(C(=O)C(C)C(F)F)CC2 C1(C(N(C(C)C(=O)OC)CC)=O)CC(NC(c2n[nH]cc2C)=O)CCO1 c1(CC)nc(C)[nH]c1C(N1CC(NC(C2(c3ccccc3)CC2)=O)CC1C)=O c1(C(N2CCC(NC(CCCc3nc(C)sc3)=O)C2)=O)cc(Br)n(C)n1 CC1(C)CN(C(=O)CCc2nc(-c3ccsc3)no2)CCO1.C(=O)(CC1CC1)N c1(CNC(=NC)NCC(C)Oc2ccc(F)cc2)cccc2ncn(C)c12 C1(C(=O)NCCNC(N(C)C)=O)CCCN(C(=O)COc2ccon2)C1 c1(C(N2C3C(NC(C4CC5CC5CO4)=O)C(C3)C2)=O)cc(F)cc([N+](=O)[O-])c1 c1(OC)ccc(F)c2c1CCN(C(=O)C(N1CCCC(CS)C1)=O)C2 n1(CC)nc(C)c(Cn2c(Cc3ccc(C)cc3)nc(-c3cscn3)n2)c1C N1(C(C23CCC(N=[N+]=[N-])C2C3)=O)CCC(C2CCCN(C(c3cocn3)=O)C2)C1 Cc1ccc(C(=O)NC23CCN(C(=O)CCSc4nnnn4C)CC2C3)cc1N C1(NC(c2c(CC)scn2)=O)CN(c2nc(CCOC)ns2)C2CCCCC12 Cc1cnc(N)c(C(N2CCC3CCC23C)=O)c1.c1(C=O)c[nH]c(C(N)=O)c1.N C12(NC(C3C(C=C)CC3)=O)CCC(C1)N(C(=O)CCc1ccc(Cl)s1)C2 Cc1ccc(OCC(=O)NCCN(C(=O)Cc2cnoc2)C(C)C)cc1 c1(C=O)c(C(F)(F)F)cccc1[N+](=O)[O-].c1(C(=O)NCC(O)C)ccc(Cl)o1 N1(C(COCCOC)=O)CC2CC(NC(=O)CCc3cscn3)C1C2 c1(C(=O)NCC(C)NC(C2(C)CCCS2(=O)=O)=O)cncc2nc[nH]c12 C1(C(=O)NCC2(NC(C(C)CC3CCC3)=O)CCCC2)Cc2ccncc2C1 N1(C(C2=NN(CC)C(=O)C2)=O)CC2CCCC1C2CNC(=O)CSC(F)F C1(n2ccc(C(=O)O)n2)CCCN(C(c2ccn(C3CC3)n2)=O)C1 C(=O)(C1=CCN(C(=O)Cc2cscn2)CC1)N1C(C(CC)C)CCC1 c1(C=O)ccnc(N2CCCC2)n1.CC(C(=O)NCC1CC1)SC(F)(F)F.C Cc1cccc(C=CC(N2CCCC(C(N3CCC(CF)C3)=O)CC2)=O)c1 C(=O)(CCCCN(C)C(C1CCC(=O)NC1)=O)NC(COC)C1(C)CC1 S(=O)(=O)(CCCC1CCC1)N(C(C(=O)OCC)Cc1ccccc1)C CC1(C)OC2CC(C(=O)NCCC3CCN(C(=O)CSC(F)F)CC3)CC2O1 C(=O)(N=c1cc(C(F)F)[nH][nH]1)C1(c2c(C(N)=O)cccc2)CCC1 N1(C(Cc2ccc(C)nc2)=O)C2CC=C(C(=O)NCC(O)C(F)F)C1CC2 Cc1ncc(CC(=O)NC2(CNC(=O)Cn3ccc(C4CC4)n3)CCC2)[nH]1 C1(C(N2CCC(NC(c3ccoc3)=O)C(F)C2)=O)C2CCC3(COC(=O)C13)O2 C=C(CNC(C1CC(n2ccnc2)C1)=O)CCNC(C1CCCN1CCC)=O N1(C(CN(CCOC)C)=O)CCC(O)(CCNC(C2CCCCC2(F)F)=O)CC1 N1(C(CN(CC)CC)=O)CCC(C)C(NC(=O)Cc2[nH]cnc2C)C1 N1(C(C2(C=C)CC2)=O)CCCC(CCC)(NC(=O)CC2(CO)CCOCC2)C1 N1(C(C(C)C2C(C)C2)=O)CC2CCCC(C1)N2C(=O)CCc1cccc(F)c1 c1(C(=O)NC2(CNC(Cc3nc(=N)[nH][nH]3)=O)CCC2)[nH]nc([N+](=O)[O-])c1Cl N1(C(C(c2ccncc2)C)=O)CCN(C(=O)C=C2CCN(C)C2)C(CCO)C1 C(=O)(C#CC(C)C)NC(C(C)NC(c1c(C)cns1)=O)C c1ccnc2ccccc12.c1(NC(N2C(C(C)C)(C(C)C)CC2)=O)cccc(Cl)c1.N CC1(C)C(CNC(=O)CN(C2CCC2)C(C2(C)COC2)=O)CC1(F)F CC(C)CC(CCO)NC(=O)CCOCCN(C)C(C1(C)SCCCS1)=O c1(C(N2C(C(=O)NCC3(C=C)CCC3)CCCC2)=O)ccc(OC)c(F)c1 CC#CCC(C(=O)NCC1COCCN1C)NC(c1ccoc1Cl)=O c1(C(N(CC(C(=O)N(CCCCCC)C)C)C)=O)c(C)cnn1CC Cc1ccc(F)c(C(=O)NC2CCC(C(N3CC4CC4C3C#N)=O)OC2)c1F C(=O)(C(O)C(F)(F)F)NC1C2CN(C(c3ccc(CCC=C)cc3)=O)C1C2 C(N=c1cc(C2CC2)nc(Cl)[nH]1)C1C(C)CN(C(c2cnc(Cl)[nH]2)=O)C1 C1(NC(c2c(NC)nc(C)cc2)=O)CC2CCCC2C1.C1(C)(C(=O)N)CCCO1 C(c1ccccc1OC(F)F)=CC(=O)N.Cc1ccnc(C(=O)NC2CCC2)n1 Cc1cccc2cc(C(=O)NCC(C)N(C(=O)C=C3CCCC3)C)cnc12 N1(C(c2ccn(C)n2)=O)CCOC(c2cn(CC3COC(=O)C3)nn2)C1 C1(N(C(c2c(C)coc2)=O)C)CCCC2CN(C(=O)Cc3ccc(Cl)cn3)CC12 N1(C(CC(=C=C)C)=O)CC2CCC(C1)N2C(C1CC(=O)N(CCOC)C1)=O C(=O)(C1=CS(=O)(=O)c2ccccc21)N1CCC(C2CCN(C(=O)CC3CC3)C2)C1 O=C(O)CC(C1CCCCC1)NC(=O)CC(O)c1cn(C2CCCCC2)nn1 C1(NC(c2cnn3c2CCC3)=O)C2CCN(C(C3CC4CC(=O)C3O4)=O)CC12 C1(NC(C(c2cnn(C)c2)C)=O)CC2(CCN(C(C3CCS(=O)(=O)C3)=O)C2)C1 C1CCOC2(CCN(C(C3CS(=O)(=O)CC(=O)N3)=O)CC2)C1.O=CC=CCO.N CCC(C#N)C(=O)NCC1CCCCN1C(c1ccnn1C(C)C)=O c1(CC(N2C(C(=O)NCC(=C)C)CSCC2)=O)ccc(Br)cc1C c1(COC)nc(NCCSCCC(F)(F)F)cc(=NCC(C)(C)C2CC2)[nH]1 c1(CCC(=O)NCC2N(C(CC)=O)CCCC2)cccc(F)c1F N1(C(c2c(Cl)cnc(C)n2)=O)CCC2(C1)CN(C(c1c[nH]cc1Br)=O)C2 C(c1ccc([N+](=O)[O-])cc1)=CC(N1CC(NC(CC(C)O)=O)CC(F)(F)C1)=O CCCCC(CCC)NC(C1(CNC(C2CC3CC2CC3=O)=O)CCCCC1)=O Cc1nc(C2CCCN(C(=O)NCC3CC4CCC3O4)C2)oc1C(=O)O C(C(C(=O)NC(c1scnc1C)C)NC(=O)CCCC1CC1)OCC c1(NC(=O)NC2CCN(C(CSC(=N)N)=O)CC2O)ccc2c(c1)OCO2 C1(NC(C(CC)(C)O)=O)CC(C2CCN(C(c3ccsc3Cl)=O)CC2)C1 c1(C2(NC(=O)CSC3CC(C4CC4)=NO3)CC2)nc2ccccc2o1 C1(NC(CCNS(CC)(=O)=O)=O)CN(C(c2csc(CO)n2)=O)CCC1CO N1(C(COCCOC)=O)C2CCC(C2)C1CC(=O)NC1CC1CCOC N1(C(CCCC)=O)CCCCCC(NC(=O)C(C)OCOC)C1 CC1CC(NC(C2CCSC2)=O)CCN1C(=O)C=C(F)c1ccccc1 Cc1cccc(Cl)c1S(=O)(=O)N1CCOCC(NC(c2ccc(F)nc2)=O)C1 N1(C(c2c(C)cc(F)nc2)=O)CC23CCCCC2(C1)CN(C(c1cncs1)=O)C3 CCC(C)(C)CCCC(=O)N1CC2CC(C(=O)NCC(C)C(C)(C)C)(C2)C1 N1(c2cc(NCCc3cccc(OC)c3)ncn2)CCC(C)(F)CC1 c1(C(Cn2cc(C(N)=O)c(O)nc2=O)=O)ccc(Br)c2nsnc12 c1(OC)cc(C(N2CCN(c3cccc(C(F)(F)F)c3)CC2)C(=O)O)ccc1F c1(C(=O)N)cccc(Nc2ccsc2)c1.C(CCCNS(=O)(=O)CC)OC C1(CNC(c2c(OC)c[nH]n2)=O)CN(C(=O)CCN(C2CCCCC2)C)CCO1 c1(CNC(c2nscc2Br)C)cccc2ccsc12 c1(C(=O)NC2CC(C)(NC(CCCN(C(C)=O)C)=O)C2)cccc(C#CCO)c1 C1(O)(CNC(C2CCNC2=O)=O)CCCN(C(c2cccc3nccn23)=O)CC1 N1(C(C2(OC)CCC2)=O)CC=C(CC)CC1.c1(C=O)ccc(S(N)(=O)=O)s1.N C(=O)(CCCCC(N)=O)NC(C(=O)NCc1c(C)c(F)ccc1)C1CCCO1 N(C1CCc2cc(F)c(F)c(F)c21)C(Cn1cc(CN(CCOC)C)nn1)=O C1(CC(N2C(CN(C(c3ccc(CCC)s3)=O)C)CCC2)=O)CCCCC12CC2 Cc1ccc(CC(=O)NCC2CCCCN2C(=O)C(C)NC(C)(C)C)cc1C CC1CCC(C(N2CCC2c2cn(CCn3cccn3)nn2)=O)S1 N1(C(C(n2cc(CCSCC)nn2)C)=O)CCN(c2ccc(F)cc2)CC1.CC.O C(=O)(C1=CC2(CCN(C(=O)CCOCC3CC3)C2)C1)N(c1ccsc1Cl)C C(c1cc(Cl)cc(Cl)c1)=CC(=O)NC1C=CCN(C(c2cc[nH]n2)=O)C1 C(c1ccc(F)cc1)=C(C)C(=O)NC1CC(O)CN(C(=O)CN2CSCC2=O)C1 C(C1c2ccsc2CCN1C(=O)COC(C)C)NC(CC1N(CC)CCOC1)=O N(S(=O)(=O)N(C)C)CC=O.CC(Cn1cccn1)C(=O)N.C1(CC)CCCC1 Cc1ncc(C(=O)NC2(C(=O)NC(c3nnc(O)o3)C)CC2(C)C)c(C)n1 c1(CC(C)C=O)ccc(C#N)cc1.C1(C(N(CC)C2CC2)=O)CC2CCC1C2.N C1(CNC(C(C)NC(CC)=O)=O)C(C2CC2)CCN1C(c1cc(Cl)no1)=O C(=O)(C(F)C(C)C(F)(F)F)N.N1(C(C(C=CC)O)=O)CCC(F)(F)C(C)C1 N1(C(c2n(C)nc(Br)c2)=O)CCCOC(CNC(C2CC3CC3C2)=O)C1 c1(CC(C)NC2(C(=O)OC(C)(C)C)CC2)ccccn1 C(=O)(C(C)(C)CC(=O)NCC)OCC.c1csc2c1CCCC2.C(=O)NC c1(CC)ncccc1C(=O)NCC(N1CCN(C(=O)C(C)C(C)O)CC1)C c1(C(=O)NC(Cc2n(C)cnn2)C(N)=O)ccncc1C(F)F c1(OC)cc(F)c(F)cc1C(N1CCC(NC(C2CC=CCC2)=O)CC1)=O C1(C)(CCC(=O)NCC(C)N(C(COCCC)=O)CC)CCC(=O)N1 c1(CCC(=O)NC(CC2CN(C(C3(CC#C)CCC3)=O)C2)C)ccc(O)nc1 Cc1cc(C(=O)NC(C)CC2CN(C(=O)C=C3CCOCC3)C2)c2nccn2c1 C1(C(=O)NC(CCC)C(=O)N2CCC(C(C)CC)CC2)CC(=O)C12CCC2 CC(C)CC(CC(=O)NCC(C)S(N)(=O)=O)NC(=O)COC.C1CCCC1 N1(C(c2cc(CCC)[nH]n2)=O)CCC(CNC(C2COCCO2)=O)(OC)C1 N1(CC(C)Nc2ccc3scnc3c2)CCCCC(N(C)C)C1=O C1(C(N2CC(C)(NC(C3(CC=C)CCCC3)=O)C2)=O)CCCCN1CCCC S(=O)(=O)(c1cccc(=NCC2(C)CC(C)(C)C2)[nH]1)NC(C)CC(C)(C)C CC1(C)CC=CCN(C(C2(NC(=O)C=CC3CCCC3)CC2)=O)C1 C(=O)(C1CCCc2ncc(C)n21)N1C(CNC(CCCCCCCC)=O)CC1 N1(C(CNC(CCC)=O)=O)CCN(C(c2cc(Cl)c(C)cn2)=O)C2CCCCC12 Cc1c(Cl)ccc(C(N2CCC(NC(C3CCCC(=O)N3)=O)CC2)=O)c1O c1(C(=O)Nc2c(C)nc(-c3cccc(F)c3O)s2)c(Cl)cc(Cl)cc1[N+](=O)[O-] C(=O)(CCC(F)(F)F)NC(COCCCNC(c1ccc(CC)[nH]1)=O)(C)C C(CC(C)C(C)C)NC(C1(OCC)CCSCC1)=O.C(=O)CCn1ccnc1.N C(=O)(CCCCCC#N)Oc1c(C(C)C)cccc1 C(=O)(C1CCCn2ncnc21)N(CCCN(C(=O)CC1CCC2(CCC2)O1)C)C C1(C2CCN(C(c3ncccc3O)=O)C2)(NC(Cc2cc(C)sc2)=O)CC1 C(c1ccc(Cl)cc1F)=CC(=O)NC1C2CCN(C(C3CC4(CC4)C3)=O)CCC12 N1(C(C2CNC(=O)O2)=O)CCC2(CCCN2C(c2cc(Cl)cs2)=O)C1 c1(CN2CCC(CC(=O)Nc3ccc(C)nc3I)CC2)c[nH]c2nc(Cl)ccc12 CC(C)C(C(=O)NC[Si](C)(C)C)NC(c1ccc(F)cc1)=O.c1nc(NC)no1 c1(C(N(C(CCNC(C(C)(C)OCC)=O)C)C)=O)ccc(Br)cc1Cl C(CC(O)C(=O)NC1CCCC1C(=O)NC1CCOCC1F)N(C)C Cc1nc2ccc(NC(=O)Nc3cccc(-c4ncccn4)c3)c(Cl)c2nc1C C1(CN(C(=O)OC(C)(C)C)CC)(CNc2nc(C)no2)CCOC1 C(CCCCCC(=O)N(C(C)CN(C)C(C1CC(C)(C)OC1(C)C)=O)C)SC N1(C(CC(n2ccc(C)n2)C)=O)CC2(CNC(c3ccc(Cl)o3)=O)CCC1C2 c1(C(C)=O)cc(C(=O)NCC2CCC2)n(C)c1.c1(C=O)ccc(=O)oc1.N C(CC(=O)NCCN(C(C1CC1(F)F)=O)C1CC1)(C(F)(F)F)OC.C C1(CNc2cn(C)nc2-c2cccc(C#N)c2)CCC2(COC(C)C2C)O1 N(C1CC(C)(C)c2ccccc21)C(=O)NC(CC(C)C)C(=O)N1CCOCC1 Cc1cc(C(=O)NCCC(C)(C)C(=O)NCCCCS(C)=O)cnc1C c1(OC(C)(C)C)cc(C(=O)N)ccn1.C1CC1(F)F.C1(C=O)CC12CC2.C c1(C(N2CCC(C(C)NC(=O)CC(C)(C)CN(C)C)C2)=O)cncc2nc[nH]c12 Cc1nn(Cc2nc(-c3cncc(Br)c3)nn2C2CCCCCC2)cc1F c1(C(N2CCC(N(C(=O)C=C(C)C)CCC)C2)=O)nc(Br)sc1C Cn1oc(C(=O)NCC2(C)CCN(C(c3sc(Cl)cc3Cl)=O)C2)cc1=O C1(NC(CCCOCCC)=O)COCCC1C(=O)NCCCCC1CCCC1 C1(NC(CCc2ccc(CC)cc2)=O)CCCN(C(C2CCN2C)=O)CC1 CCCCCCCCC(F)C(=O)NC1CC(NC(c2c(C)cnn2C)=O)C1 O=S(=O)(c1ccccc1N1CCCS1(=O)=O)c1ccc(Br)cc1 c1(C(C)C)ccnc(NCc2cncs2)n1.C12CC(c3ccccc3)CN1C2=O N1(C(C2(CNC(=O)CCc3cnco3)CC(=C)C2)=O)CCC2(CCCO2)C1 C1(CC(C)C)CN(C(=O)C(c2ccncc2)N(C)C)CCO1 C1CCC(N(C(=O)C=CCN(NC(c2ccn(CC)n2)=O)C)C)CC1 c1(C2CC(C(=O)NCC(CNC(c3cnsc3)=O)F)C2)ccc(F)cc1 c1(OC)ccsc1C(N1CCC(NC(c2csc(C3CCCCC3)n2)=O)C1)=O c1(C(=O)NCC2CN(C(C(C=C)(C)CC)=O)CC23CC3)ccc2cnn(C)c2c1 N1(C(C2(C)CCN(C(C)C)C2)=O)CCN(c2ncc(F)cn2)C(C#N)C1 C=CCC(C)(CC)C(=O)N1CC(O)(CCNC(c2cc(F)c(C)cc2N)=O)C1 C1(CCNC(C2N(CCC)CCC2)=O)CC(OC)CN1C(c1cc(C)on1)=O C(C(=O)OC)(C1=NOC2CC12)NC12CC(C(=O)NC)(C1)C2 c1(C(N2CC(C)OC(c3cccc(C(F)(F)F)c3)C2)=O)cnn2c(Cl)cccc12 S(=O)(=O)(c1ccc(C#N)c(NCCC#N)c1)N1CCN(CCC)CC1 C1(C)(CNC(c2cc(C)oc2)=O)CCN(C(=O)C(C(C)C)N2CCCC2=O)C1 Cc1ccc(C(C)C)cc1OCC(=O)OCc1cnc(Br)c(F)c1 N1(C(=O)Cc2cscn2)CCN2CCN(C(c3cc(C4CCC4)[nH]n3)=O)CC2C1 C(CCN(C)C(C1CCCC(=O)N1)=O)C(C)(C)C.CCS(=O)(=O)NCCC=O C1(C)(C=O)CC(C2CC2)=NO1.c1(C(=O)NCCC)sccc1-c1ccccc1.N c1(CC(=O)N)cn2c(C)cncc2n1.c1(C(=O)NCCCC)cnc(C2CC2)[nH]1 C=C1CC(COC)(COC(=O)CC2(C3CC3)CC2)C1 N1(C(C2(COC)CCCCO2)=O)CCC(C)C(C)C1.c1(C(=O)N)n[nH]c(O)n1 Cc1cc(-c2nc(C3CC3)nn2C2CCN(C)CC2)cc2nn[nH]c12 N1(C(c2[nH]ccc(=N)n2)=O)CCC2CN(C(c3ccc(F)s3)=O)CCC12 C(C1=NOC2CCCC12)NC(CCOCCNC(CC1C(C)=NNC1=O)=O)=O Cc1cc(C(N2CCCC(N(C)C(C3CN(C)CCO3)=O)C2)=O)cc(O)n1 c1(NC(C2CC3N(C(CCC(=O)OC)=O)C(CC3)C2)=O)ccc(S(N)(=O)=O)cc1 c1(SC)cc(C)nc(N2CCOC(CNC(=O)Nc3ccc(C)c(C)c3)C2)n1 C#CC(C)(C)C(=O)NCCC1(NC(=O)CC(C)COC)CC1 N1(C(c2nnn(CC)c2C)=O)CC(NC(=O)C(C)C2CCCC2)C2CCCCC12 c1(NC(C2CCCN2C(=O)Cc2ccccn2)=O)cc(I)ncn1 c1(NC(CC(C)NC(=O)CNC(c2cccs2)=O)C)cc(=O)n2ccccc2n1 N1(Cc2cc(C(=O)OC)n[nH]2)CC(F)CC1C(F)(F)F c1(OC)cc(CNCCCC2CCOCC2)ccc1OCCC(C)C CCCCC(C)N(C(=O)CCCN(C(=O)CC1CC(=O)C1)C)C CC(=O)C(C)CC(C)C(=O)NCc1ncc(C(=O)N(CC(C)O)CCO)cn1 [N-]=[N+]=NC1CCN(C(C2C3CN(C(=O)Cn4cc(Cl)cn4)CC23)=O)C1 C(=O)(C(C)(O)c1ccccn1)N(C(CNC(C1CC12CCC2)=O)C1CC1)C N1(C(CN(C)C)=O)CCC(C(=O)NC2(C)CC3CCC2C3)=C(F)C1 c1(C2C(CNC(C)(C)CCCl)C2)c(F)cccc1Br C(=O)(C(C(C)CC)N(C)C)NC1CCN(C(c2c(CC)ncs2)=O)C1 c1(-c2scc(NC(c3ccnc(F)c3)=O)n2)ccc(CN2CCCCC2)nc1 C1(OC)CC(Sc2ncc[nH]2)CN(C(=O)OC(C)(C)C)C1 CCC(C)CC(=O)NC1CCC1NC(C1CN(C(N)=O)C1)=O c1(CC(=O)NCC(CC)N(C(=O)CC2CCOC2)C)cn(C)cn1 C1(N(C(C(C=CCCC)O)=O)C)CCCN(C(c2ccnc(CC)c2)=O)CC1 N1(C(C(N2CCC(c3nc(C(C)C)on3)CC2)=O)=O)CC2CC(O)C(O)CC2C1 C12CC(C(N)=O)(C1)C1(CN(C(C3CC(N=[N+]=[N-])C3)=O)C1)O2.C(C)C=O.C c1(C(=O)NC2CC(C)(NC(CSC)=O)C2)ccc2c(c1)NS(=O)(=O)C2 N1(CC(=O)NCC2C3CN(CCCC4CCC4)CC23)CC(=O)NC1=O C1(C(N(C2CCN(C(=O)C(=O)Nc3ccccc3)C2)C)=O)CCOCC1 C1(O)(CC)CCN(C(C2(F)CC=CCC2)=O)CC1.C(=O)(CC(=O)N)NCC#C N1(C(C2(C)CC2)=O)CCCCC2C(NC(C34CCC(C3)C4)=O)C12 c1(CC(=O)N(CCN(C(CCN(C)CCO)=O)C)C)ccc2ccoc2c1 O=C(N=c1cc(-c2ccccc2Cl)[nH][nH]1)C1CN(c2c(Cl)cnn2C2CCC2)C1 C(=O)(C(O)CC(F)(F)F)N1CC(CC(N2CCC(O)(CC(C)C)C2)=O)(OC)C1 Cc1cc([N+](=O)[O-])ccc1C(=O)N.N1(CC)CCN(C(C2(O)CC2(C)C)=O)CC1 Cc1c(N)ccc(C(N2CC(NC(=O)C(C)(C)C3CCCCO3)C(O)C2)=O)c1Cl Cc1ccc(C(=O)NC2CCC(NC(c3csc(CO)n3)=O)CC2)c(C)c1 N1(C(c2cnc(C(=O)OC)s2)=O)CCC(NC(c2sncc2C)=O)C(CO)CC1 C1(CN(C(=O)C(F)C)C)CCCN1C(=O)CCc1cnn[nH]1.C1CC1 c1(C=O)cc(F)cc([N+](=O)[O-])c1N.N1(CC)CCCC(C(=O)NC)C1.C1CC1 c1(CNC(C(C=C)O)=O)nc(C(=O)NCc2ccoc2)c(C)o1 C#CCC(CC(=O)NCc1cn(CCOC)nn1)NC(=O)OC(C)(C)C c1(-c2n(C3CCS(=O)(=O)CC3)nc(-c3nc[nH]n3)n2)cc2c([nH]1)CCCNC2 C(c1ccccc1Sc1nn[nH]n1)=CCNC(Cc1ccn(C(C)(C)C)n1)=O C1CCCC12CC2.c1(C(C)=O)c[nH]c(C(=O)N(C(C)(C(=O)N)C2CC2)C)c1.C C(=O)(C1=CC2(CN(C(C3C4CCCC34)=O)C2)OC1)NCc1[nH]nc(C(C)C)n1 Cc1ccc(-c2ccc(NC3CCCC(C(F)(F)F)C3)cc2)cc1 c1(CN(C(=O)C(Cl)Cl)C(C)C)ccccc1Oc1ccccc1 C1(N(C)C(c2cscn2)=O)CCCCN(C(=O)CC2COCCO2)C1 c1(C(N2CCC(CN(C(C(C(C)O)N(C)C)=O)C)C2)=O)ccc2c(c1)OCCN2 Cc1cc(O)ccc1CNC(=O)CC1CC1.C12(C=O)C(=O)C3CC1C2C3 N1(C(Cc2cc(C)sc2)=O)CCC(C(N2CC(C)C(C)C2C)=O)C12CCC2 C#CCC(C(=O)NCCCCCNC(C1CC(F)(F)CS1)=O)C1CC1 CCCC(C(=O)NC(c1nnnn1C1CC1)C=Cc1ccccc1)N(C)C c1(C2C(NC3(c4ncc(C)[nH]4)CCOC3)CCC2)c(Cl)cnn1C N1(C(c2cc(C)c(F)cn2)=O)CC2(CC(C(N3CCCC3CN(C)C)=O)CO2)C1 Cc1cn2cc(C(=O)N(CC(C)N(C)C(C3CC3C3CC3)=O)C)ccc2n1 c1(C(C)=O)cc(NC(=O)CC2CN(C(c3cnc(O)[nH]3)=O)C2)ccc1O c1(N2C(C(=O)NCC3CCC(O)CC3)CC(O)C2)ccn2nccc2n1 Cc1cc(C(=O)NC2CCC(NC(=O)C(C)C3(O)CCC3)CC2)ccc1[N+](=O)[O-] c1(C(=O)OC)ccc(OC)cc1NC(C1COCCN1Cc1ccc(O)nc1)=O C1(NC(c2cncc(OC)c2)=O)CN(C(=O)C=C(C)C)C2CCCC12 N1(C(c2c(C)ccnc2C)=O)CCC2(CC(NC(C3CS(=O)C3)=O)CO2)C1 C1(C(C)NC(=O)C(C2CC2)C2CC2)CCN(C(=O)C(F)CC2CC2)C1 C1(NC(C(CC)=CC)=O)CS(=O)(=O)CC1NC(c1cc(C)sc1N)=O c1(-c2ccc(OCCCC)cc2)ccc2c(c1)CCN(C(=O)C(C)C(C)(C)C)C2 C1(NC(CNC(=O)OC)=O)(CO)CCCN(C(C2CC3(CCCO3)C2)=O)C1 C1(O)(C(C)(C)NC(C(C2CN(C(C(C)SC)=O)C2)O)=O)CCCC1 C1(C(N2CC(O)(CCNC(C(CC)CC)=O)C2)=O)CCc2nccn2C1 Cc1ccc(C(=O)C(=O)NC2COCCC2NC(C2CC(F)(F)C2)=O)cc1.C c1(C(=O)NC2CC(C)N(c3cc(C4CC4)nc(Cl)n3)C2)ccc(F)c(F)c1F CCCCCC(O)C(=O)NC1C2CC3C(C2)C13C(=O)Nn1cncn1 S(=O)(=O)(c1cccc(C(=O)O)c1[N+](=O)[O-])Nc1c2ccc(NC)cc2on1 c1(C(C2(OC)CCC2)OCC)nnnn1CCN1CC(SC)C1.CNC c1(NC(COCCNC(CCCC=C)=O)(C)C)ccc(C(=O)O)cc1[N+](=O)[O-] CC(c1cccnc1)=CC(=O)NC1CN(C(c2ccc[nH]2)=O)CC12CC2 N1(C(C2(C#C)CCN(C(c3snc(C)c3N)=O)C2)=O)CC2OC(=O)N(C)C2C1 C1(NC(C2C3CC3C3CC23)=O)CC2(CCCCC2)C1.C(=O)C(F)(F)C(F)F.N n1(CC)cncc1CN1CCC1C(=O)Nc1ccnn1CCCO CC1CCN(C(=O)NC2CCCN(c3ncccn3)C2)CCC1(F)F C1(C(N(CCCOC)C)=O)CCn2ncnc2C1.C12(CCCOC1)C(=O)N2 C#Cc1ccc(CNC(=O)CCC2CCCN(C(c3cnc(Cl)s3)=O)C2)cc1 C(CCC(N)=O)NC(C(C1CCN(C(=O)Cn2ccnc2)C1)C)=O N1(C(C(C)CN(C)C)=O)CCCC2C(NC(c3scnc3Cl)=O)C(C)(C)C12 C(=O)(C1=C(Cl)CCC1)NCC(CNC(c1c(CC)c[nH]n1)=O)(C)C C1(C)(C(N2CC(O)(CNC(c3n[nH]c(CC)c3Br)=O)C2)=O)CCN(C)C1=O C1(CC#C)(C(=O)NC(CNC(c2cc(C)c(C)[nH]2)=O)C(C)C)CCOCC1 C[Si](C)(CCCNC(c1c[nH]cc(Cl)c1=O)=O)C1CC1 C(=O)(CCCC(=O)N1CCN(C(C2SCC=C2C)=O)C(CCO)C1)OCC C1(NC(CCc2n(C)ncn2)=O)CC(NC(=O)CC2CCCC23CC3)CC1O c1(C(C)CC(=O)OCCNC(=O)C2CC2)cccc(C(F)(F)F)c1 c1(C(=O)OCC)cc(Br)ccc1Cn1cc(-c2ccc(C)c(N)c2)nn1 C1(CNC(CCCCC#C)=O)CCCC12CCN(C(=O)C(F)n1ccnc1)CC2 c1(C(=O)Nc2ccc(C)cc2O)cc2c(nc3ccccn23)s1 c1(C(N2CC(NC(c3cc(C)sn3)=O)C(F)C2)=O)ccnc2[nH]cnc12 c1(C=O)cc(Cl)cc([N+](=O)[O-])c1O.Cc1nocc1C(=O)NCC1CCCC1.N c1(OC)cc(C(N2CCOC(C)(C)C2)=O)cc(Cl)c1.C1(C(=O)N)CNC(=O)C1 c1(OC)cnc(Cl)[nH]c1=NC1CC(F)(CNC(c2cc(C)c(C)cc2Cl)=O)C1 c1(OC)ccc(C(N2CC(C)(C(=O)Nc3nc(C4CC4)cs3)C2)=O)cc1 N1(C(CCCC(=O)OC)=O)CC(C2CN(C(c3ccc(Br)o3)=O)C2)C1 c1(CN2C(C(=O)Nc3sc(C(=O)OC)c(C)c3)CC2)c[nH]c2cc(Cl)ccc12 Cc1cncc(C(N2CCC(N(CCO)C(C3CC3(C)C(F)(F)F)=O)CC2)=O)n1 N1(C(CN2CCC(C(=O)OC)CC2)=O)CC(CC(F)(F)F)OC(C)C1 C(C(C)C(=O)NOCC(C)N)c1cccc(C)c1 Cc1noc(-c2ccccc2)c1C(=O)NCCC(C)NC(=O)Cc1cnn(C)c1 C(=O)(C(C)CC#N)N(CCC(=O)NC(CCSCC)C)CC1CC1 c1(NC(C2C(C(=O)Nc3ccc(OC)c(C)n3)C2)=O)nc(Cl)c(Cl)nc1C C(CCCCCCCC(=O)NCCCCCCNC(=O)CNC(C)=O)(OC)OC N1(C(Cc2cc(C)nn2C)=O)CC2COCCC2(NC(=O)C=CC(C)(C)C)C1 C1(C(N2CC(CC(=O)NCC3C(OCC)CC3)C2)=O)Cc2cccnc2C1 C#CCC(C)(CNC(=O)CSCc1ccc(O)cc1)CO CC(C)CCCN(C)C(C1CCC(CNC(=O)C=CC(F)(F)F)O1)=O c1(C(CC)C)cccc(C(=O)OC(C)C(c2ccc(Cl)cc2)=O)c1 N1(C(C2=CC(C)(C)C2)=O)CCOC2(CCCN(C(C3(C)CCCCO3)=O)C2)C1 c1(C=O)cc(N)c(F)c(F)c1Cl.n1(CC)ccnc1C(=O)NCCC1CCC1 C(C(CC1CCCC1)C=O)NC(CNC(CN(C)C)=O)=O.c1(CC)ccns1.N c1(OC(C)C)cc(F)ccc1-c1cnc(CC(=O)Nc2nc(F)ccc2Br)nc1 O=C1CC2CC(C(N3CC(Cn4cc(C5(O)CCOC5)nn4)C3)=O)C1C2 c1(C(=O)OCC)c[nH]c(=NCC(C2CC2)NC(=O)C(F)(F)c2cncs2)s1 CC1CC(C(=O)NC(CO)C(C)(C)CO)CCN1C(=O)CCCN1CCCC1 S(=O)(=O)(c1ccc(Cl)nc1)N1C(C(=O)Nc2c(C)cc(I)c(F)c2)C=CC1 C12(C(=O)NC(C3OCCC3(C)C)C)CC1CCN2C(=O)Cc1ccco1 C1CCC2(CN(C(=O)CN3CC(C)C3)C2)O1.C1(CCOC)(C(=O)N)CC1 Cc1[nH]c2ccccc2c1CCNC(C1CCN1C(c1cccc(Br)c1Cl)=O)=O CC1CCCC=C1C(=O)NC1(CN(C(=O)CCO)C)CC1.CC(F)(F)C(F)F C(=O)(C(C)(C)C(=O)N1CCCC(C=O)C1)O.C1CC(F)(F)C1(C)C.CC(C)C c1(C=O)sc2[nH]cnc(=S)c2c1C.C(C(=O)NCC1CC1)N(C(=O)OC)C C1(CC(=O)NC)CN(C(=O)CNc2ccccc2Cl)CCN1C(=O)CC(C)CF C(CC(=O)NC(C1CCCC1)C)(CC(C)C)NC(C1C(OCC)CC1)=O c1(C(=O)NC(CCNC(C(CC)C)=O)C)ccc(C(C)C)nc1 C1(CNC(C2(C(C)(C)OC)CC2)=O)CCCCN(C(c2cc(C)[nH]n2)=O)C1 C#Cc1cccc(CC(=O)NC2CCCC(C(=O)NOCCCOCC)C2)c1 CC1(NC(=O)Cn2ccnn2)CCN(C(C23CCCC2OCC3)=O)CC1 CC(O)C(C(=O)N(C)CCc1cccs1)NC(=O)CC1CC(F)C1 C(CCC(=O)NC(Cc1ccccc1)CC)=CC.C1(=CC=O)CCN(C)C1.N C=C(Cl)CC(C(=O)Nc1cncc(SC)c1)NC(C1C2CCC(C2)C1C)=O N1(CC(C)O)CC(C)OC(C)C1.c1(C(C)NC=O)ccccc1OC(F)(F)F.N N1(C(C(C2CCN(C(CN(CCC#C)C)=O)C2)CC)=O)CCCC(CC)(C)C1.O Cc1nc(C)n(CC(N2CC(F)(CNC(=O)CSc3ccccc3Cl)C2)=O)n1 N1(C(c2ccccc2-n2cccn2)=O)CCC(NC(C2(F)CCC2)=O)C(F)C1 CCCC(CCCNC(C1CCC(=O)N1)=O)NC(=O)C(C)=C1CC1 Cc1cc(C(=O)NC(C)CCNC(=O)CC2CC2(Cl)Cl)sn1 c1(C(=O)NC2C(NC(CC(CC)SC)=O)CCCC2)cnc2c(c1)C(=O)CCC2 N1(C(CN(C(C)C)C)=O)CCC2(CC2C(N2CCN(C)CC2CO)=O)C1 N1(C(C=C(CC)CC)=O)CC(CNC(c2cnc(CC(C)C)s2)=O)C2CC12 Cc1cc(=NCC(C)N(C)C(c2csc3cncn23)=O)[nH]c(C)c1C#N CC1(C)CC(NC(=O)CSC(C)(C)C)CCN(C(=O)CC(C)(C)C(F)F)C1 N1(C(C(COC)(C)O)=O)CCCC(C)(CNC(C2C3CC4C(C3)C24)=O)C1 c1(CCNC(n2cc(C(=O)OC)nc2)=O)nc2c(s1)COCC2 C1(C(NOCCOCC)=O)CC12CC(NC(=O)CCc1ccn(C)n1)C2 C1(CC)COCCN1CCNC(=O)Nc1nn(CC)cc1Br CC1(C)CCC(CC(=O)N(C2CCCC2)CCNC(C2CCCS2)=O)C1 Cc1cc(=O)n(C)cc1C(=O)NCC1(NC(=O)CS(=O)(=O)CCO)CC1 Cc1csc(C(=O)N(CCNC(c2occc2C2CC2)=O)C2CC2)c1C C1(C)(NC(COc2ccc(C)cc2)=O)CC12CCN(CC1=CCS(=O)(=O)C1)CC2 c1(CNC(C)C(=O)NC(C)(C)C)cccc(N2CCN(C)CC2)c1 C(=O)(C1Cc2c(Cl)cccc21)NCC(C)NC(C1CC2(CCOC2)C1)=O Cc1cnc(C(N2CC(CNC(=O)C=Cc3ccccc3)CC2C)=O)c(O)c1 Cc1c(C(N2CCN(CCNC(=O)C(O)CN(C)C)CC2)=O)nn2c1OCCC2 CN1CCCC(C(N2CCCC(C(=O)NCCNC(=O)CC(F)F)C2)=O)C1 N1(C(C(=O)NCC(F)F)=O)CCCCC2(CCN(C(c3cccc(O)n3)=O)C2)C1 Cc1cnc2cc(C(N3CC4CCN(C(C5CC6CCC5C6)=O)C4C3)=O)nn2c1 c1(C(N2CC(C)(CNC(=O)CC3=CCCC3)OCC2)=O)nccc2[nH]ccc12 C1(O)(C=O)CCCC(C)(C)CC1.N1(C(C(C2CCC(=O)N2)C)=O)CCCCC1C.N C1(CNC(C=COCC)=O)CC2COCC2N1C(c1cccc2cc[nH]c12)=O N1(C(C#CC2(CC)CC2)=O)CCC2C(CCCN2C(c2coc(C(F)F)c2)=O)C1 c1(CCC(=O)NCc2ncoc2CCNC(C2(F)CC2)=O)cccc(O)n1 C1(C(N(C(C)CO)CC)=O)CCC2CCC1N2C(c1ccc(C#N)cc1)=O C(=O)(CCCCCC#N)N1C(C(=O)NCC(CC)C)CC(F)C1 Cc1sc(C)c(C(=O)NCCCCNC(=O)C(C)Cc2ccnn2C)c1C#N Cc1ccc2c(N3CCN(C(C4CCC(C)(C)CC4)=O)CC3)ncnc2c1 C1(CC)CCN(C(=O)CN2CSCC2=O)C(C(N2CCC(CC(C)C)CC2)=O)C1 N1(C(C(C)n2cnnn2)=O)CCC(C2(NC(C3CC(C)(C)O3)=O)CC2)CC1 c1(C(=O)NCC(CC)NC(c2c(C)cc(C)nc2C)=O)sc2cccc(F)c2c1C CC1CCC(CNC(c2ccon2)=O)N(C(=O)CCCc2cccs2)C1 N1(C(C2(NC(c3cc(C)cc(C)n3)=O)CCSC2)=O)CCC(C2CCC2)C1 c1(OC)sc(-c2nc(-c3csc(C#N)c3)no2)cc1Br c1(OCC(=O)NC2C3CN(C(C4CNC(=O)C4)=O)CC23)cc(Br)cc(F)c1F c1ccc2c(c1)CCCC2CCNC1(c2nnnn2C2CC2)CC2CC2C1 CCCC(F)C(=O)NC(C)CCN(C)C(C1CC1c1ccccc1)=O O=C(CCCCN1CCCCC1)NCCCOCC.C1(C(=O)N)CC(F)C(=O)N1 C1(CNC(C(CC)c2ccccc2)=O)C2CC1N(C(c1n[nH]c(C(C)C)n1)=O)C2 c1(C(=O)NC2C(F)CCN(C(C(C(C)C)C)=O)C2)cn2c(Br)cnc2s1 N1(C(c2c(CC)csc2)=O)CCN(C(c2nc(C)oc2OC)=O)CC1CCOC N1(C(c2ccc(OC)c(C)c2)=O)CCCC2(CC2)C1.C1(C)(C=O)CS(=O)(=O)C1 O=C1CCC(C(=O)NC23COC(C)(C2)C3)=NN1.C1(C=O)CCC2(CCOC2)O1 c1(C(=O)NCCN(C(C(C)Oc2ccccc2Cl)=O)C)cc2cccn2cn1 CC(C)CC(C(=O)N(C)CC1CC1)N1CCCC1=O.C(=O)C(C)(C)N(C)C.C C(C)(CC(=O)N1CC(CF)C1)NC(C(=O)NC(C)C)=O C1CN(C(C2CS(=O)(=O)C2)=O)CC2(CCC2)O1.O=C1CCC(C(=O)N)=NN1.C C(N=c1nc(N2CC3C(CO)C3C2)c2c([nH]1)CSC2)c1c(CC)nco1 N1(CC(=O)NC(CNC(CC=C(C)C)=O)(C)C)C(=O)NC(C)(C)C1=O N1(C(CC2CC(C)(C)OC2)=O)CCCC(C)(NC(=O)CC2CCC2)C1 C1(C(=O)NCc2cccc(CO)n2)CN(C(=O)C(F)OC(F)(F)F)CC12CC2 C=CC(CCC)CC(=O)NCc1nocc1C(=O)N=c1ccn(CCC)[nH]1 c1(C(=O)NCC(C)(C)NC(CC(C)(C)OC)=O)cnc2c(c1)COCC2 CC1CCC(C)(NC(=O)C=CC(C)NC(C2CCOC2C)=O)C1 c1(C(N2CCC(CN(C(=O)C(C)(C)c3ccccc3)C)C2)=O)coc2c1COC2 Cc1nnc(N2CCN(C)C(CNC(=O)C(C)(C)CF)C2)c(C#N)c1C C(c1cc(Cl)sc1Cl)=CC(=O)NC1CCCC(NC(CN(C2CCC2)C)=O)C1 c1(CC(N2C(CNC(c3c(SC)snn3)=O)CC2)=O)ccncc1Cl CC1CN2CCN1CC2C(=O)NC1CC2CC(C1)N(C(c1cnsn1)=O)C2 C(=O)(C(F)CCC(C)(C)C)NCCOC1CN(C(c2ccnc(C)c2N)=O)C1 Cc1nnn(CC(=O)NCC(C)CN(C(=O)COC(C)(C)C)C)n1 c1(CNC(C2C(NCc3c(C)n(C)nc3)C2)=O)cnc2[nH]ccc2c1 C1(N(C(=O)Cn2ccnc2C(C)C)CC)CCCCC1.C(=O)CC(F)(F)F.N C1(CNC(=O)CN2CCOCC2)CN(C(=O)CCC2CCCC(=O)N2)CC1O c1(OC)cc(CN2CCC3(CC3C(=O)Nc3cccc(F)c3Cl)C2)ccc1O C(=O)(CCCF)NC1C(CC(=O)N(CCC(C)C)CCO)C(O)C1 C(=O)(C(C)(C)C)NCC1(COC)CCC1.C(=O)C(F)OC(F)(F)F.N CCC(C)(CCC(C)C)C(=O)NCC1(OC)CN(C(=O)CC(C)C)C1.C(N)=O C1(C)(CNC(CC(CC)O)=O)CN(C(c2csnn2)C)CCO1 Cc1cc2ccccc2nc1C(=O)NC(C1CCN(C(=O)CCS(C)(=O)=O)C1)C CON(C(=O)c1cccc(SC)c1Cl)C1CCOCC1 CC1(C(N2CCOC(CCNC(=O)Cn3cnc(Br)c3)C2)=O)CCC(=O)C1 c1(C(=O)N)cnn2ccnc(N)c12.C1(C(=O)NCCC)(COC(C)C)CC1 N1(C(c2cnc(C)o2)=O)CCCC(NC(=O)CSCc2ccc(Cl)cc2)CC1 Cc1ncc(N)cc1C(=O)NC1CC(CC)C1.C1(c2cc[nH]n2)(C=O)CCC1.N C1(C2CC2)(NC(=O)CSC2CC2)CCN(C(=O)NN2CCOCC2)C1 CC(C)CCCC(=O)NCCCN(C)C(c1ccc(C(=O)C2CC2)cc1)=O N1(C(C2N(CC)CCOC2)=O)CCN(C(c2cccc(Cl)c2Cl)=O)C(C(C)C)C1 C=CCCCCC(=O)N1CCN(C(C2CC(C(C)(C)C)C2)=O)CC1CO C(=O)(CCCNC(C1CC(=C2CC2)C1)=O)NCC(=O)OCC c1(C(c2n(CCC)nnn2)NC2CCCOC2)cccc(OCCOC)c1 c1(OC)cc(I)ccc1C(N1CC2CC2(C(N2CCC(O)CC2)=O)C1)=O C(c1cc2ccccc2o1)=CC(=O)NC(C(C)NC(CSCC#C)=O)C C(c1cnc2ccccc2c1)=CC(=O)NC1CCOCC1NC(=O)C=C1CCC1 N1(C(c2cc(CC)sn2)=O)CC(C)C(NC(c2cc(C)ns2)=O)C(C)C1 C(C)(C(C(=O)N1CC(CNC(c2csc(Cl)c2)=O)C(O)C1)N(C)C)OC C1(C#CC(=O)NCC(C)(CC(C)C)NC(C23CCCC2C3)=O)(CC)COC1.O C1(CNc2ncnc(N(CCCCCC)C)c2C)CCOC12CCOCC2 C1(CC(=O)N(CC(C)C)CC(N2CC(CC(C)(C)C)C2)=O)CC(O)C1(C)C C12(NC(C(C)CN(C)C)=O)CCC(CC1)N(C(=O)C(O)CC[S+](C)C)C2 c1(C(=O)NC2(CCNC(CCCCC)=O)CC2)ccc2c(c1)C(=O)NC2=O c1(CNC(c2csc(C)c2C)c2n(C(CC)C)nnn2)c(F)c(F)cc(F)c1F c1(NC(N2CC(CS(C)(=N)=O)C2)=O)cccc(Br)n1 N1(C(C(COCC)C)=O)CCCCC1CCN(C)C(c1cc(OC)n(C)n1)=O c1(COCC)nc(C)c(C(=O)NCC2CCCN(C(=O)CC=O)C2)s1.O N1(C(C(c2ccccc2F)C)=O)CCCC(F)(C)C1.C(=O)(C(C1CC1)C1CC1)N c1(C(N(CCC)C)=O)ccc(S(C)(=O)=O)s1.C12(C(C)C)COC(C=O)(C1)C2 c1(C(C(=O)NC(CC)C)N(C)CC2CCCCO2)cccc2[nH]ncc12 c1(CC2CCCN(CC(=O)NC(CCCCC)C)C2)c(C)cccc1I c1(CN2CCC(CNC(=O)CN3CCCNC3=O)CC2)cc(=O)n2ccsc2n1 CC1(C(=O)NCC2(NC(c3c[nH]nc3Br)=O)CCC2)C=CCC1 N#Cc1ccccc1C(N1CCC(=CC(=O)Nc2cc(Br)ccc2F)CC1)=O O=C(C1CCc2nccn21)NC1CC12CCN(C(=O)C=C(Cl)Cl)C2 C(=O)(C1=NOC(C(N2CCCN(C(=O)CC(F)(F)F)CC2)=O)C1)OC(C)(C)C c1(-c2ncccc2)cccc(S(C)(=O)=O)c1.C(CCNCCCN(C)C)N(C)C.C C(CC(C(=O)NC(C(=O)NCc1ncsc1C)C(C)C)OC)OC c1(NC(C(c2n(C)ccc2)=O)=O)ccccc1.C1(C=O)(C(F)F)CC(F)(F)C1 CCC(CC(C)C)C(=O)NC1CCCCN(C(=O)C(=Cc2cccnc2)C)C1 CC(C)(CC(F)C(=O)NC1CC2OCCCC12)NC(=O)CCC(F)(F)F N1(C(C2(COC)CCOC2)=O)CCN(C(=O)Cn2cc(C#N)cn2)CC1 CCS(=O)c1ccccc1C(=O)OC1CCCOCC1 C1(CC)CCCCC1OCC(=O)NCC(C)N(C)C(C1CCOCC1)=O c1(C(=O)NC(CC)CNC(=O)C(O)C2CCC2)ccc(C)[nH]1 N1(C(C2(COCC)CC2)=O)CCN(C(C2CCCC(C(=O)O)C2)=O)CC1 c1(N2C3CCN(C)CC2CC3)nc(N2CCSC3(CCC3)C2)nc2ccccc12 C1(NC(C(C)N2CCCC2)=O)CCCC12CN(C(=O)CC1OCCC1(C)C)C2 C1(C(=O)NC2C3CC(NC(c4cnc(CC)s4)=O)CC32)CCOC(=O)CC1 C(=O)(CCC(F)(F)F)NCc1cccc(CNC(C(N2CCNC2=O)C)=O)c1 Cc1cc(CC(=O)NC(C)C(C)(C)NC(c2cccnc2O)=O)ccc1F Cc1cc(C(N2CCC(O)(CNC(=O)C(C)CN3CCCCC3)C2)=O)cc(F)c1 Cc1csc(CNC(=O)CCC2CCCC2)n1.c1(C(=O)N)ccn(C2CC2)n1 C1(CC(=O)NCC2C3CN(C(COCC)=O)C2C3)CCS(=O)(=O)CC1 Cc1cc(C(=O)NC2CCCC2NC(C2CC(CF)C2)=O)c(C)nc1C c1(-c2c(C)nc(F)cc2)ccc2cc(C(N3CCN4CCC3CC4)=O)nn2c1 C(=O)(C1CCCc2sc(C)nc21)N1C2CC(NC(CC=C(C)C)=O)C1CC2 N1(C(C)CNC(C2CN(C)CCN2C(C23CC(C2)C3)=O)=O)Cc2ccccc2C1 C(CC(=O)NC(C1CCN(C(C2(Br)CC2)=O)C1)C)(C(F)(F)F)OC c1(C(N2CCC(N(C(C(CC)F)=O)CCO)C2)=O)scc(C)c1C CC1CSc2ccc(Br)cc2C1NC1CC1c1ccc(C#N)cc1 C(=O)(C(CC(C)C)C(C)C)NCC(CC)NC(c1cc(-c2cnn(C)c2)[nH]n1)=O C1(C(N2CC(CNC(C(c3ccccc3)OC(C)C)=O)C2)=O)CCC(=O)O1 C(=O)(C1COc2cc(C(C)(C)C)ccc21)OC(c1cccc(O)c1)C Cc1cc(CC(=O)N(C)CCNC(c2nc(C(F)(F)F)ccc2N)=O)cc(O)n1 CC1C(=O)Nc2ccccc2N1C(C1CC2CC(N)C2C1)=O CCCC(C(=O)NC1CN(C(C2(C)CCCCO2)=O)CC1C)OC C1(NC(c2[nH]cc(CC)c2)=O)CN(C(=O)COc2ccc(O)cc2)CC1O N1(C(C(F)OC)=O)CCCC(N(CCF)C(c2ccc(CCF)cc2)=O)C1 c1(C(N2C(C)CC(NC(C(C)N3CCC3)=O)C2)=O)cc(Cl)ncc1Cl c1(CCCC=O)ccc(Cl)c(Cl)c1.C1(C(=O)OCC)CC(C=O)C1.C1CC1 N1(c2nnc(C(=O)N(C)CC3CCC3)n2C)CCC(F)(F)C(C)C1.CCCCC C1(CCOC)(C(N2CC(N3CCOC3=O)C2)=O)CCN(C(=O)COC(F)F)CC1 N1(C(c2cc(C(CC)C)no2)=O)CC(C)OC2(CCN(CC#N)CC2)C1 S(=O)(=O)(c1cccc(=NCC2CC3CCC3C2)[nH]1)N(C(CCSC)C)C C1(O)(C(C)NC(CC(C)(C)OC)=O)CCN(c2nc(C(C)=O)c(C)s2)CC1 C1(N(C)C)CCCC1CNC(=O)CC1CCC1.C1(CCC(=O)N)CCCN1C c1(C(N(CCC(C(C)C)NC(C(CC)C)=O)C)=O)ccccc1C#CC1CC1 C12(NC(c3[nH]cc(C)c3)=O)CCC1CN(C(=O)C=C1CCCC1)C2 c1(C2(C)C(NC(=O)NCC(C3CCOCC3)(C)OC)C2)ccc(F)c(F)c1 C12CCC(CC1)CO2.c1(C=O)cc(Cl)nnc1O.C1(CC)OCCC1C(=O)NC Cc1ccc(NC2CCC3CCNC2C3)c(C#N)c1 C1(C(N2CCC(CN(C)CC)C2)=O)C(C)CCN1C(c1cc(OC)ns1)=O C(=O)(C(C1=CCSC1)N1CCCC1C(C)C)NCCOC C1(C)(C(N2CC(N(C(=O)C=CC3CCC3)C)C2)=O)CC(C#N)C1 O=C1CCC(Nc2cc(NCC3CC3)ncn2)C(C2CCNCC2)N1 C(C(C)C(=O)N(C1(C(=O)N(C2CCC2C)C)CC1)C)OC Cc1cc(=NCc2ncoc2C2CC2)[nH]c(=NCCC(C)C(=O)OC(C)(C)C)[nH]1 c1(C(N(C2CCCCC2)CCNC(=O)CSC(F)(F)F)=O)ccsc1Cl c1(OC)cc(I)c(Cl)cc1C(N1CCCC(C(C)(F)F)C1)=O c1(C(c2n(CC=C)nnn2)NCc2ncoc2C)c(Br)n[nH]c1C c1(C(=O)NCC)cc(C(=O)NCC(c2ccccc2)N)c(C)o1.C(C)C C(=O)(C(C)(C)CC(=O)N1CCN(C(=O)Cc2cncnc2)C(C)C1)OCC C(CCN(C(=O)C(C)C1CC1)C)C(C)(C)C.c1cccc(C=O)c1.CC(=O)N c1(CN2CCC(C(N3CSCCSC3)=O)CC2)ccnc(Br)c1F CS(=O)(=O)c1ccsc1C(N1CC2CC1CN2C(=O)CCCC(N)=O)=O Cc1c(C(=O)NC2CCCC(NC(=O)C(C)(C)O)C2)c[nH]c2nccc1-2 CC1=C(C(=O)N(C)CC2CCN(C(C3CC(F)C3)=O)CC2)SCCO1 c1(CCNC(C(C)C2CN(C(=O)OC(C)(C)C)C2)=O)cc(C(C)C)nn1C C(CCC(F)(F)F)NC(c1c(C)c(C2CC2)[nH]n1)=O.C1(C(=O)N)CCCN(C)C1 C1(C(=O)NC2(C)CC(C(NOCC(=O)OCC)=O)C2)CCCCN1C N1(C(C2C(OC)C2)=O)CCC(N(CC(=O)N(C)Cc2cccs2)C)C1 C(=O)(C1=NNC(=O)CC1)N1C(CN(C)C(C2CCC23CCOCC3)=O)CC(F)C1 N1(C(C2C(C)(CC)C2)=O)CCC2(CCCN2C(C2CC3CCCC23)=O)CC1 Cc1cnc2cccc(C(=O)NC3CC4(C3)CC(NC(=O)CC(C)C3CC3)C4)n12 CN1C(=O)CCC1C(=O)NCCCN(C(c1ccoc1Cl)=O)C1CC1 Cn1ccc(=O)c(C(=O)NCc2cccc(NC(c3ncccc3O)=O)c2)c1 C1(F)(CNC(CC(C)(C)C)=O)COCCN(C(c2n[nH]c3cccnc23)=O)C1 CC1CN(C(c2[nH]nnc2C2CC2)=O)CC(CCNC(c2cccc(O)n2)=O)O1 Cc1nnccc1C(N1CCN(C(=O)CCSc2nnnn2C)CC1)=O C1(C=O)CCC(C)(C)C1.C(=O)C(C)CC1CC1.C(=O)(C)NCCOC C1(NC(CSc2cn(C)nc2)=O)CCCCN(C(=O)C(F)=CC2CC2)C1 N1(C(C(CC(C)C)OC)=O)CCCC2(C1)C(NC(C1C3COCC13)=O)CCN2C C1(C(N2C(C(N(CC(CCC=C)O)C)=O)CCC2)=O)CCCCC1(C)C CCCC(CN=c1[nH]c(=NCc2cnc(O)nc2O)[nH]c2c1CCC2)OCC CCC(C)(C)CC(=O)N1CCOC(C(C)NC(=O)CCc2cc(C)n(C)n2)C1 Cc1noc(C)c1C(=O)NC(C)CC(C)NC(=O)C=CCC1CCCC1 N1(CC#C)CCCC1CNC(=O)C(C)OC(C)=O c1(C(=O)NCC2CN(C(C(C)Cn3cccn3)=O)C2)cc(Br)cc2ccccc12 Cc1onc(-c2ccccc2Cl)c1C(=O)NCC1CCN1C(=O)Cc1ccoc1 c1(OC)cccc(CN(CCC(F)(F)F)C(=O)CNC2C(C)C2C)c1 c1(C(=O)NCCNS(C)(=O)=O)[nH]c2ccccc2c1-c1cccnc1F C12(OC)CCC(CC1N=c1nc(N(C)CCC3CCCN3C)c3sccc3[nH]1)C2 C12(CNC(CC(C)N(C)C)=O)CCC1CN(C(=O)CSc1ccc(Cl)cc1)C2 C(=O)(CC(C)C(C)C)NCc1cc(C)c(C(=O)N)o1.C1CCN1C(C)(C)C C(=O)(CCCCCCCC(=O)OC)NCC(CC)(C)NC(=O)CC(C)NC(N)=O Cc1ncn(C)c(=O)c1C(=O)NCC1CN(C(=O)C(C)(C)CO)CC12CC2 N1(C(C(C)c2ccsn2)=O)CCCCCC(NC(c2ccc(C(F)F)o2)=O)C1 C1(C(=O)NCCCCOC)CCCCN(C)C1=O.C1(C2(O)CCC2)(C=O)CC1.N C1(CC=C)(NC(C2CC(CC)C2)=O)CCN(C(=O)C(C)C2(O)CCC2)C1 C1(NC(c2c(CC)c[nH]c2)=O)CCN(C(c2cnn(C3CCCC3)c2)=O)CC1C Cc1cc(C)n2c(CNC34CNCC(C)(C3)C4)cnc2n1 Cn1c(NCCC2CCC(CNC(=O)C(C)(C)C(N)=O)CC2)cc(O)nc1=O C(C(CC(C)C)C(=O)O)NC(Cn1cc(CN(CCCCC)CC(C)C)nn1)=O C1(F)(COC)CCN(C(c2ncccc2-c2ccccc2CC#N)=O)CC1 CCCCC(CC(=O)N1CC(OCCF)C1)NC(=O)C(CC)(CO)OC CCCCC(C)(F)C(=O)N(C)CCN(C(=O)C(C)CS(C)(=O)=O)C(C)C c1(-c2ccc(CC(=O)NCCCOC)cc2)cnc(F)cc1.CCCOCCO C(=O)(C1=CC2(CCOCC2)C1)NC1C2CN(C(CCn3c(C)ncc3)=O)C1C2 c1(CC)cc(F)ccc1C(N1CCC(NC(=O)C)C1C(C)(C)C)=O.CCCF c1(C(N2CC(NC(C(C(C)(C)C)O)=O)CC3(C2)CC3)=O)cc2c(Cl)ccnc2s1 C1(CNC(c2cnn(CC)c2C)=O)CN(C(=O)C(F)C(C)(C)O)CCC12CCC2 C1(C(=O)NC(C)CCNC(=O)CC(O)CN(C)C)CC2CCC1C21CC1 Cc1ccc2ncccc2c1C(=O)NCC(C)CO.C12(C(=O)N)CC(C#N)(C1)C2 C(=O)(C(F)C(F)(F)F)NCC(C(=O)N(c1cccc(O)c1)CC)N(C)C CCCCCCNC(=O)C(=O)Nc1cccc(C)c1.C1(CC=O)CCC1(C)C.N Cc1ccc(CC(=O)N(C(C)CNC(c2c[nH]c(C(F)(F)F)c2)=O)C)c(Cl)c1 c1(CCNCC(c2ccc(Cl)cc2)(C)O)cccc(Cl)c1F CC1CS(=O)CCN1C(C1CC=CC(NC(C2(C(F)(F)F)CC2)=O)C1)=O C(CC1CCC1)(C(=O)N1CCC1)NC(C1CC(O)(Cc2ccccc2)C1)=O c1(C(=O)NC(C(C(C)C)NC(c2cc(OC)ncc2)=O)C)cc(C)ncc1C c1(C(=O)NCC(CC=C)NC(=O)CCC(=O)NCCCOC)nc(C)ccc1O C(=O)(CC(C)(F)F)NC(CC=C)CNC(c1cnn(CC(F)(F)F)c1)=O CC(C)(CCCNC(C1CCCN1N=O)=O)NC(=O)CC1CC2(CC2)C1 c1(OC)ccc(C(=O)NCC2CCN(c3ccc(Br)cn3)C2)c(F)c1F C#CCCCCC(=O)NC1CCCC(C(=O)NC(C)(C)C(=O)NC)C1 N1(C(C#CC(=O)N(C)C)=O)CCC2C(CCCN2C(=O)Cc2ccco2)C1 C1(C(=O)NCC(CNC(c2cc(C)c(F)cc2)=O)F)CC2(CCCCO2)C1 C(=O)(CCC(=O)C(C)(C)C)NC(C(C)C)C(=O)NC1(C)CCC(=O)NC1=O C1(CC)CN(C(c2ccc(Br)nc2C)=O)CCN1C(c1c(C)nn(C)c1C)=O N1(C(CCC2N(C)CCC2)=O)CC2(CNC(=O)CCC3CCOC3)CC1CO2 Cn1nc(C(F)F)cc1Cc1nnnn1C1COC1.C1CN(S(C)(=O)=O)C1.N C(CCC(=O)NCc1ccc(C)nc1)(C(C)C)NC(CS(CC)=O)=O N1(C(c2c(C)nc(C)s2)=O)CCN(C(C2(S(N)(=O)=O)CC2)=O)CC(C)(C)C1 N1(C(CCC2CCC(NC(C3CC(=O)C3)=O)C2)=O)CCCN2CCCC2C1 c1(C(N2CC(CNC(CCN(C)CC)=O)C2)=O)csc(S(C)(=O)=O)c1.C N1(C(C2N(C(COCCCCC)=O)CCC2)=O)CCC(CCC)(CO)C1 C(C1CCCCC1)=CC(=O)N(C1CCN(C(C2CC(C)(C)C2)=O)C1)CC C1(C(=O)NCC(COC)O)(NC(=O)CC2CCC2)CC(O)C1 C(CC(CC)C(=O)NC1(C)CCN(C(c2cnnn2-c2ccccc2)=O)C1)=CC c1(CC)ccc(C(N2CC3C(NC(C4(CC)CNC(=O)C4)=O)C3C2)=O)cc1C C(=O)(CCC(F)(F)F)N1CCC(CC#C)(C(=O)NCC#CC(F)(F)F)C1 S(=O)(=O)(C1CC2(CCCC2)C1)NC1C(C)CN(Cc2c[nH]c(=N)s2)CC1 C#Cc1ccc(NC(c2c(CNC(=O)C(O)CCCC)cnn2C)=O)c(C)c1 C(=O)(C(C(C)C)N(C)C)NC1C(NC(COC(CC)(C)C)=O)C1 N1(C(c2cnc(C)nc2)=O)CCCC(NC(C2(CO)CCCO2)=O)C1C c1(C(=O)NC(CN(C(C2ON=C(C)C2C)=O)CC)C)sc2ccccc2c1C c1(C(=O)NC(C(C)(C)C)CNC(C2(CF)CCOCC2)=O)csc2c1CCCC2 N1(CC(C2CCC(C)O2)=O)CCCN(Cc2ncccn2)CC1 CC#CCCCC(=O)NCC12CC(NC(C3CCC(OC)C3)=O)(C1)C(C)O2 C1(C(N(C)CCc2cnccn2)=O)COCCC1NC(C1CCCCC1O)=O Cc1[nH]nc2cc(C(=O)NCCC3CCN(C(C4CC4C(N)=O)=O)C3)ccc12 c1(OC)ccc2ccc(NC(C3C4CC(O)C3N(C(C)=O)C4)=O)cc2n1 C1(N(C(c2cccc(OC(F)F)n2)=O)Cc2ccsc2)CCCC12CCNCC2 C(=O)(C(C)(C)C(=O)NC(c1ccc(F)cc1)C)OC.c1(C=O)ccnc(C)n1 C1(C(N(CCCNC(C(CC)SC)=O)C)=O)Cc2cc(C)c(C)cc2O1 c1(C(C(=O)NCC=C)N(CC(C)C(=O)OC)C)ccc(OC)nc1OC C1(C(N2CCN(C(C3(C4CC4)CC3)=O)CC2)=O)CCCCC12CC2(F)F Cc1nc(NCC(C)NC(C2CCC(C)CC2)=O)c2c(C)csc2n1 C1(CC#C)(C(=O)N(C)CCNC(=O)C(C=C)c2ccccc2)CCOCC1 c1(C(=O)NC2C3CC(C)(C3)OC2)cccc2c3c([nH]c12)CCC3 Cc1cnc2[nH]cc(CN3CC(C(=O)Nc4ccc(I)c(Cl)c4)CC(F)C3)c2c1 C1(C(=O)NC(C2(O)CCN(C(c3cscc3Cl)=O)C2)C)CCCCN1C C1(NC(=O)C(C)N(C(=O)C(C)OCC)C)CCCN1SCCC.CC.O C1(CC)CCCCN1N1CCN(c2ccc(Cl)cc2C(N)=O)CC1 C1(N(CCC)C(c2sccc2C)=O)CCN(CCSc2ccccc2)CC1F C12(C(=O)NC(CCCC)CNC(=O)CN3CC=CC3)CC(C)(CCO1)C2 CCC(C(=O)NC1CC(OC)C1)NC(=O)CC(C)n1cccc1 CCC(CC)CCCC(=O)NCC1(F)CC(NC(C2CCC2C)=O)C1 C1(SC)CN(C(=O)Cc2ccccc2Cl)CC1NC(=O)C(C)Oc1ccccn1 c1(Cc2cccc(Br)c2)cnc(C2CN(C(C3(C4CC4)CCNC3)=O)C2)nc1 c1(SC)cc(C)ccc1-c1nc(CSC)nn1C(C1CCOCC1)C c1(C(N2CC(NC(C(C)OCC3CCCO3)=O)C2)=O)cccc2sccc12 Cc1cccc(F)c1C(N1CC2CCC2(CNC(=O)C(C)(C)C2CCC2)C1)=O CCC(C)CC(C)C(=O)NCCc1n[nH]cc1C(=O)Nc1cc(F)ccc1C C1(NC(c2n(C(C)C)ccc2)=O)CCC(C)(CNC(c2coc(Br)c2)=O)C1 S(=O)(=O)(c1cc(C)cnc1)N1CCCCC1.CC(C)S(C)(=O)=O.C(=O)(NC)N C1(NC(CC2N(C)CCC2)=O)CCS(=O)(=O)C12CN(C(=O)C)C2.c1nccs1.N C1(C(=O)NC)CC(O)CN1C(c1coc(C)n1)=O.C1(C)(CC=O)CCOC1 C=CC(C)(C)C(=O)N1CCCC(N(C(=O)Cc2csnn2)C)C1 S(=O)(=O)(c1cc(F)cnc1N)NC(C1C=C(C)CS1)=O N1(C(C(C)(C)F)=O)CCCC2CN(C(=O)CCCCc3cnn[nH]3)CCC12 N1(CC(C)NC(C(C)NC(C)=O)=O)CCN(C(c2ncc[nH]c2=O)=O)CC1 C(CC(=O)N(C(CNC(=O)CCc1ncc[nH]1)C1CC1)C)SC C1(NC(C(C)OC(C)=O)=O)CCOCC1C(N1CC(N2CCCC2)C1)=O C1(OC)(CNC(=O)CC(F)(F)F)CCN(C(=O)C(C)CC2CCCCC2)CC1 N1(C(C(n2c(C)ncc2)C)=O)CC(F)CC1CNC(c1csc(=N)[nH]1)=O Cc1ccc(CNC(=O)C(O)C2CCCC2)c(OCC2CCCO2)c1 C1(C(N2CCC(Cn3cc(-c4ncccn4)nn3)C2)=O)CCCN1CC(F)(F)F N1(C(C(C)c2cc[nH]n2)=O)CCCC1CNC(=O)C=Cc1ccco1 Cn1cc([N+](=O)[O-])c(C(=O)NCC2CCCCC2)n1.c1(CC=O)cncs1.C CCCCCC(C)(C)C(=O)NCC1CC(OC)CN1C(C1CC1CC)=O C(=O)(CC(C(F)(F)F)NC(c1ncccc1O)=O)NCc1cc(C)cc(C)c1 C1(C(=O)NCC(C)(C)OCC(=O)NCC)CCC(=O)N1 Cn1cnc2c(C(=O)NC3(C)CN(C(C4(Cl)CC4(C)C)=O)C3)cccc12 C1(C2CCN(C(CNS(NC)(=O)=O)=O)C2)CCCCN1C(C1(OC)CCSCC1)=O C1(NC(CC(CC)CN(C)C)=O)C2CC3CN(C(=O)CC4CCCC4C)C1C3C2 C(=O)(CC(C)C(C)(C)NC(=O)CN1CCC(=O)CC1)N(CCC(=O)OC)C CC(CNC(=O)CN1CCCCC1)C(F)C(=O)NC1CCN(CCCO)C1 C1(C=O)CCc2cncn2C1.N1(C(C2C(C(=O)OCC)C2)=O)CC(C)C1.N c1(C(=O)NCC23N(C(C4(C=C)CCC4)=O)CC(C2)C3)ccc2ccoc2c1 C1(OC)CN(C)C(C)(C(=O)N)C1.c1(C=O)cnc(N(C)C)nc1.C1CC1.C n1(CC(=O)NCCCCNC(C(c2cccc(C)c2)(F)F)=O)ncc(C#N)c1N N1(C(c2cnc(C)[nH]c2=N)=O)CCC2(CCN(C(c3ccc(CO)cn3)=O)C2)C1 Cn1nc(Br)c2c(NC(=O)C(N3CCCCC3c3nccs3)=O)cccc12 c1(C2(NC(c3cccc(OCOC)c3)=O)CC2)cc(OC)ccc1C N1(C(Cc2n(C)ccc2)=O)CCC2CCCC12C(=O)NC1(CCCCO)CC1 C1(C(=O)NC(C#C)CC)C(NC(c2cc(Cl)c[nH]2)=O)C1(C)C n1(CC#C)ccc(C(C(=O)NCc2cccs2)N(C(C)C(F)F)C)c1 n1(CC=O)cc(C2CC2)cn1.C1(CCNC(CSC(=N)N)=O)CCCCC1.N N1(C(C(CC(C)(C)C)O)=O)Cc2n[nH]cc2C1C(=O)NCCN1CCOCC1=O Cc1cnc(C(N2CC(CNC(C3CCCC(O)C3)=O)CC2C)=O)cc1C C(C(F)(C(=O)NCc1nc(C)cs1)C(C)C)NC(C(CC(=O)OC)C)=O C1(C)(NC(C=NOC)=O)CCCN(C(=O)CC2CCC(=O)O2)C1 c1(C(C)(F)F)ccc(C(N2CCN(CCC3CC3)CC2)=O)cn1 c1(C(C)C)cccnc1C(c1cccc(F)c1)NC1CCC1 CCCC(CC(C)C)C(=O)NCC=CC(=O)N(CCF)CCOC C(C1CCCCCC1)=CC(N1CCC(NC(C2CCC(F)(F)C2)=O)C1)=O c1(C(=O)NCC(CC)NC(=O)C(F)=CC2CC2)ccc(S(N)(=O)=O)s1 c1(C(=O)OC)cc(C2CN(C(=O)O)C2)[nH]n1.C(C)(C)C.C12CC1NC2 C1(C(=O)Nc2c(CC)nsc2)CC(O)CN1C(C1(N2CCCC2)CC1)=O C1(Nc2c(C)n(CCN(C)C)nc2)(C)CCC(C)CC1.C(C)(C)C.C(=O)N C1(O)CCN(C(c2c(F)cccc2F)=O)CC1.c1(C(=O)NC)ncsc1C1CC1 N1(C(CC2(C)OCCO2)=O)CCOC2CCN(C(=O)C(F)C3CCCC3)CC12 C1(C(=O)NCc2ncsn2)(CC)CCN(C(=O)C=CC2CCCCC2)C1 c1(C(N2CC(NC(C(C)C3CCOC3)=O)C(C)CC2)=O)ccc2cncn2c1 c1(C(N(CCCN(C)C(c2nnsc2C(F)F)=O)C)=O)cc(=N)[nH]c(Cl)n1 c1(C(N2C3C(NC(c4c(SC)ccs4)=O)C(C3)C2)=O)cc(F)ccc1N N1(C(C2CC(NC(c3cc(C)cc(O)c3)=O)C2)=O)CC(C)OC(C)(C)C1 c1(C(N2CC(O)CC(NC(c3c(CC)cccn3)=O)C2)=O)cc(Cl)c(N)cc1F C1(F)CCN(C(c2cc(-c3ccccc3)ns2)=O)CC1.C1(C(=O)NC)C2CCC12 c1cnc2c(=NCc3cncs3)[nH]c(=NC3CCN(CC4CC4)C3)[nH]c2c1 C(N=c1[nH]n(C)cc1[N+](=O)[O-])C1N(C(C2(O)CCCC(C)CC2)=O)CCCC1 c1(C(=O)NCCc2cn(C3CCCC3O)nn2)cccn(C2CCSC2)c1=O CS(=O)(=O)C(C(=O)NCCNC(c1ccc(C2CCCCC2)cc1)=O)C1CC1 N1(C(c2ccc(C(C)=O)cn2)=O)CCCC(N(C(=O)CC2C=CCCC2)C)CC1 c1(SCC(=O)NCCCOCCCNC(C2C(C#N)C2)=O)cccnc1 N1(C(C(COC(C)=O)C)=O)C(C(=O)N(CC(C)C#N)C)CCC1C1CC1 c1(C(=O)NC(CC)CNC(=O)COc2cc(C)on2)csc2cccnc12 N1(C(C(C)OC)=O)CCC(NC(c2csc(COC)n2)=O)C1C(C)(C)C c1(C(=O)NCCC(C(C)C)NC(C2C=CCC2)=O)cnc2c(Cl)cccn12 N1(C(C2CC(CC)(CC)C2)=O)CC(NC(=O)C(F)C2CCC2)CC1(C)C c1(OC)ccc(C(N2CCC(NC(C3CCCCO3)=O)C(O)C2)=O)c(I)c1 N1(C(=O)Nc2c(OC)cc(Br)cc2OC)CCC(O)CC(C)(C)C1 Cc1cc(C(=O)NCC2CN(C(c3ccn(C(F)F)n3)=O)CC2O)n(CCO)n1 CC(CC(=O)NCC(C)(C1CC1)NC(=O)C1=CCOCC1)C(C)(C)C c1(CCC(=O)NC2CC(OC)CN(C(=O)CC(C)CF)C2)n[nH]c2ccccc12 C(=O)(C1=CC(O)CCC1)N(C)CC1CCN(C(c2cc(CC)nc(O)c2)=O)CC1 N1(C(c2c(CNC(c3c(=N)[nH]cnc3)=O)ccs2)=O)CC23CCC2(COC3)C1 C(N=c1ccnc(CC(C)C)[nH]1)c1ccn(C(CCC)C(=O)OC)n1 Cc1c(C(=O)NCCC(C)(C)NC(=O)C)sc2cncn12.C(=O)CN(C)C C1(CC=C)(NC(C2CC3(CC(OC)C3)C2)=O)CCCN(C(C2CC2)=O)C1.O N1(C(c2cc(SC)oc2)=O)CCN(C(=O)C(C)(C)C2CCCO2)CC(C)C1 C(C(=O)N(CCCC(=O)NC(C)CC1CCC1)C)(C(C)C)OC Cn1nc(CC(=O)N)cc1C(F)(F)F.C1CN(C(C2CC2C(F)(F)F)=O)C1 n1(CC(=O)NC(C(=O)NCCC2(C)CC2(F)F)CO)cnc(C#N)n1 CCCCCCCCC(F)C(=O)N(C1CCN(C(=O)C(F)(F)CO)C1)CC C=CCCCC(C1CC1)NC(=O)C(C)N(C(=O)CCNC(=O)OCC)C C(=O)(C(C)(C)CNC(c1nnc(S)n1C1CC1)=O)OCC C1(C(N2CCC(N(C(c3c(C)cccc3)=O)C)CC2)=O)CCOC(C)(C)C1 c1(CC(=O)NCCCC)cc(C2CC2)on1.c1(C=O)csc(-c2ccsc2)n1.N Cc1cc2c(cc1C)C(C(=O)NC1CN(C(c3ccc(CO)c(F)c3)=O)C1)CO2 Cc1cc(C(=O)NC2(C=O)CC(F)(F)C2)cc(O)c1.c1(CC)cn(C)nn1.N C(=O)(C1=CC(O)C(O)C(O)C1)N1C(C(=O)N)CC2CC21.c1(OC)nn(C)cc1 c1(NC(C#CCNC(CCCC(=O)OC)=O)=O)cccc(C#N)c1F C1(C(=O)NCCC(CC)(F)F)CCC(O)CN1C(=O)Cc1ccnc(O)c1 c1(CC(=O)NC(C2CC2C(=O)NC)C)ccn(C)c1.C1CC(C#N)C1 C1CCSC12CN(C(c1sc(F)cc1Cl)=O)C2.C1(C(=O)N)CC(=O)N(C2CC2)C1 S(=O)(=O)(c1cc(C)cnc1NCc1ncccc1N)NCc1cc(C)cc(C)c1 Cc1ccc(O)c(C(=O)NC2CCN(C(C34CCC(C3)C4)=O)C(C)C2)n1 n1(CC)nc(C(N2CCCC2C(N2CC(n3ccnc3)C2)=O)=O)c(C)n1 c1(NC(CN2C(C)(C)SCCC2)=O)ccc(S(=O)(=O)N2CCNC(=O)C2)cc1 CC(C)C(C#N)C(=O)NC(C)CN(C)C(c1nonc1N)=O CC1CC2(CCN(C(c3cc(O)ccc3[N+](=O)[O-])=O)CC2)CN1C(=O)CC(F)F N1(C(C2ON=C(CC)C2)=O)CC2CCC2(CNC(=O)CCc2ccc(C)cc2)C1 c1(C(=O)N)ncc(C#N)cc1C.C1(NC(C2C(=C)C2)=O)CC2(C1)CC(C)C2 N1(C(c2cc3scnc3[nH]2)=O)CCC2CCN(C(=O)CCC3CC3(F)F)C2C1 c1(C(=O)NC2C(C(=O)NCC(COC)C)CCCC2)nc(C)ccc1F c1(NC(C(C2CC3CC3C2)N(C2CC(n3cccn3)C2)C)=O)ccccc1Cl N1(C(C2C(C(=O)Nc3c(OC)cc(Br)cn3)C2)=O)CCCCC(C)(F)C1 C1(C)CCCC1.C12(C=O)CC(F)(C1)C2.C(C)(C)C.CN(CC)C.C=O c1(C(=O)NCCC(C)N(C(C2CCN(CC(C)C)C2)=O)C)cc2ccccn2c1 CCCCC(O)C(C)C(=O)NC1CCN(C(=O)C(=Cc2cn(C)cn2)F)C1CC C1(CCNC(c2c(Cl)cn(C)n2)=O)CCN(C(C2C3CCCC23)=O)CCC1(F)F CC(Cn1ccnc1)C(=O)N1CC(CNC(=O)CSc2nncn2C)C1 N1(C(CNC(N2CCCC2)=O)=O)CCCC12CCN(C(c1cccnc1S)=O)C2 C(=O)(NN(C)c1ccccc1)NC(C1CCCCO1)CC C(c1ccccc1)=CC(N1C(CNC(c2scc(COC)c2)=O)CC1)=O c1(C(N2CC(SC)C(NC(=O)C=Cc3cnc(C)s3)C2)=O)cnc(C)[nH]c1=N C1(C#N)(C(=O)NCCC2N(C(C(C(C)C)SC)=O)CCCC2)CC2CCC1C2 C1(NC(C2(C=C)CCC2)=O)CCOC(C(=O)NC2(C)CCSCC2)C1 CC1(C)CN(C(c2cccc(Cl)c2O)=O)CC1NC(=O)C(F)(F)CC1CCCO1 C(C(C(=O)N1C(CO)CC1C)NC(c1nnsc1C)=O)OC CN1C(=O)CCCC1C(N1CC(C)(NC(C2C(C3CC3)C2(F)F)=O)C1)=O N1(C(=O)C2=CCSC2)CCC2CCN(C(=O)CC34CCC(CC3)OC4)C2C1 C(=O)(C(C)C(C)COC)NCC1(O)CN(C(C(CC)=CCCC)=O)C1 N1(C(c2n(C)nc(C(F)(F)F)c2)=O)CC2CN(C(=O)CC3COCCO3)CC2C1 C1(C=O)CCN(C(=O)CC2(N3CCCC3)CCC2)C12CC2.C(CO)OC.CC C1(C(=O)NC2CC3C(NC(=O)Cc4cc[nH]n4)C3C2)(CF)CCOCC1 N1(CC(=O)N(CCC)C2CC2)CCN(C(C2CCCN(C(N)=O)C2)=O)CC1 c1(C(N2C(CNS(CC(=O)OCC)(=O)=O)CCC2)=O)nc(C)ccc1.O C12(Nc3nccc(SC)n3)CCC(CNC(c3c(F)ccnc3Cl)=O)(C1)OC2 CC(CCCCNC(=O)Cc1cncnc1O)NC(c1cnn[nH]1)=O C(=O)(C1=CC(C)(CC)C1)NCC(CCCC)NC(=O)CCCCc1ccccc1 C1(CNC(C(C=CCCC)O)=O)CN(C(c2cscc2CC)=O)CCO1 c1(CNCc2ccc(C)[nH]2)ccc(C(=O)NCc2cccnc2)cc1 C#Cc1ccc(C(N2CCCC(NC(=O)Cc3ncccc3C)C2)=O)c(F)c1Cl C1(C(=O)NCC(C)O)(CC)CCN(C(=O)CNC(=O)NC)CC1 c1(C(C)C)cccc(C(N2CC(C)(NC(=O)C(C3(O)CCCC3)F)C2)=O)c1 c1(CN(C(c2ccc(OC)nc2)C(=O)NCCCC)CCC)ccc(C#N)nc1 N1(C(CC=CC=C)=O)CC2CC1CC2NC(=O)CCCC(N)=O C1(CC)(CC)CCN(C(=NCCc2ccccc2)NCC2(F)CC2)CC1 C1(C(N2CC(NC(C(C=C)CC)=O)C(n3ccnn3)C2)=O)CCn2nncc2C1 C1(NC(CC=CCNC(CCNC(=O)OC)=O)=O)CC(O)C(O)C1 C(=O)(C#CC1(C)CCCO1)NCCN(C(c1nnc(C)o1)C)C1CC1 n1(CCCNC(=O)NC2(C3CCCC3)CCC2)cnc2ccccc12 c1(C(N(C)CCNC(c2cc(Br)n(C)c2)=O)=O)c(F)ccc2ccoc12 c1(NC2CC(NC(C3CCN(CC#C)CC3)=O)C2)ncnc2cc(F)c(F)cc12 c1(OC)cc(C(N2CCCC(NC(C3CCNCC3)=O)C2)=O)ccc1Cl c1(C(=O)NCCC2(O)CCN(C(C(C)SC)=O)C2)cc2cnn(C)c2s1 C(=O)(CCCC(F)(F)F)N1CCN(C(c2cccc(C3CCCN(C)C3)c2)=O)CC1 C=CC(C(=O)NN1CCCC1C(N1CC(C(N)=O)(N(C)C)C1)=O)OC N1(C(c2cc(CO)on2)=O)CCC2(CCN(C(C3OCCCO3)=O)CC2)C1 C(=O)C(C)C(CC)CC.C1(CC)CC2(C1)CC2C(N1CCC(C=O)C1)=O.CC Cc1ccc(C=CC(=O)NC(C)(C)CCCNC(C2CCOC2(C)C)=O)s1 N1(C(c2ccc(C)nc2)=O)CCOCC(CNC(=O)C(F)(F)C(C)O)C1 Cc1ccc(C(=O)COC(=O)COC2CCCN2C=O)cc1C.C(C)(C)C c1(SCC)cncc(C(=O)N(C)CCC2CCCCN2C(c2ccc(C)s2)=O)n1 c1(CC)c(C(=O)N(C)CC2CCN(C(c3c[nH]nc3C(C)C)=O)C2)ccn1C c1(CC(=O)NCC(CN(C(C=CCOC)=O)C)O)cncc(OC)c1 C1(C(=O)NC(CNC(C2C(C)C2C)=O)CO)(COC)CCCCC1 Cc1ncccc1-c1cn(C2COCC2NC(C2CCOC2C)=O)nn1 CS(C)(=O)=NC(=O)C(=O)N.C12CCC1CCN2C(=O)CCc1ccc(Cl)cc1.C C1(N(C(C(C)n2ccnc2)=O)C)CC2CC1N(C(C1CCC(=O)N1)=O)C2 C12(C(N3CCC3)=O)CC(C)(CCO1)C2.Cc1c(C(=O)N)cnn1C(C)(C)C N1(C(c2cc(CC)on2)=O)CCC(C)(C)C1C(=O)Nc1cc(C)ccc1CO C1(C(=O)NCC(C)C#N)CC(C)(C)CCN1C(c1cccc2nccn12)=O Cc1cc(F)cc(C(=O)N(C)CCN(C)C(C2CC(=O)NC2(C)C)=O)c1N c1(NC(c2cc(CNC(C(C)C3CCC3)=O)oc2)=O)cnccc1CO Cc1ccc(C(=O)NCC2CC(C(N3CCC(CO)C3(C)C)=O)CO2)nc1O Cc1ccc(N)c(C)c1.c1ccc(C(C)(C)C)cc1.C(=O)(CC)N(CC)C.C=O c1(C(N(CCNC(c2c(Cl)c(C)n(C)n2)=O)C)=O)cc2c(nn1)CCC2 C1(NC(C(C)(C)OC)=O)CN(C(=O)C(C)(C)C2CCOCC2)CCC1C Cc1cc(O)ccc1CNC1CCC(NC(c2ccc(I)c(O)c2)=O)C1 C1(N(C(c2cc(C)cc(C)n2)C(=O)NCCC2CC2)C)CCc2c[nH]nc2C1 N1(C(=O)C(=C2CCCCC2)F)CC2CCN(C(=O)CCN3CCCC3)C2C1 Cc1c(C(=O)NCC2(F)CN(C(c3cnsn3)=O)C2)noc1C1CC1 C12(C(=O)Nc3cccc(NC(C4CC(C)(C)C4)=O)c3)CCCCC1CCCC2 c1(C(=O)NC(c2nc(Cl)cs2)C)ccc2cc(C(=O)O)ccc2c1 c1(C(=O)NC2C=CC(CNC(C(CC)(CC)CO)=O)C2)c[nH]c2cc(Cl)ccc12 C1(NC(c2cc(F)ccc2Br)=O)COCCN(C(=O)C2=COCCC2)C1 Cc1nc(O)nc(C)c1C(=O)N(C)CCN(C)C(C1CCCCS1(=O)=O)=O N1(C(c2cnn(C)c2)C(=O)NCCC)CCCC(c2ccccc2)C1 C1(CNC(c2cnn(CCO)c2)=O)(NC(C2CC2Cl)=O)CC2CCC1CC2 N1(C(C(CC)NC(C)=O)=O)CCC(NC(=O)C(C)(C)C2CCCO2)C(CO)CC1 C1(N(C(c2c(CC)ccs2)=O)C)CCN(C(=O)CC2(CSC)CC2)CC1 C1(C=O)C2CC(=O)CC12.C1(C)(COC)CCC1.C(=O)CCn1cncn1.N N1(C(CCC2C(C)C2)=O)CCC(O)C(N(C)C(C2CCCC(C)(C)C2)=O)C1 c1(CN2CCC(NC(=O)CCSc3ccccc3)C2)ccnc(O)c1 c1(C(N2CC(C(=O)N)C2)=O)cccc([N+](=O)[O-])c1.c1(NC(C)=O)ccccc1C Cc1csc(C(=O)NC(C2CC=CCC2)C(=O)NCCn2ccccc2=O)c1C N1(C(COCCCCC)=O)CCC(C)(C)C(NC(C2CCN(CC(C)C)C2)=O)C1 Cc1cc(=NCCC2CCOC2)[nH]cc1S(=O)(=O)N1CCC(OC2CCC2)CC1 c1(CNC(C(F)=CCC)=O)c[nH]nc1C(=O)NCC(C)CO c1(C(N2C(C)CN(C(C3NC(=O)OC3C)=O)CC2)=O)cnc2ccccc2n1 Cn1ncc2c(NC3CCCC(NC(=O)CC=C(Cl)Cl)C3)ncnc12 C1CN(C(c2ccnc(-c3ccc(F)cc3)n2)=O)C2CC12.O=C(CC1CC1)NC C1(C#N)(CC(N2C(CNC(C(CCC)OC)=O)CC(OC)C2)=O)CCOCC1 c1(N(C2CC3(CNC3)C2)C(CN(C)C(=O)O)=O)cccc(Br)c1.C(C)(C)C c1(C(N2C(CCC)CN(C(C3CSCCS3)=O)CC2)=O)cc(C)cc2c1OCC2 c1(C(N2CC3CC2CN3C(c2cccc(F)c2O)=O)=O)nsc2ccccc12 CC(F)CCN=c1[nH]c(=NCCc2ccncc2F)c2cccc(F)c2[nH]1 C(=O)(C(C)(F)C(F)(F)F)NCC(N(C(CCCCC)=O)C)C1CC1 C1(NC(C(C)CS(C)=O)=O)C2CC3CN(C(c4cc5ccccc5s4)=O)C1C3C2 C1(CCC)CN(C(=O)C(O)C(F)F)CCN1C(=O)COc1cc(C)oc1C Cc1ccc(C(=O)NCC2CC(C(=O)N)C2)n1C.C1CCC(C(N)=O)O1.C C1(C(=O)NCC=CC(=O)N(C)Cc2n(CC)cnn2)COCC1(C)C c1(OC)cc(C(=O)NC2CCC2)ccc1F.C1(C=O)CCN1S(C)(=O)=O.C C1(C(=O)NCCNC(c2ccc(O)cc2[N+](=O)[O-])=O)CCc2ccc(F)cc2O1 N1(S(CCOC)(=O)=O)CC2CCC(C1)N(C(c1ccc([N+](=O)[O-])cc1OC)=O)C2 C(=O)(C1=NOC(C)(C)C1)N(C1CCN(C(=O)C(C)(C)C2CCOC2)C1)C c1(C(C(=O)NCCC(C)NC(c2cscc2C(F)F)=O)=O)ccc(O)cc1 C1(CC(=O)O)CN(C(=O)C=Cc2cocn2)CCO1 C12(C=O)CCC(CC1)C(C)(C)O2.c1(C(=O)NCCC)ccc(C#N)c(Cl)c1.N N1(C(c2cc(C)[nH]n2)=O)CC2CC(C(=O)NC(C)Cc3nncn3C)C(C2)C1 O=C1COCC2CN(C(=O)Nc3cc(Br)c(C(F)(F)F)cc3F)CCN12 Cc1[nH]nc2ncc(C(=O)NC(C)CCNC(C3CCC3n3ccnc3)=O)cc12 c1(NCC2(O)CCN(C(c3n(C)ncc3)=O)CC2)nc2c(cc1C#N)COCC2 c1(-c2nc(CC(CC)C)nn2C(c2ccc(F)cc2)C)cccc2c(C)csc12 C12(NC(CC3CN(C)C3)=O)CCN(C(=O)C=CC(N3CCOCC3)=O)CCC1C2 N1(C(CCSCC)=O)CCC(NC(c2cn(C(F)(F)CO)nn2)=O)C1C CCCC(CN)C(=O)N(CC(C)(F)F)C CC1(C)CC(CNC(C2C3CC(=O)CC23)=O)N(C(C2CCC(=O)NC2)=O)C1 Cc1ccc(C(=O)NCC2CCOC2C(=O)NCC[Si](C)(C)C)s1 C1(COC)(CN)CN(C(c2n[nH]c(-c3ccccc3)c2Br)=O)CCO1 CCCC(CNC(=O)C(C)(C)c1ccno1)NC(c1c[nH]nc1OC)=O Cc1cc(C(=O)NCC2CC(O)CN2C(=O)CCCC(N)=O)ncc1C#N C#CC(C)(C)C(=O)NCc1ncc(C(N2CCC2C(=O)OC)=O)cn1 C1(NC(=O)CC2CC3(CCNC3)C2)CCCS(=O)(=O)C1 C=Cc1ccc(C(N2CC(O)(CNC(c3scc(C)c3Br)=O)C2)=O)cc1 c1(NC(C2(OCC)CCN(C(C(C)SCC)=O)C2)=O)ccc(O)c(C)c1 N1(C(c2c(CCC)occ2)=O)CC(NC(=O)C(C)(O)C(C)C)CC1(C)C c1(-c2cn(CC(C)NC(C3CC(Cc4cncn4C)C3)=O)nn2)cccc(Cl)c1 O=S(=O)(c1cccc(Br)n1)NC1CC12CCN(Cc1cnccn1)CC2 C1(OCC(C)O)CCN(CC2(c3ccccc3)CC2)C1 CCC(CC(=O)NCC(O)CNC(=O)C(N)=O)CC(C)C C1(C(=O)NCc2cc(C(=O)NC(C#C)C(C)C)on2)CC2CCC1CC2 Cn1nnc(CNC(=O)CC2OCCCO2)c1C(=O)N.c1csnc1C1CC1 c1(C(=O)NC2CN(C(C(C)Cn3cccn3)=O)CC2O)cccn2ccnc12 C(C(C(=O)NCCCCC#N)n1cc(CCNC(C)=O)nn1)OCC N1(C(C(C)OCCCCCC)=O)CCN(C(c2ccc(C)cc2OC)=O)C(C)C1 c1(C(=O)NCC(C)(C2CC2)NC(C2CCOC2)=O)ncn2c1CCCC2 N1(C(c2cn(CCC)nc2)=O)CCC(CC(=O)NCc2cnc(C)o2)CC1 C1(C(N(CCCNC(=O)CSC2CC2)C(C)C)=O)CCC(=O)N(C)C1 C1(NC(Cn2c(C)csc2=O)=O)CCCN(C(c2ccc(C3CC3)cc2)=O)C1C C1(C(=O)NCC2C(C(=O)NC(CCC)c3ccco3)C2)CCOC1(C)C Cc1ccc(CC(=O)NC2CCC2NC(=O)CCCN(C)C)cc1C Cc1ccc2cc(C(=O)NCC3C4CN(C(C5CCC(O)CC5)=O)CC34)cn2c1 C1(CCC(=O)NCCC2CN(C(COC(CC)(C)C)=O)C2)CCCOC1 C1(C(=O)NCC(N(C(c2c(C(C)C)noc2)=O)C)C2CC2)CCOC(=O)CC1 c1(CC)ccccc1C(=O)NC1(C(=O)NC2CCNC(=O)C2)CCN(C)C1 CCC(C(=O)NC1CC(C)(NC(C2CC(O)C2)=O)C1)C1CCOCC1 C(C(C)(COC)CO)NC(CCN(C(=O)CCCCN(C)C)CC#C)=O C(=O)(C(C)C(C)(C)O)N(CCN(C(C1CC(C(=O)OC)C1)=O)C)C C(=O)(CCCC(C)C)NC1CCC(NC(c2cc(C(=O)OC)on2)=O)CC1 c1(C(N2CC(NC(C3C(C)(CC)C3)=O)C(C)C2)=O)cnc2c(c1)ncn2C C(C)(C)(CCCCC(=O)NCC1CCC1)OC.C1(C=O)(N(C)C)CCCSC1.N C1(Cc2nnc(NC(C(C)Sc3ccccn3)=O)s2)CCS(=O)(=O)C1 c1(CC(C(=O)NCC(Cc2ccc(OC)cc2)C(=O)O)N)c[nH]c2ccccc12 c1(NCC(=O)NC(C)CNC(=O)CCF)ccccc1[N+](=O)[O-] C1(OC)CC(CNC(C2CC=CCC2C)=O)N(C(=O)CC(F)F)C1 c1(C(=O)NCC2C3CN(C(C(C)(C)n4cccn4)=O)CC32)cc2c(nn1)CCC2 c1(CC(=O)NC(C(=O)OC)(C)C(C)C)c(Cl)ccc(O)c1Cl c1(CC)ncncc1C(N1CCC(C(=O)N(C)CC2CCCC3CC23)C1C)=O CC(C)(C)CCC(=O)NCC(C(C)(C)C)NC(C1CC2CC1C1CC21)=O c1(C(=O)NCC(CNC(CN(C)C)=O)(C)C)ccc2ccc3ccccc3c2n1 Cc1ncn(C)c(=O)c1C(=O)NC(c1ccccc1)C.C(=O)(C(O)CC(C)C)N C1(C(N2CC(N(C(=O)C3=CCCS3)C)C(C)(C)C2)=O)(OC)CCCC(C)(C)C1 c1(C(=O)OC)ccccc1CCC(=O)NC1(CO)CN(C(=O)CC(C)F)C1 c1(C(=O)NCC(CC(C)C)NC(c2ccc(C)nc2)=O)ccc(C)c2c1CCC2 N1(C(Cc2cn(CC)nc2)=O)CCN(C(c2ccc(Cl)cc2F)=O)CC(C)(C)C1 S(=O)(=O)(c1cc(Cl)ccc1F)N1CC(CC)N(C(=O)Nc2cccc(Cl)c2)CC1 n1(CC)cc(C)c(C(N2CCC(CN=[N+]=[N-])C2)C(=O)NCCCOC)n1 Cc1cc(C(F)(F)F)nc(=NCC2CCCC(NC(=O)CCC3CC3)C2)[nH]1 C1(C(N2CCC(NC(C(C)(C)c3cnc[nH]3)=O)C2)=O)CCCC2(CCCCC2)C1 N1(C(C=C(C)C(C)(C)C)=O)CCC(F)(C)CC1.C1(C)(CC=O)CC1(F)F.N c1(C(c2n(CCCSC)nnn2)NCC2(CO)CCCC2)cc(F)c(Br)cc1F CCCCC(CCCC)C(=O)N(CCNC(C1CCCSC1C)=O)CC c1(C=O)ccc(F)c(F)c1N.C1(C(F)F)(OC)CC(C(=O)N)C1.C1CC1.C Cc1nsc2ncc(C(=O)NCCN(C(C3CCCCN3C)=O)C3CC3)cc12 c1(CC(N2CC(CNC(=O)CCF)C3(C2)CC3)=O)ccc(S(=O)C2CC2)cc1 N1(C(C(C)S(N)(=O)=O)=O)CCOC2(CCC(NC(c3cccc[n+]3[O-])=O)CC2)C1 C1(C)(NC(C2C(NC(C(COC(C)=O)C)=O)COC2)=O)CCCC1C c1(OC)ccccc1-n1cnc(NC(=O)CC(N2CCCCC2=O)C)c1 C1(C(=O)NCCC(C)NC(c2cc(Br)co2)=O)(CC)CC(F)(F)C1 c1(C(=O)NC(C(=O)NCCC(C=C)C)CCF)cnn2c1CCC2 C1(C(N(C)CCOCCC(=O)NCc2cscn2)=O)CC=CCO1 N1(C(C(COCC)(C)C)=O)CCC2C(CCCN2C(C2CC2C(=O)O)=O)C1 CCC(O)C(C)C(=O)NCC1CC(C(=O)NC(C)C(O)C(F)F)C1 C1(O)(CC)CCN(C(=O)C(F)OC(F)(F)F)C1.c1(CC(=O)N)ccc(F)cc1 C12(CNC(c3c(CC)ncs3)=O)CC(C1)C(NC(c1ccnn1C)=O)CO2 c1(OC)cncc(C(=O)NC2CCN(C(C3(CO)CC(C)(C)C3)=O)CC2C)c1C CCC(C)CCCC(=O)N1CCSCC1C(=O)NC(C(=O)OC)C1CCC1 c1(C(N2C(CNC(C3CCC(C)C3)=O)CCC2)=O)ccnc2nccnc12 C(=O)(C(C)CC(C)CC(C)C)N(CCC)CCNC(=O)Cc1cocn1 c1(C(=O)NC(C(=O)OCC)c2ccns2)cc(OC)c(OC)cc1O C1(N(C2CCCCC2)C(N2CCN(C(C)=O)C3C2C3)=O)CCN(S(N)(=O)=O)CC1 c1(NC(C2CN(c3cc(SC)ncn3)CC(F)(F)C2)=O)ccc(C#N)c(F)c1C N1(C(C(C)CN(C)C)=O)CC2(COC(CNC(C3CC3)=O)C2)C1.C1CC1 S(=O)(=O)(c1ccccc1Br)N1CCCCC1.S(C)(=O)(=O)N(CC)C.CCO.C N1(C(c2c(C)coc2)=O)CCN(C(=O)Cc2ccc(Cl)cc2F)C2CCC12 c1(C(N2CCC(C)(C(N3CCC(C(N)=S)CC3)=O)C2)=O)cccc2c1OCCO2 N1(C(C(C=C)(C)C)=O)CC2CCCC(CNC(C3CCCC(F)C3)=O)C2C1 CC1CCN(C(C2COC(C)(C)C2)=O)C(C)C1NC(C12CC(C)(C1)C2)=O c1(CC(=O)Nc2cncc(N3CCCC3)n2)cn2cc(Cl)cc(Cl)c2n1 C1(NCC(=O)NC23C4CC(CC24)C3O)CC(=O)NC(=O)C1.c1ccccc1 C(c1ccc(OCc2ccccc2)cc1)=CC(=O)NCCc1ncc(C)s1 c1(-c2cc(C)[nH]n2)ccc2c(CC(=O)Nc3ccnc(C4CC4)c3)n[nH]c2c1 C(C(=O)N1CC(C)(O)CO1)(c1cn(C)nn1)NC(=O)CCC1(C)CC1 C1(NC(c2cc(C)on2)=O)C2CCN(C(c3cccc4nc[nH]c34)=O)CCC12 c1(C(N(CCCOCCN(C)C(C2CCCCO2)=O)C)=O)ccc(F)c(N)c1F C=C1CCN(C(c2cc(CO)ccn2)=O)C(C(=O)NCC(C)(C)CSC)C1 O=C(C1=CC2CC3CC(C2)CC1C3)NCC1(NC(=O)Cc2ccsc2)CC1 C12(C(=O)NC3C(NC(CCCn4c(C)cc(C)n4)=O)C3)CCC(CC1)C(C)O2 C=C1CC2(C1)CC(C(N1CC(NC(=O)C(CC)N(C)C)C(C)C1)=O)C2 c1(C(=O)NC(CCCNC(C=Cc2c(C)cccn2)=O)C)cc(C)n(C)c(=O)c1 Cc1cnoc1C(=O)NC(C1CCOC1)CNC(=O)C(C)(C)C1CCCCC1 N1(C(C23C(CN(C(c4ccc(O)c(I)c4)=O)C2)C3)=O)CCc2cnccc2C1 c1(C=O)nsc2ccccc12.C1(CC(=O)NC(C2CC2)C)CC(=O)NC1=O.C N1(C(c2ccnc(OC)n2)=O)CCC(C)CC1C(=O)N.C1(CC(N)=O)CC1.C CC(C(=O)NC1(C(=O)NCC2(C)CC=CCC2)CCCC1)S(N)(=O)=O c1(OCC)ncc(F)c(N2CCC(NC(=O)C(O)C(C)(C)C)C(O)C2)n1 C=CC(CC)CC(=O)NCCNc1cc(OC)nc(C(F)(F)F)n1 C1(F)(C(N(CC(C)N(C(CC2(OC)CC2)=O)C)C)=O)C(C)(C)C1(C)C c1(OC)ccc(Cl)cc1-c1nc(CCCN(C)C)nn1-c1cccnc1C N1(C(CCC=CC)=O)CCCCC(C(=O)N(C)Cc2ccncc2F)C1 N1(C(C2C=CCN2C(c2cn[nH]c2)=O)=O)CCN(C2COC2)CC1 c1(NC(CCN2CCN(C)CC2)=O)cc(S(N)(=O)=O)ccc1O Cn1cccc(C(=O)NC2CCC(N(C(=O)Cn3ncnn3)C)CC2)c1=O c1(CN2C(C(=O)Nc3c(F)cc(F)cc3Cl)CC(F)C2)cc2ccccc2cn1 c1(C(=O)NC2CC3CC(NC(C(CC)=CC)=O)C3C2)cccc2nnn(C)c12 c1(CN2CCCN(C(c3cnn[nH]3)=O)CC2)cnc2c(c1)COC2 c1(CC(=O)N(CCCNC(c2c(C)noc2)=O)C)cc(C(F)(F)F)cc(F)c1 c1(NCCSC(C)(C)C)cc(Br)ccc1S(=O)(=O)N1CCCOCC1 CC(C)(CN=c1[nH]c(N2CCCC(C#N)C2)nc2c1COCC2)C(N)=O c1(-c2n(CCC(C)C)ncc2)ccc([N+](=O)[O-])c(CN2CCC(F)(F)CC2)c1 c1(C(=O)NCC2(NC(c3c(C)cncc3)=O)CC2)ccc(Cl)c(N)c1Cl c1(N(C(c2ccc(F)c(F)c2)C)C)ccc(S(=O)(=O)NCC(CO)C2CC2)cn1 N1(CCC)CCCCC1C(=O)NC1(COC)CN(C(C2CC=C(C)CC2)=O)C1 C1(NC)(CNC(=O)COCC(C)C)CCCC1.C(=O)(C)N.C(C)=O c1(CCC(=O)NC2CN(C(c3cc(O)ncn3)=O)CC2O)ccc(Cl)cc1Cl C1(NC(c2n(CC)nc(C)c2)=O)CN(C(C2CCCCC2O)=O)C2CCCC12 CCC(CC)(C(=O)NCC1CCN(C(=O)CNc2cccnc2)C1(C)C)OC c1(NC(C2CC3N(C(COCC(=C)C)=O)C(CC3)C2)=O)ccc2ccncc2c1 CCC(CC)C(C(=O)NCCC(CC)(CC)NC(=O)Cc1csc(Cl)n1)OC C1(C(=O)NC(CC=C)C2CC2)C2CCC(C2)N1C(=O)C(O)C1CCCC1 c1(C(N2CCC(C)(CNC(c3c(C)[nH]cc3)=O)C2)=O)csc(S(C)(=O)=O)c1 N1(CC2CC(F)C2)CCCC(CC2CCC2)C1 c1(NCC(=O)NC(C)C)cccc2c1COC(=O)N2 c1(NC(c2nnnn2C(C)(C)CC)C2(CC)CCC2)cc(OC)c(Cl)cc1.O CCCCC(O)CCC(=O)N1CC2CN(C(=O)C=Cc3nccs3)CC2C1 N1(C(c2c(C)cn(C(C)C)c2)=O)CCCOC(C)C1.c1(C(=O)N)cc(Cl)n(C)n1 c1(N2CCCC(C(C)NC(c3cc(C(F)F)ncn3)=O)C2)ncn(C)c(=O)c1Br c1(C(N2CCCC(CNC(CC3OCC(C)(C)C3)=O)C2)=O)cc(Cl)cc(Cl)c1F C1(C(=O)OC)OC(C(=O)NC2CCCCC2)CC1C.c1(C(=O)N)oc(C)cc1C C(C)(C(C)(C)NC(=O)C(C1(O)CCCC1)F)NC(CCSCC(C)C)=O CC1(C)CCN(C(c2ccn(C(C)(C)C)c2)=O)C1.c1(C(=O)N)c[nH]c(C#N)c1 N(C1CCCc2ccccc21)(C(=O)Cc1ccccc1SC)CC#C c1(CC(N2CC(NC(c3cc(C)[nH]n3)=O)C(F)C2)=O)cc2ccccc2c(=O)o1 O=C(C1=CCCN(C(=O)C=CC(F)F)C1)NCC1CC1c1ccccc1 c1(OC)ccc2c(c1)OCCC2NC(=O)NC1CCCSCC1 Cc1cc(Br)c([N+](=O)[O-])c(C)c1C(=O)OCC(C)O Cc1cc2ccc(C(=O)NCC3CC4CCC3N4C(=O)CO)cn2c1.CC(F)F C1(OC)CCCN(C(=O)C(N2CCOC(C(=O)N(C)C)C2)=O)C1C CC(CC(F)(F)F)C(=O)NCC1CCC2(CN(Cc3cnn(C4CC4)c3)C2)O1 CN=c1cc(C(N2CCOC(C(=O)NC(c3ccc(C)nc3)C)C2)=O)cc[nH]1 c1(C(N2CCOCC2)=O)ccc2c(c1)CCC2.C1(C(=O)N)CCCS(=O)(=O)C1.C N=c1[nH]nc(C2CC2C(=O)N)s1.C1CC(CC)C1.C(=O)C.C(=O)C1CC1 Cc1cnc(NCC2CC(C)C2)c(S(=O)(=O)NC2CC(F)C2)c1 c1(C(C)C(=O)NCC2CCN2C(=O)CC2CC=CC2)ccccn1 N1(C(C(C=C)OC)=O)CC(C(N2CC(=O)NC(=O)C2)=O)C(C)(C)C1 Cn1ncc(CNC(C2CC23CCC3)=O)c1C(=O)NCCSC(F)F C1(NC(C(C)(C)C2CCCCO2)=O)CC(NC(C2SCCCS2)=O)CC1O c1(C(=O)NCC(CNC(=O)CC(=O)N(C)C)OC)cnncc1C N1(C(c2cnc(C(C)C)s2)=O)CC(CCNC(=O)CN2CCCCC2)OC(C)C1 C1(N(C(=O)C(C)OCCO)CC)CCN(C(c2ccc(Cl)o2)=O)C1.CCO n1(CCC(=O)NCC2COCC2)cnccc1=O.c1(C(=O)N)cnn(C2CC2)c1 N1(C(c2n(CC)ncc2Cl)=O)CCN(C(c2cc(N)c(F)cc2F)=O)C2(CC2)C1 c1(C(N(C)CC2CCCCN2C(c2cscn2)=O)=O)ccc2c(c1)oc(=O)n2C N1(C(C2(C)CC(=C)C2)=O)CC2CN(C(c3ccccc3[N+](=O)[O-])=O)CC2(C)C1 CCC(C)(CNC(c1cc(CO)c(C)o1)=O)C(=O)NCc1cnn[nH]1 C1(NC(C(N2CCNC2=O)C)=O)C2CC3C1C3C2C(N1CCC(F)(CF)C1)=O O=C(C1CCCc2nccn21)NCCCc1cn(CC2CCCCC2)nn1 c1(OC)ccc(S(=O)(=O)NCC(C(F)(F)F)n2cccn2)c(CC(=O)O)c1 CN1CCCC(C)(C(=O)NCC2OCCC2C(=O)N(C2CCCC(O)C2)C)C1 N1(CC(C)C)CCCC(CNCC(C)CCc2ccc(Cl)cc2)C1 N1(C(C(=O)NCC(CNC(CC=C)=O)F)C)CCNC1=O c1(C(=O)NC2CCCC(C(=O)NCCS(C)(=O)=O)C2)cc(Br)c(F)cc1F Cc1c(Cl)ccnc1C(=O)NC1CC2CCC1N2C(=O)C(C)(O)C(C)C C(=O)(C#CC1CC(F)(F)C1)N.c1(CCC(=O)NCCC)nnc(-c2ccsc2)o1 CC(C)(C)C1=NOC(C)(NCC2CC3CCC(C2)N3C=O)C1.C(C)(C)C.O c1(OC)cc(C(=O)NC(CNC(=O)CC(C)n2cc(Br)cn2)C(C)C)on1 Cc1oc(Cl)nc1C(=O)NC1C2CC1N(C(c1cc(C3CC3)n(C)n1)=O)C2 CC1CCC(C(=O)NC2CCCCNC2=O)CN1C(=O)CN1CCSCC1 C1(C(N(C)CCO)=O)CCC(N(C)C)CC1.C(c1cccnc1)=CC=O.CC N1(C(c2c(OC(C)C)ccc(Cl)c2)=O)CCN(C(c2cc(O)no2)=O)CC(O)C1 C1(C(N2CC3C(CNC(c4c(C)nccn4)=O)(C3)C2)=O)CCCCC12OCCO2 Cc1cc(N)c(C(N2CCC3C(C2)CN3C(C2CC(Cl)(Cl)C2)=O)=O)c(F)c1 N1(C(Cn2c(CCC)ncc2)=O)CCC(NC(=O)C(C)(O)COC)CC1C c1(N2CCC(C(F)(F)F)(OC)CC2)cc[nH]c(=NCCCCCS(C)(=O)=O)n1 CC1CCCCC1CC(=O)NCCC1CN(C(=O)CN2CCCC2=O)C1 c1(N(C(=O)CN2CCN(C(=O)CNC=O)C(C)C2)C)cccc2ccccc12 N1(C(c2ccc(OC)s2)=O)CCC12CN(C(=O)CCc1ccoc1)C2 CC1CC(C(=O)N(C)CCC2CCCCC2)CCN1C(c1ccc(=O)n(C)c1)=O c1(C(N(CCNC(C2CCC(C#N)C2)=O)CC)=O)cc(C)c(Cl)cc1O C(=O)(C1COc2ccccc21)N1CCC2(CC(NC(C(C)SCC)=O)C2)CC1 c1(C(=O)NC(C(N2CC(C)C(CO)C2)=O)C2CC2)ccc(F)c(O)c1 C(C)(C(O)C(=O)OCC(=O)NCC(c1ccc(C)cc1)=O)OC N(C(=NCCN1CCC1)NC1CC1)CCOC.C1(C(C)C)C(=O)N1 c1ccc([N+](=O)[O-])cn1.C1CC(F)(C=O)C1.C1(C=O)CC1.C1CC1.CC.N CCC(CCC(=O)NC1CCCCCC1OC)NC(C1CCC2CC1CO2)=O Cc1ccc(C(=O)N)c(C)c1.C1CCN(C(=O)COCP(C)(C)=O)C(C2CC2)C1 N1(C(CCCNC(=O)OC)=O)CC2CCC(C1)CC2.c1(CCC(=O)N)ncnn1C C1(C(N(CCCN(C)C)CCNC(=O)C=CS(C)=O)=O)CCOCC1(C)C c1(OCC)cc(C(=O)N(CCCC)CC)cc(F)c1.C(=O)C(CO)N(C)C.N c1(C(=O)OCC)cc(C)c(C)c(Br)c1.C1(C)(C(=O)O)CNC(=O)N1 c1(C(=O)NC2CC(C)CN(Cc3ccc(Br)cc3)C2)cccc2c(O)nccc12 C1(COC)CN(C(c2ccc(F)c(O)c2)=O)CCN1C(C1CN2CCC1CC2)=O N1(C(c2ncc(C(C)C)o2)=O)CCN2CC3(CC3)CC2C1 N1(C(C(c2ccccc2)NC(CCc2ccc(C)o2)=O)=O)CCOC(C(C)C)C1 c1(C(N2CCCC(C)(C(=O)NC3CN(C)C3)C2)=O)ccc(Br)c(C#N)c1 C1(C(C)C)CN(C(=O)CC2CCN2C(=O)CCn2cnc(=N)[nH]2)CCCO1 N1(C(C(C(=C)C)(C)C)=O)CC(C)OC(C)(C)C1.c1(C=O)ccc(C(F)F)o1.N CCC(O)(CC)c1cn(CCCCCNC(=O)C(c2cnn(C)c2)=O)nn1 N1(C(CC=C)=O)CCC2(CC1)CC(NC(C1CCCSC1)=O)c1ccccc1O2 Cc1nccc(C(=O)NCC2CCCCN2C(=O)CCC(C)CN(C)C)c1C CN(C)S(=O)(=O)NCC(N1CC(NC(=O)CO)C(C(F)F)C1)=O c1(C(=O)NCC(N(C(C(CCN(C)C)O)=O)C)C2CC2)cnn2c1CCC2 c1(OC)c(F)cc(C(=O)NC(C2CN(C(=O)CCSC)CCO2)C)c(N)c1F c1(C(=O)OC)ccc(C(=O)NC2CCS(=O)(=O)C2C)c(F)c1 N1(C(=O)Nc2cc(Cl)nc(Br)c2)CC2(CC2)c2ccccc21 CS(=O)(=O)CCCC(=O)N1CCC2(CC1)CC2C(N1CCN(CCO)CC1)=O C=C(CO)CCNC(C1CC(c2ccccc2)C1C)=O C(CN=C(NCc1cccs1)NC)N(C(C)C)C(C)C.C1CC2(C1)CC21CC1 C1(C(=O)NC2CCC2C(=O)NCCCC(C)(C)O)(OC)CCC(C)C1 C(CC1c2ccccc2-c2ccccc21)NC(CCOC)C(C)C N1(C(c2ccc(I)cc2O)=O)CC2CCN(C(c3cc(Br)ccn3)=O)C2C1 C1(C=O)CCS(=O)(=O)N1.c1(CCC(=O)N(C(c2ccccc2)C)C)ccncn1 c1(C(=O)NC2CCC(NC(C(CCSC)O)=O)CC2)cc(Cl)cc2c1NCCC2 c1(C(N2CCC(N(C(CC(CC)OC)=O)CC)C2)=O)cccc2ncn(C)c12 C(=O)(CC(C)CC(F)(F)F)N1C(C)CN(C(C(c2cncn2C)OC)=O)C(C)C1 C1(N(C(=O)CC2(C)CC2)C)CCN(C(c2cn(CC3CCOC3)nn2)=O)CC1 C1(NC(CC2ON=C(CC)C2)=O)CN(C(C2CC(SC)C2)=O)CC12CC2 C(=O)(C(C#N)(CC)CC)N1CC2(CN(C(C(CC)CC3CCCC3)=O)C2)C1 Cc1nn(CC(N2CCCC2CNC(c2cnc(C(C)C)s2)=O)=O)c(C)c1C c1cn(C)nc1C(F)(F)F.c1(CCCC=C)cn(C2CCC(C(=O)NC)C2)nn1 C=CCC(CC)C(=O)NC(C(=O)NCC1CCCNC1=O)C1CCOC1 N1(C(c2ccn(CCOC)n2)=O)CCC2C(NC(C3CCCS3)=O)C2C1 C(=O)(C(C)=Cn1ccnn1)NCC1CCN(C(C(CCC)(C)O)=O)CC1 N1(C(N(CCC#N)C)=O)CCC2(C(=O)OC(C)(C)C)CC2C1 c1(-c2c(CN3CCCN(c4nccc(Cl)c4)CC3)cccn2)c(Cl)cc(Br)cc1Cl C1(NC(=O)C(F)C2CCOC2)CCC2(CC1)CN(C(c1cnco1)=O)C2 N1(C(CSc2n(C)ccn2)=O)CCOCC1(C)c1cn(CCC(F)(F)Cl)nn1 c1(-c2cc(SC)c(F)nc2)ccnc2ccc(NC(=O)Cn3ccc(C)n3)cc12 N1(C(c2cnc(=N)[nH]c2)=O)CCCC2(NC(c3nccc(Cl)c3F)=O)CC2C1 C=C(Cn1cc(CN(C)C(c2csc(-c3cccs3)n2)=O)nn1)C1CCOCC1 C1(CC)CCCC1C(=O)N.c1(C2C(NC(C3(CC)CC3)=O)C2)cncs1 N1(CC=O)CCC(C(F)(F)F)CC1.C(=O)(C(F)C1CCOC1)NC.C1CC1.C S(=O)(=O)(c1cc(Cl)ccc1F)N1CC2CN(C(c3ccc(Cl)c(C)c3F)=O)CC21 Cc1nc2ccc(C(=O)NC(C)CNC(c3ccc(-c4ccco4)o3)=O)cc2[nH]1 N1(C(c2ccc(Br)c(Cl)c2F)=O)CCCC2C1CCN2C(=O)Cc1ccccn1 C(=O)(C(O)CCCNC(=O)C(C)(C)N(C)C)NC(c1cccnc1)CC c1(C(N2C(C(C)O)CC2)=O)ccc(Br)cc1N=[N+]=[N-] N1(C(C=C=C(C)C)=O)CC2(CCOCC2)CC1CNC(c1ccccn1)=O C12(NC(Cn3c(C(C)C)nnn3)=O)CCC(CN(C(C3CCO3)=O)C1)C2 c1(C(=O)OC)ccccc1CCN1CCC(c2cc(C)no2)CC1 CC1C(C)N(C(c2cnn(C3CC3)c2)=O)C(C)C(=O)N1C c1(CN(Cc2cn(C(CC(=O)NC3C(C)CCC3)(C)C)nn2)O)ccc(Cl)c(Cl)c1 c1(C(=O)NCC(CNC(C(C)Cn2cccn2)=O)F)cnn(C)c1Cl c1(OC)cc(COCC(F)(F)F)c(-c2ccc(OC)cc2)c(Cl)c1O Cc1cc(CC(=O)NC(C)C)cc(C)c1.c1(C(=O)N)cccc(OC(F)(F)F)c1 O=C1CCC(C(N2CCC(Cc3cn(-c4ccccc4I)nn3)C2)=O)CN1 c1(OC)cc(C)cc(C(=O)NC2(CN(C)C(c3cnns3)=O)CC2)c1O C(C)(CCC(=O)NC(C)Cc1ccco1)NC(Cc1c(C)non1)=O c1(C(N2C(C)CC(NC(C3CN(S(C)(=O)=O)C3)=O)C2)=O)ccn2nncc2c1 C(=O)(CCC(C)(C)C#N)N(C)CCNC(c1scnc1C(F)F)=O N1(CCC(F)(F)F)CCN(CCOc2cncc(Cl)n2)CC1 C(=O)(CCCC(=O)N(C)C)NC(C(=O)NC(CCC)C(=O)OC)CCN(C)C CCCCCC(CC)C(=O)NCC(C)CN(C(=O)CC(c1cccs1)C1CC1)C C=CCCCC(C)(C)C(=O)N1C2CC1CN(C(=O)C(C(C)CC)N(C)C)C2 C(CS(=O)(=O)N(CC(F)(F)F)CC(=O)O)(C1CC(F)(F)C1)OC CS(=O)(=O)CCCC(=O)N1CCCC1C1(NC(=O)C(CO)NC(N)=O)CC1 N1(C(C(C2CCN(C(c3cc(CC)no3)=O)C2)F)=O)CCC(F)(F)C(O)C1 C1(C(=O)NC(CC(C)C)CNC(C23CC2C3)=O)CCc2nncn2CC1 C(CN=C(NCc1ccnn1C)NC1CC2CCC1O2)c1c(C)n(C)nc1 N1(C(c2c(N)cccn2)=O)CCC2(C=C(C(=O)NC3CCC(=O)NC3)C2)C1 N1(C(C)=O)CCN(C(=O)C(C)N(C(c2cc[nH]n2)=O)C2CC2)C(C)C1 C(=O)(C1=CCCC1(C)C)NC1CC(NC(Cc2c(C)cccc2F)=O)C1 c1(-c2nc(C3(CSC)CC3)on2)cc(Br)c2ccccc2c1F C1(NC(C=CC=CC)=O)COC2(CCN(Cc3cccc4[nH]ccc34)C2)C1 Cc1ncc(NC(c2cnn(CCNC(c3nnsc3N)=O)c2)=O)c(C)n1 c1(C(N2CC3CN(c4nc(C)nc(=N)[nH]4)CC3C2)=O)ccc2nnn(O)c2c1 N1(C(c2c(CC)[nH]c(=N)s2)=O)CCCN(C(=O)CC2CN3CCC2CC3)CC1 Cc1[nH]c(=N)nc(O)c1CCC(=O)NC1CCC1.C1(C)(C=O)CNC(=O)C1.C C(=O)(C(C)CCc1cccc(F)c1)N(C1CCN(C(C(CC)C)=O)C1)CC CC(C)S(=O)(=O)CC(=O)NC1COCCN(C(=O)CC2CC(O)C23CCC3)C1 c1(C(N(C)Cc2c(C)ncs2)=O)c(Cl)ccc(O)c1Cl C1(CNC(CC(C)(C)O)=O)C(C2CC2)CCN1C(c1cc(Cl)c(F)c(Cl)c1)=O c1(C(=O)NCCCCN(C)C(C2CCC(=O)N2)=O)c[nH]nc1F c1(C(=O)N)n[nH]c2ccccc12.N1(CCC)CC(C(=O)NC(C)C2CC2)CC1=O c1(C(N2CCC(NC(C(Br)=C(C)C)=O)CC2)=O)ccc2nc(C)[nH]c2c1 C(C)(C(C)C(=O)N(Cc1ccc(C)o1)OC)NC(CC(=C=C)C)=O c1(C=O)cccc2c(C#N)c[nH]c12.CCC(C(=O)N(CCC)CC)NC(N)=O.N C(CC(=O)NCCC(O)C(F)F)(C(F)F)NC(c1n[nH]c(CC)c1C)=O C(=O)(CC1CC(=O)c2ccccc21)NCC1(C)CCCC1NC(c1csnn1)=O c1(OC)ccnc(F)c1C(N1CCN(C(C2CCC23CCC3)=O)C(C2CC2)C1)=O C1(C)(NC(C2C(OC)CC2)=O)CCN(C(c2ncccc2)=O)C1.C1CCC1.N C1(C)(CNC(CCN(C(CSCCOC)=O)C2CC2)=O)CCN(C)CC1 CCCC(C)(C)CC(=O)N1CCC(CNC(C2CC=C(C(C)C)CC2)=O)C1(C)C C(=O)(C(F)(F)C(F)(F)F)NCCC(CNC(CCCOC(C)=O)=O)(C)C Cc1ccoc1CC(=O)NCCC1(O)CN(C(C2CCCS2)=O)C1 N#Cc1ccc(OC(=O)NC2CCN(Cc3ccccc3)C2)cc1C(F)(F)F C1(CNC(c2nc(C)sc2C)=O)CC(C)CN(C(c2cccn2C2CC2)=O)C1 N1(C(=O)NCc2ccc(-c3nc(=O)o[nH]3)cc2)CCCN(CC2CCCC2)CC1 CON=Cc1ccc(C(=O)NC(CNC(=O)CCOC2COC2)CC(C)C)cc1 N1(C(C(CC=CC)C)=O)CC(C)(C)OCC1CNC(C1(CCO)CC1)=O C1(C)(C(=O)N)CC(C(F)(F)F)=NO1.c1(C(N(CCCC)C)=O)c(C)cnnc1O c1(N2CC(C)C(CNC(C3CCOC3)=O)CC2)[nH]cnc2nc(Cl)cc1-2 c1(CC)nc(C)oc1C(N1CCC(C)C1)=O.c1(C(=O)N)cn(C(C)C)cc1C N1(C(c2ccc(Cl)cc2F)C(=O)NCC(=C)C)CC(C)C(P(C)(C)=O)C1 Cc1cc(C(=O)NCC(C2CCN(C(=O)Cc3cnc[nH]3)CC2)(C)O)nc(C)c1 CC1(C)CCC(=CC(N2CC(c3ocnc3CNC(=O)C)C2)=O)CC1.CCF CCCC(CC)CCC(=O)NCCCCC1CN(C(=O)CC2CC2(Cl)Cl)C1 C1(NC(C=NOC)=O)CN(C(c2cc(Cl)c(Cl)cc2C)=O)C2(CCCOC2)C1 C(C)(CCN=c1cc(C)[nH]c(=NCCc2cc(C)n(C)n2)[nH]1)N(CCC)C N1(C(C(N2CC(CC(C)NC(c3ccc(CF)cc3)=O)C2)=O)C)CCCCCC1 Cc1conc1C(=O)NCC(C)CN(C(=O)CC1C(C)C1(F)F)C N1(C(c2ccc(OC(CC)C)cc2)=O)CCC(NC(=O)C(F)=CCCF)CC1C C1(C)(NC(CCCOCC=C)=O)CCN(C(C2(C)CC(C#N)C2)=O)CC1 C1(C)(CNC(C2CC(=C)C2)=O)COCCN(C(C2CCCC(F)(F)CC2)=O)C1 N1(C(C(CC=CC)C)=O)CCCC(F)(C(=O)NCCN(C)C2CC2)C1 N1(C(C(c2ccoc2)NC(c2c(C)oc(C#N)c2)=O)=O)Cc2ccnn2CC1C c1(CCC(=O)NCC=CCNC(C2CCN(C)C2)=O)ccc(Cl)nc1 C1(C(N)=O)C(=O)NCCCN1Cc1ccc2c[nH]nc2c1 CC(C)C(C)(O)C(=O)NCC#CCNC(C1(c2ccccc2)CCCCO1)=O N1(C(CCN(CCC)C)=O)CCC2(CCCN2C(c2cc3nc(C)sc3[nH]2)=O)C1 CP(C)(=O)CNC(c1c[nH]nc1C(F)F)=O CC1(C(=O)NC2CCCC2)CC2CCC(C1)S2.N1(CC=O)C(=O)CNC1=O.C c1(C(N2CC(C(C)(C)O)(CNC(C3C(=C)CC3)=O)C2)=O)cc(Br)ccc1F Cc1nocc1C(=O)NC(CNC(=O)CC1CCCCC1)Cc1ccccc1 CN1CCn2ncc(C(=O)NCCCCNC(C3CCC(C)(O)CC3)=O)c2C1 C=CC(C)(CC)C(=O)NCC1CCC(C)N(C(c2csc3cncn23)=O)C1 c1(OC)nc(C)cc(=NC2CCCCN(C(C3CC4CCC3O4)=O)C2)[nH]1 CCC(C#N)C(=O)NC1CC(NC(c2sc(F)cc2Br)=O)C(O)C1 Cc1cc(C(N2CC(NC(=O)C(F)F)C3(CC3)C2)=O)cc(Cl)n1 C1(C=O)CCCCC(=O)N1.c1(CC(=O)N(CCC)CC)csc(C2CC2)n1.N Cc1cccn2cc(C(=O)NCC3C(C)CCN3C(C3CC3(F)F)=O)cc12 CCC(C)(O)C(=O)NC1CCCC(CNC(=O)C(C)OC2CCCC2)C1 CC(CCCNC(c1cn[nH]c1)=O)NC(C1CC1C)=O CCC(C(C)(F)F)NC(C1C=CCCN1C(=O)CC12CCC(CC1)C2)=O C1CCC2(CC1)CN(C(=O)C#CC(=O)N(C)C)CCO2.C(C=O)NC(=O)NC.N c1(C(=O)NCC(CC)(C)NC(C2CCO2)=O)coc2cc(OC)ccc12 N1(C(CCC(C)(F)F)=O)CCC(NC(c2ccncc2Cl)=O)CC(C)(C)C1 c1(C(N2CCC(O)(C(N(C)Cc3ccc(Br)cc3)=O)C2)=O)cccc2[nH]ncc12 C(CCC(N)=O)(C(=O)NCC1CCOC1)NC(C)=O.C1(C(=O)N)CCOCC1 N1(C(c2cc(OC)no2)=O)C2CCC1CN(C(=O)C)C2.C(=O)(C)N.C(C)=O c1(C(=O)NC(CN(C(CCCCC)=O)CC)C)cc2c(Cl)cccc2s1 C1CC2(C1)CS(=O)(=O)C2.C1(N(C(=O)C=Cc2cc[nH]c2)C)CCCCN(C)C1 c1(C(N(C(CNC(c2cccc(CC)n2)=O)C)CC)=O)cc(OC)cnc1F C=C(CNC(C1CC(NC(c2cnc(CC)o2)=O)CCO1)=O)C(F)(F)F c1(OC)cc(C(N2CCN(C(=O)Cc3ccc(C)o3)CC2)=O)cc([N+](=O)[O-])c1C c1(C(=O)NC(C2(O)CN(C(Cc3c(C)ncs3)=O)C2)C)cnn2cnnc2c1 N1(C(C2(F)CCCN(C(CSC)=O)C2)=O)CC2CCCCC2C1C C(CC(C(=O)NCc1cc(C)cs1)NC(C1CCCCN1C(C)=O)=O)OC c1(OC)ccc(Cl)c(C(=O)NCC2CC(F)CN2C(C2CCC(=O)C2)=O)n1 C1(C(=O)Nc2cncc(C)c2)CN(C)CCN1C(=O)CC1CCCNC1=O Fc1c(CNC2(c3nn[nH]n3)CC3CCC2CC3)ccc(Cl)c1Br C1(NC(C(n2cc(CN3CCSCC3)nn2)C)=O)CCC2(CC1)CC2 C1(c2cc(C(=O)OC)on2)CN(C(c2nn[nH]c2C(=O)O)=O)CCO1 n1(CCC)nccc1C(c1nnnn1CCCF)NCC1(c2noc(C)n2)CC1 C=C(C)c1cn(CCC2CN(C(=O)CC(C)CN(C)C)CCCO2)nn1 Cn1cnc2c[nH]c(=NCCNC(c3cc(C(N)=O)c[nH]3)=O)nc12 C1(OC)CCCC1CNC(C1(CNC(c2cc(C)no2)=O)CC1)=O c1(CC)c(C(N)=O)cnn1-c1ccc(NC(C2(c3cccs3)CC2)=O)cc1 C(N=c1[nH]c(=NC2CCS(=O)C2)[nH]c2c(F)cccc12)c1c(C)cn(C)n1 CCCCC(CC)CC(C(=O)NC(C)CC)N1CCCC1CC(N)=O C(C)(CC(C)C(F)F)NC(C(CCOC)NC(C1CC(C)N(C)C1)=O)=O c1(OC)cnnc(C(N2CC(OC)CC2CC)=O)c1.C1(C)(CC=O)CC1(Cl)Cl Cc1cc(C(N2CC3CC2C3NC(C2CCSCC2)=O)=O)oc1C C1(CNC(c2cc(C)ncn2)=O)CCCC12CCN(C(=O)C=CI)CC2 C1(NC(CCc2ccc(C)o2)=O)(CNC(=O)CC(F)(F)Cl)CCCCCC1 c1(NC(C2CC(C)CN2Cc2ccc3ccnn3c2)=O)cc(Br)ccc1[N+](=O)[O-] C(CC(N)=O)(C(=O)O)NC(c1cc(C)n(-c2ccc(F)cc2)n1)=O C1(C)(C(N(C)Cc2nnc(CC)o2)=O)CCN(C(=O)C=CC2CCCC2)CC1 N1(CC2CCC(C(N)=O)O2)C(=O)CN(CC2CCCOC2)C1=O c1(NC(=O)Nc2cccc(Oc3ccccc3)c2)ccnc2cccnc12 C1(CNC(C(n2cc(Cl)cn2)C)=O)C2CN(C(=O)Cc3ccccc3)CC12 C(=O)(CC(C)C(C)C(C)C)NCCCNCc1c(C)ccc(N)c1 C1(NC(N2CCCC(C)C2)=O)C2Cc3c(Br)cccc3C12.C(=O)(C(F)(F)F)N C1(C(N(CCN(C(=O)CCc2ncc[nH]2)CC)CC)=O)CCCC(C#N)C1 CCCCC(F)C(=O)NC1C=CCCC1C(=O)NC(CC)C(C)(C)C c1(C(N2CC(O)(C(C)NC(c3cncc(CC)c3)=O)C2)=O)cccc(N)c1.O C#CCC(O)C(=O)N(CC(C)O)CCNC(C1CC(F)(F)CS1)=O N1(C(C(C)=C2CC2)=O)CCc2cc(CNC(C3CCC(C)(C)C3)=O)ccc2C1 C1(N(CC(=O)N(C(CC)C)CC)CC)CCS(=O)(=O)C1.CCC#N N1(C(c2cn(CCC)nc2)=O)CCN(C(c2cc(COC)cs2)=O)C(C)C1C C(=O)(C(CC(C)C)n1ccnc1)N1CCC(NC(c2cc(C)ncc2)=O)C1C C(=O)(CCCC1CCCCC1)N(CC(CC)NC(C1C(=C)C1)=O)CC C1(NC(C=CC)=O)CC(CNC(c2ccc(=O)oc2)=O)C1(C)C C(CC(=O)N1CCC(c2ccco2)C1)(C(F)F)NC(c1ccc(C#C)o1)=O c1(C(=O)NC2C=CCN(C(C3C=CCC3)=O)C2)cc([N+](=O)[O-])cc2c1OCCO2 c1(CCC)cc(C(=O)NC(c2cnn(C)c2)C(=O)NC(C2CCOCC2)C)n[nH]1 N1(C(C(C(C)C)C)=O)CC2(C1)CN(C(C1CCCC(C)C1)=O)CC2CO C(C(=O)NC1CCCCC1NC(c1ccc(Br)cc1)=O)(C(C)C)OC Cc1ccc(S(=O)(=O)N2CCC3(CCCOC3)CC2)c(I)c1 C=CC(C)(C)CC(=O)NC1(C(=O)NCCO)CC1.C(C)C(C)n1cccn1 CC1(C)CC(CC(=O)NCCOCCOCC)C1.c1(C(=O)N)ccns1 CC1C(NC(=O)C(C)(C)C)CCCN1C(=O)C(F)C1CCOC1 N1(C(C(C)C)=O)CC2CCC(N=c3[nH]n(C)cc3[N+](=O)[O-])C2C1.C(=O)(NCC)N Cc1c(C(=O)NC(C)CCNC(c2cn(CCCF)nn2)=O)cncc1N C12(C(=O)NCC(N(OC)C)=O)CC(C)(CN1C(c1cc(C)ccc1O)=O)C2 N1(C(CC(CC)O)=O)CCC2(CCN(C(=O)CCc3cnccn3)C2)C1 c1(C(=O)NC2CC(NC(c3cc(OC)no3)=O)C(O)C2)cc(C)cc2c[nH]nc12 CCCCC(C(=O)N(CC(C)(C)C(=O)NCCN(C)OC)C)C(C)C C(C(F)(F)CO)NC(C1N(C(C2(C(C)C)CCC2)=O)CC1)=O N1(C(C(C)SC)=O)CCOC(C(=O)NCCSC(F)F)CC1 C1(NC(c2ccccc2C2CC2)=O)C2CCC1CN(Cc1cnc(O)nc1O)C2 CC1CC(NC(=O)CN2CCCCC2)CN1C(=O)C(F)CC1CCOCC1 CC1(O)CCN(C(C2CCN(C(=O)c3cc(C#N)cs3)O2)=O)CC1O c1(C(=O)OC)c(OC)cccc1NC(=O)NCC(c1ccc(F)cc1)(C)O CC(C)CC(CCO)NC(c1ccc(Cn2cc(C3CCCN3C)nn2)o1)=O C1(C(C)(O)CNC(=O)C(c2cccnc2)O)CCN(C(=O)CCC2CCC2)CC1 Cc1cnc(C(N2CCN(C(c3ncccn3)=O)CC2)=O)nc1 c1(CCC(=O)NC23CC(NC(C(C)CF)=O)(C2)C3)ccc(=N)[nH]c1 N1(C(CC(C)(C)C#N)=O)C(CNC(C2(C)CC=CCO2)=O)CC2CCCC12 O=C(CC1=CCCC1)NCCCCNC(c1ccnn1CCF)=O N1(C(CC2CC(C)C2)=O)CC(=O)NC2CN(C(=O)COc3cnn(C)c3)CCC12 CC1OC2(CNC(=O)CC=CC(C)(C)C)CC1C2.C(=O)(C(C)(C)CO)N C=CC(CC)C(=O)N1CCC(CC)C1C(N1CCOCC1CCOC)=O c1(OC)ccc(CO)c(NC(C2CC(C)CN2C(=O)Cn2ccnc2)=O)c1 C(=O)(CCC(=O)N1CC(O)CC1CNC(=O)C(n1ccc(C)n1)C)NCC N1(C(CC(C(C)C)C)=O)CCC2(CC1)CN(C(C1CCC(=O)N(C)C1)=O)C2 N1(C(c2cccc(Oc3ccc(C#C)cc3)c2)=O)CCC(C2(O)CCCC2)CC1 c1(CC)cc(C(=O)NC2CCCC2NC(C2ON=C(C)C2C)=O)nn1CCO C1(C(=O)NC2CCN(C(=O)CC3CC4CC4C3)CC2)CC(c2cccnc2)=NO1 CCC(C)(CNC(=O)COC1CC=CC1)C(=O)N1CC2C(C1)C2(C)C c1(NC(c2c(C)oc(-c3ccco3)n2)=O)cccc(S(=O)(=O)NC(C)(C)C)c1 C(=O)(C(C(C)C)NC(=O)CC)N1CCC(CCCC)C1 C1(CC)CN(C(c2ccc(=O)oc2)=O)CCC1NC(=O)CCc1cccnc1F C(CCC(C)CC(=O)N1CCN(C(c2sc(C)nc2C)=O)C(C)C1)=C(C)C c1(C(=O)NC(CC2CN(C(COC)=O)C2)C)ccc2c(c1)nc(C)c(=O)n2C c1(C(=O)NCC(CC)NC(=O)CC2C=CS(=O)(=O)C2)cc(C)cnn1 C12(C(N(C)Cc3ncc(C)nc3)=O)CCCC1CCN2C(c1cc(C)c(C)s1)=O CC1=C(C(=O)N2CCC(C)C(NC(c3cn(CCCF)nn3)=O)C2C)CCCO1 c1(N2C(COC(=O)NCCC)CCC2)nc(-c2ccco2)n2ccccc12 N1(Cc2c(-c3cn(C)nc3)n[nH]c2)CCCCC2(CCCCC2)C1 N1(C(CCC)=O)CCC2(CCN(C(=O)C(Cl)COC)C2)C1 c1(C(=O)NCC(C)N(C(C2(OC(C)C)CCC2)=O)C)cc2c(s1)CCOC2 C(=O)(C(C)C(O)C(C)CC)N1C2C(C(=O)NC(CC)C(=O)N(C)C)(CCC2)CC1 C(=O)(C1(C)CCn2c(C)nnc21)N1CC(NC(C(CCC)=CCC)=O)C(C)(C)C1 N1(C(c2c(C)nn(C)c2)C(=O)NCCCC2CC2)CC(C#N)C2(CCC2)C1 c1(CC)nn(C)c(C(N2CCC(NC(c3cccc(C)c3C)=O)C(F)C2)=O)c1Cl C1(C(=O)NCC(CC)NC(c2c(C(F)F)cccc2F)=O)CN2CCC1(C)CC2 C=C1CCC(C(N2CCC(C(=O)Nc3nc(N(C)C)n[nH]3)(OC)C2)=O)CC1 C1(N(C(C(CC)c2cccnc2)=O)CC)CCN(C(=O)CC2NC(=O)NC2=O)CC1 c1(C(N(CCCC)CCO)=O)csc2c1CCN(Cc1cc(O)ccc1O)C2 CCCCC(CCCC)C(=O)N1CCC2CN(C(=O)CSc3nnnn3C)C2C1 C(=O)(CS(=O)(=O)c1ccc(Cl)cc1)N1C2CCC(CNC(CSC)=O)(C2)C1 C1(CNC(C(c2cccc(C)c2)C)=O)CN(C(c2cc(C)nn2C)=O)CCC1C N1(C(CC)=O)CCC(CC2CC=CC(n3cc(-c4scnc4C)nn3)C2)C(C)C1 C1(C(=O)NCC=C)CCN(Cc2ccc(OC)c(Br)n2)CC1O N1(CC)CCCN(C(C2C3CCCCCC23)C(=O)NCC(F)F)CC1 c1(C(=O)NC2CCCN(C(c3n(C)ccc(=O)c3)=O)CC2)c(O)ccc(F)c1F CCC(C)C(O)C(=O)N1CCCC(NC(c2ccc(-c3cnc[nH]3)cc2)=O)CC1 N1(C(COCCC)=O)C2CCC1CC(N(C)C(C1CCN(C(C)=O)C1)=O)C2 N1(C(c2ccc3snnc3c2)=O)CCC2C(CCCN2C(c2n[nH]cc2F)=O)C1 CC1(C)COC(C(=O)NCCNC(=O)Cc2coc(-c3ccccc3)n2)C1 Cn1ncc(C(=O)NCC2(C)CCCN2C(C2CCOC2(C)C)=O)c1Cl N1(C(CCOC)=O)CCC(NC(=O)CCc2ccccc2)C1C(C)C.C(C)C.O C1(N(C(C2C(=C)CC2)=O)CC)CCN(C(c2cnc(C)n2C)=O)CC1 O=C1CCC(C(=O)NCC=CCNC(c2ccncc2Cl)=O)c2ccccc21 c1(CC(N2C(CNC(CCc3ncc(C)[nH]3)=O)CCC2)=O)cccc(C#N)c1 N1(C(c2sc(Br)nc2Cl)C(=O)NCCCSC)CC(c2ccccc2)CCC1C C(=O)(C(O)CC(F)F)NC1CCC(NC(c2ccnc(N3CCCC3)c2)=O)CC1 C1(C(=O)NC2(CC=C)CCC2)C=CCN(C(c2ccc[nH]2)=O)C1 O=C1NC(=O)C2(CCCC(C(=O)NCCc3nc(Br)n[nH]3)C2)N1 C=Cc1cncc(C(N2CCC(CNC(c3nc(C)nn3C)=O)(OC)C2)=O)c1 c1(CC)cccc(C(=O)N(CCC(C)(C)NC(=O)Cc2cccc(C)c2)C)n1 N1(C(c2c[nH]ccc2=O)=O)CCC2(CCCN2C(C2CC3CCC2CC3)=O)C1 C(=O)(CCCCC1CC1)NCC(C)(C1CC1)NC(C(C)Cn1ccnc1)=O CC1C(C(=O)NC2CCN(C(C3(CO)CC(C)(C)C3)=O)C2)=Cc2ccccc21 C(C(=O)NC(C(=O)OC)C1CC1)(c1cn[nH]c1)N(CCSCC)CC C1(C(=O)NC(C)CCCNC(C2(O)CC(CF)C2)=O)(CF)CCOCC1 c1(C(N2C(CC(=O)N(C3CCCC3C#N)C)CCC2)=O)cccc(CO)c1 c1(NCCCNC(C23C(C)(C)OCC2C3)=O)cccc(F)c1C#N C(=O)(C(C)CSC(F)(F)F)N(C1CCN(C(c2ccc(CO)s2)=O)C1)CC O=C1COc2ccc(CNc3ccccc3NS(=O)(=O)c3c[nH]nc3Cl)cc2N1 n1(CCCC)cc(-c2nnc(CSc3ccccc3)o2)nn1 N1(C(COC)=O)CCC2(C1)CN(C(=O)Cc1ccc(-n3cnnc3)cc1)CCO2 C(=O)(C(O)C1=CCCCC1)N.C(C(C)(O)C1CC1)N(C(=O)CCOCCC)C Cc1ccc(C=CC(=O)NCCC)cc1.C1CCCN1C(=O)CC1CN(C)C1 C1(NC(C2CCCS2)=O)CC2(C1)CC(NC(C13CCC(F)(CC1)C3)=O)C2 CC(C)CC(CNC(=O)C1=COCC1)C(=O)N(C)Cc1nncs1 c1(NC(CC2CN(C(C(COC)(C)C)=O)CC2C)=O)cnc2c(c1)CCC2 Cc1ccccc1-c1nsc(N(C2CCN(C(=O)CC(C)(O)C3CC3)CC2)C)n1 C1(NC(CC2CC(C(N3CC(F)(F)C3C3CC3)C)C2)=O)CC2CCCC2C1 CCCCC(C(=O)NCC(CC(C)C)NC(c1cc(C(F)(F)F)n[nH]1)=O)C(C)C N1(C(C2CC(F)(F)C2)=O)CCCC(C)C1.C1(CC=O)C(C)C1(F)F.CO.C c1(C(=O)NCC(CNC(=O)C(C)N(C)C)OC)ccc(-c2ccccn2)o1 C1(C)(C(N(C)Cc2ccncn2)=O)CCN(C(C2C3CCC(=O)C23)=O)CC1 C1(CC(=O)NCC(CN(C)C)O)CC(C)(C)CN1C(c1c[nH]ccc1=O)=O N1(C(=O)Cc2cc[nH]c2)CC2CN(C(c3cccn4cnnc34)=O)CC2C1 Cc1ccc(C(N2CCC(NC(=O)Cc3cn(C)nn3)C(C(C)C)C2)=O)c(Cl)c1 N1(C(CC2(OC)CN(C(=O)CCC)C2)=O)CCC(O)C(F)(F)C1.C=O.C(C)C c1(C(N2C3CC(C(=O)Nc4nc[nH]n4)CC2CC3)=O)c(O)ccc2nc[nH]c12 C(CNC(=O)C=CC1CCC1)(C(=O)NCC(c1nncn1C)C)OC c1(C(=O)NCCCC2(CNC(C(CC)(F)F)=O)CCCC2)ccc2c(c1)CC2 CC1(C)Cc2[nH]nc(C(=O)NCCC)c2C1.c1(C(=O)N)ccc(C(F)(F)F)nn1 C12(C(N3CCCC3)=O)CC1CNC2=O.Cn1ccc(C2CC2NC(=O)CO)n1 C1(O)(CN(C)C(c2ccc(O)nn2)=O)CCN(C(=O)C(O)CC2CCCC2)C1 N1(C(c2ccc(CC)s2)=O)CCCCC1CNC(c1conc1C1CCCO1)=O c1(OC)cc(C)c(C(=O)OCCS)cc1S(N)(=O)=O.CC1OCCc2sccc21 N1(C(c2c(NC)ccc(F)c2)=O)CC2CN(C(=O)Cc3cnn(C)c3)CC2(C)C1 c1(C(=O)N)ccn2cccc2c1.C1(CNC(CC2(C=C)CC2)=O)CCC(C)CC1 N1(C(c2n(CCC)ncc2)=O)CCC2C(NC(=O)Cc3ccccc3Br)C12 Cn1nnc(CNC(C2(C)CCCS2)=O)c1C(=O)N.C1CCN(C(N)=O)C1 N1(C(CSCCC(C)C)=O)CC2CC1(C(=O)N(CC(O)C1CCC1)C)C2 C1(CSCC(=O)OCCCCC)COCC1OC N1(C(C2C(C)SCCC2)=O)CC(O)CCC1C(=O)N(C)CCc1ccccn1 C1(NC(C2N(CC)CCCC2)=O)CC(F)CN(C(c2cncc(OC)n2)=O)C1 c1(C(c2n(CC)nnn2)NCC(c2cccc(C)c2)(C)C)cc(F)ccc1SC c1(C(C(=O)NCC(C2CC2)NC(Cc2cc(C)no2)=O)C)c(C)noc1C C(N=c1[nH]c(=N)[nH]c(=NCC2(Br)CC2(F)F)[nH]1)c1nccc(C)c1F c1(C(=O)Nc2nc(C)oc2)ccc(F)c(C)c1.N1(C=O)CCCC1.C(C)=O.N c1(C(=O)NCC2C3CC2N(C(=O)C2=NOCC2)C3)onc2ccccc12 C1(C(N(CC(F)F)CCN)=O)CCCCC12OCCO2 C(CC(C(=O)NCc1ccc(O)nc1)NC(=O)Cn1ccc(C)c1)SC Cc1ccc(C(=O)NC2CC2C(N2CCC3(CC2)CN(C)C3)=O)c([N+](=O)[O-])c1 c1(CC)[nH]ccc1C(=O)NC(CC1CCCC1)C(=O)N.C(CC1CCC1)CO CC1(C)CC(NC(c2ccc(CO)cc2)=O)CCN(C(C2CSC2)=O)C1 c1(C(=O)NCC2N(C(C3(C)C=CCC3)=O)CCC2)ccc([N+](=O)[O-])[nH]1 CC(CF)CC(=O)NC(C)(C)CN1CCN(C(=O)CCC2CCCC(=O)N2)CC1 N1(C(c2c(CC)c(C)sc2)=O)CCN(C(C2CC3C=CC2C3)=O)CC1C CCCCCC(C)(C)C(=O)N1CCC(CC(N2CC(N(C)OC)C2)=O)C1 C1(NC(c2cnn3c2CCC3)=O)CC2CC1CN2C(c1cncnc1)=O N1(C(C2CCC(CC)CC2)=O)CCCC2C1CCN2C(=O)Cc1cc[nH]n1 C(=O)(CC(C(C)C)NC(C1CCCC1)=O)NC(CCCC)CC C1(NC(C2(OC)CCC2)=O)COC2(CCCN(C(=O)CN3CCCOC3=O)C2)C1 c1(C(=O)NC(CC(=C)Cl)C(=O)N(C)Cc2csc(C)n2)nccc2[nH]ccc12 Cc1c(C(=O)NCC(C)NC(C2(C)CC2(F)F)=O)cccc1C(F)(F)F CC1(C)CC(=O)N(CC(=O)NC2C=CCN(C(=O)CCNC(=O)CO)C2)O1 c1(C(N2CC(C(C)NC(C(OC)OC)=O)OCC2)=O)c(F)cc(Cl)cc1F C1(C(N2CCCC(F)(CNC(c3occ(C)c3)=O)C2)=O)Cc2cncn2C(=O)N1 C1(NC(CCCNC(C)=O)=O)CC(NC(c2n[nH]cc2C)=O)C(O)C1 n1(CC)cc(CC(=O)NCC(C(C)C)NC(=O)C(C)c2ccco2)cn1 C(C)(C(=O)NCC(C1CC1)NC(=O)C(F)F)N(C(C)=O)C O=C(N=c1[nH][nH]cc1Br)C1CCN(C(C2C3COCC23)=O)CC1 CC1C(NC(=O)Cc2ccnn2C)CCCN1C(c1ncncc1Cl)=O C1(CC#C)(NC(C2C=CCC2)=O)CC=CCC1.C(=O)C=CC(=O)N(C)C c1(C(N2CCC(N(C(C)=O)Cc3coc(C(C)(C)C)n3)C2)=O)ccccc1.C c1(C(=O)NCCN(C(CC2CC(C)C2)=O)CC)ccc(CN2CCCC2)o1 N1(Cc2cnc(C(C)C)s2)CCC2(CC1)CC2NC(=O)CC1CC2C=CC1C2 C(=O)(C(CNC(c1ccoc1C)=O)CC(C)C)Nc1c(C)cc(Cl)nc1 c1(OC)c(C(=O)N(C)CC2CCCN2C(=O)CCOC2COC2)cnn1C CC(C)CCC(=O)C(=O)N(C)CC1CCCN1C(c1ccc(N(C)C)cn1)=O C(=O)(C(C)(CC)C(=O)NCCNC(=O)CC(c1ccccc1)C)OCC.O c1(C(=O)NC2CCN(C(C(c3ccc(Cl)s3)C)=O)C23CC3)ncn2ccccc12 c1(CC)c(C(c2nnnn2C(C)(C)C)NC2CC3(CC3)C2)cnn1C C12(NC(c3nc(Br)c[nH]3)=O)CCCC1N(C(c1cc(C3CC3)[nH]n1)=O)CC2 C12(n3cc(CONC(C4(C)CC4(Cl)Cl)=O)nn3)CCC(OC(F)F)(CC1)C2 C1(NC(c2nnn(CC)c2C)=O)CCC12CN(C(c1cc(Cl)ccc1Cl)=O)C2 N1(C(c2cc(C)c(C)s2)=O)CCC(C2CCCN(C(c3ncc(F)cn3)=O)C2)C1 N1(c2nccc(OC)n2)CCC2CN(C(=O)C(C)S)CC12 CC(CCS(C)(=O)=O)NC(=O)N.C1(C)CCN(C=O)C1(C)C.C(C)(C)C N1(C2CCC(NC(CC=CC=C)=O)C2)CCN(C(=O)CN2CCNC(=O)C2)CC1 C(C(C)(C)CC(F)F)NC(CC1C=CC(NC(CCOCC#C)=O)C1)=O c1(C2(C(=O)NC3CC(NC(CC4N(C(C)C)CCC4)=O)C3)CC2)ccccc1Cl Clc1ccc(-n2cc(CNC(c3ccccc3)C3CCCO3)nn2)c(Br)c1 C=C(Br)CCC(=O)NCC1(O)CC(NC(=O)CC2CC(OC)C2)C1 C1(CNC(c2ccn(C(C)(C)C)n2)=O)CCCC(NC(C2CSC2)=O)C1 Cc1ncsc1C=CC(N1CC2C(C)C2C1)=O.C(=O)CC(F)(F)F.C(=O)C.N C(=O)(C(CNC(C1CCN1C)=O)C(C)C)Nc1cn(CC(C)C)nc1 c1(C(N2CCC(NC(c3cn(CC)nc3)=O)(CF)C2)=O)ccn2ccnc2n1 c1(C(=O)NC2C(NC(=O)CCC3CCCCO3)C2)c[nH]c2ccncc2c1=O C(=O)(CCCCCO)N1C(CNC(c2cnc(C(C)C)s2)=O)CC(F)C1 C1(NC(c2c(CC)[nH]nc2Cl)=O)CC2CC1N(C(C1(CC)CC1)=O)C2 CCC(CC)C(C(=O)NC(C)(C)CNC(C1(C)CC1(Cl)Cl)=O)N1CCOCC1 Cc1cc(=NCC2(CNC(=O)CN3CC4CC4C3)CC2)[nH]c(C(C)(C)C)n1 c1(C(N2CCC(N(C(c3c(OC)nsc3)=O)C)C2)=O)cccc(Cl)c1OC CC1(C)C(NC(c2ccn3cncc3c2)=O)CC1N=c1[nH]nc(O)s1 C1(C(=O)NCCCC=CC)CCN(C(=O)CCC2CCCOC2)CC1 c1(CC)nn(C)c(C(=O)NC2C=CC(CNC(=O)CCC(N)=O)C2)c1Cl N#Cc1ncc(C(N2CC(CNC(=O)CNC(c3ccsc3)=O)C2)=O)s1 N1(C(Cc2c(C)nc[nH]2)=O)CCCC(N(C(C2CCN(C3COC3)C2)=O)CC)C1 C1(C(N2CCCCC2C)=O)Cc2nccn2C1.n1(C2(C(=O)N)CC2)cc(Cl)cn1 N1(C(C(CC)(O)c2ccccc2)=O)CCC(CNC(=O)CSC2CC2)C(C)C1 C1(NC(c2nn(CC)nc2C)=O)COC2(CCN(C(c3cnsc3)=O)C2)C1 C1(C(N2C(CC)CCOCC2)=O)CN(C(=O)C=CC2CCCCC2)CC(C)(C)C1 C(C(O)CO)NC(N(CC(C1CC1)SC)C)=O C(=O)(C(CCc1ccccn1)N1CCCC1c1ccccc1Cl)NCCOC c1(OC)ccc(F)c(CC(=O)NCCOc2cnn(C3CC3)c2)c1 C1(C(=O)NC2(CC=C)CCN(c3nnc(C(F)F)s3)C2)CCc2ccccc2O1 CC1=CC(NC(c2cccnc2-n2cncn2)c2nnnn2C2(C)CC2)CCC1 c1(C(N2CC(C(C)NC(C3CC(C(C)C)OCC3)=O)C2)=O)onc2ccccc12 C(CC(C)N=c1nc(N(C)Cc2ccns2)c2c([nH]1)CCCC2)OC C1(C(=O)NCC2(C)N(C(C(C)OCC3CC3)=O)CCC2)CC(C)(C)CN1C N1(C(c2ccc(CCC)[nH]2)=O)CCCC(C(F)F)C1 CCC(CC)C(C(=O)N1CC(NC(=O)CN(S(C)(=O)=O)C)CC1(C)C)OC C1(NC(CC(CC)C)=O)CC2CC1CN2C(=O)C(C)ONC(=O)OC(C)(C)C C1(CC(=O)NC(CNC(CCOCC)=O)C2CC2)COCC2(CCC2)O1 Cc1[nH]nc(C(=O)NCC2(C(C)(C)C)CCN(C(=O)CCC(F)F)C2)c1N CC1CCC(C)(C(=O)N)C1(C)C.c1(C(N2CC(C(N)=O)C2)=O)cccc[n+]1[O-].C c1(CC(=O)NCCNC(C2CC(SC)C2)=O)c[nH]c2ncccc12.C1CC1 C1(NCC2(C)CCC(C)C2)CC2CC1CN2C(=O)OC(C)(C)C C(C(C)C(=O)NC1CCC(CCC(=O)NCC2(OCC)CC2)C1)OC c1(NCC=CC(=O)NC)ncnc2scc(-c3ccc(C)cc3)c12 N1(C(CC)=O)CCCC(C(N2CCC(CN(C)CC=C(C)CC)C2)=O)C1 c1(C(=O)OC)cn(C)nc1C(=O)NC1CC(C)C1.C1(CC=O)CCCO1 C12(C(=O)NCCC(CCNC(CCc3c(C)nn(C)c3)=O)C)CCCC1OCC2 C12(C(=O)NCCC(C)N(C)C)CCC(CC1)N(C(c1cccc3ccoc13)=O)C2 N1(C(c2ccnc(C)n2)=O)CCCC2(NC(C3CS(=O)(=O)C3)=O)CC2C1 CC(=Cn1ccnn1)C(=O)N1CCC(C(C)NC(c2sccc2CN(C)C)=O)C1 Cc1[nH]c(C#N)cc1C(N1CCN(C)C(C(=O)NC2CCC(=O)N(C)C2)C1)=O O=C(CCCCN1CCCC1)NCC1CCC1NC(C1C2COCC12)=O C(=O)(N=c1[nH]onc1C)C1(C)CCN(Cc2ccc(C)nc2Cl)C1 N1(C(c2nc(C)sc2)=O)CCc2sc(CNC(c3scc(C)c3C)=O)nc2C1 n1(CC(C)OCC(=O)NCC(=C)C)cc(C)cn1 C(=O)(C#CC1CCCO1)N.c1(N(C(C)=O)C)ccc(C(=O)NC(C)(C)CC)cc1 CC1CC(NC(C2CCN(C)S2(=O)=O)=O)CN(C(=O)COC2CCOC2)C1 CN1CCCCC(C(N2CCCC2CNC(=O)CCCN=[N+]=[N-])=O)C1=O CCCC(CCCNC(c1nc(C)nn1C)=O)NC(C1CC12CC(C)(C)C2)=O n1(CCC(C)C)nc(CNC2CN(C(C)C)C2)c2ccccc12 C(=O)(C(C)CC(F)(F)F)NCC(CC=C)NC(=O)C=Cc1cnc(C)s1 C1(NC(C(Cc2c(C)cccc2)C)=O)COCCN(c2nccc(CO)n2)C1 Cc1cccc(C(N2CCN(C)CC2C(=O)NC2CCCSC2)=O)c1N CC1(CNC(=O)Cc2sccc2Br)CCN(C(C2CC(O)C2)=O)CC1 CC(CS(=O)(=O)c1cccnc1Cl)NC(=O)C(C)(C)c1cscn1 C1(C(=O)NC2CC3CN(C(c4cc(C#N)on4)=O)C2C3)CCc2nc[nH]c2C1 CC1CCCN(C(c2c(I)ncn2C)C(=O)NCCN2CCOCC2)CC1 n1(CC)nc(C=O)cc1C1CC1.C1CCCN(C(c2cc(C(C)C)[nH]n2)=O)C1.N CC(O)C(C)(C)C(=O)NCCC1CCCN1C(C1CNC(=O)N1)=O N1(C(CCN(C)C)=O)CCN(C2COCC2NC(=O)NC=O)CC1.C(C)(C)C c1(NC(C(CCCNC(C(C)OC2CCCC2)=O)O)=O)ccc2c(c1)OCC2 N1(C(c2cc(F)cc3c2CCC3)C(=O)NC(CC)C)C2CCC1c1ccccc12 C1(NC(CCOCC(C)C)=O)C2CC1N(C(c1c[nH]c(-c3ccncc3)n1)=O)C2 N1(C(C=C(C)Cl)=O)CCCC(C2CCN(C(c3ccnn3C(C)C)=O)C2)C1 C(=O)(C(C=O)C(C)(C)C)NC(CC)CNC(C1CN(C)C1)=O.C(C)(C)C C1(NC(CCCCC=CC)=O)COC2CN(C(c3cc(C)c(F)c(C)c3)=O)CC12 C1(C(C)NC(=O)Cc2cnns2)CCCN1C(=O)C.c1(C=O)ccccc1.N N1(C(=O)C=CSc2ccccc2)CCOC2(C1)CN(C(=O)Cc1ccsn1)C2 c1(C(N2CCCC(C)C2)C(=O)NCCCOC)cccc2c1ccn2C C1(NC(C(C)c2cccs2)=O)CCC2CN(C(=O)CC34COC(C)(C3)C4)CC2C1 N1(C(c2ccc(C)cc2F)=O)CCCC(C2CCN(C(=O)C=CCF)C2)C1 C(CCCC(=O)NC(C)(C)CC1CCCC1)N(C(COCCSC)=O)C C1(CN(C(CNC(C(CC)C)=O)=O)C)CN(C(=O)CS(=O)(=O)CC)CC12CC2 CC1CC(c2ccccc2)(C(=O)NC(C)CCN(C(=O)C=C2CCC2)C)C1 N1(C(CSC)=O)CC(C)CN(C(c2nc(C(F)(F)F)cc(C)n2)=O)C(C)C1 C(=O)(C1=CCCCCC1)NCC=CCNC(Cc1cc(C)ns1)=O c1ccc(C#N)cc1.C1(NC(CSCC(C)C)=O)CCN(C(=O)CS)C1C.C S(=O)(=O)(c1cncc(CNC)c1)NC(C1CCOCC1)C(=O)OCC N1(C(C2(COC)CCCCO2)=O)CC2C(C1)C2N=c1ccnc(C2CC2)[nH]1 C1(C(N(CCC#C)CCO)=O)CCC2(CC2)N1C(=O)C(CC)CCOC C(=O)(C1=C(SC)CCCC1)NC1CC(OC)CN(C(c2ccc(CO)cc2)=O)C1 c1(SC(C)C(N2CC(O)(C)C2)=O)ccccc1.c1(C=O)ccnn1CC(F)F.N C123CCCC1CN(C1CCCC2=CC=CC(C(=O)O)=C1O)C3 N1(C(C(C)NC(CC)=O)=O)CC2(C)CN(C(=O)Cc3ncc(C)o3)CC2(C)C1 C1(CC(=O)N(C)CC2CCN(C(C3CCCC3N)=O)CC2)CCOC(C)(C)C1 c1(C(N2C(C)CC(NC(=O)Cn3ncn(C)c3=O)C2)=O)cc2ccncc2s1 Cc1nc(C(=O)NC(C2(O)CN(C(=O)CNc3ccccn3)C2)C)c(C)s1 C1(NC(C(F)=C(C)C)=O)CN(C(=O)CCC(C)N(C)C)C2(CCOCC2)C1 CC(C)(C)C(O)C(=O)NC1(CC(=O)NC2CCSCC2)CCC1 C1(CNC(C=COCC)=O)CC2CCC1N2C(c1cc(O)ncn1)=O N1(C(C(CCOC)C)=O)CC2(CC2)CC1CNC(=O)Cc1cnns1 c1(C(NNC(c2ccc(NC(=O)OC)cc2Br)=O)=O)csc2ccccc12 C1(N(C(C(C)CC2CCCC2)=O)C)CCCN(C(=O)C(C)(C)c2cnco2)C1 N1(C(C2CC(=O)N(C3CCCCC3)C2)=O)CC(F)(F)C2(CCOCC2)C1 c1(CNC(CC2ON=C(CC)C2)=O)nc(C)cc(O)n1.C1(C(=O)N)CCCCS1 C1(NC(c2cnn(C3CC3(F)F)c2)=O)CN(C(c2ccccc2O)=O)CCC1F N1(C(c2scc(C3(C)CC3)n2)C(=O)NCC2CC2)CCCC2(CC2)C1 C1(CNC(C(C=C)(C)O)=O)CC(F)(F)CN1C(c1oc(SC)cc1C)=O N1(C(C2C(C)(C)C2(C)C)=O)CC2(NC(C3(N4CCOCC4)CC3)=O)CCC1C2 C(c1ccc2c(c1)COCC2)=CC(N1CCC1)=O.c1(CC(=O)NC)csnn1.C c1(COC)ncc(C(=O)NC2CC2)c(=N)[nH]1.C1(Br)(C=O)C(C)C1C.C C(C)(CC(=O)N1CC(NC(c2cn(C3CCN(C)C3)nn2)=O)C1)OC CN1CCOc2ccc(C(N3CCC(NC(c4cn(C)cn4)=O)C(F)C3)=O)cc21 Cc1[nH]nc(C(=O)NCCOCCCNC(C2(C(F)F)CCCO2)=O)c1C N1(C(CCCn2c(C)ncc2)=O)CCCCC1CNC(=O)C1=COCC1 C1CCS(=O)(=O)C12CN(C(C1CC3(CCOC3)C1)=O)C2.C(CC=O)SCCC.N N1(C(c2cc(C)no2)=O)CC(CNC(=O)CO)CC12CCC2.C1CCOCC1.C c1(-c2nc(C)on2)cccc(C(=O)NC2CN(C(=O)C(F)=C3CCC3)C2)c1 C(=O)(C#CC1CCOCC1)NCC(C1CCCC1)NC(C1(Br)C(C)(C)C1)=O N1(C(C2(CCC)CCC2)=O)CCC(C(C)NC(=O)CNC(=O)CC)CC1 N1(CCCn2cc(C3CCCS(=O)(=O)C3)nn2)CCC(C(F)(F)F)C(F)(F)C1 N1(C(C(C)n2ccnc2)=O)CCN(C(=O)CCCN=[N+]=[N-])CC1CF C1(C(=O)NCCC(C)(C)NC(c2cnc3[nH]ccc3n2)=O)CC2CSCC(C1)C2 c1(C(C)C)ncc(Br)c(=NC2CC3CC(C2)N(C(=O)C(F)C(F)(F)F)C3)[nH]1 CCC(C)(C)C(=O)C(=O)NC.C12(CCCCO1)C(=O)N1CC(n3cc(nn3)C2)C1 C1CN(C(C2CCCC2)=O)CC2(CCC2)O1.NC(=O)CCNC(=O)C(=O)N.C C#CC1CCCN(C(C2CCCN(C(c3c(F)cccc3F)=O)CC2)=O)CC1 C1(NC(c2c(F)ccc(C)c2)=O)CC2CN(C(C3CN4CCN3CC4)=O)CC2C1 c1(C(N2C(CCNC(C(C)=C3CCC3)=O)CCC2)=O)cccc(O)c1F N1(C(COCC(C)C)=O)CCN(C(=O)C(N2CCCC2)C2CC2)CC1C(C)C C1(C(=O)Nc2c(CN)ccs2)CCS(=O)(=O)C12CN(Cc1ccccc1)C2 C1(CNC(C(CC)CC)=O)CCC2(CN(C(C3(C)COC(=O)N3)=O)C2)O1 n1(CC)cnc2c(NCCN3CC=CC3)[nH]c(=NC(C)c3ccc(C)cn3)nc12 N1(C(CC=CCC)=O)CC(C)CCC1CNC(=O)CCCC(N)=O c1(C(=O)NCC2OCC(CNC(C(C)C)=O)C2)coc2ccc(O)cc12 c1(CNC(CCOCC(C)(C)C)=O)cscn1.C1(C)(CC=O)CCOC1.C N1(C(c2sc(C)c(O)n2)=O)CCCC(C)C1CNC(c1cc(O)n(C)n1)=O C1(NC(C(CCC(C)C)O)=O)CN(C(C2CN(C(C)C)C2)=O)CC2(CCC2)C1 C(CC(C(=O)NCC(O)C(N)=O)NC(c1nc(C)oc1C)=O)OCC Cc1ccc(CC(=O)NCC(C2CCC2)NC(C2(n3nccn3)CC2)=O)cc1 N1(CCOC)CCC(C)C1.c1(C=O)cnn(CCN(C)C)c1.C(=O)(CC)N c1(C(=O)NC2C3(CN(C(C(CCC#C)O)=O)C3)CC2)ccc(S(N)(=O)=O)s1 c1(C(=O)NCC(CC(C)C)NC(C(CCC)O)=O)ccc(C(F)(F)F)c(N)c1 c1(NC(=O)NC(C2CC3CCC2C3)C)cccc(OCCSC(F)(F)F)c1 N1(C(C2C(CC)CCN2C(C2CCCC(=O)C2)=O)=O)CC2(CCC(=O)O2)C1 Cc1[nH]nc2c1CC(C(N1CCN(C(C3(S(C)(=O)=O)CC3)=O)CC1C)=O)CC2 C1(c2ccccc2)(C(=O)NC2C(NC(C(CSC)O)=O)CC2)CC(F)(F)C1 c1(C(=O)NCC(CO)NC(C(F)=CC)=O)ccc(C)cc1.C(C(F)F)O c1(C=O)cccc2c1OC(C)C2.c1(SC)nocc1C(=O)NC1CC(F)(C)C1 N1(CC(=O)N(CCC)C(c2ncc(Cl)cc2C)=O)CCC2(COC(=O)N2C)C1 Cc1csc2nc(CC(=O)NNC(=O)CNc3ccc([N+](=O)[O-])cc3)cn12 C1(c2nnnn2C2CC2)(NC(C)Cn2ccccc2=O)CN(C2CC2)CC1C N1(C(c2c(SC)csc2)=O)CCN(C(C2CN(C(C)C)C2)=O)C2CCCC12 C(CC(C)C)(C(=O)NC(c1ncccc1C)C)NC(CCCOCC)=O C1(NC(c2c(C)nc(O)cc2)=O)COC2(CCN(C(=O)CCSC(F)(F)F)C2)C1 CC1CCN(C(=O)NCC2(n3cncn3)CCC2)C(C(=O)OC(C)(C)C)C1 N1(C(CCSC)=O)CCC(C(=O)Nc2c(C)noc2C)C(C)(C)C1 c1(OC)ccc(C(O)C(=O)N(C2CN(C(=O)CCC3CC3(F)F)C2)C)cc1 Cc1nc[nH]c1CC(O)C(=O)NCCC1CCN(C(=O)Cn2ccnc2C)C1 c1(C(=O)NCC2CN(C(=O)CC3COCCO3)C2)ccc(Br)c(Cl)c1F c1(C(N2CC(CNC(c3ccc(O)nc3)=O)C2)=O)cccc(C(N)=O)c1F c1(CC(=O)OC)cc(=NCC(c2ccsc2)N(C)C)[nH]cn1 N1(C(c2cc(COC)[nH]n2)=O)CCCN(C(c2ccc(O)nn2)=O)CC1C C(=O)(C(O)CC(C)(C)C)NCCCC1(NC(C(C2CCCC2)OC)=O)CC1 Cc1nc2cc(C(=O)NC3(c4ncc(C(=O)O)cn4)CCC3)ccc2n1C c1(C(=O)NC2C3CN(C(C(CN(C)C)(C)C)=O)C(C3)C2)cc2ccc(Cl)cc2s1 C1(NC(c2ccc(C(=O)OC)s2)=O)CCC(NC(=O)CC)CC1.CC(N)=O n1(C(C)C)ncc(C(N2CC(CNC(c3nocc3Cl)=O)C2)=O)c1F C1(C)(C(=O)NCCC(C(C)C)NC(C(C(C)C)C2CCC2)=O)CCCCCCC1 C12(C(=O)NC3C(C)CN(C(=O)CCCCCO)C3)CC=CCN1CCC2 C1CN(C(=O)C(C)(C)CF)CC(C)(C)C1.c1(OC)ccc(C(F)(F)C(=O)N)cn1 n1(CCN(C)C)cc(C2CCCN2C(c2sccc2Br)=O)nn1 C(=O)(CS(=O)(=O)CC(C)C)NC(CNC(CC(CC)C1CCC1)=O)(C)CO O=C1CC(NC(C2(Sc3ccccc3)CCC2)=O)C2(CCN(C3CC3)CC2)N1 C1(CC(=O)NCC2N(C(C(C)C3CC3)=O)CCC2)CC2(CCO1)CC2 c1(COCC=C)nc(-c2ccc(C)cc2)nn1C1CCCCC1O c1(C(=O)NC2CN(C(C3(C(F)F)CCCO3)=O)CC2CO)ccn2ncnc2c1 C1(C(=O)NC2C(CNC(=O)CSc3cn[nH]c3)C2)CCOCC12CCCC2 C1(NC(C=CCCC)=O)CC(OC)CN(C(=O)Cc2ccc(COC)[nH]2)C1 C1(C(=O)NCCC)(NC(=O)CCc2cnco2)CCCC1.C1(C=O)CCCC1 N1(C(CCCOC)=O)CC(C(=O)NC2CC(C)C2)C(C)(C)C1 C12(CNC(C(C(C)C)O)=O)CC(CO1)N(C(c1cc(N)ccc1Cl)=O)C2 C1(NC(C2(C#C)CCC2)=O)CN(C(C2CCC(OC(F)F)CC2)=O)CC1C c1(-c2cnc(CC(=O)NC(c3ccsc3)C)nc2)cccc2c1CNCC2 c1(C(=O)NCC(CN(C(C(CC#C)C2CC2)=O)C)(C)C)nc(OC)cc(O)n1 c1(OC(C(=O)NCc2cccc(SCCCC)c2)C)ccc(Cl)cc1C CN1CCC(C(F)(F)F)(C(=O)NCCCC2CN(C(C3CCSC3)=O)CCO2)C1 c1(C(=O)NCCCN(C)C(c2c[nH]c(=N)s2)=O)cc(F)c2cn[nH]c2c1 C1CC2CCC(C1)N2C(C1CCC(F)(F)C1)=O.c1(SC)cc(C(=O)N)c(C)o1 C1(CC=C)(NC(C2CCC(=O)N2)=O)CCN(C(=O)CNC(=O)NC)C1 C(N=c1[nH]c(=NCCCC#N)c2ncccc2[nH]1)C1CC(C)(C)C1 N1(C(c2c(C)sc(O)n2)=O)CCN(C(c2cn(C)nc2Cl)=O)CC1CC1CC1 C1(C(=O)NC2(C)CN(C(c3csc(C)c3N)=O)C2)Cc2ccccc2C1(C)C C(=O)CCC(F)(F)F.C1(CNC(CCNC(C2C(C)C2)=O)=O)CCCC1.C C1(CNC(C(C=CC)O)=O)CC2CC2N1C(c1ccc(OCC)cc1)=O C1(NC(C2(CO)CC2)=O)CSCCN1Cc1ccccc1Cl.N12CCCC1C2 Cc1ncc([N+](=O)[O-])cc1C(=O)NCC1CCC1.c1(C=O)cnn2c1OCC2.N c1(OC)cc(F)c(CC)c(F)c1.C1C2CC(O)C1N(C(C)=O)C2.C=O.C(C)C N1(C(CC(CC)SC)=O)CCOC2CCN(C(c3ccsc3C#N)=O)CC12 C(CC(O)CC(=O)NCC1CCN1C(c1cc(CF)on1)=O)SC C12(C(=O)NCC3(CNC(=O)Cc4ccc(Cl)s4)CCC3)CCCC1CCC2 C1(CC(N2CCOC(c3nc[nH]n3)C2)=O)CCC2(CCOCC2)CO1 C1(C(N(C2CCN(C(C3CCCOC3C)=O)C2)CC#C)=O)C2(CC2)C12CC2 c1(C(N2CC(CN(C(CSCCN(C)C)=O)C)C2)=O)ccc(F)c(O)c1F Cc1cc(=NCCCCCCN(C)C(c2ccnn2CC(F)F)=O)[nH]c(C)n1 c1(OC)ccc2c(c1)N(C(C1C3C=CC(O3)C1C(=O)O)=O)CCC2 c1(SCC(N2CC(CNC(=O)CC3CSC3)C2)=O)ccccn1 c1(N2CCC(CNC(c3c(OC)ccs3)=O)C2)cc(=O)n(C(C)C)c(O)n1 CCC(CC(=O)NCc1csc(C)c1C)N(C)C(c1c[nH]c(C)c1)=O C(=O)(C1=NOC(C)C1C)N1CCCC(C)(C(=O)NC(CC=C)(C)C)C1 CC1(CNS(=O)(=O)CC2(c3ccccc3)CC(F)(F)C2)CC=CCO1 n1(CC(=O)NCC2CC2)cc(C2CC2)c2ccccc12.C1(Br)(C=O)CC1.N c1(OC)ccccc1C(=O)NCC(=O)NC1CC1.c1(C(=O)N)ccncc1Cl N1(C(C(C=CC)O)=O)CCCC(C(=O)NCC2CCC(C)C2)C1 C1(NC(C2C(C)=CCS2)=O)C2CC1N(C(C1CC1(C)C)=O)C2 N1(C(c2nc(CC)oc2)=O)CCN(C(=O)CC2CCOC2)C(c2ccccc2)C1 N1(C(CC=CC=C)=O)CCC(NC(c2cccc3[nH]ccc23)=O)C(CO)CC1 C1CCC2CCC(C1)N2C=O.C1(C(=O)OC)CN(C(=O)C=O)C1.C(C)(C)C N1(C(C(C)C2CCC2)=O)CC(NC(c2ccc(C#N)cn2)=O)CC2(CCC2)C1 CC1CCN(C(c2ccc(=O)n(C)c2)=O)CC1N(C(=O)C(C)n1cnnn1)C C1(CC)(NC(=O)Cn2ncc(Br)c2C)CCN(C(c2cn[nH]c2)=O)CC1 c1(CC)nc(=NC2CC(CCNC(C3(C)CCC(=O)N3)=O)C2)s[nH]1 C1(C)(C(=O)NC(CNC(c2c(CCC)n[nH]c2)=O)COC)CCOC(C)C1 c1(C(C)C)nc(C(=O)NC2CC(CNC(=O)CC3(C)CCCO3)C2)cs1 CCC(C)C(O)CC(=O)NCCC1(O)CN(C(c2c(C)n[nH]c2C)=O)C1 C(C(C)(C)N=c1[nH]nc(C2CC2)o1)NC(c1nccc(SC)n1)=O N1(C(C(CC(C)C)=O)=O)CCC2(CCCCN(C(=O)COc3ccon3)C2)C1 C1CCC12CCC2.c1(C(=O)OC)cc(C=O)cs1.C(=O)CC1(N(C)C)CC1 c1(C=O)cccc2oc(O)nc12.C1(CNC(C(=O)NC2CC2)=O)COCC1.C Cc1c(C(N2CCC(NC(=O)CN3CCS(=O)CC3)C2)=O)[nH]c2c(C)cccc12 N1(C(CC2N(C)CCC2)=O)CCn2ncc(CNC(=O)CCCC(C)(C)C)c2C1 C1(O)(CN(C(CC2(OC)CCC2)=O)C)CCCN(C(c2sncc2C)=O)C1 C(CC(CC)C(=O)NC1C2CCN(C(=O)C(N3CCCC3)C3CC3)CC12)=CC C1CC2CCC(C1)O2.C1(c2cn(C(C)(C)CC(=O)O)nn2)CCCCC1O C1(CCNC(CNC(=O)OC)=O)CN(C(=O)CC(=O)OC)CCO1 C1(CN(C)C(C2CC2F)=O)CN(C(c2ccnn2CCF)=O)CCO1 C12(NC(CCN(C(C)=O)C)=O)CCCCC1N(C(c1cnc(O)c(F)c1)=O)CC2 c1(C(=O)NCC(CNC(c2c(Cl)cc(C)nc2)=O)CO)n[nH]c2c1CCOC2 C#CCCC(O)CCNC(C1(C(C)C)CCN(C(c2[nH]nnc2C)=O)C1)=O C#CCC(C(=O)NCC(C)=CCC)NC(=O)Cc1cnccc1C C1(CNC(C(C)C2CCOC2)=O)CC(C)(C)CN1C(c1ccc(Cl)c(Cl)c1)=O CC(C)C(C(=O)NC1CCC1NC(=O)CCC#N)n1cnnc1 C=CCC(CNC(=O)CSC)C(=O)NCC1OCCC1(C)C CCC(CN=c1[nH]c(=NCC2CC23CC3)c2cc(F)cc(F)c2[nH]1)C(C)(F)F C#CCCCC(C(=O)NC(C)CC)N(C1CC1C)C c1(C(N2CCCC(N(C(c3ccnnc3C)=O)CC)C2)=O)cnc(C)cc1Cl n1(COC)ncc(=NC(=O)NC2CCCN(c3cccnc3)C2=O)[nH]1 N1(C(CC(=O)NCC#C)=O)CCN(C(c2scc(C)c2OC)=O)CC1C(C)C c1(C(N2CC(CCNC(C=CC(C)(C)C)=O)OCCC2)=O)cnc2[nH]ccc2n1 N1(C(C2CC2)=O)CC2(C1)CN(C(C1(C3CCCO3)CCCC1)=O)CCO2.CCS c1(NCCCC(=O)OCC)[nH]c(=NCC2(COC)CCCO2)nc2c1cnn2C C=C(C)CN=C(NC1CCS(=O)(=O)C1)N1CC(O)C(C)(C)C1 C1(C(=O)NCCNC(c2c(Br)ccc(C)c2)=O)Cc2c(C)cccc2N1 c1(OCC)cc(C(=O)N)ccc1C.C1CC(C)N(C(=O)Cn2nnnc2C)C1.C C1(C(=O)NCC(C(C)C)NC(c2n(CC)ncc2)=O)CC2CCC(C1)C2F C=C(C)CCC(=O)N1CCC(C(C)(C)NC(C2(CN(C)C)CC2)=O)C1 c1(N2CCC3CC(C(=O)NC)C3C2)nc(=NCC2CCC2(F)F)[nH]c2c1CCC2 C1(CCOC)(NC(=O)N(C2CCCC(O)C2)C)CCNCC1 C(CCCCC(=O)NC1CC(C)(NC(c2ccc(C(C)C)cc2)=O)C1)=CC.O C1(C(=O)NCCN(C(=O)C(O)CC[S+](C)C)C)CCC(S(C)(=O)=O)CC1 Cc1cc(C(N2CC(O)(CCNC(=O)C(C)Sc3ccccn3)C2)=O)on1 N1(C(C=C(C)C(C)(C)C)=O)CCCN(C(C2CC2c2cncn2C)=O)CC1CO C(C(C(=O)NCc1cnn(CC(F)(F)F)c1)c1ccccc1)OCC=C Cc1cc[nH]c1C=O.N1(CC)CCC(C(=O)NOCCCN(C)C)C1 Cc1cc(NC(C2(C)CC(C)(C)C2)=O)cc(F)c1.C(=O)(C#CC(C)(C)C)N c1(NC(C2CN(C(c3sc(Br)cc3Br)=O)CCN2)=O)cc(Cl)nc(Cl)c1 C(=O)(CC(C)C(=O)OC)NCCN(C(=O)C=CC1CCOC1)CC C1(CC(=O)NC(C2CCCN2C(c2ccnnc2)=O)C)CC2CCC1CC2 C1(C(C)NC(c2c(C)[nH]cc2)=O)CN(C(=O)Cn2cncn2)CCO1 c1(CCCC(N2CC3C(CNC)C3C2)=O)ccc2c(n1)NCCC2 Cc1ccc([N+](=O)[O-])c(C(=O)NC2CCOCC2)c1.C1(C(=O)N)CC1C(F)F C1(NC(c2cc3ncccc3s2)=O)CN(C(=O)CC2(CO)CC2)CC12CCC2 N#Cc1ccccc1CNC(C1CC(NC(=O)CCc2cccs2)CCO1)=O N(C1CCCc2cccnc21)(CCC)C(C1COCC(C)(C)C1)=O c1(C(C)=O)cc2c(cc1NC(NC1CCc3cccnc31)=O)OCO2 N1(C(C2(NC(C(n3ncc(C)c3)C)=O)CC(F)C2)=O)CCC2(CCCC2)C1 Cc1nc([N+](=O)[O-])cn1CCC(=O)NC(C)CN(C(=O)Cc1cnccc1Cl)C c1ccccc1.CCS(=O)(=O)NC.C1(NC(=O)OC(C)(C)C)(C)CCC1.N C=CCC(C(=O)N(CCC(=O)N1CC(C(C)O)C1)CCO)OC c1(CC(=O)NCCCN(C(C(CC)(C)O)=O)C2CC2)cc(Cl)ccc1Cl C1(N(C)C)CCCN(CC(=O)Nc2cccc(Cl)c2-n2cccn2)CC1 c1(CC(=O)OCC)cc(=NCCC(C)NC(C2CCOC(CC)C2)=O)[nH]c(C)n1 CC(C)CCC(C)CNCC1CCC(=O)N1C N1(C(CC2N(C(CC(=O)OCC)=O)CCC2)=O)CC2C3C=CC(CC3)C2C1 C1(NC(=O)CCF)CC2CCC1N(C(=O)CCCc1ccccc1Cl)C2 C=CCC(C(=O)N1CCC1CNC(c1c(OC)cccc1F)=O)C(C)C N1(C(c2cc(C)oc2)=O)CC(C)OC2(CCN(C(C3CC(C(C)C)C3)=O)CC2)C1 C1(C)(COC(C(CNC(=O)OC(C)(C)C)OC)=O)CC2CCC1C2 CC(C)CCCCC(=O)NCC1(O)CCN(C(=O)CC2C=NN(C)C2=O)C1 C(=O)(C1=NOC(C)(C)C1)N1CCC(n2c(C)nnc2)CC1.c1(CCCCC)cn[nH]c1 c1(CC(=O)NCCC(=C)CNC(c2ccoc2)=O)csc2nc(C)cn12 c1(OCC)cccc(C=CC(=O)N(CCCC)C)c1.C1CCOC1.C(=O)(C)N C=CCC(C)C(=O)NC1(C(=O)N(C)Cc2nncn2CC)CCC1 C(=O)(C1=CCCN(C(c2cc(-c3cccc(F)c3)no2)=O)C1)NC(C)C Cc1cncc(C)c1C(=O)NC1CCCC1NC(c1c(C)[nH][nH]c1=N)=O O=C1CCC(C(F)C(N2CCCCC2CNC(C23CCCC2C3)=O)=O)CC1 c1(C(C(=O)N)Nc2ccc(OC(F)(F)F)cc2)ccc2nsnc2c1.C1CC1.CO C1(O)(CNC(C(=Cc2ccco2)C)=O)CCN(C(C2CCCOCC2)=O)C1 C1(OC)CN(C(c2nccc(C(F)(F)F)n2)=O)CC1NC(c1ccccc1O)=O c1(C(N2CC(N(C(c3c(C)cc(Br)c(F)c3)=O)C)C2)=O)ccc2cn(C)nc2c1 c1(C=O)cc(C(C)C)nc2onc(C)c12.C1(C(=O)N(C)CC)(CC)CCOC1.N N1(C(C2N(C(C(C(CC)C)N(C)C)=O)C(C(C)C)CC2)=O)CC2(C)CC1CCO2 CCC(C)(C(=O)NCCCN(C1CCCC1)C(=O)COC)OC c1(C(=O)NC2CCCN(C(C3CC(OC)C3)=O)C2)ccc2nc(S)oc2c1 CCCCC(C)(F)C(=O)N1CCCC(CCNC(c2ccncc2C2CC2)=O)C1 Cc1nonc1CC(=O)NC(CCCNC(C1CCC1C)=O)c1ccccc1 c1(C=O)cc(S(N)(=O)=O)n(C)c1.CC(C=O)C(F)(F)F.C(C)(C)C1CCC1 CC1CCC(=CCNC(c2cn(-c3cnnn3C)nn2)(C)C)CC1 c1(NC(C(C)O)=O)cccc(NC(c2cccc(SC(F)(F)F)c2)=O)c1 C(=O)(CCCCCBr)NC(c1ccccc1)CNC(c1c(CC)noc1C)=O C12(C(=O)NCC(C)C)CC(CO)(C1)OC21CCC1.C1(C=O)CC(C)(C)CO1 c1(OC)ccc(C(N2CCN(C(C34CCC(CC3)O4)=O)CC2CO)=O)c(OC)n1 C1(NC(CCC=C)=O)C(CNC(c2nccc(Br)c2C)=O)CCC12CCC2 C1(NC(C(CNC(CC2C(C)C(=O)CC2)=O)O)=O)CC2CCC(C1)C2O C1(C(=O)NCCCC)CN(C(c2cc(C(C)C)on2)=O)CC1C1CC1 Cc1nc2ncnn2c(C)c1C(=O)NCC1C2CN(C(c3cc[nH]n3)=O)CC12 N1(C(N2CCCC(n3nccn3)C2)=O)CCCCCC1C=Cc1ccccc1 CCC(CCC(=O)N(CCC(C)O)C)NC(=O)C(F)C(C)(C)O c1(C(=O)NCC2(C)CCN(C(C(CCC)C)=O)C2)cc(Cl)ccc1-n1cnnn1 C#Cc1cccc(C(=O)N(C2CN(C(C3C4C5CCC(C5)C34)=O)CC2O)C)c1C n1(C(CC)C(=O)N2CC(CC(C)NC(C3CS(=O)(=O)C3)=O)C2)cnc(C#N)n1 CCCC(CCC)CC(=O)NCC1CN(C)CCN1C(=O)C1=CCS(=O)(=O)C1 c1(OC)ccc(C)cc1Sc1ncccc1OCC(C)C CN1CCC(O)(CNC(=O)C(CC2CCCC2)NC(c2cocn2)=O)C1 N1(C(CC2CCCN(C(CCCC(=O)OCC)=O)C2)=O)CCC2=C(CCCC2)C1 C(=O)(C1CCCc2nccn21)NCCCC(C)NC(c1cnccn1)=O C1(C(=O)NCC2(O)CN(C(CSCC#C)=O)C2)CCN(C(=O)O)CC1 N1(C(C(C)SC)=O)CC=CC(C(=O)NCc2cnc[nH]2)C1 CCCCCCCCCC(C)CC(=O)NCC1CC1NC(=O)C(C)CC CC1=NOC(C(=O)NCCCNC(c2cc(C(N)=O)no2)=O)C1 c1(C(=O)NC2C3C(C)N(C(C4CCCCC4(C)C)=O)C2C3)ccc([N+](=O)[O-])cc1 n1(CC=O)c(C)cc(O)cc1=O.C(C(=O)NC1CC1C)N(CCOC)C C1(C(=O)NCC(C(=O)OC(C)C)C)CCC=CC1N C1(NC(CC2(N(C(C(C3CC3)SC)=O)C)CC2)=O)CCC(C)(N(C)C)CC1 C1(CNC(C2(C#C)CC2)=O)CCCN1C(=O)Cc1cc(C2CC2)no1 C1(NC(C(N2CC(C)C2)C)=O)CCC(C)(NC(=O)OC(C)(C)C)CC1 C(=O)(C(C)C(F)F)NCc1c(C(=O)NCc2[nH]nc(C(C)C)n2)occ1 C(c1ccn(C)c1)=CC(=O)N(CC(=O)N(C(CCO)C(F)F)C)C1CCC1 c1(C(=O)NC(CN(C(C2C(CCC)C2)=O)C)CC)ccc(SC(C)C)cc1 c1(SC(C)C)ncccc1C(N1CCCC(NC(=O)CC2CSC2)C1)=O Cc1ncc(C(N2CCOC(C(C)NC(=O)CCc3ccon3)C2)=O)n1C C1(C(=O)NC(C(C)C)(C)C)C2CC3C(C2NC(=O)C)C13.C1CCCO1.O c1(OCC(=O)N(C2CN(C(CCC(C)C3CC3)=O)CC2O)C)ccc(Cl)c(F)c1 c1(C=O)cc(O)nc(C)n1.c1(OC)cc(CN(C(=O)CCC2CCC2)C)on1 N1(C(CCOC)=O)CCCC1Cn1cc(CNCc2ccc(C)[nH]2)nn1 C(=O)(C(C)(C)CC)N1CC(NC(CC=CC=C)=O)C1.C(C)(C)C.C=O.N c1(C(N2CC(CC=C)(NC(c3ccc(Cl)s3)=O)C2)=O)cnc2cccnc2c1 CCC(C(=O)N)C(C)C.c1(C(N2C3CC(C2)C3)=O)cc(C(F)(F)F)cc(N)c1 C(=O)(C(F)(F)C(F)F)N1CC(CC(CNC(CCC2CCCN(C)C2)=O)(C)C)C1 C1(CC)C(CC(=O)NCC2CCC2)C1(F)F.n1(CC(=O)N)ccc(C)n1 N1(C(C2CN(c3n(C)nnn3)C2)=O)CCC(C)(NC(=O)CC2(CO)CC2)C1 N1(C(CC(=O)O)=O)CCCC12CCC2.c1(C=O)c(C(F)(F)F)oc(C)c1C.CC C(=O)(C(C)(C)C1=CCSCC1)N.N1(C(C(C(C)O)(C)C)=O)CC(C)CC(C)(C)C1 CC(C)CCC(CO)NC(C1C2CCN(C(=O)Cc3ccc4c(c3)CC4)CC12)=O C(CC(C)C(C)C)NC(C(n1ccc(C)n1)(C)C)=O.C1(C=O)CC2(CSC2)C1.N C=CC(C)(O)C(=O)NC1CCC(CCC(N2CCC(C(=O)NC)C2C)=O)C1 c1(C(N(CC(CC)NC(=O)COCCSC)C)=O)noc(C)c1[N+](=O)[O-] N1(C(C(F)=CC)=O)CCCC1CN(C)C(c1nccn1CC)=O CC(C)CCCCNC(=O)C(C)CN(C)C(C1(O)CCSC1)=O N1(C(C2(CC=C)CCCC2)=O)CC2CCC2(CC(N2CC(F)(C#N)C2)=O)C1 C(=O)(C(C)CCCC(C)=O)NCC1C(CC(=O)Nc2c(CC)noc2)C1 c1(OC)ccccc1N1CCC(NC(=O)C(=O)NCCc2nnc(S)n2C)C1 N1(Cc2c(C)noc2C(C)C)CC(C(=O)O)C(C)(C(F)(F)F)C1 C(=O)(CCCCCC#N)N1C(CCNC(c2c(C)n[nH]c2)=O)CCC1 c1(OC)cccc(C(=O)NC(C)CCN(C(=O)CCCc2ncc(C)o2)C)c1F C1(C(=O)NC(CSC)(C)C(=O)Nc2ccc(C)nc2O)CN(C)CCN1C c1(C(=O)Nc2c(OC)cc(OC)nc2)ncc2ccccn12 Cc1cnc(S(C)(=O)=O)nc1N1CC2CC1CN2Cc1cncn1C C(=O)C1=C(C)CCCC1.C(Cc1ccccc1)(C(=O)NC12CC(C1)C2)OC.C CCC(C)(C)CCCC(=O)NCCNC(C1CN(C(C2CCCOC2)=O)C1)=O c1cccc(C(N2CC(O)C2)=O)c1.C1(C)(C(NC)=O)CNC(=O)C1.C#CC.S c1(C(C)SCC)nc(-c2cnn(CCOC)c2)n(C2CCC(C)(C)C2)n1 CC(C)CCC(C(=O)NC)NC(=O)CC1CCC(=O)C1C.C1CC(N(C)C)C1 c1(C(N2CC(CCNC(=O)C(=O)N(C)C)(OC)C2)=O)cccc2nccnc12 Cn1cc(C(N2CCCC2CNC(=O)COCCF)=O)nc1-c1ccccn1 C=C(C)CC(C(=O)NCC1(O)CCC(C)C1)NC(c1cc(C)cc(F)c1)=O C1(C(NOCCC(=C)C)=O)CCCN(C(C2CC(F)C(=O)N2)=O)CC1 c1(C2C(C(=O)NC(CC)CNC(C3CCCCC3)=O)C2)ccc(Cl)cc1 N1(C(C(C(C)(F)F)F)=O)CCCC2CN(C(C3CC4CC(=O)C3O4)=O)CC12 c1(C=O)ccc2nc(O)oc2c1.c1(C(=O)NCC2(C)CC2)coc2c1CSC2 C1(NC(C(C)(C)C2CCOCC2)=O)CCC(NC(c2cnsc2)=O)CC1 c1(CNC(=O)NC2(CC#C)CCOC2)nc(C)c2ccccc2n1 c1(C(=O)NC2(C(=O)NCC(C3CC3)OC)CCC2)cnn2c1CCC2 C1(NC(C=CCCC)=O)CN(C(C2CCCN2C=O)=O)CC1OC Cc1ccccc1N(C(c1sc(=N)[nH]c1C1CC1)=O)Cc1cncn1C C1(C(=O)NC)C2CCC(C2)N1C(=O)C(n1ccc(C)n1)C C12(CC)CC1CN(C(=O)C(Cc1cn[nH]c1)NC(=O)C=CCCC(C)C)C2 C1(C=O)CC12CC(C)(C)C2.C1(OC)COCCC1CC(=O)NCC1CCCC1 CCC(C)C(C(=O)NC1CCCCC1NC(c1cnsc1)=O)NC(=O)OC c1(CC(=O)N)ccc([N+](=O)[O-])cc1Cl.C1(NC(CCNC(N)=O)=O)CCCCC1 c1cc(Cl)cc(Cl)c1[N+](=O)[O-].c1(C(=O)NCc2nc(C)sc2)nc(NC)cn1C C1(C(=O)Nc2ccc(Cl)nc2)C2CCCC1CN(Cc1cccc3c1CCC3)C2 c1(OC)ccc2cc(C(N3CCCC(NC(=O)C4=COCC4)C3C)=O)[nH]c2c1 N12CCCC(C1)C(C)C(=O)N(CC(C)C)CC2=O.c1(CC)ncc(C(=O)O)s1 c1(C(CC(=O)NC(c2cccc(Br)c2)C#C)N)ccc(Cl)c(F)c1 C1(NC(C2C(NC(c3cc(C)cc(C)c3)=O)CCCC2)=O)COC2(CCCC2)C1 C1(CCC#C)CCN(C(C2CC2CNC(c2cc(O)n(CC)n2)=O)=O)CC1 C(=O)(C#CC1(C)CC1)N(C)CC1CCCN(C(=O)C(C)(C)C2CCOC2)C1 c1(NC)ccccc1C(N1CC(C(N)=O)(C)C1)=O.c1(C(=O)N)coc(O)n1 Cn1nc(C(N2CC(C)(NC(=O)C3=C(Cl)CCOC3)C2)=O)c2c1CCC(F)(F)C2 C1(C(N2CCC(NC(c3n(C(C)C)ncc3Cl)=O)C2)=O)CC(=O)NC1(C)C c1(C(N(CCCN(C)C(c2cc(C3(C)COC3)no2)=O)C)=O)n[nH]c2c1CCC2 c1(C(N2CCC(C)(CNC(C3CC(C)OC3)=O)CC2)=O)cc(F)c2cn[nH]c2c1 C1(C(=O)NCC=CC)CC12CCN(C(=O)CC1(O)CCC1)CC2 c1(CC)noc(C)c1NC(=O)CC(CNC(c1ncoc1C)=O)C1CCC1 N1(C(C2C(C)(CC)C2)=O)CCCC(CNC(C23CC(CO2)C3)=O)C1 c1(C(=O)OCC)ccc(C(=O)N)nc1.C12CC(C1)C2.c1(C=O)nocc1Cl C=CC1(C(N2CCC2c2cc(OC)no2)=O)CCNC1 c1(OCC(=O)NC2CCN(C(COC)=O)CC2)ccccc1C(C)(C)C C1(NC(C(CSC)OC)=O)CC2(C1)CC(NC(=O)CO)C2.C1CCOC1 C(C(C(=O)N(C)Cc1cncs1)NC(=O)C(C)n1cccn1)OC N1(C(C(C)NC(=O)NC)=O)CC2(C)CC1(C(=O)NC1CCCCC13CC3)C2 C1(COC)CN(C(c2c(C)c[nH]c2CC(N)=O)=O)CCN1C(=O)CN(C)C c1(C=O)cccn2c(O)nnc12.C1(C(NCC)=O)CCCC(C(F)(F)F)C1.CC n1(CCC)nc(C)cc1C(N1CCCC(n2cc(CN3CCOC3=O)nn2)C1)=O N1(C(COC(C)C)=O)CCCN(C(=O)Cc2cc(Cl)ccc2Cl)CC1C(C)C N1(C(c2c(C(C)C)noc2)=O)CCN(C(=O)C=Cc2cn(C)nn2)CC(C)(C)C1 c1(CC)ccc(C(=O)NCCc2cn(CCSc3ccccc3)nn2)cc1Cl c1(C(=O)NC(C(=O)OCC)C2CCCC2)cncnc1.c1(CC)ccoc1.C c1(C(=O)NCCc2c(C)ccs2)ccc(OCCO)nc1 N1(CC(N2C(C(=O)NCC=C(C)C)C=CC2)=O)C(=O)CCCC1=O n1(C(C)C)cc(C(=O)N(C)CCOCC)c(O)nc1=O.c1(C(=O)N)cnn[nH]1 N1(C(C(C=C)C)=O)CC(C(N2CC=CC2C(=O)NC)=O)CC12CCC2 C(C)(C)(CCC(=O)NC1CC1CC(C)C)NC(Cn1c(C)ccn1)=O C(=O)(C1=NOC(CNC(c2cccnc2OC)=O)C1)NCC(CC)(C)C CC(C)CC(C)CC(C)C(=O)NCCCCCCNC(=O)CC1CCCOCC1 O=C1OC(C(=O)NC2COCC2n2ccnc2)Cc2c(F)cc(Br)cc21 C(=O)(C(F)F)NC1(N(C)C(C2CC2C(=O)NCCO)=O)CC1 N1(C(COC(C)C)=O)CC(NC(=O)CCOCC2CCCO2)C2(CC2)C1 C(C(=O)N1CCN(C(C2CCCN(C(=O)C(F)(F)F)C2)=O)CC1)(C(C)(C)C)SC C(c1ccc(O)cc1)=CC(=O)NCC(C)N(C(=O)C(F)=CC1CC1)C Cc1ccc(C(C(=O)NCCCC2CC2)N(C2CCCC2C#N)C)c(Cl)n1 c1(C(N2CC(C(N)=O)(CNC(C(C=C)O)=O)C2)=O)nc(C)c(C)s1 C1(C(C)C)N(C(c2nc(Cl)ccc2Cl)=O)CC12CCN(C(=O)C(C)O)CC2 C1(CNC(C(C=C)C)=O)CCCCC1NC(c1nnc(C)s1)=O N1(C(CCCC)=O)CCN(C(=O)CC2CCOC(C)(C)C2)CC1C1CC1 N1(C(CC=C(C)C)=O)CCC2(CC1)CN(C(=O)CCCc1ncc(C)o1)C2 C1(NC(c2cc(CCC)ncc2)=O)CCN(C(=O)C=C2CCC2)CC1(C)C CC(CC=Cc1ccccc1)C(=O)N1CCC(CNC(=O)CCC2(C)CC2)C1 c1(C(=O)NCC2(OC)CN(C(=O)C(C)C(F)(F)F)C2)cnc2[nH]ncc2c1 c1(C=O)cc2scc(C)c2[nH]1.c1(C(=O)OC)cccc(C(=O)NC2CC2)n1.C C12(CNC(CCCCC)=O)CC3CCC(C1C2)N3C(=O)C(F)(CC)C=O Cn1cnc2c(NCCC34CCCC3C4)nc(N3CCCC(CO)(CO)C3)nc12 CCC(C(=O)NCC1CC2(CC2)CN1C(c1cc(Cl)ccc1C)=O)C(C)C c1(CNC(C=C(C)C)=O)c(C(F)(F)F)cnn1C C1(CNC(=O)Cc2ccc(Br)cn2)C(C2CC2)CCN1C(=O)CCC(F)F CC1CN(C(=O)C(C2CC2)N(C)C(C2CC(=O)CCO2)=O)CC2(CCC2)O1 N1(C(C2CC(C(=O)OC)C2)=O)CC2CCN(C(=O)CCc3ccccc3)C2C1 N1(C(C#CC2(C)CC2)=O)CCC2(CC1)CCN(C(=O)Cc1csc(S)n1)CC2 c1(NC(COC2CCN(C(C3C(OC)(OC)CC3)=O)C2)=O)ccc(C)nc1 C1(C(N(C(C)C)Cc2c(C)cccc2)=O)CC12CCN(C1CCOC1)CC2 CC(O)CCCC(=O)NC1CCN(C(=O)O)C1.c1(-n2ccnn2)cccc(Br)c1 N1(C(C23C(CN(C=O)C2)CCC3)=O)CC(O)C2(CCCC2)C1 C1(O)CCCN(C(c2ccn3ccsc23)=O)C1.c1(CC)oc(C)cc1C(=O)NC c1(C(=O)OC)cn(C(N)C(=O)NC(c2cn(C(F)(F)CO)nn2)=O)nn1 C(=O)(C(C)(CC)C(F)F)NC1CC(CNC(CCC=CCC=C)=O)C(O)C1 C1(NC(CCNC(C)=O)=O)CCCC(CNC(=O)C#CC2(C)CC2)CC1 CC(CC(=O)N1CCC(C(C)(C)C(=O)Nc2ccccc2O)C1)C(F)(F)F c1(C(=O)NC2CCC(NC(C(C)SC(C)C)=O)CC2)cccc(F)c1O C(=O)(C(CC(N)=O)NC(c1ccc(C#N)[nH]1)=O)NCCc1cc(C)[nH]n1 N1(C(c2n(CC(C)C)ncc2)=O)CCC(N=c2[nH]nc(C(F)F)o2)C1 Cc1nc(O)[nH]c1C(=O)NCC1CCCN(C(C2CC2C2CCC2)=O)C1 C1(C(=O)NCCOCCOCC)COCCC1.C1(C)(C(=O)N)CCCC1 C1(NC(CCn2ccc(C)n2)=O)(CO)CCCN(C(=O)CCCN)C1.[SH](C)(=O)=O c1(C(N2CC(CCCNC(C3CN(C(C)=O)C3)=O)OCC2)=O)cccc(Cl)c1C C1(OCC(=O)NCC2CC2)CCC12CC(C=O)C2.c1cccs1.C=CC C1(NC(CCN(C(=O)Cc2ccc(F)cc2)CC#C)=O)CC(O)C1(C)C C(=O)(C(CO)C(F)(F)F)N1C2CC(C(=O)NC(C)(CO)C3CC3)(OC2)C1 N1(C(C(CC2CCCCC2)OC)=O)CCC(C)(NC(=O)C(C)C2CC2)CC1 c1(C=O)ccc(C2CC(F)(F)C2)cc1.C(=O)(C(C)N(C)C)NC(C)C.CC N1(C(C(C(C)OC)NC(=O)C(C)C2CC2)=O)CCCCC(COC)C1 N1(C(c2cc(OC)no2)=O)C(C(N2CCOCC2)=O)CC2CCCCC12 c1(C(=O)NCC(CNC(CC=C(C)C)=O)O)ncoc1-c1ccccc1 C1(NC(=O)CNC(C2CCCCC2)=O)CCCCN(C(=O)CSC(F)(F)F)C1 N1(C(C(C)SC(C)C)=O)CCCC1CN(C(=O)C(C)Cc1cccnc1)C c1(C(N(CC(CC)NC(=O)Cn2ccnc2C)C)=O)scnc1C1CC1 c1(C(=O)NCCC2CCCN(C(C(CC)C(C)C)=O)C2)ccnc2c1CCC2 c1(C=O)ccc([N+](=O)[O-])c(S(N)(=O)=O)c1.N1(C(C(F)=C)=O)CC2CCC1C2.CC Cn1ccc2c(N3CCOCC3CC(N3CCCC3(C)C)=O)ncnc12 Cc1ccc(C(N2CCCC(N(C(=O)C#CC(C)(C)C)C)C2)=O)cc1C(F)(F)F CC1CCCCC1CNC(c1cn2c(n1)CCC2)=O.C1(C=O)CC(F)(F)C1.N C1(C2CC2)CCCN1C(c1csc(C2CC2)n1)=O.CC(C)CCOCC(=O)N N1(C(c2cnc(O)s2)=O)CCN(C(C2CCN(CCF)CC2)=O)C(C(F)F)C1 C1(CC)(NC(=O)C(N)=O)CCN(C(=O)CC(O)C2CCCC2)CC1 c1(NC(c2n(C=C)ncc2)=O)ccc(NC(c2cccc(N(C)C)c2)=O)c(C)c1 C1(NC(C2(C)N(C(c3n(C)cnc3)=O)CCC2)=O)CCCCC12CCC2 c1(C(N2C(CNC(c3c(CCC)onc3C)=O)COCC2)=O)ccc(I)cc1O C1(C(=O)NC)CCN(C(C2CCOCC2NC(=O)Cc2cnc(C)s2)=O)CC1 n1(-c2ccn(CC)n2)nc(CCSC)nc1-c1cc(Cc2ccccc2)on1 Fc1cc(C2CCN(CC3CC4CCC4C3)C2)cc(F)c1 C1(N(C(CSCC=C)=O)C)CCN(C(=O)CC2CNC(=O)C2)C1 C1(C(N(CCCCO)C2C(C)C2)=O)CC2(CCNCC2)C1 C1(C(N(C(C)CC2CC2)C)=O)CC2CCCC2N1C(=O)C(C)O C(=O)(C(O)CN1CCCC1)NC(C)C(=O)NCCCOCC(F)F c1(COCC)nc2n(n1)CCCC2NS(=O)(=O)C1CC(C(F)(F)F)(OC)C1 Cc1cn(C)nc1C(=O)N(C(=O)CCN1CCN(C(C)(C)C)CC1)C c1(C(=O)NC(CNC(C(C(C)C)OCC)=O)C)ccc(F)cc1C1CC1 C(c1ccc(OCC2CCCCC2)cc1)=CC(=O)NCC1CNCC1(F)F N1(C(COCC(C)C)=O)CCC(C)C1CNC(=O)C(F)(F)c1ncccn1 N1(CC=O)CCCCCC1.C1(CNC(=O)Cc2coc(C(F)F)n2)CCCC1.N C(C(C(=O)N1CCCC(C(=O)OC)C1)C(C)C)NC(CC(=O)NCC)=O c1(C(=O)NC(C2CCN(C(=O)Cn3cnnc3O)C2)C)ccc2c[nH]nc2c1 O=C(N=c1[nH][nH]c2c1CCCC2)C1CCN1Cc1c(F)ccc(Br)c1F C#Cc1ccc(F)c(C(=O)NCC2CCC2)c1.c1(C=O)cnn(C(C)C)c1.N c1(C(=O)NC(C2CCNCC2)CO)ccnc2cc(F)cnc12 c1(C(=O)NC2(C(N3CC(O)(COC)C3)=O)CSC2)c[nH]c(=O)cn1 c1(CCC)ccccc1C(=O)N(CCCNC(C1CCC1(C)C)=O)C(C)C N#Cc1cc(C(N2CCCCC2C2(NC(c3ccco3)=O)CC2)=O)ccc1Cl N1(C(C(CC(C)C)OC)=O)CC2CN(C(C3CC(=O)OC3(C)C)=O)CC(C1)O2 C1(CC#C)(C(=O)NCCC2(CNC(=O)C3=CCOC3)CC2)CCCCC1 N1(C(c2sc(NC(=O)CCCF)cc2C)=O)CCCC(c2ccccc2)C1.c1ccccc1 c1(C(=O)NC(CC(C)NC(=O)COc2ccc(F)nc2)C)cccc(F)c1Cl c1(C(N(CCNC(=O)CC2C=NN(C)C2=O)CC)=O)cccc(F)c1.O c1(OC)cccc2c(C(=O)NCC(CO)NC(C3CC4CCC3C4)=O)coc12 c1(C(=O)NC2CC3(CC(NC(c4c(C)nsc4)=O)C3)C2)cccc2cc[nH]c12 C(C)(c1ccco1)=CC(N1CC(C)(C(=O)NC(CC#C)CO)C1)=O C(C)(C=O)(C(C)C)OC.c1(C(N2CCC(CCC)CC2)=O)cnc(O)c(C)c1.N C(=O)(C(CNC(c1cnn(C)c1N)=O)C(C)(C)C)N(C1CC2(CCC2)C1)C CC1(C)OC(=O)CC1C(=O)OCc1cccc(C2CC2)c1 N1(C(C(c2ccc(Cl)cc2)C)=O)CCC2(CCN(C(=O)Cc3cc[nH]c3)C2)C1 c1(C(C)C)cccc(F)c1C(=O)N(C1CCN(C(C2(C)CCCO2)=O)CC1)C N#CC1CNCCN1C(c1ccc(OC(F)F)cc1F)=O C1(C(=O)NCC2C(NC(CCC(C)C)=O)COC2)CC2CC(=O)C1C2 C(CC)(C(=O)NCC)N.C(C)C.C(C(=O)N(C)C)NC(=O)OCC C=CCCCC(=O)N1CCCCC1CN(C(c1cnncc1O)=O)CC C(CC(F)(F)Br)NC(=O)NCCNC(c1ccco1)=O C1(CCNC(CN2CC(C)C2)=O)CCCN1C(C1OCC1(C)C)=O Cc1cc(C(=O)NCC2C(C)CCCN2C(C2CC2(F)F)=O)n2ncnc2n1 c1(CNC(c2cnccn2)=O)ncc(C(=O)NCCn2cncn2)cn1 c1(C(=O)NCC2(CCO)CC2)cccn2ccnc12.CC1(C=O)CC(C)C1.N Cc1c(C(=O)OCC23CC(C2)C3)sc2cc(F)ccc12 C1(NC(C2(C=C)CCOCC2)=O)CCC2CCN(C(C3(C(=O)NC)CC3)=O)C1C2 C(=O)(CC(=O)NCC(C)N(C(=O)COCc1ccnn1C)C)NCC#C c1(CC)nn(C)c(Cl)c1C(=O)N(CC(C)NC(c1cc(C)cc(C)n1)=O)C C(C(C)(C)N=c1ccc(C#N)n[nH]1)NC(C1CCC(CC)O1)=O C1(C(=O)OC)CC(NC(=O)NC2CC2c2ccccc2F)C2OC(C)(C)OC12 c1(N(C2CNC2)C(c2cc(C)ncc2)=O)nc(C)nc2c1CCC2 C12(C(=O)NC3CN(C(Cc4c(C)nn(C)c4)=O)C3)CCCCC1CCC2 S(=O)(=O)(c1ccc(O)c(NC(=O)CN2CC(C(F)(F)F)C(C)C2)c1)NC C(C)(N=c1nc2scnc2c(NCC2CC(C)C2)[nH]1)c1scc(CC)n1 C1(CNC(c2c[nH]nc2Br)=O)Cc2ccccc2CN1C(C1C=CCC1)=O N1(C(C(CC=C)C)=O)CCN(C(=O)CN2CCC(O)CC2)CC1C N1(C(C(CCCOC)(C)C)=O)CC(NC(c2[nH]cnc2C)=O)CC2(CCC2)C1 S(=O)(=O)(c1ccc2[nH]c(=NCCOCCF)sc2c1)N1CC(C)OCCC1 C1(NC(Cn2c(CCC)ncc2)=O)CC(O)CN(C(c2nnc(O)nc2O)=O)C1 C#CCC(C)(C(=O)Nc1cccc(SC)c1)NC(C1CC2(C1)CC2(F)F)=O O=C(C1=COCCC1)NC1CCN(C(c2cc3n(c2)CCC3)=O)CC1F C1(C=O)CC(S(N)(=O)=O)C1.N1(C(CNC(CCC)=O)=O)CC(C)C(C)C1.N C(=O)(CC1=NN(C)C(=O)C1)N(C1CCN(C(C2CCC(C)CC2)=O)C1)C C1(CNC(C(COC)C)=O)CC2(CO1)CN(C(c1cc3scc(Cl)c3[nH]1)=O)C2 N1(C(c2c(C)nc(-c3ncc[nH]3)s2)=O)CCCC2(CC2)C1.C(=O)C=C1CCC1.N N1(C(COCCOC)=O)CCN(C(c2cc(C)cc(C)c2)=O)CC1C(F)F C=CCCC(C(=O)NC1CC2(CCC2)C1O)NC(C1CC2CCC1CC2)=O c1(C(N2C(C(=O)NCc3ccc(C#N)nc3)CC2)=O)c(Cl)ccc(Br)c1Cl C(C(=O)NCCCC1CC1)(C(CC)CCC)N(C(CCCC)C(=O)OCC)C C1(OCC)CCN(C(=O)C(C)C(C)NC(c2c[nH]nc2C(C)C)=O)CC1 c1(C(=O)NC2CCN(C(c3cnc(C(C)OCC)s3)=O)C2)ccc(C)s1.C c1(C(N2CCC(NC(=O)NC)C2)C(=O)NC2(C)CC2)cc2cc(Cl)ccc2o1 C1(C(=O)NCC2N(C(c3cnc(OC)s3)=O)CC2)Oc2ccccc2C1C N1(C(CCCCNC(N)=O)=O)CCC(CO)C(NC(c2ccoc2Br)=O)C1 Cc1nc2sccn2c1C(=O)NCC1CC(C)N(C(c2cnn(C)n2)=O)C1 N=c1[nH]c(C2CC2)ncc1C(=O)NC1(CNC(c2nocc2Cl)=O)CCOC1 c1(C(=O)NCC2COCCN(C(C3(SC)CC3)=O)C2)cc(C)cc(C)c1C C1(NC(=O)CCN2CCCC2=O)CC2(C1)CC2.c1(C=O)cc(C(F)F)ccn1.N c1(C(=O)OC)cccc(S(=O)(=O)NC(c2ccc(OC(F)(F)F)nc2)=O)c1 c1(OC)cc(Cl)c(CN2CC3CC3(C(=O)NC(C)C(F)(F)F)C2)c(Cl)c1 Cc1ccc2cc(C(=O)NCC3CCCC(NC(=O)CN(C)C)C3)cn2c1 C1(C(C)(C)C)CCC(C(N2CCC(c3cccnc3O)C2)=O)CC1 C1(=CCNC(Cn2nnc(C)n2)=O)CCN(C(C2CCS2(=O)=O)=O)CC1 c1(N(C)C)cnc(C(=O)NCC(C(C)(C)C)NC(C2CCCC(=O)N2)=O)cn1 Cc1cccn(CC(=O)NCCCCCNC(=O)CCNC(=O)CC(C)C)c1=O C1CN(C(=O)CC2C=NN(C)C2=O)CC1n1ccnn1.CC(C=O)=C1CCC1.N N1(C(c2cnsn2)=O)CCN(C(c2ccc(=O)n(C3CC3)c2)=O)C(CF)C1 N1(C(C(c2ccc(C)cc2)C)=O)CC2CCN(C(=O)CSc3cccs3)CC12 N1(C(CC2CC(SC)C2)=O)CCCC(C)(NC(C2CCC3(CC3)C2)=O)C1 C(N=c1ccc2c([nH]1)CCC2=O)C1OCCCN(C(c2c(C)nn(C)c2)=O)C1 CC(C)(C)C(C)(O)C(=O)N.C(=O)CS(=O)(=O)NCCO.CC(C)C1CCC1 N1(C(CS(CC)=O)=O)CC2CC(C(=O)NCCCC(=O)N(C)OC)C(C2)C1 Cn1cc2c(n1)CCCC2NC(c1cn(Cc2ccccc2)nn1)=O N1(C(C(=O)NC(C)C)=O)CCC2CN(C(C34CCC(C)(CC3)CO4)=O)CC12 C1(C(C2CCC2)NC(C2(C)CC2)=O)CCSCC1 C1(C(C)C)CN(C(C2CCSC(C)C2)=O)CCN1C(=O)Cn1cncn1 N1(CC)CC2(CN(C(=O)CC3CN(C(=O)CCOC(C)C)CCO3)C2)C1 C=CC(C)C(C)C(=O)NCC1(O)CN(C(c2cc3sccc3s2)=O)C1 c1(C(N(C2CN(C(=O)CC(C)C3CCCCC3)C2)C)=O)cn(CCCF)nn1 c1(SCC)cccc(CC(N2CC=CC2CNC(C2CC2C)=O)=O)c1 N1(C(C(C)C2CCOC2)=O)CCC2(CCCN2C(c2cccc(N)c2F)=O)CC1 Cc1cn2c(C(=O)NCc3csc(-c4ccccc4C)n3)cnc2s1 C1(CC(=O)NCC2CCN(C(=O)OC)CC2)CCOC(=O)CC1.c1ccccc1 CC(F)(CC1CCCC1)C(=O)N1CCC(O)(CCNC(C2(F)CCOCC2)=O)C1 C(C(C)CNC(=O)C(C)N1CCCC1)N(C(CSCCOC)=O)C c1(CC(=O)NC(CC)CNC(c2cc3n(n2)CCO3)=O)csc2ccc(C)cc12 C1(C(=O)O)CCC(NCc2c[nH]nc2C(F)(F)F)C1 N1(C(C2C(C(C)C)N(C(=O)CCCn3cccn3)CC2)=O)CCC2(CCCC2)C1 N1(C(CC2C(NC(C3(CC)CCCO3)=O)CCC2)=O)CCSC(C)(C)C1 C12(C(=O)NC3C(C=C)OCC3)CCN(C(=O)C=C(C)C3CC3)CCC1C2 C#CCCN=C(NCCOc1cccc(Cl)c1Cl)NCc1nn[nH]c1C1CC1 N1(C(C(C)CC(F)F)=O)CCC2(CC1)CN(C(C1CC1(Cl)Cl)=O)C2 C12(CNC(C(C(C)C)SC)=O)CC(NC(=O)CCC(N)=O)(C1)C(C)O2 c1(C(C)(C)C)cnc(Cl)c(NC(=O)NCC2CC23CCOCC3)c1 S(=O)(=O)(c1ccc(C#N)c(NCCC(Cl)(Cl)Cl)c1)NC(C)CN1CCOCC1 CC(=O)CCC(=O)N(C1(C(N2CCC(CC(F)F)C2)=O)CC1)C C(=O)(C(C1=CCCSC1)N1CCC(S(=O)(=O)N(C)C)C1)NCC=C NS(=O)(=O)c1cc(C(=O)NCCCN2CCN(C(c3cc(O)cs3)=O)CC2)co1 CCC(N=c1cc(C)nc(N2CCC(c3nncn3C)C2)[nH]1)C1CCCC1 c1(CC(=O)NCC(C)NC(C2(C)CCCO2)=O)c[nH]c2ccc(Br)cc12 Cc1ccc([N+](=O)[O-])c(C)c1C(=O)NC1CCC1.C1(C=O)C=CC=CC=C1.C c1cc(C=O)cc(F)c1.C(C)CCN(C)C(C1CCN1S(C)(=O)=O)=O.CC C1(NC(=O)NC(CCC)=O)CCN(Cn2cc(C(F)(F)F)cc(Cl)c2=O)CC1 N(C(=NCCCc1ccccn1)NCCC1CCOC1)CCOCC=C c1(CCC)ccc(C#N)c(NCCCNC(c2nc(C)n(C)n2)=O)n1 C1(CNC(CC(=O)NCC)=O)CN(C(=O)CSSC)CC1C Cn1nc2c(c1C(=O)N(c1cnccn1)C)CNC2.N1(CC)CC(O)C1 c1(C(C)=O)c(NC2CCCCC2NC(=O)CCC(C)N(C)C)ncnc1Cl Cc1cc(Br)cc(C(=O)NCC2CCC2NC(c2ccsn2)=O)c1F C(C(O)C(=O)NCCn1ccc(C(=O)NCC2CCC2(F)F)c1)SC N1(C(c2c(OC)cc(Cl)cc2)=O)CC2(CCC2)CC1CNC(=O)C(C)SC C1(C(C)NC(CCSCCC)=O)CN(C(c2cc(C(C)C)n(C)n2)=O)CCO1 c1(C(=O)NCC2C(CNC(C3CC(C)(F)C3)=O)C2)cnn(CCO)c1N O=C(CC1OCc2ccccc21)N1CCN(C(c2ccc[nH]2)=O)C(CF)C1 C(=O)(CCC(C)CN(C)C)NC1C(CC(=O)N(CC(CC)C)CC)C(O)C1 c1(N2CCCC(NC(CC(CC)(F)F)=O)C2C)ncc([N+](=O)[O-])cc1Br Cc1nc(CC(C)C)sc1C(N1CCCCC1C)=O.c1(C(=O)N)cn(C)c(O)n1 CCC(C(=O)NCC1CN(C(N)=O)C1)C(C)C.C1C(=O)N1 c1(CN2C(C(=O)Nc3cc(C(=O)OC)sc3)COCC2)cc(Cl)nc(Cl)c1 C1(NCCc2c(C)occ2C(F)(F)F)CCC2(CCCO2)CC1 CC(C)CC(C)CC(=O)N(C1CCCN(C(c2cc(F)cc(F)c2N)=O)C1)C C1(N(C)C)CC(C(=O)NC(C(=O)NC2CCC2)C2CCOC2)C1 c1(C(=O)NCC(=C)CCNC(=O)C=CC2CCOC2)cn(C)c(=O)cn1 C12(NC(C(CC=CC)C)=O)CCCC1CN(C(c1cc(C(=O)OC)no1)=O)C2 c1(C(N2CC(SC)CC2)=O)ccccc1[N+](=O)[O-].C(=O)C(C)(C)C.C(=O)(C)N C1(C)(CC)CC(NC(=O)C)CN1C(=O)C.c1cccc(Cl)c1C.C(C)=O.O c1(C(N2C(CNC(C(C)C3(O)CCC3)=O)CC(F)C2)=O)n[nH]c2c1CN(C)CC2 Cc1ccc(NC(c2nc(NCc3ccc(I)o3)cn2C)=O)c(O)n1 C1(C(=O)O)C2(CCC2)C12CC(C(N1C3CCCC1(F)CC3)=O)C2 C1(n2cc(CN(C)C3CC3)nn2)CN(C(C2(C)CC2(Cl)Cl)=O)CC1SC N1(C(C(COC)COC)=O)CCCCC2(CCN(C(=O)CCOCC(F)F)C2)C1 c1(C(C(=O)NCCCNC(Cc2n(C(C)C)cnn2)=O)O)ccc(Br)cc1 C1(c2n(CCCC)nnn2)(NCC2CC(CC)C2)CCC1C1CCC1 C#CC1(C(=O)NC2CCCC(O)C2)CCN(C(=O)C(C(C)C)C2CCC2)CC1 N1(C(C(=O)NCCOCC)C2CC2(C)C)CCC(O)(c2ncnn2C)CC1 C1(OC)CC(CNC(=O)C(c2cccc(C(F)(F)F)n2)(F)F)C1(C)C C1(C)(C(=O)N)CC2CCC1O2.N1(C(CCCNC(C)=O)=O)CCC(OCC)CC1 CC1(CNC(=O)Cc2cccc(F)c2O)CCCCC1.C1(CC(=O)N)CCSC1 CC1(O)CCCN(C(C2CC(O)CN2C(c2ccc(Cl)cc2Br)=O)=O)CC1 C=CC1COCCN1C(C(=O)NC1CC(F)(F)C1)C(C)CC1CC1 C1(C2CCN(C3CC3)CC2)(NC(=O)NC(C#C)CC2CCCO2)CC1 N1(C(c2n(C=C)ncc2)=O)CCC(NC(c2cnn(C3CCC3)c2C)=O)CC1C c1(C(=O)N)cc2n(n1)CCOC2.CC1(C)CCCN(C(C2(C(F)F)CCC2)=O)C1 N1(C(c2c(C)nsc2C)=O)CCC2(C1)CN(C(=O)C=Cc1ccco1)CC(C)O2 N1(C(Cn2nnc(=N)[nH]2)=O)CC(C2(NC(=O)CCc3nccs3)CC2)C1 C1(NC(C2(F)CN(C(=O)OC)C2)=O)CCCCC1.c1(CC=O)cccnc1.N N1(C(CCNC(C)=O)=O)CC2CN(C(C3C4CCC3(c3cncs3)C4)=O)CC2(C)C1 C=CCC(CC(C)C)C(=O)N1CCC(CCCCCNC(C2CC(O)C2)=O)CC1 CCCC(C)(O)C(=O)NC(CNC(=O)CC1(COC)CCCC1)CCOC N1(C(=O)CCSC(F)(F)F)CCN(C(c2csc(C(F)F)n2)=O)CC(O)C1 C(=O)(C(O)CCCNC(=O)C(c1cccnc1)O)N(CC(=C)C)C C(=O)CS(=O)(=O)C(C)(C)C.CC1CCC(=CC(=O)NC(C)CC(C)C)CC1.N C#CCCCCCCCC(=O)NC1CCN(C(C2(CC#C)CCC2)=O)CC1CC CCC(C)(C)C(=O)NCC(CNC(C1CC=CCC1)=O)OC Cc1cc(N(C2(C#N)CCNC2)C(=O)CCc2ccccc2C(N)=O)cc(C)c1 c1(C(CSCC)C)cn(CCC(=O)N(CC(C)(C)C)CCC2CCOC2)nn1 N1(C(C2N(S(C)(=O)=O)CCC2)=O)CC(C2CC2)C1 C1(C(N2CCN(C(C(C)=CC)=O)C(C3CC3)C2)=O)CC2CCC(C1)C2F C1(C(=O)NC2CN(C3CCC3)C2)C2COCC12 C(=O)(C1CCCc2nc[nH]c21)N1CCC(NC(C(CC)C)=O)CC1 c1(C(=O)NC2C(NC(CN(C)S(N)(=O)=O)=O)COC2)c(Cl)cc(Cl)nc1N N1(C(C(C)OCC)=O)CCC2(C1)CN(C(c1cncc(I)c1)=O)C2 C1(C=O)CCCC2(CC2)C1.C(C)(C)(CCCNC(c1cn(CC)cn1)=O)OC CCCC(CCCNC(=O)CCN(C)C(C)=O)NC(C1CC(F)(F)C1)=O.C CCC(C)CC(C(=O)NCC1(C)CC=CCC1)NC(c1ncn(CC)n1)=O C1(NC(C(C)(C)OCC)=O)CN(C(=O)CC(C)F)CCC1CO c1(C(C)NC(C2CN(C(=O)CCc3ccn(C)c3)CCO2)=O)cc(Cl)ccc1F Cc1cc(C(=O)NC(C)C(CO)NC(=O)C(C)C(F)F)c2ncccc2c1 C#Cc1ccc(C(=O)N(CCCNC(=O)C(CC(C)C)N(C)C)C)nc1 C1(C(N2CC(NC(C3(C)CC3)=O)C(O)C2)=O)CCc2c[nH]nc2C1 C(CC(C(=O)NCC1CSC1)NC(=O)CNc1ncccn1)=CC c1(OC)cc(C(N2CC(F)(C(=O)NCC(C)(O)C3CCC3)C2)=O)[nH]n1.CC c1(C(=O)NC(CNC(C(C(C)(C)C)N(C)C)=O)CO)cc([N+](=O)[O-])nn1C c1(C(=O)NCC2N(C(C=C(CCC)C)=O)CCCC2)ccc2ncccc2c1F C(=O)(C1CCCc2ccccc21)NCC(CC)NC(c1c(C)cc(CC)o1)=O C(=O)(C1=CCC(NC(c2ccc(C#N)s2)=O)C1)N(C1CCCC1)CC=C c1(C(=O)NCC2N(C(C(C)N3CCC3)=O)CC(F)C2)ccc2ccn(C)c2c1 c1(C(N2CC(NC(Cc3ncc(C)s3)=O)C2)=O)ccc(-c2ccc(F)cc2)cc1 N1(C(C=C(CNC(c2cc(C)nnc2)=O)C)=O)CCCC(CCO)CC1 N1(C(=O)CC2COCC2O)CCN(C(C2(CC3CC3)CCC2)=O)CC1C1CCC1 C1(C(=O)NC(C=C)C)CC1C1CCN(C(=O)OC(C)(C)C)CC1 C(=O)(CC(C)(C)C(C)(F)F)N.CC(C)C(C(=O)NC1CCCC1)NC(N)=O Cc1ccc(-n2cc(CNC(C)C(F)F)nn2)c(C)c1 C(c1ccc2c(c1)CCO2)=CC(N1CC2CC2C1)=O.C1(C(=O)N)C=CCC1.C c1(C(=O)NCCC2CSCCN2C(c2cnc(Cl)cn2)=O)cnn2cc[nH]c12 N1(C(c2cn(C)nn2)=O)CCC(C)(C)C(C(N2CC(Cc3ccoc3)C2)=O)C1 N1(C(c2cc(C)on2)=O)CC(NC(=O)CCOCC(C)(C)C)CC2(CCC2)C1 C1(C=O)CCCC(C2CC2)C1.c1(OCC(=O)NC(C2CC2)C)ccsc1.N C1(NC(C(CC#CC)NC(=O)C(c2cncnc2)C)=O)CCCC2(CC1)CC2 c1(C(C)=O)c(C)[nH]c(C(=O)NC2(C)CCOCC2)c1C.C(=O)C(F)C(C)(C)O N1(C(C(CC)NC(=O)C=Cc2cc(C)no2)=O)CCC2CCN(C)C2C1 Cc1ccc2c(c1)OC(C)(C)CC2NC(c1nnn(C2CC2)c1C1CC1)=O C(=O)CCC(C)(C)N1CCOCC1.c1(C(C)NC(C2CC2C)=O)ncc[nH]c1=O CCCCC(C)(F)C(=O)NCC(C1CC1)NC(c1c(N)cc(F)cc1Cl)=O C(=O)(CCC(=O)N1CCC(O)(CNC(=O)CC2CCC2)C1)N(CC)CC C(=O)CC(C)(O)C(F)(F)F.C1(OC)CCC2(C(=O)NCC)CCC12.C1CC1 CC(CC(=O)NC1(C(=O)NC2CC=CCC2)CCC1)C1CC1 C=CC(CCC)CC(=O)N1CCN(CC(=O)NCc2nnc3n2CCC3)CC1 C=CCC(CNC(c1cc(C)c(Cl)s1)=O)CC(C)C(C)(C)C C1(OC)(CNC(=O)CC2CCCC(N)C2)CCC(C)C1 c1(C(=O)NC(C)CCNC(=O)C(F)CC2CCCC2)cnc(N)c(Br)c1 C(CCC(=O)N(C1CCN(C2CC2)C1)C)N(C(CC=C(C)C)=O)C C1(NC(c2c(C)scn2)=O)CCN(Cc2cc(Br)cnc2Br)CC1F C1(C)(OCc2occ(OC)c2)CCCOC1.C1(N)CCCN1C(n1cccn1)=O N1(C(C2N(Cc3cccc(OC)c3F)CCNC2)=O)Cc2ccc(Cl)cc2C1 C1(CC(=O)NCCCOC=C)CC(C)N(C(c2cncnc2C)=O)C1 c1(C(=O)NC2CCC(NCc3cn(CCC)nc3)C2)cc2[nH]ccc2cc1Cl c1(C=O)csc(S(N)(=O)=O)c1.c1(CC)cc(C(=O)N)n[nH]1.C1(CCC)CC1 N1(C(C(C(CC)C)N(C)C)=O)CC(N=[N+]=[N-])CC1C(=O)NCCO.CCC(C)C c1(C2CCN(CC(=O)NC(c3ccccc3)C3CCCC3)C2)cncc(F)c1 C1(CC(=O)OC)CN(c2nnc(-c3cnn[nH]3)n2CC(C)C)CC1N1CCCC1 C1(NC(c2conc2C2CC2)=O)CCC12CCC2.c1(C(=O)N)n[nH]c2c1COC2 c1(C(N2CCOC(C)(C(F)F)C2)C(=O)NCCCOC)ccc(CO)cc1F Cc1nn(C)c(NC(=O)NC2CC(Oc3ccccc3)C2)c1-c1ccc(Br)cc1 CON(C(=O)CC1CC2(CC2)CN1C(c1cccc(OC)n1)=O)C1CCC1 c1(N2CC3CCCC(NC(CC(CC)O)=O)C3C2)cc(C)nc(S(C)(=O)=O)n1 c1(SCC)ccc(CC(=O)NC(C)(C)CO)cc1.C(=O)C(C)CN(C)C.N C(=O)(CC(C(F)(F)F)P(C)(C)=O)N1CCN(C(c2ccc(OC)s2)=O)C(CF)C1 Cc1ccc(C(N2CCOCC(C(=O)NC(C3CCCCC3)C)C2)=O)c(O)n1 C#Cc1cc(F)c(C(=O)NC2CCCCN(C(=O)CC3(C)OCCO3)C2)c(F)c1 c1(CC)ccc(C(N2CC(NC(=O)C(C(C)O)N(C)C)C(O)C2)=O)c(Cl)c1 C1(NC(C(=O)OCC)(C)C(C)C)COc2ccccc2SC1 c1(C=O)cnc2c(F)cccc2c1.c1(COC)ncc(C(=O)NC2CCC2)s1.N C(=O)(C1=CCC(C)(C)CC1)N1C(C)CC(CNC(=O)C2=CCCCO2)C1 CC1CC(NC(c2nnn(C)c2C(F)F)=O)CCN1C(=O)CN1CC2CCC1C2 CCC(CCC(=O)NC1(C(C)O)CC1)NC(C1CC1(F)Cl)=O C#Cc1cccc(C(=O)NCC2CCN(C(c3cncc(C=C)c3)=O)CC2)c1 C1(O)(C(=O)NC(C(=O)NC(CO)C2(O)CC2)Cc2ccco2)CCOCC1 c1(COC)nc(CNC(c2nnnn2CC2CC2)C2(CF)CC2)cs1 N1(C(CN(CC)CC)=O)CCC(C(=O)NCC2(OC)CC2)C1 N1(C(C(N2C(=O)CCC2=O)CC)=O)CCC(NC(=O)C2=CCCCO2)C12CC2 C1(CNC(CCCC#C)=O)CCN(C(c2coc(C(F)(F)F)c2)=O)C12CC2 CCC(C)C(O)CC(=O)NOCC(=O)NCCC(O)CO C(=O)(C#CCNC(=O)C(C)CN(C)C)N(C1CC(=C)C1)C N1(C(C(C=CC)O)=O)CCC(CN(C(=O)C(C)Sc2ccc(Cl)cc2)C)CC1 NS(=O)(=O)c1cccc(CCC(=O)NCC(O)C)c1.C1(O)(CC=O)CCOC1.N CC1CN(C(=O)CNC(=O)C(C)(C)C)CC(C)CN1C(=O)OC(C)(C)C c1(C(=O)OC)cc(C(=O)NC(COC)Cc2ccccc2)cc2[nH]ccc12 C=CC(C)(CCOC)C(=O)N1CC(O)(C(C)NC(=O)CC2CC3CCC2C3)C1 N1(C(C(=O)NCC)C2CC(CC)C2)CCCCC1CC(=O)NC c1(OC)c(C(=O)N(C(C)C)C)cccc1Cl.C1(C(=O)N)CC(CC(F)(F)F)C1 C1(CNC(C2CCCN2C2CC2)=O)CCN(C(=O)CCc2ccc[nH]2)C1 C=CC(=C)CCC(C(=C)C)Nc1cc(Cl)cc(Cl)c1 C1(CC=O)CCCS1(=O)=O.C1(CC(=O)NCCCN(C)C)CCCC1(F)F.C CC(CNC(c1c[nH]nc1-n1cnnn1)=O)(CO)NC(=O)C=O.CC(F)F.N C1(OC)CC(NC(c2c[nH]nc2C2CC2)=O)CN(C(c2cc3sccc3s2)=O)C1 c1(C=O)coc2c1CS(=O)(=O)C2.C(C)CC(C)C.CCC(C=O)NC(C)=O.N c1(C(=O)NCCNC(C2CCCN(C(COC)=O)C2)=O)cnc(O)c(Cl)c1 Cc1cc(C(=O)NC23CC(NC(c4cnn(C(C)(C)C)c4)=O)(C2)C3)n[nH]1 N1(C(c2cccc(C)c2)=O)CCC2CCN(C(c3nc(C(C)C)cs3)=O)CC2C1 c1(C(=O)OCC)c(C)[nH]c(C)c1S(=O)(=O)NC1CC(CC(C)(C)C)C1 C1(CNC(C2(CC)CC2(F)F)=O)CC2CCC1N2C(=O)Cn1cncn1 C12(NC(C(C=CC)O)=O)CCCC1CN(C(C1(C)CCCC1)=O)C2 CC1(C)CN(C(c2cc(CNC(=O)C(C)(C)O)on2)=O)CCO1 CC(N=c1cccc(S(=O)(=O)NC2CC3CCC(C2)S3)[nH]1)c1cn(C)cn1 C(C)(CO)(C(=O)NCc1ccsc1C(N1CCC(N2CCCC2)C1)=O)OC CC(C)(CNC(=O)CC#N)Cn1cc(CC(O)CO)nn1.N12CCCC1C2=O C1(NC(c2sc3nccnc3c2N)=O)CN(C(=O)C(F)(F)CO)Cc2ccnn2C1 Cc1cnc(C(=O)NC(CC2CCOCC2)C(=O)NCCCCC(C)C)c(C)c1 N1(C(c2n(CC#C)ccc2)=O)CC(NC(C2(F)CC=CC2)=O)C(N=[N+]=[N-])C1 C(CC(C)C)(C(=O)NC1CC2CCC1(C(=O)NCc1ncccc1Cl)C2)OC c1(CC(C)NC(=O)NC(C)Cc2nc[nH]n2)ccc(O)cc1 c1(OC)c(Cl)cc(C(=O)N(C2CN(C(=O)CC(C)C(F)F)C2)C)c2ncccc12 N1(C(C2(C(N)=O)CCC2)=O)CCN(C(c2cnsn2)=O)C(c2cccc(F)c2)C1 Cc1oc(C#N)cc1C(N1CCC(C(=O)N(C2CCOC2)C)C12CC2)=O c1(C(=O)N)cncc2nc(O)[nH]c12.C1(C(C)C)CC(C(=O)N(CC)C2CC2)C1 N1(C(C(C)n2ccnc2)=O)CC23CCCC2(C1)CN(C(c1nnn(C)c1N)=O)C3 C(=O)(C(C#N)CNC1CC1)N(C(=O)CN1CCC(n2cnnn2)C1)C c1(CC(C)N(CCOCC)CC)cccc(C)c1C Cc1cc(C(=O)NC2CCC(C(=O)Nc3c(C)csc3C)CC2)c2cc[nH]c2c1 Cc1cc(=NC(=O)C(=O)N(C2CN(C(c3sncc3C)=O)CC23CC3)C)[nH]o1 C1(C(=O)NC2CCCN(C(c3ccc(C)c(C)c3)=O)CC2)CC2CCCCN2C1 N1(C(C(C(c2c(OC)cccc2)NC)C)=O)CC2(C1)CN(C=O)C2.C(C)(C)C c1(C(=O)NCC2C(C)CCCN2C(=O)C=C2CCC2)nn(C)c2ccccc12 C(=O)(CC1=CCOCC1)NCCN1CCC(NC(CN(C(C)=O)C)=O)CC1 CC(C(=O)N(C)CC1CCCN(C(c2ccc(C(F)(F)F)nc2)=O)C1)C(F)F c1(OC)ccc(Cl)c(C(N2CCC(C)C2CNC(C2(O)CCC2)=O)=O)n1 c1(C(=O)NC(CC)CN(C)C(C2CCOC2C2CC2)=O)ccnc2c1nnn2C C(CNC(C1CC(F)(F)C1)=O)(C(C)(C)C)NC(c1ccc(OC)s1)=O c1(CC)cc(CC(=O)NC2CC(C)CC2O)n(C)n1.c1(C(=O)N)cnc(C)[nH]1 N1(C(C(CC(C)C)F)=O)CCN(C(C2COCCC2(F)F)=O)C2(CCC2)C1 C1(CC(=O)N)CCC2(CC1)CC2.CC(C)(C(=O)NCC1CC1)c1cc[nH]n1 C(=O)(C1CCc2nnc(C)n21)NCCC1N(C(CC(C(=O)OC)(C)C)=O)CCC1 C(c1ccccn1)=C.C1(C(=O)OCC)CCC(CNC(N2CC(O)C2)=O)CC1 C(=O)(C1CCCc2nnn(C)c21)N1CCC(NC(c2cccc(C#C)c2C)=O)C1 C(=O)(C(C)C(C)NC(c1cncnc1)=O)NC(C)Cc1cn[nH]c1 C1(CNC(COCC=C)=O)CC(NC(=O)COCCCC)C1(C)C C1(C(=O)NC2CCN(C(C3SCCCS3)=O)C2)(OC)CCOC1 C(=O)(C(=O)N=c1ccn(Cc2ccc3c(c2)CCC3)[nH]1)NCCC(C)CO C1(C(=O)NCc2cn(C)nn2)CC(F)(F)CN1C(C1COC(=O)N1)=O N1(C(CNS(NC)(=O)=O)=O)CCC(NC(c2cncs2)=O)C(C)C1 C1(NC(C2CC(N=[N+]=[N-])C2)=O)CN(C(=O)C(=O)NCC(F)F)CC2(CC2)C1 C(=O)(C#CC1CC1)NCC(C1CCCN1C(c1cccc(CCO)c1)=O)(C)C C1(CNC(C2C(C=C)CC2)=O)CCCCN1C(c1cnn(CC2CC2)c1)=O C1(NC(Cc2c(OC)cccc2)=O)CC12CCC(NC(C1CSCCS1)=O)CC2 C(=O)(N1CCC(C(=O)Nc2cccc(C3CC3)c2)O1)c1c(CC)ncnc1 CCCCC(CC(=O)NCC(C1CC(C)(C)C1)O)NC(C1CN(C)CCN1C)=O c1(C(N2CCCC(CCNC(c3c[nH]nc3Cl)=O)C2)=O)n[nH]c2c1CCOC2 CC1N(C(=O)CNC(C2CCCC(O)C2)=O)CCCC12CCC2 N1(C(CC#C)=O)CC2CN(C(c3ccc(F)nc3C)=O)CC2C1 C1(C(=O)NCCCOC=C)CC(OC)CN1C(=O)CC1(C)CCOC1 N1(C(C(CC)Sc2ccccc2)=O)CC(CNC(=O)C(F)=C(C)C)C(O)C1 C1(C(=O)NC2(CC=C)CCC2)CCN(C(C2(CC)CCCCC2)=O)CC1O c1(C(=O)OC)ccc(C(=O)NC(C)CN2CCN(C(=O)C=CSC)CC2)cc1Cl n1(CC(N2CCC(COC)(NC(C3C(C)C3C)=O)C2)=O)cccc(C)c1=O Cn1nnc2c1CCC(C(N1CC(C)(NC(=O)C(O)CC[S+](C)C)C1)=O)C2 C(=O)(C1=COCC1)OC.C1(C2CCC2)C(=O)N1C1(c2ccsc2)CC1 N1(C(C2C3CN(C4CCC5CCCC45)CC23)=O)CCc2cccc(Br)c2C1 C=CC1OCCC1N(C(=O)CCCF)CC.c1(C(=O)NCC)cccs1 C(=O)(N=c1[nH][nH]c(C)c1Cl)C1N(C(Cc2c(OC)ccc(Cl)c2)=O)CCSC1 C=CC(C)(C)C(=O)NCC1CC(NC(c2cccc(C(F)(F)F)c2)=O)C1 C(=O)(C1=CCCCCC1)N1CC(O)(C(C)NC(=O)C(C)Cc2cnco2)C1 C1(CNC(c2cccc(=O)o2)=O)C2CC1N(C(C1C3CCC(F)C13)=O)C2 Cc1c[nH]nc1C(=O)N(C(C)CCNC(c1c[nH]nc1-c1ccc(Cl)s1)=O)C c1(CC)cc(=O)oc2cc(NC(c3c(C)noc3C)c3nnnn3CC)ccc12 c1(SC)cccc(C(=O)NCC(C)CNC(=O)C2=NNC(=O)C2)c1Cl N1(C(c2n(C)ncc2C#N)=O)CCN(C(C2CCC3(CCC3)O2)=O)CC(O)C1 C1(C(=O)NC(C)(C)CCF)CCC(O)CN1C(=O)CCCNC(N)=O N1(C(c2ccc(CC)[nH]2)=O)CCC(C(N2CCCC(C)CC2)=O)C12CC2 C1(OCC)(OCC)CC(C)(C(=O)NCCC)C1.C1(C=O)CN(C)C1.N C(=O)(Nn1cnc2ccccc12)C1CCCN(C(C2CN(C(C)=O)C2)=O)CC1 c1(C(N2CCC(CN(C(c3c(CCC)nco3)=O)C)C2)=O)ccc(=O)oc1 Cc1ccc(C(N2CC(CN(C(=O)C(C)CF)C)C3(CC3)C2)=O)c(Cl)c1 c1(OC)ccc(C=CC(=O)N)cc1.C(=O)(CC(C)(C)O)N(C(C)C1CC1)C N1(C(c2nnc(O)nc2O)=O)CCN(c2ccnc(CO)n2)CC(O)C1 c1(C(=O)NCC2(C)CCC(NC(c3cnco3)=O)C2)c2c(c[nH]c1=N)CCC2 C1(C(N(C)CC2CCCN2C(=O)C=CC2CCC2)=O)Cc2nncn2C1 c1(OC)cccc2c(C(=O)Nc3cc(Cl)cc(C)c3N)csc12 c1(C(N(CCNC(=O)C=Cc2nc[nH]n2)CC)=O)ccnc(O)c1.CCO.O C1(C(N2C(CN(C(c3c(C(C)C)nns3)=O)C)CCC2)=O)CC1C1CC1C N1(C(COCC)=O)CC2CCOCC2(NC(c2cn(C)nc2Br)=O)C1 CCCC(CCCNC(=O)COC)NC(c1ccnc(N(C)C)c1)=O Cc1cc(C(=O)NC(C2CCN(C(C3CC3(C)C)=O)C2)(C)C)c(N)c(Cl)c1 C1(CNC(c2n(CCCOC)nnn2)c2ncoc2C(F)F)(C)CCOCC1 C=CCC(CC(F)F)C(=O)NC1(C)CC(F)(F)C1.C(=O)CC(C)(C)CC(F)F.N C1(CC)CC(CC(=O)NCC2(C)CC2)C1.C1(C=O)CC1.C(N)=O.N C=C=CCCC(=O)N(C(C)CN(C(=O)C=COc1ccc(OC)cc1)C)C c1(N2CCC(n3cc(C)nn3)CC2)cccc(S(=O)(=O)N(CCC(C)C)C)n1 C1(NC(C(CSC)(C)C)=O)CN(C(=O)Cc2ccoc2C)CC1C1CC1 CC1CN(C(C2CC3CC3N2C(=O)C(=O)C2CCCC2)=O)CCN1CCO C1(NC(c2n(C)ncc2Br)=O)CC12CCN(C(c1cc(O)ccc1O)=O)CC2 C(CCCCCO)(c1nnnn1CC1CCCO1)SCC.c1(C2CC2)ccccc1N C1(NC(c2c(C)ncs2)=O)CC2CC(NC(C3CCCC34OCCO4)=O)CC2C1 C=CCCCC(C(=O)N1CCN(CC#CC)CC1)NC(=O)CCN1CCCCC1 C1(C(=O)NCC(C)(C)Cn2cc(CC)nn2)CCC2(CCOC2)O1.C(N)=O.N c1(C(C(=O)NC(COCC=C)C(=O)O)(C)C)ccc(F)cc1F C(=O)(C1CCc2ccccc21)NCC(C)(C)OCC=O.C(C)(C)CC(F)(F)F.N c1(CC)cccc(CNC(c2c(Cl)n[nH]c2C)c2nnnn2C2CCOC2)c1 c1(OC)cc(C)cc(C(=O)NCCCNC(C23CCCCC2C3)=O)c1O c1(C(N2CC(CNC(C(C)SCC)=O)(OC)C2)=O)ccccc1.C1CC1 CC1(C)C(CC(=O)NCC2CCOCC2)CCN1C(c1n[nH]c2c1COC2)=O c1(C(N2CC(C)C(CNC(C3CC(=O)CO3)=O)CC2)=O)cnn2c1OCCC2 C(=O)(CCCOC)NC(c1n(CC)ncn1)C.C1(CC(C)=O)(C=O)CC1.N C=CC1CCCN(C(C2CCC(CNC(=O)CC3CCCC3)C2)=O)C1 C(=O)(C(O)CC(N)=O)NCCC(CC)(C)NC(c1cc(C2CCC2)[nH]n1)=O c1(C(=O)NNC(=O)c2csc(C(F)F)n2)cn2ncccc2n1 N1(C(C2CC(SC)C2)=O)CCC2CCC(NC(=O)Cc3ccc(F)cc3)C1C2 Cc1csc(=NCC(=O)NC2CCCCN(C(C3(O)CCC3)=O)C2)[nH]1 CC(O)C(C(=O)NC1CCC(NC(=O)CNC=O)CC1)N(C)C Cc1ccc(CC(=O)N(C2CC(NC(C3CC4C=CC3O4)=O)C2)C)cc1Cl c1(C(N(C2CC3CN(C(C(CCC)OC)=O)C2C3)C)=O)ccc(F)cc1SC c1(C(=O)NC2CC(NC(CC(C)N(C)C)=O)C2)cc(F)cc2nn[nH]c12 N1(C(C2(COC)CC2)=O)CC(NC(=O)Cc2cc(C)no2)C(C2CC2)C1 n1(CCOC)cc(C(=O)NC2CCC(NC(=O)CCCCSC)CC2)ccc1=O C1(C)CCCN(C(=O)C(O)C(F)(F)F)C1.c1(C(=O)OC)ccc(C(=O)N)cn1 C#CCC(CC(F)F)C(=O)NCC(CC(=O)NCCC(C)CCC)C1CCC1 C#CCC(C)(C(=O)N1CCC=CC1COC)NC(=O)C=C(C)COC Cc1ccc(C(=O)NC(C2CCCC2)CNC(C2CCCCC2(F)F)=O)c(Cl)c1 Cc1cccc2c(C(=O)NCC34CCCC(CN3C(=O)CNC=O)C4)c[nH]c12 Cc1cncn1CC(=O)NCC1CCCN1C(=O)CN(C)C(c1cccs1)=O C1(NC(CCc2cc(C)[nH]n2)=O)CCCN(C(c2cc(C)c(C)o2)=O)CC1 c1(OC)ccc([N+](=O)[O-])cc1C(N1CCC(F)C1)=O.c1(C(=O)N)cc(O)nn1C c1(NC(C2CC3(C2)CN(Cc2cccnc2Br)C3)=O)cc(Cl)c([N+](=O)[O-])cc1Cl C(C(=O)NC(C1CCCCC1)C)(C(C)(C)C)OC.C(=O)(CCCCCN(C)C)N N1(CC(=O)NCC2(c3cc(Br)ccn3)CC2)CCc2ccccc2C1=O C(C(C)(O)C(F)F)NC(CCN(C(C(C=CC)O)=O)C)=O Cc1nn(C)nc1C(=O)NCC1COC(CNC(c2sccc2C)=O)C1 Cn1cc(C(=O)NC(C)CO)nc1C(F)F.c1(C=O)cccc(C2(C)CC2)c1 C1(c2c(C(=O)NC3CC(C)(C)C3)c[nH]n2)CCCCN1C(=O)CNC(N)=O c1(NC(C(CC(C)C)NC(=O)OC)=O)cc2cc(F)ccc2cn1 Cc1c(F)ccc(C(N2CC(CNC(=O)CCC3CCC3)C3CC23)=O)c1N C1(C)(NC(CC=C=C)=O)CCCN(C(c2c(C)noc2C(F)(F)Cl)=O)C1 N1(C(C(C)(C)C)=O)CCN(CCNC(C2(C3CCCO3)CC2)=O)CC1 c1(C(=O)NC2CCC(NC(CN3CC(CC)C3)=O)C2)ccc(C#N)n1C C1(CNC(C(C)O)=O)CC12CCN(C(=O)Cc1sc(O)nc1O)CC2 C1(CNC(=O)Cc2cnns2)CC(C(=O)NCc2ccccc2O)=NO1 c1(C(C(=O)NCc2cn(CC(N3CCCC3)=O)nn2)(F)F)ccc(F)cc1 c1(C=O)cnn2ccc(O)nc12.c1(C(=O)NC2CC(C)C2)cnc(C2CC2)o1 N1(C(CC(CNC(=O)C#CC2CCC2)O)=O)CCC(O)C12CCC2 c1(CNC(=O)OC(C)(C)C)nccc(=NCC2CCCC(F)(F)C2)[nH]1 c1(C(N2CCC(NC(C3(COC)CC3)=O)C(F)C2)=O)cn2cccc(Cl)c2n1 c1(C(=O)NCCCCNC(C2(SC)CC2)=O)cnc(C(C)(C)CF)o1 Cc1nscc1C=CC(N1CCCC(N(C(=O)CC2CCC(C)(C)C2)C)C1)=O CCCCC(CC)CC(=O)NC1CC(C)(NC(c2cnc3scc(C)n23)=O)C1 Cc1cc(C=CC(N2CCOC(C(C)NC(=O)C(C)(C)N(C)C)C2)=O)ccc1F c1(-n2ncc(C(=O)N)c2)ncccc1C(F)(F)C(F)(F)F.CS(=O)C1(C)CC1 c1(C(N2CCN(CC(C)NC(C3(C)CC=CC3)=O)CC2)=O)ccnc2ccsc12 c1(COC)c(CNCC(C)(C)Cc2cccc(Br)c2)noc1C1CC1 c1(NC(C2N(C(c3ccc(C)c(F)c3)=O)CCSC2)=O)ncnc2sc(Br)cc12 N1(C(C(=O)O)C2CC2)CCN(C2CCOC2)CC1 c1(OC)ncnc(C)c1C(=O)NCC=CC.c1(C=O)cc(C(F)F)ncn1 c1(OC)ccc2c(c1)CCC2C(=O)NC(C)(C)CN(C(=O)C(F)C(C)C)C N#Cc1ccc(C(N2CCCCC2C(=O)NCC(CO)C2CCC2)=O)cc1 C(C(C)(C)C(=O)NC)SC.C1(O)CCN(C(c2n[nH]c(C(C)(C)C)n2)=O)C1 c1(OC)cc(F)c(Cl)cc1C(=O)NCC1CCC1NC(=O)CCS(C)=O CCCCCCCNC(=O)CCC1(C)CN(C(C2(C)CCCO2)=O)C1 c1(C2(C(=O)NCC(CC)NC(c3ccnc(C)c3N)=O)CC2)cccc(F)c1F c1cc(C)cc(C)c1.C#CC1CC1C(=O)NCCC1CCCC1.C(=O)(CC)N n1(C(CC)C)ncc(C(=O)Nc2ccccc2-c2nn[nH]n2)c1C N1(C(C(=O)NC)=O)CC(C)N(C(=O)C(c2cnc(Br)c(C)c2)(F)F)CC1C C1(N(C(C)=O)CC(C)C)CCN(C(=O)CC(C)(C)F)CC1.C(C=O)NC(C)=O C(=O)(C(CN(C)C)CC)NCC(C(=O)N(CC#C)CCO)C c1(CCNC(=O)CCc2ccc[nH]2)c[nH]c(=NCc2cnc(Cl)cc2F)s1 C1(C)(NC(C(CC2CCC2)NC(c2c(C)con2)=O)=O)CCCCCC1 Cc1c(C(=O)NC2CC(NCc3ccc(O)c(Br)c3)C2)cccc1F c1(OCC(C(C)C(=O)NC2(C)CCSCC2)=O)cccc(Br)c1F C1(NC(C2(C)CC=CCO2)=O)COC2CN(C(c3cc(Cl)ns3)=O)CC12 N1(C(C(C2CCCCC2)OC)=O)CC2(CCC2NC(=O)Cc2cc(C)sc2C)C1 C=C(C)C1CCC(C)=CC1CC(=O)NC1CC1.c1(C=O)ccc(C)c(C)c1O.N C1(NC(c2ncc(Br)cn2)=O)(CF)CCN(C(c2cnn[nH]2)=O)C1 c1(C(=O)Nc2cccc(-c3c(C)ccc(C#N)c3)n2)ccc2cccc(F)c2n1 N1(C(c2n(C(C)C)cnc2)=O)CC2(C(=O)N)CC1CO2.C(C)C=O.C(C)(C)C Cc1c(F)cc(C(N2CCC2C(=O)Nc2ncc(C(F)(F)F)cc2Cl)=O)cc1Br C1(C(N2CCOCC(NC(C3C(OC)CCC3)=O)C2)=O)CC2CCC(C1)C2O n1(CCC#C)c(N2CCOC(C)C2)nnc1-c1ccc(Cl)nc1 C1(OC)CN(C(=O)C(COC)OC)CC1NC(=O)CC1CCCO1 C1(NC(C(C(CC)C)N(C(=O)CCc2ccncn2)C)=O)CCC(C2CC2)CC1 N1(C(CCN(CC)CC)=O)CCN(C(=O)C(C#N)C2CC2)CC2(CC2)C1 C1(C(N2CCC(c3cc[nH]n3)C2)=O)(CNC(CSC)=O)CCOCC1 C(=O)(C(C)CC(C)(C)C)NC(CCC)CCCNC(c1ccc(F)cc1CC)=O c1(C(=O)NC2CC(C)(NC(C3CC4CC4C3)=O)C2)cc([N+](=O)[O-])cnc1N Cc1ccccc1CCc1nc(-c2ccnn2C)nn1CC1CCCO1 C=CCC(C(=O)N1CCC(NC(c2c(NC(C)=O)cccc2F)=O)CC1)C(C)C CC1CN(C(=O)Cc2ccsn2)CC1CNC(=O)C(O)(C1CC1)C1CC1 N1(C(C(N2CC(C)C2)C)=O)CCC(C)(C)C(C(=O)NCc2ccc(O)nn2)C1 C(=O)(CCC(C)NC(c1ccncc1F)=O)NCCCC(C)C C#CC1CCN(C(=O)C(CCSC)NC(=O)CCc2nc(=N)[nH][nH]2)CC1 N1(C(COCCOCC)=O)CCC2(C1)CN(C(=O)C(c1cncn1C)O)C2.C C=CCC(C)(CC)C(=O)N1CC(NC(c2cccc([N+](=O)[O-])c2)=O)C(F)C1 Cc1ncnc(C)c1CC(=O)NC1CCN(C(=O)CCc2cnc[nH]2)C1(C)C N1(C(c2cn(C)nc2Cl)=O)Cc2ccnn2CC(NC(=O)C(CO)C(C)(C)C)C1 c1(C(=O)NCC2CCN(C(C(F)OC)=O)C2)cc(C2CC2)nnc1O Cc1cncc(CC(=O)NCC(C)N(C)C(C2CC2c2ccccc2)=O)c1 CC(C)CC(O)CC(=O)NC(C)C(=O)Nc1cnccc1C1CC1 C(CC(C(=O)N)OC)OC.CC(CC1CCCC1)C(=O)N(C(C(N)=O)C1CC1)C Cc1c(C(=O)NCCC2CCC2)cnc2ccnn12.C1(CC(=O)N)CCC(C)O1 C1(C(N2CCC(C)C2CNC(c2cc(O)no2)=O)=O)CC(C2CCOCC2)=NO1 c1(C(C)=O)cc(C(=O)NC2CCCC2)c(C)o1.c1(C=O)sccc1C(C)C.C C1(NC(c2ccc(C)c(N)c2)=O)CC2CCC1N(C(=O)CCOCC(C)C)C2 c1(NC(C2CC(NC(c3[nH]cc(C)c3C)=O)C2)=O)cc(F)cc(I)c1 C1(C(N(C)Cc2ncnn2C)=O)CCOCCN1C(c1cnnn1C)=O C1(CCC)CN(C(c2nc(CC)oc2C)=O)CC1NC(=O)Cc1ccc(C)cc1 c1(NC(=O)NC)ccc(Cl)c(C(=O)N)c1.C1CCCC1.C1CC1.C(=O)C Cc1ccc(CCC(=O)NC2CCC(NC(c3ccc(Cl)o3)=O)C2)cc1C c1(C(=O)NC2C(CC)CN(C(=O)C(F)(F)C3CC3)CC2)snc2ccccc12 C(c1ccc2c(c1)CCO2)=CC(=O)NCCCCOC.C(=O)(C#CC1CCC1)N Brc1cncc2c(N3CCCN(C4COC4)CC3)ccnc12 c1(C(=O)NC2C(F)CCN(C(C3(OCC)CCOC3)=O)C2)nccc2ccsc12 CCCCCC(C(=O)NCC1CCCN(C(=O)COCP(C)(C)=O)C1)C(C)C C1(CNC(C=Cc2c(C)ncs2)=O)CN(C)CCN1C(=O)C(F)C1CCC1 C1(CCN(C(c2scc(C=O)c2)=O)C)CCCCN1C(C1CCC(=O)N1)=O.C C1(C(N2CCC(N(C(=O)CCC3CCC3)C)C2)=O)CCCc2ccccc2C1 c1(C=O)ccc(CC(N)=O)cc1.c1(C(C)OC)nc(C(=O)NC2CCC2)cs1 N1(C(CSCC#C)=O)CC(NC(c2cnc[nH]2)=O)CC12CCCC2 c1(C(=O)NCC23N(C(c4c(C)coc4)=O)CCC2CC3)ccc2oc(S)nc2c1 C1(CNC(CC(C)NC(c2c(C)ccn2C)=O)=O)CC(=O)N(C)C1=O C1(C(=O)NCCCOCCCC)(OC)CCN(C(=O)CCOC)C1 c1(C(N(C2CCN(C(=O)Cn3cccc3)C2)C)=O)ccnc(OC2CCCC2)c1 C(C(=O)N)(C1C(CC)C1)NC(=O)OC(C)(C)C.C(CN=[N+]=[N-])C1CC1 c1(C(=O)NCC2(O)CC(NC(CC(C)CF)=O)C2)cccc2ncccc12 c1(C(N2CC(C)C(C)C2)=O)cc(=NS(C)(=O)=O)cc[nH]1.c1(C(=O)N)scnc1Cl N1(C(CCC2C(C)C2)=O)CCOC2(C1)CN(C(C1CCC(F)(F)C1)=O)C2 C=CCC(CNC(C1CCCCCCC1)=O)C(=O)Nc1cccc(O)c1 C1(F)(C=O)C2CCCCC12.c1(C(N(CCC)CC)=O)cnc(C)nc1C(C)C Cc1cc(O)ccc1CC(=O)NCCC(C)NC(C1CC(C)N(C)C1)=O C(c1c[nH]c(=N)c(C)c1)=CC(N1CCCC1)=O.C(C(=O)N)(C1CCOC1)OC N1(CC)CCC(C(=O)NCC(=O)NCCc2cc(O)ncn2)CC1.C1CC1.C C1(COC)(COC)CCCN1C(C1CC1)=O.c1ncsc1C=O.C1CC1 C(=O)(C1=CCN(C(=O)C(O)C2CCCC2)CC1)N(C(C)C(N)=O)C N1(C(CCCCNC(C(C)OCOC)=O)=O)CCc2sccc2C1 c1(C(=O)N=c2cc[nH]cc2O)cc(C2=CCC(N3CCOCC3)CC2)[nH]n1 N1(C(C)C)CC(C(=O)NCCNC(c2cccs2)=O)CC1=O.c1ccccc1.C c1cn(C2CCN(C(=O)C=CCn3cncn3)C2)nn1.C(C=O)SCC=C.N C(=O)(N1CC2COCC2O1)C1CN(C(=O)OC(C)(C)C)C2(C1)CCC2 C1(CNC(CCOC)=O)CC(F)(CNC(C2CCC2c2nc[nH]n2)=O)C1 Cc1cc(O)n2ncc(C(=O)NC3(C4CCN(C(C5(C)CC5C)=O)C4)CC3)c2n1 N1(C(c2cc(CC)n(C)n2)=O)CC(C)CN(C(=O)CNS(C)(=O)=O)C(C)C1 Cc1nc(CCC(=O)NC2CCC(CNC(C3CCC(F)CC3)=O)CC2)oc1C c1(C(=O)NCC(CC)NC(C2(NC(C)=O)CCCCC2)=O)cnc(S)nc1 N1(C(C(C)N(C)C)=O)CC2CCC1C1CN(C(C3OCC4COCCC34)=O)CC21 C(=O)(CCCC(C)(C)C)N(CC(C)(C)CNC(=O)CC(F)F)C c1(OC)ncc(Nc2cc(N3CC4CSCC4C3)ncn2)cc1C#N Cc1nc(-c2ccco2)cc(=NCC(C)NC(C2CC3CCC2CC3)=O)[nH]1 CC(C)(C)CCC(F)C(=O)NCCOC1CCN(C(C2COCCO2)=O)C1 C#CCC(C)(C(=O)NCCNC1CC1)NC(C1CCOC1C1CC1)=O.C CC1(C(=O)NCCCc2ccncc2)CCCN1C(C1CC(=O)CS1)=O Cc1nnc(CC(=O)NC2(C)CC(NC(=O)Cc3c[nH]nc3O)C2)o1 Cc1c(C(=O)NC(C2CCCN2C(=O)OC(C)(C)C)C)ccc2ccccc12 N1(C(C2CN(C(C)=O)C2)=O)CCCCC1C1CC1.c1(C(=O)N)c[nH]cc(F)c1=O c1(C(=O)NC2(C)CCN(C(C(C)NC(C)=O)=O)C2)ccc2c(Br)cnn2c1 N1(C(c2cc(C)n(-c3ccccc3F)n2)=O)CC2CC1CC2NC(C1(Br)CC1)=O C(=O)(CCCCC(=O)NC1(COC)CN(C(c2nscc2Br)=O)C1)NC C12(C(N(CCC(N)=O)C)=O)CC(CN1C(=O)C(C1CCOCC1)F)C2 C1(C)(CC)CC(NC(C2CC=CC2)=O)CN1C(=O)CNC(=O)OC CCCC(C)CC(=O)NC(C1CCCN1C(=O)Cn1cnc([N+](=O)[O-])c1)(C)C c1(NC)nc(C)ccc1C(=O)NCC1CN(C(c2scnc2Cl)=O)CC1C N1(C(c2ncn(C)c2)=O)CCN(C(C2(c3ccccc3)COC2)=O)CC1CO C(=O)(CCCN=c1nccc[nH]1)N1CC(O)(C(C)NC(c2c(C)snc2)=O)C1 C(=O)(CCCC(F)(F)CO)NC(CNC(C1C(CC)CCC1)=O)(C)C c1(C(=O)N)cnc(C(N)=O)cn1.c1(CC)nnsc1C(=O)NCC1CC1 C(=O)(C1=NNC(=O)C1)N(C1CCC(NC(C2CC2c2ccccc2Cl)=O)CC1)C c1(C(=O)NC(C)CCCCNC(c2ccc(C#N)[nH]2)=O)cc(F)cc2ccoc12 C1(C(N2CCC(N(C(c3c(C)cc(F)s3)=O)CCO)C2)=O)CC2(CCCC2)CO1 C(=O)(C(N=[N+]=[N-])C(C)C)N1C(CNC(c2ccc(C)c(C)c2)=O)C(C)CC1 CCC(CC)C(C)C(=O)NC1CC(CC(=O)NC2CCCC2)C1 c1(C(=O)NC(C)(C)C(=O)NC2CN3CCCC2C3)cc2occc2[nH]1 c1(OCC)c(F)c(C(=O)NC2CN(C(C3CCSCC3)=O)CC2C)cc(F)c1F c1(C(=O)NCCCN(C(=O)CC2(O)CCCOC2)CC)nc(Cl)sc1C c1(C(=O)NC2CC(CCNC(=O)CCSc3ccccc3)C2)cccnc1O CC(C)CCC(=O)C(=O)N1CCCC1(C)C(=O)NCc1cnn(C)c1O c1(C(=O)NC(CNC(C2ON=C(C(C)C)C2)=O)C(C)C)sc2ncccc2c1N C1(CC(=O)NC(C(=O)NC(C(=O)NC)C)Cn2cncn2)CCCC2CC12 C(=O)(CC(C)C(=O)OC)NC(CNC(C(CCC)OC)=O)(CC)CC S(=O)(=O)(c1cc(C(C)C)c(C)cc1C)NC(C(=O)OC)C1CC1 N1(C(CN2CC(=O)N(C)C2=O)=O)CCN(C(C2CCCC2)=O)CC(C)(F)C1 C#Cc1cncc(C(N2CCC(NC(c3ocnc3C3CC3)=O)C(F)C2)=O)c1 N1(C(C2CC(CCNC(Cc3cnc(C)s3)=O)C2)=O)CCS(=O)C(C)C1 N1(C(Cc2c(C)nc(C)s2)=O)CCCC(C)(NC(=O)CCc2c(C)n[nH]c2C)C1 N1(C(C(C)(C)NC(CCCC2C(C)C2)=O)=O)CCC(O)CC(C)C1 c1(CC)cc(C(=O)NC(c2cn(C)nn2)C(=O)NCC2CCSC2)c(C)o1 CCC(C)C(C)C(=O)NCCOC1CCN(C(c2cnn(C)c2OC)=O)CC1 C(C)(C)(CCC(=O)NCCn1ccc(C(=O)N)c1)N(C)C.C1CC(C)(C)CO1 N(C1CCCCc2cnn(C)c21)C(=O)NC1C(COC)C1 CC(C)S(=O)(=O)C(C)C(=O)N1CCC(NC(c2c(F)cncc2Br)=O)C1 N1(C(CCCOC)=O)CCN(C(=O)Cc2cc(F)ccc2Cl)C(C)CC1C C1(C)(CNC(c2nc(OC)oc2)=O)CCCN(C(C2(C)CCC2)=O)C1 N1(C(C2CCCS2)=O)CCN(C(=O)C2=CCCCC2)C(C(F)F)C1 c1(C(=O)NC2CCC(NC(c3ccn(C)c3)=O)CC2)ccnc2c1ncn2C N1(C(CNC(=O)OC)=O)CCCCC1CC(=O)NCCN1CCCOCC1 Cc1[nH]nc(C(=O)NCC(C)CN(C)C(C2CCN(C)C2C)=O)c1C CCC(C)C(=O)C(=O)N1CC(NC(c2ccc(F)cc2C)=O)C(C)(C)C1 C1(C(=O)NC(C(CO)NC(C2(NC(C)=O)CCCC2)=O)C)CCC=CCCC1 c1(C(N2CC3(C(NC(CC(C)OC)=O)CCC3)C2)=O)ccc([N+](=O)[O-])cc1O N1(C(C(c2ccco2)NC(CCCCCN(C)C)=O)=O)CC2(CCC(=O)NC2)C1 c1(C(N(C2CCN(C(c3ccnc(C(C)C)n3)=O)C2)C)=O)cc(O)cc(Cl)c1 C=CCC(CC=C)C(=O)NCC=CCC(=O)NC1(CC=C)CCC1 c1(C(N2CC(NC(C(C)CC3CCC3)=O)C(F)C2)=O)c(O)nnc2c1CCCC2 C(CCCCCNC(C1CN(C)CCO1)=O)N(C(CNC(CCC)=O)=O)C N1(C(Cc2c(C)ocn2)=O)CCC(CN(C)C(C2(C)CC2F)=O)CC1 N#Cc1cccc(C2CC2C(N2CC(C#N)C2)=O)c1 C1(CC(=O)NCC(C)N(C(=O)C=CC(=O)N(C)C)C)CN2CCN1CC2 c1(NC(c2nc(O)sc2-c2ccccc2)=O)ccc(C(=O)NCCCO)cc1 c1(OC)cc(C(N2CCCCC(NC(=O)CC3CC=CCN3C)C2)=O)c(Cl)cn1 c1(C(c2n(CC=C)nnn2)NCCC(F)(F)F)cn(-c2cccc(C)c2)nc1C C(C(=O)N(C1CC1C1CC1)C)(C(C)C)NC(CCc1cnc(C)o1)=O C1(CN(C(CC)=O)C)CCN(N2CCC(Cc3cccc(F)c3)CC2)CC1 N1(C(C(CC)c2ccccc2)=O)CC2=C(C1)CN(C(=O)CN1CCCC1C)C2 N1(C(C(C)(C)c2ccncc2)=O)C2CCC1CC(CNC(c1cscc1Cl)=O)C2 N1(C(C2(C)CCCS2)=O)C2CCC1C(NC(c1ccc(CO)c(Cl)c1)=O)C2 C1(C(=O)NC(CC(C)C)(C)CNC(c2ccco2)=O)CCn2ccnc2C1 c1(CNCC2CCCN(C(=O)Nc3cccc(OC)c3)C2)cc2cccnc2[nH]1 C(=O)(C(C#N)C(C)(C)C)NCCn1cc(C(N2CCC(SC)C2)=O)nc1 c1(C(N2CCC(CN(C)C(C3CNC(=O)N3C)=O)C2)=O)ccc2c(ccn2C)c1 C=CCC(CC(F)F)C(=O)NCCC(C)N(C)C(c1cc(OC)cc(F)c1)=O c1(OC)cc(C(N2CCN(C(=O)CCS(C)=O)C3CCC23)=O)cc([N+](=O)[O-])c1 c1(C(N2CC3C(NC(c4c(OC)cc(C)cn4)=O)C3C2)=O)ccnc2c1CCO2 N1(C(CSc2cccc(C)c2)=O)CC2CC(NC(c3c(C)ncnc3C)=O)C1C2 Cc1cc(C(=O)NCC(C2CCOC2)NC(=O)Cn2cnnc2)c(C)o1 c1(N(C(C(C2CCN(C(CCCCSC)=O)C2)C)=O)C)ccc(C)cc1C O=C1CN(CCC(=O)NC2CC(NC(C3(Cl)CC3(F)F)=O)C(O)C2)CCN1 CC1=C(C(=O)NCC2CCCC2NC(=O)CCc2ccsc2)C(C)(C)CCC1 c1(C(=O)NC2CCC(C)N(C(C3COC(C)(C)O3)=O)C2)ccc2oc(=O)oc2c1 C1(NC(c2cn(C)nn2)=O)CN(C(c2cn(C)nc2C2CCCC2)=O)CC12CC2 CC1CC(NC(c2ccccc2SC(F)F)=O)CN(C(=O)CC2CCCOC2)C1 C1(CC(=O)NC)CC2(CCC2)CO1.N1(C(C)=O)CCC(O)C1.C(=O)OCC C(=O)(C(O)CC(N)=O)NCC(CC(C)C)NC(c1ccnc(OC)n1)=O c1(CNC(N(CCC=C)CC)=O)sc(C)cc1Br C12(CCNC(CCN(C(=O)C=COCC)CC#C)=O)CC(CCO1)C2 c1(C(=O)Nc2ccc(-c3cccc(NC4CC4)c3)s2)cc(O)c(O)c(O)c1 CC1C(NC(=O)C=CCO)C(C)CCN1C(C1(F)CCOC1)=O Cc1cc(C(c2nnnn2CCN2CCOC(C)(C)C2)NC2CCCO2)ccc1Cl C(CCC(O)C(=O)NC(c1nnc(C)o1)C)NC(C(C(C)C)NC(C)=O)=O N1(C(C2N(C(CCC#CC)=O)CC=CC2)=O)Cc2nc(C)sc2C1 C1(CC(=O)N(CCCCCCC)C)CC2(C1)CN(C(=O)CCC(C)OC)C2 C12(C(=O)OC)CN(Cc3cnn(CC4CCC4)c3)CC1S(=O)(=O)CCO2 c1(NC(C2(C)CN(C(C3C(CC)CCC3)=O)C2)=O)ccc(C(N)=O)nc1C C(CC(=O)N1CCN(C(C2CC=CC(O)C2)=O)CC1C1CC1)(C(F)(F)F)OC C(=O)(CCC(O)C(C)(C)C)NCC1CCCN(C(C2(OC)CCCC2)=O)C1 N1(C(C2(C(C)C)CC2)=O)CCCC1C1CCCN1C(=O)CSc1ccccc1F C(=O)(C1=CCOCC1)N1CCC(C)(C(=O)NCCc2cc(C)ncc2)C1 C1(C)(C(=O)NC2CCCC(NC(C(C3CCCCC3)OC)=O)C2)COC(=O)OC1 C=CC(C)(C)C(=O)NC(COC)CC(=O)NC(C)C(=O)N1CCCC1 c1(CC)cccc(CC)c1CN=C(NC1CC1)NCC(C)(O)c1ccco1 Cc1cccc(C)c1CC(N1CCC(N(C(=O)CC2(C)CC2)C)C(C)C1)=O C1(NC(C2CCC(C)(C)C2)=O)CCC12CN(C(=O)CCSC)C2.c1ccccc1 c1(OC)ccc(OS(=O)(=O)CC2CC=C(C)CC2)c(C)c1 C1(C(C(=O)NC(CC)C)N(C2CCC2(C)C)C)C2CC=CCC12.CCN(C)C Cc1[nH]c(C)c(C(=O)NCC(C)C(F)C(=O)NC(CO)CCO)c1C c1(C(=O)NC(C(=O)N(C)Cc2nc(C)sc2)CCF)cc(O)cc(F)c1 c1(C(=O)NC(C2CCN(C(C3(CC=C)COC3)=O)C2)C)cccc2[nH]nc(O)c12 O(S(=O)(=O)c1cnc(C2CC2)o1)c1ccc(C(C)C)c(C(F)(F)F)c1 C(C(=O)NCCCCCO)(C(C)(C)C)NC(c1n(COC)ncc1)=O c1(COC)nc(=N)[nH]cc1C=O.c1(C=O)ccc(C(C)(C)C)[nH]1.CCCC.N C(CC(O)CNC(c1cc(Cl)ns1)=O)NC(CCC1C(C)C1)=O CC1C(NC(C2CC3CCC3C2)=O)CCN1C(C1CCN(CC2CC2)CC1)=O C(C1CCCC1)=CC=O.C(=O)(CN(C)C(C1CC1)=O)O.C(C)=O.CC C1(C)(CN(C(C(C)n2ccnn2)=O)C)CCCC1NC(C1(F)CC=CC1)=O N1(C(C2CCC(CC)CC2)=O)CC2CCC(N=c3[nH]nc(C#N)s3)CC2C1 CN(C)S(=O)(=O)N1CCC(C(=O)NC2CCCN(C(=O)CC3CCOC3)C2)C1 c1(N2CC(OC)C(NC(C3(C)CC3)=O)CC2)ncnc2c1CC(=O)N2 c1(C(=O)NCC(CNC(C(CC)C(F)(F)F)=O)O)c[nH]c2cc(F)c(F)cc12 c1(OC)ccc(C(N2CCCC2C(=O)Nc2cc(O)nn2C)=O)cc1I C1(C(N2C(CN(C(C=CC(C)C)=O)C)CCC2)=O)CCCCC1O C(=O)C1CCCc2c[nH]nc21.C1CC2(C1)CC2.C(=O)(C(F)(F)F)NCC(=O)N CCC(CCC(=O)NC1CCN(CC)C1=O)NC(=O)CC1CCCN(C)C1 c1(C(N2C(CNC(=O)CCc3nccs3)CC(OC)C2)=O)cc2cccnn2c1 c1(NC(C(C2CCCN(C(C3CNC(=O)C3)=O)C2)C)=O)ccc(F)cc1F C(C(=O)O)C(C)(C)C.C12CCCN(C1)C(=O)CC1CCN(C1)C2=O.CC(=O)N CN1C(=O)CCCC1C(=O)NCCCn1cc(COCCN(C)C)nn1 Cc1ccc(F)c(C(N2CCC(F)(CNC(=O)CC3CCCO3)C2)=O)c1Br N1(Cc2ncc(Br)s2)CCC2(CC1)CCN(CC)CC2.c1(CC)nn(C)cc1C=O CC12CC(C1)C1(CN(C(c3ncccn3)=O)C1)O2.C1(C)(CC=O)CC1(F)Cl.N c1(NC(C2(N(C)C(c3cncs3)=O)CC(CO)C2)=O)cncc(N(C)C)c1 C(CC(C)C(C)C)NC(c1c(C)sc(O)n1)=O.c1(C=O)ccc(C(N)=O)cn1.N C1(CN(C(CC(C)c2ccco2)=O)C)CCCCN1C(c1cc[n+]([O-])cc1)=O C1(NC(c2ccccc2)=O)CCN(C(c2ccc(=O)n(CCO)c2)=O)C12CCC2 c1(CN2CCC(N(c3ncnn4cc(Br)cc34)C)C2)cc([N+](=O)[O-])c(Cl)cc1F CCC(F)(F)C(=O)NCCC(C(C)C)NC(=O)CC1(COC)CCOCC1 C(C)(C)(CS(N)(=O)=O)c1cn(Cc2cn(-c3ccc(C)cc3)nc2C)nn1 CC1(C(N2CC3CC3(NC(=O)CCc3cc(Br)cs3)C2)=O)CCNC1=O c1(C(=O)NCC(CN(C(CCC2C(C)C2)=O)C)O)cc(F)c(N)cc1F c1(C(=O)NC(C2CCN(C(CCCC#C)=O)CC2)C)ccc(C(F)(F)F)c(O)c1 C(C(C)(O)CC(=O)NC1(C(=O)NCCC2(O)CCCCC2)CCC1)OC C1(C(=O)NCC2(NC(C=C(C)C)=O)CCCCC2)CC2(CCO1)CC2 N1(C(C(c2cn(C)nc2)=O)=O)CCN(C(C2CCC3CCC2O3)=O)C(CO)C1 c1(N2C(C(=O)NC3C(C)C3C)C(C)CC2)ncnc2c(Br)cccc12 n1(CC)nnc2c(NC(c3ccc(Br)cc3)CCO)ncnc12 C1(CNS(=O)(=O)CCC2CCCO2)COc2cscc2O1 Cc1sc2nc(Br)cn2c1CNCC12CC(CO1)C2 N(C1c2ccccc2CC1NC(=O)CCCS(N)(=O)=O)C(C1(C)CC1(F)F)=O C=C(CNC(=O)C(F)C1CCOC1)CCNC(=O)CSCC C(c1cc(F)cc(F)c1)=CC(=O)N.C1CC2(C1)CN(C(c1ccnc(Cl)c1)=O)C2 C1(C(N2CCC(NC(Cc3cc(C)nn3C)=O)C2C)=O)CC2CCC(C1)C2 N1(C(c2c(C=C)cnn2C)=O)CCOCC(F)(CNC(=O)CC)C1.C1CCC1.O c1(C(N(CCC)CC)=O)cc(N)c(O)c(F)c1.C1(C(=O)N)SC2C=CC1CC2 N1(C(c2c(C)nco2)=O)CC2CCCC(CNC(=O)CC(C)CC(C)(C)C)C2C1 N1(C(c2c(C(C)C)occ2)=O)CC(NC(C2(C)CNC(=O)C2)=O)CC(C)(C)C1 C1(CNC(CCSCCC)=O)CN(C(C2COCCN2CC)=O)CCN1C c1(C(=O)NC2CN(C(CC=C)=O)C2)[nH]c2c(c1C)C(=O)CCC2 N1(Cc2n(CCC)nnn2)Cc2ccccc2CC1CNC(=O)CCC1CC1 N1(C(C2(N=[N+]=[N-])CC2)=O)CC2C(Nc3cc(C(=O)OC)ncn3)C2C1 c1(N2CC=C(C)C2)nc(=NCC2(CC#N)CCC2)[nH]c2c1CC(C)CC2 N1(C(c2ncc(OC)nc2)=O)CC(CC=O)C2(CC2)C1.C1(O)CCC(C)(C)C1.N CC1(C)CC1(C#N)C(=O)Nc1ccc(CN2C(=O)CCC2=O)cc1 C(C)(C)(CC(=O)N1CC(C)(C(=O)NC)C1)NC(C(C)OC)=O C1(CNC(c2cn(C(C)(C)C)nn2)=O)C2CN(C(c3cncc(Cl)c3)=O)CC12 c1(C(C)C)cccc(C(N2CC3CC2C3NC(c2ccn(C)c2)=O)=O)c1F N(C1COc2cc(F)ccc21)C(c1ncc(Cl)cc1Cl)c1n(C)nnn1 CC(CC(C)(C)C)C(=O)N1CC(NC(=O)Cc2c(Br)cnn2C)C(O)C1 c1(OC)ccccc1C(c1ccccc1)NC(=O)N.c1cc(C(C)(C)C)n[nH]1 C(=O)(C1=C(Cl)CCCC1)NC(C)C(C)(C)NC(c1cccc(CF)c1)=O c1(C(=O)OC)nc(NC(C2CCN(Cc3ccnc(Cl)c3C)C2)=O)ccc1Br c1(C(=O)NC2COC3CN(C(c4csc(O)n4)=O)CC23)cc2n(n1)CCCC2 c1(N2CCC(N(C(CC(C=C)(C)C)=O)CCC)C2)nc2cc(CC)ccc2n1C C1(C(N2CCCCC2)=O)CC2(C1)CC2(F)F.c1(CC(=O)NC)ccc(Cl)nc1.C N1(C(=O)CCCn2cc(COC3COC3)nn2)CCCC2(COC2)C1 C(=O)(C#CC1CCCC1)NCC(CCOC)NC(=O)Cc1nc(C)sc1Cl C1(NC(CC(CCC)C)=O)CCCN(C(=O)C(F)(F)C(C)O)CCC1 C1(NC(C2(C(C)C)CC2)=O)CC(NC(C23CCC(C2)C3)=O)C(O)C1 CC1(CNC(C2CCCCC2)=O)CCN(C(c2cnc(-n3cccn3)cn2)=O)C1 S(=O)(=O)(c1ccc(C(=O)O)cc1)N1C(C(=O)Nc2scc(C#N)n2)CC(F)C1 c1(C(=O)NC(CC)CNC(=O)COc2cc(C)on2)c(C)nsc1N C(=O)(C1=C(Cl)CCCC1)NCC(CC(C)C)NC(=O)CCc1c(F)cccc1Cl N#Cc1cc(F)ccc1C(N1CCCC(CNC(=O)CSc2ccncc2)C1)=O C(=O)(C(C)(C)C1CCC1)NC1CC(NC(C(F)=CC)=O)C1 C(=O)(CCCC(C)(C)NC(C1CC12CC2)=O)NCc1c(C)ocn1 C(C(=O)NNC(=O)CCC1CCCN1)(C1CCCC1)OC C1(C(=O)NC(CNC(C2C(C=C)C2)=O)C2CCC2)CCOCC1 N1(C(C2NCCN(C(c3ccc(O)cn3)=O)C2)=O)CCCN(CC(F)(F)F)CC1 C1(CC(=O)N(C(C)CN(C(=O)C=CC2CCCC2)C)C)CCS(=O)(=O)C1 N1(C(c2c(C)ncnc2)=O)CCOC(C(N2CCCC(C)(CO)C2)=O)CC1 c1(C(=O)NC(CNC(=O)CCc2cocn2)C2CC2)cccnc1O c1(NCCN(C)C(c2cnc(Cc3ccccc3)s2)=O)ccc([N+](=O)[O-])cc1 C=CC1OCCC1C(=O)N(CCC)C1CC1.C(=O)(CCCCN(C)C(C)=O)N CC(CC(=O)N(C(C)CNC(=O)Cn1[nH]cnc1=N)C)n1cccn1 c1(C(N2CCC(N(c3ccncn3)C)C2)=O)c(C2CCC2)cnn1C C#Cc1ccccc1CC(N1CC(NC(=O)CC2CC23CC3)C(O)C1)=O C1(OC)CC(C)N(C(c2cc(Br)n[nH]2)=O)C1.C1(CC(=O)N)COC(C)(C)C1 C1(S(C)(=O)=O)(C(N(CCCn2cc(-c3c(C(C)C)n[nH]c3)nn2)C)=O)CCC1 Cc1cc(NC(c2c(C)ncn2C)=O)ccc1NC(C1C2CC3C(C2)C13)=O C1(CNC(c2ccccc2-c2cccc(F)c2)=O)CC2CCC1CC2 c1(-c2n(C)ncc2)cnc(Cl)c(C(=O)Nc2ccc(F)nc2F)c1 Cc1cc(Cl)c(Cl)cc1C(=O)NC1CC1CNC(=O)CCC(C)(C)C N1(C(c2cc(C)oc2C)=O)CC2CCC(CNC(=O)C(C)(C)C(N)=O)C2C1 Cc1ccc(Cl)c(F)c1C(N1CC2CCCC2C1)=O.C(=O)(C1=CCS(=O)(=O)C1)N Cc1[nH]nc2ncc(C(=O)N(C(C)CCNC(C3CCOC(=O)CC3)=O)C)cc12 CC(C)CC(CN)NC(C1CCCC(C(F)(F)F)O1)=O CCC(C)C(N)C(=O)N(c1ccccc1)CCCCOCCCOC c1(C(N2CCC(C(=O)Nc3c(CC)cc(Cl)cc3)C2)=O)cccc2c1OCCO2 C1(CC)CN(C(=O)C=C(C)C)CCC1NC(=O)C(c1ccncc1)C N1(c2nnc(COC)n2CCCCCSC)CCOC(C2CC2)CC1 Cc1ccc(C)n1CC(=O)NCC1CC(O)C1.C(=O)C(C)Cc1cnc[nH]1.C CCC(C)CCCCC(=O)NCCC1CN(C(=O)C(C(C)C)NC(N)=O)C1 c1(N2CCCC(CNC(CC=C=C)=O)C2)nc2c(cc1C(=O)OCC)COCC2 C(=O)(C(C)S(=O)(=O)C(C)C)N(C)Cc1cn(-c2ccc(C)c(Cl)c2)nn1 c1(C(N(C2CCN(C(Cc3nnc(C)o3)=O)C2)C)=O)ccc(C#N)c(Cl)c1 C1(C(N2CCCC(CNC(c3cc[n+]([O-])cc3)=O)CC2)=O)CC2CSCC(C1)C2 [SH](=O)(=O)CCCC.C(C)(C)(CO)NCCC1C(=O)C(C)N1C.C(=O)C.N C1(C(=O)NCCC(C)NC(=O)C=Cc2ccco2)CC12CCCCC2 C12(NC(Cc3scc(C)c3)=O)CCCC1CN(C(c1cc(C3CC3)[nH]n1)=O)C2 N1(C(=O)CSc2nncs2)CCC(CO)(NC(C2(Br)CC2)=O)C1 C(=O)(C1CCc2ccc(C)cc21)NC1(CNC(C=CC)=O)CCC1 c1(NC(=O)CC2(NS(=O)(=O)CCCCO)CCC2)ccnc(F)c1F N1(C(CCn2ccc(C)n2)=O)CCC2(CCCN2C(=O)C2CCc3nccn32)C1 N1(C(c2cc(C#C)cc(F)c2)=O)C2CCCC1CN(C(C1CC1(C)Br)=O)C2 C1(C(=O)NC(Cc2c(C)non2)C(=O)O)CCc2cnn(C(C)C)c2C1 Cc1nc2cc(C(N3CC(NC(C4CCN(C)C4)=O)C(F)C3)=O)ccc2o1 c1(CC(C)NC(C2(Sc3ccccc3)CC2)C)cnccn1 C1(C(N2CCCC(OC3CC3)C2)=O)C2CCC(C2)N1C(n1cncn1)=O C(=O)(CCCN=[N+]=[N-])NC1(C)CC(NC(C(C(C)C)Sc2ccccc2)=O)C1 O=S(=O)(COc1ccccc1-n1cccc1)c1cc(F)ccc1F c1(NC(C2C3CC2N(C(c2cnn4cccnc24)=O)C3)=O)c(Cl)cc(Br)cc1Br c1(C(=O)NC(CNC(c2c(CC(C)C)nc(C)s2)=O)CO)ccc(Cl)cc1Cl c1(C(=O)NCC2N(C(CC3ON=C(C)C3)=O)CCC2)c(C)ncn(C)c1=O c1(C(N(C)CC2CN(C(C3=C(C)CCC3)=O)CC23CC3)=O)cncc2[nH]ccc12 N1(C(CC(C)F)=O)CCC2(CCCN(C(c3ccc(P(C)(C)=O)o3)=O)C2)C1 C1(NC2CC(n3ccnn3)C2)CCCCCO1 Cc1cc(C)c(C(=O)N(CC(C)NC(=O)C=C2CCC2)C)c(=O)o1 CCC(CC)CC(F)C(=O)N1CCC(C(C)C(=O)NC2CC(C3CCCC3)C2)C1 C(c1ccccc1Cl)=CC(=O)NCC(CNC(C1(C)CC=CCC1)=O)OC c1(C(N2C(C=C)CCC2)=O)n[nH]c2c1CN(C(C1CC1(C)CC)=O)C2 C=CC(C)(O)C(=O)NC1CN(C(=O)C(C)NC(=O)CC2C=CCC2)C1 N1(C(C(=O)NCC)=O)CCCCC1C1CCCN(C(C23CC(CCO2)C3)=O)C1 N1(C(CC2C=NN(C)C2=O)=O)C2CCC(C2)C1C(=O)Nc1cncc(C#N)c1 c1(C(N2CC(OCC#C)C2)=O)conc1CC.c1(C=O)cc(C(N)=O)[nH]n1 C(C(O)C(=O)NC1(C)CC(NC(=O)COC(C)=O)C1)SC c1(CNC(C(CCC)CC)=O)ccc2c(c1)CN(C(c1cc(C#N)[nH]c1C)=O)C2 C1(CNC(c2cc(CC)no2)=O)CN(C(=O)C(C)S(N)(=O)=O)CCCO1 c1(OC)cncc(C(=O)N(C2CN(C(=O)Cc3nocc3C)CC23CC3)C)c1C c1(C(N2CCC3(CN(C(C=C(C)C(F)F)=O)C3)C2)=O)cc2c(C)ccc(Cl)c2[nH]1 CN1CC2CC2(NC(C2COC(CNC(=O)CC3CSC3)C2)=O)C1 c1(C(NOCC(=O)N(C2CCN(C)C2)CCC)=O)cc(O)cc(F)c1 C#CCC(C)(C)C(=O)NCC1CCN(C(=O)CCc2cnn(C)c2C)C1 c1(CC)cccnc1C(N1CC(O)(CC)C1)=O.C1(C(=O)N)CCCN1C(C)C c1(C(=O)NCC2CCCC(NC(c3nccc(C)c3)=O)C2)cc(O)cc(Cl)c1Cl c1(C(N(C(CC)C)C)=O)sc2[nH]cnc(=O)c2c1C.C1(C(=O)N)(COC)COC1 N1(C(c2nnc(C)s2)=O)CC2(C1)CN(C(c1cnn(-c3nccs3)c1)=O)CCO2 Cc1cccc(OCC(N2CC(NC(=O)C(C)(C)F)C(O)C2)=O)c1 C1(CNC(c2c(-c3cn(C)nc3)cco2)=O)CCN(C(C2CC2Cl)=O)CC1 Cc1cc(F)ccc1C(=O)NCC12CCC(CC1)N2C(=O)CC(F)(F)F C1(NC(COCCSC)=O)C=CC(CNC(=O)CC23CCCC2C3)C1 C1(C)CCCN(C(c2cc(C(F)F)ncn2)=O)C1.N1(CC)CCCC1C(=O)N.C c1(NC(=O)NC2CCC23CC3)ccc(Cl)c(S(=O)(=O)NC2CCCC2)c1 c1(C(C)=O)ncc(C(N2CC(CO)(NC(=O)C(C)CN(C)C)C2)=O)s1 N1(C(C(C)c2cc[nH]n2)=O)CCOC(C(=O)NCCC2CC(O)C2)CC1 C1(NC(C=CCOC)=O)COC2(C)CC1C2.N1(CC=O)CCC(O)CC1.N C1(CC)CC(C(=O)NC2CCC(C(=O)NOCC(N)=O)C2)CCO1 C(=O)(CCCCCC#N)N1C(C(=O)NCC2CC(C)(O)C2)CCCCC1 C1(C(=O)OC(C)(C)C)C(N)C2CCCC12.C(C(F)(F)F)=CC(C)N CCC(C(=O)N1CCCC1CN(C(=O)Cc1csc(C2CCOCC2)n1)C)SC c1(OC)cc(SC)ccc1C(=O)N(C)CCNC(C1CC1CF)=O N1(C(c2onc(C)c2C)=O)CCC2(CCN(C(C3CCCC(F)(F)C3)=O)C2)C1 C1(C(=O)OCC)CCCC2CN(C(=O)Cc3cccnc3OC(C)(C)C)CC12 C(c1cccc(O)c1)=CC(=O)N(C1CN(C(C)=O)C1)C C1(C)(CNC(C2N(C)C(C(N)=O)CC2)=O)CCCN(C(=O)CC2CC2)C1 c1(C(=O)NCC2(NC(CC(COC)(C)O)=O)CC2)cc2c(s1)CCOC2 C(CC(C)C)(C(=O)N1CCC(O)(CNC(=O)C(N)=O)CC1)OC N1(C(CC(=C)C)=O)CCN(C(=O)CCOCCC)CC2CCCCC12 C1(C(N(C2CCN(C)C2)C)=O)CCN(C(=O)CC2CCOC2=O)C1C1CC1 C1(NC(C2CC(Cl)(Cl)C2)=O)CCCN(C(C2(S(C)(=O)=O)CC2)=O)C1.CC C1COC2(C1)CN(C(c1ncc[nH]1)=O)C2.Cc1ccc(C)c(COCC(=O)N)c1 CC1CCN(C(=O)Cc2cccc(Cl)n2)CCC1NC1CCCC1C C1(OC)CCC2(CCN(C(=O)CC3(C)COCCN(C(=O)CC4CC4)C3)C2)C1 N1(CC)N=C(C(=O)N(CC(C)C)C)CCC1=O.C1(C(=O)N)CC(=C2CC2)C1 C1(O)(CNC(CC(C)(C)OC)=O)CCCN(C(=O)CN2CC=CC2)C1 C1(O)(C(N2CC(CC=C)(NC(=O)C(CO)NC(N)=O)C2)=O)CCCCC1 c1(CC(N2CC(F)(CNC(C(C)CC(F)F)=O)C2)=O)ccc(F)cc1[N+](=O)[O-] N1(C(c2ccc(SC)o2)=O)CCC2CCN(C(c3c[nH]c(C)c(Cl)c3=O)=O)C2C1 c1(CC)ccc(C)cc1C(N1CC(N2CCN(C(C3CC3C3CC3)=O)CC2)C1)=O CC1CC(NC(=O)CCc2cc(Cl)cs2)CN(C(=O)CN2CCSCC2)C1 C(c1ccccc1Cl)=CCSCC(C(=O)NC(C)(C)C)NC(C)=O C1(C(=O)NCC(C)(C)NC(=O)COc2ccccn2)CCCNS1(=O)=O c1(OC)ccc(C)c(C(=O)NCC2(CC)CC2)c1.C(=O)C.CC(C)C.N CC1CN(C(c2cncc(-c3ccccc3)c2)=O)CCN1C(C1CNC(=O)C1)=O c1(OC)ccc(C(=O)NCCC2CCN(C(C3CCCS3)=O)C2)c2ccccc12 C#Cc1cc(C(=O)NC2CN(C(=O)CCC(C)C)CC2S(C)(=O)=O)cc(Cl)c1 N1(CC(=O)NCC2CCCCNC2)CCNC(=O)C1 N1(C(C(CCC)O)=O)CC(NC(c2ccnc(OC(C)(C)C)c2)=O)CC(C)(C)C1 n1(CC(=O)NC2C(NC(C(F)OC)=O)CCC2)cnc2ccccc12 CC(C(=O)NC1CN(C(C2C3CCCCCC23)=O)CC1(C)C)C(C)(F)F N1(C(C(C)OCC#C)=O)CCCCC1CCNC(C1(C2CC2)CCC1)=O CCCC(C(=O)NCC1(NC(=O)Cc2ccc(C)s2)CC1)C(C)C Cc1nc2c(N3CC=CC(NC(c4csc5c4CCC(C)C5)=O)C3)ncnc2s1 c1(OC)ccc(F)c(C(N2CCC=C(C(=O)NCc3ccc[nH]3)C2)=O)c1OC c1(C(N(CCN2CCN(C(C(CC)(C)O)=O)CC2)C)=O)ccc(Br)c(O)n1 c1(OC)ccc2c(c1C(N1CC3CC3C1)=O)CCC2.C(=O)(C(O)P(C)(C)=O)N C1(C(=O)NCC(C(C)C)(C)O)COC2(C1)CN(C(=O)CCC(C)(C)C#N)C2 C(=O)(C1CCCc2ncccc21)NCCCCCNC(c1cnn(CC)c1C)=O O=C1OC2CC(C(=O)NC3(C(F)(F)F)CC(F)(F)C3)CC2O1 C1(C(N2CC3C(NC(c4cncc(F)c4)=O)C3C2)=O)CCc2nccn2C1 CC1(NC(=O)CC2COCCOC2)CCN(C(=O)C(O)CN2CCOCC2)CC1 CCCC(CC(=O)NC1CCCC1C(=O)NC)NC(C1CN2CCN1CC2)=O c1(C(N2CC(C(C)NC(=O)CCSCC(N)=O)OCC2)=O)ccn2nncc2c1 c1(OC)cc(C(=O)NCC(n2cc(CCC(=O)O)nn2)C)c(F)cc1Br C1(OC)(OC)CCOCC1CCNC(=O)NC1CC2C(C1)C2(F)F N1(C(C2C(CCC)C2)=O)CCC(C(=O)NCCn2cc(CO)nn2)C1 N1(C(C(=Cc2ccco2)C)=O)CC(C(=O)NC(C)CC(N)=O)CC12CCC2 N1(C(C=CCC)=O)CC2(C)CN(C(c3c(F)ccc(F)c3Cl)=O)CC2(C)C1 C1(C(=O)NC(c2cncnc2)C)CN(C(=O)CC2OCCC2C)CCO1 CCC1C(=O)Nc2ccc(C=O)cc21.CCCN(C(=O)CC1(C(F)F)CC1)C.N c1(C(=O)NC(CC)CNC(C2(O)CC2(C)C)=O)cc(O)nc(Cl)c1 CC1CC(C(=O)N)CC(C)(C)C1.C(C)(C)C.C12(CC=O)CC(C1)C2.CC c1(C(=O)NC(C2CCCN(C(Cc3ncc(C)o3)=O)C2)C)nc(C)c(C)[nH]c1=O C1(NC(=O)CN2CCC(O)CC2)CCC12CN(C(=O)C(c1ccccc1)F)C2 C1(CNC(=O)C(C2(O)CN(C(C3(F)CC=CC3)=O)C2)F)COC(=O)N1 Cc1nnccc1C(=O)NCC1CN(C(=O)C(=O)NC(C)C)CC1O C#CCC(C(=O)N(C)CC)C1CC1.c1(C2(C(N(CC)C)=O)CC2)ccncc1.O N1(C(C2C(C)OCCO2)=O)CCC2(CC2)CC1C(=O)NCc1ncco1 C(=O)(CCCCN1CCCC1)NC(C1CCN(C(C(C)NC(CC)=O)=O)C1)(C)C Cc1cc(F)c(CO)cc1Br.C12CON(C(=O)Cn3cc(cn3)-c3cn1nn3)C2 C1(C(=O)NC2(CNC(CCc3c(C)noc3)=O)CCC2)C2CCCOC12 Cc1cccc(C(N2CCC(NC(C3CCCN3S(C)(=O)=O)=O)C(C)C2)=O)c1O CC(C)C(C)(O)C(=O)N(C)CCN1CCN(C(C2(C)CCCOC2)=O)CC1 c1(CNC(C2N(C(CCC3N(C)CCC3)=O)CCC2)=O)cccnc1Cl C1(CNC(CC2(CC=C)CCCC2)=O)CC(O)CN1C(=O)CCN1CCCC1 C1(NC(c2cccnc2)=O)CC2CC(C1)N(C(c1cc(O)cc(Cl)c1)=O)C2 N1CCN(C)C(=O)C1.c1(OCC)cncc(-c2ccc(C(=O)CC3CC3)cn2)c1 N1CCC(C2CCN(C(=O)CCCS(C)(=O)=O)CC2)C1.Cc1sccc1.c1ccccc1.CC c1(C(N2CC3(CN(C(=O)CCC4CCCCO4)C3)C2)=O)ccc(O)cc1[N+](=O)[O-] c1(C(=O)NCC2N(C(C(C=C)(F)F)=O)CCC2)ccc(C)c(S(C)(=O)=O)c1 CC(C)(C)CC(O)CC(=O)N1CCC2CCN(C(c3cscc3Cl)=O)CC12 CC1CCN(C(=O)CCc2nc(O)n[nH]2)C1C(=O)N(C)Cc1cnn(C)c1 C1(C(=O)Nc2c(SC)ccnc2)CCN(C(c2ccc([N+](=O)[O-])[nH]2)=O)CCO1 Cc1n[nH]c(C)c1C(C)C(=O)NCCc1ccccc1.C1(O)(C(=O)N)CCCC1 C1(C(=O)NC2CCSC2)(CC)CCCN(C(=O)CC2CSC2)C1 C(c1ccccc1)=CC(N1C(C(C)(C)CNC(c2cncnc2)=O)CCC1)=O Cc1c(C(=O)NC2CCCCCN(C(=O)C(C)C3CC3)C2)sc2ncnc(N)c12 C1(C(C(=O)NCC(=O)N(C)C)C#N)CC1C1CCCCC1 Cc1nc(NCC(C)S(C)=O)cc(=NCc2ccccc2OC(C)(C)C)[nH]1 CC1CC1(C#N)C(=O)NCC1(CC(N2CC(C)(O)C2)=O)CC1 Cc1ccc(F)c(C(=O)NC(CNC(c2c(C)ccn2C)=O)C2CC2)c1F c1(C(C)C)ncc(C(=O)NCCCN(C(=O)C(C#N)C2CC2)C)n1C N1(C(C=COCC)=O)CCN(C(=O)CC2CCC23CCC3)CC1C1CCC1 C(N=c1cccc(S(=O)(=O)NCCSc2nccn2C)[nH]1)c1c(C)csc1 C(=O)(C(C)CS(C)(=O)=O)NCCCN(C(C(CC)C(=O)OC)=O)C(C)C C1(C(N2CCC(N(C)C(c3ccc(CO)cc3)=O)C2)=O)CCCCC1(C)C n1(CC)cccc(NC(=O)CCCC2(NC(C3CC(O)C3)=O)CCC2)c1=O N1(C(c2c(CCC)[nH]cc2)=O)CCOCC(C(=O)NC(C)(C)CC(C)(C)C)C1 C1(NC(C2(COC)C=CCN2C(=O)C=CCF)=O)CC2CCC(C1)C2O n1(CCCC)nnnc1C(c1cncn1CCC)NCC1C=CCOC1 N1(C(c2n(CCC)ncc2)C(=O)NC)CCOC(c2cccc(F)c2)C1 N1(C(C(C(C)C)C)=O)CCC2CC1CN(C(c1cc3nn[nH]c3cc1F)=O)C2 C(c1ccc(F)cc1[N+](=O)[O-])=CC(=O)NC1C(NC(CC(CC)C)=O)CCCC1 C1(C(N(C)CC2N(C(Cn3nnc(C)n3)=O)CCOC2)=O)CNC(=O)C(C)(C)C1 O=S1(=O)CCC2CN(S(=O)(=O)c3ccc(C(F)(F)F)cc3Cl)CCN12 c1(OC)ncccc1CN1CC2CC2(C(=O)NCC(N)=O)C1 c1(C(=O)NC(C(C)NC(=O)CNC=O)(C)C)cc2nc(Cl)ccc2o1 C1(C(=O)NC2C(C(=O)NC(c3onc(C)n3)(C)C)CCC2)CCC(C)(C)OC1 c1(C(=O)NC2CC(NC(C(C(C)C)C#N)=O)C2)cnc2onc(C3CC3)c2c1 C1CCN(C(=O)C)C1C(C)C.c1(CC)ccccc1.N1(CC)CCC1C(=O)N C(=O)(CC1=CCCC1)N(C)CC1(O)CN(C(=O)CCC2CCOCC2)C1 N1(C(CCCC2(NC(CC3CC(=C)C3)=O)CCC2)=O)CC(O)C(F)C1 n1(CCC)c(NC(C2C3CCC2(c2cncs2)C3)=O)nc2c1CCOC2 C1(CCC(=O)NC(C)C(F)F)CCCN(C(=O)C=CCN2CCC2)C1 c1(CNC(c2c(CC)n(C)nc2)c2nnnn2C2(C)CC2)cc(Cl)ccc1.O C1(CNC(C2(CC)CN(C(=O)CC3CCCO3)C2)=O)CC2CCCC2C1 C1(SCC)CCC(C(N2CC(NC(c3c(Br)cnn3C)=O)C(C)C2)=O)CC1 CS(=O)C1CCC(NC(=O)NC2CC(c3ccc(F)cc3F)C2)C1 Cc1cc(O)n2ncc(C(=O)NC3CN(C(=O)CC4CCOCC4)C4CC34)c2n1 c1(C(=O)NC2C3CN(C(=O)Nc4c(F)ccc(C)c4)C2C3)cc(Cl)cc(Cl)c1O C1(NC(C(C)CN(C)C)=O)C2CC1CN(C(=O)CC1COCC(C)(C)O1)C2 Cc1ccc(S(=O)(=O)N2CC3(CCN3C(c3ccccc3C3CC3)=O)C2)c(C)c1 C1(O)(C(C)NC(=O)CO)CCN(C(c2n[nH]cc2Br)=O)C1.c1(CC)cccs1 C1(n2cc(CCC(CC)O)nn2)CN(C(c2c[nH]nc2C2CC2)=O)CC1C c1(OC)nc(C(=O)NC2(C)CCOCC2)cc(O)n1.C(=O)(CCCN(C)C)N C=CCC(CC(F)F)NC(C1CC1C(C)NC(C1CC(C(=O)O)C1)=O)=O c1(CC(=O)N(CC(C)NC(C2CC(SC)C2)=O)CC)cccnc1C C=CC1CCCC(c2nnnn2CC2CCOCC2)(NCCCOCOC)C1 C1(C2CCCN(C(c3ccc(N(C)C)cc3)=O)C2)(NC(C2C(C)C2)=O)CC1 C1(C(=O)NCC)CCCN(C(c2cncc(-c3ccccn3)c2)=O)C1 c1(C(=O)NC(CNC(C(C=C)CC)=O)CC)ncc(C)cc1C C=CC(C)(C)C(=O)N1CC(O)(C(F)C(=O)NCC(F)C(C)(C)O)C1 c1(C(=O)NC2C(NC(c3ccc(OC)o3)=O)CCCC2)cc([SH](=O)=O)c[nH]1 CC(C)(CC)C(N)=O.c1(Cc2n(CCSC)nnn2)c(C(C)C)nn(C)c1Cl.N N1(C(c2cc(C)c(CO)cn2)=O)CCC2CN(C(c3csc(C(F)F)c3)=O)C2C1 O(N=Cc1ccc(OC)cc1)CC(=O)NC(C1N(C(C=CCCC)=O)CCC1)C N1(C(C=C2CCC(C)CC2)=O)CCN(C(=O)CC2CC=CCN2C)C2(CCC2)C1 C1(C(=O)NC(c2nccn2C)CC)CC(NC(C2(C#N)CC2)=O)CCO1 c1(C(=O)NCCCN(C(c2cnoc2C(C)C)=O)CC)n[nH]c2c1CCCCC2 N1(C(C2ON=C(C(C)C)C2)=O)CC2CCC1CN2C(=O)C(O)C1CCCC1 N1(C(C(C(=O)NC)(C)C)=O)CCCCCC(NC(C2CC2(Cl)Cl)=O)C1 C1(NC(c2ccc(CS(=O)(=O)c3ccccc3)cc2)=O)CCCC2(CCNCC2)O1 C(=O)(C1=CCC(C)(C)CC1)NCCC1N(C(C2CC3(CC(=C)C3)C2)=O)CCC1 C#CCC(CC(F)F)C(=O)NC1(CCC(=O)NC2CC2(C)C)CCCC1 N1(C(=O)NCC2(c3cccc(C)c3)CCCC2)CCOCC(C)(F)C1 N1(C(C2(C=C)CCC2)=O)CCCC(CCNC(=O)COc2ccc(C)cc2)C1 c1(C(c2n(C(C)C)nnn2)NCCCc2ccccc2F)nc2ncccn2n1 C1(C)(C(N2CCC(C(F)F)(CNC(CC)=O)C2)=O)CCCC1(F)F C1(C)(CNC(C(C)NC(CC)=O)=O)CCCN1C(c1cn(C)cn1)=O C1(C(=O)OC)CC(C)CN(C(C2CC3CC3N2C(c2[nH]cc3c2CCC3)=O)=O)C1 C1(N(C(=O)CC2(n3ccnc3)CCCC2)C)CC2C(N)C2C1 C1(F)(CNC(CCCCCOC)=O)CCCN(C(c2ccncc2)=O)CC1 C1(C(=O)NC2(C)CN(C(C3(CCN4CCCCC4)CC3)=O)C2)CC2(CSC2)C1 C(C(C)C(C)C(=O)N1CCC(C)(CNC(C2(C3CCCO3)CC2)=O)C1)OC c1(CC(=O)N(CCC)CC)ccc(C=O)c(C)c1.C1(C=O)CC(C)CO1.N c1(NC)cncc(C(=O)NC2CN(C(c3ccn(C)c3)=O)C2)n1 C1(O)CCN(C(c2ccccc2C)=O)CC1.C=C(C)C(=O)OCCNC(=O)N N1(C(COCc2ncc(C)o2)=O)CC(NC(c2cccc(C3CC3)n2)=O)CC1C c1(C(N2CC(O)(CC)C2)=O)cc(Cl)cnn1.CC(C(=O)N)OCC1CCCO1 Cc1cc(C(F)(F)F)ncc1C(=O)NC(C)CCNC(c1ccc(O)nc1)=O c1(C(=O)NC(C)(CNC(C2CSCCS2)=O)C2CC2)cnc2cncn2c1 C(=O)(C1c2c[nH]nc2CN1C(C1CCCCCC1)=O)NCC(C(=O)NC)C CCC(C)(C#N)C(=O)N1CC=C(CNC(C2(C)CCN(C)CC2)=O)CC1 C1(NC(C2CN(C(C)C)C(=O)C2)=O)CN(C(=O)CN2CCCC2)CCC12CCC2 c1(N2CC3(C(C=O)C3)C2)nc(C)cc(C#N)n1.c1(C(=O)OCC)ccccc1.N c1(NC(CN2C3(CC(=O)O3)CC2)=O)cc(Br)cc(C(F)(F)F)c1F C1CCN(C(c2coc3c2COC3)=O)C12CC2.CS(=O)(=O)C1(C(=O)NC)CC1 Cc1cc(C(=O)NC(CNC(c2ccc(CF)cc2)=O)C2CCC2)oc1C C(C)(CCCCNC(=O)C=CC(c1ccc(C)cc1)=O)NC(CCC)=O C#Cc1ccc(C(N2CC(CNC(=O)C=Cc3ccc(C)s3)C2)=O)cc1Cl.O c1(C(C2CC2)NC(=O)NCCCc2nnc(C)n2C)ccc(F)c(F)c1 N1(C(c2ccc(C)c(Br)c2C)=O)CCC2C(CCN2C(=O)CC2CCCC2)C1 N1(c2nc(C(=O)OC)c(C)s2)CCC(NC(C2CCS(=O)(=O)N2)=O)C(F)C1 C=C(C)CC(C(=O)NCC1CCCC2(CC2)C1)NC(c1sccc1C)=O CC(C)CC(C)C(=O)N1CCC(NCC(=O)Nc2cccc(Cl)c2Cl)C(C)C1 C1(NC(=O)C=Cc2cc[nH]n2)CN(C(=O)CC2CC23CC3)CC1O C(CC=CC)(C(=O)NOCC(C)(C)O)NC(C(CC#C)C)=O c1(CNCC2CC(NC(=O)OC(C)(C)C)C2)ccc(OC(F)F)cc1Br S(=O)(=O)(c1cc(Cl)cc(Cl)c1)N(c1cnc(C#N)c(C#N)n1)C1C2CC3C(C2)C13 C1(COC)(CNC(C2CCOC2)=O)CCCN1C(=O)Cn1ncc(Cl)c1C Cc1ncccc1C=CC=O.C(C)(C)C.C(S(C)(=O)=O)C1(CC=O)CC1.N N1(C(Cc2c(C)nc(C)nc2O)=O)CC2(CCN(C(=O)C=C3CC3)CC2)CC1C c1(NC(N2CC(C)(C(N3C(C)CCCC3)=O)C2)=O)cc(F)ccc1C(F)(F)F N1(C(C2C3(CC(C)(C)C3)C2)=O)CCC(C2CC2)C1C.C(=O)C(O)C1CCCC1 C=CCC(CC(=O)NCCOCCCO)NC(c1cncn1C)=O Cc1nn(C)cc1C(=O)NC1CCCCC1CNC(=O)CCNC(N)=O Cc1cccc(C(=O)C(=O)NC(C)C(C)NC(=O)C=Cc2ncco2)c1 C#CC1(O)CCCN(C(C2(C)CCCN2C(c2cnn(C=C)c2N)=O)=O)C1 N1(C(CC2(NC(C)=O)CC2)=O)CCC2(CC2)C1.C1(C=O)(C(F)F)CCCO1 c1(C=O)c[nH]c2nc(Cl)ccc12.N1(C(C=CC(CC)=CC)=O)CC(CO)C1.N C1(CC)CC(O)CN1C(=O)C(C)=CCNC(C1CCCC(O)C1)=O C1(C(N2C3CC(C3)C2)=O)CC2(CO1)CC(F)(F)C2.CN1CCOC(C(=O)N)C1.C c1(C(N(C)CC2CCCN(C(C3(F)CC3)=O)C2)=O)cc(F)c2cn[nH]c2c1 c1(C(N2CCC(N(CCC)C(c3coc(O)n3)=O)C2)=O)ccc(OC)c(OC)n1 CC(CS(C)(=O)=O)C(=O)N1CC(NC(=O)CC(P(C)(C)=O)c2ccccc2)C1 [N-]=[N+]=NC1CC(C(=O)NCC2CCC(C(=O)NCCCn3ccnn3)C2)C1 c1(C(=O)NC(C2CCN(C(c3c(CC)noc3)=O)C2)C)nn(C)cc1[N+](=O)[O-] N1(C(C(C)OC)=O)CCN(C(c2oc(Br)cc2C)=O)CC1c1ccnn1C C1(C(N(CCOCC)C)=O)CCC2C(CC1)C2(F)F.c1cc(C)cc(Br)c1O C#Cc1cccc(C(=O)NC2CCN(Cc3cccc(I)c3O)CC2)c1 c1(N2CCC(NC(=NC)NCCC(=O)NC(C)=O)C2)ccc(Cl)c(F)c1 CN=c1ccc(C(=O)NCC2CN(C(=O)CC3CCCS3(=O)=O)C2)c[nH]1 Cc1cc(C(=O)NC2CCCN(C(C3NC(=O)CC3C)=O)C2)ccc1Cl C(=O)(CCCCCC#N)N1CCC(CC)(NC(C2CCCOCC2)=O)CC1 CC(C)(CNC(=NCCc1ccccn1)NCC1CCCC(F)C1)CC(F)F C=CCCCCCCC(=O)N1CCCC2(CCC2NC(c2cc(C)on2)=O)C1 CCCCCCCCCC(=O)NCC1CCCN1C(c1nc(Cl)cs1)=O Cc1cc(C(=O)N(C(C)CNC(=O)Cc2cnsc2)C)c2c(c1)C(C)CCN2 C1(NC(c2c(C(=O)OC)nccc2)=O)CCN(C(=O)CC2CCCCC2)CC1O CCCC(C(F)(F)F)NC(=O)C=CCN(C)C(C1CCCC(C)CC1)=O C1(NC(=O)CCn2cncn2)CC12CC(NC(=O)CN1CCCCC1=O)C2 c1(OC)ccc(CO)cc1C(=O)NCCNC(=O)CC12CC(C1)C2 N1(C(C(C(C)(C)C)O)=O)CCC2(CC1)CC2NC(c1ccc2nc[nH]c2n1)=O C(CC(C(=O)NC1CC=CC1)NC(c1cc(C)c(C)s1)=O)OC N1(CCN(C)C)CCC(N(C)N2CCCC(Cc3ccc(Br)cn3)C2)CC1 N1(C(CC2CCC(C)CC2)=O)CC(NC(=O)COCCF)CC12CCCCC2 CCC(CCC(=O)N(CC(C)C#N)C)NC(=O)C(CC)C(=O)OC N1(S(CCCC)(=O)=O)CCC(NC(c2cncc(C#N)c2)=O)C(F)C1 Cc1csnc1C(N1CC(CC(F)C(=O)NC2CCN(CCF)C2)C1)=O N1(C(C2CCN(C(N(C(C)C)CC)=O)CC2)=O)CCCC2C1CCN2C(=O)CO C12(C(=O)NC(C(=O)NCC=C(C)C)Cc3ccoc3)CCCC1C2(F)F C(CC(O)C(=O)NCCC1(C)CC1)NC(C1C(C(C)=O)C1(C)C)=O c1(C(=O)NCCCN(C(C23CCN(CC2)CC3)=O)CC)cc(Cl)cnc1O N1(C(c2ccc(OC)nc2)=O)CCOC2CN(C(=O)CCn3ccnc3C)CC12 C1(CNC(CN(CCC)C)=O)CN(C)CCN1C(C1CCOC(=O)N1)=O c1(C2C(C(N3CCCC3)=O)C2)ccc(C)cc1.C(C)(C)(C(=O)N)OCC.C CC(C)(C#N)CCC(=O)NCC1(O)CCCN(C(=O)CCCCCF)C1 C1(NC(C=C2CCC(C)CC2)=O)CC(O)CN(C(=O)C(C)CC2CC2)C1 CC1(CNC(=O)Cn2cccnc2=O)CCC(NC(=O)Cc2ccno2)C1 CC1CN(C(=O)C(C2(O)CCCCC2)NC(c2cnc[nH]c2=N)=O)CCS1=O Cc1ccc(NC(=O)CSC)cc1.C(C)C(=O)NCCCNc1cccs1 N1(C(C=CCC)=O)CC(NC(C2CCCCS2)=O)C(C)C1 N1(C(C(n2cc(Cl)cn2)C)=O)CC(CC(=O)N(C)Cc2nnnn2C)CC1(C)C c1(C(C(=O)NCCC)N(C)Cc2cc(C)cc(C)c2)cc(C)nc2ccccc12 C1(c2n(CCOCC)nnn2)(NCc2ccc(Cl)c(C)c2)CCOCC1F c1(NC)c(C(=O)OCC(c2csc(C)n2)=O)cccc1[N+](=O)[O-] N1(C(c2c(C)ncs2)=O)CC2CC1CN(C(C1(c3cccc(F)c3C)CC1)=O)C2 C(C)(C)(CC(=O)N1CC(N(C(=O)C=Cc2ccccc2)CCO)C1)SC CC(C)C(C)(CNC(=O)Cn1cc(Br)cn1)NC(=O)CCc1ccccc1 C12(NC(CSC)=O)CC(C1)N(C(c1nc(C(C)(F)F)cs1)=O)C2 C1(NC(C2N(CC)C(=O)CC2)=O)CC2CN(c3cnc(C#N)cn3)CC2C1 C1(NC(C2N(C)CCC2)=O)CCN(C(=O)Cn2cnc([N+](=O)[O-])n2)CC12CCC2 C1(CNC(=O)Cn2ncc(Br)n2)CC(NC(=O)C2CC2)C12CCC2 N1(C(c2c(OCC)ccs2)=O)C2CCCC1CN(C(=O)CO)C2.c1ncc(C)o1 N1(C(C(C)NC(=O)C2CC2)=O)CC=CC(C(=O)NCC2(F)CC2)C1 N1(C(CC(C(F)F)NC(=O)Cc2cccs2)=O)CCc2cccc(O)c21 S(=O)(=O)(c1cc(Cl)c(Cl)cc1Cl)N1C2CN(C(c3conc3)=O)CC21.COC C1(NC(C(COC(C)C)NC(c2sccc2CO)=O)=O)C=CC(C)(C)CC1 N1(C(c2c(C)n(C)cc2)=O)CCC2(NC(c3cc(F)n[nH]3)=O)CC2C1 Cc1ccc(CC(=O)NC(C)(CNC(=O)COC(F)F)CO)cc1Br C(=O)(CCN(OC)C(=O)C1(F)CCOC1C)N(CC)Cc1cnn(C)c1 N1(C(C2(COCC)CC2)=O)CC2CC1C2.C1(CC=O)CCCC(O)C1.C c1(C(N2CCN(C(c3cnns3)=O)CC2CCO)=O)cc2cc(F)cc(F)c2[nH]1 N1(C(c2c(C)cc(F)cn2)=O)CCC2CN(C(=O)CSc3ccccc3)CC2C1 C1(NC(CCC(C)OC)=O)CCN(C(c2ccc(-c3ccccc3)[nH]2)=O)CC1C C1(C(=O)NCCC2(O)CN(C(CCCCC)=O)C2)CCc2nn(C)cc2C1 N1(C(c2cccc(CC)n2)=O)CC2CN(C(c3cc(C(F)(F)F)nn3C)=O)CC12 C12(C(=O)NC3CCC(OC)C3)CC(CN1C(C1CC(=O)C1(C)C)=O)C2 c1(C=O)cc(F)cc([N+](=O)[O-])c1.c1(COC)ncccn1.C1(C(=O)N)CCC1 N1(C(c2cnc(C)s2)=O)CC2CCC2(NC(c2cc(N(C)C)nc(Cl)c2)=O)C1 C1(C(=O)NCC#CC)CCCN(C(=O)C(C#N)CC)CC1 N1(C(C2(CC#C)CCN(C(=O)C(O)C=C)C2)=O)CC2CC1CS2=O Fc1ccc(-n2nc(-c3ccsc3)nc2C2COCCN2C2CC2)c(C(F)F)c1 C1(NC(c2c(C)nc(C)[nH]2)=O)CCCN(CC2CCOC2)C1C c1(C(N2C(CCNC(C(CC)SC)=O)COCC2)=O)cc(C(C)(C)C)ccc1N c1(C=O)ccc(Br)cc1.C1(COC)CC1C(=O)NCC1(CC)CC1.N N1(C(c2cccc(C)c2Br)=O)CCCC2(CNC(c3cnn[nH]3)=O)CCCC12 N#Cc1ccc(NC(C2CCC3(CC3)N2C(c2ccnc(O)c2)=O)=O)c(O)c1 C1(NC(C2CCC(=C)CC2)=O)CC(F)CN(C(C2CCC2=C)=O)C1 CCC(CCOC)C(=O)NCCOC1CN(C(C2C(F)(F)C23CC3)=O)C1 c1(N2CC(CNC(c3ccc(C#N)cn3)=O)OCC2)ncnc2cc[nH]c12 CC1(C(N2CCCC(CNC(=O)C=Cc3ncc[nH]3)C2)=O)CC(F)(F)C1 C1(NC(CN(C(=O)C(C)C(F)F)CC(C)C)=O)CC2(COCCO2)C1 O=[N+]([O-])c1ccnn1CC1CCN(c2cnccn2)CC1 c1(CCNC(C2CCN2C(=O)CCc2ccc(Br)cc2)=O)c[nH]c2ncccc12 CCC(C)(C)CC(=O)N1CCOC(C(C)NC(=O)CSc2cccc(OC)c2)C1 Cc1ccc2c(c1)C(Nc1cc(Nc3ccccn3)nc(C(F)(F)F)n1)CO2 CCC(C)(C(=O)NC1CCCCCC1NC(=O)CCc1ccc(C)nc1)C(N)=O N1(CC=O)CCCCC1C.n1(CC)nnnc1C.c1(C2C(C=O)C2)cccs1.N N1(C(c2cc(C)[nH]c2C)=O)CCN(C(c2csc(C)c2C)=O)C2CCCCC12 CC1(C)CC(C)CO1.c1(C(=O)N)cnn(CC)c1.n1(C2(C=O)CC2)cnnn1 N1(C(C(C)(C)O)=O)CCN(C(=O)Cc2csc3ccc(Cl)cc23)C2(CCC2)C1 CS(=O)CCC(=O)N1CCOC(CNC(c2ccc(C#N)[nH]2)=O)C1 Cc1cnc(C(=O)NC(C)(C)C(C)NC(=O)C(c2nc(F)ccc2Cl)C)cc1Cl C(=O)(C(C)C(F)(F)F)N1CC(N(C(CCc2cc(C)n(C)n2)=O)C)C(O)C1 C(CCC(C)(C)C(=O)Nc1cccnc1C)NC(c1cc(C)nnc1C)=O N1(C(c2cnc(S)n2C2CC2)=O)CC2CCC(C1)N2C.C1CCS(=O)(=O)CC1 C(=O)(C1=CCc2ccccc21)NC1CC(C)CN(C(c2cn3ccnc3s2)=O)C1 C1(CC(=O)N(CC(C)O)CCNC(=O)C=C(Cl)Cl)CC(=O)NC(=O)C1 Cc1cc(CNC(=O)C(C2CCN(C(=O)C3=CCCC3)CC2)C)cc(C)n1 C1(C(=O)NCC2CCC2)(COC)CCC(=O)N1.C1(C=O)(CCO)CC1 C(C(C)(CO)NC(=O)C(O)CSC)NC(C1(CC)CCC1)=O N1(C(c2cc(-c3cn(C)nc3)[nH]n2)=O)CCOC(C)C1.C1(C=O)CC1C(F)F.N O=C(N=c1nc(Cl)nc2[nH][nH]cc1-2)C1CN(c2ccnc3ccnn23)CCC1O C(=O)(CCCCC(N)=O)N1C(CCC)CN(C(C2COCCO2)=O)CC1 C(=O)(CCC(=O)NN(C)C)N1CC2C(NC(C(C3CC3)OCC)=O)C(CC2)C1 C(=O)(CCCCC(=O)NC)N1C(CNC(C(CC)(CO)OC)=O)CC2CC21 c1(C(N2CCC(CC(=O)NCC(c3cccs3)C)CC2)=O)cncc(C#N)c1 C12(CNC(C(=O)NCC(c3cccc(F)c3)C)=O)CCC(CN)(CC1)OC2 c1(CN(C)C)ccsc1C(=O)NC1CC(C)C1.C(=O)C(F)CC1CCCC1 C12CC(CN1C(=O)CN1CC(C)(C)C1)C2.C1(C)(C=O)CC(C)=NO1.CO C1(C(N(CC(CNC(c2cc(C)nn2C(F)F)=O)O)C)=O)CCC2CC1CO2 C1(OC)CCN(C(=O)C(Cc2cnc[nH]2)NC(C2CCCC2O)=O)CC1 c1(N2CCN(CC(C)(C)NC)CC2)[nH]c(=NC2COCC2OC)nc2scnc12 Cc1csc(CCCC(=O)NC(C)CNC(C2CC2C(F)F)=O)n1 C1(O)(C(C)NC(CCNC(COC)=O)=O)CN(C(=O)C(c2cccnc2)O)C1 c1(OC)ccc2c(c1)OCC(C(=O)NCCN(C(=O)Cc1cc(C)cs1)C)C2 N1(C(C(CSC)C)=O)CC(C(N2CC3(CCC3O)C2)=O)CC(C)(C)C1 c1(SC(F)(F)F)cnc(=NCCn2ncc3ccccc23)[nH]c1 C(=O)(C(CCCCCO)N(CCC(=O)OC)C)NC(CC)C N1(C(CCSc2ccc(C)cc2)=O)CC2(CCCC2NC(c2cnc(C)[nH]2)=O)C1 C(=O)(C(C)C(O)C(C)CC)N(CCC(=O)NC(c1[nH]c(C)nc1C)C)CC#C CCCC(C)CCCC(=O)NCCCCCNC(=O)C(F)CC1CCC1 c1(CC)c(C(N2CCCC2C)=O)cnc2ncnn12.C(=O)C(C)(C)C(F)(F)F.N C(=O)(CC(C)NC(c1ccnn1-c1ccncc1)=O)OCC c1(CC(=O)NCCC(=C)CNC(=O)C(C)C)cncc(F)c1.c1ccccc1 C(=O)(C1CCCc2cccnc21)NC1CC(C)N(C)CC1 c1(C(=O)NC2C3(NC(C4CCC(C)O4)=O)CCC(C2)C3)cc2ccccn2n1 C1(C(C(C)C)NC(CCC)=O)CCN(C(=O)C(C)Cc2ccccc2C)CC1 N1(C(c2c(C)nn(C(C)(C)C)c2)=O)CCCCC(C)(C)C1.C1(C(=O)N)C=CCC1 C1(CNC(C=Cc2n(CC)ncc2)=O)CN(C(=O)C(C)C#N)CC12CC2 C12(C(N3CC4C(NC(CCC=CCC=C)=O)C4C3)=O)CC(CO)(C1)OC2C c1(NCC(CNC(c2sccc2-n2cnnn2)=O)O)c(Cl)cccc1[N+](=O)[O-] c1(C(N2CC(NC(C=CCCC)=O)C(O)C2)=O)cccc(C(N)=O)c1N C1(C(=O)NCCC(C)(C)CO)C2CCC(C2)N1C(c1ncccc1O)=O c1(CC(=O)NC(CCOC)CNC(c2cnn(C)c2Cl)=O)ccc(Cl)cc1C c1(C(=O)NC(CNC(C2C(C)C2)=O)C2CCC2)conc1C1CCCC1 C1(NC(CC2(C)CCCO2)=O)CC2(CCCCN2C(c2cc(Cl)ncc2Cl)=O)C1 C(CC(F)F)(C(=O)NCCC1CCCC2CC12)NC(c1cc(CC)oc1C)=O C1(C(=O)N)CC(c2cccc(Cl)c2F)=NO1.CCCCNC(=O)C=CCOC C=CCCC(C(=O)NCC(C)(C)C(F)(F)F)NC(C1CCCC(O)C1)=O c1(C(N2CC(OC)CC2)=O)csc(=NC2CC2)[nH]1.C1(CC(=O)N)CN(C)CC1O N1(C(c2c(CC)onc2)=O)CCOC(C(C)NC(C2(N=[N+]=[N-])CC2)=O)C1 c1(C(c2nnnn2Cc2cccs2)NC(C)CF)ccccc1F C(=O)(C#CC(C)(C)CNC(c1ccnnc1)=O)NC(C#C)C(C)(C)C C1(CNC(=O)C=CCN2CCOCC2)CCCCN1C(=O)CCC1CCC1.C c1(C(N(CCNC(CC2CC(OC)C2)=O)C)=O)c[nH]c2ccc(O)cc12 N1(C(C(CSC)C)=O)CCC(C(=O)N(C)Cc2cnn(C)c2)CC1(C)C C(C)(C(C)(C)C(=O)NC(C)CC#C)NC(CCCCOCC#C)=O N1(C(C=C(CCC)C)=O)CCN(CC(C)NC(c2cncc(Cl)c2)=O)CC1 c1(OC)cc(C#N)c(COC(c2cnn3ccccc23)=O)cc1OC C1(CNC(CC(C)F)=O)CCCC2(CN(C(c3ccc(C(F)(F)F)s3)=O)C2)O1 C1(C(=O)NCCNC(c2nnn3c2CCC3)=O)CC2CCC(C1)C2(F)F Cn1nccc(C(=O)NCC2CCCOC2c2ccccc2)c1=O N1(C(C(C(C)C)SCC)=O)CCOCC(CNC(C2CN3CCN2CC3)=O)C1 Cc1cc(O)c(C(N2CCOCC2C(N)=O)=O)cc1Br n1(CC)ncc(NC(C2CC(F)CN2C(c2cnc(SC)nc2)=O)=O)c1C C1(CNC(c2cc(C)on2)=O)CCC2CN(C(C3CCSC3)=O)CCC2C1 N1(C(C2CC(NC(c3ccncc3)=O)C2)=O)CCOCC(C2CC2)C1 c1(CNC(C2CC(OC)C2)=O)cc(C(=O)NC(c2cn(C)cn2)C)cs1 CC1CC(NC(=O)COCCN(C)C)CCN1C(c1cc(Cl)cs1)=O C(C(C)(O)C(=O)N(CCNC(c1ncncc1Br)=O)C1CC1)OC Cc1cc([N+](=O)[O-])ncc1C(=O)NCCC1(O)CCN(C(=O)C2=CCCS2)C1 C(=O)(N1CCC(C(=O)NCc2ccc(Cl)cn2)O1)c1cnc(C)o1 C1(CN(C(C=COCC)=O)C)CCN(C(C2(C)CS(=O)(=O)C2)=O)CC1 CC1CCN(C(c2cc(N)cnc2Cl)=O)CC1NC(c1cscn1)=O N1(C(C2C(C)CC(=O)N2)=O)CCC(C2CCCN(c3cc(Cl)ncn3)C2)CC1 C1(NC(c2cc(=O)cc[nH]2)=O)C2CCN(C(C3(CF)CCOCC3)=O)CCC12 C1(CNC(CN2CCC(C)C2)=O)(CNC(C2(C)CCC2)=O)CC12CCC2 N1(C(CSCC#C)=O)CCC(C2CCCN(C(=O)CC3CCCC3(F)F)C2)CC1 C1(C(N(C)CC2(N(C)C)CC2)=O)CC12CCC2.CCCN=[N+]=[N-].C(=O)C.N C(=O)(CCCS(N)(=O)=O)N1CC(C)C(NC(c2cc3n(n2)CCCC3)=O)CC1 O=C(C1=CCCCC1)NC1CCC(NC(C2CC2CF)=O)C1 c1(C(C)(C)C)ncc(C(N2CCC2Cn2cc(-c3cnccn3)nn2)=O)[nH]1 CCCC(CC(C)C)C(=O)N1CC2C(C(=O)Oc3c(C)cncc3[N+](=O)[O-])C2C1 c1(OC)cc(C(=O)NCCCN(C(=O)C(C)(Cl)Cl)C)nc(Br)c1 C(C(CC(C)C)C(=O)NCCOCC)OC.c1(C=O)c(C)cc(C)oc1=O.N CC1CN(C(=O)C(C)C(C)(C)C)CC2(CCN(C(c3coc(Br)n3)=O)CC2)O1 c1ncccc1SC(F)(F)F.c1(CCCC)ncc(CN2CC(NC(=O)N)C2)[nH]1 C1(NC(c2cn(CC)nc2)=O)CN(C(C23CCC(CC2O)C3)=O)CC12CCC2 c1(CN(C(CCO)C(F)(F)F)C=O)ccc(O)c(Br)c1 NS(=O)(=O)c1coc(C(N2CC(CO)(NC(C3CC34CC4)=O)C2)=O)c1 N1(C(CCCSC)=O)CC(C)(C)CC1CNC(=O)CC(C(F)F)c1ccccc1 CCCCC(O)C(=O)N1CC2CC1(CNC(c1ccc(C)cc1C1CC1)=O)C2 N1(CC(=O)NC(C)C(C)NC(C2(C(F)F)CCOCC2)=O)CCC(C)(C)C1 CS(=O)CCC(=O)NCC(C)(C1CC1)NC(c1cnn(C(F)F)c1)=O C1(C)(CC=O)CC(F)(F)C1.c1(C(C)NC(Cc2c(C)nc[nH]2)=O)ccccc1F Cc1cc(C(=O)NC2(CF)CCN(C(c3ccnn3CCF)=O)C2)n(C)n1 C1(NC(c2nc(Cl)ccc2F)=O)CC12CCN(Cc1cc(Br)cc(F)c1F)CC2 CC1CCC(CNC(c2cc(F)ccc2F)=O)N(C(c2cc(C(N)=O)co2)=O)C1 c1(CNC(=O)NC2C(C(=O)OC)CCC2)csc2cc(Cl)ccc12 c1(C(=O)NC(C2CCCN2C(=O)CC(C)c2ccco2)C)cc2ccccn2n1 C1(NC(c2nccc(OC)c2)=O)COC2C(NC(c3[nH]ccc3C)=O)COC12 c1(C(=O)NC23C(CCN(C(C(CSC)(C)C)=O)CC2)C3)ccccc1S(C)(=O)=O c1(-c2sccc2)nnc(N(C2CCCCC2)C)n1CC1COCCO1 N1(C(=O)C=Cc2ccccc2)CCN(C(c2cncc(Br)c2)=O)C2CC12 c1(OC)cc(Br)cnc1C(=O)N(CC(O)CNC(=O)CCF)C C(=O)(C1CCc2cccnc21)NCC1CN(C(c2ccccc2)=O)CC(C)(C)O1 c1(OC)cc(C(=O)NC2C=CCN(C(c3c(Cl)cccc3Cl)=O)C2)ccc1Cl C1(NC(C2N(C(C=CCN(C)CC)=O)CCC2C)=O)CN(C)CC1(F)F c1(CC(=O)NCC2N(C(C(CC)F)=O)CCCC2)cc(F)c(C)cc1F c1(NC(CC)CNC(C2(N(C)C)CCCC2)=O)ncnc2[nH]ccc12 C(=O)(C1CCCCc2ccccc21)NCCCCN(C(=O)C=CS(C)=O)C c1(C(N2C(CNC(CCCC(C)=O)=O)C(O)C(O)C2)=O)cc(C)c(F)cc1Cl CCCC(CCNC(=O)C=CC(C)NC(=O)CC1CCOC1)C1CC1 C123CCC(CC1)(CC2)CCNC(=O)C1CCN1C3=O.c1(CC)ccc(F)nc1 CN=c1[nH]ccc(C(=O)N(C)CC2CCCN2C(C2CC2C(C)O)=O)c1N CC(C)C1=NOC(C(=O)NCC2CCN2C(=O)Cc2ccncc2Cl)C1 c1(C(=O)N)cc2cccnc2cc1F.C1(CC)CC2(C1)CNC2.C12(CC1)C(=O)N2 c1(-c2nnc(N3C(COC)CCC3)n2CC2CCCO2)cc(F)c(N)c(F)c1 N1(C(C(CC)O)=O)CCC2(CCCN(C(c3cc(Cl)n[nH]3)=O)C2)CC1 N1(C(=O)OC)CCC(OC)CC1.C12CC(C)N1C(=O)C2 N1(C(c2cc(OCC)ncc2)=O)CC2(C)CN(C(=O)C(C#N)CCC)CC2(C)C1 c1(OC)ccc([N+](=O)[O-])cc1.C1(NCC)COCCN1C(=O)OC(C)(C)C N1(C(=O)Cc2sccc2Cl)CC2CN(C(C3(C4CC4)CC3)=O)CC2C1 Cc1n[nH]cc1NCC(C)(C)NC(=O)OC(C)(C)C C1(NC(C2SCCS2)=O)CN(C(c2cc3nn[nH]c3cc2F)=O)C2(CCOC2)C1 c1(OCC(=O)NCC2N(C(CN3C(C)CC3)=O)CCOC2)cccc(Cl)c1Cl Cc1cccc(C=CC(=O)NC2(C)CN(C(=O)C(CO)N(C)C)C2)c1 N1(C(COc2cccc(CC(=O)OC)c2)=O)CC(F)(F)CC1CCO N1(C(C2COCCN(Cc3sccc3Cl)C2)=O)CC2CC(C1)C1CCCCN1C2 N1(C(c2cc(C)nc(O)n2)=O)CCC(C2(NC(c3cc(Br)nn3C)=O)CC2)C1 CCCC(O)CC(=O)N1CC(F)(F)CC1CCNC(=O)COc1ccccc1Cl N1(C(=O)CO)CC2(C1)CN(C(C1(C(F)(F)F)CCC(F)C1)=O)C2.C1CCOC1 CC(CS(C)=O)C(=O)NCC1(O)CN(C(c2ccc(OCCO)cc2)=O)C1 c1(C(N2C(CCN(C)C(C3CC4CC4C3)=O)CCCC2)=O)ccc([N+](=O)[O-])o1 c1(C(N2C(CNC(C3C=CC(C(=O)OC)C3)=O)CC2)=O)c(Cl)cccc1Cl c1(NC(C2C(NC(C3C(C)C3)=O)C2)=O)cncc(Cl)n1 c1(C(=O)NC2CCCC(NC(C3ON=C(CC)C3)=O)C2)cc2ccc(C)cc2[nH]1 c1(CCOC)ccc(S(=O)(=O)N(C)CCN(C)C)cc1.c12ccc(cc1)[nH]2 N1(C(C2(C#C)CCCC2)=O)CC2(C1)CN(C(c1c(C(F)F)nn(C)c1C)=O)C2 C1(N(C(=O)CCC2CC(C)C2)CCNC(c2c(C)scn2)=O)CCCCCC1 C(c1cccc(O)c1)=CC(N1CCC(CN(C(CCC#C)=O)C)C1)=O Cc1c(C(N2CCCC3CN(C(=O)CCCC#N)CC23)=O)sc2[nH]cnc(=S)c12 c1(C(N2C(C(N3CC(C=C)C3)=O)CC2C)=O)cc(C)c(C)[nH]1 c1(OC)cccc2c1CC(C(=O)N(CC(C)NC(=O)CCC)C)CO2.C(N)(=O)N C(CCC(C)(C)C(=O)NCCC(CNC(C1(C)CCCCC1C)=O)OC)OC c1(C(N(CC(C)NC(C2C(CC)OCC2)=O)C)=O)cc2cc(Br)ccc2[nH]1 Cc1cncc(C)c1C(=O)NC1CCCCC1CNC(c1cc(O)ccc1Cl)=O c1(C(N2CCN(C(c3c(C)ccs3)=O)C(C)CC2)=O)cccc2c1COCC2 c1(CNC(C2CCN(C(C3CCC(=O)N3)=O)C2)=O)cncc(O)c1 N1(CCC)CC(NC(=NCc2ccccc2C)NCC2CCOC2)CC1=O C=CC1CCN(C(=O)CC(CNC(c2ccc(F)s2)=O)C2CCC2)CC1 C(CC(C(=O)N1CCC(F)(F)C1)NC(=O)C(C)N(C)C(C)=O)=CC C#CC1(O)CC(C(=O)NC2CCCC2NC(=O)Cc2ccco2)C1 N1(C(CC(=O)NCC#C)=O)CCCC1(C(=O)NCC(C)OCC)C=O c1(C(=O)NC2CC(C)N(c3nc4ccccc4s3)C2)ccc2cnccc2n1 c1(C(=O)NC23CCC(NC(C(C)(C)Br)=O)(CC2)C3)ccc2ccoc2c1 c1(C(=O)NCC(CO)NC(C(C(CC)C)O)=O)c(Cl)nc2sc(C)cn12 c1(C(=O)NCC(C)C)cc(-c2ccc(Cl)s2)[nH]n1.C1(CC(=O)N)CCOC1=O c1(OC)cc(CNc2cncc(C(=O)NCCc3cnc[nH]3)c2)cc(O)c1O N1(C(C(C)CO)=O)CC(NC(C2(CF)COC2)=O)CC12CCCCC2 c1(C(=O)NCC2CCC(NC(C(C(CC)O)C)=O)CC2)cccc2ccncc12 Cc1c(Cl)ccnc1C(=O)NC1CCN(C(C2CCC=CCCC2)=O)C1 O=S(=O)(c1ccccc1F)NC1CN(S(=O)(=O)c2cccs2)CC1F C(=O)(C(C)(C)C(=O)N(C)CC)OC.c1(C=O)ccn(C2CC2(F)F)n1.CC N1(C(C2CC3(CCC3)C2)=O)CCC(O)(C)CC1.C1(C=O)CC(O)(C(F)F)C1 Nc1cccc(C(=O)NC2CCCC(CNC(c3ccc(F)cc3Cl)=O)C2)c1F c1(C(C)(C)C)nsc(CNC(c2cnn(C3CCOCC3)c2)=O)n1 N1(C(CC(C)n2cccn2)=O)CCC(NC(=O)C=CC(C)(C)C)CC(C)(C)C1 N1(C(c2c(C)nn[nH]2)=O)CC2(CCN(C(c3cncnc3C(C)(C)C)=O)C2)C1 C(=O)(CC(CC)C(C)(C)C)N1CCC(CCCCNC(C(CCC)OC)=O)CC1 c1(C(CNC(c2n[nH]cc2C)=O)NC(CCSCCC)=O)ccc(F)cc1 N1(C(CN(C(CNC(CC)=O)=O)C2CCC2)=O)CCC2(C1)CC2(F)F C12(COC)CCCC1N(C(C1CN(c3ncncc3Br)C1)=O)CC2 c1(C(C)C)ccc(O)c(C(=O)NCCC2CC2)c1.C1(C(=O)N)CCN(C)C1C C1(NC(c2c(CC)onc2)=O)CC2(CCN(C(c3ccc(NC=O)cc3)=O)C2)C1 c1(OC)ccc(C(=O)NCC(C)(CO)NC(c2cnn(C)n2)=O)nc1Br CC1CCN(C(=O)C=CCC2(NC(C3CC4CCC3C4)=O)CCC2)CCS1 C(=O)(C(C)(CO)NC(=O)CCCC1CCCC1)NC1(C(COC)O)CC1 c1(C(=O)NCC2(C)CCN(C(C3(C)CC(=C)C3)=O)C2)sc(C)c(Br)c1C N1(C(c2ncc(I)s2)C(=O)NCc2ccccc2)CC(CO)C(C(F)(F)F)C1 Cc1c(C(=O)NCCC(C)N(C(=O)CSCC(C)C)C)cc(C)c2ncccc12 C=Cc1ccc(C(=O)N(C2CC(NC(=O)CN3CCCC3CO)C2)C)cc1 C1(C=O)CC2C=CC1CCC2.C1(NC(COCC(=O)NC)=O)CCCCC1.C C(=O)CC(C)O.C1(CC)CN(C(=O)Cn2ccnn2)C1.N(C)C.C(N)=O.N C1(O)(CNC(C2(C#N)CCCC2)=O)CCN(C(=O)Cn2ccccc2=O)CC1 c1(CC(=O)NCC2CCN2C(C2C=CCC2)=O)n[nH]c2ccccc12 N1(C(C2CCOC2)=O)CCC2(CCCC2NC(C23CCC2CC3)=O)CC1 C1(NC(CC=C)=O)CC2CCC1N(c1ncnc(C)c1F)C2 c1(CC(=O)N)cn2cc(F)ccc2n1.C1(NC(CC(=O)OC)=O)CCC12CCC2 Cc1c(C(=O)NC2CN(C(c3cccnc3Br)=O)C2)cccc1F C1(NC(Cc2c(C)noc2C)=O)CCC2CN(C(=O)C(O)CC3CCCC3)CC12 c1(CCC(=O)NCC(CC=C)NC(=O)CCC2CC(C)C2)ccc(Cl)c(F)c1 c1(C(N2CCCC(C(C)NC(C(C(C)C)(C)C)=O)C2)=O)cc2c(O)cccc2[nH]1 c1(C(=O)NCC2(CNC(c3cocc3)=O)CCCC2)cccnc1OCF n1(CCCF)nnnc1C(C1CC2CC2C1)NCC1(n2cncn2)CCC1 C1(CC(N2CCN(C(c3sc(CC)c(Br)c3)=O)CC2)=O)CC2C=CC1CC2 c1(C(C(=O)NCCOC)N(c2ccccc2OC)C)ccc(C(C)C)cc1F N1(C(CC(CCC)O)=O)CC23CCCCC2(C1)CN(C(c1nc(Cl)sc1Cl)=O)C3 c1(C(=O)NC2CCN(C(COC3(C)CCOCC3)=O)C2)cc(C(F)F)ccc1Cl C1(NC(c2cccc(F)c2F)=O)CC2CC(NC(C3CCC(F)(F)C3)=O)CC12 c1(C(=O)NC2C3CN(C(c4n(C)ccc4)=O)CC32)cc(Cl)cnc1O c1(C(=O)NC2C(CNC(c3csc(C)c3C)=O)C2)[nH]cc2c1CCCC2 c1(C(=O)NC(C)C(N2CCOCC2)C)ccc2nc(C3CCCCC3)oc2c1 C(=O)(C1CCN(C)c2ccccc21)NCC1CC(C)N(C(=O)C=CCO)CC1 c1(C(=O)NCCC2CCCN(C(=O)CCC3CC3)C2)cnc2c(c1)COC2 C1(C(=O)NC(C)CNC(c2cc(C#N)cs2)=O)CC2(C1)CS(=O)(=O)C2 O=C(CCC(=O)c1ccccc1Br)NCCNC(C1CC2CCC1C2)=O CC1CCN(CC(N2CCC(OCCNC(c3ncoc3C3CC3)=O)C2)=O)C1 c1(CCC(=O)N(CC(C)NC(=O)Cc2ccnn2C)C)cnc2ccccn12 N1(C(COc2c(C)nn(C)c2C)=O)CCN(C(C2CCC(=O)NC2)=O)CCC1C CC1CCC(C(=O)NCCCNC(c2cnc(-c3cnccn3)s2)=O)C1 C1(CNC(C(C)OCC=C)=O)CC2CC1CN2C(c1c[nH]nc1OC)=O C1(C(N2CCN(C(c3cnc(Br)s3)=O)C(CF)C2)=O)Cc2nccn2C1 C1(CC(=O)N(C2(C)CCOCC2)CCC)CCN(C(c2cscc2C)=O)CC1 C(=O)(CC1CCc2ccccc21)NC1CC(F)(CNC(CSC)=O)C1 Cc1cc(N(C)Cc2ccc(C)o2)nc(NCC2(C)CCC(=O)N2)n1 N1(C(c2n(C)ncc2)=O)CC2(CC2C(=O)NC(Cc2ccc(O)cc2)CO)C1 C1(NC(c2cn(C)[nH]c2=N)=O)CCC12CCC2.c1(C=O)ccsc1C(F)(F)F c1(C(N(CCNC(CC(CC)(O)c2ccccc2)=O)C)=O)ccn2c1CCCC2 N1(C(C2CCN(C)C2=O)=O)CC2CC(C(=O)NCCCN3CC=CC3)(C2)C1 c1(OC)ccc(O)cc1CN1CC2(CC(C(=O)Nc3ncn(C)n3)C2)C1 C1(NC(CCNC(COC)=O)=O)CCCC(C)C1.C12(C(=O)N)CCCC1C2 N1(C(c2n(CC)nnc2)C(=O)NCc2ccco2)CC(C(F)(F)F)CC1CO C(=O)(CCCC(=O)OC)NCC1CCC(NC(COCCCC#C)=O)CC1 C(CC1(C)CC1)(C(=O)NCCCO)N(C(C)CCC1CC1(Cl)Cl)C.C1CC1 c1(CC(C)N(C)C(C2CC2Cl)=O)ccc(O)cc1 CC1(CNC(C2(CF)CCOCC2)=O)CCCN1C(=O)CCC1CCCC(=O)N1 C1(N(C(C(COCC)NC(=O)CO)=O)C)COC(C)(C)C1.CC(F)(F)F C1(C)(NC(C(CC)O)=O)CCC(NC(=O)CCCc2ccc(C)cc2)CC1 C(CO)(CCCNC(C12CCCC1C2)=O)NC(CC1(OCC)CC1)=O c1(-c2c(OC)ccnc2)cc2cc[nH]c2cc1C(=O)Nc1ccc(CO)cc1 c1(OC)cc(C(=O)NCC(C)C)cc2c(C)c(C)[nH]c12.C1(C=O)CNC(=O)N1 C1(C(N(OC)C2CCC2)=O)CN(C(C2C=CCS2)=O)CC(C)(C)C1 C=CC1OCCC1C(N1CCC(N(C(=O)CSCc2ncc[nH]2)CCO)C1)=O N1(C(C)=O)CCC(C)(C=O)C1.C(=O)(C(C)n1cccn1)N(CCC)C(C)C.N N1(C(CCC(=O)NCCC)=O)CCC(C(=O)N(C)CCN2CCCC2)CC1CC Cc1cn2c(C(=O)NCCC3CCCN(C(C4C5CCCCC45)=O)C3)cnc2s1 C1(C2CCC2)(C(N2CCC(C)(CNC(C3(SC)CC3)=O)C2)=O)CC1(F)F C(=O)(C(C)CC(F)F)NC(C(C)C)CNC(c1cnn(C(C)C)c1)=O C(c1cnc(C(C)(C)C)s1)=CC=O.c1(CCC)n[nH]cc1C(=O)NCCCO S(=O)(=O)(c1ccc(NNC(=O)c2ccnn2CC=O)nc1)NC(C)(C)C.C(N)=O c1(N2CC(C(=O)OC)C2)ccc(-c2ccc(Br)cn2)nc1 C1(NC(C(C)n2ccnc2)=O)CN(C(=O)Cn2ncnn2)CC1CO N1(C(CCc2cnc(C)s2)=O)CC(NC(c2sc(CO)nc2C)=O)C(O)C1 c1(CC(N2C(CCNC(C(C)C)=O)CCC2)=O)ccc2nonc2c1 N1(C(c2c(C(C)C)sc(Cl)n2)=O)CCCCC(N2CCOCC2)C1 C1(C)(CC)CC(NC(=O)C(N)=O)CN1C(=O)Cc1ccc(C)nc1Cl C1CC2CC1N(C(C1CC1c1ccc(Cl)cc1)=O)C2.C(C=O)(C1CC1)OCC C1(NC(CCOCCC)=O)CC2CC1CC2C(=O)N(C)CCc1cc[nH]n1 Cc1cc(C(=O)NC(C2CCCN(C(C3CC(F)(CO)C3)=O)C2)C)nnc1C Cc1ccc(SC(C)C(=O)N2CCC2C)cc1.C1(C=O)CCC(C(N)=O)O1.N CC1CCCCC1(CNC(c1nnsc1N)=O)NC(=O)C1=C(Cl)CC1 CC(CC(=O)N1CC2CCC(C1)C2C(N1CCCC(C)(C)CC1)=O)CC(C)(C)C CC(C)CC(C)CC(=O)NC1CCCC12CN(C(C1(C)CCN(C)CC1)=O)C2 CC(C)CC(O)C(=O)N1CCC1C(=O)Nc1cnn(-c2ccc(Cl)cc2Cl)c1 C1(NC(C(C(C)C)OCC)=O)CC(O)CN(C(c2cnn(C(F)F)c2)=O)C1 N1(C(c2c(C)nsc2C)=O)CCCN(C(c2cn(CCCC#N)nn2)=O)C(C)C1 c1(CN2C(C(=O)Nc3ncc(C(C)(C)C)cn3)COCC2)c(F)cc(F)cc1F C#Cc1ccc(Cl)c(C(=O)NCC2CCCCN(C(=O)CSC(C)C)C2)c1 C(=O)(CC1=CCOCC1)N1CCC2(C(C(N(C)Cc3onc(C)n3)=O)C2)C1 c1(C(=O)OC)nccnc1N1CCC(CN(C(=O)C=Cc2cscn2)C)CC1 C(=O)(C1CCc2cccc(O)c21)N1CCN(C(Cn2c(C)nnn2)=O)CC1C C1(C(N2C(C)(C)CC(NC(c3cc(N)ccc3F)=O)C2)=O)CCn2nccc2C1 N1(C(CCNC(C)=O)=O)CCC(CCNC(=O)CCn2nc(C)cc2C)CC1 C(=O)(C(O)C1=CCCCC1)N1CC(CC(=O)NCC2(n3nccn3)CC2)OCC1 N1(C(=O)CC2(O)CCOC2)CC2CCC(C1)N2C(=O)CC(O)CC1CC1 C1(c2n(CCSC)nnn2)(NCCc2ncn(C)n2)CSCC1C C1(OCC(=O)N(CCCC)C)CCN(S(C)(=O)=O)CC1.C(=O)C.C1CC1 c1(N2C(CNC(CCCOCCC)=O)CCCC2)ncnc2sc([N+](=O)[O-])cc12 N1(C(C2CC2)=O)CCC(CCC)CC1.C1(CC=O)CCSC1.CC(=O)OCCC S(=O)(=O)(c1ccc(S(=O)(=O)C(C)(C)C)cc1)NC1CC(OCC)C1C c1(OC)cc(Cl)c(Br)cc1CNc1cc(O)c(C)cc1C C1(C(N(CCCC)CC)=O)CCC2(CC2)N1C(c1ccc(CO)nc1)=O c1(CC(=O)NCC2(NC(=O)CC3CC=CCC3)CC2)csc2nccn12 C(N=c1[nH]c(=NCCCN(C)C)[nH]c2c1CC(C)CC2)c1cccc(C)c1N C1(CNC(c2c(CC)nns2)=O)CCN(C(C2CC3(CC3)CO2)=O)CC1(F)F C=C=C(C)CC(=O)NC1CN(C(=O)CSCCC(C)C)C2CC12 C1(CNC(C(C)OCC#C)=O)N(C(c2nnn3ccccc23)=O)CCCC1(C)C C(C(F)(F)C(=O)NCC1CCC(C)C1)OC.c1cccc(C)c1.C(=O)C=O C#CC1(NC(=O)C(Cn2cncn2)NC(=O)CCC(C)(C)F)CCCCC1 [SH](=O)(=O)c1ccc(C(N2C3CCC2CC3)=O)cc1.CC(C)(C)N.C(=O)C1CC1 N1(C(CC(CC)OC)=O)CCC(C2(NC(=O)C(F)CC3CCCC3)CC2)C1 CC(C)P(=O)(CC(=O)N1CC(NC(=O)CCn2cc(Cl)cn2)C(F)C1)C(C)C C#CCC(C)(C(=O)NCC(N1CCOCC1)=O)NC(c1nn(C)cc1Cl)=O CCCCCC(O)CC(=O)NCC1(C2CC2)CCN(C(C2COC(C)C2)=O)C1 N#Cc1cc(C(N2CCC2CNC(=O)CC2CCCC2(F)F)=O)c(F)cc1F N1(C(C(CC)O)=O)CCC2(CCCN2C(C2CCC3CCC(=O)N3C2)=O)CC1 Cc1cc(C(=O)NC2CN(C(=O)C(N3CCNC3=O)C)CC2F)nn1C(C)C C1CC12CCN(C(=O)CC1CCC(=O)N1)CC2.c1(CN=[N+]=[N-])ccc(C(=O)N)o1 c1(CC(=O)N(CC(=O)NCC2CC(NC)C2)CCC)cc(C)oc1C C1(C(N2CC(NC(CCC(=O)c3cn(C)nc3)=O)C2)=O)CCCC(F)(F)C1 CC1C(NC(c2cnc(Cl)c(C3CC3)c2)=O)C(C)CCN1C(c1cn[nH]c1)=O CCCC(CCO)NC(c1nccc(OC)n1)c1nnnn1CCC1CC1 c1(CC(=O)NCCOCCCC)ccc2c(c1)CN(C(=O)C(C)(C)F)CC2 C1CC(C)(C)CCC1.c1(CC)cc(C(=O)NC)n[nH]1.C1(C=O)CC(C)(C)C1 c1(CC)cc2c(CC(=O)NC3CC3CNC(c3cnn(C)c3)=O)csc2s1 C12(NC(=O)CC3CCOC3)CC1CN(C(=O)CN1CCCC1=O)C2 Cc1nc(-c2cccs2)ccc1C(N1CCCC1c1cc(O)nc(O)n1)=O CCCCC(O)C(=O)NC1(C2CN(C(=O)C(C)Cc3ccnn3C)C2)CC1 N1(C(c2c(CC)n(C)cc2)=O)CC(C(=O)N(CCCO)CCCO)CC(C)C1 c1(C(=O)NCC2CCC2)ccnc(F)c1O.N1(C)CCCC1.C1(C=O)CC1F c1(C(N2CCC(NC(C(C)NC(CC)=O)=O)C2C)=O)cc2c(Cl)cc(Cl)cc2[nH]1 Cc1ccc(C(N2CC(CNC(c3ccc(CF)cc3)=O)CC2C)=O)c(N)c1F c1(C(=O)NCC2CCN(C(c3onc(C)c3C)=O)CC2C)cccn2cnnc12 N1(C(Cc2c(C)ccs2)=O)CC(C)(C)CCC1C.C(=O)C(F)(F)C(O)C1CC1.N C(C)(CC(C)(C)CO)NC(C(C(C)OC)NC(C1CCOC1C(C)C)=O)=O CCCC(CCC)CC(=O)N1CCOC(CC(=O)NC(CCO)C2CCC2)C1 Cc1cc(C(N2CCCC(C)C2CN=c2ccnc[nH]2)=O)c2c(n1)CCCC2 CN(Cc1cccc(OC(F)(F)F)c1)N1CCCC1(C)c1ccccc1 N1(C(C2(CC=C)CN(C(=O)CC(CC)C3CCC3)C2)=O)CCC2(CC(OC)C2)C1 Cc1nc(CO)sc1C(=O)NC(C)CCNC(=O)CC(C)c1cccnc1 c1(C(CC)N(C(=O)NC2(C#C)COC2)CC)cccc(Cl)c1 c1(C(=O)OC)c[nH]c(C)cc1=NC1CN(C(C2(N(C)C)CCCCC2)=O)CC1C Cc1cc(N)n2ncc(C(=O)NC(C)CC(C)C)c2n1.N(S(N)(=O)=O)CC=O c1(C(=O)N)ccc2c(c1)C1CCC2O1.C(=O)(C(F)C(F)(F)F)N1CC(F)C1.C c1(C(C(C)NC(=O)NCC2CC(OC(F)F)C2)C)ccccc1Cl c1(C2CC(=C)C2)nc(CN(C)C(=O)OC(C)(C)C)nn1-c1cccnc1 c1(CC(=O)OC)cn(CC2CN(C(C3SCCCS3)=O)C2)nn1 Cc1cccc(OCC(=O)NC(C)(C)CN(C(=O)CC(C)F)C)c1 Cc1cc(C(N2CC(NC(C3(C)CCC(F)(F)C3)=O)C(O)C2)=O)c(O)c(C)c1 C1(C(=O)NCC(CC)(C)C(=O)N2CC3CC2CN3C(=O)NC)CCn2nncc2C1 CCC(C)CCCC(=O)NC1CC(NC(=O)C(c2ccccc2Cl)(C)C)C1 C(=O)(C1=CCSC1)N(C(C)C)CCNC(C1(C)CCOC1)=O CCCC(CC)C(=O)NCC1(C(N2CCC(CN(C)C)C2)=O)CCC1 C=CCC(CC(C)C)C(=O)N(CCCOCCN(C(=O)CC(C)(C)CC)C)C Cc1ccnnc1C(=O)NCCN(C)C(c1ccccc1OC1CCCC1)=O N1(C(CN(C)Cc2ccccc2)=O)CCCC(NC(=O)CCCCCF)CC1 Cc1nc(-c2cc(C(=O)NC3COCC3NC(=O)COC(F)(F)F)co2)cs1 CC#CCCC(=O)NC1CCOCC1NC(=O)C(C(C)C)N1CCCC1=O C1(CNC(C2C(c3cn(C)nc3)C2)=O)C2CCCC1N(C(=O)CC(F)(F)F)C2 c1(C(N2CCN(C(=O)CC(F)(F)F)CC2CC(F)(F)F)=O)ccc2c(c1)COC2 N1(C(Cc2n(C(C)C)cnn2)=O)CCC(O)(Cn2cc(CN(C)C)nn2)C1 CC1=C(C(=O)NC2CC(NC(C3CC(C)CO3)=O)C2)CCC1 O=C1CCCCC(C(=O)NCc2ocnc2C(N2CCCC2C2CC2)=O)C1 N(C1CCOc2cc(F)ccc21)C(C1CC1NS(=O)(=O)CCCCl)=O C1(C(C)(C)C)COCCN(CC2(c3ccc(Cl)cc3)CCC2)C1 C1(C(=O)N)CC(=O)N(C)C1.Cc1nc(CC(=O)NCc2csc(C)n2)cs1 n1(CCC)ncnc1CNC(=O)CCCN(C)C(c1cn(C)nn1)=O C(CCC(=O)N1CCCC1C(C)NC(=O)C(O)CC1CCOCC1)OCC=C Cc1ccc(CN2CCCCC2C(N2CCS(=O)(=O)CC2)=O)cc1Br C1(C(=O)NC(C)(C)CNC(c2cc(C(F)F)ccc2F)=O)CCn2ccnc2C1 C1(C(=O)NCCCCCC)CN(C(=O)C=Cc2cc[nH]n2)C2(CCC2)C1 C1(n2ccnn2)CCN(C(=O)C=CC2CCCC2)CC1.C(C)(C(=O)N)OCC S(=O)(=O)(c1ccc(-c2ccc(F)cc2)cc1)NCC1CC(C)SC1 N1(C(CSCC)=O)CCOC(CCNC(C2(OC)CCCOC2)=O)C1 C1CN(C(C2(F)CCC2)=O)CC(C)(C)C1.C=C1CC(C(F)(F)F)(C(=O)N)C1 c1(-c2nc(C(c3ccccc3)(F)F)c(Cl)s2)cccc2ncoc12 N1(C(C(C)(C)c2cscn2)=O)CCCC(C)(CNC(=O)Cc2cncnc2O)C1 c1(C(=O)N)cc(C)c(C)cc1Cl.C(C(=O)N(C)CC1CC1)(C1CCCC1)OC C=CCCCCCNC(=O)C(CCC1CCC1)NC(=O)Cc1ccn(C)c1 CC(F)(F)C(C(=O)N1CC(CNC(=O)CCC2CC2(F)F)C1)c1ccccc1 c1(CC(N2C(CNC(c3cc(C)sn3)=O)C(C)CCC2)=O)cn2c(n1)CCCC2 Cn1nc(C(N2CC(O)CC2C(=O)Nc2ccnc(O)c2)=O)cc1Cl C(=O)(CCCS(C)(=O)=O)N(C1CCCN(C(=O)CN2CCCCC2=O)C1)C c1(NCc2cc(C)c(Br)cc2)nc(N2CCOCC2)nc2scnc12 N1(C(c2c(C)c[nH]c2)=O)CC(C(=O)N(CC(N2CCCC2)C)C)C2(CCC2)C1 CC(C)(C)CC(O)CC(=O)N1CCC(C(CO)NC(=O)COCCCF)CC1 C1(NC(CCc2cc(C)[nH]n2)=O)(CF)CCN(C(=O)CN2CCOCC2)C1 Cc1cn2c(n1)CN(C(=O)C1=CCN(C(C3CCCO3)=O)CC1)CC2 C=CCC(CC)C(=O)N1CC=CC1(C(=O)N(C)CC1(F)CCC1)COC c1(CCC(N2CCC(O)(CCNC(CCOC)=O)C2)=O)c(Cl)cccc1Cl c1(C(=O)NC(CNC(c2c(OC)ccc(C)c2)=O)C)ccc2ccc(C)cc2n1 c1(C(N(C2CCCCC2)CC)=O)ccc(C2CCCCC2)c(F)c1 C#CCC(C)(C(=O)NCc1nnsc1CC)NC(=O)CC1CCCC(O)C1 CCC(C)C(O)CC(=O)NC1CC(C(=O)N2CC(OC(=O)NC)C2)=CC1O c1(CC)cccc(C(N2CCC(N(C(=O)CC(C)F)CC3CC3)C2)=O)n1 C1(C(=O)NC(C2N(C(COC(C)=O)=O)CCC2)(C)C)CCN(C(C)=O)CC1 CC1(C)CCC1CC(N1CCCC1C1(NC(c2cc(Br)cs2)=O)CC1)=O C1(CCNC(CC=CCC)=O)CCN(C(C2CC(C#N)C2)=O)C1 C1(C(C)C)C(NC(=O)CC(C)F)CCN1C(=O)Cn1cnc(=N)[nH]1 N(C(=NCCCF)NCCOc1ccc(Cl)cc1)CC(N(CC)OC)=O N1(C(CC2C3CN(C(C4(C)CCCS4)=O)CC32)=O)CCCCC2(CCC2)C1 c1(OC)cnc(N2CCCC(CC(N)=O)C2)[nH]c1=N c1(COC(=O)NC(CC=C)C2CC2)c[nH]nc1C(N1CC2CC2C1)=O C(N=c1ccc(Br)c(S(=O)(=O)NC2CCCC(F)(F)C2)[nH]1)c1c(C)c(F)ccc1 c1(C(N2CCC(NC(c3cc(OCC)no3)=O)C2)=O)cc2n(n1)CCC2 C#CC1(C(=O)NCC(C2CCCN2C(=O)CC2CCCN2CC)(C)C)CCCC1 N1(C(Cc2cc(C)on2)=O)CC2CN(C(c3n[nH]c(C)c3C)=O)C2C1 c1(NC(c2n(CC)nnn2)(C)CCN2CCCCC2)ccc2nc(SC)sc2c1 c1(C(N2C(C)CC(NC(=O)C3=C(Cl)CCC3)C2)=O)cc2c(ccn2C)s1 Nc1c(C(N2CC(NC(c3c[nH]nc3F)=O)CC(F)C2)=O)cccc1C(F)(F)F C(=O)(C#CC1CCCCO1)NCC1C(C)CCN1C(c1ncc2ccccn12)=O N1(C(C2COCCO2)=O)CCCN(C(c2cc(C3CC3)nnc2O)=O)CCC1 N1(CC)OCC(N(C2CCN(C3CCOCC3)CC2)C)C1=O C(CC(=O)N1CCCC(N(C)C)CC1)(C(F)F)NC(C(C)(C1(C)CC1)OC)=O c1(C(N2C(C3(NC(CC4(C#N)CC4)=O)CC3)CCCC2)=O)n[nH]c2c1CC1CC21 Cc1coc(C(C)C)c1C(N1CCC(CNC(c2c(C)n[nH]c2C)=O)CC1)=O c1(CC(=O)O)cncc(NC(=O)CCCNC2(C3CCCO3)CCC2)c1 N1(C(CC2C(C)CC2)=O)CCCC2CN(C(C3CC4COCC4C3)=O)CCC12 N1(CC(=O)N(C2CCC2)CC=Cc2c(C)noc2C)CCC(C#N)CC12CC2 C(=O)(C1SCCc2ccccc21)N(CC(CO)(CO)NC(C(C)C(F)(F)F)=O)C c1(OC)ccc(O)cc1NC(c1ncoc1CNC(=O)C1=CCCSC1)=O c1(CC)cc(Br)ccc1C(N1CC(NCc2cc(C)cnc2Cl)C2(CC2)C1)=O c1(C(=O)NCC(C)NC(C2(C(C)(C)C)CCCC2)=O)ccc2c(c1)NCC2 C(c1ccccc1Cl)=CC(=O)N.C1C2CCC(C2)N1C(=O)CC1(C(F)F)CC1 c1(OC)c(C(=O)NCc2cncc(C(=O)NC3CCS(=O)CC3)c2)cnn1C N1(C(C=Cc2c(C)ccs2)=O)CC(NC(=O)C=CC2CCCO2)CC(C)C1 n1(CC(N2CCC2)=O)nnc2c1CCCC2.C1(CN(C)C)CC1C(=O)N.CC C=CCCCCCCC(=O)NC(Cc1ccccc1Br)C(=O)NC1CC(CO)C1 C1(C(=O)NCC(CC=C)(C)C)CN(C)CCN1C(C1SCCS1)=O N1(CC(N2C(CNC(C(CC)C=O)=O)CC2)=O)C(=O)Cc2ccccc2C1=O.O C#Cc1cc(NC(C2CC(NC(c3ccnnc3O)=O)C23CCC3)=O)ccc1C c1(C(=O)NC2CC(C)N(C(C3CNC(=O)N3C)=O)C2)ncc(C#N)cc1Cl C1(NC(C2CCC(C)(CC)O2)=O)CN(C(=O)Cc2ccccc2)CC12CCC2.N C=CCCCCCC(=O)N1CC(CC=C)(NC(c2oc(CC3CC3)nc2C)=O)C1 C=CCC(C(=O)NCCOCC1CCCC1)NC(C1COC(=O)N1C)=O c1(CN(C(C(c2cccc(F)c2)NC)=O)C)coc2cc(F)cc(F)c12 c1(C(=O)NC2CC(NC(C3C4CCN3CC4)=O)C2)cc(Cl)cc(Cl)c1O C1(CC(=O)NCCN(C(CN(CCC)C)=O)C(C)C)CCC2CC12 c1(C(=O)N)ccc(=O)n(C2CC2)c1.C1(CC(C)C)(C(=O)N(C)CC)CCC1 CON(CCC(=O)NC1CC1C)C(=O)CCN1CCCC1 c1(C(N(CC)CC)=O)c(C)noc1C(F)(F)F.c1(C(=O)N)ccn(C)n1 C12(NC(c3cc(C)sc3)=O)CCN(C(C3C(C)(C)C3(C)C)=O)CCC1C2 C1(CNC(C(C)SCC)=O)CC2CCC1N(C(C1CC(OC)CC1)=O)C2.O O=C(N(O)Cc1cn(CC2CCCO2)nn1)c1cc(C2CC2)on1 N1(S(CC)(=O)=O)C2CCC1CC(C(=O)NC(c1ccccn1)CO)C2 Cc1oc(-c2ccccc2)cc1C(=O)NC1CCN(C(=O)CC2CCCCC2)C1 C1CCN(C(c2cc[nH]n2)=O)C(C2CC2)C1.c1(C(=O)N)cc(F)ccc1C(F)F N1(C(CC(C)(F)F)=O)CC2(CCN(C(c3ccncc3N)=O)CC2)C2COCC12 c1(NC(C2N(Cc3c(C)c(O)ccc3)CC2)=O)cc(Cl)c(F)cc1Br c1(C(N(CC(CNC(COCCOCC#C)=O)O)C)=O)cc(O)ncn1 CC1CC(C(=O)N(C2CN(C(C3CC(C(=O)O)C3)=O)C2)C)=NO1.C(C)(C)C c1(OC)ccc(S(C)(=O)=O)cc1C(=O)N(C1CC2CCC(C1)N2)C CCCC(C(=O)N1CCC(CNC(c2cccc(F)c2Cl)=O)C1)S(N)(=O)=O C1(CNC(=O)CCc2cccnc2)CN(C(=O)CCc2ccc[nH]2)CC1(F)F N1(C(c2cnc(CC)s2)=O)CCCN(C(=O)C(C)N(CC(F)(F)F)C)CC1C C1(O)(CCC)CCN(C(C2CSCN2C(=O)C(N2CCNC2=O)C)=O)CC1 Cc1nc2[nH]c(C(=O)NCC3CC(C)(C)CN3C(=O)CCCC#N)cc2s1 CCCS(=O)(=O)C(C)C(=O)N1CC(CC(C)NC(c2c(C)nn(CC)c2C)=O)C1 N1(C(Cc2ccc(OCC)cc2)=O)CCN(C(=O)CC2(CC)CCC2)C(C)C1 C1(C(=O)NC(CC)CN(C(c2ccsc2OC=O)=O)CC)CCN(C)CC1 c1(C(N2CC(O)(CNC(C(C=C)(C)O)=O)C2)=O)ccc(OC(F)F)cc1.O Cc1ccsc1C=CC(=O)N.C1(C(N(CC(C)C)C)=O)CCC(=O)N1C(C)C c1(OC)cc(C)c(C(=O)NC(C)C(C)NC(=O)CC2CCCCC2)c(C)c1 C1(NC(CNC(C)=O)=O)C2CC1CN(C(c1c(C)coc1-c1ccccc1)=O)C2 C1(CNC(C(C)OC)=O)CN(C(c2ccc(OC)nc2)=O)CCO1.C1CC1 C12(CNC(C(CC(=C)C)C)=O)CN(C(c3cnoc3C)=O)CC(F)(C1)C2 C1(C(N2CC=CC2CF)=O)(CC)CCCN1C(c1cccn1CCOC)=O Cc1cc(F)cnc1C(=O)NCC(C1(O)CN(C(=O)C2=CCSC2)C1)(C)C C(=O)(CC(=O)N(CC(C)NC(=O)CC(C)n1ccnc1)CC)NCC#C.C CCCCCC(C)(CC)C(=O)NC(CNC(C1(Cl)CC1)=O)C1CC1 C1(C)(NC(CC2C(C)=NOC2=O)=O)CCN(C(=O)CC2C=CCC2)CC1 C1(N(C)C(C2CC3C=CC2C3)=O)CC2CCC(C1)N2C(=O)CC1CC2CC1C2 Cn1c(C(N2CC3C(C(N4CC5C(C4)C5(C)C)=O)C3C2)=O)cc2ccccc12 c1(N2CC3C(NC(c4c(OC)nc(C)cc4)=O)C3C2)nc(C(C)C)ccc1C#N c1(C(=O)NC(CNC(CCn2ccc(C)n2)=O)CO)cnnc(O)c1 C1(C(=O)NCCC(C)N2CCCC2)(CC)CCCN(C(=O)C(C)OCC(C)C)C1 C(CCNC(c1cc[nH]c1C)=O)(C(=O)NCCC(O)CO)OC CC(C)CC(C(=O)NCCCC(N)=O)NC(=O)CCCC1CC1C Cn1cc(Br)cc1CN1CCC(n2cc(C(=O)N(C)C)nn2)C1 c1(CC)ccc2c(c1)CN(C(c1csc(=NC)[nH]1)=O)C2.C1(C=O)(CC)CCC1.N N1(C(C2N(C(c3ccc(C)s3)=O)CCCC2)=O)CCC2(CNC(=O)N2)C1 C12(CNC(c3cnns3)=O)CC1CN(C(c1coc(-c3ccccc3)n1)=O)C2 C=CCC(CC=C)C(=O)NCc1cnn(C)c1C(=O)NC(C)(C)C(C)O C(C1=CCN(C(c2ccccc2Cl)=O)CC1)NC(c1c(C)occ1)=O Cc1cccc(C(C)(C)C(=O)NC2CCOC(C)C2)c1.C1(C)(C(=O)N)CCCO1 c1(C(c2nnnn2C2CCOC2)NC(c2noc(C(F)(F)F)n2)C)ccccn1 CCCCCC(O)C(=O)NCC=CCC(=O)NC(C)Cn1ccnc1 N1(C(CC(C=C)(C)O)=O)CCC2CCC(C1)N2C(c1ccc(S)cc1)=O N1(C(Cc2n(C)nnc2)=O)CCCCC1CNC(C1(n2cccn2)CCC1)=O Cc1cc(C)n2cnc(C(=O)NCCCO)c2n1.C1(C=O)CC1.CC.C1CC1 Cc1ccc(NNC(=O)Cc2c(-c3ccccc3C)noc2C)c(C)c1 Cc1cn2ccnc(C(=O)N(CC(C)NC(C3CCn4ncnc4C3)=O)C)c2n1 C(=O)(C(C)C(F)(F)F)N(CCOC)CCNC(=O)CSC1CC1 CN1CCN(C(c2ccco2)=O)C(CNC(C2NC(=O)OC2(C)C)=O)C1 c1(C(=O)NC(CNC(C2C(C)C2C)=O)(C)C2CC2)ccnc2c1CC(=O)N2 CC(C)CC(N)CC(=O)N1CCC(Oc2ccc(I)cc2F)CC1 c1(C(N(C(C)CNC(=O)C(C)(C)CCCO)C)=O)ccc2c(c1)SCCN2 N1(C(C2CC(C(C)C)OCC2)=O)CC2CCC1C(CNC(c1cscn1)=O)C2 CC#CCC(C(=O)NCCCCN1CCC1)NC(C1CCC2(CCC2)O1)=O C#Cc1cc(NC(=O)CC2CCN(C(=O)CC3(OC)CCC3)C2(C)C)ccc1C CC(C(C)(C)C(=O)NCCCc1cn[nH]c1)NC(C1CCCSC1)=O c1(CN2C(C(=O)N(CCO)Cc3ccccc3)COCC2)n[nH]c2cccnc12 C12(C(=O)NC3CCN(CCCNC(C(CC)COC)=O)C3)CCC(CC1F)C2 N1(CCNC(Cn2c(C)cnc2)=O)CCCN(C(C2CC3(CCOC3)C2)=O)CC1 C1(C(=O)NC2(CO)CN(C(c3c(C)ccc(C)n3)=O)C2)CCC12CCOCC2 C(=O)(C1CCSc2ccccc21)N1CCCCC(NC(=O)Cn2cncn2)CC1 C1(NC(N=S(C)(C)=O)=O)CCCN(c2ccc(OC(F)F)cc2)C1=O N1(C(c2n(C(C)C)ncc2Cl)=O)CCN(C(=O)C(C2CC2)C2CC2)CC12CC2 C1(CNC(c2c(C)nco2)=O)CCN(CCCC2CCOC2)CC1 N1(C(CC2CN(C)C2)=O)CCOC2(CCCN(C(c3cc(Cl)cnc3O)=O)C2)C1 CC(C)CC(CNC(c1sccc1F)=O)NC(C12CC(F)C1C2)=O N1(C(COc2cccc(C)c2)=O)CC2(CCN(Cc3ccn(C(C)C)n3)C2)C1 CC(CCN=c1[nH]c2ccccc2s1)NC(=O)C(C1CCCCCC1)O N1(C(CC(C)N(C)C)=O)CCC2CCC(C1)N2C(=O)CCn1cnccc1=O N1(C(C2C(OC)CC2)=O)CCCCC1CN(C(=O)CCc1nc(=N)[nH][nH]1)C N1(C(c2cc(C)[nH]c2C)=O)CCC(C)(C)C1CC(=O)NCC(C)C(C)C C1CN(C(c2cc(O)cs2)=O)CC12CC2.C(C)(CC(=O)NC)(C1CCC1)N(C)C c1(C(=O)NC2C(NC(C(C=C)(C)O)=O)CCOC2)cc(F)cc(F)c1 N1(C(C2(C)CCOC2)=O)CCC2(C=C(C(=O)NC3CCS(=O)CC3)C2)C1 CN1N=C(CC(=O)N2CCCC(N3CCC(=O)NC3=O)C2)CC1=O N1(C(C(=Cc2cccnc2)C)=O)CCC(F)C(NC(=O)C2=NOCC2)C1 CC#CCCCC(=O)NC(C1CCCCN1C(c1cn(C(C)C)cc1C)=O)C C1(CNC(CCOC)=O)CCCCC1NC(=O)Cc1ccc(OC(F)F)cc1 N1(C(CC2CCCN(C(c3ccc(C(C)=O)o3)=O)C2)=O)CC(C)OC2(CCC2)C1 C1(C(C(C)NC(C2OCCO2)=O)NC(c2cocn2)=O)CCCCC1 CC1CN(C(=O)C2=CCC(NC(C3CC(O)C3)=O)C2)CCN1C N1(C(CN(c2ccccc2)C(C)=O)=O)CCCC(CC(N)=O)C1 C1(C(=O)NCC(CN(C(c2c(C)nc(CC)s2)=O)C)O)CC(C)(C)CN1C c1(C2C(C(N3CCCC4CCC34)=O)C2)c(F)cccc1Cl C=C(C)CC(C(=O)NCC1CC2CCC2C1)NC(C1C(C#N)C1(C)C)=O N1(C(C(C(CC)O)C)=O)CC(C)CN(C(=O)C=CCN(CC(F)(F)F)C)CC1C CC(C)CC(C)(CNC(C1CC=CC1)=O)NC(=O)CSc1n[nH]c(=N)s1 Cc1cc(Br)cc(C)c1S(=O)(=O)NCc1cccc(Cn2cncn2)c1 C1(C(=O)NCC2(CNC(C3C(C)CC=CC3)=O)CC2)CCCC2CCCN12 c1(C=O)nc2cnccc2s1.CC(C(=O)NC(C)C1CC1)NS(C)(=O)=O.N Cc1nc2c(C(=O)NCCCCCNC(=O)C(C3CCOCC3)C)cccc2o1 C#CCCC(C(=O)N1CC(C(=O)OC)(CC)C1)NC(C1CC(C)=NO1)=O C(CC(C)C(=O)N)=CC.c1(C(N2CCC2)=O)csc(N(c2ccccc2)C)n1.C N1(C(C2C(NC(C3(C(N(C)C)=O)CC3)=O)CCCCC2)=O)CCc2ccsc2C1 C1(NC(c2c(CC)non2)=O)C2CC(NC(=O)C(C(C)C)C3CCC3)CC12 C1(c2n(CCOCC)nnn2)(NCCOC(C)=O)CCCC2(CCC2)C1 N1(C(C(CC)n2ccnc2)=O)CCCCC1CN(C)C(C1CC(N(C)C)C1)=O C(=O)CCCC(C)(C)C#N.C(=O)C(C)N(C(=O)CC1CCOC1)C1CC1.CO C(CC#CC(C)(C)C)NC(C1CC(OC)CN1C(c1nc(=N)cc[nH]1)=O)=O C(=O)(CCS(=O)(=O)NC)N1CCC(N(C(=O)CCN(C)CC)CCC)CC1 C1(C2CN(C(c3cc([N+](=O)[O-])c[nH]3)=O)C2)CC1.c1(SC)cc(C=O)n(C)n1.N C1(C(=O)NCC(c2c(Cl)cccc2Cl)N)CN2CCC1CC2 CC(C)C(CCN(C)C(c1csc(Cl)c1Cl)=O)NC(=O)Cc1cn[nH]c1 C1(C)(C(=O)NC(CC(C)C)CNC(=O)Cc2cscn2)CCC(=O)NC1 c1(CNC2C(C(=O)NCc3ccc(C(C)C)cc3)C2)cn2c(Br)cccc2n1 c1(N2C(CN(C)C(c3cc4n(n3)CCC4)=O)CCC2)ccc(F)cc1[N+](=O)[O-] n1(CC(N2C(CC)C(NC(=O)C(C)c3cccs3)CC2)=O)cnc2c1CCCC2 CCS(=O)(=O)CC(=O)NC(CC(=O)N1CCC1C(C)C)C1CC1 c1(C=O)cccc2c1CCC2.C1(SCC)CCC(C(=O)NCC2CC2)CC1.N C(CC(=O)Nc1c(C)cc(C)nc1C)(C(F)(F)F)NC(C1CCC(N(C)C)C1)=O C1(CNC(C(CC)C)=O)CCN(c2cc(OC3CCOCC3)ncn2)CCC1(F)F c1(CN(C(=O)C(=O)N(C)CCC2CC2)C)cc(Cl)ccc1Cl c1(C(=O)NC(C2CCN(C(C3C4(CC4)C34CC4)=O)C2)(C)C)ccc(Cl)cn1 C1(NC(c2n[nH]cc2F)=O)CCN(C(C2CCCN2Cc2ccccc2)=O)C1 N1(C(c2cc(N)c(Cl)cn2)=O)CCC(F)(F)C(CNC(c2ccccn2)=O)C1 N1(CC)CCN(C(=O)C(c2cccs2)NC(c2coc(C)n2)=O)C(C)C1 c1(C(N2CC(O)C2)=O)cc(S(N)(=O)=O)co1.CC1(C)CC1CC(=O)NC CCC(CCC(=O)NC1COCC1S)C(=O)OC(=O)Cc1ncccc1F C(=O)(C1=Cc2ccccc2C1O)N1CCN(C(C(=O)N(C)C)=O)CC(C)(C)C1 c1(C=O)ccc(S(C)=O)cc1.N1(C(c2n(CC)ncn2)=O)CC(C)CC1(C)C.N N1(C(CCCOC(C)=O)=O)C(C(=O)N(CC(O)C2CC2)C)CCC12CC2 N1(C(C(C)C)Cc2nn[nH]n2)CCC(c2ccccc2)CC1CO C1(C(=O)NC(CC)CNC(=O)C(O)CN(C)C)(N(C)C)CCOCC1 C(=O)(C(C)(F)C(F)(F)F)N1CCOCC(NC(c2ccc(C)c(F)c2)=O)C1 N1(C(C(CSC)(C)NC(=O)Cc2cc[nH]c2)=O)CCSC2(CCC2)C1 c1(C(N2C(CCC)CN(C(C3COC(=O)N3)=O)CC2)=O)n[nH]c2nccc(Cl)c12 N1(C(C(=O)NC(C2CCC(N3CCOCC3)CC2)=O)=O)CCC2(C1)OCC1CC21 N1(CC(C)NC(c2ccncc2)=O)CCN(C(C2CCC(=O)N2)=O)CC1 N1(C(C=CCN(C)C(C2(O)CCOC2(C)C)=O)=O)CCOC2(CCCC2)C1 c1(OC)ccnc(-n2cc(CC3CCCC3NC(c3c(C)ncn3C)=O)nn2)n1 C1(NC(C2CCN(C(C(C)C)=O)CC2)=O)CCN(C(=O)C2CC2)C(C2CC2)C1 N1(CCn2c(C)ncc2)CC(=O)N(CC2C3CCC23)C1=O Cc1cc2c(cc1C)C(C(=O)NCCC(C)NC(=O)C1=CCOC1)CO2 C1(C(N(CCCN(C(C2C(C)CC2)=O)C)C)=O)CCN(Cc2ccccn2)CC1 N1(C(c2cc(OC)no2)=O)CC2CCC1C(NC(=O)C(C)(C)N1CCOCC1)C2 c1(C(=O)OC)c[nH][nH]c1=NC(=O)C12CC1CN(C(c1cc(C)n(C(F)F)n1)=O)C2 CCCC(F)C(=O)NC(C)CCCCNC(c1ncn(CC)n1)=O CC1CN(C(c2cc(F)c[nH]2)=O)CC1CCNC(c1cccnc1O)=O c1(C(N(C2CCN(C(=O)CCn3cncn3)C2)C)=O)cnc(O)c2cncn12 C(=O)(C(C)(C)CF)N(CC(C)(C)CNC(=O)C(C)CC1CCCC1)CC C(=O)(CC(c1nccs1)NC(N1CCOCC1)=O)OC.c12cc(no1)CO2 c1(C2C(C=O)C2)ccc(O)cc1.C1(N(C)C)CC(C(=O)NCC)C1.C1CC1 c1(C(=O)OCC)cccnc1NCC(CC)NC(=O)Cc1cnc(CC)[nH]1 C1(O)(CC(=O)Nc2cncc(Br)c2)CCN(C(=O)COC2CCCCC2)CC1 C12(OCC)CN(C1)C2=O.C1(CNC(c2cocn2)=O)(OC)CCOC1 CCC(CC(C)C)C(=O)NC(C(=O)N(C)CC1CCCN1C)c1ccco1 Cc1cc(C(=O)NCC2CCN2C(=O)C)cc(C)c1.[SH](=O)(=O)C1CC1.N c1(C(C)(F)F)ccc(Cl)c(NC(=O)Cc2scnc2-c2ccccc2)c1 N1(C(C(CNC(CC(CC)(C)C)=O)C(C)C)=O)CC2CCC(O)C2C1 n1(CCC)ccc(C(N2CCC2(C)CC(=O)N(CCF)CC)=O)n1 CN1CC(C)(C)CC1C(=O)NCC.c1ccc(F)cc1.C(=O)(C)N.C1CC1 Cc1cnc(C(=O)NC(C)Cn2cc(C3CCCN3C)nn2)n1C CCC(CC)(C(=O)NCC#CCNC(c1csc(C)c1)=O)OC Cc1ccc2c(N(CCCN3CCCC3)C)nc(=NC(C)c3cc[nH]n3)[nH]c2c1 N1(C(C2N(C(C)=O)CSC2)=O)CC(NC(=O)CCCc2nccs2)C(C2CC2)C1 C1(C(N(CCNC(c2c[nH]cc(F)c2=O)=O)CC)=O)Cc2cccnc2C1 N1(C(C2=C(C)CC2)=O)CC(C)(C)OCC1CNC(=O)CC(C)n1cccc1 CC(CC(=O)NCC1CN(C(=O)CC2CCC2)C1)C1CC1 c1(C(=O)NCC(CNC(CC2N(C(C)=O)CCC2)=O)C)ccc(Cl)c(Br)c1 CCC(C)(C(=O)N(CC(n1cc(CO)nn1)C)CN1C(=O)COCC1=O)C(N)=O S(=O)(=O)(c1ccccc1)N1CCN(CC=O)CC1.n1(C(C)c2ccco2)ccnc1C CCCCC(O)CC(=O)NCC1(C(=O)N)CC2(CC2)C1.CCCN(C)C1CC1 c1(CC(=O)NCCN(C(=O)CC2CC3CCC2C3)C)ccnc(O)c1 Cc1cc(C(=O)NC2(CCCNC(c3cc(Cl)ccn3)=O)CC2)c(O)c(C)n1 C1(NC(N2CCCCC2CC(C2CCCCC2)=O)=O)C2CCC1(c1cnco1)C2 N1(C(c2c(C)csc2)=O)CCC2(CC1)CC(NC(c1cnsc1C)=O)CCO2 CC1CN(C)CC(c2nc(-c3ccnc(-n4cncn4)c3)nn2CCF)O1 c1(C(=O)NC(C2CCCN2C(=O)C2=NOC(C)C2)C)ccc2c(c1)nc(O)n2C c1(CN2CCC(C(=O)Nc3cc(C(=O)OC)ncc3)C2)c(Br)ccc(Cl)c1F C#CCC(C)(CC)C(=O)N1CC(O)CC1C(=O)N(C(C)CC(N)=O)C C(C1=CCN(C(=O)Cc2c(C)cccc2F)CC1)NC(C1(CC)CCCO1)=O C(=O)(C(C)S(N)(=O)=O)N1CCC(OC)(CNC(=O)Cc2ccno2)C1 c1(C(=O)NC(C2CCCN2C(=O)CN2CCCC2=O)(C)C)ccc2[nH]ccc2c1 c1(C(CC)NC(=O)NCc2nc(-c3ccco3)oc2C)ccc(F)c(F)c1 CCC(COC)C(=O)N(CC(O)CNC(=O)CCn1cccc1)C c1(CC)ccccc1CNC(c1cscc1)=O.C1(C=O)CCC1.C1CC1.C C1(CCNC(c2cnnn2C2CC2)=O)CCCN1C(=O)CC(Cl)Cl Cc1cc(NC2CCC(C)(C)C(C)C2)ncc1S(=O)(=O)NC1CC2(CC2)C1 C1(c2n(CC)nnn2)(Nc2ccc(Oc3ccncc3)cc2)CCCOC1.C1CC1 C(=O)(C1=CC2(CCOCC2)C1)N1CCN(C(C2(S(C)(=O)=O)CC2)=O)CC(C)(F)C1 C1(C(=O)NC2CC(C)OC2=O)CC2CC1CC2NC(c1cnc(O)o1)=O C1(C(N2CCC(N(C(=O)C(F)=CC3CC3)CCO)C2)=O)CCn2cnnc2C1 c1(N(C)Cc2ccc(Br)cc2)nc2cc[nH]c2c(=NC2CCC2N2CCCC2)[nH]1 c1(NCC(CC)(CC)NC(=O)CC2CCCNC(=O)C2)cc(=O)n(C)c(O)n1 c1(CN2CCC(N(CC(CC)C)C)C2)cccc2c1OCC2 N1(C(c2cc(C(=O)OC)no2)=O)CC2CC2(NC(c2ccco2)=O)C1 Nc1ccc(Cl)cc1C(=O)Nc1cccc(NC(C2(F)CC3(CCC3)C2)=O)c1 S(=O)(=O)(c1c(Cl)cc(F)cc1Br)NCc1ccc(CCC(=O)OCC)cc1 c1(C(=O)NCC2OCCN(C(CC(=C)Br)=O)C2)cccc2c1OC(C)C2 CCC(CC)C(C(=O)NCc1ccoc1C(=O)NC(CC)CC)OC N1(C(CCSCCCC)=O)CCOCC(CNC(=O)CCc2cc(C)[nH]n2)C1 C1(CC(N2C(CCNC(c3scc(C)c3C)=O)COCC2)=O)CC2CCC1CC2 C(=O)(N=c1[nH]oc2ncccc12)C1N(C(c2ccc3c(c2)NC(=O)C3)=O)CC=C1 N1(CC(=C)Br)Cc2ccccc2CC1CNC(=O)CCCNC(N)=O C(=O)(CC(F)(F)C(F)F)N(CCC(=O)NCCCN(C)OC)CC=C C(C(CC1CCCC1)C(=O)N1CCOCC1CCO)NC(c1cc(O)ncn1)=O c1(OC)c(NC(N2CCCCC2c2nc[nH]n2)=O)cccc1C#N c1(CNC(CCN(C(=O)CC2CCC(O)C2)CC#C)=O)cc(C)ccn1 C1(C(N(CCN(C(c2nc(C(C)OC)sc2)=O)C)C)=O)CCc2c[nH]nc2C1 C1(CNC(c2nc(OCC)oc2)=O)CCN(C(=O)C(C)O)CC1O C1(C(=O)NCc2cnn(C)c2C)(COC)C=CCN1C(=O)CC(C)C C1(C=O)CCC(=O)N(C(C)C)C1.C1(C=O)CC1(F)F.CC=CC.CO.C c1(CN2C(C(=O)Nc3cc(OC)ncc3F)CC(F)C2)c(F)ccc2occc12 N1(C(c2c(CC)nn[nH]2)=O)CCOCC(C(=O)NCCc2ccnc(OC)c2)C1 Cn1ncc(S(N)(=O)=O)c1C(=O)NCC(C)(C)NC(=O)Cn1ccnn1 n1(COC)nc(C)c(NC(C2CCC(NC(c3ccc(I)cc3)=O)CO2)=O)c1C c1(C(=O)NC2CN(C(C(C)c3ccco3)=O)C(C)(C)C2)cc(F)c(F)c(N)c1Cl c1(OC)cc(C(N2CCOC(C(C)NC(c3c[nH]ccc3=N)=O)C2)=O)ccc1Cl C(CC(=O)NCCC1CCCN1C(=O)CN(C)CCO)(C1=CCCC1)OCC C1(C)(CCNC(C(C)(C)OCCC)=O)CCN(C(c2cn[nH]c2C)=O)CC1.C N1(C(CC(c2c(F)cccc2F)NC(C)=O)=O)CC2(C)CC1C2.C(=O)(C(C)C)N CC(C)C(C(=O)N(C1(C(=O)N(C2CCCC2)C(C)C)CC1)C)n1cncn1 C1(c2n(C)ccn2)CN(C(C2CCC(=O)C2)=O)CCN1C(=O)C(F)=CCCF CCCC(O)CC(=O)NC1CCCC1CNC(=O)CCc1ncc(C)[nH]1 C1(O)(CN(C(C(C=C=C)C)=O)C)CCCN(C(C2(S(C)(=O)=O)CC2)=O)C1 c1(COC)ncc(C(=O)N(CCC)C)c(=N)[nH]1.n1(CC(=O)N)ccc(C)n1 N1(C(C(=O)NCCN2CCCC2=O)=O)CCNC(=O)C12CCCCC2 N1(C(c2cn(CCC)nn2)=O)CC2(CC2)CC1C=O.C1CC(C(F)(F)F)C1.N Cc1cccc2c(C(N3CCC(N(C(=O)Cc4ccc(Cl)cc4)C)C3)=O)n[nH]c12 O=c1cc[nH]c2c(CNc3ccc(C(N4CCNC4=O)O)cc3)cccc12 C#CCC(C)(C(=O)N1CCC(C2(C)N=N2)C1)NC(C1CCC(C)C1)=O Cc1cc(CNC(=O)C(F)C(C)C)cc(O)c1.C(C(F)(F)F)=CC(=O)N C#CC(C)(C)C(=O)N1CC(O)(CCNC(=O)C(CC)n2cccn2)C1 C1(COCC(=O)NC(c2ccccc2)CCO)CCOCC1Oc1ccccc1 C1(NC(C(C)Cc2cccc(Cl)c2)=O)CN(CCc2cnn(C)c2)CC1(C)C c1(C(=O)NCC(C)CNC(C23CCCN(CCC2)C3)=O)cc2ccncc2o1 c1(CN)cccc(NC(=O)C(=O)NCC2CCC(c3ccccc3)O2)c1 CC1(NC(=O)CCCCNC(C2(C)C=CCC2)=O)CCCCC1 c1(CN2CCCC(C(=O)Nc3cncc(C)c3)CC2)cccc2c1OCCO2 c1(CNC(c2n(CC=C)nnn2)c2ccc(I)s2)cncc(C(=O)OC)c1 N1(C(c2ccn(CC)n2)=O)CCC2(CCC2)C1.c1(C(=O)N)cncc(N(C)C)c1 CC1(CC(=O)NCCC2CCCN2C(=O)CC2(N(C)C)COC2)CCCC1 N1(CC)CC(N=c2[nH]c3c(c(=NC4CCCc5c(F)cccc54)[nH]2)COC3)C1 C1(NC(c2ccc(CC)s2)=O)CCCOC12CCN(C(=O)C(C)(CC)CO)CC2 C#Cc1ccc(CC(N2CCSCC2C(=O)NC2C(O)C3CCOC23)=O)cc1 N1(C(C(N2CCCC(C)C2)=O)=O)CCN(C(=O)CCNS(C)(=O)=O)C(C)C1 C(C)(C(C)C(C)C)NC(c1c(CC)cncc1)=O.c1(C(=O)N)cc2cscc2s1 C1(SCC(=O)OC(C(=O)NC2CCOCC2)C2CC2)CCC=CCCC1 N1(C(C2CC3(C(OC)CC3)C2)=O)CCC2(CC1)CC(NC(=O)CCCN=[N+]=[N-])C2 C(=O)(C(O)C(C)(C)C)NC1CC(NC(CC(C)CF)=O)C1 CCC1=NOC(CC(=O)NC(C)CO)C1.C1(c2ccccc2)(C(=O)N)CC(=O)C1 CC1CC2(CC(C(=O)NC(CCF)C(=O)N3CC(NC(N)=O)C3)C2)C1 CCCC(C(=O)N1CCC(C(=O)NC2(C)CC(F)C2)(CC)C1)N(C)C N1(C(CC2CCN(OC)CC2)=O)CCC2CCN(C(=O)CO)CC2C1 C1(C2CCCCO2)(C(=O)NCCCC(C)NC(CCOC(C)C)=O)CCOCC1 N1(C(C2CC(=O)C23CCC3)=O)CC2COCC2(c2ccccc2)C1 C1(c2nc[nH]n2)CCCN(C(c2ccc(C(N)=O)nn2)=O)C1.NC(=O)C(=O)NC c1(NC(=O)N(CCCn2cc(CO)nn2)CCO)nc(C(F)(F)F)cs1 C(CC(O)C(=O)NC(C)(C)C(O)CO)NC(C(C)C#N)=O c1(C(=O)NCC2C3CN(C(CCCCN(C)C)=O)CC32)cc(N)c(F)c(F)c1F CC(O)C(C)(C)C(=O)NC1CC(C)(C)C1.c1(C=O)ccc(-c2cc[nH]n2)s1.N CC1CN(C(=O)CC2CSC2)CCN1C(c1cccnc1)=O C1(OCC(N)=O)CCN(C(c2ccn(CCNC(c3cc[nH]n3)=O)c2)=O)C1 C1(C(=O)NC(C2CCCC2)C#C)C(NC(=O)CCCC2CC2C)C1(C)C Cn1cc(OCC(=O)NCC2(F)CC(NC(=O)C(F)n3ccnc3)C2)cn1 c1(C(N2C(C)CC(NC(=O)CC3(C#N)CC3)CC2)=O)ccc(=O)n2c1CCC2 CC(CC(C)(C)C)C(C(=O)NCCN1CCOCC1)N1CCc2nn(C)cc2C1 C1(F)COCCN(C(c2cc[nH]c2C2CC2)=O)C1.NC(=O)CSCC(=O)N.C CN1N=C(CC(=O)N2CCC2CNC(c2cc(C(N)=O)no2)=O)CC1=O C#CCCCC(C)C(=O)N1CCCCC1CNC(=O)Cn1ccnn1 Cc1cnc(NC(C2CC3CC3N2Cc2cccc(CC(=O)O)c2)=O)nc1Cl c1(C(N2CCC(CC)(NC(c3ncccn3)=O)CC2)=O)cnn2c1C(C)CCC2 C1(CC(N2CCC2)=O)CC(C)(C)OC(C)(C)C1.c1(SC)ccsc1C(=O)N N1(C(c2cn(CCC)nc2C)=O)CCN(C(C2CCO2)=O)CC(CO)C1 C1CN(C(=O)Cn2ccnn2)CC2CC12.c1(C(=O)OC)ccc(C=CC=O)o1 N1(C(CC2(C#N)CC2)=O)CC2(CCC2)CC1C(N1CCCCCCCC1)=O c1(NC2C(NC(=O)OC(C)(C)C)CCOC2)ncc2[nH]ncc2n1 C1CN(C(C2(n3nccn3)CC2)=O)CC1(F)F.C(C=O)=CCN(CC)CC c1(C(N2CC(CC(=O)NC3(C(N(OC)C)=O)CC3)OCC2)=O)occ2c1CCCC2 c1(C(=O)NC2CC(C)(NC(c3csc(CO)n3)=O)C2)ccccn1.C1CC1.O CCC(C)(CC)C(c1nnnn1CC1CCCO1)NCC(C)C(F)F c1(OC)ccc2c(C)c(C(N3CCN(Cc4cccnn4)CC3)=O)oc2c1OC C(=O)(CN=c1[nH]c2ccccc2s1)N1C(CNC(C2(C)C(C)C2)=O)CCC1 CCCCC(C(=O)NC(c1nc[nH]n1)C1CC1)NC(c1cn(CCC)nn1)=O C1(C)C(=O)N1.C(C)(C(=O)N(C)C)N(C(C=CCCC)=O)C c1(CC(=O)NC(C(C)C)CNC(=O)CCc2cnoc2)c(F)cccc1C#N Cc1cccc2c1N(C(=O)NCCC1(C)CCCO1)CCCC2 Cc1cc(N2CCC(n3cc(Cl)cn3)CC2)nc(=NCCc2ccncc2)[nH]1 C1(CCC)CN(C(=O)C(C)(COC)CC)CCN1C(c1cc(OC)cnc1F)=O c1(OC)ccc(F)cc1C(=O)N.C1(C=O)COCC(C)(C)O1.C1(C)CCC1.C c1cnn(-c2ccccc2)c1.C(CCO)NC(C1(COC)CC1)=O.C(=O)C.N c1(SCCC(N2CCC(C)(NC(C(F)=C(C)C)=O)CC2)=O)ncnc2[nH]cnc12 O=C1NC2(C(=O)NC3CCC3)CC3CC1C2C3.C1(C(=O)N)CCCC(F)(F)CC1 C1(C2CCC2)(C=O)CC1(F)F.C(CC1CC1)(C(=O)N(C)CC1CC1)OC CC1(CNC(=O)C(=O)NCc2cccc(-c3ccccc3)c2)CCCC1O c1(C(N(C(CNC(C(C)OCC=C)=O)C)C)=O)c(F)ccc(O)c1F C1(C(=O)NCC2(C(N(C)Cc3ccccn3)=O)CC=CC2)CCCOCC1 c1(CC(=O)NC(C(=O)NCCC2CCC2)C2CCC2)nc(O)n[nH]1 N1(C(C2(CNC(C3CCCC(C)CC3)=O)CC2)=O)CCC(C)(C#N)CC1 C1(C(=O)NCC(=C)CC)CC(C(F)F)(NC(=O)OC(C)(C)C)C1 Cc1cc(CN2CCN(C(=O)Nc3cc(C(N)=O)ccn3)C(=O)C2)c(C)cc1O c1(CNC(C(C)N(C(Cn2c(C)nnn2)=O)C2CC2)=O)cc(Cl)ccn1 c1(C(=O)NC2CCC(NC(C3(C)CNC(=O)C3)=O)C2)ccc2cnccc2n1 Cc1nc2c([nH]1)CN(C(C1(F)CCN(C(c3cncc4[nH]ccc34)=O)C1)=O)CC2 C(=O)(C1CCCc2sccc21)NCCOCCNC(C1(C#N)CCN(C)CC1)=O C1(C(N2CCC(c3ncncc3F)CC2)=O)(OC)CCCC(C)(C)C1 C=CC(C)(C)CC(=O)NC1CC(C)(NC(=O)Cc2coc(C)n2)C1 C1(NC(c2n(CCC)nc(C)c2)=O)CN(C(=O)C=CCCC(C)C)CCC1C C(=O)(C(CO)(CO)NC(=O)Nc1cccc(NC=O)c1)OC c1(C(N2CCC(N(C(c3cccc(CCC)c3)=O)C)CC2)=O)cnn(C)c1C#N CCC(CC)CCC(=O)NC1CCN(C(c2cc(C(C)C)n(C)n2)=O)C12CCC2 c1(C(=O)NC2CCC(NC(c3c(F)ccc(N)c3)=O)CC2)ccc2n[nH]cc2c1 N1(C(C(C)NC(C=C)=O)=O)CCC2C1CCN2C(c1ccc(N(C)C)cn1)=O N1(C(c2cc(C)cc(C)n2)=O)CCC12CCN(C(c1cnccc1C#N)=O)CC2 C1(CC(=O)OCC)(C=O)CCCCC1.C1(C=O)CC(C)CO1.CC.CC.N N1(C(CCCN(C)C(c2cccn3cncc23)=O)=O)CCOCC(C)(F)C1 CN1CCC(C(N2CCC(OCC(=O)NCCC(C)(C)CO)C2)=O)CC1 Cc1cc(C(c2nnnn2C(C)(C)C)NCc2ccc(Br)c(Cl)c2)nc(Cl)c1Br N1(C(=O)CSc2cc(F)ccc2F)CC2(CCN(C(C3CCCCC3)=O)CC2)C1 Cc1cc2c(CC(=O)NCC(C)(C)CNC(c3cnc(S)nc3)=O)csc2s1 C(=O)(CCC(F)(F)F)NC(C1CN(C(C2CCC2c2ccc(F)cc2)=O)C1)C N1(C(=O)CC2CC(O)CN2C(c2ccsc2Cl)=O)CCn2cncc2C1 N1(C(C2(C)CCN(Cc3c(C)cccc3)CC2)=O)CCc2ccc(Cl)cc2C1 N1(C(Cc2c(C)con2)=O)CC(NC(=O)C(C)CC(C)(F)F)C2(CCC2)C1 C1(CCNC(CCOCCN(C(C(C)=CC2CC2)=O)C)=O)CCC(C)O1 C1(COC)CN(C(=O)C(C)(C)n2cnc(C)c2)CCN1C(c1cc(C)sc1C)=O C1(NC(C(CC)C)=O)CCCCC12CCN(C(c1cc(C)[nH]c1C)=O)CC2 c1(NC(C2CCCN(C(=O)C(Cl)(Cl)Cl)C2)=O)ccc(Cl)c(Br)c1 c1(C(=O)NC2C(CC)N(C(c3sccc3OC)=O)CCC2)ccc2c(c1)COC2 CCCC(C#N)C(=O)N(CC(=O)NCCC1CCC(=O)N1)C(C)C c1(C(N2C(CNC(C=COCC)=O)CC2)=O)ccc(-c2csnn2)cc1 Cc1cc(F)c(CN2CCC(NS(=O)(=O)c3ccncc3)C2)c(Br)c1 c1(CC)cccc2c1OCCC2NC(=O)NCCCN(C)C(C1CCC1)=O N1(C(C(C2CC2)OC)=O)Cc2ccccc2C(Nc2nnc(O)s2)C1 Cc1c(NC(=O)C(C)Sc2ccccc2)cccc1C(=O)Nc1nc(Cl)sc1Cl c1(C(N2C(C)CC(CNC(CN(CCOC)C)=O)C2)=O)ccn2ccsc12 c1(CCC=O)cn(CC(F)(F)C)nn1.C1(CC=O)(CC(=O)O)CC1(C)C.C c1(C(=O)NC)cccc(C(=O)N(C2CCC(Nc3ccncn3)CC2)C)c1 c1cncc(C)c1.C12(C(=O)Nc3cc(C(=O)OCC)[nH]c3)CC1CN(C)C2 N1(C(=O)OCC)CCC(C(=O)NCCN(C(c2cn[nH]c2)=O)CC)CC1 C1(C)CCCCO1.n1(CC)ccnc1C(c1cccnc1)NC C1(NC(c2c(C)n(CCO)nc2)=O)COC2(C1)CN(C(C1CCCN1N=O)=O)C2 N1(C(C(C)N2CCC2)=O)CCC(C2CCN(C(=O)C#CC3CCCCC3)CC2)C1 N1(C(c2c(C)ccnn2)=O)CC(C)CN(C(c2sc3nccn3c2C)=O)CC1C Cc1nc(O)ccc1C(=O)NCC(CO)NC(=O)C(F)CC1CCCC1 N1(C(C(CCCOC)N)=O)CCCC12CCC(C)(C)CC2 C1(CNC(c2c(C)noc2)=O)CCN(C(C2CC(O)CN2C)=O)C1(C)C C1(NC(C(C)=CC2CC2)=O)CN(C(C2(C3CCOCC3)CC2)=O)CC12CCC2 C(CC(C)(C)CC(=O)N1CCN(C(C2CCc3cnnn3C2)=O)CC1CO)OC N1(C(CC2(OCC)CCC2)=O)CCC2(CC1)CC2C.c1(C=O)nccc(C)n1 c1(OCC)cnc(C(=O)NCCCCCN(C(=O)Cc2ccsc2)C)c(Cl)c1 N1(C(CNC(N)=O)=O)CC2(CCCC2NC(c2coc(O)n2)=O)C1 N1(C(c2c(C)cccn2)=O)CCC(C)(NC(C2CC(F)(F)C2(C)C)=O)CC1 C1CC2(CCN(C(C3(C4(C)OCCO4)CC3)=O)C2)CO1.C(CC(=O)N)=CC=C C(=O)(CC(C)NC(C1(NC(c2cncn2C)=O)CCSC1)=O)NC C#CCCCCCCC(=O)NCCC(CNC(C1CN(C)C1)=O)OC N1(C(C(C(C)C)(C)O)=O)CCOC2(CCC(NC(C34CCC(CC3)C4)=O)CC2)C1 C1(n2c(C(c3ccccc3)C)nc(-c3ccc(OC)cc3)n2)CC(C)OC(C)C1 N1(c2ccc(NC(CC)C(c3cc(OC)ccn3)=O)cc2)C(=O)CCCC1=O CCCC(CC(=O)NC(c1cccnc1F)C)NC(C1CC1(C)C)=O C(=O)(CCC(C)(C)[N+](=O)[O-])N1CC(C)(C(N(C(CC)C2CC2)C)=O)C(C)C1 C=CC(C)(C)C(=O)NCC(C1CCCC1)NC(=O)CSCCC C(=O)(C1CCc2c[nH]nc21)N1CCN(C(C(c2ccc(C)o2)C)=O)CC(O)C1 C1(NC(CC2CC(=O)C2)=O)CN(C(c2c[nH]c3nccc-3c2)=O)CC2CCCC12 c1(-c2nc(C3NCC(C)(C)C3)on2)cnn2cc[nH]c12 c1(N2CC(=O)N3C(C2)CCCC3)nc2c(c(=NCCN3CC=CC3)[nH]1)COCC2 Cc1ccc(Cl)cc1NC(C1(NC(C2CCSC2)=O)CCCC1C)=O C1(C(=O)OC)CN(C(=O)CC2CCC3(CC3)CO2)C2(CCCOC2)C1 C(C(C(=O)NCC(C)(O)CNC(c1n[nH]c(C)c1C)=O)C(F)(F)F)OC C(=O)(N=c1[nH]oc2cnccc12)C1N(C(C(C)C)=O)C2C(C1)CCCC2 N1(C(C2CCOC2)=O)CCCC2(CCN2C(c2ccc(Cl)nc2)=O)C1 c1(C=O)ccc(S(C)=O)cc1.C1(C(=O)OC)CC1C(=O)N(CCC)CCO n1(CC=O)cc(Cl)cn1.C(=O)(C(C)(c1cccs1)N(C)C)N(CC(C)C)C.N c1(OC)ccc(C(CNC(c2ccnnc2O)=O)NC(=O)C=CC)cc1.O C=C(C)C(CC(=O)Oc1ccc(OCC)cc1)OCc1nccc(C)n1 CC(C)CC(C)CC(=O)NCCN(C(=O)CNc1ccccc1Cl)C(C)C CN1CCC(C)(C(N2CCCCC(CNC(c3ccc(C(F)F)s3)=O)C2)=O)C1=O CCCCC(C(=O)N1CC(OCC)C1)NC(=O)CN1CCC(=O)CC1 C=C(Br)CC(=O)N(CCC(C)NC(=O)Cn1cncn1)C C(C1c2ccccc2CN1C(C1OCCC1(C)C)=O)NC(CCC)=O N1(C(C=C(C)c2ccsc2)=O)CCOCC(C)(CNC(=O)CCCCC2CC2)C1 c1(CC(=O)NC2(CO)CN(C(C3CC(C)C3)=O)C2)ccc(C(F)(F)F)cc1 N1(C(C2(CSC)CCC2)=O)CC2(CC(CC=O)C2)C1.C1CCOC(C(C)C)C1 Cc1nc(Cl)ccc1C(N1CCC(C(C)NC(c2cc(Cl)nnc2Cl)=O)CC1)=O C1(NC(C=C(C)C)=O)CC12CCN(C(c1cccnc1SC(F)F)=O)CC2 C(C(C)(C)CC(=O)NCC1CC(NC(C2(F)CCCC2)=O)C1)N(C)C c1(C(N2CC3C(C(N4CCS(=O)(=O)CC4)=O)C3C2)=O)ccc(Br)c2cc[nH]c12 n1(CCCC)nnnc1C(c1sccc1C)NC(c1nc(C)cs1)C [SH](=O)(=O)c1ccccc1.C1C2CN(C(=O)CC)CC12.C(=O)(CC(=O)N)OC.C N1(C(C(=O)NC(c2ccccc2)C)CCC2CC2)CC2NC(=O)OC2C1 C1(NC(c2cnsn2)=O)CCCC(NC(C2CCC(C(F)(F)F)O2)=O)C1 c1(C(N(C)CC2CCN(C(c3cc(C)cc(C)c3)=O)C2)=O)cn(C)c(C)cc1=O C1(C)(CNC(C(C)(C)C2CCOCC2)=O)CCN(C(c2cncs2)=O)C1 C1(C=O)Cc2c(C)cccc2O1.c1(SCC)cncc(C(=O)NC(C)CC)n1.N c1(CC)nc(C)n(C)c1C(=O)NC1CC(F)C1.C(=O)C(C)C(C)(C)C.C c1(C2N(C(C(NNC(C)=O)=O)C)CCC2)ccc2ccccc2c1 N1(C(c2c(CC)[nH]cc2)=O)CCCN(C(=O)C(C(C)C)NC(C)=O)CC1C C(=O)(CC(C)(C)C(F)(F)F)NCCN(C)C(C1CC12CCCOC2)=O CCCCCC(CC)C(=O)NCC1(CNC(c2c[nH]c(C#N)c2)=O)CCCC1 C#CCCN=C(NCc1c(C)coc1C)NCC1(OC)CCCSC1 N1(C(CCCSC)=O)CCCCC1CCC1CCCN1C(=O)CC(=O)N(C)C CC1C(NC(=O)CCC2CC2(C)C)CCCN1C(=O)CC1CCC(=O)N1 c1(CC)nc(C(=O)NCCCN(C(=O)C(O)CN(C)C)C(C)C)cs1 C#CCC(O)C(=O)NC1(CNC(=O)Cn2cncn2)CC1 CCCC(C)(O)CC(=O)NCC1CN(C(=O)C(c2cscn2)N(C)C)C1 N1(C(CC2CCCN(C)C2)=O)CCCCC(N(C)C(C2CC3CCC2CC3)=O)C1 N1(C(C2C(C)(C)N(C(C3CC=CC3)=O)CC2)=O)CCCC(C)(O)CC1 c1(C(N2CCC(NC(CC(CC)SC)=O)C(O)C2)=O)c(C)ccc(Cl)c1F c1(NC)ccc(C(=O)NC(C)C(C)NC(C2(n3cccc3)CCOCC2)=O)nc1 C(CN=c1ncc(C(N)=O)c[nH]1)=CCNC(c1ccc(OC)c(OC)c1)=O Cc1csc(C(N2CC=CC2CNC(=O)CCOCC2CCCO2)=O)c1 c1(SC)nc(C)cc(=NCCCONC(=O)OC(C)(C)C)[nH]1 CC1CC(C(=O)NC2CCN(c3ccc(OC(F)F)cc3)CC2)OC1C(=O)O c1(C(=O)NC2C(C(=O)NC(c3nn[nH]n3)CC)CCOC2)cc(O)nc(O)n1 c1(C(=O)NC2C(NC(c3cc(C)on3)=O)CCC2)cc(C)oc1C(F)(F)F Cc1cc(C)n(CC(=O)N(C)CCNC(C23CC(CF)(CO2)C3)=O)c(=O)n1 c1(C(N(CCNC(C2C(C)(COC)C2)=O)C)=O)ccnn1C1CCC1 CC(CC(=O)NC1CCCC(NC(c2ccc3n[nH]cc3n2)=O)C1)C(C)(C)C c1(C(=O)NCC(C)(C)NC(c2c(C)nncc2)=O)cc(O)cc(Cl)c1 Cc1cc(F)cc(C)c1C(=O)NC1CCN(C(C2CCC(O)CC2)=O)C1C1CC1 C(=O)(C(C(C)O)N(C)C)NC1C(CNC(C(n2cc(Cl)cn2)C)=O)COC1 C1(C(N(C)Cc2ccns2)=O)C(NC(=O)CCc2nncn2C)C1(C)C n1(CC(=O)NC(C(=O)NCCC)C2CCCO2)ccc(C)n1 c1(C(C)C)ccc(C(N2CC3CCC2C3)C(=O)NCCOCC2CC2)c(Br)c1 Cc1cc(C(N2CCOCC2(C)c2cn(CCF)nn2)=O)n2nccc2n1 c1(C(N(C)CC2CCN(C(c3nc[nH]n3)=O)CC2)=O)cccc2c1CCCO2 N1(C(=O)CC2CCCC(c3nn[nH]n3)C2)CCCC2(C=CCO2)CC1 c1(CC)cc(CC(=O)NCCC(O)C)n(C)n1.c1(C(C(=O)N)C)cccc(C)c1 C1(CCCC)CN(C(=O)CC(C)N(C)C)CCN1C(=O)C=Cc1cocn1 N#CC1(C(=O)NCCc2ocnc2C)CCOC1.C(=O)C=CSc1nc[nH]n1.N CCC(C)C(O)C(=O)N(CCNC(=O)CN1CCCNC1=O)Cc1ccccc1 N1(C(C2(CCNC(c3n(C=C)nnc3)=O)CCC2)=O)CC2CC3CC2C1C3 N1(C(COCc2nnc(C)s2)=O)CCCC(C2CCCN2C(=O)CC2CC2)C1 Cc1cccc(OCC(=O)N(CCCCN(C(=O)C(C)N2CC(C)C2)C)C)c1C c1(C(=O)NC2CC(CNC(C(C)(C)C3CCOCC3)=O)C2)cn2ncccc2n1 C1(NC(C(CCSC)NC(c2ccc(CC#N)cc2)=O)=O)CCOC(C)(C)C1 Cc1ccc2cc(C(N3CC(S(=O)(=O)N(c4ccccc4)CCO)C3)=O)[nH]c2c1 c1(C(N2CCCC(NC(=O)CC3CCC3(F)F)(CO)C2)=O)ccc([N+](=O)[O-])cn1 C1(CC)CN(C(=O)C(C)n2cnnn2)CCN1C(=O)COC.c1nnc(S)n1C C1(c2nnnn2CCCF)(Nc2c(C)ncc(F)c2)COCC(C)(C)C1 c1(C(=O)NC(C(=O)NC2C3COCC23)C2CCCC2)cncc(F)c1 c1(CCNC(CCOCCN(C)C)=O)cccc(Cl)c1.C1(C(=O)N)CCCOC1 C(CC(N=c1ccn2ccnc2[nH]1)C(C)C)N(C(C1N(CC)C(=O)CC1)=O)C C(c1cccc([N+](=O)[O-])c1)=CCOC(=O)Cc1ccc(I)c(Br)c1 C1(C=O)CCC(C)(C)CC1.C1(OC)CN(C(=O)C)CC1.c1(C(=O)N)ccoc1 C1(CNC(c2cccc[n+]2[O-])=O)CCN(C(c2coc(O)n2)=O)CC1(F)F CC1CCCc2c(C(N3CCCCCC3CNC(c3cnc(O)o3)=O)=O)cnn21 O=C(C1=CCCOCC1)NC1CC(O)CN(C(c2cn(C3CCC3)nn2)=O)C1 S(=O)(=O)(c1cc(F)ccc1Cl)NC(c1nccc(C)c1)C c1(CC)ccc(C)c(NC(C2CC2C(C)NC(c2[nH]cc(C)c2C)=O)=O)c1 c1(CCC(=O)NC2CC2NC(C23CCC(CC2)N3)=O)ccc2ccccc2c1O CC1CCc2ccccc2N1C(=O)CN1CCCCC(SC(C)(C)C)C1 C1(CCNC(N(CCOC(C)C)C(C)C)=O)COCCO1 C1(CCNC(CC)=O)CCN(C(=O)COCC(C)(C)C)CC1(F)F N1(C(C(=O)NCc2cccs2)C2C(CC)C2)CCOC(C2CCOCC2)C1 c1(C(N2CC(NC(CC(=O)NCC)=O)C2)=O)cc2c(F)c(F)c(F)cc2[nH]1 N1(C(Cc2c(C)cco2)=O)CCCC2CCN(C(C3SCCCS3)=O)CC12 CCC(CC)CC(F)C(=O)NCC1CC2CCC1N2C(C1CN(C(C)=O)C1)=O C(=O)(C(=O)N=c1ccn(C(C)COC)[nH]1)NC(c1ccc(F)c(F)c1)CC c1(C2(CNC(CCCn3cc(-c4c(C)ocn4)nn3)=O)CC2)cc(Cl)cc(Cl)c1 C(CNC(=O)C(C)(C)n1cccn1)(CCNC(=O)CC(C)N(C)C)OC C=CCCCCC(=O)NC1CC(CNCc2cccc(N3CCCC3)c2)C1(C)C N1(C(C(C)(C)OCC)=O)CCN(C(=O)CCCC(=O)NCC)CC(CO)C1 C#CCC(C)(C(=O)N(C)CCn1ccnc1)NC(=O)Cc1cccnc1O C(CN(C(=O)CC#N)C)(CO)(CO)NC(C1CC(SC)C1)=O c1(CNC(c2ccc(OC)cc2)c2cccs2)cnc2[nH]ccc2c1 Cc1cc(F)c(C(=O)NC(C)CN(C)C(C2C3(CC3)C23CC3)=O)c(Cl)c1 C1(C(=O)NC2CC(NC(C3CC(C#N)C3)=O)C2)CCC(F)(F)CC1 c1(NC2C(C)CN(C(=O)CCCN3CCCCC3)C2)cncc(C#N)n1 C(=O)(CCCC(=O)OC)NCC1(CO)CCN(C(C2CC(CCC)C2)=O)C1 CS(=O)c1ccc(C(N2CCSCC2CCNC(c2csnn2)=O)=O)cc1 C1(C)CN(C(c2cnc(Cl)s2)=O)C(C)(C)C1.Cc1cc(C)c(C(=O)NC)cn1 C#Cc1cncc(C(=O)NCC2CCCN2C(=O)CCC2(C)N=N2)c1 c1(C=O)ccc(N)c([N+](=O)[O-])c1.N1(CCNC(C2C(C)(Br)C2)=O)CCCCC1 c1(Nc2sc(C(=O)Nc3c(C)ccc(Br)n3)c(C)n2)ncnc2cc(Br)sc12 c1(C(=O)NCC2N(C(C(c3ccc(C)cc3)O)=O)CC2)cc2n(n1)CC(O)CO2 C(=O)(CC(C(C)C)C(C)C)N1C(CNC(c2cc(C)c(C)o2)=O)CC(O)C1 N1(C(C2CCCCC(=O)C2)=O)CCOCC2(CCSCC2)C1 Cn1c(C(N2CCC(CCC(=O)NCCC(O)C(F)F)C2)=O)nnc1S C1(NC(c2cccc(C)c2F)=O)CCN(C)C12CCCN(C(c1ccc[nH]1)=O)C2 Cc1nc2ccccc2n1CC(=O)NCC1CCCC1.C(=O)C(C)S(N)(=O)=O.N CCC(C)(C(=O)NCCC1(O)CN(C(c2c(N)cc(Cl)cc2Cl)=O)C1)C(N)=O C1(C2CC2)(CNC(=O)C=Cc2ccncn2)CCN(C(=O)Cc2nccs2)C1 C1(NC(=O)Cc2ccoc2)CC(NC(=O)Cc2c[nH]nc2O)C(O)C1 CC1CC(=O)NCC1C(=O)N(C)CCO.c1(C(N(CC)C)=O)ccc(C#N)[nH]1 c1(C(=O)N)cc2c(nn1)CCC2.CC(C)C(C(=O)NCC1CCCCO1)N(C)C N1(C(C2CC(OC)C2)=O)CCCC(C)C1CCNC(=O)Cc1ccsc1C N1(C(CC(=O)NCC)=O)CC(NC(=O)C(C)S)CC2(CC2)C1.c1ccccc1 c1(C(=O)NCC(C)(C)NC(CCCOC)=O)ccc(Br)c(C)c1F CC(C)CC(C(=O)NCC1(CO)CCN(C)C1)NC(C1CCC(=O)NC1)=O c1(CC(N2C(C(=O)NCc3cnc(C)s3)CC(C)C2)=O)cc(F)cc(F)c1F C12(CNC(CCOCC#C)=O)CC(CO1)N(C(C1(C)CNC(=O)C1)=O)C2 c1(N2CCN(C(CC)C)CC2)nc(=NC)nc(N2CCC(S(C)(=O)=O)C2)[nH]1 N1(Cc2ccc(N(C)C)nc2)CCCC(C(N2CCCC2C2(O)CC2)=O)CC1 c1(NC(=O)CC2CC(CNc3nccc(-n4ccnc4)n3)C2)c(F)cccc1F N1(C(C(C)SCCCC)=O)CCC2(CCN(C(c3cc([N+](=O)[O-])n[nH]3)=O)CC2)C1 C1(CC)(NC(c2ccc(C)cc2C)=O)CCCN(C(=O)C(C)O)C1 Cc1cccc(Br)c1C(C(=O)NC(C)C(=O)NO)NC(c1csnc1C)=O CC1(C)C(C(=O)N(CC)CCc2ccccc2)C1(F)F.C(=O)(CCS(C)=O)N C(C(C)(O)C)NC1CN(C(=O)OC(C)(C)C)C1.C1(CC=O)CCCCC1.O c1(C(=O)NCC23C(NC(=O)C(Cl)=CCl)CC(CC2)C3)csc2ccccc12 N1(C(c2ccc(C)o2)=O)CCC(CNC(=O)CCN2CCN(C)CC2)C12CCC2 c1(-c2cn(CC3N(C(c4cnc(CCC)s4)=O)CC=C3)nn2)ccc(C)cc1C c1(CNC(=O)COC2COC2)ccccc1.C(=O)C(F)Cc1ccccc1.C C12(CNC(CSC)=O)CC(C1)C(NC(=O)CC1CSCCS1)CO2 C=C(C)C(O)CC(=O)N1CCC(C2CCCCN2C(c2cnn(C)c2N)=O)CC1 C(=O)(CC(CC)CC(C)C)N1C2CC(C(=O)NCC)C1CC2 C1(NC(c2c(=N)[nH][nH]c2)=O)CCCCCN(C(=O)C2=CCCOCC2)C1 N1(C(C(C(C)C)OC)=O)CC2CCN(C(c3cc(C)nn3C3CCC3)=O)CC2C1 c1(OC)nccc(C(N2CCN(C(C3CCCCS3(=O)=O)=O)C(C)C2)=O)c1F Cc1cc2nccnc2cc1C(N1CC2(NC(=O)C(O)C(C)C)CCC1CC2)=O c1(OCC)nc(C)ccc1C(N1CC=CC1C)=O.C(=O)CC.CCC(C)C.N c1(C(=O)NC2CC(C(=O)OC)C2)cncnc1.n1(CC=O)ccccc1=O.C c1(C(=O)NCC(C)CNC(=O)CN(C2CCC2)C)ccc(F)c2cnccc12 N1(C(c2nc(C)sc2C)=O)CCC2CC(C1)CN(C(c1cn(C(F)F)cn1)=O)C2 Cc1ccc(C2CC2C(=O)NC2CC(NC(=O)C(c3cccnc3)O)C2)cc1 c1(C(=O)NC2(C)CCN(C(c3ccc(OCCO)cc3)=O)C2)c(N)cccc1Cl CCCC(C(=O)N1CC2(CC2)CC1CNC(c1cncc(CO)c1)=O)C(C)C N1(C(C2(C)C(C)C2)=O)CCC(C)N(C(c2cc(C(N)=O)[nH]n2)=O)CC1 CC1CN(C(c2cn3c(n2)CCCC3)=O)C(C)CN1C(c1coc(C2CC2)n1)=O N1(C(C(=O)Cc2cccs2)=O)CC2CCCN(C(c3cncc4ccsc34)=O)C2C1 c1(C(C(=O)NC(CNC(c2nc(C)nn2C)=O)(C)CO)C)c[nH]c2ccccc12 CCCC(C(=O)N1CCN(C(c2ccnc3c2CCC3)=O)C(CC)C1)S(N)(=O)=O CC(CNC(=O)C(O)CC(N)=O)C(F)C(=O)N1CC(CC23CC(C2)C3)C1 C1(C(=O)NCC2CN(C(c3c(C)nc(CO)s3)=O)CC2C)CCC(C)(C)OC1 C1(C(=O)NC(C)CCN(C)C(C2CCCS2)=O)CCCCN1C N1(C(C=C(C)C(F)F)=O)CCC(NC(c2ccnc(-n3cccc3)c2)=O)C(C)C1 C1(NC(CC(CC)OC)=O)CC2CCC(C1C)N2C(c1cc(CO)[nH]n1)=O C=C(C)C(C)(C)C(=O)NCC1CCN(C(c2cc(C)c(F)cn2)=O)C12CC2 c1(C(=O)NCC(C)NC(C(CC2CCCCC2)OC)=O)ccn(CCO)c1C N1(C(C2C(=C)CC2)=O)CCOCC(NC(c2cc(CO)c(C)o2)=O)C1 N1(C(=O)NC(c2nccn2C)CC)CC(C)(OCC2CCCCO2)C1 CC1(C)CC(CC(=O)NCC(C2CCN(C(=O)C3CC3)CC2)(C)C)CC(C)(C)O1 c1(C(=O)NC2C3CN(C(C(C)CC(C)(C)C)=O)CC32)cccc2nn(C)cc12 Cc1cc2ccccc2nc1C(=O)NCC(C)CN(C(=O)C1=CCSC1)C N#Cc1cncc(-c2cn(CC3CCN(C(C4CC=CCO4)=O)C3)nn2)c1 C(=O)(CCCC(=O)NCC(O)CCNC(=O)C=Cc1cc[nH]n1)NCC C(=O)(CCCCCCc1ccccc1)N1CCC(NC(C(CC)=CCC)=O)C1C C(c1cnc(O)nc1O)=CC(N1C(CCCNC(c2cncs2)=O)CCC1)=O N1(C(CNC(c2cscn2)=O)=O)CCN(C(C2C3CCCOC23)=O)C2CCC12 C1(C(=O)NCC2CN(C(c3n[nH]cc3C)=O)C2)(COC)CCCO1 c1(COCC(=O)NCCC2CC(NC(C3CCC3)=O)C2)ccccc1.C C1(CC)C(C(=O)NCC(C)(O)C2CC2)CCCN1C(=O)CCO.C(N)(=O)N n1(CC(=O)NCc2scc(CNC(CCC(N)=O)=O)n2)nc(O)ccc1=O Cc1cn2cc(C(N3CCCCC3CNC(c3cscc3Cl)=O)=O)nc2s1 N1(C(COC(C)=O)=O)CCOC2(C1)CN(C(C1CC(C(C)(C)C)C1)=O)C2 C=C(Cl)CC(C(=O)NC(C)COC)NC(=O)CN1CC(C)(C)C1 C1(NC(c2cc(C)n(C)n2)=O)(CNC(=O)CCC2CCCO2)CC2CCC1CC2 c1(CC)cccc(C(=O)NC2CC(CO)N(C(=O)CCC3CCC3)C2)c1F C(=O)(C(CC)C(C)C)N1CC2C(CNC(c3cnc(OCC)s3)=O)C2C1 Cc1cc(C(=O)NC(C)CCNC(c2cncc3sccc23)=O)cc(C)c1F C12CCC(CC1)C2.N1(CC(=O)NC2CCN2C(=O)C(F)C2CCCC2)CCCC1 C1(CNC(=O)CC2CC(F)(F)C2)CN(C(=O)CC2CC=CCC2)CCC1(F)F C(CCNC(=O)CCCCN(C)C)(C(C)C)NC(C1(CC=C)CC=CC1)=O Cc1cccc(C(C)(C)C(=O)N(CCCCN(C(=O)CC(C)NC(N)=O)C)C)c1 C(C(C)(C(=O)N1CCOC(CN(C)C(c2cc(Cl)n(C)n2)=O)C1)OC)OC C(=O)(C1CCCc2c[nH]nc21)N1C(C(C)(C)NC(c2cc(C)sn2)=O)CCC1 Cc1nc(-c2ccc(Cl)cc2)sc1Sc1ccccc1CC1(SC2CCOC2)CC1 C(=O)C(F)(F)C(O)C(C)C.c1(COC)cncc(C(=O)N)c1.C(C)(CC)CC CN1CC(NC(c2ccccc2C(=O)NC(C)(C)C)=O)C(F)C1 C1(C)(OCC(=O)N(CC=C)CCOC)CN(C(C2C=CCC2)=O)C1.C C1CCN(C(C2(C)CNC(=O)C2)=O)CC1.N1(C(C)(C)C)CCC1C(=O)N.CC C1(C(C)C)CC(C(=O)NCC2CC2C(=O)N(C)CCOC(F)F)CO1 N(C1CCCc2n[nH]cc21)C(C1N(C(C2CC(N=[N+]=[N-])C2)=O)CCSC1)=O C=C(C)CCC(=O)N(C)CCN(C)C(c1ccnc(-c2ccccn2)n1)=O CC1Cc2cc(F)ccc2CN1C(C1CCSC1(C)C)C(=O)NC1(C)CC1 C1(NC(CCOC(C)=O)=O)CN(C(C2CCc3nncn3C2)=O)CC2(CCC2)C1 C1(OC)CN2CCCC2(C(=O)NCC2(C)CCC2)C1.C(=O)C.C(C)C.N c1(CNC(CN(C(c2ccnc(C)n2)=O)C(C)C)=O)c(F)cccc1F C1(C(N2CC3CC3C2)=O)CS(=O)(=O)CC(=O)N1.CCCCOCC(=O)N.C C1(CN(C)CC2(Cc3cccnc3)CC2)CCN(C(c2nnnn2C)=O)CC1 N1(C(C2C(CCC)C2)=O)CCCC(C)(C)C1.C1(CC=O)CC(N(C)C)C1.C c1(OC)ccc(O)cc1CN1CCCC(NC(=O)Cc2ccc(Cl)s2)C1 c1(C(N2C(CC)C(NC(=O)C(C)(F)F)CC2)=O)cc(OC)c(Cl)cc1Cl C(=NOC1CCC1)c1ccc(-c2ccccc2)c(C#N)c1 C1COC(C(F)(F)F)CN1C(C1(C(N)=O)CC1)=O.c1(CC)[nH]ccc1C=O c1(N(CCC)C(C2(N(C)C(c3ccns3)=O)CC2)=O)cncc(C)c1 c1(C(N2CCC(C(C)(C)NC(C(CSC)C)=O)C2)=O)ccc(C2CC2)cn1 c1(C(N2CCC(c3ncc[nH]3)C2)C(=O)NCC2CC2)cc2c(s1)CCOC2 C1(NC(CSC)=O)CC(=O)N(C2CN(C(C3(C)CCCC3C)=O)C2)C1 c1(C(N2CCC=C(Cl)C2)C(=O)NCCC2(C)CC2)ccn2nccc2c1 C1(CCOC)(NC(c2cnc(C(C)C)[nH]2)=O)CCN(C(=O)CCC=CBr)C1 C1(N(C)C)Cc2ccccc2N(C(=O)NC2CCCCC2F)C1 N1(C(c2cnc(C)s2)=O)CCC(C)(C)C(CNC(=O)C(F)(F)C(C)O)C1 c1(C(N2C(C(=O)Nc3ccc(Br)nc3)CC(O)C2)=O)ccc([N+](=O)[O-])nc1 C1(C)(CNC(C(C)=C(C)C)=O)COCCN(C(=O)C(c2cccc(Cl)c2)C)C1 Cc1oc(C(N2CCCC2C2CCN(C(c3cocn3)=O)C2)=O)cc1Br C(=O)(CCCC(C)(C)C)N1C2(CNC(C3CCN(C)C3=O)=O)CCC1CC2 N1(C(CNc2scc(C)n2)=O)CCC(NC(=O)Cn2ncnn2)C(F)C1 CC(C)C(CCC(=O)N(CC(N1CCCC1)C)C)NC(=O)CCC(F)(F)F CC1CCCC1(C(=O)NCCN1CC=CCC1)NC(C1C(C#N)C1(C)C)=O N1(C(c2cc(OC)n(C)n2)=O)CC2CCN(C(c3cc4n(n3)CCCO4)=O)CC12 CCC(C)(C(F)(F)F)NC(=O)C(CCF)NC(=O)COc1ccsc1 C1(CC)(NC(=O)CCc2ccncc2)CCCN(C(c2cnc(C)[nH]c2=N)=O)C1 C(=O)(C[SH](=O)=O)N.N1(C(C2CN(C(C)=O)C2)=O)CCC(n2cc(C)nn2)C1 C(=O)(C1OCCc2ccccc21)N1CCC(CC=C)(NC(=O)CC(C)(C)F)C1 c1(CCNC(=O)NCc2ccc(C(=O)OC)c(OC)c2)cnn2c1CCCC2 N1(CCNC(=O)CCC2CCCCO2)CCC(NC(=O)Cc2cnsc2)CC1 C=CCCC(C(=O)N1CCC(c2ccon2)C1)NC(=O)COC(C)(C)C C(C(=O)Nc1cncc(C(N)=O)c1)(C(C)O)NC(C(CSC)C)=O C(C(C)(C(=O)NCCCOCCNC(C1CC1(F)F)=O)OC)OC C(=O)(C(CCC1(C)CC1)N(C)Cc1ccn(C)c1)NCCC c1(CC)nn(C)c(C(=O)NC2C=CCN(C(=O)C(=O)Cc3cccs3)C2)c1Cl C1(C)(C(C)(C)C)CCCN(c2nnc(CCSc3ccc(C(=O)O)cc3)s2)C1 C=CCC(C(=O)N1CC(C2(NC(c3ccn(CCO)c3C)=O)CC2)C1)C(C)C C1(Cc2ccc(C#N)cc2)CCN(N2CCCC23CCOCC3)CC1 C1(NC(CCOC)=O)CC2C1CCN2C(c1cc(C)c(Br)cn1)=O N1(C(CC(COC)NC(c2c(CC)cns2)=O)=O)CCC2CN(C)CC2C1 c1(C(=O)NC2(CNC(CC(C=C)C)=O)CC2)cc(S(C)(=O)=O)ccc1C N1(C(CCOCCOC)=O)CCN(C)C(C(=O)NCC(COC)OC)C1 c1(C(=O)NCC(CC)NC(c2noc(-c3cccc(F)c3)n2)=O)ccnnc1C N1(C(CCC(C)OC)=O)CCCC(C)(C)C1CNC(=O)CCc1cccnc1Cl CN1CCC(NC(=O)CC2(C)CC2)C1=O.C1(CC(=O)N)CCC(C)(C)C1 C1(C(C)C)CN(C(=O)CSCCNC(=O)CCCCN(C)C)CC(=O)N1 c1(C(N(CC)Cc2ccc(N(C)C)cc2)=O)cc(OC)c(OC)c(Cl)c1 c1(C(NNC(C2(C)CCCN2C(N2CCCC2)=O)=O)=O)ccc([N+](=O)[O-])cc1 N1(C(c2cc(OCC)n[nH]2)=O)CC(O)CC1(C)CO.C1(CC2CC2)C(=O)N1 c1(C(=O)NC2CCN(C(C34CCCC3C4(F)F)=O)C2)cccc2c1CCCC2=O CCC(C(=O)N1CCC(CO)(NC(c2ccc(C(C)C)nc2O)=O)CC1)C(C)C c1(C(=O)NC2CCCCN(C(c3cc(C)sn3)=O)C2)cnc2cc[nH]c2c1 c1(N2CCC(NC(c3cccc(SC)n3)=O)C(C)C2)nc(Cl)nc(C2CC2)c1F N(C(=NCCC(C)N1CCCCC1)NC1CCC1)Cc1cn(CC)nn1 C1(NC(C(C)OCC=C)=O)CC(C)(NC(c2c[nH]nc2I)=O)C1 c1(C(=O)OC)cc(Br)cnc1NC(C1CCN1Cc1cc(F)ccc1O)=O CC(C)C1=CCC(C(=O)NC(C2(O)CCN(C(c3ccn(C)n3)=O)CC2)C)CC1 CC1C(NC(c2cn(C(C)(C)C)nn2)=O)CC2CCC1N2C(=O)CS(N)(=O)=O C1(C(=O)NCCC2(C(=O)NC(C)(C)C=O)CC2)(CC)CCCCCC1.O N1(C(c2ccc3nn[nH]c3c2)=O)CC2OCCN(C(C3CCS3(=O)=O)=O)C2C1 C1(CNC(c2nnc(C(F)(F)F)s2)=O)CCCCN1C(=O)CC1CSC1 c1(C(=O)NC2CCN(C(C(CC)(F)F)=O)CC2CO)ccc2nncn2c1 Cc1cc(C(F)F)nn1CC(=O)N(CCCCCNC(C1(C)CC2CC2C1)=O)C C=CCC(CNC(=O)Cc1ccn(C)n1)C(=O)NC(C1CCCC1)CC c1(-c2ccon2)ccc(Cl)cc1.C(=O)(CC(=O)NC1CC(C=O)C1)OCC.N Cc1cc(C(N2CCCOC(CNC(C3CC4CC3CO4)=O)C2)=O)c(O)c(C)c1 c1(C(N(C(c2ccc(Br)s2)C)CCO)=O)c(Br)c(Br)nn1C C(CNC(=O)CC)(CC(F)(F)F)NC(C1CCN(C)C1=O)=O.c1cccnc1.O c1(OC)ncc(C(N2CC3CC2C(=O)O3)C(=O)NC(C)(C)C)cc1F CC(CC(=O)NCC(O)CN(C(=O)Cc1ccco1)C)c1ccccc1 C1CN(C(=O)CN(C)C(C)=O)C2(CCC2)C1.c1cccc(CC=O)c1.CCO C(=O)(C1CCc2snnc21)Nc1cccc(-c2c(C)nn(CC(F)F)c2)c1 N1(C(C2(F)CN(C(C(CC=CC)C)=O)C2)=O)CC(N(C)C)C2(CC2)C1 C1(F)(CNC(CC#C)=O)CCCN(C(c2cncc(-c3ccccc3)c2)=O)C1 Cc1cc(C(N2CCC(CN(C)C(c3cc[nH]c3C(C)C)=O)CC2)=O)c(C)o1 N1(C(c2scc(C(C)=O)c2)=O)CC2CCC(C1)N2C(C1CC2CC2C1)=O C1(NC(C2CC3CCC2O3)=O)CN(C(c2ccc(SC3CC3)cc2)=O)CC1O C(C(C)(C)CNC(c1coc(O)n1)=O)N(C(C1CC(C)=NO1)=O)CC C(CCOC(=O)C(N)=O)(C1CC1)OC C(C(=O)N(CC(=O)NC1CC1)C)(c1ccoc1)NC(CN(C)CC)=O CCC(CC1CCCCC1)C(=O)NC1CCN(C(c2ccc(C(F)F)cn2)=O)C1 c1(CC=O)csc(Cl)c1.c1(CC)cccnc1.CCS(=O)(=O)NC(C)C=O.N c1(CCCC(=O)N2CC(CC(C)NC(=O)C3=CCCC3)C2)ccc(F)cc1F N1(C(c2cn(C)nc2)=O)CCC2CN(C(c3cc(C(F)F)ncn3)=O)CC2CC1 C=CC1(C(N2CCCC(C(=O)N(CCCCCC)C)C2)=O)CCOCC1 C1(NC(C(CCC)(C)C)=O)CC2CC(C1)CN(C(C1OCC1(C)C)=O)C2 C(=O)(C(O)CCC(C)C)N.c1(SC)cn(C)nc1C(=O)NCC(=O)NCC c1(CC)c[nH]c(C(=O)NCCC(C)NC(=O)CCCc2cnccn2)n1 CC1(C)CN(C(c2ccncc2F)=O)CC1CNC(=O)CCn1cnnn1 C(=O)(C(C)CC(F)(F)F)N(C(CC)CNC(c1nc(=N)cc[nH]1)=O)C C(=O)(C(C)C(O)C(C)C)N1CC(C(=O)N)C(F)(F)C1.c1(CC)nn(C)cc1C CC1(C)CN(C(c2n[nH]c(O)n2)=O)CC2(CN(C(=O)CCN3CCOCC3)C2)O1 N1(C(C2C(C(C)C)CCO2)=O)CC(C(=O)NC2CC2c2cncs2)CC1(C)C C1(N(C(=O)C=CBr)C)CCC2CN(C(=O)C3=COCC3)CC12 c1(CNC(c2ccn(CC)n2)=O)cc(C)c(C(=O)NC2(C)CCSC2)o1 c1(C(N2CCC(NC(C#CC3(C)CC3)=O)CC2)=O)ccc(N=[N+]=[N-])cc1 c1(C(NCC)=O)cncc(C(F)(F)F)c1.O=CCCOC1CCC1.C1CC1 c1(C(N(CC=C)CC=C)=O)cc2cccc(-c3ccc4c(c3)CCOC4)c2[nH]1 N1(C(CC(C)(C)C(F)F)=O)CCCC(C2CCN(C(=O)CC3CCC3)CC2)CC1 CCCC(C(=O)OC)N(CC(=O)NCCc1nc[nH]n1)C C(N=c1nc2c(Br)csc2c[nH]1)C1CN(C(c2nnn(CC)c2C)=O)CC1(C)C c1(C(N2CCOCCC2C(=O)O)C(=O)NCC(=C)C)cc(OC)cc(CC)n1 c1(CC2CN(C(=O)Cn3cc(C4COCC4O)nn3)C2)ccc(F)cc1 CC(C)CC(CNC(=O)CN1CCCCCC1)C(=O)N(C(C)C(F)F)C C1(OCC)CC2(C1)CC2NC(C1CCN(C(c2csnc2Cl)=O)C1)=O CC(C(=O)NCC1CCOC1C(=O)NCC1CCC(=O)NC1)C(C)(C)C c1(C(=O)NCC2CCC(NC(C(CC)=CC)=O)C2)cc(Br)cn1CC N1(C(c2n(CCC)ncc2)=O)CCN(C(=O)C(CC)C2CCOCC2)C(CC)C1 C(=O)(C(CN(C)C)C(C)C)NC(COC)CC(=O)N1CCC=C(Cl)C1 Cc1coc(C(N2CCCCC2CCN(C(=O)C(O)Cc2cnc[nH]2)C)=O)c1C C(=O)(CCCC(=O)NC(C1CCN(C(=O)CCc2nc(C3CC3)no2)C1)C)OC CC1(C)CN(C(c2ccccc2C(C)(C)C)=O)CCN(C(C2CC(F)C2)=O)C1 C1(N(C(C(N)=O)C(N)=O)C(c2nc(C)sc2)=O)CC2(CNC2)C1 CCC1c2cccn2CCN1C(C1CC12CCN(c1nc(=N)[nH]cc1C)CC2)=O c1(C(=O)NCC2CCN(C(c3cscc3Cl)=O)CC2O)cnc2[nH]ncc2c1 NS(=O)(=O)C1(C(N2CCC(CNC(=O)C(c3ccccc3F)O)C2)=O)CC1 C(=O)(CC(C(F)(F)F)NC(=O)C1CC1)N(C(c1cn[nH]c1)C)CC C1(CNC(C(N2C(C(=O)OC)C(O)CC2)=O)=O)CCCC12CCNCC2 N1(C(C(C=CC)O)=O)CCC2CN(C(C3(Cl)CC4CCC3O4)=O)CC2CC1 N1(CC(c2c(C)ccc(Cl)c2)=O)CCC(O)(CO)C(O)C1 C1(COC)(NC(=O)NC2CC2)CCN(c2ncc(C)c(C)n2)CC1 C(=O)(C1=CCCCO1)NC1C(C)(C)C(CC(=O)NC2(CCF)CCC2)C1 c1(C(N2CC(C(=O)Nc3cnncc3Br)OCC2)=O)cc2ccc(Br)cc2s1 Cc1cc(CC(=O)NC2CCOCC2NC(C2CC(C)C2)=O)ccc1Cl c1(N(C2(CO)CCNCC2)Cc2cccc(C)c2)ncnc2cc[nH]c12 N1(C(c2c(CC)nc(C)s2)=O)CC2(CCCC2NC(=O)CC(C)CC)C1 C1(c2nnnn2C)(N(C(=O)CCCn2ccnc2)C)CC2CC1CC2(O)C(F)(F)F C1CCCCC1.C(C)(C)(C(=O)N)OCC.N1(CC=CC=O)CCCCC1.C N1(C(C2C(C)C2)=O)CC(CO)C2(C1)CN(C(=O)Cc1nncs1)C2 CC(N=c1[nH]c(=NCc2ccccc2S(C)(=O)=O)[nH]c2cc[nH]c12)C1CC1 C1(NC(c2cc(-c3cccc(Cl)c3)ns2)=O)CCCN(c2cncs2)C1 CC(C)C(C(=O)NC(c1ccc(Br)cc1)C(F)F)c1cc(O)no1 c1(C(C(N2CCC(NC(c3c(OC)n[nH]c3)=O)C2)=O)N(C)C)ccccc1Cl C=C(C)C1CN(C(C2(C3CCCN3C(=O)CN3CCOC3=O)CC2)=O)CCO1 c1(SCCN2CC(=O)N(CCCC(F)(F)F)C2=O)nc2ccccc2s1 N1(C(c2c(OC)scc2)=O)CCCC(CNC(=O)CCCn2ccnc2C)C1 N1(Cc2c(OC)cccc2Cl)CCC2C1CCCN2C(c1cccc(O)c1C)=O C(CC(C)(C)C)(C(=O)N1CCC(C(N2CCOC(C(C)C)C2)=O)C(C)C1)OC C(=O)C(O)C(C)C.CC(C)CCNC(=O)C(C)(C)C.C(C)(C)C.C=O.N C(=O)(CC(O)C(Cl)(Cl)Cl)N1C(C)CCC(NC(c2cc(F)cnc2O)=O)C1 CC1CCN(C(c2cc(C3CC3)no2)C(=O)NC2(C)CC2)C1(C)C c1(C(N2C(CNC(C(CCOC)C)=O)CC2)=O)cccc2c1COCCN2 c1(OC)ccccc1OCC(=O)N(CC(O)C)C.c1(CC=O)ccc(Cl)cc1.N Cc1ccc2nc(N3CC4CC3CN4C(C3(C)CCN(C)CC3)=O)sc2n1 c1(C=O)ccc(N=S(C)(C)=O)cc1.N1(CC)CCOCC1C(N1CC(C)C1)=O.N C1(NC(Cc2scc(C)c2)=O)CCCCC1NC(C1CCC(C)O1)=O C=CC(C)C(=O)NC1(CC(=O)NCC(C)(C)CSC)CCC1 N(C(=NCCC(CO)CO)NC(c1ccc(Br)cc1)CF)CCOC C=CC(C)(CCOC)C(=O)N1CCC(CCNC(=O)C(C)CO)C1 c1(CC)cc(C(=O)N(C2CCN(C(c3coc(C(N)=O)c3)=O)C2)CCO)on1 C#CCC(C(=O)NC(C)CCCCNC(=O)CN1CCOC1=O)C1CC1 c1(SC)ccc(C(=O)NC2C=CC(C)C2)cc1[N+](=O)[O-].C(=O)C(C)CC(N)=O C1(O)(CNC(c2ccc3c(c2)CC3)=O)CCCN(C(C2CCC2)=O)CC1 N1(C(C=C(COC)C)=O)CCN(C(=O)C(c2csc(C)n2)=O)CC(C)(C)C1 N1(C(CC2N(C(CC=CCC)=O)CCC2(C)C)=O)CCSC2CCCC12 CCCCC(F)(F)C(=O)NC(CCC)CC(=O)NC1CCCCCCC1 c1(NC(c2ccc(Br)cc2)=O)ccnc(S(C)(=O)=O)n1.C12CCC(N)(CC1)C2 N1(C(CC2ON=C(C)C2)=O)CCCC(CN(C)C(C2NC(=O)OC2C)=O)C1 N1(C(=O)CCCC(F)F)CCC2(CC1)CCN(C(C1(Br)CC13CCC3)=O)C2 c1(C(=O)OC)cc(C)nn1C.C1(N2CC(C=O)C2)CCN(C)CC1.C(C)CC n1(CC)nc(C(=O)NC(C)CC(C)NC(C2(N(C)C)CC2)=O)ccc1=O c1(OC)ccc(C(C)NC(C2CC(NC(c3cc(Br)c[nH]3)=O)C2)=O)cc1F S(=O)(=O)(c1nccs1)N1CC(CNC(Cc2nc(C(C)C)on2)=O)C1 CC1CCN(C(=O)C=C2CCC2)C1CNC(c1ccccc1)=O.C1CC1.O C1(CC(=O)N(C2COC(C)(C)C2)C)CC2(C1)CN(C(C1(O)CCC1)=O)C2 c1(CNC(C(C)OCC#C)=O)cccc(C(=O)NCC)n1.C(C)(C)C c1(CN(C(C2CCOC2(C)C)C(=O)NCC(=C)C)C)ccc(C)c(OC)c1 C=CCCC(=O)NC1(C(=O)NCC2(CC)CCCC2)CC1C C(=O)(C1Cc2ccc(C)cc21)NCC(CC)NC(c1ocnc1C1CC1)=O c1(N2CCC(NC(C3CCCNS3(=O)=O)=O)C2)ncnc2sc(C(F)(F)F)nc12 N1(C(c2cc(O)cc(F)c2)=O)CCC2(CCCN(Cc3cccnc3O)C2)C1 N1(C(C(C(=C)C)(C)C)=O)CC2=C(C1)CN(C(=O)CC13CCCCC1C3(F)F)C2.C n1(CCC(N2CC(CN(C(COC)=O)C)OCC2)=O)c(C)c(C)sc1=O Cc1cccc(C(=O)N(C2CCN(C(C34CC(CC(F)(F)F)(C3)C4)=O)CC2)C)c1 c1(C(N2CCC(F)(C(N3CCC(N(C)C)CC3)=O)CC2)=O)cccc2[nH]ccc12 c1(C(N2CC3(C)C(C2)CN(C(=O)C(F)(F)CF)C3)=O)cc(Cl)cc([N+](=O)[O-])c1O N1(C(C(CCOCCO)NC(c2cc(C)[nH]c2)=O)=O)CCC(C2=NOCC2)C1 CC(C(F)(F)C(F)(F)F)=CC(=O)NCCCC(C)NC(c1cn2ccsc2n1)=O c1(C(=O)NCC(C)CNC(=O)CC(C)c2ccco2)cccc(CN=[N+]=[N-])c1 C(=O)(C(F)C(C)(F)F)NC(C(=O)NC(CCCC)(C)C)CCC1CC1 Nc1nn(C2CCCCC2)cc1C(=O)NCC(=O)NC1CC1 CN=c1[nH]c(C(=O)NCC(C)N(C)C(c2ccc(-n3cncn3)cn2)=O)cs1 Cc1ccc(-c2cc(C(=O)NCC(O)CCNC(C3CC(CF)C3)=O)n[nH]2)s1 c1(C(=O)NCC2C(NC(C(CC)OC)=O)CCC2)cc(Br)c(C)n(C)c1=O C1(NC(c2cnc(C3CC3)nc2O)=O)CCN(C(=O)CCCCCO)CC1F c1(C(=O)NCC(CNC(C(Br)=C(C)C)=O)C)ccc2nn[nH]c2n1 N1(C(C2(F)CCCN(C(C#CC3(C)COC3)=O)C2)=O)CC23CCC2(COC3)C1 C(=O)(CCC(C)NC(c1csc(C(C)C)n1)C)OCC C(c1ccc(C(C)(C)C)cc1)=CC=O.C1(NC(C=C(C)C)=O)CC(C)C1 C1(CC(=O)NCCOC2CN(C(C3C(=C)C3)=O)C2)CC2CC2C1 CC1CCCc2ncc(C(N3CCN(C(c4coc(O)n4)=O)C(C)C3)=O)n21 C(C1=NOC2CN(C(=O)C3=NNC(=O)C3)CC12)NC(C(C)=C1CCC1)=O C1(NC(C2N(C)CCN(C(C3OC4CCC3C4)=O)C2)=O)CCc2n[nH]cc2C1 c1(CN(CCC(=O)O)Cc2cccnc2)ccc2c(c1)CCCC2O C(=O)(C1=C(C2CCOCC2)N(CC)C(=S)NC1c1ncc(C)s1)OCC N1(C(C(CC)SC)=O)CC2CCCC(NC(=O)CC3(O)CCCCC3)(C2)C1 CCCCCC(=O)NCC(=O)NCC1COC(C)C1.C(=O)CCc1ccsc1.N C(CCCC(=O)N1CC(OCCC(=O)NCC=CCl)C1)N(C)C C1(C)(CC)C=C(C(=O)NCCCOCCNC(c2cnn(C)c2N)=O)C1 C1(N(C)C)CN(C(=O)CC2CCCN(C(=O)CC(C)(C)C)C2)CC1(C)C c1(N2CCC(CNC(CC=C)=O)C(C)C2)nc(CC)nc(Cl)c1F Cc1cc(CC(N2CCC(O)C2C(=O)Nc2cccc(I)c2)=O)cc(C)c1 c1(C(=O)OC)cc(CNC(=O)C(=O)C(N2CCC3CCC23)=O)n2c1CNCC2 c1(C(=O)NCC(C)N(C(=O)C=CC2CCCO2)CC)ccc2occc2c1 c1(C(N2C(C(=O)Nc3c(C)c(Cl)ccc3)CC(O)C2)=O)cccc2c1OCCO2 N1(C(c2c(C)scn2)=O)CCC2(CCCN(C(c3nc(Cl)cs3)=O)C2)CC1 C(C1CN(C(=O)OC(C)(C)C)Cc2ccccc21)NC(CC(CC)CC)=O CCCS(=O)(=O)CC(=O)N1CCC(NC(=O)C(c2ccccc2)F)C12CCC2 c1(C(N2CC(F)(F)CC2CC#N)C(=O)NC(C)(C)C)ccc(Br)c(F)c1 c1(C(=O)NCC2C(CNC(C(C)C(C)(F)F)=O)C2)cccc2nn[nH]c12 CCCC(C(=O)NCC1(O)CN(C(=O)C(=O)NC2CC2)C1)NC(C)=O CN1CCCCC(C(=O)NCCC(C)(C)NC(c2ccc(N)c(Cl)n2)=O)C1=O C1(C(=O)Nc2cn(CC)nc2)CC(C)(C)CCN1C(=O)C(=O)NCC(F)F N1(C(CC(C)C)=O)CCCC(C)(CNC(C2CN(C)CC(C)O2)=O)C1 C=CCCC(CC(C)C)C(=O)N1CCCC12CCN(C(C1C(OCC)C1C)=O)C2 N1(C(c2cc(C)[nH]n2)=O)CCCC12CN(C(C1CNC(=O)C1)=O)C2 c1(C(N2C3C(NC(CNC(CCC(C)C)=O)=O)C(C3)C2)=O)ccc(F)c(F)c1F O(S(=O)(=O)c1sc2cccc(F)c2c1C)c1cccc(OC)c1 N1(C(c2cnc(Cl)s2)C(=O)NCCOC)CCCC2(C1)NC(=O)N(C)C2=O N1(C(CCCOC)=O)CCCC2C1CCCN2C(=O)CN(C)CCO CC1(C)CCN(C(=O)Cc2ccco2)C1C(=O)NCCn1cnnn1 C1(C(N2C(C(C)C)C(NC(c3cccs3)=O)CC2)=O)CN=C2N=CNN2C1 CC1(C)C(NC(C2CCCN2C2CC2)=O)CCN1C(=O)CCCF c1(C(N2C(C(=O)OCC=C)CCCC2)=O)ccc(CN(C)C)cc1CC C1(CNC(CCC#C)=O)CN(C(c2ccc(OC(F)F)cc2)=O)C2COCC2O1 c1(C(=O)NC2(C)CC(NC(Cc3c(C)ocn3)=O)C2)cccc2nc(O)n(C)c12 c1(NCCC2CCN(C(C3C(C)(C)S(=O)(=O)CC3)=O)C2)ncnc2cccnc12 C(=O)(C(C)=C1CCCC1)N(CC(=O)N(CCCC)CCCO)CCOC C#CCCC(O)C(=O)NC(C1CCCC1)CNC(=O)C(F)(F)CO N1(C(C#CC(=O)N(C)C)=O)CCC2CCN(C(c3cc(Br)n(C)n3)=O)C2C1 Cc1c(NC(=O)C(C)(C)CCCl)cccc1S(=O)(=O)NC(C)(C)C C1(C(=O)NCCN(C(C(C=C)C)=O)CC(C)O)CCc2n[nH]cc2C1 Cc1cc(NC(=O)CC2CN(C(=O)Cc3ccc(Cl)s3)CCO2)cc(Cl)n1 C1(NC(C=CC(C)C)=O)CCCC12CN(C(=O)C(C)(C)c1ncco1)C2 C12(C(N3CCCC(CNC(=O)CCc4cnoc4)C3)=O)COC(CCO1)C2 c1(C(=O)NC2C(NC(C(C)(C)c3ccsc3)=O)CC2)ccc(-n2ccnc2)cc1 N1(Cc2cnc(SC)nc2)CC2CN(C(c3ccc(I)cc3Br)=O)CC12 C(=O)(C1=CCN(C)C1)N(CCCOCCNC(c1c(C)nc[nH]1)=O)C c1(-n2cc(C3CN(C(c4n(C(C)C)cnc4)=O)C3)nn2)cccc(CO)c1 C(=O)(N=c1ncnc2[nH][nH]c(C)c1-2)C1N(c2nc(C)nc3c2CCC3)CCSC1 CC(CN(C)C)C(=O)NCCNC(c1ccsc1C(F)F)=O c1(C(=O)NCCCCCNC(c2c[nH]cc(F)c2=O)=O)cnn2c1OCCCC2 c1(C(N2CCCC(NC(C3COC(=O)O3)=O)CC2)=O)cc2ccccn2c1 Cc1o[nH]c(=NC(=O)C2CCCN(Cc3c[nH]c4ncccc34)CC2)c1Br N1(C(CCCN=[N+]=[N-])=O)CCC2(CCC2NC(=O)C2CCc3nccn32)CC1 CC1(C)CC2CC2C1.c1(C(=O)N)cc(CC)on1.C(=O)CC=CC(C)(C)C O=C(C1=C(Cl)CCCC1)NC1C2CC3C1C3C2C(=O)NC1CCn2ncnc2C1 C1(C)(C(N(CCC(C)NC(C(C=C)OC)=O)C)=O)CNC(=O)C1 C1(C(=O)NCC2C3CN(C(c4cn(C)[nH]c4=N)=O)CC32)CCC2(CCC2)CO1 N1(C(c2cc(C)sc2)=O)CC2CC(NC(=O)CCc3cccc(F)c3)CC2C1 c1(C(N2CCN(c3cc(Cl)ncn3)CC(O)C2)=O)ccc2nccnc2n1 CC(C(=O)NC1CC(CCNC(c2csc(C(F)F)n2)=O)C1)C(C)(C)C N1(C(CN2C(C)CCC2)=O)CCC(O)(Cc2cn(C3CCCNC3=O)nn2)CC1 C(CCCCC(=O)NC1CCCCC1(F)F)N(C)C(C1CCC(F)(F)C1)=O C1(NC(C2(CSC)CC2)=O)COCCN(C(=O)CCc2ccc(C)cc2)C1 C12CCN(C(c3cccn3C)=O)CC1C2.n1(CC)nc(C(=O)N)cc1C(F)(F)F c1(C(C)NC(N(CCCF)CCOC)=O)nc(N(C)C(C)C)no1 C(CCCCC(=O)NCCC1(NC(=O)CCc2nccn2C)CCOCC1)=CC C1(C)(C=O)CC1(F)Cl.C1(CNC(CNC(=O)OCC)=O)CCC1.N Cc1[nH]nc(C(=O)NCC2CC(O)CN2C(C2C(C)C2C)=O)c1O Cc1cncc(CC(=O)NCC2CCCC(CNC(=O)C(C)C)C2)c1 C1(CC(N2CCCC(O)C2)=O)SC2=NCCN2C1=O.C(C(=O)N)=CC=CCC Cc1sc(Br)cc1C(=O)NCC1CC(F)CN1C(C1CC1[N+](=O)[O-])=O C(CCCCC(=O)NC1CCCN(C(c2ccc(C)cc2C2CC2)=O)C1)OC c1(C(=O)NC(C(N2C(C#C)CC2)=O)(C)C)c[nH]c2cccnc12 c1(OCC(=O)NCC2CCCCS2(=O)=O)ccc(C(=O)O)cc1[N+](=O)[O-] N1(C(CCCCCCC)=O)CCCC2C1CCCN2C(c1cnc(O)cc1C)=O CC#CCCC(=O)N(C1CCC(NC(=O)Cc2ccc(C(C)C)cc2)CC1)C S(=O)(=O)(c1cccs1)NCCC(=O)NC1CCCC1O.c1(C(=O)N)n[nH]cc1Cl CCCC(CCCNC(c1cccc(=O)o1)=O)NC(=O)C(O)CC1CCOCC1 c1(CC)nc(C(=O)NCc2ccoc2C(=O)N(C(C)C)CC)cs1 C(=O)(CCCC(C(=O)NCC1CCOCC1)N1CC(C)(C)CC1CC(=O)N)OC CCC(C)C(C(=O)NCC1(NC(=O)C(Cl)=CCl)CC1)NS(C)(=O)=O CC1CCN(C(=O)CC(C)(C)CN(C)C)CCN1C(=O)C(F)=CCCF c1(C(=O)N)cnc2scc(C)n12.C1(CNC(C2(CC#C)CC2)=O)CCOC1 C(CC(=O)NCC(C)=CCC)(C(C)(C)C)NC(C(C=C)OC)=O c1(C(N2CCOCC(CNC(c3cnc(C)n3C)=O)C2)=O)cnn2ccn(C)c12 CC1CCC(NC(=O)C(N2C3CCCC2CC(O)C3)=O)Cc2ccccc21 c1(CN(C)C)nc(-c2ccc(C(=O)NCC3CC3(F)F)cc2)cc(=N)[nH]1 C1(N(C(c2c(C#C)c[nH]n2)=O)C)CCCN(C(C23CC(C)C2C3)=O)CC1 c1(C(=O)NCC(C)NC(=O)Cc2ccnnc2O)c(F)cc(F)cc1Cl C1(NC(c2nn(CC)c(=O)cc2)=O)CN(C(c2cc(C)oc2C)=O)CC(F)(F)C1 N(C1CN(C(c2cc(C#N)cs2)=O)CCc2ccccc21)C(C(CC=C)CC)=O c1(C2(C(=O)NCCCCN(C(C(CC)C)=O)C)CC2(Cl)Cl)ccc(OC)cc1 Cc1nc2c(s1)CC(C(N1CCN(C(c3cnsn3)=O)CC(O)C1)=O)CC2 CC1CCCCC1(CNC(=O)C1=CCCC1)NC(C1CCCCN1C)=O C1(C(C)C)CCC(NC(=O)Nc2ccc(C3CC3)nc2)CC1 C#CCC(C)(C(=O)NCc1cccc(OC)n1)NC(c1nc(CC)oc1C)=O Cc1ccc(CCCNC(C2CCN(c3ccccc3F)C2=O)=O)c(Br)c1 c1(C(C(=O)N(C2CCC(CNC(=O)OC(C)(C)C)O2)C)O)ccccc1Cl C(C(=O)NCCCOC1CC1)(C(C)C)NC(Cc1c(CC)con1)=O N1(CC)CCCC(ONC(=O)NC2CS(=O)(=O)C2)C1 CCCCCCNC(=O)C(C)NC(N)=O.c1(C=O)ncccc1C(F)(F)F.N c1(C(C(=O)NCCOCCCN(C(C#CC(C)C)=O)C)C)cc2ccccc2s1 N1(C(CC2CCN(Cc3ccc(CC)cc3)CC2)=O)CCC12CCCC2 CC1CCN(CC(N2CC3C(CC(=O)NCCCCC(N)=O)C3C2)=O)CC1 N1(C(C2CC2)=O)CC2CN(C(C3CC(=C4CCC4)C3)=O)CC2(C)C1.COC N1(C(C=Cc2ccc(OC)cn2)=O)CCN(C(C2CC(OC)C2)=O)CCC1C CCCC(CNC(=O)Cc1cncnc1)C(=O)Nc1ccc(N(C)C)cc1 CN=c1nc(N2CCCC(C)(N(C)C)C2)[nH]c(=NC(C)c2cnsc2)[nH]1 N1(C(C2CN(C(c3nc(C)c(C)s3)=O)CC2(F)F)=O)CCOc2ccccc21 N1(C(C(CC#CC)NC(=O)C(C)CC)=O)CCC2(CC1)CC2C#N N1(C(CSCC=C)=O)CC(O)CC1(C)C(=O)NC1CC(O)CC1O N1(C(CCOC(C)=O)=O)CCN(C(c2cc(Br)cs2)=O)CC(CO)C1 CN1CC(O)CC1(C)C(N1CCC(C(C)(C)NC(c2cc(O)n(C)n2)=O)CC1)=O CCCC(F)(F)C(=O)NC1(CCCC(=O)NCC(O)CF)CCC1 S(=O)(=O)(c1ccc(S(=O)(=O)N2CCC(=O)N3CCCC23)cc1C)NC C1(N(C(C2C(C(=O)OC)C2)=O)C)CCN(C(c2ccncc2F)=O)CC12CC2 c1(C(N2C(CNC(CCCOC)=O)CCC2)=O)cc2nccnc2cc1F C(CCCCCN=[N+]=[N-])NC(C1(SC)CN(C(c2oc(C)nc2C)=O)C1)=O C1(C(=O)NC(CC(=O)NCC(CC)n2cccn2)(C)C)CC2C=CC1CC2 c1(C(N2CCC(CC(=O)NCC(C)OC)C2)=O)cnn2c1OCC2 c1(C(N(C2CCN(C(c3c[nH]c(=N)o3)=O)C2)CC)=O)cc2ccc(F)cc2[nH]1 C(CC1=CCC2CC1C2(C)C)NCc1c(C)nco1 c1(CC)ccc(C(C)=CC(=O)N(CCC)C)cc1.c1(C=O)ccsc1C(F)F.N CCC(C)(C)C(=O)NC1CCC1NC(C1CC(C(F)F)C1)=O C=C=CCCC(=O)NC(CC=C)C(=O)NCC1(OCC)CN(C)C1 C12(NC(=O)C(O)C3CCCC3)CC1CN(C(c1cccc(C3CC3)c1)=O)C2 C1(C(N(C2CCOCC2)CC#C)=O)CCCC(NC(C2CCCCC(=O)N2)=O)CC1 c1(C(N2CC(NC(C3N(C(C)=O)CCC3)=O)C(F)C2)=O)cc2c(ccn2C)[nH]1 Cc1oncc1C(=O)NCC(N1CCC(N(C(=O)C(F)C2CC2)C)C1)=O N1(C(c2cccc(SC)c2)=O)CCn2nnc(C(=O)NCC3CCC(O)C3)c2C1 N1(C(C2C(OCC)C2)=O)CCN(C(c2cn(CC3CC3)nn2)=O)CC1 c1(C(C)NC(C2(CN)CC2(F)F)=O)noc(C(C)(C)C)n1 [SH](=O)(=O)c1ccc(Cl)cc1.C1C2CC1N(C(=O)C)C2.C#CC1CC1C(=O)N C(=O)(C(O)C(C)C)NC(CNC(c1c(COC)ccs1)=O)(C)C1CCC1 CCCC(C)CC(=O)NCCC1CNC(=O)CCNC(=O)O1.O(C)CC c1(C(=O)NC2(CN(C(=O)Cn3nccn3)C)CC2)ccc(C(N)=O)[nH]1 N1(C(CC2CCCC(=O)N2)=O)CCCN(C(c2cc(O)cc(=O)o2)=O)CC1 C=CCC(CNC(=O)CC1CCC(=O)C1C)C(=O)Nc1ccc(O)cc1C c1(CC)ccc(C(N2CC3CC(NC(=O)C=C4CCN(C)C4)C3C2)=O)cc1N C#CCCCC(C)(c1nnnn1C)NC=O.C1(CC)CCN(C(C)=O)C1.C(C)(C)C C1(CNC(C(C=C)O)=O)CC2(CO1)CN(C(c1cn(CC)nc1C)=O)C2 N1(C(C2C(C(=O)NC3(C=C)CCCC3)C2)=O)CC2CC(OCC)C2C1 C=CCCC(C(=O)OC)NC(=O)C(CNC(=O)CCCF)CC1CCCC1 CC1CN(C)CC1N=c1[nH]c(=N)[nH]c(=NCc2cccc(-n3cncn3)c2)[nH]1 Cc1cccn2c(C(=O)NCC3CC4CCC3N4C(c3cc(O)cs3)=O)cnc12 C1(NC(=O)COC2CCC2)CC2(C1)CN(C(C1CCC(C3CC3)C1)=O)C2 N(C1CCCc2ccoc21)C(COC1CC(NC(C(CC(=C)C)OC)=O)C1)=O N1(C(c2n(CC)ncn2)=O)CCC(C(C)CNC(c2cc(O)[nH]n2)=O)CC1.C CC(C)(C)C(CO)C(=O)NC1CN(C(c2ccc3ccoc3c2)=O)CC12CC2 Cc1[nH]c2ncccc2c1C(N1CCCN(C(=O)CN2CC3CC3C2)CCC1)=O C12(C(C)NC(CC3N(C(CCOC)=O)CC3)=O)CC(CO1)C2 c1(C(CC)OC)cn(CCCNC(C2CSCN2C(C)=O)=O)nn1 S(=O)(=O)(c1ccc2c(c1)COCC2)NC1CN(c2c(OC)cccc2)C(=O)C1 N#CC1Cc2cccc(C(=O)NCC3CC3)c21.c1(CCC(=O)N)cc(Cl)no1 C1(C(N(C2CCN(C(c3cnnn3-c3ccccc3)C)C2)C)=O)CC2CCC1C2 C12CCC(CO1)C2.c1(C(=O)NCCC)conc1NC.C(C)(C)C.C=O C(C1CCCCC1)=CC(=O)NC(C(=O)N1CC(=CC)C1)Cn1cccn1 S(=O)(=O)(c1cc(Cl)c(Cl)cc1Cl)NCCN(C(C)C(C)(C)C)C N1(C(Cn2cc(C(C)O)nn2)=O)CCN(C(=O)C2=COCC2)C(C)C1 N1(C(CCCCOCCC=C)=O)CCCC(NC(C2CC(C3CC3)=NO2)=O)CC1 N1(C(=O)CCc2nccs2)CCC(CNC(C23CCC(CC2)CO3)=O)C12CC2 CCC(N=c1[nH]c(=NCC2(CO)CCOC2)[nH]c2cccc(F)c12)c1ccncc1 c1(C(=O)NCC2C=CC(NC(CCOC(C)C)=O)C2)cnn2ccn(C)c12 c1(CNC(=O)CC2CCSC2)cnn2c1CN(C(C1(F)CC=CC1)=O)CC2 N1(C(C(n2c(C)cc(C)n2)C)=O)CC(NC(c2cccs2)=O)CC(C)C1 C1(NC(c2ccc(F)cc2)=O)CC2(C1)CC(NC(=O)C(c1cccnc1)O)C2 Cc1c(NCC=CC2CC2)nc[nH]c1=NCC1(CO)COCC2CCCCN12 c1(C(=O)OC)cc(C(C(=O)NCCCF)N(C)Cc2cccc(C)n2)n(C)n1 Cc1nn(C)c2c(N3CCOC(C4CC4)C3)nc(=NC3CCC(O)C3)[nH]c12 c1(CCCNC(c2scnc2C2CC2)=O)cnc2ccnn2c1 C1(CC(=O)NCC(CNC(c2cc(C)c(Br)o2)=O)O)CCC(C)(C)CO1 C(=O)(C(O)CC(N)=O)N(CCNC(C(C)Cc1ccncc1)=O)C1CC1 Cc1ccc(C)n1CC(=O)NCC1CC1NC(=O)C=Cc1cc[nH]n1 c1(N2CCCC(CC(N3CCCCC3CO)=O)C2)ncc2sccc2n1 N1(C(c2cc(C)on2)=O)CCC(O)(CNC(=O)C(C)OC)C1.c1ccncc1 c1(OC)cccc(C(N2CC(NC(=O)Cn3cc(C(C)=O)nn3)CC2C)=O)c1 c1(CC(=O)NCC(C)N(C(c2n(CC)ncn2)=O)C)coc2ccc(F)cc12 N1(C(c2cn(CCC)nc2)C(=O)Nc2ccccc2)CCC(C#N)C1 CC1(C)C(C(N2CCC2(C)CC(=O)NC2CC(n3cccn3)C2)=O)C1CO C1(CNC(CCSCC)=O)(NC(=O)CC)CCCCC1.c1ccc(F)cc1.O C(=O)(CC(F)(F)F)N1CCC(CC=C)C1.c1(C(=O)N)cnn(C)c1N.C(C)=O N1(C(c2cc(C)n(C(C)C)n2)=O)CCN(C(=O)Cn2cnc(C(N)=O)n2)CC1C c1(C(=O)NC2(c3c(C)ccs3)CC2(C)C)cccn(CC(C)C)c1=O N1(CC)CCOC(C(=O)N(CCCN(C(=O)C=Cc2cccnc2)C)C)C1 C1(C)(C(=O)NCCCN(C(=O)CCCCC(N)=O)C)C2CCC(C2)C1(C)C c1(CCC(=O)NCC(C)(C)NC(c2c(CC)ocn2)=O)ccc(CO)cc1 CC(C)C(N=c1cc(Cl)nc(-c2cccnc2)[nH]1)C1=CCCC1 C1(C(N2C3(C(=O)NCc4cc(C)ncn4)CC3CC2)=O)CCC(C)(C)CC1 c1(C(N2CCCC(NC(C(CC)=CC)=O)C2)=O)c(C)nc(C2CC2)nc1O C1(C(=O)NCCn2cncn2)CCOCCN1C(=O)COC1CCOCC1 n1(CC)nnc(C)c1CNC(=O)CC(O)C.C1(CC(=O)N)CCCC(C)O1 Cc1cn2c(CC(N3CC(C)CC3C)=O)csc2n1.C(=O)(C(C1CC1)C1CC1)N Cc1ccc2ccccc2c1NC(=O)NCC1CC2CCC1CC2 C1(C)(CNC(c2nnn(C)n2)=O)CCCN1C(C1CCC(CCO)CC1)=O C=CC(CC)CC(=O)N1CCC(O)CC1C(N1CCC(c2nn[nH]n2)C1)=O N1(C(c2c(NC)cccc2)=O)CCN(Cc2cccc(OCOC)c2)C(C)C1 C1(C(=O)NC(C=C)C2CCC2)CCN(C(c2cc(C)ncn2)=O)C(C)(C)C1 N1(C(CSCC)=O)CCCC2C1CCN2C(=O)CSC(C)(C)C C1(CNC(=O)CCC2CC2)CC2(CCN(C(C3(CO)CC3(F)F)=O)CC2)CO1 C#Cc1ccc(C(=O)NC2CN(C(=O)COC3CCC3)C(C)(C)C2)c(C)c1 C(=O)(CC=C(Cl)Cl)N(C)CC1(CNC(=O)CCC2CCCO2)CCCC1 C(=O)(CC(CC)CCCC)N(CCCOCCN(C(CC(C=C)CCC)=O)C)C c1(C(N2C(CNC(COCCOC)=O)CN(C)CC2)=O)cc2cnccc2[nH]1 N#Cc1ccnc(S(=O)(=O)N=c2cc(COc3ccccc3Br)[nH][nH]2)c1 CCC(C)C(CC(=O)NCC(CC)n1cccn1)NC(=O)C(C(C)C)C(C)C Cc1oc([N+](=O)[O-])cc1C(=O)N(CC(O)CN(C(=O)CS(C)(=O)=O)C)C.C n1(CC=C)cc(C(=O)NC23CC2CN(C(c2cnccn2)=O)C3)c2ccccc12 CC(C)CCC(C)NC(C1(N(C(=O)C(C)CO)C)CC1)=O C(=O)(C(C(C)NC(c1nccc(C)c1F)=O)C(C)C)NCCc1c(C)cccc1 N1(C(CCOCCOC)=O)CCCC(C)(NC(C2COC(C)(C)CO2)=O)C1 c1(C(=O)NC(C)C2CCC2)cnn2c1OCC2.C(=O)(C(F)(F)c1ccccc1)N N1(C(c2c(F)ccc(CC)c2)C(=O)NCc2cccs2)CCC2(CNC(=O)O2)C1 C1(CCNC(CC=C)=O)CN(C(C2CCC(=O)N2c2ccccc2)=O)CCCO1 C1(NC(=O)CC2CCC(C3CC3)O2)CC2CCC1N(C(=O)CC1=CCCCC1)C2 Cc1ccccc1CCC(N1CCC(NC(C2(C#N)CCOC2)=O)C1)=O c1(COC)ccccc1NC(=O)C#CCNC(c1csnn1)=O c1(Cc2n(CCCSCC)nnn2)cc(F)c(Cl)cc1Cl.C1(CC)CC1(Cl)Cl.N c1(NC)ccc(S(=O)(=O)NCc2cc(C3CCC3)nn2C)cc1[N+](=O)[O-] C1(C(N(C2CCNC2=O)C)=O)CN(C(c2nocc2Cl)=O)CC1(C)C N1(C(=O)NC(C2CCC3(CCC3)O2)c2ccoc2)CCOC2COCC12 C#Cc1cc(NC(C23CC(NC(=O)C(C)C4(O)CCC4)(C2)C3)=O)ccc1C C=CCCCC(C)(C)C(=O)NC1COCCC1NC(=O)C(CC)CC=CC c1(C(=O)NC2CCCC(NC(CSCCOC)=O)C2)c(C)ccc2c1CCCN2 CC1(C)CN(C(C2(C)C=CCC2)=O)CC1NC(c1ccc(Cl)nc1)=O N(C1CCc2ccccc21)C(C1N(C(c2cccc(C(=O)O)c2)=O)CCC1O)=O N1(C(c2n[nH]c(C)c2C)=O)CC(NC(C2(Br)CC2(C)C)=O)CC12CCC2 c1(OC)ccc([N+](=O)[O-])c(N2CCN(C(=O)NC3CCCC3S(C)(=O)=O)CC2)c1 CC1CN(C(C2(C(F)(F)F)CCC2)=O)CC1NC(C1CC1F)=O C(=O)(C(C)C(=O)NCC(F)CNC(c1cnc(C(C)(F)F)s1)=O)OC c1(C(N2CCC(=CCNC(CC(CC)C)=O)CC2)=O)ccc2[nH]c(=N)oc2c1 c1(C(=O)NC2CCCC(CC(=O)N(CCO)C3CC3)C2)ccc(Cl)cc1O C(CC1CCCC1)(C(=O)NOCCC(F)F)NC(CCc1cn(C)nn1)=O c1(NS(CCC)(=O)=O)ccc(C)c(C(=O)Nc2cnc(F)c(C)c2)c1 C1(O)(CCNC(C(CC)F)=O)CCN(C(c2ccc(Br)c(OC)c2)=O)CC1 C1(CNC(C2CCCN(CC)C2)=O)CC(C)(C)CN1c1cc(C2CC2)ncn1 C1(NC(C(C(CC)O)C)=O)CC2CC1CN(C(c1cccn1C)=O)C2 c1(OC)ccc(OC)c([N+](=O)[O-])c1C(=O)NC(C)CC.C1(C(=O)N)CC1F N1(C(C=CC=CCC)=O)CCC2(CC1)CCS2(=O)=O.C(=O)C(C)C(C)C.N C(=O)(C1=NNC(=O)CC1)N(C(C)C)CCN(C)C(C1CCC2(CC2)C1)=O.C C1(C(=O)NCCN2CCC(NC(C(CN(C)C)O)=O)CC2)OCC2CCCCC12 c1(OC)c(Cl)ccc(C(=O)NC2C3CC4CN(C(=O)C(C)C(C)C)C2C4C3)c1F Cc1cc2c(N(C3CNCC3O)C(c3cc(F)cc(Br)c3C)=O)ncnc2[nH]1 C(=O)(C(C)(O)CC(F)F)NCc1cn(C2CN(C(C(COC)OC)=O)C2)nn1 N1(C(CC(C)(C)OC)=O)CC(CNC(=O)CC=C(Cl)Cl)C2(CCC2)C1 c1(OC)cccc2sc(C(N3CCC(CNC(=O)CCCC#N)C3)=O)cc12 c1(C(=O)NCCCOCCNC(C2CN(C)C2)=O)cn(C2COC2)nn1 C12CN(CCO1)C(=O)CN(CCCCCC)C2=O.N1(CCSC)CCNCC1 c1(C(N2CCC(NC(Cn3ccc(C)n3)=O)(CF)C2)=O)cnc2n1CCC(C)C2 c1(N2C(C)CC(NC(=O)C(O)CCc3ccccc3)C2)ccc([N+](=O)[O-])cc1F c1(CC(=O)NC2(CO)CN(C(C3C(C)OCCC3)=O)C2)ccc2oc(O)nc2c1 C(=O)C1=C(C)CCCC1(C)C.C1(C(N2CC(CC)C2)=O)(COC)C=CCC1.N CCCC(CNC(c1nnsc1C)=O)C(=O)N1CC(C)(C)C1C(C)C C1(C)(CN(C(=O)CCn2ccnc2)C)CCCC1NC(c1ccc(F)cn1)=O CC1CC(C(=O)NCC2COC2)CC(C)C1.c1(C2(C=O)CCC2)ccccc1.N c1(C(=O)NC2CCN(Cc3ccc(OC)nc3OC)C2)cc(F)c2cn[nH]c2c1 C1(NC(c2n[nH]cc2[N+](=O)[O-])=O)CCN(C(=O)C(c2cccc(F)c2)O)CC1F C1(NC(CCN(CCC)C)=O)CCCC(CNC(=O)CC2CC3CC3C2)C1 c1(C(=O)NC(CNC(=O)CC2CN3CCC2CC3)C2CC2)cnc2ccccc2n1 O=S1(=O)CCC2(CC(NCc3ccc(C4CC4)o3)CCO2)C1 N1(C(=O)OC(C)(C)C)CC(NC2CN(CC(F)F)C2)C2CCCC12 c1(CC(=O)N)ncc(F)cc1F.C1(CC)CCC(C(N2CCC(F)(C)C2)=O)CC1 C(C(O)(CO)CO)NC(c1scc(CNC(c2c(CC)nn[nH]2)=O)c1)=O C(=O)(C1CCCc2sc(C)nc21)N1CCC(F)(CNC(CCCOC)=O)C1 C12(C=O)CC(C1)C(C(F)(F)F)O2.C1(NC(=O)CCc2nccs2)CCCC1.C c1(C(=O)N)ccc2c(c1)COCO2.C(C)(C(=O)NC1(C)CCC1)OCC#C CCCCC(C(=O)NCC(C)(C)C1CC1)NC(=O)CCC1CCCO1 N1(C(C(C)C#N)=O)CC(C)(CNC(=O)C2CC2)CC1(C)C N1(C(C2(C)CCN2C(=O)C=Cc2cscn2)=O)CC(O)C(O)C1 CCC(C(=O)NCCc1nc(C)no1)NC(C1CCCN1CC)=O c1(C(N2CCC(NC(C(CC)C(C)O)=O)(CO)CC2)=O)cc(Cl)c(F)c(Cl)c1 c1(C(=O)N)cc(C)c(S(N)(=O)=O)cn1.C(C)(CCC(=O)N(CC(C)C)C)SC CC1(C)CNC(=O)c2c(C(N3CCC(CNC(C4CCCO4)=O)C3)=O)coc2C1 N(C(=NCCC(C)=O)NCC1(OCC)CCOC1)CC(c1ccc(C#C)cc1)=O c1(OC)cc(OC)c(CNCC2(c3ccccc3)CC2(C)C)c(C)c1Br C1(NC(CCC(C)(C)N(C)C)=O)CC2CC(C1)N(C(c1cccc(F)c1Cl)=O)C2 C1(CC(=O)N(C23CC(C2)C3)CC)CCN(C(C2CS(=O)(=O)C2)=O)C1 c1(C(=O)NCC2(F)CCC(F)(F)CC2)cnc2c(c1)CNC2 c1(C(=O)NC(C)CCNC(c2ccnn2CC(F)F)=O)cnc2c(cnn2C)c1 N1(C(c2ccccc2)=O)CC2=C(C1)CN(C(=O)C=CSc1nc[nH]n1)C2.C(C)=C.C Cc1cc(C(=O)N(C2CCCN(C(c3cccs3)=O)C2)C)c(F)cc1Cl CCC(CC)C(C)C(=O)NC1CC12CCN(C(c1cc(C#N)no1)=O)CC2 O=C(N=c1cc2n([nH]1)CCOC2)C(=O)OCCc1ccccc1OC(F)(F)F c1(C(=O)NC2CC(C)(NC(c3ccc(C)o3)=O)C2)ccc(-c2ccco2)nc1O N1(C(Cc2n(C)ccc2)=O)CCCCC(CNC(=O)C(C)(C)C)CC1 C1(C(=O)NCCC(=C)CNC(c2cc(C3CC3)ns2)=O)(OC)CCCSC1 N1(C(C(C)NC=O)=O)CC2C=CC1C(C(=O)N(C)Cc1ncc[nH]1)C2 N1(C(C2CC(C#C)(O)C2)=O)CCC2(CC2NC(=O)Cc2cnnn2C)C1 C1CC2C(C1)C2(F)F.c1(C(=O)NC(C(=O)N)C2CCC2)ccc(C2CC2)o1 C(=O)(C1=C(Cl)CC1)NC(CSCC)C(=O)NCCC(O)C(C)C C1(CC(N2C(COC)C=CC2)=O)CC(C)N(C(=O)C=C=C(C)C)C1 c1(C=O)cnc2[nH]ccc2n1.C(C(=O)NC(C)(C)CC(C)C)(C(C)(C)C)OC.N N1(C(CCC#CC)=O)CC(CC(=O)NCC2(OC)CCC(C)C2)C2(CC2)C1 C(=O)(C(C)(C)C(=O)OC)NCC(C(=O)NC1(CC=C)CCCC1)C N1(CCCNC(C(=O)N(C)C)=O)CCN(C(=O)C(C)SC(F)(F)F)CC1 N1(C(c2n(CC)nc(C)c2)=O)CC2(C1)CN(C(=O)CCn1cncn1)CC2CO c1(OCCC(=O)NCC(CC)NC(=O)C(O)CC2CCCCC2)ccccc1Cl c1(OC)cc(N2CCC2C(N2CCC(c3ccnn3C)C2)=O)nc(OC)n1 C1(C(N2C(CNC(=O)Cn3nnc(=O)[nH]3)CC2)=O)COCCOC1 C(=O)(C(C)(C)CC(C)=O)N1CCN(C(C(CC)N(C)C)=O)C(CC2CC2)C1 CC1CN(C(c2n[nH]c(C3CC3)n2)=O)CCC1CNC(c1cnc(Cl)[nH]1)=O c1cn(C2CCN(C(C3CC3F)=O)C2)nn1.c1(C(=O)NC)nc(C(F)F)cs1 c1(C(N2CCN(C(C(CC#C)O)=O)C(CCC)C2)=O)cc(C)nc2onc(C)c12 Cc1cc(C(=O)N(C(CNC(=O)CC2(O)CCOC2)C2CC2)C)cc(Cl)c1 C1(C(N2CCCC(CCC#C)C2)=O)CN(C(C2CC(=O)CS2)=O)CC1C1CC1 C1(NC(C(C2CC2)OC)=O)CS(=O)(=O)CC1.c1ccnc(C)n1.C(C)C.N CC1=C(C)CN(C(c2cc(CNC(C3(C)CC4C=CC3C4)=O)cs2)=O)CC1 C(C(C)(C)C#CC(=O)N(C)Cc1nncs1)NC(c1cc(C(C)=O)[nH]n1)=O N1(C(C23C(C(N)=O)(CCC2)C3)=O)CC2CCC1C2.c1(CC=O)cncn1CCC CC(C(C)(C)C(=O)NCCCCC(F)(F)F)NC(c1cccc(F)c1F)=O C#CCC(O)C(=O)N1CCCC(CCNC(=O)C(C)=CC=C)C1 c1(C(=O)NC(COCC)C(=O)NCCCCCN(C)C)cn(C)c(=O)cn1 C1(NC(C2(C)CCCCC2)=O)COC2C(NC(=O)C(F)(F)c3cscn3)COC12 CC(C)(C)CCCNC(=O)C(C1CCC1)NC(C1CC1)=O.C(C)(=O)O c1(NC(C(CC)OC(C2CCCN2c2cnccn2)=O)=O)ccc(F)cc1 c1(C(=O)NC(Cc2cnc(O)nc2O)C(=O)O)cnn2ccc(CO)cc12 c1(C(=O)NC)cccc(C(=O)NC2CCC2)n1.C1(C=O)CC(O)C(F)C1.C c1(C(=O)NC(c2ccncc2)C)ccc2[nH]nc(C3=COCCC3)c2c1 c1(OC)ccccc1CC(N1CC2CC2(NC(C2CCOC2)=O)C1)=O.C(C)C.O CC1CN(C(C2CC2Br)=O)CCN1C(c1cccc(CC#N)c1)=O C(c1cccc(F)c1F)=CC(N1CCC(NC(C2CC3CCC2O3)=O)C12CC2)=O c1(C(=O)OC)c(C)ccc(C)c1C(N1CCC1)=O.C1(C=O)CC12CC2.CC C1(NC(c2nc(C)oc2)=O)C2CC3CN(C(C4CCC5CC4C5(C)C)=O)C1C3C2 c1(C(N2C(CNC(CCCCC#C)=O)COCC2)=O)ccc(C)c(S(C)(=O)=O)c1 c1(OCC)ccccc1C(=O)NC1CC(C)N(C(c2oc(Br)nc2C)=O)C1 c1(C(N2CC(O)CC(C)(C)C2)=O)cc(F)cc2[nH]ncc12 C1(C(=O)NC(C)C(C)(C)NC(c2cnc[nH]2)=O)CC(C2CC2)=NO1 C1(CC(=O)NCCSCC(C)(F)C(C)C)(C(=O)OCC)CCCNC1=O CCC(C)(C(=O)NCC(C)(CO)NC(c1ccc(C)c(F)c1)=O)C(N)=O Cc1cc(C(N2CC(NC(C3CC(=O)NC3(C)C)=O)C(C)C2)=O)c(Cl)cc1F C1(C(=O)NC(C)Cc2ccc(C)cc2)(OC)CCCCCC1.C(=O)C(C)(F)F CC(Cc1nccn1C)N=c1nc(N(C)CCC2CN(C)C2)c2ncccc2[nH]1 CCCC(CC(C)C)C(=O)N1CCCC1CNC(C1(O)CCCC1)=O Cc1cc(C(N2CCOC(C(C)NC(c3sc(=N)[nH]c3C)=O)C2)=O)sc1C CCCC(C)(CCC)C(=O)NC1CC(CNC(=O)C2=CCS(=O)(=O)C2)C1 CS(=O)(=NC(=O)C1COC(C(F)(F)F)CN1)c1ccccc1Cl c1(C(N2C(CCNC(C(C)SCCCC)=O)CCC2)=O)ccncc1O CC1(C)CC(N2CC(OCCF)C2)c2ccccc21 N1(C(C2CC(C#C)(O)C2)=O)CC(C(N2CCOC(C#N)C2)=O)OC(C)C1 c1(C(N2CC(C(=O)NC(c3n(C)cnn3)CO)OCC2)=O)cc(C#N)ccc1N n1(CCNC(=O)CC2(O)CCC2)cc(NC(c2cnc(C3CC3)s2)=O)cn1 C(C(=O)N1CCC(C(N2CCC(n3c(C)cc(C)n3)C2)=O)O1)NC1CC(=O)NC1=O c1(C(=O)N)c(F)ccc(N)c1F.Cc1nc(C(=O)NC(C)(C)C(C)C)n(C)n1 c1(OC)ccc(C(=O)NCCCC(C)NC(C2CCCC(F)C2)=O)cc1C1CC1 c1(OC)ccc([N+](=O)[O-])c(C(=O)N(C)CCNC(C2CCCCO2)=O)c1 c1(C(=O)NCCC2(O)CCCN(C(COC)=O)C2)coc2c1CCCC2 N1(C(CCNC(=O)OCC)=O)CCN(C(c2cc(C)n(C)n2)=O)C2COCC12 Cc1nc(C(=O)NCC2(C)CC23CCC3)c(=O)[nH]c1C.C1(C=O)CC1(C)C CN1CCC(NC(C2(CC(=O)O)CCC(F)(F)CC2)=O)c2ccccc21 S(=O)(=O)(c1c(Cl)nc2sccn12)N(CC(=O)OCc1ccccc1)C c1(C(=O)NC2C(CNC(c3cnsc3)=O)CC2)cc(O)cc(Br)c1 Cc1ccc(OC2CCCC2)cc1OCc1cccc(COc2nccn2C)c1 C1(C#CC(=O)NC2(C)CCN(C(=O)C=CC(C)(C)SC)C2)(CC)CC1 Cc1cc(C(=O)NCc2n[nH]cc2C(=O)NC)cc(O)c1.C1CC12CCOC2 CCC(C)(C)CCCC(=O)NCC1COC(CNC(c2ccc(F)cn2)=O)C1 C(=O)(C(F)C(F)(F)F)N1CCC(NC(C(F)=CCC)=O)(COC)C1 C=C(C)CCC(=O)NCCOCCN(C)C(c1ncccc1NCC)=O N#CC1CC=C(c2ccc3c(c2)COC32CN(C(c3cc(O)no3)=O)C2)CC1 C(=O)(C(C)(C)CC(=O)NCC1CCCC1)OCC.c1(C=O)cnccc1C.N Cc1cc(C(=O)NCCC(C)N(C)C(c2coc(N(C)C)n2)=O)cc(O)n1 n1(CC(=O)NC2C(CNC(COC(CC)C)=O)C2)c(C)csc1=O Cc1nc(C)c(C(=O)NCC(C)(C)CCNC(=O)C)c(C)n1.C1CCOC1=O C1(NC(C2C(C(=O)O)C23CC3(F)F)=O)CCC2(CCCN2)CC1 Cc1c(C(=O)NC2C3CC2N(C(=O)Cc2csnn2)C3)sc2ccc(F)cc12 C=C(C)CCC(=O)NCC1CN(C(C2CCC2c2ccc(F)cc2)=O)C1 Fc1cc(CNC(c2ncco2)Cc2ccccc2)c(Cl)cc1I N1(C(C2N=C(C)SC2)=O)CC(NC(=O)CC2CC=CCC2)C2CCCCC12 C12(CNC(COC)=O)CCC(CN(C(=O)CP(C)(C)=O)C1)C2 N1(C(CCC2CC(C)C2)=O)CCC(C(C)NC(=O)CC2CC2)CC1 C=CCCC(F)(F)C(=O)NCC(CC(F)(F)F)NC(=O)Cc1cncnc1 C1(NC(c2cccc[n+]2[O-])=O)(CNC(C2(NCCO)CC2)=O)CCCCCC1 CN1CCC(CNC(C2CCCN2C(=O)CC2CCCSC2)=O)C1 c1ccc(O)c(C)c1.C1CCC(=O)NC1.C12(CC=C)CN(C1)C2=O.C(=O)(C)N CC(C)CC(O)C(C)C(=O)NC(C)CCC(=O)NCCCCCCN(C)C N1(C(c2c(C)onc2C2CC2)=O)CCC(NC(c2c[nH]nc2[N+](=O)[O-])=O)C(O)C1 c1(C(=O)NC(C(C)NC(CCCCCOC)=O)C)nc2ccccc2nc1C c1(C(=O)NCCCCNC(C(C)(C)C(F)F)=O)cccc2c1C(=O)NC2=O Cc1nc(C)c(CC(=O)N)s1.C1(O)(CC)CCN(C(c2c[nH]nc2C2CC2)=O)C1 Cc1cc(C(N2CC3C(CC(=O)NC(C)CCCO)C3C2)=O)ccc1F c1(C(N2CCn3cncc3C2)C(=O)NCC(=C)C)cc(F)cc(Br)c1OC N1(C(c2cc(CC)ncn2)=O)CCC(C)N(C(c2nccc(OC)c2F)=O)CC1 c1(C(C(=O)NC(CC)C)N(C(C)CC(N)=O)C)cnc(OC)c(Br)c1C C(=O)(C1=C(Cl)CCC1)N1CCC(CC(=O)NCC(c2n(C)ncc2)O)CC1 c1(C(=O)NCC(CCOC)NC(=O)CC2C=CCC2)cccn2ccnc12 Cc1cc(C)c(C(=O)NC2CCC2NC(=O)C(C)(O)Cc2ccccc2)cc1N N1(C(C(c2cn(C)nn2)NC(CC)=O)=O)CCC(OC)CC1.c1nc(C)c(C)s1 c1(CC)cn2c(n1)CCC(C(=O)NCCC1CSCCN1C(=O)CCF)C2 c1(C(=O)NCC(n2cc(C(CC)CC)nn2)C)ccnc2[nH]ncc12 Cc1cc(CC(C)NC(=O)CCOCCCNC(=O)C)n[nH]1.C1CCCO1.S CC(C)CC(C)(CO)NC(c1coc(CNC(=O)CCC2CCCC2)c1)=O Cc1c(Cl)ccnc1C(N1CC(NC(c2ccc(OCF)cc2)=O)C1)=O N1(C(CC(CC=C)NC(C2CCC=CCC2)=O)=O)CCC(C)C(C)(C)C1 c1(-c2c(SC)cccc2)cc(C)c(S(=O)(=O)Nc2cccc(Cl)c2)cc1C C#CC1(C(=O)NCC2CC(C)C2)CCN(C(c2cc(O)nc(C)n2)=O)C1 c1(C(N2CCCC2)=O)cn(C)ccc1=O.CC(C(=O)N)NC(c1ccco1)=O.C C1(F)(C(N(CC(C(=O)N(C(CC)C2CC2)C)C)C)=O)CCCCCC1 C1(C(N(C2CCN(C(=O)CC(C)(C)C)CC2)CC#C)=O)CN=C2N=CNN2C1 N1(C(=O)COc2ccsn2)CC2(CCCN(C(C3(F)CC3)=O)C2)C1 C(CCCSCCC(=O)N)NC(C1C(C)C1)=O.n1(CC=O)ccnn1.CCC c1(C(C(=O)NCC=C)N(C)CC2CCN(C(C)=O)C2)ccnn1COC c1(C(N(CCCNC(C2C=CCC2)=O)CC)=O)csc(C)c1 C(=O)(C(C)(C)C(O)c1cc(Cl)cc(Cl)c1)OCC(c1cc(C)on1)=O Cc1c(C(=O)NCC2CC2)ncn1C.c1(C=O)ccc(N(C)C(C)C)cc1.C N1(C(Cc2cnc(C)s2)=O)CC2CC(C)NC2C1 c1(Oc2ccc(OCCC)c(C(C)C)c2)ccc2c[nH]nc2c1 Cc1scc(C(=O)NCC(C)C(=O)NC2CCSCC2)c1C c1(CNC(C2C3CNCC23)=O)ccc(-c2cscn2)nc1 C1(C(=O)NC(c2cccc(O)c2)C)CC12CCN(C(=O)Cc1cncnc1O)C2 N1(C(C2(C#C)CCC2)=O)CCN(C(c2nn(C)cc2S(N)(=O)=O)=O)CC(C)(C)C1 CC1C(NC(=O)CSC(F)(F)F)CC2CCC1N2C(=O)CC1CC2CCC1O2 CCCCCC(C)CC(=O)NC1CC2(C1)CC2NC(c1cc(C)c(CO)cn1)=O C(=O)(CC(CO)C)N1C(CN(C(c2cc(CC)on2)=O)C2CC2)CCC1 C(=O)(C(CC)C(=O)OC)NCC1(NC(c2c(CC=C)cccc2)=O)CCC1 c1(NC2CC(OC(C)(C)C)C2)nccc(N2CCC(Cc3ccc(N)cc3)C2)n1 N1(C(CCC)=O)CC2CN(C(=O)Cc3ccc(CCC)cc3)CC2C1 c1(OC)ccc(Br)c(OC(=O)CC2CCC(=O)N2Cc2ccccc2)c1 c1(N(C)C(c2c(C(F)(F)F)cncc2F)=O)cccc(S(C)(=O)=O)c1 C12(CNC(CNC(c3snc(C)c3N)=O)=O)CC=CC(C1)OC2 n1(CC)c(C(=O)N(C)CCO)cc2ccccc12.C(=O)(C(C)(C)O)N(CC)C c1(CN2CCC(NC(C3C(C)CCC3)=O)C2)ccc(C(=O)O)c(F)c1 c1(NC(C2N(Cc3sc(C)c(Br)c3)CCNC2)=O)cc(Br)ncc1[N+](=O)[O-] C(=O)(CCCC(=O)C(C)(C)C)N1CCC(CCOC)(NC(C(CCC)C)=O)CC1 c1(C(=O)NC2CC3CN(C(C4C(OC)CCC4)=O)CC32)ccc2n[nH]cc2n1 c1(OC)c(Cl)cc(C(=O)NC2(C)CC(NC(c3cnc(O)n3C)=O)C2)cc1Cl CC(C(=O)NCC12CCC(C1)N(C(c1csc(Br)n1)=O)C2)C(C)(C)C C12(C(=O)NCCC(CC)(CC)NC(c3ccco3)=O)CCCCC1NC(=O)CC2 C(=O)(C(C)(O)CCN(C)C)NCC=CCC(=O)Nc1c(C(C)C)nsc1 C12(NC(CCCNC(=O)OC)=O)CCC(CC1)C2.C1(C=O)CCOC(C)C1.N C=C1CC2CCC(C1)N2C(=O)CCC1CCCN(C(=O)C(C)CCOC)C1 N(C(=NCCCF)NCC1(CO)CC1)CC1CC(=O)N(C2CCCCC2)C1 N1(C(CC(C)C(C)(C)C)=O)CCC(C2CCCN(C(C3(C)COC3)=O)CC2)CC1 CC(CCCc1ccccc1)C(=O)NC1CCN(C(C2(F)CCCCC2)=O)C1 N1(C(C(CC=C)OC)=O)C(C)CN(C(c2c(C)cc(C)nc2O)=O)CC1C N1(C(C=CC(C)(C)NC(c2ccc(OC)o2)=O)=O)CCC(F)(C#N)C1 N1(C(CC(C=C)(C)C)=O)CC(C)N(C(C2CC3(C2)CC32CC2)=O)CC1C C(c1cc[nH]n1)=CC(=O)N(CC(C)C)C.C(=O)CN(C)C1CC1.C=O.C CC(C)(C(=O)N1CCC1)C1CCCN1C(=O)CCc1ccncc1 c1(CC)occc1C(=O)NCc1nocc1C(=O)NOCC(=O)N(C)C c1(C(=O)NC(C(N2CCOCC2)=O)C2CCCO2)cnc(S)nc1 C(=O)(C#CC1CCOC1)N(CC(C)NC(Cc1c(C)nn(CC(C)C)c1C)=O)C c1(C(N2C(CCCNC(=O)CC(F)(F)F)CCCC2)=O)ncnc(O)c1F c1(C(=O)N)cc2c(nc1O)CCN(C)C2.CC1CC(=O)NC1C(N1CC(C)C1)=O C1(C(F)(F)F)(OC)CC(C)C1.C12(C=O)COCC1C2.C1(C=O)CC(O)C1 C(=O)(C1CCc2nccn21)NCCNC(CC(C)N(C)C)=O C1(NC(C=C(C)C)=O)C2CC3CN(C(c4cscn4)=O)C1C3C2 C=CCCCC(C(=O)N(C)CC1CC1(C)C)NC(c1ccsc1)=O C1(C(=O)NCC2(NC(C3C(C)OCC3)=O)CC2)CC(F)(F)CCC1(C)C N1(C(c2cc(C)nnc2)=O)CCC2(NC(c3occ4c3CCC4)=O)CC2C1 C(=O)(C(C(O)C(C)C)NC(c1coc2c1CCCC2)=O)OC c1(OC)ccc(C)cc1C(N1CC2CC1CN2C(c1cccc(Br)c1)C(N)=O)=O Cc1cc(C(=O)NCC(CNC(=O)COC2CCOC2)CO)c(C)cn1 C1(CC)CCN(S(=O)(=O)Cc2nccn2C)C(CO)C1 c1(-c2ccc(C(=O)NC(C3CCOCC3)C)nc2)cccc2c1OCCCO2 C(CC(C)(C)NC(C1(COC)CN(C(=O)C(C)C2CC2)C1)=O)OC c1(C(=O)NC(C(C)NC(C2(C(=O)OC)CC2)=O)C)ccc(=O)n(C)n1 C1(CNC(CC2C(CNC(C(C3CCCCC3)C)=O)C2)=O)CN2CCC1C2 Cc1ccc(CC(=O)NC2CC3(C2)CC3)c(F)c1.C1(CC=O)CC(C2CC2)C1 C(=O)(C1=NOC(C)(C)C1)NC1CCN(C(C2C(OCC)C2)=O)CC1CO c1(CC)ncc(C(N2CCCC(NC(C3CCSC3)=O)C2)=O)c(C)n1 C(=O)CC(F)(F)F.Cc1nc(CSCCC(=O)NCCC)cs1.C(=O)(C)N CN1CCC(O)(C2(C(N3CCN(C(=O)CCC4CC4)CC3CCO)=O)CC2)CC1 N1(C(CCCOCCC)=O)CCC2CN(C(=O)Cn3cc(CO)nn3)CC2CC1 C(=O)(CCCCN1CCCCC1)NCCC(C)(C)NC(=O)CC1(C)CCC1 C(=O)(CCCCCCC(=O)N(C1CN(c2ncc(Br)c(C)n2)C1)C)OC c1(C(N2CC3CCC2CC3)=O)[nH]nc2c(-c3cccc4ccccc34)cccc12 CC1CC(C(N2CCC(CCNC(=O)COC3CCCOC3)C2)=O)CC(=O)N1 c1(CN2CCC(OCC)C2(C)C)n[nH]c2ccc(Br)cc12 N1(C(c2c(C)c(Br)cnc2)=O)C2CCC1CC(NC(=O)C(C)CC(F)F)C2 CC1CCC(C)CN1C(=O)C(C)Cc1cnc[nH]1.C1(CC=O)CC(C)(C)CO1.N C12(NC(=O)CC3CC4C=CC3C4)CCC(NC(c3cnco3)=O)(CC1)C2 C(=O)(CCCC(=O)NCC(C)NC(=O)C(c1cccc(OC)c1)C)NCC N1(C(c2cn(CCOC)nc2)=O)CCCC(C)C1.CCC(F)(F)F.C(=O)(C)N C1(C(=O)N)CC2(C1)CC2F.C(C)(CO)NC(CNC(=O)OCC=C)=O CC1CN(C)C(C)CC1N(C(c1ncc(Cl)cc1Cl)=O)C(C(C)(C)C)=O N1(C(c2n(CC)cnn2)=O)CCN(C(=O)C(C)(F)C(C)(C)F)CC(C)(C)C1 N1(C(c2c(C)nncc2)=O)CCC2(CC1)CC2C(=O)NCC1CC12CC2 c1(C(N(C)CCNC(=O)CC2CC3C=CC2C3)=O)ccn2nccc2n1 N1(C(c2cnc(CC)[nH]2)=O)CCC2(CNC(=O)C(C)N(C)C)CCCCC12 C(CC(CC)C(=O)NC(C)CC(=O)NC1CC2CC2C1)=CC C1CCCOC1.c1(C(=O)N)ccc(C(F)F)o1.CC(C=O)NCC1(C)CC1 CN=c1[nH]cc(C(=O)NC2(C(=O)NOCCCN(C)C)CCSC2)o1 C(=O)(C(C)(C)C(=O)NCC(C)C(=O)NCC(C)(O)C1(C)CC1)NC C(=O)(C1=CCC(NC(c2nonc2N)=O)C1)NC(CCSCC)C Cc1nnccc1C(=O)NCCC(=O)NCCS(N)(=O)=O c1(C=O)cn2ccccc2n1.C(C)(C(=O)N(C)CC1CC1)NC(=O)OC.N c1(C(N(C)Cc2c(C)nsc2)=O)ccc(C2(O)COC2)cc1 c1(C(=O)NC2(CC)CCCN(C(C3(C)CC(=C)C3)=O)C2)cc2c([nH]1)CCCC2=O N1(C(=O)C=Cc2cccc(Cl)c2)CCCCC1C1CC(N=c2[nH]nco2)CCO1 C1(NC(c2cc(Cl)c(Br)s2)=O)CCC2(C1)CN(C(c1onc3ccccc13)=O)C2 C1(C(N2CC(C3CC3)C2)=O)CCS(=O)(=O)C12CCC2.c1(C=O)cccc(=O)o1 n1(CC(N2C(C(=O)Nc3nccc(C)c3Br)CC(O)C2)=O)cc(C)c(O)nc1=O N1(C(c2cnc(CC)s2)C(=O)NCCC2(C)CC2)CCCC2(C)CCCC12 n1(CCC(=O)N(C)C)cc(CCCNC2CSC(C(F)(F)F)C2)nn1 C1(CNC(CCCCC#C)=O)COC(C)(C)CN1C(C1CCOC1C)=O n1(CCC(N2C3CN(C(=O)C=C4CCOCC4)C(C3)C2)=O)ccc2cccnc12 C(CC(=O)N(C(C)CNC(C1CCC(C)CC1)=O)C)(C(C)C)OCC C12(C(=O)NCCOCCN(C)C(C3CCCCCC3)=O)CCC(CC1)OC2 c1(CSC)cc(C(N2CCN(C(=O)Cc3ncc(C)s3)C3CC23)=O)ccc1F CCCC(CNC(C1(OCC)CCOCC1)=O)C(=O)N1CCC1CO CC1(C)C(CC(=O)NCC(CO)NC(c2ccoc2C(F)(F)F)=O)CC1O Cc1nc(NCC2CC(NC(=O)C(c3ccc(F)cc3C)O)C2)c(C)c(O)n1 C1(C(=O)NCCCCCNC(CSCC)=O)CCCC(F)C1 C=C(C)CC(C(=O)N(C(C)CC(F)(F)F)C)NC(C1CCCN1C)=O Cc1cccc(CC(N2CCC(NC(c3cc(CO)ccc3Cl)=O)CC2)=O)c1C c1(COC)n[nH]c(=NC2(C3CN(C(C4CC(C)OC4C)=O)C3)CC2)s1 C(=O)(CC(C)CC(C)C)N1CC(CCCC)N(C(=O)Cc2nccn2C)CC1 C1(CCNC(C#CC(C)C)=O)CC(F)(F)CN1C(c1cc2n(c1)CCC2)=O O(NC(=O)C(CNC(=O)C(C)(C)CC(F)F)CC1CCCC1)CCCOC Cc1ccccc1C(C)C=O.C1(CC(=O)N(CC)CC)CC(F)(F)C1.CCO c1(NC(=O)NCCCn2c(C)cnc2)ccc2c(c1)CCCN2C c1(COC(CCSC)=O)ccc(C)c(OC(F)F)c1 CN1N=C(C(=O)NC23CC(CNC(=O)C4=NOCC4)(C2)C3)CCC1=O Cc1cc(C(=O)N=c2ccn(CCC(C)C)[nH]2)c2c(c1)CCC2 Cc1sc2nc(CC(N3CCC(C(c4nn[nH]n4)(C)C)CC3)=O)nc(O)c2c1C c1(C=O)cc(Cl)ccc1F.c1(CC)[nH]c(=N)sc1C(N1CCCC1C1CC1)=O.N c1(OCC(=O)OC)cc(C(=O)O)ccc1.C1(C=O)CCC(C(C)(C)C)N1 c1(C(n2nccc2C(=O)NC(=O)C(N)Cc2cocn2)C)ccc(F)cc1 C1(C(=O)NCC(C2CCC2)NC(C(CSC)(C)C)=O)CN2CCN1C(C)C2 Cc1ccc2c(C(=O)NC3(CNC(=O)CCCS(N)(=O)=O)CCOC3)c[nH]c2c1 c1(OC)cc2c(c([N+](=O)[O-])c1)N(C(=O)Nc1ccc(O)nc1)CC2.C1CC1.C N1(C(c2n(C)ncc2)=O)CCC(C(=O)O)C(C(C(=O)O)C(c2ccccc2)=O)C1 c1(OC(C)C(=O)NC2CCCC2)cccc(C#N)c1.c1(C(=O)N)csc(C#N)c1 C1(CN2CCC(CC(=O)OC(C)C)C2)C2CN(Cc3ccncc3)CC12 C(=O)(CC(C)(C)C1CC1)N(C1CN(C(c2cc(CC(C)C)on2)=O)C1)C N12CCCC(O)(C1)CCC2=O.N1(S(CC)(=O)=O)CCCC1C.C(=O)(CC(F)F)N c1(CC)ccc(C(=O)NCCC2(OC)CN(C(=O)CCC3CC3(C)C)C2)s1 C1(NC(CCSCC)=O)CC2CCC1C(NC(C1(CO)COC1)=O)C2 c1(OC)ccc(CC(=O)NCCCN(C)C(C2(C)CCCC2C)=O)c(Cl)c1 C1(NC(c2oc(C)c(CO)c2)=O)CCN(C(c2cc([N+](=O)[O-])n[nH]2)=O)CC1(C)C C1(CCNC(=O)COC2CCCC2)CCCN(C(=O)C2=COCC2)CC1 CC(CC(N)=O)C(=O)NC1CN(C(=O)CCC(F)(F)F)CC1O C(C)(C)(CC(=O)NCCC1(C)CCOC1)NC(C1N(CC)CC1)=O Cc1ccncc1C(N1CCC(C)(C(N2CCC(O)(CO)C2)=O)C1)=O c1(OC)ccc2c(c1)OCC(C(N1CCCC1C)=O)C2.c1(C(=O)N)cc(Cl)no1 C1C2CCCC12.c1(C=O)cnn(C)c1C(F)F.C1(C(N(C)C)=O)(C=O)CC1 C12(C(N(C)CC3CCN(C(C(C)OCOC)=O)C3)=O)CC3CC(CC(C3)C1)C2 c1(C(N2CCCC(NC(C(C)SCC)=O)C2)=O)c(C)c2cc(O)ccc2oc1=O CC1CN(C(=O)Cc2ccccn2)CCN1c1nc(Cl)c(C#N)s1 c1(C(=O)NCC(=O)NCC=C)c[nH]nc1CC.C1(C(C=O)F)CCCCC1 c1(NC2CC(C)N(C(=O)CCc3cncnc3)C2)ncc2ccsc2n1 Cn1ncc2c(C(N3CCC4(NC(=O)CCCCCF)CC4C3)=O)cccc12 C1(N(C(=O)CC(C)(C)O)CC)CCCN(C(c2cccc[n+]2[O-])=O)CC1 N1(C(C(Cc2cn(C)nc2)O)=O)CC2CC2(CNC(=O)CCc2ccc(Cl)s2)C1 c1(OC)ncc(F)c(=NC(=O)C2CCCN(C(C34CC(C3)C4)=O)CC2)[nH]1 C(=O)(CC(F)(F)C(C)C)N.n1(CC)ccc(C(N2CC(OCC)C2)=O)cc1=O C1(C)(COC)CCCN1C(c1csnc1C)=O.c1(C(=O)N)cnc(N(C)C)s1 Cc1ccc2c(C(=O)NCC3C(Cn4cc(CCO)nn4)C3(F)F)coc2c1 CC(CC(=O)NC1CC2CN(c3nc(C4CCCC4)nc(=N)[nH]3)CC12)C(F)(F)F C1(OC)CCC12CC(C(N1CCN(C(=O)CCn3cncn3)CC1CCO)=O)C2 c1(C=O)ccnn1C(F)F.c1(C(=O)N)ccn(C(F)F)n1.C1(CC)CCCC1 C1(C(N2CCN(C(CCC=C)=O)C3C2CC3)=O)CCn2c(C)nnc2C1 c1(OC)cc(C(=O)NCC(C2CCCCN2C(C2CCC2)=O)(C)C)cc(N)c1O C1(NC(CC=C)=O)(CNC(c2cnn3c2OCCC3)=O)CCC(F)(F)CC1 CCCCC(CC)C(=O)N(C(CC)C(=O)NCC(N)=O)C CCC(C)(C)CC(=O)NC1CC(OC)CN(C(=O)C=Cc2ccc(Cl)s2)C1 c1(OCC)n[nH]cc1NCc1ccccn1 C12(COC)CN(C(=O)NCCCCn3cnnc3)C(C(=O)O)(C1)C2 CC(C(=O)NC(C)(C)CN(C)C(C1(C)CC1)=O)n1ccnc1 n1(CC(N2CC(NC(COC)=O)C(n3cccn3)C2)=O)ccc(C)cc1=O c1(CN(C)C)ccc(C=O)cn1.CC(C)(O)C.C1(C(F)(F)F)(C=O)CC1.N C1(NC(C(C=CCCC)O)=O)CCCN(C(=O)CSCC2CCCCO2)C1C c1cccc(F)c1Cl.c1(CSCCCNC(CCN(C)C)=O)cn(C(=O)N)nn1 C(=O)(C(C(C)OC)NC(=O)CCc1ccccn1)NCC(CSC)OC CC1(C)CC(NC(=O)COCC)CC(O)C1.c1(C=O)coc(C(F)F)c1.N C(=O)C1=NN(C)C(=O)CC1.Cc1cnn(C(C)C)c1C(=O)NC(CC)C(C)C C(=O)C(C)(C#N)CC.c1(C(C)C)ccc(CCNC(C2(C3CC3)CC2)=O)cc1 CCC(COC)C(=O)NCCN(C(=O)CN1CC(C)(OC)C1)C(C)C C1(C(=O)NCc2nccs2)(OC)CCN(S(=O)(=O)CCCCCl)CC1 N1(C(CCCNC(C)=O)=O)CCC(NC(c2ncn3c2COCC3)=O)C(C)(C)C1 O=C(C1=CCCS1)NCC1(O)CCN(C(c2cc(Cl)cnn2)=O)C1 C1(NC(C(C)OC)=O)CN(C(c2cccc(C3COC3)c2)=O)CC2(CC2)C1 CC(c1ccccc1Cl)=CC(N1CCN(C(=O)C=CC(C)C)CC1CN(C)C)=O N1(C(Cc2c(C)scc2)=O)CCCCC(CNC(=O)CC(O)C(C)C)C1 N1(C(COCCOCC)=O)CCC(F)C(NC(c2cccc(C)c2C)=O)C1 C1(NC(C(F)=CCC)=O)CCN(C(=O)C(C)Oc2ccccc2F)CC1C C12(C(N(C)CCC3CCOCC3)=O)CCC(CN(C(=O)CC3CCOC3)C1)C2 c1(-c2ccc(C)c(SCCO)c2)n[nH]c2cc(C(=O)NCCN(C)C)ccc12 C(C)(N=c1ccnc(NCc2nnnn2C2CCC2)[nH]1)c1c(C)cc(Br)cn1 C(C(C(=O)NCCS(N)(=O)=O)NC(=O)C1CC1)N(C)C Cc1c(CC(=O)NCC2C(C(=O)NCC(Cl)C(C)(F)F)C2(C)C)cnn1C C(CN=c1nc(O)c2ccccc2[nH]1)(C1CC1)NC(c1ccn(C(F)F)n1)=O N1(C(c2c(C)ncnc2)=O)CC2=C(C1)CN(C(=O)Cc1csnc1C)C2 C1(O)CCN(C)C1.C1(N(CC(=O)N)C(C2(CCCC)CC2)=O)CC(C#N)C1 Cc1cccc(CC(CO)NC(=O)NCCc2cocn2)c1 N1(C(CCC)=O)CCC2(CC1)CCN(C(c1nncn1C1CC1)=O)C2 N1(C(C(CC=C)C)=O)CCCCC(NC(c2csc(C)c2Br)=O)CC1 c1(C(N2CC3C(NC(c4cncc(C#N)c4)=O)C3C2)=O)ccc2ncnn2c1 N1(C(C2(COC)CC=CC2)=O)CCN(C(c2cnc(Cl)s2)=O)C(CC(F)F)C1 C12(C(N3CCCN(C(C=C4CCC(C)C4)=O)CC3)=O)CC(C)(C1)OC21CCC1 N(C(=NCCCc1ccccc1)N1CC2CCOC2C1)C(CC)C N1(C(C2(OC)CCCOC2)=O)CCCC(C)(CNc2cncc(C#N)n2)C1 n1(CC(=O)NC2CCN(C(C(CC)O)=O)CC2)cc(Br)ccc1=O N1(C(C2(F)CN(C(c3nc(C)n(C)c3)=O)C2)=O)CCOC(C)(C)C1 c1(C(N2C3CCC(NC(CC(C)(C)O)=O)(C3)C2)=O)sc2sccc2c1Cl N1(C(C(C)(C)C2CC2)=O)CCCC2(CCN(C(c3cc([N+](=O)[O-])c[nH]3)=O)C2)C1 CCC(C)C(C(=O)NC(CC1CC1)C=O)N(C)C(C1CC(=O)CC(=O)N1)=O C(=O)(C(C)CCCOC(=O)C(c1ccc(C)cc1)=O)N(CC=C)CC=C N1(C(c2c(C)snc2)=O)CCOCC1CCNC(=O)CCC1CC1 c1(OC)cccc2[nH]c(C(=O)NC3CC3)cc12.c1(C=O)c[nH]cc1C(F)(F)F Cc1nc(C2CCC2)oc1C(N1CC2CC2(CNC(=O)C=CS(C)=O)C1)=O C(=O)(CC1=CC(=O)OC(C)(C)O1)Nc1onc(-c2ccc(C)c(F)c2)n1 c1(C(=O)OC(C(=O)NCCC)(C)C)cccc(Oc2cc(F)cc(F)c2)c1C O=C1CC(CC(=O)NC2CCC2NC(c2ccn3ncnc3c2)=O)=NN1 C1(CCCC)C(=O)NCCN1C(CC1CCC(C)(C)O1)C(=O)NCCOCC c1(N2C(C)CC(NC(COCc3onc(C)n3)=O)C2)cc(C(N)=O)nc(Cl)n1 c1(OC(C)C)ccc(C(=O)NCC2CCN(C(C3CC3(C)C)=O)C2)cc1N c1(C(CNC(=O)Cc2cccc(Cl)c2)NC(C2CCCC2O)=O)ccccc1Cl N1(C(C(COC)(C)C)=O)C2CCC(C2)C1C(=O)NC(C)Cc1nccn1C c1(C(N2CC3C(C=O)C3C2)=O)cc(F)c(C)c(F)c1.c1(OC)cc(Cl)ncc1.N Cc1c(NC(=O)NCC2(c3ccc(Cl)cc3)CCC2)oc2ccccc12 n1(CCOC(c2c(OC)oc(C)n2)=O)cccc(C)c1=O O=C(C1CCCc2nn[nH]c21)NCC1CCN1C(C1CCS(=O)(=O)N1)=O C1(CNC(CC=CC=C)=O)(NC(=O)Cc2ccc(S)cc2)CCCCC1C C1(NC(C(CCC)NC(N)=O)=O)CCN(C(c2snnc2CC)=O)CC1C c1(C(C(=O)OC)(C)C)cccc(NC(=O)C(C2CCCOC2)OC)c1 S(=O)(=O)(c1ccc(N)c(Br)c1)N1CCC(C)(N(C)CC)C1.C1CCCC12CC2.C Cc1cc(N(C)CC2CCCN2S(C)(=O)=O)nc(C)n1 CCC(C(=O)N1CCOCC1CNC(=O)C1=CCCCCC1)C(F)(F)F CCCC(C)(CC)C(=O)N1CC2CC1CC2CNC(c1c(C)noc1CC)=O C12(CNc3scc(COC)c3)CCCC1N(C(=O)OC(C)(C)C)CCC2 c1(C(=O)NCc2c(C)nccn2)cccc2[nH]nc(-c3cccc(C(N)=O)c3)c12 C1(C(N(C)CC2CN(C(c3cnoc3-c3ccccc3)=O)C2)=O)CCCCC1O c1(C2C(C(=O)NCC(C)(C)NC(C3CCCO3)=O)C2)cccc(Br)c1 C(=O)(C1=CCC(C(F)(F)F)OC1)N.c1(OC)cccc(CC(=O)NC(C)C)c1 c1(CC(=O)N)cccc(C(F)F)c1.C1(O)CCN(C(C23CCC(C2)C3)=O)C1.C CCCC(C(=O)N1CC2CC(NC(=O)CCCCCOC)C2C1)C(C)C C(CC)(C(=O)NCc1csc(C(=O)NCC(C)(C2CC2)OC)c1)=CC CCC(C)C(C#N)c1nc(C(=O)NCCC(C)(C)NC(=O)Cn2nccn2)cs1 c1(COC(C2(CC(C)C)CC(=O)C2)=O)ccc(F)c(C#N)c1 CC1CCN(C(c2csc(F)c2)=O)C1CNC(C1CCC(N(C)C)CC1)=O C(=O)(CC(C)C(C)(C)NC(C1CCCN(C)C1)=O)N(CC(CCC)O)C N1(Cc2cnc(OC)nc2)CCC(F)(F)C(NC(c2nc(Cl)sc2Cl)=O)C1 n1(CC=O)cc(F)ccc1=O.CCCCNC(=O)C.n1(CC=O)cncn1.N Cc1oc(C2CC2)cc1C(N1CCCCC1C1(NC(c2c[nH]cc2Br)=O)CC1)=O c1(OC)c(C(N2CCCC2Cn2cc(CCO)nn2)=O)ccc(I)c1F CC1(C)CC(C=O)C(C)(C)O1.C12CC1CN(C(=O)C(C)C)C2.CC(F)(F)F.N C=CC(C)(CC)C(=O)N1CC(CNC(c2ccc(C(N)=O)[nH]2)=O)(OC)C1 C(C(C)(CCO)NC(C1CN(C(=O)C(c2ccn(C)c2)C)CC1F)=O)OC CCCC(CC)CCC(=O)NC(CCNC(c1ccc(=O)n(C)c1)=O)C(C)C c1(C(N(C2CCCN(C)C2)C(CC)CC)=O)ccc2snnc2c1 c1cc(C=O)ccc1F.c1(NC(C(C)OCC=C)=O)nc(C)c(C(=O)N)s1 C1(CC(=O)N)COCCN1C(c1cnc(C)cn1)=O.c1(COC)ncc(C)s1 N1(C(c2csc(C)c2C)=O)CCC(C(=O)NC(c2ncccn2)C)C12CCC2 n1(C2CC(NC(CN(C)C=O)=O)C2)cc(C2CCC=CO2)nn1.C(C)(C)C.O C12(c3ccc(C(C)=O)cc3)C3C4C1C1C2C3C41CNC(=O)C(F)(F)Br c1(OC(C)C)ccc(C(=O)Nc2ccsc2C(=O)Nc2cn(C)cn2)cc1F N1(C(c2sc(Br)nc2Cl)C(=O)NCCCF)CCCC2(CC=CCO2)CC1 Cc1c(C(=O)NC2(CCO)CN(C(=O)COCc3cccnc3)C2)ccn1C C(=O)(C1CSc2ccccc21)NCC(C(C)(C)C)NC(c1cccc(=S)n1O)=O C1(NCCC(C)N2CCC2)COC2(COC2)C1 Cc1cc(C(C)C)ccc1C(=O)NCCCO.c1(CCC(=O)N)cc(C)n(C)n1 C1(C(N(CCNC(CC(=C)C)=O)CCO)=O)CCc2cc(F)ccc2O1.CCO C(=O)(C(C)(C)C(C)(C)O)NC(CC)CC(=O)N(C1CCN(C)C1)C c1(OC)cc(CN2CCCC2(C)C(=O)NC(c2ccc(Br)cn2)C)ccc1C#N Cc1cnc(N2CCC(NC(C3(Br)CC3)=O)C(CO)CC2)nc1S(C)(=O)=O CC(C)(C(=O)NC1CC(C)C1)c1ccccc1.c1(C=O)cc(C(F)(F)F)no1 C1(C=O)C2CC3C(C2)C13.c1(CC=O)cccnc1C.C1(C=O)CC1.CC.N c1(N(C)Cc2scc(C)n2)nc(N(C)CC2CCOC2)c2c(n1)c(C)nn2C c1(C(=O)NC2C(C(=O)NCc3ccc(C)cc3F)CC2)cccn2ccnc12 c1(CC)cc(=NC(=O)C2CSCCN2C(c2nc(O)nc(O)c2F)=O)[nH][nH]1 C1(COC)(CNC(=O)CC(C)N(C)C)CCN(C(c2cc(C)ncn2)=O)C1 c1(C(=O)NCCOC2CN(C(C(F)OC)=O)C2)ccc(O)c(C(C)=O)c1 C1(CN(C)C)CC(N=c2[nH]c(N3CCC(Nc4ccccc4)C3)nc(=N)[nH]2)C1 N(C(=NCCN1CCCC(C)C1)NCc1ccc(C)cc1)C(C=C)C CCC1c2ccc(OC)c(OC)c2CCN1Cc1cccc(C(F)C(F)(F)F)n1 c1(CC(=O)OC)cn[nH]c(=NC(C)c2ccc(O)c(C(C)(C)C)c2)c1 c1(C(=O)NC)cccc(C(C(=O)NC2CCOC2)N(C)Cc2cn[nH]c2)c1 n1(CC)ccnc1C(c1nnnn1CC(F)F)NCC1(CC(C)C)CCCC1 Cc1cc(C(=O)NCC23CC(NC(c4cnncc4O)=O)(C2)C3)cc(O)c1 C(=O)(C(F)(F)C1=CCOCC1)N.CCC(C)(CC)C(=O)NCc1ncccc1C CC(C)(C)CC(O)C(=O)N1C2CCC1CC(NC(c1nccc3ccsc13)=O)C2 C1(C(N(CC)C)=O)CCN(C)C(=O)C1.CC(CC1CC1)C(=O)NCCCO C=C1CC2CC1CN2C(=O)CC=CCNC(C1CNC(=O)CC1C)=O n1(CC)nc(C)c(CC(=O)NCCC2CCCC2)c1C.C1(C)(C(=O)N)COC1 C(=O)(C1=CNS(=O)(=O)N=C1C)N.C#Cc1ccc(C(N2CCC(O)(C)C2)=O)o1 C(C1CCOCC1)=CC(=O)NC12CC1CN(C(=O)C(N1CCCC1)C1CC1)C2 C#CCC(C(=O)NC1(CF)CC1)NC(=O)Cn1ccnc1 c1(CC(N2CC3(OCC(NC(c4cnc[nH]4)=O)C3)C2)=O)coc2cc(F)ccc12 Cc1ccc(Cl)c(N)c1C(N1CCC(NC(c2cc(C(N)=O)no2)=O)C1)=O Cc1ccc(C=CC(N2CCC(CN(C(=O)CCn3cccnc3=O)C)C2)=O)o1 C1(C2CCCCO2)(C(N2CCCC2CF)=O)CCCO1 C1(C(=O)OC)CC(CN)CN(C(=O)C(=O)N)C1.C1CC(=O)N(C2CCCCC2)C1 Cc1cc(NC(C23CC(F)(C2)C3)=O)ccc1NC(C1CCCOC1C)=O Cc1[nH]nc(C(=O)NC(Cn2cncn2)C(=O)N2CCC(n3cnnn3)C2)c1Cl C=C(C)C(CC(=O)N1CCCC(C)(NC(=O)Cc2ccnc(C)c2)C1)OCC C1CC2(C)CCCN2S1(=O)=O.CC1(C)OC(c2cccc(C(=O)OC)c2)OC1(C)C N1(c2n(CCC#C)c(-c3cccnc3)nn2)CCN2C(=O)N(C)CC2C1 CC(F)(F)CCC(=O)N(C1CC1)CC1CCCN1C(C1CC2CCC2C1)=O N1(C(C2(CC=C)CCCN2C(=O)CC(=O)N(C)C)=O)CC(C)OCC(C)(C)C1 c1(C(=O)N)c(C)cc(C)nc1O.C1(C)(CC)C=C(C(=O)NC(C)C(C)C)C1 N1(C(CCc2cncc(C)c2)=O)CCN(C(C2CC(C)(C)CO2)=O)C(CCO)C1 c1(CC)c(C(=O)NC2(CNC(=O)CC(C)C3CCCO3)CCOCC2)cnn1C C(CC(O)CO)N(C(=O)C(C1(C)CC1)NC(=O)C(F)C1CCCC1)C C1(CNC(C(c2ccccc2Cl)C)=O)CN(C(=O)Cc2nccs2)CCC1(F)F Cc1nn(C)c(Br)c1C(c1nnnn1CC(F)F)NCC(C)Cc1cccs1 C1(CC(=O)NCCNC(CC2(C=C)CC2)=O)CC2(CC2)CO1.C1CC1.C C1(NC(C2CCCN(CC(F)F)C2)=O)(CF)CCN(C(c2cc[n+]([O-])cc2)=O)C1 c1(C(=O)NC23CCCC(NC(CCC)=O)(C2)C3)cc(S(=O)(=O)N(C)C)c[nH]1 C(=O)(CC(F)(F)C(F)F)N1CC2C(CC(=O)NCC3(C)CCN(C)C3)(CC2)C1 Cc1ncc(C(N2CC=CC(NC(=O)COc3cccnc3)C2)=O)cc1C#N c1(OC)cc(C(N2CCC(C3(NC(c4ncoc4C)=O)CC3)C2)=O)cc(N)c1O C1(C(=O)NC2(CC3CCC3)CC2)CC12CCN(C(c1ccc(F)s1)=O)C2 CC1(C)CC(C)(C(=O)NCc2ncco2)CN1C(=O)C=Cc1cnccn1 CCCCC(CNC(=O)CCc1ncc(-c2ccccc2F)o1)NC(=O)CSC N1(C(c2[nH]cc(CC)c2)=O)CCN(C(c2cccn3ccnc23)=O)C2CCCC12 C1(C2(O)CCOCC2)(CNC(C2CC(C)OC2C)=O)CCC1 CC1(C)CCN(C(c2cccc(OCC(N)=O)c2)=O)CC1.C1(C=O)CC(O)C1.N N1(C(c2c(C)nsc2Cl)=O)CCC2(CC1)CCN(C(=O)C(F)C1CCOC1)C2 C(C)(C(C(C)C)NC(=O)CCO)NC(C1(CC(C)C)CC1)=O.C1COC1 c1(C(N2CCCC(C)(NC(C(C)NS(C)(=O)=O)=O)C2)=O)cc2cccnc2[nH]1 N1(C(C2CCN(C(C)=O)CC2)=O)CCC2(CC1)CCN(C(=O)C(F)C(C)(C)O)C2 c1(CN2CC(O)(C(=O)NCc3cnc(C)s3)C2)ccc(SC(F)(F)F)cc1 N1(C(c2ccc(C(N)=O)s2)=O)CCCC2(NC(c3cnc(Cl)cn3)=O)CCCC12 CCC(C)CC(CO)NC(C1CCC(NC(C2(C#N)CC(F)(F)C2)=O)C1)=O CC1CCCCN1C(=O)C(C1CCCO1)C1CC1.C12(C=O)CC(C)(C1)OC2C.N Cc1ccnc(C(=O)NC2CCC(CNC(c3cccc(CC#N)c3)=O)C2)c1 CCC(C)C(=O)N(C)CC1(O)CN(C(C2(n3ccc(C4CC4)n3)CC2)=O)C1 CP(C)(=O)c1ccc(C(=O)NC2(C)CCC2)s1.C1(CC(=O)N)CC=CCC1 c1(C(=O)N)nccc(Cl)c1F.CC(CCNC(=O)Cc1cc(C2CC2)no1)CC C(=O)(C1=CCN(C(C2CCOCC2)=O)CC1)NCC(C)C1CCC1 c1(C(N2CCC(N(C(c3ccc(OC)cc3)=O)C)C2)=O)cc(N)cc(O)c1F C(=O)(C(F)CCC(C)C)NC(C(=O)NCc1c(C)cc(C)s1)Cc1ccco1 N1(C(CCN(C(=O)CCc2csnn2)CC#C)=O)CCc2nccnc2C1 C1(OC)CCCCCC1N=c1ccnc(NC2CC(C(C)C)C2)[nH]1 N1(C(CC(CNC(C(n2c(C)ccn2)C)=O)(C)C)=O)CC2CCCC(O)C2C1 C(CC(C)C)(C(=O)NC1CCC(O)C1)OC.c1(C=O)n[nH]c(C(C)(C)C)n1.C N1(C(c2nccc(C)c2)=O)CCCCC(NC(=O)C2=C(Cl)CCC2)CC1 c1(C(N2CCC(CC)C2)C(=O)N)ccnn1CC(F)F.C(=O)(CC)OCC Cc1[nH]nc2c1CC(C(N1CCCCC1CN=c1[nH]nc(C3CC3)o1)=O)CC2 C#CC1(C(=O)NCCn2ccnc2C)CCN(C(=O)CC(C(=C)C)OCC)CC1 c1(C(=O)NC2C3CN(C(c4c(C)cc(O)cc4)=O)CC32)cc2ccc(O)nc2s1 c1(C(N2CCN(C(c3c(C)ncs3)=O)CC2CC#N)=O)cccc(S(N)(=O)=O)c1 N(C(=NCCCc1cnn(C)n1)NCC(c1ccccc1)O)CC(C)C c1(CC)nc(C(=O)NCC(CO)NC(=O)CC(C)N(C)C)cs1 c1(-c2nc(C)nn2-c2ccc(F)nc2)sc2cccc(F)c2c1C C1(CCNC(CC=C)=O)CCCN(C(=O)CCCc2nc(C)no2)CC1 C(=O)(C1CSc2ccccc21)NCC1N(C)CCN(C(C(C)(C)OCC)=O)C1 C(=O)(C#CC1CCCCO1)N1C(CNC(C2CCN(C(CC)=O)C2)=O)C(C)CC1 CCCCC(O)C(=O)NC1(c2ccccc2)CCN(C(C2CCC2)=O)C1 C1(COC)CN(C(C2CCC(C)O2)=O)CCN1C(c1cc(C)c(C)s1)=O c1(NC(C(N2CCCC(C(C)(C)C)C2)c2ccoc2)=O)ccc(Cl)cc1F C1(NC(c2ccc[nH]2)=O)CN(C(C2CCCSC2)=O)CCC1CO N1(C(CCc2cc(C)on2)=O)CCC(O)CC1C(=O)NOC1CCN(C)C1 c1(C(N2CCC(n3cc(CNC(C(C=C)O)=O)nn3)C2)=O)ccc2ccoc2c1 c1(C=O)cc2cccc(Cl)c2o1.c1(OC)ccc(C(=O)NCC2CC2)c(F)n1 CON1CC(C(=O)NCC=C2CCN(C(C3CCCCO3)=O)CC2)CC1=O c1(C(=O)NC(C=CC(=O)NC2CN(C(C)=O)C2)C)ccn2cncc2c1 CC(C)CC(C)CC(=O)NCc1cccc(C(=O)NCCc2cscn2)n1 c1(OC)cccc(C)c1C(=O)NCC(C)(CNC(c1c[nH]c(=N)o1)=O)O CN1CC(NC(=O)C(C(C)(C)C)NC(=O)CCC2CCCOC2)C(F)(F)C1 C(C(C(=O)N1CC(CNC(=O)C(C)(C)SC)(OC)C1)OC)OC CN=C(NCC(=O)Nc1nc(C(F)(F)F)cs1)N1CCOC(CF)C1 N#Cc1ccc(CCC(=O)NC2CCC(CNC(C3C4COCC34)=O)C2)c(F)c1 Cc1ccc2cccc(S(=O)(=O)NC3COC(C4CNC4)C3)c2n1 CCS(=O)(=O)NCCC(=O)NCC=CCNC(c1ccsn1)=O N1(C(C(N2CCCCC2=O)C)=O)CCC(NC(C2(O)CCCCCC2)=O)C(O)C1 C1(F)(CN)COCCN(C(c2coc(Cn3cccn3)n2)=O)C1 C1(C(=O)Nc2ccc(OC(C)(C)C(F)(F)F)cc2)CCN(C(=O)CO)CC1O N1(C(C(CCCC)CC)=O)CCC2CN(C(=O)Cc3cccc(F)c3F)CC2C1 C1(C(=O)NC2C(OC)CN(C(c3ccc[nH]3)=O)C2)CCOCC1(C)C N1(C(c2n(COC)ncc2)=O)CCOCCC1C(N1CC(CO)(CF)C1)=O c1(C(N2C(CNC(=O)CC3CC4(CCC4)C3)C=CC2)=O)cc2ccoc2cc1F C(=O)(C1=NNC(=O)CC1)N(C1CCC(NC(c2cc(C(C)=O)cn2C)=O)C1)C N1(C(c2scc(OC)c2)=O)CCC(CNC(=O)CO)C(F)(F)C1.C(C)C C1(CC)(NC(C2CCCC(F)C2)=O)CCN(C(=O)C(F)(F)COC)CC1 C1(NC(=O)C2=CCCCC2)CN(c2ncnc(-c3ccccc3)n2)CC2(CC2)C1 C(CCCCCNC(C1COCC1NC(c1ccc(C#N)[nH]1)=O)=O)N(C)C CC1=NOC2(CCN(C(=O)C(N3CCSC(c4ccccc4)C3)=O)CC2)C1 c1(CC)c(N2CCN(CCN(C)C(C3COCCO3)=O)CC2)ncnc1Cl c1(C(=O)NC2C3OCC(NC(c4cocn4)=O)(C3)C2)cccc2nc(C)[nH]c12 C(=O)(C(N)C(C)C(C)C)NC(C(=O)OCC)CCO N#Cc1ccc(C(=O)NC2CC2C)o1.c1(C(=O)N)cn[nH]c1Cl.c1ccccc1 c1(C=O)ccn2cc(C(F)(F)F)nc2c1.C(C)(C)C.C1CC1C=O.COC C=CCC(C(=O)N1CCCC(CC(=O)NCC2CCN(C3CC3)C2)CC1)C(C)C c1(C(=O)NCCC(=C)CNC(c2cc(Cl)c[nH]2)=O)ccc2cnccc2n1 N1(C(=O)OC(C)(C)C)CC2CCC1CN2C(=O)OC12CCC(C1)C(=O)N2 CCCCCCCCCC(=O)N1CC2(CCCCN2C(=O)C(F)OC)C1 Cc1nc2ncc(C(=O)N(C(C)CNC(=O)CC3COCCO3)C)cc2o1 c1(C(N2CC(N(C(=O)C)C)C2)=O)cccc(-c2nn[nH]n2)c1.C(=O)C(F)(F)F Cc1c(C(N2CCC(C(c3ccccc3)=O)C2)=O)sc2ccc(F)cc12 c1(C(=O)NC2C(NC(c3ccoc3C3CC3)=O)C2)cccc(=S)n1O CCC(F)(F)C(=O)NCC(C)(C1CC1)NC(c1cc(CO)[nH]n1)=O c1(OCC(=O)NCCCN(C(=O)CC(Cl)Cl)C2CC2)cccc(O)c1 c1(NC(C)Cc2cn[nH]c2)cncc(CN(C)C)c1 CS(=O)CCC(=O)NCCC1COCCN1C(c1ccc(Br)s1)=O c1(C(=O)NC(c2occ(C(=O)NC(CC)C)n2)C)ccccc1C#N CN1CCCCCC1c1nc(-c2ccncc2)nn1-c1ccc(F)cc1 c1(NC(c2c(C)scc2)=O)cccc2c1CC(C)(C)C2 C(=O)(C(F)C(=O)N(CCCC(=O)NCC(C1CCCC1)OC)C)OCC c1(CCC(=O)NC(C2(O)CN(C(C(CC)F)=O)C2)C)ccc(C)c(Cl)c1 Cc1cccc(OCc2nc(-c3cc(O)nnc3O)no2)c1F C1(CNC(=O)C2=CCCCO2)(NC(c2cc(O)nc(O)n2)=O)CC2CCC1CC2 C1(CC(=O)NC(c2cn(C)nc2)CO)COCCN1C(c1ccc(N)cn1)=O C(c1sc(Cl)nc1Cl)=CC(N1CC(N(C(C(C)CO)=O)C)C(O)C1)=O C(c1cncc(O)c1)=CC(=O)N(C1CCCC1)Cc1ccccc1Cl N=c1[nH]c(=NCC2OCC3CCC2C3)[nH]c(=NC2CC(CC(N)=O)OC2=S)[nH]1 c1(C(N2CCCC(N(C(C(CCC)OCC)=O)C)C2)=O)ccc2c(cnn2C)c1 Cn1ncc2c(N3CCN(C(c4cn(C5CC5)cn4)=O)CC3CCO)ncnc12 CN=c1[nH]c(=NCc2ccnn2C2CCC2)[nH]c(=NC2COCC2C2CC2)[nH]1 c1(OC)cccc(CCC(=O)NCC(C)NC(c2cnn(C)n2)=O)c1OC N1(C(C(C)N)=O)CCCC(C)(C)C1.C1(C=O)CC2C(C1)C2(C)C.[SH](C)(=O)=O CC1(C)CCc2nc(NC(=O)NC(c3cccs3)(C)C)sc2C1 CON=Cc1ccc(C(N2CCCC3(NC(=O)CC4(O)CCC4)CC3C2)=O)cc1 c1(C(C(=O)NC2CC(C(C)NC(=O)Cc3ccsn3)C2)C)cccnc1 C(=O)(CC(C)C(F)(F)F)NCc1c(C(=O)OC)cnn1C C(C(C(C)(C)C)NC(c1ccc(C(F)F)s1)=O)NC(C(n1c(C)ncc1)C)=O C1(C(CNC(C2CC(CNC(=O)CN3CCCC3)C2)=O)O)CCCCC1 C(=O)(C1=CCCC(C)(C)C1)N1CC2C(CCC2)C1.c1(CC)cc(C(=O)NC)n[nH]1 C1(NC(c2c(CC(C)C)nc(C)s2)=O)CN(C(=O)CCc2ncc[nH]2)CCC1O c1(C(=O)NCCOCCNC(C2(CCC)CCCC2)=O)cccc(OC)c1 C1(NC(c2c(CNC(COCCC=C)=O)cco2)=O)CCN(C)C1C c1(C(=O)NC2C(C)N(C(c3ccn(C(F)F)n3)=O)CC2)cc2ccc(Cl)nc2s1 C#CC1CN(C(C2C(O)CCN2C(c2ccsn2)=O)=O)CCO1 C1(C(N2CC(CCCCNC(=O)CSC(F)(F)F)C2)=O)CCCC2CCCN12 O=C(C1=NOC2(CCC2)C1)NC1(CCNC(C23CC=CCN2CCC3)=O)CCC1 n1(CC)cc([N+](=O)[O-])c(C(=O)NCC2COCCN2C(=O)C(C)OC)n1 S(=O)(=O)(c1cccc(N2CCCC(C(N)=O)C2)n1)N1CCC(C(CC)CC)C1 C1(NC(c2n[nH]cc2C2CCC2)=O)CN(C(=O)C2=CCCC2)Cc2ccnn2C1 C1CN(C(c2cc(Cl)cc(Cl)c2O)=O)CCC1(C)C.C1(OCC)CC(C(=O)N)C1 Cc1cnc(C(=O)N(C)CC2CCCN2C(C2(C)CCCCCC2)=O)c(C)c1 C(CC)C(C)C.c1(C=O)nc(O)c(C)s1.c1(COCC)nc(C=O)cs1.N C1(CCC)CN(C(c2cccc(CSC)c2)=O)CCN1C(=O)CSCC CC(C)C(F)C(=O)NC1CN(C(c2cnn(-c3ccccc3)n2)=O)CC1O c1(OC)ccc(F)c(C(N2CC(F)CC2CN(C(=O)CC(C)(C)C)C)=O)c1 c1(C(N2CC(NC(CCCC(C)=O)=O)C(C3CC3)C2)=O)cc2c(Cl)ccnc2s1 c1(C(N2CC(C(=O)Nc3n(C(C)C)ncc3)OCC2)=O)ccc(Br)nc1Br c1(SC)ncc(C#N)c(N2CCCN(Cc3nccc(Oc4ccccc4)n3)CC2)n1 N1(C(c2ccc(C(C)(C)C)[nH]2)=O)CC(NC(c2nc(Cl)ccc2N)=O)CC1(C)C C#CCCCCC(=O)NC1CCCC1(C)CNC(C12CC(F)(C1)C2)=O S(=O)(=O)(c1cc(C(=O)NC(C2CCCCC2)CO)cc(C)c1C)NC c1(NC(C(C)CN(C(=O)CCc2ccccn2)C)=O)ccc(F)cc1F C1(C(=O)NCC2(OC)CN(C(c3ccsn3)=O)C2)CCC(=O)NC1 CCCC(C(F)(F)F)NC(C1(CO)CCN(C(c2ccoc2Cl)=O)C1)=O C1(COC)CCCN1C(=O)C.C1(C)(CC=O)CCCCC1.CCN(C)C.C C(=O)(C(CC)(CC)CO)CC(CCC=C)N.C1(C(=O)N2CCCO2)CC12CCC2 N1(C(C(CC)C#N)=O)C2CCC1CN(C(=O)C(C)C1CCCC1)C2 C1(C(=O)NC2CCN(C(CCC(=O)N(C)C)=O)C2)CC12CCCCC2 c1(C(=O)NC2C(NC(CC3ON=C(C)C3)=O)C2)cc(Br)n2ccccc12 Cc1c(C(N2CCCC(N(C(=O)CC3CCCSC3)C)C2)=O)nnn1C c1(C(=O)NCC2CC(NC(c3c(C)scn3)=O)C2(C)C)cc2c(ccn2C)[nH]1 c1(CC)cnc(NC2CCCC(C(=O)N)C2)nc1.n1(CCC2CC2)cc(Br)cn1 C1(CNC(c2cccs2)=O)(NC(c2c(Cl)nsc2Cl)=O)CC2CCC1CC2 C=C1CC2CC1CN2C(=O)C(=O)NCc1cccc(SC)c1 C1(CNC(CC=C)=O)CCC2(CN(C(=O)CCCOC(C)=O)C2)O1 c1nc(Cl)ncc1C(N)=O.c1(SC)ccc(C(=O)NC2CCC(C)CC2)cc1.N C=C1CN2C(=O)CCC2(C(N2CCC(C)C2)=O)C1.c1(C(=O)N)cc(N)nc(Cl)c1 C1(NC(C2(C(=O)OC)CC2)=O)C2CC1CN(C(=O)CC1OCCC1(C)C)C2 Cc1cc(C(N2CCN(C(C3CNC(=O)C3)=O)CC2)=O)n2nccc2n1 c1(C(N(CC(C)(C)NC(C2(C(CC)(F)F)CC2)=O)C)=O)cc(OC)nn1C N(C(=NCCCF)N1CCC(CS(C)(=O)=O)C1)Cc1c(C)nc(C)c(C)n1 c1(CN2CCC(O)(C(=O)NCC3(C(=O)OC)CCC3)C2)cnc(Cl)cc1Br CC1CN(C(=O)CC(C)(C)C2CC2)CC(C)N(C(c2cnn(C3CC3)c2Cl)=O)C1 c1(C(=O)NC2CN(C(C3C(OCCC)CCCC3)=O)C2)ccc(CC)c(N)c1 N1(C(C2CCCN2C(=O)CCNC(=O)CCCc2cccnc2)=O)CCOCC1 C12(C=O)C3C4C1C1C2C3C41.CCC(C)(C)C.CNS(=O)(=O)NCC(=O)N N1(C(C2C(C(C)C)C2)=O)CC2(CCC2)C1.C1(CC=O)CN2CCC1CC2.CC c1(C(N(C2CN(C(=O)C)CC2F)C)=O)cc2nnn(C)c2s1.C(=O)(C1CC1)N c1(C(N(C2(C(=O)NCC)CCC2)C)=O)cc(F)cnc1O.C1CC[Si](C)(C)C1 C(=O)(C1CC=Cc2ccccc21)NC(CCCNC(c1c(N)cn(C)n1)=O)(C)C C1(C(=O)OC)CCCC(C(=O)NCC(C)C2CC2)C1.c1(C=O)ccncc1F.N c1(NCC2(C(N)=O)CCCC2)ncc(S(=O)(=O)NC2CC(CO)C2)cc1Cl C(C1OCc2ccccc21)NC(=NCCF)NCC(Cl)C(F)(F)F C12(C(N3CCC(O)(CN(C(c4ccc(SC)o4)=O)C)C3)=O)CCCN1CCC2 N1(C(CC(CC)OC)=O)CCCCC(NC(c2ccc(CC(C)C)s2)=O)C1 C(=O)(CCCCC(C)(C)C)NCC(C)NC(C1CNC(=O)CC1(C)C)=O c1(CNC(C(CO)NC(C=C(CC)CC)=O)=O)ccc(F)c(C)c1 S(=O)(=O)(c1ccc(NC(CCO)C2CC2)c(Br)c1)NC1CC(=O)NC1=O C1CC2(CC2)CN1C(C1CC(O)C1)=O.n1(C(C)(C)C)nnc(CC(=O)N)n1.C C(=O)(C(CNC(C1CCCC(O)C1)=O)CC(C)C)NC(CC)(C)C(N)=O n1(C(CC)C)ccc(=NC(=O)C2COC(C)C2)[nH]1.C1(CC(=O)N)CC(C)(C)CO1 N1(C(c2ccn(C(C)C)n2)=O)CC2(CCC2)CCC1C.C1(C=O)CC1C(F)F C1(C(=O)NCC(N2CCOCC2)=O)CN(C(=O)Cc2cncnc2)CC12CC2 C1CN(C(c2cc(N)c(F)cn2)=O)CC(C)(C)C1.c1(CC)nc(C)c(C=O)s1.N CC1=NNC(=O)C1CC(=O)NC(C)(C)CC(=O)NC1CC1c1ccco1 N1(C(C=C(CNC(C(COC(C)=O)C)=O)C)=O)CCCC[Si](C)(C)C1 N1(CCC(=O)NC2CCC2C(=O)Nc2cccnc2)CCOC1=O c1(CCC=O)nnc(S)nc1O.O=NN1CCCC1C(=O)NC12CC(C)(C1)C2 CC1(C)C(C(=O)Nc2c[nH]nc2-c2ccccc2)C1N C(=O)(CC(O)C(C)C)N.c1(C(=O)OC)ccc(C(N2CC3CC3(C)C2)=O)cc1 Cc1ccc(C(=O)NCC2CC3CC3N2C(=O)CSC(C)C)c(O)n1 C1(C(CNC(C(C)CC2CCCC2)=O)(C)C)CCN(C(c2cnn[nH]2)=O)CC1 N1(C(C2N(C(CCC)=O)CCC2)=O)CC2(CCC(F)(F)CC2)C1C(=O)OC N1(C(C2C(C)(C)CO2)=O)CCC2CCN(C(=O)CC3CCC4(CCC4)O3)CC2C1 C1(C(=O)NC(C=O)C2(C)CC2)CCCN(C(=O)CC2(C)CCC2)C1.C1CC1 C(CNC(=O)CCc1cccc(O)c1)(C(C)(C)C)NC(CNC(C)=O)=O C1(NC(C2C(CC)CCCC2)=O)CCN(C(C2CCS(=O)(=O)N2)=O)C1(C)C c1(C=O)sc2cc(F)ccc2c1C.c1(OC)ccnc(C(=O)NC2CC2C)c1.N C(=O)(C(C)(CSC)NC(c1ccncn1)=O)NC1(CC(=O)OC)CC1 CCC(C(=O)NCC1CCN(C(=O)C(n2nnnc2C(C)(C)C)C)CC1)C(C)C Cc1nc2cc(-c3ccc(CNCc4ccc(C(=O)O)[nH]4)cn3)ccc2s1 C1(C(=O)NCC2CCCN2C(=O)Cn2ncc(Br)n2)(OC)CCSCC1 C1(CC(N2C3CCC2CC3)=O)CC2(CCC2)CCO1.C(C)(C=O)OCC#C.N Cc1nnc(CN(C(=O)CCO)C)s1.C1(CCC(N2CCC2)=O)CCC(=O)C1 C1(C(N2C(C(N3CC(CC)OCC3)=O)CC(O)C2)=O)CC(=O)NC(=O)C1 N1(C(CC(C)NC(C2(CCCC)CC2)=O)=O)CCNC(=O)C1C c1(NC(C2(C)CCN2C(=O)CNC(=S)NC2CCCC2)=O)ccc(Cl)c(F)c1 N1(C(=O)NC2CCC(NS(C)(=O)=O)CC2)CC(O)CC12CCOCC2 C1(NC(C(C)c2cc[nH]n2)=O)CC2C1CCN2C(=O)C=CC1CCCCC1 c1(NC(c2c(CNC(c3cc(CC)ncc3)=O)noc2)=O)cncc(C#N)c1 C1(C)(C(=O)NCC(CC)NC(c2nn(C)c(C)c2Cl)=O)CCCNS1(=O)=O Cc1[nH]nc(C(N2CC(NC(=O)Cc3cccc(Cl)c3)C(C)C2)=O)c1Br C1(CNC(c2[nH]cc(CC)c2)=O)CN(C(=O)CCCC)C(C)(C)C1.C(N)=O C(C(CC(C)C)C(=O)Nc1cccc(CC)c1F)NC(C(C)NC(CC)=O)=O Cc1oc(C)c(C(=O)N)c1C.CC(C)CC(C)C.C(=O)CC1CC1C(F)(F)F N1(C(c2ccc(CCC)s2)C(=O)NC(C)CC)CCOCC2(CCC2)C1 c1(C(=O)NCCCC(C)NC(Cc2cc(OC)ncc2)=O)cnc2cc[nH]c2c1 N1(C(C(COC)OC)=O)CCN(C(=O)CC23CCCCC2C3(F)F)CC(C)(F)C1 N1(C(C(C)NC(N)=O)=O)CCCCC12CN(C(C1CCC(C(F)(F)F)O1)=O)C2 c1(C(=O)NC2CN(C(CC(C)F)=O)CC23CC3)nccc2c(Br)cccc12 c1(CC)cc[nH]c1C(=O)NCC1CCCC1C(=O)NC(C)(C)C(C)O CC(C)C(CNC(C1(CCCF)CC1)=O)C(=O)NCC1(F)CCN(C)C1 C1(CCC(N2CC(OCC#C)C2)=O)CCN(C(C2(CC#C)CCC2)=O)CC1 CC(C)CS(=O)(=O)CC(=O)N1CCCC1.N1(CC(=O)NC2CC2)CCCC1.C Cc1ccc(CCC(=O)Nc2ccc(C(=O)NCCF)cn2)cc1F N1(C(C2ON=C(CC)C2)=O)CC2CCCC2C1C(=O)NCc1nc(C)c(C)o1 c1(NCC(C2CC2)NC(c2scnc2Cl)=O)nccc(C(F)(F)F)n1 c1(C(=O)NC2C3CN(Cc4ccc(Br)cc4)CC23)c[nH]c2ncccc12 c1(C(C)C)ccoc1C(N1CC(O)(C(F)C(=O)N)C1)=O.c1(C(C)O)cn(C)cn1 C1(C(C)NC(=O)CCn2cccn2)CCN(C(=O)Cc2cnnn2C)C1 C(CC(C)CC)(C(=O)NCc1cnc(C)o1)NC(c1n(CC#C)cnn1)=O C(CC(C(C)C)NC(c1ccc(=N)[nH]n1)=O)N(C(C1CC(SC)C1)=O)C O=C1CCCC(CCCC(=O)N2CC(O)(CNC(c3cnc(Cl)[nH]3)=O)C2)N1 c1(CC)occ(C)c1C(=O)NC1(C2CCCCN2C(=O)C(O)CSC)CC1 c1(N(CCCC=C)C)nc(NC2COCC2Cc2ccncc2)c2ccsc2n1 c1(C(=O)NCC#CCNC(c2ccc(Cl)cn2)=O)cc2c([nH]1)CCOC2 c1(C(=O)NCc2cncnc2)cc2n[nH]cc2cc1-c1cc(F)c(F)c(F)c1F N1(C(C2CCCN(C)C2)=O)CCCC(NC(c2ccc(C3CC3)c(Cl)c2)=O)CC1 C(=O)(C(C)(C)CCF)NCC1(OCC)CN(C(C2CCOC2(C)C)=O)C1 Cn1c(C(F)(F)F)ccc(NC(C2CCCCCC2c2ccccc2)=O)c1=O c1(OC(C)C)cnccc1C(N1CC(CC(C)NC(=O)CC(C)N(C)C)C1)=O C1(C(N2CCC(F)(C(N(CC=C)CCO)=O)C2)=O)CCCCCCC1 c1(CCN2CC(O)(CNC(=O)CCC3CCOCC3)C2)ccccc1F C1(CC)CN(C(=O)CC(C)(C)N(C(=O)C(c2ccnn2C)O)C)CCO1 C1(CN2CC(C)(C(=O)Nc3nc(OC(F)(F)F)cs3)C2)CC12CCCOC2 C1(F)(CNC(C2C(=C)CC2)=O)CCCN(C(c2c(C)nn(CC)c2Cl)=O)C1 c1(CC)conc1C=O.C1(C(N)=O)CN(C(=O)Cn2cc(C3CC3)cn2)C1 C1(C2CCC2)(C(=O)NCCC2(O)CCN(C(c3cc(C)ns3)=O)C2)CC1(F)F CC1(CNC(=O)Cc2cccs2)CN(C(c2sccc2I)=O)C1 C(C)(CCC(=O)NC12CC(C1)N(C(c1csc(C(C)(C)C)n1)=O)C2)SC n1(C2CCN(C(C)C)C2)c(N(C)CC2CCOC2)nnc1C(N)=O c1(C(=O)NC2C3CN(C(C(CC(N)=O)O)=O)C2C3)cc(S(N)(=O)=O)co1 S(=O)(=O)(C1CCC(=O)CC1)N1CCC2(C(C(=O)Nc3c(C#N)c(O)cs3)C2)C1 c1(C(=O)NCCn2cc(Br)cn2)ccc(OC(F)(F)F)cc1 C1(C2CCC2)(NC(=O)NCC2(c3cccc(C)c3)CC2)CCC1 O=C(CC(C(F)F)N1CCOCC1)NCc1nc(-c2ccncc2)no1 C(=O)(C1=CC(O)C(NC(C2(N(C)C)CC2)=O)C1)NCCC(C)N(C)C C(CC(F)F)(C(=O)NCC(O)C(C)(C)O)N(C(=O)Cn1cccn1)C CC1=C(C(=O)N2CCC(O)(CN(C)C(c3ccccc3C)=O)CC2)CCC1 CC(C)CCCCC(=O)NCC1CC(C)CN1C(C1CCCC(C)CC1)=O C1(NC(Cc2nc(C)sc2)=O)CC2CN(C(c3cnc4[nH]cnc4c3)=O)CC2C1 Cc1ncnc(C(=O)NC(CC2CCC2)C(=O)NCC(c2ccco2)O)c1C C1(C)(CC(=O)OCC)CCN(C(=O)C(C)Cc2cnc[nH]2)C1 C1(C(N2CC(F)(C)C2)=O)(COC)CCCCC1.C(=O)CCC1CC(C)C1.N N1(Cc2c(C)n[nH]c2)CCC(=O)N(CCOc2ccncc2)C1=O N1(C(CC=C)=O)CCC2CCCC12C(=O)NCC1OC(=O)NC1(C)C c1(CC)cc(C(=O)NCC(C)NC(C2(CCOC)CC2)=O)nn1C c1(C(N2C(C)C(NC(=O)Cn3cnnc3O)CCC2)=O)cncc2sccc12 N1(C(COCC(=O)NC)=O)CCCN(C(c2nn(C)cc2[N+](=O)[O-])=O)CC1C C1(CC(N)=O)(NC(CCN(CC)CC)=O)CCN(C(=O)C2=CCCC2)CC1 c1(C(N2CC(CNC(C3CCC(=O)NC3)=O)OCC2)=O)cc2ccc(O)cc2o1 C12(C=O)CCN(C(=O)CC3CCCC(=O)C3)CCC1C2.C1(C(C)N(C)C)CC1 C(=O)(C1Cc2ccccc21)NC(C)CCc1ccc(Br)cc1 CC1(C#CC(=O)N2CCCCC(NC(C3(c4ccno4)CCOCC3)=O)C2)CC1 Cn1cc([N+](=O)[O-])cc1C=O.C1(C)CCC1.c1(C=O)ncn(C(C)(C)C)n1.N n1(CCNC(C=CC(=O)N(C)C)=O)ccc(C(=O)N)c1.C1CCC1(F)F c1(C(N2CC(C(C)NC(C(CCCOC)C)=O)C2)=O)cnc2c(c1)NC(=O)CS2 C(=O)(C1=C(Cl)CCC1)N(C1CCC(O)C1)C.C1(N2CC(C(=O)N)C2)CCCCC1 Cc1noc(C)c1C(C)C(=O)NCC(O)CCNC(c1cc[nH]n1)=O c1(C(N2C(CNC(C3N(CC)CCC3)=O)C(C)(C)CC2)=O)cccc2sncc12 c1(OC)ccc(C(=O)N(C2CN(C(c3cncnc3)=O)C2)C)c(Cl)c1.C(C)C.O N1(C(C2C(CC)OCC2)=O)CC(NC(c2cnc(C)s2)=O)C(C)(C)C1 C1(CN(C(CN(C(=O)Cc2ccc(C)s2)CCOC)=O)C)CCOC1C C(CCN=C(NC1CC1)NC1CCCC(F)C1)NC(c1ccccc1)=O C=CCCCCC(=O)N(CC(=O)NCC(=O)OC(C)(C)C)CCOC C1(C(N2CCCC(O)C2)=O)CCc2nnc(O)n2C1.C=C1CC(C)(C(=O)NC)C1 N1(C(c2ncn(C)n2)=O)CCC(CNC(=O)Cc2ccc(OC(F)F)cc2)CC1 C1(C(=O)N)C2CC(F)C(C2)N1C(c1sccc1Cl)=O.c1(OC)ccc(OC)cc1 c1(CCNC(=O)NCc2c(Br)cc(C)s2)c(F)cccc1Cl CC1CCN(C(c2ccc(N)cc2)=O)C1c1cn(Cc2ccccc2)nn1 N1(C(c2c(OC)cc(C)s2)=O)CC2CC(C)C2C1.C1(C2CC2)(C(=O)N)CC1 c1ccc(C#N)cc1.Cc1conc1C(=O)N(C1CC(NC(=O)CO)C1)C.C c1(C(=O)NCC(CNC(=O)CC(C)C)OC)c[nH]c2cc(C#N)ccc12 n1(CC)nc(C)c(CC(N2CC(NC(=O)CC3CCCC3(F)F)C(C)C2)=O)c1C C(=O)(CCCC(=O)N1CCCC(CN(C)C(C2COC(=O)N2)=O)C1)N(C)C Cc1ccc(S(=O)(=O)N2CCc3cc(F)c(Br)cc3C2)c(Cl)c1Cl C(=O)(C1=CCc2ccccc21)NC1C(NC(c2cc(COC)[nH]n2)=O)C1 C(=O)(C(CC1(C#N)CCC1)N(CC(N1CCCC1)C)C)NCCOCC c1(CNC2C(C(=O)NC(c3cccnc3)CO)C2)cc(Cl)c(F)c(Cl)c1 CC1(C)CC(NC(=O)CC2=CCOCC2)CCN(C(c2cccnc2N)=O)C1 C1(CC)CN(C(c2cnsc2)=O)CCN1C(=O)C.C(c1ccccc1)=CC=O.N C1(NC(C(N2CCC(C)CC2)=O)=O)CC(C)CN(C(=O)C(C)n2ccnc2)C1 CC1CN(C(C2CCCC(=O)N2)=O)CCC1.c1(CC(=O)N)cnn(C(C)(C)C)c1 N1(C(CNc2c(C)cccc2)=O)CCn2nc(C(N3CCC3)=O)cc2C1 C1(CNC(c2cc3c(s2)CCSC3)=O)CCC2(CN(C(C3CCOC3)=O)C2)O1 C1(C(=O)NCCC2(C(N3C(C(C)C)CC3)=O)CC2)COC(=O)N1 C1(COC)CCCN(C(=O)C)C1.N1(CC(=O)N)CCCS1(=O)=O.C(C)=O C1(NC(Cc2c(C)noc2)=O)CN(C(=O)CN2CSCCSC2)CC1S(C)(=O)=O C1(NC(CCC(=O)NC)=O)CC2CC1CC2C(=O)N.c1cc(C(C)C)on1.C C1CCN(C(=O)CC23CCC(CC2)CC3)C12CCC2.C(=O)(CCC(=O)NC)NC N1(C(c2[nH]cc(C#N)c2)=O)CC2(C1)SCCC2NC(C1(C2CCCO2)CCC1)=O c1(C(N(C2CCN(C(=O)CCCC(F)F)CC2)CC)=O)sc2ncccc2c1Cl C1(C(N(CCC(C)NC(=O)COC2(C)CCCC2)C)=O)CC2(CCOCC2)C1 c1(C(=O)OC)nc[nH]c(=NCCCN(C)C(c2cc(O)n(C)n2)=O)c1OC C1(NC(C2(C)CCC3CC3C2)=O)CC2CCC1CN(C(=O)COCCCF)C2 C1(COC(c2ncc(Br)cc2C(F)F)=O)CCC2(CCC2)O1 CC1C(C(=O)NC2CCC2NC(=O)Cc2cccnc2)OC2CCCCC12 C1(C(N2C(C)(C(=O)OC)CCC2)=O)CCC2(CC2)N1C(=O)C1=NOC(C)C1 N1(C(c2nc(OC)nc(O)c2)=O)CC2CCCC1C2C.C1(C)(C(=O)N)CCCC1 NC(=O)CCCCC(=O)NC1CCN(C(=O)CCCn2ccnn2)CC1O S(=O)(=O)(c1ccc(F)cc1F)N1CC(C(N2CCC(Br)C2)=O)C(O)CC1 C(=O)(CCCC(=O)N1CC(C)(C)CC1)OCC.C(=O)C(C)(C)C.C(=O)C.C CN1CC=C(C(=O)N2CCCC2C(C)(C)C(N2CCC3(CCC3)C2)=O)C1 C1(C(N2CCC(NC(=O)C=CCOCC(F)(F)F)C2)=O)CCc2cnnn2C1 C1(C(=O)NC2CC(NC(c3c(C)nn(C)c3)=O)C(O)C2)CCCCNC1=O C1(NC(C2(CC=C)CC2)=O)CN(C(=O)CO)CC1C1CC1 N1(C(C(=O)NCC2CC(=C)C2)=O)CCC(Cl)=C(Cl)C1 c1(N(CC(C2CC2)OC)C)cc(N(C)CCN2CCOCC2)nc(C(F)(F)F)n1 C#CCCCCCC(=O)N(CC(C)(C)NC(=O)CC(C)(C(F)F)N(C)C)C N1(C(C2(COC)COC2)=O)CCOC2(CCN(C(C3(CO)CC3)=O)CC2)C1 [SH](=O)(=O)CCC(=O)N1CCC1.C1(C=O)OCCOC1(C)C.CC(=O)NCCN c1(CN2CCN(C(C(=C)C)C)CC2)c(F)cc(C)cc1Br c1(C(=O)NCC2N(C(c3[nH]cc(C)c3)=O)CC=C2)cnn(C(C)C(C)C)c1C C1(F)(CNC(Cc2cn(C)nc2)=O)COCCN(C(=O)CCc2cccs2)C1 C(CCCCC(=O)NC(CNC(=O)C(N1CCOCC1)C)C(C)(C)C)NC(C)=O c1(C(=O)NCC(CC)NC(c2ccnc(OC(F)F)c2)=O)ccc(C#N)cc1O Nc1cc2c(cc1Br)CN(C(=O)NC1CC(C(F)(F)F)C1)C2 N1(C(C2(C)ON=C(C)C2)=O)CC2(CCCC2NC(c2nc(C)c(C)[nH]2)=O)C1 c1(C(=O)NC2CCN(C(Cc3cc(C)sc3)=O)C(C)C2)c(F)ccc(C)c1F Cc1cc(C)c(S(=O)(=O)Nc2cc(C(F)(F)F)cc(C3CC3(F)F)c2)c(F)c1 C1(C)(OC)CCC1(C)C.c1(C(=O)N)cc[nH]n1.N1(CC=CC=O)CCCC1 CC(C)C(C(=O)NOCC1CCCN1C(=O)CC1CCN(C)CC1)NC=O C=CCCCCCCCC(=O)NC(CNC(C1(OC)CCSC1)=O)CO CCCC(CCCNC(=O)CC(C)C1CCCCC1)NC(=O)CCC(=O)OC C1(C(=O)NC2C=CCCC2C(=O)NCC2CC(C)C2)CC2(CCO1)CC2 c1(C(=O)NC2CCN(C(CCC=CC)=O)CC2CO)ccc2c(c1)CCCO2 C(C)(C)(CCC(=O)NCC1(C)CCC(NC(=O)CCC2CC2)C1)OC c1(C(N(C2CCCC2)CC)=O)cc(Cl)c(Cl)n1C.CC(C=O)OC1CCCC1.N C1(CC)CN2CCCC2CN1S(=O)(=O)Cc1ccc(C#N)cc1OC c1(OC)cccc(F)c1C(=O)NCC(C)(C(C)C)NC(=O)Cc1cnc[nH]1 C(=O)(C(C)(C)CC#N)NCC1CC(NC(C2C(c3n(C)c(S)nn3)C2)=O)C1 C(=O)(C(O)CC(F)(F)F)NCCCN(C(CC(N1CCCCC1=O)C)=O)C CCCCC(O)C(=O)NC1CCC(NC(=O)C(C)Cn2ccc(C)n2)CC1 C1COCCC1.N1(C(=O)OC(C)(C)C)CSCC1C(=O)N.C(=O)C.C1CC1 Cc1cc(C)n(CCNC(C2CCN(C(=O)CCc3ncnn3C)CC2)=O)n1 C1(C(=O)NC(C2CCN(C(C3(C4CC4)CC3)=O)C2)C)CC(F)(F)C1 c1(C(=O)NCC(CC)NC(=O)C(C)NC(C)(C)C)ccc2cc(C)cn2c1 N1(C(CNC(=O)NC)=O)CC2(C1)SCCC2NC(=O)C(c1cncn1C)=O c1(CC(C)C)nc(C(=O)NC2COCC2NC(=O)Cc2cscn2)cs1 Cc1ccc(C(=O)NCCCCNC(=O)CO)c(O)n1 C1(CC)C(C(=O)N)CCN1C(=O)Cc1cccc(O)c1.c1cccc(N(C)C)c1 c1(C(N2CCC(CO)C(O)CC2)C(=O)NC(CC)C)nc2ccc(OC)cc2s1 CC1=C(C(=O)N)CCC(C)(C)C1.C1(C(N2CCC(O)C2)=O)CC(C)(C)CN1C.C CC12CN(C(c3ncn4c3CCC4)=O)C(C(=O)NC3CC4(CC4)C3)(C1)C2 C1(NC(CSCC=C)=O)CCN(C(=O)C(=O)NCC)C1C CC1CN(C(c2cccc(O)c2F)=O)CC(CCNC(=O)CC2CCCSC2)O1 CCC(CC(=O)NC(c1cn(-c2ccc(C)cn2)nn1)CSC)SC CCCCC(CC(=O)N(C(C)C(C)(C)C)C)NC(C1COCC1(C)C)=O C1(C)(CNC(CC(=O)OCC)=O)CCCN(C(=O)CC2CCC2(F)F)C1 c1(C(N2C3C(NC(C4C(C)(Br)C4)=O)C(C3)C2)=O)cc2n(n1)CCCCC2=O Cc1cnc(N2CCC3CC3C2)c(S(=O)(=O)NCCc2cnccc2C)c1 c1(C(=O)NCC2CN(C(c3nc(C)oc3C)=O)C(C)(C)C2)cc2sccc2cn1 N1(c2c(C)ccc(C)c2)CCN(N2CC(c3ccccc3)OC(C)(C)C2)CC1 C(=O)(CCC(C)(C)N(C)C)NCC(C(C)C)NC(COCC(C)C)=O CC(CC(=O)N1CCOC2CN(C(C3(F)CCCCC3)=O)CC12)CC(C)(C)C C1(C(=O)NC)CCC2C(C1)C2(F)F.C1CC2CC2N1C(=O)Cc1ccccc1 N1(C(CCC(=O)N(C)C)=O)CC2CCCC2(CNC(=O)C(c2cccn2C)=O)C1 CS(=O)(=O)c1cnc(O)c(C(=O)NCC2CCN(C(=O)C3=CCCC3)C2)c1 C(=O)(C1=NN(C(C)C)C(=O)CC1)N(CC(CO)CO)C.C(C)C=O.C#CC.O N1(C(=O)Cn2cccc2)CCC(NC(C23OCCCC2C3)=O)CC1C1CC1 N1(C(c2nocc2C)C(=O)NC)Cc2ccnn2CC1C(C)C N1(C(CC(C)C2CC2)=O)CCC2(CC1)CN(C(=O)C=Cc1cncs1)C2 CCC(C)(F)C(=O)N1CC(CNC(c2cnccc2C(F)(F)F)=O)C(O)C1 N1(C(c2nccc(C)c2)=O)CCC2CCC12CNC(c1ccc(C)n1C)=O c1(C(N2C(CCCNC(CC=CC)=O)CCC2)=O)ncc(F)cc1C N1(C(CCSC)=O)CCCC2CCN(C(c3ncn4ccccc34)=O)CC12 CC(O)CN(Cc1ccccc1)N1CCCC(C)(C)C1 C(=O)(C#CC1CCCCC1)NC1C(NC(C(c2ccc(OC)cc2)O)=O)CCC1 C1(C(C)C)CN(C(c2ccc(C3CC3)s2)=O)CCN1C(=O)CC1COCCOC1 CC1(C)COCC(CS(C)(=O)=NC(=O)c2cc(F)cc(F)c2)O1 CCC1=C(C(=O)NC2CC(NC(c3c(C)ncn3C)=O)C2)SCCO1 C1(C(=O)NCCCCCF)(CNC(Cc2c(C)non2)=O)CCCCC1 c1(CC)cc(Cl)ccc1C(=O)N(CC)C(C)C.C1(C=O)CCN(C(C)C)C1 C(=O)(C1CCc2cccnc21)NCCCN(C(c1cc(C(C)C)[nH]n1)=O)CCO c1(C(N(CCN(C)Cc2cnc(C)o2)C(C)C)=O)cccc2c1COCC2 C1(C(=O)O)CCC2(CCCN2C(=O)CSc2cncc(-n3cccn3)n2)CC1 O=C(CC1=Cc2ccccc2C1)NCCNC(c1cnncc1O)=O C(CCC(C)(C)C)N(C(=O)CC(=O)N(C)C)C.C(C)(C)C(F)(F)F.C(=O)C Cc1nnc(=NCC2CN(C(c3cccc(Br)c3C)=O)CC23COC3)[nH]c1C C1(C(N2CCC(CNC(C(C)OC3CCCC3)=O)C2)=O)CN2CCCN1CC2 n1(-c2cn(C)nc2)nc(CCc2ccc(Cl)cc2)nc1CC1CCCC1 C1(=CC(N2CCCC2)=O)CC2CCC(C1)N2C.c1(CC)nnc(C(=O)N)s1.C C12(NC(CCNC(C)=O)=O)CCC(F)(F)CC1CN(C(=O)C(O)CC(F)F)C2 N1(C(C(n2c(C)ccn2)C)=O)CCCC2(CCC2)C1.C(=O)(C(=O)N=S(C)(C)=O)N C(=O)(C1CCCc2cncn21)NC1CCN(C(c2c(OC)nn(C)c2)=O)C1 c1(C(N2C3CN(C(c4ccc(Br)c(F)c4)C)C(C3)C2)=O)cn2c(n1)COCC2 C=C(C)CCCC(=O)N1CCC(C(=O)NC2(C)CC(F)(F)C2)C1C c1(C(=O)NC2(c3cn(CC4CCCC4)nn3)CCCOC2)c[nH]cc(Br)c1=O N1(C(c2cc(CC)no2)C(=O)NCC(F)F)CCc2ccc(S(N)(=O)=O)cc2C1 c1(C=O)ccn2ccsc12.C1(S(C)(=O)=O)(C(N2CCC(CC)CC2)=O)CCC1.N C(=O)(C(C)(O)C(C)C)N(CC(CC)NC(c1cc(Cl)cnc1C)=O)C c1(CN=C(NC(c2cc(C)sc2C)C)NC2CC2)ccc2c(c1)OCO2 c1(C(=O)OC)c(F)ccc(S(=O)(=O)NC2CCC23CNC3)c1F C1(CC(=O)NC2CCN(C(=O)C(F)F)C2c2ccccc2)(CCO)CCCCC1 S(=O)(=O)(c1ccc(N2CCCC(F)(F)C2)c([N+](=O)[O-])c1)N(CC)C.N(C)C C12(C(=O)OC)CCCC1(C(=O)NC1(C)CN(C(C3C4COCC34)=O)C1)C2 S(=O)(=O)(c1ccc(S(N)(=O)=O)cc1)NC1CCC(CN)CC1 C1(C(=O)NCC(C(C)C)OC)(NC(c2ccnn2C)=O)Cc2ccccc2C1 N#Cc1ccc(S(=O)(=O)N2CC(O)CC2C(N2CCC2c2cccs2)=O)cc1 CS(=O)CCCCNC(c1nnnn1CCCF)C1(OC)CCCC1 N1(C(Cc2nc(=N)[nH][nH]2)=O)CC2CC(NC(=O)CC3CC4C=CC3CC4)CC2C1 C(C(=O)NCC(C)OC)(c1ccoc1)NC(C1C(CC)C1)=O C(C)(N=c1[nH]c(N(CC(=O)N(C)C)C)nc2ncn(C)c12)c1cc(OC)ns1 N1(C(C(=O)NCCOC)=O)CCOCC1CNC(=O)CC.c1ccccc1Cl N1(C(C2(CC)CC2)=O)CC=CCC1.c1(CC=O)cc(=O)n(CC(C)C)[nH]1.C C1(C(N2CC(CC=C)(C(=O)NCc3cnn(CCF)c3)C2)=O)CCCCC1C CCC(CCOC)C(=O)NCC(O)CNC(=O)C=Cc1c(C)coc1C c1(C(=O)NC2C(NC(C(C)OCOC)=O)CCC2)cnn2c(Br)cccc12 c1(NC(C2CCN(C(N)=O)C2)=O)ccc(Cl)c(F)c1F CC1(C)C(C=O)CCS1(=O)=O.C1CC(F)(F)CC1.C(c1ccoc1)=CC=O.N C(c1cnn(-c2ccccc2)c1)=C(C)COC1CCN(C(=O)C(C)C(C)O)CC1 c1(OCC)cnc(OCC)c(C)c1.c12nc(no1)CN1CCC1C2 Cc1c(C(=O)NC(C)CO)cccc1S(N)(=O)=O.c1(C(=O)N)cc(CCO)on1 N1(C(c2cc(CC)ncn2)=O)CCN(C(c2ccc(CO)c(F)c2)=O)CC1CF CC1(C(=O)NCCNC(=O)C=CCF)CC2CC2C1 C1(C(=O)NCC2N(C(c3cc(N)c(Cl)cn3)=O)CC2)CCCCC12CCC2 N1(C(c2nc(COC)[nH]n2)=O)CCc2ccccc2C1CNC(C1CC12CC2)=O N1(C(Cc2n[nH]c(=N)s2)=O)CC2C(CNC(C34CCCC3C4)=O)C2C1 C1(C(N(CC=O)CC)=O)CCC(C2CC2)N1C(=O)Cc1ccco1.CC c1(C(=O)NCC(c2cccc(F)c2)C)cccn2cnnc12 C1(CNC(COCC(=C)C)=O)CC(NC(c2cnccc2Cl)=O)CC1O c1c(C)cccc1C.c1(COC)nocc1C(=O)N.C1C=CCN1C(=O)C.C N1(C(=O)NC2(CCNC(C(C)C)=O)CCC2)CCN(C2(C)CC2)CC1 C12(CNC(CC(C)SC)c3nnnn3Cc3ccccc3Cl)CCC(CC1)CC2 C1(C(=O)NCc2ccc(C(=O)NCC(C)C(F)F)nc2)CC12CCOCC2 CP(C)(=O)CC(=O)NC1CCCCC1NC(C1CC2(CC2)C1)=O C1(OC)CN(C(=O)C(F)(F)c2cccnc2)CC1NC(c1cncc(Cl)c1)=O C1(C(=O)NC(CCC)CO)CC12CCN(C(c1cc(OC)ns1)=O)C2 c1(COC)cc(C(=O)N)c(C)o1.C1CCCCC1.c1(C=O)cnc(C2CC2)s1 C(=O)(C1=CCC(C)(C)CC1)NC(C(=O)NC1C(O)CCN(C)C1)Cn1cncn1 c1(C(=O)NC(C)CN(C)C(C2CC3CCC3C2)=O)cc(Cl)c(N)cc1F Cc1n[nH]c(C)c1CC(=O)NC1C2CCN(C(=O)C(F)n3cccn3)C12 n1(CC)c(C(=O)N)cnc1O.c1(C(N(CCC)C)=O)cc(C2(C)COC2)no1 c1(CC(=O)NCC(C)N(C(COCCC)=O)CC)n[nH]c2ccccc12 C(=O)(CC1=NNC(=O)C1)NCC1(O)CCCN(C(Cc2c(C)occ2)=O)C1 Cc1cccc(-c2cn(C(C3CCC4(CC4)CO3)C3CC3)nn2)c1F C1(NC(C(CC)CO)=O)CCC2CCN(C(c3cc(C)sc3C)=O)C1C2 c1(C(C(N2CCCC(N(CCNS(CCC)(=O)=O)C)C2)=O)C)ccc(F)cc1F c1(C(C)(COCC)NC2(CC)CC2)nnnn1CCC1(OC)CCC1.S c1(C(N2C(CCC)CN(C(c3cnnn3C)=O)CC2)=O)n[nH]c2ccc(F)cc12 C(=O)(C(CC1CCCCC1)C(C)C)NCCN(C(=O)C(C)n1cncn1)CC C1(NS(=O)(=O)Cc2ccc(Cl)cc2)CN2CCC1CC2 c1(C(=O)NCC2(NC(c3c(C#C)c[nH]n3)=O)CCOC2)cnc(N)c(Br)c1 C1(C(=O)NCc2c(C)ccs2)(NC(C2COCCC2C)=O)CCCCC1 N1(C(=O)OCC)CCN(c2nnc(-c3ccc(F)cc3F)n2CC)C(C(C)C)C1 Cc1cc(N)cnc1C(N1CCC(O)(CNC(c2cscc2Br)=O)C1)=O N1(C(c2c(C)noc2)=O)CCC(C)N(C(=O)CN2CCCC(N(C)C)C2)CC1 c1(NC(C(C(=O)OC)C)=O)cnc2c(c1)CN(C(c1ccc(I)c(F)c1)=O)CC2 c1(C(N2CCN(C(=O)Cc3cscn3)C3C2C3)=O)c[nH]c2cnccc12 C(=O)(C1CCc2nccn21)NC(C(=O)N(C1CC2CC2C1)C)C1CC1 CCC(C)CC(CO)NC(=O)CCC(C)(C)NC(=O)C(C)=CC1CC1 n1(NC(CCNC(C2C(C)C2)=O)=O)cc(C(N2CCCC2)C2CC2)nn1 C1(C(C)(C)C)CCOCCN1CC1CCNC(=O)C1 C1(CNC(=O)CCCF)COCCN(C(=O)CC2CC2c2ccc(F)cc2F)C1 C(=O)(CCCCCN=[N+]=[N-])NC(C(CC)C)C(=O)Nc1ccc(N(C)C)cc1 N1(C(C2CCc3c[nH]nc3C2)=O)CCC2(CCN(C(C3CSCCS3)=O)CC2)C1 CCC(C)C(C(=O)NC)N1CCCC1c1cn(C2CC2)nn1.c12nc(cs1)C2 N1(C(C(C)C#N)=O)CCC2(CCC(CNC(C3(C(F)F)CCCCC3)=O)O2)CC1 C#CC1(C(=O)NC(C)Cn2ccnc2)CCN(C(c2nocc2C)=O)C1 Cc1c(C(=O)N(CCCNC(=O)C=Cc2cnc[nH]2)CCO)ccn1CCO c1(C(C)(C)C)ccc(Br)cc1C(N1CC(CC(=O)Nc2cc(Cl)c(Br)cn2)C1)=O CC1=C(C)CN(C(C2CCC(CNC(c3cc(C4CC4)on3)=O)O2)=O)C1 c1(OC)cc(C(=O)NC)n(C)n1.C1CCN(C(c2cc(C3CC3)no2)=O)C1 C(=O)(C(C(C)(C)C)c1ccc(C)cc1)N1CC2C(CN(C(CC=C)=O)C)C2C1 C(=O)(C1=CCN(C)C1)NC(C(C)NC(C1(COCC)CCC1)=O)C c1(C(C(=O)NC(Cn2cc(-c3c(C)c[nH]n3)nn2)C)(C)C)ccc(F)c(F)c1 C(CC(CC)C(=O)NCC(CC)NC(=O)COC1(C)CCCC1)=CC Cc1cc(Cl)c(C(N2CC(C)(c3cn(CC4CCC5CC5C4)nn3)C2)=O)s1 Cc1ccc(C(=O)NC(c2cccnc2)C(N2CCC2(C)CCO)=O)n1C c1(OC)ccc(C=CC(=O)NC2COCC2NC(C2CC2C)=O)cc1 C=CCN=C(NCCc1cc(Br)ccc1F)N1CCC(NC(C)=O)C1 N1(C(c2c(C)[nH]cc2)=O)CCCC(NC(c2cnc(CCC(F)(F)F)s2)=O)C1C CCC(C)CCC(=O)NCCN1CCCN(C(=O)CCc2nc(C)cs2)CC1 C1(NC(C=C(C)C(C)C)=O)CC(C(=O)NCC2(CO)CC3CC3C2)CC1O N1(C(C(CCC)O)=O)CC2CCCC1C2CNC(=O)C(CC)(CC)OC C1(CCSCC(C)C(=O)Nc2ccccc2)CCCN(c2nnc(C#N)s2)C1 n1(CC)nnc(C)c1C(=O)NCC1(COC)CN(C(C2CCOC2)=O)C1 C1(NCCNC(C(C)(C)CO)=O)CC2CCC(C1)N2C(=O)CN=[N+]=[N-] Cc1nc(C2CCCO2)sc1C(N1CC(NC(C2CC3CC3C2)=O)C1)=O c1(OC)ccc2nccc(CNC(=O)N(C3CCSC3)CCN(C)C)c2c1 c1(C=O)ccc([N+](=O)[O-])s1.CCC(CNC(C1C=CC1C(=O)OC)=O)CC C1(C(=O)Oc2ccc(NC(C)=O)c(Cl)c2)Nc2ccccc2C1(C)C C1(C)(NC(CN(CCC)C)=O)CCN(C(=O)Cc2ccnc(OC)c2)C1 Cc1csc(NC(C2CN(C(=O)CCc3ccccc3F)C2)=O)c1C#N N1(C(C(C)Oc2ccccc2Cl)=O)CC2(CCCC2NC(C2CC=CCC2)=O)C1 C(=O)(CC=C(Cl)Cl)NCC(C1CCOC1)NC(c1c(C)csn1)=O Cc1cccc([N+](=O)[O-])c1C(=O)NC(C)CCN(C)C(C1COCCN1C)=O C1(C(=O)NCC2(NC(C(C)CF)=O)CCCCC2)CCc2ncccc2C1 N1(C(c2ccc(OC)nc2)=O)CCC(CO)(NC(c2csc([N+](=O)[O-])c2)=O)CC1 c1(CNC(C(CC)C#N)=O)cccc(F)c1.C1(F)(C=O)CCN(C(C)(C)C)C1 C(=O)(CCC(=O)N1CC(O)CC1)NCC.c1(C=O)sc(C(C)(C)C)nc1C.C N1(C(c2c(C)scn2)=O)CCC2CC12C(=O)N(C(C)CO)CC1CCC1 C(=O)(C1CCCc2cn(C)nc21)N(CCCOCCO)C N1(C(C2(C#N)CCC2)=O)CCCCC(NC(=O)CN2CCCC2=O)C1 Cc1ccc(C(=O)NCC(F)CNC(c2ccc(-c3ncon3)cc2)=O)nc1C Cc1cc(C(=O)NC2CCC(O)CN(C(=O)C(C)C(C)(C)C)C2)c(F)cc1Cl c1(C(=O)OC)csc(C(N2CCCC2c2cn(CC3CCCOC3)nn2)=O)c1 C(=O)(C1=Cc2ccccc2C1)NCCCCC(C)(C)NC(c1cc(F)c[nH]1)=O N(C1CC(C)n2ccnc21)C(CC1(CSCC)CC1)=O C(=O)(CN=c1cc[nH]cc1)N1CC(NC(C(CN(C)C)N(C)C)=O)CC12CCC2 N1(C(C(C(C)C)C)=O)CCC2CC1CN2C(c1onc2ccccc12)=O C1(C(=O)NCC(C(C)C)(C)F)CC2CC1CN(C(=O)C(C#N)C(C)(C)C)C2 C1(NC(CCOC(C)C)=O)CN(C(C2CCS(=O)(=O)N2)=O)CC1C C1(NC(CSc2ccc(OC)cc2)=O)C2CC3CN(C(=O)CNC)C1C3C2.C C1(C(N2CC3C(NC(CCCCSC)=O)C(C3)C2)=O)CCCCC(F)(F)C1 C1(O)(C(=O)NCC2(O)CN(C(c3[nH]c(=NC)sc3)=O)C2)CCCC(C)(C)C1 N1(C(c2n(C)cnn2)=O)CCC2(NC(C3CSCCS3)=O)CCCC12 C1(NC(CN2C(=O)NCC2)=O)CC2CCC1N2C(C1CCCSC1)=O N1(C2CCN(C(=O)OC(C)(C)C)C2)CCN(C(C2C3CCC2CC3)=O)CC1 c1(CCC(=O)NC(CNC(C(F)OC)=O)C(C)C)csc2nc(C3CC3)cn12 N1(C(C2(C)CCCC2)=O)CC2CCCC(CNC(=O)C(Cl)=CCl)C2C1 Cc1cc(C(C)(C)NC(=O)CC2CCCC2NC(=O)C)on1.C1CC=CC1 C(CCCC(=O)NCC1(O)CCSC1)NC(=O)C=CCN1CCC1 C1(COC)CN(C(=O)CN=S(C)(C)=O)CCN1C(=O)CC1CCCC1 n1(CC)c(C)cc(C(=O)N)c1C.c1(C(N(CCC)C)=O)cc(C2CC2)nn1C C#Cc1nc(C(=O)NCCC(C)NC(C2CCN(c3ncccn3)CC2)=O)cs1 c1(C(=O)NC2(CNC(CS(CCC)(=O)=O)=O)CCOC2)ccc2c(c1)CCCC2 C1(C(N(C2CCN(C(C3CCCO3)=O)CC2)C)=O)NC(=O)C2CCC12 C(C(C)(CC)C(=O)NCC(C)C(F)F)NC(C=C(CC)CC)=O c1(Nc2ccnc(CN(C)Cc3ccc(OCC)cc3)n2)c[nH]c2cccnc12 c1(C(=O)OC)cc([N+](=O)[O-])cc(Cl)c1NC(c1cc2c[nH]nc2s1)=O CC(CC(=O)N1CCC(C)(CNC(c2cc(C#N)ccc2F)=O)CC1)P(C)(C)=O C1(C(=O)NC(C2(O)CCN(C(c3cn(C)[nH]c3=N)=O)C2)C)OCC2CCCC1C2 C1NC(=O)OC1(C)C.N1(C(C2C(OCC)CC2)=O)CCOC(CC(=O)N)C1.C c1(C(N2CC(CC=C)(C(=O)N(C(C=C)C3CC3)C)C2)=O)cn(C)ccc1=O Cc1cc(CO)oc1C(=O)NC(C)CN1CCN(C(c2ccsc2C)=O)CC1 C(CN=c1cc(C(F)(F)F)nc(Cl)[nH]1)(c1ccccc1F)NC(C1(C#C)CC1)=O CN1CC2(CCCN(C(C3CCCN(C(=O)Cc4cnc[nH]4)C3)=O)C2)OC1=O O(NC(=O)CC(O)CNC(=O)CCSC)CC(=C)Cl c1(OC)nc(=NCCC(C)NC(c2ncoc2C(C)C)=O)nc(OC)[nH]1 C1(C)(C(N(C)C)=O)CCC(=O)N(C)C1.CC1=NOC(C(N2CC(O)C2)=O)C1C c1(C(=O)NC(Cn2cc(-c3c(C)cn(C)n3)nn2)C)oc2ccccc2c1Cl c1(C(=O)NC2CC(O)CN(C(c3cc(Cl)ccn3)=O)C2)cnc2ccccc2n1 CC(C(=O)N1CCOC(CCCNC(=O)CN2CC3CCC2C3)C1)S(N)(=O)=O C(=O)(CCCCC(N)=O)NCCC12C(CN(C(C(F)=C(C)C)=O)C1)CC2 C1(O)(C(=O)NCC2CC(C)N(C(=O)CC3(C(F)F)CC3)C2)CCCCCC1 Cc1cc(F)c(N)cc1C(=O)N(CC(C)NC(=O)CCc1cn[nH]c1)C N1(C(c2c(OC)nn(C)c2)=O)CCC(C)(C)CC1C(=O)NCC1=NOCC1 C(=O)C(C)CC(C)C.C1(CC)CCC(C)CC1.c12cccc(c1)C(=O)N(C)C2.N C1(COC)CN(C(c2nc(C)no2)C(=O)NCCCSC)CCO1.C1CC1.O C=C1CCN(C(=O)C=CC(F)F)C(C(=O)N(C)CC2(CC(C)C)CC2)C1 Cc1c(F)ccc(C(N2CCC(CNC(=O)CC3COC(C)(C)C3)C2)=O)c1N N1(C(CCSC)=O)CCC2C1CCCN2C(=O)C(c1ccc(C)cc1)=O c1(C(C)C)ccccc1COC(=O)CC1(C)CC1(F)Cl C(=O)(CC(F)(F)C(F)F)N1C(CCNC(c2cc(=O)cc[nH]2)=O)CC(OC)C1 c1(NC(=O)NCC(C)(C)O)cccc(OC(F)F)c1.c12cnn(c1)C2 C1(c2n(CC=C)nnn2)(NCC2(CO)CCOC2)CCN(C2CC2)CC1 N1(C(C(F)=CCC)=O)CC2(COC(CNC(=O)C(C)NC(N)=O)C2)C1 C1(CC(=O)NCCCNC(c2cncn(C)c2=O)=O)Cn2ccnc2NC1=O N1(C(C(C(C)(C)O)(F)F)=O)CCc2c(CC(N)=O)cccc2C1.C(=O)CN C(CC(=O)NC(c1scnc1C)C)(CC(C)C)NC(CCC(C)=O)=O c1(OCCNC(CCN(C(=O)C(C)(C)O)C)=O)cccc(F)c1 C1(NC(c2nc(C)oc2C)=O)CCCC12CCN(C(C1(C)CCCCO1)=O)CC2 C1(C)(C(=O)NC2CC(C)(NC(c3cccn(C)c3=O)=O)C2)CCCC(F)(F)C1 N1(C(C(C=C)(C)CC)=O)CC2(NC(c3cnc(SC)nc3O)=O)CCC1CC2 Cn1nc2c(c1C(N1CC3CCC(C1)N3Cc1cc(C#N)ccc1F)=O)CCC2 C1(C(C)NC(C2(OC)CCC2)=O)CCN(C(C2CC(C)OC2C)=O)CC1 c1(C(=O)NCC2CCN(CC(C)C)C2)nc[nH]c2ncnc1-2 c1(C(=O)NCCC2(O)CN(C(c3c(C)cno3)=O)C2)cccc(CO)n1 CC1(CNC(C2CC=CCN2C(=O)CNC(=O)C2CC2)=O)C=CCCC1 CCCCCC(O)CC(=O)NC1C2CN(C(=O)CCSC(F)(F)F)CC12 C(CC(C)C)(C(=O)NC1CN(C(C2CC3CCC(C2)C3)=O)CC1C)OC c1(OCC)ccc(C(=O)NC2(C)CCN(C(=O)CCc3ccccc3F)C2)nc1 CC1CCCCC1N(C1CN(C(c2ccc(CNc3cnn(C)c3)o2)=O)C1)C c1(C(=O)N)cc2c(s1)CCC2.N1(CC)CCOCC1C(=O)N(CCC)C1CC1 c1(C(=O)NCC23CC(NC(C(C(CC)C)C)=O)(C2)C3)cc2c(ncn2C)s1 c1(NC(C(CC)=O)=O)ccc(C(=O)Nc2csc(-c3ccsc3)n2)c(F)c1 CC1(C)CCCC(CNC(C2CCN(C(=O)CSC(F)F)CC2)=O)C1 c1(CNC(c2c(OC)ccc(C(=O)O)c2)=O)cc2ccccc2oc1=O N1(C(Cn2c(C)csc2=O)=O)CCN(C(C2CCC(C)(C)C2)=O)C2COCC12 C1(C(=O)N)C(C=O)CCN1C(=O)CC.C1(COC)CC1.CCN(C)C N1(C(C(C)Cc2ccccn2)=O)CCCC(NC(C2(C#N)CCSCC2)=O)CC1 N1(C(C2C(CCC)C2)=O)CCCC(N(C(C)=O)Cc2cc(CF)on2)C1 n1(CC=O)nc(C)cc1C.C1CCS(=O)(=O)C1.C1(OC)CN(C(=O)C)C1.C N1(C(c2c(CC)onc2)=O)CCC(C)C(NC(C23COC(CCO2)C3)=O)C1 C1(C(N2CC(N(C(C(C)(C)SC)=O)C)C2)=O)CCn2nnnc2C1 C1(C(N(C)Cc2cc[nH]n2)=O)CC2CCC1O2 Cc1ccc(CC(=O)NC2CCN(C(=O)CCC(C)(F)F)C2C)c(F)c1 N1(C(CCC=C=C)=O)CC(NC(c2cc(C)nn2C2CCC2)=O)CC12CCOC2 N1(C(=O)CCn2cncn2)CCCC(C2CCCN(C(c3cccs3)=O)C2)C1 C(=O)(CCCC(C)(C)C)N1CC(CC(C(=O)NC(c2cnc[nH]2)C)F)C1 C(=O)(CCCCN(C)C)NCCCCCN(C(C(c1ccc(F)cc1)C)=O)C N1(C(c2snc(C)c2N)=O)CCN(C(c2cscn2)=O)CC2(CC2)C1 c1(C(N2CC(O)(CCNC(C(C=C)(C)C)=O)C2)=O)cc(=O)c2ccccc2o1 N1(C2(C(N)=O)CCOC2)CCN(C(c2cnc(-c3cncnc3)nc2)=O)CC1 C#Cc1cn(C)nc1C(=O)NC1CCC1C.C(=O)C1=NNC(C(F)(F)F)C1 C1(C(N(C)CC2C(NC(C(C=C=C)C)=O)CCC2)=O)CC12CCOCC2 c1(C(=O)N)cnc(C)cc1C.C1(OC)(C)CCN(C(=O)CNS(N)(=O)=O)C1 C1(CCC(=O)NC(CC2CCCC2)C(=O)N2CCCC2CF)CCCOC1 c1(C(N2CC=CC2)=O)cn(C)c(O)n1.C(C)(C)(C=O)NC(=O)NCCC CC1C(C(=O)NC23CC(C2)C3)=NOC1C.C1(C=O)CC(=O)N(C(C)C)C1.N C(=O)(CS(=O)(=O)CC(C)C)N1CCC1.c1(OCCC)nc(C)ccc1C(=O)N c1(SC)ccc(O)c(C(=O)NCC2CC2NC(=O)C)c1.c1ccccc1C N1(C(C2C(C)CCOC2)=O)CC2(CNC(=O)Cc3ccnc(O)c3)CC1CO2 C(=O)(CC(F)(F)C(F)F)N1C(CC(=O)NCCSC(F)F)C2CCCC21 c1(CC(=O)NC2CC3CC(NC(C4(F)CCOCC4)=O)C2C3)ccc(O)c(Cl)c1 Cc1nc(C(=O)NCC2C(C)CCN2C(c2sccc2C#N)=O)ccc1[N+](=O)[O-] C1(F)(CNC(C(=O)OCC)=O)CCN(C(=O)C(C)OC)CC1 C1(CC)C(NC(=O)CCn2cncn2)CCCN1C(=O)CCCc1cc[nH]n1 C=CCCCCCCCC(=O)NC12CCC(CC1NC(c1n[nH]c(C)c1Cl)=O)C2 C#CC(CNC(=O)C(C1CCCC1)NC(c1cc(C)c[nH]1)=O)C(C)C c1(CC(=O)NCC(C)NC(C(C(=O)OC)OC)=O)cn2ccsc2n1 c1(C(=O)NC2C(NC(Cc3c(C)nc(S)s3)=O)COC2)ccc(Cl)c(F)c1O C1(C(=O)NC2(C(=O)NCCCCCCCO)CCCC2)CC2C=CC1CC2 C1(NC(C2N(CC)CCC2)=O)CCOC(C(=O)N)C1.C1CCC(C(C)(C)C)O1 C(=O)(C(O)CCC(C)(C)N)N(C(c1ccccc1)C(=O)OC)C C1(CNC(C2(C)CC(C)C2)=O)CC12CCC2.C(=O)C(O)(C1CC1)C1CC1 c1(C(N2CCCN(C(C=Cc3c(C)nccc3)=O)CC2)=O)ccc(P(C)(C)=O)o1 C(=O)(C1CCOc2c(F)cccc21)N1C(C)CCN(C(CCCOCC)=O)CC1 C(C(=O)N=c1cc(C)cn[nH]1)C1CN(c2nc(OC)nc(OC)n2)C1 c1(NCC(C2CCCC2)OCC)ccc(S(=O)(=O)N2CCCC(C)CC2)cc1Br O=S(=O)(c1c(Cl)cc(F)cc1Br)N1CC2CNCC2(CCC(=O)N2CCCC2)C1 N1(C(CCCN(C)C)=O)CCCC2C1CCN2C(C1CC12CC(F)(F)C2)=O c1(C(N2C(CC)CCC2)=O)cc(F)c(C)cc1Cl.C1(C=O)(OCC)CCOC1.N N1(CC)CCC(NC(=O)CCC(C)NC(=O)CCc2ccncn2)C1=O c1(C(=O)NC(CCOC)CNC(=O)Cc2ccnn2C)cc2n(n1)CCCC2O c1(CCC(N2CC=CC(NC(C(C=CC)O)=O)C2)=O)c(C)[nH]c2ccccc12 C1(O)(C(=O)NC2CC(NC(c3c(C)ncnc3C)=O)C2)CCCC(C)(C)C1 C1(C(N2CCC(C)C2)=O)CS(=O)(=O)CC(=O)N1.Cc1nnnn1CC(=O)N.C c1(C(CC)NCC2OCCC2C)cnnn1CC C(=O)(C(=O)N=S(C)(C)=O)N(C(C)C)C.C(=O)(CCO)N.C(=O)C.C1CC1 c1(NC(C2C(C(C)NC(C3CN(C(C)=O)C3)=O)C2)=O)n[nH]c(O)n1 C1(COc2c(OC)cc(C(=O)O)cc2)Cc2ccc(F)cc2C1 c1(C(N(CCNC(CCC2CCC(C)O2)=O)C2CC2)=O)ccnc(F)c1O Cc1cc(NC(=O)COCCc2cn(C(C)C(=O)N3CCCC3)nn2)nn1C CCCC(CC)C(=O)NC1(CN(C(=O)C(=O)Nc2ccc(C)cc2)C)CC1 c1(OC)cn(CC(=O)N(CCCN(C(=O)CC2CCC(C)C2)C)C)c(C)cc1=O C1(NC(C2(CCCC)CCCC2)=O)CC(NC(=O)C(c2ccnn2C)O)C(O)C1 C1(NC(c2ccc(-n3cccc3)cc2)=O)CN(C(C2CCCCC2)=O)CC1CO C1(C(C)N(C(=O)C(C2CCN(C(C3CC4(CC4)C3)=O)C2)F)C)CCOCC1 c1(OC)ccccc1CCNC(=O)C(O)CN(C)C.C(=O)C=CC1CC1 C1(NC(c2cnnc3ccccc23)C)Cc2ccc(C(=O)O)cc2C1 c1(-n2c(Cc3ccoc3C)nc(CC(CC)C)n2)cc(F)cc(F)c1 C(=O)(CCCCC(C)(C)OC)N1CC2C(N(C(C(CC=C)C)=O)C)C2C1 c1(OC)cncc(C(=O)NCCC2CCCC2)c1.C(=O)(CCC=CC(C)C)N N1(C(C(=O)NCC)=O)CC(C)CN(C(C2CC(OC)(OC)C2)=O)CC1C N1(C(C(C)(C)CC2CC2)=O)CC(C2CCCCN(C(c3cc(CO)[nH]n3)=O)C2)C1 c1(CN(C(C(C)=C2CCCC2)=O)C)cccc(C)c1.C1(O)(C(=O)N)CCOC1 Cn1cc(S(C)(=O)=O)c(C(=O)NCCC(C)(C)C)n1.C(C)(C)C.C(=O)N c1(C(N2CC3C(CNC(c4c(C)cco4)=O)(C3)C2)=O)cccc(C)c1I N1(CC)CCOCC1CNC(=O)CC1(C)CCN1C(c1cnc(C)n1C)=O C(CCC(C(=O)NCC1CCCC(C)O1)NC(c1coc(C2CC2)n1)=O)OC C(=O)(CC1=NN(C)C(=O)C1)N1CC(CC(=O)NCc2c(CC)nn[nH]2)C1 NS(=O)(=O)C1(C(=O)NC2CCC(CC)C2)CCC1.c1(CC(=O)N)cnns1 C1(C2N(C)CCC2)CN(C(=O)C#CC2CC2)C2(CCOC2)C1.c1ccccc1F N1(C(C(OC)OC)=O)CC2CCC1CN(C(c1cccc(F)c1F)=O)C2 N1(C(CC2CC(NC(CCC=CCC=C)=O)C2(C)C)=O)CC2CCC(CO)(C2)C1 C1(C(=O)NCC23C(CN(C(CCC(=O)OC)=O)C2)C3)CC2C=CC1C21CC1 C=CCCCC(C(=O)N1CC(O)(C2CCC2)C1)NC(C1CC2C=CC1O2)=O CC(C)C(C)(C)C(=O)NCC1(O)CCCN(C(=O)CN2CCN(C)CC2)C1 N1(C(C(=O)NCCSC)C2=CCCCCC2)CCOc2c(F)cc(F)cc2C1 CC(=O)CC(C)(C)C(=O)N1CC=C(CNC(C2CSC2)=O)CC1 C#CCC(CC(=O)N1CCCC1C(C)(C)OC)NC(c1ncc(F)cc1C)=O c1(CNC(C2(C(C)NC(c3csc(F)c3)=O)CC2)=O)cnn(C)c1O C1(C(=O)NC(CC#C)C)CCCN1NC(=O)C1CC(=O)OC1(C)C c1(CC)cc(-c2ccc(C(=O)NCc3cc(Br)c[nH]3)cc2)ccn1 C1(C2CC2)(CNC(C(C)CO)=O)CCN(C(C2CCCC23CC3)=O)C1 N1(C(=O)Cn2cnnc2)CCC2(CCCN2C(c2ccncc2O)=O)C1 N1(C(c2cc(C)n(C(C)(C)C)n2)=O)CCC2CN(C(c3ccncc3Cl)=O)CC12 c1(OC)cccc(Br)c1CN(C)CC1CCCN(C(c2ncc(Br)cc2Cl)=O)C1 Cc1ccc(C(N2CCN(CCN(C(=O)CC3(C)CC(F)(F)C3)C)CC2)=O)n1C C(=O)(C1=NOC2(CCC2)C1)NC(C1CCN(C(c2cccc(OC)c2C)=O)C1)C N1(C(COCCC)=O)CCN(C(=O)CCCCC(=O)NC)CC(C)C1 c1(C(=O)NC2(C(=O)NCCC3CCCC3)C(C)C2)[nH]nnc1CN c1(NC)cnc(C(N2CC(C)(CC(=O)Nc3ccc(C)nc3)C2)=O)cn1 N1(C(C(CC=C)NC(C)=O)=O)CCCOC(CC)C1.C1(C=O)(C(N)=O)CC1.N C(=O)(C1=CC2CCCCCC12)NC(C)CCCNC(=O)COC1(C)CCOCC1 C1(C(=O)NCCCCN(C(=O)CC2CC(C)(C)CO2)C)CCN(C)C(=O)C1 c1(N2C(C)CC(NC(=O)CC3OCCC3(C)C)CC2)nc(Cl)nc2[nH]ccc12 N1(C(C(COC)(F)F)=O)CC2CC(NC(C3CCCC3c3nc(S)n[nH]3)=O)C1C2 N1(C(CCCSC(C)(C)C)=O)CC=CC(NC(=O)C(c2ccc(F)cc2)(C)C)C1 N1(C(CC=CCNC(C2(SC)CC2)=O)=O)CCn2c(C)cnc2C1 C1(CNC(C=CC(C)(C)NC(c2sccc2CO)=O)=O)CC2CC1CC2O CN1CCN(c2ccccc2C(=O)NC2CCC(NCc3csc(Br)n3)C2)CC1 C(=O)(C(F)C(F)(F)F)NCC1(C)CCCN1C(=O)CCc1cncs1 c1(CN2CCC(NS(CC)(=O)=O)CC2)ccnc2c(OCC(F)(F)F)cccc12 N1(C(C2CC(SC)C2)=O)CCC=C(C(=O)NC(c2ccncc2)C)C1 N1(C(CC=CC)=O)CCC2(CCCCC2NC(=O)C)C1.C1(CC=O)CCCC1 c1(SC)ccc(Cl)c(C(=O)NCCN(C(C2CC2(F)Cl)=O)C2CC2)c1 Nc1c(C(N2CCC3(CCC3)C(NC(c3cn[nH]c3)=O)C2)=O)cc(F)c(F)c1F CC1(C)CC(C)(C(=O)NCC2(CO)CC3CC3C2)CN1C(c1csnn1)=O C1(NC(=O)CCN2C(=O)CNC2=O)CC2CC1CN2C(c1ccccn1)=O C=CCC(F)(F)C(=O)NC(CNC(C1CC(OC)C(OC)C1)=O)CC(C)C CC(C)(C(=O)NNC(=O)c1nccs1)n1cc(-c2ccccc2)nn1 c1(NCCCC(CCCC)CC)ccc(S(=O)(=O)NCc2ncoc2C)cc1Br C12(C(=O)NCc3c(COC)noc3)COCC1CN(C(=O)CS(=O)CC)C2 N1(C(c2[nH]cc(C(C)(C)C)c2)=O)CCOC(CNC(c2cc(O)ncn2)=O)C1 N1(C(C2C(C=C)OCC2)=O)CCc2ccccc2C1CNC(=O)CCSCCC Cc1nn(CC(N2CCC(NC(c3cnc(Cl)c(Cl)c3)=O)C(C)C2)=O)c(=O)n1C N1(c2c(C)cccc2)C(=S)NC(c2ccnn2C2CC2)C2=C1C(C)(C)NC2=O N1(C(COC)=O)CCC2(CNC(c3nc4nccc(C)n4n3)=O)CCCCC12 N1(C(CCC(CC)C)=O)CCCCCC(NC(=O)CC(Cl)Cl)C1 C(CC(C)C)(C(=O)NC1CC(C)OC1=O)NC(c1cncc(CC)c1)=O C1(CC(=O)Nc2cc(Br)c(F)cn2)CC2CCC1CC2 N1(c2nc(C)cc(OC)n2)CC2CCCC1C2CNC(=O)Cn1ncn(C)c1=O O=CN1CCN(C(=O)CC2CCCN2C(=O)Cc2cc(F)cc(Cl)c2)CC1 C(C(=O)NOCCC(F)F)C1(N(C(=O)C(C)C#N)C)CC1 Nc1ccc(C(=O)NCC2CC2C)nc1Cl.c1(C=O)cccnc1.N(C)C.N CC(C(F)C(=O)NC1(C2CCCN(C(=O)CCCC3CC3)C2)CC1)C(F)(F)F C#CCC(C(=O)N1CCC(OCC2CC2)C1)NC(C1CC(C)N(C)C1)=O c1(C(CC)(C)C)ccccc1C(=O)N(C1CCN(c2ncc(F)cn2)CC1)C CCCCCC(F)C(=O)NCc1ccnc(OC(C)(C)C)c1 CC1CC(NC(c2cc3sccc3[nH]2)=O)CN(C(=O)C=Cc2cc[nH]c2)C1 C1(CC(=O)NCCCCCC)COCC(C)(C)O1.c1(C(=O)N)cn(C(F)F)cn1 C(C)(C)(C(=O)NCC1CCN1C(C1CC1C(C)C)=O)OC(C)C C12CC(C1)C(C)(C)O2.C1(C=O)CCCC1(F)F.C(CC(=O)N)N(C)CCO.C C1(C(=O)NCC2N(C(C3(CC(C)C)CCCC3)=O)CCC2)CCC(N=[N+]=[N-])C1 c1(OC)cccc(N2CCCOC(CNC(=O)C(F)(F)C(C)O)C2)c1[N+](=O)[O-] C(=O)(C(=O)N(O)C(C)C)NC1CCCN(C(C(C(C)C)OC)=O)C1 C1(CCNC(=O)C2CC2)C2CCC1CN(C(=O)CNc1cncc(Br)c1)C2 C(C1CN(C(C2(O)CCOCC2)=O)CC1C(=O)N(CC(=O)OC)C)=CC Cc1cc(C(=O)N(C)CC2CC2)c2occc2c1.c1(CC(=O)N)ccc(F)cn1 C1(NC(=O)CC23CCCC2C3)(NC(=O)CON)CCOCC1 CCC(C)CC(=O)NCCC1CCN(C(=O)CC2CCN(CC(F)(F)F)CC2)C1 c1(C(=O)OC)cnc(N2CCCC(CO)(NC(c3cnn(C)c3)=O)C2)cc1C N1(C(C2C(C)C2C)=O)CC2CCC(C1)N2C(c1cc(C(F)(F)F)ccc1F)=O N1(C(=O)NCC2CC2C2CC2)CCCCC1c1cn[nH]c1 Cc1ccc(-n2nc(CCn3cncn3)nc2CC2CCCCC2O)c(C)c1 C(=O)(C1=C(C(C)F)N(c2ccc(Cl)cc2F)C(=S)NC1c1ncc(O)s1)OCC C1(NC(C(CC)=CC)=O)CN(C(c2cc(C)nn2C2CCC2)=O)CC1N=[N+]=[N-] c1(C(=O)NC(C)C(C)NC(c2nncs2)=O)ccc2ccc(Cl)cc2n1 C(CN=C(NCC12CCCC1C2)NC1CCCS(=O)(=O)C1)OCC CCCCC(C(=O)NCc1cnc(C)c(C)c1)NC(c1cc(O)cs1)=O C#Cc1cc(C(N2CCC(NC(C3(CC4CC4)CCCO3)=O)CC2)=O)cc(F)c1 c1(NC(C2C(NCc3ccc(C(=O)OC)cn3)C2)=O)ccc(C#N)cc1F C(CCCCC(=O)NC(C)CCC(=O)NC(COC)CCO)=CC C1(O)(CNC(C2(C)ON=C(C)C2)=O)CCN(C(=O)C(F)OC(F)(F)F)CC1 c1(OC)cc(O)ncc1C(N1CCC(NC(C2C3CC(F)(F)CC23)=O)C1)=O C1(NC(=O)NC(C)C(=O)O)CC(=O)N(c2ccc(F)cc2)C1 c1(C(=O)NCC(C)CNC(c2cccc3nsnc23)=O)ccc(O)cc1[N+](=O)[O-] c1(C(N2CCC(O)(C(C)NC(C34CCCC3C4)=O)CC2)=O)cn2ccnc2cn1 C1(CNC(Cn2c(N)ccn2)=O)CCCCC1NC(c1cscc1Cl)=O n1(C(C)C)ccc(=NC(=O)C2(NC(=O)C3=C(Cl)CCCC3)CCCCC2)[nH]1 n1(CC)ncc(C(=O)NC2CCCC2(C)CN(C)C(c2cncs2)=O)c1C C1(C2CN(C(=O)Cn3nnnc3C(C)C)C2)(NC(C2ON=C(CC)C2)=O)CC1 C1(C(=O)NCC(COC(C)C)O)CCCCN(C(=O)CC2CCCC(=O)C2)C1 C=CCCC(C)(C)C(=O)N1CCC(NC(c2cc(F)cc(C)c2N)=O)C(CC)C1 c1(C2(C(=O)OC)CC2)ccc(C(F)(F)F)s1.C1C(F)(F)C2(CCC2)N1 Cc1ncc(CN)[nH]1.c1(Cc2nnnn2CCC2CC2)cncn1C(C)(C)C c1(C(=O)N)coc2ccc(F)cc12.C(CCCC)NC(C1(C)CC1C(F)(F)F)=O Nc1nccn2ncc(C(N3CCOC(CNC(=O)CC4CC4(Cl)Cl)C3)=O)c12 c1(NC(c2ccc3occc3c2)=O)ccc(=NCc2cc3cccnc3[nH]2)[nH]c1 c1(CCNC(c2cccnc2)C(=O)OCC)ccc(Cl)cc1 CC1COCCC1C(=O)NCC1(CNC(c2nc(Cl)cs2)=O)CCC1 c1(C(C)NC(CN(C(c2csc(C)c2)=O)CC)=O)ncc(C)o1 C1(CC)(NC(=O)C#CC2CC2)CCN(C(C2CCC2c2ccc(F)cc2)=O)CC1 C1(NC(C(C2CCOC2)NC(C2CCC(CC)O2)=O)=O)CC12CCCCCC2 N1(C(C(C(C)C)SC)=O)CC2CCC2(CNC(C2(n3cnnn3)CC2)=O)C1 C1(C(=O)NC(C2(O)CCC2)C)(CC)CCN(C(=O)Cc2csc(C)c2)CC1 C1(CC)(NC(=O)CCC2CCN(C(=O)CSCCC(C)C)C2)CCOCC1 CCC(C(=O)NCC1(F)CCN(C(=O)C=NOC)CC1)C(C)O C(=O)(CC(CC#C)NC(=O)C(C)(COC)CC)N1CCN(CCC#C)CC1 C(C)(CNC(C1COC(C)C1)=O)(CC(C)C)Nc1cc(OC)ncn1 N1(C(C2CC(CC)C2)C(=O)NC2COC2)CCC(CO)(Sc2ccccc2)CC1 c1(CC(=O)N(CCNC(c2n(C=C)ncc2)=O)CC)ccc2c(c1)CCCN2C C1(CCNC(C(COC)(C)OC)=O)CN(C(=O)C2=CCCOC2)CCS1(=O)=O C1(C(N2CCN(C(Cn3c(C)nnn3)=O)CC2CCO)=O)CS(=O)(=O)CC12CC2 N1(C(C(C=CC)O)=O)CCC(c2cn(CCCN3CCCC3)nn2)(N(C)C)CC1 N1(C(CC2CCCC(=O)N2)=O)CCC(NC(c2cnc(S)nc2)=O)C(F)(F)CC1 CCCC(CCCNC(=O)C(C)(CO)OC)NC(=O)C(C)=C1CC1 C1(O)(CNC(CCC)=O)CC2CCC(C1)N2C(C1(C(C)C)CCCO1)=O c1(CC(C(=O)Nc2cncc(C)c2)NC(=O)CC(=O)N(C)C)ccc(Cl)cc1Cl Cc1ccc(S(=O)(=O)N2CCCC2C(=O)N(CCON)C(C)C)s1 c1(-c2ccc(NC(c3cc(CC)[nH]n3)=O)nc2)cccc2ccncc12 c1(C(N2CCC(O)(CNC(C3CCN(C(C)=O)C3)=O)C2)=O)occ2c1CCCC2 C(CC1=CCN(C(c2sccc2F)=O)CC1)NC(c1ccc(C(O)CF)cc1)=O C=CCCCCNC(=O)C(c1ccoc1)NC(=O)C(C)COC N1(C(c2ncn(CC)n2)=O)CCOCC1C(N1CCC(c2cnco2)C1)=O Cc1ccc(-n2nc(Br)cc2C(N2CCN(c3n[nH]c(Br)n3)CC2)=O)cc1 N1(C(c2ccon2)=O)CC2CCC1C(NC(=O)C(C1(O)CCCCC1)(F)F)C2 C#CC(C)(C)C(=O)N(CC(C)(C)CNC(c1ccc(C2OCCO2)cc1)=O)C N1(C(C(C)OCCCC)=O)CC=CC(C(N2C3CSCC2C3)=O)C1 N1(C(COC(C)(C)C)=O)Cc2ccccc2CC1C(=O)N=c1cc[nH]cc1 C12(NC(c3cccc(CC)c3)=O)CCC1CN(C(c1c[nH]nn1)=O)C2.C1CC1.C C1(NC(=O)C2=CSCS2)CN(C(c2[nH]nnc2C2CC2)=O)C2(CCOC2)C1 C1(NC(C2CCC(OC)CC2)=O)CCC(C)N(C(c2ncccc2Cl)=O)C1 C(CCCCC(=O)N1CCC(NC(c2ccc(C(N)=O)nc2)=O)C(F)C1)OC Cc1nn[nH]c1C(=O)NCc1cc(C(=O)NC2CC2)no1 CC1CC(C(=O)NC(C)CN(C)C(c2c[nH]nn2)=O)=NO1.c1cccc(F)c1.C c1(C(N(C2CCCN(C(C=CC(CC)C)=O)CC2)C)=O)cc(S(N)(=O)=O)oc1Cl C#CCCCCCCC(=O)N1CC(CNC(=O)Cc2cnn(CC)c2)CC1(C)C CCCC(C)C(C(=O)NN1CCCCCC1)N(CCCSCC)C C1(NC(CCCC(=C)C)=O)COC2(C1)CN(C(C1CCN(S(C)(=O)=O)CC1)=O)C2 c1(OC)nccc(C)c1NC(C1C2CCC(C2)N1C(c1c[nH]nc1OC)=O)=O c1(C(=O)NCC=CCNC(CCC=CC)=O)c(Cl)c2ccc(Cl)cc2n1C CC(C(=O)NC(CNC(=O)CCN1CCOCC1)CC(F)(F)F)C1=CCCC1 O=C1CC(C(=O)NC2COCCN(C(c3cc4ncccn4n3)=O)C2)=CC=N1 C1(NC(CC(CC=C)NC(=O)C=Cc2cnn(C)c2)=O)CCOCC12CCC2 N1(Cc2ccc(OC)cc2)CC2(CC2)CC1C(=O)NCCc1cccc(F)c1 C(C)(C)(CC(=O)N1CCC(C(C)NC(c2cccc(NC=O)c2)=O)C1)OC Cc1ccc(=NCCC(=O)N(CCC(C)NC(=O)C#CC2CCCCC2)C)[nH]c1 C#CCC(O)C(=O)NC(C1(O)CCCCC1)C(=O)NCC(=O)N(C)C C1(C(=O)NC2C(NC(C(=O)NCC)=O)C2)CC1C1CC(F)(F)C1 n1(CC=O)cnccc1=O.c1(C(C)OC)nc(C(=O)NC2(C)CCC2)cs1.N C1(NC(c2sccc2-n2cnnn2)=O)CCSC12CN(C(c1cc(Cl)no1)=O)C2 S(=O)(=O)(c1cc(Cl)ccc1Cl)N1CCCC(C(=O)Nc2ccc(C)cc2F)CC1 C(C(C(C)(C)C)NC(=O)CN(C)CCO)NC(C1C(CC)C1)=O N1(C(c2c(OC)c[nH]n2)=O)CCC2(CC1)CC(C)N(C(=O)C#CC1CCC1)C2 c1(C(C(=O)N(CC(C)O)C)F)ccc(C)cc1.c1(C(C(=O)N)OC)cnn(C)c1 c1(NC(C(COC)NC(C(F)=C(C)C)=O)=O)cnc(Cl)c(C)c1 CC(C)C(C(=O)N1CC(C(=O)N)C(O)C1)NC(=O)C(C)(C)C.c1cnncc1O N1(C(Cc2c(C)nn(C)c2)=O)CC2(CC2)CC1CNC(C1(C)CCCCC1)=O c1(C(=O)NC2(CNC(C3C=CCC3)=O)CCC2)cc(=O)c2ccccc2[nH]1 C1(NC(C2(CNC(=O)C3CC3)CCCCC2)=O)CCc2c[nH]nc2C1 c1(C(N2CCC(NC(CC(CC)C)=O)C2)=O)cc(Cl)c(C)c(Cl)c1 CC1CN(C(=O)CC2(C)CCCCC2)CC(C)C1NC(c1ccc(Cl)nc1N)=O C(=O)(CC=C(Cl)Cl)NCc1c(C2CN(C(CCc3ccn(C)c3)=O)C2)ocn1 c1(C(N2CC(F)C2)=O)ccccc1-n1cncn1.CCS(=O)(=O)NCC(=O)N C(C(=O)OC1CCCNC1=O)(C(C)C)NC(=O)OCC CCCCCCC(C)C(=O)N1CC(C)CN(C(c2ccccc2SC)=O)C(C)C1 N1(C(c2c(C)nc(O)[nH]2)=O)CCN(C(=O)Cc2ccn(C)n2)C2CCC12 Cc1cccc(N)c1C(N1CCC(NC(=O)Cn2cnc([N+](=O)[O-])c2)C(F)C1)=O C1(C(=O)NC(C)CCCCNC(C2CCOCC2)=O)CCCC(=O)N1C N1(C(CC)=O)CCCC(C2CCCN2C(=O)CCN(c2ccccc2)C)C1 CC(CNC(C1C=CCN(C(C2CCCC(CF)C2)=O)C1)=O)S(C)(=O)=O C1(NC(C(C(C)C)SCC)=O)CC2(NC(=O)C=C3CCC3)COC1C2 C(CCC(C)C)(C(=O)NC(C)CCCCNC(C1COC(=O)N1)=O)NC(C)=O C(=O)(C(C)C1=CCCC1)N1CC2(CN(C(C(CC=CC)C)=O)C2)C1 C1(C(=O)NCC2CCC(NC(c3ccncn3)=O)C2)(CC)CC(C)(C)C1 C1(CN(C(C2CC(OC)C2)=O)C)CCCCN1C(C1CCCSC1)=O N1(C(CC2N(C(C(c3ccnn3C)C)=O)CC2)=O)CCCC(C#N)C1 Cc1cc(N)c(F)c(C(=O)NC(CO)C(O)C2CCCCC2)c1F Cc1ccc(Cl)c(CNC(=O)NCc2cc(C)cc(F)c2)n1 C(c1cnccn1)=CC=O.Cn1nccc1C1CC1C(=O)NCC=CC.N S(=O)(=O)(c1ccc(NC2CCN3CCCC23)c(F)c1)N(C1CC(C(N)=O)C1)C CCC(CC)CCC(=O)NC1CCCC1NC(=O)Cc1cn2ccccc2n1 C1(CC(=O)N(c2ccccc2)CC#C)CCCN(C(c2cnn(C)c2)=O)C1 c1(C(N(C(c2csc(COC)n2)C(=O)NCC=C)C)C)cccc(Cl)c1 O=C1CCc2ccc(C(N3CC(NCc4cc(O)ccc4Cl)C(F)C3)=O)nc2N1 N1(C(c2cc(CCC)c(C)s2)=O)CC23CCCC2(C1)CN(C(=O)CCS(C)=O)C3 CC(C)CC(=O)NCCN(CCc1ccccc1)C(c1ccnn1CC(F)F)=O C(=O)(C(F)CC1CCOC1)N(C(C=O)C1CC1)C.N1(C(C)C)CC(C)C1.N CC(C)CC(C)(C)CNC(=O)C(C1CCCO1)NC(=O)CCN1CCCC1=O c1(OC)cccc(CN2CC3CC3(C(=O)Nc3ccnn3C)C2)c1O Cc1cc(NC(=O)NCCC2CCCC(C)C2)c(C)s1 c1(COC(c2cn(C3C(OC)CCCC3)nn2)=O)ccc2c(c1)CCC2 C(=O)(C(CC)C(=O)NC1CCCC1CNC(=O)CS(C)(=O)=O)OCC c1(OC)ccc(OC)c(CN(C)Cc2nc(OC)ccc2F)c1 Cc1cc(=O)n(CCC(N2CCCC(N(C(=O)CC34CC(C3)C4)C)C2)=O)cn1 N1(C(=O)NCC(c2ncc[nH]2)C)CC2C3C=CC(C3)C2(C)C1 N1(C(C2(NC(c3csc(C#N)c3)=O)C(C)CCC2)=O)Cc2cncnc2C1 C1(C2CC2)(C(=O)NCC(C)(C2CC2)OC)CN(C(c2cc(Cl)ns2)=O)C1 c1(C(=O)NC(CSC)C)ccccc1-n1cc(-c2ccc(-n3cccn3)cc2)nn1 N1(C(CCN(C(=O)C(C)C=C=C)CC#C)=O)CC(C)CC1(C)C C1(C(NOCC(CC)C)=O)CN(C(=O)CCOC)CC1(C)C c1(CC)c(C(N2CC(OC)CC2C(=O)NCCC2CCCC2(C)C)=O)ccn1C C1(CNC(CC=C(C)C)=O)CCCCN(C(c2cc(=N)[nH]cc2Br)=O)CC1 N1(C(c2cc(C)ncc2)=O)CCC(O)(C2(NC(=O)CN3CCC3)CC2)CC1 CCC(CNC(=O)C(CO)NC(N)=O)(CC)C(=O)N.C1CCCN1C(C)=O CC(C)(Cc1ccccc1)C(=O)N1CCCC(CNC(C2(C)CCOC2)=O)C1 C1(N(C)CCN2CC3CCC2C3)CC12CCN(C(=O)CC(=O)NC1CC1)CC2 N1(C(C2(CC=C)CCCN2C(=O)CSCC(N)=O)=O)CCCC[Si](C)(C)C1 C1(C2CCN(C(c3cc(F)cc(F)c3N)=O)CC2)(NC(C2(F)C(C)C2)=O)CC1 C1(C(N(CCC(F)F)CC)=O)COCC(C)N1C(=O)OC(C)(C)C c1(OC(Cc2c(C)ccc(C)c2)=O)ccc(C)c(C)c1Cl c1(C(=O)NCC(CCNC(c2ccc(F)cn2)=O)OC)cc2cnccc2[nH]1 c1(CC)cc(C)ccc1NC(=O)CCCCCN(C)C(C1(OC)CCCOC1)=O c1(C=O)ccc(O)c(C(C)=O)c1.C1CN(C(=O)CC2CC2(Cl)Cl)C1.CO.C C=C1CON(C(=O)C(CC2CC(F)(F)C2)CC(C)C)C1.C(=O)C(C)C(C)C c1(CCC)occc1C(N1CCCC1CCNC(=O)C(O)CN1CCCC1)=O C(=O)(C(C)C(C)(C)C)NC12CC(NC(CC=C(C)C)=O)(C1)C2 c1(CC)ccc(C(N2CCCC2CNC(=O)CC(CC)OC)=O)c(C)c1 C1(N(C(CSc2n(CC)c(-c3ccc(Cl)cc3)nn2)=O)C)CC(OC)C12CCC2 C1(OC(C)(C)C)CCN(C(c2ccc(-c3csc(=N)[nH]3)cc2)=O)CC1 C1(C(=O)N(CCC)C2CC2)CC1(F)F.c1ccon1.C(=O)(C)N.C1CC1 C1(C)(CC=O)CC(F)(F)C1.c1ccc(C(N2CCCC2CC)=O)o1.CSC c1(C(N(C2CCCN(C(C3C4C5CCC(C5)C34)=O)CC2)C)=O)cccc(N)c1O N1(C(C(C2CCCOC2)OC)=O)CC(C2(NC(=O)C=CC(F)(F)F)CC2)C1 C(=O)(C(O)C(F)(F)F)N(C1CCN(C(c2cc(Cl)cnc2C)=O)C1)CC#C c1(SC)nccc(=NC2CCC(C(=O)N=c3[nH]onc3C3CC3)CC2)[nH]1 c1(C(=O)NCC2CN(C(C3CC4CCCCC34)=O)C2)cc(O)nc2ncccc12 CS(=O)(=O)CCC(=O)NC(Cn1ccnn1)C(=O)NCCCc1ncco1 c1(C(=O)NC2CCC2CNC(C2CC3CC3C2)=O)ccc([N+](=O)[O-])[nH]1 C(=O)(CC(O)CC(C)(C)C)N1CCCC(O)(CN(C(=O)CCCS(C)(=O)=O)C)C1 c1(C(C(=O)NC(CCNC(C(CC)C)=O)C(C)C)(C)C)cc(OC)cc(OC)c1 N1(C(C(CC)F)=O)CCC(c2nnc(CNC(=O)C(F)C(C)C)s2)CC1 c1(CC)nc(C(=O)NCCNC(c2ccccc2Cl)=O)nn1-c1ccccc1F C(N=c1[nH]nc(O)s1)C1CCC(CNC(C2CC23CC(O)C3)=O)CC1 N1(C(C=C(C)Cl)=O)CCCC(CN2CCN(C(=O)CCc3cc(C)no3)CC2)C1 C1(NC(C(C)C#N)=O)C2CCCN(C(c3cc4cc[nH]c4cn3)=O)C2C1(C)C C1(CNC(=O)CN2CC=CC2)CC2(CO1)CN(C(=O)C1=CCSC1)C2 CCC(CC(=O)NC1CCC1NC(=O)CCCNC(N)=O)c1ccc(C)cc1 C1(NC(c2ccc(OC)cn2)=O)CN(C(c2cc(C)ccc2F)=O)CC12CCC2 C(C1CCCN1)=CC(=O)OCCSCc1ccccn1 C(=O)(C1=CCCCCC1)N(CC(C)C(=O)NCCCC1CCOC1)C CCCCC(F)C(=O)N1CCCC1(CNC(C1CCC1)=O)COC C1(C)(CNC(Cc2ccc(C)c(F)c2)=O)CN(C(c2cccs2)=O)C(C)(C)C1 CC1(C)CC(CNC(=O)C2=C(Cl)CCC2)N(C(C2CCCNC2=O)=O)C1 c12nc(n[nH]1)C(C)N2C(C)CNC=O.c1cc(C)on1.C(C)(C)C.CC c1(C(C(=O)NCCCNC(c2cc(-c3ccccc3)[nH]n2)=O)O)cccnc1 C1(NC(C2(C)CCCN2)=O)CC2CCC(C1)N2C(c1nccc2nc[nH]c12)=O c1(C(C=O)(C)C)cccc(Cl)c1F.c1(C(C)C)cc(C(=O)NCC2CC2)n[nH]1 C1(C)(CNC(c2cccc(CC)c2F)=O)CC(F)(F)CN1C(=O)C(C)C.S CC(=O)C(C)(C)CC(=O)NC1CCCCCC1C(=O)NCC(C)N=[N+]=[N-] C12(CNC(CCC=CCC=C)=O)CC(CN1C(c1sccc1OC)=O)C2 CCCCC(CCCC)C(=O)NC(CNC(C1CCC(=O)N(C)C1)=O)CCCC O=C1CCC2(CCN(S(=O)(=O)CCCS(=O)(=O)NCC3=CCCOC3)C2)N1 CCC1=NN(c2ccc([N+](=O)[O-])cc2)C(=O)C1OCc1[nH]nc(C(F)(F)F)c1C CCCCC(O)CCC(=O)NC(C1(O)CN(C(c2nc(C)ccc2C)=O)C1)C c1(CC(N2CCCC2(C)C)=O)cn2cc(F)ccc2n1.C(C=O)(C1CC1)SC.N c1(OC)cc(C)sc1C(N1CCC1Cc1ccccc1)=O C1(NC(=O)CC2CC=CCC2)COCCC1C(=O)NCC1(O)CCCCC1 O=C1NCCC2CCN(C(C3(c4ccno4)CCOCC3)=O)CC12 C1(CC(=O)N(CCNC(c2nc(COC)oc2)=O)C)COC(C)(C)C1 N1(C(=O)Nc2ccc(N=[N+]=[N-])cc2)CCOc2cccc(F)c2C1 C(CC1=CCN(C(=O)CSC(F)(F)F)CC1)NC(c1cccc2nn[nH]c12)=O C1(CN(C(=O)Cc2ccccc2CO)C)CCN(C(C2(C#N)CC2)=O)CC1 Cc1cccc(OC(C)C(=O)NC(CNC(=O)CCC2CCCC2)C(C)C)c1 C1(C(N(CCNC(C(C)C)=O)C)=O)CC(O)CN1C(c1ccncc1)=O c12cccc(c1)OC(c1cn(CC(C)C)nn1)COC(=O)C2.CCC(C)(C)S C1(C(=O)NCC2CC2Cl)CC12CCN(C(c1cccn3ccnc13)=O)CC2 c1(C(N2CC(CNC(C3(CCC)CC3)=O)C(C)C2)=O)ccn2ncnc2c1 N1(C(C2(CC)CCOC2)=O)CC(CC(=O)N(C)Cc2ccncc2C)C(C)C1 Cc1cc(C(N2CC(C)(NC(=O)C(F)CC3CCC3)C2)=O)on1 CC(C(=O)N(CCCNC(=O)CCc1ncc[nH]1)C)S(=O)(=O)c1ccc(F)cc1 C#CC1(C(=O)NC(CSCC)C(=O)NC2CCOC2(C)C)CCCC1 C1CCN(C(c2ccn(C)c(=O)c2)=O)CCC1(F)F.C(C(=O)N)=CC=CCC N1(C(c2cnn(C)c2C(C)(F)F)=O)CC2CN(C(C3CCC(=O)C3)=O)CC2(C)C1 c1(C(=O)NCCCN(C)C(C2CCN3CCOCC23)=O)cccn2nccc12 N1(C(c2c(C)cn(C)n2)=O)CCCC(C)C1.C(O)(C(F)(F)F)C1(C=O)CCC1.N C(C1=NOC2CC12)(c1nnnn1CC(F)F)NC(COC)(C)C c1(NC(c2cncc(-c3ccc(OC(F)F)c(F)c3)n2)=O)cnc2sccc2c1 c1(OC)ccccc1C1CC1C(=O)NCc1cn(C(C)CO)nn1 C1(C)CCCC(C)(C)C1.CN1CCOC(C(=O)NCCn2cc(C(=O)N)cn2)C1 O=C(CS(=O)C(F)(F)F)NC1CCC1CNC(c1cc2c(s1)CCCC2)=O Cc1oc(C(=O)NC2CC(C)CN(C(=O)CC(C)C)C2)cc1S(C)(=O)=O C1(NC(c2c(C)cccc2Cl)=O)CC2CCC(C1)N2C(c1cc(Cl)cnn1)=O N1(c2snc(C(=O)OC)n2)CCC2(CC1)CC(C)N(C(=O)CSC1CC1)C2 c1(CC(=O)NCCCN(C(C(CCC)=CCC)=O)C2CC2)ccccc1Cl.N C1(CNC(CCN2CCN(CC)CC2)=O)CCC(C)N(C(c2cnc(O)s2)=O)C1 c1(C(=O)NC(CC)CNC(C2CC(OC)C2)=O)cn(C)c(=O)cc1OC C(CCCCC(=O)N1CCSCC1CCNC(C1OCCC1C)=O)OC c1(C(=O)OC(C)(C)C)cc(NC(=O)C(CC(F)F)c2ccc(F)cc2)ccc1F C1(CC(=O)NC2CCN(C(CNC(=O)C3CC3)=O)C2)COC2CC1C2 Cc1cc2nc(NC(=O)N(C)C(c3ccc(-c4csc(Br)c4)o3)=O)sc2cc1F c1(CC(=O)NCC(CNC(C(C(C)C)O)=O)F)cc(Cl)c2c(c1)OCCO2 C1(NC(C=CCCC)=O)CN(C(c2nc3ncccn3n2)=O)CC12CCOCC2 C(CC(N)=O)(C(=O)NCc1cnc(C)s1)NC(CCc1onc(C)n1)=O C=CCC(CNC(=O)C(C)(CC)OC)C(=O)NC(C)COC(F)(F)F C(=O)(CC(C(F)F)N1CCOCC1)N1CC(CCNC(C2(C)C=CCCC2)=O)C1 Cc1ccnn1CC(=O)NC1CCC(NC(=O)CCC2CCCCO2)C1 N1(C(Cn2c(C)ccn2)=O)CCCCC1C1CCN(C2CC2)C1 Cc1cc(F)cc(C(=O)NC(C)CNC(=O)C(c2ccc(F)cc2)(C)C)c1C c1(CN2C(CNC(C(c3cccc(Cl)c3)CC)=O)CC2)cc(Br)ccc1F c1(OC)ccc(C(=O)NC(C)(CNC(=O)C(C)N(C)C(C)=O)CO)s1 c1(C(=O)NC(C)C(C)(C)NC(=O)COC2CC(F)(F)C2)cc(O)ncn1 c1(COC)cccc(C(=O)NCC2(F)CCC2)c1C.C1(C(=O)N)CCOC1 c1(CNC2C(C(=O)N(c3nccs3)CCO)C2)ccc(Br)cc1 N1(C(C(CC(C)C)C)=O)CCN(C(=O)CN(C)CCO)CCC1C C(=O)(C1CCCc2nncn21)N1C2CN(C(CNC(=O)C3CC3)=O)CC1CC2 c1(CC)nc(C)ncc1C(=O)NC(C)CC(C)NC(c1cc(N)cc(O)n1)=O c1(C=O)ccccc1S(C)(=O)=O.C1(CC)CCC(C(=O)NCC2CCCC2)O1 N1(C(Cc2ncc(C)o2)=O)CCC(C(N)=O)(N(C)C)C1 C(=O)(CCCCCCC)N1CCN(CCCCCC=C)CC1 C1(NC(CCC(CC)OC)=O)CCCCC12CCN(C(c1ccccn1)=O)CC2 c1(CC(=O)NC2CN(C(CC(C=C)C)=O)CC23CCC3)coc2cc(Cl)ccc12 c1(CC(=O)N(C(C)C(=O)NCCCC2CCOC2)C2CC2)ncccn1 Cc1nc2ncnn2c(C)c1CC(=O)NC1CCCN(C(C23CC2C3)=O)C1C c1(C(=O)NC(CCN(C(c2ccc(NC)cn2)=O)C)C)cccc2nn[nH]c12 C1(C)(CNC(C=C2CCN(C)C2)=O)CCCC1.C1(C=O)COCC1C(N)=O c1(C(N2CCN(C(c3n(C(C)C)cnc3)=O)CC2)=O)cc([N+](=O)[O-])c(O)cc1N C(CCCCC(=O)NCC12CC(CO1)N(C(c1cc(F)ccc1N)=O)C2)N(C)C CC1CCC(CO)(NC(=O)CSCCNC(C2(O)CCCC2)=O)C1 c1(N2C(C)CN(C(c3coc(C(F)F)n3)=O)CC2)nc2ncc(Cl)cc2o1 N1(C(c2cc(C)ncn2)=O)CCCC(C)(NC(=O)CCCC2CCCCC2)C1 c1(CC(=O)NC(CC=C)CNC(=O)C(C)c2ccon2)ccc(Cl)cc1C C1(C#N)(C(=O)NCCCCCCNC(C2(F)CCCN(C)C2)=O)CC12CCCC2 CC1CCCC1(C)Cn1cc(-c2cccc(N)n2)nn1 C1(c2cn(C)nc2)C(NC(C2SCCCS2)=O)CC(=O)N1C1CC1 Cc1cncc(CCC(N2CCCCC2CCN(C)C(C2CC2C(F)F)=O)=O)c1 c1(C(N2C(CNC(c3ccc(C)cc3)=O)C(C)CC2)=O)cccc([N+](=O)[O-])c1 c1(C(=O)N)ccc2c(c1)NC(=O)CS2.CC(CC(=O)N(C(C)C1CC1)C)C(F)F N1(C(C(C=CC)O)=O)CC(C2CCCN(C(c3nn(C)nc3Br)=O)C2)C1 C1CN(C(=O)C(c2ccc(F)cc2)C)C2(CCC2)C1.C(C)(C)(CC(=O)N)OC.C C1(C(=O)NC2CCN(C(C#CC(C)C)=O)C(C)C2)CCCCC(C)(C)C1 c1(N(C)C)ccc(NC(C2CC(F)(F)C2)=O)cc1F.C(=O)(CC)N.C(=O)CO CCC(C)CCCC(=O)N1CCOCC1c1cn(-c2cccc(Cl)c2Cl)nn1 N1(C(C2C(C)C2)=O)CC2(C1)CN(C(C1(C3CCCO3)CCCC1)=O)CCO2 c1(C(=O)COC(c2csc(Cl)n2)=O)cccc(O)c1 C12(C(=O)NC3CN(C(CCC4N(C)CCC4)=O)CC34CC4)CCC(C)(CC1)OC2 C1(C(=O)Nc2c(C(=O)OC)cccc2F)CCN(C(=O)CCBr)C2CCOC12 N1(C(c2noc(CC)c2C)=O)CC(NC(=O)COCC(C)C)CC(F)(F)C1 c1(OCC)ccnc(NC2CCCCC2NC(=O)CC2CSCCS2)n1 CN1CCN(C(c2ncc(Cl)cc2O)=O)C(CNC(C2COCCN2C)=O)C1 O=C(CCC=CBr)NCC1(F)CC(CNC(=O)CC2C=CCC2)C1 c1(CCNC(N(CC=C)CC2CCCO2)=O)ccc(OC)cn1 c1(C(=O)NCC(CC)NC(C2(C(F)F)CCCC2)=O)cc(C2CC2)ccn1 c1(C=O)coc(S(C)(=O)=O)c1.c1(COC)nc(C)ncc1C=O.CCCO.N c1(C(N2CC(F)CC(NC(CC(C(C)C)C)=O)C2)=O)ccc2ccc(Cl)cc2n1 C(=O)(C(F)(F)C(O)C(C)C)N1CCC(NC(CC=C(C)C)=O)C(CO)C1 Cn1nc(C(=O)NC2CCN(C(=O)C=C3CCCC3)CC2F)c2c1CCC2 C1(C(N(C2CCCCC2)C)=O)C2CN(C(=O)CN3CCCCC3)CC12 C1(C(=O)NC2CC(NC(CC(C)(O)c3ccccc3)=O)C2)CCCCCC1(F)F C1(C(N(C)CC2CCCN2C(c2cnoc2C2CC2)=O)=O)CN2CCC1CC2 c1(C(=O)NC2CN(C(C3C(=C)CC3)=O)CC2F)cnc2sc(C)cn2c1=O C(=O)(NNC(=O)C1CC1c1ccccc1OC(F)F)N(C)CCn1ccnc1 c1(C(N(CCCN(C)C(C2SCCCS2)=O)C)=O)ccc(OCCO)cc1 Cc1c(C(C2CCC2)NC2CCC(Cc3ccccc3)C2)cnn1C C1(NC(C(CC)F)=O)CCCC(NC(c2nc(Br)sc2C2CC2)=O)C1 O(S(=O)(=O)N1CCC(C)(C)CC1)c1ccc(C(CC)=O)c(F)c1 C1(NC(Cc2cccc(C)c2)=O)CCC(O)CN(C(c2cc(O)cc(=O)o2)=O)C1 C1(C(N(C(c2ccccc2)C)C)=O)CCN(Cc2cccc(OC(F)F)c2)CC1 C=CC1(C(=O)NCCc2cnccn2)CCN(C(c2ccn(C3CC3)n2)=O)C1 C(=O)(C(C)C(O)C(C)CC)C1CCC(C)NC(=O)C(CC=CC)NCC1 CCCCC(O)CC(=O)NCCCNC(C1CC2(C1)C(F)(F)C21CC1)=O c1(C(N(CC(C)NC(=O)Cn2ccnn2)CC)=O)cc(OC)ncn1 c1(CCC(=O)NCC(CN(C(C(C)OCCC(C)C)=O)C)C)ccc(F)nc1 N1(C(c2c(C#C)cnn2C)=O)CCC2(CCCCC2NC(=O)Cn2ncnn2)C1 C1(CC#C)(C(=O)NCC(O)C=O)CCN(C(=O)C(c2ccc(Cl)cc2)=O)C1.N c1(C(N2CCCC(NC(C3(CC#C)CCCCC3)=O)C2)=O)cccn2ccnc12 c1(OC(C)C(N2CC(C(C)(C)O)C2)=O)cccnc1.C(=O)C(F)CC1CC1.C C(C)(N=c1[nH]c(C#N)c(Cl)s1)C1CCCN(C(C(C)Cc2cnn(C)c2)=O)C1 C1(C)(CC)CC(C(=O)NC(C)C2CCC2)CCO1.C1(C=O)CCC(=O)N1C.N N1(C(c2c(OC)ccc(C)n2)=O)CCN(C(c2occ(C)c2C)=O)CC1C N1(C(C2(C(C)(C)O)CC2)=O)C2CCC1CN(C(C1(C)CC=CCO1)=O)C2 C(=O)(C1=NOC(C)C1C)N1CCC(C(C)NC(c2cncc(C(C)C)c2)=O)CC1 C(CN=C(NCc1ccc(C)cc1)NCC1CCCC(F)C1)N(CC)CC C1(C(=O)NCC2CCC2)CC(=O)N(c2ccccc2Br)C1.C1(C=O)CCO1.N c1cc([N+](=O)[O-])ccc1C(N1CC2C(C(N)=O)C2C1)=O.Cn1cnc(C=O)c1.N c1(C(N(C2CN(C(C=CSC)=O)CC2F)C)=O)ccc(F)c2[nH]ccc12 c1(C(=O)NCCC(C)NC(c2c(C)[nH]c(=N)s2)=O)cc(O)nc(O)n1 N1(C(C2CC3C=CC2C32CC2)=O)CCC2(CC1)COC(C)C2.C(=O)C(F)(F)F.N c1(CC)[nH]c(C(=O)NCCC(C)NC(c2cn(CCN(C)C)nn2)=O)nc1Cl c1(C(=O)NC2CCC(NC(C3CC34CCOC4)=O)CC2)cc2scnc2[nH]1 c1(C(=O)NCC(CN(C(CC)=O)C)(C)C)ccnc(C(C)(C)O)c1 N1(C(C2CC(C)(C)C2)=O)CCC2(CC(C(=O)N)C2)C1.C1(CC2CC2)CCC1 N1(C(C=C(CCC)C)=O)CCC2(CCC2)C(NC(c2coc(OCC)n2)=O)C1 C1(C(N2CC(CN=c3[nH]cnc(=N)[nH]3)OCC2)=O)CC2CCCCCCC12 c1(C=O)ccc(S(N)(=O)=O)o1.C1(N(C(COCCN(C)C)=O)C)CCCCC1 c1(C(N(CC(C)C)C)=O)cccc2c(C)c(C)[nH]c12.C1(CC)CC1C(=O)N C1(NC(CSCC#C)=O)CCC(N(C(=O)CCCSC)C)CC1.C(N)(=O)N c1(CC)c[nH]cc1C(=O)NC(C(=O)NC1(C)CC1)c1cccs1.C1CCC1 c1(N2CCC(C(=O)Nc3c(CC)nc[nH]3)CC2)ncnc2c1ccn2C c1(CC)cccc(C(=O)NCC(CC)NC(=O)Cc2nocc2C)n1 CCC(C)C(=O)NCC(=O)N(CC(O)CNC(c1ncn(C)n1)=O)C c1(CNC2(CC(=O)Nc3cccc(F)c3Cl)CCC2)ccc([N+](=O)[O-])o1 N1(C(C=C(C)C(C)C)=O)CCCCCC1CNC(c1conc1C(C)(C)C)=O N1(C(C2C(C(=O)OC)C2)=O)CCC(OCC(=O)N(C2CCC2)C)CC1 C1(CC=C)(NC(=O)CS(C)(=O)=O)CCCN(C(c2cc(C)ccc2O)=O)C1 CC1CCCCC1(CNC(C1CC12CCCC2)=O)NC(c1cnns1)=O C1(C(=O)NCCCN(CC(C2CCC2)OC)C(C)C)CCC(O)CC1 C1(NC(C)=O)CN(C(c2coc(C3CCC3)n2)=O)CC1C c1(C(=O)NC2C3N(C(c4cnc(C)n4C)=O)C(CC3)C2)cc2c([nH]1)CCCC2 C1(NC(c2n(CCC)ncc2)=O)CC(C(=O)NC2(C(N)=O)CCC2)CC1O C1(C(=O)NC2C(CC=C)CCC2)CCCN(C(C2CC3(C2)CC32CC2)=O)CC1 CC(CCCC(=O)Nn1ccccc1=O)NC(=O)CN(C)C(N)=O C(C(C)C)(C(O)C(=O)NC(CCC(=O)NCc1nc(C)co1)C(C)C)OC N1(C(CN(CC)CC)=O)CCCC2CN(C(=O)CC3=NN(C)C(=O)C3)CCCC12 c1(CC(=O)NC(CN(C(C2C3CC4C(C3)C24)=O)CC)C)ccc(O)nc1 N1(C(C(CCF)NC(C2ON=C(CC)C2)=O)=O)CC2(CC=CC2)C1 C12(CSC)CC(C(=O)NCCC3CCCN3C(=O)C(C)SC)(CO1)C2 C1(C(N(C(C)C)CCNC(c2ccc(Cl)c(F)c2)=O)=O)CC1C1CCOCC1 N1(C(Cn2nnc(C)n2)=O)CCN(C(=O)C(F)C2CC2)C2(CCC2)C1 C#Cc1cccc(NC(C2(C)CCN2C(=O)Nc2cc(Cl)cc(Cl)c2)=O)c1 C1(C(C)(C)O)CCN(C(C2CC=CCN2C(=O)CC2CC3CCC2O3)=O)CC1 c1(C(=O)NC(C)C(C)NC(=O)Cc2cn[nH]c2)ccc(Cl)cn1 C1(C(N2CC(F)CC(NC(c3csc4cncn34)=O)C2)=O)CCC(=C(F)F)CC1 c1(C2CCN(C(C#CCC)=O)C2)ccc(NC(=O)O)cc1F.C(C)(C)C.C(N)=O CCCCS(=O)(=O)CC(=O)NC1CCN(C(c2cnc3scc(C)n23)=O)CC1O CC(C)C(CNC(=O)C1=CCCCC1C)C(=O)Nn1cnnc1 N1(C(c2cnc(C(C)C)n2C)=O)CC(C)N(C(=O)C2=CCCS2)CC1C CC(C(=O)NCC1CCCN(CC2CN(C(=O)C3CC3)C2)C1)C(C)(C)C c1(OC)cn(CC(=O)NC2CCSC23CN(C(=O)CC(=O)OC)C3)c(C)cc1=O CC1C(CO)OCCN1N(C)CC(=O)N(CC(F)(F)F)CC1CC1 N1(C(CSCCCC)=O)CC2CCCCC2(CNC(c2cnc[nH]c2=N)=O)C1 C12(C(=O)N)CC3CC(C1)CC(F)(C3)C2.C1(C(=O)NCCCC)CC12CCOC2 c1(OC)ncc(Br)c(=NCC2C3CN(C(C4CCc5nn[nH]c5C4)=O)CC23)[nH]1 C1(CCC(=O)NCC2(O)CCCOC2)CCCCN1C(=O)CC=C(Cl)Cl n1(CCC(=O)NC2C(NC(C3(F)C(C)C3)=O)C2)nnc2ccccc2c1=O C1(C(=O)NCCCCNC(=O)Cc2cnoc2)CCN(c2ccc(Cl)cc2)C1=O c1(OC)ccc(C)c(CC(=O)NCc2ccc(C#N)cn2)c1 N1(C(Cn2nc(C)c(Cl)c2)=O)CCC(CO)(CNC(C2COCCC2C)=O)CC1 N1(C(c2c(C)c(F)cnc2)=O)CCN(C(C2CCCC2O)=O)CC(C)C1 Cc1cc(C)c(C)c(C(=O)NC(C)CN(C(=O)C(F)=CCCF)C)c1C C1(C(=O)OC(C)(C)C)CC(F)CN1C(C1CC=CCC1)=O.C12CC(C1)C2.N C(CC)(CCCC)(c1n(CC=C)nnn1)NCC(=O)N(C(C)(C)C)C.CC c1(CCC(=O)N(CCOC)CCNC(C2C=CCCC2)=O)ccc(C)nc1 c1(-c2c(NC(c3cccc(=O)o3)=O)ccs2)ccc(COC2CCNCC2)cc1 Cc1ccnc2nc(C(=O)NC(C)C(CO)NC(c3scnc3C(F)F)=O)nn12 C1(CNC(C(C=C)OC)=O)CCN(C(C2(OC)CCCSC2)=O)CC1(F)F Cc1cc(NC(c2csc(NC(c3cc4ccccc4[nH]3)=O)n2)=O)c(C)cc1O C1(O)(CN(C(=O)CN2CCNC(=O)C2)C)CCCN(C(=O)CS(C)(=O)=O)C1 c1(OC)cc(Br)c2c(c1)CN(Cc1cn(CC3(O)CCC3)nn1)CC2 C12(NC(C(N)=O)=O)CN(C(=O)Cc3ccc4ccccc4c3)CC1CS(=O)(=O)C2 Cc1cc(CNC(=O)NCCC(C)N(C)C)c(C)c(C)c1 Cc1ccc(CC(N2CCC2C(=O)Nc2cccnc2-c2ccncc2)=O)cc1 N1(C(c2csc(C(F)(F)F)n2)=O)CCCN(Cc2cncc(Cl)c2)CC1 N1(C(=O)C=Cc2ccco2)CCOC(CCCNC(C2(C3CC3)CCCO2)=O)C1 N1(C(CCOCCN(C(C(C)n2ccnc2)=O)C)=O)CCCC(CCO)CC1 c1(C(N2CC(O)CCC2C(=O)OC)C(=O)NC)cc2cc(Cl)ccc2s1 c1(C(=O)NCCCC=C)ccc(S(C)(=O)=O)s1.c1(C=O)ccc(F)c(F)c1.N C(=O)(CC1OCCc2ccsc21)NCCC1CCN(C(CC(CC)OC)=O)CC1 C(CCCC(F)(F)F)NC(CCCNC(C1(CC=C)CCCC1)=O)=O c1(OCC(=O)NCCCCCNC(c2c(CC)con2)=O)ccccc1C C1(C(N(C2CN(C(C3CCC3c3nc[nH]n3)=O)C2)C)=O)CCCC1(F)F c1(OC)ccc(C)nc1C(N1CCC(NC(=O)COCCC(C)C)C12CC2)=O CCC(C)C(O)CC(=O)N1CC(F)(CNC(C2(C(F)F)CCN(C)CC2)=O)C1 O=C1CC2OCCC2(C(=O)NC2CCCC2NC(=O)Cc2ccoc2)CN1 C(=O)(C(F)C(C)CNC1CCCC1C(=O)OC)NC Cc1cc(C(N2CCC3CC23C(=O)N(C)Cc2ncccn2)=O)c(C)n1C C(C)(CC(F)(F)F)NC(c1cnccc1C(F)(F)F)=O.C1(C=O)CC(O)C1 C1(CC)CC(O)CN1C(C1CCN(C(c2cnn(C3CC3)c2)=O)C1CC)=O N1(C(c2c(C)nns2)=O)CC=CCC1C(=O)NCC1CCOC1 c1(CC(=O)NC2CC3CN(C(=O)CC4NC(=O)NC4=O)CC23)nc2ncccn2n1 C1(CC)(CC)CC(NC(c2cc3cscc3s2)=O)CN1C(=O)C(C)OC c1ccc2c(=NC3CC4CCC3C4)[nH]c(N(C)CCOc3ccccc3)nc2c1 N1(C(CCCNC(CCC2C(C)(C)C2)=O)=O)CCCC12CCOCC2 C(=O)(C1CCCc2cncn21)N1CC2CN(C(c3c(C)cc(Cl)cc3)=O)C2CC1 c1(C(N2CC(F)(CNC(c3onc(C)c3C)=O)C2)=O)cc(O)c2cnn(C)c2c1 C(=O)(C(=O)N=S(C)(C)=O)NC(CCNC(C(C(C)c1ccccc1)O)=O)(C)C C(=O)(C(F)(F)C(O)C(C)C)N1CC(C(C)NC(CC(c2ccccc2)OC)=O)C1 c1(NC(=O)Cn2ccnc2)ccc(-c2cnn(CC)c2)cn1.c1ccsc1 N1(C(CNC(C)=O)=O)CCC(C)C(NC(=O)COCc2ccco2)C1C c1(CC=O)ccc2c(cnn2C)c1.N1(C(C(C)=CC)=O)CCC(CO)(C)C1.N Cn1cnc2c(NCC34CC(C(F)F)(CO3)C4)[nH]c(=NCc3cnc[nH]3)nc12 CCC(O)C(F)(F)C(=O)NCC1(OC)CCN(C(=O)CC(CC)C2CCC2)CC1 N1(N(C2C(C)CCNCC2)C2(C(F)(F)F)CCC2)Cc2ccccc2C(O)C1 C1(CCC=C)(C(=O)NCC2CC2)CN(C(C2CCOC2C(C)C)=O)C1.C Cc1cc(F)c(C(N2CCC(NC(C3CC(C(C)C)C3)=O)C2)=O)cc1F C12(NC(CN(CC)CC)=O)CCC(CN(C(c3cc(F)cc(Br)c3)=O)C1)C2 C(=O)(CC(C)CC(C)C)NC1C(NC(COc2ccc(C)cc2)=O)CCOC1 c1(C=O)ccccc1.c1(C(N(CC)CC)=O)sccc1C(F)(F)F.C(C)C C1(CC)CN(C(C2CC2(F)F)=O)CCC1NC(=O)CC12CC(C1)C2 C(c1ccccc1C#N)=CC(=O)NC(C1CCN(C(c2ccc(Cl)cn2)=O)C1)C CCC(C(=O)N(C)CCNC(=O)C(O)Cc1cnc[nH]1)C(C)(F)F c1(CNC2C(C(=O)NCC3(C)CCOCC3)CCC2)cc(F)c(Cl)cc1Cl C1CC12CCN(C(c1cnn(CC(F)(F)F)c1)=O)CC2.O=C(COC1CC1)N C(=O)(C1=C(NC(C2CN(C(=O)C(F)(F)Cl)CCO2)=O)CCC1)OCC c1(C(=O)NCC(CNC(c2c(CC)n(C)cc2)=O)CO)c[nH]c2cc(Cl)ccc12 N1(C(C(C)NS(CCC)(=O)=O)=O)CCC(NC(c2sccc2C#N)=O)CC1 CC1CN(C(=O)CSCCCc2ccccc2)CC1C.c1(C=O)coc(Cl)n1.N c1(C(N(CCCNC(C2(C)CCOC(C)C2)=O)CC)=O)cc[nH]c2nccc1-2 C(=O)(C(C)(CC)CO)NCCC1(O)CN(C(c2c(OCC)n[nH]c2)=O)C1 C(C(C)(C)CN=c1[nH]c2c(c(=NCCC3CCS(=O)(=O)C3)[nH]1)CCC2)N(C)C c1(CN2CC3C(C(N(CCn4cccn4)CC)=O)(C3)C2)cc(Br)c(C)cc1F CC(C)CC(F)C(=O)NC1CC(=O)N(C2CN(C(c3cnc(O)s3)=O)C2)C1 c1(C(N2CC(CNc3nccc(C#N)n3)OCC2)=O)c(F)ccc(O)c1F Cc1cc(O)ccc1C(=O)NC1CCCC(NC(=O)CC2(C3CC3)CC2)CC1 c1(OC)ccc(CC(C)C(=O)NCC(C)C2CC2)cc1.C(=O)C=C(C)Cl.N C#CCC(C)(CC)C(=O)NCC(CC)NC(C1(c2cccc(C)c2)CCC1)=O C(C)(C(C)(C)CC)NC(C1(CC=C)CN(C(=O)C(COC)CC)C1)=O CC1CCN(C(C2CCCC(=O)N2C)=O)C(C)C1NC(C1CC2CC1C1CC21)=O CC1CN(C(c2cn(C)c(C(F)F)n2)=O)CCN1C(=O)CCc1cc(Cl)cs1 CN1CCC(C)(C(=O)NC2CCC2)C1=O.c1(C=O)cnc(C(F)(F)F)c(F)c1 C1(NC(c2cn(CCF)nn2)=O)CCCC12CN(C(C13C=CC(CC1)C3)=O)C2 c1(C(=O)NCC2CCC(NC(C3CC4CCC3O4)=O)C2)ccn2cnnc2c1 Cc1cc2cc(C(=O)N)oc2cc1C.CC(C)CN(C(=O)C(C1CC1)N(C)C)C Cc1nc2c(C)cc(C(=O)NCC3CCN(C(C4CC45CCC5)=O)C3)cn2n1 C=CCC(Cc1ccccc1)C(=O)NCC1(NC(=O)C)CCC1.C1CC=CC1 c1(C(=O)NC23CCC(CN(C(c4cccnc4)=O)C2)C3)ccnc2ncccc12 N1(C(C2OCC(C)C2)=O)CCN(c2nc(C(F)(F)F)cs2)CC1 N1(C(Cc2cc(OC)c(C)cc2)=O)CCCCCC(N=c2[nH]nc(C)s2)C1 CC1(C(=O)NC2C=CCN(C(=O)C=C3CCC3)C2)CCOc2ccccc21 [N-]=[N+]=Nc1ccc(C(=O)NC2CC2NC(c2cnn(CC(F)(F)F)c2)=O)cc1 c1(CC)nn[nH]c1CNC(C1(NC(C2C=CCC2)=O)CC(F)C1)=O C1(C#N)(C(=O)NC2C(NC(CCc3scc(C)n3)=O)COC2)CCN(C)CC1 C1(C(=O)NCC2N(C(c3c(C(=O)OC)nccn3)=O)CC2)CCN(OC)CC1 Cc1nccnc1C(N1CCCC(CNC(c2c[nH]nc2C2CC2)=O)C1)=O C(CCN=c1[nH]nc(C(N)=O)s1)N(C)C(c1cn(C2CCOC2)cn1)=O c1(NCCC(CC)C)ccc(S(=O)(=O)N2CC(O)C(C)(C)C2)cn1 CCC(CC)CC(c1nnnn1C)NCc1cccc(CN2CCN(C)CC2)c1 c1(C(=O)NCC(C)N(C)C)ccc(Cn2cc(C)nn2)o1.C1(N)CCCCO1 N1(c2nccc(OC3C(C)CCCC3)n2)CCCC2(CCCCCC2)C1 N(C(=NCC(O)COCc1ccccc1)N1CC(F)(F)C(F)(F)C1)C(CC)CC c1(C(=O)NCCC(C)NC(Cc2ccc(C)cc2)=O)cnn2c1OCC(F)C2 N1(C(C(C)CS(C)=O)=O)CC2(CCN(C(C3(C(C)(F)F)CCC3)=O)CC2)C1 Cc1ccc(F)c(C(=O)N(CC(C)NC(=O)CC(c2c(C)noc2C)C)C)n1 N1(CC)CCCC(ONC(=O)C=CCNC(=O)Cc2cnn(CC)c2)C1 N1(C2(C(N(CCCNC(=O)Cn3ccnn3)CC)=O)CCC2)CCOCC1 c1(OCCN(C)C)ccc(CCNC(=O)CC2CCC23CNC3)cc1 C#Cc1ccnc(C(N2CCC(N(C(C3CC34CC4(F)F)=O)CC)CC2)=O)c1 CCCCCCC(C)C(=O)NCC1C(CC)CCN1C(c1ncn(C(C)C)n1)=O C1(NC(C=CCC)=O)CCC(N2CCN(C(c3n[nH]cc3Cl)=O)CC2)CC1 N1(C(C(C)C2CCC2)=O)CC2CC1CN2C(c1cc(-c2cccc(F)c2)on1)=O C1(NC(C(CNC(C(C(C)O)N(C)C)=O)O)=O)CNC(=O)C1(C)C CC1(C(=O)NCCc2cn(CC3CC4CC4C3)nn2)CCOC1 C(=O)(C1=CCC(NC(c2conc2C)=O)C1)N(C(C(=O)OC)C)C C1(CCC)CCN(C(C2COCC2NC(=O)C(CC)SC)=O)C1 C1(CNC(CC(C=C)CC)=O)CC12CCC(C(C)(C)CC)CC2 C1(CNCC)CC2(C1)CC(F)C2.Cc1nc(C2CC2)sc1CC=O.C1CC1 c1(C(=O)NC(C(C)C)CNC(=O)C=Cc2cocn2)cnc2scnc2c1 CC1CCCN(C(C2CC3CC3N2C(=O)CSc2ccc(F)cc2)=O)C1 C12(C(N(CCCC(=O)NC3(COC)CC=CC3)C)=O)CCCC1OCC2 C1(CN(C)C(c2cnn(-c3ccccc3)n2)=O)COCCN1C(=O)C.C1CC1.S N1(C(c2c(C)ccs2)=O)CC2CCC1C1CN(C(C3(CCF)CCC3)=O)CC21 c1(CCNCC2CCN(Cc3cccc(Cl)c3)CC2)c(C)nc(C)nc1O C1(CC(N2CC3C(NC(c4nc(C(C)=O)sc4)=O)(C3)C2)=O)CCCC(C)(C)C1 N1(C(C(CC(=O)OC)C)=O)CCN(C(=O)CN2CCC(CO)CC2)CC(C)(F)C1 Cc1cnc2n1CCC(C(=O)NC1CC(CCNC(C3CCCS3)=O)C1)C2 CCCCC(CN=c1[nH]c(C)nc(=N)[nH]1)NC(C1CCC2CC2CC1)=O N1(C(c2ccn(C(CC)CC)n2)=O)CC(NC(c2cnc(C(C)C)[nH]2)=O)C(C)C1 C1(NC(C(CCCC)NC(CCCOCC=C)=O)=O)CCc2nncn2C1 N1(C(CN(C(C(C)C)=O)C)=O)CC2CC(C(=O)Nc3cc(Cl)cnc3O)(C2)C1 N1(C(c2cc(F)c(Cl)cc2Cl)=O)CC2CCC(C1)N(Cc1cccc(F)c1O)C2 C(=O)(C(C)(F)C(C)(C)F)N1CCC(C)(CNC(C(Cn2ccc(C)n2)C)=O)C1 CC(C)C(C(=O)NCc1ccc(-c2nnc(O)n2C)cc1)c1ccc(Cl)cc1 N1(C(C(C)NC(C=C)=O)=O)C(C(N2CCC(N3CCC(C)CC3)C2)=O)CC2CC12 Cc1cnccc1C(=O)NC1CCC(NC(C2CN(CC(C)C)C2)=O)CC1 c1(-c2onc(C(=O)NC3CC(NC(c4n(C)ccc4)=O)C3)n2)cccc(F)c1F C=CC(C)(O)CC(=O)NC1COCC1CNC(=O)CC(F)(F)c1ccccc1 C1(F)(C(=O)NCC(C(C)C)NC(=O)CC2CC3CC2C3)CCCCC1 N1(C(=O)OC(C)(C)C)CCCN(C(c2csc(Br)c2)=O)CC(F)(F)C1 CN1CCN(C(c2ccc3c(c2)CC3)=O)C(CNC(c2nccc(Cl)c2O)=O)C1 Clc1cc(Br)cc2c1OCC2Nc1cnc2ccnn2c1 O=C1CN(C(C2(CO)CCN(C(C3CCCC(O)C3)=O)C2)=O)CC2(CC2)N1 C(c1ccc(O)cc1)=CC(N1CCC(C2N(C(C(CC)=O)=O)CCC2)C1)=O N1(C(c2ccc(CC)cc2)=O)CC2CC(NC(c3c(C)noc3N)=O)CC1C2 C1(CNC(c2cc(CC)[nH]n2)=O)CC(C(=O)N)=NO1.C1C(=O)NCC1(C)C C1(C(=O)NCC2C(C(=O)NC3C(C)C3(C)C)CCO2)CC(O)CN1C C1(C(N)=O)CCC(NC(=O)CC2C=CCC2)CC1.C(=O)(CCCC1CCCC1)N c1(SC)nc(N(c2cc(-n3cncn3)ncn2)c2ccc(=N)[nH]c2)ncc1F C1(C(=O)NC(C)CNC(=O)CC2CCOC2)C2CCC(=O)C12 c1(N2C(C)C(NC(C3CC4(CC4)C3)=O)CCC2)ncc2c(n1)CCCCC2 Cc1cc(=O)ccn1CC(=O)N(C1CCN(C(C2(S(N)(=O)=O)CCC2)=O)CC1)C C(=O)(C#CC1(C)CC1)NC(C1CCN(C(C23CCC(OC)C2C3)=O)CC1)C C(C)(C(C)C(C)C)NC(c1cc(CC)n(C)n1)=O.n1(C2(C=O)CC2)cncn1 c1(C(N2CCCSCC2C2CC2)C(=O)NCC(=C)C)cc(C)ccc1Br c1(NC(CCC)C(=O)OC)sc2c(c1C(=O)OC(c1ccccc1)C)CCCC2 c1(C(C(=O)NCCCC)N(C)Cc2cc(C)ccn2)ccc(OC)cc1F N1(C(c2c(OC)n(C)nc2)=O)CC(C(N2CCCCC2CO)=O)C(C)(C)C1 CCCCCC(O)C(=O)N1CCCCC1CN(C(=O)CCc1cn[nH]c1)C c1(C(N2CC(C3(NC(c4c(C)n[nH]c4)=O)CC3)C2)=O)ccc2c(n1)CCCC2 CCCC(C(=O)NCC1(C)CCN(C(C2CC(O)(C(F)F)C2)=O)C1)N(C)C C(CCCCCC(=O)N1CC(C(C)NC(=O)C(C(C)C)NC(N)=O)C1)SC NS(=O)(=O)c1cccc(C(N2CCCN(C(c3csc(Cl)n3)=O)CC2)=O)c1 C1(CC(N2CCN(C(=O)Cn3cnnn3)CC2CF)=O)CSc2ccccc2O1 c1(CNC2C(C(=O)NCc3cc(F)c(F)cc3F)C2)ccnc2ccccc12 C1(NC(C(C)N(C(CC=CC)=O)CCC)=O)CCC(=O)NC1C C#CCCCC(C)C(=O)N(CCC(=O)NCC(C)(C1CC1)OC)C(C)C C(CN=c1[nH]c(=NCc2ccn3cnnc3c2)c2sccc2[nH]1)NC(N(C)C)=O C(CS(C)(=O)=NC(=O)C(C)CS(C)=O)C1CC(N(C)C(=O)OC)C1.C(C)(C)C N1(C(C(CC)(F)F)=O)CCC2(CCN(C(=O)C(C3CCCCC3)O)CC2)C(C)C1 c1(NC(c2ccncc2F)=O)cccc(Cl)c1[N+](=O)[O-] c1(CC(=O)N)ccc([N+](=O)[O-])cc1.C1C2CC1N(C(c1cc(C(F)F)no1)=O)C2 c1(C(=O)NCC(C(C)C)(C)NC(=O)C2=CCC2)ccnc2c(F)cccc12 c1(C(N2CCC(CCC(=O)NCC3(OCC)CC3)C2)=O)c(C)n[nH]c1C c1(C(N(C(C)C)CC)=O)cccc(C#CCO)c1.c1(C(=O)N)cc([N+](=O)[O-])n[nH]1 c1(C(=O)NC(C)(CNc2nccnc2F)C2CC2)n[nH]c2c1CCSC2 Cc1c(C(=O)NCC(C)CC(C)C)cccc1CO.C1(CC(=O)N)CC2CC2C1 C1(C(=O)NC(CN(C(C(CC)=CC)=O)CC)C)CCOC(C)(CC)C1 C=Cc1ccc(C(N2CCC(N(C(C3CCC4CC4CC3)=O)CC)C2)=O)cc1 C(CN=C(NCC1CCC1)NCC1(N2CCOCC2)CCSC1)SCC(F)(F)F C1CC(F)(F)CN1C(C1COC(=O)O1)=O.c1(OCCC(=O)N)ccccc1F.C C1(C(N(CC)Cc2ccncc2)=O)CC(NC(=O)CCCC(=O)O)C12CCC2 C1(CCNC(c2cc(CCC)on2)=O)CCCN(C(C2CCCCO2)=O)C1 c1(C(=O)NCCC(C)NC(C2CC2)=O)ccnc(-n2ccnc2)c1.C1CC1.C C(CC(C)CC)NC(C1(SCC)CC1)=O.c1(C(=O)N)ccc(C(C)C)nc1 CC(C)C(C(=O)NC1COCC1NC(=O)C(C)(C)O)N1CCCS1(=O)=O C(N=c1ccnc(C2CC2)[nH]1)C1CCCCN(C(c2csc(O)n2)=O)C1 O=C1COc2ccc(C(N3CC4C(C3)N4C(c3cccnc3Br)=O)=O)cc2N1 N#Cc1c(F)ccc(Br)c1OC1(c2ncc[nH]2)CC1 C#CCCCC(C)C(=O)N(C1CCN(C(c2ccc(F)c(OC)c2)=O)C1)CCC c1(CC)ccc(C(=O)NC(C)CCCNC(c2cc(OC)n[nH]2)=O)cc1CC CC(C)C(N=[N+]=[N-])C(=O)N1CC(C(N2CCCC(C(C)(C)C)C2)=O)C(C(C)C)C1 c1(CC)ccc(C(=O)NC(C)CCNC(=O)CSCc2cscn2)o1 CC1CCN(C(=O)CC2CCS(=O)(=O)C2)CC1.c1(C=O)cnn(CC(F)F)c1.N c1(C(N2CC(CNC(C(C)=C(CC)C)=O)C2)=O)cc(Cl)cc(Cl)c1OC c1(C(=O)NC2C(NC(=O)CC3CC34CC4)CCC2)cc2ccc(F)cc2[nH]1 c1(C(=O)NCC(CNC(=O)C2=C(Cl)CCCC2)OC)cnc2ncnn2c1C CC1C(C(=O)NOCCC(F)F)CCN1C(c1cnnn1C1CC1)=O C=CC(C)(O)C(=O)NCCC(C(C)C)NC(=O)C=CC=C(Cl)Cl CN1CCc2cc(C(N3CC4(CC(NC(C5CC5(F)Cl)=O)C4)C3)=O)ccc2C1 N1(C(Cc2cnc(C)[nH]2)=O)CCC(N(C(=O)CC2CCC(C)C2)C)CC1.C1CC1 C=CC(C)(CC)C(=O)N1CCC1CNC(c1cnn(CCC#N)c1C)=O C(CO)(CCCCNC(=O)CNc1ncccn1)NC(C1(C)CCCCO1)=O C(CC(C(C)C)NC(c1cccc(OC(F)F)n1)=O)NC(Cc1cnc(C)s1)=O Cc1ccc(CC(N2CCC23CN(C(=O)CC(C)C(C)C)C3)=O)c(Cl)n1 Cc1ccc2c(c1)CCC(C(=O)NC1CCCN(C(=O)CN=S(C)(C)=O)C1)O2 c1(C(=O)NC(CNC(CC)=O)(C)CO)ccc(CC(F)(F)F)cc1 N1(C(CCC2(NC(c3c(C)scn3)=O)CCCC2)=O)CCCCCCCC1 N1(C(c2cn(CC)nn2)=O)CC(C(=O)NC2COCCC2(F)F)C(C)(C)C1 N1(C(=O)NCC2(Cc3ccccc3Cl)CC2)CCCC12CC1CCC2C1 CCCC(CNC(c1c[nH]nc1CNC(=O)C(F)C(F)(F)F)=O)CCO C1(NC(Cc2cnc(C)o2)=O)C2CC1N(C(c1ccccc1SC(C)C)=O)C2 N1(C(C2C(CCOC)C2)=O)CCCCCC1C(=O)NCCc1cccc(F)c1 N1(C(C(CNC(CCC(C)(C)OC)=O)(C)C)=O)CCC2(CCC(C)C2)C1 N1(C(Cc2ccc(C(C)=O)s2)=O)CCC(COC)(NC(c2cccnc2)=O)CC1 C(=O)(C1SCCc2ccccc21)N.C(C(C)(C)C)N(C(C1CNC(=O)N1)=O)CC CC(C(=O)N1CCOCC(CNC(=O)CNC)C1)P(C)(C)=O.c1ccccc1.C N1(CC)N=C(C(=O)NC2CN(C(C3CCC4CC4CC3)=O)CC2O)CCC1=O CS(=O)(=O)C1CCCCC1.C1(C(N2CC(c3c[nH]nn3)C2)=O)C2CC3C(C2=O)C13 c1(NS(C2C(OC)CCC2)(=O)=O)cc2c(cc1F)CCC(=O)N2 N1(C(C(C)CC2CCCO2)=O)CCOC2(C1)CN(C(c1cccc(Cl)c1N)=O)C2 c1(N(C)C)cc(NC(=O)CCCn2ccc(C(=O)O)n2)cc(F)c1 c1(N2CC(C)C(CNC(=O)CCC(N)=O)CC2)ncnc2[nH]c3ccccc3c12 c1(C(=O)NCCNC(C2N(C(C)=O)CCOC2)=O)cc(S(N)(=O)=O)cs1 C1(C(=O)NCC2CC2(Cl)Cl)(CC)CCCN(C(C2(CC(C)C)CC2)=O)C1 C(=O)(C(CC)CCOC)N1CC(C)(NC(CCc2ncc(CC)o2)=O)C1 c1(NC(C(Cn2ccc(C)n2)C)=O)nc2ccc(I)cc2[nH]1 C1(NC(c2c(C)onc2)=O)CN(C(c2cc(=O)n(C)cn2)=O)C2(CCOCC2)C1 C1(CCNC(CCOC)=O)CSCCN1C(=O)CCOc1ccc(N)cc1 N1(C(=O)OC(C)(C)C)CCC(C=O)CC1C1CC1.[SH](=O)(=O)C(F)(F)F.N CS(C)(=O)=NC(=O)C(=O)NCC1CC(C)CO1.c1(C=O)cnc2ccccn12 CCCCC(=O)C(=O)NCC(C)(O)CNC(c1cnn(CCC)c1)=O C(=O)(CCCN=c1nccc[nH]1)NC1C2(CCN(C(CC(=C)C)=O)C2)CCCC1 C1(NC(C2C(CC)C2)=O)CCCCN(C(=O)C2CC2)C1 CC(C)(C)C(C)(O)C(=O)NC1CCC(C)C1.c1(CC=O)ccc2c[nH]nc2c1.N C=C(C)CC(C(=O)N1CC(c2cc(O)no2)C1)NC(c1ccc(C)cn1)=O c1(NC)ccc(C(=O)NCC2CCCN2C(=O)CC2CSC2)nc1 N1(C(Cc2c(CC)con2)=O)CC(C(=O)NC2CC=C(C)CC2)CC1(C)C C(=O)(C#CC1(C)CC1)NC(C(C)C)CNC(C1CCC=CCC1)=O N1(C(C(=O)N(CC(C)C(F)(F)F)C)=O)CCC(O)C(C)C1 C#Cc1ccc(C(=O)N(C(C)C(=O)N(CC(O)CO)CC)CC)o1 C1(NC(C(c2cccnc2)C)=O)(CF)CCN(C(C2(CO)CCCCO2)=O)C1 c1(C=O)cc(C)c(F)cc1F.c1(COC)nc(C(=O)NC2CCCC2)cs1.C c1(C=O)ccncc1.C1(C(C)N(C)C)CCCC1.CC(F)(F)C1CC1C(=O)N C1(NC(c2cncc(C#C)c2)=O)COC2(C1)CN(C(=O)CCc1nc(=N)[nH][nH]1)C2 Cc1cc(C(=O)NCC=CCNC(=O)C(C)C(F)F)nc2[nH]nc(O)c12 Cc1ccccc1CC(=O)NCCn1cc(C)nn1.C(=O)CC(O)CN(C)C.N N1(C(CNC)=O)CCN(C(C2CCC(C(=O)N(C)C)CC2)=O)CC1C1CC1.CC CC1CC(C(=O)Nc2ccc(O)cc2)CCN1C(=O)CC1CSCCO1 Cn1cc(CN2C(C(=O)NCC3CCSCC3)CC3CC23)c2ccccc12 N1(C(CN(C(COC)=O)C)=O)CCC(C2(NC(=O)CC(O)CSC)CCC2)CC1 CCCC(C)(O)CNC(c1cc(CCNC(=O)C(=O)N)on1)=O.CC(F)F CC1=NOC(CC(N2CCC(NC(=O)CCc3nc(C)cs3)C2)=O)C1 Cc1cccc2c1CC(C(=O)NC1CCN(C(=O)CSC(F)F)CC1CO)O2 CC1CC(O)CCN(C(C2CC23CC(NC(=O)C=Cc2cocn2)C3)=O)C1 c1(CC)ccc(C)cn1.C1(C=O)CC=CC1.C1(CC(=O)N)(NC(C)=O)CC1 Cc1cncc(C)c1C(=O)NC1CCC(F)(CNC(=O)CC2OCCCO2)C1 c1(C(=O)NC2CCN(C(c3cc(Br)n[nH]3)=O)CC2O)nc2cnccc2s1 C1(NC(CC2CCN(C(CN(C(C)C)C)C)C2)=O)CCc2n[nH]cc2C1 c1(C=O)ccnc(C(F)(F)F)c1.C(C)(C(=O)NC1CCC1)NC(=O)OC C1(C(=O)NC2(C)CC(C(=O)OC)C2)(NC(=O)C(C)C)CCCC1C C(=O)(C(CCc1ccccc1F)N1CCCC1c1ccccc1Cl)NC(C)(C)C n1(C(CC)CC)cc(SC(C2CN(C(=O)OC(C)(C)C)C2)C)nn1 C(=O)(C1(C)CCc2ccccc21)NC(CNC(c1c(CC)sc(=N)[nH]1)=O)CC c1(C(=O)NC2CCC(NC(c3c(=N)[nH]cnc3)=O)CC2)ncc(Cl)cc1Cl O=C1Cc2c(C(=O)NC3(C4CCCN4C(c4scnc4Cl)=O)CC3)ccnc2N1 c1(C(N2CC(C(C)NC(c3nccn3C)=O)OCC2)=O)cnc(F)c(Cl)c1 N1(C(CCCOCC=C)=O)CC(NC(=O)C=CCN2CCCCC2)CC(C)C1 N1(C(Cc2c(C)nn(CC)c2C)=O)CCCN(C(C2CCCS2(=O)=O)=O)C(C)C1 c1(OC)ccc(Cl)c(C)c1C(N1CCCN(C(=O)C2=CCCCO2)C(C)C1)=O C1(NC(C2CCS(=O)(=O)N2)=O)Cc2ccccc2C1NC(C1CC(O)C1)=O c1(C(N2CCC(C#C)C2)C(=O)NCCCCCC)cccn2cc(C)nc12 N1(C(c2cc(OCC)no2)=O)C2CC1CN(C(=O)C(F)C1CCOC1)C2 CC1(C)CCN(C(c2cnc[nH]2)=O)CC1NC(C1(N2CCOCC2)CC1)=O N1(c2cnc(C(=O)OC)c(C)n2)CCCC(CO)(NC(C2CCC2(C)C)=O)C1 C12CC(C1)CCO2.C(CC(=O)N)NC(=O)NC.C(=O)CN(C1CCC1)C c1(C(C(=O)NC(CCNC(COCCC)=O)C)O)ccc(Cl)c(Br)c1 Cc1ncc2ccc(C(=O)NCC3(CC)CC3)cn12.N1(CC=O)CC=CC1.N C(CC1CC1)(C(=O)NC1(CO)CN(C(c2coc(Cl)c2)=O)C1)OC CS(=O)(=O)c1ncc(C(N2CC(NC(=O)CC3CCCO3)C3(CC3)C2)=O)s1 c1(C(=O)NCC2CC2NC(c2ncc(F)cc2F)=O)cc(Cl)c(F)cc1Cl C1(NC(C2CCC=CCC2)=O)CN(C(=O)CSCc2cscn2)CCC1O C(=O)(CCCC(F)(F)F)NC(COCC)C(N1CCCCC(F)(F)C1)=O c1(NC(c2ncc(CC3CC3)s2)=O)ccc(C(=O)O)c(C(F)F)c1 N1(C(C)=O)CCN(C(=O)C2CC2)CC1.c12ccc(cc1)SCC(=O)N2 C1(C(=O)NCC(CN(C(c2c(C)ncn2O)=O)C)O)CC2CC(O)CC(C1)C2 C(=O)(C1=CNC2=NCCCN12)N1CCN(C(c2cccc(C)n2)=O)C2C1C2 C1(CC(N2C(COC)CC2C)=O)C2CCC1CN(C(=O)OC(C)(C)C)C2 N1(C(c2n(CCC)ccc2)=O)CCCC1(C(N1CC(SC)C1)=O)C(C)C C1(NC(C(C)=C(CC)C)=O)CCC2(CCCN2C(c2cc(C#N)c[nH]2)=O)CC1 C1(NC(N2CCN(C(c3ccccc3Br)=O)CC2)=O)C2CC3(CC3)CC12 c1(C(=O)NCC(CNC(c2n(CC)ncc2)=O)(C)F)c(C)cccc1Cl C1(CNC(=O)C(=O)NC2CC2)CC2(CCOCC2)CN1c1nc2cccnc2s1 N1(Cc2scc(C(C)C)n2)CCNCC1C1CCC1 CC1(CNC(=O)CC2CCC2)CCCN(C(=O)CCN2CCCC2=O)C1 CCC(CCCC(=O)N1CCN(C)CC1C(C)C)NC(c1[nH]cc(C)c1C)=O C(=O)(CC(=O)N)NCC#C.c1(C=O)cnn(C(C)C)c1.C1(CC)CCCCC1 C1(CC)CCCN(C(=O)CC2OCCCO2)C1C(N1CC(OCC(C)C)C1)=O c1(C(N2CC(CC(C)NC(C3(CCO)CC3)=O)C2)=O)ccc(C2CCOC2)cc1 c1(OC)ccc2cccnc2c1C(=O)NCC1(NC(=O)CC(C)C(C)C)CC1 NC1C2CC3CC(C2)CC1(CNS(=O)(=O)C1(Cc2ccccc2)CC1)C3 CC12COCC1CN(C(C13CCC(CC1)N(C(C1CCC(C4CC4)C1)=O)C3)=O)C2 CC(C)CC(C(=O)N(CC(C)O)CCNC(=O)C=Cc1cc[nH]c1)C(C)C C(c1ccc([N+](=O)[O-])s1)=CC(N1CC2C(C2)C1)=O.c1(C(=O)N)sccc1Cl.C C1(CNC(=O)CCCF)CC2(CCN(C(=O)CCc3cccc(F)c3F)CC2)C1 c1(C(C)C)ccc(C(O)CNCCC2COCC2O)cc1 CC1(CNC(c2csc(CO)n2)=O)CCN(C(=O)COc2ccccc2O)CC1 N1(C(C(C)c2cccs2)=O)CC2CC(NC(c3cnc(O)o3)=O)C1C2 n1(C2CC(C(N(C(C)C)C(C)C)=O)C2)cc(CCSCCO)nn1 c1(C=O)ccccn1.C(C)C(=O)N(CC)C(C)C.[SH](C)(=O)=O.C=O.C C12(NC(c3n(CCC)ncc3)=O)CCN(C(=O)CN3CC(C)(C)C3)CCC1C2 c1(OC)nc(=NCCCNC(=O)Cc2cc(Cl)ccc2OC)nc(OC)[nH]1 c1(C(=O)NC(CCNC(C2CN(OC)C(=O)C2)=O)C(C)C)cc(F)cc(N)c1F c1(C(=O)NC(CNC(C(N2CCCC(C)C2)=O)=O)C)cc2c(s1)CCSC2 Cc1ccnc(C)c1C(=O)NC1CC(n2cc(-c3c(C)nn(C)c3Cl)nn2)C1 C1(C(N2CCC(C(C)(C)O)C2)C(=O)NCC(=C)C)CCCN(C(=O)OC)C1 c1(OC)ccnc(C(=O)NC2CCCN(CCOC3CCC3)C2)c1F N1(C2CCN(C(C3(C)CN(C(COC(C)(C)C)=O)C3)=O)C2)CCNC(=O)C1 c1(N2CCC(CC=C)(NC(c3ccc(Cl)cn3)=O)C2)cc(S(C)(=O)=O)ncn1 C(=O)(CS(=O)c1cccc(OC)c1)N(CCNC(C(C(=C)C)(C)C)=O)CCC CC1COC(C(=O)N(C)CCNC(=O)C(=O)NCC2CC2)CO1 c1(C(N(C)CC2(O)CCCN(C(C3(C)CCCO3)=O)C2)=O)cc(F)c(F)cc1F CC(C(C)(C)C(=O)NCCc1noc(=O)n1C)NC(=O)C(O)C(F)(F)F C(=O)(C#CC1CCCC1)NC1(C)CCN(C(C2CC(CC3CC3)C2)=O)CC1 Cc1cc(C(C(=O)NCC2CCOC2)N(C)CCc2ncccn2)c(C)s1.C c1(C(N2CC(NC(Cc3cc(OC)c(F)cc3)=O)C2)=O)cc2cnc(Cl)cc2s1 c1(C(=O)Nc2ccc(C)c(NC(C)=O)c2C)ccc(C)c(S(=O)(=O)CCO)c1 c1(C(=O)NCCOCCNC(C(n2ncc(C)c2)C)=O)cc2cnccc2o1 C1(C(N2CC(C)(C)C(NC(c3ccns3)=O)C2)=O)CC2CC1C1C2C1(F)F c1(OC)cc(NCC2CN(C(c3sncc3C)=O)CC2C)nc(C(F)(F)F)n1 c1(OC)c(C(=O)NC2CC(OC)CN(C(=O)C(C)(C)CF)C2)ccc(Cl)c1Cl CC1CCCc2c(C(=O)OCC(n3cccn3)C)cnn21 C12(NC(Cc3c(C)occ3)=O)CC3CCC(C1C2)N3C(=O)C(C)C1CCC1 Cc1cc(N)c(C)nc1C(N1CCCC(NC(c2ccc(Cl)cc2)=O)C1)=O C1(CNC(c2ccc(OC)o2)=O)CC2CN(C(=O)C(F)OC(F)(F)F)CC12 c1(C(N2C3C(NC(C(c4n(C)ncc4)(F)F)=O)C(C3)C2)=O)cc(F)ccc1Cl N1(C(=O)CSc2cccs2)CCC2(CCC2CNC(C23CCC2C3)=O)CC1 C1(C(F)(F)F)(C(N(CC)CC)=O)CC2CCC1C2.Cc1nc(C=O)n(C)n1 CCCC(CC(C)C)C(=O)N1CC(O)(CNC(C2CC2(F)F)=O)C1 C1(C=O)CCc2n[nH]cc2C1C.C1(OC)CN(C(=O)CC2CS(=O)(=O)C2)CC1.N C(=O)(C1CCCc2n[nH]cc21)NC1C(CN=c2c(CC)c(Cl)nc(C3CCC3)[nH]2)C1 c1(OC)cc(C)nc(N(C)CC2CCCCN2C(c2cc(C)c(C)nn2)=O)n1 CC1CCC(C)N1CC(=O)NCC1(CNC(c2ccc(F)cc2)=O)CCC1 C(C)(CCC(C)(C)C)(c1n(C)nnn1)NCC12CCC(CC1)O2 c1(C(N2CCC(CNC(C3CC(C)OCC3)=O)C23CC3)=O)cccn2nnnc12 CC(C)C(F)C(=O)NCC1(F)CC(NC(=O)C(C)S)C1.c1ccccc1.C N1(C(C(C)(C)O)=O)CC2CCCC2(NC(=O)C(=O)NC2CC2)C1 Cc1cn2nc(C(=O)NNC(N3CCC(C(=O)O)C4(CCC4)C3)=O)cc2c(=O)[nH]1 N1(C(CSCCC)=O)CC2CCC(C1)N2C(c1cnc(OC)cc1C)=O c1(OC)cnnc(C(=O)NCc2nc(C=O)c(C)o2)c1.CC(N)=O.CC.N CCC(C)(C(=O)NCC1CCCCN1C(=O)CCCn1ccnc1C)C(N)=O N1(C(C(C(=O)OC)C)=O)CC(C)OC(C)(C)C1.N1(CC(=O)N)CC2CC2C1 N1(C(C2C=CC(=O)N=N2)=O)CCCC2(CCN(C(c3cc(F)ccc3F)=O)C2)C1 N1(C(C(CC)OCC)=O)Cc2ccccc2CC1CNC(=O)C(C(C)C)O.C N1(C(C(C)NC(=O)C2CC2)=O)CC=C(CC(=O)N)CC1.C1(C2(O)CCC2)CC1 C(C(C(=O)NC1CSC(C)C1)C(C)C)NC(C(=O)NCC)=O C1(NC(c2ccnc(C(C)C)n2)=O)CCCN(C(c2cn(C)ccc2=O)=O)C1C C#Cc1ccc(C(=O)N(CCCCCNC(=O)C(C)c2ccon2)C)c(OC)c1 C1(NC(C(CCC)NC(N)=O)=O)CCC2CCN(C(C3(CO)CCOCC3)=O)C1C2 C(=O)(CCCCC(=O)N1C(C)C2CC1C2NC(c1csc(C2CC2)n1)=O)NC N1(C(C(CCC)OCC)=O)CC(CNC(C2(c3ccno3)CC2)=O)CC12CCC2 N1(C(C2C=C(C)CS2)=O)CCC(O)C(N(C(=O)CCC(C)CN(C)C)C)C1 c1(C(N2CCC(NC(C3C(C)(C)C3C(F)F)=O)CC2)=O)cncc2sccc12 c1(C(CN(C(=O)NCC2C(C=C)C2)C)(C)O)ccccc1 C(CC(O)C(=O)N1CC(CNC(=O)C)C(O)C1)SC.c1ccccc1.C=O.N N1(C(c2cc(C)c(C)s2)=O)CC(CNC(C2CCC2(F)F)=O)CC(C)(C)C1 C1(CC(C)C)CCN(C(=O)CSC2CCCC(C)C2)C1(C)C C=CC(C)(O)C(=O)N1CC(F)(CNC(=O)C(CC)n2cccn2)C1 N1(C(c2c(CCC)[nH]cc2)=O)CCCC(COC)(NC(C2CC2(C)C)=O)C1 c1(C(=O)NCCCN(C(CC(C)CF)=O)C)cc2c(nc1O)CCC(C)(C)C2 C(C)(CC(F)(F)F)NC(c1ccc(F)s1)=O.C(=O)C(N1CCCC1)C1CC1 N1(C(c2ccc(OCC)nc2)=O)CC2CN(C(C3C=CC(=O)N=N3)=O)CC2C1 C(=O)(C1=CCC(C)(C)CC1)N(CC(O)CNC(c1ccc(C#N)o1)=O)C c1(C(=O)NCC2CC(NC(C(N3CCNC3=O)C)=O)C2)cccn2ccnc12 c1(Cc2n(-c3cc(F)ncc3)nc(-c3cc[nH]n3)n2)ccc(Cl)cc1Cl c1(C(=O)NC(c2cc(C)[nH]n2)C2CCOCC2)oc(C2CC2)nc1C c1(C(N2CCCCC2Cc2ccc(F)cc2)=O)cc2c([nH]1)CCNC2 C1(CN(C)C(c2cncc(Br)c2)=O)CCCC(NC(c2ccon2)=O)C1 Cc1cc(Cl)n[nH]c1=NC(=O)C1CC1C(=O)Nc1ccc(Cl)nc1C#N c1(C(N2CC3CN(Cc4cn(C(C)C)nc4)C3C2)=O)c(Cl)cnc(Cl)c1Cl c1(-c2scc(OCC)c2)nc(C(C)N(C)C)nn1Cc1ccc(Cl)cc1 C1(NC(C(C)OC2CCCC2)=O)CCCC(N(C(=O)Cn2cnnc2O)C)C1 C1(CNC(C=NOC)=O)CC2CCC1N2C(c1ccn(C2CCCC2)n1)=O Cc1cc(C)n(C(C)C=O)n1.C1(C(C)C)CCCN1C(=O)Cc1cnc(C)o1.N c1(CC)ccc(C(=O)N(C2CN(C(=O)COCC(=O)OC)CC2F)C)cc1Cl Cn1cc(C(=O)NCC(C2(O)CN(C(=O)C(O)c3ccco3)C2)(C)C)c(=N)[nH]1 c1(N2CC3C(CNC(Cc4c(OC)ccc(C)c4)=O)C3C2)ccc(C#N)cc1F N1(C(Cc2ccc(C)o2)=O)CCOC(C(N2CCCOCC2C)=O)CC1 c1(CCC(c2n(CCC)nnn2)NC2(C)CCC(C)CC2)ccc2c(c1)CCO2 C(=O)(CCC(=O)N1CCOCC1CNC(c1c(C)ncn1O)=O)OCC N1(C(C(CC)F)=O)CCC2(CCCC2CNC(c2cccn3nnnc23)=O)CC1 C(=O)(CC1=NN(C)C(=O)C1)N1CCCC(F)(C(=O)NCC(COC)OC)C1 CN1CCC(F)(C(=O)NCC2CCN2C(=O)CCc2cn[nH]c2)CC1 CC1(C)CN(C(=O)C(O)C(C)(C)C)CC1C(=O)NC1(C)CCOC1=O C1(C)CCCN1C(=O)CC1CN(C2CCCCC2)C1.C(=O)C(F)F.CCO.C C1(NC(c2cncc(O)c2)=O)CC2CCCC(C1)N2C(C1(O)CCCCCC1)=O C1(C(=O)NCCN2CCN(C(CCNC(=O)OC)=O)CC2)CC2CCC(C1)S2 N1(C(CCC(C)OC)=O)CC2CC(C1)C2NC(=O)Cc1ccc(F)cc1Cl C1(C)(CC(=O)NCC(=O)NCC(CO)Cc2onc(CC)n2)CCCCCC1 CC1(C#N)CCCN(C(C2CCN(C(C3CN4CCC3CC4)=O)C2)=O)C1 c1(C=O)cc(Cl)c([N+](=O)[O-])[nH]1.C1(NC(=O)COCC(F)(F)F)CCCCCC1 c1(C(=O)NCCc2c(C)nc[nH]2)coc2c1CN(C(c1ccnn1C(C)C)=O)C2 C#CCCCC(C)C(=O)NC(CNC(c1cnn(C(C)C)c1)=O)CC c1(C(=O)NC2CC(CNc3ccc([N+](=O)[O-])cn3)C2)coc2c1C(O)CCC2 N1(C(C(c2cccnc2)C)=O)CCN(C(C2CC3CC2C2CC32)=O)CCC1C N1(C(CN(C(C)=O)C)=O)CCN(C(c2cn(C(F)F)cn2)=O)C(CO)C1 C1(C(NOCC=CC)=O)COCCN1C(=O)CC1(N(C)C)CC1 C1(NC(c2sccc2S(=O)(=O)N2CCC(O)CC2)=O)CCOC12CCCCC2 c1(C(N2C3C(NC(C(Cn4ccc(C)n4)C)=O)C(C3)C2)=O)ccc(S(C)=O)cc1 N1(C(CCCOc2ccc(C)cc2C)=O)CC(C)N(C(c2ccsn2)=O)CC1C N1(C(CSCC(=O)OC)=O)CCCC(C2CN(C(=O)CC(C(F)(F)F)O)C2)C1 CCC(C)(C#N)C(=O)NC(C)CN(C)C(c1ncc(C)cc1OC)=O Cc1cc(NC(C2CC(F)CN2C(=O)C(C)c2ccon2)=O)c(C)s1 C(C)(C(=O)N=c1[nH][nH]c2c1CN(C(c1cnc(Cl)c(I)c1)=O)C2)OCC=C c1(CC)ncccc1C(=O)NC1(C(N2CC(COC)C2)=O)CSC1 c1(OC)cc(C)c(C(=O)NC2CN(C(=O)CC(C)C3CC3)CC2O)cc1OC N1(C(Cn2cnc(C#N)n2)=O)CC(C2CC2)(C(=O)NCC2NC(=O)NC2=O)C1 C(=O)(C(C)(C)C(C)(F)F)NCCCCC.N(CP(C)(=O)OCC)C(=O)C Cc1cc(N2CCOC(C)(C)CC2)ncc1S(=O)(=O)NCC1CCCOCC1 N1(C(C2C(OCC)C2C)=O)CC(C)CN(C(C2CC(OC)C2)=O)C(C)C1 C1(C(N)=O)(OC)CCN(C(c2cncc(C)c2)=O)C1.c1(C=O)ccsc1C#N.N N1(C(C2(SC)CC2)=O)CCCC(O)(C)CC1.C1(C(=O)N)(C(F)F)CCCCC1 Cc1cc(O)ccc1CC(=O)NC(C1CCCN(C(C2(O)CCSCC2)=O)C1)C C1(C(=O)NCCCNC(=O)NC)CCN(C(c2cc(O)cs2)=O)C1C c1(C(N(CCNC(C(C(C)OC)O)=O)C(C)C)=O)csc2c(F)cccc12 c1(NCc2c([N+](=O)[O-])cccc2)ccc(S(=O)(=O)N2CCC3=C(CCCC3)C2)cn1 c1(C(=O)NC(C(C)NC(=O)C(C)(C)n2cccn2)C)nnc(O)nc1O C1(C(N(CC(C)NC(=O)CC2CCC=CCC2)C)=O)CCC2CCCCN12 N1(C(c2oc(C)c(CO)c2)=O)CCC(C(=O)NC2CC(=O)N(C)C2)C1(C)C N1(C(C(C2CC2)OC)=O)CCC(NC(C2CCCC(O)C2)=O)C(CO)CC1 c1(C(=O)NC(C(=O)OC)C(C)c2ccccc2)cc(C)nc2ccnn12 C(C(=O)N=c1ccn(C)[nH]1)NC(=O)NC(CC(=O)OC)C C1(NC(Cc2ccc(C)nc2)=O)CC2CCC1CC2C(=O)NCc1ncoc1C C1(C(=O)NC2CCCC(O)C2)CC(O)CCN1Cc1cnc(O)nc1O C=C(C)CCCC(=O)NC1CCCCN(C(=O)CSc2ccncc2)C1 c1(C(=O)N)cc(C(F)(F)F)cnc1C.c1(CC)c[nH]nc1C(N1CC(C)C1)=O C1(CNC(CC(CC)C)=O)CCN(C(=O)COCc2nnc(C)s2)C12CC2 C12(NC(Cn3ccc(C)n3)=O)CCCCC1CN(C(c1cc[nH]c1C)=O)C2 n1(CC(=O)N)nc(C2CC2)n(C)c1=O.CC1CCCC(Cn2cc(CC)nn2)C1 C1(C)(CC)C=C(C(=O)N2CCCCCC2C)C1.C1(C=O)(CCN(C)C)CC1 N1(C(c2ccc(CC)[nH]2)=O)CCOCC(C(=O)NC(C)(COC)CCO)C1 C(C#Cc1cccc(F)c1)NC(=O)NC(C)(CO)C1CC1 CCCCCCCC(=O)N1CCCC(N(c2cc(C)ncn2)C)C1 c1(OC)cccc2c1CCC2(C(=O)O)NC(=O)C1CCCc2c1ncn2C N(C1c2ccccc2CC1O)C(=O)NCc1cccc(C)n1 c1(C(=O)NC(CCCN)CO)oc2ccccc2c1Cc1ccc(Cl)cc1 C(=O)(C(F)C(C)(C)O)N1CCC(C(C)CNC(=O)Cc2cn[nH]c2)CC1 C1(C(F)F)(CNC(=O)C(=O)N)CCN(C(c2ncc(F)cn2)=O)C1.C1CC1 N1(C(Cn2c(C)cnc2)=O)CCN(C(=O)CC2OCCO2)CC1C C(C1OCCc2sccc21)C1C(O)COCC1 c1(C(=O)NC2CC(NCc3ccc(F)c(Br)c3)C2)ccnc2ncccc12 c1(C(=O)NCC(C)C2CC2)cc2c([nH]1)CCCC2.C1(C=O)SC2C=CC1CC2.N CC1(C(=O)NCCC2CCCCCC2)CCN(C(C2CCCS2)=O)C1 c1(C(=O)NCC(C)N(C(CS(CC)(=O)=O)=O)C)ccc(OC)c(F)c1N c1(C(C)NC(c2cc(Br)ccn2)=O)ccc(Br)nc1 C1(NC(c2cncc(O)c2)=O)C2CC1CN(C(C1CC1(Cl)Cl)=O)C2 Cn1cc(S(N)(=O)=O)c(C(N2CCC(NC(=O)Cn3ncnn3)C2)=O)n1 c1(C=O)cn(C)[nH]c1=NC=O.C(C)CC.CC(C)CC1CC1C=O.C(C)C.N c1(N(C)CC2(CC)CC2)nnc(-c2nc(-c3ccncc3)no2)n1CCC#N CCCCCC(O)C(=O)N(CCCCCCNC(C1CCC2CC1CO2)=O)C C1(O)(CC(=O)N)CCCCC1.C1(NC(C(N2CC(C)C2)C)=O)CC(F)(C)C1 C1(NC(C2C(CNC(C3CCC4(CCC4)C3)=O)CCO2)=O)CN2CCCC1C2 N1(C(C2CC(C)C2)=O)CCCC(CCNC(c2ccc(CC(C)(C)O)s2)=O)C1 C1(CNC(Cn2c(C)ccn2)=O)C(C)CCN1C(c1cccnc1O)=O n1(CC)ncc(Br)c1C(=O)NC1CC1CNC(c1cnccc1OC)=O c1(C(N2CCCC(CC(=O)NOC3CCCCC3)C2)=O)cc2ccccn2c1 N1(C(C(n2cc(C)nc2)(C)C)=O)CC2C(C)C2C1.N1(CC=O)CCC(C)(O)C1 S(=O)(=O)(c1cccc(C(=O)N(CC(C)(C)C)C)c1)NCCCC n1(CC)nc(C)c(C=O)c1C(F)(F)Cl.C(=O)(C(O)C1CCCC1)N(CCC)C N1(C(c2c(C)c(Br)cc(F)c2)=O)CCC2CN(C(C3CN(C)C3)=O)CCC12 Cc1cc(F)c(C(N2CCC(O)C2C(=O)Nc2cnc(C#N)c(C)n2)=O)cc1F n1(CC)cc(Cl)c(C(=O)NCC2CN(C(=O)CCCC3CCCCC3)C2)n1.O N1(C(c2n(C)cnn2)=O)CCN(C(c2n[nH]c(C(C)(C)C)n2)=O)C2(CCC2)C1 c1(C(=O)NC2CN(C(c3c(CC)cno3)=O)C(CO)C2)cnn2c1OCC(O)C2 C1(CNC(c2cncc(C)c2Cl)=O)CCC2CN(C(=O)CCCC#N)CCC2C1 C1(Cc2cc(C(C)NC(CCCCC)C)[nH]n2)OCCN(C)C1c1ccccc1 c1(C(=O)N)nnc(O)nc1O.C1(NC(C(C)SCCCC)=O)CCC(F)(C)C1 N1(C(C2C(C)(NC(C(C)SC(C)C)=O)CCCC2)=O)CCC2C(=O)NCC2C1 c1(OCC)cccc2c1CCC2N1C(=O)C2CCC(C(=O)O)CN2C1=O N=c1[nH]c(NCC2(N)CCCCCC2)ncc1Cl C1(NC(CC2CC(C)(NC(CC3C(CC)C3)=O)C2)=O)CCCC1C#N c1(C(=O)NCC(CCCC)NC(C2(C)CCCS2)=O)ccc2nc(O)sc2c1 Cc1cnc(C(=O)NC(C)CC(C)NC(=O)CCc2cncc(C)c2)c(C)c1 N1(C(c2c(OC)cccc2)=O)CCC(C(C)(C)C)CC1C.c1(C=O)ccon1.N c1(CC(C=O)O)ccc(F)cc1.C12(NC(CCC3(C)CC3)=O)CC(C)(C1)C2 Cc1noc(C2CC2NC(=O)CC2CCCSC2)n1.C1(C)(C)CNC1=O c1(CNC(C2N(C(CC3CCC(C)O3)=O)CCC2)=O)ccc(F)c(F)c1 Cc1ccc(F)c(C(N2CC(NC(C3(F)CC3C)=O)CC(F)C2)=O)c1 N1(C(C(CC)(C)COC)=O)CC(C(=O)NCCO)CCC1(C)C.C1CCCC1.C C=CCC(C(=O)NCC1(n2cccn2)CC1)NC(c1nc[nH]n1)=O N1(C(Cc2c(C)nn(Cc3c(OC)cccc3)c2C)=O)CC2C3C=CC(CC3)C2C1 c1(N2CCC(CCNC(C(CC)F)=O)CC2)nc2c(cc1Cl)C(=O)OC2 C1(NC(N2CCCC(C)C2CCO)=O)CC1C1(C)CCOCC1 N1(C(C2CCN(C(CNC(C(CC)C)=O)=O)C2(C)C)=O)CCCC2(CCCO2)C1 C=CCC(CC)C(=O)N1CCC(N(C(=O)Cn2cc(C)cn2)CC2CCCO2)CC1 CC1(CNC(c2nn[nH]c2C(F)(F)F)=O)CCN(Cc2cc(Cl)ccc2Cl)CC1 N1(C(c2oc(C)c(CO)c2)=O)CC(C)CN(C(=O)CNC(C2CCC2)=O)CC1C C1(N(C(CCOCCNC(C(CC#C)O)=O)=O)CC=C)CCCOC12CCC2 C1(C(=O)NCCCC(C)(C)NC(C(CN(C)C)O)=O)C2CCC1(C)C2(C)C C1(CCCNC(C2(C)CC(=C)C2)=O)CCCCN1C(=O)C(CCC)=CCC c1(-n2c(NC(=O)NCc3cc(C4CCC4)n[nH]3)ncc2)ccccc1Cl Cc1nn(C)c(C)c1OCC(=O)NC(C1CN(C(C2(C)CC2)=O)C1)C C1(N(c2ccc3cc[nH]c3c2)C(=O)NC2C(C)C2C)CCc2ncccc2C1 C(CCCCCC(=O)N1CC(C)(C)C1C1CC1)NC(C1CC(C)OC1)=O C#CC1(OCC(=O)NCC(C)(C)NC(C2CCC(N(C)C)C2)=O)COC1 C(C)(C(=O)NCC(CO)OC)NC(C1(CCCC)CC1)=O c1(C(=O)NC(C(C)C)CNC(=O)CC2CCC2(C)C)cc2c(F)cccc2s1 C1(CNC(c2n(C(C)C)nnn2)C2(SC)CC2)CC12CCCCC2 c1(C(=O)NCC(C)(O)C2(C)CC2)cc(C)ccn1.C1(C(=O)N)CCCCC1O C(C(CO)C(F)(F)F)NC(=O)CC1CN(C(=O)CC=C(Cl)Cl)CCO1 c1(OC)cc2[nH]ncc2cc1NC(C1CC12CN(Cc1cccc(F)c1Br)C2)=O c1(CCC)cc(C(N2C(C)C3CC2C3NC(=O)CCc2cnc[nH]2)=O)cc(O)n1 C(C)(C)(CC(=O)NCC1CCOC1=O)N(C(COCC(=O)OC)=O)C C1(CCNC(=O)CC2CCCCC2)(NC(c2cc(C(C)C)sn2)=O)CCOCC1 C(=O)(CCCC(=O)c1cccs1)N1C(Cc2cncc(C(=O)OC)n2)C=CCC1 C(=O)(C1CCc2ccccc21)N1CC2CCN(C(COCCOCC)=O)C2CC1 O=C1COc2ccc(C(=O)O)c(F)c2N1CCc1nc(C(F)(F)Br)no1 C1CN(C(=O)C(C(C)C)N2CCCC2=O)CC1C.C1(C(=O)N)(OC(C)=O)CC1 c1(C(=O)NCC(C)N(C(C=CC=CC)=O)C)cccc(C(N)=O)c1 C1(NC(c2cnc(C(C)C)[nH]2)=O)CCCN(C(=O)CCC2CC2)C1C C1(CC(=O)OC)CCC2CN(C(c3ccc(OC)nn3)=O)CCC2C1 [SH](=O)(=O)c1ccccc1N.CCC1=NOC(C(=O)N(CC(C)NC(=O)C)C)C1.N c1(C(N2CCC(CN(C(C(SC)SC)=O)C)C2)=O)ccc(C(C)(C)C)nc1 C1(N(C(CSc2nc(C)[nH]n2)=O)C)CN(C(c2c(C)noc2C(C)C)=O)CC1F c1(C(N2CCC3C(NC(c4cc5ccccc5[nH]4)=O)C32)=O)cnc2[nH]cnc2c1 c1(C(=O)NC2CCN(C(C3(C#C)CCC3)=O)C2)cccc2nc(C)sc12 Cc1cccc2cc(CN=C(NCC(=O)NC3CCC3)NC3CCC3)c(Cl)nc12 N1(C(CN2CC(C)(C)C2)=O)CCC(C2N(C(C3COCCO3)=O)CC2(C)C)CC1 C1(C(N(CC(CNC(c2nccc(C)n2)=O)C)C)=O)Cc2ccccc2N1 Cc1nsc(Br)c1C(=O)NCC1CC1NC(=O)C(C)n1cccc1 N1(C(CCCOCCOC)=O)CCC2CN(C(c3cc4sccc4[nH]3)=O)CC2C1 C(=O)(CCC1=CCCCC1)NC1(C2CC2)CCN(C(C(C)(C)N(C)C)=O)C1 C(=O)(CC1CCOc2ccccc21)NC1CC2C(NC(C=CC)=O)C(COC2)C1 C(=O)(C#CC1CCOCC1)N1C(C(N2CCC(C)(C#N)C2)=O)CCC1 C1(CC)(CC)CC(NC(C2(O)COC2)=O)CN1C(=O)C(=Cc1cccs1)C C1(CNC(c2nc(C)n(C)n2)=O)CC(C)CCN1C(c1ncn(C(C)C)n1)=O c1(C(=O)NC2CN(C(c3c(CC)nn[nH]3)=O)C(CO)C2)cc2nnn(C)c2s1 c1(-c2c(OC)ccc(Cl)c2)ccc(S(=O)(=O)NC2CC3CCC2N3)c(Cl)c1 C12(C(N3C(CC)CCC3)=O)CC(CO)(CN1C(=O)C(C)CCN(C)C)C2 N1(C(c2nn(CC)c(O)c2)=O)CCCC(N=c2ccc([N+](=O)[O-])c(O)[nH]2)CC1 c1(CC(=O)N)cccc2sccc12.c1(CC)conc1CC(=O)NC1CC1C S(=O)(=O)(c1cc(F)c(C)c(F)c1)N1c2ccc(CC)cc2CC1 CC(CC(F)F)C(=O)Oc1ccc(C(=O)O)cc1CN1CCCCC1 C1(NC(=O)CC2CNC(=O)O2)CCC2(CCCN(C(=O)Cc3cnns3)C2)C1 C1(C)(CC(=O)NC2(COC)CN(C(=O)CN3CCOCC3)C2)CCCCC1 c1(C2C(C=O)C2)ccccc1OC(F)F.CCC(C)CNC(c1csnn1)=O.N N1(C(CNC(C2(c3cc[nH]n3)CC2)=O)=O)CCCC1C(O)CO n1(CC=O)c(=O)oc2ccccc12.Cc1nc(C(=O)NC2CC(C)C2)n(C)n1 CC1CC(NC(=O)CCCC2CCCO2)CCN1C(=O)C(C)C1CCOC1 Cn1nnc2c(C(=O)NCCC3CCCCN3C(C3CC(O)C3)=O)cccc12 C(=O)(CCC(=O)N1CCC(CO)(CNC(=O)C=C2CC2)C1)NCC c1(C(C(=O)NCC2CCN(C(CCC)=O)C2)(C)C)cccc(F)c1.C(N)(=O)N c1(NC)ncccc1C(=O)NC1CCC(N(C)C(c2ccsc2OC)=O)C1 N1(C(CC(C)NC(=O)OC(C)(C)C)=O)CCCC(CCl)C1 C(=O)(CCC(C)(C)C=O)N.C(CCC(=O)NC1CC(C)C1)=CC.C(C)(C)C CCC(CC)C(F)C(=O)N(CC(=O)NCCN1CC(OC)C1)C(C)C c1(C=O)c(F)c(F)cc(F)c1F.C1(OC)CCC1C(=O)NCC1CCC1.N c1(C(N2CCC(N(C(CCCCC(=O)NC)=O)C)C2)=O)c(F)ccc2nc[nH]c12 N1(C(c2ccnc(C)c2N)=O)CC2CCCC2(NC(c2cnsn2)=O)C1 C(=O)(C(C)C(CC)CC)NCCC1(C(=O)NC(CCCC)C)CC1 c1(C(N2CCC(CCNC(c3cc(CN(C)C)on3)=O)C2)=O)cc(F)ccc1N c1(C(=O)NC2C=CCN(C(C(C)NC(C)=O)=O)C2)cc(C)cc(C)c1 C#CCCCC(=O)NCC=CC(=O)NCC(O)C(C)C c1(C(=O)N)cc2ccc(Cl)c(F)c2o1.CCC(C(=O)NCCC1CCC1)N(C)C C(=O)(CN=c1ccc(C#N)c[nH]1)N(C)CC1C2CN(C(=O)C3=CCCCC3)CC12 C(C(COC)C(=O)NC1(C)CCN(C(=O)C(C)(CO)NC(C)=O)C1)OC CCCCC(CC(=O)NCC1CCCCC1O)NC(=O)C(C)(C)C1CC1 N1(C(CCc2cc(C(=O)OC)[nH]c2)=O)CCOC(C)C1.C(=O)(C(C)N1CCC1)N N1(C(C(C2CC2)OC)=O)CC2CC(C1)CN(C(=O)C(O)C1CC1)C2 C1(c2n(CCCOC)nnn2)(Nc2cccc(C#N)c2)CCCOC2(CCC2)C1 C=C(Cl)CCC(=O)NC1CC(CC(=O)N(C)Cc2cc(C)nn2C)C1(C)C C1(C=O)CCN(S(=O)(=O)NC)CC1.CCCCN(C(=O)CC1CC(F)C1)C Cc1c(CC(=O)NCC2(F)CC(NC(=O)C3=CCCCC3)C2)oc2ccccc12 C1(CNC(CCC(C)C)=O)CN(C(=O)CC2CCCNC(=O)C2)CCN1C c1(C(C(N2CCN(C(C=C(CCC)C)=O)C3C2C3)=O)C)ccc(S(C)(=O)=O)cc1 c1(CC)cc(F)c(C(N2CCCC(N(C)C(c3ncccc3Cl)=O)C2)=O)c(F)c1 C(=O)(C(O)CCNC(c1csc(CO)n1)=O)N(C(C)CO)CC C1(C(=O)NC2(CCCNC(C3(C)CCSCC3)=O)CC2)COCC2(CCC2)O1 c1(C(=O)NCC(CNC(C2(C#N)CCCO2)=O)O)ccc2c(c1)CC(=O)N2 C1(O)(C(=O)NC(C)CCN(C)C(C2CC(CC3CC3)C2)=O)CCCCC1 N1(C(C2C(C)OC(=O)N2)=O)CCC=C(CNC(=O)CCCc2ncco2)C1 N1(C(c2c(C)n(C3CC3)nc2)=O)CCCC(NC(c2csc(C(F)F)c2)=O)CC1 c1(C(N2C(CN(C(C(C)NC(N)=O)=O)C)CCC2)=O)cccn2c(C)nnc12 c1(C(N2CCN(C(C3NC(=O)OC3)=O)CC2C2CC2)=O)cc2n(n1)CCCC2O c1snc(Cl)c1Cl.c1(COCC(=O)NCCCSC2CC2C)ccccn1 N1(CC(CC)OC)CC2(C)CN(C(=O)Cc3cnn(C(C)(C)C)c3)CC2(C)C1 c1(CCC(=O)NCC(C)NC(C=C(CCC)C)=O)cc(C)no1 N1(C(C(N2CC(O)(c3cscc3CO)C2)=O)=O)CC2(CCC2)C1c1ccccc1 C1(NC(Cc2c(C(C)C)con2)=O)CCOCC1NC(C1CC2CCC1C2)=O C1(OC)(CNC(C2CC(=O)C2C)=O)CCN(C(=O)C(F)OC(F)(F)F)CC1 C(=O)(C#CC(C)(C)CNC(C1(C)CC1)=O)NC(C#C)C(C)(C)C C1(C(N2CC(NC(=O)COc3ccc(Cl)cc3)C2)=O)CCn2nncc2C1 N1(C(CSCc2nc(C)sc2)=O)CCC(O)(C(N2CCCC2CCO)=O)CC1 Cc1ccccc1C1(C(=O)NC(CNC(C23CCC2CC3)=O)C(C)C)CC1 c1(C(=O)NCC2COCCN(C(c3cc(C)[nH]n3)=O)C2)cc(P(C)(C)=O)ccn1 N(S(=O)c1ccccc1F)c1c2[nH]cc(COCC)c2ccc1 c1(OC)nccc(C(=O)NCC2CN(C(c3ccsc3OC)=O)CCO2)n1 N1(C(CNS(N)(=O)=O)=O)CCN(C(=O)Cc2cccc(CCC)c2)CC2(CC2)C1 C1(O)(CNC(c2c(OC)c[nH]n2)=O)CCCN(C(C2(C)CC2(F)F)=O)CC1 NC(=O)C(CNC(=O)CCOc1ccccc1)Cc1ccccc1Cl C(CCCCCNC(=O)CC1CC2(COC2)C1)NC(C1N(C(C)C)CCC1)=O N1(C(c2cc(C)[nH]n2)=O)CC2CCCC2(NC(=O)C=Cc2ccc(Cl)s2)C1 c1(C(N2CCC(NC(CCC(=C)Cl)=O)(CO)C2)=O)cccc(F)c1Br C1(C(N2C3CC4C(C2CC3)C4)=O)Cc2ccccc2S1(=O)=O.C1(C(=O)N)CCC1 C1(CCC)CN(C(=O)CC=C(Cl)Cl)CCN1C(C1CC1CC)=O c1(CN2CCN(C(=O)NC(c3ccccc3)=O)C3C2C3)cc(F)c(F)c(F)c1 c1(C(=O)N)c(Cl)csc1Cl.c1(COC)csc(C(=O)N(CCC)C2CC2)c1 C1(C(=O)NCC(O)CNC(c2coc(O)n2)=O)(NC(N)=O)CCCCC1 Cn1ccc2cccc(-c3c[nH]c4ccc(C(=O)NC5CCC(F)(F)C5)cc34)c12 C1(C)(CCC)CCCN(C(C2CCOCC2NC(=O)C=C(CC)CC)=O)C1 CCC(CC)CC(=O)N1CC(CCNC(=O)Cc2ncn(C)c2C)OC(C)C1 N1(C(C2(C(CC)=O)CC2)=O)CCCC(C(=O)NC(C2CCCCC2)CO)CC1 C(=O)C(C(C)C)n1ccnc1.C1(CC(=O)NC(C2CC2)C)(CC)CCC1.N n1(CC=O)cnc(C(F)(F)F)c1.N1(CC)CCC1C(=O)NCC1CC1 c1(NCCC(CCC)O)cc(=NC(CC)CC(C)O)[nH]c(C(F)(F)F)n1 C1(OC2CN(C(C3C(SC)CCC3)=O)C2)CCN(C(C2CCS(=O)CC2)=O)CC1 CC1CCN(CCC(=O)N(C)CC2CC(F)CN2C(=O)CNC(N)=O)CC1 C(=O)(C(CC(N)=O)NC(=O)C(C)n1ccnn1)NCC(CC)O C1(C(=O)NC(CC)CN2CCCC2)C=CCN(C(=O)C(CO)OC)C1 C(=O)(C(C)(N)C1CCC1)NC(c1csc(C2CCCO2)n1)C N#CC1(C(=O)NCC2CCC2)CC2CCC1CC2.C(c1ccco1)=CC(=O)N [N-]=[N+]=NCCCC(=O)NCCC1CCCN1C(c1cc(F)n[nH]1)=O N1(C(C=CCOC)=O)CC(CC(=O)NC2CCOCC2C)CC1C C1(S(=O)c2ccccc2)(C(=O)NCc2ccc3c(c2)CNC3)CCC1 c1(OCC)ncccc1C(=O)N(C1CCCN(C(=O)CCCc2cnn[nH]2)C1)C C(N=c1cc(NCCCc2ccc(Br)cc2)nc[nH]1)c1c(OC)ccc(Cl)c1 c1(C(N2CCC(F)C2)=O)cc2cc(F)ccc2o1.C(C)(CCC(=O)NC)OCC N1(C(CS(C(C)C)(=O)=O)=O)CC2CN(C(=O)C(C)(C)CCC#N)CC2(C)C1 c1(C(N2CC(O)C2)=O)c(C)nn(C)c1-n1cncn1.C#CCC(O)C(=O)N(C)C c1(C(N2CCCC2)=O)cc(C(N)=O)ccn1.C1(COC)CC1CC(=O)N.C c1(-c2nc(C(C3CCOC3)OC)n(-c3ccc(C)c(C)c3)n2)ccc(F)c(C)c1 C(=O)(C(C#N)C(C)C)NC1C(NC(c2c(C)nn(-c3ccccc3)c2)=O)CCC1 c1(C=O)ncnc2ccsc12.c1(OC)cc(C=CC(=O)NC2CC(C)C2)sn1 Cc1c(C(=O)NCCCn2cc(C3CCCS(=O)(=O)C3)nn2)cncc1Br C(=O)(C(F)(F)C(F)F)NC(C)C(CO)NC(=O)C(C)Cc1ccc(O)cc1 CCC(COC(C)(C)C)N=c1nc(N2CCCN(C)CCC2)c2c([nH]1)COC2 c1(CC(N2C(CNC(=O)CC=C(Cl)Cl)CC2)=O)ccc2ncccc2c1 CC1(C)CC(NC(c2n[nH]cc2[N+](=O)[O-])=O)CN(C(c2cc(CF)on2)=O)C1 c1(C(=O)NC2CC(F)(CNC(C(CC)SC)=O)C2)cc2cc[nH]c(=O)c2s1 Cc1c(NC(c2n[nH]cc2-c2cccc(O)c2)=O)cccc1N C1(NC(CN2CCN(Cc3ccc(C)o3)CC2)=O)CCC2(CC1)OCCO2 c1(NC(c2ccc(Br)cc2O)=O)cccc(F)c1C(=O)Nc1nc(Cl)nc(Cl)n1 c1(C(=O)N)ccc(C)cc1N=[N+]=[N-].N1(C(C=CC=CC)=O)CC(O)(CC)C1 CC(C)(C(=O)N1C(CO)CC1CO)C(F)F.C1CCC(=O)N1 N(C(=NCCS(=O)(=O)C(C)C)NC1CCS(=O)(=O)C1)Cc1c(OC)cccc1 C(=O)(C1=NOC(CNC(C2CCCSC2)=O)C1)N(C1(CCO)CC1)C C1(C(N2CCC(CC=C)(NC(c3cnc(OC)o3)=O)C2)=O)CC(O)C12CCC2 Cc1nc(C)c(C)o1.C1(CC=O)CC(C)N(C(C2OCCC2C(C)C)=O)C1.N CC1(C)CCC1C.C1(F)(C=O)CCCCC1.C(=O)(CC(C1CC1)C1CC1)N CN1C(=O)N(C2CC=CC2)C(=O)C1c1ccc(Br)cc1F N1(C(C(CCOC)C)=O)CC2(CCC2)CC1C(=O)OC Cc1csc(C)c1C(N1CCOC(C(C)NC(C2CCCC(=O)C2)=O)C1)=O C(=O)(CS(=O)(=O)C1CC1)N(C1CCCCC1)CCNC(CC1CCC(C)O1)=O C1(CNC(NC(C=C)C)=NCc2c(Br)nnn2C)CCC2(CC1)OCCO2 C(CC(=O)NCC1CC(F)CN1C(c1cc[nH]n1)=O)(C(F)(F)F)OC C1(C=O)CC2(C1)CC(F)(F)C2.C1(CC=C)CCCN(C(=O)CCC(F)(F)F)C1.N c1(C(N2C(C)CC2C(N2CCCC2CC2CC2)=O)=O)cc(CO)ccn1 c1(C(N2CC(F)CC(C(=O)Nc3cc(C)c(Br)cn3)C2)=O)cc(Br)c(F)cc1F C#CCC(C)(CC)C(=O)NC1CCOCC1NC(c1nnsc1SC)=O CN1CCN(C(c2ccc(C(N)=O)nc2)=O)c2cnccc21 C(=O)(CCCC(C)(C)O)NC(C)CC(=O)c1ccco1 c1(C(N2C(C(C)NC(CCCOCC=C)=O)CCCC2)=O)ccc(C)c(F)c1 C(CC(F)F)(C(=O)N(C)CCC1CCCO1)N(C(c1ccc(C)[nH]1)=O)C CCCC(C(O)C(=O)NC(CO)C(=O)OCC)NC(C1CNC(=O)N1)=O c1(CNC(c2cnc(C(C)O)s2)c2nnnn2C2(C)CC2)ccc(O)nc1 Cc1nn(C)cc1CCC(=O)NC1CCC(N(C(=O)C2=CCSC2)C)C1 N1(C(CCSC)=O)CC2CCC2(CCNC(c2cc(-c3cn(C)nn3)on2)=O)C1 CC1(O)CCN(C(c2cc(CNC(=O)C(F)C(C)(F)F)ccn2)=O)CC1 Cc1occc1CC(=O)NC1CC(O)C1CC(N1CCC(OCCO)C1)=O N1(C(C2(Cl)C(C)(C)C2)=O)CCCC(C2(NC(C3CC4(CCC4)C3)=O)CC2)C1 N1(C(C(C)N(CCC)C(C2CC3CC2CC3=O)=O)=O)CCc2c[nH]nc2C1 C1(CCC)CN(C(=O)C(=O)N(C)C)CC1NC(C)C(c1ccccc1)C OC1CCCC2CN(CC3CCC=CO3)CCC12 C1(C(=O)NCCOC2CN(C(Cc3cn(C)nc3)=O)C2)CCCC(F)C1 CCC(C)CC(C)C(=O)N1CCCCC(NC(=O)C(O)Cc2ccccc2)C1 C1(NC(C2(COC)CC2)=O)CC2(CCCCN2C(C2CCCC23CCC3)=O)C1 N1(C(C2(OC)CCOCC2)=O)CCC(C)N(C(C2CC23CC(C)(C)C3)=O)CC1 CCC(C)C(C)C(=O)NCC1CC(C)N(c2ncc(Cl)c(O)n2)C1 CC(C)C(CNC(=O)C(C)c1ccsc1)NC(c1coc(C2CCOCC2)n1)=O CCC(C)CCCCC(=O)NC1CN(C(=O)C(F)C2CCOC2)CC2(CC2)C1 C(CCC1(C)CC1)(C(=O)NCCOC)N(CCCCC)C(C)C.C1CCOCC1 Cc1csc2c(=NCC(C)N(C)C(c3cc([N+](=O)[O-])cn3C)=O)[nH]cnc12 N1(C(c2cc(C)c(C#N)[nH]2)=O)C2CCC1CN(C(c1n[nH]c(C)c1Br)=O)C2 C#Cc1cncc(C(=O)NC(CNC(c2ccc(Cl)nc2O)=O)C2CCC2)c1 c1(NC(c2ccc(C(C)(C)C(N)=O)cc2)=O)cc(S(C)(=O)=O)ncn1 c1(C(C(=O)NCCN(C(=O)C(C)(CC)CO)CCC)C)ccc(Br)cc1F C1(NC(C(CC(C)C)C)=O)CN(C(c2ccc(F)c(N)c2F)=O)CC2(CCC2)C1 C1(CC)C(NC(=O)C(C(C)C)n2cccc2)CCN1C(c1cc(C)c(C)s1)=O Cc1cc(C(=O)NC(C(=O)N(CC(O)CF)C)C2(C)CC2)ccc1O C1(C(N2CC3(CC(NC(C(C)(C)CCC#N)=O)C3)C2)=O)CCc2ncncc2C1 C(=O)(C(C#N)C(C)(C)C)NCC1CCN(C(C2(C)CCC(O)CC2)=O)CC1 Cc1cc(C(=O)NCC=CC)c(N)c(Cl)n1.c1(C=O)cn(C2CCC2)nc1C C#CCCCC(C)C(=O)N(C1CN(C(=O)CCc2ccc[nH]2)CC1(C)C)C C1(CC(N2CCCC2)=O)CC(O)C12CCC2.C(C(=O)NCC)N(C1CCC1)C N1(C(CC=CCC)=O)CCCC(C)C1CNC(c1ccc(C)nc1OC)=O C1(C(N(C)CC2(O)CN(C(C(CCCOC)C)=O)C2)=O)CC2CC1CC2(F)F N1(C(C(C)SC(C)C)=O)CC2CC2(NC(c2ccc(Cl)cc2)=O)C1 C(=O)(CC(F)(F)C(F)(F)F)N1C2C(NC(CC3CCC(C)(C)CC3)=O)C(CC2)C1 Cc1ncc(C(F)(F)F)cc1C(=O)NCC(O)CNC(C1(C#N)CCC1)=O CCCC(C#N)C(=O)N1C(C(N2CCN(CCO)C(=O)C2)=O)CCC1C1CC1 CC1(NC(=O)CC2(O)CCCOC2)CCCCC1C(=O)NCC1CC=CC1 C(=O)(CCS(=O)(=O)Cc1c[nH]nn1)N(CC(C1CCC1)OC)C.c1cocn1.C Cc1cc(C(N2CCC(C(C)CNC(=O)CC(C)C)CC2)=O)c(F)cc1F c1(C(N2CC(NC(C(CCC)C)=O)C(CC3CC3)C2)=O)cc([N+](=O)[O-])ccc1Cl c1(NC)cc(C(N2CCN(C(c3sncc3C)=O)CC2C)=O)cc(Cl)n1 CC1COc2c(C(=O)NCc3ccccc3CN(C(=O)C=C(Cl)Cl)C)cnn2C1 N1(C(c2c(C)cc(C)nc2)=O)CCC2(C1)CN(C(C13CCC1CC3)=O)CCO2 C1(C(N2CCN(C(c3n(OC)cnc3C)=O)CC2)=O)CCC(=C(F)F)CC1 C1(S(=O)(=O)c2ccccc2)(C=O)CC1.CC(C)C(C)C(=O)NC1(C)CCC1.N Cc1ccc(=NCCC(=O)N2CCOC(CN(C(=O)C(O)C(F)(F)F)C)C2)[nH]c1 CCC(C)CC(=O)NCC1(NC(c2sc(-n3cccc3)nc2C)=O)CC1 CC(C)C(F)(CNC(=O)C(C1CCCCC1)F)C(=O)N(C)Cc1nccs1 C1(CNC(C2(OC)CCOC2)=O)CCCC2CN(C(c3cn(C)nc3C)=O)CC12 N1(C(C2CN(C(c3ncn(CC)n3)=O)C(C)CC2)=O)c2ccccc2CC1C Brc1ncc(C(c2nnnn2CCc2ccccc2)N)s1.c1(CC2CC2)cscn1 O=C(NNC(=O)N1CCC(c2nnc(O)o2)CC1)c1ccccc1Br c1(C(N2C(C3CCN(C(CC(C)C)=O)C3)CCC2)=O)cc(Cl)cc(Cl)c1 C1(C(N2C(C3(C(N(C)Cc4nc(C)sc4)=O)CC3)CCC2)=O)C2CCC(F)C12 N1(C(C(=O)NCC)=O)CC2C(C(=O)NC(c3cccc(F)c3)C)C2C1 c1(C(=O)NCCNC(c2nc(COC)sc2)=O)nn(C)c2c1COCC2 N1(C(C(C)=C2CCCC2)=O)CCCC(C2CC2NC(c2sccc2C)=O)C1 C1(CC(N2CCC(O)C2)=O)CC(=O)NC(=O)C1.C(c1cscn1)=CC=O.CC Cc1nc2n(n1)CCN(C(c1ccc(CC(C)(C)O)s1)=O)C2 Cc1cc(NC(N2CCC(C)(C)C2C)=O)n2nc(C)c(Br)c2n1 c1(C(=O)OCc2nccn2C(F)(F)F)nncc2ccccc12 C1(CC=O)CCC(=O)CC1.C1(C(N(CCCCC)CC(N)=O)=O)CCOC1C c1(C(=O)NCC2COCCN(C(c3c(C)coc3)=O)C2)cccc(C=C(F)F)c1 N1(C(CSc2ccc(OCC)cc2)=O)CCN(C(c2oncc2SC)=O)C2CC12 c1(NC(=O)CC2CCN(Cc3ccc(I)cc3O)CC2)nc2cc(F)ccc2s1 N1(C(c2c(CNC(=O)OC(C)(C)C)cccn2)=O)CC2(CCC1CO)CC2 CN1CCN(C(=O)C2=COCC2)CC1CNC(=O)CSC1CC1 Cc1cc(Cl)cc(C(=O)NCC2(C)CCCN(C(c3coc(Cl)c3)=O)C2)c1N C1(CC)OCCCC1C(N1CCC(CC=C(C)C)CC1)=O CC(CN(C)C)CC(=O)N(CC(C)CNC(c1c[nH]nc1C(F)(F)F)=O)C c1(NC2CCCC(C(C)C)C2)ccc(S(=O)(=O)NCCCC(C)(C)C)cc1F C1(CNC(C(C)Cc2ccc(C#N)cc2)=O)CCc2cn(C)nc2C1 C(=O)(CC1CCCc2ccccc21)NCCCNC(CN(S(N(C)C)(=O)=O)C)=O N1(C(c2ccc(CC)cc2)=O)CCC2(NC(=O)CCS(C)(=O)=O)CCCCCC12 C12(CNC(CSCCC#N)=O)CC(CN1C(C1CC1)=O)C2.c1ccsc1 N1(C(CSCC#C)=O)CCCCCC1C(=O)N(CCOC)CC N1(C(C(COC)C)=O)CC=CCC1C(=O)NCc1ccncc1F C(=O)(C(O)CC(F)(F)F)N(CCC(c1cccs1)NC(c1cncc(Cl)c1)=O)C C(=O)C(F)C(F)(F)C(F)(F)F.c1(OC)c(C(=O)N(CC)CC)cnn1C.N C(=O)(C1=CCc2ccccc21)N.CC(C)(C)C(C(=O)NC1(CC)CC1)C1CCC1 C1(C(=O)NC(c2cnsc2)C)(CC)CCN(C(=O)Cc2cccc(C)c2)C1 N1(C(C2(CC=C)CCC2)=O)CCC2CCC(C1)N2C(=O)C(C)Cc1cnc[nH]1 C=CCC(CNC(c1csc(C2CCCO2)n1)=O)NC(c1ccccn1)=O C1(OC)CN(C(=O)CNC(c2ccccc2)=O)CC1.c1(CC=O)cnsc1.C CC1=C(C(=O)N(CC)C2CC2)C(=O)OC1(C)C.c1(C(=O)N)cc2sccc2s1 Cc1ccc(O)c(C(N2CCCC(NC(C3CCC34CCC4)=O)C2C)=O)c1 S(=O)(=O)(c1cnn(C)c1)N1CC(C)C(NC(=O)C=Cc2cccc(O)c2)C1 CC1CCOC1CC(=O)NC1CCC(CNC(c2scnc2C(F)F)=O)C1 N1(C(c2ccc(CC)nc2)=O)CCCC2(CCCCN2C(C2CC2(F)Cl)=O)C1 N1(C(C2C(C)(C(F)F)C2)=O)CCN(C(=O)CCOC2CCCC2)CC1 O=C1CC(C(N2CCCC(N(CCO)C(c3ccoc3Cl)=O)C2)=O)NC(=O)N1 N1(CC)CCCC1CC(N1CC(n2cc(C)nn2)C1)=O.C1(C=O)CC(C)CO1.N N1(C(COc2ccc(C#N)cc2)=O)CCC2(CCOC2)C(CNC(=O)C2CC2)C1 C1(N(CC(N2CCCC2)C)C(=O)NC23OCC(C)(C2)C3)CCC(O)C(O)C1 c1(C(=O)NCC(C)NC(=O)CC2CCC(=O)C2C)ccc([N+](=O)[O-])o1 N1(C(c2ccn(C)c(=O)c2)=O)CC(NC(c2csc(=N)[nH]2)=O)CC12CCOC2 CCCCC(=O)C(=O)NCCCN(CCCNC(c1nc(C)n(C)c1C)=O)C O=S1(=O)CC2CCN(Cc3ccc(C4CCCCC4)s3)CC2C1 Nc1c(C(N2CCN(C(C3CC=CC3)=O)C(CF)C2)=O)cc(Cl)cc1Cl C=C(C)CCCC(=O)N1CC2CC1CN2C(=O)C(c1cccc(F)c1F)(F)F c1(CC)ccc(C(=O)NC2(CO)CCN(C(=O)C=CC3CCC3)C2)cc1O C12(C(N3C(C(N4CCC(C(CC)CC)C4)=O)CC3C)=O)CC1CNC2=O C1(CC(N2C(C)(CNC)C=CC2)=O)CN(C(=O)CO)CCC1C.C1CCCC1 c1(CCC(=O)NCC(CNC(c2cc(C)no2)=O)O)ccccc1C(F)(F)F C1(CC=C)CCCN(C(=O)Cn2nc(C(F)F)cc2C)C1.C1(C(=O)N)C=CCC1 C(=O)(CC1=NNC(=O)C1)N1C(C)(CNC(c2ccc(C)cc2F)=O)CCC1 C1(C(=O)OC)CCN(C(=O)C(F)CC(C)(C)NC(=O)CCCC)O1.C(C)(=O)N N1(C(CN2CCC(OC)C2)=O)CC2(C(=O)NCC3(O)CCOCC3)CC1CCO2 c1(OC)nccc(C(=O)N(CCCNC(c2csnc2Br)=O)C2CC2)n1 c1(C(=O)NCCN(CC(C)O)C(C2CC2F)=O)cc(O)c2ccoc2c1 c1(C(N(CC(C)C)C)=O)cc2c(=O)[nH]ccn2c1.c1(C(=O)N)cc(F)cc(Cl)c1 C1(NC(C(C)OCCOC)=O)CCN(C(c2ccc(C)c(F)c2)=O)C12CC2 C=CC(CCC)CC(=O)N1CC(C)N(C(=O)C(=O)NCC)CC1C N1(C(=O)C2=COCC2)CC2OCCN(C(c3cncc(F)c3)=O)C2C1 C1(NC(c2cc(O)no2)=O)CCCCC12CCN(C(=O)C(O)C1CC1)CC2 C(=O)(C1CSc2ccccc21)NC1CCN(C(c2c(OC)cncc2)=O)C1(C)C c1(CCCCC)ccc(C(=O)NCC23CC(C2)C3)o1.c1(C(=O)N)nccn1C N1(C(C2OCC(C)(C)C2)=O)CCCC(C)(NC(=O)C=Cc2cccc(CO)c2)C1 C12(NC(c3csc(CO)n3)=O)CCN(C(c3cnn4ccsc34)=O)CC1C2 c1(C(=O)NC(C2CCN(C(COc3cc(C)oc3C)=O)C2)C)cc(F)ccc1Cl c1(C(=O)NCC23C(CN(C(C(CC)O)=O)C2)C3)ncc2c(F)cccn12 c1(OC)cccc(NCCNC(=O)Cn2nccc2C)c1[N+](=O)[O-] c1(C(N2CC(NC(CSC(=N)N)=O)C2)=O)ccc(COCCO)cc1 n1(CC)nc(C2CC2)cc1C=O.C1C=CCN(C(=O)CC2COC(C)(C)C2)C1 c1(CC(=O)NCC2(C(C)(C)O)CN(C(C=NOC)=O)C2)cccc(C)c1F Cc1ncccc1CC(=O)NC1(CF)CCN(C(=O)C(c2c(C)n[nH]c2C)C)C1 c1(C(=O)NC2C3(CC(NC(CC(C)c4ccncc4)=O)C3)C2)cccc(Cl)c1N C(=O)C1=NOC2(CCC2)C1.C1(N(C)C(c2cccnc2C)=O)CCCC(C)(C)C1 Cc1cc(C(=O)NC(C)(CNC(C2CCCOC2)=O)C(C)C)c(Br)cn1 Cc1ncc(C(N2CCC2)=O)c(C2CC2)n1.c1(C(=O)N)ccc(C(C)(C)C)cn1 c1(C(N2CCC(CC(=O)OC(C)(C)C)CC2)=O)cc2c(s1)CCN(C=O)C2.O c1(C(=O)NCCC(CNC(C2ON=C(C)C2)=O)O)csc2cccnc12 C1(CN(C)C(c2nonc2N)=O)CCN(C(=O)C(C)(C)CC2CCOCC2)CC1 C(=O)(CC1COc2ccccc21)NCC1(CNC(CCCCCC)=O)CC1 c1(CC(=O)N(CCNC(CC(C)F)=O)CC2CC2)ccc2c(c1)CCCO2 N1(C(CCCC(=O)N(C)C)=O)CC(N=[N+]=[N-])CC1C(N1CCOCC2(CC2)C1)=O CNS(=O)(=O)N1CCN(C(C2CCCN2C)=O)CC1 c1(C(=O)NC(C2(O)CN(C(C3CCCCC3O)=O)C2)C)cc(Cl)nc(Cl)c1 c1(C(=O)NCC(C(=O)Nc2cnn(C)c2C(N)=O)O)cc(C#N)ccc1N N1(C(C(CC)NC(N)=O)=O)CCC(C)(C)C(C)C1.c1(CC(=O)N)[nH]cnc1C C1(CCNC(=O)C=CC2CCCO2)CCN(C(=O)CO)CC1.c1cccnc1.C C(CN=c1nc(O)c2c(ncn2C)[nH]1)C1(O)CCN(C(CSCCCC)=O)CC1 C1(NC(C2CC(CNC(=O)CN3CC=CC3)OC2)=O)CC12CCCCC2 N1(C(C(C)N(C(=O)Cc2csnc2C)CCC)=O)CCC(C)(C2CC2)C1 N1(CCNC(c2cnc(S)nc2)=O)CCN(C(=O)CC2OCCO2)CC1 c1(CC)nc(C)c(C(=O)NC2CCN(C(=O)CC(C)(O)COC)C2)c(C)n1 C(=O)(C#CC1CCCCO1)N(C(CN(C(c1c(C#C)cnn1C)=O)C)C)C CC1(C)CCCOC1C(=O)NCC(CC1CC1)C=O.c1cncc(C(N)=O)c1.N c1(OC)ccc(C(=O)OCc2cnn(-c3ccccc3)c2C)cc1C C1(COC)(NC(C2CC2Cl)=O)CN(C(c2cnc(CC(C)C)s2)=O)C1 c1(C(=O)NCC2CCC(N(C(c3[nH]cc(C)c3)=O)C)CC2)cc(N)c(C)cc1C N1(Cc2onc(C(C)SCC)n2)CC=C(c2cccc(F)c2)CC1 C1(CC=C)(C(N2CCC2c2ccccc2)=O)CCCN1C(=O)C(O)CCN(C)C Cc1c(C(=O)N(CCCNC(=O)CC2COCCO2)C)cc(C(C)(C)C)n1C c1(CN(C)CCN(C)C(C2(C)CC2F)=O)ccc(OC(F)F)c(OC(F)F)c1 CN1N=C(CC(=O)N2CCC(C(=O)NC3CN(C)C(C)(C)C3)C2)CC1=O N1(C(C(C)CC2CCCC2)=O)CCC(C(=O)NCC(=O)NCCO)C(C)(C)C1 C(C(C)(F)C(C)(C)F)n1cc(C2N(C(C(COC)O)=O)CCC2C)nn1.C1CC1 CC1CCN(C(=O)CN2CCNC(=O)C2)C1CNC(C1CCC(=O)N1C)=O Cc1n[nH]c(=NC(C)CNC(C2(Oc3ccccc3)CC2)=O)s1 N1(C(C2CN(OC)C(=O)C2)=O)CCC2C(C1)CN2C(=O)Cc1cc(C)no1 C1CN(C(C2CCC(C(F)(F)F)O2)=O)C1.CCS(=O)(=O)NCC(=O)N.C C12(NC(=O)CC3(O)CCOCC3)CCCC1N(C(=O)CN1CCCCC1=O)CC2 C1(C(=O)N)CCC(=C2CCC2)CC1.c1(OC)cc(CC(=O)NC(C)CC)on1 N1(C(C2(CCC)CCC2)=O)CCOCC(F)(CNC(=O)CN2CCCCC2=O)C1 C1(C(N2CC(F)(C(=O)NOCC(O)C(C)C)C2)=O)(COC)CCCC1O CCCC(C(=O)N(C(C)(C(=O)NC1CC(c2ncc[nH]2)C1)C1CC1)C)OC C12(C(N3C(CNC(=O)CCC4CC4(F)F)CCC3)=O)CCC(CC1F)C2 CC1=C(C(=O)N2CCC(CCNC(=O)C(N3CCC(O)CC3)C)C2)CCS1(=O)=O CC1=NOC(C(=O)N(C)CCNC(=O)Cc2ccc(Br)s2)C1 c1(C(=O)N)ccco1.C(=O)(CC)N(CCC)CC.[SH](=O)(=O)CC.C1CC1 N1(C(C(C(C)O)N(C)C)=O)CCC2(CCCN(C(c3cc(Cl)cs3)=O)C2)C1 C(CC(C(C)(C)C)NC(c1cnc(C)cn1)=O)N(C(CC(=O)OC)=O)C N(C(=NCCC1CC(F)C1)NC1CCS(=O)(=O)C1)CC1CC(C)(C)C1 C1(C(N(C)C)=O)COCC(C)(C)O1.N1(C(CN(CCOC)C)=O)CCC(O)C1 N1(CC(=O)NC(CNC(C)=O)C)CC(C)C1 c1(C(=O)NCCCOCCC(=O)NCC2CC(C)C2)cn(C)c(=O)n1C Cn1nnc2cc(C(=O)NC3(C)CCCN(C(c4ccccc4F)=O)C3)sc12 C(C(C)(C)C(=O)NC1CCC(N(C)C(c2nc(Br)c(C)s2)=O)C1)SC c1(CC)cc(C(=O)NCCC2CN(C(c3nocc3Br)=O)C2)cc(O)n1 N1(C(CC2C(C)C2)=O)CCCC(C)C1CNC(c1cnn(CC2CC2)c1)=O CCCC(C(=O)N1CCC(CC(=O)NC(C(=O)OC)c2ccoc2)C1)OC N1(c2nccc(-n3c(C)cc(C)n3)n2)CCC2(NC(=O)C=CCF)CCCC12 C1(n2cc(C3(C#N)CC3)nn2)CCCN(C(C23CCCC2C3)=O)C1 C1(C(=O)NCCOCCN=[N+]=[N-])CCCN(C(=O)C(F)n2ccnc2)C1 CCC(C(=O)NC1CN(C(c2ccn3ccnc3n2)=O)CC1O)C(F)(F)F C(c1ccccc1F)=CC(=O)N.C1(C(=O)NC2CCC2)(OCC)CCSCC1 Cc1c(C(=O)N(C)CC2COCCN2C(=O)C(n2cc(Cl)cn2)C)cccc1Cl c1(NC(=O)NCC2(C)N(C(CC(CCC)C)=O)CCC2)ccc(S(C)(=O)=O)cc1 C1(NC(C(C)(C)OC(C)=O)=O)CCCC(C(=O)NC)CC1.c1ncc(C)o1.C C1(CC(N)=O)(NC(CC(C=C)C)=O)CCN(C(c2cc(C)n(CC)c2C)=O)CC1 C1(O)(C(C)CNC(=O)Cc2cnc[nH]2)CCN(C(c2cnc(C3CC3)s2)=O)C1 Cc1cc(CN2CC3C(C(=O)NCc4cn(C)nc4C)C3C2)ccc1Br Cc1nc(C(N2CCC(N(C(=O)CSc3ccc(F)cc3F)C)C2)=O)c(C)n1C CC(C)S(C)(=O)=O.c1(C=O)sccc1CC#N.C1(N(C)C)CC(CC(=O)N)C1 C(=O)(C1=C(C)CCOC1)NC1CCCC(CC(=O)Nc2cccc(SC)c2)C1 CCCC(CC)C(=O)NCC1(O)CCN(C(c2oc(C3CCC3)nc2C)=O)CC1 c1(CS(C)(=O)=O)nc(C(N2CCCC2)=O)cs1.c1(C=O)cnc(C2CC2)o1.N c1(C(=O)NC2CCN(C(C=C(C)Cl)=O)CC2C(C)C)c[nH]c2cc(Cl)ccc12 N1(C(C(n2ncc(C)c2)C)=O)CC=C(CCNC(=O)CCc2cncs2)CC1 Cc1cc(C(=O)NOCC(=O)NC(C2CCOC2)(C)C)cnc1C c1(C(N2CCC(CNC(C(CC)(C)O)=O)C2)=O)cc(C(F)(F)F)ncc1OC C1(COC)CN(C(=O)C(O)CSC(F)(F)F)CCN1C(c1ccc(O)cc1)=O c1(C(=O)NCC2C(NC(c3ccn4c3CSCC4)=O)C2)cccc2[nH]ccc12 Cc1noc(C(N2CCCC2C(C)NC(=O)C=Cc2ccsc2)=O)c1C N1(C(C2CCc3ccnn3C2)=O)CC2CC(C1)C2N=c1ccn2c(Br)cnc2[nH]1 C(CCC)(CCCNC(=O)CCC1CC1(C)C)NC(CCN(CCCCC)C)=O c1(N2C(C)CCC(OC)C2)ccc(S(=O)(=O)N2CCC=CC2C(=O)OC)cc1F c1(CC(=O)N(C2CCCCC2)CC)cccc(O)c1F.CC1(C)CC1(Cl)C(=O)N CCC(C)C(C)C(=O)NCc1cccc(OCC(=O)NC2CC(O)C2)c1 Cc1ccccc1CC(=O)NCC1CC(O)CN1C(c1ccc(CCF)cc1)=O N(C(=NCCCc1cccc(Cl)c1)NCC1CC(C)(C)CO1)CCSC CCCCCC(O)CNC(C1(NC(c2nc(C)ccc2C)=O)CC1)=O N1(C(CC(C(F)(F)F)OC)=O)CCC2CCN(C(=O)C=C(C)c3ccsc3)C2C1 C(c1cnccn1)=CC(=O)NC(CC)CNC(=O)Cc1cnc(C(C)C)[nH]1 c1(C(=O)NCC(CC)(N)CC)cc(Br)ccc1Oc1ccncc1 C1(C(N2CCC(N(C(c3cnc(O)n3C)=O)CC)C2)=O)CCOC(=O)CC1 c1(NC(C2CC(NCc3cc(F)ccc3F)C2)=O)cn2c(Br)cccc2n1 C1(C2CCCN(C(=O)C(O)c3ccsc3)C2)(NC(c2c(CC)ncnc2)=O)CC1 c1(C(=O)NC2C(NC(C(C)N(C)C)=O)CCCC2)cc(Cl)c2c(c1)OCCCO2 c1(C(N2CCCC(CN(C)C(C3(C(N)=O)CCC3)=O)C2)=O)cccc2ccsc12 Cc1nc(C(N2CC(C3(NC(c4cnc(C#N)s4)=O)CC3)C2)=O)c2ccccn12 N1(C(CC(C)(F)F)=O)CC(NC(c2ccc(Cl)c(F)c2)=O)C2(CCOCC2)C1 Cc1c(F)ccc(CN2C(C(=O)Nc3c(F)cc(Br)cc3F)CC3CC23)c1F c1(C(N2CC(CNC(C3C(C)N(C)CC3)=O)C2)=O)cc(Cl)cc([N+](=O)[O-])c1O N1(C(CCn2c(C)ncc2)=O)CC=C(CC(=O)NC2CCCC2C)CC1 N1(C(CC2OCC(C)(C)C2)=O)CC(NC(=O)CCC2CCOCC2)CC2(CC2)C1 N1(CC(=O)N(C2CCN(C(C3ON=C(C)C3)=O)C2)C)C(=O)NC(C)(C)C1=O C1(NC(c2ccns2)=O)CC2(C1)CN(C(c1cccc(=O)o1)=O)C2 C#CC1CCC(CNC(=O)C(CNC(=O)CCc2ccn(C)c2)C(C)C)CC1 C1(C(=O)NCC(C)(O)CNC(=O)C)(CC)CCCO1.c1ccco1.C=O N1(C(c2cncc(C)c2Cl)=O)CCN(C(=O)Cn2ccnc2C(C)C)C2(CC2)C1 CCCS(=O)(=O)C(C)C(=O)N1CCC(O)(CNC(C2(C3CC3)CC2)=O)C1 C(CCC(CCC)NC(C1(Br)CC1(C)C)=O)NC(c1n(CC#C)ccc1)=O CC(C)CCC(=O)NC1CCC(NC(=O)C(c2ccccc2)O)C1 N#Cc1ccc(S(=O)(=O)N2CCC(C(N3CCCC(O)C3)=O)C2)cc1 C1(C(=O)NCCOC(C)=O)CNC(=O)CN1C(c1cc2n(n1)CCC2)=O C1(C=O)CC(C(C)C)=NO1.C(COC(C)C)(C(=O)N)NC(C)=O.CCC CC1CC=CCC1NC(=O)CC1(CO)CCC1 N1(C(c2c(C(C)C)con2)=O)CCCC2(CCN(C(=O)C(C)CF)C2)C1 C1(NC(c2ccc(COC)o2)=O)(C)CCN(C(C2CCC2C(F)F)=O)C1 Cc1onc(C(=O)NC2CCC2)c1[N+](=O)[O-].C1(C=O)CC2(C1)CC(F)(F)C2.N C1(NC(=O)CCCn2ccnc2)CCCCN(C(c2cccc(C(F)F)n2)=O)C1 C1(O)(C(=O)NCC(C2CC2)NC(=O)CP(C)(C)=O)Cc2ccccc2C1 c1(CC)nc(C)ncc1C(N1CCCC(NC(=O)C2=NOCC2)C1)=O CN1CCCC(F)(C(=O)NCCCCCNC(c2n[nH]cc2F)=O)C1 c1(C(=O)NC(CC)CN(C(=O)CC2(O)CCC2)C)cc2sc(C)cc2s1 c1(-c2onc(CC)n2)ccc(NC(c2nnnn2C)C2C3COCC23)cc1 C1(c2cc(OC)c(F)cc2)CCN(N2CCc3ccc(CO)cc3C(C)C2)C1 C(=O)(N=c1ccc(-c2ccccc2F)n[nH]1)N1CC(N(C)C)C(C(=O)O)C1 Cc1cnc(C(=O)NCC2(C)CCCN(C(=O)C(N)=O)C2)c(O)c1 C1(NC(C(=O)Nc2ccc(CCOC)cc2)=O)CC(N(C)C)C12CCC2 CCC(C)C(C(=O)NCc1ncco1)NC(=O)C(C1CC1)SC c1(CNC(C)CC2CCOC2)cnc(C2CC2)[nH]1 C1(NC(=O)Nc2ccc(CNC(C)=O)o2)CCCC(S(C)=O)C1 N1(C(C2C=C(C)CS2)=O)CCCC(CC(N2CCCC2C2CCCC2)=O)C1 CCC(C)(CC)C(=O)NC1CC(O)CN(C(c2ncncc2Br)=O)C1 c1(SC)nc2c(s1)CCN(C)C2.c1(-c2sccc2)nc(C=O)c(C)s1.c1ccccc1 Cn1ncc2cc(C(=O)NCCC3CCN(C(=O)Cc4cnns4)C3)cc(O)c12 C#CCCCC(=O)NC(CC(=O)N1CCC(n2ccnc2)C1)C1CC1 c1(C(N(C2CCN(C(C(CC=C)C)=O)C2)C)=O)cnc(O)n(C2CC2)c1=O C#CC1CN(C(=O)COCCNC(C2CCC(C)O2)=O)CCN1C c1(C(C(=O)OCCCc2c(C)ccnc2)O)cc(Cl)cc(Cl)c1 c1(NC(c2ccccc2C(F)F)=O)cc(-c2ccc(Cl)cc2)nc2ccccc12 C1(NC(CCC(=C)Cl)=O)(CO)CCCN(C(C2(C)CC=CCC2)=O)C1 C1(NC(CC2(C)CC2)=O)CN(C(c2cccc3c2CCC3)=O)Cc2nccn2C1 C=Cc1cncc(C(N2CCC(O)(C(C)C(=O)Nc3cnn(C(C)C)c3)C2)=O)c1 Cn1[nH]nnc1=NCC1CN(C(=O)CC2CCNC2=O)CCC1C(F)(F)F Cc1csc(=NCC(=O)N2CC3(CCCC3NC(c3ccc(C)c(F)c3)=O)C2)[nH]1 C(=O)(C(C(C)C)N(C)C)N(C(CNC(COCC=C)=O)C)CC C(=O)(C(C(C)(C)C)n1cc(-c2cncs2)nn1)N(CC)Cc1cc(F)ccc1F c1(CC(=O)NCC2(C(C)NC(C3CC(C#N)C3)=O)CC2)cncn1C C1(=CC(=O)NC2C(NC(C(CCC)=CCC)=O)C2)CCC(C)(C)CC1 CCCC(C)(CCC)C(=O)N1CCC(C(C)CNC(=O)C(C)n2ccnc2)CC1 c1(CNC2C(C(N3CCCC(C)C3)=O)C2)c[nH]c2cc(C#N)ccc12 c1(NC(CC)CC#N)ccc(S(=O)(=O)NC(C)CCCCO)c(Cl)c1 c1(CC(=O)NC(CNC(C=CC=CC)=O)C(C)C)cc(Br)ccc1O C1(C(=O)OC)CC(O)CC2C(=O)N(Cc3nnc(C)o3)C(=O)N12 C(C(CNC(=O)CCC1CCCC1)C(C)C)OC.C1(CCC(=O)N)CCCCO1 c1(C(=O)NC(CN(C(c2ccc(OC(F)F)cc2)=O)CC)C)cnc(S)nc1 Cc1c(CC(=O)NC(CNC(C2CC(C)N(C)C2)=O)C2CC2)cccc1Br C1(NC(c2c(F)cc(F)cc2F)=O)CN(C(c2ccccc2O)=O)CC(F)(F)C1 C(=O)(C(CC)CCC)NCC1(CNC(C(CCC)OCC)=O)CCC1 Cc1ccc(C(N2CCC(C(=O)O)C(F)C2)=O)c2c1CCC2 CC(C)CC(C)(CNC(c1ccns1)=O)NC(C1CC1(F)F)=O CON(CCC(=O)NC1(C2CCCO2)CC1)C(=O)Cn1cnnn1 CC1CCN2N=C(C(=O)NCC(C)(C)CNC(c3ccon3)=O)NC2=N1 c1(C(N2C(C(N3CC4COCC4C3)=O)CSCC2)=O)cc(Cl)cc(Cl)c1 c1(C(N2C(C)CN(C(C3(F)CC=CC3)=O)CC2)=O)cc(F)c(Br)c(F)c1 CC(C)CC(O)CC(=O)NC1COCC1NC(=O)C(C)(C)C(C)O N1(C(c2ccc(OC)nc2)=O)CCC(C(=O)NC2CCOCC2F)CC1C c1(C(N2CCC(C)C(CNC(C3(C)CCNC3=O)=O)C2)=O)cc2c(s1)CCCC2 c1(NC(CC(C)CNC(C2CN(C(N)=O)C2)=O)=O)cncc(C#N)c1 CON(C)C(=O)C(CNC(C1CC=C(C)CC1)=O)C(C)C N1(C(C2CCS(=O)(=O)N2)=O)CC2CC(NC(C3(C4CCC4)CC3)=O)CC2C1 C1(CNC(c2cccc(-c3cnco3)c2)=O)C2CCC1CN(C(C1CC1F)=O)C2 C1(NC(c2cc(C)c(C)[nH]2)=O)CC(C)CN(C(C2(C(C)C)CC2)=O)C1 CCC(C)C(C(=O)NCCC1CN(C(C2CC(F)CN2C)=O)C1)OC c1(NC(C2CCN(C(CCC)Cc3ccccc3)C2)=O)ccc2c(c1)CCCO2 Cc1ccc2scc(C(C(=O)NCC3CCOCC3)N(C(C)CN(C)C)C)c2c1 c1(CC(=O)NCCC(C)NC(c2c(C)ccnc2)=O)ccc(Cl)c(F)c1 N1(C(c2cc(C)ncc2C)=O)CCN(C(c2coc(Cl)n2)=O)C(C)CC1C O=C1CC2CCC(C(=O)NCCCOc3ccc(Br)cn3)C2O1 CCCCCCOCC(=O)NC1CC1NC(c1cnn(-c2ccccc2)c1)=O CC1(CNC(=O)C(C2CC2)NC(=O)CC2CCCSC2)CCCC(=O)N1 N1(CCC)CCCC(C(=O)N(CC(O)C)C)C1.C1(CS(N)(=O)=O)(C=O)COC1 c1(C(N2CC3(CC(C(=O)NCC4CCO4)C3)C2)=O)cc(Br)cc(Cl)c1F N1(C(CS(N)(=O)=O)=O)CC2(C1)CN(C(=O)CCC1CCCO1)C2 Cc1cnc(C(=O)N(CC(O)CN(C(=O)C(C)C#N)C)C)cc1Br c1(C(=O)NC(CCN(C(CC(CC)C2CCC2)=O)C)C)cc(S(N)(=O)=O)oc1C N1(C(C2ON=C(C(C)C)C2)=O)CC2(CCN(C(c3nnn4ccccc34)=O)C2)C1 CC1(C)CCCCCC1NC(C1CN(C(c2ccc(C#N)o2)=O)CC12CC2)=O C(C(C)(C)C(=O)N1CCC(n2ccnn2)C1)NC(C1C(=C)C1)=O N(C1COc2ccccc21)C(C1N(C(CNC(NCC)=S)=O)C2CCC1C2)=O c1(C(=O)NC23CC(NC(CCCC=C)=O)C(OC2)C3)cc2cccnc2nc1C CC(CC(F)(F)F)C(=O)N1CC(F)CC1CN(C(=O)CCCNC(N)=O)C C1(NC(c2cn3ccnc3s2)=O)CCN(C(c2nc(C3CC3)cs2)=O)CC1F N1(C(Cc2c(C)noc2)=O)CCN(C(=O)CN(C)CCO)CC1C Cc1nc2[nH]c(C(=O)NC3CCCN(C(C4(C)CC(F)(F)C4)=O)C3)cc2s1 C(=O)(C#CC(=O)NCC1CCN(C(=O)CCCC2OCCO2)C1)N(C)C C1(NC(CCCCCOCC)=O)COC2CN(C(=O)C(C)CC3CCC3)CC12 c1(C(C)C)ccc(CC(=O)N(C)CCOCCNC(C2C(C)C2C)=O)cc1 N1(C(c2cc(CCC)[nH]n2)=O)Cc2nccn2CC(NC(C2CCCSS2)=O)C1 CCC(CC(=O)NCC(O)CCNC(=O)Cc1cc[nH]c(=N)c1)SC C1(C(=O)NCC(C(C)C)NC(CCOC(C)=O)=O)CCc2nnn(C)c2C1 CN1CCCCC1C(=O)NC(Cc1ccoc1)C(=O)NCCNS(N)(=O)=O CS(=O)(=O)c1cccnc1N1CCC2CCC12CN Cc1ccc(C(N2CCC(NC(=O)Cc3c(C)ncnc3C)C(C)C2)=O)cc1O C(=O)(C1=C(F)CN(C(c2cc(F)n(C)n2)=O)CC1)N1CCC(CCC)(CO)C1 c1(NCC2C(NC(C3CCC(NC(C)=O)CC3)=O)CCCC2)nccnc1C#N C1(CC(=O)N(c2ccccc2)CC(O)COCC2CCOC2)Cc2ccccc2C1 Cn1nc([N+](=O)[O-])cc1C(=O)NC1CC1NC(C1CCS(=O)(=O)N1)=O N1(C(C2(NC(C(C(CC)C)=O)=O)CC2C)=O)CCCC2(C=CCO2)C1 C1(C(=O)NCC(CC)NC(C2CCN(C)C(C)C2)=O)CCC(F)(F)CC1(C)C N1(C(CCCC)=O)CC2(CCN(C(c3ccc(C(=O)OC)cn3)=O)CC2)CC1C N1(C(=O)OC)CCC(C(=O)NC2CC(C(N)=O)N(C(=O)CCCC)C2)CC1.S C1(NC(C(CC)O)=O)(CF)CCN(C(=O)Cc2coc(-c3cccs3)n2)C1 c1(C(CC)Oc2ccccc2)nc(CC(N)=O)nn1-c1ccccc1SC c1(C(=O)NCC2CCN(C(C3(C)CCOCC3)=O)C2)cnc2c(c1)CNC2=O c1(C(N2C3C(NC(=O)C4=COCC4)C(CC3)C2)=O)nccc2ccsc12 N1(C(C(CCOC)OC)=O)CCC2(C)CN(C(=O)CCCCC(F)(F)F)CC12 c1(C(N2C(CNC(CC(COC)(C)C)=O)CCCCC2)=O)ncc(Cl)c(N)c1Cl c1(OC)cccc(SCC=O)c1.CCC(C)(C)C.C1(CC=O)C(C)C1(F)F.N Cc1cc(C(=O)NC2(C)CC(NC(C3CC(C)CO3)=O)C2)cnc1O c1(OC)ccc(CNC(c2ccc(Cl)cc2)c2ccccn2)cc1I C1(OC)CCC(C(=O)NCc2cc(C(=O)NCC(Cl)Cl)ccn2)CC1 C12(C(=O)NCC(C)C3CCC3)CC=CC(C1)OC2.C1(CC(=O)N)CCCCC1 CC(=O)NNC(=O)COc1ccc(OC(F)(F)F)cc1 N1(C(c2cc(OCC)no2)=O)CCC(=CC)CC1.C(=O)C(O)CN(C)C.N C1(NC(CC2(CC)CC2)=O)CCOC(C(=O)N(C)CCc2ccccn2)C1 Cc1cc(C(=O)O)ccc1C(N1CC2CCC1C2)=O.c1(C(=O)N)cc(C)n(C)n1 C(=O)(C1CCSc2ccccc21)NC1CN(C(C2(CC)CC2)=O)CC2(C1)CCC2 C=CCCC(C(=O)NC1C2CCN(C(c3cc(OC)cs3)=O)C12)c1ccccc1 c1(C(=O)NC(C(C)C)C(C)NC(C2CC3(CCC3)C2)=O)cccc(N)c1Br CC1CCN(C(=O)CN(C)C(N)=O)CC1NC(C1(c2ncccc2F)CC1)=O C1(C(N2C(C(=O)NCC3CC3[N+](=O)[O-])CC(C)C2)=O)CC2(C1)CC2(F)F C(=O)(C(CC1CCOCC1)N(CC(C)C)C1CC1)NC1(CC)CCC1 C1(NC(C)=O)CCS(=O)(=O)C2(C1)CCC2.C1(CC=O)CCC(C)C(C)C1.C N1(C(C(=O)NC2CCOCC2)c2ccco2)CCC(C(F)(F)F)(N2CCCC2)C1 N#CC1(F)CCN(C(=NCCc2cccs2)NCc2ccc(Cl)cc2)C1 C#CCC(CC(=O)OC)NC(C1CC12CCN(C(C1(Cl)CCCCC1)=O)C2)=O S(=O)(=O)(c1cccc(Br)c1)NCCCC(=O)NC1CCOC1 C1(C(=O)NC2CCCN(C(=O)OC(C)(C)C)C23CC3)CNc2cccc(Br)c2O1 c1(C(=O)NC(C)CNC(=O)C(c2cccc(F)c2F)(F)F)ccc2ocnc2n1 C12(C(=O)N)CCC(C)(C1)OC2.Cc1csc(CCC(=O)N(C)CCOCC)c1 C(=O)(CCC(=O)C(C)(C)C)NC(C(=O)NCC(CC)CC(C)C)CN(C)C C1(C=O)CN(C)CC(C)O1.C(=O)(CC(O)CNC(=O)CCC1CCCC1)OC Cc1cc(C#N)cc(C)c1CC(N1CCC(C)C1C)=O.C(=O)C=C1CCC1.N c1(OCC)cccc(C=O)c1.C1(C=O)CC(=O)N(C(C)C)C1.CCC(C)C.N c1(OC)c(C(=O)N(CC(C)(C)CNC(c2cccs2)=O)C)ccc2c1CCC2 c1(C=O)c(N)cc(Cl)cc1Cl.Cn1ccc(C(C)(C)C(=O)NCC(C)(C)C)n1.N c1(C2(OC3CN(C(C(C)OC(c4ccccc4)C)=O)C3)CC2)ccn(C)n1 C1(CC)CCCN(C(=O)CC2CC2)CC1.C(=O)(C(C=O)C1CC1)O.CC(C)C N1(C(COC)=O)CC2CCC(CNC(c3ccc(C(=O)OC)n3C)=O)(C2)C1 N1(C(C(CC)SC)=O)CC2(C1)SCCC2NC(=O)CCOC(N)=O N1(C(Cn2ccc(C)n2)=O)Cc2[nH]nc(C(=O)NC(c3nnc(C)o3)C)c2C1 C(=O)(C1=CCCOC1)NCC1CCC(NC(=O)Cc2ccc(O)c(F)c2)CC1 C#CCCCC(C)C(=O)N(C1CCCC1)CCCNC(=O)C(O)CCC(C)C c1(C(N2CCCC(N(C(C3CC34CCC4)=O)CC)C2)=O)cnc2ccccn12 C12(NC(CCc3c(C)cccc3)=O)CCCN(C(c3ccncc3F)=O)CC1C2 N1(C(COC)=O)CC2CCCN(C(C3CCCCC3C)=O)C2C1 C(=O)(C(C)C1CCCO1)N(CCOCCN(C)CCF)C N1(C(C(c2cscn2)N(C)C)=O)CC2(CCC2)CC1C.c1(C(=O)N)ccc(F)s1 N1(C(Cn2ncc(C#C)c2)=O)CC(NC(=O)C=CCO)CC(O)C1 c1(CC(=O)N(CC(CC)NC(CCSCCCC)=O)C)cnc(Cl)cc1C CC1CCC(NC(=O)C=CC2CCCCCC2)CN1C(=O)CC1(N(C)C)CC1 c1(NC(CC2CN(C(c3cncc(OCC)c3)=O)C2)=O)cc(C)c(Br)cn1 C1(CNC(C(CC)CC)=O)CC(C)(C)CCC1NC(C1(O)CCCCCC1)=O Cc1cc(C=O)cc(F)c1.C1(C2CC2)CCCCN1C(=O)CC1CS(=O)(=O)C1 C1(NC(CCCOC(C)C)=O)CC(C)CN(C(=O)CCc2ccon2)C1 C(=O)C#CC1CCC1.CC(C)(CNC(=O)OC(C)(C)C)C(=O)NCCC C1(OC)CCN(C(=NCCNS(C)(=O)=O)N)CC1C.C1(F)CN(C(=O)CC)C1 Cc1cnc(NC(=O)CC2CCCN(C(c3ccc(O)cc3C)=O)C2)c(I)c1 C(CC(C)C)(C(=O)N1CC(OCCNC(=O)C(F)(F)C(C)O)C1)OC C1(NC(c2nc(C(C)C)sc2)=O)CCC(N(C(=O)CO)C)CC1.C1CCC1.C c1(C(N2C(C(=O)NCCC3CC(C)(C)OC3)COCC2)=O)cncc(C#N)c1 N1(C(C2(CC)CCCC2O)=O)CCC2(CC1)CN(C(=O)Cn1ncnn1)C2 Cc1cc(O)c(C(=O)NC(CNC(c2nccn2C)=O)CO)nn1 CCC(CC(C)CO)N=c1nc(N(C)Cc2cnc(C)s2)c2c([nH]1)CCS2 N1(C(CCc2ncc(C)[nH]2)=O)CC(CNC(c2sc(Cl)cc2Cl)=O)C(C)C1 N1(CCC)CCCC(C(N2CCOC(CN(C)C(C34CCC(CC3)C4)=O)C2)=O)C1 c1(N2CC(CO)CC(C)C2)[nH]c(=NCC(Br)=C(C)C)nc2sccc12 C1(C(=O)NC(c2ccc(C)s2)C)COCCN(C(c2ccncn2)=O)C1 C1(C(=O)NCC2CC(N(C)CC)C2)CC(C)C1.C(=O)(C)N.CC(F)F C1(C(=O)NCCCc2ccco2)(OC)CCN(C(C2CCCN(C(C)C)C2)=O)C1 CC1CCC(CNC(=O)C(F)F)N(C(=O)CCN2CCCC2)C1 CCC(CC(=O)N(C1CN(C(C2(Br)CC2(C)C)=O)C1)C)C1CC1 Cc1cc(C(N2CCN(C(=O)CC(C)(F)F)C3CC23)=O)cc(C)c1N C1(C(N2C(CC)(CC)CC2)=O)CN(C(c2c[nH]nc2C(C)C)=O)CC1(F)F c1(OC)ccn2ccnc2c1C(=O)NC1C2CN(C(=O)C(C)(C3CC3)O)CC12 C1(C(=O)NCC2CCCN2c2nnc(C(F)(F)F)s2)CCCC2CCCN12 c1(C(N2CC(NC(CCC(=C)Cl)=O)C(F)CC2)=O)ccc2c(c1)NC(=O)C(C)S2 C(=O)(CCCN(C)N=O)NCC(CO)NC(c1cc(C)nc(N(C)C)n1)=O C(C(COC)CC(=O)NC1CC(CCC(=O)NC2(C(N)=O)CCCC2)C1)OC N1(C(C(C)N(CC(F)(F)F)C)=O)CCN(Cc2cn(-c3cccc(F)n3)nn2)CC1 N1(CC)CCN(C(c2cn3ccnc3s2)=O)C(C)C1 N1(C(C(CSC)C)=O)CC(C)(C)CC1CNC(c1cc(C(C)=O)oc1C)=O N(S(=O)(=NCC(=O)O)N(C)C)C(c1ccc(CC)c(CC)c1)=O c1(CC=O)csc2c(Cl)cccc12.N1(C(C(C)O)=O)CCCC(C)C1.C(C)(C)C.N C(c1ccc(C(C)C)cc1)=CC(=O)NCC1N(C(C)=O)CCCC1 N1(C(c2n(C(C)(C)C)ncc2)=O)CC2(CCC(CNC(C3CCCO3)=O)O2)C1 C(=O)(C1=CCCC1)NC(C(=O)NC1C(c2n(C)ncc2)C1)c1cccs1 C=CC(C)(O)CC(=O)NC1CCCC1NC(c1cncc(OC2CCC2)c1)=O N12CC(C1)SCCOCC2=O.C1C(=O)N1.C(COC)SC N1(C(c2c(C(C)C)ocn2)=O)CCC(NC(=O)CC(C)CF)CC(C)(C)C1 C1(CNC(=NC)NCC(C)Sc2ccccc2)CC2(CCCCC2)CO1 C1(NC(C=CC=CCC)=O)CC2CC1CN2C(=O)CCn1ccccc1=O C(CCN=c1nc2ncn(CC)c2c(NCc2cnn(CC)c2)[nH]1)SCC c1(C(=O)NCCCCCCNC(C2=NOC(C)C2C)=O)ccc([N+](=O)[O-])cc1F C#CC1CC2(CC2)CN1C(C1(NC(=O)CC2CC2)CCOCC1)=O C1(NC(=O)COCCCF)CC2CC1CN(C(C1CCc3nn[nH]c3C1)=O)C2 CC(CC(N)=O)NC(=O)C(CO)NC(=O)Cc1cnsc1 N1(CC(=O)NCCC(C)N(C(C2CC(CCC)C2)=O)C)CCNC(=O)C1 C(=O)(C(C)CN(C)C(c1csc(C)n1)=O)NC(c1nccs1)CC C1(C(N2C(CO)CC(C)(C)C2)=O)CCN(C(=O)C2=CCCC2)CC1(C)C N1(C(C(CCC)N(C)C)=O)CC2CCN(C(c3cscc3C(F)F)=O)C2C1 C(=O)(CCOC(C)C)NCC(COC)O.c1(C=O)cc(C(C)C)no1.N C(=O)(C1=COCCO1)N(C1CCN(C(C2CCS2(=O)=O)=O)CC1)CC(C)C c1(CC)noc2ncc(C(=O)N(C)CCOCC)cc12.C1(C)(C=O)COC1.N N1(C(=O)CC2OCCCO2)CCC2(CC2C(N2C3COCC2C3)=O)C1 C(=O)(C#CC1CCOC1)N(C(CN(C1CCCC1)C(C)C)=O)C1CC1O c1(C(N(CCCCC=C)C)=O)nc(CNC(=O)C(C)c2ccsc2)oc1C c1(C=O)cnc(S(C)(=O)=O)s1.Cc1c(C=CC(=O)NC2CCCC2)cnn1C c1(C(=O)OC)cc2cc(-c3cccc(Cl)c3)ccc2o1 C1(NC(c2ccn(CCF)n2)=O)CCN(C(c2cnc(S)nc2)=O)CC1CO C1(C(=O)N)(OC)CCCCC1.C1CN(C(=O)CCC(C)C)CC1F.C(=O)C(F)(F)F C1(C2CC2)(NC(=O)CC23CCCN2CCC3)CCN(C(C2(Cl)CC2)=O)C1 c1(SC)nc(N2CCCC2CNC(=O)CC2CCC3CC23)c2scc(C)c2n1 CCCCC(CC)C(=O)NCC(CNC(C1(SCC)CC1)=O)CO c1(C(c2nnnn2C)NCc2n(C)nnc2)cnc2cc(Br)ccn12 c1(C(C)NC(C2CCC(NC(=O)NCC(=O)OC)C2)=O)ccccc1Cl C(=O)(CC(C)(C)C)NC(C(=O)N(C1CCC(C)(C)C1)C)CC1CC1 c1(N2CC3(CO)C(C2)CC3)cc(NC2CCCCC2)nc(C(F)(F)F)n1 C1(COC)(C)CCCN1C(=O)C(C)(O)c1ccccn1.c1(C=O)coc(Cl)n1 C1(C(N(CC(=O)N(C)C)CC)=O)CC12CCN(C(c1ccncc1O)=O)C2 N1(C(C2CCOC(C)(C)C2)C(=O)NC(CC)(C)C)CC2CCC1CC2 N1(C(=O)CC2CCCCC2O)CC2CC(C(=O)NC)(C2)C1.c1n[nH]cc1C1CC1 Cc1cc(NC(=O)C(C)C(C)O)ccc1NC(C1(C(N)=O)CC1)=O N1(C(CCC)=O)CCC(C)C1.C(=O)C.C(C=O)NCC.C(C)(C)C.C1CC1 Cc1cc(C(=O)N(C2CCN(C(=O)OC(C)(C)C)C2)C)sc1Br c1(C(N2CC3CN(C(CC4CC(CC)C4)=O)CC3C2)=O)c[nH]c2ccc(Cl)cc12 c1ccccc1[N+](=O)[O-].N1(C(C=CC(C)C)=O)CC(CNC(=O)C)CC1(C)C C#Cc1ccnc(C(=O)NCc2c[nH]nc2C2CCN(C(C3COC3)=O)C2)c1 C(=O)(CCC(F)(F)F)NCCOCCCNC(=O)CC(O)C1CCCC1 c1(C2(C(N(CC)C3CC3)=O)CC2)ccc(F)cc1Cl.O=C(C(F)C1CCC1)N Cc1oc(CNC(=O)CCC2CC2C)nc1C(=O)NC(c1ccncc1)C CC1CC(C(=O)NC2(C(=O)NCC(C3CCCO3)O)CSC2)=NO1 c1(N2C(CN(C)C(C3CCCC(F)(F)C3)=O)CCC2)cc2nncn2cn1 CC1(C)CN(C(C2(C(F)(F)F)CCC2)=O)CCC1.C1(CC=O)CC(=O)NC1=O O=C(C1=COCCC1)N1CCN(C(C2(C3CC3)CCC2)=O)CC1c1ccccn1 c1(C(N2C(CNC(C(COC)(C)C)=O)C(C)CC2)=O)cc2sccc2cn1 C1(NC(C2CC2F)=O)CC2CC(C1)N(C(c1ccc(OC(F)F)c(Cl)c1)=O)C2 n1(C(CC)C)ccc(=NC(=O)c2cocc2C)[nH]1 C=C(C)c1cn(CC2CCCC(CNC(=O)C(O)CC3CCCC3)C2)nn1 CCCCCC(O)C(=O)NCC1C2CC1N(C(C1(COC(C)C)CC1)=O)C2 c1(C(N2CC(O)(C(C(=O)N)F)C2)=O)cc(F)ccc1F.c1(COC)ccccc1 C1(c2n(C)ccc2)CCCCCN1C(C1(Cl)CC1(C)C)=O C1(C(=O)NC(C)C(C)(C)c2ccccc2)CCOCC12CCCC2 Cc1oc(Cl)nc1C(=O)NC(C1CN(C(=O)Cn2nccc2C)CCO1)C N(C1CCc2cc(CNC(=O)C=CC=C(Cl)Cl)ccc21)C(C1N(C)CCCC1)=O C#CC1(O)CCN(C(C)C(N2CC(O)(CC)C2)=O)CC1.c1(CC(=O)N)cccs1 N1(C(c2ncc(C)s2)=O)CCCC2(C1)CN(C(C1CCCO1)=O)CCO2 c1(NC2CCCC(NC(=O)C(C3CC3)C3CC3)C2)ncc([N+](=O)[O-])cc1F c1(C(=O)NC(C(=O)NCCOC(CC)CC)c2ccco2)cc(F)c[nH]1 CCCCCC(CC)C(=O)N1CCN(C(=O)CC2CCCN2C)C(C)C1 C(C)(C)(CC(F)C(=O)NCC1(S(C)=O)CC1)NC(C(C)CO)=O N1(C(=O)Cn2ncnn2)CCCC2C1CCCCN2C(c1cnc(Cl)s1)=O N1(C(COCC)=O)CCC2OCCN(C(=O)CCC(C)(C)C)C2C1 Cc1cc(C(N2CC3CC3C2C(=O)NC2(C3CCC3)CC2)=O)[nH]c1C c1(C(C=O)N)ccc(S(C)(=O)=O)o1.CC(Cl)C(C)(F)F.C1(C=O)CCC1 c1(C(N2CCCC(F)(CNC(C(C)C(F)(F)F)=O)C2)=O)ccc(O)cc1[N+](=O)[O-] c1(C(=O)NCC2N(Cc3cnc(CCC)s3)CCC2)ccnc(F)c1 c1(C(N2CCN(Cc3cccc(OC)c3)CC2)=O)nc(Cl)ccc1N Cc1ccc(CC(N2CCC(NC(C3C4CCCC34)=O)C2C)=O)c(Br)c1 C1(NC(c2c(C)csc2)=O)CCCN(C(c2c(C(F)F)nn(C)c2C)=O)CC1 c1(OC)cccc(O)c1NC(C1(C)CCN1Cc1cccc(Cl)c1F)=O N1(C(CC(C)C2CCCO2)=O)CC(F)CC1CN(C)C C1(C(=O)NC2(CC=C)CCN(C(C3CCC3)=O)CC2)CCC2(C1)CC2(F)F.C C(N=c1[nH]c(=NC2CCCCC2C)[nH]c2cc[nH]c12)c1c(C)noc1C C1(CNC(c2c(COC)scc2)=O)CC(C(=O)N=c2ccn(C)[nH]2)=NO1 C1(CNC(CCCCOC)=O)CC2CCC1N(C(=O)CC1CCCC(C#N)C1)C2 c1(SC)nc2ccccc2c(=NCC23CCC(CC2)OC3)[nH]1 CC1N(C(=O)CC(O)CNC(=O)CCC2(C#N)CCC2)CCCC12CCC2 N1(C(Cn2c(C)ncc2)=O)CCCCCC(NC(=O)C=CCF)C1 Cc1cc(OCC(=O)N)cc(C)c1Cl.CC(C)(C)CN(C(=O)Cc1cocn1)C C1(O)(CC(N2CC3CC3(Cn3cc(CO)nn3)C2)=O)CCOCC1 CS(=O)(=O)C1CCCC1n1cc(CC2CCN(C(=O)C=CC3CC3)C2)nn1 N1(CC(=O)N)C(=O)CCCC1=O.n1(CC)ccnc1C(=O)NCC(C)(C)C c1(-c2ccc(C(N3CCC(CNC(=O)C(Cl)Cl)C3)=O)o2)cccc(Cl)c1 c1(CC(N2CC3C(C3)C2)=O)cccc([N+](=O)[O-])c1.C1(C(=O)N)(SC)CC1.C S(=O)(=O)(c1ccc2nc(NCC(C)C(F)(F)F)ccc2c1)NC(COC)C(C)C c1(N(CCNC(c2cc(C(F)F)on2)=O)CC)ncnc2c1cnn2CC CCC(COC)C(=O)N1CCCC1CNC(C1(C)CCC1)=O C(=O)(C(C)(C)CC(F)(F)F)N1CC(N(C)C(C2CC3CC3C2)=O)C(O)C1 Cc1cn2c(n1)CC(C(=O)NC1C3CC1N(C(C1CC(C)C1)=O)C3)CC2 C1(N(C(CC=C)=O)CCO)CCCN(C(C2CC(N(C)C)C2)=O)C1 CCCC(C)(O)CC(=O)NC(C)(C)CC(N1CC(=O)NC(=O)C1)=O c1(C(c2n(CC)nnn2)Nc2cnn(CCO)c2)c(C)sc(C)c1S(N)(=O)=O N1(C(Cn2c(C(F)F)cc(C)n2)=O)CC=C(C)CC1.C1(C(=O)N)C2CC2C2CC12 C1(NC(C2CCC(=O)N2)=O)C2CC1CN(C(=O)CCOCC1CC1)C2 C1(C)(CCNC(CCC2CC(OC)C2)=O)CCN(C(c2cccc(F)c2)=O)C1 c1(C(=O)NCC2C(C)C2(F)F)ccncc1Cl.C1(C(=O)N)CC(F)(F)C1 N1(C(C)=O)CCOCC1C(=O)NC1CCN(C(C23CCC(CC2)C3)=O)CC1 c1(CC)cnoc1C(=O)N(C)CCOCCC(=O)N.C1(CC)CC(F)(F)C1 CCC(C)(C(=O)NCC1CCCCC1)C(N)=O.C1(CC=O)NC(=O)NC1=O.C CCCCC(O)C(=O)NC(C1(O)CCN(C(=O)C(C)COC)C1)C c1(OCC)ncc(C(=O)NCC(O)CN(C(=O)CS(=O)(=O)NC)C)cc1Cl c1(CCC(=O)NCC2(C)OCCN(C(C(OC)OC)=O)C2)cnc2ncccn12 N1(C(C2C(C)C2)=O)CCN(C(=O)COc2ccc(Cl)c(F)c2)CC1C C(=O)(CCC(=O)NC(CO)C(N1CCC(C)(CN(C)C)C1)=O)N(C)C N1(C(c2cc(C(CC)C)no2)=O)CCC(C)(C)C1CNC(C1(C)CCC1)=O C1(CC)CN(C(C2CC2COC)=O)CCN1C(=O)CC1(CSC)CC1 C1(N(C)C(C2CC2C(F)F)=O)CCCN(C(=O)C=Cc2cccs2)C1 c1(C(=O)NC(C)CC(C)NC(c2nncn2C2CC2)=O)[nH]ncc1C#N N1(C(C(CC#C)NC(c2cnncc2C)=O)=O)CCC2(C=CCO2)CC1 c1(C(=O)NC)cnn2ccccc12.C1CC(O)C1.C1(C=O)CC(=C2CC2)C1 C(CNC(C1CCC1(F)F)=O)(CC(F)(F)F)NC(CCC=CC)=O CCC(c1ccccc1)=CC(=O)NC1(C2CN(C(=O)C(C)C(C)COC)C2)CC1 c1(CSC)ccc(C(=O)NCC#CCNC(c2csnc2Br)=O)o1 C(CCC(=O)NCc1conc1C1CC1)(C(C)C)NC(CC(CC)C1CCC1)=O C(=O)(C1=C(c2sc(C3CC3)nc2)N(C)C(=S)NC1c1cn(C)nn1)OCC.O N1(C(=O)Cn2ccnn2)CCCC12CCN(C(C13CCCCC1C3)=O)CC2 CCC(O)(CC(=O)NC1COCCN(C(=O)Cc2ccsc2)C1)c1cccs1 C1(CC)(CC)CC(NC(C2CCC=CCC2)=O)CN1C(c1ccn(CCF)n1)=O C(C)(CNC(=O)C(C)(C)c1csc(C)c1)(C(C)C)NC(C(CC)OC)=O C1(C(=O)NCC2(C=O)CC(C)(C)C2)CC2(CCC2O)C1.C1CCOC1(C)C.N C(CCCC(CO)NC(=O)CN1CCC(C)(O)C1)NC(C(C)(C)n1cnnn1)=O C1(C(NOC(COC)COC)=O)CN(C(c2cccc3ccnn23)=O)CC(C)(C)C1 c1(OC)ccnc(C(N2CCC(C(N3CCC(CCCO)C3)=O)(OC)C2)=O)c1 C(=O)(CCC(CC)CC)N1CC(NC(C(C=C=C)C)=O)(CO)C1 CCCC(CCC)C(=O)N1CCC=C(CNC(=O)C(C)c2ccco2)C1 CCCCCCC(c1ccccc1)NC1(c2nnnn2CCCOC)CCOC1 c1(OC)ccc(C)nc1C(=O)NCCCC.c1(C(=O)N)cn(C)c(C(F)F)n1 N1(C(C)C)CCOC(C2CCC2)C1.C1(=O)CCCC2(CCC2)N1C(=O)C(C)(F)F N1(CC(=O)NC2CCCN(C(C3CCC3)=O)C2)CCC(C)(O)C1.C1CC1.C N1(C(CC(c2scc(C)c2)O)=O)CCCC(C)(NC(=O)CCCc2cccs2)C1 c1(CNc2ncnc(N3CCCCC(SC)C3)c2C)c(C)nc2c(N)cccn12 N1(C(C(n2ccc(C)n2)(C)C)=O)CC2CC2(NC(=O)CCc2nccn2C)C1 c1(OC)ccc(Cl)cc1C(CNC(c1cc(C(F)F)ncn1)=O)OC C1(NC(Cc2c(C)occ2)=O)CN(C(C2CCC(CC#N)CC2)=O)CC1C C1(C(=O)NCCS(=O)CC)(NC(C2(CCC=C)CC2)=O)CCCCC1 c1(C(=O)NCCCC2CCCN2C(=O)CC2C=CCC2)cc(=O)cc(Cl)[nH]1 c1(C(C(=O)NCCCCNC(c2csc(C(F)F)n2)=O)(F)F)ccc(F)cc1 c1(C(=O)NCCOC2CCN(C(c3n(C)c(S)nn3)=O)C2)ccc2[nH]ccc2c1 S(=O)(=O)(CC(=O)NCCC1CCC1)NCC.C1(C(=O)N)COC(=O)N1 C12(C(=O)NC3CCC(CNC(CC=C(C)C)=O)CC3)CCOC1CCOC2 c1(NC(C2CCN2C(C2(CCF)CCC2)=O)=O)c[nH]ccc1=O C(=O)(CCCC(C)NC(C1(c2ccno2)CC1)=O)NC(COC)C1CC1 N1(C(c2nc(C)sc2)=O)CCC(NC(C2CC(=C3CCC3)C2)=O)C(CO)CC1 N1(C(CC2(C)CCOC2)=O)CCC=C(C(=O)N2CC3(CNC(=O)N3)C2)C1 CC(CC(C)(C)C)C(=O)N1CCSCC1C(=O)NC1CCCN(C(C)C)C1 C(=O)(CC(C)(C)CC)N1CCC(O)(C(CNC(CCN(CCC)C)=O)C)C1 CC1OC2(C)CC1(C(=O)NC1CCN(C(C3Cc4nccn4C3)=O)CC1O)C2 C1(C(=O)NCCCN(C(C(CC)CN(C)C)=O)CC)CC(C)CC(C)(C)C1 C(c1ccc(F)cc1F)=CC.CCCS(=O)(=O)NCC1N(C(CC)=O)CCC1.N C1(C(N2CCC(Oc3ccc(Cl)cn3)CC2)=O)OCCOC12CCC2 C(=O)(C1=C(Cl)CC1)N(C(C(=O)NCCC1(O)CCC1)C1CC1)C C1(CC(=O)NCC(CN(C)C(C2CCOC(C)(C)C2)=O)O)CC2C=CC1CC2 Cc1ncc(C(=O)NC2(C3CCCN3C(C3CC(n4cnnc4)C3)=O)CC2)s1 C1(NC(c2cccc(C3COC3)c2)=O)CC2CC1N(C(c1cnc[nH]1)=O)C2 N1(C(CSCCOC)=O)CC(F)(F)CC1(C)CNC(C1CCC1(C)C)=O CONC(=O)C(=O)NCC(CC1CC1)C(=O)NC1CCCC1C#N Cc1nccc(C(=O)NC2CCC(C)N(C(C3CC(C)(C)CO3)=O)C2)c1C CCCC(CC1CCCCC1)C(=O)N(C1CCN(Cc2ccc(Br)cc2O)C1)C c1(C(=O)NCC2OCCN(C(CCC3N(C)CCC3)=O)C2)ccc(C#N)nc1O c1(N2CCOCC(NC(C3(C)CCCCC3(F)F)=O)C2)ccc(F)cc1[N+](=O)[O-] Cc1cc(C(=O)N(CC(O)CNC(=O)C(C)CC(F)F)C)nnc1O C1(NC(CC(C)F)=O)CCCCN(C(c2cncc(C(C)(F)F)c2)=O)C1 C#CCCC(C(=O)NCC(CC)CCO)NC(C1OCCCC1(C)C)=O CC1CCN(C(c2cnnc(C3CC3)c2)=O)CCN1C(=O)CSC1CCCCO1 C(=O)(C(C)CN=c1[nH]c2c(c(=NCCC3CCC4(CCC4)O3)[nH]1)CSC2)NC CC1(C)CC(F)(F)CN1C(=O)CC1CC(O)C12CCC2.C1(C(=O)N)CCOC1 c1(OC(C2C(C=CC)C2(C)C)=O)cc(F)ccc1F C(=O)(CC(F)(F)C(F)(F)F)N1CCC(C)N(C(=O)CCc2cccc(O)c2)CC1 Cc1cc(N)cc(C(N2CC=CC(NC(=O)C(CO)N(C)C)C2)=O)c1F CCCCC(CN=c1[nH]cc([N+](=O)[O-])cc1C)NC(=O)C(CCC)OC N1(C(C(C)OCCOC)=O)CCN(C(c2cc[nH]c(=N)c2)=O)CC1C1CCC1 c1(C(=O)NCC(CNC(c2on(C)c(=O)c2)=O)O)cc(Cl)cc(Cl)c1N CCCC(CNC(=O)CC1CCC(=O)C1)C(=O)NCC1CCC(=O)N1 C(N=C(NCC(=O)N(C)C)NC1CCN(c2ccc(F)cc2)C1)c1cc(C)ns1 N1(C(C(COC)NC(C2CN3CCN2CC3)=O)=O)CCC(O)C(F)(F)C1 C(CCC(C)C)(C(=O)N1CC2(C1)CN(C(=O)C(O)CC1CC1)C2)OC Cc1ccc(C=CC(=O)Nc2cccc(C)c2)c(C)c1.c1(C=O)cc(C)c[nH]1.N CC(CN(C)C)CC(=O)N(C)CCOCCN(C)C(C1COCCO1)=O c1(NCCCCOC(C)(C)C)ccc([SH](=O)=O)c(Cl)c1.C(CO)CC(F)(F)F.N N1(C(C2CC3CN(C(c4cc(C)sc4)=O)CC2C3)=O)CCC2(COC(=O)N2)C1 CON(C)C(=O)CNC(=O)CC1CCCN(C(C2(Cl)CC2)=O)C1 C1(NC(C(C)Oc2cccc(F)c2)=O)CN(C(c2ccoc2)=O)CCC1(C)C C(C(=O)N=C1CCN(C)N1)=C1CN(C(COC)=O)C1 N1(C(CN(C)C(N)=O)=O)CCCC(CCCCNC(=O)Cc2ccnn2C)C1 O(NC(=O)CN(C(=O)CC(C)SC)CCC1CC1)CC(CC)C N#Cc1ccc(C(=O)NCC=CCC(N2CCCCC2C2CC2)=O)s1 N1(C(c2cc(C)n(C)n2)=O)Cc2ccc(O)cc2CC1C(N1CC2CC2C1)=O c1(CC(=O)N)csc(CCC(F)(F)F)n1.C=CCCOCC(=O)NC1CC1 C(C(C)(C)C(=O)NC(C)CNC(c1c[nH]nc1C(C)(C)C)=O)SC Cc1nc2ncnn2cc1C(=O)NCC1CCN1C(=O)C(N1CCC(O)CC1)C c1(C(=O)NCC2(F)CN(C(c3cc(OC)ncc3)=O)C2)ccc2ocnc2n1 c1(C(N(CCCNC(C(c2ccc(Cl)s2)C)=O)CCO)=O)cccn2cnnc12 C(C)(CC(=O)NC1(CCC(=O)NC(C)C(C)C)CCC1)OC C#CC1(C(N2CCC(F)C(F)C2)=O)CCN(C(c2cnc(O)cc2C)=O)C1 c1(OC)cc(CCOC(=O)C(c2cccc(N(C)C)c2)C)ccc1Cl N1(C(CCC(=O)O)=O)CCC(C(N2CCC(CCO)(CO)C2)=O)C(O)C1 N1(C(c2cc(C)no2)=O)CC2(CC(NC(=O)Cc3cnco3)C2)C1 CC1CCCc2nc(C(=O)NC3CCC(NC(C4CCC(=O)O4)=O)CC3)cn21 C#CC1CN(C(=O)C(C)OCC)CCN1C(c1cc(C)c(O)c(N)c1)=O C1(C(=O)NCCC2(C)CCN(C(c3cccnn3)=O)C2)CCCN(S(N)(=O)=O)C1 C(C(C)CC(C)C)NC(C1C(NC(C2C(CC)C2)=O)CC1O)=O N#CC1CN(C(c2c(O)cccc2O)=O)CCN1C(=O)C=Cc1ccccc1 C(C)(c1ccco1)=CC(N1CC(NC(C(C)(C)NC(=O)OC)=O)C1)=O C1(C(=O)Nc2cncc(Cl)c2)CCN(C(C2CCC=CCC2)=O)C12CC2 CC1(C)CCC(C(N2CCCCC2CO)=O)CN1C(C1(CC2CC2)CC1)=O N1(C(Cc2nnc(C)o2)=O)CCOC2(C1)CN(C(=O)CCC1CC(F)(F)C1)C2 c1ccc(C)cc1.C(=O)(CC)NCCCN(C(C1CC1C(F)F)=O)CC c1(C(N2CCCC(COCC#C)C2)=O)ccc(F)c(C)c1C#N C1(NC(c2ncc(C)nc2)=O)CN(C(=O)C(C(C)(C)C)c2cc[nH]n2)C(C)(C)C1 C(C(F)(F)C(C)(C)O)NC(C1(C)CC(NC(C2N(CC)CCC2)=O)C1)=O C1(C(N2CCC(C)CC2CNC(c2cnc(S)n2C)=O)=O)CCn2cncc2C1 Cc1ncc(NC(c2ccc(-c3cn(C(C)C(=O)O)nn3)nc2)=O)n1C(C)C n1(CC)cnc2c(N3CCC(CCNC(=O)C#CC4(C)CCCO4)C3)ncnc12 C(CNC(=O)C(Cc1cn[nH]c1)NC(C1CCCC1O)=O)(C(C)C)OC C#CC1(C(=O)NCC2CCCO2)CCN(C(c2cc(C)sn2)=O)C1 C1(NC(=O)CCc2cnn[nH]2)CN(C(=O)Cn2cccn2)CCC12CCOCC2 C(C(O)C(=O)N(CC(C)(C)NC(c1coc(Cl)c1)=O)C)SC c1(C(NOCC(=O)N(CCCSC)C)=O)cc(C)co1 CCC(CCCC(=O)NC1CC2COCC(C1)C2)NC(=O)C(O)CCN(C)C CCS(=O)(=O)CC(=O)NC1(CO)CN(C(=O)C(O)CC2CCCCC2)C1 C1(CC#C)(C(=O)NC2CCC(CNC(=O)CC3CC3(Cl)Cl)C2)CCOC1 C1(NC(c2ccc([N+](=O)[O-])nc2)=O)CN(C(c2nocc2Cl)=O)CC(F)(F)C1 N1(C(CC2CCC(=O)NC2=O)=O)C2CCC1CN(C(c1ncc[nH]c1=O)=O)C2 N1(C(C2N(C)CC2)=O)CCC(CO)C(NC(c2n[nH]c3c2CCC3)=O)C1 c1(C(=O)NCC(CNC(CCC2C(C)=NOC2=O)=O)O)cc(C)nc(Cl)c1N S(=O)(=O)(c1ccc(NCC2CCCC23CCC3)c(F)c1)NC(CCC)C(=O)NC N1(C(CNS(C)(=O)=O)=O)CCCN(C(=O)Cn2nccn2)CCC1 c1(C(C(C)C)O)ccc(C(C)C(=O)NC2CC2)cc1.C(=O)C(C)(C)C1CC1.C C1(c2ccc(OC)cc2)CS(=O)CCN1CCCC1CCCCC1 C1(CC(=O)NC(c2n(CC)ncc2)C)CCCN(C(c2cnc(C)s2)=O)C1 N1(C(CC)=O)CCCC(C2CCCN2C(C2(c3cc[nH]n3)CCC2)=O)C1 Cc1nc2ccccc2c(C(N2CC(CO)(NC(C3CC3C)=O)C2)=O)c1O c1(C(=O)NCC2N(C(CCCCCC=C)=O)CC2)oc2ccccc2c1OC CC1CCC(NC(c2cccc(CO)c2)=O)CN1C(c1cn(C(C)(C)C)cn1)=O N1(C(CCCCOC)=O)CCCC(NC(=O)C2=C(C)OCC2)CC1 c1(C(C)(C)OC)nc(C)c(C(=O)NCC2CC(NC(=O)CF)C2)s1.O c1(C(N(CCC)CCNC(C2CCCC2)=O)=O)[nH]c2c(c1C)CCCC2 c1(CC)cc(=NC2CN(C(c3c(Cl)csc3Cl)=O)CC2C)[nH]c(CC)n1 c1(C(=O)OC)ccc(O)c(C(C)=O)c1.c12c(cnn1C)CCNC2=O c1ccc([N+](=O)[O-])cc1C(C)=O.CC(C)C(C)CCNC(=O)CC1C=CCC1 C(=O)(CCN(OC)C(=O)c1cnsc1)N1C(CC)CC1 Cc1cc(CNC(C2(CNC(=O)CC3CCOC3)CC2)=O)c(C)s1 C1(NC(C(C)(CO)NC(c2n[nH]c(C)c2O)=O)=O)CCCC(C)(C)C1 c1(C(c2n(CC)nnn2)NC(CCO)c2ccco2)c(C)nc2cc(Cl)ccn12 C1(C(N(C(C(=O)NC(C)C(C)(C)O)(C)C2CC2)C)=O)CCC(F)(F)C1 C(=O)(CC1CCc2ccccc21)N1C(CC(=O)Nc2cc(CC)no2)CCC1 C1(NC(C=CCCC)=O)CCCC(NC(c2cc(C(C)C)ccc2O)=O)CC1 Cc1nn(CC(=O)N(C(C)CNC(=O)COCC2CCCO2)C)c(C)c1Br c1(CC(=O)NCCSCc2cc(F)ccc2Br)cnc2c(=O)[nH]ccn12 Cc1cc(Cc2ccncc2)n2ncc(C#N)c2n1.c12nc(C)c(s1)CC(=O)S2 c1(C(N(CCNC(c2c(C)nn(C)c2)=O)C(C)C)=O)cc2scnc2[nH]1 C1(CC(=O)NC2(C)CCN(C(=O)CN3CC4CC4C3)C2)CCCCCC1(F)F C(=O)(CC(F)(F)C(C)(F)F)N.N1(C(C(C)NC(CC)=O)=O)CCC(CCC)CC1 C1(C(=O)OC)(CO)CCCN1Cc1cnc(C)n1C C1(C(N(C2CCN(C(=O)C(C)=NOCC#N)C2)CC#C)=O)CCCOC1C C1(CNC(CC(C)OC)=O)CCCC2(CN(C(c3ccno3)=O)C2)O1 N1(C(CC(C(C(C)C)C)C)=O)CCC2(CC1)CN(C(=O)CSS(C)(=O)=O)CCO2 N1(C(COCCC#C)=O)CCC=C(C(=O)NC(c2nnnn2C)C)C1 Cn1nnc2cc(C(N3CCC(C)(C(=O)NCC#N)C3)=O)ccc12 C(CC1=CCCCC1)N(C(C1N(C(c2ccc(C)[nH]2)=O)C(C)C1)=O)C c1(NC(=O)NCC2CCCN2Cc2ccccn2)ccc([N+](=O)[O-])cn1 n1(Cc2n(CC)ncn2)c(N(C)Cc2cc(C)cs2)nnc1C1(OC)CCOC1 C1(NC(C2CC3C=CC2CC3)=O)CC(C=O)C12CCC2.C1CC(C(F)(F)F)C1 N1(C(C(=O)NC)C2CC2C(=O)OCc2cc(CO)no2)CCOCC1 Cc1cc(C(N2CCN(C(=O)CC(C)c3cccnc3)CC2C)=O)ncc1N C(=O)(C#CC1CCCC1)NC1CC=C(C(=O)NCC(=O)OCC=C)C1 C1(CC)CCN(C(=O)CCCNC(C)=O)C1C(N1CC(CO)C(C)C1)=O c12ncc(s1)C(=O)NCC(C)(CO)NC(=O)OC2.C(C)(C)(C)OC C1(CC)CC(C(=O)NC(C)CN(C(=O)C2=CCOCC2)C)CCC1=O c1(C(=O)N)ccc(P(C)(C)=O)nc1.C1(NC(c2c(C)cno2)=O)CC2CCC2C1 c1(C(N2CC(CNC(C3CCC(F)(F)CC3)=O)OCC2)=O)csc2cnccc12 c1(C=O)ccccn1.C(=O)(CCC)OCC.c1(C2C(C=O)C2)cnn(C)c1.N C1(NC(c2cc(SC)oc2)=O)CC(C)N(C(=O)CC2(n3cccn3)CC2)C1 C1(C#N)(C(=O)NC2CCN(C(c3ccc(CCC)[nH]3)=O)C2)CC(C)C1 C1(C(=O)NCC2C(C)CN(C(=O)CNC=O)C2)CCn2c(O)nnc2C1 C1(CNC(CCCOCCC)=O)(OC)CCN(C(c2nc(=N)cc[nH]2)=O)C1 c1(CC(=O)N(C2CN(C(=O)CN3CCNC3=O)CC2F)C)cncc(Br)c1 C=Cc1cc(C(=O)NCC(CC)CC)cc(F)c1.C(=O)C(C)C=O.C(C)(C)C.N c1(C(N(C2CC(NC(c3cccc(OC)c3)=O)C2)C)=O)ccc(F)c2ccoc12 C(=O)CC(C)(C(F)F)N(C)C.c1(SCC)cc(C(=O)NC2CCCC2)ccn1 c1(NC(C2CCCN(c3ncc(C4CC4)cn3)C2)=O)cnc2ccc(Br)cn12 N1(C(=O)CC2CC2C(F)(F)F)CCC2(CCCCC2)CC1.C1(C=O)CC12CC2.N N1(C(C(=O)NC(CC)C)CCc2ccc(F)cc2)CCSC2(CCOCC2)C1 Cc1[nH]c(-c2ccco2)nc(=O)c1C(N1CCC1C)=O.C1(C(=O)N)CC(F)C1 c1(C(N2CC(CC=C)(C=O)C2)=O)cnn(C)c(=O)c1.N1(CCC)CCCC1.N N1(C(CC2N(CC)C(=O)CC2)=O)CCC(O)(c2ccc(Br)cc2)CC1 CC(CF)CC(=O)NCC1(NC(c2cccc(N3CCOCC3)c2)=O)CC1 N1(C(CCC=C)=O)CC(CNC(=O)C(C)OC2CCCCC2)C2(CC2)C1 c1(COCC(CN(C(=O)Cc2nccn2C)CCOC)O)ccccc1 C1(N=c2[nH]nc(C3CC3)o2)(CNC(c2cnn3c2CCCC3)=O)CCOCC1 CC1(C)CCC=C(C(=O)Nc2ccc(C3CNC(=O)C3)cc2)C1 c1(C(C)C)nccc(NC(=O)C(=O)NC(C)C(c2cccc(Cl)c2)O)n1 c1(OC)cccc(CNC(=O)C(C2CCCN(C(c3c[nH]c(=N)o3)=O)C2)C)c1 C#CCC(C)(C)C(=O)N1CCCC(CN(C)C(c2csc(Br)n2)=O)C1 Cc1c(C(=O)NCC(C(C)C)NC(=O)C(C)C2CCC2)noc1-c1ccccc1 c1(CN(C(=O)C(=O)N(C)C(C)C2CC2)C(C#C)C2CCC2)ccccc1 N1(C(C(CCCC)C)=O)CC(CNC(=O)CNC(=O)CC)OC(C)(C)C1 c1(C(=O)NC(CC=CC)C(=O)NCC(C)F)ccc2n[nH]cc2c1 c1(C(N2CC(C)(CC(N3CC(O)C(F)C3)=O)C2)=O)ccc2cccc(Br)c2n1 c1(OC(C)C#N)cccc(CC(=O)NCc2ncccc2O)c1 c1(OC)c(C(N2CC=CC(NC(=O)CC3CC3)C2)=O)cccc1C(F)F.O CC1CC(C(=O)NCC2(F)CC(NC(=O)COC3CCOC3)C2)=NO1 C(=O)(C(C)CCCC(C)C)N1C(C)CN(C(C=C(C)c2ccccc2)=O)C(C)C1 C1(CCNC(COCC#C)=O)CCCN(C(C2C(C#C)C2(C)C)=O)C1 N1(C(c2conc2CNC(C23CSCC2C3)=O)=O)CCC(CO)CC1 Cc1cc(C=CC(=O)NCC2CCC2)c[nH]c1=N.C1(CC=O)CCC(C)CO1 C1(NC(C2CCCCO2)=O)CCOC(CNc2nccc(O)n2)C1.C1(Br)CC1 N1(C(Cc2c(SC)cccc2)=O)CCCCC(C2CN(C(=O)CNC(C)=O)C2)C1 O=C(CCCCNC(=O)CC12COC(C1)C2)NC1COCC1NC(N)=O C1(C(=O)OC)CN(C(=O)CSc2cccc(S(N)(=O)=O)c2)C2(CCOCC2)C1 C(=O)(CC(C)(C)CN(C)C)NC1(C(=O)NC(C(CC)C)C)CC(O)C1 C1(NC(COCCCC#C)=O)CCC(C)N(C(=O)Cc2c(C)noc2C)C1 Cc1ccc(C=CC(=O)NCC2C(C)CCN2C(=O)CCn2cncn2)nc1 Cc1ccc(OCCCC(=O)NC2CCN(C(=O)C(C)(O)C3CC3)C2)cc1 O=S(=O)(CCC(F)(F)F)N1CCOC(CNCc2c(Cl)cc(Cl)cc2Cl)C1 Cc1ccc(C(=O)NCC2CCC2C(=O)NC(c2ccncc2F)C)c(C)c1 C(=O)(C1CCc2c(Cl)cccc21)NC1C2(c3cccc(C(F)(F)F)c3)CC(C1)C2 Cc1c(C(=O)NC2CC(C)CN(C(=O)C=CCO)C2)nn2c1CCCC2 N1(C(C2N(CCC)CCC2)=O)CC(NC(c2cc(CO)[nH]n2)=O)C2(CC2)C1 N12CCCC(CC1)N1CCC(C1)CC2=O.C1(Cc2c(C)n[nH]c2)CCC(O)C1O CCC(CC(=O)N1CCCC(N(C)C(c2ccc(N)cc2O)=O)CC1)C(C)(C)C C1(NC(C(c2cccc(F)c2)C)=O)CCN(C(c2coc(Cl)c2)=O)CC(O)C1 C1(C(N2CC(C(C)NC(c3ccc(C(N)=O)cc3)=O)C2)=O)CCn2ncnc2C1 CC(C)C(CNC(=O)C=CC1CCOC1)N=c1nc[nH]cc1C#N c1(C(N(C)CC2CN(C(=O)C)C2)=O)ccc([N+](=O)[O-])cn1.c1ccc(F)cc1 CC(C)(COC1CCCC1)C(=O)N1CCC(C)(CCNC(=O)CCF)C1 C(C)(CCC(=O)NC1C2CC1N(C(=O)CSCC1CCCCO1)C2)SC C1(C(N2CC3C(CNC(=O)Cc4ccccc4I)(C3)C2)=O)CCCCC1(F)F Cc1cc[nH]c1C(=O)NC1CC1CNC(=O)Cc1nccn1C N1(C(C(Cc2c(C)n[nH]c2C)C)=O)C2CCC1C(F)C(NC(=O)C=CCF)C2 C1(OC)CC2(C1)CC2NC(C1CCCN(C(C2CC(F)(F)C2)=O)C1)=O N1(C(C2C(OC)C2)C)C(=O)NC(C(C)C)C1=O C1(CN2C(CCCNC(C3(c4ccn(C)n4)CC3)=O)CCC2)CCC2CC2C1 c1(N(C(C2N(C(C3N(CCC)CCC3)=O)C(C)C2)=O)C)ccc(C)c(F)c1 n1(CC(=O)NC2C(CNC(C(C=C)O)=O)CC2)cnc2ccccc12 c1(CC(N2CCN(C(c3c(C)scn3)=O)C(C)CC2)=O)c[nH]c2nccc(Cl)c12 c1(CC)ccc(O)cc1C(N1CCC2(CC2NC(c2cccc(S)c2)=O)C1)=O C12CCCC1CCN2C(c1ccc(Cl)o1)=O.c1(C(=O)NC)cnc(C(F)F)nc1 C1(C)(CCNC(C2(OC)CCCOC2)=O)CCN(C(c2nc(C)oc2C)=O)CC1 Cn1ccc(C2(C(=O)NCCC3(O)CN(C(C4(CF)CC4)=O)C3)CC2)n1 C1(NC(CNS(N(C)C)(=O)=O)=O)CCCC12CN(C(C1CC(C)(C)C1)=O)C2 O=C(C1=CCCN(Cc2ccc(O)cc2)C1)Nc1ncc(Cl)cc1Br c1cc(C(c2nnnn2C2CCCC2)NC2CC(C3CCC3)C2)c2c(c1)CCC2 O=C(C1CCCc2ccccc21)N1CC2CC(CO)CC12 c1(OC2CCCN(C(=O)Nc3ccsc3Cl)C2)ccc(F)c(F)c1 CCCC(O)(CCC)CC(=O)N1CCC(CCNC(c2ccn(C)n2)=O)C1 N1(C(c2cnc(C)o2)=O)CC(C)OC(C)(C)C1.C(=O)C(C)(C)C.C(=O)CC.N c1(OC)nc(C(N2CCCC(CC(N)=O)C2)C(=O)NCC(C)C)ccc1C C(=O)(N=c1cc(Cl)cn[nH]1)c1cncc(NC(C2C(C(N)=O)C2)=O)c1 N1(C(C(C)NC(CC)=O)=O)CCCC12CCC(NC(c1cnc(O)n1C)=O)CC2 Cn1ncc(CC(N2CCC(O)C2)=O)c1C(F)F.c1(C(=O)N)conc1C1CC1 c1(NCCN(CCCC)C(=O)C2CC2)ncc(Br)cc1C#N C(=O)(C1=CCCOC1)NC1CCCN(C(C(C)CN2CCCCC2)=O)C1 Cc1nccc(C(N2CCN(C(=O)CC3COC(=O)C3)CC2CF)=O)c1C c1(C(=O)NCCCNC(c2[nH]c3cc(C)sc3c2)=O)cnn2c(C)c(C)ccc12 C(CCCC(F)(F)F)NC(=O)CCC1CCCN1C(=O)C=Cc1ccoc1 C(CNC(c1csc(C)c1)=O)(CC(=O)NCc1cccnc1Cl)OC c1(NCc2c(C(C)C)noc2)ncccc1S(=O)(=O)NC1CC(CF)C1 c1(CNC(C(O)OCC)=O)ccc(C(=O)N)nc1.N1(CC)CCCC(F)C1 C(=O)(C(O)CC(C)(C)C)N(C1CCC(NC(c2sccc2CO)=O)CC1)C C1(NC(c2cc(C)no2)=O)CCC2(CCN(C(c3ccc(C)n(C)c3=O)=O)C2)C1 C(CCCC(=O)NOC(CC(C)C)C(=O)NC(C)CC(C)C)SC c1(C(=O)NCC(CO)NC(c2ccc(CC)nc2C)=O)ccc(O)c(F)c1F c1(C(N(C2CCN(Cc3ccccc3)C2)C)=O)cc2c(nc3ccccn23)s1 CC(C)CC(C(=O)NC(C(=O)Nc1cnn2c1CCCC2)C(C)(C)O)C(N)=O Cc1cn2ccc(C(=O)NC3(C)CCC(C)(C)CC3)cc2n1.C(=O)C(C)(F)F.N c1(C(=O)NC23CN(C(C(C)(O)C4CC4)=O)C(C2)C3)ccc2nc(S)oc2c1 [N-]=[N+]=NC1CCC(C(=O)NCC2CC(NC(=O)C#CC3CCC3)C23CCC3)CC1 C(C(C)CC(C)C)NC(CNC(=O)OC)=O.C(=O)C(C)=CC(C)(C)C.N C1(C)(C(N(C(CNC(c2[nH]nc(OC)c2Cl)=O)C)C)=O)COc2ccccc2O1 N1(C(COCC(=O)OC)=O)CC=C(C(=O)NC(C(O)CO)C2CC2)C1 O=C(CC1CCCCN1C(c1cncc(O)c1)=O)Nn1cnnc1 C1COCC2(CCN(C(C3(O)CC3)=O)CC2)O1.C1(C(=O)NC)(C(F)F)CC1 C(=O)(C(C)CCC(C)(C)C)N1CCC(CC(C)NC(c2c(C)n(C)cc2)=O)CC1 C1(CC(=O)N(CCOC)CC)CCOC1C.C1(C=O)CN(CC(F)(F)F)C1 C(=O)(C1=CCCOC1)NC(C(=O)NCC(C(C)C)C)CO N1(C(C(c2n(C)c(Cl)cn2)(F)F)=O)CCC2(CCN(C(C34CCC3C4)=O)C2)C1 C(=O)(C(C(C)(C)O)NC(c1csc(O)n1)=O)N(CC(O)C1CC1)C C(C(C)(C)CCNCc1cnc(C(=O)O)s1)OC c1(C(=O)NCC(CNC(C2(C#N)CCN(C)CC2)=O)O)cc2ccccc2cn1 C12(Cn3c(N4CCC(c5n(C)ncc5)C4)nnn3)C3C4C5C3C1C5C24 C1(C)(CC)CC(NC(=O)CC2CCC2O)CCO1.c1(C(=O)N)cnn2c1OCC2 C(=O)(C1=CCCC1)NC(C)C(C1CCCCC1)NC(c1nn(C)cc1Br)=O Cc1ccncc1C(N1CC2C(CNC(=O)CCC(C)C)C2C1)=O c1(-c2scc(C)n2)ccccc1NC(c1cccc(Cl)c1)c1nnnn1C(C)C C1(NC(c2cc(CC)no2)=O)C2CCCC1CCC2.c1(CC=O)nc(=N)[nH][nH]1.N C1(C(N2CCN(C(c3n[nH]c(C)c3F)=O)CC2C(C)C)=O)CC2CCCC(C1)C2 O=C1OCC(C(=O)NC2CC2NC(c2ccc(Cn3cccn3)o2)=O)O1 c1(SCCN(C(C2CCC2c2nncn2C)=O)CC)ccc(Cl)cc1 c1(-c2nc(CCOC)on2)ccc(C(=O)OC2CCNC2)cc1 C1(C(=O)NC(C)C(CO)NC(c2c[nH]c(=N)s2)=O)CCCN(c2ncccn2)C1 N1(C(c2cc(CC)[nH]n2)=O)CCN(C(=O)CCCCCF)C2CC12 c1(C(=O)NCCN(C(c2cc(SC)ccc2C)=O)CC)c(N)sc2ccccc12 C=C1CC(C)(C(=O)NCC(O)CNC(c2cn(CCOC)nn2)=O)C1 C1(C(=O)NCCc2cn(-c3ccc(Br)cc3)nn2)CCOC2(CCS(=O)(=O)C2)C1 c1(C(=O)NCC2CN(C(CN(C)CCO)=O)C3C2C3)ccc2[nH]ccc2n1 CC1CN(C(=O)CC(C)(C)N(C(=O)C=CCN2CCC2)C)CCC1CO c1(OC)cc(Cl)ncc1CN1CCOCC1CC(=O)NCCc1ccncn1 C1(NC(C2(C(N)=O)CC2)=O)CC2CCC(C1)N2C(c1ccc(F)nc1F)=O c1(CC)ccc(CC(=O)NC2CCCCC2CNC(c2cnc(O)s2)=O)cc1 CC1CC(C(=O)NNC(=O)C2CC(C)C2)CCN1CC1CC1.C(C)(C)C.C=O c1(C(N2CC3C(CCNC(=O)CCC(F)F)(CC3)C2)=O)cccc2sncc12 C1(C(=O)NC(c2ccco2)C)CCCCN(C(c2cn(C3CC3)cn2)=O)C1 O=C1CC2CCC1(C(=O)NCC1(C3CC3)CCOC1)C2 CC1=C(C(=O)NCC=CC(=O)N(C)CC2(C)CC2)COCC1 Nc1cc2c(cc1C(=O)NC1(c3ccc(Cl)cc3Cl)CCCC1)CCCC2 Cc1cccc(C(N2CC(O)(CN(C(=O)C(O)C(C)(C)C)C)C2)=O)c1Cl c1(C2(C(=O)NC(C)CCNC(=O)CNS(C)(=O)=O)CC2)ccnn1C C(C(=O)NC)(C(C)C)SCC.C1CCOC1.c1(C=O)cccn1C1CCCC1 C1(NC(c2scc(C)c2Cl)=O)CCN(C(=O)Cc2cccc(F)c2O)CC1CO C1(NC(C2(C#C)CC2)=O)CCN(C(=O)CCc2ccc(SC)cc2)CC1F c1(C(N2CCC(C(C)(C)C)(CNC(=O)CO)C2)=O)cccc(C(N)=O)c1F c1(C(N2CCC(NC(=O)COc3ccc(F)c(Cl)c3)C2)=O)ccn2nccc2c1 c1(C(N(C)CCN(C)C(c2ccc(Br)o2)=O)=O)cc(I)n(C)n1 c1(N(C)C)nccc(=NC(=O)C2(F)CCN(C(c3c(F)cncc3Br)=O)C2)[nH]1 c1(C(=O)NCCC(CNC(C)=O)(C)C)cc2c(C)ccc(Br)c2[nH]1 c1(CC)cccc(C(=O)N(CCCNC(=O)CC2C=CCC2)CC)c1N c1(CC)ccc(C(=O)NCC2(C(N3CCC(C(F)(F)F)C3)=O)CCCO2)[nH]1 N1(C(C(c2cccs2)NC(CCC2C(C)C2)=O)=O)CCC(O)C(C)(C)C1 CC1CC(C)CN(C(C2C3CC4C(C3=O)C24)=O)C1.c1(C=O)cccn1C1CC1 c1(C(=O)NCCC(N)Cc2ccccc2)cc2c(cn1)[nH]c1ccccc21 C1(NC(CC(C)SC)=O)C=CCC(C(=O)NC2(c3n[nH]c(C)n3)CC2)C1 C1(CNC(C2Cc3nncn3C2)=O)CC(F)(F)CN1C(=O)Cn1cccn1 CCC(CO)(C(=O)NC1CC=C(C(=O)NCC2(Cl)CC2(F)F)C1)OC C1(CNC(C2N=C(C)SC2)=O)CC2CCC1N2C(=O)C=CC(N)=O C(=O)(C1=C(Cl)CCC(C)C1)N(CC(C)CNC(C1(CF)CCC1)=O)C N1(C(c2n(C=C)nnc2)=O)CC2(CCN(C(C3CC(C)CO3)=O)CC2)C1 c1cc(F)cc(Cl)c1Cl.c1(C(=O)OC)ccn(C)n1.C1(O)(CC(=O)N)CNC1 N1(C(COC2(C)CCCC2)=O)CCC(C2(O)CN(C(=O)CN3CCCC3)C2)CC1 C1(NC(C2C(C)(C)C2)=O)CCCCC1NC(=O)Cc1cnns1 N1(C(c2ccc(C)s2)=O)CC2CN(C(=O)C=CCN3CCCC3)CC2C1 C(CC(=O)NCCCOC(=O)NC)(CC(C)C)NC(C1CCC(=C)CC1)=O Cc1ccc(CCC(=O)N(C(CNC(=O)CC2CC2(C)C)C2CC2)C)cc1 C1(C(=O)NCCc2cc(C)[nH]n2)CC2CC1CC2NC(c1nscc1C)=O CC(CNC(=O)Cc1cncn1C)CC(=O)NCC1CC(C(C)(C)C)C1 Cc1ccc2cccnc2c1C(=O)NC1CCN(C(c2cc(F)c[nH]2)=O)CC1C Cc1cc(NC(c2cncn2C(C)C)c2nnnn2C(C)(C)C)cc(Cl)c1 CN1N=C(C(=O)N2CC3CCC3(C(=O)Nc3nnnn3C)C2)CCC1=O N1(C(CCC=C)=O)CC(CNC(c2cnn(C(C)(C)C)c2)=O)C2CC12 CC(C)C(F)(F)CC(=O)NCCN1CCC(NC(C2COC(=O)N2)=O)CC1 C1(CC)CCCCC1C(=O)NC(c1cn(C)nn1)C(=O)NCc1ccccc1F c1(NC(CNC(c2ccc(Oc3ccccc3)cc2)=O)=O)cnc2[nH]ncc2c1 C1(F)(CNC(C(C)C#N)=O)CCN(C(=O)C(c2ccccc2Cl)(F)F)CC1 c1(C(NOCC2CCCC(=O)N2)=O)ccc(F)cc1I C1CCN(C(=O)C(C)(C)C2(C)CC2(F)F)C1.C1(CC)CN(CC(=O)NC)C1 C(CC(C)N=c1ncnc2[nH][nH]c(C)c1-2)NC(C(CCC)OC)=O c1(C(N2CCC(NC(C(C)SC(F)(F)F)=O)C(O)C2)=O)cnc2n(c1=O)CCS2 C#CC1(NC(=O)C=CC(c2cc(Cl)nc(C(C)(C)C)n2)=O)CCOCC1 c1(SCC)cc(C(N2CCCC(C(=O)NCCC(=O)OC)C2)=O)ccc1OC C=C(C)CC(C(=O)N1CCCC(O)(C(C)C)C1)NC(c1cc(C)nnc1C)=O n1(CC)[nH]nnc1=NC(=O)N1CC(C2CCCN2C(C)=O)C1 c1(OCC)cncc(NC(=O)C(F)CC2CC(F)(F)C2)c1 Cc1cc(C(N2CCC3CN(C(=O)CC4CCOCC4)C3C2)=O)c(C)nc1C N1(C(CCOC)=O)CC2CCCC2(NC(=O)CCC(C)(C)c2ccccc2)C1 C(C(COC)CC(=O)N1CC2CC1C2CNC(=O)CC)OC.c1nnnn1C.S S(=O)(=O)(c1cccs1)NC(C)C(N1CCCC(c2cccnc2)C1)=O C1(C(N(CCCCC)C)=O)CCCN(C(C2(C(=O)OC)CC2)=O)C1 c1(CC)nn(C)c(CC(N2CC(c3cn(C4CCOC4)nn3)C(O)C2)=O)c1Br C1(NC(C2(C(=O)NC)CC2)=O)CN(C(c2[nH]ccc2C)=O)CC1CO N1(C(C2(C)CCN(C)C2)=O)CC(CO)C2(C1)CN(C(=O)Cc1c(Cl)cnn1C)C2 C=Cc1ccc(C(=O)NCC2CCCN(C(C3CCCCC3)=O)C2)cc1 N1(C(CCNC(=O)NC)=O)CC(NC(c2ccncc2Cl)=O)CC1C C(=O)(C#CC1CCCC1)N1C(C(N2CCC(C(C)O)CC2)=O)C(C)(C)CC1 CCC(CC(F)F)C(=O)NCC1(O)CCN(C(=O)C(c2ccccc2Cl)C)CC1 C=CCC(CC=C)C(=O)N1CCC(C)CC1C(=O)N(CCO)CCOC C1(CNC(C(CC)N(C)C)=O)CCC2(CN(C(=O)Cc3ncc(C)o3)C2)O1 C(=O)(CC(CCc1ccccc1)C(F)(F)F)NC1CN(C(C(C)CN(C)C)=O)C1 C(=O)(C1(C)CCn2c(C)nnc21)NC1CC2(CN(C(C(F)=CC)=O)C2)C1 C1(C2CCN(C(C34CCC(OC)(CC3)C4)=O)C2)(NC(C(CC)OC)=O)CC1 C=CCC(C(=O)NCCCC1(NC(=O)C(F)OC(F)(F)F)CC1)OC CC1(C)CC1(C(=O)NCCN1CCCCC1)NC(c1nocc1Cl)=O C#CC1(NC(C2CN(C(=O)CC(C)CN(C)C)CC2(F)F)=O)CCC(C)(C)C1 C=C(CNC(=O)CC12CCC1CN(C(C1CCCCC1)=O)C2)c1ccccc1 C#CCCCC(C)C(=O)NC(C)(C)CC(=O)NCc1nc(N(C)C)n[nH]1 C(=O)(C1=CNS(=O)(=O)N=C1C)N(CCC(C(C)C)NC(CC(C)OC)=O)C Cc1c(NC(=O)NC2CCCC3(CCC3)C2)ccc(Cl)c1Cl CCCC(C(O)C(=O)NCC1CC(=C2CC2)C1)NC(=O)C(C)(C#N)CC N1(CCC(=O)NC(C2CN(C(c3c[nH]nc3Br)=O)C2)C)CCCCC1 C(C)(C)(CCCC(=O)NCC1(CO)CC1)NC(CN(CC(C)(C)C)C)=O C#Cc1ccccc1CC(=O)NC(C(=O)NC(c1csnn1)C)C(C)(C)C N1(C(CC(CNC(C(C)S(N)(=O)=O)=O)(C)C)=O)CC2(CCC2)CC1CO C=C(C)CCCN=c1[nH]c(=NC(CNC(=O)C(F)(F)F)C(C)C)c2sccc2[nH]1 c1(SC)cccc(N2CC(C(=O)NCCNC(C3(C)CCCO3)=O)CC2=O)c1 c1(OC)ccc(-c2cnc(F)c(C(N3CCN(CCN(C)C)CC3)=O)c2)cc1F CC1(C)CC(NC(c2ccc3cc[nH]c3c2)=O)CN(C(=O)CS(=O)(=O)CCO)C1 N1(C(C=COCC)=O)CCC2(CC1)CC2NC(c1ccc(Cl)c(F)c1F)=O N1(C(CC2CC(=C)C2)=O)CCC(CO)(C)C1.c1(C(=O)N)cncc(C(C)=O)c1 C12CC(C1)N(C(=O)C)C2.Cc1nccn1C(C)C(=O)N.C(=O)C.C(C)=O c1(CNC(C2C(C=C)C2)=O)nc(CNC(=O)C(C)C#N)cc(O)n1 c1(C(=O)NC2CN(C(c3cc(CC)oc3C)=O)CC2O)csc2cccnc12 n1(C2CC(C(=O)NC(C)(C)C)C2)nc(-c2cccs2)nc1C1CC(OC(F)F)C1 N1(C(CCn2ccc(=N)[nH]2)=O)CCOCC(NC(C2CC3CCC2O3)=O)C1 C1(F)(CNC(c2cn(C)nc2)=O)CCN(Cc2cnc(Cl)c(F)c2)CC1 N1(CC(=O)NC)CCC(NC(=NCC2CC2(C)C)NCC2CCCO2)CC1 C1(C(=O)NCC(C(=O)NC2CC(C)(C(N)=O)C2)N(C)C)CCCCC1O c1(C(N2CCCC(CNCc3cc(C)cc(Br)c3)C2)=O)n[nH]c2ccc(Br)cc12 C1(C(=O)NC(CNC(c2nccc(C)c2)=O)C2CC2)CCc2nnc(C)n2C1 c1(C(=O)NC2C(NC(=O)CC(C(F)F)c3ccccc3F)C2)cccc(F)c1Cl C(=O)(C(C(C)NC(c1cc(C)n(CC)n1)=O)C(C)C)NCC=C=C N1(C(c2n(C)ncc2)=O)CCCC2(NC(C3CCCCNC3=O)=O)CC2C1 c1(C(=O)NC2CCCC(NC(CC=C=C)=O)C2)c(-n2cccn2)cccc1F N1(C(CC(C(F)F)NC(C2N(C)CC(O)CC2)=O)=O)CCN2CCCC2C1 c1(C(=O)NCC2C(NC(C3CC(N(C)C)C3)=O)CCC2)cccc2nsnc12 Cc1c(C(=O)NCC2(C)CCCN2C(c2cccs2)=O)c[nH]c1C#N C(=O)(C1=COCCC1)NC(C)CN(C)C(C1CCCN1C)=O CCC(C(=O)NC(CNC(c1ncn(C(C)(C)C)n1)=O)C(C)C)n1cncn1 c1(C(N2CC3(N(C(C(C)NC=O)=O)CCC3)C2)=O)ccccc1S(C)(=O)=O C1CC(=O)N(CC)C1.C1(NC(C2(SCC)CC2)=O)CCC(CC=O)C1.N CCC(F)(F)CC(=O)N1CCC(C)C(NC(c2ccccc2O)=O)C1 Cc1cnc2cccc(C(=O)NCCCCNC(=O)CCC(C)C#N)n12 CCC(CC(=O)N(C)CCn1cc(C)cn1)N(C(=O)C(CO)OC)C C(C(C)CC(=O)N1CCCC1C(C)(C)C=O)OC.C(CC1CC1)CC1CC1.N N1(C(C2C(=C)C2)=O)CC(=O)NCC1C(=O)NCC1(C)CCC1 Cc1cc(C#N)cnc1N1CCC(NC(c2nc(=O)n(C)[nH]2)=O)C(F)C1 Cc1ccccc1CC(=O)NCCN(C(=O)CC1COCC(C)O1)C.C1CC1 C(=O)(CCC(C)(C)C#N)N(C)CC1C(NC(C=CC=CC)=O)CCC1 N1(C(CCCOCC)=O)CCCN(C(C2C(C)C2(F)F)=O)C(C(C)C)C1 c1(C(N(CCC(C)NC(c2cc(C)c(F)cn2)=O)C)=O)cc(Cl)c(N)cc1F c1ccc(Cl)cc1.CCC1(C)Cc2cn1nn2.C(=O)(COCC)OCC.CCO c1(OC)cc(C(=O)NC(c2ccccc2)CNC(=O)C)c(Cl)cn1.C1CC1 CCC(C)CC(=O)NCCCN(C(=O)C(C)C(C)C)C(C)C N1(C(C(C)OC)=O)CCCC(N(C(=O)C(C)OCCc2ccccc2)CC)CC1 C(=O)(C(C)(C)C(=O)N1CCC2(NC(c3cn4ccnc4s3)=O)CC2C1)N(C)C CC1C(C)N(C(c2cccc(-n3cncn3)n2)=O)CCN1C(=O)Cc1cnsc1 N1(C(C(CO)NC(N)=O)=O)CCN(C(=O)Cn2cccnc2=O)CC1C(F)F c1(OCCC)ccc2ccccc2c1CNCc1cc2cccnc2[nH]1 C(=O)(C(C)OC(=O)CC)NC(CN(C(=O)C(C)C1CC1)CC)C c1(CN2CC3C(C(N4CCC(C(=O)OC)C4)=O)(C3)C2)c(Br)ccc(Cl)c1F C1(CC(=O)NC2CN(C(c3cc(C)c(N)cc3)=O)C(C)C2)CCC2(CCC2)CO1 C1(C(=O)O)CCCN2C(=O)N(CCS(=O)(=O)N3CCCC3)C(=O)C12 Cc1cc(C(=O)Nc2ccc(O)cn2)cc2nc[nH]c12 C=CCC(CC(C)C)C(=O)N1CCC2CCN(C(c3ccc(OC)s3)=O)CC12 C(=O)(C1c2c[nH]nc2CCC1C)N1C2C(NC(C(C(=C)C)(C)C)=O)C(C2)C1 N1(C(CC(C)C)=O)CC(F)CC1C(N1CCN(c2ncccc2Cl)CC1)=O c1(OCC)ccc(C(=O)Nc2ccc(NC(C3CCC3)=O)cc2C)cc1C Cc1cc(C(=O)NCC2CC23CCC3)c(C)n1C.C1(C=O)CC(C)(C)CO1.C c12ccc(F)c(c1)C(=O)NC2.O=C1CSC(=O)N1Cc1ccccc1 c1(C(N(CC(CCC)O)C)=O)cccnc1CNC(=O)CN(C1CCCC1)C c1(C(N2CC(O)(CN(C(C(CC#C)O)=O)C)C2)=O)coc2ccccc12 c1(C(=O)NC2CC(NC(c3c(CC)cc[nH]3)=O)C2)cc(C(F)(F)F)[nH]n1 S(=O)(=O)(c1ccc(O)cc1)N1C(C(=O)NC2CCCCC2(F)F)COCC1 N1(C(c2c(CCC)occ2)=O)CCCN(C(=O)C(C)S(C)(=O)=O)C(C(C)C)C1 C1(NC(C2(CC)CC2)=O)CCN(Cc2nc(-c3ccccc3)no2)CC1O CCCS(=O)(=O)C(C)C(=O)N1CCCC1CN(C)C(c1cnc2[nH]ccc2n1)=O C(=O)(CC1=CCN(C(c2cccc3cc[nH]c23)=O)CC1)N(CC(C)C)CCC CC1(C(=O)NC2CCN(C(=O)CC3CC4CC3C4)C2)CCSCC1 CCC(C)CC(C(=O)N(CCCCCO)C)NC(=O)CC(C)C c1(N(C)C)noc(CCC(=O)NC2CC(CNC(c3c[nH]cc3Br)=O)C2)n1 C(=O)(C1CCc2cccnc21)NC1CC(CCNC(CC(C=C)CCC)=O)C1 N1(C(Cc2c(C)cccc2)=O)CC2CCC(N(C(=O)CC(C)C)C)C2C1 c1(NCC(CC(C)C)N(C)C)ccc(S(=O)(=O)NCCc2cnoc2)cc1C#N Cc1cccc2c(CCC(N3CCN(C(=O)COC4CCCC4)CC3)=O)c[nH]c12 Cc1nn2ccccc2c1C(N1CC(CC)C1)=O.C1(C=O)CC(S(C)(=O)=O)C1.N C1(NC(c2nc(CCC)oc2)=O)CN(C(C2CC2(C)C(F)F)=O)CCC1(C)C C(=O)(C1=COCCO1)N(CC(C)NC(C1CC1c1ccncc1F)=O)C N1(C(C=CSC)=O)CCN(C2CCCN(C(=O)CC3CC(F)(F)C3)C2)C(=O)C1 C(=O)(C1CCCn2ccnc21)OC1CC(C)(C)OCC1 C1(NC(c2ccc(C(C)(C)C)[nH]2)=O)CCC(O)CN(C(=O)Cc2ccsc2Cl)C1 CCS(=O)(=O)c1ccc(CC(N2CC(NC(=O)C#CC3CCCCO3)C2)=O)cc1 C1(C(N2CCCC2)=O)CC2(CCCC2)CO1.c1(CC(=O)N)cc(Cl)n(C)n1.C C1(C(=O)NCCOC(CNC(CCC(=C)C)=O)(C)C)CCC2(CCOCC2)CO1 c1(C(=O)NCC(CC)NC(=O)C(C2CCC(=O)N2)C)cc(C)cc2c1OCC2 N1(C(CC(C)F)=O)CCC2OCCN(C(C34CC(c5ccccc5)(C3)C4)=O)C2C1 Nc1ccc2oc(C(=O)NC3(C)CCCC3)cc2c1.C1(CC(=O)N)CCC2CC12 C1(CC(=O)NC)CN(C(c2ccnnc2O)=O)CCN1C(c1ccncc1O)=O C1(C(=O)NC(c2ccnn2C)CC)CC2CC1CC2.C1(C=O)CCC1.C1CC1.N c1(CCC(N2C(COC)C(OC)C(C(=O)OC)C2)=O)ccc2ncccc2c1 c1(C(=O)NC(C2CCCCC2)CNC(CCOC)=O)nc[nH]c1C(C)(C)C O=C(C1CCCc2cncn21)NC1C(Cl)COC1 C(=O)(C#Cc1ccccc1)N1CC(C(N2CCN(CC(C)C)CC2)=O)NCC1 C=CCC(C(=O)N1CC2CC1CN(C(c1cnc(C)cn1)=O)C2)C(C)C C(=O)(CC(C(C)C)NC(=O)CC12CCCC1C2)NCc1nc(CC)oc1 Cc1nc2c(s1)C(NS(=O)(=O)Cc1csc([N+](=O)[O-])c1)CCC2 C1(CC=O)OC(C)(C)OC1=O.c1(CCC(=O)N(C)CCO)ncccn1.CC C1(F)CCN(C(C2COC(C)(C)C2)=O)CC1.C(C1C(C(=O)N)C1(C)C)=C(C)C c1(C(=O)NCC(C(C)C)NC(=O)C(C)(C)C(F)F)ncc2cc(Cl)ccn12 CC1CC(CNC(c2c(Cl)cnn2C)=O)CCN1C(C1CC12CC(C)(C)C2)=O c1(C(=O)NCC(CCCC)NC(c2ccnnc2C)=O)c(N)cccc1Cl N1(C(c2cc(C(C)=O)sc2)=O)CC2CCN(C(c3scnc3Cl)=O)C(C2)C1 Cc1cc(C(=O)NCC(C)(C)CCNC(=O)C(F)n2ccnc2)sc1Cl C(=O)(C1=NOC2COCC12)N1C(C(C)NC(C(CCC=C)(F)F)=O)CCC1 c1(C(N2CCC3CN(C(c4n(C)c(S)nc4)=O)CC32)=O)coc2c1CS(=O)(=O)C2 CCC(CNC(=O)C(CO)NC(=O)C=CC1CC1)C(C)C C12(C(N3CCC(CCCC)C3)=O)CCN(C(c3cccc(F)c3C)=O)CCC1C2 C(C)(C)(CCCC(=O)NCC1CN2CCC1CC2)NC(c1ccc(CC)nc1)=O c1(COC)cccc(C(N2CC(NC(C3CC(O)(C#N)C3)=O)CC2C)=O)c1 C#Cc1ccc(C(=O)NC2CC23CCN(C(=O)C(CC)OC)C3)c(F)c1 N1(C(C2(C)CC(C)C2)=O)CC(C2(NC(=O)CC3CCC(=O)NC3)CC2)C1 c1(C(N2CC(C)(C(=O)NCC3(CC)CCCC3)C2)=O)cccc(NC)n1 n1(CC(=O)N(CC(CNC(CCSC)=O)O)C)cc(C(F)(F)F)nn1 C=CC1(C(=O)NC2CNC(=O)C2(C)C)CCN(C(=O)C=C2CCC2)CC1 c1(C(N(CC)C)=O)ccc(C#N)n1C.c1(C(N(C)CCO)=O)ncc(Cl)cc1F c1(C(=O)NC(CC=C)CNC(c2cc(=O)cc[nH]2)=O)nncc2c1CCCC2 c1(OC)ccc(C(F)(F)CNC(=O)CC2CCC3CC23)cc1 CC1CN(C(=O)COc2cccnc2)CC1NC(=O)Cc1cccc(Cl)c1 N1(C(C(C)CC2CC2)=O)CCC(CO)(CNC(=O)C(N)=O)CC1 CCC(CC)C(F)C(=O)N(CCC(=O)NC(C)CCCO)CC Nc1cnc(C(=O)NC(C(=O)NCC2CCOCC2)C2CCOC2)cn1 c1(OC)ccc(S(=O)(=O)NC2CCSC2)cc1-c1ccc(C=O)o1 C(=O)(CC(=O)N(C(CNC(=O)CC)C1CC1)C)NCC.c1ccccc1.O CC(C)CS(=O)(=O)CC(=O)NC(C)(CNC(=O)C(C)C(F)F)CO c1(C(=O)OC)ccc(C(=O)NCC(C2CCCN2c2ncncc2C)(C)C)cc1 C(C)(c1ccsc1)=CC(=O)NCC1N(C(CC2(C=C)CC2)=O)CC1 c1(OC)ccccc1CC(=O)NCC1CCCCC1.c1(C=O)nc(O)c(C)s1.N N1(c2ccnc(N3CCC(OCC(C)C)C3)n2)CCc2n[nH]cc2C1 C(=O)(CC(C)CCC=C(C)C)N1CC(CC)CCC1.C(=O)(C(C)(C)CC(F)F)N Cc1nnc2n1CCC2(C)C(=O)N(CC(C)(C)NC(c1ccc(C#N)[nH]1)=O)C C1(C(=O)NC2CCN(C(c3cc(C(C)=O)sc3)=O)C2C)Cc2c(F)cccc2O1 c1(C(=O)NCC(CNC(C2CCCNC2=O)=O)OC)ccc2sccc2c1 c1(CCNC(=NCC=C)NCCOC)ccc2c(c1)CCO2 C1(NC(CN(C(C(C)C)=O)C)=O)CC2CCCC2C1.C(=O)(CC(C)n1cccn1)N CC1CC2(CC(C(=O)NC3CCCC(C(N4CCCC4(C)C)=O)CC3)C2)C1 N1(C(C2(C(N(C3CC4CC4C3)C)=O)CC2)=O)CCSCC1c1ccccc1 CC1(C)CCOC1CNC(=O)C(C1CCCC1)NC(c1ccc(Cl)s1)=O N1(C(C(CC)C#N)=O)CCC(C)(C)C(CNC(c2cc(NC)ccc2Cl)=O)C1 C1(O)(CNC(=O)C(O)C2CCC2)CCCN(C(=O)CN2CCCC2)CC1 C1(N(C(c2cccc(C)c2)=O)C)CC(C)CC(C)C1.c12cn(nn1)CC(=O)N2 c1(C(=O)NC2CCC2NC(C2(O)CCOCC2)=O)cnn2ccccc12 O=C(CC(F)(F)F)NC1CCCN(Cc2cccnc2F)C1 C(=O)(C1CCCc2c[nH]nc21)NC1CN(C(C(C)N(C)C)=O)C(C)C1 c1(C=O)cc(O)cc(=O)o1.C1(COC)N(C(=O)CCC2CCCC2)CC1(C)C c1(CC(=O)NC2CC(n3cc(CC(CC)(C)O)nn3)C2)cc(Cl)c(Cl)cc1C N1(C(c2ccccc2)=O)CCC(C2(NC(C3CC(c4ccccc4)O3)=O)CC2)C1 Cc1c[nH]c(C(N2CCCC2CCC(=O)Nc2ccnc(C(F)(F)F)c2)=O)c1C c1(N2C(CNC(c3cncc(OC)n3)=O)CCCC2)nc2c(C)cccc2o1 c1(C(=O)NC(CN(C(c2occ(C)c2)=O)C)(C)C)nn(C(C)(C)C)cc1Br CCC(CC)CC(=O)NCC1C2CN(C(C3COC(=O)O3)=O)CC12 c1(C(=O)NC(CC(C)NC(c2cnc(O)s2)=O)C)n[nH]c2c1CS(=O)(=O)CC2 c1(C(N2C(C)(C(=O)NCC3(OC)CCOC3)CCC2)=O)cc(C)cc(O)c1 Cc1ccc(CNC(c2ccccc2)=O)cc1.N1(CC=O)C(=O)C=CC1=O.C Cn1c(C(N2CCCC3(CCCC3)C2)=O)cc2ccccc12 CC(C)C(Cc1ccccc1)C(=O)N(CC(C)CNC(C1(O)CCOC1)=O)C S(=O)(=O)(c1ccc2c(c1)OCO2)NC1C(C(=O)Nc2ccc3ncsc3c2)C1 CC1=NOC(CNC(c2cc(CNC(c3conc3C)=O)[nH]n2)=O)C1 C(=O)(C1CCc2nccn21)N1C(CNC(CCc2cc(OC)no2)=O)COCC1 c1(CC(N2CCC3CN(C(C4CCSC4)=O)CC3C2)=O)noc2ccc(F)cc12 c1(C(N2CCC(NC(CCOC)=O)CC2C2CC2)=O)cc2cccnc2s1 C(=O)(C(C)CC(C)(F)F)N(CCC)CCNC(C1CNC(=O)N1C)=O Cc1cc(C(=O)N(C(C)CC(=O)NC(C)Cc2cccs2)C)nnc1C CCC(C)(C)C(=O)NC1CCC(NC(C2(C)CC2(C)C)=O)C1 N1(C(c2c(SC)snn2)=O)CCN(C(C2CC3(C2)CC3F)=O)CC1C C1(CC)(NC(c2cc(C)nc(O)c2)=O)CCN(C(=O)C=C(C)C(F)F)CC1 C12(C=O)COCC1C2(F)F.c1(CC(=O)OC)ccccc1C(=O)N.CC(O)C C1(NC(C(C)SCC)=O)CCCC12CN(C(c1cc(C)c[nH]1)=O)C2 c1(OC)ccc(C)cc1CC(=O)NC1CCC(C)C1.c1(C=O)cnc(C)cn1.N N1(C(C(C)=C2CCC2)=O)CC2(CCN(C(c3cc(C)ccc3F)=O)CC2)CC1C C1(NC(C2(CCCC)CC2)=O)CN(C(=O)COc2cccnc2)CC1F C(=O)(C1=CC2CCCCCCC12)NC1CN(c2c(CC)cnc(Cl)n2)CC1(C)C O=C(C(O)CC1CCCCC1)NCC1(O)CN(C(c2cnc(Br)s2)=O)C1 N1(C(C23CC(C)C2C3)=O)CC2CC1CN2C(c1cc(CS(C)(=O)=O)on1)=O C1(CC(=O)NCC2(C(=O)NCC(C)(CO)OC)CC2)CCCCC1O CC(C(=O)NCc1cc(C(=O)OC)no1)C(C)(F)F Cc1nc(-n2cc(C3CN(C(=O)C(C)(C)C)CCO3)nn2)sc1C N1(C(c2cc(Br)c(F)cc2F)C(=O)NCCOC)CCOCCOCCOCC1 C1(NC(c2ccc(C)c(O)n2)=O)CNCC2(CCOCC2)C1 c1(C(=O)NC(C)C(=O)NCC2C=CCCCC2)cccc(F)c1N C1(CNC(c2csc(C)c2N)=O)COCCN(C(=O)C2=NOC(C)C2)C1 C(CCCC(=O)N(CCC(=O)NC1CC(CO)C12CCC2)CC1CC1)(OC)O N1(C(CCOCCC)=O)CCCC(C)(C(=O)NCc2ccc(C)nn2)C1 c1(C(N(C)CC2N(C(COCC=C)=O)CCCC2)=O)ccc(=N)[nH]c1Cl c1(C(N2CCCCC2)=O)ccc2c(c1)OCC(=O)N2.CC(C)(C)OC(=O)NC c1(C(=O)NC(CC)C2CC2)cc(CNC(=O)C(C)SC)ccn1 c1(NC(c2cnc(C(OCC)OCC)s2)=O)ccnc(N2CCC(C)C2)c1 C1(C(N2CC(C(=O)N)C2)=O)CCC2(CC1)CC2.C=CC(C)(O)C(=O)NCC C(c1ccco1)=CC(=O)NC1CCCC1NC(=O)COCC1CCC1 N1(C(C2(n3cc(CCCCCCCC)nn3)CC2)=O)CC2CC1(CC)CN2C c1(C(=O)NC2(CC(=O)Nc3ncnc4[nH]ccc34)CCC2)cnc2[nH]ncc2c1 C1(c2ccc(OC)cc2)NC(=O)N(CC2CCOCC2)C1=O C1(C(=O)NC2CCC(CNC(CC3CC(OC)C3)=O)C2)CCCOC1C c1(CNC(CC2(COC)CCCC2)=O)cc(O)ncn1.C1(C=O)CCC1C.C c1(C(=O)NC2C(CNC(C3CCCN(C)C3)=O)CC2)ccc2[nH]nc(Cl)c2c1 C(C)(CC)(CCC)NC(c1nc(C(C)NC(CC=C=C)=O)oc1)=O CC1CC(NC(c2c[nH]cc(Cl)c2=O)=O)CCN1C(=O)CC1COC2CC1C2 C1(CC)(CC)CC(N=c2cc(NCCCC(N)=O)nc(C3CCOCC3)[nH]2)C1 c1(CC(N2CC(N(C(=O)C=CC(F)(F)F)C)C(F)C2)=O)cccc2c1OCO2 c1(-c2n(-c3ccn(CC)n3)nc(CCSC)n2)c[nH]c2cc(OC)ccc12 C#CCC(C)(C(=O)NC(c1nncn1C)CO)NC(C1CN(C)CC(C)O1)=O Cc1ccc(C(=O)N(C)CC2CCCN2C(C2CCCC2O)=O)c(=O)n1C Cc1cc(Br)cnc1C(=O)NC1(C)CCN(C(=O)C(c2cnn(C)c2)O)CC1 c1(OC)cncc(C(=O)NC2CN(C(c3csc(CC(F)(F)F)n3)=O)CC2F)c1 C1(NC(c2n(CC#C)ccc2)=O)CN(C(=O)C(O)Cc2[nH]cnc2C)CC1C c1(OC)cc(F)ccc1C(N1CCCC(C)(CNC(C2CC2F)=O)C1)=O N1(C(CONC(c2cncc(F)c2)=O)=O)CC(C2CC2(F)F)C1 N1(C(C)=O)CS(=O)(=O)CC1C(=O)NC(CO)C(C)NC(c1nn[nH]c1Cl)=O CP(C)(=O)CC(=O)NC1CC(NC(=O)C(C2CCC2)C2CCC2)C1 N1(C(c2ccc(CN(C)C)o2)=O)CC(NC(C2CC2(Cl)Cl)=O)CC12CCOCC2 c1(C(=O)NC(CN(C(c2n(C(C)C)cnc2)=O)C)C)ccc(F)c2occc12 c1(C(=O)NCC2CN(C(C3C(C)N(C)CC3)=O)CC2O)cc2n(n1)CCCC2 C(=O)(CC(C(F)F)NC(C1C2CC(=O)CC12)=O)N(CC1=CCCOC1)C CC(CC=Cc1ccccc1)C(=O)NCCC(O)CNC(=O)CCc1ncc[nH]1 c1(C(N2CCOCC(CNC(C34CC(C3)C4)=O)C2)=O)cccc([N+](=O)[O-])c1 CC(C(=O)NC1CN(C(=O)C(C2CCCC2)C2CCCC2)CC1O)C(F)F C1(C(=O)NCC(CC)NC(c2sncc2Br)=O)CN2CCC1CC2 C(=O)(C1=NOC(C)C1)N1CC2C(NC(COCCCOC)=O)(C2)C1 C1CC2(CCC2)CN1C(C1CCCCO1)=O.c1(COC)cccnc1C(=O)N.C Cc1ccc2nsnc2c1C(N1CC2C(NC(=O)CN3CSCC3=O)C2C1)=O c1(C(=O)NCCC2CC(NC(C(C)=C(C)C)=O)C2)cn2cc[nH]c(=O)c2n1 c1(C(=O)N(C2CCCCC2)Cc2ccoc2)ccc(Cl)c2c1OCCO2 C=CC(CCC)CC(=O)N1CCC2C(C(N3CCC(CCO)CC3)=O)C2C1 c1(C(C(=O)NCc2cccs2)N(C(c2ccco2)C)C)ccc(C2CC2)cc1F Cc1cc(CC(=O)NCC2(NC(C3C4CCC(=O)C34)=O)CCCC2)n(C)n1 c1(OC)ccncc1C(=O)NC1(C(=O)N(C(CO)C(C)C)C)CCC1 C1(NC(C=CC=CC)=O)(C)CCC(F)(F)CC1.C(=O)CCC1CCCO1 c1(C(N2CCOCC(CNC(C3(Cl)CC3)=O)C2)=O)cnc2n1CCC2 C(=O)(C(CO)NC(C1(F)CC1)=O)N1C(C)CC1 CC1CCN(C(c2cnns2)=O)C1C(=O)NCC1CC1 Cc1ccc(C(=O)NCCCCCNC(=O)COC(F)F)cc1C(C)(C)C c1(C(N2CCC(NC(C3=C(C)CCCC3)=O)C2(C)C)=O)cc2ccnc(Cl)c2s1 C1(CC=O)CCCNC(=O)C1.c1(COC)cc(C(N2CC(C)C2)=O)on1.N Cc1cnc(C(N2CCCCC2CNC(C2CCC(=O)N2C2CC2)=O)=O)nc1 N1(C(C2N(C(N)=O)CCC2)=O)CCCCC(NC(=O)C(O)c2ccsc2)C1 CC(C(C)(C)C(=O)N1CC(OC(F)F)C1)NC(=O)CC(O)C1CCCC1 N1(C(C)=O)CCOC(C(=O)NCC2CN(C(=O)Cn3[nH]cnc3=N)C2)C1 N1(C(=O)NCc2cc(C(C)C)nn2C)Cc2ccccc2C2CCC1C2 C(=O)(C(CCC)=CCC)NC(CNC(Cc1cn(CCC=C)nn1)=O)(C)CO C(=O)(C1CCCn2cnnc21)NC(CNC(c1c(C)nc(C2CC2)[nH]1)=O)C(C)C N1(C(C2(NC(C3CN(C4COC4)C3)=O)C(C)(C)C2)=O)CCCC[Si](C)(C)C1 N1(C(=O)COCCOCCO)CC2CC(C1)N(C(=O)CC1CCCCCO1)C2 CCCC(CCCNC(c1c(C)noc1C(C)C)=O)NC(c1scc(C)c1C)=O CCC(F)(F)CC(=O)NC1CCCN(C(c2sc(Br)cc2F)=O)C1 c1(C(=O)N)ccc2nn[nH]c2n1.c1(SC)cc(C)c(C(=O)NCCC(C)(C)C)o1 Cc1cc(C)n2ccc(C(=O)NCC(CNC(=O)CC3CCCC3O)CO)c2n1 C(=O)(C(C)(C)C(C)NC(C1CN(C2CCC2)C1)=O)NCC(CS)OC C1(C(=O)Nc2ccc(CO)nc2)CC(F)CN(Cc2cc(I)ccc2F)C1 C(Cc1cc[nH]n1)(C(=O)NCC(=O)NCC(F)F)NC(COCC)=O CC1CC(NC(=O)C(C)(C)C)CN1C(=O)CCCCc1ccc(Cl)cc1 c1(C(=O)NC(c2cc(Cl)cc(Cl)c2)CCO)cc2cc(Cl)c(Cl)cc2[nH]1 Cc1cc(C(N2CCC(C(=O)N)(CO)C2)=O)nc(O)c1.c1ccn(C)c(=O)c1.C c1(C(=O)Nc2cc(O)ccc2O)ccc2c(c1)CN(C(=O)CCn1cncn1)C2 c1(C(N(CCNC(=O)C(C)(CC)O)CC)=O)cnn2c1NCCC2C(C)(C)C N1(C(=O)OC(C)(C)C)CCC2(CC2)C1.c1(C=O)ccc(Cl)c(C(=O)O)c1.C C1(CCC)(C(=O)N(C)CC2COCCN2C(c2cc(Br)n[nH]2)=O)CCNC1=O CC1CSCCN(C(C2(CNC(c3cn(C)nn3)=O)CC23CCC3)=O)C1 C1(NC(CSC(C)C)=O)CCC2(CC1)CCN(C(C1CC13CCCC3)=O)C2 N1(C(C(CCF)NC(CCOCCC)=O)=O)CCCC(C)(C#N)C1 C1(NC(c2c(C)nn(C)c2)=O)CCC12CCN(C(c1ccc(N)c(F)n1)=O)CC2 Cc1nnsc1NCCNC(=O)NC1CC(C(F)CO)C1 c1(CNC(c2cncc(-c3ccc(C)c(C)c3)c2)=O)ccc2nnnn2c1 n1(CC)cnnc1C(=O)NC(CNC(=O)CCC1CC1(C)C)CC Cc1c(-c2nnc(CNC3(CNc4ccccc4)CC(F)(F)C3)o2)cnn1C Cc1[nH]nc(C(=O)NCc2cc[nH]c2C(=O)NCC2CC3(CCC3)C2)c1C c1(C(=O)NC2C(F)CCN(C(c3c(C)cncc3)=O)C2)cnc2c(Cl)cccn12 Cc1nn(C)cc1C1=NOC(C(N2CCOC(CO)CC2)=O)C1 C1(C(=O)NCC(C)NC(=O)CCOC2CCCCC2)CC2C=CC1CC2 c1(SC)nc(C(F)F)cc(=NCC2CCCCN2C(=O)CC2(C)CC2(F)Cl)[nH]1 C(=O)(C(C)C(=O)N1CC(F)CC1CC(=O)NC1(CCCCO)CC1)OC C(=O)(C1=CCC2CCC1N2C(=O)C(CO)C(F)(F)F)N1CC(=CC)C1 N1(C(c2[nH]c(CC)c(Cl)n2)=O)C2CCC1CC(CNC(=O)C1=C(Cl)CCC1)C2 c1(C(=O)NCCCN(C(c2n[nH]cc2Cl)=O)CC)cncc2c(O)nccc12 C(C)(CCNC(C1CCN1C(=O)C(C)N1CC(C)C1)=O)SC C(=O)(CC(C(F)F)n1ccnc1)N(CCC)CC.c1(C=O)cscc1C(F)F.N Cc1cc(C(N2CCSCC2C(=O)NC(C(C)C)c2nc[nH]n2)=O)ncn1 n1(CCOC)nccc1C(=O)NC1CC(CCNC(C2(C)CC2F)=O)C1 C(=O)(C1=CS(=O)(=O)CCC1)N1CCN(C(C(C(C)O)(F)F)=O)C(C)C1 c1(C(=O)N)ccc(OC(F)(F)F)cc1.C1(F)CCC1.C(=O)C(F)C1CCC1.C N1(C(C(CNC(CC(C=C)(C)O)=O)(C)C)=O)CC2CCC(C1)C2C#N Cn1ccc2ccc(CCC(N3CC(NC(=O)CNC=O)C(O)C3)=O)cc12 C(=O)(C(C(C)(C)C)OC)N1C(C(N(C)Cc2ccc(CC)o2)=O)CC2CC21 C1(NC(CCCOCCC)=O)CCCN(C(=O)C(F)CC2CC2)C1C N1(C(C2(C=C)CC2)=O)CC(CNC(=O)CC=CC)C(F)(F)C1 N1(C(c2ccccc2)C)CCN(C(c2oc(C3CC3)nc2C(F)F)=O)CC1 c1(C(N2CC(c3ccccc3)(NC(CC(C)F)=O)C2)=O)cccc2sncc12 CC1(C)CN(C(C2(CCF)CC2)=O)CCC1NC(=O)C1=C(Cl)CCOC1 CC1C(NC(C2CCOC2)=O)CCCN1C(=O)Cc1ccccc1N1CCCC1 C1(C(N2CC(CCCCNC(CC=C)=O)C2)=O)COc2cc(Cl)ccc2C1 CCC(O)C(F)(F)C(=O)NCCCN(C(c1ccsc1)=O)Cc1ccccc1 Cc1cc(C(=O)NCC2CCN2C(C2CC3CCCCC23)=O)cc(O)n1 N1(C(C=C(C)C(C)C)=O)CCOCC(NC(=O)CCNC(=O)C=CCl)C1 c1(C(=O)OC)cc(N(C)CC2CCN(C(c3ccoc3Br)=O)C2)nc(C)n1 N1(C(C2CCN(C(C)=O)C2)=O)CCN(C(c2ccc(Cl)c(Cl)c2)=O)CC1C1CC1 C(=O)(C#CC1(C)CCCO1)N1CC(O)(CN(C)C(C2OCCOC23CCC3)=O)C1 C1(CNC(C2C(C)C2)=O)CN(C(c2ccc(N3CCCC3)c(F)c2)=O)CCC1C CCCCC(CNC(=O)Cc1coc(C(F)F)n1)NC(=O)C(=O)N.C1CC1 CCCCCCc1ccc(COC(C)(C)C)s1.c12noc(n1)CCNC2 n1(CC(=C)C)c(N2CCC(C3CCCO3)CC2)nnc1-c1cccc(O)n1 c1(CNC(c2c(C)onc2-c2ccccc2)=O)nnc2ccccn12 c1(C(N(C)CC2(O)CCCN(C(C(CC)OC)=O)C2)=O)cc(C)ccc1[N+](=O)[O-] C#CC1(NCc2cc3ccccc3nc2OCCCC)CCc2cc(Br)ccc21 C1(C(=O)NCC(C)(C)OCC(=O)N(CC)CC)CCCC(OC)C1 N1(C(C=NOC)=O)CC2CCC1CN(C(c1cnc3occc3c1)=O)C2 Cc1cc(C(=O)N(C)CCNC(C2(Cl)CC2(C)C)=O)cc(C)c1C#N CC1OCCC1C(=O)N(CCCNC(c1ncoc1-c1ccccc1)=O)C1CC1 c1(C(=O)OC)ccc(F)c([SH](=O)=O)c1.C1(O)CCCN(C(=O)C(C)(F)F)C1.N C(=O)(C1=C(Cl)CCCC1)NC1CCC(CNC(c2c(C(C)C)nns2)=O)CC1 C#CC1(O)CC(C(N2CCC(C)(NC(c3ccccc3COC)=O)C2)=O)C1 C1(C(=O)NC2(C(N(C)CC3CC3(F)F)=O)CSC2)CCCCC1 c1(C(N2CCCC(C)(NC(CC(C)CN(C)C)=O)C2)=O)cc(O)c2ccsc2c1 c1(C(=O)NC(c2nn[nH]n2)C)ccc2c(C3=CC(C)(C)CC(C)(C)C3)c[nH]c2c1 Cc1nc2c([nH]1)C(NC(N1CCC(OC(C)C3CC3)CC1)=O)CCC2 Cc1c(NCc2cnc(O)[nH]2)ncnc1N1CCN(Cc2ccccc2)CC1 C#Cc1cn(C)nc1C(=O)NNC(=O)c1ccc(I)cc1 c1(NC(N(C(C)CF)C)=O)ccsc1-c1ccccc1 n1(CC(=O)N(CCC)C)c(C)c(C)sc1=O.Cc1ccc(C(C)CC(=O)N)cc1 c1(C(=O)Nc2c(C)nn(C)c2C)sc(=NCc2c(Cl)cc(O)cc2Cl)[nH]c1C Cn1cc(C(N2CCCC(Cn3cccn3)C2)=O)c(=O)n(C)c1=O c1(CC(=O)N(C(C)C)CC)cccc(C#N)c1.c1cnc[nH]1.C1(C=O)CC1.N CC1CCC(NC(c2cccnc2N)=O)CN1C(=O)CC1CC2CCC1O2 C1(C(N(CC=O)CCOC)=O)CCOC1C1CC1.C(C)S.C1CC1.N c1(C(N(CC(C)N(C)C(c2nc(Cl)cs2)=O)C)=O)ccc(N=[N+]=[N-])cc1 Cc1ncsc1CCC(=O)N(C)CCN(CC(C)O)C C(=O)(C1SCCc2sccc21)N1C2C(NC(c3ccc(C)cc3)=O)CC(CC2)C1 CCC(C)(C#N)C(=O)N1CCC(C)C(NC(=O)C(c2ccc(C)cc2)(C)C)C1 C1CCN(C(C2(C)CC(C)C2)=O)CC1(F)F.n1(CC=C)cc(C(=O)NC)cn1 CC(C)(C#N)CC(=O)N1CCN(C(c2cnc(S)n2-c2ccccc2)=O)C2CC12 C1(CC)CC(CC(N2CCC(CCNC(=O)COC3CCOC3)CC2)=O)CCO1 c1(C(N2CCN(C(C(C3CCC3)OC)=O)C(C(C)C)C2)=O)c(C)ncn(C)c1=O C(C)(C)(CCCCC(=O)N1CC(NC(c2ccc(C)c(C)n2)=O)CCC1C)OC N1(C(c2nn(C)c(O)c2)=O)CCN(C(c2cc3ccoc3s2)=O)C(C(F)(F)F)C1 c1(CC)ocnc1C(=O)NC1(C)CN(C(=O)Cn2nnc(C)n2)C1 S(=O)(=O)(CC(=O)N(C)CC)NCC.c1(CCC=O)ccc(C(F)F)cc1.N C(c1cnc2ccccc2c1)=CC(N1C(C(=O)O)CC2(CC2)C1)=O N1(C(C(C)OCC)=O)CCCC12CCCN(C(=O)CCS(=O)(=O)N(C)C)C2 c1(NC(c2c(OC)cc(Br)cc2)C)ccc2onc(C)c2c1 C1(C(=O)OC)NC(=O)N(C(C(=O)Nc2cccs2)C(C)CC2CCC2)C1=O C1(C(=O)NC(C2CCN(C(C3CC34CC(O)C4)=O)C2)C)CC2CCCCN2C1 [N-]=[N+]=NCCCCCCC(=O)N1CCC(Nc2ccc(C#N)nc2)C(CO)C1 C(=O)(C(C)CC(F)F)N.C1(C(=O)OC)CCC(C(=O)NC2(C)CCCC2)C1 CCCC(C(=O)NC1(C)CCCC1C)NC(c1nn(C)cc1C)=O c1(C(N2C(CO)CC(NC(C(C)(C)OC)=O)C2)=O)c(Cl)cnc(Cl)c1Cl Cc1cc(C(N2CCC(N(C(=O)Cc3ccncc3Cl)C)C(C)C2)=O)cc(N)c1 c1(CC)ccc(C(=O)NCC(C)(C)CNC(=O)C=CC(C)C)c(O)c1 C=C(CNC(C1CN(C(=O)C(C)=CC2CC2)CC12CCC2)=O)c1ccccc1 c1(CC(=O)NC2C(CNC(C(COC)OC)=O)CC2)c(C)nc(C)nc1O C#CC1(N(C(=O)CC(=O)Nc2nc(C)c(C)s2)C)CCCC1 Cc1ncc(NC(C2(CNC(c3cc(O)ccc3I)=O)CC2)=O)c(Cl)n1 C(c1csc2ccccc12)=CC(N1C2CN(C(CNC=O)=O)CC1CC2)=O C1(CCC)CC(C(=O)NCCCC2CCCN2C(c2ccoc2C)=O)CCO1 c1(C(=O)NCC(C)NC(=O)CC(C)(O)C2CC2)nc[nH]c2nccc1-2 c1(N2CCCC(C(CC)=O)C2)ccc2cc(Cl)ccc2n1 C(=O)C(C)CC(N)=O.n1(CC)cc(C(=O)NCCCCCC)c(C(F)(F)F)n1.N C1(NC(N(C2CCN(c3cc(C)nc(Cl)n3)CC2)CCC)=O)CCC12CCCO2 O=C(C(F)(F)C1(O)CCC1)NCCCCCn1cc(-c2ccccc2)nn1 c1(CC(=O)NC2CN(C(=O)COCCCF)C2)ccccc1O C1(C(N2CCC(N(C(=O)CCc3cnn(C)n3)C)C2)=O)CC2(C1)CC1(CC1)C2 C1(N(C(C2C(COC)C2)=O)C)CCN(C(c2cc(C3CCOCC3)on2)=O)C1 C(=O)(C(F)CC(C)(C)NC(c1cc(Cl)c[nH]1)=O)N1CC(C)(C(C)C)OCC1 C(c1ccccc1)=CC(=O)N.CC1=NOC(CC(=O)NCC2CC2C)C1 CC(C)C(CC(=O)N1CC(N(C(=O)CCF)C)C(O)C1)c1ccccc1 C(=O)(C(O)C1=CCCCC1)NCC(C)NC(c1c(Br)ccc(C)n1)=O c1(C(=O)NC2CN(C(C(C)CN)=O)C2)ccc2[nH]nc(Br)c2c1 N1(C(Cc2nc(C)[nH]n2)=O)CC2(NC(=O)CCNC(=O)CC(C)C)CCC1C2 C(=O)(CC(C(F)(F)F)NC(=O)C(O)CN(C)C)NCCc1c(C)n[nH]c1 C1(CNC(CCN(CC=C)C(C2CC(C)C2)=O)=O)CCCCCCC1 N1(C(CCC=CCC=C)=O)CC2CN(C(C3CSC3)=O)CCC12 N1(C(C(CC=C)C)=O)CCC2CN(C(c3ccc(-c4cscn4)cc3)=O)CCC12 C1(CNC(c2ncc(CC)s2)=O)C(C)CCN1C(c1ccn(C)c1C)=O C=CCC(C)(C)NC(=O)C(CSC(C)(C)C)NC(=O)CC(O)C1CCCC1 CC#Cc1ccc(OC(F)(F)F)cc1.Cn1[nH]nnc1=NCCNC(=O)C(N)=O C(c1cccc(F)c1)=CC(N1CC(NC(=O)C(F)CC2CC2)C1)=O CC1CC(C)(C(=O)NCC(C)(C)CNC(=O)C(=Cc2cccnc2)F)CCO1 CC(C)(CC(F)F)C(=O)NCC1CN(C(c2cc(F)c(N)cc2F)=O)C1 c1(C=O)n[nH]c2c1CC(F)(F)CC2.c1(C(=O)NCC2CCC2)c[nH]c(=O)cn1 CC1CC2(CCN(C(c3ccncc3Cl)=O)CC2)CN1C(=O)CN1CCCC1=O c1(CC)ccccc1Cn1cc(C(CC)N(C(=O)C(F)F)CCO)nn1 CC#CCCC(=O)N1CC(NC(=O)CC(O)CN(C)C)C(c2cnn(C)c2)C1 c1(C(N2C3CC(NC(c4c(OC)n[nH]c4)=O)C(C3)C2)=O)scc2c1OCCO2 N1(C(C(CSC)O)=O)CCC(C(N2CCC(C)(C)CC2)=O)CC1C C=CCC(CNC(C1(C(N)=O)CC1)=O)C(=O)NCc1cc(O)cc(F)c1 Cc1nc(O)ccc1C(=O)NC1CCCC(N(C(=O)CCC(C)(C)C)C)C1 c1(-c2nc(CC(C)(C)O)on2)cnc(C=O)cn1.c1ccccc1C(=O)N(C)C.N C(=O)(CC(F)(F)C(F)F)NC(C)(C)CNC(C1CCNC(=O)C1)=O c1(C(=O)NC2C3(CCC(NC(C(N)=O)=O)CC3)C2)ccc2cccnc2c1O CCC(CC(=O)NCC(CC(=O)NCCC(COC)OC)OC)C1CCC1 C12(CNC(C(C)(C)F)=O)CCC(CC1)N2C(=O)COc1ccc(F)cn1 C1(CNC(=O)CCCC2CCOCC2)CCN(C(=O)C(O)CC2CC2)CC1 N(C1CN(C(c2cc(Cl)c[nH]2)=O)CCc2ccccc21)C(C(CO)N(C)C)=O c1(OCC)cc(CN=c2ccc(CO)c(F)[nH]2)ccc1[N+](=O)[O-] CN1CCC(CCC(N2CCCC2CN(C(C2CC=CC2)=O)C2CC2)=O)C1 C1(C2CCC2)(C(=O)OC)CCN(c2ncnc3c2ccn3C2CC2)C1 N1(C(C(C)=C2CC2)=O)CC(C(N)=O)(C)C1.c1(C=O)cc(C2CC2)[nH]n1.N C1(=O)C(CCSC)N2CCC(C2)N1.c1(C(=O)OC)cc(C(=O)C(C)C)c[nH]1 c1(C(N2CCC(CC(=O)NCC3(O)CC(C)(C)C3)C2)=O)cc(F)cnc1O c1(CC)ccc(C(=O)NC2CN(C(=O)C=CC(C)C)C(C)(C)C2)c(F)c1 C=CC(C)C(C)C(=O)N(CCCNC(=O)CP(C)(C)=O)Cc1cccnc1 c1(C(N(C2CCN(C(C3C(CF)C3(C)C)=O)CC2)CCC)=O)cncc(O)c1 c1(OC)ccc(C(=O)NC(C)C(=O)N)cc1.C1CCCN1C(C1CC=CC1)=O Cc1ncc(NC(C2CC(O)CN2C(=O)Nc2ccccn2)=O)nc1Br c1(-c2nc(C(C=C)(C)N(C)C)on2)ccc(C)c(Br)c1 N1(C(C2CC(N(C(c3c(C)csn3)=O)C)C2)=O)CCN(C)C(C)C1 C1(C(F)(F)F)(NC(=O)Nc2ccnn2CCF)CCSCC1 C=C(C)CCC(=O)NCC1(CNC(C2(CF)CC2(F)F)=O)CC12CCC2 n1(CC(=O)N)c(C)cc(O)cc1=O.Cc1ncc(C(N2CC(CO)C2)=O)c(C)n1 C1(C#CC(=O)NC2CN(C(c3cc(C)c(-c4ccccc4)s3)=O)C2)(CC)COC1 c1(C=O)cc(C)nc(C)c1O.C1CS(=O)(=O)CC1.c1(CC)ncoc1C(=O)N Cc1[nH]c(C(=O)N)c(C)c1S(N)(=O)=O.C1CC(C)N(C(c2cccnn2)=O)C1.C N1(C(Cc2cn(CC)nc2)=O)CC(=O)NC2CN(C(=O)CC(O)C(C)C)CCC12 C1(NC(c2cc(CC)[nH]n2)=O)C2CCN(C(c3c[nH]nc3C3CC3)=O)C12 CC1(C)OC(=O)CC1C(=O)NC1CCC(O)C1.C1(C(=O)N)CC2(CSC2)C1 Cc1nc2cncc(C(N3CCN(C(=O)CC4CC5CCC4O5)C(C)C3)=O)c2[nH]1 c1(OC)c(C(=O)NCCC2CN(C(=O)CC(C)C3CCCCC3)C2)csc1C C(C(CO)N=c1[nH]c2ccc(O)cc2s1)NC(C1(C)CC(C)OC(C)C1)=O c1(OC)cc(C(=O)N)cc([N+](=O)[O-])c1.C1(C=O)CC(C2CC2)=NO1.CC(C)C CC1(CNC(=O)CC2CCC(F)(F)CC2)CCC(NC(=O)CNC=O)CC1 C1(OCC(=O)NCCC2CCCN2C(c2csc(COO)c2)=O)CCCOC1 Cc1cc(F)c(N)cc1C(=O)NCCN(C(=O)C)C(C)C.C1CCCC1.O N#CC1(C(=O)NC2CC2)CCS(=O)(=O)CC1.C1(CC=O)CN2CCC1CC2.N c1(C(=O)NC(C2CCCN(C(c3coc(Cl)c3)=O)C2)C)cnc(O)c(F)c1 CC1CC(F)(F)CN1C(C1CC(F)(F)CN1C(=O)CCc1nccs1)=O c1(C(=O)NCC2(F)CN(C(C3CC(O)C(F)C3)=O)C2)coc2ccccc12 CC(c1ccccc1C)=CC(=O)NC1CC2CCC1CC2NC(c1cn[nH]c1)=O C(c1ccccc1OC)=CC(N1CC(C(C)NC(C2C(CCC)C2)=O)C1)=O c1(C(N2C(CNC(c3c(C)n[nH]c3)=O)CCC2)=O)cc2c(Cl)cccn2n1 C(CC(CO)NC(C1CCC(CNC(C2CCC2)=O)C1)=O)OC.C1CC1.C c1(C=O)cc(S(N)(=O)=O)c[nH]1.c1(OC)cc(CC(N2CCC2C)=O)ccn1.N C#CCC(C)(C(=O)NCCC(C)CO)NC(=O)COC C(=O)(C(O)CC(C)C)N1CC(CCCCN(C(C(F)=CCC)=O)CCO)C1 C(=O)(C1COc2ccc(Cl)cc21)N1CC2C(NC(C3CCC(O)CC3)=O)C(C2)C1 N1(C(Cc2c(C)nc(SC(F)F)s2)=O)CCCC(O)(CCNC(=O)C(C)C)C1 c1(C(N2CCC(C)(CNC(c3c(C)ccn3C)=O)CC2)=O)ncc2n1CCCC2 c1(C(N(C2CN(C(C(COC)C)=O)CC23CC3)C)=O)cc2c(C)cc(Cl)cc2[nH]1 c1(NC(C2CN(C(=O)NC3CC4CCC3C4)CCO2)=O)ccnc2ncnn12 N1(C(CCOCC(C)C)=O)CC2CC(NC(=O)COc3ccccc3Cl)CC1C2 Cc1ccc2c(c1)C(=O)NCCN2C(C12CC(C)(C1)OC21CCOCC1)=O c1(C(=O)NCC#CCOC)cc(CNC(=O)Cc2ncccc2C)ccn1 c1(C(=O)NC(C)CCNC(c2cnns2)=O)ccc(-n2cncn2)c(N)c1 C1(C(=O)NC2CCN(C(c3ccc(CC(C)C)s3)=O)CC2)CCOC(C)(C)C1 c1(C(N(CC)C2CC2)=O)ccc2c(O)nccc2n1.CC(C=O)OC.C1CC1 C1(C(C)C)CN(C(c2cc(Cl)no2)=O)CCC1NC(C1(C)CC=CC1)=O C1(C(N(C)CC2N(C(C3C(C)C(=O)C3)=O)CCC2)=O)CCC2(C)CC12 c1(C(=O)NC2CN(C(CC(C=C)(C)C)=O)CC3C2C3)ccc(S(C)(=O)=NC)cc1 c1(CSCC(=O)NCCCCCN(C(CCC=C)=O)C)cccc(C)c1 c1(CN(C(COCCCCC)=O)C)cccc(C)c1.n1(CC(=O)N)ccnc1C C(=O)(C1=NOC2COCC12)N1C(CC)C(NC(=O)CNC(C)=O)CCC1 Cc1c(C(=O)NC(C2CCN(C(=O)C(C)O)CC2)C)cccc1C#N N1(C(C=C(C)C)=O)C2CC1CN(C(=O)Cc1ccc(C)cc1)C2 C1(NC(C2C(C)CC(C)O2)=O)(CO)CCCN(C(c2cncc(Cl)n2)=O)C1 c1(C(=O)NC(C(C)NC(c2cc(=NC)[nH]cc2)=O)C)cc2n(c1)CCCC2 c1(CN(C2CCCCC2)CCO)ccsc1Br C1(C(F)(F)F)(OC)CC(C)C1.C1(C)(C=O)C=CCC1.C1(C=O)COC1.N CC1C(NC(=O)C(C)(C)CNC(=O)CN2C(=O)CNC2=O)CCCN1C C12(CC)CN(C(c3ccnc(C)c3O)=O)C(C)(C1)C2.C1(C=O)CC2C=CC1C2 Cc1ccc2c(c1)CC(C(=O)NOCC1C3C4CCC(CC4C1)C3)N2C1CCC1 c1(C(N(CCC(=O)NC(C#C)C(C)OC)CCCO)=O)cnn(C)c(=O)c1 [N-]=[N+]=NC1CN(C(c2c[nH]nc2[N+](=O)[O-])=O)CC1NC(=O)Cn1cccn1 N1(C(C2N(C(c3ccc(I)cc3F)=O)CCSC2)=O)CCN2CCOCC2C1 c1(NC(C)C)nnccc1C(=O)NCC(O)CNC(c1ccnn1C)=O N1(C(C2C(CCC)C2)=O)CCCC1C(=O)NC(C1CCCCC1)C.C(=O)CO c1(C(C(N2CC(CN(C(CC3CC(=C)C3)=O)C)OCC2)=O)C)cc(F)cc(F)c1 C1(CNC(C2CC3C=CC2CC3)=O)CN(C(c2cnccn2)=O)CC2(CCC2)O1 c1(OC)cccc(C(N2CCN(C(C3(OC(C)C)CCC3)=O)CC2C)=O)c1OC C1(NC(C2N(C)CCCC2)=O)(CNC(=O)CC2CCOC2)Cc2ccccc2C1 C#Cc1ccccc1CC(=O)NC1CCN(C(c2ccc(F)c(Cl)c2)=O)CC1 C1(CNC(C(C(=O)OCC)F)=O)CC2(C1)CN(C(=O)CCCCCF)C2 C(=O)(C(F)C(F)(F)F)N(CC(=O)NCCc1ccco1)CCOC C(=O)(C(CCC(N)=O)n1cc(C2CCC2)nn1)Nc1ccc(CC)c(F)c1 C1(CNC(Cc2ccc(C(C)=O)cc2)=O)CC2CCC(C1)N2C(c1cncs1)=O CC1CN(C(C2CSCC(=O)N2)=O)CC(C)N(C(=O)CCOCCN(C)C)C1 C1(NC(C2(CC=C)CC2)=O)CN(C(C23CCC(C)(CC2)OC3)=O)CC1C1CC1 O=NN1CCCCC1C(=O)NC1COCCC1NC(=O)Cc1cn[nH]c1 c1(C(N(C2CC(C(=O)NC(c3nnc(C)o3)C)C2)C)=O)ccccc1O Cc1cc(C=CC(=O)NC(C)(C)C(N2CCC(O)(C(F)F)C2)=O)on1 CN1CCC(NC(C2CCC(CNC(c3cc(O)cs3)=O)CC2)=O)C(C)(C)C1 c1(C(N2CC(C3CC3)C2C2CC2)C(=O)NCC)cc2cc(Br)ccc2o1 N1(C(C)=O)CS(=O)(=O)CC1C(=O)N.C1CCCCC1.C(=O)C(C)(C)N(C)C N1(C(c2ccc(C(N)=O)[nH]2)=O)CCCC2(CNC(c3cc(Cl)c[nH]3)=O)CCCC12 C1(n2cc(C(C(C)(C)C)O)nn2)CC2CCC1(NC(c1cc(Br)c[nH]1)=O)C2 N1(C(C2CCCN(C(C)=O)C2)=O)CCC(NC(=O)CCOCC(F)F)CC1C Cc1cnc(Cl)c(NC(C2CN(C(c3cc(C4CC4)on3)=O)CCC2O)=O)c1 CC(C)C1=NOC(C(=O)NCC(CO)NC(c2cc(C3CCC3)on2)=O)C1 c1(-c2cn(C3CN(C(=O)C4=CCCCC4)CC3O)nn2)cccc([N+](=O)[O-])c1 N=c1cc(C(=O)NCC2CC(NC(=O)C(F)C(F)(F)F)C2)c(Br)c[nH]1 c1(C(N(C(CC(c2ccc(C(C)C)cc2)C)=O)C2CC2)C)cccc([N+](=O)[O-])c1 c1(COC)n[nH]c(=NCC2CN(C(C3CC4(CC(=O)N4)C3)=O)CC2C)s1 c1(C=O)cc(C)nc2ncnn12.CC(C)C1CC1.C1(C=O)(OC(C)=O)CC1.N C#CCC(O)C(=O)NC(C1CC(NC(c2cscc2CC)=O)C1)C C(=O)(C1CCCc2nncn21)NC1CCN(C(C2=C(C)OCCS2)=O)CC1(C)C c1(C(N(CCN2CCCC2)CC)=O)cccn1CC(=O)OC(C)(C)C N1(C(c2nc(COC)oc2)=O)CCC(C(=O)NCC2CCCCC2)C(O)C1 C1(CNC(C(CC(C)C)O)=O)CCC2(CN(C(=O)CN3CCCS3(=O)=O)C2)O1 c1(C(=O)NC(C2(O)CN(C(C(C)OC)=O)C2)C)ccc(F)c(F)c1F c1(C(N2CCC(NC(C(N3CCNC3=O)C)=O)C2(C)C)=O)cc2cccnn2n1 N1(C(c2c(C(C)C)ncs2)=O)CCCC2(C1)CN(C(C1(O)CC1(C)C)=O)CCO2 c1(C(N2CC(CNC(C(C(CC)C)O)=O)OCC2)=O)ncc2ccccc2c1N N1(C(c2cscc2Cl)C(=O)NC(CC)(C)C)CCC2(CSC2)C1 N(C1CCCc2n[nH]cc21)C(CC1C2CN(C(C3CC4CCC4C3)=O)CC21)=O N1(CC(=O)N)C(=O)C(=O)N(C)C1=O.c1(C(=O)NC(C)CC)cncc(F)c1 c1(C(N2CCC(C)(NC(=O)CC3CCCO3)CC2)=O)cc2c(nc1O)CCOC2 N1(C(c2cc(C)on2)=O)CCC(C)C(NC(=O)CN2CCS(=O)(=O)CC2)C1 c1(C(=O)NC(C2CCCN(C(c3c[nH]c(Br)c3)=O)C2)C)c(F)ccc(O)c1F c1(C(=O)NCC2N(C(=O)C=C3CCC3)CCC(C)C2)cc2c(ccn2C)[nH]1 CCCCCS(=O)(=O)CC(=O)N1CCC1CNC(C1SCCCS1)=O c1(NC)cnc(C=O)cn1.C1(C)CCN(C(C2CC(=O)N(C(C)(C)C)C2)=O)C1 Cc1ccc(C)c(CC(=O)NCC(O)CC(=O)NC(c2ccsc2)C)c1 Cc1c(Cl)ccc(S(=O)(=O)N2CC3COCC3(C(=O)N3CC(C)CO3)C2)c1Cl C#CCC(C(=O)N1CCN(C2CCC2)CC1)NC(C1CC12CCC2)=O CC1CCCC=C1C(=O)NC1(C2CCCN2C(=O)Cc2ccc(F)cn2)CC1 c1(-c2cn(C3CCN(C(C4C(C(=O)OC)C4(C)C)=O)C3)nn2)cccc(F)c1 C(=O)(C#CC1CCCC1)N1C2(C(=O)NCCC3OCC(C)(C)C3)CC(C)(C1)C2 C(=O)(C1=C(C)CCOC1)NC1C(CCC)CN(C(c2cc(C)c(C)cn2)=O)C1 C(c1ccc(F)cc1)=CCC=O.C1(C(C(=O)NCC2CC2)OC)CCCOC1 Cc1c(C(=O)N(CC(C)(C)NC(C2CCC3(C2)CC3(F)F)=O)C)sc2ccsc12 C(=O)(CC(C)CC(=O)NC)OC.C1C2CN(C(=O)C)CC12.C(=O)CCC(C)C C=CCC(C(=O)NCC(=O)NC(C)(C)C)NC(C1C2CC(=O)CC12)=O C1(C(N(C2CC(=C)C2)C)=O)(CF)CCN(C(=O)CCOC)C1 CCC(C)C(C)C.C12COC(C=O)(C1)C2.C(=O)CN(C1CCC1)C.COC CCCC(CC)CC(=O)N1CCN(C(=O)C2=COCCC2)CC(CO)C1 CCCCC(O)C(=O)N1CC2(CCN2C(C2CCC2(F)F)=O)C1 CCC(CC)C(F)C(=O)NC(C)CCNC(C1CCC2CC12)=O C1(F)(CNC(CC=CC)=O)CCC(CNC(=O)Cc2ccccc2Br)C1 CN(C)S(=O)(=O)N1CCC(C(=O)NCC(C)C(F)(F)F)CC1.C(=O)C(F)F.N C1(C(=O)Nc2ccnc(N3CCCC3)n2)CCCCC12CC2(F)F C(c1cc[nH]n1)=CC(=O)NC(C1CCN(C(=O)C=C(Cl)Cl)C1)C Cc1cccc(N2CCN(C(C)C(=O)NCCCC3CCC3)CC2)c1 C(C(=O)N=c1cc(C)o[nH]1)N(C(C12C(C(=O)OCC)OC(C)(C1)C2)=O)C C1(CC(=O)NCCCC2CCCCO2)C=CC(NC(=O)Cc2cccs2)C1 Cc1c(C(=O)NC2CCCC2NC(=O)CCCn2ccccc2=O)ccn1C C(=O)(C1Cc2c(Cl)cccc21)NCC(C)(C)CNC(=O)CSS(C)(=O)=O C(=O)(C(C)(C)C=O)NC1CCCC(NC(c2ccc(OCC)cc2)=O)C1.N c1(OC)ccc(NC(C2CCCN2C(=O)C(N2CCC(C(=O)O)C2)=O)=O)cc1 c1(C(=O)NCCN(C(=O)CO)CC)cc(C(F)F)cs1.c1nccn1C C1(NC(=O)COC2CC2)CN(C(C2CCCCC2O)=O)CC2CCCC12 CC(C)CCCNC(=O)COC1CCCCCC1.c1(C=O)cnc(C(C)O)s1.N N1(Cc2ccc(CC)s2)CCC2(CCN(S(=O)(=O)c3cnc(Cl)nc3)C2)C1 c1(C(=O)NC2C3CN(C(C4=CC(C)(CC)C4)=O)C2C3)ccc2cc[nH]c2c1F C12(C(=O)NCC3N(C(C(C4CC4)OC)=O)CCOC3)CCCC(C1)OC2 N1(C(CC(C)C2CC2)=O)CC2(CC(NC(=O)C(C)Cc3ccc(Cl)cc3)CO2)C1 N1(C(CSc2n[nH]c(=N)s2)=O)CCN(C(=O)CCC2CCCOC2)CC12CC2 C1(C(=O)NC(c2nnc(C)s2)C)CCN(C(c2c[nH]cc2C)=O)CC1O C(C(C=O)N(C)C)OC.[SH](=O)(=O)C1CC1.C(=O)(C)N(CC)C1CC1.N c1(C(CNC(=O)CC2CCSC2)NC(C2CC3C=CC2C3)=O)ccc(F)cc1F c1(C(=O)NCC2(NC(c3c(C)nco3)=O)CCOC2)cccnc1C1CC1 C(=O)(CCCCC)N1CC(CCC=C)(C(=O)NC(C2CCCCC2)CO)C1 CCC(F)(F)CC(=O)N(C1CCN(C(C2CCCN(CC(F)F)C2)=O)C1)CCO Cc1[nH]c2ccnn2c(=O)c1CC(=O)N.N1(CC=O)CC(C)(C)C1.C1CC1.C N1(C(Cc2nnc(C)o2)=O)CC(C(=O)O)C2(C1)CN(C(=O)CCc1cn[nH]c1)C2 c1(OC)ccc(C)nc1C(=O)NCC1CCCN(C(=O)C(CO)OC)C1 c1(CC(=O)N(CCNC(C2CC(n3cnnc3)C2)=O)CC)cnccc1Cl N1(C(CC(C)(F)F)=O)CC2(CC(C(=O)NC3CCOCC3(C)C)CO2)C1 N1(C(c2ccc(CC)[nH]2)=O)CCC(CNC(C2CCCC23CC3)=O)CC1 C(=O)(C1=CC2C=CC(C1)C2)N1CCCC(N(C(CCCC(C)(C)C)=O)CCF)C1 c1(CNC(Cc2ccn(C)n2)=O)ccc(C(=O)NC2CC2c2cc[nH]n2)cc1 C#Cc1ccc(F)cc1C(=O)NCC1CC(C)N(C(c2ccnn2CCF)=O)C1 C1CCC(O)C1.C(C)(C(=O)N)OC.C(=O)C(F)=CC.C(C)(C)C.C=O n1(CC)nnc(C(N2CCCC2C(C)(C)C(=O)NC2CC(C)C2)=O)c1C C1(CNC(C2(OCC)CCOC2)=O)CCCCN(C(C2CC(=O)C2C)=O)C1 C1(C(N2CCC(OCC(=O)NCc3ccc(F)cc3)C2)=O)CC2(CCC2O)C1 N1(C(c2c(C)sc(Cl)n2)=O)CC(C)CN(C(c2ccc3oncc3c2)=O)CC1C c1(-n2c(CF)nc(C3CCCC3)n2)ccc2nccnc2c1 N1(C(C2(NC(C3CC(OC)C3)=O)CC(F)(F)C2)=O)CCCNC(=O)CC1 C(=O)(C(C(C)(C)C)N(C)C)N1CC(C(C)NC(CC2ON=C(CC)C2)=O)C1 N1(C(c2n(C)ncc2C#N)=O)CCC2CCC(C1)N2C(c1ccncc1Br)=O C(=O)(C(CNC(C1CC1(C)C)=O)C(C)(C)C)NC(c1cncs1)C C(CCCCCC(=O)N1CCN(Cc2sccc2C)CC1)SC C(=O)(C(CN=[N+]=[N-])NC(C1CCCC1C1CC1)=O)Nc1c(C)n(C(C)C)nc1 N1(C(CCN(C(C(C(C(C)C)OC)O)=O)CCCO)=O)CCCC2(CCC2)C1C c1(C(N2CCCC(CNC(COCCC#C)=O)C2)=O)ccc2[nH]c(=N)oc2c1 O=S(=O)(c1ccccc1N(CC(F)F)CC1CCCC1)N1CCCC1 CCCCCC(C)(C)C(=O)NCC1(CNC(=O)C(CCSC)OC)CCC1 c1(C(=O)NCC2(C)CCN(C(c3csc(Cl)n3)=O)C2)cnc2nccn2c1 c1(C(=O)NCC(CO)NC(Cc2c(C)ccnc2)=O)ccc(Cl)c(N)c1 c1(C(=O)NCC(CN(C(c2cnn(CC)n2)=O)C)O)nc2cncnc2[nH]c1=O N1(C(c2c(C)ccnn2)=O)CCC(C)(C)C1C(=O)NCc1cc(O)ncn1 N1(Cc2cccc(OC)c2)CCC=C(c2ncccc2C(=O)Nc2cc[nH]n2)C1 C(=O)(C(O)CCC(C)C)NCC=CC(N1CCC(NC(=O)OC)C1)=O C1(C)(CC)CC(NCc2cn(-c3cc(F)cc(Br)c3)nn2)CCO1 c1(C(C(=O)NC2CC(NC(COC)=O)C2)NC(C)=O)ccccc1 CCCCC(CNC(c1nsc(OCC)n1)=O)NC(c1cnc(C)cn1)=O N1(C(C(C)Oc2cccnc2)=O)CCCC1(C)CNC(=O)C(C)(C)CO c1(OC)cccc(C(N2CCCC2CCNC(c2ccc(Cl)s2)=O)=O)c1 c1(CC(N2C(CCNC(C3C(C)CC3)=O)CCC2)=O)c[nH]c2ccc(Br)cc12 N1(C(CC(CC)C)=O)CCC2(CCC2)C(CNC(c2cncc(C)c2C)=O)C1 c1(C(N2CC(O)C2)=O)c(F)ccc(Br)c1F.C1(S(=O)(=O)N)(CC=C)CC1.C N1(C(C(CC2CCC2)NC(C(C)OCC)=O)=O)CCCC2CN(C)CC12 C1(c2nc(CSCCOC)n(CC(C)CO)n2)CCOC2(CCOCC2)C1 c1(C(=O)NCCNC(c2cc(C)sn2)=O)c(O)nnc2c1CCCC2.C1CC1.C Cc1[nH]c2cccc(Cl)c2c1C(C)NC(C1CCN(c2ccc(CN)cc2)CC1)=O C1(NC(Cn2ccc(C)n2)=O)CCC(O)CN(C(c2cc(Cl)c(Cl)[nH]2)=O)C1 c1(-c2n(CC3C(C)C3)nc(-c3ccccn3)n2)ccc2c[nH]nc2n1 CCC(CC(=O)N(C1CCN(C(c2ccc(N3CCCCC3)cc2)=O)C1)C)OC C(=O)(C#CC1CCCO1)N(CCN(C(=O)Cc1ccccc1Cl)CC)CC C1(CN(CCCO)Cc2ccc(OC)cc2)C2CCCC1NC2 C1(NC(COCC)=O)CN(C(c2ncc(OCC)cc2Cl)=O)CCC1(C)C CN1CCC(NC(C2(NC(c3ccc(C(N)=O)o3)=O)CC2)=O)C1 c1(OC)ccc(C(=O)NCC(C)(CC(C)C)NC(c2ocnc2C)=O)c(F)n1 n1(CC(=O)NCCC(C)NC(=O)C(Cl)=CCl)cc(S(N)(=O)=O)cn1 CC(F)(F)F.O=C(O)COCC(=O)N(CCCO)CC C(N(O)C(=O)C(C)C1CCC1)c1cn(-c2c(C(C)C)cccc2)nn1 CCCS(=O)(=O)C(C)C(=O)NC1CC2CC1N(C(=O)CSCCN(C)C)C2 CC(C(=O)NCC1CCCN1C(=O)CN1CCS(=O)CC1)C(C)C(C)(C)C N1(C(CCCC=C)=O)CCC2(CCCN2C(C2CC(=O)NC(=O)N2)=O)C1 C(=O)C(C)C(O)C(C)C.n1(CC)ccnc1C(=O)NCc1cn(CCC)nn1 C(=O)(C(F)C(F)(F)F)NCC1CCN(C(C2CC2(Cl)Cl)=O)CC1 C=Cc1ccc(C(=O)N(C(C)CN(C(=O)CC2CC(OCC)C2)C)C)cc1 C1(C(=O)NC2(C(=O)NC(c3c(C)nn(C)c3)C)CC2)CC2(CCO1)CC2 N1(C(C(C)c2ccco2)=O)CC2(CC(CC(=O)NC(C)(CO)C(F)F)C2)C1 C=CCCC(C)(C)C(=O)NCCC1CCC(NC(=O)CC(F)(F)CC)C1 c1(C(N(CC(CC)NC(C2CNC(=O)N2)=O)C)=O)ccc2ncn(C3CC3)c2c1 C(c1cccc(F)c1Cl)=CC(N1CCC1)=O.C1(C(=O)N)(OC)CCC(C)(C)C1 C(=O)(C(CC(C)C)N(C1(C(=O)OC)CC1)C)NC(C)CO N1(C(C(N2CC(C)C2)C)=O)CCCC(C2CN(C(=O)C#CC(C)(C)C)C2)C1 Brc1ccoc1CNC(c1nnnn1CC1CCOCC1)C1CC=CC1 C(=O)(C1CCSc2ccccc21)N1CC(N(C)C(c2cc(=O)cc[nH]2)=O)C(O)C1 C#Cc1cccc(C(c2nnnn2CC2CCOC2)NCC2=COCCO2)n1 c1(CC)ccncc1NC(c1csc(CNC(C2CCC(C)C2)=O)c1)=O CC1CN(C(=O)CCc2ccccn2)CC(C)C1.C1(C(=O)N)CN(S(N)(=O)=O)C1 c1(C(=O)NC23CCN(C(c4csc(C5CC5)n4)=O)CC2C3)ccc2cncn2c1 c1(C(N2CCC(C)C(NC(C3CC3(Cl)Cl)=O)C2)=O)cc(F)cc2nc[nH]c12 c1(C(=O)NC2CC(CNC(=O)Cn3ccnn3)C(O)C2)ccc(Cl)c2occc12 N1(C(Cc2c(C)nc[nH]2)=O)CC(NC(=O)CCC(=O)N(C)C(C)C)CC1(C)C c1(C(=O)NC2C(C)CN(C(c3cc(F)ccc3Cl)=O)CC2)ccc2n[nH]cc2n1 C(=O)(CC1=CCN(C(C23CCCC(CO2)C3)=O)CC1)N(C)Cc1cnc[nH]1 N1(C(CSCC)=O)CCC2(CC2)C1.c1(C(=O)N)cnn(-c2ccc(O)nn2)c1C C=CCC(CC(=O)N=c1ccn(CCC)[nH]1)NC(=O)CC(=O)N(C)C N1(C(C(C)N(C(c2cnc(=N)[nH]c2)=O)CC)=O)CC2CCC(C1)O2 c1(C(N2C(CN(C(CC=C)=O)C)CCC2)=O)c(F)ccc2occc12 N1(C(C)C)CCN(CCCNC(=S)NC2CCCC2)CC1 CC(C)CC(O)C(C)C(=O)N1CC(CC(F)C(N2CCc3n[nH]cc3C2)=O)C1 N1(C(CCC2N(C(CCC(C)N(C)C)=O)CCCC2)=O)CCC2(CNC(=O)O2)C1 C1(NC(c2c(CC)n(C)nc2)=O)CCCC12CCN(C(=O)Cc1csc(C)n1)C2 CCC(C(=O)NCC(C)CNC(c1cccc(Br)c1O)=O)C(C)C N1(C(CCCCSC)=O)CC2(CNC(=O)CCC(C)(C)C)CCC1CC2 Fc1c(C(c2nnnn2CC2CC2)NCC2(n3nccn3)CC2)cccc1I C1(C(=O)NC23CCC(CN(C(=O)C(F)F)C2)C3)COc2c(F)cc(F)cc2C1 C(=O)(C(N)CCC(C)(C)F)N1CCCN(Cc2onc(C(C)OC)n2)CC1 c1(C(=O)NC2(CF)CN(C(CC3(C)CCC3)=O)C2)ccc(C2CC2)nn1 c1(OC)ccc(Br)c(C)c1C(N1CSCC1C(=O)NCC(C)C)=O N1(C(CCCc2onc(CC)n2)=O)CCCC(C)(C)C1.C1(CC(=O)N)CC(F)C1 C#CCC(CC(F)F)C(=O)N(CC(O)CNC(=O)CC(=O)NC1CC1)C N1(C(c2cc(CC)on2)=O)CC2CN(C(=O)C(C)C3CCCC3)CC(C1)O2 c1(C(=O)NCC(c2n(C)ncc2)O)ccc(CNC(C2CCC2)=O)cc1.C N1(C(CC(=O)NCC#C)=O)CC(NC(=O)C(C)NC(C)=O)C(C)(C)C1 C1(N(C(C2C3CN(C)CC32)=O)C)CC2CCC(C1)N2C(C1CC2CCC(C1)S2)=O N1(CC)CCC(CN(C(c2nocc2COC)C(=O)NC(C)(C)C)C)CC1 C1(N(C(=O)CC2CC(N(C)C)C2)CC#C)CCN(C=O)CC1.c1ccsc1.N C(=O)(N1CCCCCO1)C1N(C(c2ccc(C)cc2O)=O)C(C(C)C)CC1 c1(C(=O)NCCC(C)N(C(=O)Cc2n[nH]c(=N)s2)C)cc(C2CC2)nn1C c1(C(N2CCC(NC(c3c(C)ocn3)=O)C2)=O)cncc(N(C)C)n1 c1(C(=O)NC2C(NC(c3c(C)ocn3)=O)COC2)cc2ccccc2o1 c1(C(=O)NCC(CC(=O)NC2CCCC2(F)F)O)ccc([N+](=O)[O-])o1 C1(C(N(C2(C)CCCC2)C)=O)C2CCC(C2)C1.C1(CC=O)CCC(=O)N1C.N C1(CC(C)NC(CSCCC)=O)CCN(C(=O)C(n2ccc(C)n2)C)CC1 O=C(C1=CCCCC1)NC1CCCC1CNC(c1cc(F)cc(F)c1)=O N1(C(CCc2[nH]cc(C)n2)=O)CCCn2c1nc(C)cc2=O CC1CC(CNC(=O)CCC2CCC(NCCc3nnc(Br)n3C)C2)=NO1 Cc1cc(Br)cc(Cl)c1C(N1CCN(C(C2CC2C)=O)CC1CCO)=O CC(C)CCC(=O)NC1CC2(C1)CC2NC(c1ccc(C(O)CF)cc1)=O c1(C(=O)NC2C(NC(C(C)OCC)=O)CC2)ccc(OC)c(Cl)n1 CCC(CCC(=O)N1CCC(O)C1C(C)(C)C)NC(=O)Cc1c(C)noc1C c1(NC(=O)NCC(CC)(CC)c2ccccc2)nc2c(cc1C#N)CCC2(C)C Cc1cc(C=CC(N2CCN(CC(=O)N(C(CO)CO)C)CC2)=O)on1 C(CC(C)(C)C(=O)NCCOC1CCN(C(=O)CC(F)(F)F)C1)OC N1(C(CC2N(C)CCCC2)=O)C2CCC(C2)C1CNC(=O)Cc1ccsc1 C(CCN=c1[nH]c(=N)[nH]c(=NCC(CCO)c2cncn2C)[nH]1)SCC CC(=O)C(C)(C)CC(=O)N(CCCNC(=O)CS(=O)(=O)CCO)C c1(OC)ccc(F)nc1NC(C12CC1CN(C(c1ccc(C)nc1)=O)C2)=O c1(NC(C2N(C(c3c(OC)ccnc3F)=O)CC2)=O)ccc2nccnc2c1Br c1(C(C)C)ccc(C)cc1NNC(=O)c1noc(-c2ccccc2C(F)(F)F)n1 CC1CC(CNC(=O)CC2CCCCC2)CN1C(=O)CCc1ccc(O)nc1 N1(CC(C)O)CCN(C2(C(=O)O)CCCC2)CC1.C1(CNC=O)CCCCO1.N C(=O)(C#CC1CCOC1)N1C(CNC(C(C=C)CC)=O)CC(C)CC1 CCCCCC(O)CC(=O)NC1CCN(C(c2ccc(=NCC)[nH]c2)=O)CC1O Cc1ccn2nc(C(=O)Nc3c(Cl)c(F)nc(F)c3Cl)nc2n1 C1(C(=O)NC(CN(C(c2c(C)nn(CC)c2C)=O)C)C)CCCC2CCCN12 N1(C(C(C)OC2CCCCC2)=O)CC=C(C)CC1.C1(CC(=O)N)CC(C)(C)CO1 C1(OC)CC(C(=O)N(C2CCCCCC2)C)N(C(C2CCCN2C=O)=O)C1 C(=O)(CCCCCN=[N+]=[N-])N1CCC(F)(C(=O)Nc2c(CC)csc2)C1 c1(OC)c(C)cc(C(=O)NC)cc1C.C1C(C)CCN1C(c1cccc(N)c1)=O N1(C(c2cnc(C)s2)=O)CCCC2C(CCCN2C(c2csnn2)=O)C1 C1(O)(CNC(C(=O)NC(c2ccccc2)CC)=O)CCOC1C c1(C(N2CCCC(C(C(=O)NC)(F)F)C2)C(=O)N)cc2ccc(Br)cc2s1.C1CC1 c1(CCC(=O)NCC#CCNC(C2(CC#C)CCCO2)=O)nc2ccccc2[nH]1 c1(C(=O)NCCC(C)N(C)C)coc2c1CN(C(=O)CC13CCC(CC1)C3)C2 N1(C(C2CN(CCOC)C(=O)C2)=O)CCCC12CCN(C(c1cccnn1)=O)C2 C(CC(C)C(=O)NC1CCN(C(c2cccn2C2CC2)=O)C1)=CC N1(C(C2(OC)CCCSC2)=O)CC2CC(C1)CN(C(=O)C(C)N(C)C)C2 CCC(CC(=O)NC1(CNC(C2(SC)CC2)=O)CC1)C1CCC1 c1(C(=O)NCC2C(NC(C(CCCOC)C)=O)CC2)cnc(O)n(C)c1=O N1(C(C2(C#C)CCCC2)=O)CCCN(C(=O)C(c2cn(C)nc2C)C)C(C)C1 Cc1cnccc1C=CC(=O)NCC1CCN1C(=O)C(C)Sc1nncn1C CC(C)C(C(=O)NCC1C(C)CCCN1C(C1CCC=CCC1)=O)C(C)C c1(C=O)ncc(C(N)=O)cc1Cl.C1CN(C(=O)CC2CCC3CC23)C1.COC n1(CC(=O)NC2CC(NC(C34CC(CF)(CO3)C4)=O)C2)ncc2ncccc12 C1(CNC(=O)COC2COC2)CC2CCC1N2C(=O)C(F)(F)CO Cc1oc(CNS(C)(=O)=O)cc1C(=O)NCC(=O)NC.C1CCCO1 CC1CCCc2c(C(=O)NC3CCCCC3NC(=O)CC3CCOCC3)cnn21 N1(C(C2N(C(C(CC)N(C)C)=O)CC(OC)C2)=O)CC2C3CCC(C3)C2C1 c1(C(=O)NC2C(NC(c3cc(F)c[nH]3)=O)CCC2)c(Cl)sc2nnsc12 N1(C(CCCOCC)=O)CC(COC)CC1C.c1(C=O)cnn(C(C)C)c1C Cc1nc(O)nc(C)c1C(=O)NC1CC1CNC(=O)CCCN(C)N=O Cc1cc(CC(=O)NC2(C(=O)NCCN3CC(CF)C3)CC2)nn1C C1(CNC(CN(C(=O)Cc2cccnc2F)CC#C)=O)CCCC(C)C1 CC(C(=O)NC1CC(C)(NC(c2ccncc2)=O)C1)S(N)(=O)=O.C1CCC1 Cc1cccc(F)c1CC(=O)NC(C1CN(C(c2csnn2)=O)C1)C c1(C(C)=O)cc(C(=O)NCC2(CC(=O)NC(C)(C)CO)CC2)n[nH]1 C1(NC(C2(CC#C)CCCCO2)=O)CC(O)CN(C(=O)C(C)(C)CF)C1 C1(NC(CCNC(c2c(C)sc(O)n2)=O)=O)CCC12CCCC2 c1(NC(CN2CCOCC(C)(O)C2)=O)ccc(NN2C(=O)CCC2=O)cc1 C1(NC(C(C)OCC)=O)CC2CCC(C1)N2C(c1scc(C)c1C)=O c1(C(=O)NC(CCN(C(c2c(CC)scn2)=O)C)C)cnn(C2CCC2)c1C Cc1nc2c([nH]1)CN(C(C13CC(CN1C(C1(C)CCNC1=O)=O)C3)=O)CC2 N1(C(c2ccccc2)C)CCCCC(NC(=O)CN2CCN(C)C(=O)C2)C1 c1(CC(=O)N(CCC)CC)c[nH]c2c(C)cccc12.N1(CC(=O)N)CC=CC1 Cc1cc(CC(=O)NCC(C(C)(C)C)NC(=O)CCC=CBr)cc(F)c1 N1(C(C2COCC2)=O)CC=C(C(C)(C)C)CC1.n1(CC)cccc1C(=O)NC c1(C(=O)NCC2OCCN(C(C3CC(C)(C)C3)=O)C2)cc(Cl)ncc1F C1(C)(CC2CCN(CC(C)(C)CN3CC(N4CCCC4)C3)C2)CCS(=O)(=O)C1 Cc1c(NCc2c[nH]nc2C(F)F)ncnc1NC1CCOCC1C c1(CC(=O)C(=O)Nc2cnn(CCO)c2)cccc(O)c1 C(CCCC(=O)NCC1CCN1C(=O)C(c1ccc(F)cc1)=O)SC CCCCCCOC(C)C(N1CCC(NC(c2cc(COC)cs2)=O)C1)=O C=CC1(NC(=O)CSCCNC(=O)COCC(C)(C)C)CCCCC1 c1(C(=O)NCC(=C2CN(C(C(CC)(C)OC)=O)C2)F)cccc2c1OCCO2 c1(CC(=O)OC(c2ccnn2C)C)cccc(OC(F)F)n1 c1(C(N(CCCNC(C(C)OCCN(C)C)=O)C2CC2)=O)cnnn1C Cc1nc(C)n(O)c1C(=O)NCC1CC(F)CN1C(=O)C1=CCCCO1 CCCC(C)CC(=O)N1CC=CC(NC(=O)C(C)CSC)C1 c1(C(=O)NCCCn2cc(C3(OC)CCOC3)nn2)sc(Br)cc1C O=C1c2ccccc2C(=O)N1C(CO)CC(O)C1CCC1.[nH]1nnc2ccccc12 c1(C2(C(=O)NCC(C)N(C(C(CC)n3cncn3)=O)C)CCC2)ccccc1Cl C1(CC)CN(C(=O)Cc2ccc(OC)nc2)CCC1NC(c1cc(C)ns1)=O CCCC(C(=O)NCC1C(C(=O)NCCC)C1)N(C)C.[SH](=O)(=O)CCC N1(C(CN2C(C)CCC2)=O)CC(N=[N+]=[N-])CC1C(=O)NCCCS(C)=O C(C(=O)N1CC2CC1C2CNC(=O)C(C)O)(C(C)C)SCC.CC(C)C c1(NC(C2(CC#C)CCCOC2)=O)ccc(-c2n[nH]c(C)n2)cc1Cl N1(C(CC2ON=C(C)C2)=O)CCN(C(=O)CCc2cscn2)C2(CCC2)C1 C1(NC(CNS(CC)(=O)=O)=O)CCCN(C(=O)C(C)OC)C1.c1ccncc1 C1(NC(c2c(OC)noc2C)=O)CN(C(c2c[nH]c(=N)s2)=O)C(C)(C)C1 C1(NC(c2cnn(CC)c2C)=O)C2CCN(C(c3cncnc3)=O)CCC12 CCC(CC(=O)NCc1n[nH]cc1C(=O)NCC1CCC=CCC1)C(F)F C=CC(C)(C)CC(=O)NCC1COCCN1C(=O)C(C)Oc1ccc(Cl)cc1C C1(C(C)(C)CNC(=O)CCSC(F)(F)F)CCCCN1C(C1CC1F)=O N1(C(=O)Nc2ncc(C)s2)CCC(OCC(F)C2CCC2)CC1 c1(C(N(CCOCCNC(COCC#C)=O)C)=O)[nH]c2ccccc2c1Cl c1(C(=O)NCC2CN(C(c3ccc(C)o3)=O)CC2C)cc(F)cc(Br)c1C C(CCS(C)(=O)=O)(C(=O)NCC1CCN1C(c1ccco1)=O)OC C1(CNC(CCN(C(C(C)N2CCCC2)=O)CCCO)=O)COCC1O c1(CC(=O)NC2(CN(C)C(c3cnc(S)n3C)=O)CCC2)ccc(O)cc1 c1(C(=O)NC(CC)CNC(c2cncc(OC)n2)=O)cc2sccc2s1 N1(C(c2n(C=C)ncc2)=O)CCC(NC(=O)Cc2cc(O)nnc2O)C12CC2 c1(CNC(C(F)=CCC)=O)cnn(C)c1C(=O)NC(C)C(C)(C)OC c1(OC)cncc(C(=O)NC2CN(C(=O)CC)CC2C)c1C.C1(C(=O)N)CCC1 c1(C(N2CCC(NC(COCC=C)=O)(CO)C2)=O)ccc2ccncc2n1 C(=O)(CC(C)CNC(c1cnc(CNC(C2CCC2C)=O)nc1)=O)OC c1(-c2cn(CC=C)nc2)c(C(N2CCn3cncc3C2)=O)[nH]c2ccccc12 c1(C(=O)NCC2CC(O)CN2C(c2ccccc2Cl)=O)c[nH]c2ccc(F)cc12 C1(C)(CNC(COc2ccc(OCCC)cc2)=O)CN(C(=O)CO)CCO1 N(C(=NCC1(C(C)(F)F)CCOCC1)NCC(Cl)C(F)(F)F)C(C)C c1(NC(c2nc(-c3cn(C(C)(C)C)nc3)c(F)cc2)=O)c[nH]c2nccc(Br)c12 N1(C(c2nccc(OC)c2)=O)CCC(O)(C2(NC(=O)C(CO)N(C)C)CC2)CC1 CC1CN(CCc2ccc(Cl)cc2)CCC1NC(c1cc(C2CC2)n(C)n1)=O Cc1ccc(CC(=O)NCC2(C)CCN(C(=O)CC3OCCC3(C)C)C2)cc1 C(c1ccc2c(c1)COCC2)=CC(=O)NC(CC)CN(C)C(C1CC(F)C1)=O O=S(=O)(c1ccc(NC2CCC=CCC2)cc1Br)NC1CCCSCC1 C1(C(N(CC(N)=O)C)=O)CCN(C(C2CC23CC3)=O)CC1 Cc1cc(C(N2CCOC(CN(C(=O)CO)C)C2)=O)cc(C)n1.c1nc[nH]n1.C C#Cc1ccc(C(=O)NC2CCC(C)(NC(c3cc(C)n(C)c3C)=O)CC2)cc1 C1(NC(C=Cc2n(C)ncc2)=O)CN(C(C2CC3(CSC3)C2)=O)CC1C1CC1 Cc1c(O)ccc(C(N2CCC23CN(C(=O)C2=CCCCO2)C3)=O)c1C C1(CC(=O)NCCCN(C(C)C)C)CCCN1C(C1C=CCCC1)=O C12(C(=O)NC(C3CCCN3C(c3cscn3)=O)C)CCC(C(F)F)(CC1)C2 N1(C(C2C(C)C2C)=O)CC(F)CC1CNC(=O)CCOc1ccccc1Cl c1(C=O)cc2c(=O)[nH]ccn2c1.C(=O)(CCC)N(C(C)C)CC.C(C)(=O)N CN1CCN(C)C(C(=O)N(C)CC2CCCCN2C(c2cnnn2C)=O)C1 CCCC(C)(O)CC(=O)NCC(C)(C)C(=O)Nc1cnsc1 CON(C(=O)C1(N(C(=O)C2=COCC2)C)CC1)C1CCOCC1 Cc1csc2ncnc(N(C3CNCC3F)C(c3cccc(Br)c3)=O)c12 CC1CC=C(C(=O)N2CCCCC(N(C)C(c3cc(C(C)(C)C)on3)=O)C2)CC1 CCCCC(C)CCC(=O)NCC1CCCN(C(c2ccc(C(N)=O)[nH]2)=O)C1 N1(C(CCC(=O)NC)=O)CC(CNC(c2coc(C(=O)OC)c2)=O)CCC1C Brc1cncc(C(c2ccoc2)NC2CCCNC2)c1 C1(C)(NC(C(C)OCC)=O)CN(C(=O)CC2CCOC2)C1 c1(CC)onc(C)c1C(=O)N(C(C)C=O)C1CC1.c1nc(C(C)C)n[nH]1.N C(=O)(N1C(C)CCCN1C)C1C2(CCN(C(c3ccc(OC)nn3)=O)CC2)C1 C1CN(C(C2CC(=C3CC3)C2)=O)C(C)C1.C(=O)CCC=O.C1CC1.CC.N CCCC(C)(O)C(=O)N(CC(C)CNC(=O)Cc1c(F)cccc1Cl)C CC(C)(C)CC(F)C(=O)NCC1(CC(=O)NC2CC(C(F)F)C2)CC1 c1(C(=O)NCC2CN(C(=O)C=Cc3ccccn3)C3CC23)ccc2ncnn2c1 N1(C(CCCN(C(C(C(C)C)NC(C)=O)=O)C)=O)CCCCC(C)C1 n1(-c2c(OC)cccc2Cl)nc(-c2cccs2)nc1C1=NOC(C(C)(C)C)C1 c1(C(=O)NC2C(NC(c3ccn(CC)n3)=O)COC2)cc2c(s1)CCSC2 C1(CC)(NC(C2CCCC2CNC(=O)CCC2CCCCO2)=O)CCCCCC1 C1(CC(=O)NC(COCC)C(=O)NC2CC(O)C2O)CCC(=O)NC1 C1(NC(COCC=C)=O)CN(C(c2cn(C)nc2-c2cccs2)=O)CC1C C(=O)(C(F)C(C)(C)O)NCC1C=CC(NC(C2(F)C(C)C2)=O)C1 CC1OCCC1(C)C(=O)NCCC1(CNC(=O)C=CBr)CC1 CC(=O)C(C)CC(C)C(=O)NOCC(N1CC(Cc2ccco2)C1)=O Cc1oc2nc(Cl)ccc2c1C(N1CC(NC(=O)C2=CCCC2)CC(O)C1)=O N1(C(c2cscc2Cl)C(=O)NC(C)(C)C)CCCC2(C)CCCC12 C1(NC(COCCOC)=O)COCCN(C(C23CCC(CC2)CO3)=O)C1 C1(C(=O)NC(CCC)C)C(NC(=O)C=NOC)C1(C)C Cc1onc(C(=O)NCc2cc(C(=O)NC(c3ccccc3)C#N)ccn2)c1C Cc1cnncc1C(=O)N(C)CC1COCCN1C(C1CCCN1CC(C)C)=O Cc1cccc(C(O)C(=O)NC2COCC2NC(c2cccnc2S)=O)c1 C1(C(=O)NCC2(CNC(c3sccc3F)=O)CCCCC2)CCC2CCC1O2 C1(NC(C(CC)SC)=O)CN(C(c2cccc3nonc23)=O)C2(CCC2)C1 Nc1c(F)ccc(C(=O)NCC(CO)NC(c2cncc(C(F)(F)F)n2)=O)c1F c1(C(N2CC(CC(C(=O)NC3(CCC)CCOC3)F)C2)=O)cnncc1C c1(C(=O)NCC2CC(NC(CCc3n(C)ncc3)=O)C2)cc2c(F)cccc2s1 c1cc(C)ccc1C=O.c1(C(=O)OCC)cc(NC(C2CC2)=O)on1.C CC(CC(C)(C)C)C(=O)N1CCC1C(=O)NC1C2CCCC12 C#Cc1cccc(OCC(=O)N(C)C)c1.C1CCCN1C(=O)CC1CCC(=O)N1 c1(C(=O)NC(CN(C(c2cccc(C(C)C)c2)=O)CC)C)ccc(F)cn1 c1(C(N(CCC)C)=O)cc2c(Cl)cc(Cl)cc2[nH]1.C1(C)(C(=O)N)CCC(=O)NC1 c1(C(=O)NCC2CCCN(C(c3n(C(C)C)ncc3)=O)C2)cc2cn[nH]c2cn1 Cc1cc(OCC(=O)NC2CC(C)C2)cc(C)c1.C(=O)C(C)(C)C1CCOC1 Cc1cccc(-n2cc(CC3CCN(C(=O)CSc4nnnn4C)C3)nn2)c1 C(c1ccc2ncccc2c1)=CC(=O)NCC(C(C)C)NC(=O)CCCCF CP(C)(=O)c1cccc(C(=O)NC2CC(NC(c3nccc(F)c3Cl)=O)C2)c1 N1(C(C2C(C)(C)CO2)=O)CC(CNC(=O)CN2CCOCC2)C2(CC2)C1 N1(C(c2n(C)c(S)nn2)=O)CC(C)(C)CCC1CNC(=O)C(C1CCOCC1)F Cc1ccc(C(N2CC3CC3(CNC(c3cccn3C(C)C)=O)C2)=O)c(Cl)c1 c1(CC)ccc(C(=O)NC2CC(NC(=O)CCc3cnoc3)C2)cc1OC N1(C(c2cc(OC)c(F)cc2)C(=O)NCc2cccs2)CCCC(C)(OC)CC1 C1(C(=O)NC2CCCCC2Oc2ccccc2)CCc2nc[nH]c2C1 N1(C(c2c(C)csc2)=O)CC(CNC(c2cccc(C3CC3)n2)=O)C2CC12 Cc1cc(C)c(C(N2CC3(NC(=O)CCC(C)CN(C)C)CC2C3)=O)c(C)n1 C1(NC(c2n(CC)ccc2)=O)CCCN(C(c2sc(N(C)C)nc2C)=O)CC1F CC(C)(F)C(C)(F)C(=O)NC1CCC(NC(c2ccc(F)c(C#N)c2)=O)CC1 C1(C(=O)NCCCCNC(c2c(C)oc(CO)c2)=O)CCS(=O)(=O)C1(C)C C#CCC(CC(F)F)C(=O)NC(C(=O)NCC(C)(C)CC#C)c1ccoc1 C(=O)(CC1=CCCCC1)NC1C(NC(Cc2c(C)scc2)=O)CCC1 CCCCC(O)CC(=O)N1CCCN(C(=O)CNC(=O)CC2CCCC2)C(C)C1 c1(SCC)nccnc1C(=O)NCC1(O)CCC1.C(C)(C)C.C(=O)N c1(SC)ccc(CCC(=O)NCC2CC2NC(C2CCOC2C)=O)cc1 C1CCC(C)CN1C(c1ccon1)=O.c1(CC)occc1C(=O)NC.C1CC1 C(=O)(C1=NOC(C)C1C)NC(CC#C)C(=O)NCC1(F)CC(CO)C1 C1(C(C(C)C)NC(Cc2nc(C)oc2)=O)CCN(C(=O)CCF)CC1 CC1(CNC(=O)CSCC(F)(F)F)CCN(C(=O)C(O)P(C)(C)=O)CC1 c1(C2C(NC(C(N3C(CCC(=O)OCC)CCC3)=O)=O)C2)ccc(C)cc1 n1(CC(=O)NC(C2CC2C(=O)NCCCCF)C)cc(COC)nn1 c1(-c2c(C)cc(C(=O)Nc3c(F)cc(Cl)cc3Br)nc2)scc2c1OCCO2 C1(NC(c2c(SC)csc2)=O)(CO)CCN(C(=O)CCC(=O)N(C)C)C1 Cc1oc(S(C)(=O)=O)cc1C(N1CCC(NC(C2CC(CCO)C2)=O)C1C)=O c1(CC(N2CC3C(CNC(C(C)CC(F)F)=O)C3C2)=O)ccc([N+](=O)[O-])cc1 C(=O)(C(C)(C)C1CCCCO1)NCCC(C)N(C(=O)COc1cnn(C)c1)C CCCC(C(=O)NC1(C(=O)N)CC1)OC.C12CC1C(=O)NC2.C(C)C C1(O)(CNC(COCCC=C)=O)CN(C(C2(CCO)CCC2)=O)C1.C Cc1c(C(=O)NCC2(F)CC(NC(C3CCCC3C)=O)C2)sc2nnc(S)n12 N1(C(c2nc(CC)oc2)=O)CCN(C(=O)C(C)S(C)(=O)=O)CC1CC1CC1 C1(NC(c2c(C)snc2)=O)CCC(NC(=O)C(F)(Cl)c2ccccc2)CC1 C(=O)(C1CCCc2c[nH]nc21)N1CC(NC(Cc2cc(C)on2)=O)(CO)C1 CCC(COC)C(=O)N1CCC(CCNC(c2cnnn2C)=O)CC1 N1(C(C(C(C)C)O)=O)CCC2(C1)CN(C(c1csc(Br)n1)=O)CCO2 C(=O)(CC(F)(F)F)NCC(N1CCC(N(C)C(c2ccn(C)c2)=O)C1)=O c1(C(N(CC(CC)NC(c2csc(C(C)=O)n2)=O)C)=O)ccc(OC)cc1Cl N1(C(c2c(CC=C)cccc2)=O)CC2CC(NC(=O)C(CC)OCC)C(C2)C1 N#CC1C2CC2CN1C(C1(O)CCN(C(c2ccc(Cl)cc2)=O)C1)=O C1(C(=O)NC(CCC)C)CCCC12CCN(C(=O)C(C)(F)F)C2 C(C(C)(O)CC(=O)NC(C)(C(N1CCCN(C)CC1)=O)C1CCC1)OC c1(OC)ccc(F)c(CN2CCCC(C(=O)Nc3cc(N(C)C)ncn3)CC2)c1 c1(C(=O)NC2CCCCC2NC(c2cscc2Cl)=O)cc2cccnc2[nH]1 N1(C(C2CCOC(C)C2)C(=O)NCCC(=O)OCC)CCC(F)(CO)CC1 C=CC1(C(=O)NC2CC3CSCC3C2)CCN(C(=O)C(C)=C(C)C)CC1 N#CC1(C(N2CC3CC2CC3NC(=O)C=C2CCC2)=O)CCOCC1 CP(C)(=O)c1ccnc(CN=C(NCc2cccs2)NCC2CC2Cl)c1 C1(C(C)(C)CNC(C2CCC2CF)=O)CCCCN1C(c1c[nH]c(=N)o1)=O c1ccc(Br)c(C)c1.c1(CCCNCc2n(CC)nnn2)ccccc1F C(=O)(CCCC(C)(C)C)NC(C(=O)NCC(CC(C)C)CO)(C)CO c1(C(=O)NCC(C)NC(C(C2CCCCCC2)C)=O)ccc(C2COC2)cc1 C1(C(N(C)CCn2ccnc2)=O)CC(C)(C)CN1C(=O)C(Cl)Cl C(C1CC1)(C1CC1)=CC(=O)N(CC)CCO.c1(C=O)c[nH]nn1.C1CC1 Cn1ncc(CNC(C2(NC(=O)CCc3ccoc3)CC(O)C2)=O)c1O N1(C(COCCCCCC)=O)CCC(COC)(NC(C2CCC(=O)N2)=O)C1.C c1(NCC(CC)NC(c2ocnc2C2CC2)=O)ccc(S(=O)(=O)NC)cn1 Cc1cc(C(=O)NC2CCC(CNC(c3cccc(CC#N)c3)=O)C2)ncc1Cl C1(C(=O)NCC2CC23CCC3)(COC)CCCOC1.c1(C=O)ccccn1.C c1(C(=O)NC(CC)C(F)(F)F)c(C(=O)NCc2nn[nH]n2)nn2ccccc12 N1(C(C2CCCN(CCC)C2)=O)CCCC(F)(CNC(c2nc(C)oc2C)=O)C1 N1(C(C(CC)OC)=O)CCC(C2(NC(c3cccc(NC(C)=O)n3)=O)CC2)CC1 CC1(C)OC(=O)C(CC(N2CCCC(C)(CNC(=O)COCCF)C2)=O)O1 c1(SCC(=O)NC(CNC(C(C2CCCC2)OC)=O)CO)ccc(Cl)cc1 CCC(C)C(O)C(=O)NCC(C1CCCC1)NC(C1CC1C1CC1C)=O C12(NC(c3n(C)ccc3)=O)CCN(C(c3c(Cl)ccc(Cl)c3O)=O)CCC1C2 Cc1cc(C(=O)NCCOCCNC(C2CCCCS2)=O)nnc1O Cc1c(C(=O)NC2CCCCC2CNC(C2(CF)CC2)=O)ncn1C N1(C(C2C(C)COCC2)=O)CC2CC(C1)N(C(C1CN3CCC1CC3)=O)C2 C1(C(N2CCCC(N(C)C)C2)=O)CN(C(C2CCC2)=O)C(C)(C)C1 C1(NC(C(COC)OC)=O)C=CCN(C(c2c[nH]nc2C(C)(C)C)=O)C1 n1(CC(=O)NC(CC)CNC(C2(O)CC2(C)C)=O)nc(C)nc1C C1(C(=O)NC2CCN(C(C)=O)CC2)CC(CC)CCN1C(=O)C=CC(F)F Cc1cc(C)c(C(=O)NC2CCCC(C)C2)c(N)c1.C(=O)(CN=S(C)(C)=O)N N1(C(C(CC)(C)CO)=O)CCn2nc(CNC(c3ccc(=O)n(C)n3)=O)cc2C1 N1(C(C2C(C)OCC2)=O)CC2CC(C1)C2NC(=O)Cc1csc(Br)c1 C(=O)(C1=C(Cl)CCC1)N(C1CCN(C(C2CCC(F)C2)=O)C1)CC#C C1(CC=C)(NC(=O)C2=CC(C)(C)C2)CCN(C(=O)C(C)C(C)O)CC1 Cc1cc2cccc(-c3nc(C(C)O)nn3C3CCOC(C)C3)c2o1 CCN(CCSc1cccc(OC)c1)N1CCC2(C1)C(=O)Nc1ccccc12 Cc1ccc(Cl)c(O)c1C(=O)NCCN(C(=O)CC1CCCCC1O)C C=CC(CC)C(=O)N1CCC(C(C)C(=O)N(CC(C)N(C)C(C)=O)C)CC1 C(=O)(C(CC(C)C)N1CCC(C(C(=O)OC)OC)CC1)NCCOCC N1(C(C=C(C)C(F)F)=O)CCCC2(CNC(=O)C=Cc3sccc3C)CCCC12 N1(C(COCC)=O)CC2CC(NC(=O)CC3CC(C4CC4)C3)C(C2)C1 C1(C(N(C2CCCCC2)CC)=O)CN(S(N)(=O)=O)C1.CC(CC=O)C1CC1.N C1(C=O)CC2CC(=O)C1O2.C1(C)(C(=O)NCC(C)(C)OCC)CC=CC1 C1(C(=O)NCC(=CC(NOCC=C)=O)C)CCC(C2CC2)C1 CC(C)(O)C(O)CNC(C1CCOC1CNC(c1cscn1)=O)=O C(=O)(CC1=CCCCC1)N1C2C(NC(c3cnnn3C3CC3)=O)CC(C2)C1 C(C(CC(=O)N1CC(O)(CNC(c2cc(Cl)cnn2)=O)C1)C(F)(F)F)N(C)C C1(NC(C(CC)(C)C)=O)CCN(Cc2ccc(C)c(F)c2)CC1C c1(C(C)=O)cc(C(=O)N(CC(O)CN(C)C(c2ccc[nH]2)=O)C)co1 n1(CCC(=O)NC2CC(C)(NC(c3c(CC)ocn3)=O)C2)ccccc1=O c1(OC)ccc(CNc2ncccc2C(N2CCOCC2C)=O)c(C)c1OC c1(C(C)(C)C)n[nH]c(=NC2CCCCCN(C(=O)Cn3cc(CO)nn3)C2)o1 C=CCC(C)(C)CC(=O)NC(C)CC(=O)NCC1CCCC(OC)C1 CC(C)=C=CC(=O)N1CC(O)CC1CC(N1CCC(OCCO)C1)=O c1(C(CC)NC(c2ccc(OC)nc2C)c2nnnn2C)ccc2c(ccn2C)c1 N1(C(c2c(OC)cc(N)c(Cl)c2)=O)CC(C)CN(C(c2cnc(O)s2)=O)CC1C C1(C(NC2CCN(C(=O)Cc3cncc(O)c3)C2)=O)CCCC(C(N)=O)C1.C C1(C(=O)NCCCCC)CCC(O)CN1C(=O)CCNC(C)=O C(=O)(CCCCCCN=[N+]=[N-])N1CCC(C)C(NC(=O)CC(F)(F)C(F)F)C1C CC1CC(C(=O)NC2CCCN(C(=O)Cc3cc(C4CC4)no3)CC2)=NO1 n1(CC)cc(S(=O)(=O)N2CCC3C2CCN3C(=O)CNC=O)cn1.C1CC1 c1(C(N(CC(C)NC(c2n(CCC)ncc2)=O)C)=O)cc(=O)c(OC)cn1C C1(C(=O)NCC2(CNC(c3nc(Cl)sc3Cl)=O)CCCC2)CC12CCOC2 C1(NC(c2ccc(C)nc2)=O)CN(C(=O)CC(C)C(F)F)CC(F)(F)C1 c1(NCC2CCC(C)O2)cc(S(=O)(=O)NCc2ccc(CO)cc2)ccc1C#N c1(C(N(CCC(C)NC(C2CC(N(C)C)C2)=O)C)=O)sccc1-n1cnnn1 c1(C=O)cc(Br)cc(F)c1F.Cc1nc(C(=O)NCC2CC2C)c(C)o1.N Cn1nc(CNC(=O)Cn2ncnn2)c2c1CCN(C(=O)CCC(F)F)C2 C1(O)(C(C)NC(CC2CC(=C)C2)=O)CCN(C(C2CCCC(C)(C)O2)=O)CC1 N1(C(CN(C)C(c2ccsc2)=O)=O)CC(C2CCN(C(=O)C(O)C3CC3)CC2)C1 N1(C(c2ccc(OC)nn2)=O)CCC2(CCCN2C(=O)CC2CC(=O)NC2=O)C1 N(C1CCCn2ccnc21)C(C1(C(C)C)CCN(C(c2ccsn2)=O)C1)=O Cc1ccc(C(N2CCOCC2CN(C)C(c2c[nH]nc2C)=O)=O)c(N)n1 c1(C(=O)NCC2N(C(c3c(C)nc(OC)s3)=O)CCC2)ccnc(OC)c1Cl c1(C=O)c(F)cccc1[N+](=O)[O-].C1CCC12CCC2.C(=O)(C(C)(C)C(=O)N)NC c1(OC)cc(C(=O)NC)cc(C)n1.C1CN(C(=O)Cn2nccc2C)CC12CC2 c1(C(=O)NC23CCN(C(CC(=C)C)=O)CC2C3)ccc([N+](=O)[O-])cc1O C1(CC(=O)NCCCOCC=C)CCN(C(C2(C)CCCOC2)=O)CC1 c1(CN(C(CC2ON=C(C)C2)=O)C)ccccc1CNC(c1cccs1)=O.C C=CC(C)(CC)C(=O)NC1CC(NC(c2ccccc2)CC)C12CCC2 Cc1nc(NCC2CC2)ncc1C(=O)OCCC(N1CCCCC1)=O.C(N)=O C(=O)(CC(C)(C)C)NC(CCC)CNC(C1(CC2CC2)CCCO1)=O CC1(C)CCC(C(=O)NCC=CC(N2CCC23CCCC3)=O)CO1 C(=O)(CCC(C)CC(=O)OC)N1CC(NC(Cc2nc(CC)sc2)=O)C(O)C1 c1(C(=O)NC(C)CCC2CCN2)cc(F)cc(Cl)c1Cl N1(C(C2C(C(C)C)C2)=O)CCN(CCN(C)C(c2cc(Cl)ns2)=O)CC1.CC CC1CC=C(C(=O)NC2CCC2NC(=O)C=Cc2cc(F)cc(F)c2)CC1 c1(C(N2CCN(C(CCC(CC)C)=O)C3C2CC3)=O)cc2ccc(F)cc2s1 N1(C(CC2C(CC)C2)=O)CCN(C(c2cc(C)cc(F)c2N)=O)CC(O)C1 C(C1=CCCN(C(C2CCOC2CC)=O)C1)NC(C=C(CCC)C)=O CCC(C(=O)N1CCC(Cn2cc(CN(C)CC)nn2)C1)NC(C)=O C1(C(=O)NCCCNC(c2cn(C)nc2C(F)F)=O)COc2cc(F)ccc2O1 C(=O)(C=CS(C)=O)NCC#CCNC(CCCOCCOCC)=O CCC(CCCC(=O)NCC1CCN(C(N)=O)C1)NC(=O)Cn1cccnc1=O N1(C(CC=C)=O)CCC(OCCNC(C23CCN(CC2)C3)=O)CC1 c1(C(=O)NC(C2CC=CCC2)C(=O)NC(c2nccn2C)CC)n[nH]c(=N)[nH]1 C1(CC(=O)NC2(C(=O)NCCCSC(F)F)CCSC2)CCCCO1 c1(C(C)=O)ccc(F)c(NC(N2CCOCC2)=O)c1.C(=O)C(Cl)(Cl)Cl.C=O.N c1(C(=O)NC(C)CCCNC(=O)C(C)Sc2nncn2C)cccc2nn[nH]c12 C1(OC)CCC2CN(C(=O)C(O)C3CN(C(=O)C(C)(C)CCC#N)C3)CC12 CCCCCC(=O)NC1CCCC1NC(C1CCC(=O)C1)=O n1(CC)ncc(C(=O)NCC(C)(C2CCC2)NC(=O)C(C)C)c1Br c1(C(=O)NC2(CN(C(=O)CC3CCCO3)C)CC2)cccs1.C1CC1.C C1(NC(=O)C2=C(Cl)CCC2)CCN(C(=O)C2=COCC2)CCC1CO C=CC1CCCN1C(=O)C(C)(C1CCC1)NC(c1ccnnc1C)=O c1(CNC(CN(C)CC)=O)ccc(CNC(=O)C(C)CF)cc1 C1(C(N2C3(CNC(C(CC)C)=O)CCC2CC3)=O)Cc2ccccc2S1 C12(C(N3CCC(C)(CCNC(=O)CCS)C3)=O)CCCC(CO1)C2.C1CCCC1 C1(C(=O)NC(CCCNC(C2(C(=O)NC)CC2)=O)C)CCc2ccccc2C1 C1(OC)CCC(C(=O)N(C)CC2CCCN2C(=O)C(c2ccnn2C)C)CC1 O=C1CNC(=O)c2ccc(C(=O)NCC34CC3CN(C(=O)C3=CCC3)C4)cc2N1 CC1(CCCC(=O)NC2(C)CC2)NC(=O)NC1=O.c1(C(=O)N)cnn2ccsc12 CC(CCC(=O)N1CC(c2cc[nH]n2)C1)NC(C1CCCC1)=O CC(C)C(CCC(=O)NCCN(CCCF)C)NC(=O)CC(C)C1CC1 c1(CC)cc(F)ccc1C(=O)NC(C1CCCCN1C(c1c(Cl)cnn1C)=O)C c1(-c2cn(CCOCCNC(c3[nH]cc(CC)n3)=O)nn2)ccc(C#N)s1 N1(C(CNC(N)=O)=O)CCN(C(=O)CSc2nnc(S)s2)CC(CO)C1 C(=O)(N=c1ccn(CC(N)=O)[nH]1)C1CCN(C(CC)=O)C1C(C)C Cc1nn(C)c2c(N3CCn4nncc4C3)nc(=NC(C)C(F)F)[nH]c12 C1(CC(N2CC(C(=O)NCC)C2)=O)CCCCC1.C(=O)(CCC1CC1C)N C#CC1(NC(c2cccnc2CNC(=O)Cc2cnccc2C)=O)CCOC1 Cc1ccc(SC(C)C(=O)N2CC(N(C(=O)CSC3CC3)C)C2)cc1C N1(C(C2CCC(C(=O)OC)C2)=O)CC=C(CNC(=O)C(O)C(F)(F)F)CC1 N1(C(C(C)=C(C)C)=O)CCC(C)(C)C1C(=O)NCC12CCN(CC1)CC2 N(C(=NCCCF)NCC1CN(C2CC2)CC1C)CCC(C)=O NS(=O)(=O)c1csc(C(C(=O)N)N(C2CCS(=O)(=O)C2)C)c1.C1CCOC1.C C1(O)(CNC(CCCC)=O)CCCN(C(=O)C(COC)NC(C)=O)CC1 C1(N(CC(c2cnc[nH]2)C)C(=O)C=CCN(C)C(C2CC2Cl)=O)CCCC1 n1(C(C)(C)C)cc(Cl)c(C(=O)NC2(C)CCOCC2)n1.c1(C(=O)N)cncs1 CCCCC(C(=O)NC1CCCCN(C(=O)C(C)(O)C2CCC2)C1)C(C)C c1(C(=O)NC2CCN(C(CCNC(=O)NC)=O)CC2C)c(C)cnc(O)c1Cl c1(C(=O)NCC(C)F)cc(O)nc2c1CN(C(=O)C(C)CC(F)F)CC2 C(C)(CC1=CCCCC1)NC(C1CC(N(C(=O)CN2CCC(F)CC2)C)C1)=O CCC(C(=O)OC)C(=O)NC(CC1CC1)CC(=O)NCc1nnc2n1CCC2 N(C)(S(=O)(=O)N(C)C)CC=O.N1(C(C)=O)CC(O)CC1.C(C)OCC.O CC1(C)CC(C(=O)NC2CCC(C(=O)NC3(CF)CCC3)CC2)CCO1 C(CCC)(CCCNC(=O)CCN(C)CCC)NC(C(C=C=C)C)=O C(=O)(CCCCC(F)F)N1CCC(C(C(=O)OCC)(F)F)C1 Cc1cc(C(=O)NC(C)CC(C)NC(=O)C=Cc2nnn(C)n2)c(C)s1 CC12CCC(C(=O)NCC(C(C)(C)C)NC(C3(C)CC=CCC3)=O)(CC1)CO2 C=Cc1cc(C(=O)N(C2CC(NC(C3CN(C)CCO3)=O)C2)C)cc(F)c1 O=C(C1=NOC2(CCCN(C(c3coc(Cl)n3)=O)C2)C1)Nc1cccnc1Cl CC(C)(C)CCC(F)C(=O)N1CCC(C(=O)NCC2(CCO)CCCC2)O1 Cc1cscc1CNC(=O)C#CCNC(C1(C(C)C)CCC1)=O N1(C(C2(c3cccs3)CC2)=O)CCCC(CNC(C23CCC(CC2)C3)=O)C1 c1(C(=O)NC(CNC(c2ccc(C(C)=O)[nH]2)=O)(C)C2CC2)nnn2c1CCC2 c1(OC(C(C)C)C(=O)N2CC(NC(=O)CCC(N)=O)C2)ccccc1C#N c1(C(N2CC(N(C(CN3C(C)CC3)=O)C)C2)=O)cc(CO)on1 O=C1NCC2CN(C(c3nc[nH]c3C(F)(F)F)=O)CCC2N1 C1(C(=O)NCC(CNC(c2cnc(OC)s2)=O)F)CCc2cnnn2C1 N1(C(=O)OC(C)(C)C)CCCOC(CNCc2ccccc2-n2ccnc2)C1 N1(C(c2c(Cl)ccc(C)c2)C(=O)NCC2CCOC2)CCCC(C2(C)CC2)C1 c1(-n2c(Cc3cc(C)n(CC#N)c3C)nc(C3CC3)n2)ccc2[nH]ncc2c1 N1(C(C(C)n2ccnc2)=O)CCC(NC2CN(c3cc(C(F)F)ncn3)C2)CC1 C1(C2CCN(C(=O)CC(C)CC)C2)(NC(C2CCC(CC)O2)=O)CC1 N1(C(C(CCC=C)(C)C)=O)CC2(CCN(C(C3CC(F)CN3C)=O)CC2)C1 c1(C(=O)NCC2(C(N)=O)CN(C(C3CC34CCCC4)=O)C2)ccc[n+]([O-])c1 c1(CC(=O)NC2(C)CN(C(c3cc(OC)ns3)=O)C2)c(C)nc(O)nc1C C(=O)(C(C)(C)C(=O)N1CCCC(CC(=O)NCC2CCCCO2)C1)OC C1(C=O)(COC)CCCN1C=O.c1ccccc1C1(C)CC1.C(C)(C)C.N N1(C(C2(COC(C)C)CC2)=O)CCCOC(C)C1.C12(C(=O)N)CCCC1C2 c1(C=O)cc(Cl)ccc1F.CC(C)(C(=O)NCc1ocnc1C)C1CCCO1.N c1(CNC(c2cnn(Cc3ncccn3)c2)=O)cn(C2CCCC2O)nn1 C(CC(C)(C)NC(=O)CC(C)C)=CC(=O)NC(c1cccnc1)CC n1(CC(N2CC(C(C(=O)NCC3CCC(C)C3)OC)C2)=O)ncc(Cl)c1C C(c1sc(Cl)nc1Cl)=CC(=O)NCC(C)OC.c1(C=O)c(C)cccc1C.N c1(C(=O)NC2CCN(C(c3sc(CC)c(C)c3)=O)CC2C)cnc2cc[nH]c2c1 N1(CC=O)CC(=O)N(C)C1=O.N1(C(CC2(CSC)CC2)=O)CCCC1C.C C(CC(=O)N1CC2CCC(C1)N2C(=O)C(C(C)(C)C)SC)(C(F)(F)F)OC CC1CCC(NC(C2CC=CC2)=O)CN1CCSc1nc(C2CCCC2)no1 c1(CC)cccc(C(N2CCCC(C)(NC(=O)CC3COCCOC3)C2)=O)c1C N1(C(COC2CCN(C(C(CCC)OC)=O)C2)=O)CCC(O)(CC)CC1 C(C)(CCNC(C1CC(OC2CC2)C1)=O)OC.C1(C)(C=O)CCCS1.N c1(C(N(CCNC(=O)C(O)CC2CCCCC2)CC)=O)cc2c[nH]cnc-2n1 CC(C)(C#CC(=O)Nc1cc2ccncc2[nH]1)CNC(=O)NC1(C)CCOC1 c1(C(N(CCS(C)(=O)=O)C)=O)ncn2c1CCNCC2 Cc1nnccc1C(=O)N(CCNC(=O)C(c1ccccc1)=O)C(C)C O=C(CCS(=O)(=O)NC=O)NCCC1CCN(C(=O)C(c2ccc(F)cc2)F)C1 CN1CCCC1CC(=O)NC1CC1NC(=O)C(=O)NCC1CC1 n1(CCC=C)cc(C(=O)NCCC2(O)CN(C(C3CC3(F)Cl)=O)C2)nn1 c1(OCCNC(CC2CCN(CC)C2)=O)ccc(OC)cc1.C1CCNC1 C(C(C(=O)NC(c1cccnc1F)C)C(C)C)NC(CC=CCC)=O Cc1cc(O)nc(C)c1C(=O)NCCCCCCN(C(=O)C=CS(C)=O)C Cc1nccn1CCC(=O)NC(C(=O)NCC(c1cccs1)O)C1(C)CC1 N1(C(CCC(=O)NCC)=O)CCCC2(CC(NC(=O)C3=NOC(C)C3C)C2)C1 Cc1ccn(CCC(=O)NC2CCC(CCNC(c3cnoc3C)=O)C2)n1 N1(C(CCCN(C(C(COC(C)C)(C)C)=O)C)=O)CCN(C)C(=O)C1 C1(CNC(c2c(C)scn2)=O)CC(C)(C)CN1c1cc(C(C)C)nc(Cl)n1 N1(C(c2ncn(C(C)C)c2)=O)CCOCC(NC(=O)C=Cc2cccc(Cl)c2)C1 S(=O)(=O)(c1cccc(NC(=O)CN(C)CCO)c1)N1C(C)CCC1C Cc1ccc2nc(N3CC(NC(c4conc4C(F)(F)F)=O)C3)sc2n1 CC1CCN(C(=O)C(O)C(C)(C)C)CCN1c1ccc([N+](=O)[O-])cn1 C(=O)(CC1CNc2ccccc21)Nc1cncc(S(C)(=O)=O)c1 c1(NC(CC)CC#N)ccc(S(=O)(=O)NCC23CC=CC(C2)OC3)cc1F C1(C(=O)NCC(CNC(CCN(CCC)C)=O)C)CC2(CCC2OC)C1 c1(C(N2CCCC(NC(CCC(C)(C)OC)=O)C2C)=O)ccc(C=NOC)cc1 Cn1ccnc1Cc1nc(C(F)(F)F)cs1.N12CC(O)(C1)CNC2=O N1(C(=O)NCCCC)CC(C)C(C(N2CC(F)(F)CC2CC#N)=O)CC1C N1(CCCNC(=O)CCNC(c2ccoc2)=O)CCCCCC1=O C1(CC)(NC(c2[nH]cnc2C#N)=O)CCN(C(C2CCCC(O)C2)=O)CC1 N1(C(c2c(C)nc(Cl)s2)=O)CCC2(CCCC2C(=O)NCc2cnn(C)c2)C1 C1(C(=O)OCC)CN(C(=O)C(C)CS(C)(=O)=O)CC12COC2 CC(C)C(CCNC(=O)C(O)C1CCC1)NC(=O)CC1OCCO1 C(=O)(C(=O)C(C)(C)C)NCCC(C(=O)N(CCCC)CC(N)=O)O C#CC1CN(C(c2cc(C(C)C)no2)=O)CCN1C(c1cc(Cl)cs1)=O C(=O)(C1=CCCN(C(=O)CC2COCCOC2)C1)NCC1C(C(=C)C)OCC1 c1(C(=O)NC2(CC)CN(C(C(CC)N(C)C)=O)C2)ccc2cnoc2c1 N1(CCC)CCCC(C(=O)NCCN(C(=O)C(C)CC)CC2CC2)C1 C1(NC(c2ccc(Br)cn2)=O)CC2CC1CN(C(=O)C=Cc1cnccn1)C2 c1(N2C(C(=O)NC(c3ccccc3)CC)CC(O)C2)ncnc2ccccc12 C1(NC(C(=O)NCC(N2CCC(OC)CC2)(C)C)=O)CCNC12CCC2 C1COC2(C1)CN(C(=O)CCS(N)(=O)=O)C2.Cc1nnc(COCC=O)n1C.N C(=O)CCC=O.c1nccs1.C(C(=O)N(CCCOCC)C)=CC=CC.N c1(CC)n[nH]c(=NC(=O)Nc2ccccc2Cn2ccnn2)s1 n1(CC(=O)NCCCCNC(c2csc(C)c2N)=O)nnc2ccccc2c1=O n1(CC(N2CCC(O)(CNC(C(CCC)N(C)C)=O)C2)=O)cc(F)ccc1=O C1(NC(C(c2cn(C)nc2)NC(c2ccsn2)=O)=O)CCC(CC2CC2)CC1 C1(CC)CN(C(c2cc(Cl)nnc2O)=O)CCC1NC(c1csnn1)=O N1(C(CCC=C(C)C)=O)CC2=C(C1)CN(C(C1CCC(C)(C)CC1)=O)C2 c1(C(=O)NCCCC)ccc(OCC2CC2)cc1.C1(C=O)CCC(F)(F)C1 C(c1cccc(Cl)c1)=C(C)C(=O)NC1(C)CN(C(c2cncc(C)c2Cl)=O)C1 CCCC(C(=O)N1CCC(CNC(=O)CC2(O)CCC2)(COC)C1)C(C)C C1(C(=O)NC2CCC(NC(c3cc4n(n3)CCO4)=O)C2)CCC2(CC1)CC2 N1(C(C(C(C)C)CNC(c2c[nH]nc2Cl)=O)=O)CC(O)CC12CCC2 C(CNC(=O)CCCCSC)(CC)(CC)NC(c1c(CC)ccs1)=O C(=O)(C(C)(F)C(=O)N1CCC(C)C(CC(N2CCS(=O)C(C)C2)=O)C1)OC Nc1cnc(Cl)c(C(=O)NCC(O)CNC(C2C=CCS2)=O)c1 N1(C(CN(CCC)C(c2cccc(C#N)c2)=O)=O)CCC(O)CC(C)(C)C1 C1(CC)C(=O)NCCN1C(C1CCCCCC1NC(C1CC2COCC2C1)=O)=O N1(C(C(C)OCOC)=O)CCC(C(C)NC(c2ccoc2C2CC2)=O)CC1 C1(N(C(CSCCCC)=O)C)CN(C(C2CCCCC2(C)C)=O)CC12CC2 C(C)(C)(CCCCC(=O)NC(C)CNC(=O)C(C)(C)C1CC1)OC C1(C=O)CCC2(CC1)CC2.C1(CNC(=O)CSCC2CCCO2)CCOC1 c1(C=O)cc([N+](=O)[O-])ccc1O.c1(C(=O)NC2CC(F)(C)C2)cccc(O)n1 CC1CCCC(C)CN1C(C1(NC(=O)CN2CCCC2)CC(CO)C1)=O c1(C(=O)NCC(C)OC)cccc(C(F)F)n1.C(=O)C(F)OC(F)(F)F.N CC1=CCC(C(=O)NCCn2cnc(C(=O)NCC3=NOCC3)c2)CC1 Cc1ccc(F)c(C=O)c1.C1C2CC1N(C(c1cn(C)nc1C(C)(C)C)=O)C2.N CN=c1nc(N2CCC(N(C)CCO)CC2)[nH]c(=NCC(C)CC2CC2)[nH]1 c1(C(=O)NC2(C)CCN(C(c3ccc(Cl)[nH]3)=O)CC2)ccc(P(C)(C)=O)o1 N=c1nc2c(c[nH]1)CC(C(N1CCOCC(NC(c3cc(F)cs3)=O)C1)=O)CC2 N1(C(C2(C(C)NC(=O)C=CC3CCOC3)CC2)=O)CCCN(C)CCC1 N1(C(CC(C)C2CC2)=O)CCC(NC(=O)C=CCOc2ccccc2)CC1C N1(C(c2ccc(C#C)o2)=O)CCCC(NC(=O)CCc2ccccc2F)CCC1 C(=O)(CC1OCc2ccccc21)NC(CCOC)CNC(=O)Cc1cnccn1 C1(CC(=O)N(CC=C)CC2CC2)COCCN1C(=O)CC1CC=CCN1C C1(CC(=O)NC(C#C)C)CN(C(=O)CC2CCOC2(C)C)CCO1 C1(C2CC2)(C=O)CC(=O)C1.C(CC(O)C(=O)NCc1ncoc1CC)SC CC(C)(C)CC(c1ccc(Cl)cc1)NCc1cnn(CCO)c1 C1(C(=O)NCC(N2CCCC2)C)CN(C(=O)C(Cl)Cl)CC1F Cc1c(CC(N2CC(CNC(=O)C(c3ccccc3)C)C2)=O)cccc1Br CN1C(=O)Cc2cc(-c3ncsc3C(=O)Nc3cccc4cccnc34)ccc21 N1(C(CNC(CN(C)C)=O)=O)CCC(C(=O)NC(c2ncc[nH]2)CO)C1 CCCCC(=O)NCCC(C)(C)NC(=O)COC1CN(C(=O)COC)C1 c1(C(=O)NCCCC)csc(C(C)(C)C)n1.C1(C2CCCO2)(C(=O)N)CCC1 S(=O)(=O)(c1cccc2scnc12)N1CC(C)N(C(c2ccc(Br)nc2)=O)CCC1 C=CCC(C)(CC)C(=O)NCC(C1CC1)NC(c1cnc(C2CC2)cc1C)=O C1(CC=C)(NC(c2csc(-c3ncc[nH]3)n2)=O)CCN(C(=O)CCC(=C)C)C1 N1(C(CC(C)F)=O)CC(NC(=O)C)C2(CCOCC2)C1.C1(CC(=O)N)CCCC1 N1(C(C(CC=C)C)=O)CCN(C(c2cc(C)ccc2CC)=O)C2CS(=O)(=O)CC12 CCC(CCOC)C(=O)NC1CC2(C1)CC2C(N1CCCC1(CCF)CO)=O c1(C(=O)NCCC(C)NC(C2CC23CC(O)C3)=O)ccc(F)c2occc12 C(CCC(O)C(=O)NCC1(F)CCC1)NC(C(C)N(C(C)=O)C)=O C(=O)(C(C)(C)Br)NCCN(C(=O)CC1CCC(C)C1)CCC C(CCCCC(=O)NCC(O)C1CC1)NC(c1c(C)csn1)=O C1(CC(C)NC(c2ccn(CCC)n2)=O)CCN(C(=O)OC(C)(C)C)CC1 C1(CC(=O)NCCC2CCOC2)CN(C(C2CCCCC2O)=O)CC12CC2 c1(CCC(=O)N)cn(C)cn1.C1(CC)CCN(C(C2CC(n3cnnc3)C2)=O)C1 Cc1nnc2cc(NC3(CNC(=O)CC4CCC(=O)N4)CCCC3)ncn12 N1(C(c2cc(C(N)=O)oc2)=O)CC(NC(C2CC3(CCC3)CO2)=O)C2(CC2)C1 Cc1cc2c(cc1C(=O)NCCCOCCCNC(C1(O)CC1)=O)OCO2 c1(OC)ccccc1C1(C(=O)OCC2(c3cccs3)CC2C)CC1 C(CC(C)(C)CC(=O)NCCn1cc(C(=O)NCC(C)(O)CO)cn1)OC c1(C(C)=O)ccc(C(N2CCN(C(C34C=CC(CC3)C4)=O)CC2C)=O)cc1F c1(C(N(C(C(=O)NC2(C)CC2)C2CC2)C)=O)ccc(C2CC2)nc1 N1(C(C2CCCO2)=O)CCC2(CC1)CC(NCc1cc(O)ccc1O)C2 c1(C(=O)NCC2(NC(COCCC)=O)CCOC2)n[nH]c2cc(Cl)ccc12 C1(NC(C=C(CC)CC)=O)CN(C(C2CCC(=O)N2C2CC2)=O)CCC1O C1(C(C)C)CN(C(C2CC(C)(C)C2)=O)CCC1NC(=O)CC.CC(F)(F)F.O CCC(C(=O)NC1CC(C(C)NC(C2CC(=O)N(C)C2)=O)C1)C(F)(F)F c1(C(=O)NCC(C)NC(c2c(C)cc[nH]2)=O)cc(F)cc(F)c1 C1(C(=O)NC(CC)(CC)CO)CCN(C(c2ccc(CO)o2)=O)C(CC)C1 CC1CC(NC(=O)C(C)Sc2nccn2C)CN1C(=O)CCOC1CC1 Cc1cnc(C)c(C(=O)NC2CC(O)(C)C2)c1.C12(CC(=O)N)CCCC1C2 C12(C(=O)NC3CCN(CCNC(c4ccc(C)n4C)=O)CC3)CCCC1C2(F)F c1(-n2ccc(C)n2)ccnc(C(=O)NCC2CN(C(C3SCCC3C)=O)C2)n1 c1(C2COCCN2)cccc(OC)c1.N1(CCC)CCCC1C(F)(F)F Cc1cc(C(=O)NCC(Cc2ccccc2)C(C)C)nn1CCN N1(C(C(CC)OCC)=O)CC2CC1CN(C(=O)CCOC1CC1)C2 C1(O)(CC)CCCN(C(=O)C(C)=C2CC2)C1.c1(C=O)cscc1CC=O.CO c1(C(C2(n3ccnn3)CC2)NCCCCC)nnnn1CCSC1CCOC1 c1(C(N2C(C)CCCC2)=O)ccc2c(c1)C(=O)C(=O)N2.Cc1cc(C(=O)N)ns1 c1(CCNc2cc(N(C)Cc3ccc(Cl)s3)ncn2)cc(Cl)c2ccccc2n1 c1cc[nH]c1.N1(CC)CCC1C(=O)NCCC1(C(=O)N(CC)C)CC1 c1(SCC(=O)NC2CCCCN(C(C3C(C)C3C)=O)C2)ccc([N+](=O)[O-])cc1 C1(Cn2cc(CC3CN(C(c4cncs4)=O)C3)nn2)CCC2C(CC1)C2(F)F N1(C(c2c(S(N)(=O)=O)cn(C)n2)=O)CC2CCC1C1CN(c3ccccc3)CC21 N1(C(C(CC=C)CC=C)=O)CC(O)(C2CCN(C(=O)C(C)(C)C(C)C)CC2)C1 C(=O)(C1=CN(C)S(=O)(=O)N=C1C)NC1CN(C(c2c(OC)csc2)=O)C1 c1(C(c2nnnn2CC2CC2)NCC=C)cccc(-c2ccccn2)c1 C12(C(N(CC(=O)OC)CC#C)=O)CC(CN1C(=O)C(C1CC1)OC)C2 C(C(=O)NC(C)(C)CNC(=O)C(C)(C)c1ccc(Cl)s1)(C(C)C)SC CC(C)CC(C)(O)C(=O)N1CC2CC(NC(c3cc4cccnc4[nH]3)=O)C(C2)C1 N1(C(CC)C(=O)NCCC(C)NC(c2cc(CCCO)on2)=O)C(=O)CCC1=O n1(C(CC)C)ncc(C(=O)NCCCCCCNC(C2CN(C(C)C)C2)=O)c1C Cc1cc2ccc(C(=O)NC3CCC4(C3)CN(C(C3C5COCC35)=O)C4)cc2[nH]1 c1(CC(N2CC(F)CC(NC(C(CC(C)C)C)=O)C2)=O)ccc2c[nH]nc2c1 S(=O)(=O)(c1c(Cl)cccc1Cl)N1C(C(N2CC(=O)NCCC2)=O)CC(F)C1 CCCCCC(CC)C(=O)N1CC2CC1CN2c1nccnc1F C(=O)(C1=CCCOCC1)NCC(CNC(CN(C(C)C)C)=O)C(F)(F)F N1(CC)C(=O)CCC1C(=O)NCC(C)(C)O.c1(C=O)ncc(F)cn1.CC C1(C2=CCCCCC2)(C(=O)OC(c2cccc(C#N)c2)C(=O)OC)CC1 c1(OC)ccsc1C(C)NCC(C)O C(C)(CCC)NC(CNS(CC)(=O)=O)=O.c1(C=O)c[nH]nc1-c1cnn(C)c1 N1(C(C2(C)CC3CCC2C3)=O)CC2(CCN(C(=O)CC3CC=CC3)CC2)C1 c1(SC)cc(C(=O)NC2CCCN(C(=O)C(C(C)O)NC(C)=O)C2)ccc1N c1(-n2c(C)cnn2)ccc(C(=O)NCCCNC(C2C3CCC2CC3)=O)cc1 c1ccc(O)cc1F.N1(C(C2CC(CC(=O)OC)C2)=O)CC(F)CC1C(=O)N c1(OC)ccc(C)cc1C=CC(=O)NCC(C)NC(c1ccc(C)nn1)=O Cc1cnc(C(N2CCC(NC(c3cc(N)ccn3)=O)CC2C)=O)cc1C C(=O)(CCS(=O)(=O)C1CCCC1)NCCCOCCN(C(C(CC#C)O)=O)C CC(C)CC(C(=O)NCC1C2COCC12)ONC(=O)C1CC1Cl Cc1cccc(C(N2CC(O)CC2C(=O)Nc2nccc(I)n2)=O)c1F C(=O)(CCCCC(C)C)N1CCC2(NC(CC3(C=C)CCOCC3)=O)C(C1)C2 O=C(C(Cc1cnn[nH]1)CC(F)F)NCN1CCN(c2cc(Cl)c(Br)cc2F)CC1 Cc1ccc(Br)c(C(=O)NCCC(C)NC(C2CCC(=O)C2)=O)c1F C1(CC(=O)NC2CC(NC(=O)CCC3CCC(O)CC3)C2)CN2CCC1CC2 N1(C(C2C(OC)C2)=O)CC2=C(C1)CN(C(=O)Cc1csnc1C)C2 C1(n2cc(C(C)N(C)C)nn2)CC2CCCC(C1)N2C(=O)COc1ccsn1 c1(C(=O)NCC(C)C)ccc2c(c1)CCOC2.C1(C(=O)N)CCC1c1nc[nH]n1 n1(CC)nc(C(=O)NC23CC2CN(C(C2CCN(C(=O)NC)C2)=O)C3)cc1C C1(CCOC)(NC(=O)CC2CCCCN2C)CCCN(Cc2cc(C)no2)C1 N1(C(C(F)OC)=O)CC(C2CN(C(c3c(C(F)(F)F)noc3C)=O)C2)C1 O=C(C1=CC2C=CC(C1)C2)NCC#CC(=O)NCC1CCOCC1 CC(C(C)(C)C(=O)NCc1ccc(F)cn1)NC(C1CC12CC2)=O C=CCC(C(=O)NCC(CO)NC(C1CC1c1nc[nH]n1)=O)NC(C)=O C1(N(C(=O)Cc2cc(CCC)no2)CC#C)CCN(C(=O)CC2CC2C)CC1 C(=O)(CC1=CCN(C(C2CC23CC3)=O)CC1)N(c1c(C)ccc(C)c1)C c1(C(N2C3C(NC(=O)C4=CCC4)CC(C3)C2)=O)ncnc2c1CCCC2 N1(C(C(C(C)(C)C)OC)=O)Cc2cccc(CNC(c3ccc(C)s3)=O)c2C1 N1(C(c2c(CC)noc2)=O)CC2(CCC2)CC1CNC(c1nncn1C)=O C=CC1CN(C(=O)CC(C)n2ccnc2)CC1NC(=O)CCn1cnnn1 C1(CC)C(NC(=O)Cc2c(F)cccc2F)CCCN1C(=O)C1=NOCC1 C1(NC(=O)C=CSc2ccccc2)COC2(C1)CN(C(C1CC=CCO1)=O)C2 c1(C(N2CCC(c3cc(OC)n[nH]3)CC2)=O)cnc2sc(C)c(C)n2c1=O N1(C(Cc2c(C)con2)=O)CCC(C)(CNC(c2cc(O)nn2C)=O)C1 Cc1c(CNC2(C)CCC(C)CC2)cc(I)cc1C(F)(F)F N(C(=NCCC1(C)CC1)NCC(C)(O)CC1CCCC1)Cc1cc(C)on1 N1(C(C(C(C)C)C(C)C)=O)CCc2nc(O)cc(C(=O)NCC(C)O)c2C1 c1(C(=O)O)cccc(CN2CCCC(OCC(F)(F)F)C2)c1F C1(NC(=O)C=CCCc2ccccc2)CCN(C(C2CCCS2)=O)CC1 CCC(CC(=O)NCc1nc(CNC(=O)C=O)cs1)CC(F)(F)F.C1CC1 c1(CC)cc(C(=O)NC2CCCCC2C)ncn1.S(S(C)(=O)=O)CC=O.N c1(C(N2CCCC(CC=C)C2)C(=O)NC2CC2)ccc(OC)c(COC)c1 c1(C(N2CCCC(CC=C)C2)C(=O)NCC(=C)C)ccc(F)c(Br)c1F CC(C)CC(C)CC(=O)N(CC(O)CNC(C1(O)Cc2ccccc2C1)=O)C C1(CN(C(C2(C)C(C)C2)=O)C2CC2)CCCN1C(=O)CC1COCCO1 C1(NC(=O)CCc2cccs2)CC2C(NC(c3cccc(O)n3)=O)C2C1 C1(CCC)(NC(=O)C(C2(C)CC2)NC(c2ccn(C)c2C)=O)CCNC1=O CC(CC(=O)N1C2CCC1CN(C(C1CC(OC(F)(F)F)C1)=O)C2)C(C)(C)C c1(C(N2CCC(C)C2CC)C(=O)NCC(=C)C)cc(C(=O)OC)cc(F)c1 N1(C(c2cncc(OCCN(C)C)c2)=O)CCS(=O)(=O)C2CCCC12 C1(NC(=O)CCCc2cnn[nH]2)C2CC3C1C3C2C(=O)NCC(F)Cl N#Cc1ccc2c(c1)CN(C(c1cc(=O)cc[nH]1)=O)C2 C(=O)(CCCNC(=O)C(c1ccn(C)c1)C)NCC(COCC)C S(=O)(=O)(c1cc(Br)ccc1C)NCC1C(F)(F)CCN(c2nc(C)cc(C)n2)C1 Cc1cc(C(=O)NCCC2CCCCC2)n(C)n1.C(=O)(C(C)Cc1cnc[nH]1)N Cc1csc(C(=O)NC(C2CCCN2C(=O)CC2CCCCO2)C)c1 C1(CC#C)CCN(C(c2sccc2CNC(C2CCCC2CCC)=O)=O)C1 C1(CC=C)(NC(=O)C(C)CCOC)CCCN(C(=O)CCC2(O)CCC2)C1 Cc1cnc(Cl)c(C(=O)N(C(C)CNC(c2c(C)cccc2N)=O)C)c1 c1(C(=O)NC2CC(C(C)NC(CC(C)OC)=O)C2)ccc(C)cc1F C(=O)(C(C)(C)C(C)(C)c1ccccc1)NCC(CN(C)C(c1cnsc1)=O)O C(=O)(C(=O)N=c1cc(C)o[nH]1)N1C2CCCN(C(C3CC(CC)C3)=O)C2CC1 N1(C(c2scc(CNC(C(CC(C)C)O)=O)c2)=O)CC2(CC(CO)CO2)C1 C1(CCC(=O)N(CC)CC2CCOC2)CCCN(C(C2(C#N)CCCC2)=O)C1 N1(C(C(C)NC(N)=O)=O)CC2CN(C(C3(F)CC3(Cl)Cl)=O)CC2C1 C1(NC(c2nc(C)c(C)s2)=O)CC2(C1)CC(NC(C1C(C)C1C)=O)C2 C=CCC(C)C(=O)N1CCC(C(=O)NCc2nc(N(C)C)no2)C1 Cc1ccc(C(N2CCC(CNC(C3CC3(F)F)=O)C2(C)C)=O)c2c1CCC2 c1(CC)ccc(C(=O)NCc2ocnc2C(=O)NC)s1.C1(CCO)CC1 C1(C(c2nnnn2C(C)(C)CC)NC(c2ccncc2)CC)CCCCCCC1 c1(CCC(=O)NCC(N2CCC2)C)cnn(C)c1O.c1(C(=O)N)cc[n+]([O-])cc1 N1(c2c(Cl)cnc(OC)n2)CCCC(C)(C)C1.c1(CC(=O)N)nc(F)c(F)cc1F C1(C(N(C)CC2CCSC2)=O)CCN(C(=O)Cn2cc(CO)cn2)C12CCC2 C(=O)(C(C)(CC)C(=O)N)OCC.c1(CCC(N2CCCC2)=O)cccc(C)c1 N1(C(=O)NCc2cccc(C(=O)OC)n2)CC(C(=O)OC)OC(C)(C)C1 N1(C(C2(C(C)NC(=O)Cc3ccc[nH]3)CC2)=O)C2C=CCC1CC2 C1(NC(C2C(C)CC(C)O2)=O)CN(C(C2(F)CCOC2C)=O)CC2(CCC2)C1 c1(NC(CC(C(F)F)NC(C(C)(C)OCC)=O)=O)cc(C#N)ccc1F N1(C(C(C)NC(N)=O)=O)CCC(F)(F)C(CNC(C2CCC2)=O)C1 c1(C(N2C3C(C(=O)Nc4n(C)cc(Br)n4)C(C3)C2)=O)ccnc(Br)c1Cl CC1CN(C(C23CCC2C3)=O)CCN1C(=O)CC1CCOC1=O c1ncc(Br)cc1C(F)(F)F.N1(C(C2(CC)CC2)=O)CC(F)CC1C(=O)N C1(C(=O)NC2(c3cn(C(c4ccccn4)CC)nn3)CC2)CCCCC(=O)C1 C=CCC(CNC(=O)CCc1ccsc1)C(=O)NC(CC)CC(=O)OC N1(C(C(C)(F)F)=O)CC2CC1CC2CNC(C1CCC=CCC1)=O N1(C(C(C)NC(C=C)=O)=O)CC2CCC(NC(c3cnn4cccnc34)=O)C2C1 c1(NC(C2CC(NC(=O)C=CCO)C2)=O)ccc(O)c(CO)c1 Cn1cccc(-c2cnc(CNCc3ccc(C#N)cn3)c(C(F)(F)F)c2)c1=O Cc1cccc(C)c1C(=O)NCC1CCC(NC(C2CCC2C)=O)CC1 N1(C(c2ccncc2)=O)CC2CC(NC(C3(F)CCOCC3)=O)C2C1 N1(C(c2c(C)nc(CC)o2)=O)CC2(CCN2C(=O)CCc2ccon2)C1 C1(CC(=O)N(CC(C)C)C)CC(=O)c2ccccc2C1.C(=O)C(F)(F)C(F)F.N C12(NC(=O)CC3CCCCCC3)CCCC(NC(=O)C3=CCCSC3)(C1)C2 C(=O)(C(O)CN1CCOCC1)NCC(n1cc(C2CCCN2C)nn1)C c1(C(N2CCC(O)(CN(C(C(C=C)(C)C)=O)C)C2)=O)cnc(C2CC2)nc1O N1(C(C(n2cc(CC(c3ccccc3)C)nn2)C)=O)CC(C2CC2)CC1C1CC1 C=CCC(F)(F)CN(C(=O)CCOC1CN(C(C2CCN(C)CC2)=O)C1)C c1(C(N(C)CC2(CNC(=O)CCCF)CC2)=O)c(O)nc2ccccc2c1Cl C1(C(N(C2CS(=O)(=O)CC2O)C)=O)COCCN(CCc2cc(F)ccc2F)C1 CON(C)C1CCN(C(C2CCN(C(=O)C(O)CC3CCC4CC34)CC2(C)C)=O)CC1 c1(CC)cc(C(=O)NCCC)cn(C)c1=O.N1(C(C=CC=O)=O)CCOCC1 C1(C(=O)NC2CC(C)(NC(c3coc(Cl)c3)=O)C2)CCN(c2nncs2)CC1 C1(C(=O)NCCN(CCC)C(c2ccc(Cl)s2)=O)CCCC(C(F)(F)F)C1 C1(OCC)(OC)CCN(C(c2cnc[nH]2)C=O)CC1.C(C(C)C)C1CC1.C(C)C c1(CC)nc(C)cc(=NC(C)C2CCCCN2C(=O)CC2(OC)CCOCC2)[nH]1 C(=O)(C(C)(C)CC(=O)N1CCC(CC(=O)Nc2cc(I)ncn2)C1)OC c1(C(N(CCNC(CSCC)=O)C)=O)csc2cccnc12 N1(C(c2c(C)cc(C(C)(C)C)cc2)=O)CCCN(C(=O)C=CC(C)C)C(C)C1 c1(NC(CNC(c2n[nH]c(CC)c2[N+](=O)[O-])=O)C)ncnc2scc(C)c12 C(C)(C)(CCC(=O)N(CC(C)(C)NC(=O)C(C#N)CC1CC1)C)OC C1(C(=O)NOCC2(F)CCC2)CCCC(NC(C2C3CCCC23)=O)CC1 N1(C(=O)OC(C)(C)C)CC2(CCCCO2)C1.C(C(O)C(C)(C)C)ONC(=O)N N1(C(C(OCC)OCC)=O)CCCC(C)(C)C1C=O.c1cnn2c1CCCC2.N N1(C(CC=CCC)=O)CC2C(C(=O)NCCCN3CCCC3)C2C1 c1(C(=O)NCC(CNC(CC(CC)CN(C)C)=O)F)[nH]c2cc(F)ccc2c1C C1(C=O)CC(=O)C12CCC2.CN1CCC(CO)(CNC(C2(C)CC2)=O)C1 C1(CC(=O)N(C(C)CO)C)CN(C(C2(C)CC2C)=O)CCO1 C1(CCC)(NC(=O)CC(COC)COC)CCCN(C(=O)CC(CC)OC)C1 C(=O)(C1=CCN(C(=O)C(C)C#N)C1)N(C)Cc1ccc(CC)o1 C1(C(=O)NC2(C3N(C(c4c(C)nns4)=O)CCC3)CC2)CC1C1CCCC1 N1(C(c2cn(CC)nc2)=O)CC(C)OC2(CCN(C(c3csnn3)=O)C2)C1 c1(C(=O)NC(CNC(C2CC2(F)F)=O)C2CC2)cc(-c2ccccc2)ns1 CC1CCN(C(=O)CCCCN(C)C)C(C)C1NC(c1cnc(O)cc1O)=O CC1CN(C)CC(C(=O)NC(C(=O)Cc2ccccc2)c2ccccc2)O1 C1(C(N2CCCC(NC(C(C)c3ccsn3)=O)C2)=O)CC(S(C)(=O)=O)C1 c1(C(C)N(C(=O)NC2CC(CCn3ccnc3)C2)C2CC2)ccccc1 N1(C(c2cc(CC)ncn2)=O)CC(NC(c2cnn(C)c2)=O)CC(O)C1 c1(NC(=O)NC2(c3ccccc3)CC(F)(F)C2)c(Br)cc(Cl)cc1Br N1(C(C(C(C)O)NC(C)=O)=O)CCCOC(CNC(C2CC3CCC2CC3)=O)C1 Cc1ccc(C(N2CCN(C(c3cccc(OC(C)C)c3)=O)CC2C)=O)c(O)c1 C1(CNC(c2c(C)oc(Cl)n2)=O)CCC(F)(C)CC1.C1(C=O)CCCC(C)C1 CN1C(=O)c2cc(Br)ccc2NC1c1ncoc1C N(C1COCc2ccccc21)Cc1cn(C2CCN(C(C3CCS3(=O)=O)=O)C2)nn1 CCC1=C(C(=O)N2CCCCC2C(C)NC(c2cnc(Cl)n2C)=O)SCCO1 N1(C(Cc2nc(CC)sc2)=O)CCC(C)(NC(=O)COC2CCOC2)C1 CC1CCCCC1C.c1(C=O)cccc(C2CC2)c1.C(=O)(CCC1(C)N=N1)N N1(C(c2cn(C(C)C)nc2)=O)CC2CCN(C(c3cc(C(N)=O)c[nH]3)=O)CC12 c1(C(N2CC(C)(NC(c3ccc(SC)cc3)=O)C2)=O)cccc2c1CCC(=O)N2 c1(OC)ccc(C(C)C)cc1CN1CCCCC1c1cncnc1 c1(C(N2CC(C)(C)C2C2CCN(C(=O)C#CC3CC3)CC2)=O)cc2occc2[nH]1 CC1CCCC(C(=O)NCCC2(NC(c3cn(C(F)F)cn3)=O)CCC2)C1 Cc1ccc(F)cc1CNCc1ccc(Sc2ccccc2)cc1 C1(CC#C)(C(=O)NC)CCCOC1.C12CC(C1)C2.c1(CCC=O)nccn1C CC1(C)CC(C(=O)NCC=Cc2ccccc2)N(C(=O)C(C2CCCCC2)O)C1 C1(C(=O)NCCNC(C(CC)N(C)C)=O)CCCN(c2ncccn2)C1 c1(C(=O)Nc2ncc(-c3cccc(OC)c3OC)s2)cccc2c1CCCC2 C1(n2cc(C(=O)O)nn2)CCC(C(=O)NCCCCc2ccc(Br)nc2)CC1 C(=O)(C(C)(C)C(C)(F)F)N1CCCC(NC(C(C(=C)C)(C)C)=O)CC1 C1(C(N(CCC(=O)NC)C)=O)CCN(C(=O)C(C)C(F)F)C1C c1(CCC(N2CCC(N3C(NC(C)=O)CCCC3)C2=O)=O)c(C)nc(O)nc1O C(C(C)C(C)(c1nnnn1C(C)(C)C)NCc1ccnc(C(F)(F)F)c1)OC CCC(C)(C)C(O)C(=O)NC(C)C1CC1.c1(C(=O)N)ncsc1-c1ccccc1 N1(C(CN2CC(C)(OC)C2)=O)CCC(C)C(CNC(C2(C)CCCC2C)=O)C1 N1(C(CC(C)(F)F)=O)CCC2(CCC(NC(=O)C(C)(C)Cc3cnn[nH]3)C2)CC1 c1(NCc2nc(CC)sc2)[nH]c(=NCCCF)nc2c1cnn2C c1(CN2CCCC(C(C)NC(C(C)OC3CCCC3)=O)C2)ccc(F)c(C#N)c1 c1(NC(C2N(Cc3c(C)nc(F)cc3)CCCC2)=O)cccc(S(C)(=O)=O)c1 C1(C(C)C)CN(C(=O)Cc2ccsc2)CCCN1C(=O)CN1CC(=O)N(C)C1=O CCCC(C)CC(=O)NC(C1CCCN1C(c1cnn(CC2CC2)c1)=O)C CC(C)(C)S(=O)(=O)CC(=O)NC1CC2CCC1N(C(c1cc(CO)[nH]n1)=O)C2 C1(C(=O)NC2(CCC(=O)NCCC(CC)C)CCCC2)CC12CCCC2 C1(CN(C)C(C2C=CCCC2)=O)COCCN1C(=O)CC1COCCOC1 c1(N2CC(COC)N(Cc3ccncc3O)CC2)cc2ncnn2cn1 c1(C(=O)NCC(C)NC(c2c(F)ccc(C)c2Br)=O)nccc2ncncc12 C1(NC(c2c(CC)c(C)sc2)=O)CC2CCC1CN(C(=O)CS(=O)CC)C2 c1(C2C(C(=O)NCC3(NC(C(C)c4cccs4)=O)COC3)C2)ccccc1 c1(NC(CC(COC)COC)=O)ccc2ncnn2c1 c1(C(=O)O)ccc(SCc2cc(-c3ccccc3)cs2)c(F)c1 N1(C(C(CC)C2CCOCC2)=O)CCN(C(=O)C(=O)NCC(F)F)CC(C)(F)C1 CCCCC(C(=O)NC1CC2(CCC2)C1OC)NC(=O)CC1CC2C=CC1C2 Cc1cc(C)c(C(=O)NC(CNC(C2(c3ncco3)CCC2)=O)CO)cn1 c1(CC(=O)NCCN2CCC(NC(C(CSC)O)=O)CC2)cccc2c1OCO2 N1(C(=O)OC(C)(C)C)CCS(=O)(=O)CCC1.c1(C=O)ccc(F)c2ccoc12.N c1(C(N(C)C)=O)cccc(NC(c2ccc(CSc3nncn3C)o2)=O)c1 Cc1cc(C(C)Nc2ccc(-c3ccc(C(N)=O)o3)cc2)c(C)o1 C1(C(=O)NCC(F)C2CCC2)C2CCC(C2)N1C(C1CC2(CCO1)CC2)=O N1(CC=O)CCCCS1(=O)=O.C1(O)(CC(=O)N(C(C)C2CC2)C)CCOC1 N1(C(C(COC)O)=O)CCC(CCCCNC(=O)C=C2CCC(C)C2)CC1 N1(C(c2c(C)noc2N)=O)CCCCC(NC(c2cnc[nH]2)=O)CC1 CC1(C)CN(C(=O)CC2CCCO2)CC(C)(C)C1NC(=O)CCC1CCCO1 c1(C=O)cc([N+](=O)[O-])n(C)n1.CCC(C)(CO)C(=O)NCC1CCCC(C)C1 c1(C(=O)NCC(CNC(C(CC)NC(C)=O)=O)O)nccnc1C(N)=O N1(C(c2nc(OC)nc(O)c2)=O)CCOC2CN(C(C3CCN(C)C3=O)=O)CC12 c1(CC(=O)NCCOCCNC(C2N(CC)CC2)=O)sccc1Br N1(CC)CC(C(=O)NC(C)CN(C)C(c2cnn(C3CC3)c2)=O)NC1=O N1(C(CCC2(C)CC2)=O)CC(CCO)(NC(CC(Cc2ccccc2)CO)=O)C1 c1(CC)ccc(C(=O)N(CCC(C(C)(C)C)NC(C2C=CCC2)=O)C)cc1O c1(C(=O)NCCCC(C)NC(=O)CC(C)C2CCCCC2)nnc(O)cc1O N1(C(c2c(CC)cno2)=O)CCC(C)C1C(=O)NCc1ccccc1C N1(C(C2C(C)(C)C2c2ccncc2)=O)CCCC(CNC(C2(O)CC2)=O)C1 N1(C(CC)CC)CC(C(=O)N(C(C)CNC(=O)Cc2ccccc2)C)CC1=O N1(C(CCCCC#C)=O)C2CCC1CN(C(C1(C(C)(F)F)CC1)=O)C2 C1(C(N(CCCCN(C(c2c(C)cn(C)n2)=O)C)C)=O)CC2CSCC(C1)C2 C1(NC(c2ccc[nH]2)=O)CN(C(c2c(F)cc(F)cc2F)=O)Cc2nccn2C1 C(c1cnc[nH]1)=CC(=O)N(CCC(C)NC(C1CCCCC1)=O)C c1(C(=O)NC(CNC(C(C(C)C)C)=O)C)ccn2ccnc2c1 O=C(O)CC(O)C(=O)NCCCS(=O)(=O)N1CCCC1 C1(COC)C2CN(C(C3CCCCC3c3ccc(C)cc3)=O)CC12 N1(C(c2cc(CC(C)C)on2)=O)CCC2(NC(C3CCCCN3C)=O)CCCC12 c1(NCCC(C)NC(C(C)=C(CC)C)=O)cc2nc(-c3ccccc3)nn2cn1 C1(C(N(C2CCN(C(=O)CN3CCC(OC)C3)C2)CC#C)=O)OC2CCC1C2 c1(C(=O)NC2C(NC(C(CC)F)=O)CC2)ccc(OC2CCCCC2)cc1 C(=O)(CC1COc2ccc(Br)cc21)N1CC(CCO)(OCC)C1 N1(C(C(C)CO)=O)CCCC(CCC(=O)Nc2cnn(C(F)F)c2)C1 C1(C(N2CC=C(CNC(C3(C(N)=O)CCC3)=O)CC2)=O)Cc2ccccc2N1 c1(C(=O)NCC(CNC(c2ccc3nnnn3c2)=O)O)ccc2nc(O)cn2c1 CCCCCCC(C)C(=O)NCCOCCN(C(=O)CC(C)(C)COCC)C N1(C(c2c(C)cccc2F)=O)CC2CC(C1)CN(Cc1cccc(O)c1Br)C2 N1(C(Cc2ccc(C)nc2)=O)C2CC1CN(C(=O)CC1SC(=N)NC1=O)C2 c1(C(=O)NC(C(C)NC(C2(C=C)CCC2)=O)C)cc2ccccc2c(OC)n1 C1(CNC(Cc2n(C)ncc2)=O)CCN(C(C2CCCN2C(N)=O)=O)CC1(F)F C1CC2(CCN(C(=O)C)CC2)C1.O=C(CCOCC1CC1)N.C1CCC1.C N(C1CN(C(=O)C(F)n2ccnc2)Cc2ccccc21)C(C1(C)CCCC1)=O Cc1cccc(C(=O)NC2CCCCC2NC(=O)Cn2ccc(C3CC3)n2)c1O Cc1c(C(N2CC=CC2(C)C(=O)NCC2C3COCC23)=O)cncc1F C1(NC(C#CCNC(C2OCCN(CC)C2)=O)=O)CC2COCC(C1)C2 n1(CC)c(C)cc(C(N2CC(CC(C)(C)C)C2)=O)c1C.N1(CC=O)CCSCC1 Cc1cc(=NCCN2CCN(CCN(C)C)CC2)[nH]c(=NCc2nccs2)[nH]1 N1(C(CC=CCC)=O)CCOC(C(=O)NC2(C(O)CO)CC2)CC1 Nc1cccc(C(=O)NC(Cc2ccccc2)CCNC(c2ccoc2)=O)c1O CC(CC(C)(F)F)C(=O)N1CC(C)(C)CC1CNC(c1ccc2occc2c1)=O N1(C(Cn2ncc(CC)c2)=O)CCC(C)(C)C(C(=O)NC2(C(N)=O)CC2)C1 C1CC2(CCN(C(C3CCC(=O)N3CCC)=O)CC2)C1.C1(C=O)CC(Cl)(Cl)C1 N1(C(C2C(C)(C)C2)=O)CCOC(CC(=O)NCc2ccc(F)nc2)C1 c1(C(N(CCCNC(c2ccc(-c3cccs3)s2)=O)CC)=O)cnc(O)cc1O Cc1nn(CC(F)(F)F)cc1-c1nc(-c2ccncc2)nn1CCc1cnc[nH]1 Cc1cccc(F)c1CC(N1CC(N(C(=O)CC2CCOCC2)C)C(F)C1)=O C1(C(N(CCCCC)C(C)C)=O)CCN(C(C2CC3C=CC2C3)=O)C(C)(C)C1 C1(CCC)(C(=O)NCC2CC2C(=O)N(CC)CC2CCC2)CCC1 C1CC2(C1)C(F)(F)C21CC1.c1(N(CC)CC)ccc(CNC=O)cc1.N C(c1cccnc1C)=CC(=O)N(CCCNC(C1CC1(C)Br)=O)CC n1(Cc2cc[n+]([O-])cc2)c(-c2cnccn2)csc1=Nc1ccc(Br)cc1 CC1CCc2c(C(N3CCCC3(C)CNC(=O)C(C)n3cccc3)=O)csc2C1 CC(CC(=O)NC1CC(C)(NC(c2cnc(C3CCC3)nc2O)=O)C1)C(F)(F)F N1(C(=O)NC2C(C)=C(C)CCC2)CC2(CO)CCCCC2(CO)C1 C1(NC(CCNC(COC)=O)=O)CCN(C(c2coc(Br)c2)=O)CC1F N1(C(c2cncc(CNC(COC3(C)CCC3)=O)c2)=O)CCC2CCCCC12 C1(Nc2cc(NCC3(CCC=C)CCCC3)nc(C)n2)CCc2ccccc2C1 C(=O)(C(O)(C(F)(F)F)C1CC1)NCC(CCCC)NC(c1cn(C)nc1C)=O N1(C(c2c(CC)scc2)=O)CC2OCC(NC(C3OCCOC34CCC4)=O)C2C1 c1(C(N2C(C)(CNC(C(CCC)OC)=O)CCC2)=O)ccc(OC)c(Cl)n1 c1(C(N2CCCC(C(=O)NC)C2)=O)coc2c1CN(C(c1occc1C)=O)C2 c1(C(N(CC(C)CNC(C23CCC(CC2)C3)=O)C)=O)ccc2cncn2c1 N1(C(C=CCN(C)CC)=O)CCN(C(=O)C(c2ccccc2F)C)C(C)C1 CCC1=NOC(CC(=O)NC(C2CCCN2C(=O)CCCN)C)C1.[SH](C)(=O)=O C1(C(=O)NCC)CCCCC1.C(=O)C(CN(C)C)N(C)C.C(CC)OCC c1(CN2CC(C(=O)Nc3cccc(CO)n3)C(O)CC2)ccc2sccc2c1 C1(C2N(C(COCCC)=O)CCC2)CCCN(C(c2cc(C(F)(F)F)n[nH]2)=O)C1 c1(COC)nc(C(N2CC(C(C)NC(C3(C(N)=O)CC3)=O)C2)=O)co1 c1(-c2cn(C3CN(C(C(c4ccc(F)cc4)C)=O)C3)nn2)cnc(O)nc1 N1(C(c2cnc(C)c(N)c2)=O)CCC2(CCC2CNC(=O)C(O)CC2CC2)CC1 c1(CC=O)ccc(C#N)cc1.N1(C(C(C)NC(=O)C)=O)CCC(CC(N)=O)C1 C12(SCCC(C)C)CCOC(C)(C1)C2.c1(C2C(C=O)C2)ccccc1.CCCO.O Cc1cc(C(N2CCCC2C(C)(C)NC(c2cnn(C)c2)=O)=O)nc(C)c1 CCC(CC)C(C)C(=O)NC1(C)CCCCC1.c1(C=O)nn(C)cc1C(C)=O.N C(C)(C(C(=O)NCc1cncc(Cl)c1)C(C)C)NC(c1scc(C)c1C)=O N1(C(CCN(C(C2CCC(=O)O2)=O)CC2CC2)=O)CCC2(CSC2)C1 c1(CN(C)C)cc(C(=O)NCC2CCN(C(=O)C)C2)no1.c1ccccc1.S c1(C(=O)N)ccc2c(c1)C(=O)N(C)C2=O.CCCCCCNC(=O)CC(C)(C)O C1(C(=O)NCC2OCCN(C(C(C)C3CCCO3)=O)C2)CCCCN1N=O c1(C(=O)NCC2C(CNC(c3c(C)nsc3)=O)C2)nccc2nn[nH]c12 N1(C(C2C(NC(CCCC(=O)OC)=O)COC2)=O)CCC2C(O)C(C)(C)C12 C(C)(C(=O)NCc1nccs1)NC(C1C(CCOC)C1)=O c1(C(N2CC(OCCNC(C3CCCC3O)=O)C2)=O)cnn2ccsc12 C1(COC)CC(CNC(c2c(C)ncn2O)=O)N(C(=O)Cc2cncs2)C1 CCC(C)(CNC(C1CC1C)=O)NC(c1cc(-c2cn(C)nn2)on1)=O c1(CS(N2CCCC(C=O)C2)(=O)=O)cccc([N+](=O)[O-])c1.c1ccc(=O)oc1.N C1(OCC=C)CCN(C(C2CC23CC(NC(=O)C(O)C=CC)C3)=O)CC1 N1(C(C2(CC#C)CCCO2)=O)CC2CC(C1)C2NC(C1CC1CC)=O N#CC1CC2(CC(NC(C3CC4CC4N3C(c3csc(F)c3)=O)=O)C2)C1 C=C1CCN(C(=O)CC(F)(F)CC)C(C(=O)NCC(O)COC)C1 c1(CC(=O)NC2(CNC(C(CC=C)C)=O)CC2)c(C)ncnc1C CCCCC(F)C(=O)NCC(C1CC1)NC(c1cc(C)ccc1CC)=O c1(C(=O)NC)ccn(C)c1.c1(CC)nn[nH]c1C.C12CC1C(C)NC2=O C1CC12CCN(C(=O)C(C)(F)F)CC2.c1(OCCOC)cccc(C(=O)N)c1C N1(C(c2c(C(C)C)ocn2)=O)CCC(CCNC(c2cc[nH]c2)=O)CC1 C(=O)(C1c2ccccc2C2CC1C2)NC(CNC(C(C)(C(C)C)OC)=O)C N1(C(CC2C(C)=NNC2=O)=O)CC(C(=O)NC)C(C2CC2)C1.C1C2COCC12 c1(C(=O)NC2C(C(=O)NCCCC)COCC2)cc(O)cc(=O)o1 C1(NC(Cc2ccc(OC)cc2)=O)CN(C(=O)CN2C(=O)CCC2=O)CCC1F c1c(F)cc(Br)cc1Br.c1(C(C)NC(c2csc(C(=O)N)n2)=O)ccc(Br)cc1 C(=O)C(C(C)C)S(=O)(=O)C1CCCCC1.N1(C(C2C(=C)C2)=O)CCOCC1C.N c1(C(=O)NCC(CCCC)NC(=O)C(F)CC2CC2)cnn2c1CCCC2 C1(NC(CSCCN(C)C)=O)CCN(C(c2ccc[n+]([O-])c2)=O)C1C1CC1 c1(OC)c(C(=O)Nc2nc(-c3nn(C)c(C)c3Cl)no2)sc(C)c1Br C1(C2CCCC(C)(C(=O)OCC)C2)CCc2ncc(Br)n2C1 n1(CCOC)nccc1C(=O)NCC1CCC(NC(c2occc2C)=O)C1 C(=O)(C(C)(C)C1CCCCO1)NCCCN(CC(=O)NC(C)(C)C)C c1(C(N2CCCCC2)C(=O)NC)ccccc1OCCN(C)C.n1(C)ccnn1 CC1(C)C(CNC(c2ccc(CO)cn2)=O)CCN1C(C1C=CCCC1)=O C12(C(=O)NC3CC(C(N4CCC(C)C4)=O)C3)CCN(CC1)C2 C1(NC(c2cnn[nH]2)=O)CC2CC(C1)CN(C(=O)Cc1cccc3occc13)C2 N1(C(CC(CCC)O)=O)CC2CCCCC2(NC(c2cnc(O)n2CC)=O)C1 N1(C(C(C2CC2)OCC)=O)CC2CC1CN2C(C1CCCSC1)=O N1(C(C2C(OC)CCC2)=O)CCC2CCN(C(=O)CC3CC(OC)C3)C2C1 Cc1nc(Cl)ccc1NC(C1CC(C)CN(C(c2csc(C#N)c2)=O)C1)=O C1(CC(=O)NCC2N(CC)CC2)CCCN(C(=O)CCNC(=O)C)C1 c1(C(N2CCC(CN(c3ccc(C(C)=O)cn3)C)C2)=O)c(C)ccnc1O C1(SCC)CCN(C(=O)Cc2c(F)cncc2Cl)CC1O.c12ncc(s1)c(=O)[nH]2 C(=O)(C(F)CCCCC)NC1CCC(CC(=O)NCc2ccc(CCC)[nH]2)C1 N1(C(CCCOC(C)=O)=O)CCCC(C(C)(O)CNC(=O)Cn2ccnn2)C1 Nc1ccnc2c(C(N3CCCC3CNC(=O)CSc3ccccc3)=O)cnn12 C(=O)(C(F)C(C)CNC(=O)Cc1cccnc1)NC(CC)C(C)(F)F Nc1ccc(C(N2CC(OCCNC(c3ccnc(Cl)c3)=O)C2)=O)c(F)c1F C=CCC(CNC(c1cc(-c2ccccc2)co1)=O)NC(=O)C(F)n1cccn1 C1(NC(C(CC)C(C)O)=O)CCCCC12CCCN(C(c1cnc[nH]1)=O)C2 C1(C(=O)NC2CN(C(C3(S(C)(=O)=O)CC3)=O)C2)(OC)CCCOC1 CC(C(C)(C)C)=CC(=O)NCC(C1CCC1)NC(=O)C=C1CC1 Cc1cnc(C(=O)NC2CC(NC(c3ccccc3)=O)C2)cc1C#N.C1(O)CC1 CC1CCCN(C(=O)Cc2cnns2)C1CNC(=O)COC1CCCCC1 c1(C(=O)N)cnn2ccn(C)c12.N1(C(C2N(CC)C(=O)CC2)=O)CCCC(F)C1 c1(C(=O)NCC2(C(=O)N)CC(=C)C2)cn(C)nc1CC.C1CCCC1.C C1(C)CCN(C(c2cscc2Br)=O)CC1.C(C)(C(=O)NC)OCCOCC N1(c2cc(C)nc(NC(C)CCCO)n2)CC2CCC(C1)C2(F)F C(=O)(C(F)C(C)(F)F)NC(COC)CNC(c1[nH]nnc1C)=O C(=O)(C(CC(C)C)NC(=O)C=Cc1cn(C)nn1)Nc1ccc(SC)cc1 C12(C(N(CCCNC(C3CSC3)=O)C)=O)CC(c3ccc(F)cc3)(C1)C2F C1(OC)(C)CCN(C(=O)C=Cc2cnc(C)s2)CC1.n1(CC=O)[nH]cnc1=N CCCC(CCCNC(C1(c2n[nH]cc2C)CC1)=O)NC(c1cnc(C)n1C)=O C1(C(N2CCC(C)(NC(C(C)C3CCCC3)=O)C2)=O)COC2COCC2O1 c1(NC(C2NC3CC2C3)=O)cnc2ccc(Br)cn12 N1(C(C2(NC(CCCC3C(C)C3)=O)CC2(C)C)=O)CCc2ccncc2C1 c1(CCC)ccc(CC(=O)NCC2(NC(c3cscn3)=O)CCOC2)cc1 CCC(O)C(C)C(=O)NCC(C)CNC(c1sc(F)cc1Cl)=O c1(N2CCCC(CNC(C3(C(F)F)CC3)=O)CC2)ncnc2c1COC2 C1(NC(CC(CC)OC)=O)CCCN(C(c2cccc(N(C)C)n2)=O)C1CC c1(C2(C)CC2)ccccc1C(N1CCC(C2CCCN2C(c2ccno2)=O)C1)=O C1(CN(C(c2ccc(O)nn2)=O)CC)CCN(C(C2CCC(CC)C2)=O)CC1 N1(C(C(C)n2cncn2)=O)CCC2CN(C(=O)COc3ccc(Cl)cc3)CC12 Cc1oncc1S(=O)(=O)NC1(CO)CN(Cc2ccc(O)c(O)c2O)C1 CCCCC(C)CCC(=O)N(C)CC1CCCN1C(c1cncc(OC)n1)=O c1(CC(=O)NCCC2OCCN(C(C3=CC(C)(C)C3)=O)C2)ccc2nonc2c1 n1(CCOC(C)=O)cc(C2CCCN2C(c2cc(CO)[nH]n2)=O)nn1 CC1=C(C(=O)N2CCC(O)(C)C2)C(C)(C)CCC1.C(=O)(C(F)OC(F)(F)F)N Cc1cc(=NCC2(C)CCCN(C(=O)CC3CC4CCC3O4)C2)[nH]c(C)c1C#N C(=O)(C(F)(F)Cc1ccccc1)N(CC(CN(C(C(COC)C)=O)C)O)C C12(CNC(C3(F)C4CCCCC34)=O)CCC(CO)(CC1)CC2 C#CC1CCCN1c1nnc(C(C)O)n1CC1CCCO1 N1(C(C2=CC(C)(CC)C2)=O)CC2(CCCN(C(C3(C#N)CC3)=O)C2)C1 C1(CC)(CO)CCN(C(=O)CCCn2cc(C3C4COCC34)nn2)CC1 Cc1cc2c(Br)ccc(C(=O)NCC(S(C)(=O)=O)C3CC3)c2o1 N1(C(CCc2onc(C)n2)=O)CCN(C(=O)Cc2nc(C(C)(C)C)cs2)C(C)C1 C1(OC)COCC1NC(c1ccc(CNC(=O)CCc2cnccn2)s1)=O C=CC(C(=O)N(CC(O)CNC(c1ncn(C(C)C)n1)=O)C)OC C1(C(=O)NCC(C)(CC(C)C)NC(c2sc(C)c(O)n2)=O)CCn2nnnc2C1 C1(NC(Cn2ccc(C)n2)=O)CC12CCN(Cc1cccc(Br)c1Br)CC2 N1(C(C2(CC)CCN(C(C3CC(F)CN3C)=O)C2)=O)CC2C=CC1CC2 c1(C(N2C(C)(C(=O)NCC(C)(C)SC)C=CC2)=O)n[nH]c2c1COC2 C#CCC(C(=O)NC1CCC(NC(C2(C)CCOC2)=O)CC1)C1CC1 C12(CNC(c3c(C)snn3)=O)CC(CCO1)C2.C1(CC=O)CCCC(C)C1.N c1(CN(C(C(=O)NC(CC)C)CC2C=CCC2)C)ccncc1F c1(C(=O)NCC(C)N(C(=O)CCCCC(C)(C)C)C)cnc2n1C(C)CCC2 N1(C(C(C)CF)=O)CC(C)OC2(CCC2)C1.c1(C(N(CC=O)C)=O)ccoc1.N N1(C(CC2N(C(COCCCC)=O)CC2)=O)CC2C(C1)C2(F)F C(C)(CCC(=O)NC(C)CNC(c1cccc(C(C)(C)C)n1)=O)OC CC(C(=O)NCCC(C)(C)NC(c1cccc[n+]1[O-])=O)C1OCCc2sccc21 CC(C)(CC(=O)N1CCCC(CCC2CCCN(C=O)C2)C1)C1CC1.C(C)(C)C.O C1(NC(C(CC)F)=O)CC2(C1)CC(NC(=O)Cc1nonc1C)C2 C1(CNC(C=C(C)CN2CCOCC2)=O)CN(C(c2cc(F)cs2)=O)CCO1 C1(C(=O)NCC(C(=O)N(CCC)C)OC)C2CCCC(=O)C12 C(=O)(C(=O)N=c1cc(C)o[nH]1)NC1CCN(Cc2ncc(C)nc2)CC1O C(=O)(CCCCCF)NCC1CC(F)(CNC(C2(C)CCC(C)C2)=O)C1 Cc1cc(CCC(=O)NC2CC(C)(CNC(C3(Cl)CC3(C)C)=O)C2)no1 Cc1ccc2c(c1)C(C(=O)N1CCC(C)C(CNC(c3n[nH]cc3Cl)=O)C1)CC2 N1(C(=O)NC2C(C(N)=O)CCC2)CCC(Oc2ccccc2)CC1 c1(C(=O)NC(C)CCNC(c2cnc(C3CC3)[nH]2)=O)cnc2n1CCCC2C c1(C(N(CCC(C)NC(C2CC=CCO2)=O)C)=O)c(Cl)cc(Cl)nc1N C1(C(=O)NCC2C3CN(C(Cc4cn(C)nc4)=O)C2C3)CC(C2CC2)=NO1 C(c1cnccn1)=CC(=O)NCC(C)C(=O)N(CC(c1cccc(O)c1)=O)C CC(C(C)C(=O)N1CC2C(CO)C2C1)NC(=O)COCc1cccnc1 C1(c2c(OCCC)cc(O)cc2)NC(=S)N(CCC)C2=C1C(=O)NC21CCOC1 CC1(C)CCCC(C)(CNC(=S)NC2CCC2)C1 c1(OC)nc(Cl)ccc1C(=O)NCCC(C)NC(C1CC(=O)NC1(C)C)=O C1(C(=O)Nc2cc(C(C)C)nn2C)CCCC2CN(c3ncncc3I)CC12 CC1CN(c2cc(O)ncn2)CCC1NC(c1c[nH]nc1C1CCCCC1)=O c1(NC(C2C(C)CN(C(C3(n4cnnn4)CC3)=O)CC2)=O)ccc2cnccc2c1 c1(NC(c2c(C)coc2)=O)c(Cc2cn(C(C)C(=O)O)nn2)noc1C C(=O)(CCP(C)(C)=O)NC(C1OCCN(C(C2(CC)CC(C)(C)C2)=O)C1)C N1(C(CCSCCC)=O)CCCC1CNC(=O)CCc1csnn1 c1(OC)nc(C)cc(=NCC2CN(C(c3cc(C)c(O)nn3)=O)CC2C)[nH]1 c1(C(N2CCN(C(CCOCC)=O)C3C2CC3)=O)ccc2nnn(C)c2n1 C1(NC(CCc2cc(OC)no2)=O)CCOCC1NC(=O)CC1CCSCC1 c1(C(=O)OCC)nnc(Sc2ncsc2C(C)C)n1C CC(C)CCN=C(NCc1ccc(F)cc1O)N1CCCC2(C=C2)C1 c1(C(N2CCCN(C(CCC=C=C)=O)C(C)C2)=O)ccc2c(n1)NC(=O)CO2 c1(OC)cc(C(=O)NC(C)CCN(C)C(C2CC2O)=O)cc([N+](=O)[O-])c1 C1(C(=O)NC(CN(C(=O)C=CC2CCOC2)CC)C)CC(C)(C)C1 c1(OCC)ccccc1C(N1CCOC(c2cn[nH]c2)C1)C(=O)NC N1(C(C(CC)CC)=O)CC(N)CCC1(C)C C1(CC(N2CC(C)C(CNC(C3CCC(=O)N3)=O)C2)=O)CCC2(CC1)CC2 N1(C(C(CNC(Cc2c(CC)con2)=O)O)=O)CCSCC1C N(C(=S)NC1CCCn2c(CO)nnc21)CCCCCCC CC1=C(C(=O)N2CCCC2C(C)NC(c2cc(C3CCC3)nn2C)=O)CCO1 C1(C(=O)NC(c2ccc(Br)cc2)C(=O)OC)C2CN(Cc3[nH]cnc3C)CC12 C1(CNC(CCC)=O)CN(C(=O)Cc2csc(-c3ccccn3)n2)C2(CCC2)C1 N1(C(CC=C=C)=O)CCC2CCC(C1)N2C(c1coc(Cl)c1)=O c1(C(N2CCC(NC(c3cc(C)cc(O)n3)=O)C2)=O)cc(Cl)c(O)cc1C C(=O)(CC(C(F)F)C(C)(C)C)N1CC(NC(c2cc(C)c(O)nc2)=O)C(F)CC1 N1(C(CSCC=C)=O)CCN(C(c2ccccc2-c2nc(S)n[nH]2)=O)CC1CC C(C(O)C(=O)NC1CC(CNc2ncccn2)C1)=CCCC c1(CC(N2C(C)CCC(C)C2)=O)ccc2oc(O)nc2c1.C(=O)(CS(C)(=O)=O)N C1(CCC)CN(C(c2cncnc2CC)=O)CC1NC(C1CC(C)(O)C1)=O CC(C)C(C(=O)NC(C(=O)N(C1(C)CC1)C)C(C)C)C(C)C Nc1ccc(F)c(C(=O)NC2COCC2CNC(C2CCCSC2)=O)c1F CC(C)CC(C(=O)NCC1CCC1)C(N)=O.c1(C=O)ccc(C(C)(F)F)cn1 N1(C(c2coc(C)n2)C(=O)NCC=C)CCCC(c2nccs2)C1 C(CCCC(=O)NCCNC(=O)C(CC)SC)OCC C=CCCCC(C)Nc1cc(N2CCC(C)(CCO)C2)ncn1 C(CCCCNC(=O)C)N(C1CN(C(C2CCCCC2)=O)C1)C.C1(C)CCC1.O Cn1cnc2ccc(-c3csc(C(=O)N=c4cc(Cl)n(C)[nH]4)c3)cc12 n1(CC=C)cc(C(=O)NC(C)CC(C)NC(=O)CC2(C)CCCC2)nn1 N1(C(C2CC(=O)OC2)=O)CCCC2(CCc3ccccc32)C1 CN=c1ccc(C(=O)NC2CN(C(C3CCC(F)(F)C3)=O)CC23CC3)c[nH]1 C(=O)(CN=S(C)(C)=O)NCC1(C)CCCC1.c1(C=O)ccc(C(F)F)cc1.N C#CCC(C)(CC)C(=O)NCC1CC(OC)CN1C(=O)C=C(CCC)CCC c1(SC)ccc(CNC(=O)CC2CCN(C)C2)s1.c1cnc(N2CCOCC2)s1 C(CC(C(=O)NC(COC)C1CC1)NC(=O)CCNC(N)=O)=CC C1(N(C(C(C)OCCC#C)=O)C)CCN(C(=O)C(N)=O)C1 Cc1nc2cc(C(=O)N(C)CCNC(c3c(C)cc(O)cc3C)=O)cnc2[nH]1 c1(CCC(=O)NCC(CNC(c2c(C)occ2)=O)(C)O)ccc(N(C)C)nc1 CC(C)(C)C(CNC(=O)CC1C(NC(=O)Cn2cccnc2=O)CC1O)CO N1(C(C(C=CCCC)O)=O)CCN(C(C2C3CCCC23)=O)CC1C(C)C c1(C(=O)NC(CNC(c2nccc3ccsc23)=O)CO)coc2c(F)cccc12 N1(C(c2cncc(OC)n2)=O)CCCC1C1CCCCN1C(=O)C1=CCCSC1 C#CC1CCC(C(=O)N(CCNC(=O)C(c2cccc(C)c2)C)CCO)CC1 C#CCC(CC(=O)N(C(=O)CC(CC)C1CC1)CC1CC(Cl)(Cl)C1)c1ccccc1 C=C1CC(C(=O)NCCC2CC2)N(Cc2cccc(C(C)(C)C)c2)C1 C1(C(=O)NC(CO)CCF)CCOCCN1C(c1cc(O)ccc1F)=O c1(C(N(CCCCN(C(C2(CC#C)CCCC2)=O)C)C)=O)ccncc1C(F)F O(NC(=O)C=C1CCCC1)CCOCC#C.c12ccn(n1)CCNC2=O Cc1cc(C)n2nc(CCCNC(=O)C(F)Cc3ccccc3)c(C#N)c2n1 c1(C(=O)NC2C(NC(C(CC)(C)C)=O)CCCCC2)cnc2sc(C)nc2c1 C1(CNC(Cc2cc(C)sc2)=O)CCC2(CC1)CC(NC(c1ccoc1C)=O)C2 CC1(C)CCC(C)(NC(=O)CCC2(C)CCCN2C(=O)CC2=CCCC2)C1 c1(C(N2C3C(N(C(=O)CC4CCCO4)C)CC(C3)C2)=O)c(F)ccc2occc12 CCC(CC(=O)NC(C)(C)CN1CCN(C(c2ccc(Cl)s2)=O)CC1)SC N1(C(C2CCC(C)S2)=O)CCCN(C(c2c(F)cncc2Cl)=O)CC1 C1(CC)CCN(C(C2CN3CCN2CC3)=O)C(CC)C1 Cc1ccc(F)c(C(=O)NCC(C)NC(c2cnoc2-c2ccccc2)=O)n1 C1(C(=O)OC)CCN(C(=O)Cn2cc(C)nn2)O1.C1(C)(C(=O)N)CCCC1O Cc1cn2c(n1)CC(C(=O)N(C)CC1CC1)CC2.c1(C(C(=O)N)F)ccccc1 n1(CC)c(C(N2CCC(CF)(NC(=O)CS)C2)=O)nc2ccccc12.C(C)C N(C1CCCn2nccc21)C(C(CCC)NC(c1ccc2occc2c1)=O)=O N1(C(CC(CC)(C)C)=O)CC(C)(CNC(=O)CCc2cn(C)cn2)CC1(C)C c1(N2C(CCC(=O)NCC(F)CO)CCC2)ncnc2c1ccn2C1CC1 N1(C(C2CC2F)=O)CCOC2(CCC(NC(=O)C(F)(F)c3ccccn3)CC2)C1 CC1CCN(C(c2cc(CC3CC3)on2)=O)C1CNC(C1CS(=O)C1)=O Nc1cc(F)c(C(N2CCC(O)C(NC(C3C=CCCC3)=O)C2)=O)cc1F Cc1ccccc1CC(=O)NCC1CCOC1.C(=O)C(C)(C)C.C(=O)(CC)N C(CNC(c1cc(CNC(C2CCOCC2)=O)on1)=O)(C(F)(F)F)OC C(C(F)(C(=O)NCC(F)C(C)(C)O)C(C)C)NC(c1n(CC)ccc1)=O C1(C(N(C(C)C)CCN(C(=O)CCc2cnoc2)C)=O)C2CCCC12 c1(C(=O)NCC2(CC#N)CCC2)cc2c(O)nc3ccccc3c2s1 CC1CC(C)N(C(=O)CSC(F)F)CCN1C(=O)C=CSc1nc[nH]n1 CC1CC(NC(c2ccoc2)=O)CCN1C(c1cc(C(F)F)n(C)n1)=O n1(CCOC)cc(NC(=O)NC2(CCO)CCCSC2)ccc1=O N1(C(c2cccc(C(=O)NCC(C)C)c2)C(=O)NC)CC(CO)CC12CCC2 N1(CC2=NC(C)(C)CO2)CCOC2(CCSCC2)CC1 Cc1nc(C2CCCNC2)sc1C(=O)NC1CCS(=O)(=O)C1 CS(=O)(=O)c1cccnc1C(N1C2CCC1C(CNC(=O)C(F)(F)CO)C2)=O C(=O)(C(CC(F)F)NC(c1cn(C)c(=O)n1C)=O)N(CCC)CC C1(C(=O)NCCN(CCO)CC)CN(C(c2cc(C)[nH]c2C)=O)CC12CC2 c1(CNC(c2c(CCC)n[nH]c2)=O)cccnc1C=O.CC(C)(C)N(C)C.N c1(N2C(C)CC(NC(=O)C(c3ccc(F)cc3)(C)F)C2)nc(C#N)ncc1Cl Cc1cc(=O)c(C(N2CC(C)(NC(c3ccc(CF)cc3)=O)C2)=O)cn1C c1(C(=O)NCC2OCCN(C(c3n(C)c(S)nc3)=O)C2)ccc(O)nc1Cl C1(CC(=O)NCC2CN(C(c3cnnc(O)c3)=O)C2)CCCC2CCCCC12 C1(C(=O)NCC(COC)C)CN(C(C2CC3CC2CC3O)=O)CC(C)O1 c1(C(N(CCNC(CC=C(C)C)=O)C2CC2)=O)c(C)nn2c1CCCC2C n1(CC(=C)CC)cc(CN(C)C(c2cnn(C3CCOCC3)c2)=O)nn1 C1(C(=O)NC2C(NC(C=CC(C)C)=O)C2)CCC(=O)N(C)C1 Cc1cc(=N)[nH]cc1C(=O)NC1CCCCCC1NC(c1c(C)cnn1C)=O C1CCC(O)CN(C(=O)Cc2ccc(Cl)cc2)C1.C1(C(=O)NC)(C=O)CCC1.N c1(COC(c2cn(-c3ccccc3)cn2)=O)ccc2ccccc2n1 C(=O)(C1=CCCCC1C)N1CCCC(N(C(c2cc(C)on2)=O)C)CC1 N1(C(c2ccsc2)=O)CCC(O)C1.C1(C(NC)=O)C(C)(C)C1(F)F.COC Cc1cc(CCNC(c2cc(CCNC(c3ccncc3)=O)on2)=O)nn1C N1(C(CCC(=O)N(CC)CC)=O)CC2CCCCC2(CN=c2nc[nH]s2)C1 C#Cc1ccc(C(N2CCN(C(=O)CC(C)(F)F)C(C3CC3)C2)=O)cc1F.C(=O)N c1(CC(N2CCC(C(C(=O)O)(C)C)CC2)=O)cnc2c(=O)[nH]ccn12.C(C)OC N1(C(CN(C(=O)CC(C)SC)CC)=O)CC(C)=CC(C)C1 c1(C(N2C(C(=O)Nc3c(C)nsc3)CSCC2)=O)cc2cccn2cn1 CCCCC(C)C(=O)NC(CN(C(c1cnn(C(C)(C)C)c1C)=O)CC)CC c1(C(=O)NCC2CCC(CC)O2)cc(C(F)(F)F)nc(C2CC2)c1 C1(c2ccccc2)(CS(=O)(=O)NCC(C)C2CC2)CCCO1 C(=O)(C(CNC(=O)CC1(CSC)CC1)OC)NC(C#C)C CCC(CC)C(F)C(=O)NCC1CCCCC1C(=O)Nc1cnccc1C C1(NC(c2cncc(OC)c2)=O)CCCCCC1NC(=O)CCC1CC1(F)F c1(COC)nc(=NC(C)C2CCCN(C(c3cn(C(C)(C)C)nn3)=O)C2)s[nH]1 C1(NC(CC(C)n2ccnc2)=O)COC2(C1)CN(C(C1(CCF)CC1)=O)C2 C#CCC(C)C(=O)NC1CC1CNC(c1ccnc(SC(C)(C)C)c1)=O CC1CC(O)CCN(C(=O)CCN(C)C(c2cnn(C3CC3)c2)=O)C1 N1(C(c2c(C)n(C)cc2)=O)CCC(C(=O)NCCC(F)(F)Cl)C1(C)C c1(CC)c(C(N2CCN(C(c3cc(C)n(C(C)CC)n3)=O)CC2)=O)cccc1F S(=O)(=O)(CC(=O)N1CCCC1C1CCN(C(=O)C)C1)NC.c1cccc(Cl)c1.S N1(C(C=CC(CC)C)=O)CC2=C(C1)CN(C(=O)CC)C2.C1C=CCC1.C(=O)C C#Cc1ccc(C(N2CCCCC2CCNC(C2CCCOC2)=O)=O)c(F)c1Cl C(=O)(C1CSc2ccccc21)N1CC(NC(c2ccc(C(=O)OC)o2)=O)C1 c1(C(=O)NC(C(C)NC(c2cc(O)ncn2)=O)(C)C)cc2ncccc2[nH]1 C1(C(=O)N)CCN(C=O)C1(C)C.c1(OC)ccc(CC)cn1.C(C)(C)C.CC CN1CCCC(NC(c2cc(CNC(C3COCCOC3)=O)[nH]n2)=O)C1=O c1(NCC2(C)CCN(C(C3CC3(C)C)=O)CC2)c(F)cc(C#N)cc1[N+](=O)[O-] N1(C(c2cc(C)ncc2)=O)CC2OCCN(C(c3cc(Br)ccn3)=O)C2C1 C#CC1(O)CCN(C(=O)C(C2(C)CC2)NC(=O)CCc2ncnn2C)C1 C1(NC(CCc2cn(C)nn2)=O)CCC(C)(CNC(c2cccc(N)c2)=O)C1 C1(C(=O)NCc2ccc(C)cn2)(NC(C2COCOC2)=O)CCC(C)(C)C1 C1(CCC)(C=O)CCN(C(c2ncc(C(=O)O)cc2F)=O)CC1.C(=O)C1CC1.O CC1(C)CCC(O)(C)C1.C1(CC=O)CC(O)CN1C(=O)CCCn1ccnc1.N C(=O)(C(O)CC(F)(F)F)N1CC(C(=O)NCc2ccc(Cl)cn2)C1 N1(C(Cn2ncc(CC)c2)=O)CCC(C(C)NC(C2CCOC2)=O)CC1 Cn1cc(C(=O)O)cc1C(=O)NCCCCc1cn(CCc2ccccc2)nn1 C(=O)(C(C)(C)CC(F)F)N1CC(CN(C(C(C)Cc2ccccc2F)=O)C)C1 C1(C(C)(C)C)CSCCN1C(=O)CCCCc1ccc(C(=O)O)cc1 N1(C(CNc2c(OCC)cccc2)=O)CC(NC(C)=O)CC(C)(C)C1 C1CC2(C1)CCC2.Cn1cc(C=CC(=O)N)nn1.N1(C2(C=O)CC2)CCCC1 c1(C(=O)NCC2(NC(=O)CCC3CC3)CCC2)ccnc2ccc(F)nc12 C(=O)(C(Cc1ccccc1)NC(C)=O)NC(CC)CNC(c1cnsn1)=O N1(C(c2ccnc(CC(C)C)n2)=O)CCN(C(C2CCC2(C)C)=O)CC1CO Cc1ccc(C2C(C)CN2C(=O)Nc2nccn2C(C)C)cc1 C=CCCCCCC(=O)NC(CNC(c1ccoc1C1CC1)=O)CCOC CN1CCCCC(COC(=O)Cc2csc(-c3ccc(Cl)cc3)n2)C1=O C(=O)(C(COC)CC(C)C)NCCN(C(CC=C)=O)CC(C)O Cc1nc2c(N(C3CCN(C(=O)Cc4cnns4)C3)C)ncnc2s1 c1(C(=O)OC)c(C(N2CC(NC(C3(C)CCOC3)=O)C(O)C2)=O)cnn1C c1(CCC(=O)NCCCCCCCC#C)n[nH]c2ccccc12 C1(C)CC(F)(F)CN1C(=O)C.c1(SC)ncc(C=O)c(O)n1.[SH](C)(=O)=O C(CC(F)F)(C(=O)N(C)Cc1nc[nH]n1)N(C(C(C)SC)=O)C C1(C(=O)NC2CN(C(C3(C(F)F)CCOCC3)=O)CC2F)CC12CCOCC2 C(=O)(C1=CCCCO1)NC1C(CNC(C2N(CCCC)CCCC2)=O)COC1 N1(C(Cc2c(C)nc[nH]2)=O)CCN(C(C2(C)CCN(C)C2=O)=O)CC1CCO c1(C(c2n(C)nnn2)Nc2ccc3ncnn3c2)c2c(nn1C)CCOC2 Cc1ccc(C(N2CC(NC(=O)CSc3cccs3)C(O)C2)=O)c(N)c1 Cc1cc(C(F)(F)F)ccc1-c1ccc(NC(c2cc(O)cc(Br)c2)=O)cc1O C(CCCCCCCC1CC1)(c1nnnn1CCC1CC1)NCCCCCCC Oc1cc2ccccc2cc1CNCC1CNCCO1 c1(CC(CN(C)C(c2cnc(S)[nH]2)=O)NC(c2ccc(Cl)s2)=O)ccccc1 S(=O)(=O)(c1c(F)c(F)c(F)c(F)c1F)N.CC1(CNC2CCCC2)CCOCC1 C1(CC(=O)NCCOCCNC(CC=CC)=O)CCCCCO1 c1(C(C)Nc2ccnc(C)n2)ccc(OC2CCC2)c(Br)c1 C1(C(=O)OC)(C(=O)N(C2CC(O)C2)CC(C)NC)CC1C.C(C)(C)C.O C1(CNC(c2cc(C)c(C)[nH]2)=O)CCC2CN(C(C3C=CCS3)=O)CC12 N1(C(c2c(C)occ2)=O)CC2CC1C2NC(=O)CCCN1CCCCC1 N(C1CCCc2n[nH]cc21)C(CC1C(NC(c2ccc(CC)cc2)=O)CCC1)=O C(=O)(CC(C)C(F)(F)F)N(C1CCN(C(c2cnn(C(C)C)c2N)=O)CC1)CC C1(C(=O)NCC2C3CN(C(=O)C=CCF)CC23)COc2ccccc2O1 N1(C(C2CC2(Cl)Cl)=O)CCC2CCN(C(C3(C(F)F)CCCO3)=O)CC12 C1(C(N2CC(C(N)=O)C2)=O)C2CCC(C2)C1(C)C.CC1OCCC1(F)C(=O)N c1(C(=O)NC2C(NC(c3nc(OC)oc3)=O)CC2)ocnc1C.C(C)(C)C N1(C(C(=O)N(C)C)=O)CCC(NC(=O)Cc2ccnc(Cl)c2F)C(C(N)=O)C1 c1(CSC)ccc(C(=O)NCC#CC)o1.c1(C=O)c[nH]cc1-c1csc(C)n1 N1(C(CCC(CC)OC)=O)CCC(C)(C)C(CNC(=O)CCc2cn[nH]c2)C1 N1(C(C(CC(C)C)ONC(=O)Cn2ncn(C)c2=O)=O)CCC12CC(C)(CO)C2 c1(-c2occ(C(N(CCCN(C(=O)CN3CC=CC3)C)C)=O)n2)ccc(F)cc1 CCC(O)C(F)(F)C(=O)NC(C1CCN(C(c2c(Cl)ccc(F)c2C)=O)CC1)C CC(CC(C)(C)C)C(=O)NC1(C(N2CCOC(CO)C2)=O)CC1C Cc1cc(C(N2CCCCC2CN(C)C(C2(C)CC2)=O)=O)c(Cl)cc1N C(C(C)(C(=O)NCCC1CC(NC(C2(C#N)CC2(C)C)=O)C1)OC)OC c1(N(C(C)CNC(=O)OC(C)(C)C)C)coc(OCC(F)F)n1 c1(C(N2CCC(C)(COC)C2)C(=O)NC2CC2)cc2ccc(Cl)cc2n(C)c1=O Cc1[nH]c2ncnc(NC3CCN(C(c4cc(F)n(C)n4)=O)C(C)C3)c2c1C c1(NC)nc(C)ccc1C(=O)NC(CCNC(=O)CC(C)CF)C(C)C C1(NC(C(COC)O)=O)CN(C(c2c(F)cc(F)cc2Cl)=O)Cc2ccnn2C1 c1(C(N2CCC(O)(CNC(=O)Cc3nccs3)CC2)=O)ccc2nc[nH]c2c1 C(C(CC1CC1)C(=O)NC)NC(CC1(OCC)CC1)=O.C1CN(C)C1.C c1(C(N2CC(NC(c3nn(C)c(Cl)c3)=O)C3C2C3)=O)cc2c(nc1N)CCCC2 c1(C(N(C(C)C(=O)NCC2CN(C)CCO2)CCC)=O)cnc(OC)nc1 CC(CCCCNC(=O)CCCCF)NC(=O)CNC(c1ccccc1F)=O C1(NC(c2c(C)nsc2)=O)CCCN(C(=O)CC2CCCC23CC3)CC1 n1(CC)nccc1C(=O)NCC1(CC)CC1.C(=O)(CC=O)N.CC(F)F C(=O)(CCC1=CCCCC1)NC1COC2CN(C(CCCC(C)=O)=O)CC21 Cc1noc(C)c1.C(CC(C)C)OCC=O.C(C(=O)N(CCC)C)SCC.N C(=O)(C1=CCC2(COC2)OC1)N1CCCCC(NC(CCCOCC)=O)C1 N1(C(C)C)CCN(C(=NCc2ccnc(C(=O)N(C)C)c2)NC2CCCC2)CC1=O c1(C(=O)NCCC(C)NC(c2cnn(C(C)C)c2F)=O)ccc(S(C)=O)cc1 Cn1ccc(C=CC(=O)NC(CNC(=O)C(c2ccc(Cl)cc2)O)CO)c1 C1(C)(CNC(CSCCN(C)C)=O)CCCN(C(c2ccc(F)cc2O)=O)C1 C1(CC=C)CCCCN1C(C1CC1CNC(=O)CC1CCCO1)=O Cc1ccccc1CC(C)N(C(=O)C(c1ccc(Br)cc1)=O)C c1(C(=O)NC(C2CCN(C(c3c(CC)nns3)=O)C2)C)oc(CO)nc1C CC1(C)CC(O)(CC(=O)N)CO1.C1(CC)CCCCN1C(C1C2CCC(=O)C12)=O c1(-c2n(C)cnc2)cc(C(=O)Nc2csc3ccncc23)c2cc[nH]c2c1 n1(CCCC)nnnc1C(CC)(C1CC1)NC(C)(C)COC(C)C c1(Cc2cccc(OCCN(C=O)SC)c2)cccc(SC)c1[N+](=O)[O-] c1(CC(=O)NC(C2CN(C(=O)COc3ccsn3)C2)C)cn(C)nn1 C(=O)(CCCCC(F)F)N1C(CN(C(C2CNC(=O)N2)=O)C2CC2)CCC1 CCC(O)C(C)C(=O)N1CC(CCNC(=O)C(C)N(C)C(C)=O)(OC)C1 c1(CNC(c2c(C(C)(F)F)cc(F)cc2)=O)ccc(S(N)(=O)=O)o1 C#Cc1cccc(C(=O)Nc2cccc(C)c2)c1Cl C1(NC(c2cc(CC)nn2C)=O)CC(C)CN(C(C2(C)CCN(C)C2=O)=O)C1 C(=O)(CC(=O)NCC(C)NC(C1CCCSS1)=O)OC CCCCC(O)CC(=O)NCC1CC2CCC(C1)N2C(=O)CSC.c1cscn1 N1(C(=O)CC23CC(C2)C3)CC(NC(c2cccc3cnsc23)=O)CC12CCOC2 CC1(C(=O)NC2C3CC(NC(=O)CCCN=[N+]=[N-])CC23)CCCCCC1 C1(NC(C2N(C(CCCOCCOC)=O)C3C(C2)C3)=O)CCC(C)(O)CC1 c1(C(=O)NS(CCCC)(=O)=O)ccc(S(=O)(=O)NC2C=CC(C)(C)CC2)cc1 C1CS(=O)(=O)CC1.c1(OC)ccccc1SCC=O.c1(CC=O)cnc[nH]1.N Cc1cccc2nc(C(N3CCOC(CNC(C4CCCCC4O)=O)C3)=O)cn12 c1(OC)cccc(C(C)NC(C2CCN(C(=O)CCCn3ccnn3)CC2)=O)c1 C=CCC(CC(=O)N(C1CCN(C)C1)CC)NC(=O)CC(C)C n1(CCOC)nnnc1C(c1coc(Br)n1)NCCC(C)SC c1(C(N2CC(C)(C)C(NC(=O)COC(F)F)C2)=O)csc2ncnc(O)c12 C1(C(=O)NCCCCCN(C(=O)Cc2cnc(C)[nH]2)CCC)NC(=O)OC1C N1(C(c2cccc(COC)n2)=O)CCCC12CCN(C(=O)CC1CC3CC3C1)C2 C1(C(=O)NC2C(C)CN(C(C3CCCCN3C)=O)CC2)CCS(=O)(=O)C(C)C1 c1(C(=O)N(CCO)CCO)n[nH]c2cccc(-c3cncc(O)c3)c12 c1(CC(=O)NC(COC)C(=O)NCCCN2CC=CC2)cccc(F)c1 CCC(C)C(C(=O)NC(C)CC(C)C)NCCC(C(C)=O)NCCC=O N1(C(c2c(CC#N)cccc2)=O)CCCN(C(=O)CCN2CCC(F)C2)CC1 C=CCC(C(=O)NCCN(C(=O)C(C1(O)CCCC1)F)C(C)C)C(C)C C12(C(=O)N)CCOC(C)(C1)C2.CCC(CC(=O)NC(C)(C)C(C)C)C1CCC1 N1(C(c2ccnc(C)c2C)=O)CC2(CCCC2NC(=O)C2=CCCOC2)C1 CCCCC(F)C(=O)NCC(C1CCN(C(=O)CCc2c[nH]c(=N)[nH]2)CC1)C N#CC1CCCN(C(C2CCC2CNC(=O)CC2CCCC3CC23)=O)C1 CC1CCCC(OCC(=O)N(C2C3CN(C(=O)C=C(Cl)Cl)CC23)C)C1 c1(C(N2CC3(CN(Cc4ncc(C)nc4)C3)C2)=O)cc(O)c(C)c(O)c1 O=C(CS(=O)(=O)CC(F)(F)F)NCC1CCCN1C(c1n[nH]c2c1CSCC2)=O c1(C(N2CCC(NC(CC(C)F)=O)C2(C)C)=O)ccc(S(=O)(=O)N(C)C)o1 c1(C(CC)OC(c2cnn(C3CCC3)c2)=O)cccc(Br)c1 C1(NC(C2(OCC)CCC2)=O)C2CC1N(C(C1CCOCC1)=O)C2C c1(C(=O)NCCN(CCC)C(C2(C)CC(O)CN2C)=O)ccnc2cc[nH]c12 C12(CC(=O)N(CC)C3CC3)CCC(CC1)CC2.C1(OC)CCCC(CC=O)C1 CC1(NC(c2cscn2)=O)CCCN(C(C2COC2)=O)C1 Cc1cnn(C)c1C(=O)NC1CC(C(=O)NOCC(O)C(C)C)CC1O N1(C(CCC=C=C)=O)CCC2C(CCN2C(C2CCCC23CCC3)=O)C1 CC1CN(C(C2CC3(CC(NC(=O)CCc4ccn(C)c4)C3)C2)=O)CC(C)C1O C=CC1(C(N2CCCC(CC(=O)NCCCCN(C)C)C2)=O)CCCC1 C1(NC(C2C(C)(C)CC2)=O)CCC2CCN(C(c3ccc([N+](=O)[O-])cn3)=O)C12 C12(C(=O)NCC3(NC(C4C(C)C4)=O)CCC3)CCCCC1NC(=O)CC2 CC(C)CC(O)C(=O)N(CC(O)CNC(=O)CCCOc1cccc(F)c1)C CCS(=O)c1ccccc1C(=O)NC1C=CC(CNC(=O)CC)C1.C1CCC1 N1(C(CNC2CC2)=O)CCN(C(=O)C=CC2CCCCC2)C(C2CCC2)C1.CC N1(C(C(C)=C2CC2)=O)CCOC2(CCN(C(=O)Cn3c([N+](=O)[O-])cnc3C)C2)C1 N1(C(c2cc(CC)on2)=O)CCC2C(C1)CN2C(=O)CC.C(=O)C1CC1.CO C1(NC(C=C(C)C(F)F)=O)CN(C(=O)CCOCC2CCCO2)CC1N=[N+]=[N-] N1(S(CC)(=O)=O)CCC(C(=O)NCCC2(CNC(=O)CC)CCC2)CC1 O=C(CCCCCF)NCCn1cc(C(N2CCOC3CC23)=O)cn1 c1(OC)cc(C(=O)NC23CC(C2)C3)c(F)c(Cl)c1.c1(C(=O)N)ccnnc1 c1(C(=O)NCC(CNC(c2n[nH]c(CC)c2Br)=O)C)c(C)ccc(C)c1O N1(C(CNC(CCCOC)=O)C)CCN(C(c2csc(C(C)=O)n2)=O)CC1 Cc1nc(C)c(C(N2CCC(=O)C(C)C2)C(=O)NCC2CC2)nc1C C=CCCCCCCNC(C1CCCN1C(=O)C=C(CCC)CCC)=O C1(NC(c2c(C)nc(CC)o2)=O)CC2CC1N(C(C1(CC(C)C)CCC1)=O)C2 C(=O)(C(C)C(F)F)NCC(=O)NCC(=O)NC.C1(O)(S)CCCCC1 N1(C(c2c(C)nc3sccn32)=O)CCC2(CCN(C(=O)CC3(O)CCC3)C2)C1 c1(C(=O)NC2(CC=C)CN(C(C3(C)COCCO3)=O)C2)ccc2nc(=N)[nH]n2c1 C1(NC(C(C(C)OC)NC(=O)CN(C)C(N)=O)=O)CC2(C1)CC(C)C2 n1(CCC)nc(C)cc1C(N1CCOC(CCN(C)C)C1)C(=O)NCC(C)C N1(C(C=CS(C)=O)=O)CCN(C(=O)CNC(=O)C2CC2)CC(C)(F)C1 n1(CC)nc(C(C)C)cc1C(=O)NC.c1(C(N2CC(C)C2)=O)cnccc1 N1(C(C(CC#C)O)=O)CC(C(=O)Nc2cc(C)sc2C)C(C2CC2)C1 C(CC(=O)NC1C=CCC1)(C(C)(C)C)NC(C(C)=NOCC#N)=O C1(C(=O)NCC(c2ccccc2Cl)O)C2CN(C(C3(F)CC3)=O)CC12 C(CCCCC(=O)NC1CC(C)(CNC(=O)C(F)(F)C2CCCC2)C1)OC c1(C(=O)NCC2(SC)CC2)[nH]ccc1CNC(=O)C(O)C1CCC1 C(=O)(C1=COCCC1)NCCN(C(COc1ccc(OC)cc1)=O)C1CC1 C1(O)(CC(C)C)CN(C(C2CC(N(C)C(c3cc(C(N)=O)[nH]n3)=O)C2)=O)C1 C1(CC(=O)NC)CC2C=CC1CC2.C1CCCCN1C(=O)Cn1nnc(=N)[nH]1.C N1(C(=O)OC(C)(C)C)CCc2ccc(C(=O)NC3CCCNC3=O)cc2C1 N1(C(CC=CC(C)(C)C)=O)CCCC(CC)CC1.C(=O)(CC=CC(C)(C)C)N CCC(C)(C)C(=O)N1CC(CC(C)NC(=O)C=Cc2nccn2CC)C1 C(=O)(C1=CCCCO1)N1CCC(C(C)(C)C)(CNC(c2c(C)[nH]cc2)=O)C1 c1(C(=O)NC(C)CCNC(c2cc(Cl)ncc2O)=O)c(F)ccc2ccoc12 C1(NC(c2n(CC)ccc2)=O)(C)CCCCC1C.c1(C=O)ccc(C)c(Cl)c1.N C(=O)(C(CC)(CC)CO)NCC1(OC)CCN(C(C(C=C)(C)C)=O)C1 N1(C(CCNS(CC)(=O)=O)=O)CC(NC(=O)C=C(C)c2ccco2)CC1C N1(C(c2ncc(C)s2)=O)CCC2(COCCN2C(=O)Cn2ccncc2=O)C1 c1(C2(O)CC(CNC(C3(CC(C)=O)CCCC3)=O)C2)ccccc1Cl C=CC(CCC)CC(=O)N1CCCOC(CNC(c2c(C)cc(O)cc2C)=O)C1 C1(C(=O)NC(CNC(CN(C)C)=O)=O)(CO)CCC1.C1C(C2CC2)N1 N1(C(C(CC)C)=O)CCC2(C=C(C(=O)NC3CCC(O)C(O)C3)C2)C1 C(C)(CN=c1ncc(C(F)F)c[nH]1)NC(c1cc(OC)cc2c1OCC2)=O Cn1cc(C(N2CCCC(C)C2)=O)c(O)nc1=O.C1(C(=O)N)CC(=O)NC(=O)C1 C1(C(C)C)CN(C(=O)C=Cc2ccsc2)CCC1NC(C1CCCCC1(C)C)=O Cc1cc(Br)oc1C(=O)CN(C(C)C(=O)NC(C)(C)C)C C1(N(C(C(C)CN2CCCC2)=O)C)CCN(C(=O)C(C)n2cccn2)CC1 N1(C(CC(=O)N(C)C)=O)CCC(F)CC1C(=O)NCc1ccnc(C#N)c1 C1(NC(CCOC(C)=O)=O)CN(C(C2CC=CCO2)=O)C2(CCCC2)C1 C=C(C)CCCC(=O)N1CCN(C)C(C(=O)NCc2c(F)cccc2F)C1 Cc1c(C(N2CC(NC(c3ccccc3OC3CC3)=O)C(C)C2)=O)cnn1C CCCC(CC)C(=O)N1CCC(C(C)(C)NC(=O)CC(C)(C)COC)C1 O=C(CCCCC(F)F)NC1CN(C(c2cc3c(s2)COCC3)=O)CC1O c1(C(N2CC(N(C(=O)C(c3cccnc3)O)C)C2)=O)cn(C)c(=O)nc1O Cc1ncc(Cn2cc(-c3ccc(C(C)(C)C)cc3)nn2)c(C)c1Br CCC(CC(=O)NC(CO)C(C)NC(=O)CN1CCNC(=O)C1)C(F)F N1(C(C2CN(OC)C(=O)C2)=O)C2CCC1CN(C(c1ccc(C)c(O)n1)=O)C2 N1(C(=O)Cc2nc[nH]n2)CCCC(NC(C2(n3cccc3)CCCC2)=O)CC1 CC(C(N)=O)(c1ccccc1)NS(=O)(=O)CC1CCOC1 c1(COC)ccc(NC(=O)CC2CCN(C(=O)Cc3cncs3)C2)cc1 C(=O)(C1Cc2ccc(Cl)cc21)Nc1n(CC(=O)OC)nc(C)c1 N1(C(C(Cc2cnc[nH]2)NC(c2cc(C)sc2C)=O)=O)CCn2nc(C)nc2C1 c1(-c2ccc(OC)cc2)nc(=O)c(C(=O)NC2CCN(C3CNC3)CC2)c(C)[nH]1 S(=O)(=O)(c1cccc(S(C)(=O)=O)c1)N1CCC(C(=O)NCCCCCC)CC1 N1(C(C(C(C)(C)C)OC)=O)CCOCC(C)(C)C1.C1(C=O)CC(=C2CC2)C1 C(c1cn(C)cn1)=CC(=O)NCCCN(C1CCNC1=O)CCC CCC(CO)(C(=O)N1CCC(C(=O)NC(C)CCSC)C(C)C1)OC N1(C(c2cc(N)cc(N)c2)=O)CC(NC(=O)C=C2CCSCC2)C2CCCCC12 N1(C(C2(COC)CC2(F)F)=O)CC2CCCC(C1)N2C(=O)CC(C)n1cccc1 c1(N(C)Cc2ccncc2F)nc(N2CCN3C(=O)OCC3C2)nc2scnc12 N1(C(C2CC(C)C2)=O)CCC(CNC(=O)C(O)C2CCC2)C(C)C1 c1(C(=O)NC(CC)CNC(=O)CC2CCCC2C)ccc(N(C)C)cn1 C(CCCC(=O)NCCn1cnnc1)N(C(C(CC)OC)=O)C C(=O)C(C)CC(F)(F)F.C(CC(=O)NC(C)(C)CC)(c1cccs1)NC(C)=O Cc1c[nH]cc(C(=O)NC(C2CCN(C(=O)C=CCN3CCOCC3)C2)C)c1=O CC1CC(CNC(=O)CSC(F)(F)F)CN1c1nnc(C(F)F)o1 C=CCCCCC(C)(c1nnnn1CCOC1CC1)NCc1cc(Br)ccc1F C=CC(F)(F)C(=O)NC(C1CCCCC1)CNC(=O)C=CC=O.C1CC1 N1(C(c2c(CCNC(C)=O)cccc2)=O)CCN(C(C2CCCCC2)=O)CC1C C1(O)CCN(C(C23CC(C)C2C3)=O)CC1.n1(CC)nc(C)cc1C(=O)NC.C N1(C(c2cc(C)sn2)=O)CCCN(C(=O)C(C)NC(N)=O)CC1C N1(C(C(CC)NC(C)=O)=O)CCC2CN(C(=O)Cc3cc(C)ccc3C)CCC12 CCS(=O)CC(=O)N1CC(F)(CNC(=O)CCOc2ccccc2Br)C1 N1(C(c2cnc(OC)nc2)=O)CC(C(=O)Nc2ccc(OCF)cc2)CC(F)C1 C#CCC(C(=O)OCC)NC(=O)C(C)NC(c1cnnn1CC)=O c1(SC)ccc(C(=O)NC2CCCC(CNC(c3cnco3)=O)C2)c(Cl)c1 N1(C(C=C(CC)CC)=O)CCC(C(F)F)(CNC(C2(CC)CCC2)=O)C1 CC(C)C(O)C(C)C(=O)NC1CCN(C(=O)C=C2CCC(C(C)(C)C)CC2)C1 c1(-c2ccc(NCCCN3C(C)CCCC3)cc2)cccc2c1OCO2 C1(C(N2C(C(C)NC(C(CC)F)=O)CCC2)=O)CCC(OC)CC1 C(=O)(C(C#N)C(C)C)NCCC1CCN(C(c2n(CCOC)ncc2)=O)CC1 C(C1CCCCCC1)=CC(=O)N(CC(C)N(C(CCCCSC)=O)C)C N1(c2nc(C)nc(=N)[nH]2)CC23CCCCC2(C1)CN(C)C3 N1(C(C2C(C=C(C)C)C2(C)C)=O)CCCCC(NC(C2C3COCC23)=O)C1 C(CS(=O)(=O)CC(=O)NC(C)C)OC.c1(C(=O)N)sc(-c2ccccc2)cc1N C(=O)(C1CCCn2nccc21)NCCC(C)NC(CC(C=C)(C)O)=O CC(C)C(O)C(C)C(=O)N1CC(C(C)(C)O)(CNC(C2CCCCO2)=O)C1 Cc1cncc(CCC(=O)N(C)CC2CCCN2C(C2(c3ccsc3)CC2)=O)c1 C1(C(=O)NCCCCCSC)C2CC2CN1C(=O)CC(C)(C)N(C)C c1(CN2CCC(Cc3nc(COCC)on3)C2)cc(F)cc(Cl)c1 CC1C(NC(C2COCC(C)(C)O2)=O)CCCN1C(=O)C=Cc1cc[nH]n1 C1(N(C(CNCC)=O)CC)CCN(C(=O)C(C)C)CC1.N1(C(C)=O)CCCC1 C1(CCNC(C(C)N(CC(F)(F)F)C)=O)CCCN1C(=O)CCc1ccco1 c1(OC)cccc2c(CC(N3CC(NC(c4occc4C)=O)C4CC34)=O)c[nH]c12 Cc1ccc2c(c1)CC(C(=O)N(CCNC(C13CCC1CC3)=O)C(C)C)S2 C=C1C(N(C(=O)C(C)C(=O)N2CCOCC2)CC)CC2CC1C2(C)C c1(C(=O)NC2C(CNC(c3ccc(=N)[nH]c3)=O)CCC2)cnc2c[nH]nc2c1 N1(C(Cc2cn(C)nc2)=O)CCCCC1CNC(C1(O)CCOC1)=O c1(C(N2CCN(CC(C)NC(CCOCC)=O)CC2)=O)ccc2nc(C)cn2c1 CCC(=O)CCC(=O)N1CCOC(CCCNC(=O)CN2CCCC2C)C1 N1(C(C2(c3ccc(OC)nc3)CC2)=O)CCC(NC(=O)CC(F)F)C(C)C1 C(=O)(CC(C(F)F)C(C)(C)C)NCCCCOC.C1(=CC(=O)N)CCOCC1 O=C(C(F)CC1CCOCC1)N1CCC(NC(C2(F)CCOC2)=O)C1 Cc1[nH]c2c(C(=O)NCCC3CC3)cccc2c1C.C12(CC(=O)N)CCCC1C2 CC1(C(=O)NC2CCC(CNC(C3CCC(=O)NC3)=O)CC2)COCCO1 C1(NC(c2c(C(C)C)cnn2C)=O)COC2(C1)CN(C(=O)CC=C(Cl)Cl)C2 C=CC(CCC)CC(=O)N1CC2CC1CN2C(=O)CCCn1c(C)csc1=O c1(CC)cccc(CNC(C2CN(C(c3ccc(C)o3)=O)CC2C)=O)c1 c1(COC)cccc(NC(C2C3CN(C(=O)C(C)CCN(C)C)CC23)=O)c1 c1(CC)cccc(NC(=O)C(C(C)OC)NC(=O)C(n2nccc2C)C)c1O N1(C(c2cnc(O)s2)=O)CC2CN(C(C3CCCCC3c3nc[nH]n3)=O)CC2C1 c1(C(N2C(CNC(c3c(C)csc3)=O)CCCC2)=O)ccc(Cl)c(F)c1N c1(CCCCC)nc(C(N2CCCC2)C)n(-c2ccn(CCC)n2)n1 C(=O)(CCC(N)=O)NCCNC(N)=O.c1(CC(=O)N)ccccc1F.C=O c1(C(=O)NCC2C3CN(C(c4cc(C)n(C)n4)=O)CC32)ccc2c(c1)CC(C)O2 N1(C(C(C)(C)OC)=O)CCc2nc(CNC(=O)C(C)C(C)C(C)(C)C)sc2C1 N1(C(C(C)n2ccnn2)=O)CCC2CCN(C(C3CNC(=O)N3)=O)C2C1 C12(C(=O)NC(C3(O)CN(c4ncc(C)c(O)n4)C3)C)CC3CC(C1)CC(F)(C3)C2 c1(CNC(C2C(C)(C(F)F)C2)=O)cc(C(=O)NC2CNC(=O)C2)co1 C#CCCCCCC(=O)NC1CN(C(=O)C(C)CC(C)C)CC2(CC2)C1 C1(NC(CC=C=C)=O)CC(CNC(=O)CC(=C)C)C1(C)C C1(CC(=O)NC2(C3CCCN3C(=O)CC3CC4(CC4)C3)CC2)CCCCCCC1 N1(C(c2ccc(OC)nn2)=O)CC2(C(N3CCc4ncccc43)=O)CC1CCO2 c1(C(N2CCN(C)C(CNC(C3CC34CC(O)C4)=O)C2)=O)nccc2occc12 Cn1ncc(Cl)c1CC(=O)NCC1C(C(=O)NCc2ncc[nH]2)C1(C)C c1(N(C(=O)COc2cccnc2C)CCC)ccc2c(c1)CCNC2 C1(O)(C(N(C(CC)CC)CCC)=O)CCN(Cc2ccc(O)nc2)CC1 N1(C(CCC(=O)NC)=O)CCN(C(C2CC2(C)C(F)F)=O)C2CS(=O)(=O)CC12 C1(NCCn2cc(-c3cn(C)nc3)nn2)CN(C(=O)Cc2cc(Cl)sc2Cl)CCO1 O=C(C1CCCc2nn[nH]c21)NCC1C2CN(C(c3cnco3)=O)CC12 c1(C(N2C(CNC(c3c(C)oc(C)c3Br)=O)CCC2)=O)ccn2c(O)nnc2c1 c1(C(=O)NC2CCN(C(c3c(C)[nH]nc3Cl)=O)CC2)nc2n(c1Cl)CCCC2 CC1CCC(C)N1C(c1cccc(F)c1)C(=O)NCCC1CC1 CN(CCCC(=O)NCC1CN(C(C2CCCCS2)=O)CC1(F)F)N=O Cc1ccc(O)c(CC(=O)NC(CNC(C2CCCSC2)=O)C(C)C)c1 c1(C(c2n(CC)nnn2)NCCc2ccccc2Cl)cc2cnccc2o1 N1(C(C2N(CCC)C(=O)CC2)=O)CCC2(CC(NC(=O)C3=CCCCC3)C2)C1 C1(NC(C(C2CC2)NC(C2CC(=O)NC2)=O)=O)CCn2nnnc2C1 N1(c2nc(COC)nc(C)c2)CCN(C(=O)CC(C)c2cnn(C)c2)CCC1C N1(C(C(C)OCC)=O)CCCOC(CNC(=O)Cc2cc(Br)ccc2C)C1 C1(c2cn(C(CC)C)nn2)CCCN(C(C2C(c3ccccc3)C2C)=O)C1 C12(NC(=O)CC3CSCCS3)CCC(CN(C(C3(O)CCC3)=O)C1)C2 c1(C(N(CCCN(C(=O)CCC(C)(F)F)C)C)=O)cccc(C(F)(F)F)c1Cl c1(CC)ccc(C(=O)NC2CCN(C(c3ccc(C)cc3O)=O)CC2F)cc1Br C1(C)(C(N2CC(NC(CCC(C)C)=O)C2)=O)CCN(c2ccncc2)CC1 c1(-c2n(Cc3cccc(OC)c3)nc(CC3CC3)n2)ccc(C)c2ccccc12 C(N=c1nc(N2CCC(O)C(F)C2)c2cc(F)cc(F)c2[nH]1)c1cnc(CC)s1 C1(C(N(C(C(=O)Nc2cccc(C(C)=O)c2)C)C(C)C)=O)CCCCCCC1 C#CC1CCCCN1C(C1(F)CN(C(=O)CC2CSC2)C1)=O C1(CNC(C2CC(OC)C2)=O)CCCCN1C(=O)CCc1ccc(C)s1 C1(C(=O)NC(C2CCCCC2)CNC(=O)CCN2CCOCC2)CC2(C1)CC2F C(=O)(CCC(C)(C)[N+](=O)[O-])NCC1(F)CN(C(C(CCOC)OC)=O)C1 CCC(C)C(C(=O)NC1(C)CCN(C(c2ncc(F)cn2)=O)C1)OC C1(NC2(C(=O)OCC)CC(C[Si](C)(C)C)C2)CC2CCCCC2C1 c1(NC(C2CCN(C(c3ccncn3)=O)CC2O)=O)c(Br)ccc(F)c1F C1(NC(CC2(CCC#N)OCCO2)=O)CCCCC12CCNC2 CC(C)CC(C)CC(C)(c1nnnn1CCCC1CC1)NCCOC1CC1 C(=O)CS(=O)(=O)C(C)(C)C.c1(C=O)cccc(C(F)(F)F)n1.CCC(C)C.N C1(C(N(CCNC(c2c(CC)scc2)=O)C2CC2)=O)NC(=O)C2CC12 c1(CN(C(CN(C(=O)C(C)COC)CCOC)=O)C)ccc(OC)cc1 c1(C(C(=O)NCC(F)F)N(C(C)COC)CC)ccc(C)s1 CC1CCCC(C(=O)NCCCCN2CCC(C(N)=O)CC2)O1 c1(C(=O)OC)cc(F)cc(Cl)c1.C1(C=O)CC2CC2N1C(=O)CN1CCCC1 N1(C(Cc2nc(C)[nH]n2)=O)CCN(C(=O)Cn2ncccc2=O)C(CCO)C1 C1(C(=O)NCC(CN(C)C(C2(C)CCC3CC3C2)=O)O)CCCCC1(F)F C(=O)(CC(C)(C)C(F)(F)F)NC1CC(CNC(C=C(C)Cl)=O)C1(C)C C1(N(C(CCC2CCCO2)C(=O)Nc2ccccc2)CCC)CC2CCC1CC2 CCCCCCc1ccc(C(=O)NC(C2CCCN2C(C2C=CCC2)=O)(C)C)s1 c1(C(N2CC3C(CC(N4C(CC=O)CC4)=O)C3C2)=O)cn(C)ccc1=O.CN C(=O)(N1CCC(C(=O)OC)O1)c1ccc(CNC(c2nc(CC)oc2)=O)s1 c1(OC)nc(C(=O)N(CCCN(C)Cc2ccccc2)C)[nH]c(=N)n1 Cn1ncc(CN2CCOCC2)c1C(=O)NC(c1ccc(F)cc1)C(F)F c1(OC)ccc(N2CCC(CN3CCCC3)C2)cc1.c12cc(cs1)C2 C1(C2CCCC2)(C(=O)N)CCNC1=O.CCC(C)=CC(=O)NCC1CC1C C(N=c1nc(N2CCCC(OCCO)C2)c2c([nH]1)CCCC2)C1OCCC(O)C1 CC(CF)CC(=O)NC(C)(C)CCC1CCCCN1C(c1ncc(F)cn1)=O C(=O)(CCCC(C)(F)F)N1C(C)CCC(NC(C2=C(C)CCC2)=O)C1 c1(OC)cc(NC(C2CC2C(=O)NCc2cncnc2)=O)cc(Cl)n1 Cc1c[nH]cc(C(=O)NC(C2CCCCN2C(=O)CSC)C)c1=O.c1cscn1 Cc1nn(CC(=O)NC23CCC(CC2NC(=O)C=CS(C)=O)C3)c(C)c1C=NO Cc1cc(C(N2C(C)CC3CC23)=O)cc(C)c1.C1(n2cccn2)(C(=O)N)CCC1 c1(N(C)C)ccnc(C(N2CC(CNC(=O)CCC3CCCCO3)C2)=O)c1 N1(C(C2C(c3n(C)ncc3)C2)=O)CC=C(C)CC1.c1(C(=O)N)cc2n(n1)CCO2 Cc1cc(C)c(C(=O)NC2CCCC2C(=O)Nc2c(C)cc(Br)nc2Cl)cc1C Cc1noc(C)c1C(C)CC(N1CC(C)C(O)C1)=O.C1(=CC(=O)N)CCCC1 N1(C(c2c(NC)cccc2)=O)CCC(C)N(C(c2ccn3ccnc3c2)=O)CC1 CN=c1[nH]c(=NCc2ccc(=N)[nH]c2)[nH]c(=NC(C)Cc2ccc(C)c(F)c2)[nH]1 c1(C(N2C(CC(=O)NCC)CCC2)=O)ccoc1C.C1(C)CC(C=O)C1.C CC1CC(C)CN(C(c2ccc(C#N)s2)=O)C1.C1(C(=O)N)CC(=C2CCC2)C1 c1(NCc2c(C)cns2)ccc(CN(C)C)cc1 C1(NC(C(C2CC2)SC)=O)C2CCC1CN(C(c1csc3nccn13)=O)C2 c1(NCc2ccc(OC)c(C)n2)ccc(S(=O)(=O)NCc2cncnc2)cc1Cl Cc1cc(N)c(C(N2CCN(C3COCC3NC(=O)CC3CC3)CC2)=O)c(F)c1 Cc1nscc1CNC(c1ccc(C)o1)=O.c1(C(=O)N)cnn(C2CC2)c1 CC1CC(C(N2CC3CC2CN3C(=O)C(c2ccc(F)cc2)(F)F)=O)CC(=O)N1 C1(CC)CCN(C(=O)Cc2cc(C)on2)C1C(=O)NCCC(C)O CCCCC(O)CC(=O)NCCNC(=O)COCC(F)(F)F.c1ccccc1.C C1(C(=O)NCC(C)CN(C(=O)C(F)(F)c2cscn2)C)CCC(=O)N1 N1(C(CCC2(CCC#C)N=N2)=O)CC(NC(=O)C(C)(C)C2CCCCC2)CCC1C N1(C(C(C)=C2CC2)=O)CCC2(NC(c3cc(Br)cn3C)=O)CCCCCC12 N1(C(c2c(C)ccc(N)c2)=O)CCCC2(NC(=O)CC=C(Cl)Cl)CC2C1 C1(C(F)(F)F)(C(N2CCCC2)=O)CC(F)(F)C1.C1(C)(CNC)C=CCCC1 N1(c2ncnc(N3CC(CC)SCC3)c2C)CCc2ccc(Cl)cc2CC1 C1(NC(C=CCC)=O)CN(C(C2CC2c2ccc(F)cc2)=O)C2(CCCC2)C1 c1(C2OCCN(CC(C3(CO)CCOCC3)O)C2)ccc(Cl)c(Cl)c1 c1(CC)cc(C(=O)NCC(C)(C2CC2)NC(=O)CC2CCCNC2=O)nn1C C1(C(N2C(CNC(c3c(COC)noc3)=O)CCCC2)=O)Cc2nncn2C1 N1(C(c2cc(OCC)n[nH]2)=O)CC2CCC2(NC(c2cncnc2)=O)C1 c1(OC)cc(CO)ccn1.C1(C=O)CCC(C(N)=O)C1.CC(=O)N(CCC)C N1(C(C2N(C)CCCC2)=O)CCC(O)C(NC(=O)CCF)C1 c1(C(N2CCC(N(C(C=C(C)C(F)F)=O)CCO)C2)=O)ccc(C)cc1C N1(C(CN2CCN(C)CC2)=O)CC2CCCC2(NC(c2cc(O)cc(=O)o2)=O)C1 C1(C(N2C3CC(C2)C3)=O)OC(C)(C)OC1(C)C.Cc1ccc(F)c(C(=O)N)n1 c1(CC(=O)NCC(CNC(c2ccc(C#N)s2)=O)O)c[nH]c2cnccc12 C1(CNC(c2c(SC)noc2)=O)CN(C(c2n[nH]c(C)c2O)=O)CC1(F)F c1(C(N2C(C(CNC(CSC)=O)(C)C)CCC2)=O)cc(C(F)F)cc(C)c1 CCCCC(C(=O)NC1CC2CC1CN(C(c1csnc1C1CC1)=O)C2)C(C)C c1(CCC(=O)NCC2CCC(NC(C(C)=CC)=O)C2)nnc(S)nc1O c1(OC)cc(C(N2CCCC2)=O)cc(F)n1.C1(C=O)CCCN(C(=O)C2CC2)C1 N1(C(C(C2CCCCCC2)C)=O)CCOCC(NC(c2csc(C#N)c2)=O)C1 c1(C(N(CCCN(C)C(C2(F)CCCC2)=O)C)=O)nn[nH]c1C(F)(F)F.C c1(CC)cc(C(N2CCN(Cc3cn[nH]c3)CC2C)=O)cc(C)n1 C(CCCCC(=O)NCC(O)CC(=O)NCC(C#N)CC)=CC C1(C(=O)NCC2OCC(C(=O)NCCCC=C)C2)COCCC1C C#CC1CCC(C(N2CCN(C(=O)C(=O)NCC3CCCCC3C)CC2)=O)CC1 c1(OC)ccc(C)cc1C(N1CC(NC(c2cc(C)sc2C)=O)C2CC2C1)=O N1(C(CCC)=O)CCOCC(F)(CNC(c2c(C3CC3)cccc2F)=O)C1 C#Cc1c[nH]nc1C(=O)N(CCC(=O)NOCC1CC2C=CC1C2)C1CC1 C1(NC(C(CC)(C)O)=O)CC(F)CN(C(=O)Cc2cc(C)cc(F)c2)C1 N1(CC#C)CCN(C(=O)C(CCCC)NC(=O)C(C)C#N)CC1=O c1(C(C(=O)NCC2C(NC(CCCSC(C)C)=O)C2)C)ccccc1Cl C(N=c1[nH]c(=NCCC(F)(F)C(F)F)c2ccccc2[nH]1)c1c(CCC)nns1 C1(CC=C)(NC(=O)C(C(C)C)n2cnnc2)CCN(C(=O)C(CC)=CCCC)C1 Nc1c(C(=O)NCCCCCCNC(=O)CC23CCCC2C3)cnc(Cl)c1F N1(C(CCCC=C)=O)CCC2(CC1)CC2NC(=O)C1=CCCC1C c1(CC)ccc(C(N2CCOC(CC(N3CCC(F)C3)=O)C2)=O)nc1 c1(C(=O)NCC2C(NC(C(C(C)C)(C)C)=O)CCCC2)cccc2ccnn12 C1(C(N(CC(C)CNC(=O)C(O)CC2CCCCC2)C)=O)CCCCC12CCC2 C=CCCC(C(=O)N1CCC(CC(N)=O)C1)NC(=O)CC1CCC(=O)CC1 c1(C(N2CCC3(NC(CCC(N)=O)=O)C(C2)C3)=O)cc(F)cc2ccoc12 CC(C)S(=O)(=O)CC(=O)NC.C1CCN(C(=O)CN(CC(C)(C)C)C)CC1O CCC(O)C(C)C(=O)NCCC1(O)CN(C(=O)C(C)OC2CCCCC2)C1 N1(C(C2N(CCC)CCC2)=O)CCN(C)CC1CNC(=O)COCCO C(=O)(CCS(=O)(=O)C(F)(F)F)N1C(CNC(C23CC(C)C2C3)=O)CCC1 C(C)(CC(=O)C(F)(F)F)OC(c1sc(CC)c(C)c1)=O c1(CN2C(C)(C(=O)NCCC3N(C)CCC3)CCC2)ccc(N(C)C)cc1Cl C(=O)(C1=COc2ccccc2O1)N1CC(C)(NC(C(CC=C)C(C)C)=O)C1 C1(CNC(C2(C3CCC3)CC2)=O)CC(O)CN1C(=O)Cc1cc(Br)cs1 C(C(CCC)C(=O)NC(Cc1ccco1)CO)NC(C(C=C=C)C)=O C1(CNC(C2CS(=O)(=O)C2)=O)CC2(CCC2)CN1C(c1ccoc1Br)=O c1(C(N(CCCC#C)C2CC2)=O)cc2ccccn2c1 CC1OC(C)C(C(=O)NC2CCN(C(=O)CC3CC(C(F)F)C3)C2(C)C)C1C Cc1ncnc(N2CCC(N(C)C(C3CCOC3)=O)C2)c1C#N Cc1ccc2occ(C(=O)NC(CNC(=O)CC3CCCCO3)C(C)(C)C)c2c1 Cc1ncncc1C(=O)NC1C=CCN(C(C2(c3cccc(Cl)n3)CC2)=O)C1 C(C(C)(C)CNC(=O)CC1C=CCC1)N(C(=O)CCC1CC1(F)F)C N1(C(COc2c(OC)cccc2)=O)CCCN(C(C23CC(F)(C2)C3)=O)CC1C c1(C(=O)NC2CN(C(CC(=O)OCC)=O)C(C)C2)csc2ccccc12 C1(C(=O)NCC(C)CO)CN(C(=O)CNc2nccs2)CC(C)(C)C1 N#Cc1ccnc(NCC(=O)N(C2CC2)Cc2ccncc2)c1.N12CCC(C1)C2 N1(C(c2ccc(C3CC3)c(F)c2)=O)CCCCC2(CCN(C(C3(F)CC3)=O)C2)C1 C(=O)(C1c2ccccc2C2CC1C2)NCCN(C)C(C1CCS(=O)CC1)=O C(=O)(C(C)(C)CS(C)(=O)=O)NCC(CC=C)NC(=O)CCc1cscn1 C1(CNC(C(C)N(C)C)=O)CCN(C(=O)CCCc2cccc(Cl)c2)C12CC2 N1(C(CCC(C)(C)C)=O)CCC2CN(C(=O)C(c3ccc(Cl)cc3)O)CC12 c1(CC(=O)OCC)cccc(N)c1.C1CC=C(C)CC1.C(C)(C)C.C=O.N c1(C(N2C(C(N3CC(C)C3)=O)CCC2C(C)C)=O)cc(C)nc(O)n1.CS.C N1(C(CCC(CC)NC(=O)Cc2cc[nH]n2)=O)CC(CO)C(C2CC2)C1 N1(C(C2C3(CCN(Cc4ccc(C)s4)CC3)C2)=O)CCCC(C)(O)C(C)C1 c1(C(=O)NCC(CC(=O)NC(c2cn(C)nn2)C)O)ccc(=O)n(C)n1 c1(C(=O)NC(C)CCNC(=O)C(F)F)cc2sc(Br)cc2[nH]1 C1(CNC(c2ccnc(C)n2)=O)CC2CCCC2N1C(C12CC(C)(C1)OC2C)=O [SH](=O)(=O)c1ccccc1.N1(CCOC)CCCC(C(C)N)C1.[SH](=O)(=O)C1CC1 C(C)(CCCC(=O)NCC1OCCC1(C)C)NC(C(C)CC1CC1)=O Cn1cnc2c1CCCC2C(=O)N1CCOCC1CNC(=O)CNC(N)=O N1(C(C=NOC)=O)CCC(NC(c2coc(C(F)(F)F)c2)=O)CC1 n1(CC)cc(CC(N2CCC2CNC(=O)C)=O)c(C)n1.C1(C)CCCC1.O C1(C(=O)NCCCCOC)C(C)CCN1C(=O)Cc1csnn1 C(CC(=O)NC(C)(CNC(C1CCSC1)=O)C1CC1)SCCC CC1=CCC(NC(C2CC(CNC(c3ccc(Cl)s3)=O)C2)=O)CC1 C1(NC(c2ncc(CC)cn2)=O)CC(O)CN(C(C2CCC(CC)CC2)=O)C1 C1(CC)(NC(c2cc(CC(C)C)nn2C)=O)CCN(C(C2(C)C=CCC2)=O)CC1 C(CCC(C)C(=O)NCC#CCNC(c1sc(N(C)C)nc1C)=O)OC N1(C(c2n(C)ncc2[N+](=O)[O-])=O)CC(NC(c2nc(Cl)cs2)=O)CC2(CCC2)C1 CCCC(C(=O)NCc1cn(CC(C)NC(=O)C2=CCCO2)nn1)OCC CONC(=O)C(=O)NC(C)C(C)C(=O)NCCC1NC(=O)NC1=O n1(CC)cnc(C(C(=O)NCCC2(C)CC2)N(CC(=O)NC)CC)c1 C1(CN(C(C2N(C(C)=O)CCC2)=O)C)CN(C(=O)C(C)(C)n2ccnn2)CCO1 n1(CC=O)cc([N+](=O)[O-])cn1.C(C(F)(F)C(=O)NCCC1CCCC1)N(C)C c1(C(=O)NCC2CN(C(COCCOC)=O)CC2C)cc2n(n1)CCC2 c1(OC)nc(=Nc2ccsc2C(N2CCCC(C(N)=O)C2)=O)nc(OC)[nH]1 N1(C(c2cc(C)oc2C)=O)CC2(CCCN2C(c2cc(Cl)c(F)c(Cl)c2)=O)C1 C1(C(N(c2ccccc2)CC)=O)CCCN1C(=O)C(=O)Nc1nccn1C N1(C(c2cc(C)cc(Cl)c2)=O)CCC2(NC(C3CC(O)C3)=O)CCCC12 C(=O)(C(C)S(C)(=O)=O)N(CCN(C(=O)CC1CCC1(C)C)CC)C C1(NC(Cn2cc(C(C(C)C)N(C)C)nn2)=O)CCCCC1O.c1ccc(F)cc1 N1(C)CCCCCC1.c12cccc(c1)C(=O)N2.C(C(O)CO)N(CC(=O)N(C)C)C C(CC(=O)NC1CCC1NC(=O)Cc1cc(CC)no1)(OCC)OC c1(C(=O)NC2CCC(N(C)C(c3csnc3Cl)=O)C2)ccc2c(c1)NC(=O)CS2 CC1(NC(c2ccncc2N)=O)CCN(C(=O)CSCC(N)=O)C1 c1(C(=O)Nc2cc(OC)c(N3CCCCCC3)cc2)cnc2n1CCC(CN)C2 C#CC1(C(N2CCC(CN(C)CC)C2)=O)CCN(C(C2CCC(F)CC2)=O)C1 C(=O)(C1=NOC(C)(C)C1)N1CCC1.S(=O)(=O)(c1ccccc1)NC(C)C(=O)N Cc1c[nH]c(C(=O)NC2CCC2C)c1.C(=O)(CCCc1nc(C2CC2)no1)N c1(C=O)ccc(F)c(F)c1.O=C(CCn1ccnn1)NC.C1CN(C(=O)C)C1 C1(C(=O)OCC(=O)NC(=O)NCC)CCn2nncc2C1 C12(C(N3CCC(C(C)NC(=O)CCOC)C3)=O)CC3CC1C2C3.C1CC1 N1(C(C(CC)F)=O)CCCC(O)(CNC(c2nccn2C)=O)CC1 C1(C(N(CCC(=O)NC(C)(C)CC2CC2)CC)=O)CCC(C(N)=O)O1 c1(NC(C2CNCCN2Cc2ccc3ncsc3c2)=O)c(F)cc(Br)cc1Br N1(C(C(C)N)=O)CC2(C1)CN(C(=O)CC1CCC(C)C(C)C1)C2.Cc1cscn1 N1(C(C(C)NC(CC)(C)C)=O)CCN(C(=O)Cn2cc(C3CC3)nn2)CCC1C CC1CC(O)CCN(N2CCC(n3cnnc3)CC2)C1 C1(C(=O)NC)CCN(C(c2coc(CNC(=O)Cc3cn[nH]c3)n2)=O)C1C N1(CC(=O)NC(c2ccc(C(C)C)cc2)C)CC(N)CC(F)(F)C1 C12CC(C1)C(C)(C)O2.c1(C(C=O)(F)F)ncc(Cl)n1C.C(C(=O)N)=C(C)C N1(C(C(CC#C)O)=O)CC2CC1CN2C(=O)COc1ccc(CC#N)cc1 c1(CC(=O)Nc2ccccc2Oc2cccc(Br)c2)ccc(I)cc1 c12nc(cc(C)n1)OC1CN2C1.C1(CCC)CC(C(=O)OCCSC)CCO1 c1(C=O)cnc([N+](=O)[O-])n1C.CC1CCN(C(=O)CSCCC(F)(F)F)C1C N1(C(CC)=O)CCC(O)(C2CCN(C(=O)Nc3cccc4cn(C)nc34)CC2)C1 C(c1ccco1)=CC(N1CC(CN(C(=O)CSc2nnnn2C)C)C1)=O C(N=c1[nH]cc(Br)cc1C#N)C1(O)CCN(C(C(CC)CC(C)C)=O)CC1 N1(C(CC=CC)=O)CCC2(CCC(CNC(C3CC4CCC3CC4)=O)O2)CC1 Cc1cc(O)cc(C)c1C(N1CCC(C)C(CNC(c2ccnnc2)=O)C1)=O c1(OCC)cccc(CN(c2nc(-c3cnn(C)c3)cs2)C)c1 C1(NC(C(C)CC2CC2)=O)CN(C(=O)C=Cc2ccnn2C)CC12CCC2 CC(C)C1=NOC(C)(C(=O)NCCCC2CCCN2C(=O)COCCCF)C1 N1(C(CCC#CC)=O)CCN(C(c2oncc2CC)=O)C(CC(F)(F)F)C1 c1(C(=O)NC2CCC(C(N(CCC(C)(C)C)C)=O)C2)c[nH]c2ncccc12 C12(NC(c3n(C)nc(C(C)(C)C)c3)=O)CCCCC1N(C(=O)CC(C)(F)F)CC2 C1(Cn2cc(C(C)(C)C)nn2)CCCN(C(=O)C2CC2)CC1 C1(C(=O)NC2C(NC(=O)C=Cc3cscn3)CCC2)Cc2ccccc2CO1 N1(C(C(C)SC(C)C)=O)CCC2CCCC12C(N1CCC(N2CCC2)CC1)=O c1(C(=O)NC(C2N(C(C3C(C)C(=O)C3)=O)CCC2)(C)C)cc2ncccc2[nH]1 N1(C(C2C(c3cn(COC)nn3)C2)=O)CCC(C)(Oc2sccc2C#N)CC1 N1(C(C(C)OCC=C)=O)CC(O)CC1C=O.c1ccccc1.[SH](C)(=O)=O.N N1(C(C(=O)NCCCSCC)C2CC2Cl)CC2C(C)C2C1 c1(NC(=O)NC(C)CCC2CCCC2)nc(Cl)cn2ccnc12 C1(N(C(=O)C(C)(C)CNC=O)CC=C)CCC12CCNCC2.C(C)(C)C.O C1(NC(C2(NC(=O)CCC3CCCC3)CC2)=O)CC2(CCC2)C1O C1(C(N2CCN(C(c3c(C)scc3)=O)C(C3CC3)C2)=O)CS(=O)(=O)CC12CC2 CC(CC(F)(F)F)(c1ccccc1)NC(=O)C(F)F C(CC(C)C)(C(=O)NCCC(C)NC(c1ccc(CC(F)(F)F)cc1)=O)OC C12(C(=O)NCC(C)(C)C(N)=O)COCC1CN(CCC(c1ccccc1)O)C2 c1(C(=O)N)ccc(-c2nnc(C(F)F)o2)cc1.CC1CC2(C(=O)NCC)CC12 N1(C(c2c(OC)c(Cl)ncc2)=O)CCOCC(F)(CNC(c2cnn[nH]2)=O)C1 C(=O)(C(C(C)CC)c1ccccc1)NCC1(CNC(CC=C)=O)CCOCC1 C(C(CSC)Cc1cccnc1)N(CCN(CC)CC)CC N1(C(c2n(C)cnn2)=O)CCCC(C)(C)C1CNC(C12CCCCN1CCC2)=O c1(C(C)(C)C)cnc(CCC(=O)NCCCN(C(=O)CN(C2CCSC2)C)C)o1 C1(C(=O)NCC2CN(C(COCC)=O)CC2O)CSC(c2ccccc2O)=N1 C(=O)(C(C)C(F)(F)F)N(CC(CC)NC(=O)C=C(C)C(C)(C)C)C N#Cc1cc(-c2csc(NC(c3ccc(Cl)nc3)=O)n2)cc(F)c1 CC1CN(C(=O)CN(C)C)CC2(CCN(C(=O)C3CC3)C2)O1 C1(NC(CC2N(CC)CCC2)=O)CCN(C(=O)Cc2cc(C)on2)CC1 C=C(C)C1OCCC1C(N1CCC(C(=O)N)(CC)CC1)=O.C1(C(F)(F)F)CC1 CCCC(C)CC(=O)N1CCOCC(NC(C2CC3CC3CC2C)=O)C1 c1(C(=O)NC2CN(C(=O)C(F)F)C3(CCCC3)C2)c[nH]c2cc(F)c(F)cc12 N1(C(C2(C)CCC(C)C2)=O)CC2(CCC(NC(=O)COc3cccnc3)CC2)C1 C#Cc1cnn(C)c1C(=O)NCC1CC(NC(=O)C=O)C1(C)C.C1CC1 C1(CC(=O)N(CC)CC2CCN(C(=O)C(C)O)CC2)CC2(CCCC2)CO1 c1ccc2c(c1)OCCO2.CC1OCCC1C(N1CC(CCNC(=O)CS)C1)=O c1(C(N(C(C)CCNC(=O)C(O)C2CCC2)C)=O)ccc2c(c1)CCCS2(=O)=O C1(C(=O)NCCCSc2ccc(C)nc2)CC(O)CCN1C(=O)N(C)C Cc1c(C(=O)NCC(C)Cn2ccnc2)cccc1Br Cn1cnc2c(NC3CCSC(C)(C)C3)[nH]c(=NC3C4CCCC3CC4)nc12 N1(CC)CCOCC1C(=O)NCCc1ocnc1CNC(=O)C(O)C(C)C c1(CC(=O)N(CC)C)ccc(O)c([N+](=O)[O-])c1.C(C(=O)N(C)CC)=CCC c1(C(=O)NCC2(CNC(C3(O)CC3)=O)CC2)ncc2cc(Cl)ccn12 C1(CCNC(CCS(C)=O)=O)CN(C(=O)C=CC(C)(C)C)CCCO1 C1(C(N2CCCN(CC(=O)Nc3ccccn3)CC2)=O)CCc2nc[nH]c2C1 C#CCC(C)(C(=O)NC(c1cccc(O)c1)C)NC(=O)CC(C)CN(C)C N1(C(c2ccn(C)c(=O)c2)=O)CCN(C(=O)CCC2CC2(C)C)CC12CC2 c1(C=O)cc2c(cnn2C)nc1C(F)F.C(=O)(C(C)(F)C(F)(F)F)NCCC c1(C(N2CCC(CC=C)C2)=O)cc(C)nc2nc(C(F)(F)F)nn12.C(=O)C(F)F C(CC(=O)NOC1CCCCC1)N(C(C(CC)n1ccnc1)=O)C(C)C c1(CNC(C(C=C)O)=O)ccc(CN(C(=O)CCc2cccc(C)c2)C)cc1 c1(C(=O)NC2CN(C(C(CC(C)C)NC(C)=O)=O)C2)cc2c([nH]1)CCCC2 c1(OC)cc(N(C)C)ccc1CNc1cccc(Cc2ccccc2)c1 Cc1ccc(N)cc1C(N1CC(NC(c2n[nH]c(C3CC3)c2Cl)=O)CC1C)=O N1(C(C=CC(CC)C)=O)CCC2(C)CCCC12.N1(CC=CC=O)CCCC1.N C(CC(O)CNC(=O)CCC1CC1(C)C)NC(CNC(CCC)=O)=O N1(C(C=CC=CCC)=O)CC(C)CN(C(=O)C(Br)=C(C)C)C(C)C1 C1(C(=O)NCC(C2CCC2)OC)CCCCN(C(C2CCCC2C(C)C)=O)C1 N1(C(c2cnn(C)c2N)=O)CC2CCCC2(NC(c2ccc(C3CC3)cn2)=O)C1 N1(C(C2(N(C)C)CCCC2)=O)CCCCC(CNC(=O)CCc2cnc[nH]2)CC1 C1(O)(CCNC(C=CC(CC)C)=O)CCCN(C(c2nccc(OC)c2N)=O)C1 N1(C(c2c(O)ccc(N)c2)=O)CC2(COC(C)C2)C1.c1(CC=O)ccc(Cl)s1.N c1(N2CCC(C)(COC)CC2)nc2c(c(=NCc3ccc(F)c(Cl)c3)[nH]1)CSC2 c1(C(=O)NC(C2(O)CCC2)C)ccnc(CNC(c2nc(Cl)cs2)=O)c1 C1(C(=O)NCC(C)(C)O)CCC2CCC1N2C(c1ccc2[nH]ccc2c1)=O C(=O)(CCCCCS(N)(=O)=O)NC1CCN(C(COCC)=O)C1C1CC1 C1(NC(=O)CNS(=O)(=O)C2CC2)CC2CCC1CC2.c1(C=O)nsnc1O.N c1(CNC(C(C)OCCCC)=O)cc(C(=O)N(CCC)C(C)C)no1 C1(NC(c2cc(SC)oc2C)=O)CCN(C(c2ccccn2)=O)CC1CO c1(CCC)nc(CSc2csc(NC(=O)Cc3ccccc3)n2)no1 C1(OC)CC(C)C1.C1(C(=O)N)CC2(CC2)C1.c1(C=O)ccc(C2CC2)o1 C12(C(=O)NCC3N(C(CCC)=O)CCC3)CCC(CC1=O)C2 c1(C(N2CC(C(C(=O)NCC(CCC)C)O)C2)=O)ccc(NC)cn1 c1(OC)ccc(Cn2nnnc2C(CC(C)C)Nc2cnn(CCO)c2)cc1 N1(C(C2(CCNC(C3CC(C)N(C)C3)=O)CCC2)=O)C2CCC1COC2 C1(C(N(CCCCCNC(=O)C(O)Cn2cncn2)C)=O)CC2C=CC1C21CC1 Cc1n[nH]c(C)c1CCC(=O)NCC1CN(C(c2oc(CO)nc2C)=O)CC1C C(=O)(C(O)CC=O)NC1(CNC(C(C)=C2CCC2)=O)CC1.C(C)(C)C C1(F)(CNC(=O)Cc2ncsc2Cl)CCN(C(C2(CO)CCCO2)=O)CC1 c1(OCC)ccc(OCC(C(CNC(=O)C)(C)C)=O)cc1.C1CCCCC1.O Cc1ccc(-n2nnc(C(=O)NCCC(C)NC(=O)Cc3cn[nH]c3)c2C)cc1 c1(CCCN2CCC(N(CCC)C)C2)c(F)cccc1F c1(C(=O)NC2(CCOC)CCN(C(=O)C3=NOC(C)C3)C2)cccn2cnnc12 C(C)(C(=O)NCC(C)(C1CCC1)NC(c1snc(O)c1Cl)=O)(C(C)C)OC c1(OC)ccc(C)c(C)c1.CC(F)(F)F.C(=O)C.CC(C)N(C(=O)C)C.N C1(C(=O)NCC2CCN2C(=O)C(C)=O)(COC)C=CCC1 N1(C(Cn2c(C)cnc2)=O)CCCC2(CC(NC(c3coc(Cl)n3)=O)CO2)C1 CCC(N=c1[nH]c2c(c(=NCCCc3cc[nH]n3)[nH]1)CCCCC2)C1CCCO1 c1(CC)cccc(C(N2CCCC(N(C)C(C3C(Cl)(Cl)C34CC4)=O)C2)=O)c1 N(C(=NCc1ncnn1C)N1CCC2(CC1)CNC(=O)O2)CC(=O)NC(C)C c1(C(=O)NC2C(NC(Cc3n(C)nnc3)=O)COCC2)cc2ccccn2n1 Cc1cccc([N+](=O)[O-])c1N(C)Cc1cc(Cl)c(O)c(Br)c1 N1(C(C2(CC=C)CCC2)=O)CC(NC(c2cn(CC(O)CC)nn2)=O)CC1C C1(NC(CCSC)=O)COC2(C1)CN(C(=O)C(c1cccc(C)n1)(F)F)C2 Cc1cccn2cc(C(=O)NCC3CC3NC(c3c[nH]cc(F)c3=O)=O)nc12 CC1=C(C(=O)NCC2(O)CCCN(C(c3cc(F)ccc3N)=O)C2)CCO1 c1(C(=O)NCC2CN(C(C3(SC)CCC3)=O)CC2C)cc(C)n(C)c1C C(C(C)C(=O)N(CCNC(=O)C(C1CCOCC1)O)C1CC1)SC c1(C(C(=O)NC(C)CCCNC(c2nc(Cl)cs2)=O)O)ccc(C#N)cc1 C1(C(=O)NCC(COC)O)C=CCN1C(C1SCC=C1C)=O N1(C(c2c(C)nsc2C)=O)CCC2C(C(=O)N(C3CC4CCC3O4)C)C2C1 N1(C(CS(=O)(=O)NCC)=O)CCCCCC1C(=O)NCC(C)C(=O)OC c1(CCCC(=O)NCCC(O)CNC(c2ncoc2C2CC2)=O)ccc(F)cc1 C1(CC)CCN(C(=O)CC2CCN2C(c2ccc(COC)s2)=O)CCO1 c1(C=O)c(F)ccc(Cl)c1[N+](=O)[O-].C(CSC)(C(=O)N)OC.C1CC(CC)C1 COn1cnc(C)c1C(=O)N(CCCNC(=O)C(=O)N)C1CC1.CC(F)F O(NC(=O)C(CC1CC1)NC(=O)CC1(O)CCCOC1)C(c1ccccn1)C c1(OCC)nn(C)cc1NC(C1CCCCC1)=O.c1(C(C=O)C)ccccc1.N CC(C)C(F)C(=O)NCC1CC1CC(=O)NC1C(C)(C)C1(C)C c1(CC(=O)NC(C)CNC(=O)COC2CCC2)ccc2nc[nH]c2c1 C=CC1(C(=O)NCC2(O)CCN(C(=O)C(C)CC(N)=O)C2)CCCCC1 CCCCCCC1CC1.C(C)(C)(C=CC(N1CC(CC=O)C1)=O)SC.CCCC.N c1(C(=O)NCC(CC=C)NC(c2csc(C)c2C)=O)ccccc1OC(F)(F)F c1ccc(O)cc1C.n1(C2CC2)nnnc1C(C1COC(=O)C1)(C)CCC Cc1nc(CNC(C2(C)CC2(C)C)=O)oc1C=O.C(CC1CCC1)CO.N C(C1CCCCCC1)=CC(=O)NC1C2CN(C(C3C(C)OCC3)=O)C1C2 S(=O)(=O)(c1ccc(C#N)cc1)N1C2(CN(C(C=CC=CC)=O)C2)CC1 CCC(N=c1cc(C)nc(N2CC3OCCC3(CSC)C2)[nH]1)c1ccc(OC)cc1 C1CN(C(c2csc[n+]2[O-])=O)CC1C(F)(F)F.C1(C=O)CC(C(F)(F)F)C1.N CC1(C)COC(C(=O)NC2C=CC(CNC(c3cc(Cl)c(Cl)s3)=O)C2)C1 N1(C(COCCOC)=O)CC(C)N(C(c2ccc(C#N)cc2)=O)CC1C c1(C(=O)OC)c[nH]c(C)cc1=NC1CC(C)N(C(c2cc3n(c2)CCCC3)=O)C1 c1(C(C=O)O)ccc(Cl)cc1Cl.C(C)(C)(C)NC(CNC(=O)OCC)=O N1(C(CCNC(C2C(COC)CC2)=O)=O)CC2(CCOC(=O)N2)C1 C=CCC(CNC(C1CC1C(C)C)=O)NC(=O)C(C)(C)n1cnc(C)c1 N1(C(c2nc(C)sc2C)=O)CCCC(NC(c2ccc(C(N)=O)cn2)=O)C1C Cc1cc(C(N2CCC(O)(C(C)C)C2)=O)cc(F)c1.C1(C)(C)CS(=O)(=O)C1 c1(CC)cc(CC(=O)NC2CCCC(N(C(=O)CC3CC3)C)C2)n(C)n1 C(CCCCC(=O)NCCN(C1CCCC1)C(c1cc(Cl)sc1Cl)=O)OC C1(NC(C2CCC(NC(C(CCC)F)=O)C2)=O)C(O)C2CCCC12 Cc1c(NC(=O)N(CC(C2CCC(F)(F)CC2)O)C)cncc1Cl N1(C(C2C(C)(C)C2)=O)CCOC(C(=O)Nc2cc(-c3ccccc3)no2)C1 CC1(C)CN(C(c2cc(Cl)ncc2N)=O)C(CNC(=O)CC2(O)CC2)CO1 C(=O)(C1CCCc2nc[nH]c21)N1CC2=C(CN(C(=O)C=CCO)C2)C1 CCC(F)(F)CC(=O)NC1CCCC(C(=O)NC(C)CCc2cn[nH]c2)CC1 C1(C(=O)OC)CCN(C(C2(OC3(CNS)CCOC3)CC2)=O)C1 C1CCC2(CC1)CC2.N1(C(C(C)OCCOC)=O)CC(C)(C(=O)NC)C1 Cn1ccc2c(C(N3CC4CN(C(c5cccc(Cl)c5)=O)CC34)=O)cccc12 C1(NC(C(CC)C)=O)CC12CCN(C(=O)Cc1ccnc(Br)c1)CC2 C1(C(N2CC3CC(NC(=O)C4=CCOCC4)CC3C2)=O)CCn2c(O)nnc2C1 Cc1nc(CNC(C2COCOC2)=O)oc1C(=O)NCCC(C)(C)C n1(CC)ncc(C(=O)N(C)CC2CCN(c3nnc(C(C)C)o3)CC2)c1C N1(C(COCC)=O)CC2CCN(CC(=O)NCc3cc(C)cc(F)c3)CC2C1 C(CC(C(=O)NC1CC(NC(c2[nH]nnc2-c2ccccc2)=O)C1)OC)OC c1(C(=O)NCCN(C(=O)C(F)OC(F)(F)F)CC)cncnc1 C(N=c1ccc(S(C)(=O)=O)c[nH]1)C12OC(C)C(NC(=O)CCC(F)F)(C1)C2 N1(C(c2cc(C)cc(C)c2)=O)CCCC(N=c2[nH]c(Cl)c(C#N)s2)(CO)C1 c1(C(=O)NCC2N(C(C(CCCC)C)=O)CC(C)(C)C2)cc(N)c(F)cc1C N1(C(c2c(C)ccs2)=O)CCCC(CNC(c2cscc2C(C)C)=O)C1 O=C(C1=CSCCO1)NC12CC(NC(c3cnc(CC4CC4)s3)=O)(C1)C2 N1(C(CC(C(=O)OC)C)=O)CCC2(CC1)CC2C(=O)NC1CCCCCC1OC c1(N2CCC(C(N(CCCC)CCCC)=O)C2)nc(SC)ncc1C(=O)OC c1(C(N2C3CN(C(C)C)C(C3)C2)=O)nnn2c1CSCC2 C1(NC(CNC(CNC(C(CCC)F)=O)=O)=O)CCc2cnn(C(C)C)c2C1 C(c1ccc(=N)[nH]c1)=CC(N1CC(NC(CC2C(C)CCC2)=O)C1)=O CCC(C)(CNC(C1(CCNC(=O)CCC(C)C)CCCC1)=O)C(C)O C1(C(N2C(C)C(C(=O)NCc3nnc(O)n3C)CC2)=O)CCCCC1(C)C N1(C(C2(OC)CCCOC2)=O)CCCCC2(CCN(C(=O)CC(O)C(C)C)C2)C1 C(=O)(C(F)CC1CCCC1)NCC(CC)N(C)C(C1CC1OC)=O CC1CCC(NC(C2CCS(=O)(=O)N2)=O)CN1C(c1sccc1F)=O C1(NC(c2c(OC)ccs2)=O)CN(C(c2ccc(N)c(Cl)c2)=O)CC12CCCC2 Nc1cc(C(=O)NC2COCC2CNC(=O)Cc2c(F)cccc2F)cnc1Cl N1(C(CC)CC)CC(C(=O)NCCCNC(=O)C(F)=CC2CC2)CC1=O N1(C(c2noc(CC)c2C)=O)CC(CC(=O)NC)C2(CC2)C1.C1CCCC1(C)C N1(C(c2oc(CC)c(C)c2)=O)CCC(C(=O)NC(c2n[nH]c(C)n2)C)C12CCC2 c1(CC)nonc1C(N1CCC(C(C)NC(C2(COC)COC2)=O)C1)=O C1(C=O)CCCCC1c1nc[nH]n1.c1(C(=O)NCCOCC)ccc(Cl)o1.N N1(CC(N2CCC(C)CC2)=O)CCN(C(c2csnn2)=O)C(C)C1 N1(C(CC2C(CC)C2)=O)CC2CCCN(C(c3ccoc3Cl)=O)C2C1 C1(C(=O)OC)CC12CN(C(=O)C(C)CC1CC1)C2.c1(C=O)cnc(=N)[nH]c1 Cc1c(Cl)cnn1CC(N1CC(NC(c2ccc(Br)cn2)=O)C(O)C1)=O C1(C=O)COCC(C)O1.C1(CC(=O)N(CCC)CC)(C(F)(F)F)CCC1.N CCCC(C)(O)C(=O)N(C)Cc1ccc(C)cc1.c1(C=O)cc([N+](=O)[O-])c[nH]1.N Cc1ccc(Cl)c(C(N2CCCC(NC(c3cncn(C)c3=O)=O)C2C)=O)c1 C1(CNC(CC=CC)=O)CCCC2CN(C(c3sccc3CO)=O)CC12 C(=O)(CCC(CF)CF)NCCCCCC(=O)NCCC1(C)CC1(F)F C(=O)(C(C)(C)C(=O)N1CCOC(CNC(C2CCCC2(C)C)=O)C1)OCC c1(C(=O)NC2CC(C)CN(C(=O)C(C)OCCN(C)C)C2)cccc2c1OCC2 c1(NC(C23C4C5C6(C(N7CCC(N)C7)=O)C4C2C6C53)=O)cnc2ccccc2c1 C(=O)(C1=NOC2COCC12)N1C(C(=O)Nc2ccc(C#C)nc2)CC1C C1(NC(CC(=O)NCC)=O)CCN(C(c2ncncc2Br)=O)CC1O CC1CCCCC1CCNC(=O)N(CC(F)Br)C1CC1 Cn1ncc(CNC(=O)CCCC2CC2)c1C(=O)NCCCS(N)(=O)=O C1(C(=O)OC)CN(N2CC3(CO)CCOCC3(CO)C2)CC12CCC2 C(=O)(C(CC1CC1)NC(c1cocc1C)=O)N1C(C(=O)NC)CC1 N1(C(C(C)N(C(=O)COCC(F)F)CC)=O)CC2CCC1C(O)C2O O=C(CCc1ccc[nH]1)NCC(F)CNC(C1(n2cnnn2)CC1)=O c1(C(N(CC(C)(C)C)C)=O)cc2cc(Cl)ccn2n1.[SH](=O)(=O)CC=O.CCN n1(CC)nc(C(=O)NC2C3CN(C(C4CC(C)CCO4)=O)CC23)c(Cl)c1Br N1(C(=O)C=CCCc2ccccc2)CC2CCOC2(CNC(C2(Cl)CC2)=O)C1 c1(C(N2CC(NC(C3C(CC)OCC3)=O)C2)=O)c(F)ccc(OC)c1OC N1(C(C(C2CN(C(c3cc(C)nc(C)c3)=O)C2)O)=O)CC(=O)NC(=O)C1C C(c1cscn1)=CC(=O)NCCN(C(=O)C(F)n1cccn1)CC(C)O N1(C(CN(C)C)=O)CC2CC(CNC(=O)CSc3ccc(F)cc3F)C2C1 C(=O)(C(C)CN(C)C)N.CCCCN(C(C1CCC1C(=O)OC)=O)CC C1(OC)CN(C(c2c(Cl)c(C)nn2C)=O)C(C)(C(=O)O)C1 CC(CC(=O)NC(C)(C(=O)O)c1ccsc1)c1ccccc1 c1(C2C(NC(c3cncc(C)c3)c3nnnn3C)C2)ccc(F)c(F)c1 O=C1CC2C(CCCN2C(c2cc(CNC(=O)C(Cl)Cl)no2)=O)N1 C(=O)(CCCCC(N)=O)N1CC(C(=O)NCC(c2cnc[nH]2)C)C(F)C1 C(=O)(C1CCCc2nn[nH]c21)NCCOCCN(C)C(c1cc(CF)on1)=O N1(C(C(C(CC)O)C)=O)CCCN(C(c2ccc(F)cc2F)=O)C(C(C)C)C1 c1(C(=O)NC2CCC(C(=O)NC3CCNC3=O)CC2)cnc(O)nc1O CC(C)C(CCN(C)C(c1ccccc1OCCF)=O)NC(=O)C(C)N(C)C c1(CC(=O)NCC=C2CCN(C(CC3(C)CC3F)=O)CC2)ccnc(Cl)c1F C1(C2CCN(C)CC2)(C=O)CC1.CC(C(=O)NC(C)(C)CCC)S(C)(=O)=O.N c1(C(=O)NCCCN(CCCNC(c2c(C)c[nH]n2)=O)C)c(O)cc(Cl)cc1F C1(c2nccc(OC)c2)CCN(C(=NCCF)NCC(C)C2CCC2)C1 c1(C(N2CC(C)N(C(C3CC4CC3C3CC43)=O)CC2)=O)cn(C)c(=O)nc1O c1(-c2n(CCC=C)nc(-c3ccccn3)n2)cc2ccc(Br)cc2c(=O)o1 C(C)(C(=O)NNc1cc(C)nc(Cl)c1)n1cc(-c2ccc(OC)cc2)nn1 c1(C(=O)NCCC2CCC(NC(c3ccsn3)=O)C2)ccc2ncccn12 N12CCC(C1)OC(C)C1CC1C2=O.C(C(=O)NCC1CC1)=CCC C(=O)(C1=C(F)CN(C(c2cnc(OC)nc2)=O)CC1)NC1CCC(CCCC)C1 c1(C(N2CCC3CN(C(C4CC=CC4)=O)C3C2)=O)cc2c(=O)[nH]ccn2n1 N1(C(COCCCC)=O)CCC2CC2(C(N2CC=CC2CF)=O)CC1 N1(C(C(C)c2ccsc2)=O)CCCC(C(=O)N(C2CCCC2(F)F)C)C1 Cc1cc(C(C)C)ccc1C(=O)NCC1CCN(C(=O)C(F)CC(C)C)C1 c1(C(N2CC(C)C(NC(C3CCCCC34CCC4)=O)C2)=O)cccc2c1OCO2 C(C(CC(C)C)NC(c1ccc(N(C)C)nc1)=O)NC(CC1C(CC)C1)=O c1(N2C(C)CCC(NC(c3c(C)n[nH]c3)=O)C2)ccnc2ncnn12 Cc1ccc(C(=O)NCC2CCCC2C(=O)N)n1C.c1noc(C2CC2)n1.C N1(C(c2ccnc(OCC)c2F)=O)CCC2(CCCN2C(=O)C=C2CCC2)C1 CC1=C(c2cscc2C(N2CCC(n3cccn3)CC2)=O)CCCC1 C1(NC(Cc2cccc(OCC)n2)=O)CN(Cc2c[nH]ccc2=N)CC1(F)F C=CCC(C(=O)N1CC(NC(c2cnn3cccnc23)=O)CC(F)C1)C(C)(C)C N1(C(C(CNC(C2(C)CCCOC2)=O)OC)=O)CCCN(C(C)C)CC1 C#CC1CC2CCC1N(C(=O)C(n1cc(-c3ccc(OC)nc3C)nn1)C)C2 N1(C(CC2CC(C)(C)OC2)=O)CCOCC(CNC(c2cccc(CO)c2)=O)C1 Cc1cc(=NCCCC(c2ccccc2)NC(C2CC2C(C)C)=O)[nH]c(CO)n1 c1(C(=O)NCC2CC(NC(C3N(CC)CC3)=O)C2)cc2ccccc2o1 c1(CCCC)ccc(C(C(C)C)NC(N2CCC2C(N)=O)=O)cc1 C(=O)(C1CCCn2nccc21)Nc1cccc(NC(c2c(COC)ncs2)=O)c1 C=C(C)CC(C)C(=O)N(CC(O)CNC(=O)CSCCCc1ccccc1)C N1(C(c2cc(OC)cc([N+](=O)[O-])c2)=O)CCn2c(nc(C)c2Br)C1C CC1CC2(C(=O)NC3CC(C(=O)NC)C3)CC12.c1nnc[nH]1.c1ccccc1 C1(C(CC)C)CCN(C(c2cn(CCNC(c3cc(CO)on3)=O)nn2)=O)CC1 C1(NC(CCc2c(C)ncs2)=O)CN(C(C2CCCOC2)=O)CCC1CO Cn1cc(Br)c2c(N3CC4C(C(=O)Nc5cc(F)cc(F)c5Br)C4C3)ncnc12 N1(C(COC(C)=O)=O)Cc2ccccc2CC1CNC(=O)Cc1ccon1 CCC(COC)C(=O)N1C(C(=O)NCc2c[nH]nc2C(C)C)CC2CC12 C(=O)(C(C)(C)CNC(=O)C=CCNC(=O)CC(C)(F)F)NCC N1(C(C(c2cc(C)oc2C)C)=O)CCC2(C1)CN(C(=O)C(C)(C)F)CC(C)O2 c1(C(=O)NC(C2CN(C(c3c(Cl)cncc3Cl)=O)C2)C)csc2nccn12 N1(C(C(C(C)C)CN(C)C)=O)CCN(C(=O)Cn2ncn(C)c2=O)CC(O)C1 C1(OC)CCC(NC(c2n[nH]cc2CNC(c2cc(F)c[nH]2)=O)=O)C1 CCC(C(=O)NCC1CC(F)CN1C(C1CC(N(C)C)C1)=O)C(F)(F)F C1(C(=O)N)CN2CCN1CC2.CC1CN(C(=O)C=CCN2CCCC2)CC1CC N1(C(C(C(CC)C)NC(C)=O)=O)CCC(C)N(C(c2ccc(C(F)F)o2)=O)CC1 C(CC(=O)NCC1CCC1NC(=O)C(F)C1CCCC1)OCC#C Cc1scnc1C(=O)NCC1(O)CC(C(=O)NC(C)Cn2cncn2)C1 N1(C(=O)NCC2(OC)CCC(C)CC2)CCC(S(N)(=O)=O)C1 CC1CN(C)CC(C(=O)NCC2CC(F)(C)C2)O1.N1(CCC=O)CCOCC1 C(CN=C(NCC(C)F)NC1CC(=O)N(c2ccccc2F)C1)OCC c1(C(=O)NCC23C(CN(C(CCC=C=C)=O)C2)C3)ccc(C=NOC)cc1 c1(C(=O)N)cnn2ccncc12.C(=O)(CCCc1ccc(C)s1)N(C(C)C)CC C1(C(=O)NC2(CC=C)CN(C(c3ccc(OCC)s3)=O)C2)SC2C=CC1C2 N1(C(CCCOCCOC)=O)CCC(C(=O)NCc2c[nH]nc2C2CC2)CC1 C(=O)(CC(C)CC(C)C)N1CC(N(C(CCOCC(C)C)=O)C)C(C)(C)C1 N1(C(C(=Cc2cn[nH]c2)C)=O)CCC2(CNC(=O)O2)C1.C(C(=O)O)N1CC1 Cc1ccc(C)n1CCC(=O)NCC(CO)NC(C1CC(CC(F)F)C1)=O C(C)(CCC(=O)NC(CCC1CC1)C(=O)NCCc1nncn1C)SC Cc1c(Cl)c(C(N2CC3CCC3(NC(=O)C=Cc3ncc[nH]3)C2)=O)nn1C OCC(Cc1ccoc1)CN=C(NC1CC1)N1CCC2(CC1)CC2(F)F c1(OC)ccc2ccccc2c1C(=O)NC1CN(C(C23CCCN2CCC3)=O)C1 CN1CCC(C(=O)NC2CCCC(NC(=O)C(C)(C)C3CCCCC3)C2)CC1 C1(O)(C(N2CCC(NC(c3ccoc3)=O)C(O)C2)=O)CCc2ccccc2C1 CC(C)(CCCNC(C1CCCOCC1)=O)C(=O)NCC1C(CO)C1(F)F C1(NC(C2CC(CNC(c3n(C=C)ncc3)=O)OC2)=O)CCCN(C)CC1 C(=O)(C(CC(C)C)CC(C)C)N1CCC(NC(C(CC#C)C)=O)C1C1CC1 C=C(C)C(C)(C)C(=O)NCC(=C)CCNC(C1(OC)CCCC(C)C1)=O c1cnn(C)c1.C1(C(C)NC(=O)COC(C)(C)C)CCN(C(=O)O)C1 CC1=C(C(=O)NC(C)(C(=O)NCC2CC2C)C2CCC2)CCC1 C1(C(N(CCCC)CC)=O)CCC2(CCC2)OC1.c1(C=O)cc(=O)cc(Cl)[nH]1.N c1(C(C(=O)NCCNC(=O)CCC2CC2(Cl)Cl)O)ccc(O)c([N+](=O)[O-])c1 C(C)(C)(CCCCNC(C1CCC1C)=O)NC(CC(CC)C1CC1)=O C1(CNC(c2c(C)nc(=N)[nH]c2)=O)CN(C(c2cscc2Cl)=O)C(C)CC1C C1(C(=O)OC)C2CCC(C2)N1C(c1cc(OC)cc(C)c1)=O c1(CN(C)CCO)ccc(C(=O)Nc2cn(CC3CCN3)nn2)cc1 c1(CC(=O)NCC)c(Cl)cccc1Cl.n1(CC=O)cc(CC)nn1.C(N)=O Cc1c(C(=O)NCC2CCN(C(C3CCC(C4CC4)C3)=O)CC2)ccc(F)c1F c1(CC(N2CCC(N(C)C(c3ccncc3)=O)C2)=O)cccnc1C(F)(F)F C(=O)(C(CC1CCOCC1)NC(C12CSCC1C2)=O)N1C(C(C)O)CC1 c1(C(=O)NC2CC(N(C)C(=O)C3CC3)C2)cnn(C2CCCC2)c1C(F)F N1(C(c2cnc(S)[nH]2)=O)CC(C2CCCCN(C(c3cccnc3S)=O)C2)C1 c1(SC)cc(F)ccc1C(N1CC(CCNC(=O)Cc2nonc2C)C1)=O c1(C(N2CCC(NC(Cc3cc(C)sc3C)=O)CC2C)=O)ccn2ccccc12 Cc1ccc(CC(=O)NC(C)(C)CCNC(C2(C)CCCO2)=O)cc1Br CC(=C)C1CCOCC1.C(CCC(=O)CC=C)O.C12CC(C1)C(F)C(=O)N2 C1(CC)(NC(c2cnc(CO)nc2C)=O)CCN(C(=O)CC2CCCOC2)CC1 N1(c2nc(C)nc(O)c2)CC(NC(C2(O)CCC2)=O)C2CCCCC12 C1(C(=O)NCC(CCC)(C)C)CN(C(C2(C)CCC(=O)C2)=O)CCN1C c1(NC)ccc(C(N2CC3C(NC(=O)C#CC4CCCO4)C3C2)=O)cc1[N+](=O)[O-] CC1(CNC(=O)NCC2(C(c3ccc(F)cc3)O)CC2)CCCCC1O c1(OC)nccc(C(=O)NC(c2cccnc2)C(=O)NC)n1.C1CC2C=CC1O2 Cc1ccc(C(N2CCOCC2CC(=O)N(C)CC2CN(C)CCO2)=O)nc1 C(=O)(C1CCCc2ncnn21)N1CC(C)C(CNC(C2(C)CNC(=O)C2)=O)C1 C(C)(c1ccccc1Cl)=CC(N1CCC(N(C(=O)C(C)CCOC)CC)CC1)=O c1(C=O)c(C)cc(C)oc1=O.C(C(=O)N1CCC(F)(F)C1)(C(C)(C)C)SC.C n1(CC=C)nc(C(C)CCC)nc1-c1ccc(C(F)(F)F)nc1 c1(C(=O)NC(CCN(C(CC(COC)C)=O)C)C)cc(Cl)ccc1Br c1(C(=O)NCC2(NC(CCC(C)N(C)C)=O)CCOC2)ccc2c[nH]nc2n1 n1(CCCC)nccc1C(=O)NC(C)(C)CC.C1(C=O)CCCN1C(C)=O.N C1(CC=C)(NC(C2C=CCN2C(=O)CC2(N(C)C)CCC2)=O)CCCCC1 Cc1nc(NC(=O)NCC(c2nc(C3CC3)no2)O)sc1F C1(C(N2CCN(C(c3ccccc3I)=O)CC2)=O)CCC2CNCCN12 C1(C)(NC(C(C)O)=O)CCCN(C(=O)Cc2ccn(C)c2)C1 Cc1csc(C(F)(F)C(=O)N2CC(N(C(=O)CCCn3ccnn3)C)C2)n1 c1(C2C(C(N3CCC3)=O)C2)cccc(F)c1F.c1(C(=O)N)ccc(C(F)F)cc1 N1(C(c2cnc(C)n2C)=O)CCCC(C)(NC(=O)C(C)C2CCOC2)C1 C1(NC(c2n(C)ncc2)=O)CN(c2nc(-c3cccc(Cl)c3F)ns2)CC1(C)C C1(CC(=O)N(C(C)CS(C)=O)C)CC2(C1)CN(C(=O)CCc1cn(C)nn1)C2 c1(SC)cnc(N2CCC(C(C)C(=O)N(C)Cc3cccnc3)CC2)nc1 N1(C(C(CCCNC(C(C)(C)NC(C)=O)=O)O)=O)Cc2ccncc2C1 N1(C(c2ncn(C)n2)=O)CC2CC1CCC2NC(c1ccnc(C(N)=O)c1)=O C(=O)(C1(C)CCc2ccccc21)N1CC(NC(c2ncc(C)cn2)=O)C1 Cc1ccc2nc(N3CCCC3CN(C(=O)Cc3cncnc3)C)sc2n1 Cc1ccc2c(c1)CCC(C(=O)NCCN(C(=O)CC13CCC(CC1)CC3)C)O2 C1(NC(C(COC)(F)F)=O)CC(O)CN(C(=O)C(C)(C)COCC(F)F)C1 c1(OC)cnc(F)cc1C(=O)NCCC(C)NC(C1CC(C)C1)=O C1(NC(c2cn(C)c(O)n2)=O)COC2(CCN(C(c3ccc(N)c(O)c3)=O)C2)C1 CC(CNC(C1(C2CC2)CC1)=O)C(F)C(=O)NCc1cccnc1F C1(NC(C(C)=C2CCCC2)=O)CCCN(C(=O)CC2CCCC(C#N)C2)CC1 C1(NC(=O)C=Cc2cocn2)CC2CC(NC(c3nccc(Cl)c3Cl)=O)C2C1 C(=O)(CC(O)CC(C)(C)C)N1CC(CC)C(NC(=O)C)CC1.c1cc(C)on1.O CCCCCC(O)CC(=O)NCc1cc(C(=O)NC(C)COC(C)C)n[nH]1 C(=O)(C(C)CC(=O)NCC1(CC(=O)NCCC(C)C(F)(F)F)CC1)OC C1(NC(=O)CCCNC(c2cncc(C3CC3)c2)=O)C=CCCCC1 N1(C(C)=O)CCc2c(CNC(=O)COC3CCCC3)cccc2C1 c1(C(N2C(CNC(CC=C(C)C)=O)CCCC2)=O)cc2c(C)ccc(C)c2[nH]1 C1(CNC(c2ccc(F)s2)=O)CCCN(C(C2CCS(=O)(=O)N2)=O)C1 C1(N(C(CCOCCN(C)C)=O)C)CCCN(C(=O)CCSc2nnnn2C)C1 c1(NC(C2COCCN2C(=O)CCOC2CC2)=O)ccc2n[nH]cc2c1 c1(OC)ccc(O)cc1C(N1CC2CC(NC(=O)C(c3ccccc3)O)C1C2)=O C(CC(C)C)(C(=O)N1CC(NC(=O)C=CC2CCOC2)CC(O)C1)OC C1(CC(=O)N(CC(=O)NC(C)CCSCC)CCOC)CCSC1 c1(OC)ccc(CC(=O)NC2CC2CNC(=O)CN2CC=CC2)cn1 c1(C(=O)NCC(C)NC(=O)Cn2cc(Cl)cn2)nccc2ccncc12 n1(CC(=O)NCCCN(C(=O)CC2CC2)CC)nc2ccccn2c1=O.C N#CCCCCCC(=O)N1CC2CC2C1C(N1CCCCC1CCCO)=O C#CCC(O)C(=O)N(C(C)C(N1CCCC(CC2CC2)C1)=O)C C1(NC(C2CC23CCOC3)=O)CCN(C(=O)CN2CCCC2=O)CC1F N1(C(CN(C(=O)CCC2CC2(C)C)CC#C)=O)CCCCC1CC=C C=CC(C)(O)C(=O)N(C1CCC(NC(=O)C=Cc2ccccn2)CC1)C c1(C(=O)Nc2cc(C)cc(O)c2)sc2cc(C3=CCC(O)CC3)ccc2c1O c1(C(=O)OC)cncc(C(N2CC(NC(c3cnc(C)o3)=O)CCC2C)=O)c1C c1(C(N2C(C(N(C(CCCC)C)C)=O)CC2C)=O)cc(C)sc1C C(=O)(C1=NOC2(CCC2)C1)N1CC(C(=O)NC2(C)CCCC2)OCC1 c1(C(N2CC3C(CNC(C(CC)C)=O)C3C2)=O)ccc2nnn(O)c2c1 C1(C(=O)NCc2nc(COC)[nH]n2)CN(C(=O)CP(C)(C)=O)CC1(F)F N1(C(=O)NC(CC)CCOC)CCC(C(F)C(N)=O)CC1 C=CC1CCN(C(=O)C(C)(C)CN(C)C(C2CCOC2)=O)C1 N1(C(c2n[nH]cc2C2CC2)=O)CC(CNC(C2(O)CCC2)=O)C(F)(F)C1 Cc1ccc(CC(N2CC(NC(c3ccn(CCF)n3)=O)CC2C)=O)c(Cl)n1 N1(C(C2(C)CC(=C)C2)=O)CC(NC(=O)Cc2cccc(CO)c2)CC(C)C1 C=CC(C)CC(=O)NCc1ncccc1C(=O)NC1CCN(CCF)C1 c1(C(=O)NCC(C2CC2)NC(c2nc(C)sc2)=O)cnc(N)c(O)c1 CCCCC(C(=O)NC(CC)(CC)CCNC(=O)C)N(C)C.C(=O)C(C)CC.N N1(C(CNC(C(C)NC(C2CC(F)(CF)C2)=O)=O)=O)CC2CCC1C2 CCC(C)N(OC)C(=O)C1CCCC(C)(C)CC1 C1(C(N2C(CC(=O)NC)CC2)=O)CCN(C(=O)CSCC(F)F)C1(C)C CC(=Cn1ccnn1)C(=O)NC1CCN(C(=O)C=Cc2ncc(C)[nH]2)C(C)C1 C1(NC(c2cn(-c3cccc(Cl)c3)nn2)=O)CCCN(C(c2cc(Br)co2)=O)C1 C1(C(=O)NC(C(C)C)CCO)C2CCC(C2)C1NC(C12CCCC1OCC2)=O N1(C(CNS(CC)(=O)=O)=O)CCC(NC(=O)C(C)NC(=O)NC)C1(C)C C1(CNC(=O)CS(=O)(=O)N2CCCCC2)CC(F)(F)CN1C(C1CC1F)=O c1(C(=O)NC2CCN(C(Cc3cnc(C)[nH]3)=O)C(C)C2)cc2occc2n1C N1(C(C2C(C)(NC(CC=CC=C)=O)CCCC2)=O)CCC2(CCN(C)C2)C1 c1(C(N(CCCN(C)C(C2CC(CN(C)C)C2)=O)C)=O)cc(C#N)c[nH]1 C#CCCC(=O)NC(C(=O)N(C)CC1CCSC1)C1CCCO1 c1(SC)cc(CN=C(NCc2ccc(C)nn2)NCc2cccs2)ccn1 C(CCN(C(=O)CCn1cncn1)C)(C(C)C)NC(C1ON=C(C)C1)=O C(=O)(C#CC1CCCCC1)N(CC(C)(C)NC(c1cc2cccnc2[nH]1)=O)C c1(C(N(CCN(C(C)C)C(C2CC2C)=O)C)=O)cc2sc(Cl)cc2s1 c1(C(=O)NC2CC23CC(NC(=O)C(O)c2ccsc2)C3)cc2ccccc2s1 N(C1C(=O)Nc2cccc(Cl)c21)C(=O)NCc1c(OCCOC)nccc1 C1(C(=O)NCC(C(C)C)NC(C2SCCS2)=O)(CN)CC12CCC2 c1(CC(=O)OC(C)(C)C)ccc(NC(C2COC(Cn3cccn3)C2)=O)o1 c1(N2CCC(NC(c3cc(Cl)nc(Cl)c3)=O)(CF)C2)ncnc(O)c1Br C(C(CCO)NC(=O)CC1(NC(C2SCC=C2C)=O)CC1)OC C(=O)(C1CCCc2sccc21)NC1C2(CN(C(C3CCCN(C)C3)=O)C2)CCC1 c1(C(=O)NC2(C)CCCC2)cncc([N+](=O)[O-])c1.C1(C=O)CC=CC(O)C1.N CCCCC(CNC(c1cc(C2CC2)nn1C)c1nnnn1CCSC)CCC C1(NC(CCCC(N)=O)=O)CC1C1CCCN(C(=O)CCSc2ccccn2)C1 c1(NC(c2ncc(Cl)cc2Br)=O)cnc2c(c1)CN(Cc1scc(Br)c1Br)CC2 c1(-c2c(OC)ncc(C(N3CCC(=O)C(C)C3)=O)c2)cc(Cl)c(O)c(Cl)c1 N1(C(C2CC(C#C)(O)C2)=O)CCCCC2C1CCCN2C(=O)CC(C)=C=C N1(C(c2c(C)nc(CO)s2)=O)CC2CC(N=c3[nH]nc(C)s3)C2C1 c1(CC(=O)NCC(CNC(CCC=CC)=O)OC)ccc(Cl)nc1 N1(C(Cn2ncc(C#N)c2)=O)CCCC2(CC(NC(=O)Cn3cncn3)CO2)C1 c1(CC(=O)NC(c2nc(C(C)(C)C)no2)C)cc(Br)cnc1F c1(NC(CCCSC)c2nnnn2C2CCCCC2)ccc(C(N)=O)c(F)c1 CC(C)(C#N)CCCC(=O)N1CCC2CC2(C(N2C3COCC2C3)=O)CC1 c1(CC(=O)N(CC(CC)NC(=O)CN2CC(C)(OC)C2)C)ccc(C)nc1Cl C1(C(=O)N(CC(C)C)C)(OC(C)C)CCOC1.C1(C(=O)N)(C(N)=O)CC1 Cc1cc(=NCC2(C)CCN(C)CC2)[nH]c(N2CCC(F)(F)C(C)C2)n1 CCCC(C#N)C(=O)N1CC(NC(=O)CCn2cccn2)C(c2cncn2C)C1 C1(CNC(C(CC#C)CC#C)=O)CCCC2(CCN(C(C3CC3C#N)=O)CC2)O1 c1(COC)nc(N(C)CC2CCN(C(=O)CC3OCCC3C)C2)cc(C)n1 C1(NC(c2c(C)nc(COC)s2)=O)CN(C(=O)CCC(C)SC)CC1C1CC1 c1(N2CCCC(C)(NC(c3cc(CF)on3)=O)C2)ncnc2scnc12 C1CC2CCC(C1)N2C(=O)C=C(C)Cl.C1(C=O)(COCC)CCC1.N c1(C(=O)NC(C)Cc2cnccn2)ccncc1N=[N+]=[N-] c1(C(N(CCC(C)NC(CC=C)=O)C)=O)cnc2c(c1)CCCO2 c1ccc(Cl)cc1.C1(C#N)(C(N(C)CC2(NC(=O)CC)CC2)=O)CCCO1 CC(O)C(C(=O)N1CCC(C(C)(C)NC(=O)CN2CC3CC3C2)CC1)N(C)C C(N=c1nc2sccc2c(NCc2ccnnc2)[nH]1)c1cccc(C)n1 c1(C(N2CCC(SC)CC2)=O)cn2c(n1)CN(C(c1c(I)ccnc1F)=O)CC2 C1(O)(CC(=O)NC(C(=O)NC(C#C)C)CSCC)CCCCC1 N1(C(COCCC)=O)CC2(CC2)CC1CNC(=O)CSCC(N)=O C1(NC(Cc2n(C)ccc2)=O)CCCC(C(N2CCOC3CCC23)=O)CC1 N1(C(c2nccc(C#C)c2)=O)CCC2(CCC2NC(=O)CCOCC)CC1 C1(NC(C(CCCC)C)=O)C(C)CCN(C(c2cc(C)sn2)=O)C1C Cc1nnc2n1CC(C(=O)NC1CCC(NC(=O)C=CSc3nc[nH]n3)CC1)C2 c1(SCC(=O)OCC)nc(CSc2ccc(C(C)(C)C)cc2)nn1C c1(NC)ccc(C(N2CC(NC(C3CCOC(C)(C)C3)=O)CC(F)C2)=O)c(Cl)c1 CC(CC(=O)N1CC(C)CN(C(=O)CN2CCC(F)(F)C2)CC1C)C(C)(C)C CC(C)(C)C(CO)C(=O)NC1(CO)CCCN(C(c2c[nH]cc(Cl)c2=O)=O)C1 C(=O)(C1=NNC(=O)CC1)NCCOCCNC(C1C(SC)CCC1)=O N1(C(C2C(CC)OCC2)=O)CCN(C(C2CCC3CC3C2)=O)CC1 c1(OCC)cccc(CC(=O)NC2CCCC(NC(=O)C(F)=C(C)C)C2)n1 CC1(C)OCC(CCC(N2CCN(CCCNC(=O)C=CCF)CC2)=O)O1 c1(C(=O)NC2(CNC(c3cc(C(N)=O)[nH]c3)=O)CCOC2)n[nH]c2c1COC2 C=CC(CC)CC(=O)NC12CC(CNC(=O)Cc3cccc(C)c3)(C1)C2 c1(C(N(CC(CNC(CCCC(C)=O)=O)(C)C)C)=O)cc(F)c2nc(C)cn2c1 C(=O)(C(C)(C)CCC#N)N1CC(C)(CNC(CN(CCOC)C)=O)OCC1 N1(C(COCCOCC)=O)CCOC(C(=O)NC(C)(C)C(C)O)CC1 C1COCCN1C(=O)C(C)Cc1ccc(F)cc1.c1(CC)cc(C(=O)NC)no1 C1(C2(O)CCC2)(CNC(CC2N(C(CCC=CC(C)C)=O)CCCC2)=O)CC1 N1(C(CCN(C(CC2C(C)(C)CCO2)=O)C2CC2)=O)CCc2cncnc2C1 CC1CC(C(=O)N(C2(CC(N3CCCC34CC4)=O)CC2)C)=NO1 CCCC(C=O)N1CCN(C(=O)OC(C)(C)C)CC1.C(=O)(C(=O)N)NCC C1(CCNC(C2(NC(CCOCCOC)=O)CC2)=O)COC(C)(C)C1 c1(OC)cc(F)c(NC(=O)COCC2CCC2)cc1Cl N1(C(CC(=O)N(C)C)=O)CCN(CC(=O)NCC2CC2)CC1 c1(C(=O)NCCCC2(NC(Cn3c(C)ccc3C)=O)CC2)cccc2ccoc12 N1(C(COCCC=C)=O)CC2CCC2(NC(C2CCCN2C(=O)CCC)=O)C1 c1(C(N(C2CCCN(C(=O)C(F)C(F)(F)F)C2)CC)=O)ccc(OC)cc1O C1(NC(c2nnn(CC)c2C)=O)COC2(CCCN(C(c3cc(C)no3)=O)C2)C1 Cc1nc(=NC(=O)C2(F)CCN(C(c3n[nH]c(C)c3C)=O)C2)s[nH]1 c1(CCC=O)ccc(O)nc1.C1(CNC(C=C(C)C(C)C)=O)CC(F)C1.C c1(NCC2(C(C)(F)F)CC2)[nH]c(=NCC2COC(=O)N2)nc2sccc12 c1(C(N2C(C)CN(C(=O)C=CC3CCCO3)CC2)=O)cccc2scnc12 N1(C(c2ncnn2CCF)C(=O)NCCOC)CC2CN(C)CC2C1 Cc1cc(F)ncc1C(N1CCC(CC(N2CCC(C(F)(F)F)C2)=O)C1)=O O=c1ccc2cc(S(=O)(=O)N3CCCC(C4CCO4)C3)ccc2[nH]1 N1(C(CNC=O)=O)CCN(C(C2(c3cc[nH]n3)CCC2)=O)CC1c1cccnc1 c1(C(=O)OC)ccc(Cl)cc1S(=O)(=O)N(C)Cc1nc2c(s1)CC(C)CC2 C12(C(=O)OC)COC(C=O)(C1)C2.C1(=C(C=O)F)CCCCC1.C1CCC1.N C1(NC(CCN(C(=O)Cc2ccns2)C)=O)CCOC12CCOC2 c1(C(N(C(CC)CC)C)=O)cc(CNC(C2CCC2(F)F)=O)nn1C N1(C(C(C)n2cnnn2)=O)CCC2(CC1)CN(C(C1CC(O)CN1)=O)CCC2O Cc1[nH]c(C(N2CCC(C(C)NC(c3ccnc(C4CC4)c3)=O)C2)=O)c(C)c1C c1(C(=O)NCC2CCN(C(CC(COC)C)=O)C2)cc2ccc(Br)nc2[nH]1 C1(C(=O)NC2C(NC(c3c(CC)noc3C)=O)CCC2)CC2COCC2C1 O=C(O)CC(CNC(=O)Nc1ccns1)c1ccccc1 C1(NC(c2c(C)nn(C(C)C)c2)=O)CCC(O)CN(C(=O)CC23CCCC2C3)C1 c1(C(=O)NCC2N(C(CCCN(C(=O)OC)C)=O)CC2)ccc2ocnc2c1 N1(C(C(C)=O)=O)CCC(F)(C(=O)NCCc2cccs2)C1 c1(C(N2CCC(c3nncs3)C2)C(=O)NC2COC2)cc([N+](=O)[O-])sn1 N1(c2n(C3CC(CC#N)C3)nnn2)CCC(O)(C2CCOC2)CC1 c1(C(=O)NCCC2CCCN(C(c3cnn(CC)c3C)=O)C2)ccc(C)c(Cl)c1 c1(C(=O)OCC)ccccc1Cl.C1(C(=O)N)C2CN(C=O)CC12.C(C)(C)C c1(C(=O)NC2CCCC2NC(=O)C(O)CC2CCCC2)cc2ncccc2o1 N1(C(c2cc(OC)no2)=O)CC=CC(NC(=O)CC=C(Cl)Cl)C1 Cc1cnc(C)c(C(=O)NC(C2CCCN2C(=O)CC2OCCOC2(C)C)C)c1 C1(CNC(C(CC)F)=O)CCCC12CCN(C(c1sccc1C)=O)CC2 C1(CCC#C)CCCN(C(=O)C(C)N(C(=O)CCC(=O)NCCC)CCC)C1 C(C(C)(C)C(=O)N(C1CCN(C)C1=O)C)NC(CCN(C1CCCCC1)C)=O Cn1ncc(C(=O)NC(CNC(C2CC(N3CC(O)C3)C2)=O)C2CC2)n1 C(CC(C)C(F)(F)F)NC(C(CN(C(CCCC)=O)C)C)=O CCCCC(O)CC(=O)N1CC(NC(c2cnc(Br)s2)=O)C(O)C1 c1(C(=O)NC(CC)CNC(c2n[nH]c3cccnc23)=O)nccc2ccncc12 c1(C(=O)NC(C)C(N2CCC(O)C2C)=O)cc(O)cc(F)c1 c1(OC)cc(C(=O)NC(C2(O)CN(C(=O)CCc3nc[nH]n3)C2)C)cnc1.O N1(C(c2cc(CC)n(C)n2)=O)CCC2CCC(C1)N2C(=O)C(C(C)C)OC C(=O)(C(O)C1CN(C(=O)COc2ccsn2)C1)NCC1(CCC)CC1 N1(C(CC=CC=C)=O)CCN(C(=O)C(C2CCCOC2)OCC)CC1C N1(C(c2cc(C)nc(C)c2)=O)CC2(CCCC2CC(N2CCCCC(O)C2)=O)C1 C(C1=NOC2CN(C(C3CCC=CCC3)=O)CC12)NC(c1ccc(C=C)cc1)=O c1(OC)ccc2c(c1)OCC2CC(=O)N1CCCc2c(F)ccc(Cl)c21 C1(C(=O)O)(CC)CCCN1C(=O)CC1CCN(C)CC1.c1cccc(C(C)C)c1 C1(NC(CCC(=C)C)=O)CC2CCC(C1)N2c1nc(-c2cc(Cl)cc(Cl)c2)no1 N1(C(C(c2ccccc2Br)NC(CNC(N)=O)=O)=O)CC=C(CO)CC1 C1(C(=O)NCC=CCNC(C(CCOC)C)=O)CC2(CCC2)CCO1 C=C=CC(C)C(=O)NC1(CN(C(=O)CCc2cccnc2C)C)CC1 C(=O)(CC(C)OC)N(CC(CC)NC(=O)CCc1ccc[nH]1)C C(CC(C(=O)N1CCC(CCF)CC1)NC(c1ccc(N)cn1)=O)OC C=C=CC(C)C(=O)N1CCC1CNC(c1ccnc(OC(F)(F)F)c1)=O c1(C(=O)NCC2C3CC2N(C(=O)Cc2ccns2)C3)[nH]cc2c1CCCC2 C#Cc1ccc(C(N2CC(C)(C)CC2CNC(C2CCN(C)CC2)=O)=O)cn1 CC1CN(C(c2ccc(CN(C)C)s2)=O)CC1CC.C(=O)CCC1CCCO1.N c1(C(C)C)ncc(Br)c(NC2CC(NC(=O)CC(C)c3ccccc3)C2)n1 CC(C)C(C(F)(F)F)NC(C1CCCCCN1C(=O)CN1CCCNC1=O)=O c1(OC)cccc2c(C(N3CCCC4(CCN4S(=O)(=O)C(C)C)C3)=O)cncc12 C1(C(=O)NCC(C)N(C)C(C2(CF)CC2)=O)CCCN1CC(F)(F)F c1(OC)ccc(NC(=O)CC2CC(O)CN2C(c2cnn(CCF)c2)=O)cc1C C(C(CO)(CO)NC(c1cnc(Cl)s1)=O)N(C(C(C)n1cncn1)=O)C C1(NC(c2c(C)cc(F)s2)=O)C2COCC1CN(C(c1cccc(C)c1C)=O)C2 C(c1ccc2c(c1)CCO2)=CC(=O)NC1CCN(C(c2cc(Br)co2)=O)C1 C(=O)(C(C#N)C(C)C)N1CCC(NC(c2nc(C(F)(F)F)sc2C)=O)CC1.CC CC(C)C(CNC(=NCCN1CC2CC2C1)NC1CCS(=O)(=O)C1)C(C)C C(C(O)(CNC(C1CCCCN1C(c1cc(O)nn1C)=O)=O)CO)OC CC1C=C(C(=O)NC(C)(Cc2ccccc2)C(F)F)C1 c1(C(=O)NC2CCCN(C(CSCC(C)C)=O)C2C)cccc2oncc12 C1(CC(=O)NCC(C)Cc2cn[nH]c2)CN(C(C2CCC(=O)NC2)=O)CCO1 C#CC1(C(=O)NCC2CC2)CCCC1.C(CC(C)(C)C)N(CCC(=O)N)C c1(NC(c2c(-c3ccn(C)n3)cccn2)=O)cc(F)cnc1Cl CC(CC(=O)NC1CCN(C(c2cc(C(N)=O)c[nH]2)=O)C1)c1ccccc1 C1(CC(N2C(CC)CCCC2)=O)CCN(C(=O)C=Cc2ccc[nH]2)C1(C)C C1(NC(Cc2c(C)non2)=O)CN(C(=O)Cc2noc(C)c2C#N)CCC1CO C1(NC(C2CC=CC(NC(c3c(C)nn(C)c3)=O)C2)=O)CCCC2(C1)N=N2 n1(Cc2n(CCCC)nc(-c3cc(C)oc3C)n2)nc(C)c2ccccc2c1=O Cc1ccc(CNC(c2ccn(C)c2)c2nnnn2C(C)(C)C)c(F)c1F C1(c2nnnn2-c2cccc(OC)c2)(NCCCC)CCCCC1N(C)C Cc1nc(NCCC2CCCC(C)C2)cc(=NCc2cncc(C(F)(F)F)c2)[nH]1 c1(NC(c2csc(=NCc3ncc(Cl)cc3Cl)[nH]2)=O)nc(Cl)ccc1O c1(OC)ccc(CC(N2CCC(NC(C34CC(C)(CO3)C4)=O)C2C)=O)cc1O N1(C(CCCOCCC)=O)CC(C(=O)N(C)CC2(CO)CCC2)CC(C)C1 c1(CC)ccc(C)c(C(=O)N(C(C)CC)C)c1.c1(C=O)ncn(C(C)(C)C)n1 Cc1cc(F)c(C(=O)N(CC(C)NC(=O)CCN2CCCCC2)C)cc1F C1(C(=O)O)CCCC2(CN(Cc3cc(F)c(F)c(F)c3F)C2)O1 N(C1CCc2c(Br)cccc21)C(=O)C(N1CCCCC(CO)C1)=O C1(NC(C(C2CCCCC2)C)=O)(CO)CN(C(=O)CCc2ccccc2)C1 N1(CC)CCN(C(C2CCCN(C(=O)C3=C(C)CC3)C2)=O)CC1C N1(C(C2CCN(CC(C)C)CC2)=O)CC2CCCC(NC(C3C=CCC3)=O)(C2)C1 c1(CC(=O)N)ccc(Br)c(O)c1.C1(OCC)CC(C(=O)N(C(C)C)C)C1 c1(CC)ccccc1C(=O)N(CCC(N1CC2CC1CS2)=O)C1CC1 c1(C(N2CCCC(N(C(C3CC4CC4C3)=O)CC)C2)=O)cnc2n(c1=O)CCS2 C1(C(N2C(C)CNCC2)=O)CCC2(CCN(Cc3ccnc(Cl)c3)CC2)C1 C1(C(=O)N)(COC)CCOCC1.C1CCCCN1C(=O)C(n1ccc(C)n1)C.C C#CCCC(C(=O)N(C1CCC(C)(C)C1)C)NC(c1nc(Cl)cs1)=O C1(NC(C2(CC#C)CC=CCC2)=O)CC2CCC1CC2NC(C1(C)CC1F)=O c1(C(=O)NC2CCC(CCNC(c3cc(C#N)oc3)=O)C2)ccn2nccc2c1 C1(CNC(C(C)=CC2CC2)=O)CC12CCN(C(c1c(N)cccc1Cl)=O)CC2 C1(O)(c2c(C(=O)OCC(=O)Nc3c(C)non3)cco2)CCOCC1 c1(C(N2CCOCC2)=O)ccc(C(F)(F)F)c([N+](=O)[O-])c1.NC(=O)C(=O)NC n1(CC=O)cc([N+](=O)[O-])ccc1=O.CC1(O)CC(C(=O)NCCC2CC2)C1 c1(C(N(CC(CO)(CO)NC(C2C(C)C2)=O)C)=O)cnn(C)c(=O)c1 Cc1nn(C2CC2)c(C)c1COC(=O)CN1CCC(n2cnc(C#N)n2)CC1 C1(C(=O)NCC(C2CC2)N(C)C(C2CC(C)CO2)=O)(OC)CCSC1 CCC(C)CCCC(=O)N1CCN(C(=O)CNC(C2CCC2)=O)C(CCO)C1 Cc1nc(C(=O)NC2CCC(NC(C3COCC(C)O3)=O)CC2)c(C)s1 CC(O)C(C)C(=O)NCCC1CCN(C(c2cccc(-c3ccc[nH]3)c2)=O)C1 C1(NC(CN(C(CCC=C)=O)CC)=O)C=CCCCC1 C1(C(N2CCCC(N(C(CCC(=O)NC)=O)CCO)C2)=O)C2C3CCC(C3)C12 C12(C(N(C(C)C)CCN(C(=O)C)C)=O)CC(C#N)(C1)C2.c1cccs1.S Cc1cc(C(F)(F)F)cc(-c2ccc(CN(C)CC3OCCO3)cn2)n1 CCCC(CNC(=O)CC1CCCC1)C(=O)NCCN1CC2CC2C1 C(=O)(C#CC1CCOCC1)N1C(C)CCC(CNC(=O)C2=NNC(=O)C2)C1 Cc1ccc(Cl)c(C(=O)NC2CN(C(=O)CSCC(N)=O)CC2C)c1O c1(C(=O)NC2CCC(NC(c3cc(CC)ncc3)=O)C2)oc2ccccc2c1C C1(C(=O)NCC2CCN2C(C2CCCCO2)=O)COCCN1C1CCCC1 C1(C(N(CCC(=O)NCC2=CCSC2)C)=O)CCCCC1(F)F N1(C(C)=O)CCC(C(=O)NCC2(c3ccc(Br)cc3)CCOCC2)CC1C c1(SC(C)(C)C(=O)NC2CCC2)nc2ccccc2[nH]1.C1(C)(C(=O)N)CCCO1 Cc1n[nH]c(C)c1CC(=O)NCC1CC(NC(=O)C)C1(C)C.c1ccccn1 C(=O)(CC1OCc2cc(F)ccc21)NCCC(C)(C)C#N c1(C(=O)Nc2ccc(C(=O)NC3CC4CC4C3)cc2)ccc2c(c1)OCO2 c1(Nc2c(OC)cc(Br)cc2OC)ncnc2c1cnn2C c1(C(=O)OC)ccc(C)nc1N1CC2(CN(C(C3(C4CCCCO4)CC3)=O)C2)C1 c1(C(C)=O)ccc(C(=O)NCC2(O)CN(C(c3cccnc3S)=O)C2)nc1 CC(C)CC(C(=O)NC1CCN(C(=O)C(C)C)CC1F)C(C)C C(=O)(C(F)CC1CN(C(=O)C(C)C2CCCO2)C1)N(CC)CC.c1ccccc1 C1(C(=O)OC)CCCC1C(=O)N(CCCN1CCOCC1)C CC(CNC(C1(C#N)CCOC1)=O)S(C)(=O)=O c1(C(C)NC(=O)NCc2cn(CCC)nc2C)c(F)cccc1I C(=O)(C1=CCSC1)NCCCCN(C(C(C)OC1CCCC1)=O)C Cc1csc(=O)n1CCC(N1CC(F)CC1C)=O.c1(C=O)ncc(C(F)F)s1.N CN=c1[nH]c(=NCC2(C)CC(F)(F)C2)[nH]c(=NC2CC3CC(O)C2C3)[nH]1 Cc1cccc(C(=O)NCC23CC(CN2C(=O)Cn2ncnn2)C3)c1Br c1(OC)ccnc(N2CC(C)(C)C2C2CCN(C(=O)CN3CCC3)CC2)n1 C1(N(C(=O)C(c2ccccc2)C)CC)CCCN(C(=O)C(C)NC(=O)OC)C1 C(=O)(C(=O)NOC)NCC(CCC)NC(=O)CC1CC2(CCC2)C1 c1(C(CC)C)nc(-c2coc(OCC(F)F)n2)n(-c2ccn(C)n2)n1 C1(C=O)COCC(C)(C)O1.Cc1nc(CC2CC2)oc1C(=O)NC1CCCC1 C(=O)(C(CC1CCCOC1)N(Cc1ccoc1)CC1CC1)NC CC1(C)CC(NC(=O)CC2CN(C(=O)CN3CCNC3=O)C(C)(C)C2)CCO1 Cc1nn(C)c2sc(C(=O)N(C3CCC(C(=O)O)CC3)C)cc12 c1(C=O)c(C)nc(C)n1O.c1(OCC)ncccc1C(N1CC(C)C(O)C1)=O CC(O)C(C)C(=O)N1CCCC1CNC(C1(C)CCC(=O)C1)=O CC1(C)Cc2cccc(C(=O)NC3CCOCC3NC(C3CSCCS3)=O)c2O1 Cc1ccc(Br)cc1NC(=O)C(=O)NC1(c2cccc(Cl)c2)CC1 C1(NC(CCN(C(=O)Cn2cccn2)CC=C)=O)CC(C)(C)C12CCC2 C(=O)(C1=C(Cl)CCC1)NCC(C)CC(=O)N1CCC(F)(C(N)=O)C1 c1(C(=O)NC2(CC=C)CCN(C(C3COCOC3)=O)C2)ccc([N+](=O)[O-])o1 C1(F)(C(=O)OC)CC(NC(=O)CCC2CCC2)C1.C(C)(C)C.C(=O)N CCC(C)(F)C(=O)NC1CC(NC(c2c(SC)cnn2C)=O)C1 CC(C)C(O)CC(=O)N1CCC(C)(C)C1.c1(CCC(=O)N)nc(C(C)(C)C)no1 c1(C(=O)N)ccccc1SC(F)F.C1(C(N2CCC2)=O)COCC1C(F)(F)F CCCC(C(=O)NCc1cc(C(=O)NCCOC2(C)CCCC2)ccn1)OC Cc1nc(C(N2CCC(N(C)C(c3ccc(N)c(F)c3)=O)C2)=O)c2ccccn12 c1(SCC(=O)NCC2CN(C(=O)Cc3ccon3)CCO2)ccccc1Cl N1(C(C2CC(CC(F)F)C2)=O)CCCC(C)C1.C1(C(F)(F)F)(C=O)CC1.N CC(O)C(F)(F)C(=O)N1CC2(CCNC(=O)C(C)(C)F)CCC1C2 Cc1ccc(C=CCC(N2CC3(CC3)CC2C)=O)cc1.C1(F)(C(=O)N)CCC1 CCC(CCC(=O)N1CCCC1CCCNC(=O)CC(C)SC)OC C(CCCC(=O)NCCNC(C)=O)N(C(CNC(CC=C)=O)=O)C C1(CC)CN(Cc2cc(OC)ccc2Br)CCN1c1ncc(I)cn1 c1(OC)ccc2[nH]cc(C(=O)NCC(CO)NC(C3C4COCC34)=O)c2c1 N1(C(CCC2CCN(C(C=CCOC)=O)C2)=O)CCCCC1CF c1(CC)nc(CN(C(C2CC23CCC3)C(=O)NC2COC2)C)cs1 Cc1cc(C(=O)NCCCCC2CN(C(=O)C(C)(C)CC#N)C2)c(O)nc1C Cc1ccc(=O)n(CC(N2CC(O)(C(C)NC(c3occc3F)=O)C2)=O)n1 Cc1c(Cl)ccnc1C(=O)N.C1(O)CCCN(C(C2CCC(C(N)=O)C2)=O)C1.C C1(NC(CCCC(=C)C)=O)CCC2(CC1)CC2NC(c1cc2occc2[nH]1)=O N(C1c2ccccc2C2CC1C2)C(C(=O)NCCN1CCc2ccccc21)=O c1(C(C(=O)NCc2csc(C(F)F)n2)(F)F)cccc(C(F)(F)F)n1 C(C(C)(CC)CO)NC(C(C)N(C(=O)CN(C)C)CCC)=O C(CCCC(=O)NNc1ccc(F)cc1Cl)(N(C)C)OC CC1CC(NC(=O)C(O)CF)CN(C(c2ccc(Cl)o2)=O)C1 Cc1cccc(C(F)(F)C(=O)NCC2CCCN2C(=O)C(c2cnn(C)c2)O)c1 N1(C(C(C)OC)=O)CCN(C(c2ccc(Br)cn2)=O)C(C(F)F)C1 C(=O)(C1=CCC2CCC1N2C(C1CC(OC)(OC)C1)=O)Nc1cccc(C#C)c1 c1(N(C)Cc2ncc(C3CC3)o2)nccc(=NCc2c(F)cccc2Br)[nH]1 CCC(O)C(F)(F)C(=O)NC1CN(C(c2ccc3cncn3c2)=O)CC(C)(C)C1 CC1(C)CC(CNC(=O)Cc2cnsc2)N(C(c2nc(Cl)c(Cl)s2)=O)C1 N1(C(C2C(CC)C2)=O)CC(NC(c2n[nH]c3c2COC3)=O)C(C)(C)C1 N1(C(c2c(CC)n[nH]c2)=O)CCC(NCc2cc(F)ccc2F)C(C)C1 N1(C(c2c(CNC(c3c(C)scc3)=O)cc[nH]2)=O)CCCC(C)C1C(N)=O c1(OC)nc(Br)cnc1NC(C1CCN(C(C2CCN(C)C2)=O)C1)=O.C(C)O c1(NC)cc(=NCc2cccc(N(C)C)n2)[nH]c(C)n1 C1(CNC(c2c(C)coc2)=O)CCCCN(C(c2cccc(N(C)C)n2)=O)C1 Cc1cc(C)n(CC2CCCCN2C(c2cc(Br)nn2C)C(=O)NC2CC2)n1 N1(C(C(C)OCC)=O)CCC(O)(C2(NC(c3n[nH]c4ccccc34)=O)CC2)CC1 c1(NC(c2ccc(C)nc2)=O)ccc(NC(=O)C(C)C2CCOC2)cc1C Cc1nn(C)cc1NC(=O)C(Cn1cncn1)NC(=O)Cc1ccon1 N1(CC(=O)NC(COC)C(=O)NC(c2cncc(F)c2)C)CCC(O)CC1 CCCC(C(=O)N1CCCCC1CNC(=O)C(C)(C)Cc1cccc(Cl)c1)OC Cc1cnn(C)c1C(=O)NCC1CC(F)(CNC(=O)C2=CCSC2)C1 CC1CC(C=O)CN1C(=O)C.N1(CC(=O)NC(=O)CO)CCCOC1=O.C C1(N(C)C(c2ccc(-c3cccs3)s2)=O)CN(C(C2C3CCCC23)=O)CC1O c1(N(C)CC2(c3cccc(Cl)c3)CC2)nccn2nccc12 C1(C)(CNC(C2(C)CC(F)C2)=O)CCCN1C(C1CC1c1ccccn1)=O C1(CN(C(C2CC(OC)(OC)C2)=O)C)COCCN1C(=O)Cn1cnnc1O c1(C(N2C(C)CC3CN(C(CS(CC)=O)=O)CC32)=O)cccc(C#CC2CC2)c1 N1(C(C2C(CCOC)C2)=O)CC2(C=C(C(=O)NC3CC4CCC4C3)CO2)C1 c1(OC)cc(C)cc(C(=O)NC(C)C(C)NC(c2nccn3ccnc23)=O)c1O C(=O)(CCCC(=O)OC(C)(C)C)N1CC(CC)C(C(NCP(C)(C)=O)=O)C1 C1(C)(C(=O)NCC(c2cccs2)OC)CCCN(C2CCNC2(C)C)C1 CC1(C)CCC(C(=O)NCC(O)CNC(C2(C(F)F)CC(=O)C2)=O)CO1 C1(NC(Cn2c(C)ccn2)=O)CCCCC1CNC(c1coc(C(C)C)n1)=O c1(C(=O)NC2CC3C2CCN3C(c2ccc(Cl)o2)=O)cccc2c1OCCO2 N1(C(C(=O)NCCC)C2CCC2)CCC2(CC(=O)c3ccccc3O2)C1 N1(C(C(CC=C)(F)F)=O)CCC(C2(O)CN(C(=O)COCCCCCC)C2)CC1 c1(OC)cc(OC)c(S(=O)(=O)N2CCN(C(C)=O)CC2)cc1Cl C(CCN=c1nc2c(ncn2C)c(NCCCOc2cccc(F)c2)[nH]1)N(C)C C1C(C)CCCN1C(=O)Cc1ccnc(F)c1.c1(CSC)ccc(C(=O)N)o1 c1(CC(=O)NCC2C3CN(C(c4csc(Cl)n4)=O)CC23)cccc(F)c1F C1(N=c2[nH]c(Cl)c(C#N)s2)(CN(C(c2cccc3cnn(C)c32)=O)CCO)CCC1 CC1CCC(C(N2CCN(C(=O)C=Cc3cn(C)nn3)C(C)C2)=O)CC1C Cc1ccc(C(=O)NC(C)CCC(=O)NCC(n2cccn2)C)c(C)c1 C(CN=c1nc2ncn(C)c2c(NCCSC(F)(F)F)[nH]1)c1c(C)n(C)nc1 Cc1cnc(CC(=O)NCC2CCCN2C(C2(CCN(C)C)CC2)=O)s1 N1(C(C(c2cccc(OC)c2)C)=O)CC2CCC2(NC(=O)C=CCF)C1 N1(C(c2c(C)[nH]c(C)c2C)=O)CC2(NC(c3cn(C)c(=O)n3C)=O)CCC1CC2 C(CC(C(C)C)NC(c1ccncc1OC(C)C)=O)N(C(c1c(C)csc1)=O)C CCC(C)(CCNC(=O)CCCCC1CC1)NC(=O)CC(C)c1ccccc1 CC(CO)CCCNC(=O)CC1CCCC1NC(=O)C(C)(C)CC1CC1 c1(C(N(C)CC2CN(C(CC(C=C)C)=O)CC23CC3)=O)c(C)sc(C)c1C#N Cc1cc(C)c(C(N2CCC3(NC(c4ccc(F)c(N)c4)=O)CC3C2)=O)c(C)n1 C1(O)(C(N2C(C(N3CCC(F)(C(=O)NC)C3)=O)CC2)=O)CCOC1(C)C C1CCCCCC1.CC(C)(CNC(=O)C)C.c1(C=O)cnc(C(C)(C)C)s1.O C1(OC)CN(C(c2cnc(O)cc2O)=O)CCC1NC(c1[nH]cc(C)c1C)=O c1(OC)ncc(F)cc1C(=O)NCC1(O)CCCN(Cc2cn(C)cn2)C1 c1(C(=O)NC2(C(N(CCCCOC)C)=O)CC2(C)C)[nH]cc(C)c1C N#Cc1ccc(C=O)cc1.c1(C(=O)NCC2CC(C(F)F)C2)ccc(C)cc1 CC(CN(C(=O)C(C)(O)CCC1CC1)C)C(=O)NOCC(O)CO C=CC1CCN(C(=O)C(Cn2ccnn2)NC(C2CC3CCC(C2)C3)=O)CC1 c1(C(N2CC(CN(C(c3cccc(CC)n3)=O)C)C2)=O)[nH]nc([N+](=O)[O-])c1Cl c1(CC)cc(C(=O)NCC(CC)NC(=O)CC2CCCSC2)n(C)n1 CCC(C)C(C(=O)NC1(C)CC(C)C1)N(C(=O)CC1(O)CCCCC1)C CN1CC2CCN(C(=O)COC(C)(C)C)C2C1.c1(C(=O)N)ccc(O)c(F)c1 N1(C(c2c(C)csn2)=O)CC(N=[N+]=[N-])CC1C(=O)Nc1cnn(CC(N)=O)c1 Cc1ccc(O)c(C(=O)NC2CCCCC2)c1.C(=O)(C(N1CCCC1)C1CC1)N C1CC(C(=O)N(CCC)C2CC2)CC(=O)N1.c1(C=O)snnc1C(C)C.C Cc1cc2c(cc1C(N1CCCCC1c1ccon1)=O)C(C)(C)CCC2(C)C N1(C(C(N2CCOCC2)C)=O)CCCC1(C(=O)NC)C(C)C.C1(N(C)C)CC1 c1(CONC(C2C(C)CN2C(=O)CC2C=CCC2)=O)ccc(F)nc1 C(C#Cc1cccc(F)c1)NC(C(N1CCSC(C)(C)C1)C)=O c1(N(CC(C)NC(C23CCC(CC2)C3(C)C)=O)C)cnc2cc(F)c(F)cc2n1 O=C1CC2(CCCN(c3ccnc(NCc4cnn(-c5ccccc5)n4)n3)C2)CN1 CC1CCN(C(=O)CN2CCOCC2)C(C)C1NC(c1cnn2c1CCCN2)=O c1(-c2ccc(CNC(C(C(C)C)=O)=O)cc2)nnc2n1CCOC2 N1(C(CC2CC(=C)C2)=O)C(CNC(C2(C)CC(F)C2)=O)CC2CCCC12 N1(C(C(C(C)C)O)=O)CCC(C2CC2)(CNC(c2c[nH]c(Br)c2)=O)C1 C(C)(C(=O)NC(C)CN(C(=O)C=CC(C)(C)C)C)N(CC)CC N1(C(COC)=O)CC2=C(C1)CN(C(c1sc(-c3cnn(C)c3)nc1C)=O)C2 Cc1coc(C(C)C)c1C=O.C1CC2(C1)CC2.C1(C=O)CN(C(N)=O)C1.N c1(C(=O)NCC2OCCN(C(C(C)CC(F)F)=O)C2)cnc2ncccc2c1 C1(C(N(CCC)CCO)=O)C2C3CCC(C3)C12.n1(C(C)(C)C)cnc(C=O)n1 C1(C(=O)Nc2cc(F)ccc2O)C2CCCC2CN1C(c1ccns1)=O C1(NC(=O)NCC2CC(COC)OC2)CCN(CC2CC2)CC1 N1(C(CC(C=C)C)=O)Cc2ccccc2C(CNC(c2ccn(CCC)n2)=O)C1 N1(C(C(CC=C)(F)F)=O)CC2CCCC(CNC(=O)Cc3cn(C)nc3C)(C2)C1 c1(C(N2CCC3C(NC(c4ccc(C(C)C)cn4)=O)C32)=O)nccn2nccc12 CC(C)C(C#N)C(=O)NCC(C(=O)N1CC(c2nc(=O)o[nH]2)C1)C(C)C C1(CC)CN(C(=O)CC2CCC(=O)N2)CCN1C(c1csc(C(C)=O)n1)=O c1(C(=O)NCC(CC)NC(C(C)=C(CC)C)=O)ccsc1C(F)F N1(C(CC2CCCN(C(c3ccn(C)c3)=O)C2)=O)CCC(N=[N+]=[N-])C1 C1(C(=O)NCC#CCNC(c2ccc(C(C)C)nc2)=O)CC(C2CCC2)C1 C1(CCC=O)C(=O)NN=C1C.C1(CC=C)CN(C(c2n[nH]cc2C(C)C)=O)C1 C(=O)(C1=CCC(C)CC1)N(C(C)CNC(=O)C(C)(C)c1sccc1Cl)CC Cc1c(F)cc(C(=O)NCC(O)CN(C(=O)C(C)C(C)(C)C)C)c(F)c1N N1(C(CC(CC#C)NC(C2(O)CC(CF)C2)=O)=O)CC(=O)N2CCCC2C1 C1(NC(C(F)OC)=O)(CO)CCN(C(=O)CN(C2CCSC2)C)CC1 Cc1c(Cl)ccnc1C(N1CC(NC(=O)COCCCF)CC(O)C1)=O N1(C(c2scc(C)n2)C(=O)NC2(C)CC2)CCC(O)C1c1ccccc1 c1(C(N(CCCNC(C2(CO)CCC2)=O)CC)=O)cnc(C(C)OC)s1 N#Cc1ccc(NC(=O)NCCc2cnccc2C(F)F)nc1F C1(CNC(C=CC)=O)CN(C(=O)Cc2cccc3nonc23)CCC1(F)F c1(C(C(=O)NCC2C(NC(=O)NC)C2)(F)F)ccccc1C.c1ccsc1 CC(CC(=O)NCC1CCN(C(=O)C(Cl)=CCl)C12CCC2)C(F)(F)F C1(CC(N2C(CNC(c3sc(C)c(C)c3C)=O)CC2)=O)COc2ccccc2O1 c1(C(N2CC(CNCC3(CF)CC3)C2)=O)cc(OC2CCCC2)ccn1 C1(NC(c2cccc(CC)c2)=O)CC(C)CN(C(c2cnc(C)nc2C)=O)C1 C1CN(C(C2COC(=O)N2C)=O)CC(C)(C)O1.Cc1cccc(C)c1C(=O)NC C(CN=C(NCc1ccc(N(C)C)cc1)N1CCc2c(F)ccc(F)c2C1)OC C1(N(C(c2c(C)nco2)=O)C)CCN(C(=O)CC(=O)NC2CCC2)CC1 C(=O)(C1CC(=O)Nc2ncn(C)c21)N1CCCC1.C(=O)(C(=O)N)NCCOC c1(C(N2C(C)C(NC(=O)CNS(N)(=O)=O)CC2)=O)ccc([N+](=O)[O-])[nH]1 CCC(CC)C(C)C(=O)N1CCCC(CN(c2ccnc(CO)n2)C)C1 c1(C(=O)NCCN(C)C(C2CC(CCO)C2)=O)cncc(N2CCCC2)n1 Cc1nn(C)c(C)c1S(=O)(=O)N1CCCCC1CNC(c1cc(Cl)n(C)n1)=O C(C(C(C)C)NC(=O)C)NC(C(n1cc(Cl)cn1)C)=O.c1nncn1C1CC1 C1(CC#C)(NC(=O)C(CC2CCC2)NC(=O)CC(CC)SC)CCCCC1 C(=O)(C(O)CCNC(=O)CC1CN(C)C1)NC(C)Cn1cccn1 N1(C(CC(=O)Nc2ccsc2)=O)CCOC2CCN(C(=O)COC3CC3)CC12 c1(N(C)CCc2ccccc2Br)nc(N2CCC3C(C2)C3(F)F)nc2c1COC2 C#CC1(C(=O)NCC2CC3(CC3)CN2C(=O)C(O)CCCC)CCOCC1 C=CCCCC(c1nnnn1CCOC)NC(C)CC(C)(C)OC Cc1ccc2c(c1)C(C(=O)N1CCN(C(=O)Cn3cccn3)C(CCO)C1)C2 N1(C(c2c(C)c(O)ccc2)=O)CCc2nc(C(=O)NC(C)CO)ccc2C1 c1(C(C)NC(=O)Cc2coc(C(F)F)n2)ccc(F)cc1C(F)(F)F C(C(C(=O)NCCCCNC(C1CC1F)=O)C(F)(F)F)OC C1(C(=O)OC)CN(C(=O)C=CSc2ccc(OC)cc2)CC(C)(C)S1(=O)=O c1(CNC(C(C)OC(C2(CC)CC2)=O)=O)ccc(F)cc1F N1(C(C2C(NC(C3CC(O)C3)=O)CCOC2)=O)Cc2cccc(F)c2C1 c1(CC)ccc(CC(=O)NCCCCCCNC(C2CCCCC2O)=O)cc1 c1(CNC(=O)C(Cl)Cl)ccc(C(=O)NCC(O)C2CCC2)cn1 CCC1=NOC(C(=O)NCCCN(CCCNC(c2cc(CC)ccn2)=O)C)C1 c1(C(=O)NC(CC=C)CNC(c2cc(F)ccc2N)=O)cn2ccc(C)cc2n1 Cc1cccc(C(N2CCC(O)CC2C(=O)NC2CC23CCC3)=O)c1N C1(C(=O)NC2CN(C(c3c(C)scn3)=O)CC2F)CC12CC(C)(C)C2 c1(C(=O)Nc2cc(OCC)ncn2)ccc2c(c1)CN(CC1CCCN(C)C1)C2 Cc1nc2ccc(S(=O)(=O)NCC(C)(C)OC(c3ccccc3)C)cc2[nH]1 C1CCCCC1.C(C)(C)(C=CC(=O)NC1CC1CNC(=O)CC)SC c1(COCC)nc(N2CCC(C)C23CC3)cc(Cl)n1.C(=O)(COC(F)F)N C(=O)(C1CCOc2ccc(F)cc21)NC1CCN(C(c2onc(C)c2C)=O)C1 C1(NC(CCCOCCOC)=O)CN(C(c2nnccc2C)=O)CCC1C CCCCS(=O)(=O)NC(C)C(=O)N.c1(C=O)ccc(C(C)=O)o1.C1CCC1 N1(c2snc(COC)n2)CC2(CCCC2)C1.c1(C(=O)N)cc(C(F)(F)F)no1 c1(OC)cnccc1C(=O)NCC1CC(NC(C2CCO2)=O)C1 N1(C(C(CC)COC)=O)CC2CN(C(C3(C)CC3)=O)CC2(C)C1 c1(CC(N2CCN(c3cccc(C)c3)CC2)=O)cc(NC(=O)C2CC2)ccc1O C(=O)(CCCC(F)(F)F)N(C)CC1CCN(C(=O)CC(C2CCC2)C2CCC2)C1 C1(NC(C(C)CCO)=O)CCCCC12CCN(C(=O)C(C1CC1)C1CC1)CC2 c1(CNC(C(C)CNC(=O)C=CC(F)F)=O)ccnc(CO)c1 C=Cc1cncc(C(C(=O)N)N(CCCSCC)C)c1.N(C)CP(C)(C)=O C1(N(C(=O)CCNc2ncccn2)C)CN(C(c2cocn2)=O)CC1F Cc1c(Cl)ccc(C(=O)N(CC(C)NC(c2cc3sccc3[nH]2)=O)C)c1N C(=O)(CS(=O)(=O)CC)N1C2CC(C1)C2.n1(C(C)(C)C)nnc(C(=O)N)n1.C Cc1cc(C(=O)NCC2CCCC2NC(=O)Cc2n[nH]c(C)n2)on1 c1(N(C(=O)CC2CCNCCC2(F)F)CCN2CCCC2)nc2c(s1)CCCC2 C1CCN(C(c2cn(C(C)(C)C)cn2)=O)CC1O.c1(OC)nn(C)cc1C(=O)N N1(c2snc(CC)n2)CCC(NC(c2cnc3n2CCCCC3)=O)C2(CCC2)C1 c1(CCNCC(c2ccccc2Br)C)c(C(F)(F)F)cccc1Cl n1(CC)nc(C(=O)NC2CC(F)(F)C2)c(C)n1.c1(CCC=O)ccc(C)s1 C(=O)(C(C)(C#N)CC)NCC(CC=C)NC(=O)CN(C)C(c1ccoc1)=O c1(C(CNC(c2c(C)nn[nH]2)=O)NC(c2nnn(C)c2C)=O)cccc(Cl)c1Cl Cc1ccc(C=CC(=O)NC2(CCCNC(=O)C(C)C(F)F)CC2)cc1 C(=O)(C1=CCCC1C)Nc1c(C)oc(-c2ccco2)n1 c1(N(C2CC(c3ccc(Cl)cc3)C2)C(C2(C(F)F)CCC2)=O)cc(F)ccc1Br c1(CC)cc(C=O)n(C)n1.C1(CC=O)C=NN(C)C1=O.CC=CC.CC CC1CCN(C(c2cnc(C3CC3)s2)=O)CC1NC(=O)Cc1cccc(F)c1F c1(OC)cc(N2C(=O)NC(CO)C2=O)ccc1N(C)C c1nnn(C)c1C=O.C1(=CC)CCCCC1.C(C(=O)NC)(c1cccs1)SC C1(C(N(C2C(C)CC2)C)=O)CC(N=[N+]=[N-])CN1C(=O)CC1CCOCC1 C1(CNC(=O)C=Cc2cccs2)CCCN(C(=O)CC2CCC(O)C2)CC1 c1(C(N2CC(C3CN(C(c4c(C)nsc4)=O)C3)C2)=O)c(F)ccc(Cl)c1[N+](=O)[O-] C1(C(=O)NC(C)CNC(=O)Cn2cnnn2)CCc2nnn(C)c2C1 c1(C(N2CC(NC(C3N(C(C)=O)CSC3)=O)C(C)C2)=O)oc2ccccc2c1Cl C(=O)(CCCCCF)NCCCN(C(CC(c1ccc(CC)cc1)C)=O)C c1(C(=O)NC2CN(C(C(COC)N(C)C)=O)CC(C)C2)cnc2c(c1)nnn2C C1(CC(=O)N(CC(=O)NC2CC2c2ccsc2)C(C)C)CCC(C)C1 CCCCCC(C)C(=O)N1CC2CN(C(=O)C(c3ccc(F)cc3F)O)C2C1 N1(C(C(CC(C)C)C)=O)CCCC(C2CC2NC(C2(C)CNC(=O)C2)=O)C1 N1(C(C(c2cc(F)cc(F)c2)C)=O)CCC(O)C(NC(C2CCC2)=O)C1 c1(-c2n(C)c(N3CCC34CCC(C)(C)C4)nn2)ccc(Br)c2ccncc12 c1(C(N2CCCN(C(C3C(=C)CC3)=O)CC2C)=O)cc2c(C)c(F)ccc2[nH]1 c1(C(N2CCN(CC(C)NC(=O)CC3CCOC3=O)CC2)=O)ccc(Cl)cc1Cl N1(C(C2(C)CCNC2=O)=O)CC2(C1)CN(C(c1cccc3ccnn13)=O)CCO2 C(=O)(C(CC)(CC)OC)N1CCC(CC(=O)NCC(CC)OC)CC1 c1(C2(C(=O)NC3C(C(N(CCO)CC)=O)CCC3)CC2)ccccc1F C1(C)(C=O)CC(F)(F)C1.n1(CC#C)cccc1C(=O)NC1CC(C)C1.N Cn1cc(Cl)c(C(=O)NCC(Cc2ccccc2)NC(C2CCCC2)=O)n1 C1(F)(C(=O)NC(C(C)(C)C)CNC(C2CSCCS2)=O)CCCCCC1 C(C(C)(C)CSC(c1nnnn1C1CC1)C)N(CCC)CC c1(NC(C2CC23CCN(C(=O)CN2C(=O)CSC2=S)C3)=O)cc(F)cc(F)c1 C1(O)(C(C)NC(CSCCC)=O)CCN(C(c2cncc(C3CC3)c2)=O)CC1 Cc1cc(C(=O)NC2CCCC2)nnc1C.C(C(F)(F)F)N(CC=CC=O)C c1(C(N2C(C(=O)NCCCOCCOC)CN(C)CC2)=O)cccc2[nH]ccc12 Cc1ccc(C=CC(=O)N(CCCOCCN(C(=O)CNC=O)C)C)cc1Cl c1(C(N2C(C(=O)NC3C(C(=O)OC)CC3)CCC2C)=O)cnnc(C)c1C N1(C(C2(CC)CCCC2O)=O)CCC(F)(C(=O)N)CC1.c1(C(C)C)noc(C)n1 C(CC(F)F)(C(=O)N(C(CO)C1CC1)C)NC(C(COC)COC)=O Cc1[nH][nH]c(=NC(=O)c2cccc(-c3cc(=O)c(O)c[nH]3)c2)c1Cl C(C(O)CNC(=O)COCC1CCCC1)N(C(=O)CCc1cnco1)C c1(OC)nn(C)cc1C(=O)NCC(C)CN(C)C(C1C2COCC12)=O C=CC(C)C(C(=O)O)NC(C1CSCN1C(C)=O)=O c1(CC)cc(F)cc(Cl)c1.C(C)(C(=O)N)SC.C(=O)C=CC=O.C1CC1 c1(C2(NC(C3C(C(N4CCCC4c4ccncc4)=O)C3)=O)CC2)cccnc1 C#CC1CN(C(=O)CN2CCCCC2C)CCN1C(=O)C(C1CCC1)OCC CCCCC(CC(=O)N(C)Cc1ccccc1O)NC(C1CCCCC1)=O O=C1CC(C(=O)N2CCOC(CNC(=O)C(c3ccccc3)O)C2)=CC=N1 N1(C(c2c(C)nns2)=O)CCCC(C(=O)NCC)C1.C(=O)(C(F)n1cccn1)N C(=O)(C(O)CCNC(=O)CC(CC1CC1)NC(=O)C(C)(C)CO)OC C1(OC(C(CCC)OCC)=O)CC(C(=O)O)N(c2ccccc2)C1=O C(=O)(C1=NOC2COCC12)N1CC2C(NC(C3C4CN(C)CC43)=O)C(CC2)C1 C(=O)(C1=NOC2COCC12)NCC1N(C(c2cccc(OCC)c2)=O)CC=C1 c1(OC)ccn2ncc(C(N3CCC(CNC(C4CCS(=O)CC4)=O)C3)=O)c2c1 CC(CC(C(=O)NCCCF)N(C)Cc1ccsc1)C(C)(C)C Cc1nn(C)c(C)c1C(=O)C(=O)N(C)CC1CCCN1C(c1ccon1)=O Cc1ncc(C(N2CC=CC2C(N2CCC(C(C)O)CC2)=O)=O)cn1 C1(NC(c2cccnc2)=O)CN(C(=O)CCOCC2CC2)C2(CCC2)C1 C#CCC(C)C(=O)NC1CC(CNC(=O)Cc2cccc(F)c2)C1 C1(C(N2CCC3(C(CNC(c4ccns4)=O)C3)CC2)=O)CCCCC12OCCO2 N1(C(C#CC2(C)CC2)=O)CCCC2(CC(NC(c3ccc4snnc4c3)=O)C2)C1 N1(C(c2ccc(C(C)=O)[nH]2)=O)CC(C)OC(C)(C)C1.C(=O)(C(F)C1CCC1)N C1CN(C)CCN1C(c1cnc(O)c(Cl)c1)=O.C1(C(=O)N)(OC(C)=O)CC1 C1(O)(CC)CCC(NC(C2CCCCCC2NC(c2coc(C)c2)=O)=O)CC1 C1(CC=C)(NC(c2ccncc2)=O)CN(C(C2(C(F)F)CC2(F)F)=O)C1 N1(C(C2C3(CCN(C(C(C(C)C)O)=O)CC3)C2)=O)CC2CCCN2C(=O)C1C N=c1cc[nH]c(C(=O)NC2(CC(=O)NCCc3ccns3)CC2)n1 c1(OC)cccc(C(C(=O)NC(c2ccccc2)c2nc(C)no2)C(C)C)c1 CC1(C2CCC2)CN(C(C2CCC(n3cc(CCNC(N)=O)nn3)CC2)=O)C1 c1(CCC(=O)N(C(CNC(CC(=C=C)C)=O)C2CC2)C)nc2ccccc2s1 N1(CC)CC(NC(c2ccc(CNC(c3csnn3)=O)cn2)=O)CC1=O CC(C)C(C(=O)NCC1CCCCC1CO)c1ccccc1.C12CN(C1)C2=O c1(OC)ccc(C(=O)NCC2CC2)c(C(F)F)c1.c1(C=O)onc(C)c1C c1(OC)ccc(C(=O)NC2CCN(C(=O)C(C)c3cccs3)C2)c(Br)c1OC N#Cc1c[nH]c2ccc(C(=O)NCCC(O)CNC(=O)C(F)(F)CO)cc12 c1(C(N(C2C(C(=O)OC)CCCC2)C)=O)ccc2c(c1)NS(=O)(=O)C2 N1(C(C(CC)C)=O)CC2CCC1C1CN(C(=O)C(C)Cc3ccc(C)cc3)CC21 c1(C(=O)NCCCCC(C)NC(C2CCCN2C)=O)cccc(Cl)c1F c1(C(=O)NC2CCCCC2C)ccc2c(c1)CCC(=O)N2.c1(C=O)cn[nH]c1.N N1(C(c2c(CC)sc(=N)[nH]2)=O)CC2CCC1C1CN(C(=O)C(C3CC3)S)CC21 c1(NCCC(C=C)C)nccc(=NCC2CCS(=O)(=O)CC2)[nH]1 N1(C(c2c(CC)cncc2)=O)CC(NC(=O)CC(C)n2cccc2)CC(C)(C)C1 CCC(CC)C(=O)N1CCCC(CCC(=O)NC(COC(C)=O)CO)C1 c1(NC(c2c(CC)ccc(C(F)(F)F)c2)=O)cccc2nc(O)ccc12 O=c1cc(Cc2nc(C3CN4CCCCC4CO3)no2)[nH]c2ccccc12 C(=O)(C1=NN(C)C(=O)CC1)NC(C(=O)NCc1nnc(C)s1)C1CCOC1 C1(NC(COC(CC)C)=O)C2CCC1CN(C(=O)CSc1cccs1)C2 N1(C(C(C)CC(N)=O)=O)CCC2CCN(C(=O)CCS(C)(=O)=O)CC2C1 C1(C(N2CCC(C)(NC(C3CCN(C)C3)=O)CC2)=O)CN2CCCC2CO1 N(C1CCCc2ccc(C(C)C)cc21)C(=O)N.C12(C(=O)OCC)CCC(CC1)C2 CCC(C)(C)C(C)CC(=O)NCC1CCCN1C(=O)CCCN(C)C(C)=O Cc1c(Br)c(C)n(NC(=O)CCCOc2ccc(Cl)cc2)c(=O)c1C#N c1(COC)cccnc1C(=O)NC1CCN(C(C2CC(F)(F)CS2)=O)CC1 C1(C(N(CCNC(CC2ON=C(C)C2)=O)C)=O)C2CCCCC12 Cc1nc(C(=O)NCCN2CCN(C(=O)C=CC3(C)COC3)CC2)cc(O)n1 C12(C(=O)NC3C4CN(c5cc(SC)nc(SC)n5)CC43)CCC(F)(CC1)CC2 N1(C(c2c(C)ccnc2)=O)CCN(C(=O)CCC2CCCN2C)CC1C(C)C C1(C(=O)NCC2(F)CCN(C(CCC)=O)CC2)CC2OC(=O)OC2C1 C(=O)(C(C(C)C)C(C)C)NC(CNC(C(C)=C1CCCC1)=O)C(C)C Cc1cc(C2CCC2)ncc1C(=O)NCC(C)NC(C1CC(C)CO1)=O c1(C(=O)NCCCCCN(C(=O)C(F)n2cccn2)CCO)cccc(CF)c1 c1(NC(c2c(CC)cnn2C)=O)cccc(OC)c1Cl c1(CC(=O)NCCCCNC(=O)CCCc2cccs2)ccc2nn[nH]c2c1 c1(C=O)cc(C(=O)NC2C(NCC)CC2)n(-c2ccccc2)n1.C(C)(C)C O=C(C1=CCC2CCC1N2C(=O)Cn1cnnc1O)NC1CC(=O)N(O)C1 n1(CCC)cc(C(N2CC(N(C(=O)C=Cc3ccc(SC)s3)C)C2)=O)c(C)n1 CC1(CNC(c2cc(O)cc(O)n2)=O)CCCN(C2CCc3c(Cl)cccc32)C1 c1(OC)ccc(CC(N2CC(C)C2)=O)nc1.C1(C=O)C(C=C(C)C)C1(C)C CCC(C)(C)CCCC(=O)N1CCC(OCC(N2CCC2(C)C)=O)C1 C1(C(F)(F)F)(C(=O)NCCCc2cn(CC(CC)O)nn2)CCCCO1 c1(C(=O)N)cscc1S(C)(=O)=O.CCCC(C(=O)NC(C)CCO)NC(C)=O c1(NC2CC(C(=O)SC)C2)ccc(S(=O)(=O)N2CCOC(C)C2)cn1.C1CC1 CN1CCN(C(=O)CCCNC(c2cncc(C#N)c2)=O)C(CCO)C1 N1(C(CC2CC(SC)C2)=O)CC2(C1)CN(C(C1CC(O)CN1C)=O)C2 C12(NC(c3ccn(C(CC)CC)n3)=O)CCN(C(C3(C4CCC4)CC3)=O)CC1C2 c1(C(N(CCCC)CCO)=O)c[nH]c2ccc(-c3ccc(F)s3)cc12 N1(C(c2onc(CC)n2)=O)CCC(N(CCOC)C(C2CC23CCOC3)=O)CC1 C1(NC(CC2(CC)CCC2)=O)CN(C(c2ccccc2S(C)=O)=O)CCC1(C)C C1(C(=O)NC(C(=O)NCc2c(C)csc2)CO)COC(=O)N1C C(=O)(CS(=O)(=O)C(C)C)NC1(C2N(C(CCc3c(C)cccn3)=O)CCC2)CC1 CC(C)C(CNC(=O)C(F)(F)c1cccnc1)NC(=O)CS.C1CCC1.C C1(C(N2CCN(C(C(C)(C)N3CCOCC3)=O)CC2)=O)CC(C)(C)OC1(C)C C1(C(N2C(CCCC)CCC2)=O)(OC)CCN(C(c2cccc(CC)c2)=O)C1 CC1C2CCCN2CCN1C(=O)C(F)CC1CN(C(c2cnnc(O)c2)=O)C1 C1(CNC(c2cc(C(F)F)no2)=O)CC2CCC(C1)N2C(=O)CCF N1(C(CCOCC)=O)CCN(C(=O)C(CCSC)N(C)C)CC1c1cnn(C)c1 N1(C(c2c(OC)cccn2)=O)CC2(COC(C)C2)C1.C(=O)(C(F)(F)C(C)O)N C(=O)(CCCCC(N)=O)N1C(CNC(=O)C(=O)NCC(F)(F)F)CCC(C)C1 c1(C(=O)OC(C)C=O)ccc([N+](=O)[O-])c(C)c1.c1(N(C(C)=O)C)nccs1.S C=CCN=C(NCc1cc(CC)no1)NCC1(COC)CCCC1 CCC(C)CCC(=O)N1CCN(C(c2cn(CC)nc2C)=O)CC1CC(F)F CC1(CNC(c2ccsc2Cl)=O)CCN(C(=O)CCCNC(N)=O)CC1 CC1CCN(C(=O)CCCOc2ccccc2N)C1c1cccc(F)c1 C1(CC(=O)NC2CC(NC(c3cc(C(F)(F)F)cs3)=O)C2)CCCC1O N1(NC(C2C(CC)CN(C(c3cc(C)nnc3O)=O)C2)=O)CCC12CCCCC2 Cc1ccnc(O)c1C(=O)NCc1cncc(C=O)c1.C1CC(C(C)(C)O)C1 Cc1cc(F)c(C(=O)NC2CN(C(c3cncn3C)=O)CCC2CO)cc1F C1(CC)CN(C(c2cncc(Br)c2C)C(=O)NCc2ccccc2)CCN1C C1(NC(c2cc(CNC(CN(CCC)C)=O)oc2)=O)CCN2CCCC12 N1(C(C(CCC#C)O)=O)CCCC2CN(C(c3cccc4oncc34)=O)CC12 CN=c1ccc(Br)c(C(=O)NC2(CNC(C3CNC(=O)C3)=O)CCC2)[nH]1 c1(C(N(CCN(C)C)CC)=O)cc(CNC(=O)C)no1.C1CCCOC1 c1(CCNc2cc(OC)nc(C)n2)nnc2c(=O)[nH]ccn12 c1(C(=O)NC(CC)CNC(=O)C(C)C2CCCC2)cc(C)nc2[nH]nc(O)c12 C#CCCCCC(=O)NC1CC(O)(CNC(=O)CC(CC)C2CC2)C1 c1(SC)cc(C)c(C(=O)N)o1.C1C2CN(C(=O)C(C)(C)c3ccn(C)n3)CC12 C1(C(N2CCN(C(=O)COC3CCSCC3)C(C3CC3)C2)=O)C#CCCCCC1 C1(NC(CCSCC)=O)CN(C(c2cc3n(n2)CCCCO3)=O)C2(CCCC2)C1 CCCC(C(=O)NCCc1ccc(CNC(=O)C(C)C)cc1)S(N)(=O)=O.S n1(C(C)(C)C)c(NC(=O)NC2COCC23OCCO3)nc2cc(Br)ccc12 C(CC(C)(C)CC(=O)N1CCOCC1C(=O)Nc1csnc1C)OC CC1(CNC(C2CC(F)(CO)C2)=O)CCN(C(=O)Cn2cnc(=N)[nH]2)CC1 N1(C(C(CC#C)(C)NC(c2cc(C)on2)=O)=O)CC(CO)C2(CCC2)C1 c1(C(=O)NC2C(NC(c3cc(C4(C)CC4)on3)=O)CCC2)ccccc1C#N C(=O)(C1CCCc2cccnc21)N1CC=C(CCNC(C2C(C)CCC2)=O)CC1 CC1(C)CCN(C(C2CCOC(=O)N2)=O)CC1CNC(=O)C.c1cccnc1.O C1(NC(C(F)=C(C)C)=O)CCCC1CNC(=O)C(C)C1CCC1 C1(CNC(C2CC=CCC2)=O)CCC2CN(C(=O)C(F)C3CCOC3)CCC2C1 C1(C(N2CC(O)(C(C)C)C2)=O)CCC2(CC2)N1C(C12CCCN1CCC2)=O CN1CC(NC(c2ccc(C3CCCCC3)o2)=O)C(=O)N1 C(c1nc2ccccc2s1)=CC=O.N1(C(C(C)(C)SC)=O)CCC(C)(CC)C1.N C1(C(=O)NCC2C(NC(CC(C)(C)O)=O)CC2)COC2(CCC2)C1 c1(C(C)C)cc(C(=O)NOC2(C)CC(C(=O)N(C)Cc3ccccc3)C2)n[nH]1 C1(C(N2C(C(N3CC(C4CCCO4)C3)=O)CC(C)C2)=O)CN2CCC1CC2 CC(C)C(C)(C)C(=O)N1CCC(n2cc(-c3cnn(C(C)C)c3)nn2)C1 c1(NC2(CNC(c3cn(CCOC)nc3)=O)CCCC2)cc(OC)ncn1 C1(NC(C2CCN(C3COC3)C2)=O)CCCN(C(c2cc(C3CCCC3)[nH]n2)=O)C1 c1(C(=O)NCCC(C)OC)c(C)nn2ccccc12.C1(C=O)COC(=O)N1C.N C1(C(N2CC(NC(c3c(NC)cncc3)=O)C2)=O)CC2CCCCCCC12 c1(C(N2C(CC)CCCC2)=O)cc2ccccc2o1.C1(C(F)(F)F)(C(=O)N)CC1 c1(CC)ncc(C(N2CC(CNC(c3cnnn3C3CC3)=O)C2)=O)cn1.C CC1(C)CN(C(C2CN(C(=O)CNc3ncccn3)CC2(C)C)=O)CC(C)(C)O1 CC1CCC(O)(C(=O)NC(C2CN(c3ncncc3Br)C2)C)CC1 C(=O)(C1=C(Cl)CCOC1)N(C)CCOCCCNC(c1ccc(F)cc1F)=O CCCCCC(O)C(=O)NCCC1(O)CCN(C(c2ccc(NC)cn2)=O)CC1 N1(C(C(CC=C)C)=O)CCN(C(c2ccc(=N)[nH]c2Cl)=O)CC1C c1(NC(CNC(C#C)C(C)(C)OC)=O)ccc(Br)cc1Cl C1(C(N2CCC(N(CC#C)C(c3cc(C(C)C)[nH]n3)=O)C2)=O)CCNC1=O.C c1(C(N(c2ccn(C)n2)C)=O)ccc(-c2ccc(Cl)s2)cn1 c1(NC(C2CN(C)CC2c2cccnc2)=O)cccc(S(=O)(=O)N(C)C)c1 N1(C(CCCCNC(C)=O)=O)CCC(CNC(C2CCCN(C)C2)=O)C12CCC2 C(=O)(C(C)(CO)NC(=O)CCc1nc(=N)[nH][nH]1)NCC(C1CC1)OC CC(C)N=c1[nH]c(=NCCc2ccc(C(N)=O)cc2)c2c(F)cccc2[nH]1 Cc1cc(C2CC2)ncc1C(N1CCC(O)(C(C)NC(C2SCCS2)=O)CC1)=O Cc1cc(C#N)cc(C)c1C(N1CCOC(CN(C)C(C2(F)CCOC2)=O)C1)=O CCCCCC(C)(C)C(=O)Nc1ccc(NC(=O)Cc2cncc(C)c2)cc1C Nc1nccnc1C(=O)NCC(O)CCNC(=O)Cc1ccc(Cl)cc1 C1(=CC(=O)NC2CCN(C(=O)CSC)CC2F)CN2CCC1CC2.C1CCCO1 c1(C(N(CCN(C)C(c2cccc(F)n2)=O)C)=O)cnc2cccnn12 c1(N(CC(C)(C)OC)C)ccnc(N(CC2=CCCOC2)C)n1 C1(CNC(=O)COc2ccccn2)CC2CCCC2N1C(c1c[nH]ccc1=O)=O c1(C(=O)NCC2(NC(=O)CC3CSC3)CCCC2)cc(Br)cnc1O N1(C(C(C=C)O)=O)CCCC12CCN(C(=O)COc1ccc(F)c(F)c1)C2 CC1CN(C(=O)C(C)(C)Oc2ccc(Cl)cc2)CCC1.C1(C=O)CC(C)(O)C1.N C1(C(=O)NC(COC)COC)CCN(C(C2CCCNC2)=O)CC1 c1(C(N(CC(C)NC(C2CN(CC)C(=O)C2)=O)C)=O)ccc2nn[nH]c2n1 c1(C(=O)N)c2c(nn1C)CCOC2.N1(C(CC2(CSC)CC2)=O)CC(CC)C1 N1(C(C(C(C)C)C)=O)CCN(C(=O)COc2cccc(F)c2F)CC1C N1(C(c2nccc(C#C)c2)=O)CCN(C(=O)C=Cc2ccncn2)C(C)C1C c1(OC)ccc([N+](=O)[O-])c(NCC(C)NC(=O)Cc2cc(C)[nH]n2)n1 N1(C(c2c(C)nsc2C)=O)CCCC(C(=O)NC2CN3CCC2CC3)CC1 C1(NC(CC)=O)C2CC3C(C2)C13C(=O)Nc1ccc(C2CC2)cc1 C(=O)(C1=CSCS1)N(C1CCN(C(c2cccnc2-n2cncn2)=O)C1)C Cc1nc(=NC2CC(Oc3ccccc3)C2)n(-c2cccc(F)c2)[nH]1 CC1(C)C(NC(c2ccnc(C3CC3)c2)=O)CCN1C(=O)CCc1cncs1 C1(CCOC)CN(C(=O)CCc2ccc(C)cn2)CCN1C(c1cc(C)cs1)=O C1(NC(C=C(C)C(C)C)=O)CC2CCC1CN2C(=O)C(C)(C)CCCF N1(C(C=C)=O)CCC2(CC1)CN(C(=O)C(CCCCC)C(C)C)CCO2 Cc1cc(C(=O)NCCN(C(=O)C=Cc2cscn2)C2CC2)c(F)cc1F c1(CC)noc(C)c1NC(C1CC(C)N1C(C1CCOC1C1CC1)=O)=O N1(C(CCn2ncc(C)c2)=O)CC(C)(C)CCC1CNC(=O)C(F)=C1CCCC1 c1(C(=O)NC(C)C(C)(C)NC(=O)CCCS)c2ccccc2nn1C.C(C)(C)C CC(CC(C)(F)F)C(=O)N(C1CCN(C(c2cccnc2-n2cncn2)=O)C1)C C(=O)(CC(C)(C)C(=O)NC)OC.C(=O)(C(CN(C)C)C(C)C)N1CC(O)C1 N1(C(c2n(CCOC)ncc2)=O)CCC2CN(C(=O)C(C)CO)CCC12 c1(OC)cc2c(cc1OC)CC(C(N1CC3OCC(NC(=O)C(C)C)C3C1)=O)C2 c1cn2c(n1)CCCC2C.N1(C(C2(SC)CC2)=O)CC2C(C)C2C1.C(=O)C.N c1(C(N2CCCC(CCC(=O)NC(CC)CCCO)C2)=O)cnn(C)c1C#N c1(C(N(CC(=O)NCC(O)CO)CCC)=O)c[nH]nc1C c1(C(N2CCC(N3CCCC3)C2)C(=O)NC(CC)C)ccnc(F)c1OC c1(CC)cc(C(=O)NCC(CCOC)NC(=O)CC(C)C2CC2)c(C)o1 C(=O)(CCCN(C)N=O)NC(C)CC(C)NC(=O)Cc1ccnn1C1CCC1 N1(C(c2cn(CC)nc2C)=O)CCCC(C)(C)C1.C(=O)(CCC1CC1(C)C)N c1(C(N2C(CN(C(C3(CC)CCC3)=O)C)COCC2)=O)cc(Cl)cc(Cl)n1 C1(C(=O)Nc2cccc(CS(N)(=O)=O)c2)CCc2ncc(Br)n2C1 C1(NC(C(CC=C)C)=O)CCC12CCN(C(c1ccc3c(c1)CNC3=O)=O)CC2 N1(C(C23CC(CCC)(C2)C3)=O)CC2(CCC(C)O2)C1.c1(C(=O)N)cnco1 c1(NCCC2N(C(C)=O)CCOC2)cc(OC(C)C)cc(OCC2CC2)c1 Cn1ncc(Br)c1CC(=O)NC1CC1NC(=O)CC(C)(C)C N1(C(C2CC(C(C)C)C2)=O)CC2CC(NC(=O)CCSC(F)(F)F)C1C2 CS(=O)(=O)CCC(=O)NCCOC1CCN(C(=O)C(F)(F)C(F)F)C1 C(=O)(C1CCc2cccc(O)c21)NCC(CO)NC(Cn1c(C(C)C)nnn1)=O S(=O)(=O)(c1ccc(Br)cc1N1CCN(CC(C)(F)F)CC1)N1C(C)CC(C)C1 c1(C(=O)NCC(CO)NC(C2N(CCC)CCC2)=O)ccc(-c2cnn[nH]2)cc1 C1(C2CCN(C(C=CCC)=O)C2)CCCCN1C(C1CCC(CCC)CC1)=O O=C(C1=CCS(=O)(=O)C1)N1C2CCC1CC(CNC(C1(C3CC3)CC1)=O)C2 C(CC(C(=O)NC1(C)CC(F)C1)NC(=O)C(F)CC1CCOC1)=CC N1(C(C(CCC)OC)=O)CC(NC(c2cc(CC(C)C)nn2C)=O)CC1(C)C CC(C)CCCC(=O)N1CCOCC1CN(C)C(c1cn(C(C)(C)C)cn1)=O C1(C)(NC(CCCSC)=O)CCCN(C(=O)CNc2ccccc2O)C1 c1(OC)ccc(C(C)C)cc1C(=O)NC1CC1C(=O)N.c1cc(O)ccc1C C1(C2(O)CCOCC2)(C(=O)NC2CCCC(NC(=O)CC3CCOC3)C2)CC1 C(=O)(C(F)CC(CC)CC)NCC(CCC)NC(c1sc(F)cc1C)=O CCCC(C)CCCC(=O)N(CCN(C)C(C1CCCC1C(C)C)=O)C(C)C N1(C(C(=O)NC2(C)CC2)CC2CCC2)CCC2(CCOC2=O)CC1 CC1CC(NC(=O)Cn2cc(C3CCOC3)cn2)CN1C(c1coc(CO)c1)=O C1(C(C)C)CC=C(C(C(=O)NCCC#N)N2CCC(C(C)(C)C#N)CC2)CC1 N1(Cc2ccc(NC)cc2)CC2CCC(C1)C2NC(c1cc(F)ccc1C#N)=O N1(C(c2cnc(COC)s2)=O)CCCC(CN(C(=O)CC(F)(F)Cl)C)C1 CCCC(C)(CC)C(=O)NC1COCCC1C(N1CCC(CN=[N+]=[N-])CC1)=O C1(C(=O)N(C2CCOC2=O)C)(NC(CCOCC(C)C)=O)CCCC1C C(=O)(C1COc2ccc(Br)cc21)N1CCCN(C(C(C)OCC)=O)CCC1 CC1CN2CCN1C(C(=O)NC1CC3CC(NC(c4ccc(O)nn4)=O)CC13)C2 Cc1cc(C(c2nnnn2CC2CC2)NCCCC2NC(=O)NC2=O)oc1C N1(C(CC(C)(C)F)=O)CC(NC(C2CC2(F)F)=O)C(C)(C)C1 n1(CC(=O)NCC(N2CCc3ccccc32)=O)c(O)nc2ccc(F)cc2c1=O Cc1sc(O)nc1C(N1CCC(O)(CCNC(=O)CSCC(F)F)C1)=O c1(NC(C2N(C(C(C3CCCCC3)C)=O)CCN(C)C2)=O)cnn2c1CCCC2 CCCC(CCC)C(=O)NC1CC1NC(c1cnc(Cl)[nH]1)=O C(CC(=C)C)(C(=O)OC)NC(C(C(C)NC(COCC#C)=O)C)=O C(=O)(C1CCCc2c[nH]nc21)N1CC(CNc2nc(C)c(Br)cn2)OCCC1 c1(C(=O)NC(C)CCCCNC(C2CCCC(O)C2)=O)ccc2oc(=O)oc2c1 C1(C(=O)NCc2occ(C(N(C3CCCN(C)C3)C)=O)c2)CCC(C)(C)C1.S O=C(CCS(=O)(=O)C(F)(F)F)NCC1CCC1NC(C1(F)CCCCC1)=O N1(C(CCC(=C)C)=O)CCCC(C2CCN(C(C3CN(S(=O)(=O)C(F)F)C3)=O)C2)C1 C1(C(=O)NC2(COC)CN(C(=O)Cn3cc(C)nn3)C2)CCC2CC2CC1 CCCCC(C)CCC(=O)N1CCC(O)CC1C(=O)NC(CCO)C1CCC1 c1(CC)ccc(C(=O)N(CCN(C(=O)C(C)O)C)C(C)C)[nH]1 c1(-c2nc(NC(C3CC4CCC3O4)=O)sc2)ccc(F)c(Cl)c1 C(=O)(CCC(=O)N(C)CC1CCCN(c2ccc(Br)cn2)C1)NC C(CCCCCCC(=O)NC1CCC2CCN(C(=O)CC3CC3)C1C2)SC C(=O)(CCCS(N)(=O)=O)N1CC(CN(C(C2(OC)CCCC2)=O)C)C1 N1(CC)CC2CC1CN2C(=O)C(C)(C)CNC(c1ccc([N+](=O)[O-])[nH]1)=O C(=O)(C#CC1(C)CCCO1)NC1C=CCN(C(Cc2c(OC)ccc(C)c2)=O)C1 C(=O)(C1=C(Cl)CCCC1)N(CC(O)CN(C)C(C1CC(CF)C1)=O)C N1(C(C2(CC#C)CCC2)=O)CCOC2(CCC(NC(=O)C#CC(C)(C)O)CC2)C1 N1(C(c2c(C)[nH]cc2)=O)CCOC(CC(NC[Si](C)(C)C)=O)C1 c1(OC)ccnc(C(C(=O)NCSc2ccccc2)N(C2CCC2)C)c1 C12(NC(C3CC(=C)CN3Cc3cccc(F)c3O)=O)CCC(C#N)(CC1)CC2 c1(OC)ccc(C)cc1.C(=O)C(CCC1CC1)N1CC(C)(C)C1c1ccco1.N CC1CC(NC(c2cccnc2Cl)=O)CN1C(c1cscn1)=O C12(CNC(=O)CCF)CC3CC(CC(C3)C1)C2.c1(C(=O)N)ccc(Cl)c(Cl)c1 N1(C(c2c(C)cccn2)=O)CCC(CNC(=O)CCC2CC2(C)C)C12CCC2 c1(CN(CCC)C(c2sccc2I)=O)ccccc1-c1cncnc1 CCC(C)C(CC(=O)NCc1nc(C)ns1)NC(C1CC2CCC1O2)=O N1(C(CCC(C)C)=O)CC2CCN(C(c3cc4c(F)cccc4[nH]3)=O)CC2C1 C(C(=O)N1CC2C(CN(C(=O)CSC(F)F)C)C2C1)(C(C)C)n1ccc(C)c1 CC(C)CC(C)C(=O)OC(c1ccc(Br)cn1)C N1(C(C2C(=C)C2)=O)CCN(C(=O)CCn2c(C)c(C)sc2=O)CC1CC(=O)N C(=O)(C(C)S(=O)(=O)C(C)C)NCC(C)NC(c1ccn(C(C)C)n1)=O C(=O)(CC1=CCN(C(=O)C(C)NC=O)CC1)NC(C)CSCC.CCF C1(CC(=O)NC2(c3ccccc3)CC(NC(C3CC4CC4C3)=O)C2)CCCCO1 C(C(CC(F)(F)F)NC(C1(CC)CCC1)=O)NC(C1CN(CC)C(=O)C1)=O c1(C(=O)NC(CCNC(C(CCC)OCC)=O)C)[nH]c2cc(C)cc(C)c2c1C C1(C(=O)NCc2c[nH]nc2C(=O)NC2CCSC2)(OC)CCOC1 c1(NC(C2CN(Cc3ccc(Br)c(F)c3O)CCO2)=O)cc2ccccc2[nH]1 CC1(C)CCC(O)(C(=O)NC)CC1.c1(C(N2CCC2)=O)csc(-c2nc[nH]n2)n1 CC1CCCC1(C(=O)NCCCc1nncs1)NC(=O)CCCC1CC1C CC1(C(N2CC(C3(NC(c4ccc(=N)[nH]c4)=O)CC3)C2)=O)CCNC(=O)C1 c1(NC(c2cccnc2F)c2n(CCCC)nnn2)cc(C)cc(S(N)(=O)=O)c1 N1(C(CNC(C)=O)=O)CC(C)C(C(F)(F)F)C1.C(c1cnccn1)=CC=O C1(C(N(CCNC(COC(CC)C)=O)C)=O)OCC2CCCC12 N1(C(C2C(c3cc(C)sc3)C2)=O)CCOCC1CN(C)C(C12CCCC1C2)=O c1(C(N2CCCC(NC(C3CCS(=O)(=O)CC3)=O)C2)=O)nc(Cl)ccc1Cl c1(C(=O)NC2CCC(NC(C(C(C(C)C)O)C)=O)C2)ccc2c(c1)N(C)CC2 N(C1CCc2ccccc21)(CCOC)C(=O)NC12CCCC1(OC)OCC2 C(=O)(C(CS(C)(=O)=O)c1ccccc1)NC(C1CN(C(c2ccncn2)=O)C1)C c1(C(N2CCCCC(CNC(C(CCC)(C)C)=O)C2)=O)cc2ccsc2n1C C12(C(=O)NCc3c(C)c[nH]n3)CCCC1CCN2C(=O)CC1CCN(C)CC1 CC(C)C(CNC(=O)CCC(C)(C)F)C(=O)NCC(O)C(F)(F)F c1(C(N2C(CN(C(CC(COC)C)=O)C)CCCC2)=O)cnc2ncnn2c1C CC1CN(C(c2cc(C3CC3)no2)=O)CC(C(N)=O)O1.C1(CC=O)CC(=O)C1 CC1CC(NC(=O)C=Cc2cncs2)CCN1c1nccc(C#N)n1 c1(C(=O)NC(CC)(C)CC(=O)OC)c2c(nn1C)CCCC2 CC(C)C(C#N)C(=O)N1CC(CNC(C2CCC(C)CC2)=O)CC1(C)C N1(C(C2C3CCN(C(C4N(C)CCC4)=O)CC32)=O)CCc2nccnc2C1 C1(C(=O)OCC)(NC(C2CN(C(c3ccc(F)cc3)=O)C2)=O)CCOCC1 c1(NC(C2CC(Cn3cccn3)C2)=O)cc(C(F)(F)F)ncc1Cl N1(C(c2cnccn2)C(=O)NCCCC)CCN(C(C)CO)CC1 N1(C(c2cnn(C(C)(C)C)c2Cl)=O)CC2CN(Cc3cc(Cl)ccc3Br)C2C1 C1(CC(=O)NC2C(C)N(C)CC2)CC2(C1)CN(C(=O)C(F)=CC1CC1)C2 c1(C(=O)NCCCCCCC(=O)OC)cn(CCCC#N)c2ccccc12 c1(C(=O)NS(=O)(=O)C2CCOC2)cc2n(n1)CC(F)C2 N1(C(c2c(CC)nc[nH]2)=O)CC(NC(c2ocnc2C(F)F)=O)C(C)C1 C1(NC(c2cc(CCC)on2)=O)CCC(C)N(C(=O)CCC=CC(C)C)C1 c1(C(=O)N)cc(F)cc2c1C(=O)CC2.C(CC(=O)NCCOCCC)=CC c1(C(N)=O)ccc2c(n1)N(C(c1ccc(F)c(Cl)c1)=O)CCC2 c1(C(=O)NC(CNC(C(C(C)C)OCC)=O)CC(C)C)cc(C)ccc1Cl N1(C(=O)OC(C)(C)C)CC(F)(F)CC1C=O.c1c[nH]nc1C=O.N1CCC1 S(=O)(=O)(c1ccc(=NCC2CC(CC(C)(C)C)C2)[nH]c1)NCc1nn(C)c(O)c1 Cn1c(Cl)nc2nc(Cl)nc(N3CC4(COC(CNC(C5CSC5)=O)C4)C3)c12 C1(C(N2CC(CC(C)NC(c3cccc(Cl)c3)=O)C2)=O)(CO)CC(F)(F)C1 C1(C2(O)CN(C(=O)C(O)c3ccco3)C2)CC1.C(c1ccccn1)=CC(=O)N.C C1(C(NC2CCN(C(c3ccc(C(C)(C)C)[nH]3)=O)C2)=O)Cc2nccn2C1.CC C1(NC(C2C(F)(F)C23CCC3)=O)CC12CCN(C(c1cnn[nH]1)=O)CC2 c1(NC2CCC(CC)(CC)CC2)[nH]c(=NCCn2ccnn2)nc2scnc12 c1(C=O)cc(=O)n(-c2ccc(Cl)cc2)[nH]1.CC1C(C(=O)NCC(O)C)C1(F)F N1(C(c2nc(C)nn2C)=O)CCn2nc(CNC(C3(C)CCCOC3)=O)cc2C1 C(=O)(CCC(=O)NC1(C)CN(C(c2conc2C(C)C)=O)C1)NC c1(C2CC(NC(N(CC(OC)OC)C(C)C)=O)C2)cccc(Br)c1 N1(C(C2CC(N(C)C)C2)=O)CCCC(NC(=O)Cn2ccccc2=O)C1 c1(CC(=O)NC2CN(C(c3c(OC)cccn3)=O)CC2F)ccc(F)c(C)c1 C1(n2cc(C)nn2)(C(=O)NC(c2ccn(C)n2)C(C)C)CCOCC1.C(N)=O Cc1cnsc1C(=O)NCCCC1(NC(=O)C(C)SC(F)(F)F)CC1 Cn1cnc2ccc(-c3ccc(C(=O)NCc4ccc5c(c4)OCO5)nn3)cc12 N1(C(C(CC)=CC)=O)CC(NC(=O)C(c2ccc(C3CC3)cc2)O)CC(F)C1 C1(NC(COCC(=O)NC)=O)CCCCCC1C(N1CC2(CCC2)C1)=O CC1=CC(C(=O)NCCOC2CN(C(c3ncsc3C)=O)C2)SC1 c1(-n2cc(C3(O)CC(C(=O)NC(c4ccncn4)C)C3)nn2)cc(Cl)ccc1F N1(C(CC2(CC)CC2)=O)CCC2(C(=O)NC3CCCCCC3)CCCC12 CN(C)NC(=O)CCC(=O)NCCO.C1(CC(N2CCCC2)=O)COC(C)(C)C1 c1(C(=O)NC(C(C)NC(=O)CCF)CCc2ccccc2)c(Cl)cncc1Cl c1(C(N(C)CCNC(C2CCCCNC2=O)=O)=O)ccc2c(c1)OCCN2 c1(C=O)cc(-c2ccoc2)on1.c1(C(=O)NCC)cccn1C1CC1.CC.O C1(CC)CC2CCC(C1)N2C(C)C(=O)Nc1ccc(Cl)cc1Cl C(=O)(N=c1ccn(C2CCCCC2)[nH]1)Nc1ccc(C(=O)NCCOC)cn1 C1(NC(C2CC(O)(CC#C)C2)=O)CC2CN(C(C3CCC(=O)N3)=O)CC2C1 CC1(C)CCN(C(=O)C(F)CC2CCOC2)C1C(=O)NC1C(C)(C)C1(C)C N1(C(COc2cccc(C(C)=O)c2)=O)CC=C(c2c[nH]c3cc(C)ccc23)CC1 C1(N(C(CCN(C(C)=O)C)=O)C2CCC2)C(C)OCC12CCNCC2 C1(F)(CNC(CC=C)=O)CCC(CNC(C2CCCO2)=O)C1.c1ccccc1 N1(C(c2cccc(=O)o2)=O)CCN(C(=O)CCC(F)F)C2CCCCC2C1 C1(OC)CN(C(c2cnc(OC)s2)=O)CC1C(=O)NC(C)C=O.C(C)C.N C1(C)(CC)C=C(C(=O)N2CCC(CNC(=O)CC)C2(C)C)C1.c1ccccc1 N1(C(C(C)OCCCC)=O)CCCC1C1(NC(=O)C=CCF)CC1 N1(C(c2cnc(NC(C)=O)o2)=O)CCN(C(c2n[nH]cc2F)=O)C2CCCCC12 C(CNC(=O)C(=CC1CCCC1)C)(CC(=O)NC1CCC(O)C1)OC C1(C#N)(CC(=O)NC(C)CNC(c2cncc(Cl)c2)=O)CCOCC1 CCC(C)(C)CC(=O)N1CCCCC1CN(c1ncc(Cl)cn1)C C(=O)(CCCC#N)NCC(C)(C1CC1)NC(C1C(c2cn(C)nc2)C1)=O c1cncs1.C1(CC(=O)N(CCC)C2CC2)CCCC1.N=C(N)SCC=O.N CC1CC(=O)CCC1C(=O)N(CC(=O)NCCC1=CCCCC1)C1CCC1 C1(CC(=O)OCCCNS(C)(=O)=O)CCC(OCc2ccccc2)CC1 Cc1cc(C(=O)NCCCN(C)C(C2CC2C)=O)c(N)cc1F CCCCCS(=O)(=O)CC(=O)NCC(C)CN(C)C(C1CCN1CC)=O c1(C(N2CC(CC=C)(NC(c3c(Cl)cnn3C)=O)C2)=O)ccc2c(c1)CCC2 C1(NC(C2C(OC)(OC)CC2)=O)CCC(C)N(C(c2cnn(C)n2)=O)C1 CCC(CC(=O)NC(C1CN(C(c2cccc(C3(F)COC3)c2)=O)C1)C)C(C)C c1(C=O)cnc(O)n(C2CC2)c1=O.CC1CCCC1C(=O)NCC1CC1.C C(C)(CCC(=O)N(C1CCN(C)CC1)C)NC(C1CC(=C)C1)=O O=C1CCc2ccc(C(N3CCC(CNC(=O)Cc4ccc(O)cc4)C3)=O)cc21 C1(NC(C2N(CC)C(=O)CC2)=O)CCN(C(=O)CN2CCCC2=O)C12CC2 C(=O)(C1=CC2CC(C1)CC2O)NCC1(O)CN(C(CCC(CC)C)=O)C1 CC(CNC(=O)Cc1ccon1)CC(=O)NCC(O)CF C1(CNC(c2ncnc3c2CCCC3)=O)CC2(CCN(C(C3CC3F)=O)CC2)C1 C(C)(CCN(C)C(c1cocn1)=O)NC(C1(SCC)CC1)=O CC1CCC2(CO1)CN(C(=O)C(CNC(C1CCCSC1C)=O)CC1CC1)C2 N1(C(C2C(C)CC3CC3C2)=O)CCC2(CC1)OCCC2NC(=O)Cc1cnsc1 C1(NC(C(C)(C)OC)=O)CN(C(c2ccc(F)cc2Cl)=O)CCC1C(F)(F)F C=C1CCN(C(=O)CC2(OCC)CC2)C(C(N2CCC2C(C)O)=O)C1 N1(C(C(C)C)=O)CCCC(C2CCCN(C(=O)C(C)C(C)(C)C)C2)C1 N1(C(COCCCC#C)=O)CCC(C)(C(N2CCC(C(=O)OC)CC2)=O)C1 N1(C(C2CCC(CO)CC2)=O)CC2CN(Cc3c(O)cc(Br)cc3F)CC2C1 N1(C(C(C=C)(C)O)=O)CCCC2(CC(NC(=O)CC(C)C3CCCO3)C2)C1 C(C(=O)NCCC1CC(C)(C)CO1)(C(C)(C)C)NC(C=CCCC)=O N1(C(C2CC(OCC)C2)=O)CC(NC(=O)Cc2cc(Cl)ccc2O)CCC1C C1(C(N(C2CN(C)C2)CC)=O)CCC(C(F)(F)F)N1 N1(C(c2c(C)ncnc2)=O)CCC2CCCC12C(=O)NCC1CCC2CC12 CC(C)(C)C(CNC(c1ccc(C#N)cn1)=O)C(=O)NC1CCCOC1 C1(C(=O)NCc2ccc(C(=O)O)o2)C2CC1N(C(c1cccs1)=O)C2 CC(C)C(F)C(=O)N1CCC(N(C(=O)CN2CCC(C(N)=O)CC2)CCO)C1 c1(C(C)=O)ccc(C=O)nc1.C1(C(N2CCC(C(C)C)C2)=O)C(F)(F)C12CC2 N1(C(c2c(OC)cc(Br)cc2)=O)CCC(F)(F)C(C=O)C1.C1CCC(F)(F)C1.N N1(C(CCC(C(C)C)NC(CCOCCOC)=O)=O)CCC2(CCCCC2)C1 c1(C(=O)NC(C2CCN(C(Cc3c(C)con3)=O)C2)C)cncc(S(N)(=O)=O)c1 c1(CNC(C2C(C)(CC)C2)=O)cc(C(=O)N)on1.CC(C)(C)O.CC CC1CCN(C(C2CCC(F)(F)C2)=O)CC1NC(=O)CCc1ncccn1 Cc1csc2ncc(C(N3CC4(CC)CCC3C4)=O)c(=O)n12.C(=O)(CN(C)C)N c1(C=O)cn(C)nc1C(C)C.C1(CC(=O)N(CC(C)OC)C)CCC1O.N C1(NC(C(CCSC)NC(N)=O)=O)CCN(c2ncncc2C#N)CC1C c1(OC)ccc(Cl)cc1CN1CCC(NC(=O)CCc2nnc(C)o2)C(O)C1 c1(-c2c(C(N3C(C(=O)OCC)CCC3)=O)n[nH]c2)ccc(C(F)F)c(F)c1 N1(C(C(C(C)C)=O)=O)C(C(=O)Nc2csc(C(F)(F)F)n2)CC2CCCCC12 C12(NC(c3cncc(COC)c3)=O)CCCC1CN(C(=O)CC1CCCCO1)C2 CC1Cn2nccc2CN1C(C1(F)CCN(C(c2ccc[n+]([O-])c2)=O)CC1)=O C1(NC(CC(C)n2cccn2)=O)CN(C(=O)Cc2c[nH]nc2O)CC1S(C)(=O)=O c1(CC)nccn1CCC(=O)N(CC(CC)n1cccn1)CCCSC(C)C c1(C(=O)NC2C3C(C(=O)NC(CC)CCO)C4C(C3)C24)ccc(C)c(C#N)c1 CC1CN(C(c2ccnn2C(F)F)=O)CC1NC(=O)CSc1nc[nH]n1 NC(=O)CCCCC(=O)NCC=C1CCN(C(C2CSCCS2)=O)CC1 c1(C(=O)N)c(C)nc2sc(C)nn12.C=CC(C)(O)C(=O)NC1CC(F)(C)C1 N1(C(C(C)OCCCC)=O)CCCN(C(c2cccn2C)=O)C(C(C)C)C1 CC(C)CC(O)C(=O)N1CCOCC1CNC(=O)Cc1ccoc1 N1(C(Cc2nnc(C)o2)=O)CCC(C)(CNC(C2(F)CC2(Cl)Cl)=O)C1 CC(C)C(CC)NC(=O)CCN1CCC(O)CC1.N1(CC=O)CCCS1(=O)=O.N c1(C(N2CCN(C(CCCC)=O)C(CS(C)(=O)=O)C2)=O)n[nH]c2ccc(F)cc12 c1(CC(=O)N(CCNC(c2cn(C3COC3)nn2)=O)CC)ccccc1.O c1(CC)cc(Br)ccc1CC(N1CCN(C(C2CC3CC3C2)=O)C(C)C1)=O C1(NC(C(C)=C2CC2)=O)(CO)CCCN(c2cc(C(C)C)nc(C)n2)C1 C1(CC=C)(NC(=O)C(C)C(O)CC)CCN(C(C2CC2(C)Br)=O)CC1 C1(c2cn(C(COCC)C(=O)N(CC(F)F)CC)nn2)CCCN(C)C1 C1(c2n(C(C)C)nnn2)(NCc2ccc(Br)s2)CC(C#N)C1 C1(NC(CCCOCC=C)=O)CN(C(C2(C)CC(OC)(O)C2)=O)CCC1(C)C N1(C(c2csc(CO)n2)=O)CCC2CCC(C1)N2C(c1sccc1C(F)F)=O Cc1cc(C(=O)NC)c2c(O)nn(C)c2n1.C1CN(C(=O)CC(F)F)C(C)(C)C1 Cc1ccc(C(=O)O)cc1CN1CCC(C)(NC(=O)Cc2ccc(F)cc2)CC1 C=CC1CCCN(C(=O)CN2CCN(C(C3CC4(CCC4=O)C3)=O)CC2)C1 C(=O)(C1=NOC2(CCOC2)C1)NCCCCNC(Cc1c(F)ccc(OC)c1)=O c1(C(=O)NCC(CC)(CC)NC(C2CC23CCCOC3)=O)c(C)cc(F)cc1C N1(C(c2c(C)oc(CO)c2)=O)CC(C)(C)CC1C.CC(F)(F)F.C(=O)(C)N Cc1ccc(C(=O)NCC2CCCC2NC(=O)CO)cc1[N+](=O)[O-].C1CC1 CC1CN(C(=O)CCc2ccccc2Br)CCN1C(=O)C(F)CC1CC1 c1(OC(C)C)ncc(C(N2CCCC2C)=O)cc1Cl.c1(C(=O)N)cccc(=O)o1 C1(C)(C(N2CCCC3(C2)CC3)=O)CC(C(C)(C)C)=NO1.C(C=O)N(C)CC.N C(CC(O)C(=O)NCc1ccsc1C(=O)NC(C)CSCC(C)C)SC c1(CC=C)cccc(-c2nc(C(C)(F)F)no2)c1 C1(NC(C=C2CCN(C)C2)=O)(CNC(=O)CC)CC2CCC1C2.C(=O)CO c1(CCNC(C(C2CCCO2)NC(=O)COCC(F)F)=O)ccc(O)nc1 C1(N(C(C(CSC)C)=O)C)CCCCN(C(c2cnc(-c3cnn(C)c3)s2)=O)C1 C=CCC(C(=O)NC1CCC1CNC(c1ccc(=O)n(CC)c1)=O)C(C)C C1(C(N2CC(NC(c3c(CC)ccs3)=O)C(F)C2)=O)CNC(=O)CC1(C)C c1(C(=O)NC(CC)(C)CCNC(c2cscc2OC)=O)cn(C)c(=O)n1C C1(C(=O)NC(C)CC#N)CNCCN1C(c1ccc(C(C)N)cc1)=O CC(CS(C)(=O)=O)C(=O)N1CCC(NC(C23CCC(C)(CO2)C3)=O)CC1 c1(C(C)NC(=O)NCc2c(OC)cc(C)nc2)cccc(S(C)(=O)=O)c1 N1(CC(=O)N)CCCCCC1.c1(C(N(C(C)C2CC2)C)=O)cnc(N(C)C)o1 C1(NC(N2CCC(F)(F)C(C(F)(F)F)C2)=O)CC2(CCC(CO)CC2)C1 N1(C(CC)CO)CCN(C(C23CC(C(F)(F)F)(C2)C3)=O)CC1 c1(NC(COCCNC(=O)Cc2cccs2)=O)ccc(O)c(=O)cc1 N1(C(C(CC2CN(C(C(C)=CCC)=O)C2)F)=O)CCCCCCC1C C(=O)C(O)P(C)(C)=O.C=CCC(CNC(=O)CC1CC1)O.c1ccccc1 C1(OCC)COCCC1CC(=O)N.C1(C)CN(C(c2cc[nH]c2C2CC2)=O)C1 c1(C(=O)NCC2(CO)CCN(C(CCNC(N)=O)=O)CC2)cc2ccncc2s1 c1(C(=O)OC)cc(C)n(CC=O)n1.c1(C2C(F)(C=O)C2)ccccc1.CC.N Cc1cc(C(=O)NC2(C)CC(NC(C3CC3)=O)C2)cn1C.c1ccccc1.O C(=O)(C(C#N)C(C)(C)C)NC1(CNC(C(CC=C)OC)=O)CC(OC)C1 C1(NC(C(Cc2ccsc2)NC=O)=O)CCC(F)(C)C1.c1(C=O)cscn1.N CC1(O)CCN(C(C2C=CCN2C(c2ccc(C#N)s2)=O)=O)CC1 c1(C(N2CCC(CNC(CC3CN(C)CC3O)=O)C2)=O)ccc(O)c(N)n1 Cc1nn(C)c2ncc(CN=C(NCC3(O)CCC(C)C3)NC3CCCC3)cc12 N1(C(CS(CC)=O)=O)CCC(C2CCCN(C(c3cc4n(n3)CCCO4)=O)C2)C1 Cc1cccc(C)c1CC(=O)NC(C)CCNC(c1ccc(-c2ccco2)s1)=O c1(NC(=O)NC(C2CCCOC2)COC)cc(Br)ccc1Br N1(C(CCC=C)=O)CCC2(CC(NC(=O)CCCC(=C)C)C2)C1 C1(NC(c2c(C)scn2)=O)CC2(C)CC1CO2.C(=O)(C(C)(C)N1CCOCC1)N Cc1c(C(=O)NC2(C(=O)NCCCCS(C)=O)CCSC2)ncn1C c1(C(N2CC(C(=O)NCCO)C2)=O)cc(=O)n(C)cn1.c1(CC)cncnc1 C(CCCC)(CC(=O)NC1CCC(C(C)O)CC1)NC(C(C=C)OC)=O c1(CNC(C2CC(F)C2)=O)ccc(C(N2CC(c3nncs3)C2)=O)s1 Cn1nnc2c1CC(C(=O)NC1CC1NC(c1c[nH]cc1C(C)(C)C)=O)CC2 Cc1cc(C(=O)NC(c2cccnc2)C(=O)NCC2CNC(=O)C2)c(C)s1 CC1(C(=O)NCc2ccc(Cl)cc2)CCCN(C(C2CC(O)C2)=O)C1 CN(Cc1cccc(Br)c1)N1CCCCC1c1ccc(C(F)(F)F)cc1 CC1CC(C)(C(N2CC(C)(C)CC2C)=O)CCO1.C12(C=O)CC(C)(C1)OC2C N1(C(c2ccc(OC)s2)=O)CC(NC(=O)CCc2ccc[nH]2)CC(O)C1 Cc1ccc(O)c(C(=O)NC(CCF)C(=O)NCc2ocnc2C)c1 N1(C(c2c(C)nc(SCC)s2)=O)CCCC(NC(=O)C(C)c2cccs2)C1.O N1(C(Cn2cc(-c3c(C)ocn3)nn2)=O)CCN(CCOCCO)CC1 c1(NC(CCCC(=O)NCCNC)=O)c([N+](=O)[O-])ccc(C)c1C c1(C(N2CCOCC(COC)C2)=O)ccc2c(c1)CCCS2(=O)=O C(c1cc(Br)ccc1F)=CC(=O)NC1(C(O)CO)CC1 c1(N(CC(O)C2CC2)C)cc(Br)ccc1S(=O)(=O)N1CCCCC(CO)C1 c1(C(=O)NC2CCC(CCNC(c3ccc(CC)o3)=O)C2)ccnc(CO)c1 c1(C(=O)NCC2CCC(NC(c3c(C)cc[nH]c3=N)=O)C2)ccc2cccnn12 C12(C(=O)NCCCN(C)C)CCCC(O)(CC1)C2 c1(C(=O)NC2CN(C(CCCOCCOC)=O)C(C)CC2)cccc(F)c1C#N C(C(CNC(c1cc[nH]n1)=O)S(C)(=O)=O)NC(C=Cc1nc(C)sc1)=O C1(NC(C23CC(C)(C2)C3)=O)C(CNC(c2ccccc2)=O)CCC12CCC2 CON(CCC(=O)N1CCC(F)(CO)C1)C(=O)C1CCC(C#N)CC1 C1(CNC(c2ncn(C)c2)=O)CCCCN(C(C2CCC(F)(F)C2)=O)CC1 C1(CCNC(c2c(C)cncc2)=O)CC(F)(F)CN1C(=O)C(C)n1cccn1 C1(NC(C(COC)O)=O)CC2CCC(C1)N2C(C1(CO)CCCC1)=O CC1CCN(C)C(=O)C1NC(=O)Nc1ccc(COc2ccc(Cl)cc2)cc1 c1(CCC(=O)NCCN(C(C(C=CCCC)O)=O)C)cc(F)ccc1Br c1(C(c2noc(C3CC3C)n2)C)cc(Cl)ccc1F N1(C(C(CC#C)O)=O)CCN(C(C2(F)CCCC2)=O)CC1c1cc(F)ccc1F CC(CCCCO)NC(=O)C(Cn1cncn1)NC(=O)CCc1ncnn1C c1(C(N(CCN(C(c2ncsn2)=O)C)C(C)C)=O)cc2c(C)cccc2[nH]1.C Cc1c(C(=O)NC2CC2)ccc(F)c1F.c1(C(N(C)C)=O)cnn(C(C)C)c1 CC(C)CC(C)(C)C(=O)N1CC(C(=O)NCCO)CC(C)(C)C1.C1CC1(F)F CCCCC(C(=O)NC)NC(=O)C1=NOC(CNC(c2c(C#N)ncn2C)=O)C1 c1(OC)ccc(Br)c(CN2CC(C(=O)Nc3cccc(Br)c3CO)CC(F)C2)n1 c1(C(C)C)nc(-c2nccnc2Br)n(C(C)C)n1 N1(C(C(CC=C)(C)C)=O)CC(C(=O)N(C)CC2(OC)CCCC2)C2(CCC2)C1 c1(OC)cc(CN2CCCC(C(C)NC(c3cc(I)ccc3Br)=O)C2)ccc1F c1(OC)cc(CNC2CC2C(=O)Nc2cncc(O)c2)c(F)cn1 C=CCCC(C(=O)N1CC=CCO1)NC(=O)C(C1CCCCC1)O C(=O)(C1CCc2snnc21)N(C)CC1CCN(C(C2C(C)OCCC2)=O)CC1 c1(C(N2C(C(C)NC(C(CC=CC)C)=O)CCC2)=O)cccc(N)c1C c1(NC(c2ccc(I)c(O)c2)=O)ccc2c(c1)C(=O)OCC2 c1(CC)nc(C(=O)NCc2cc(C=O)cs2)cs1.C(C(C)(C)C)=CC.N C1(C(N2C(C)(CCO)CC2)=O)CC1C1CN(C(=O)CC23CCC(CC2)C3)C1 CCN=c1ccc(C(=O)NCCC2CN(C(c3snnc3C)=O)C2)c[nH]1 Cc1cnn2cc(NC(C3CCNC34CC4)=O)cnc12 n1(CC)nnc(C(N2C(CNC(c3ccon3)=O)CC3CC23)=O)c1C Cc1cc(OCC(=O)NCCC(O)CNC(C2(C(F)F)CCCC2)=O)ccc1Cl c1(C(N2CCC(NC(=O)Cn3nccn3)C(F)C2)=O)cc2c(F)c(F)ccc2s1 Cc1nc2ncc(C(=O)NC(C)C(C)C)cc2o1.c1(C(=O)N)ccc(=O)n(C)n1 c1(CC(C(=O)NCCCNC(C(c2ccc(F)cc2)OC)=O)O)ccccc1Cl Cn1cncc(C(=O)NCC(C)(C)NC(C2CC(F)(CO)C2)=O)c1=O c1(CN2CCC(O)(C(=O)NC(c3ccncc3)CC)C2)c(C)cc(F)cc1C c1(-c2cn(C(C)C(=O)NCC3COC(=O)O3)nn2)cccc(F)c1Br CCC(C(=O)NC1(c2cc[nH]n2)CC1)NC(c1cc(C(N)=O)c[nH]1)=O C1CC2CCC(C1)N2C(=O)CC1CCC(=O)C1C.CCC(C)C(C(=O)NC)OC c1(C(N2CC3(CC(C(N(C)C)=O)C3)C2)=O)c[nH]c2cccnc12 N1(C(c2c(CC)nn(C)c2)=O)CC2CC1CN(C(c1ccc(C)nc1NC)=O)C2 c1(C(=O)NC(CCNC(CC(C)SC)=O)(C)C)cc2c(cn1)CCCC2 c1(CN2CCN(C(C)=O)CC2)cc(N)c([N+](=O)[O-])cc1Br C1(C2CC2)(NC(c2n[nH]cc2Cl)=O)CCN(C(C2(C)CC2)=O)C1.c1cccnc1 c1(C(=O)NC2CC3(C(NC(C(CC#C)C)=O)C3)C2)cc(Br)c(C)cc1OC Cc1ccc(C(N)=O)cc1NC(=O)C(c1ccc(Br)cc1)N1CCCC1 CC(C)CCCCCC(=O)N1CC=CCC1C(=O)NCC1C(C)(C)C1(F)F N(C(=NCCCC1(O)CCC1)NCC)C1CCC(SCC)C1 C1(NC(c2c(C(C)C)occ2)=O)CCCC(CN(C)C(c2cnc(O)n2C)=O)C1 c1(OC)cc(CCC(N2C3CCC2C(NC(=O)Cc2cnsc2)C3)=O)ccc1O C#Cc1ccc(C(=O)NC2CCCN(C(c3occc3C(C)C)=O)CC2)c(F)c1 C1(CC(N2CC3CSCC3C2)=O)C2CCCC2N1C(c1sccc1Cl)=O c1(-c2cnc(CC(=O)NCc3cn(C)nc3)nc2)ccc(F)c(C(F)(F)F)c1 C(CC(=O)NC(CC1CC1)C(=O)N)(C(F)F)NC(C1CC(C#C)(O)C1)=O N1(C(C(C)OCOC)=O)CC(O)CC1CNC(=O)Cc1ccccc1.C(C)C C1(C)(C(=O)NC(CC)CSC)C=CCN1C(=O)C(CSC)OC C1(NC(c2c(CC)ncs2)=O)CN(C(C2C=CCC2)=O)CC1CC(C)(C)C C12(C(=O)NC3C(CNC(COC(C)C)=O)CC3)CCC(O1)c1ccccc12 Cc1cccc(C)c1S(=O)(=O)N1CCC(CC(=O)Nc2ccc(O)cc2)C1 C(=O)(CCCC(C)(C)C#N)N1CCC2CN(C(c3c(CC)nccc3)=O)CC21 C1(NC(c2ccc(-n3cc(CCC(=O)OC)nn3)cc2)=O)CC2CC1CC2CO c1(CC)ncccc1C(=O)N(C)CC1C2CN(C(=O)C(F)C3CCCC3)CC12 C=CC(F)(F)C(=O)NCC1(NC(=O)C(C(C)C)n2cccc2)CCCC1 N1(C(C(C)NC(CC)=O)=O)CCC(NC(=O)CCc2ccsc2)C12CC2 Cc1cccc2[nH]c(C(N3CCC(NC(C4CCC4C(F)F)=O)C(O)C3)=O)cc12 Cc1cc(NC(CCN(C)C(C2CC23CC(O)C3)=O)C(C)C)n2nc(C)nc2n1 c1(CC(=O)NCC2CCCCN(C(c3cc(C)no3)=O)C2)c(C)cc(O)cc1C c1(C(N2CCCC(NC(c3[nH]cc4c3CCCC4)=O)C2)=O)cn2cnnc2cn1 C(=O)(CC1OCCc2ccsc21)NC1C(C)CCN(C(COCCCC)=O)C1C N1(C(c2c(C)ccs2)=O)CCCC(N(C(=O)C=CC2CCCO2)CCF)C1 C1(CNC(=O)NCc2ncn(C)c2)CC2CCC(C1)N2c1ncccn1 Cc1ccc(O)c(C(=O)NC(C)(C)CC(=O)NCCC(C)N(C)C)c1 C(=O)(C(C)(C)CC(F)F)NC1CN(C(C(CC#C)(C)C)=O)CC1C C#CCCCC(C)C(=O)NCCC1(C)CCN(C(c2cnc(N)cn2)=O)CC1 c1(CNC(N(CC(=O)N(CC)CC)C)=O)cc([N+](=O)[O-])cnc1C C1(S(=O)(=O)NC2(CO)CN(C(=O)C(C)n3ccnc3)C2)(CC=C)CC1 N1(C(C(=O)N)=O)CCC(C)C(N(C(=O)Cc2cc(C3CC3)on2)C)C1.CCC C(=O)(C1CCc2c[nH]nc21)NCC(CO)NC(c1c(OC)ncc(Cl)c1)=O C1(C(=O)OC2(C3CC3)CC2)CCCCN1C1CCCC1 c1(C(C(=O)NC2(C)CC2)N(CCC)CCC)cnn(CCC2CC2)c1 C1(C(=O)NC2C(CNC(C(CCC)C)=O)C2)CCc2nnc(O)n2C1 C(=O)(C1=NOCC1)NCCC(C)N(C)C(c1coc(C(F)F)c1)=O C(c1cccc(F)c1)=C(C(N1CC(O)C1)=O)F.C1(C(N(C)C)=O)CCC1(F)F CCC(C)C(C(=O)NCC1CCC(C(N2CCS(=O)CC2C)=O)CC1)OC C1(NC(CCC)=O)CCOCC1NC(=O)Cc1ccccc1CC c1(CN2CC(CNC(=O)CC(C3CC3)C3CC3)C2)cccc2c1OCCO2 C(=O)(CCCCC(=O)OC)NC(CC(=O)NCCCOCC#C)C(C)C C1(NC(CCCOCC=C)=O)CC2CCC1N(C(c1ccc(C)cc1N)=O)C2 C(=O)(CC(CC)CC(F)(F)F)NC(CC=C)CNC(c1ccc(F)c(F)c1)=O C1(NC(C(=O)NC2CSCSC2)=O)COCC1Oc1ccccc1 C1(C(NC(C)C=O)=O)CCC2(C1)N=N2.c1ccccn1.C1(C2CC2)CCCC1.C CC1CN(C(=O)C(C)(C)O)CCC1C(=O)NOCc1c(F)cccc1F c1cnnn1C1CC1.C(C)(C(=O)NCC=O)N(CC(=O)NCC)CC.N Cc1c(C(N2CCC(C(N3CC(F)(CF)C3)=O)C2C)=O)cccc1C#N C(=O)(C(O)CC[S+](C)C)NCC1(O)CC(NC(c2[nH]c(=NC)sc2)=O)C1 c1(C(=O)NC)ccc(=NCCC(C)(C)COC)[nH]c1 C(=O)(CCCCCCNC(=O)CCC1CC1(F)F)NCCNS(CC)(=O)=O c1(C(N(C2CN(C(C(CN(C)C)O)=O)CC2(C)C)C)=O)cc2ccc(O)cc2[nH]1 C(=O)(C(CCCC)C(C)C)NC(C(C)NC(CCC=CCC=C)=O)CO C1(C#N)(C(N2CCC(C)(NC(C(C)Cc3ccc(F)cc3)=O)C2)=O)CCSCC1 c1(OC)ccc(CC(C)C(=O)NC2CC(c3cccc(Cl)c3)C2)cc1F C1(CNC(CC(C)c2ccco2)=O)CC2CCC(C1)N2C(c1cnc(O)s1)=O C1(C(=O)NCCC(C)O)(CNC(c2c[nH]c(=O)cn2)=O)CCCCC1 C1(CC(=O)N(CCNC(c2cn(C)cn2)=O)CC)CCC2(CC1)CC2.C c1(C(N(CCCNC(C(CCC)N(C)C)=O)CC)=O)ccc2c(c1)CCC2=O c1(C(=O)NCCCN(C(=O)CCc2cn(C)cn2)CCC)cc2ccncc2[nH]1 NS(=O)(=O)C1CCCN(CC(=O)Nc2cnccn2)C1 c1(C(C(=O)NCCCCCC)N(C2CCCCCC2)C)n[nH]c2c1CCCC2 N1(C(c2ccc(CNC(Cc3c(C)ccnc3)=O)o2)=O)CCCc2occc2C1 C(N=c1[nH]c(=NCC2CCCC2)[nH]c2ccsc12)C1C(C)COCC1 Cc1cccc(OCC(=O)NC2CC(NC(C34CCCCC3C4)=O)C2)c1 C1CCN(C(=O)C(C2CCCO2)C2CC2)C1C1CC1.C12(CC=O)CC(C1)C2 N1(C(C(CC)C)=O)CCC(O)CC1C(=O)NCC(C)(C)N(C)C c1(OC)ccncn1.N1(CCN)CCC(CN(C(=O)CC2CCC3CC23)C)CC1 C1(C(=O)NCc2cc(CC)no2)CC(NC(=O)CCc2csnn2)CCO1 C=CC1(C(=O)N(C(C)C(=O)OC)C)CCN(C(c2cc(C(N)=O)c[nH]2)=O)CC1 C1(C(=O)NC2(C)CN(C(C3(C(=O)OC)C(=C)CC3)=O)C2)CC2CCC1C2 c1(C(=O)O)[nH]c(=NCCCc2c(F)cccc2F)sc1Cl c1(CC(C)C(=O)N(C(C)CNC(=O)COc2cn[nH]c2)C)ccccc1F C(=O)(C(O)C1=CCCCC1)N1C(CN(C)C(c2cncnc2)=O)CCCC1 c1(C(N2CC(CNC(CCNC(C)=O)=O)C(C)C2)=O)cncc(C)c1C c1(CC)ccc(F)c(C(=O)NC2(C)CCN(C(C3(C)COC3)=O)CC2)c1 C(=O)(C(O)C1=CCCCC1)N(CC=CC(=O)N(CCCCC)CCO)C c1(SC)cc(C(=O)NC(C)CNC(c2cccc(N)c2C)=O)ccc1F c1(CN(C(=O)NCc2ccc(OCC)nc2)C)c(C)cc(C)cc1C C1CN(C(=O)Cn2cnc(C#N)n2)CCN1C(=O)C.C1(C=O)CCC1.CO.C Cc1c(C(=O)NCCNC(c2cccc(N(C)C)n2)=O)cnn1C1CCC1 c1(OC)ccc(C(=O)N(C2CN(C(=O)CC3CC3)CC2(C)C)C)c(C)n1 Cc1ccc2c(c1)CC(C(=O)NC13CC1CN(C(c1nnc(O)cc1O)=O)C3)S2 N1(C(c2oc(C)c(Br)c2)=O)CC2(C1)CN(C(=O)CN(C)C(C)C)CC2CO c1(NC(C2(CNC(C(CC=C)CC)=O)CC2)=O)c(C)ccc(O)c1C C1(CNC(CC=CC=C)=O)CN(C(=O)Cc2cc(CC)no2)CCC12CCC2 c1(C(C)NCCC23COC(C(F)(F)F)(C2)C3)cc2cccc(F)c2o1 CC(C)(C)S(=O)(=O)C1CCN(CCCN(c2c(O)nc(=O)n(CCF)c2N)C=O)C1 C=CC(C)(CC)C(=O)N(CCCC(C)(C)C)C.c1(C(=O)N)csc(C(F)(F)F)n1 c1(SC)c(C(=O)NC2CCC(CCNC(c3c(C)noc3N)=O)C2)cnn1C C1(C(=O)NC(CCOC)C)COCCN(C(=O)Cc2cccnc2F)C1 c1(C(C)NC(=O)C2=C(Cl)CC2)ccc2c(c1)CN(C(=O)C#CC1(C)CC1)C2 N#Cc1csc(C(N2CC(NC(c3ccn(-c4ccncc4)n3)=O)C(O)C2)=O)c1 C1(CC(=O)N(CCNC(CCSCC)=O)C(C)C)CCCC2(CC2)C1 c1(C(=O)NC2CCC(c3ccc(F)cc3)C2)ccc2c(c1)C(=O)NCCO2 CC1CN(C(=O)C=CBr)CCC1CNC(=O)CCc1cn[nH]c1 C1(N(C(CNC(=O)OC)=O)C)CN(C(=O)CCN2CCCC2=O)CC1F CCC(C)(CO)C(=O)NC1C2CC(NC(C3NC(=O)OC3(C)C)=O)CC12 N1(C(C2CC(CC)C2)=O)CC(C(N)=O)(C)C1.C(=O)CCC1CC1(F)F.N N1(C(CN(C(c2ccc(C#C)cc2)=O)C2CC2)=O)CCCC(C)(C#N)C1 CCCC(CCNC(C1CCN1C(C1CNC(=O)N1)=O)=O)C1CC1 c1(CC(N2C3CC2CN(Cc2cc(Cl)c(Cl)cc2O)C3)=O)cc(F)c(F)c(F)c1 Cc1nc(C)c(C(=O)NCC2(C)CN(Cc3ncsc3Br)CCO2)c(C)n1 CCC1=C(C(=O)N2CC3C(NC(=O)CC4CCCO4)C3C2)CCCO1 N1(C(CN2C(=O)CCC2)=O)CCC(C(=O)Cc2ccccc2)CC1 c1(C(=O)NCC2OCCCN(C(C3(C#N)CC3)=O)C2)cc2c(=O)[nH]ccn2n1 N1(C(CC(C=C)CC)=O)CC2(CC(NC(=O)CC(C)c3ccncc3)CO2)C1 N1(C(C=O)C)CC2C(C(=O)N(CCCN(C)C)C)C2C1.[nH]1nccc1C.CCC.N c1(C(N2CCN(C(CCCC)=O)CC2CCO)=O)ccc(N=S(C)(C)=O)s1 N1(C(=O)OC(C)(C)C)CC2(CCN(c3ccc([N+](=O)[O-])c(F)c3)CC2)C1 C#CCC(C(=O)N1CC(F)CC1CNC(=O)CCc1ccn(C)n1)C1CC1 C1(C(=O)NC(C)CCCCNC(=O)C=Cc2cccs2)CC(C2CC2)=NO1 C=C(Br)CC(C)(C)C(=O)N1CCC(NC(c2cnc(CC)[nH]2)=O)C(O)C1 C=C(Cl)CC(C(=O)NCc1csnn1)NC(C1CCCS1)=O C(=O)(C(C)(C)S(C)(=O)=O)N.C1(CC)CCN(C(=O)CC2COC(=O)C2)C1 C1(CN=c2ccnc(NCC3(OC)CCCCC3)[nH]2)COC2(CCCCCC2)O1 C1(NC(CCOCCC)=O)CN(C(c2c[nH]nc2-c2cnn(C)c2)=O)CC1(C)C C(CC(=O)NOCC1(C)CCC1)N(C(C1CN(C)C1)=O)CC CC1CN(C(=O)CCC2CCOCC2)C(C)CN1C(=O)CC1COCCOC1 c1(C(N2CC(NC(C(C)CO)=O)CC2(C)C)=O)cccc2ccn(C)c12 c1(C(=O)NC2(CCNC(C3C(C)N(C)CC3)=O)CCCC2)cnn2cccnc12 c1(C(=O)N)cc([N+](=O)[O-])nn1C.C1(OC)CC(C)N(C(=O)C)C1.C1CCOC1 N1(C(C2(CC)CN(C(=O)C(C)Cn3cccn3)C2)=O)CCCC(CN(C)C)C1 C(=O)(CC(F)(F)CC=O)NCC(C1CC1)NC(c1c(CC)nn(C)c1)=O N=c1ccc(C(=O)NCC2(C(N3CCOCC3)=O)CC23CCC3)c[nH]1 C12CCC(CC1)C2.c1(C=O)ccccc1.O=C(CC)NC1CC1.C(=O)C1CC1 N1(C(CC(=C=C)C)=O)CCC(O)(C(C)NC(=O)CC2CCCC(=O)N2)CC1 C1(NC(C2CCCC(=O)N2)=O)CC2CC(C1)N(C(c1cnc(F)c(Cl)c1)=O)C2 C1(CC(=O)NCCNC(C2(CC3CCCC3)CCC2)=O)COc2ccccc2O1 n1(CCC)cccc1C(=O)N(CC(C)(C)CNC(=O)C(c1ccnn1C)C)C N1(C(CCC(C)=O)=O)CC2CCCN(C(c3csnc3C)=O)C2C1 C1(NC(c2cccc(C)c2F)=O)CC2CCC(C1C)N2C(=O)CCC(C)O c1(OC)ccc(C(O)CNC(C2CCCN(Cc3cccnc3OC)C2)=O)cc1 c1(C(=O)NC(C)CNC(c2snc(O)c2Cl)=O)c(O)cc(=O)n2c1CCCC2 C1(NC(=O)C=CC2CCC2)CCOC(C(=O)NCCC2(CO)CCC2)C1 N(C(=NCC(C)c1ccsc1)NC1CCC1)CC1CCN(C(C)C)CC1 Cc1cccc2c1OC(C(N1CCOCC1CCNC(=O)COCC(C)C)=O)C2 C(CC(C)C(=O)N(C(CC)C(N1CCN(C2CC2)CC1)=O)C)=CC c1(C(N2CC(NC(=O)C3=CCCOCC3)C(O)C2)=O)cccc2cccc(O)c12 C1(C)(CC)CCC(C(=O)N(C2CN(C(c3ccc(COC)cc3)=O)C2)C)O1 C1(N(c2cc(O)ncn2)C(c2c(C)ccn2C)=O)CCCC12CCNCC2 c12cc(C)nc(n1)NC2.c1(CC)n[nH]c(CC)c1CC(N1CCCC(NC)C1)=O C1(N(C)C(C2(N3CCCC3)CC2)=O)CCCCN(C(c2cc3n(n2)CCC3)=O)C1 C(=O)(C(CC(C)C)ONC(=O)CC1(C)CC1)N1C(C(=O)OCC)CCC1.S Cc1ccc2c(N3CCSC(C)(C)C3)nc(=NCCS(C)=O)[nH]c2c1 C1(NC(CSCC)=O)C(C)CN(C(=O)Cc2scnc2-c2ccccc2)CC1C c1(OC)nccc(C(=O)N(C)CCC2CCN(C(=O)CC3CC=CC3)CC2)n1 CC(C)CC(C(=O)N1CCCC1CNC(c1cscn1)=O)c1ccccc1 c1(N2CCN(C(CCC)=O)CC2)[nH]c(=NC2CCCC(F)C2)nc2scnc12 C(C)(C(C(=O)N(CC(C)(C)C)C)C(C)C)NC(c1c(C)oc(CO)c1)=O CCCCCCCC(=O)NC(CC(=O)NC1C2CCC1CC2)C(C)OC N1(C(C2C(NC(CCOC)=O)CC2)=O)CC2CC1CC2C(=O)OC c1(C(N2CCCC(NC(C(C)NC(N)=O)=O)C2)=O)ccc(F)c(C(F)F)c1 C1(CNC(C2OCC(C)C2)=O)CCN(C(c2ncnn2C)=O)CCC1(F)F c1(NC(C2CN(C(c3n(C)ncc3C3CCC3)=O)C2)=O)nc[nH]c2ncnc1-2 S(=O)(=O)(c1cccnc1NCCCc1nc(C)cs1)NCC(=C)CC O=C1CC(CC(N2CCC(CNC(=O)CCC(=O)c3cccs3)C2)=O)CCCN1 C1(O)(C(=O)NC2CCC(CNC(CC3(C#N)CC3)=O)C2)CCOCC1 c1(CN2CCC(O)(C(=O)Nc3c(Cl)ccnc3Br)C2)c(F)ccc(Br)c1Cl C(=O)(CC)NC(C)C.C1(CC=CC(=O)N)CCC1.C(=O)C(O)C1CC1 C#CCCCCCC(=O)NC12CC(C(=O)NC3CCCCCC3C)(C1)C2 C1(C=O)CCCS1(=O)=O.Cc1occc1C1CC1C(=O)NC1CC(C)C1.N C1(CC)CN(C(c2ccoc2Cl)=O)CCC1NC(c1cc(C(C)C)ccc1F)=O Cc1cn2cc(CC(N3CC4CC3C4NC(c3ccn(CCF)n3)=O)=O)nc2s1 c1(CN2CCCN(C(C3N(C)CCC3)=O)CC2)c[nH]c2ncc(Br)nc12 c1(-c2nc(C(C)SCC)nn2C(C)C(C)C)ncnc2c(C)csc12 C12(CNC(COCC)=O)CC1CN(C(=O)CCOCC1CCCO1)C2 C#Cc1ccc(F)cc1C(=O)N(C)CC1CCCN1C(=O)COCCOC Cc1nc(O)ccc1C(N1CCCCC1CN(C(=O)CCc1ccnn1C)C)=O N=c1[nH]nc(CC(N2CC(n3cnnc3)C2)=O)s1 c1(C(=O)NCC2(CNC(=O)CCCC3CC3)CCCC2)ncc2ccccn12 N1(C(CS(=O)(=O)NC)=O)CCC(C2CC2)C1C(=O)NCc1cnn(C)c1C c1(OC)cc(CC(=O)NC2CC2C(N2CCCCC2C)=O)cc(C(F)(F)F)c1 C1(C(=O)NCc2ncn(C)n2)C2CC(O)C(C2)N1C(C1(CCF)CCC1)=O C1(C2CCN(C(C3C(C)C3C)=O)CC2)OCCCC1N=c1cc[nH]cc1[N+](=O)[O-] N1(C(C=C(CCC)C)=O)CCOC(CCNC(=O)CCC(=O)OC)C1 C1(O)(CCNC(C(C)C2CCCC2)=O)CCN(C(=O)C=CCN(C)C)CC1 Cc1noc(C2CC2)c1C(=O)NC(C)C1CC1.C(=O)(CCCC)N.C(N)=O CCC(C(=O)NCC(=O)NCCO)NC(=O)Cc1cc(C)cs1 c1(C(N2CCCC(NC(C(F)=C(C)C)=O)C(F)C2)=O)cc2ccc(F)cc2s1 Cc1cc([N+](=O)[O-])ncc1C(=O)NCC1CCC1.C1(C=O)CCCC(=O)O1.N C1(NC(CC(C=C)C)=O)CN(C(c2cc(F)ccc2OC(C)C)=O)CC1(C)C S(=O)(=O)(c1cc(C)cc([N+](=O)[O-])c1)N1C(c2n(CCCOC)ncc2)CCC1 C1(C(N(CC(C(=O)NC)C)C)=O)CC2(CC2)CN1C(C1C2COCC12)=O CC(N=c1[nH]c(=NCCc2ccoc2)c2ncccc2[nH]1)c1cnn(C2CC2)c1 c1(C(=O)NC2C(NC(Cc3c(OC)ccc(C)c3)=O)C2)cnn2ncccc12 C1(C(=O)NCC2CN(C(C3CCC(N(C)C)C3)=O)C2)(CC)CCCCC1 N1(C(c2c(F)ccc(C)c2)=O)CC(C(=O)NCCCS(C)=O)C(C2CC2)C1 Cc1cc(CN2CCOCC2CC(=O)NC2CC2c2ccc(Br)cc2)c(C)s1 c1(N2CC3C(CNC(C4CCCC(OC)C4)=O)C3C2)nc(C)cc(C)c1C#N N1(C(C2ON=C(C)C2C)=O)CCCN(C(c2cn(CCO)nn2)=O)CC1C N1(C(Cc2c(C)nc(C(CC)C)nc2C)=O)C2CCC1C(CO)N(C(=O)CO)C2 C(=O)(C(C)(C)C(C)C)NC1C(NC(C2OCCN(C(C)C)C2)=O)CCCC1 c1(C(N2CCC(O)(C(CNC(CC=CCC)=O)C)C2)=O)nccc(Cl)c1Cl N#Cc1ccc(-n2ccc(=NC(=O)c3cnc(CC4CCNCC4)s3)[nH]2)c(Cl)c1 N1(C(c2c(C)n(C3CC3)cc2)=O)CCOCC(NC(c2n[nH]cc2Cl)=O)C1 C1(CNC(C(=Cc2ccccc2)CC)=O)N(C(c2cnsn2)=O)CCCC1(C)C CCCCCC(C)NC(=O)C(CNC(=O)CCc1csnn1)N(C)C C1(C(N2C(C(=O)NC)CC2)=O)CN(C(c2nc(C)oc2C)=O)CC1(C)C C1(CC(=O)NCc2cc(C)sc2C)CN(C(c2cnn[nH]2)=O)CCC1C C1(NC(CC(C)n2ccnc2)=O)CN(C(=O)CCCNC(N)=O)CCC1O c1(OC)cc(N)c(C(=O)NC(C(=O)O)C(C)c2ccccc2)cc1OC C1(CNC(C2OCCN(C)C2=O)=O)CN(C(c2n[nH]cc2Br)=O)CC12CCC2 C(=O)(CCC(F)(F)F)NC1C(OC)CN(C(C23COCC2C3)=O)C1 C(=O)(C(C)CCCOC)N1CCC(O)(CCNC(c2c(CC)cc[nH]2)=O)C1 CN1CCN(C(=O)CN2C(=O)NC(C)(c3ccccc3Br)C2=O)CC12CC2 CCC(C)(C)C(O)C(=O)NCC1CCCCC1C(=O)Nc1ccc(F)cc1C CCCCCC(O)C(=O)NC(c1cnn(C)c1)C(=O)NC12CC1CN(C)C2 C1(C)(C(=O)Nc2cn(CC(C)C)nc2)CCN(C(=O)CCCCC2CC2)C1 N1(C(CC(CCC)C)=O)CC(C(=O)Nc2cc(O)ccc2C)C2(CCC2)C1 N1(C(c2c(C)[nH]nc2Cl)=O)CCC(NC(C23CCCCC2C3)=O)CC1C N1(C(C2CC(=C)C2)=O)CCCC(CC(=O)NCC2CC3(C2)CC(O)C3)CC1 C(CNC(C1CC(=O)NC1(C)C)=O)(CC(F)(F)F)NC(C(CC)N(C)C)=O C(N=c1nc(O)c2c(ncn2C)[nH]1)C1CCN(C(c2c(C)nn(C)c2C)=O)C1 Cc1oc(CNC(C2CCCCN2C)=O)nc1C(=O)NCC(C)C(F)F C(=O)(N=c1[nH]onc1C)C1(CNCc2cnc(SC)nc2)CC1 c1(OC)ccc(C(C)NC(=O)CSc2ncccn2)c(C)c1.C(=O)C1CC1 n1(CC)cnc2[nH]c(=NCCc3nc[nH]c3Br)nc(N3CCC4(CC3)CSC4)c12 c1(C(C)(C)C)ccc(C(=O)NCC2CC(CNC(=O)C=C(Cl)Cl)CO2)[nH]1 c1(NC(Cc2cnc(C)s2)=O)ccc(N2CC(C)(C)C2=O)c(Cl)c1 Cc1c(NC(=O)N(C)CC2COCCO2)cnn1C(F)F C1(CC(=O)NC2CCC3CCC23)CCN(C(C2C3CCC(F)C23)=O)CC1 N1(C(C2(CC=C)CCC2)=O)CCCC(C(C)C)C1.c1(CC=O)ccc(F)cn1.N CCC(C)(COC)C(=O)NCC1CCCCO1.c1(C=O)cccnc1.C(C)C.N C1(C(=O)OC)CCCC1C(=O)NC1CC(NC(c2cc(Br)no2)=O)C1 c1(C(=O)NC2CCCC(N(C(=O)CNC=O)C)C2)ccc2ocnc2n1 CC(C)(C)C1=NOC(C(N2C3CCC2CC(NC(c2cc(=O)cc[nH]2)=O)C3)=O)C1 C1(C(=O)NC2(CNC(C(C)SCC)=O)CCCC2)CNC(=O)CC1C C(=O)(C1=COCCC1)NC(C(=O)NC(CCOC)CO)C1CCCC1 c1(OC)ccncc1C(=O)NC1CCCC1CNC(c1cccn1C)=O C(=O)(C1=NNC(=O)CC1)NC1C(F)CCN(C(c2ccc(C)c(F)c2)=O)C1 N#Cc1ccc(C(=O)NC2COCC2NC(c2ccc(CO)cc2)=O)s1 C1(CC)CN(C(=O)C(c2cccnc2)N(C)C)CC1C.C(C=O)(C1CC1)SC.N c1(OC)cnc(F)cc1C(N1CCN(C(C2(C)C=CCCC2)=O)CC1C1CC1)=O C#CCCCC(=O)N1CCC(NC(=O)CCOc2cccc(C)c2)C1 C1(CC=C)(C(=O)NCC2CCN2C(=O)C(O)CC2CCCC2)CC=CC1 c1(C(N2CC(CC(=O)OC)C(O)C2)=O)sc2cc(C)cc(C)c2c1Cl C1(NC(CC2C=CC(NC(c3c(C)non3)=O)C2)=O)CCCC(O)CC1 C1(NC(c2cnc(CCCC)s2)=O)CC2CN(C(C3(C(F)(F)F)CC3)=O)CC12 c1(C(N2CC(C3N(C(CCCOC)=O)CCC3)(O)C2)=O)cc(C(F)(F)F)ncn1 C(CC(N)=O)(C(=O)NC1CCCCC1(C)O)NC(C(C)n1cncn1)=O C1(CC)CN(C(=O)Cc2ccc(Cl)s2)CCC1NC(c1cc(OC)ncn1)=O c1(CC(=O)NC2CN(C3CN(C(C(CC)(F)F)=O)C3)C(=O)C2)ccc(F)c(Cl)c1 c1(NC(c2c(CC)cncc2)C)nccc(=NC(C)c2csc(C3CC3)n2)[nH]1 C1(CN=C(NC(C=C)C)NCc2snnc2C)CCCCC1(F)F C1(CC(N2CC(CC)(OC)C2)=O)CCCC(F)(F)C1.C1(C(=O)N)CC=CCC1 Cc1c(C(N2CCN(C(C3(C(F)F)CCC3)=O)CC2)=O)c(Cl)nn1C C1(O)(CCNC(c2cc[n+]([O-])cc2)=O)CCN(C(=O)Cc2cscn2)CC1 c1(C=O)ncc(C)cc1F.c1(CC)cc(C)c(C(=O)NCCC2CCCC2)o1.N Cc1cc(CC(=O)NCCN2CCN(C(C3CCCN3C(N)=O)=O)CC2)n(C)n1 c1(CNC(C2CCC3C2C3(F)F)=O)cc(O)nc(C)n1.C1(Cl)(C=O)CC1 Cc1cc(CC(=O)NC2CCOCC2NC(=O)CC(C)C(C)C)ccc1Cl C(=O)(C(CCC1CC=CCC1)N1CCOC(C2CCCOC2)C1)NCCCSC c1(CNCCC(C=C)C)cccc2c1NCCC2 n1(CC)ccc(C(N2CCC(NC(=O)CN3CSCC3=O)C2)=O)n1 c1(C(=O)NCC(C2CCN(C(CCC(C)(C)F)=O)CC2)F)cccn2cncc12 C#CCC(C)(C)C(=O)N1CCCC(O)(CNC(=O)CC(C)(C)c2ccccc2)C1 C1(C(=O)NCc2ccc(C)cc2)CN(C(=O)CCC2CCCCC2)CCC1(F)F C(=O)CC1=CCN(C)CC1.c1(C(=O)OCC)c[nH]cc1C(=O)N.C1CC1.C CCC(CN(C)C)CC(=O)NCC1(C)CCCN1C(=O)C=CSC C1(CC(=O)N)COCC1(C)C.C1(O)(C(C)C)CCN(C(c2csc(C#N)c2)=O)C1 C=CC1(C(=O)NC(C2CCCC2)CNC(=O)C(C)(C)CF)CCOCC1 N1(C(C=CCC)=O)Cc2ccnn2CC(NC(=O)C(CC)CC(F)(F)F)C1 c1(NC(CC2CCCN(C(C(CC(C)C)O)=O)C2)=O)cccc2ccncc12 c1(OC(C)(C)C(=O)NCCCO)cc(Cl)cc(Cl)c1.C(=O)(CCc1ccc[nH]1)N c1(CC(=O)NC(CC(=O)N(CC(O)CF)CC)C2CC2)ccc(O)cc1 C1(C(=O)NCC(=O)N(CCC)CC2CC2)CNC(=O)C1 n1(CC(=O)NCC(C)NC(=O)CCSC(F)(F)F)nnc(-c2ccsc2)n1 O=C1NCCCN(Cc2nc(-c3ccncc3)cs2)CC1(F)F CCCC(CCCNC(=O)C(CCC)NC(N)=O)NC(C1CC(N(C)C)C1)=O N1(C(C(CC)=CCCC)=O)CC(F)CC1CC(=O)N(CCC(=O)NC)CC C1(C(N(CC(C)NC(C(CC)=CC)=O)C)=O)CCN(CCC)CC1 c1(N(CCC)C(N2CCCC2)=O)ccc(C)cc1Cl.C(=O)(C(F)OC(F)(F)F)N c1(-c2cccc(C3(C)CCO3)c2)cc(O)cc(F)c1 N1(C(C2CC(F)CCN2C(C23CC2CNC3=O)=O)=O)CC(C2CCCCC2)C1 c1(CC(N2CCCC(CCNC(C(CSC)O)=O)C2)=O)c[nH]c2ccc(C)cc12 N1(C(CCCC)=O)CC2CC1CN(C(C1C=C(C)CS1)=O)C2 C(=O)(C(C)(C)CC#N)NC1C(CC(N2C(CC)CC2C)=O)CCCC1 CCC1=C(C(=O)N2CCCC2C(C)NC(=O)Cc2ccnc(F)c2F)SCCO1 c1(C(=O)O)cc(=NCC2CN(C(=O)C(CC3CCCC3)C(C)C)C2)[nH]cn1.CC c1(C(N(C)CC2(CNC(CC(C=C)CC)=O)CC2)=O)c(F)ccc2ccncc12 NC1CN(C(c2cc(C3CCCCCC3)no2)=O)CC12CC2 c1(C(N2CC(CNC(CC(CC)SC)=O)C(O)C2)=O)ccc2c(c1)CNC2=O C(=O)(C(CC)CCOC)NC1C2CC(NC(C3(OCC)CCC3)=O)CC21 N1(C(c2c(C)nc(C)s2)=O)CCN(C(=O)C(C)(C)O)CC1c1ccnn1C c1(C(=O)NC(CCOC)CNC(=O)C=Cc2ccsc2)cn2ncccc2n1 c1(OC)cc([N+](=O)[O-])cc(CN2CCC2(C)C(=O)Nc2cccc(I)c2)c1O C(=O)(NNc1ccccc1C(F)(F)F)NC(C)C(C)Oc1ccccc1.C(C(F)F)N C1(NC(C2C(C=C)CC2)=O)CCC(CNC(=O)CCc2cncs2)CC1 C1(C(=O)NCCc2scc(C)n2)CN(C(=O)CC2(O)CCOCC2)CCN1C C1(C=O)CC(=O)NC(=O)N1.CC(C)(C(=O)NCC1CC(O)C1)c1ccno1 C1(NC(=O)CC23CC(C2)C3)CCC2(CC1)CN(C(=O)CCF)C2 CCC(C)CCC(=O)NCC1(F)CC(NC(=O)C=Cc2cnc[nH]2)C1 C(CC(C)(C)C)(C(=O)NCC(C)CNC(C1CCC2(CC1)CC2)=O)OC N1(C(c2ccco2)=O)CCSCC1.C1(C2CC2)CC1.C=C1C(C=O)C1C=O.N CC1COCCN(C(=O)CC2CN(C(=O)C=C(C3CC3)C3CC3)CCO2)C1 C1(N(C(C=CCCC)=O)C)CCN(C(c2cc(C)c(C(F)F)cn2)=O)CC1C C1(CCC(C)C)CCN(C(c2ccc(C)s2)=O)CC1.c1(OC)ncc(C(=O)N)s1 S(=O)(=O)(C1CC(C(F)(F)F)C1)NCc1cc(CC)no1 c1(CC(N2C(C)CC(NC(=O)CCc3ccc(F)nc3)C2)=O)c(O)ncnc1O c1(C(NNC(c2c(C)nc(Cl)cc2)=O)=O)ccc(N)c(Cl)c1O CC1(C(N2CCCC2CNC(=O)Cc2ccno2)=O)CCC2CC2C1 C(=O)(CCCC(=O)C(C)(C)C)N1CCC(C)(CNC(C2C3CCCC23)=O)CC1 CC1CNc2c(C(N3CCCC(O)(Cc4nncn4C)C3)=O)cnn2C1 N1(C(C(CCC)C(C)C)=O)CC2(C=C(C(=O)N3CC(O)C(O)C3)CO2)C1 CC1(C(N2CC3CC(C2)N3C(C2CCC(F)(F)CC2)=O)=O)CC2(CCC2)C1 C(=O)(CC(O)CNC(C1CCC1)=O)N1CCC(N(C)C)C1 c1(-c2ccc(C)nc2)cccc2c(C(=O)Nc3cc(Cl)c(C#N)cc3F)c[nH]c12 c1(C(=O)NC2(CC=C)CN(C(=O)Cn3nc(C)nc3C)C2)cc(OC)ccc1F C1(NC(C(C2CCCCC2)OC)=O)CCCCC1CNC(=O)CCc1nccs1 C=C=C(C)CC(=O)NCC1(C)CCOCC1.c1(C(=O)N)cnc(C(N)=O)s1 C1(CNC(C(CC)OC2CCCC2)=O)C(C2CC2)CCN1c1ncc(O)cn1 C#Cc1ccc(C(=O)NC(C)CCNC(C2CC3(CCC3OC)C2)=O)nc1 Cc1ccc(CCC(=O)NCCOC2CCN(c3ncccn3)C2)s1 c1(NC(C2(F)CCN(C(C3CC(=C)C3)=O)C2)=O)ccc2cccc(Cl)c2n1 C1(NC(=O)C#CC2CC2)CCN(C(c2cnc(C(F)F)nc2)=O)CCC1CO C1(C#N)(NC(c2c(C)c[nH]c2)=O)CCN(Cc2ccc(C(C)(C)C)cc2)C1 c1(CN2CCCC(C(C)NC(c3c(C)nns3)=O)C2)cc(Br)c(O)cc1O c1(C(=O)NC2CN(C(C(C(C)C)N(C)C)=O)CC2C)cc2c(O)cc(Cl)cc2[nH]1 CCCCCC(CC)C(=O)NC1(CNC(C2CCCC2O)=O)CC(OC)C1 c1(Nc2ccc(-c3scc(C)c3)nn2)ccc(Cl)c(C2CC2)c1 C(=O)(CCCCCCC(=O)NCCC1(O)CN(C(C2(C)CC2C)=O)C1)OC CC1OC(C)C(C(=O)N(C)CC2CN(C(C3(C4CCCO4)CC3)=O)C2)C1C c1(OC)nccc(I)c1C(N1CC2CC2(CNC(=O)C)C1)=O.C(C)(C)C C1(NC(C2N(CC)CC2)=O)CCC(NC(=O)C(F)n2cccn2)CC1 c1(C(N2CCC(CC=C)(NC(=O)C3=CSCCO3)C2)=O)cccc(Cl)c1OC c1(C(=O)NC2COCCN(C(C(F)=CC)=O)C2)cc2c(s1)CCC(C)C2 C(CC)(C(=O)NCC1(OC)CN(C(=O)CO)C1)=CC.C1CCCOC1.C N1(C(COCCN(C)C)=O)CCCC(C2CC2NC(c2cccc(F)c2F)=O)C1 CC1CC(NC(c2cccc(-n3cccn3)c2)=O)CN1C(C1CC(CF)C1)=O C(C(C)(C)C(=O)NCC(C1CCCN(C(=O)C(Br)=C(C)C)C1)(C)O)SC c1(C(N2C3C(NC(C4C(C)=CCC=C4)=O)CC(C3)C2)=O)c(N)cc(Cl)cc1Cl C(c1c(F)ccc(Cl)c1F)=CC(=O)NCC(C)(C)NC(c1coc(Cl)n1)=O N1(C(c2c(CC)nc(C)o2)=O)CCC2C(C(=O)N(CC(C)C#N)C)C2C1 c1(CC(N2CC(C)C(CC)C2)=O)ccc(O)cc1Cl.C1(C2CC2)(CC=O)CC1.N CC1COCCN1CCNC(C1C=CC(NC(c2nc[nH]n2)=O)C1)=O C1(C)(CNC(c2c(CC)n(C)cc2)=O)CCC(NC(=O)CS)CC1.CC C1(C(=O)Nc2scc(-c3cc(OCC)ncc3)c2)CCC2CCC(=O)N2C1 c1(C(N2CCN(C(C(C)n3cnnn3)=O)CC2CCO)=O)cc(S(C)(=O)=O)co1 c1(C(=O)NC2C(NC(C(CC)(C)C)=O)CCC2)coc2c(F)cc(F)cc12 CCCCC(C(=O)NCCC1CCC(C)(C)O1)NC(=O)CCn1cccn1 c1(-c2cc(C=O)n[nH]2)cccc(Cl)c1.C(C(=O)NC1CC1)NC(=O)NC.N C1(C(=O)NCC(CC)(C)NC(=O)CCn2cccn2)(CO)CC(F)(F)C1 c1(CC=O)cnc(C)nc1O.C(C1CCCCC1)=CC(=O)N.C(C)(C)(C)OC C1(NC(CC(CNC(c2sccc2C)=O)OC)=O)CC(=O)N(C)C1=O N1(C(c2ccc(C#N)o2)=O)CCC2CN(C(=O)CCC3CCC3)CCC12 C1(Cn2cc(C3CC(NC(C(CCC)C)=O)C3)nn2)COCCC1(F)F c1(C(N2CCC(NC(C(COCC)N=[N+]=[N-])=O)C2(C)C)=O)cnc2c(c1)CCC2 C12(NC(C(C)SC)=O)CCC(CN(C(=O)CC3(C#N)CC3)C1)C2 C1(CC)CCC(n2nc(-c3cccc(C(F)(F)F)c3)nc2CCC(F)(F)F)CC1 c1(C(=O)NC(C2CCOC2)CNC(C(C#C)(C)C)=O)cnc(O)c2cnccc12 N1(C(c2cc(CC)ncc2)=O)CCC(CNC(=O)Cc2cnccc2Cl)C12CC2 C(=O)C(O)CC(C)C.C(CC(=O)N)C1(CCC#C)N=N1.C1(CC)(C=O)CCC1 C(CC(=O)NC1C(O)C2CCOC12)(C(F)(F)F)NC(c1c(C)cnnc1)=O c1(C(C(=O)N2CC(NC(C3(C(=O)NC)CC3)=O)C2)N(C)CC)ccccc1 C1(C(C(=O)NC2(C)CC2)N(C2CCOCC2)C2CC2)CC12CCOCC2 c1(NCC)ccc(C(=O)NCC(CO)NC(c2cc(N)nc(Cl)c2)=O)cc1F c1(COC(c2cc(OC)cc(F)c2)=O)ncn2ccccc12 C1(NC(C2(C)CCN(C(c3c(C)cc(N)cn3)=O)C2)=O)CC(C)N(C)CC1C c1(C(=O)N)cc2cnccc2[nH]1.C1C(O)C(O)CN1C(C1CC1C(F)(F)F)=O O=C1CCC(CC(=O)NCC2(CNC(C34CSCC3C4)=O)CC2)O1 c1(C(N2CCCCC2C2(O)CC2)=O)cnn2c1OCC1(CC1)C2 Cc1ccc(C(N2CCOC(CCNC(=O)CCC(=O)N(C)C)C2)=O)cc1O c1(C(N2CCC(C(C)NC(c3cnc(C)s3)=O)C2)=O)coc2cc(C)c(C)cc12 C(=O)(CC1=CCN(C(c2coc3ccccc23)=O)CC1)N(CCCO)CCC C(=O)(C(CCC(C)C)NC(C1CCC2(CCC2)O1)=O)N(CCCOC)C N1(C(C2(CCOC)CCC2)=O)CCC2(CC1)CN(C(c1cnn(C)c1)=O)C2 C=CCN=C(NCC12CCC(CC1)OC2)N1CCC(C(=O)N(C)C)C1 N1(C(C(CCOC)NC(c2cc(C)ncn2)=O)=O)CC(C2(C)CC2)C1 N1(C(CCn2c(C)ncc2)=O)CC(NC(c2ccn(C3CC3)n2)=O)C2CC12 C1(O)(CC(=O)NCCC(C)NC(COCC(=C)C)=O)COC(C)(C)C1 C=CCC(C)(CC)C(=O)NCCN(C(=O)CC1=CCOCC1)C C=C=CCCC(=O)N1CCC(NC(c2scc(C)c2C)=O)C1CC c1(NC(c2ncc(-c3cnc(OC)nc3)nc2)=O)cc(F)c([N+](=O)[O-])cc1F C=C1CCN(C(=O)C(=O)CCCC)C(C(=O)NCC(C)(O)C(=O)OC)C1 CC1(C)CC(CC(=O)NCC2CCCN2C(c2c[nH]nc2)=O)C1.C(C(F)F)O C(=O)(N1CCC(C(=O)NC2(CC(N)=O)CCC2)O1)c1c(OC)cncc1 c1(CC(=O)N(CCC)CCN(C(=O)C(C)OC)CC)ccc(F)cc1F.O n1(C(C)C)cc(C(=O)NC2CC2C(N2CC(NS(C)(=O)=O)C2)=O)cn1 Cc1ccc(C(N2CCCC(C(=O)NCC3(Cl)CC3(F)F)C2)=O)n1C N1(c2ccnc(S(C)(=O)=O)n2)CCc2ccccc2C1CNC(C1C2COCC12)=O C1(C(=O)OC)CCCN(N2CCCC(O)(C(F)(F)F)C2)C1C C(=O)(C1=CCOCC1)N(CCC(=O)NCC(O)CO)CC=C c1(C(N2C(C)CN(C(=O)CC3COC(=O)N3)CC2)=O)ccc2scnc2c1 C1(CCNC(CSCC=C)=O)CC(OC)CN1C(c1scnc1CC)=O c1(C(=O)NC(C2CN(C(=O)C3=COCC3)C2)C)cc2c(F)cccc2[nH]1 N1(CCOC)CC(C(=O)NCC2(F)CN(C(=O)C(C)CC)C2)CCC1=O.O C(=O)(C(CC)CCCC)N1CCC(CC=C)(C(=O)NC2C3CCC4C(C3)CC24)C1 c1(OCC)cccc2cc(C(C)NCC3(N4CCOCC4)CCSC3)oc12 N1(C(CSCC(C)C)=O)CCCN(C(C2CC3CCC(C2)C3O)=O)CC1C(C)C C1(C(=O)NC2(C#C)CCOC2)(NC(c2cc(C)no2)=O)CCC(C)(C)C1 c1(C(N(C(CCNC(C(CCSC)O)=O)C)C)=O)csc2c1CCCC2 CN1C(=O)OCC1C(N1CC2CC2(NC(=O)CC2(C)CC2)C1)=O Cc1nc(C(=O)Nc2ccnc(Oc3ccc(F)cc3F)c2)c2ccnc-2[nH]1 CC(CC(C)(C)C)C(=O)N1CC(NC(c2ccn3ccnc3c2)=O)C(F)C1 C1(S(N)(=O)=O)(C=O)CCCC1.Cc1cnccc1C=CC(=O)NC1CCC1.C c1(OC)ccnc(C(=O)NC(c2ccc(F)cc2)c2ccccn2)c1C C(=O)(CC1=CCOCC1)N1CCCC(N(C(c2ccc(C)c(Cl)c2)=O)C)CC1 Cc1cc(C)c(C(=O)NCCC2(NC(=O)CCCc3nncn3C)CC2)o1 N1(C(C2=C(C)CC2)=O)CC2CCC2(CCNC(c2cncc(Cl)c2)=O)C1 C1(CCC2N(C(CC3CCC(OC)CC3)=O)CCCC2)CCC(=O)NC1=O C1(CNC(CCOCCOC)=O)CCN(c2nnc(C)o2)C1 N(C(=NCCCN)NC1CCn2ccnc2C1)CC(C(=O)NC)(C)C.[SH](C)(=O)=O C12(NC(c3c(CC)scc3)=O)CCCCC1N(C(c1cnc(S)n1C)=O)CC2 Cc1nnc(CCNC(c2cc(CNC(c3csc(Cl)c3)=O)on2)=O)n1C C(=O)(C1=CCC2(COC2)OC1)N1C(CN(C)C(C2CCC(C)(C)C2)=O)CCCC1 C1(CNC(COCCC)=O)CC(F)(C)C1.C1(CC(=O)N)CC2CC2C1 C(=O)(C(C(CC)CC)OC)N1CCC(=C)CC1C(=O)NCCCN1CCCCC1 C(=O)(C(F)(F)CO)NC(C1CCN(C(Cc2n(C(C)C)cnn2)=O)C1)C c1(COC)cc(C(=O)NCCCCN(C(=O)C(C)(C)COC)C)ccc1F C(CC(=O)NC1CCOCC1C)(C(C)OC)NC(C1CC(O)(CC#C)C1)=O C1(C#N)(SC)CN(C(c2conc2C(C)NC(C2CCCN2C)=O)=O)C1 Cc1ccc(C(=O)NC2(C(=O)NCCN(CCCF)C)CC(CO)C2)c(O)n1 c1(OC)ccc(-c2cn(C3CCCN(C(=O)CCCCCSC)C3)nn2)cn1 N1(C(c2cccc(CC)n2)=O)CCC(C)(C)CC1C(=O)NCC(C)C1CC1 Cc1cc(=O)oc(C)c1C(=O)NC1CC2CCC1N2C(=O)C(C)C1CC1 C(=O)(CC(N)CCCCN)N1CCC(C(=O)OC)CC1 CCC(C)(C(=O)NCC1CCCCC1C(N1CC(N(CC(C)C)C)C1)=O)OC C1(NC(CCCC(C)=O)=O)Cc2ccccc2C1NC(C1(C#N)CCCCC1)=O Cc1cccc(C)c1C(O)C(=O)NCC1CCCCN1C(c1nnn(C)c1N)=O C1(CNC(c2nc(CC(C)C)sc2)=O)C2CCCC1N(C(c1ccco1)=O)C2 N1(C(C2(CC)CC2)=O)CCCC(C2CC2NC(c2c[nH]c(C)cc2=O)=O)C1 c1(CNC(C2OCCN(C(COc3ccc(C)cc3)=O)C2)=O)cccc(C)c1F C1(CNC(CCC(=O)NC)=O)CCN(C(=O)C(=Cc2ccncc2)C)CC1CO c1(OCCC(N2CCC(c3nc[nH]n3)CC2)=O)ccc(-c2nn[nH]n2)cc1 Cn1ccc2c(C(N3CCC4(NC(=O)C(=O)NCC(F)F)CC4C3)=O)cccc12 Cc1ccc(C)n1CCC(N1CCC(NC(=O)C(N2CCCCC2=O)C)CC1)=O C(CC(=O)NC1CCC(C2CC2)C1)(CC(C)C)NC(C=Cc1cc(C)no1)=O C=CC1(C(=O)NC(C2(O)CCC2)C)CCN(C(=O)CSCC(N)=O)CC1 c1(C(=O)OC)cncc2cc(C(N3CC(NC(=O)C(C)SC)C(C)C3)=O)ccc12 c1(CC(=O)NC2CN(C(CCC=C)=O)CC(C)C2)c(O)nc2[nH]nc(O)c2c1C N1(C(C(C)N(c2ccccc2)CC)=O)CCN(C(=O)CCC(N)=O)C(C2CC2)C1 C1(C2CCN(C(c3cc(C(C)C)cnc3O)=O)C2)CC1.C1(CC(=O)N)(OC)CC1 N1(C(C2OCCN(CC)C2)=O)CC2CC(NC(=O)CC)CC(C2)C1.C(C)(=O)O Cn1cc(S(=O)(=O)NC2CCCC2C(=O)Nc2cccc3nc[nH]c23)cn1 c1(C(=O)N)noc2c1CCCCC2.C1(F)(CNC(=O)CCC2CC2(F)F)CCC1 N1(C(C(C2CCC2)OCC)=O)CC(CO)(NC(=O)CO)C1.C1CC=CC1 c1(C(N2CCC(C(C(=O)NCC(C)OCC#C)F)C2)=O)ccc(O)c(C)c1 C1(NC(c2c(OC)n(C)nc2)=O)CCCCCC1NC(c1cc(O)nn1C)=O N1(C(c2ncc(C)nc2)=O)CCC2(CO)CN(C(=O)C(F)(F)CN(C)C)CC2C1 c1(OC)cccc(Cl)c1CC(=O)NC1CCCN(C(c2nnnn2C)C)CC1 c1(C(=O)NC(C)CCNC(=O)CCC(C)C#N)c(F)ccc(Br)c1Cl C1(OC2CN(C(C3(N=[N+]=[N-])CC3)=O)C2)CCN(C(=O)Cc2cccc(F)c2)CC1 CN=c1nc(N2CC(c3ccccc3)C(F)C2)[nH]c(=NCC2CC=CCC2)[nH]1 C(=O)(CCP(C)(C)=O)N1CC(C)C(NC(c2ccc3c(c2)CC3)=O)C1 N1(C(CC)=O)CCCC(C(=O)N(C2CCCCC2N(C(=O)CC(=O)NC)C)C)C1 C1(NCCC)CN(C(=O)CNC(=O)N(C)C)CC12CCC2 C(C1=CCN(C(=O)CC2NC(=O)NC2=O)CC1)NC(C1CCC(C)CC1)=O C(=O)(C1=COCCO1)NCCC1(NC(c2c(C#N)ccs2)=O)CCC1 c1(N(CCC)C)ccc(C(=O)NC2CC2NC(C2CCC2)=O)cc1 CC1=C(C)CC(C)(C(N2CCC3(CCC3)C2)=O)CC1.c1(CC=O)cc(C)cs1.N N1(C(c2cc(CCCC)oc2C)=O)CC2(CCN(C(C3CC3F)=O)CC2)C1 N1(C(CC(C)O)=O)CC(C)OC2(CCN(C(c3cn(C4CCCC4)nn3)=O)C2)C1 C#Cc1cnc(C(=O)NC2(CCNC(=O)C3=COCCC3)CCC2)c(C)c1 N1(C(CC2N(C)C(=O)CC2)=O)CCCOC(CNC(=O)C=CBr)C1 C(C1CN(C(=O)OC(C)(C)C)CC1C(=O)N(C)Cc1ncco1)=CC N1(C(c2c(C)cc(OC)nc2)=O)CCN(C(c2cccc(O)c2C)=O)CCC1C N1(C(Cc2cc(C)on2)=O)CC2CN(C(c3cccc(F)c3Cl)=O)CCC12 c1(OC)cnc(Cl)c(NC(C2C=CCN2C(c2cncc(C)n2)=O)=O)n1 C(CCC(O)C(=O)NC1(C)C(C)(C)C1(C)C)NC(CC1(C)CCC1)=O N1(C(Cc2ccc(C)c(F)c2F)=O)CC2CCCC1CN(C(C1CCCC1)=O)C2 c1(C=O)cc(F)ccc1C#N.C1(C=O)CC(F)(F)CN1C(C1CC1)=O.CC.O N1(C(c2[nH]c(=N)sc2)=O)CC2CCCC(CNC(C3CCCC34CC4)=O)(C2)C1 C1(OC(C2(CC(C)=O)CCCC2)=O)CCC2(CCCCC2)C1 c1(C(=O)NC2CN(C(C(C)SCC)=O)C(C)(C)C2)sc(S(N)(=O)=O)cc1C N1(C(C(C)(C)OCC(F)(F)F)=O)CC(C2CCCN(C(=O)C(F)C3CCC3)C2)C1 C1(NC(c2cc(Cl)ccc2O)=O)CN(C(=O)Cn2ncnn2)CC1C1CC1 C12CC(C1)C(C)O2.C1(C=O)CCOC(C)(C)C1.CC1CCOC1CC(=O)NC N1(C(c2cc(Cl)ccc2O)=O)CCC2(CC1)CN(C(C1CCCCC1O)=O)C2 c1(CNC(=O)NC2CC2)ccc(C(F)(F)F)cc1C#N.C1CCCCC1(F)F c1(OC)cc(OC)c(C(=O)NCCC(C)NC(c2nnc(S)n2C)=O)cn1 c1(C(N(CC(C)O)C)=O)ccn2cccc2c1.C(C)(C=O)OCCOCC.N C(C(C(=O)NCC1CCN1C(=O)CCN1CCCCC1)N(C)C)OC CC1SCCCC1C(=O)NCc1occc1C(=O)NC(C)C(F)(F)F c1(C(=O)NCC23C(CN(C(CC(=C)C)=O)C2)C3)cccc(OC(C)C)c1C C(CCCC(C)NC(c1cc(Cl)sc1Cl)=O)NC(COCCC=C)=O c1(COCC)nc(C=O)cs1.c1(C2C(C)(C(N3CCC3)=O)C2)ccccc1 N(C(=NC1CCCC1)N1CCC(C2CCC2)C1)C1C(C)C1.C12(CC1)C(=O)NC2 CCCCCC(CC)C(=O)NCC1(C)CCCN1C(=O)CC1CCCC(C#N)C1 c1(C(=O)O)cc(C2CC2)nnc1N1CCC(C)C1.C(=O)C(C)C(C)(C)C.CC C1(C(=O)OC)CCCC(NC(=O)NC2CCN(C=O)C2)CC1.C(C)(C)C.N c1(C(CNC(C=CCC)=O)NC(C2(SC)CC(O)C2)=O)cccc(O)c1 N1(CC(C)C)CCN(C(=O)C(C2CC2)NC(c2ccc(N)cn2)=O)CC1 c1(C2(C(N(CCCC)C)=O)CC2)cnccn1.c1(C=O)c[nH]cc1C(F)(F)F.N C1(NC(C2(C(C)C)CC2)=O)CCCC1NC(=O)C=C1CCC1 C(=O)(C(C)CCC(C)(C)C)NC1CC2CN(C(CN(CCOC)C)=O)CC21 c1(CC(=O)NCC23C(CN(C(c4cc(OC)no4)=O)C2)C3)cc(O)ccc1Br N1(C(C2(Cl)C(C(C)=O)C2)=O)CC(C(=O)NOCC(N)=O)C(C)C1 N1(C(c2c(C)cn(C)n2)=O)CC(C)CCC1CNC(=O)C(F)(F)c1ncccn1 c1(C(N2CCC(c3cn(C4CCCC4)nn3)C23CC3)=O)ccc2c(c1)OCCO2 N1(C(COCC(=C)C)=O)CCC2CN(C(C3CCC(=O)N(C)C3)=O)CC2C1 N1(CC(=O)N)CCC(O)(C2(c3ccccc3)CC2)CC1.C1(OC(C)(C)C)CCC1 c1(NC(c2c(CNC(CCn3ccc(C)n3)=O)cco2)=O)ccc2c[nH]nc2c1 N1(C(C(F)=CCC)=O)CCC(C)(C)CC1C(=O)Nc1cc(OC)ccc1C N1(C(C(CC)C)=O)CCOCCC1C(=O)NOCC(O)C(C)C c1(NC(C(C2CC2(C)Br)N(CCOCC=C)C)=O)ccccc1C C1(NC(c2nc(C)c(Br)cc2)=O)CCC12CCN(C(C1CCCO1)=O)CC2 N1(C(c2ccn(CCOC)n2)=O)CCCC2(CC2)C1.C1(C2CC2)(C=O)CC1.N CCC(C)C(O)CC(=O)NCC1CC1CC(=O)N(CCC(=O)NC)C C12(C=O)CC1COC2(C)C.c1(OC)oc(C)nc1C(=O)NC1(C)CCC1.N c1(N2CC(CO)CC(C(C)(C)C)C2)cccc(P(C)(C)=O)c1 CCS(=O)(=O)c1ccc(CN2CC(NC(c3ccc(I)c(Br)c3)=O)C(F)C2)cc1 N1(C(C2(CCNC(C3C(C)=CCS3)=O)CCC2)=O)CCCCC(C)(F)C1 c1(OC)ccc(C(=O)NC(CO)C(C)NC(=O)CCc2ccno2)c(Cl)c1.O c1(C(=O)NC2CC(F)(C)C2)ccc2nsnc2c1.C1(O)(C(=O)N)CCCCCC1 C1(CC#C)(NCCC2CCOC2)CCCCC1 CCC(CC(C)O)NC(=O)C=CCNC(=O)C=CC(=O)N(C)C N1(C(C(C(=O)OC(C)(C)C)C2CC2)=O)CCCCCC1.c1(CC=O)ccon1.N N1(C(CC(C)(C)O)=O)CCC2(CC1)CCN(C(c1cnc(N)c(N)c1)=O)CC2 c1(C(N2CCC(N(C)C(C3Cc4nnsc4S3)=O)CC2)=O)cnc2cc[nH]c2c1 c1(SCC)cnccc1C(=O)NCC1CCC(N(C)C(C2CC2C)=O)CC1 Cn1cnc(CCC(=O)NC2CC(CCC(=O)NCC(C)(O)C3CCCC3)C2)c1 S(=O)(=O)(c1cccc2cccnc12)NC1CN(C(C(=O)OCC)=O)CC(C)C1 C1(C(C(=O)NCC(C)C)N(CCn2cncn2)CC)CC2CCC1O2 N1(C(C(CCC(C)C)F)=O)CC2(CCCN(C(c3ccc(F)cc3)=O)C2)C1 c1(OCC)cccc(OCCCn2c(-c3cccc(C)c3)noc2=O)c1 C=CC1(CC(=O)NCC2C(C)CCCN2C(=O)CSCC(F)F)CCCCC1 C=CC(C)CC(=O)N1CCC(COC)(NC(=O)Cc2csc(Cl)n2)C1 C(=O)(CC1=CCOCC1)N.N1(C(C=CC(=O)OC(C)(C)C)=O)CCCC1C C1(NC(c2c(CNC(c3ccon3)=O)n[nH]c2)=O)CC2COCC(C1)C2 CCCC(C)(C)CC(=O)NCC(C)(C)NC(c1nc(CC)oc1C)=O C(=O)(C1CCc2nccn21)NC(CCC)C(O)C(=O)NCC1(CN(C)C)CC1 C1(F)(C(N(C)CC2OCCN(C(c3ccc(C(C)C)o3)=O)C2)=O)CCN(C)CC1 c1(CC)ccc(NC(=O)NC2CCCN(c3nccn3CC)C2)cc1Cl Cc1nc(C)c(CC(=O)N(C2CCC(CNC(=O)CC(F)(F)F)CC2)C)c(O)n1 Cc1ccc(CCNC(=O)C(=O)N(C2CCS(=O)(=O)C2)CCO)c(Br)c1 N1(C(c2cc(C)sc2C)=O)CCC(CCNC(C2(CO)CCOCC2)=O)CC1C N1(C(c2c(CC)occ2)=O)CCC2(CCCN(C(=O)C(C)C(=O)OC)C2)C1 c1(C=O)cccc(O)c1[N+](=O)[O-].C1(NC(=O)COC2CCC2)CC(CC)C1.N c1(C=O)cc(C(F)(F)F)ncc1F.N1(C(C2(OC)CCC2)=O)CCOC(C)C1.N C(=O)(C(C)CC(C)(C)C)N.C1(CC=C)CCN(C(=O)CC2CC(O)C2(C)C)C1 c1(CC)cccc2c1OCCC2NC(=O)NCC(=O)N(CC)CC N1(C(C2OCCN(C(c3c[nH]c(=NC)o3)=O)CC2)=O)CCC12CCCCC2 C12(NC(C(C)OCC#C)=O)COC(C1)C2.c1(C=O)ccc(-c2cc[nH]n2)s1 N1(CC)N=C(C(=O)N2CCN(C(=O)CC3CCCOC3)CC2C2CC2)CCC1=O N1(C(=O)Nc2ccc(CSC)o2)CCC(NC=O)C12CCCC2.C(C)(C)C c1(OC)ccc(C(N2CCCC(CN(C(=O)Cc3ccsc3Cl)C)C2)=O)nc1 C1(NC(C(C)C)=O)COC2CN(C(C3CC3[N+](=O)[O-])=O)CC12 N1(C(CC2(C)CC2)=O)CC(NC(=O)Cn2cc(Cl)cn2)CC(O)C1 N1(C(c2ccc(C)cn2)=O)CC2(CNC(=O)C(C)n3ccnc3)CCC1C2 C(C1c2ccccc2CCN1C(=O)C1=C(Cl)CC1)NC(C1(C(=O)NC)CC1)=O Cc1cc(=NCCn2ccnn2)[nH]c(=NCCOC2CCS(=O)(=O)C2)[nH]1 CCCCC(C)CCC(=O)N(CC(=O)NCCF)C(C)C C=CCC(C)C(=O)N(C1CCN(C(c2n[nH]c(C)c2C(=O)OC)=O)CC1)CC c1cn(C2CN(C(=O)CC3CCC3)C2)nn1.C(=O)(C=CC=O)OCC.N Cc1nn(C)c(Cl)c1C(N1CCC(F)C(NC(=O)C(C)OC2CCCCC2)C1)=O C=CCC(CC)C(=O)N1CCN(C)C(C(=O)N(C)CC2CCCCO2)C1 C1(NC(Cc2n(C)ccn2)=O)CC12CCN(C(=O)CC1OCCOC1(C)C)C2 C#CCCC(O)C(=O)NCC1(C(N)=O)CN(C(=O)C(n2ccc(C)n2)C)C1 Cc1c(C(=O)NCC2(F)CCN(C(C3CC(O)C3)=O)C2)cccc1CO N1(CC(=O)O)C(=O)NC(c2nc(-c3cccc(Cl)c3)no2)C2=C1COC2=O n1(C2CCCS(=O)(=O)C2)cnc2c(N3CCCC4(C=CCO4)C3)ncnc12 CCCCCCC(C)(C)C(=O)N1CC(N(C(=O)C(C)n2ccnn2)C)C(O)C1 c1(CC)ccc(C)cc1NNC(=O)c1nc2ccccc2nc1N Cc1nc(CCC(=O)NC(CNC(=O)C=CC2CCCO2)C(C)C)cs1 C1(C(=O)NC2CN(C(Cn3c(C)c(Cl)cn3)=O)CC2C)CCC2(CCCC2)CC1 C(=O)(CCCCCn1cnnn1)NCCN(C(=O)C=CCO)CC C1(CN(C(CNS(CC)(=O)=O)=O)C)C2CN(C(=O)C(C)c3ncco3)CC12 c1(CC)ocnc1C(=O)NC1(CNC(c2cocc2)=O)CCC1.N(C)C N1(C(c2c(OC)ncc(C)c2)=O)CC(C2CN(C(=O)CC(C)(C)C)C2)C1 C1(C(=O)NCCC)CCN(C(c2cn(C)cc2C)=O)CC1O N1(C(C(CC)(F)F)=O)CCC(NC(=O)C(O)C(C)CC)C(C)C1 N1(C(Cn2cc(C(=O)OC)nc2)=O)CC2CC(NC(=O)C(C)c3cc[nH]n3)C1C2 c1(OCCCC)cccc(C(N2CCC(N3CCOCC3)C2)CNC(=O)CC)c1 CC(C)C(C)(O)C(=O)N1CCC(F)(CNC(c2ccc(F)nc2F)=O)CC1 C=C1CCN(C(C(=O)NC2CC2)c2ncco2)CC1 C(CNC(=O)CC1(CC(=O)OC)CCCC1)(CCCC)NC(C(C=C)O)=O C12(NC(C=C=C(C)C)=O)CCC(NC(=O)CSCCN(C)C)(CC1)C2 n1(CC(=O)NCC(O)CCNC(c2nn[nH]c2Cl)=O)nc2n(c(=O)c1=O)CCC2 CCCCC(O)C(=O)NC12COC(C1)C(NC(c1cc[nH]c1C1CC1)=O)C2 c1(CC=O)ccccc1.C1(NC(CSCC)=O)CC(F)(C)C1.N(C)C.N N1(C(C2(OC)CCSC2)=O)CC2(CCCN(C(c3csc4ccncc34)=O)C2)C1 CC1CCC(Cl)=C(C(=O)NCCC(C)N(C)C(c2ccc(Cl)c(N(C)C)c2)=O)C1 c1(C(=O)NC2C(NC(C(CC)(C)OC)=O)CCCC2)ccc2oc(=N)[nH]c2c1 N1(C(c2scc(C(C)(C)C)n2)=O)CCC(O)(C(=O)NCC2CC3CC3C2)CC1 Cn1nnc2c1C(C(=O)NC1COCCN(c3ncc4ccsc4n3)C1)CCC2 C1(OC)CC(O)CN(C(c2ncc(C3CC3)o2)C(=O)NC2CCC2)C1 c1(CNCc2c(OC)ccc(C)c2)c(OCCO)nnc(C)c1C.C1CCCCC1 C1(C(=O)N)(CNC(C(C=C)OC)=O)CC2(CC2)C1.c1cc(C)c(C)o1.C c1(NC(=O)NCCC2CC2(Cl)Cl)ccc(Cl)c(N2CCCC2=O)c1 C1(CNC(c2cncc(C)c2)=O)CCC(C)CN1C(=O)COC1CC=CC1 N1(C(C2CCN(OC)CC2)=O)CCN(C(c2cc(Cl)cs2)=O)CC(O)C1 c1(OC)ccc(CC(=O)NC2CC2NC(=O)CCc2cn(C)nn2)cc1 Cc1cccc(C(=O)NC(C)C(C)NC(c2sc(N3CCCC3)nc2Cl)=O)c1O C1(OCCC)CCCC1C(=O)NC1CC(C)(NC(=O)CC2C=CCC2)C1 N1(C(CC2CCN(OC)CC2)=O)CCN(C(C2(C)SCCCS2)=O)CCC1C N1(C(CC(=C=C)C)=O)CCCC2(C1)CN(C(=O)C(c1cccc(OC)c1)O)C2 n1(CC)nccc1C(=O)NC(c1cn(C)nn1)C(=O)NCC1CCCO1.C c1(CCCC)cc(C(=O)NOCc2cn(Cc3cscn3)nn2)c(C)o1 N1(C(C2CC(NC(c3ccc(C#C)cn3)=O)C2)=O)CC2CCCCC2C1C CC(C)(CNC(C1(F)CCN(C(C2CC(=O)CCO2)=O)C1)=O)CCCO C(=O)(CCC)NC12CC(NC(CC)=O)(C1)C2.C(C)(C)C.CCO.C=O.O C1(OC)CN(CC2(c3ccc(Cl)cc3)CC2)C(C(=O)O)C1SC C1(CNC(C(CC)F)=O)CC(c2ccccc2)CN1C(=O)CCC(=O)OC C1(NC(c2n[nH]cc2[N+](=O)[O-])=O)CC12CCN(C(C1C=CC=CC=C1)=O)CC2 Cc1cnn(CC(=O)NC(CO)C(C)NC(=O)C(C2CCOCC2)C)c(=O)c1 C1(O)(CC(N2C(C(N3CC(CF)C3)=O)CSC2)=O)CCOCC1 C1(CC(N2CC(CCO)(NC(c3cc(C)nn3C)=O)C2)=O)CCC(C)(C)CO1 C(CN=c1[nH]c(=NC(C)CS(C)=O)c2[nH]ccc2[nH]1)c1c(C)[nH]nc1O c1(OC)cc(Cl)ccc1N1CCN(C(=O)C(N2CCOCCOCC2)=O)CC1 N1(C(C2C3(CC(NC(C4C(C(C)C)OCC4)=O)C3)C2)=O)CCOCC(C)(C)C1 CCCCC(C(=O)NCc1cc(Cl)no1)NC(c1cc(C)ccc1C)=O N1(C(c2cc(C)ncc2C)=O)CCC2(CC1)CCN(c1nnc(C(C)(C)C)o1)C2 C1(NC(CCC(=C)C)=O)COC2(C1)CN(C(C1CC(C(C)(C)C)=NO1)=O)C2 c1(N2C(C(=O)Nc3ncc(F)c(Cl)n3)CC(O)C2)ncnc2[nH]ccc12 CC1(CNC(c2ccccc2Cl)=O)CCN(C(=O)Cn2cnnc2)C1 N(C(=NCCCCn1ccnn1)NC1CCCCC1C)CC(N(OC)C)=O N1(C(=O)CSc2ccccc2)CC(NC(C2CCCNC2=O)=O)C(C)C1.C1CC1 C1C2CN(C(c3ccc(Cl)cc3)C3CC3)CC12.O=C(CCCC1CCOCC1)NC c1(NC(=O)Nc2cc(OC(C)(C)C)c(O)cc2)cc2c(nc1O)CCCC2 C(=O)C(C)(C)S(=O)(=O)C1CC1.CC1CCCCN1C(=O)Cc1c(Cl)cnn1C.N c1(C(N2CC3C(NC(C(CCCC)C)=O)C3C2)=O)ccc(Cl)c(C)c1OC N1(C(c2cc(CC)c(F)cc2)C(=O)NCC2CCCO2)CC(C)C12CCOCC2 C1(CC(NOCC#C)=O)C2CCCC2N1C(c1ccco1)=O N1(C(C2CC(C)(C(=O)OC)C2)=O)CC2CC(NC(C3C(C)C3C)=O)C1C2 C=Cn1nncc1C(=O)NC1COCC1C(=O)NC1(C(=O)NC)CCC1 N1(C2CCCN(C(C(CC)SC)=O)C2)CCN(C(c2ccnn2CC)=O)CC1=O c1(NC(N2CCC(NC3COCCC3(F)F)CC2)=O)cnn2c1OCC(O)C2 N1(C(C(C)(C)c2ccccc2)=O)CCOC(CC(=O)NC23CC(C2)C3)C1 c1(C=O)cc(C(F)(F)F)ncc1-c1ccc(C(F)(F)F)nc1.C1(CC)CCC1.N C1(CNC(CCCC(C)C)=O)CCC2(CCC2)C1NC(c1cscc1F)=O c1(C(=O)NC2C(NC(c3cc(C)c(C)nc3C)=O)C2)cnn2cccc(C)c12 C(=O)(C1SCCc2ccccc21)NC1CN(C(CCC=CC)=O)C2(C1)CCC2 N1(C(C(C)C(F)F)=O)CCC2(NC(=O)COc3ccn(C)n3)CCCC12 CC1(C)CN(C(=O)C#CC2CCOC2)CCC1NC(=O)COC1CCCCC1 Cc1ccc(C(N2C(C(=O)NCc3ccc(C)c(C)n3)CC2C)=O)c(O)n1 c1(CC)c(C(=O)N(C2CCN(C(=O)CC3CNC(=O)C3)C2)C)csc1C c1(C=O)ccccc1.c1(OC)ccc(C(N2CC(O)(C)C2)=O)s1.CC(N)=O.N c1(OC(C)C)cccnc1C(=O)NCCCN(C(=O)C(C)C1CCOC1)C c1(CNC(C2(CC#C)CC2)=O)cnn2c1CN(C(=O)C(C)N=[N+]=[N-])CC2 CC(C(C(=O)NCC1CC1)N1CCCCC1(C)C)C(C)(C)C N1(C(C2C(C)OCC2)=O)CC2CC(C1)N(C(=O)CC(O)c1ccccc1)C2 CCCC(C)CCCC(=O)NCC1CN(C(c2cnc(C)nc2COC)=O)C1 Cc1ccc(C)c(C(N2CC3(C2)CN(C(C2OC4CCC2C4)=O)C3)=O)c1N c1(C(N2CC(CNC(=O)CC3CCCO3)OCCC2)=O)cccc2c1CCOC2 N1(C(c2nc(CNC(CC(COC)C)=O)oc2)=O)CC2CC=CC1C2 c1(NC(C2CCN(C(c3ccccc3)=O)C2)=O)ccc(C2(CO)CCC2)cc1O C1(NC(c2c(C)ocn2)=O)(CO)CCCN(C(=O)C(=O)N(C)C)C1 C1(COC)C(OC)C(OC)CN1Cc1ccccc1OC(F)F N1(CCC)CCCC(C(=O)NCCCCCNC(c2ccc(CF)cc2)=O)C1 C#Cc1ccc(C(=O)NC2(C(N3CCC3CC(C)(C)C)=O)CCSC2)cn1 c1(C(=O)NC(Cc2ccco2)CCNC(C2(F)CCC2)=O)ccc(O)nc1 CN1N=C(CC(=O)NCC2OCCC2C(=O)NCCC(Cl)Cl)CC1=O Cc1nc2ncc(C(N3CCC4C(NC(=O)CN5CCSCC5)CC34)=O)cc2o1 C=CC(O)C(=O)N(C(C)C(=O)NC(C)(C)CO)CCC c1(OC)ccc(CC(=O)CNC2CCCN(c3cccc(N(C)C)c3)C2)cn1 C1(Nc2cc(N3CCC(COC)C3)ncn2)CCC(S(C)(=O)=O)CC1 N1(C(CNC(C)=O)=O)CC(NC(=O)CC2CCC(C)(C)CO2)CC12CCC2 C1(NC(CN(C(c2nc(C(C)C)oc2)=O)C(C)C)=O)CCC(C)(C)C(C)C1 CC(=NO)C1CC(C(=O)NCC(C)C2CC2)C1(C)C.C(=O)(C(C)C1CCC1)N Cc1ccc(C(O)C(n2cc(CN(C)C(c3nc(Cl)c(Cl)s3)=O)nn2)C)cc1 Cc1ccc(CC(=O)NCCOCCN(C)C(C2(C#N)CC(C)C2)=O)cc1C N1(C(c2cc(COC)no2)=O)CCCC(C)(C)C1C(=O)NC1CNC(=O)C1 C#Cc1cccc(OCC(=O)NCCNC(=O)CCc2ncco2)c1 c1(-c2cn(CCN(C(C(C3CCCC3)OCC)=O)C)nn2)cccc(OC)c1F C1(C)(C(=O)NCCN(CCC)C(c2ccc(Br)cc2)=O)CNC(=O)C1 c1(C(C)=O)cnn(C)c1C(=O)NCC(C)(C)NC(=O)C(C)c1cccs1 c1(C(=O)NCC2(F)CCN(C(CCn3ccc(C)n3)=O)C2)ccc2ncccn12 C(=O)(C1CCN(C)c2ccccc21)NC1CCN(C(C=COCC)=O)CC1C C1(C(=O)NC(c2cccc(Cl)c2)CC)CCCN(C(=O)CCOC)C1 C1(CC)CCCN(C(=O)CC2COCC2O)C1C(N1CC2CC1CS2)=O N1(C(CCSc2n(C)ccn2)=O)CC2(CCN(C(=O)COC(F)(F)F)C2)C1 c1(C(N2CCCCC2c2nnc(C3CCC3)o2)=O)ccc2c(n1)CCOC2 Cc1[nH]c2ccc(CNC(c3nccc(Br)c3F)=O)cc2c1C C(N=c1[nH]c(=NC2CC(CCO)C2)[nH]c2cc[nH]c12)c1c(C)n[nH]c1C Cc1nc(C(=O)NCC2CCCN2C(=O)CC2CCC(F)(F)C2)n(C)n1 C1(NC(C2CC(=O)N(c3ccc(F)cc3)C2)=O)CC2CC1N(C(=O)CCF)C2 C1(OCCCNC(C2(CC(=O)OC)CC2)=O)CCOCC1 C1(NC(C(F)=CC)=O)(CO)CCN(C(=O)CC)C1.C(=O)(CC(C)(C)C)N C=CC(C)(CC)C(=O)NC(C)C=CC(=O)NC1CCCC(O)C1 S(=O)(=O)(c1cc(C)cnc1NC1CCS(=O)(=O)C1)NCCCOC n1(CC)cnc(CCNC(c2cccs2)=O)c1.C(=O)(CO)NC1CC1 N1(C(c2ccc(C(C)=O)cc2)=O)CCC(CNC(C2CCCC2(C)C)=O)C1(C)C CCCCS(=O)(=O)CC(=O)NCC1C(C)CCN1C(C1CC1(Cl)Cl)=O c1(C(=O)NCCC=C)cc(C)c(-c2ccc(OCC(F)F)cc2)cn1 N1(C(CN(CCC)C)=O)CC=CC1(C(=O)N)COC.C1CCC(C(N)=O)O1 C(C1CCCCC1)=CC(=O)NCc1ncc(C(=O)NC)cn1.C1CCC1(F)F CC(CO)C(=O)NC1(C(=O)NC2CCNC2=O)CSC1 N1(C(C2(C)CC(C)C2)=O)C2CCC1C(CNC(c1ccsc1)=O)C2 CCC(CC(=O)NCC1CC2CC2N1C(=O)C(c1cn(C)nc1C)C)C(C)C c1(C(N2CC3N(C(C(CC)(C#N)CC)=O)C(CC3)C2)=O)cnc2ncc(Cl)cn12 C12(C(=O)NCCCOC)CCC(CC1NC(=O)Cn1cc(C#N)cn1)C2 C1(C(N(CC(F)F)CCOC)=O)CCN(C(=O)C23CCCC2C3(F)F)O1 Cc1cnc(NC(=O)C(c2cncn2C)N(C)C)nc1C CCCC(C)CCCC(=O)N(C1CC2CCC(C1)N2C(c1cc(C)c(C)o1)=O)C N1(CC(C)(C)NC(C2CCC2(C)C)=O)CCN(C(c2ccc[nH]2)=O)CC1 Cc1ccc(C(=O)NC2COCC2NC(=O)C(O)Cc2ccccn2)nc1 C=CCC(F)(F)C(=O)NCC(CC1CC1)C(=O)Nc1cnc(C2CC2)nc1 c1(-c2n(C(C)C(F)(F)F)nc(-c3cc[nH]n3)n2)[nH]c2ccccc2c1Cl CC1CC(C(=O)NCCc2cccnc2F)CN(C(=O)CN2CCNC(=O)C2)C1 N1(C(c2cc(OC)c(Cl)cc2)=O)CCC2C(=O)OCC2C1 c1(C(N(CCC(=O)NCCCC2C(C)C2)C)=O)coc2c1COC2 c1(NC(N(C2CCC3CC3CC2)CC2C#CC2)=O)cnc2ccnn2c1 c1(C(N2CCN(C(=O)COC3CCCC3)CC2)=O)cc(F)c(F)c(F)c1F N12CCC3(CC1)COC(C3)CNC2=O.c1(OC)cc(CN(C)C)ccc1CO C12(C(=O)Nc3ccc(CCN4CCOC4=O)cc3)CCC(F)(F)C1C2 CC(C)CC(O)C(C)C(=O)N(C(CC(C)C)C(=O)NCC1COC(=O)N1)C CCCCC(CNC(=O)C(O)CCCNC(C1CC(=O)C12CCC2)=O)CCC C1(C(=O)NCCCC2N(C(c3c(C)cn(C)c3)=O)CCC2)C2CCCCCCC12 C1(C(=O)N)Cc2cc(F)ccc2O1.n1(C(C)C)cc(C(=O)NC2CC(C)C2)nn1 c1(C(N2CCN(OC)CC2)=O)c(C)ccc(Br)c1F c1(CC)ccc(C(CC)(C(=O)O)NC(=O)N(C2CCOC2C)C)cc1 C#CCC(C)(C(=O)N1CCC1C1CCOCC1)NC(=O)CCn1ccnn1 N1(C(C(C)CC2CCCC2)=O)CC2CCN(C(=O)CCc3ccoc3)C2C1 C(=O)(CC(=O)N1CC(CC(=O)N(C2CC2C)C)(OC)C1)NCC#C C1(CC(=O)N(C(c2ccncc2)C)C)CCC(=O)N1C N1(C(C=CC)=O)CC2(CCC2)CC1CNC(c1cnc(NC)c(C)c1)=O c1(CN2C(CC)COCC2)cc2c(NCc3ccccc3Cl)cc(Br)cc2[nH]1 N1(C(C2N(CC)CC2)=O)C2CCCC1CC(NC(=O)CCC1CC1C)C2 C(=O)(C(C)(C)C(=O)N1CCC(COC)C1)NC.C1(CC=O)CC2CCC1CC2 c1(SCc2ccc(Cl)c(C)c2O)ccc(C#Cc2cn[nH]c2)cc1 c1(C(N(CCNC(CN(CCC#C)C)=O)C)=O)cc(N)ccc1F.C1CC1 c1(C(=O)N)cccc(-n2[nH]nnc2=N)c1.c1(CC)ocnc1C(=O)NC1CCC1 C(=O)(C(O)CCC(F)(F)F)NC1C(NC(c2cccc(OCC)c2)=O)CC1 C(C)(CNC(=O)C=Cc1scnc1C)(C(C)C)NC(CCCc1cc(C)no1)=O C1(CC(C)NC(C2(C)CCCC2)=O)CCN(C(=O)C(F)C2CCC2)CC1 c1(-c2cn(CC3CN(C(c4sc(C)c(Br)c4)=O)C3)nn2)ccc(S(C)(=O)=O)cc1 C1(CNC(C(C)(CO)OC)=O)CC(C(=O)N2CCCCCC2)=NO1 c1(C(=O)NCCOC(CNC(C)=O)(C)C)coc(O)n1.C1C(=O)N1 c1(C(=O)OC)cnn(C)c1NC(=O)CC1CN(Cc2cncs2)CCO1 c1(OC)cccc(C(=O)NC2CN(C(=O)Cn3cnccc3=O)C2)c1OC C1(NC(CCN(C(C(C)OCCN(C)C)=O)C)=O)CC(C2CCCC2)C1 C#CC(C)(C)C(=O)N1CCC(C(=O)Nc2cnccc2C)O1 O=C(C1=CCCOC1)NC1CCCC(NC(=O)C(c2ccc(F)cc2F)=O)CC1 CCC(CCC(=O)N1CCCC1CCNC(=O)CCC(=O)N(C)C)OC C1(C)(CC)COCCN1C(c1cnc(C)s1)C(=O)NC1CCOCC1 C(=O)(CS(=O)C(F)(F)F)N1CCN(CCCNC(CC(CC)(F)F)=O)CC1 n1(CC(C(=O)NCCC(CNC(C(C(=C)C)(C)C)=O)O)C)ccc2ccccc12 CC1CCCC1N=c1[nH]c(=NCCc2ccns2)[nH]c2c1CSC2 CC(C)C(C(=O)NCCCn1cc(CCN2CCCCC2)nn1)n1cnnn1 C1(C(N=S(CCOC)(C)=O)=O)COCC2(CCC2)O1 c1(NC(=O)Nc2cccc(-c3n(C)cnc3)c2)nccc(C#N)c1[N+](=O)[O-] C(=O)(C(C)P(C)(C)=O)NCC1CC(OC)CN1C(c1ccc(O)cn1)=O O=C(CCCCCBr)N(c1ncc(Br)c(N2CCOCC2)n1)CC1CCNCC1 c1(OC)ccccc1CN=C(NCC(N1CCCCC1)=O)NC1CCCCC1 C1(NC(c2cc(NC(C)=O)ncc2)=O)CC(F)CN(C(=O)Cc2ccnn2C)C1 C1(C(N2CC(O)(CC=C)C2)=O)CCCCCCN1C(=O)CCOC1CCC1 C1(CNC(CSc2n(C)ccn2)=O)CCCCN(C(c2ccc(CO)cc2)=O)C1 C1(O)(C(N2CCC(CN(C(CC(=C)C)=O)C)C2)=O)CCSCC1 N1(C(N(C)C)=O)CC2C(NC(c3cccnc3)=O)C2C1.c12cccc(c1)NC2 Cc1ccc(Br)c(OC(C2CCN(CC(F)(F)F)CC2)C)c1 C12CCCN(C(=O)Cc3cc(C4CC4)on3)CC1C2.N1(C(C)=O)CC(C=O)C1.N C=CC1CN(C(C2CCSC2)=O)CC1NC(=O)Cc1cncc(Br)c1 C1(C(N2CC(n3cc(C(C)=O)nn3)C2)=O)CCCCCCC1 N1(C(C=CC=CC)=O)CCN(C(C2CCC(C)CC2)=O)CC1CO c1(C(=O)OC)ccccc1C(F)(F)C(=O)N.C1(C=O)C2CCCC12.C1CCC1 c1(CC)cnc(O)c(C(N2CC3CC3(NC(=O)C(C)C#N)C2)=O)c1 C1(CC(=O)NC)CC2(CC2)CN1C(C1CC2(CC2)CO1)=O.C1CCCCC1O.C O=S(=O)(Nc1ccc(F)c(C(F)(F)F)c1)N1CCN(CC(F)(F)F)CC1 CCC(C(=O)N1CC(F)CC1CN(C)C(c1nc2ccccc2s1)=O)C(F)(F)F C1(C=C)(C(=O)NC2C(C#C)CCC2)CCN(C(c2nc(C)c(C)s2)=O)C1 C1CN(C(C2CC2(F)F)=O)C(C)(C)C1.C1(CC=O)(C=O)CCCC1.CC.O N1(Cc2ncc(C)s2)CCC(C2CCN(C(=O)Cc3cccc(C)c3Cl)CC2)C1 C(=O)(CCCC(C)(C)C)N1CCC(CCNC(c2c(C)noc2C(F)F)=O)C1 N1(CC(=O)N(CC(C)C(=O)N2CCC(OCCF)C2)C)CCN(C)CC1 c1(OC)ccccc1S(=O)(=O)N1CC(CO)(NCc2ccc(I)cc2O)C1 C(CCCCCC(=O)N1CCC(CF)C1)NC(c1ccc(C)nc1)=O N1(C(=O)CCc2cc[nH]n2)CCC2(C1)CN(C(C1CN=C3N=CNN3C1)=O)C2 c1(OC)ccc(C(=O)N(C)CC2CN(C(c3cnn(C)c3C#N)=O)C2)cc1C c1(C(N2CC3N(C(C(C=C=C)C)=O)CC(C3)C2)=O)cc(C)c2c(c1)CCC2 N1(C(C2C(OC)CC2)=O)CCCC(CNC(=O)CSCCC(F)(F)F)C1 c1(OC)cc(OC)c(C(=O)OCCS(=O)(=O)Cc2ccccc2)c(OC(F)F)c1 CC1CN(C(=O)CCNC(=O)C(N)=O)C12CCOCC2 n1(CC(=O)N(C2CCCCC2)C(=O)C(C)=C2CCC2)ccc(=O)n(C)c1=O Cc1ccc(F)c(C(=O)NCC2CCC(NC(C3(CCF)CC3)=O)CC2)c1 C(=O)(CCS(C)(=O)=O)N1CC2C(C(=O)NCCC(=C)CSC)(C2)C1 C1(C(=O)NCC2(CN(C)C(c3ccc(O)cc3)=O)CC2)C2CCCOC12 C(c1ccc(Cl)cc1)=CN1C(CNC(=O)C(c2cccc(Cl)c2F)F)CCCC1 c1(C(=O)OCCCN(C)C)cc(Cl)nn1-c1ncccc1Cl CCCCC(CNC(=O)C(CC(F)F)N(C(=O)C=CC(F)F)C)CCC c1(C(N2CCC(N(C(c3ccsc3OC)=O)CC)C2)=O)cc(C2CC2)ccn1 C1(NC(c2cc(C)n(C(F)F)n2)=O)CCN(C(C2(Br)CC2)=O)CC1O C1(O)(C(C)NC(CCN(C(CC)CC)C)=O)CCN(C(=O)CC2CC(OC)C2)C1 C1(C(C)C)(C(=O)NCC(=O)N(C)C2CC2)CCCN1C(C1C=CCS1)=O CCN=c1[nH]c(C)c(C(N2CC3CC(NC(c4cc(C)oc4C)=O)C(C3)C2)=O)s1 c1(OC)c(C)nc[nH]c1=NCC1CC(NC(c2cc(C)c(C)s2)=O)C1 C(=O)(CC(C)(C)C(F)F)N.Cc1ccc(CSCC(N2CCC(CC)C2)=O)cc1 c1(C(N(C(=O)NC2CCC2NC(C2CCC2)=O)CC)C)ccccc1 C(=O)(C1CCCn2nccc21)N1CC(NC(CCC)=O)CC1(CC)CC C1(NC(C2CC=CCC2)=O)COCCN(C(c2cc(C(F)(F)F)on2)=O)C1 c1(C(N2CCC=C(C(=O)N(c3cccnc3)CC)C2)=O)cc([N+](=O)[O-])ccc1F C(=O)(C1=NOC(C)C1C)N1CCC(OCC(=O)NCC(=C)F)C1 c1(C(NCCNC(c2ccc([N+](=O)[O-])o2)=O)=O)ccc2c(n1)CCC2.CC CS(=O)C=CC(=O)NC1CC(C)C1.c1(CCC=O)ccccc1OC(F)(F)F.N CCCCC(C(=O)N(CCCCNC(=O)C(C(C)C)OCC)C)C(C)C CCCCCCC(C)CC(=O)N1CC2CC1CN2C(c1c(F)cc(C)cc1F)=O C=C(Cl)CC(C(=O)NC1CCC(N(C)C)C1)NC(=O)CCCCC#N Cn1nccc1C(=O)NC1CCCC1CNC(C1(C)CC1(C)C)=O c1(CC)nc2c(C(N3CCC4CN(C(c5cccnc5)=O)CC34)=O)ccnc2[nH]1 C1(CC(=O)NC2CCN(c3cc(C(C)C)nc(Cl)n3)C2C)CC2(CCCC2)CO1 C1(C(=O)NC2C(C)CN(C)C2)CN(C(=O)CC2C=CCCC2)CCN1C Nc1cc(C(=O)NCC2(C(C)(C)C)CCN(C(C3CC34CC4)=O)C2)ccc1O Cc1nn(C)cc1C(N1CC=CCC1C(=O)N(C)Cc1ccnn1C)=O C=CC1(C(=O)NCC2(C)CC(C)=NO2)CCN(C(=O)C(C)n2ccnc2)CC1 CC(C)C(C)CNC(C12CCC(C1)C2)=O.C1(C(=O)N)CCC1c1nc[nH]n1 N1(Cc2c(C(C)(C)C)noc2)C(=O)CCN(CC2CC23CC3)C1=O N1(C(c2n(CC)ccn2)=O)CCOCC(NC(=O)Cc2cnn(C(C)C)c2)C1 C(C(N=c1ccnc(S(C)(=O)=O)[nH]1)C1CC1)NC(C1C(C)(C)CCC(F)(F)C1)=O C12(CNC(CN(C)C)=O)CCC(CN(C(c3cn(C)nc3C(F)F)=O)C1)C2 C(=O)(C(CC1CCC1)NC(c1ccn(CC)n1)=O)NCCCC=CC Cc1cccc(F)c1C(=O)CN1CC(CO)C(c2ccccc2)C1 N1(C(C2CC(OC)C2)=O)CCC(F)(CNC(C2(Cl)CC2(C)C)=O)CC1 Cc1ccc(F)c(C(=O)NCc2nc(C(=O)N(C3(CO)CC3)C)c(C)o2)c1 c1(OC)nc(C(=O)N(C2CCN(C(c3snnc3C)=O)C2)CC2CC2)ncc1F c1(OC)cc(C(=O)NNC(=O)Cn2cc(C3CCOC3)nn2)cc(OC)c1OC CC(C)CC(C(=O)NC(C1CCC(F)(F)CC1)CCO)NC(=O)C(C)(C)C c1(C(=O)NCCC(=O)N(C2C(OC)COC2)C)cnc(C)cc1C N1(C(CC2(C(=O)N(C3(COC)CC3)C)CCC2)=O)CCCC(OC)CC1 N1(C(C2CC(=O)NC2)=O)CCC(C(F)(F)F)CC1.C1(C=O)CC(=C(F)F)C1.C CCCCCC(CC)C(=O)NC1CCN(C(=O)Cc2c(C)nn(C)c2C)C(C)C1 C1(C(N(CC(C)NC(=O)C(C)(Cl)Cl)C)=O)CC(=O)N(C)C1c1ccnn1C Cc1cc(C)c(-c2csc(C(=O)NC(C)(C)C)n2)cc1C.c12ccccc1N2 C1(Oc2ccc(OC)cc2)CCOC12CCCCC2.C1(C)CC(=O)O1 C(=O)(C(C)C(C)NC(c1ccc(C)o1)=O)OC.C(=O)(C=CC(F)F)N C(=O)(C1Cc2ccccc21)NC(CC1CCN(C(CSCC#C)=O)CC1)C C1(CC)(CC)CCN1C(c1nc[nH]n1)=O c1(C(=O)NCC2C(C(F)(F)F)CN(C(CC)=O)C2)ccc(C#N)cc1F c1(C=O)ccc(C(F)(F)F)c(C)c1N.N1(C(C=CC=CC)=O)CCCCC1.C C(C)(C)(CN=c1cc(C)[nH]c(=NCC(C)C(C)(F)F)[nH]1)SC Cc1sc(N)c(C(=O)NC(CNC(C2C3CCC2CC3)=O)C2CC2)c1C c1(C(=O)NC(C2(O)CN(C(C3SCCCS3)=O)C2)C)cnc2occc2c1 c12cc(cc(OC)c1OC)CNC(=O)c1cccc(c1)CS(=O)C2.C=CC C(C(C)(C)CC(=O)N(C)C(c1ncccn1)C)NC(CN1CCC(C)C1)=O c1(C(N2CCC(CNC(C(N3C(=O)CCC3=O)CC)=O)C2)=O)cc(O)nc(O)n1 c1(C(=O)N)ccc(=O)n(CC)c1.C1(CC(=O)N(C(C)C)CC)CCCC1 CN1CCOCC1C(=O)NC1CC2(C1)CC2NC(=O)C=Cc1cncs1 N1(C(C(C)(C)C)=O)CC2C(C(N3CCCC(C(N)=O)C3)=O)C2C1 c1(C(=O)NCC(CC)C(C)C)ccc2c(n1)CN(C(=O)C1=CCCOCC1)CC2 CCCC(C)(O)CNC(C1CC(=O)CN1C(C1(C)CC(F)(F)C1)=O)=O C1(NC(C(CN(C(COCCC(C)C)=O)C)C)=O)CN2CCC1(C)CC2 c1(C(N2C3C(NC(=O)C4=NOCC4)C(C3)C2)=O)cnn2c1CCC2 C1(OC)CN(C(C2CC(O)CN2C(c2ccc(I)cc2)=O)=O)CC1OC C(=O)(C1=C(C)OCC1)N1CCCC(N(C(c2c(CC)n(CC)nn2)=O)CCF)C1 CC1(CNC(C2CCSCC2)=O)COCCN(C(=O)COC2CC2)C1 C(=O)(CCCCCCCCC1CC1)N1CC(CNC(Cc2c(C)cc(C)s2)=O)C1 CC(CCS(C)(=O)=O)(c1nnnn1C1CC1)NCC1(CO)CCCOC1 C#CC1CCC(NC(=O)C(C)(C)NC(=O)C=CCO)C1 C1CN(C(=O)C=Cc2cnc[nH]2)C(C)(C)C1.C1(C(=O)N)(SC)CCOCC1.C N1(C(C(C(CC)C)O)=O)CCOC2(C1)CN(C(=O)C=Cc1csc(C)n1)C2 c1(C(N2CC(N(C)C(C3CC3C(N)=O)=O)C2)=O)ccccc1CO CC(C)C(C(=O)N(C)C)NC(=O)COCC(=O)NC1C2CC(CO)CC12 C1(C(C(=O)NCCOC)N2CCC2c2cccc(F)c2)CCC2COCCC2C1 c1(C(=O)NC2(COC)CN(C(C(C(=C)C)(C)C)=O)C2)cn2cnnc2cn1 CCC(CCCC(=O)N1CCCCCC1CCO)NC(c1c(C)nn(C)c1C)=O N1(C(c2n(C)ncc2C(F)(F)F)=O)CCOCC(NC(C2(C)CC3CC3C2)=O)C1 C1(C(=O)NC(CNC(c2c(N)cncc2)=O)CO)CCCCN1N=O c1(C(N2CCC(NC(C=COCC)=O)C(C)C2)=O)cccc2c1OCC2C c1(C(=O)NC2C(NC(Cc3c(CC)con3)=O)CCC2)nc(C)c(C)s1 N1(CC(=O)N)CCC(=O)NC1=O.c1(CCC(=O)NCC2CCCC2)ccccc1 C1(CNC(C(CC)F)=O)CC2(CCC2)CN1C(c1nn(C)cc1C)=O C1(NC(C2(C(=O)NC)CC2)=O)COC2CCOC12.C1CCCCO1.C(=O)C.N C(=O)(CC(F)(F)C(F)(F)F)N1CC(NC(c2ccn(C3CC3)n2)=O)C(F)C1 N1(C(C(C)=C2CCC2)=O)CC=C(C(C)(C)C(=O)N2CCC(CCN(C)C)C2)C1 c1(C(=O)NCC(C)(CNC(C2COCCN2C=O)=O)OC)cccc2nn[nH]c12 N1(C(C=CS(C)=O)=O)CC(NC(=O)C=Cc2ccc(Cl)cc2)CC2(CC2)C1 c1(C(N2CCCC(C)C2)=O)n[nH]c2ccccc12.C1(C(F)(F)F)(C(=O)N)CCC1 N1(C(CCCOCC)=O)CC2(CC(NC(c3nsnc3O)=O)CO2)C1 N1(C(CC2N(C(C(C)NC(=O)OC)=O)CCC2)=O)CCC(O)CC1C C1(CCNC(CCNC(=O)OC)=O)CN(C(=O)CCc2ccsc2)CC1C C(=O)(C(CO)NC(=O)C(C1CCN(C(=O)Cc2cccn2C)C1)F)N(C)C Cc1ccc2[nH]cc(C(=O)NC3CCC(C)N(C(C4CC4C(F)F)=O)C3)c2c1 c1(OC)cc(C(C)NC2CC=CC(N)C2)ccc1OCCC(C)C N1(C(COc2c(CC)cccc2)=O)CCOCC(NC(C2(C)CCN(C)C2)=O)C1 C(=O)(C(N)C(=O)NCc1ccc(N2CCSCC2)cc1)OC C#Cc1cc(NC(=O)C(CCSC)NC(c2cc(Cl)n[nH]2)=O)cc(F)c1 C1(CC(=O)NCCOCCC(N2CC(C)(O)C2)=O)CCCC12CC2 C1(C)(COC)CC(NC(=O)C)CN1C(c1ccoc1)=O.[SH](C)(=O)=O.N C12(CN=c3nc(C(C)(C)C)[nH]s3)CCCCC1CN(C(=O)CCCNC(N)=O)C2 N1(C(CC=CC=C)=O)CCN(C)CC1CNC(=O)CC1(C=C)CCC1 c1(CNC2CC(C(=O)Nc3ccc(N(C)C)cc3)C2)ccc([N+](=O)[O-])cc1F C=CC1(C)COCCN1C(C(=O)NC1CC1)C1COC1 C=CC(C)(CC)C(=O)NCCCNC(=O)C(C)Cc1ccc(O)cc1 N1(C(c2c(C)nc(CC)o2)=O)CCN(C(c2ccc3ccoc3c2)=O)CC(O)C1 c1(C(N(C2CCN(C(=O)C#CC3CCOC3)CC2)CC)=O)n[nH]c2c1NCCC2 c1(C(=O)OCC)n[nH]c2c1CN(C(=O)NCCc1c[nH]c3ccc(C)cc13)CC2 N1(C(C(C)NC(C(C)=NOCC#N)=O)=O)CCN2CCCC2C1 C(=O)(CN=c1cc[nH]cc1)N(C(CC)C(=O)N1CC(C)(c2ccccc2)C1)C c1(C(=O)NCC2C(NC(CNC(CC)=O)=O)CC2)ccc(Br)cn1 CP(C)(=O)c1ccccc1C(N1CC(C2(NC(C3CC3C#N)=O)CC2)C1)=O C1(CC=O)CCC(C)(O)CC1.N1(C(C2CC(SC)C2)=O)CCC(=CC)CC1.N Cc1noc(C)c1NC(=O)CN1CCN(C(=O)COc2ccncc2)CC1 C(=O)(C1CCCc2nc[nH]c21)NC(c1c(OC)cccc1)CNC(C1CCC1)=O c1(C(CCc2ccccc2)N(CC)CC)ccccc1OC(=O)CC1CC=CC1 C1(C(N2CCCC(C(C)C)C2)=O)CCCN(C(c2ccncn2)=O)CC1 C1(NC(CCC=C(C)C)=O)CCCC(NC(c2cccc(C(N)=O)n2)=O)CC1 Cc1ccc(C(=O)NCC(C)NC(c2cccc3nonc23)=O)c(Cl)c1C N1(C(C(c2ccc(CC)cc2)(C)C)=O)CCC(C)(C)C1.C1(O)(C=O)COC1.C N1(C(c2nccc(CC)c2)=O)CCN(C(c2ccc(Br)cc2O)=O)C(C2CC2)C1 Cc1cc(C(=O)N(C2CN(C(C3(CC4CC4)CCC3)=O)CC2F)C)c(C)s1 c1(CC=O)ccc2c(c1)CCO2.c1(C(=O)NC(C2CCC2)C)ccc(Cl)[nH]1.N c1(C(N(C2CCN(C(C(C#C)(C)C)=O)CC2C)C)=O)cc2ccccc2cn1 N1(C(C2CCc3c(ccc(C)c3)O2)=O)CC(C)C(N=c2[nH]c(Cl)ncc2Cl)C1 C1(C(=O)NC2(C(=O)OC)CC2)CCC(O)CN1C(=O)CC1(O)CCCC1 N1(C(C(C)(c2ccccc2)OC)=O)CCC(NC(=O)CCCC2CCC2)C(C)C1 c1(CC(=O)N(CC#C)CC)c(C)cccc1Br.c1(C=O)cc(C)c(N)cn1.O C1(S(C)(=O)=O)(C=O)CCC1.CC(C)C(C(=O)NC(C)C1CC1)N(C)C.N c1(C=O)ccc([N+](=O)[O-])cc1Cl.C1(CC(=O)N(CCC)CC)CNC(=O)C1.N C1(C(N2CCN(C(c3ccnc(C)n3)=O)CC2)=O)CC2CCC1C21CC1 C=C1CC(C(N2CC(OC)C2)=O)(CNC(=O)CC(C)n2cccc2)C1 c1(C(N2CCN(CCNC(=O)C=Cc3cnc[nH]3)CC2)=O)ccc(Br)c(Cl)c1 c1(N2CCC(NC(C(C3CCCCC3)OC)=O)C2)ncncc1Cl c1(N2C(CNC(c3cc(C)[nH]n3)=O)CCCC2)nc(O)c2c(ncn2C)n1 C1(NC(c2[nH]cc(C#N)c2)=O)CCCCCCC1NC(c1ncc(Cl)cc1O)=O c1(C(N(C2CN(C(C3CCCS(=O)(=O)C3)=O)C2)C)=O)cc(=O)cc(Cl)[nH]1 C1(C(N2CC(OC)C2)=O)CCC(NC(=O)COC(F)(F)F)CC1 CC(=NO)C1CC(C(N2CCN(C(=O)CCCC(C)C)CC(C)(C)C2)=O)C1(C)C Cc1cc(C(N2CC3CCC2C(NC(C2CCC=CCC2)=O)C3)=O)c(N)c(C)c1 N1(C(C2(Cl)C(C(C)=O)C2)=O)CCN(C(C2C=C(C)CS2)=O)C(C)C1 c1(NC(C(C(C)NC(=O)CN2CCCCC2)C)=O)ccc(Cl)cc1O N1(C(COCCC)=O)C2CCC1CC(NC(=O)CC1CN3CCC1CC3)C2 N1(C(c2c(C3(C)CC3)cccc2)=O)CC2=C(C1)CN(C(c1ccc(F)cc1)=O)C2 CCCC(CC)C(=O)Nc1cccc(CNC(c2cscc2Br)=O)c1 C1(NC(C(C2CC=CCC2)NC(CCCC)=O)=O)C2CCCC1CC2 C(=O)(CC(CC)C(F)F)N1CCC(NC(CNC(CCC)=O)=O)C(O)C1 C#CCCCCCCC(=O)N(C(C)CCNC(c1ccc(C(=O)NC)cc1)=O)C N1(CC)CCN(C(C2C3(C)CCC(C3)C2(C)C)=O)CC1(C)C C(C(C(=O)N1CC(C)(O)CO1)C(C)(C)C)NC(C=CC(=O)OCC)=O CP(C)(=O)C1CCCN1C(c1cccc([N+](=O)[O-])c1)C(=O)NC1CC1 c1(OC)nn(C)cc1CNC(=NCC1CC1)NCCc1ccncc1C C1(COCC(=O)NCC2CCN(C(c3ccncn3)=O)C2)CCCOC1 c1(C(=O)NC2CCCN(C(CCN(C)CCO)=O)CC2)coc2cc(F)ccc12 C1(C(=O)NCCN(C(CCCCC#C)=O)CC(C)O)CC2(CCC2)CCO1 C1(C(=O)NC2(CC)CCCC2)(NC(c2cnccn2)=O)CCCC1C c1(CCC(=O)NC2CC2NC(C2CCC2)=O)cc(Br)nc(Br)c1 Cc1c(C(=O)NCC2CCC(F)(F)CO2)cccc1S(N)(=O)=O c1(OC)ccc(C(=O)NC2CC(C)CN(C(c3cc(Br)nc(Br)c3)=O)C2)cc1I CCC(CCCO)N=c1nc(N2CC3C(CO)C3C2)c2c([nH]1)c(C)nn2C c1(C(=O)NCC23OCCC(C)(C2)C3)cnn2c1CCCC2 N1(C(=O)NC(C)Cc2nc[nH]n2)CCC2(CCCN2C)C1 Cc1sc(C=O)cc1S(N)(=O)=O.C1(C)(C(N2CC(F)C2)=O)C(C)(C)C1(C)C C=C(C)CC(=O)N1CC(CNC(C2(CC)CCCC2)=O)(OC)C1 C=CCCCC(=O)NCC1CC(NC(c2ccccc2)=O)C1(C)C.C(C)=O.C N1(C(C(CCC)C)=O)CC2OCC(NC(c3nc4ncccn4n3)=O)C2C1 c1(NC(C2CN(C(c3ccn(C(C)(C)C)n3)=O)C2)=O)cc(F)c(C#N)cc1F C1(C(N(C)Cc2cncn2C)=O)CN(C(c2c[nH]c(=N)o2)=O)CCO1 c1(C=O)cnn2c1OCC(C)C2.C1(CC)CCC1.C(C(=O)N)N(C1CC1)CC c1(C2CCCN2C)cc2c(s1)CCC2.c1(N(CC(C)(C)C)C(=O)C)ccccc1 N1(c2ccc(C#N)nn2)CCC(F)(F)C(CNC(C2CC(=O)NC(=O)N2)=O)C1 CC1=C(C(=O)NC(CC(C)(C)C)C(=O)NC(c2ccncc2F)C)SCCO1 c1(C(N2C(CN(C(C=CSC)=O)C)CCCC2)=O)cncn(C)c1=O c1(CC)ccnc(C(=O)NC(C)CCCNC(C2CCC(OC(F)F)CC2)=O)c1 c1(OCC=C)cccc(C(N2CCC(c3ccc(Br)cc3)C2)=O)c1O N1(C(c2c(CC)non2)=O)CC(CCNC(C2(CCO)CC2)=O)OC(C)C1 CC1CCc2[nH]nc(C(N3CC(C4CN(C(C5(Cl)CC5(C)C)=O)C4)C3)=O)c2C1 C(=O)(CCCCC(C)C)NC1CCC(NC(C2CC(C)(C(=O)OC)C2)=O)CC1 C(C(C)(O)CNC(c1nonc1N)=O)NC(C=CC(CC)C)=O c1(N2C(CCCNC(CSSC)=O)CCC2)cc(C)nc(C(C)(C)C)n1 CCCCCCCCC(=O)N1CCN(C(c2cc(Cl)n[nH]c2=N)=O)CC(O)C1 c1(C(=O)NCC(O)CNC(C2CC3C=CC2C3)=O)cc2c(s1)COCC2 Cc1ncc(C(=O)NC2(C(=O)NC3C=CCCC3)CC2C)n1C N1(C(c2cc(C)n(C)n2)=O)CC2(CCN(C(c3cc(Cl)sc3Cl)=O)C2)C1 C1(c2n(CCOC)nnn2)(Nc2ccc(Cl)c(Cl)c2)CCN2CCCC2C1 CCCC(O)C(=O)N1CC(NC(C2CC(CF)C2)=O)C(C)C1 CCCCC(C(=O)NC)NC(C1(C)C=CCN1C(=O)CCn1ccc(C)n1)=O CS(=O)CCC(O)C(=O)NCC1(F)CCN(C(=O)CCF)CC1 CCN=c1[nH]c(C(=O)NCC2CC3CN(C(c4cnc(C)cn4)=O)CC23)cs1 C1(C(=O)OC)C2CC1N(C(=O)C#CCNC(C1CCC=CCC1)=O)C2 Cc1ncc(-c2cn(C3CN(C(=O)Cc4ccn(C)n4)C3)nn2)n1C c1(NCC(c2ncc[nH]2)C)cc(NCc2cnc(CN(C)C)s2)ncn1 N1(C(C2C(c3ccc(C)o3)C2)=O)CC2(CC(NC(=O)Cn3ccnc3C)CO2)C1 c1(OC)ccc(C(=O)NC(CNC(c2c[nH]cc2Br)=O)C(C)(C)C)c(C)c1 C1(NC(C(=O)NCC2CC2)=O)CN(C(=O)Cn2cnnn2)Cc2ccnn2C1 C1(C(N2CC(OC)C(C(=O)N(C(C)CSC)C)C2)=O)CC2CCCC2C1 c1(C(=O)NC2C(CC)CC2)cc(CNC(=O)CC2CCC(C)CC2)ccn1 Cc1ccc(O)c(C(N2CCC(NC(C3CC4OC3C3CC43)=O)CC2)=O)n1 N1(C(CCSCC(N)=O)=O)CCC2CCCCC12.C(=O)(C1=CS(=O)(=O)CCC1)N C1(NC(CCSC)=O)CCN(C(C2(CC3CC3)CCCO2)=O)CC1 C12(NC(=O)CC3CCC4CC34)CCC(CC1)N(C(c1nnc(O)nc1O)=O)C2 c1(C(C)C)cccc(N(C(C)(C)C)CC#N)n1.C(=O)O C(=O)(C(C(C)(C)C)NC(=O)Cn1ccnn1)NC.C(=O)CCCN(C)C.C c1(N(C)CC2CCC(OCC)CC2)ccc(S(N)(=O)=O)cc1C N1(Cc2n(CC)c(C)nc2)C(=O)CCN(CC2CC(N(C)C)C2)C1=O O=C1NCc2c1ccnc2C(=O)NC1CCN(C(=O)Cc2ccc(O)c(F)c2)C1 CC1CC(NC(c2cnn(C)c2-n2cnnc2)=O)CN1C(c1ccsc1)=O Cc1nc(N2CCC(CNC(=O)CCc3cnoc3)C2)cc(SC(C)C)n1 C1(OC)CN(Cc2n[nH]cc2Cl)CCC1NC(c1cc(Cl)ccn1)=O C1(C(N)=O)Cc2nc[nH]c2CN1C(=O)NCC1OCC2CCC1C2 Cc1ccccc1CC(=O)NCCCNC(C1OCCC1(C)C)=O N1(C(CC(CNC(c2cnc(C)s2)=O)O)=O)CC2CC2C2CC12 C1(C(=O)OC)C(O)C(O)CN1C(c1ccc(C2CC2)cc1Cl)C(=O)N.CC(F)F O=C(CC1CCc2cc(Br)ccc21)NC1CCCC12CCN(C(=O)C1CC1)CC2 c1(NC)ccc(C(=O)NCC2(C)CCCN(C(c3nnn(C)c3N)=O)C2)cc1F CCC1=C(C(=O)NC2CC3C(NC(C4(Cl)CCC4)=O)C3C2)CCCO1 C(=O)(C1=CC(O)C(O)C(O)C1)N1C(C2CCN(C(C(C)NC=O)=O)C2)CCC1 c1(OC)ccccc1C(C)CC(N1CCC(NC(=O)C(=O)C2CCCC2)C1C)=O c1(C(=O)NC(CNC(CCc2cc(OC)c(O)cc2)=O)C)ccc(F)c(Cl)c1F C(C(=O)NCc1ccco1)(C(C)Cc1ccccc1)N1CCC(CC#C)C1 N1(C(C2C(C)(C)Nc3ccccc32)=O)CC(N)C2CCCC2C1 c1(NC(=O)C(c2ccc(F)cc2)c2ccccc2)ccc([N+](=O)[O-])nc1 c1(CC(=O)N)ccc2n[nH]cc2c1.CC1(C)COCC1C(=O)NCCOCC Cc1c(CNC(C2CC(F)CN2Cc2cc(Br)c[nH]2)=O)cccc1F CCC(C)(COC)C(=O)NCc1cc[nH]c1C(=O)N(C1CC1(C)C)C N1(S(CC)(=O)=O)CCC(C)(C(=O)Nc2ccncn2)CC1 N1(Cc2cc(C)on2)CCCN(CC2CC(=O)N(C)C2c2nccn2C)CC1 C1(CC=C)(NC(=O)CSC2CCCCO2)CCN(C(c2nccnc2N)=O)C1 N1(C(C(F)=C(C)C)=O)CCOCC(F)(CNC(=O)Cc2cccc(C)c2F)C1 C1(C(=O)NC2C(C)(CNC(c3ccc(C)n3C)=O)CCC2)CCCCN(C)C1=O C1(N(C(CCc2cnc(C)o2)=O)C)CN(C(=O)C(F)=C2CCCC2)CC12CC2 C(=O)(C(C#N)CCC)N(C1(Cc2ccc(F)cc2)CCOC1)CCCC C#CC1CCC(C(=O)NC(CNC(C2CCCCO2)=O)CC)CC1 C(=O)(C1=CCN(C(c2cccc(=O)o2)=O)CC1)NC(CC(CC)C)CO CC(=Cn1ccnn1)C(=O)OCC1CCN(c2ccncn2)CC1 C1(C(=O)NC2CCN(C(C)C)C2=O)(CC)CCN(C(=O)NC2CC2)CC1 C1(C=O)CC(=O)N(OC)C1.C(CC=O)NC(COC)=O.C(C)(C)C1CC1.N C1(C(N(CC=C)Cc2ccccc2)=O)CC(C)CN1C(=O)C(C)COC C(=O)(CCC(C)(C)[N+](=O)[O-])N1CCN(C(C2(C(F)F)CCCC2)=O)CC(C)C1 c1(C(N2CCC2)=O)cnn(C2CC2(F)F)c1.C1(C(=O)N)(SCC)CC1.C Cc1cc(OCC(=O)N(CCC(=O)N(C)Cc2c[nH]nc2C)C)no1 N1(C(c2n(CC)ncc2)=O)CC(C(=O)NC(CO)CCF)C(C)C1 CC1(C)CCC2(CC1)CC2NC(c1ccc(OC(F)(F)F)cn1)=O Cc1cc(C(=O)NCC2CC(CNC(=O)C(Cl)=CCl)CO2)c(N)cc1F C1(C(=O)NC2(CCNC(=O)CSc3cccs3)CC2)CCC(F)(F)CC1 c1(COC)cccc(C(=O)NCC2CN(C(c3n[nH]cc3F)=O)CCO2)n1 c1(C(CN(CC#C)Cc2ccc(C)cc2)C)ccc(F)cc1Br CC1CCC(C(=O)NC(C)(C)CC=O)N(C=O)C1.C(C)(C)C.CCC1CC1 N1(C(C(C)OCCOC)=O)CC2(C(=O)N(CCCO)OC)CC1CCO2 O=C(C1=C(Cl)CCCC1)NC(C(=O)NCC1CCCO1)C1CC1 C1(NC(CCCSC)=O)CN(C(=O)C=Cc2ccncc2C)C2(CCCCC2)C1 C12(NC(C3(NC(c4ccc(C(C)C)o4)=O)CCSC3)=O)CC3CC(CC1C3)C2 Cn1c(C(=O)NC2C3CCN(C(c4cn(C5CCC5)nn4)=O)C23)cc2sccc12 C(C(C)C)(C(O)C(=O)N)OC.C1(C(N2CCCC2)=O)CC2(CC2)C1.CCO.C C1(C(=O)NC(CCN(C(c2c(C)coc2)=O)C)C)CCCN2CCCCC12 N1(C(C2OCCN(C(c3c(C)csn3)=O)CC2)=O)CC(O)C2(CCCC2)C1 N1(C(C2(C)CC=CCC2)=O)CCOC2(CCC(NC(=O)CSC(F)F)CC2)C1 C(=O)(CC1=NNC(=O)C1)NC1CC(NC(c2ccc(OCOC)cc2)=O)C1 Cc1cccc(CC(=O)NC2CCN(C(c3ccc(O)nc3)=O)CC2F)c1C c1(CN(C(c2cc(C)sc2C)=O)C)cnn2c1CN(C(C1CSCN1C)=O)CC2 c1(NCC(=C)CC)[nH]c(=NCC2CCCC2O)nc2scnc12 C=CCC(CNC(C1(CC)CCCN1C(C1CC1(C)C(F)F)=O)=O)CC(C)C Cc1cc(C(=O)NC2CCC(N(C)C(c3cc(C)ccc3C)=O)C2)nc(C)c1 Cc1ccc(-c2nnc(SCCSCCNC(=O)Nc3cccnc3O)o2)cc1 c1(C(=O)NC(c2cscn2)C)conc1C(C)NC(c1cscn1)=O c1(-c2scc(C(=O)O)n2)ccc(C)c(F)c1.N1(C2(CC(=O)N)CC2)CCNCC1 c1(C(=O)OCC)ccc(C(=O)NC(C)(C)CC(F)F)nc1C c1(C(N2CCC(C(C)NC(=O)CO)C2)=O)ccnc2[nH]c(O)nc12.C1CCOC1 C(=O)(CC1=Cc2ccccc2C1)N1CC2C(NC(C3C=CC=CC=C3)=O)C2C1 C1(NC(CCc2scc(C)c2)=O)CC12CC(NC(=O)CCn1cnccc1=O)C2 N1(C(C(CCCC)O)=O)CCC(C)C(NC(C23CC=CCN2CCC3)=O)C1C C1(OCCC)CCN(C(=O)C=CCNC(=O)C(O)CN2CCCC2)CC1 CCC(C)C(C)C(=O)NCC#CCNC(=O)CCc1cscc1Br C1(O)(CNC(C2(Cl)C(C)(C)C2)=O)CCN(C(=O)C=CC2CC2)CC1 n1(Cc2ccc(C)cc2)cc(Br)c(=NC(=O)C2Cc3ccccc3C2C)[nH]1 N1(C(c2cc(CC)nn2C)=O)C2CCC1CC(C)C2.c1(CC(=O)N)scnc1C O=C(CC1=CCOCC1)NCCCCNC(c1cc2sccc2[nH]1)=O c1(C(N(CC(C)(C)NC(=O)CC2CSCCS2)C)=O)cc(F)cc2nc(S)[nH]c12 CC1CN(C(C2CC3(CC3)CO2)=O)CCC1C(=O)NC(C)Cc1cn[nH]c1 C12(C(=O)NCCC3CCN(C(c4c(C(C)C)con4)=O)CC3)CCCC1OCC2 c1(C(N(CC(C)(C)CNC(=O)CC2CCCC2(F)F)C)=O)cccc2[nH]ccc12 C(CCCC=C)(C(=O)N(C1CC(=C)C1)C)NC(CCC#C)=O C1(CC(=O)N(C)CCOCC)CCCCCC1(F)F.C(=O)(CS(N)(=O)=O)N C#CCC(C)(C(=O)N1CCCC(CC)CC1)NC(=O)Cc1cnoc1 C1(CNC(=O)C(F)=CC2CC2)C(C2CC2)CCN1C(c1nc2cccnc2s1)=O Cc1cc(C(C)C)ccc1C(=O)NCC(C)(C)CC.C1(C)(C(=O)N)CCOC1C c1(C(=O)NCC(CN(C(CCCC#C)=O)CC)(C)C)cc(Br)ncc1OC c1(C(N2CC(CN(C)C(C34CC(CO3)C4)=O)C2)=O)c(O)cccc1Cl CC(C)CC(CS(C)(=O)=O)N=c1[nH]c2c(c(=NCC3CC(O)CN3C)[nH]1)CCC2 C1(NC(CN2CC(=O)NCC2)=O)CC2CC1CC2C(N1CCNC(=O)C1CO)=O c1(C(N2C(C(=O)OCC)COCC2)=O)cc(-n2cccc2)cc(Br)c1 C(C)(C)(CCCC(=O)N1CC(N2CCNC2=O)C1)NC(C(CCSC)O)=O N1(C(C2C(OC)CN(C(c3cccc(=O)n3C)=O)C2)=O)CCC2(CCOC2=O)C1 N1(C(c2ccon2)=O)CCC(O)(CC)C1.c1(C=O)cncn1C1CC1.COC C=C1CC2(C1)CC(C(=O)NCCN(C(C1CCC(C)O1)=O)C(C)C)C2 C1(C(N2CCC(NC(=O)Cn3cc([N+](=O)[O-])cn3)C2)=O)CC2COCC(C1)C2 C1(F)(CNC(c2cncc(C)c2)=O)CCCN(C(c2cn(C)c(=O)cn2)=O)CC1 CC1(C(=O)NC2(C)CN(C(c3cccc(CN4CCCC4)c3)=O)C2)CC=CCO1 C=CC1(C(=O)NC(Cc2ccco2)CO)CCN(C(=O)CC2CCOC2=O)CC1 c1(C(=O)NCC#CCNC(c2ccc(C)nc2O)=O)ccc(=O)n2c1CCCC2 C1(NC(CC2(CSC)CC2)=O)CCC(N(C(=O)Cc2ccccn2)C)CC1 C1(NC(c2nnnn2-c2ccc(O)cc2)(CSCC)C)CC(=O)N(C2CC2)C1 C(C(CC=C)NC(c1ccsc1-n1cnnn1)=O)NC(C1C(C#C)C1)=O c1(C(N2CC(C)(OCC(=O)NCCC(O)C(F)(F)F)C2)=O)cncc2[nH]ccc12 Cc1cc(=O)c(C(=O)NC(CCC2CC2)C(=O)NC(CO)C2CC2)c[nH]1 N1(C(c2cccc(OC)c2)=O)CCC(C)C(NC(C23CC4CC2C3C4)=O)C1C N1(C(c2c(=N)cc[nH]c2)=O)CC=C(CCNC(=O)CCC=CBr)CC1 N1(C(C2(C)CCC(C)C2)=O)CC2(CCN(C(C3CC4(CCCC4)CO3)=O)CC2)C1 [SH](=O)(=O)c1ccc(C)cc1.C(CC)(C(=O)N1CCC(NC(=O)C)C1)=CC.N C12(CCCCC1)C(=O)N2.C1(C(C(=O)NC)C)CCCN(CC2(O)CC2)C1 c1(OCC(C)C)ccc(C(=O)NC2CCCC2NC(=O)C(C)C(C)O)cc1 n1(CC(N2CC3CC3(C)C2)=O)ncccc1=O.C(C(F)(F)F)C1(C(=O)N)CC1 C1(NC(c2c(C)nc(C)o2)=O)CN(C(c2ccc(=N)[nH]n2)=O)CCC1(C)C c1(-n2c(C(C)(CCI)NCC(C)(C)C3CCC3)nnn2)cccc([N+](=O)[O-])c1 c1(CC(C(=O)NC)N(C)CC2(C)COC2)ccc(F)cc1F.C1(O)CCOCC1 c1(C(N2CC(CCNC(c3nc(C)[nH]n3)=O)OCC2)=O)cc2cc(Cl)ccc2s1 CCCCCC(=O)N1CC(NC(=O)CC2CCC2C)C(C)C1 c1(NC(C)C(=O)NC2CC(NC(=O)C=CC3CC3)C2)c(F)cccc1F N1(C(C2(C)C(C)CN(C(CS(CC)(=O)=O)=O)C2)=O)CC2CSCC(C2)C1 Cc1cc(NC(=O)N(C2COC2)C)ccc1OC(F)F C1(C(N(CCC)CCNC(C2CCC(CC)CC2)=O)=O)Cc2nccn2C1 N1(C(C(CCC)CCC)=O)CC2CCCC(C1)N2C(=O)C(CC)C(C)O C(=O)(C1=NN(C2CC2)C(=O)CC1)NCC(CNC(c1cnn(C)c1N)=O)O N1(C(C(C)NC(=O)C(C)(C)C)=O)CC(NC(c2cnsn2)=O)CCC(O)C1 N1(C(Cn2c(C)ccn2)=O)CC(NC(c2ccncc2Cl)=O)C2(CCC2)C1 c1(N2CCC(CNC(c3cnc(CC)nc3C)=O)C2)ccc([N+](=O)[O-])cc1C#N C12(COC(C3CCC(F)(CS(=O)(=O)NCCC)C3)=O)CCCN1CCC2 CC1CCCc2c(C(=O)NCCC3(NC(c4ccc(CO)o4)=O)CCC3)cnn21 C(=O)(CCC(=O)CC)NCC1C(C(NOCCC#C)=O)CC1 C1(C(=O)N)Cc2nccn2C1.CC(C)(C)CCNC(C1(P(C)(C)=O)CC1)=O C(=O)(CC(C)C(=O)OC)NCC1(C(=O)NC(COCC)CO)CCOCC1 Cc1ccc(C(=O)NC2CCN(C(=O)C3=CC(C)(C)C3)C2C2CC2)c(C)n1 c1(CCCC)cnc(NCc2ccc(CC#N)cc2)nc1 c1(NC(C(C2CCC(=O)N2)C)=O)coc(C2CC2)n1 N1(C(C2(C)CC2)=O)CCCC(NC(c2ccccc2NCc2ccco2)=O)C1 N1(C(CN(CCOC)C)=O)CCN(C(c2cn3c(n2)CCCC3)=O)C(C)C1C C1(C(=O)NC(C)CCNC(C2CC2c2cn[nH]c2)=O)CC2CCCC(C1)C2 CON(CCC(=O)N(C1COCC1(C)C)C)C(=O)CC(O)CC(C)(C)C N1(C(c2cn(C)nc2Cl)=O)CCN(C(c2cnns2)=O)CC1C1CCC1 c1(C=O)ccc(Cl)c(CCN(C)C)c1.Cc1cnc(CC(=O)NC2CCC2)o1.C c1(OC)cc(F)c(N2CCC(N3CCC(C4(C)NC(=O)NC4=O)C3)CC2)c(F)c1 CCC(C)(CNC(c1cccc(C#N)c1)=O)C(=O)NC1CC12CCCCC2 c1(C(N2CCC3CN(C(C(C(C)(C)O)F)=O)CC32)=O)coc2c(F)c(Cl)ccc12 C(=O)(C(C1CCC1)NC(=O)CCC1CC1(C)C)NCCOCCCC Cc1cc(CCNC(c2nnnn2CCCF)C2CC2)n[nH]1.C1CCCO1 c1(C(N2CC(CCNC(C3CCC(C)(CC)O3)=O)C2)=O)c(F)ccc(F)c1Cl C1(C(=O)NC2C(C(=O)NC)CCC2)CC2(CC2)C1.C(=O)CCc1ccoc1 c1(C(=O)NCCCC2(NC(Cc3c(C)scc3)=O)CC2)ccc([N+](=O)[O-])o1 c1(-n2cc(C(CCCC(=O)NOC3CCC3)C)nn2)ccc2c(c1)ncn2C C1CCC2(CC1)CN(C(C1CC1C(F)(F)F)=O)C2.CC1CCC(C)(C(=O)N)C1 c1(C(=O)NCC(C)NC(c2c(C)ocn2)=O)c[nH]c2c(C)c(F)ccc2c1=O C(=O)(CC(CC)CC(C)C)N1CC2C(CC(=O)NCCCOCC=C)C2C1 c1(-c2ccc(NC(C3(C)ON=C(C)C3)=O)cn2)ccc(-c2nn[nH]n2)cc1F c1(COC)ccc(C(=O)NCCCC(C)NC(=O)COCC(C)(C)C)o1 c1(C(=O)NC2(C3CN(C(=O)CC4CCOC4)C3)CC2)ccn2c1CCCC2 C#CCC(C(=O)N1CC=CC(CO)C1)NC(=O)COCC=C O(NC(=O)C(CC(F)F)NC(c1ccn2ccnc2n1)=O)CC(=O)OCC c1(C(N2CC(CC(=O)Nc3cnnc(Cl)c3Cl)C2)=O)cn2cc(F)ccc2n1 C(C(C(C)C(C)C)NC(=O)C#CC1CC1)NC(c1c(C)c[nH]c1CC(N)=O)=O Cc1cccn2cc(C(N3CCC(C)(C)C3)=O)nc12.c1(CC(=O)N)nc(=N)[nH][nH]1 C(CC(C)(C)CC(=O)N1CCCC1(C)CNC(=O)CN1CC2C=CC1C2)OC N1(C(C2CN(C)C(=O)C2)=O)CCN(C)C(CNC(=O)CCC2CCCCO2)C1 CC(CC#N)C(=O)N1CCC(O)(CCNC(=O)Cc2cnccc2Cl)C1 CCC(CC(=O)NCC(C)(F)CNC(=O)C(N1CCCC(C)C1)=O)OC c1(CC(=O)N(C2CCN(C(=O)CC(C)OC)CC2)CC)ccc(OC)cc1F C1(C(N(C2CC(NC(CC=C(C)C)=O)C2)C)=O)CC2(COC(=O)N2)C1 N1(CC(=O)N(C2CCC(F)(F)CC2)C)C(C(=O)O)CCC12CCC2 N1(C(c2c(C)cncn2)=O)CCCC(F)(C(=O)NCCC2CCC(=O)N2)C1 C12(C(=O)NC3CCC(N(C(CCc4cc(C)[nH]n4)=O)C)C3)C3C4C1C1C2C3C41C C(=O)(CC(C)CC(C)(C)C)N1CCC(C(N(C(C#C)C2CCC2)C)=O)CC1CC c1(C(N(C2C3CN(C(C4CCC4)=O)CC32)C)=O)n[nH]c2cc(C)ccc12.CCO n1(CC)ncc2c(N3CCCCC(CC4CC4)C3)[nH]c(=NCc3ccoc3)nc12 C1(NC(C(N)=O)=O)CS(=O)(=O)CC1NC(c1ccc([N+](=O)[O-])[nH]1)=O C1(NC(c2ccc(CNC(CCCC)=O)cn2)=O)CCCC2(C1)N=N2 C1(N(C2CCS(=O)(=O)C2)C(=O)Cn2cc(CN)nn2)CCC(C(F)(F)F)CC1 C(CCC(=O)NCCC(C)(C)NC(c1cc(-c2cnn(C)c2)no1)=O)=CCC=C CCCCCCC(C)C(=O)N(C(C)CNC(=O)C(F)(F)C(C)O)C C1(NC(c2ccc(CNC=O)cc2)=O)CN(c2ncc(Br)cn2)CC1(F)F.N C1(C)(CNC(CCC2CCC(C)O2)=O)CCCN(C(=O)CSc2nncs2)C1 CC1C(NC(c2cncc(C(C)(C)C)c2)=O)CCN1C(=O)CCCCN(C)C C1(C(=O)NC(C)C(C(C)C)NC(=O)Cc2cscn2)(OCC)CCCCC1 n1(CC)c(C(=O)NC2CN(C(c3c(C4CC4)noc3C)=O)CC2O)cnc1O N1(c2c(OC)cncn2)CCC2(CC1)CC2(C)C(=O)N(CCCO)C c1(N2CCC(C(=O)Nc3cccc(CC)n3)C2)ncnc2[nH]c(C)nc12 c1(C(=O)NCC(N(C(CC(C)N(C)C)=O)C)C2CC2)ccc2cccnc2c1 N1(CC)CCN(C(c2sc(C)cc2Br)C(=O)N(C2C3CCCC23)C(C)(C)CC)CC1 CC(Cc1cnc[nH]1)C(=O)N1CCCC1CN(C)C(C1CCCCS1)=O C1(C(=O)Nc2ccc(C#C)nc2)N(C(=O)CC(C)(C)C(C)=O)CCCC1(C)C C1(CC)(NC(c2csc(C3CC3)n2)=O)CCN(C(=O)C(C)C#N)CC1 c1(CC)ccnc(C(=O)NCCNC(C2CC(C)OC2=O)=O)c1 CC1CN(c2ccnc(-c3nccs3)n2)CCC1NC(C1(C)CC1(F)Cl)=O N1(C(CC(C(C)C)O)=O)CC2CC(NC(=O)C3=CCCC3)CC1C2 CCCC(C(=O)NCCC1CCN(C(C2CCNC(=O)C2)=O)CC1)NC(N)=O CC1CCN(C(=O)C(C)C(F)F)C1C(=O)NCC(C)(C)C(F)F c1(C(=O)NCCN(C(=O)Cc2csc(Cl)c2)CC)cnn2ncccc12 c1(C(=O)NC2C(NC(C(C)(C)C3CCCC3)=O)C2)cccc(CC(F)(F)F)c1 c1(CN(C(c2cn(C)nn2)C(=O)Nc2ccccc2)C(CC)C)ccccc1Br C1(C(N(C(C(N2CC(CCCCC)C2)=O)C2CC2)C)=O)CCCSC1C C1(NC(CCCOCCOC)=O)(CF)CCN(C(=O)CCN2CCC(F)C2)C1 c1(C(N(CCCN(C(c2n(CC=C)ccn2)=O)C)C)=O)cc(C)ccc1[N+](=O)[O-] N1(C(C2CN(C(c3cc(C)nnc3)=O)CC23CC3)=O)CCCC(N=[N+]=[N-])CC1 c1(C(=O)NC23CN(C(C(C)OC)=O)C(C2)C3)ccc2nc(C)n(C)c(=O)c2c1 c1(CC(=O)NCCCn2cc(C(C)NC)nn2)c(C)c2ccc(O)cc2oc1=O c1(C(N2C(CNC(c3cc(CC)c(C)s3)=O)C=CC2)=O)cnc2ccccc2c1 C1(NC(C(C(CC)C)O)=O)CN(C(c2ccc(=O)n(CCF)n2)=O)CC(C)(C)C1 c1(C(N2C(C)CC(NC(c3nncs3)=O)CC2)=O)ccc2c(c1)C(=O)OCC2 c1(C(=O)NCC(C2CCOC2)NC(COC)=O)ccc(NC2CC2)nc1 C(=O)(N=c1[nH]nc(C2CCCO2)s1)NC1(C(=O)NC)CCCC1 C1(N(C(CNC(CCC)=O)=O)C)CCCN(C(C2(OC)CCCSC2)=O)CC1 N1(C(C(C)NC(C)=O)=O)CC(F)(c2nn[nH]n2)C1 c1(C(N2CC(CNC(C(C)(C)F)=O)C3C2C3)=O)cc(O)ccc1Cl c1(C(=O)NCC2(N)CCC3CCCC23)cc(=O)c2ccc(Br)cc2o1 C=CCC(CC(=O)N(CC(C)(C)O)C1CC1)NC(=O)C(c1ccn(C)c1)C c1(CC)ccc(C)c(C(N2CCN(C(=O)C(C)CCOC)C(C3CC3)C2)=O)c1 N(C(=NCCc1cc(C)ccc1OC)NC1CCCC1)Cc1n(CC)ncc1 Nc1cc(=O)nc(C(N2CCCC(N(C(c3cscn3)=O)CC3CC3)C2)=O)[nH]1 c1(C(=O)NCC2CN(C(C3(C)CC3)=O)CC2O)nc2ncc(CCO)cn2n1 N1(c2n(CCC#C)c(C(C)C(O)CC)nn2)CCC(O)(COCC=C)CC1 c1(NC(C(CCC=C)NC(C2C3CCCC23)=O)=O)ccc2ccoc2c1 c1(C(=O)NC2CC3CN(C(c4n(C)cnc4)=O)CC3C2)cc2c(nc1O)CCC2 C1(CC(=O)N)CC2CC2C1.C1(O)CN(C(=O)Cn2ccnn2)C1.C1CCC1.C C1(C(N(C(CC)C(=O)NCCCc2nc(C)no2)C)=O)COCC(C)O1 C1CC2CC1N(C(C1(S(N)(=O)=O)CC1)=O)C2.c1(N(CC(=O)N)C)ccccc1 c1(SC)nc(C(F)F)cc(=NCC2CN(C(c3c[nH]c(=O)cn3)=O)C2)[nH]1 N1(C(c2cnc(CC)[nH]2)=O)CC2CCC(C1)C2.c1(C(=O)N)c([N+](=O)[O-])cnn1C C1(C(=O)NC(C)CCNC(=O)C=CC2C(C)C2(Cl)Cl)Cc2ccccc2C1 c1(C(N2CCCC(NC(c3c(CC)c(C)sc3)=O)C2)=O)c(C)c(C)nn(C)c1=O C12(CNC(C(CC)(F)F)=O)CCCC1N(C(c1cccc(O)c1C)=O)CCC2 N1(C(CCN(CCCCC)C)=O)CC2CCC(C1)N2C(C1CCC(=O)N(C)C1)=O c1(C(=O)NC(CCC)C(=O)N2CCC2C(N)=O)ccc2[nH]nc(Cl)c2c1 N1(C(Cc2c(C)cccc2)=O)CCC(C)C(O)C1 c1(CC(=O)NCC(CO)NC(C2(C)COCCO2)=O)cc(O)nnc1O N1(C(Cc2c(C)con2)=O)CCCCC1C(=O)NCC(C)CC1CC1 Nc1cc(C(=O)NCC2(O)CCCN(C(=O)C3=COCCC3)C2)c(F)c(F)c1F Cc1cc(C(=O)NC2CCC(C)N(C(c3cc(Cl)nnc3O)=O)C2)nnc1O n1(C(C(=O)NCCCN(C(C2CCC(=O)N2)=O)CC)C)cc(C)cn1 C1(NC(C(F)=CC)=O)CCN(C(C2(CC)CCCC2)=O)CC1 C1(C(N2CC(CCO)(NC(=O)C=Cc3cc[nH]c3)C2)=O)CCCN(CCO)C1 Cc1ccc(-c2cc(C(N3CC4C(C)C4C3)=O)on2)cc1.C(=O)(C(C)N(C)C)N C(CNC(C1CC1)=O)(CC(F)(F)F)NC(COCCC)=O.N(C)(C)C C1(C(=O)NCC(C)NC(CCCC(OC)OC)=O)CC(C)(C)OC(C)(C)C1 c1(C(C)C(=O)NCCCNC(C2(c3cccc(Cl)c3)CC2)=O)cccc(C#N)c1 c1(NC(C2CN(C(c3c(CC)nco3)=O)CC23CC3)=O)cccc2occc12 CC1CC(S(=O)(=O)NC(COc2ccccc2)CN)CC(C)O1 C1(CC)CCN(C(=O)CCc2nc(O)n[nH]2)C1C(=O)NC(C)C=O.C(C)C N1(C(C(C)O)=O)CC(C(=O)N(C(C)CO)C2CC2)C(C2CC2)C1.C(C)(C)C c1(C=O)c(C)nn(C)c1-n1ccnc1C.C(C)(CCC)NC(C1(SC)CC1)=O N1(C(c2ccc(CC)cn2)=O)CC2(CCCCN2C(C2CC23CCSCC3)=O)C1 CCC(C)(C(=O)N1CCC(C)N(C(c2nc(O)sc2C)=O)CC1)C(F)F c1(OCC)ccnc(NC(C)CN(C)C(c2ccccc2)=O)n1.C(C)=O.C N1(C(C(C)C2CCCO2)=O)CC2(CC(NC(c3snc(Cl)c3Cl)=O)CO2)C1 C1(NC(Cc2ccc(C)c(C)c2)=O)CCCC2CN(C(=O)CN(C)C)CC12 CC(C)CC(CC(C)C)C(=O)NCC(O)CN(C(=O)C(c1ccc(Cl)cc1)C)C N1(C(C2CC2)=O)CCC(C2CC2)C1.C1(C=O)C2(CC2)C12CC2.CC(C)C.O C1(NC(Cc2n(C)ccn2)=O)CCC(F)(C)C1.C(=O)(C(O)CN1CCOCC1)N C1(C(N2CC3CN4CC3(C2)C4)=O)C2C3CC4C1C1C2CC3C41.C1(N)CCCCNC1 C1CCCCC1C.C(C(C)(C)C)N(C(=O)C)CC.c1(CC=O)cc(Cl)cs1.N c1(OC)c(C)csc1C(=O)NCCCCCNC(=O)C=Cc1cccs1 C1(c2nnnn2CC(F)F)(NC2(SC(F)F)CC2)CCCC(C(F)(F)F)C1 CC#CCC(C(=O)NCc1nnc(CC)o1)NC(=O)C(C)CC=CCC C(CCC(=O)NCC1CCC1NC(=O)C(O)COC)OC.c1ccccc1 C(=O)(C(O)CC(C)(C)C)NC(c1n(C)ncc1)C(=O)NCC1CCCCCCC1 Cc1noc(CCCNC(C2(F)CN(C(c3ccoc3)=O)C2)=O)n1 Cc1nc2ccccn2c1C(=O)NC(C1CCCN(C(c2cc(F)n[nH]2)=O)C1)C CCCCCCC(F)C(=O)NCC1(CNC(=O)Cc2cccc(O)c2)CCC1 Cc1csc(C(=O)NC2(CNC(C3CC(C)OC3C)=O)CC2)c1Cl c1(C(=O)NCCN(C(C)C)C(C2C(C)CC2C)=O)cn(-c2ccccc2)nn1 C1(C(=O)NCC(C)NC(=O)C(C)C(F)F)COCC2(CCC2)O1 c1(C(=O)Nc2ccc(CC)cc2)cccc(C)c1C.C1(C=O)CC1.C(C)=O.N N1(C(c2c(C)nc(CC3CC3)s2)=O)CCC(C2CC2)C1.C(=O)CC(F)(F)F.C C(=O)(CCCCC#N)N1CCC(C)C1C(=O)NCC(n1cccn1)C C1(NC(c2nc(C)c(C)s2)=O)CN(C(=O)C=CBr)CC1N=[N+]=[N-] Cc1nc2c(F)cccc2cc1C(=O)NC1CCN(C(C2OCCO2)=O)C(C)C1 C1(CNC(=O)Cc2ccsc2)CN(C(=O)CSc2ccncc2)CCO1 N1(C(C(=O)NC(C)C)C(C)C)CC(=O)N(C)C(C)C1 C1(NC(C2CCS(=O)(=O)N2)=O)CN(c2ncnc3cccnc23)CCC12CCC2 C1(C(=O)N)CCc2ccccc2CC1.C(C(=O)NC(C)C)N(C(=O)OCC)C C1(NC(CC(CCC)NC(=O)C(CN(C)C)C(C)C)=O)CCn2cncc2C1 c1ccc2c(c1)CCC2.C(C)(CC(=O)NCC1CC(NC(=O)C)C1)SC.S CC1CC2CC2CC1C(=O)NCCC1(O)CN(C(=O)CCc2ncc(F)cn2)C1 N1(C(C(COCC)NC(C(CCC)F)=O)=O)CCC2(CCCC2)CC1 c1(C(=O)NC2CN(c3c(F)cnc(C)n3)C(C)C2)cc2ncccn2n1 C1(C2(N)CC2)CCCCN1C(c1cscc1C(F)F)=O.C1(C=O)C2CCC1CC2 C1(CCC(=O)NCC=CCC(=O)NC2(CF)CCCC2)CCCCO1 N1(C(CN(C(COC)=O)C)=O)CC(C)N(C(c2cc(C)nc(O)n2)=O)CC1C c1(C(N2CC(OC)C(NC(c3sc(C)cc3C)=O)C2)=O)coc2c1C(=O)CCC2 CC1CCN(C(C2CC2C(F)F)=O)C(C(=O)NCCSCC(C)(C)O)C1 CON1CCC(C(=O)N(C2CCN(C(=O)C(C)OCC(C)C)CC2)CCO)CC1 C=CC1CC(N=c2[nH]c3c(c(=NCC(F)(F)c4ccc(Cl)cc4)[nH]2)COCC3)C1 c1(C(=O)O)cc2n(n1)CCCN(Cc1cc(CF)on1)C2 N1(C(c2c(=N)[nH][nH]c2)=O)CCC12CN(C(C1CCN(C3CC3)C1=O)=O)C2 CCC(CCC(=O)N1CCCC1C(C)(C)NC(c1ccnc(OC)n1)=O)OC CCN=c1[nH]c(C)c(C(=O)NC2C3CCC2N(C(C2CNC(=O)C2)=O)C3)s1 C(=O)(C(C)CCC(C)(C)C)NCCC(CC)(CC)NC(C1ON=C(CC)C1)=O c1(C(=O)OCC)cnc(C(=O)Nc2cccc(-n3nncc3C)c2)cn1 CC(C)(CCC(=O)N=c1ccn(C2CC2(F)F)[nH]1)c1ccccc1 C=CCC(CNC(c1cc(C)sc1C)=O)C(=O)NCCCc1ncc[nH]1 C=CCC(CC=C)C(=O)NC1CCCCC1CNC(C1CC(C)C1)=O S(=O)(=O)(c1ccc(OCC)cc1)N1CCC(CCCC)C1 CCCCCCC(CC)NC(C1(NC(C2CN3CCN2CC3)=O)CC(O)C1)=O CC1CN(C(=O)Cc2cccnc2)CC1NC(=O)CCn1ccccc1=O Cc1cc2ccc(C(N3CCN(C(C4CC5CC5C4)=O)CC3CF)=O)cn2c1 CN1CCN(C(c2ccc(OCCF)cn2)=O)C(CNC(C2(C)CCOC2)=O)C1 C1(CNC(c2c(C)ncnc2)=O)CCCCCN1C(=O)C(=Cc1c[nH]cn1)F c1(C(N(C(c2ccc(Cl)cc2)C)C2CC2)=O)cc2c(F)ccc(Br)c2[nH]1 c1cc(C)c(C#N)cn1.N1(C(C(C)=CC2CC2)=O)CC(C(F)(F)F)C(CN)C1 n1(C(CC)C)ccc(=NC(=O)CC2CN(C(=O)C(C)OCCOC)CCO2)[nH]1 C(CCC(C)C)(C(=O)NC1CCCNC1=O)NC(Cc1c(C)cccc1)=O C1COC2(C1)CN(C(C1(CS(C)(=O)=O)CCC1)=O)C2.Cc1cc(C(=O)N)co1 c1(C(N2CC(CC(=O)OC)OC(C)(C)C2)=O)ccc2c(c1)NC(=O)CO2 N1(C(c2ccnc(OC)n2)C(=O)NC2CCCC2)CCC(F)C(O)C1 Cc1cc(C(C2(C)CC2)NC(C2(C)CCCN(Cc3nncs3)C2)=O)ccc1F C1(CNC(C(C)c2cncs2)=O)C=CC(NC(=O)C(c2ccccc2)=O)C1 Cc1cc(C)n(CC(=O)NC2CCCC2C)n1.c1(C=O)ncoc1C1CCC1.N c1(C(=O)NCC=C)ccc(C(=O)NCCC)cc1.C(=O)CC.C(C)(C)CC c1(C=O)c(Cl)ccc(F)c1N.c1(CC)nn(C)c(Cl)c1C(=O)NC(C)CC.N C12(C(=O)NC3C(CNC(CCC#CC)=O)CCC3)CCC(C1)OC2C Cc1cc2c(C(=O)N(CCNC(C3(C)CC4CC4C3)=O)C(C)C)nccn2n1 c1(N(C)C)cccc(C(=O)NCC(C)(C)CNC(C2(C#N)CC2(C)C)=O)c1 CC(C)C(CCc1ccccc1)C(=O)OCC1(CC(F)F)CCC1 N1(C(C2C(C)CCC2)C(=O)NC2CCCCC2)CC2CSCC(C2)C1 C(=O)(C1=C(C)OCCS1)N(CC)CC.c1(C2(C=O)CCCC2)cccc(C)c1.N C(=O)(N1OC2CCC1CC2)C1(NC(C(C)n2cncn2)=O)CSC1 CC1(C)CNCC(C(=O)NCc2ccncc2Oc2ccc(F)cc2F)C1 C1(C(C)C)OCCC1C(=O)NC1CCC(C(=O)NCCCCC2CC2C)C1 CC1C2CC(C2)N1C(C1CNC(=O)C1)=O.c1(C=O)cccc(CCN(C)C)c1 C1(OC)CCCC1C(N1CCCC1C(C)NC(c1cnn(CCF)c1)=O)=O C1(C(=O)NC(C2CCCCC2)CNC(C2(C(C)C)COC2)=O)CC=CCO1 c1(CNC(=O)NCC2C(C)CC2)cccc2c1OCO2 c1(C(=O)NCc2cc(C)cc(C#N)c2)cc2n(n1)CCCC2O c1(C(=O)NCC2OCCN(C(C(CC)=CC)=O)C2)cn(C)c2ncccc12 N1(CC)CC(C(=O)N2CCCC(CNC(=O)CCCC(N)=O)C2)c2ccccc21 c1(-c2occ(C(=O)NC(CCNC(c3cnn(CC)n3)=O)C)n2)ccc(F)cc1 C1(COC)CN(C(=O)C=Cc2ccc(Br)s2)CCC1(CO)OC C1(NC(=O)C=Cc2cncs2)CC2CC1CN(C(C1CCC=CCC1)=O)C2 C(=O)CC(C)O.n1(CC(N2CC(C)(CC=O)C2)=O)nc(C)cc1C=O c1(C(N)=O)ccc(Cn2cc(CC(CN)C3CC3)nn2)cc1 C12(CNC(C(F)=C(C)C)=O)CCC(CN(C(c3ccc(C)c(O)c3)=O)C1)C2 c1(C(N2C(C)(CC(=O)NCc3ncc(C)[nH]3)CC2)=O)cccc(F)c1N C1(C(=O)NC2(C(N(CC(F)Cl)C)=O)CCC2)C2CC3C(C2)C13 CC(C)(C)C(CNC(C1C2(CC2)C12CC2)=O)C(=O)N1CC=CCO1 C1(C(=O)Nc2sc(C(C)=O)c(C)n2)CCc2nc(O)[nH]c2C1 C1CCCC(C(N)=O)C1.Cc1cc(CC(=O)NCCn2cc(C(=O)N)nn2)no1 CCCCCCN(CC(=O)NCCN(C)C(c1cc(-c2cccs2)on1)=O)C N1(C(C=CC=CCC)=O)CC2(CCC2)CCC1CNC(C1CCCCC1O)=O CC1(C)CN(C(=O)NCC2CCCC3(CCC3)O2)C(CO)CO1 c1(C(N2CCC(C(=O)O)C2)=O)ccc(-n2cc(CC(O)C3CC3)nn2)cc1 N1(C(C(CCCC)F)=O)CC2(CCN(C(c3nnn4c3CCCC4)=O)CC2)C1 c1(NC(c2cnc(NC(c3cnccc3I)=O)o2)=O)ccc(F)c(F)c1 C(=O)(C1=CCSC1)NCC1CCC(NC(C(C)C2CCCO2)=O)C1 c1(CN2CCN(CC(=O)NCCCS(N)(=O)=O)C(=O)C2)c(F)cc(I)cc1F C1(C(=O)NC2CN(C)C(=O)C2)CCN(C(c2ccc(=N)[nH]c2)=O)C1(C)C C#Cc1cnn(CC(=O)N(C)CC2(CNC(C3(C)CCCOC3)=O)CC2)c1 N1(Cc2c(C)nccc2)C2CCC1CC(NC(c1ccnc(F)c1)=O)C2 c1(C(N2CC(CNC(C3CCN(CC)C3)=O)C(C)C2)=O)c(Cl)cccc1[N+](=O)[O-] N1(C(C(C)N(CCC)C(c2cc[nH]c(=NC)c2)=O)=O)CCC2(CNC(=O)O2)C1 C1(NC(CC(C)C(C)(C)C)=O)CC2COCC(C1)N2C(=O)C(O)C(C)(C)C C(C(C)CC(=O)N1CCCCC1CNC(c1ccns1)=O)OC n1(CC)ncc(Cl)c1C(=O)N.C1CC(C)N(C(=O)C=CC=O)C1.C(C)C c1(C2N(C(N(C)CCc3ccccc3)=O)CC2)ccc(Cl)cc1 c1(OCC)ccc(CN2C(C(=O)N)CC3CC23)cc1Cl.N1(CC)CCC(C)CC1 CC(C)C(C(=O)N1CCC(NC(C2CN(C)C(=O)N2)=O)C1C)NC=O C#CCCCOCC(=O)NC(C)C(=O)N(C(C)C(=O)OCC)C C=CCC(C)(C)C(=O)N1CCC(CNC(=O)CC(C=C)CC)(COC)C1 C1(NC(CN(CCOC)C)=O)C=CC(C(N2CC(C)(N(C)C)C2)=O)C1 Cc1cc(O)cc(C)c1C(N1CC2CCCC2(NC(=O)C=CCF)C1)=O C(=O)(CC(F)(F)C(F)F)NCCCCC(N1C(C(=O)OC)CC=CC1)=O Cc1c(C(N2CC=CC2CNC(C2CC3OC2C2CC32)=O)=O)oc2ccccc12 C(=O)(C(CNC(=O)CCN1CCCC1=O)C(C)(C)C)N(C)Cc1ncnn1C N1(C(c2cncc(SC)c2)=O)CCCC(NC(C2CC(C)(C)CO2)=O)CC1 C(=O)(C1=C(Cl)CC1)N(CCC(=O)NC1C(CC)C1)C(C)C Cc1cc(C)n(C(C)CC(=O)NCCNC(=O)C(O)Cc2[nH]cnc2C)n1 N1(CC(=O)N(C)Cc2nccs2)C(C)(C)CC(O)CC1(C)C N1(Cc2c(CC)scc2)CCCC(C2CCCCN2C(=O)Cn2cncn2)C1 C1(C(C2CCC(F)(F)C2)=O)Cn2cnnc2CN1CC1CCCCO1 c1(OC)cc(C(=O)Nc2cc(C(F)F)nc(C)n2)cnc1Br C(C(=O)Nn1nnc(C)c1C)N(C(=O)CC1CC2CC2C1)CCOC c1(C(=O)NCC2C(NC(c3ccc(Cl)s3)=O)C2)nc(Cl)cs1 C(=O)(C(CC)C(F)(F)F)NCCn1cc(C(N2C(CC)CC(C)C2)=O)nn1 Cc1ccnc(C(=O)NC2CCCCC2NC(c2c[nH]c(C#N)c2)=O)n1 c1(NCC(CCSC)OC)cc(N(C)C)nc(C(C)C)n1.C1CC2(CCC2)C1 N1(C(c2nnc(C(C)C)s2)=O)CC(C)OC2(CCN(C(c3cc(O)cs3)=O)C2)C1 N1(C(COCc2n(C)ccn2)=O)CCC2CCN(C(=O)C3=CCCSC3)C2C1 CC1(C)CCC(C(F)(F)F)(C(=O)NC(C(=O)O)C2CCCC2)C1 c1(OCC)ccccc1.C(C)(C)(C=O)O.c1(C(N(CCC)C)=O)csc(C)c1 CCCCC(O)C(=O)N1CCC(C)C(CNC(c2cnn(CCN(C)C)c2)=O)C1 C1(NC(C(C2CCN(C(C(C=C)O)=O)CC2)C)=O)(CO)CC2CCCC12 C#CCCCCCC(=O)N1CCN(C(=O)CC2CNC(=O)C2)CC1CS(C)(=O)=O C(=O)(C1CC=Cc2ccccc21)NC(CNC(=O)Cc1ccccc1O)CO C12(CNC(=O)CCF)CC3CC(CC(C3)C1NC(C1CCCC1C1CC1)=O)C2 N1(C(CC(C2CC2)NC(C(c2cn(C)nc2)=O)=O)=O)Cc2n[nH]cc2C1CO C(=O)(C(O)CC1CC1)N1CC(CCNC(=O)C(F)n2cccn2)C1 c1(C(C)=O)ccc(C(=O)NC(C)C)c(O)n1.C(=O)C(C(C)C)N1CCCCC1.N c1(C(N(C(CNC(CNC(=O)OC)=O)C2CC2)C)=O)ccc(O)nc1Cl c1(NC2CC3CN(C(Cc4ccc(C)cc4)=O)CC32)ncc([N+](=O)[O-])cc1C#N CC1=C(C(=O)NCC2(C)CC2)CCC(C)(C)C1.C12(CC=O)CCCC1C2 N1(C(c2n(CC#C)ccn2)C(=O)NC2CC(F)(F)C2)CCCC2CC12 c1(OC)cc(C(=O)N)ccc1C(F)(F)F.C1(F)CCC1.C1(C=O)CCC1.C c1(CCC)c(C(=O)NCC(C)(O)C)nnn1C.c1(C(C(=O)N)C)cccc(F)c1 c1(C(N2C(CNC(C=Cc3ccn(C)c3)=O)CC2)=O)cc2ccc(F)cc2s1 Cc1c(Cl)ccnc1C(=O)NC1CC(NC(=O)C(CO)c2ccccc2)C1 CCCC(C(=O)N1CCC(CN(C(=O)C(C)(C)Cc2ccccc2)C)CC1)OC C1(NC(C(C#C)(C)C)=O)CCN(C(c2nn(C)cc2C(C)=O)=O)CC1O C(=O)(CC(F)(F)C(F)(F)F)NCCCCCNC(C1(C)CC1C(F)(F)F)=O CS(=O)(=O)c1ccc(F)c(C(N2CCC2C(=O)NCC2CCCCO2)=O)c1 S(=O)(=O)(c1cc(Br)c(Cl)s1)N1CCC(c2ccc(C#N)cc2)C1 N1(C(c2c(CC)cno2)=O)CCCC(F)(C(=O)N(CC(C)(C)C)C(C)C)C1 C(=O)(C1CCCc2sccc21)NCC1CCCCN(C(C(C(C)C)O)=O)C1 C(CC(=O)N1CCC(C)(NC(c2nnsc2SC)=O)CC1)(C(C)C)OCC CCCCCCCCCC(=O)NCCN(CC(C)O)C(c1sccc1CC#N)=O CS(=O)C=CC(=O)NCC1CN(C(c2ccccc2-n2cnnn2)=O)C1 c1(C(=O)NC(CC(C)C)CNC(c2cccnc2)=O)cc(O)ccc1Br C1C2CN(C(C3CC(C(C)(C)C)C3)=O)CC12.c1(OCC)sccc1C=O.N C1(C(N2CC(CCNC(C(CC)c3ccccc3)=O)C2)=O)CCc2nnnn2C1 Cc1nn(C(C)C)c(C)c1CC=O.C1(C)CCN(C(C2CC2C(C)C)=O)C1.N c1(C(N2CC3C(NC(c4cc5ccccn5n4)=O)(C3)C2)=O)cc2nc[nH]c2cn1 C(CO)(CCCCNC(=O)C(F)=CC)NC(C(C)OCCC#C)=O CC1C(NC(=O)CCC2CCCC(=O)N2)CCCN1C(C1COCCO1)=O Cc1nncc(C(=O)NC(C(=O)NC(C)CC(C)C(F)F)C2CCCO2)c1C C(C(C)(CC(C)C)NC(=O)Cc1csc(C)c1)NC(C1N(CC)CCC1)=O C1(C(=O)NCC(n2cc(C(n3cccc3)(C)C)nn2)C)CCC2(CCOC2)O1 CCC(C)(C)C(=O)C(=O)NCC(CC(C)C)C(=O)NCC1CC(C)(O)C1 C1(CC)CCN(C(C2(C(C)NC(c3ccc(C(C)C)o3)=O)CC2)=O)C1 C1(SC)CN(C(c2cc(Cl)n(C)n2)=O)CC1NC(C1(C)CC(F)(F)C1)=O c1(CN2C(C)(C)C=CC2)c(F)cc(C(F)(F)F)cc1Br c1(C(N2CCC(CC(=O)Nc3c(C#N)nc[nH]3)CC2)=O)cc2[nH]ccc2cc1Cl N1(C(C(C(=O)OC)C)=O)CCc2c(C(=O)N(CCCO)C(C)C)n[nH]c2C1 Cc1[nH]nc(Cl)c1C(=O)NCCCCCN1CCN(C(=O)C=CC2CCC2)CC1 C1(CC(=O)N)CCN(C(c2ccc(C)c(F)c2)=O)C1(C)C.C(C)(C)(CC)OC C1(C(=O)NCCC(C)N(C)CC)CC12CCN(C1CCCNC1)CC2 CC1CC(C(=O)N)CC(C)C1.C1CC(F)(F)C1.n1(CCC=O)cnc(=N)[nH]1.C c1(CCNC(N2CC3CCCC2C3)=O)c[nH]c2cc(F)c(Cl)cc12 C1(C(=O)OC)CCCCCCC1NC(c1ccccc1Cn1ccnn1)=O C(C)(C)(CCC)NC(c1cc(C(C)=O)oc1)=O.C1(C(=O)N)CS(=O)(=O)C1 C(C)(CNC(=O)C(F)(F)C1CC1)(C(=O)O)OC O=C(CS(=O)(=O)C1CC1)NC12CCCN(C(c3nnsc3C(F)F)=O)CC1C2 c1(SCC(=O)N(CC(C)NC(c2ncccc2F)=O)CC)ccsc1[N+](=O)[O-] N1(C(CC(CC2CC2)NC(CC(CCOC)(C)C)=O)=O)CCOCC(C2CC2)C1 C=C1CCC(CNC(c2ccncc2)(c2nnnn2C)C)C1 N1(C(=O)CCCc2ccsc2)CCC2(C1)CN(C(=O)CCSC(F)(F)F)C2 c1(C(N2CC3(C(NC(CCSCC(C)C)=O)CC3)C2)=O)ccc(Cl)c2occc12 C12(C(N3CC4C(C4)C3)=O)CCC(F)(CC1)CC2.c1(C(=O)N)nc2c(s1)COCC2 C1CN(C(=O)Cc2cnc[nH]2)CCC1C.c1(C(=O)OC)cn(CC(=O)NC)nn1 C(C1=CCCCC1)NC(c1ccnc(CNC(c2n[nH]cc2Cl)=O)c1)=O c1(C(CCC2CCCO2)N(C)CC=CCF)cccnc1.C(CC(=O)OCCO)O c1(OC)ccc(CN2CCN(C(c3c(Br)cncc3Br)=O)CC2)cc1OC N1(C(CC(=CC(F)(F)F)Br)=O)CC2C3CCC(C3)C2C1 C1(C(=O)NCCC2OCCN(C(C=C(COC)C)=O)C2)CCc2nc(O)[nH]c2C1 N1(C(c2c(C)c(F)ncc2)C(=O)NCc2ccco2)CCCC2(C=CCO2)C1 C1(C(=O)NC(C)CC(C)NC(C2CCCC2)=O)(NC(=O)OC)CCCC1 c1(CC(=O)NC2CCN(C(=O)COCc3cccnc3)CC2)cc(O)nnc1O Cc1c(C=O)ccn1C1CC1.[SH](=O)(=O)C(F)(F)F.C1CCC1.C(=O)CC.N c1(C(N2CCCCC2C)=O)cnc(O)n(C)c1=O.C1(OC)(OC)CCC1C=O.N N1(C(c2cc(C)sc2C)=O)CC(C)OC(C)(C)C1.C1(C=O)CCCC(C)(C)C1.N Cc1cc(C(=O)NC2CCCN(C(=O)CSCC(N)=O)C2)n(C)n1 C(=O)(C(C)(C)C(F)F)NCC(CNC(C1(CC#C)CCOCC1)=O)C C(c1ccc(F)c(Cl)c1)=CC(N1CCCCC(NC(=O)CCc2cc[nH]n2)C1)=O c1(CNC(c2c(C)cc[nH]2)=O)nc(C)c(C(N2CCC2CF)=O)o1 C1(C(N(C23CCC(CC2)CC3)C)=O)COCCN(C(C2(n3nccn3)CC2)=O)C1 Cc1cc(C(N2CCN(C(C)C)CC2)=O)nc(O)c1.C12CC3CC1CC3C(=O)N2 c1(C(=O)NC(C)CC#N)cc(OCCc2ccccc2)ccc1F Cc1nc(N(CC(F)(F)Cl)C)cc(N2CCOC(C)(C(F)(F)F)C2)n1 c1(C(N2C(CNC(c3coc(C(F)F)c3)=O)CC2)=O)cnc(Cl)c(Cl)c1 CC(C)C(C(=O)N1CCN(C(C2CC2(Cl)Cl)=O)CC1)c1ccc(Cl)cc1 C12(CC(=O)NCCCCN(C)C(C34CC(C3)C4)=O)CCCCC1C2(F)F.C CCC(CC)(CO)C(=O)N1CCCC(N(C(=O)C(COC)COC)CCF)C1 c1(C(C(=O)NCC(CNC(C2C(C)C2)=O)CO)=O)cc(Cl)cc(Cl)c1 C1(OC)CC(C)N(C(=O)C2=CCOC2)C1.CC(F)(F)F.C(=O)(C=CC)N Cc1ccccc1OCC(C)(C)CNC(c1csc(CC(F)(F)F)n1)=O C1(C(N2CC(CC(CNC(C(CC)O)=O)(C)C)C2)=O)CCCC12CCOCC2 C1(CNC(COCc2[nH]c(=N)sc2)=O)CCCC(C)C1.C1(C=O)CCSC1 C1(NC(C(C)NC(CC)=O)=O)CC2CCC(C1)N2C(c1cccc(C)n1)=O c1(C(N2CC3CC(CNC(CCC)=O)C3C2)=O)n[nH]c2ccccc12 c1(OCC2N(Cc3[nH]nc(CC)n3)CC2)cccc(OC(C)C)c1 N1(C(C(CCN(C)C)NC(c2cnc[nH]c2=N)=O)=O)Cc2c[nH]nc2C1 c1(OCC)ccc(Cl)c(C(=O)NC2CC3CC2N(C(c2ccco2)=O)C3)n1.O N1(C(c2nn(C)c(=O)cc2)=O)CC2CC(C1)CN(C(=O)C#CC1CCCCO1)C2 C1(OC)(OC)CC(C)(NCC(F)(F)Oc2cccc(Br)c2)C1 C1(N(CC)C)CCCN(C(C)(C)C)C1=O.C1(C(N(C)CCO)=O)CCC(O)C1 CCC(CC)(CCNC(c1cnc(S)nc1)=O)NC(=O)Cn1nnnc1C c1(C(=O)NC2C(NC(C3(CCC)CCC3)=O)C2)cnc2[nH]ncc2c1 C1(NC(C(C)NC(CC)(C)C)=O)CC2(C1)CCC2.c1(C=O)ccnn1CCF C1(NC(c2c(CCC)n[nH]c2)=O)CN(C(=O)C(N2CCNC2=O)C)CCC1O N1(C(C)=O)CCC(C)(C(=O)NCC(C)N(C)C(C2CCNC(=O)C2)=O)CC1 c1(C(N(CCNC(C2CCC(O)CC2)=O)CC)=O)cc(C#N)c(N)cc1O C1(C(=O)NC2CCN(C(c3cccs3)=O)C2C2CC2)CCCCCCC1 C(=O)(C(C#N)C(C)(C)C)NC1C(C)N(C(=O)CCCN=[N+]=[N-])CCC1 N1(C(c2c(SC)cccn2)=O)CCN(C(=O)C(O)CC(C)C)CC1CC(F)(F)F c1(NC(C)CC(N)=O)cc(S(=O)(=O)NCCc2ccoc2)ccc1C#N O=C1CCC(c2cn(CCNC(=O)COCC(F)F)nn2)CC1 N1(C(c2n(C(C)C)ncc2Cl)=O)CCCCC(NC(C2(C)CCCC2(F)F)=O)C1 N1(C(CCC=CC)=O)CCn2nc(CNC(=O)C(C)Oc3ccccc3)cc2C1 c1(C=O)ncc2ccccn12.C(C(C)(C)CC(=O)NCC1CC(C)CO1)OC.N N1(C(C2CC(C3CCC3)C2)=O)CC(O)(C2CCN(C(C3CC3F)=O)CC2)C1 C1(NC(C2(CNC(c3c(C(C)C)onc3)=O)CC2)=O)CC2C=CC1C2 N1(C(CN(C)C(c2cccs2)=O)=O)CCC(c2cn(C3CCOC3)nn2)C1 C=CC(C)(O)CC(=O)N(CCC)C1CC1.c1(C(=O)N)nccnc1C(F)(F)F C1(C(=O)N(C2CN3CCC2CC3)C2CC2)CC2(CCCCN2)C1 Cc1ccc(CNC2CC(CNC(=O)CC(C)C(C)C)C23CCC3)cc1F CC(C)(CC(=O)NCC1COCC1NC(=O)COc1cccnc1)C1CC1 N1(N(c2cccc(O)c2)C(C)=O)CCC(NC(=O)C(F)(F)F)CC1 C=CC1(C(=O)NCCOCCC2CC2)CCN(C(=O)C#CC2CCCC2)CC1 CC(C(=O)NC1CC1C(F)(F)F)C(C)(C)c1ccccc1 c1(CNC2CC(C)CN(C(=O)Cc3cccc(C#N)c3)C2)csc2ccccc12 Cc1n[nH]cc1CN(C(=O)C(c1ccco1)NC(c1csc(F)c1)=O)C c1(OC)nc(=NC2CCCN(C(=O)C(C)CO)C2)[nH]c2[nH]cnc12 C=CCC(C(=O)N(CC1=CCSC1)C)NC(=O)CCc1ccncc1 C1(CC)CN(C(c2ccc(C)nc2O)=O)CCC1NC(=O)CN1CCCCC1=O N1(C(CC(C)C2CC2)=O)CCN(C(=O)Cc2cc(F)ccc2O)C(C)C1 CC1ON=C(C(=O)NC2CCCN(C(c3ccc(=O)n(CCO)c3)=O)C2)C1C c1(NC(C2N(Cc3ccc(OCC#C)cc3)CCC2)=O)ccc2nc(C)cn2c1 CC(CC(C)(C)C)C(=O)N1CCC(CO)(CNC(=O)Cc2ccon2)CC1 CC(N=c1[nH]c2cc(Cl)c(S(=O)(=O)NC(C)CCO)cc2s1)c1nnc(CO)s1 CCC(CC(=O)N1CC(N(C(=O)C=C2CCOCC2)C)C(C)(C)C1)C(C)(C)C Cc1[nH]nc2ncnc(N3CCN(C(c4c[nH]nc4[N+](=O)[O-])=O)CC(O)C3)c12 c1(OC)ccc(OC)c(CC(=O)N(C2CC2)Cc2noc(C)n2)c1 C1(O)(C(=O)NC(C)CN(C)C(C2CC3CC3C2)=O)CCOCC1 c1(NC(C2CCN(C(COC(C)=O)=O)CC2)=O)ncc(Br)cc1C c1(C(N2CCCC(CC(C)C(=O)O)C2)=O)cccc2occc12 c1(CC)onc(C)c1C(=O)N(CCC(=O)NC1CC2CCC1C2)C Cc1ccc(C(=O)N(CCC(=O)NC(CO)CCO)CCO)s1 c1ccc(Cl)c(C)c1.C1(CNC(C(c2ccccc2)OC)=O)C2CN(CC)CC12 N1(C(c2nc(CC)oc2C)=O)CCN(C(c2sccc2C)=O)C2CCCCC2C1 C1(C(NOCC(C)(C)O)=O)CCC(NC(c2cc(C(N)=O)[nH]n2)=O)C1 C=CCC(CNC(=O)CN1CCCNC1=O)C(=O)NC1CCC(=O)N(C)C1 C(=O)(CC(C(F)(F)F)c1ccon1)NCC(CO)NC(c1c(C)n(C)nc1)=O N1(C(c2c(CC)noc2)=O)CC(CNC(C2CC2C2CCC2)=O)C(C)C1 C(C#Cc1cn(CCO)nn1)NC(CN(C)C(N)=O)=O.C1CC2CC1C1C2C1(F)F N1(C(Cc2cn(C(C)C)nc2)=O)CCCC2(CCC(NC(C3(F)CCC3)=O)C2)C1 c1(C=O)c(O)cc(=O)n2c1CCCC2.n1(CC(=O)NC2CC2)nnc(=O)[nH]1.C N1(C(CNC(CCC)=O)=O)CC2CCC(CNC(=O)CCS(C)(=O)=O)(C2)C1 c1(C(=O)NC2CCCC(NC(C3(CCC=C)CC3)=O)C2)ccc2c(O)n[nH]c2c1 C1(NC(C2CC=C(C)CC2)=O)CC(C)CN(C(c2ccnn2CC(F)(F)F)=O)C1 C1(COC)CCN(C(c2cc[nH]n2)=O)C1.c1(CC(=O)N)cnn(C(C)C)c1 C1(C(N2CCC(NC(C(CC)OC)=O)C2)=O)CCN(C(=O)N(C)C)CC1 C1(C(N2C(C(C)NC(C=CSC)=O)CCC2)=O)CCCN(C(C)(C)C)C1=O C#Cc1ccc(NC(C2CN(C(C3CCC(CC)O3)=O)CC23CC3)=O)cc1 N1(C(C(CC#C)O)=O)CCOC2CN(C(=O)C(F)(F)C(F)F)CC12 C1(NC(c2n(CC)cnn2)=O)CC(NC(c2cc[n+]([O-])cc2)=O)C(O)C1 C1(CC)CN(C(=O)Cc2cccc(OC)c2OC)CCN1C(c1sncc1C)=O c1(NCC(CNC(c2c(CC)[nH]nc2Cl)=O)O)cc(C(C)C)nc2ncnn12 N1(C(CC2(C=C)CC2)=O)CCN(C(=O)C=Cc2cc[nH]c2)CC12CCC2 c1(C(N2CC(CCC)C2)=O)c(N)cc(C)cc1F.C(C)(C)C1(C=O)CC1.C C12(C=O)CCCC(C1)OC2.C1(CC(=O)NCc2nc(C)cs2)CCCOCC1.N C12(CNC(C(C)(C)NC(C3C(OC)CCCC3)=O)=O)CCC(CC1)CC2 C1(NC(=O)NCCCc2cccc(C)c2)CCC=CCCC1 CCCCCC(C)(CC)C(=O)NC1CCN(C(=O)C(C)COCC)CC1 N1(C(C=CSC)=O)CC(NC(=O)CCc2n[nH]c(=N)s2)CC12CCOC2 N1(C(C(C)S(N)(=O)=O)=O)CC2CCN(C(c3cc4c(s3)CCSC4)=O)CC2C1 C(C(CNC(c1n[nH]c(C)c1O)=O)C(F)(F)F)NC(C(C)SCC)=O c1(C(N2CCOC(C(F)(F)F)C2)C(=O)NC(CC)C)cc(Cl)ncc1Cl C#CC1(C(=O)NCc2c[nH]nc2C(=O)NC2CNC(=O)C23CC3)CCCCC1 c1(C(=O)NC(C(=O)N(CCCCOC)C)C2(C)CC2)sc(O)nc1C C(=O)C1=CN(C)S(=O)(=O)N=C1C.C1(NC(C2CC(SC)C2)=O)CCCC1.C C(=O)(CCC(C)(C)C)NCC(C)N(C(=O)CC1(C(F)(F)F)SCCS1)C c1(CC)cccc(C)c1NC(=O)C(c1cccc(C)c1Br)N1CCCC(CC)C1 c1(N2C3CC(NC(c4ccn(C)c4)=O)CC2CC3)ncc([N+](=O)[O-])cc1CO c1(CCC(N2CCC(NC(C=CC)=O)C2C)=O)c(C)nc2c(C#N)cnn2c1C C1(CNC(=O)C2=C(Cl)CC2)CN(C(=O)CN2C(=O)CNC2=O)CCC12CCOC2 C1(NC(c2cc(C(C)C)c(F)cc2)=O)CCN(C(=O)Cc2cocn2)CC1(C)C C1(NC(C(C(=C)C)(C)C)=O)CN(C(C2CCC(=C3CCC3)CC2)=O)CCC1(C)C c1(C(N2CCN(C(C(Br)=C(C)C)=O)C(C)C2)=O)cc2c(O)ccc(F)c2[nH]1 c1(N2CC(CNCc3ccc(O)c(O)c3)OCC2)ncnc2cc[nH]c12 CCC(C)C(C)C(=O)NCC(C)(C)NC(c1cn(C)nc1OC)=O C(=O)(CC(O)C(C)C)NC1C(CNC(c2c(C)coc2-c2ccccc2)=O)C1 CCCCC(C)C(=O)N1CCSCC1CCNC(=O)C(O)COC C1(C(C)NC(=O)O)CCCCN1C(C1CCC1C(F)(F)F)=O.C(C)(C)C c1(C=O)cnc(O)c([N+](=O)[O-])c1.Cc1cc(CC(=O)NCC2CCCC2)no1.N C1(C2CCC2)(C(N2CCC3(CC3)C2)=O)CC1(F)F.NC(=O)CSCC(=O)N N1(C(C(C)C(F)F)=O)CCc2nc(O)cc(C(=O)Nc3c(O)cccc3Cl)c2C1 C(N=c1[nH]cnc(Cl)c1[N+](=O)[O-])C1CCC(NC(C2(C)CNC(=O)C2)=O)CC1 c1(OC)ccc(CN2CCCC2(C)C(=O)Nc2cc(F)ncc2F)c(Br)n1 N1(C(Cn2nnc(C)n2)=O)CC(N(C(=O)Cn2nccc2C)C)C(O)C1 C1(c2cn(CCNC(C3(CCCOC)CCCC3)=O)nn2)CCCC(O)C1 C1(N(C)C(=O)C2CC2)(OCCNC(CN(C)C(N)=O)=O)CCC1 c1(-c2n(C)nnn2)ccc(S(=O)(=O)N2CC3(CCC3)C2)cc1 C1(C(NOCCOC(C)C)=O)C(C)OCCN1C(c1sccc1F)=O C1(COC)CC(C)CN(C(=O)CC2(C)CCN2C(c2cc(C#N)[nH]c2C)=O)C1 CN=c1[nH]c(C(N2CC3C(CNC(c4cncc(OC(F)F)c4)=O)C3C2)=O)cs1 c1(C(=O)NC2CN(C(CC3(C)CCC3)=O)CC23CCC3)ccc2c(c1)OCCO2 C(=O)(CC1=CCCCC1)N1CCN(C(C2(COC)C=CCC2)=O)CC1C(F)F c1(CONC(=O)C2(c3ccccn3)CCC2)c(F)c(F)c(F)c(F)c1F N1(C(C(C2CC2)OC)=O)CC(C)C2(CCC2)C1.C1(C=O)CCC1.C(C)C.N c1(OC)ccc(Br)cc1CC(=O)OCC(C)Cc1ccccc1 C1(C(=O)NC(C(=O)N(CC=C)C)(C)C2CCC2)CCCCC(=O)C1 C(=O)(C1=CC2CCC(C1)C2)NCc1ccc(C(N(C(CCSC)C)C)=O)o1 Cc1cc(C(=O)NC2(CO)CCN(C(c3cncnc3)=O)C2)ncc1C#N N1(C(c2c(C)n(CC3CC3)cc2)=O)CCC2CN(C(c3coc(Cl)c3)=O)CC12 c1(OC)nc(Cl)c(-c2nnc(CC(N3CCCCC3)=O)n2CC(C)C)s1.C1(S)CC1 N1(C(CN(C)CCO)=O)CCC1(C)C(=O)N(c1ccn(C2CC2)n1)C c1(C(N2CC(F)(C(=O)Nc3ccc(-c4ccco4)s3)C2)=O)cncc(Cl)n1 N1(C(=O)OC(C)(C)C)CCC2C(NCCc3cnc[nH]3)CC12 N1(C(c2c(NCc3cc(OC)ncc3)c[nH]n2)=O)CC2CCC(C1)O2 c1(SC)ccc(CN2CCC(C(C)NC(c3nccn3C)=O)C2)cc1 C1(OCC(C)NC(=O)CN2CCCC2)CCN(C(C2CCCCN2C)=O)CC1 CC1CN(C(c2cc(C(F)F)n(C)n2)=O)CCN1C(c1c(Cl)cnn1C)=O C1(NC(=O)CCN2CCOC2=O)CN(C(c2cnc(C(F)(F)F)cn2)=O)CC1O c1(C(=O)NC(C)CCNC(c2ccn(C)n2)=O)scc2c1CCCC2 C1(C)(C(=O)OCC)CCN(C(=NCCC=C(C)C)NCCC2CCCCC2)C1 CC1(C)CN(C(=O)CCn2cccc2)CC(C)O1.C1(C(=O)N)CCS(=O)(=O)N1 CC1(F)CCCN(C(=O)COC2CN(C(=O)CCc3nc[nH]n3)C2)C1 N1(C(CNC(CC)=O)=O)Cc2n[nH]cc2C1C(=O)N1C2CCC1CC(CC)C2 C1(NC(CCc2scc(C)n2)=O)CCC(N=c2[nH]nc(C3CC3)o2)CC1 c1(C(N2CC=CC(NC(c3cnc(OC)c(C)c3)=O)C2)=O)cc([N+](=O)[O-])cn1C CC(C)CC(CNC(=O)C(C)NS(C)(=O)=O)NC(c1cc(Cl)cs1)=O C=CCC(F)(F)C(=O)N1CC2(CCC2NC(c2cccc(C)c2F)=O)C1 c1(C(=O)NCC(CN(C(CC(c2cccc(F)c2)C)=O)C)O)ccc(N)cc1O Cn1ncc2c(C(=O)NC3CCCCN(C(C4(C)CC4(F)F)=O)CC3)ccnc12 C12(C(=O)Nc3cccc(OC)c3)CCN(C(=O)Cn3[nH]cnc3=N)CCC1C2 c1(OC)cc(Cl)c(C(C(=O)NC2CCOC2)N(C)Cc2ccc(C)nc2)cc1Cl N1(CCNC(C(c2ncn(C)n2)N(CC(F)Br)C)=O)CCOCC1 c1(NCC(=O)NC(CSC)C(=O)N(C)C(c2ccccc2)C)cccnc1 N1(C(CC(C)c2ccccc2)=O)CC(NC(=O)CCCCCF)CC(C)(C)C1 c1(C(=O)N)ccc(F)c2occc12.c1(CC)sc(C(=O)NCC2CC2)cc1C C=Cn1nccc1C(=O)N(C(CC)CC(=O)NCCCC1CCOC1)C c1(C(N2CC(NC(c3cn(CCF)nn3)=O)C(F)C2)=O)cnc2cccnc2c1 C1(CNC(C2(C(C)(F)F)CCC2)=O)CCCC1.N1(CCC(=O)N)CCCCC1 c1(C(N2CCC(CN(C)C(C3CC(F)C3)=O)C2)=O)cc(Br)ccc1N Cc1cncc(CC(=O)N(CC(CO)(CO)NC(=O)COC(F)(F)F)C)c1 C=CC(C)CC(=O)NCCCC1(NC(c2cn(C(F)(F)CO)nn2)=O)CC1 C1(OC)(C)CCN(C(c2cccc(N(C)C)c2)=O)C1.C1(C=O)CCC2(CC2)C1 CCCC(CC)C(=O)N(C)CCOCCC(=O)NCC1CC12CC2 C1(NCc2cn(CCNC(=O)NCCO)nn2)CCCCS1(=O)=O CCCCS(=O)(=O)NC1CCCC1C(=O)Nc1cnncc1Br c1(C(=O)NCCN(C(C2C(CC)CCC2)=O)CC)ccc([N+](=O)[O-])nc1 N(C1c2ccccc2CC1NC(=O)C(F)C1CC1)C(c1sccc1F)=O C1(C(=O)NCC(C)NC(C(CC)Oc2cccc(C)c2)=O)CC(C)(C)CN1C C=CCC(C)(O)C(=O)NCc1cc(C(=O)NC2CN(C(C)=O)CC2C)no1 C1(C=O)CC2CCC(C1)N2C1CC1.Cn1cc(Cl)cc1C(N1CCC(C)C1)=O.N C1(C(=O)NCC(C)NC(C2Cc3nccn3C2)=O)CCC(C)(F)CC1 c1(C(N(C(C=C)C2CC2)C)=O)ccc(CNC(c2c[nH]cc2CC)=O)o1 C1(NC(CCCOC)=O)CN(CCc2scnc2C)CC2(CCOCC2)C1 c1(C(N2CCCCC2CC)C(=O)NCCC)cnc2cccc(C)n12 CC(CN(C)C)CC(=O)NCc1cc(C(F)(F)F)cs1 c1(C(=O)NC2(C)CCN(C(=O)C=C3CCOCC3)C2)ccc(N=[N+]=[N-])cn1 N1(C(c2cc3nc(C)sc3[nH]2)=O)CC2CC(C)N(C(=O)CC3CC(F)C3)C2C1 C12(CNC(Cc3nc(C)sc3)=O)CC1CN(C(C1NC(=O)OC1C)=O)C2 C(=O)(C1=COCCO1)N(CCCO)C.C(=O)(C(C)(C)O)N(CCCCO)C N1(C(C)=O)CC(N(C)C(c2ccnc(C(C)(F)F)c2)=O)C(C)(C)C1.CCC=O.N CC(C)(CC(F)F)C(=O)NCC1CC(NC(c2cncc(N)c2)=O)C1 c1(C(=O)NC(C)CCCNC(C2CC(O)C2)=O)cc(Cl)sc1Cl c1(C(=O)NCC(CNC(C(C=C)(C)C)=O)C(F)(F)F)cc2cncc(C)c2s1 Nc1c(C(=O)NCC(O)CNC(=O)COc2ccon2)ccc(Cl)c1Cl CCC(C#N)CNC(C1(NC(=O)CCCNC(N)=O)CC1)=O C1(C(=O)NC(C)CNC(c2ncoc2C2CC2)=O)CC(F)CN1C Cc1cnc(C(=O)NC2(CNC(=O)C(C)(F)F)CCC2)c(Br)c1 C1(C(N2CCCC(NC(CC(CC)(C)C)=O)C2)=O)CCC2(CCCCC2)C1 c1(OC(C)COC2CCOC2)ccc(S(=O)(=O)N=C2CCCN2C)cc1 C1(C(=O)OC)CC(F)(F)CN1C(C1CC1)=O.c1(C=O)ccc(Cl)c(F)c1.N C(=O)C1CCCc2ncnn21.CC(C)(C(=O)NCC1CCC1)NS(C)(=O)=O CC(CO)(C(=O)NCC1COCC1N(C)C)NC(=O)COC1CCC1 c1(C(=O)NC(CNC(C(CC#C)C2CC2)=O)CC(C)C)c(Cl)ccc(F)c1C Cc1ccc(F)c(C(=O)NC2CN(C(=O)CCNS(C)(=O)=O)CC2C)c1Cl C1C(C2CC2)CCN1C(=O)C=Cc1ncc[nH]1.c1(C(=O)N)cc2sccc2s1.C CC1(C)CN(C(c2cc(Cl)no2)=O)CC1CNC(=O)CCC.C(=O)C1CC1 C(CCN=C(NCCCN(C)C1CC1)N1CC(C)C(C)C1)N(C(C)C)C N1(CC)CCCN(C(C2CCN2C(=O)C(C)n2cccn2)=O)CC1 N1(C(c2csc(Cl)c2)C(=O)Nc2c(C)cccc2)CCCC2CC(O)CCC12 N1(c2ncc(C)c(O)n2)CCC(NC(c2cc3ncccc3[nH]2)=O)C(C)(C)C1 N1(C(c2cncc(C)n2)=O)CCCN(C(c2n[nH]cc2C(F)(F)F)=O)CC1CO c1(OC)cccc(C#N)c1NC(C1(F)CCN(C(c2ccc(Br)cc2)=O)CC1)=O C(=O)(C1=C(Cl)CCCC1)N1CC2C(CNC(CNS(NC)(=O)=O)=O)(C2)C1 c1(C(=O)NCC2(O)CN(C(c3ccc(Br)c(Cl)c3)=O)C2)ccc2ncncc2c1 C(=O)(C(C)S(N)(=O)=O)NCC1N(C(C(C)=CC2CC2)=O)CC1 C(C(F)(F)C(=O)N1CC(CC(C)NC(c2nc(C(C)(F)F)cs2)=O)C1)OC C=CCCCCC(O)CNC(=O)C.c1(C(=O)OCC)ccc(C2CC2C)o1 C1(NC(C2CC23CC3)=O)CCS(=O)(=O)C12CN(C(=O)CC1OCCCO1)C2 C(=O)(CC(C)C(C)C)NCC1(O)CN(C(c2n[nH]c(C)c2O)=O)C1 n1(CC)ncc(C(=O)N(C2CN(C(C3(CCO)CC3)=O)CC2O)C)c1C C1(C(=O)NCC(CCNC(c2cnn(C)c2Cl)=O)O)CC2C=CCC(C1)C2 C1(C(=O)NC2C=CCN(C(c3cn(CC)nc3)=O)C2)CCC2(C1)CC2(F)F N1(C(=O)CCc2cnn[nH]2)C2CCC1CC(CCNC(C1(F)CCCCC1)=O)C2 N1(C(CCCC(=O)NCC)=O)CCC2(CCCC2)CC1.C(=O)(C=CS(C)(=O)=O)N c1(CC)cc(C(N2CCCC(C)C2CNC(=O)Cn2ccnn2)=O)cc(Cl)n1 c1(C(=O)NC2CCN(CCNC(CC(=C)C)=O)CC2)ccnc(C)c1C c1(NC)cnc(C(N2CCOC(CNC(C3CCCCN3C)=O)C2)=O)cn1 C(=O)(C(O)CC(N)=O)N(C)CC1(NC(=O)CN2CCCS2(=O)=O)CC1 c1(CN(C)C(c2n[nH]cc2CNC(=O)CC2C=CCC2)=O)ncncn1 C#Cc1cncc(C(=O)NC(CCNC(C2(Br)CC2(C)C)=O)C(C)C)c1 N1(C(C(CCC)NC(N)=O)=O)CCN(C(=O)C(C2CC2)OC)CC12CC2 CC1CCC2(CCC2)CN1C(=O)C(=O)N(C)Cc1cc(C(C)(C)C)n[nH]1 CCC(O)C(C)(C)C(=O)N1CCN(C(=O)C=Cc2ccncn2)C(CCOC)C1 CCCCCCC(C)NC(=O)C(C1CN(C(c2c[nH]c(=S)cn2)=O)C1)OC c1(CC)cc(C(=O)N(CC(=O)NCCN(C)CC)CC)ns1 C1(C(=O)NCCCC(CO)NC(=O)CCC2CCCO2)Cc2ccccc2O1 c1(C(N2CCCCC(N(C)C(c3ccco3)=O)C2)=O)cccc2c1CCO2 Cc1ccc(C(=O)NC2CC(C(N3CC(CO)OC(C)C3)=O)C2)cc1F C1(CC)CCN(C(c2c(C)cnn2C)=O)C1C.c1(C(=O)N)cc(C2CC2)on1 C1(N(C(C=COCC)=O)C)CCC(CNC(C2(F)CCCOC2)=O)CC1 C1(C2N(CCOC)CCC2)CCN(C(=O)C(C)OCCOc2ccccc2)CC1 C1(C(=O)OC)CC(n2cc(C3CC3)nn2)CN1C(c1csc(=N)[nH]1)=O Cc1c(CN2CC3C(CNC(C4CCC(F)(F)CC4)=O)C3C2)cccc1Br Cc1nc2[nH]ccc2c(=NCC2CN(C(C3CCC(C)(C)C3)=O)CCO2)[nH]1 c1(C(N(C(CCNC(c2cc(C)n(C)c2)=O)C)C)=O)ccc(C(N)=O)c(Cl)c1 c1(N(C)C)ncc(C(N2CC(N(C(=O)CCc3cnccn3)C)C(O)C2)=O)cn1 C1(NC(C(COCC)C)=O)C(C)(C)CN(C(C2OCC2(C)C)=O)CC1(C)C C1(C(=O)NC2(CNC(c3scc(OC)c3)=O)CCCC2)CCc2cncn2C1 N1(C(C(C)C(C)(F)F)=O)CCOC2(CCN(c3cc4c(cn3)C(=O)CCC4)C2)C1 CC1(C)CN(CCC(N2CCCC2CCNC(C2(C)C=CCCC2)=O)=O)CCS1 CCCC(C)C(=O)N1CC(NC(C2CC(SC)C2)=O)C(CO)C1 C(=O)(C1=NOC2(CCOC2)C1)NCC1N(C(Cc2cn(CC)nn2)=O)CCC1 C(C(F)(C(=O)N(CC(C)(C)C#N)C)C(C)C)NC(C(C(C)C)C)=O c1(OC)ccc(Cl)c(CC(N2CCCN(C(=O)C(C)SC)C(C)C2)=O)c1F C(=O)(CC(C(F)(F)F)n1cccn1)NC1C(NC(C(C(C)C)F)=O)CCCC1 C1(OCC)CN(C(c2nc(Cl)sc2C)=O)CC1C.C1(C=O)CN(C)C(=O)N1 Cc1cc2sc(C(=O)NCC3CC(F)C3)cc2s1.C(=O)C(C(C)O)N(C)C.C c1(CCC(=O)NC2(c3ccccc3)CCN(C(C3CCO3)=O)C2)ccc(Cl)cc1 C1(C(N2C(C(=O)NC)CCC2)=O)CCCCCCN1C(C12CC1CNC2=O)=O Cc1cc(NC(=O)C(C)SC(F)(F)F)ccc1NC(=O)Cc1cncnc1 c1(CSCC(=O)N(CC(C)NC(=O)C(F)C2CCC2)C)cccnc1 N1(C(c2c(CC)noc2C)=O)CC(C)CN(C(C23CC(C2)C3)=O)C(C)C1 O(NC(=O)CCCF)CC(N1C(CN=[N+]=[N-])CC1)=O Cc1nc(CC2CC2)oc1C(=O)NCC1C2CN(C)CC12.c1cnn(C)c1 c1(OC)ccc2c(c1)C(C(=O)N(C(C)CNC(=O)CCc1cccnc1)C)CC2 C#Cc1cccc(C(=O)NC2CCC(CC)C2)c1F.C(C)(C(C)C)=CC(=O)N C1(C(=O)NCC2(CNC(C(C)n3cccc3)=O)CCC2)CCOCC1(C)C CC(C)C(C(C)NC(C1C=CC=CC=C1)=O)NC(c1ncc[nH]c1=O)=O C(=O)(C1=CCC(C)CC1)N1CCN(C(C=CC=CC)=O)C(COC)C1 C1(NC(CC=CCC)=O)CCC(CNC(=O)C(C)(C)OC)CC1 c1(C(=O)NCCC2CC(NC(CC(C)CF)=O)C2)cc2n(n1)CCCC2 Cc1cccnc1C=CC(N1CCCC(O)(C)C1)=O.C1(C=O)CCS(=O)(=O)N1.N c1(C(N2CCC(O)(n3cc(-c4c(C)ccnc4)nn3)C2)=O)nccn(C)c1=O C1(C(=O)NC(CC)CNC(c2sc(C)cc2Br)=O)CCC(F)(F)CO1 CCCCC(O)C(=O)N1CCC(O)(CNC(c2cnc(S)[nH]2)=O)CC1 c1(-c2cn(CCC)nn2)cnn(C)c1C.C1(C(=O)OCC)CCC(C(=O)N)C1 c1(C(=O)NC2(CC=C)CN(C(=O)C3=CCCC3)C2)ccccc1CSCC Cc1cc(C(=O)NCC(C)(C)CN(C(=O)CCNC(=O)CC(C)C)C)no1 N1(C(Cc2ccc(C)o2)=O)CC(C)(C)CC1C(=O)NC1CN(C)CC1C C1(C(NNC(c2cnn(C)c2C(F)F)=O)=O)C(C2CC2)CCN1C=O.C(C)(C)C C(c1ccccc1OC)=CC(N1CC(NC(C2N(CCC)CCC2)=O)C(F)C1)=O C1(NC(C(CC=C)C)=O)COC2(CCN(C(c3cc4nc(C)ccc4o3)=O)C2)C1 c1(C(N2CCC(NC(CN(C)CCO)=O)C(F)C2)=O)cc2ccc(Cl)c(F)c2o1 c1(OC)ccc(Cl)cc1CC(=O)NC1CCOCC1.C1(C(C)(C)O)(C=O)CC1 C1(C(C)NC(c2cc(C(C)C)on2)=O)CCCN(C(c2coc(CO)c2)=O)C1 Cc1cc(NC(c2scnc2Cl)=O)ccc1NC(c1nnc(O)nc1O)=O c1(C(N2CC3(C(NC(c4cn(C5CC5)nn4)=O)CC3)C2)=O)[nH]nc2cnccc12 N#Cc1nc(NC(c2cscc2C2CCCC2)=O)ccc1Cl C(=O)(C1=CC2C=CC(C1)C2)N1CC(CCC)N(C(=O)COCCSC)CC1 Cc1nc(NCc2cnn3ccn(C)c23)cc(=NCc2nc(C3CC3)n[nH]2)[nH]1 c1(C(N2C(C(C)C)CN(C(C3CCC3(C)C)=O)CC2)=O)cncc([N+](=O)[O-])c1 C(=O)(C(C)(C)C(=O)NC)NC.C1(C(N2CCCCC2)=O)CCN(C)S1(=O)=O.C C1(Nc2c(OC)cncn2)CCC2CN(C(C3(C)CC(O)CN3C)=O)CCC2C1 c1(C(=O)NC(CCC)C(=O)NC(COC)C(C)C)cc(C)cc(C)c1 C=CC(C)CC(=O)N(C1CCN(C(=O)Cn2cnc(-c3ccccc3)n2)CC1)C N1(C(CC)C(N)=O)CCCC2(CCN(C(c3ccc4nnnn4c3)=O)C2)C1 c1(CN2CC(CC(N3C(C(N(C)C)=O)CCC3)=O)C2)ccc(N(C)CCO)cc1 c1(CN2CC3C(NC(CN4C(C)(C)CCC4)=O)C3C2)cc(F)ccc1F N1(C2CN(C(C3CCC(C)S3)=O)C2)CCN(C(c2cc(Br)c[nH]2)=O)CC1 C(CN=[N+]=[N-])(C(=O)NCC1CCCO1)NC(c1nc(C)sc1)=O c1(C(=O)Nc2ccc(C(N3CCOCC(O)C3)=O)nc2)nc2ccccc2o1 c1(C(=O)OC)ccc(NC(C2CN(C(c3sccc3Cl)=O)CCC2O)=O)c(O)c1 Cc1nc(Cl)nc(N2CCCC(NC(c3scnc3C(F)F)=O)C2)c1F c1(OCC)cccc(CC(N2CCCC2CN(C)C(c2[nH]c(C)nc2C)=O)=O)n1 C(=O)(CCS(=O)(=O)NC)N1CCC(N(C(=O)CC(=O)OC(C)C)CC)CC1 C1(C(=O)NC(c2ccc3ncsc3c2)C)CC(C(=O)O)=NN1c1ccccc1 CC1C(C(=O)NCCCNC(=O)C(C)Oc2ccccc2Cl)=Cc2ccccc21 c1(SC)cc(C(F)(F)F)ccc1NC(N1CCC1CNC(C)CO)=O c1(C(=O)Nc2c(C(=O)OC)scn2)n[nH]c2c1CN(C)CC2.c1(C=O)ccns1 c1(C(=O)NCc2cc(C(F)(F)F)ccc2Cl)cn2cnnc2cn1 C1CN2CCCC1C2.C1(C=O)(CNC(CCC=CC(C)C)=O)CC(C)(C)C1.N Cc1cc(C)c([N+](=O)[O-])cc1C(=O)NC1CC2CC1N(C(C1CC=CCO1)=O)C2 C(=O)(CCC(C)(C)N(C)C)NC(CC)CNC(=O)Cc1nn(C)cc1Cl Cc1csc(C(N2CC(C)CC2C(=O)Nc2cccnc2C)=O)c1Cl Cc1nn(C)c(C)c1NC(=O)C(c1ccc(C(c2ccc(Cl)c(Cl)c2)=O)cc1)C C1(NC(C(=O)N(C2CCCC2)CC(C)C)=O)CCN(CC(O)CO)CC1 c1(C(=O)NC2C(NC(C3(F)C(C)C3)=O)COC2)cccc(C2(O)COC2)c1 c1(CC)cnc(O)c(-c2nc(CC(C)OC)nn2-c2ccnc(Cl)c2)c1 C1(N=c2ccn(C(C)C3CC3)[nH]2)(c2n(C(CC)(C)C)nnn2)CCCCC1C CC1(C(N2CCC23CN(C(c2c(Cl)cncc2Cl)=O)C3)=O)CC(C2CC2)=NO1 Cc1cc(C(=O)NC2CCCC2C(=O)NCc2ccc(C(N)=O)o2)ncn1 N1(C(CC)=O)CC2(CCCCN2C(=O)Cn2nc(C)n(C)c2=O)C1.C=CCCO c1(OC)cnc(Cl)cc1C(N1CCN(C(=O)C#CC(C)C)C(C2CC2)C1)=O C1(CC(=O)NC2(CNC(CC(=C=C)C)=O)CCOCC2)CCC(C)(C)CC1 c1(C(N(CCC(=O)O)CCOC)=O)nnn(-c2cccc(Cl)c2)c1C(C)C c1(C(N(C)CC2(O)CCCN(C(=O)CCC(N)=O)C2)=O)sccc1S(C)(=O)=O C1(CNC(C2CCCC2)=O)CCN(c2cc(NC3CCCCC3)ncn2)C12CC2 N1(C(C(C)O)=O)C(C(=O)NCC(=C2CCCCC2)F)CCC12CC2 C1(CC(=O)NC2(C)CCC2)CC2(CCO1)CC2.C1(C=O)CCOC1C1CC1.N CC(C)(O)CC(=O)NC(C(=O)NC1COC(C)(C)C1)C1CCCC1 C(=O)(CC(C)(C)C(=O)N1CCC(C)C(NC(c2[nH]nnc2C)=O)C1)OC N1(C(=O)CC2COCCO2)CCN(C(c2cc3n(n2)CCO3)=O)C(CC2CC2)C1 C1(NC(=O)Cn2cccc2)CCCCCCC1NC(C1CCn2cnnc2C1)=O C12(C(N(CCCC(=O)OC)C)=O)CC1CCN2C(c1nc(Cl)oc1C)=O n1(CC=O)c(C)cc2ccccc12.C(C(C)C)NC(C1C(COC)C1)=O.N c1(C=O)ccc(C#CC2CC2)cc1.c1(SC)ccc(C(=O)NC2(C)CCC2)o1.N Cc1ccc(C(N2CC=C(Br)CC2)=O)c(-n2cc(C(O)C(C)C)nn2)c1 N1(C(C2(c3cc(F)cc(F)c3)CC2)=O)CCN(Cc2cccs2)CC1CCO C=CC(C)(C)CC(=O)N1C(C(=O)NCc2cc(C)nc(O)c2)CC1C C(=O)(CC(C)OC)NCCSCC(=O)NC(c1cccnc1)CC CC1=C(C(=O)N2CC3CC3C2C(=O)NC2CC(CN(C)C)C2)CCC1 C(=O)CC(C)C(F)(F)F.c1(CC(=O)N(C(C)C)C)cscn1.[SH](C)(=O)=O Cc1nn(C)cc1C(C)NC(C1CC12CCC2)=O.C1(CCC(=O)N)CCOCC1 Cc1ccc(C(=O)NC(C2CC=CCC2)C(=O)NCc2cccnc2O)c(O)c1 Cc1[nH]nc(C(=O)NC2(C(=O)NCC(n3cccn3)C)CCCC2C)c1O c1(C(N(C(CNC(C(C)N(C)Cc2ccccc2)=O)C)C)=O)c(O)cccc1Cl C(C(C(=O)NC1COCC1CO)NC(=O)CN1CCCC1C)OC c1(OC)ccc(C)cc1CC(=O)NC1(C)CCN(C(=O)C(c2ccccc2)F)C1 C(=O)(C#CC(C)(C)O)N1CCCC(N(C)C(c2cnn(CC(F)F)n2)=O)C1 CC1Oc2ccc(C(=O)Nc3ccc4c(c3)CN(C(=O)CC#N)C4)cc2NC1=O C(=O)(CS(=O)(=O)CCO)N.Cc1ncccc1C(=O)N(C)Cc1ccc(C)cc1 C1(NC(CN(c2cnccn2)C)=O)CCN(C(c2cnn[nH]2)=O)CC1F c1(C(=O)NC(C)C(C)(C)NC(c2cnccn2)=O)cccc2c1CC(C)(C)C2 c1(C(=O)N)ccc(C)[nH]1.C(C)(CNC(=O)C=CCC)NC(=O)OC C1(NC(=O)NCCC=C)C2CCC(C2)C1C(=O)Nc1ccc(Br)nc1I n1(CC)nc(C)cc1C(=O)NCCCC(C)C.c1(C(=O)N)ccc(C(F)F)s1 c1(C(=O)NC2CCCN(C(CCCC#C)=O)C2)ccc2c(c1)OCC2 c1(N(CC(C)CNC(C2CC3(CC3)C2)=O)C)cc(Cl)nc(S(C)(=O)=O)n1 Cc1ccc(C=CC(N2CCC=CC2C(=O)NCC2CCC(C)(C)O2)=O)o1 Cc1ccsc1CC(=O)NC(CN(C)C)C(=O)NC(C)Cc1cn[nH]c1 c1(C(N2CCCC(NC(=O)CCc3ccccn3)C2)=O)n[nH]c2nccc(Cl)c12 C=CCCCCC(=O)N1CCC(CNC(C2(CF)CCOCC2)=O)C1(C)C CCCC(C)(O)CC(=O)N1CC=C(CNC(c2nc(OC)cc(OC)n2)=O)CC1 N1(CC=O)CC(=O)NC1=O.C(C(O)CC)NC(COCCOCC)=O.N C1(C)(OC)CCN(C(C2(F)CCN(C(C3CCC(C)O3)=O)C2)=O)CC1 c1(CNC2C=CC(NC(=O)OC(C)(C)C)C2)ccc(C2CCC2)cc1 C=Cc1cncc(C(=O)NC2COCC2NC(C2CCCO2)=O)c1 C(=O)(C(F)(F)C(F)(F)C(F)F)N.C1(NC(c2n(C)cnc2)=O)COC2CCOC12 c1(C(=O)N)cnc2sccc2c1.C12CC1CN(C(C1CC(=O)N(C3CC3)C1)=O)C2 c1(C(=O)NC2CCN(c3cc(OC)nc(C)n3)C2)ccc2ccn(C)c2c1 N1(C(C2(C(=O)NC)CCC2)=O)CCOCC(CNC(=O)CCc2cnco2)C1 C=CC1(C(N2CCC(CN(C)C(c3ccc(N)c(Cl)n3)=O)C2)=O)CCCCC1 c1(CC(=O)NCCN(c2cc(C(=O)O)ncn2)CCC)ccc(Cl)c(F)c1 Cc1cc(C)c(C(=O)NC2(CO)CN(C(C3(C)CCC(=O)C3)=O)C2)cn1 c1(OC)ccccc1C(C)C(=O)NC1(C)CCN(C(c2coc(C)c2)=O)C1 CC1(CC(=O)NC(C)(C)CCCNC(=O)Cn2nnc(=N)[nH]2)CCOCC1 c1(C(=O)NCC(CO)NC(C2CC(C#N)(OC)C2)=O)cc2occ(Br)c2[nH]1 C1(CCC(=O)NCC2(F)CCN(C)C2)CCCCN(C(=O)C=C2CCCCC2)C1 C1(C(=O)NC2CN(C(C3SCCCS3)=O)CC23CC3)Cc2cc(Cl)ccc2O1 CCC(C(=O)N1CCC(CN(C)C(C2CC23CC3)=O)C1)N(CC)CC c1(CNC(=O)CC2CCN2C(c2cc[n+]([O-])cc2)=O)cccc(F)c1F S(=O)(=O)(c1c[nH]ccc1=NCC(C)C1CCC1)N(C)Cc1c(Br)cnn1C N1(C(c2n(C)cnc2Br)=O)CCC2(CC(NC(=O)CSC3CC3)CO2)C1 CC1(C(N2CC(O)(CCNC(=O)CCS)C2)=O)CCCC1(F)F.c1ccccn1 c1(CC)cccc(C(=O)NC(CNC(C2(O)CC2(C)C)=O)CO)c1 C(CC(C(CC)CC)OC)NC(=O)NC1(CC)CCC(C)(C)C1 N1(C(C(C(C)C)SC)=O)CC2(CC2)CC1C.C(c1cnc(C)s1)=CC=O.N n1(CC)c(C(=O)N(CCNC(=O)C(C)C)Cc2cccc(Cl)c2)cnc1O C1(C(N2CC(CCNC(C3=CC(C)(C)C3)=O)OCCC2)=O)Cc2ccccc2S1 c1(OC)ccc2c(N3CCCCC(CO)C3)nc(N3CCC(F)C3)nc2c1 n1(CC(N2C(CNC(=O)CCC3CC3)CCC(C)C2)=O)cnc2c1CCCC2 c1(CCC(=O)NC2(COC)CN(C(=O)C)C2)ccc(O)nn1.CC(C)C.S C(=O)(CC(O)CC(C)(C)C)N1CCCCCC1.C1(C(=O)NC)(CC)CNC(=O)C1 n1(CC)ncc(CNCCC(C)(C)O)c1C N1(C(CC(=O)NCC#C)=O)CC(O)CC1C(=O)NCC1(C)CCCC1O C1(NC(C2(CCC)CC2)=O)CCCCN(C(c2cccnn2)=O)C1 C1(NC(c2csc(C)c2C)=O)CN(C(C2CC2C(C)C)=O)CCC12CCC2 C1(CNC(c2cc3c([nH]2)CCC3)=O)CC2(CCC2)CN1C(=O)C1=CCCC1 S(=O)(=O)(c1ccc(Br)cc1N1CCC(Cc2ccc(F)cc2)C1)N(CC=C)C CN1C(=O)CCC1C(=O)N.C12CC1CN(C(c1ccn(CCC(F)(F)F)n1)=O)C2 Cc1cc(C(N2CCC(CNC(c3cnn(C)c3N)=O)CC2)=O)ccc1C(C)C N1(c2ccnc(SC)n2)CCC(NC(c2ncoc2C(C)(C)C)=O)CC1C C=CC1(C(=O)NOCC2CCCO2)CCN(C(=O)C(CC(=C)C)OC)CC1 N1(C(c2n(C)cc(Br)c2)=O)CC(CNC(C23CCC2C3)=O)C(C)(C)C1 CC(C)C(O)C(F)(F)C(=O)NC1COCCC1NC(c1scnc1C(F)F)=O Cc1ccn(C)c(=O)c1NC(C1CC(C)N1C(C1(C(C)C)CCC1)=O)=O Cc1cc(N)cnc1C(=O)NC1CCC1NC(C1CC(C)(C)CCO1)=O c1(C(N2CCN(CCN(C(=O)CCC(F)F)C)CC2)=O)cccc2nc[nH]c12 C1(NC(CCNC(COC)=O)=O)CCCCC1C.c1(CC=O)cncc(F)c1 N1(C(C2CC(C)(F)C2)=O)CC2CCC1C1CN(C(c3ncc(F)cc3F)=O)CC21 c1(C(C)=O)cccc(OCC=O)c1.C1(C)CCN(C(C2CC3(C2)CC3F)=O)C1.N C(=O)(C(O)CC1CCOCC1)NC(CNC(C(C)NC(C)=O)=O)C C(CC(=O)N1CC(C)C1)(C(C)C)OCC.C(=O)C(C)Cc1cnn(C)c1.O C(=O)(C(CC)C(F)(F)F)NC(CC#C)(C)C(=O)NCC(C)C(C)O S(=O)(=O)(C1CCN(C(=NCCOC2(C)CCC2)NCCF)C1)N(C)C C1C2CN(C(C3(n4cnnn4)CC3)=O)CC12.c1(C(=O)N)cncc(C2CC2)c1 c1(C(=O)NC(CNC(C(CCCC)O)=O)C)cc(OC)c(O)c([N+](=O)[O-])c1 Cc1ccc(C(=O)NCC2CCN(Cc3ccc(Cl)cc3C)C2)c(C)c1 c1(C(=O)NCCC2N(C(C=C(C)Cl)=O)CCCC2)cc(N)nc(Cl)c1 C1(NC(C2(C)C(C)CCC2)=O)CC(N=c2[nH]nc(C3CC3)o2)C1 C1(N(C(c2nc(CCC)sc2)=O)C)CCC(NC(c2occc2C)=O)CC1 C(=O)(C(CCC1CC1)NC(=O)CC1CCCC12CC2)N(CC(CC)(F)F)C c1(CC)ccc(Br)cc1C(=O)NCC1(O)CCCN(C(=O)C=NOC)C1 c1(SC)nn(C)cc1C(N1CCC(F)(CNC(=O)C(C)N2CCCC2)C1)=O C(=O)(CCCCCCNC(=O)C=Cc1cocn1)N1CC(CC)OCC1 C(=O)CC(C)C.CCCC(C1CCC1)NC(=O)C(c1ccco1)NC(=O)C C(c1cnccc1C)=CC(=O)N(C1CCCCC1NC(=O)CO)C.C1CCC1 CCC(C)C(CC(=O)NCC1CC(C)(O)C1)NC(=O)CC1CC=CCC1 CC(C)C(C(=O)NC(C1CCN(C(c2ccncc2C(F)(F)F)=O)C1)C)C(C)C N1(C(c2c(SC)csc2)=O)CC(C2CN(C(C3(O)CCCC(C)CC3)=O)C2)C1 n1(CC(N2CC=CC(NC(c3c(C)ocn3)=O)C2)=O)[nH]cc2c(=O)ncnc1-2 N1(CC(=O)NCC(C)CO)CCCC(CC(=O)OC(C)(C)C)C1 N1(C(C(C(C)C)SCC)=O)CCCC(C)(C)C1C.c1(CC=O)cscn1.N c1(CC)ccc(C(=O)NCC(F)CNC(=O)C(c2ccc(F)cc2)CO)cc1 C1(NC(C)=O)C(C)(C)C(NC(C23C(=O)C4CC2C3C4)=O)C1(C)C CC1CN(C(=O)CN2CCCCC2)CC1C.C(=O)(CC(C1CCC1)C1CCC1)N N1(C(CC)=O)CCC(Cn2cc(CNC3CCC3)nn2)C1 C(c1cnn(C)c1)=CC(=O)NCCCCN(C(=O)CN1CCCNC1=O)C C#CCC(CC(F)(F)F)NC(=O)NC1CCC2(C1)OCCO2 CC(C)C(C)CN(CCC(N1CC(O)(C)C1)=O)C.C(=O)(C(F)(F)C1CC1)N c1(CC#N)ccc(CNC(=O)NCc2ccnnc2O)cc1 CCCCCC(CNc1ncccc1-c1ccccn1)CO c1(C(=O)NCC(C(=O)NCCC2CC3C=CC2C3)N(C)C)cccc2[nH]ccc12 n1(CC)c(O)nc2ccc(NC(N3CCC(C(=O)O)C3)=O)cc12 c1(C(=O)NCC(CNC(c2c(C)ncc(N)c2)=O)CO)cnc2[nH]cncc1-2 c1(C(=O)Nc2cccc(CC)n2)cc(-c2cc(F)cc(F)c2F)cc2[nH]ccc12 NC1COC2(CCN(C(C3CC4CCC3N4C(C3CC3F)=O)=O)CC2)C1 N1(C(CCNC(=O)OCC)=O)CCCC(C)CC1.c1(C=O)cc(Cl)nc(Cl)c1 C(C(O)(CNC(C1(NC(=O)CCn2ccnc2)CC(O)C1)=O)CO)OC CC1CN(C(=O)CN2CCCCCC2)CC1OCCNCCN(C)C CCC(C)N=c1ccnc(NC2CCOC(c3ccccn3)C2)[nH]1 c1(C=O)n[nH]c(C)c1C(F)(F)F.C(CC)C(=O)N(CCC)C(C)C.CC.O N1(C(c2c(C)c[nH]c2)=O)CC(N(C)C(c2cc(-c3ccns3)on2)=O)C(O)C1 c1(C(=O)NC(C)(C)C(=O)NCC2CCCC(=O)N2)ccc(Cl)cn1 c1(C(C)=O)cc(C(N2CC(F)(C)C2)=O)n(C)c1.c1(C(C=O)C)ccccc1C.N C1(NC(c2c(C)coc2C)=O)CC2(CCN(C(=O)C(C)C(F)(F)C(F)F)CC2)C1 C(=O)(C1CCCc2sc(=N)[nH]c21)NCC(CC(C)C)(C)NC(C12CCC1CC2)=O C1(N(C(=O)Cc2cncnc2)CC#C)CCN(CC(Cl)=CCl)CC1 C1(NC(c2c(C(C)C)c[nH]n2)=O)CC2CC1N(C(C1(c3ccncc3)CC1)=O)C2 c1(C(=O)NCC2N(C(C3C(C=C)C3)=O)CC2)ccc2cc(Br)ccc2n1 C(CC(C)NC(=O)C=CCN(C(=O)C(OC)OC)C)SCC C1(CCCNC(=O)COC(F)(F)F)(CNC(CCOCC)=O)CCCC1 Cc1cc(C=CC(=O)NCc2n[nH]cc2C=O)on1.c1(CCC)c[nH]nc1C.N C(=O)(C(C)(C)CCC(=O)OC)NC(C1CCN(C(c2cnc(CC)s2)=O)C1)C Cc1c(C=O)nnn1-c1cnn(C)c1.C1C2CC1N(C(=O)C=CC(F)(F)F)C2 C#CC(C)(C)C(=O)N1CCC(CC=C)(NC(=O)CCSCCOC)C1 c12cnc(nc1)oc2=O.C(CCNC(=O)CN(C)CC)OC.C(C)(C)C C12(C(=O)NC(CN(CC)CC)C)CCCC1CCN2C(=O)CNC=O C(=O)(CCCC(C)C)NC1CC(C)(OC)C1(C)C.n1(CC(=O)N)cccnc1=O C(=O)(CCC(=O)c1cnn(C)c1)NC(C(C)NC(C(F)=CCC)=O)C c1(OC(C(=O)NCC2(F)CN(C(CCC#CC)=O)C2)C)ccc(F)c(F)c1 C1(CC(=O)NC(C(C)C)C2CCC2)CN(C(=O)CCc2ncccn2)CC12CC2 c1(C(N2C(C)CCN(C(=O)CC3CCCOC3)CC2)=O)cccc(C=C(F)F)c1 C1(C)(C(N(C)CC2N(CC)CCC2)=O)CCN(C(c2cncc(OC)n2)=O)C1 c1(C(=O)NCC(C)N(C(C(COC)O)=O)C)c(C#N)cnn1C Cc1ncc(C(=O)NC2CN(C(C3(N(C)C)CCC3)=O)CC2C)c(C(C)C)n1 C(=O)(C1=CCCC1)N(CC(N1CC(CN=[N+]=[N-])C1)=O)Cc1ccccc1 c1(C(=O)N)cc(F)ccc1Br.C1(N(C(=O)C(=O)NC(C)(C)C)C)CCCCC1 C1(C(=O)NCCN(CC(C)O)C(C2COC(=O)N2)=O)CC2CC(=O)C1O2 C1(CN(C(CCOCC#C)=O)CC)CCCC1NC(=O)CC1CC1C CC1(C)CCN(C(=O)COCCF)CC1C.c1(C(=O)N)ccccc1.C1CC1 c1(C(=O)NC2CC(C)N(Cc3cscn3)CC2)cc2c(cc1Cl)OCCO2 C=CCC(C)C(=O)NCC1CN(C(=O)CCCc2ccsc2)CC1C c1(C(C)=O)cn(C)nc1C(=O)NC.C1CCN(C(C2(C(N)=O)CC2)=O)C1 N1(CC)CCCC1C(=O)NC(CC1CCCC1)C(=O)NCC(C)O N1(C(c2c(C)nc(C)[nH]2)=O)CCN(C(C2(N3CCCC3)CCC2)=O)CC(O)C1 N1(C(C(C(C)O)C)=O)CC(C)CN(C(=O)COc2cc(F)cc(F)c2)C(C)C1 Nc1cnccc1CN1CCOCC1CC(c1ccco1)O c1(CC)c(C(=O)NC2CC(CCC(=O)Nc3cccnc3C(C)C)C2)ccn1C C(=O)(C(C(C)(C)C)NC(=O)CCCC(=O)OC)NCC1(CO)C(C=C)C1 CCC(C)(CNC(c1c[nH]c(C(N)=O)c1)=O)C(=O)N.c1cncn1C1CC1 C1(C2CCCC2)(C(=O)NC(CC=C)CNC(c2ncsc2C)=O)CCNC1=O C1(C(N2CC3(CO)CC2(C(N2CCC24CC(CO)C4)=O)C3)=O)CN2CCN1CC2 C1(C(N(C)CCc2ccccc2)=O)CCC(F)CC1 Cc1cccc(-n2cc(C(N3CCC(N(C)C(C4CC=CCO4)=O)C3)=O)nn2)c1 N1(C(c2cn(CC)nc2C)=O)CC(NC(c2cc(C)sc2C)=O)C2CCCCC12 C#CCC(C(=O)OC)NC(C1COCC1NC(=O)CCc1cn(C)cn1)=O O=C(CS(=O)(=O)NC1CC1)NCC1CCC1.C12(C(=O)N)CCCCC1C2 c1(C(=O)NCC(CNC(CC(C=C)(C)C)=O)F)ccc2c(c1)NC(=O)CN2 c1(C(N2CC(C)c3c2cccc3)=O)ccc(C#N)c([N+](=O)[O-])c1 c1(OC)nc(Cl)c(C(=O)N(CCCCN(C)Cc2cn(CCF)nn2)C)s1 C(=O)(C1Cc2ccccc21)NC1CN(C(C(CCCC)O)=O)CC1CCC CC(CC(=O)N(CCC(O)CO)C)C(C)(C)NC(=O)Cn1cccnc1=O c1(CCC(=O)NCCC(CNC(CC)=O)O)ccc(NC)cn1 C(=O)(CC(O)C(C)C)N(C1CC(NC(c2c(C)nc(CO)s2)=O)C1)C N1(C(c2c(F)ccc(OC(C)C)c2)C(=O)NC2CCC2)CCC(C)C(F)(F)C1 Cc1cc(-n2cccc2)ccc1C(=O)NCCCN(C)C(C1CCC(C)O1)=O N1(C(=O)OC)CCCC(C(N2CCC(CCC)CC2)=O)C1.C1(C(=O)N)CC(F)C1 C1(C(N(CCN(C(C(C2CCOC2)OC)=O)C)C(C)C)=O)COC(C)(C)C1 N1(C(C(C)CC(F)F)=O)CC(C(=O)NCCCN2CCOCC2)C(C2CC2)C1 C1(NC(c2nccc(C)c2)=O)CS(=O)(=O)CC1.c1(C=O)csnc1C1CC1.N N1(C(C(CNC(c2c(CCC)[nH]cc2)=O)C)=O)CCOCC1C C1(CCNC(CNC(CC)=O)=O)CN(C(=O)CNC=O)CC1C.C1CC1 C(=O)(CC(C)COC)NCC(C1CC1)NC(CNC(CC)=O)=O C1(NC(C=CC)=O)CC(C)CN(C(c2cc(C(F)(F)F)nn2CC)=O)C1 c1(C(CC)(C)C)ccc(C(=O)NCC2CCCCN2C(=O)Cc2cnsc2)cc1 N1(C(C2(CCC)CCC2)=O)CCCC(C)(c2cn(C(c3cccnc3)C)nn2)C1 S(=O)(=O)(c1cccc(C(=O)NC2COCC2NCc2ccnn2C)c1)NC C1(C(N2CC(C)CC(NC(CC(=C=C)C)=O)C2)=O)COc2ccc(Cl)cc2C1 CC(C)C(N=c1nc[nH]s1)C(C)NC(=O)Cc1ccc2oc(O)nc2c1 N1(C(CSC)=O)CCC(n2cc(CNC(C3(C#N)CCC3)=O)nn2)C1 C1(C(N2CCCC(C(N)=O)(NC)C2)=O)CC2(C1)CC(O)(C(F)(F)F)C2 C(=O)(C(F)C(C)C)NCCC1(OC)CN(C(C23CSCC2C3)=O)C1 N1(C(c2ccc(C=O)cc2)C(=O)NCC=C)CCS(=O)C(C)C1C.C1CC1.N Cc1nc(C(=O)OCc2cc(F)c(F)cc2Br)c2ccnc-2[nH]1 N1(C(c2c(CC)nc(=N)[nH]c2)=O)CC(C)OC2CCCC12.C(=O)(C)N.C(C)C N1(C(CC2C(CC)C2(F)F)=O)C(C)CN(C(c2cccn2C)=O)CC1C c1(C(=O)OCC)cc(S(=O)(=O)NC(c2ccc3c(n2)CCCC3)=O)ccc1F CC(C)(O)C(F)C(=O)NC1CC(NC(=O)CCc2ccc(Br)s2)C1 N1(C(Cc2cc(C)sc2)=O)CCC2(C(=O)NC3CCCC34CCC4)CCCC12 Cc1cc(=O)c(C(=O)N(C)CC2CN(C(c3ccnn3C)=O)C2)cn1C1CC1 C(=O)(NN1CCCC1C(=O)NC1C(=O)NCC1(C)C)c1cnc(C(C)=O)s1 c1(C(=O)NCC(CNC(c2ccon2)=O)F)cccc2cncn12 CC(=Cn1ccnn1)C(=O)NC1CN(C(C2CCCC2C)=O)C1 c1(C(=O)NCCOCCNC(C2CCC(C)S2)=O)cc2ccc(O)cc2[nH]1 CCCC(CCC)CC(=O)N1CCC(CNC(c2nn(C)cc2N)=O)C(CC)C1 C(=O)(CC(O)C(C)C)NCC1C(NC(c2c(C)snc2)=O)CC1 c1(CC)ccc(CNC(=O)C=CCN(C(=O)C(F)(F)C2CC2)C)nc1 C12(C(N3CC(NC(c4cc(CCCO)on4)=O)C(O)C3)=O)CCCC(C1)OC2 c1(C(=O)NC(C)Cn2cc(CN(C)C3CC3)nn2)ccc2c(c1)B(O)OC2 c1(C(N2CCCC(CNC(CCCCOCCC=C)=O)C2)=O)cc(F)cc(F)c1 C(c1cc(Cl)ccc1Cl)=CC(=O)NCC(CNC(CSc1nc(C)[nH]n1)=O)F c1(OCC)oc(C)nc1C(=O)NCC1(F)CCC1.C1(C(=O)N)CC1F C1(NC(Cn2c(C)ccn2)=O)CC(C(=O)NCCC(F)(F)CO)C12CCC2 Cc1ccc(C)c(CC(=O)NC(CO)CCCCNC(=O)C(O)CC(C)C)c1 N1(C(CC)=O)CC(N(C)C(C2CCC(C)CC2)=O)C(O)C1 CC(C)CC(C)(O)c1cn(Cc2ccc(C(=O)NCc3csnn3)o2)nn1 c1(OC)ccc(C(C(N2CCC(N(C)C(c3cnc[nH]c3=N)=O)C2)=O)OC)cc1 C=C=CCN=c1nc2scnc2c(NCCCOC(=O)NC)[nH]1 CC(C)C(C(=O)NCC1(NC(=O)CC2CC2)CC1)Nc1cccs1 Cc1ncc2n1CC(C(=O)NCCCCN(C)C(C1CCC(C)CC1)=O)CC2 C(C)(c1ccccc1F)=CC(N1C2CC(NC(CC(C)(C)OC)=O)C(C2)C1)=O Cn1nc(C(=O)NCCCn2cc(-c3ccncc3Cl)nn2)cc1Br c1(C(=O)NCC(CC=C)NC(C2CCCN2CCC)=O)cccc2nc(C)nn12 C(=O)(CC(C)CC(=O)NC1CCCC1C(N1CC(OC)CC(C)C1)=O)OC C1(C(=O)NCC2(C(N)=O)CN(C(C3(O)CC3)=O)C2)Cc2ccccc2N1 N1(C(C2(F)CCC(C)CC2)=O)Cc2[nH]nc(C(N3CC4(CSC4)C3)=O)c2C1 CC1CN(C(c2cncc(C(F)(F)F)n2)=O)CCC1.n1(CC(=O)N)cnc(=N)[nH]1 c1(C(N2CC(N(C)C3CC3)C2)=O)coc(C)c1.C1(C(C(=O)N)F)CCOCC1 C1(NC(=O)OC)CCC(C(=O)NCCCc2cn(-c3ncccc3C)nn2)CC1 CC(O)CCCC(=O)N(C(CNC(=O)C=CC)C1CC1)C.CC(F)(F)F.O c1c(F)cc(Br)cc1F.C1(NC(c2ccco2)=O)CC2(C1)CC(C(=O)N)C2.C C1(O)(C(=O)N)CC(C)(C)C1.c1(C(=O)OC)ccc(-c2cn(C(C)C)nn2)o1 CCC(C)(COC)C(=O)NC(C)CCCC(=O)N(CCCCN(C)C)C c1(C(N2CCC(NC(CC3(C)CCCO3)=O)C2C2CC2)=O)cnc2sccn12 C12(C(N3C(CC(=O)N(c4cn(CCC#C)nc4)C)CCC3)=O)CC1CNC2=O N1(C(C(C(C)(C)O)NC(=O)C=CC2CC2)=O)CC(=O)NC2(CC2)C1 c1(C(=O)NC(CCCC)CNC(c2ncncc2Cl)=O)c[nH]c2cc(C)ccc12 C#CCCCC(C)C(=O)NCC1(CNC(c2cc(N)cnc2Cl)=O)CC1 C1Cc2ccccc2C(C)(C)C1.C1(C)(CC=O)CCS(=O)(=O)N1.CC=O.CC.N c1(NC(=O)NC2CCCN(c3cc(Br)cc(F)n3)C2)ccc(F)c(F)c1F CCC(CC)C(F)C(=O)NC1CN(C(C2CC(=O)N(C)C2)=O)C2(CCC2)C1 c1(C(=O)NC(C)CC(C)NC(C2CCC(=O)C2)=O)ccc(Br)cc1F c1(C(=O)NCC(CC(C)C)NC(c2cccn(C)c2=O)=O)cc2scc(Cl)c2[nH]1 C=C(C)C(CC(=O)N(CC(C)(C)C(=O)NCCCOCCCC)C)OCC.N C(CCCO)(c1cccnc1)NC(=O)C(N1CCC(C(N2CCCCC2)=O)C1)=O Cn1c(C(=O)NCC2CCN(C(C3CCCS3)=O)CC2)cc2c(O)cccc12 O(NC(=O)C(CC1CCCC1)CC=C)C1C(C#C)CCC1.c1cc(F)cc(F)c1 C(=O)(C1=CCC(C)CC1)NC(C(C)C)(C)CNC(C1CCC=CCC1)=O N1(C(C#C)(C)C)CCN(C(=O)COC(C2(c3ccc(F)cc3)CCC2)=O)CC1 C1(C=O)CCCN(C(=O)CC2CCC2)C1.CC(C)(C)OC(=O)N.C1CC1 C1(CCOCC)(CNC(=O)CCOCC2CCCCO2)CCCC1 c1(OC)cccc2c(C(N3CCN(C(=O)CCOC(C)=O)C(C)C3)=O)coc12 N1(C(C(C)OCC#C)=O)CC(CC(=O)N(CCCO)CC)CC1(C)C CCC(CNC(C1(C)CN(C(c2n[nH]c(O)n2)=O)CC1C)=O)(CC)CC C1(C(C)NC(C2(SCC)CC2)=O)CCCN1C(=O)CC1CCN(C)C1 N1(C(C(C)S(N)(=O)=O)=O)CCC2(NC(=O)COC3(C)CCC3)CCCC12 c1(C(N2CCCC(NC(c3csc(C(F)(F)F)c3)=O)C2)=O)cn2ccnc2cn1 N1(C(c2ncn(CC)c2)=O)CCCCCC(NC(=O)Cn2nc(C)oc2=O)C1 CC(C(=O)NCCN(C(=O)CC1C=CCC1)C)N(C(=O)CON)C C(=O)(C(COC)C(F)(F)F)N1CCC(N(C(=O)CC(Cl)Cl)CCC)CC1 S(=O)(=O)(c1ccc([N+](=O)[O-])c(F)c1)N1CCC(NC(C2=NNC(=O)CC2)=O)C1 c1(CC)cccc2[nH]c(C(=O)NC3CC3C)cc12.C1(CC=O)C=CCCC1.N C12(CNC(C(=O)NC3(COC)CNC3)=O)CC(C)(CO1)C2 c1(C(=O)NCCN2C(C)COCC2)n[nH]c2c1CN(C(=O)CC=C(Cl)Cl)C2 c1(SC)ncc(C(=O)NCC2(C)CCCC2)n1C.C(=O)C=O.CC(F)(F)F c1(-c2nnc(N3C(c4ccc(OC)c(OC)c4)CCC3)o2)cccc([Si](C)(C)C)c1 c1(C(C=O)O)ccc(Cl)c(Cl)c1.C(C(=O)NCC=CC)(c1cscn1)N(C)C C(C)(CC(C)C)NC(c1cnc(CCCC)s1)=O.C1(CC(C)C)(C(=O)N)CC1 C12(C(=O)NCCC3(OC)CN(C(=O)CCCN(C)C)C3)CCCCCC1OCC2 C1(CC(=O)NC(C#C)(C)C2CC2)(OC)CN(C(=O)CC2C=CCCC2)C1 N1(C(Cc2c(Br)ccc(C)c2)=O)CC2(CCC(C)O2)C1.N1(CC(=O)N)CC=CC1 C1(C(=O)NCCCN(C(c2ccc(OC)s2)=O)C)OCCOC1(C)C C1=CC(=O)Nc2c(C(F)(F)F)ccc1c2.C1(C(C)(C)C)CC(C(=O)O)CO1 N1(c2nnc(C)s2)CCC(NC(c2cc(-c3cccs3)on2)=O)C2(CCC2)C1 N1(C(C(CC)OCC)=O)CC2CCCC2(C(=O)NCCn2cnnc2CC)C1 C#Cc1ccc(C(=O)NCCC2(C)CCN(C(=O)CCC(C)SC)C2)cc1 C=CC1(CC(=O)NCC2COC(CNC(=O)C3=C(Cl)CC3)C2)CCOCC1 C1(O)(CCNC(c2ccc(CCC)s2)=O)CCN(C(=O)CCCN2CCCC2)C1 c1(CC)cc(C(=O)NCCC)sc1C.C(=O)(C(F)CC1CC1)N.C1CCCC1 Cc1ccc2c(c1)C(C(=O)N(c1ccccc1)CC)C2.C(=O)(C(C#N)C1CC1)N CN1CC(C(=O)NCC2(O)CN(C(c3cc4ncccc4o3)=O)C2)OCCC1=O N1(C(c2c(CC)n[nH]c2)=O)CC(CNC(c2ccon2)=O)C(C)C1 c1(C(=O)NCC2(O)CN(C(C(C)(C)CO)=O)C2)cc(F)ccc1C(F)(F)F C(=O)(CC(C)CC(C)C)N1CCCC(N(C(c2sccc2Cl)=O)CC)C1 O=C1CN(CCC(=O)N2CC(NC(=O)CN3CCC(CO)CC3)C2)CCN1 N#Cc1cc(S(=O)(=O)NCc2ncc(Cl)cn2)ccc1NC.C1CCCC(F)C1 C1(NC(C(COC)C)=O)CCN(C(c2cc(Cl)ncc2Cl)=O)C(C)C1 N1(C(C)C(=O)Nc2cccc([N+](=O)[O-])c2)CCc2ccncc2C1 N1(C(C(=O)N(C)C2CC2)=O)CCCC12CCOC2.C(c1ccccn1)=CC(=O)N Cc1c(C(N2CCCC(NC(=O)CCCF)C2)=O)sc2[nH]cnc(=S)c12 C1(NC(CN2C(C)CC2)=O)C2COCC1CN(C(=O)CCCn1cccc1)C2 C1(C=O)CCCC1.c1ccccn1.c1(CC(=O)NCC2(C)CC2)nc[nH]n1.N C(CCC(=O)NC1(C)CCC1)NC(=O)OCC.C1(CC=O)CC2CC2C1 C1(c2nnnn2C)(Nc2nc(C)c(C)[nH]2)CCN(CC(F)(F)F)CC1 CC(C)CC(CC(C)C)C(=O)N1CC(C)CN(C(C2CC(Cl)(Cl)C2)=O)CC1C c1(C(=O)NC(CC=C)CNC(=O)C(N2CCOC2=O)C)cn(C)c(C)n1 Cc1cc(Br)ccc1SCC(N1CCC(NC(=O)C(F)n2ccnc2)C1)=O C1(CC)CCCN(C(C2CN(C(C)=O)C2)=O)C1.c1(C(=O)N)c[nH]c(C=O)c1 CCCCC(C(=O)NC1CC(C)(NC(c2ccncc2OC)=O)C1)C(C)C N(C(=NCCCOC)NCc1cc(F)cnc1Cl)CC(C(CC)CC)OCC Cc1nn(C)c(N)c1C(N1CCCC1c1ccc[nH]1)=O c1(OC)ccc(C=CC(=O)NCCC2(C)CCN(C(C3CCO3)=O)C2)cc1 C1(C(=O)NC2C(C(C)C)C2)CCCCN(C(c2cc(F)ccc2O)=O)C1 C#Cc1cccc(C(N2CC(N(C)C(C3CN(C(C)C)C3)=O)C(F)C2)=O)c1C c1(C(N2CCOCCC2)=O)cnc(S(C)(=O)=O)s1.C(C(=O)NC)(C(C)C)OC CC(C)(C)C(CNC(=O)CC1CN(C(=O)CC23CCC(CC2)C3)CCO1)CO Cc1cc(C(=O)NCC2(F)CCC2)c2c(O)n[nH]c2n1.C(=O)C(O)C(F)(F)F C(CO)(C(=O)N1CCC(NC(C2(n3ccnc3)CCCC2)=O)C1)N(C)C CC1(C)CCN(C(=O)CSc2n[nH]c(O)n2)C1C.C1(C=O)CCC=CCCC1.N c1(CC)ccsc1C(=O)NCc1occc1C(=O)NC1CCN(C)C1 c1(C(CC)C)nc(C(CC(C)C)OC)n(-c2cccc(C(F)(F)F)c2)n1 c1(C(=O)NC2(C3N(C(c4cc(C)oc4C)=O)CCC3)CC2)cnc2sccc2c1 N1(C(c2cccc(-c3nc(C)on3)c2)=O)CCC(C)(NC(c2ccoc2)=O)CC1 c1(C(=O)NC2CCCC(NC(COCC=C)=O)CC2)cc2n(n1)CCCC2 C1(CN(C)C(C2CCCC2F)=O)CCCC1NC(C1CC12CCC2)=O C1(F)(CNC(c2ccc(OC)cc2)=O)COCCN(C(=O)C#CC2CCCC2)C1 CCC(C(=O)NCC(N1CCCC1C1(C)CC1)=O)C(C)C c1(C(=O)NC(CC(C)C)CNC(=O)CC2CCOCC2)cccc2c1C(C#N)C2 C1C2CCC1N(C(=O)C(c1ccc(OC(F)(F)F)cc1)(C)C)C2.C(C=O)=CC.N C(=O)(C1=CCC(NC(=O)Cn2cccnc2=O)C1)N(C(C)C)CC1CCCO1 C1(C(=O)OC)CC(OC)CCN1CCC(=O)Nc1ccc(OC)cc1F c1(NCCC(c2ccccc2)O)nc2ccccc2nc1N1CC2C=CC2C1 C=CCC(F)(F)C(=O)N(CC(=O)NCC1CCCCN(C)C1)C C(=O)(C1=C(Cl)CCCC1)N1CCC(N2CCN(C(C(C)NC(N)=O)=O)CC2)CC1 C1(C(N2CC(F)CC(NC(CCN(C(C)=O)C)=O)C2)=O)CC(F)(F)CCC1(C)C C1(CNC(=O)CC(O)c2ccccc2)CC2CC2N1C(c1nc(Cl)c(Cl)s1)=O c1(C(=O)NCC2C(NC(C(C=C)(C)C)=O)CCC2)ccc(Br)nc1N C(C(C)(O)CC(=O)NCC1CCCCC1)OC.c1(CC=O)cn(C2CC2)cn1 N1(C(CCc2cccc(C)c2)=O)CC(NC(C23CC(C)C2C3)=O)CC12CCCC2 c1(CC(=O)O)c(C)nc2nc(=N)[nH]n2c1C.C(=O)(CCC1CC(F)(F)C1)OC N1(C(C(C)(C)C(F)F)=O)CCCC2(CCC(NC(=O)CSCC(F)(F)F)C2)C1 c1(C(=O)Nc2cc(C)cc(Br)n2)cnn2cc(-c3ccnn3C3COC3)ccc12 c1(OCC)ccc(CC(=O)NCC2CCCN(C(=O)CCC(N)=O)C2)nc1 C1(C(=O)NC2(CCCNC(=O)CCc3cnc[nH]3)CC2)CC12CCCC2 C1(NC(C2(OC)CC2)=O)CCCC(NC(=O)C(CO)N(C)C)C1 c1(C(=O)OC)cnc2c(CNC3CCC(Sc4ccccc4)CC3)c(C)nn2c1 c1(C(C(=O)NC2CCCC2NC(C2(CF)COC2)=O)OC)ccc(F)cc1 C(=O)(C(O)C(F)(F)F)NC(CCC1N(C(c2n(C)cnc2)=O)CCCC1)(C)C c1(C(N2CC(C(C)NC(Cc3c(C(C)C)cccc3)=O)C2)=O)cn2c(n1)CCC2 c1(C(C)=O)c(C)[nH]c(C(=O)NC23CCC2CN(C(c2cnnn2CC)=O)C3)c1C C1(C=O)CC2(C1)C(F)(F)C21CCC1.c1(NC(=O)C)cc(Br)ccc1F.C1CC1 C1(NC(C2N(C)CC(O)CC2)=O)CC12CCN(C(=O)CN1CCC(C)(C)C1)CC2 C1(C(C)NC(=O)C(F)C2CCCC2)CCCN(C(=O)C(N)=O)C1 CC(CC(=O)N(CC(O)CNC(=O)CC)C)C(F)(F)F.c1(C=O)cnccn1.N C1(C(CNC(c2cc(C(C)=O)on2)=O)C)CCN(C(=O)CS)CC1.c1ncc[nH]1 Cc1nc(S(=O)(=O)NCC(=O)N)cn1C.C1(C=O)CC2(CCC2)C1.C(C)CC N1(C(C2N(C)CC(F)C2)=O)CC2CCC(NC(=O)CC3CCCCCC3)(C2)C1 N1(C(CC(C)OC)=O)CC2(CCOCC2)CC1C.C1(C=O)CC2C(C1)C2(C)C.N c1(CC)noc(C(N2CCCC(CCCCNC(=O)CCCCSC)C2)=O)c1C C1(C(N2CCC(C(C)NC(C(COC)O)=O)CC2)=O)CCC2CCCCC2C1 N(C(=NCCCc1nnc2n1CCCCC2)N1CCC(N2CC=CC2)C1)CCF CC1(Cc2cn(CC3CCCN(CN4CCCC4)C3)nn2)NC(=O)NC1=O N1(C(CCc2ccn(C)n2)=O)CC2CCN(C(C3CC3C(N)=O)=O)CC12 C(C(CC(C)C)C(=O)N1CCC=CC1C(=O)NCC1CN(CC)C(=O)O1)OC CC(O)CCCCCC(=O)N(C1CCC(NC(c2cn(C)c(=O)cn2)=O)CC1)C C1(CC(=O)NCc2ccc[nH]2)CC2(C1)CN(Cc1cc(F)ccc1Br)C2 Cc1nc(C(=O)NC2(C)CCN(C(=O)C=CCN(C)C)C2)[nH]c1C C1(NC(c2cnn(C)c2Br)=O)CC2CCC1N2C(=O)Cc1ccsc1 Cc1ccc(O)cc1CNC(C1C=CC(NC(=O)C(C)(C)C(C)O)C1)=O c1(C(N2CC(CNC(c3c(Cl)cccc3Br)=O)OCC2)=O)ccc(Cl)nc1Cl c1(OC)cc(C)c(C(=O)NC2CN(C(c3ccsc3C)=O)CCC2CO)c(F)c1 CN1CCCC(C(=O)NCc2ccc(CN(C(=O)CS(N)(=O)=O)C)cc2)C1 c1(C=O)ccc2c(c1)COCO2.C(C(=O)N)(C(C)C)NC(COC)=O.C1CC1 N1(C(COCCOCC#C)=O)CCCC2(CCC2)C1.C1(CC=O)CCCC1.N CCCC(C(=O)NC1CCCC1CN(C)C(C1(O)CC1)=O)NC(N)=O C(=O)(C(F)(CNC(C1CC2CC2C1)=O)C(C)C)NCC(C#C)C(C)C c1(C2(C(=O)NC(CC)CN(C)C(c3cc[nH]n3)=O)CC2)ccccc1Cl O=C(C1=CCCOC1)NC1CCC(NC(C2(F)C3CCCCC23)=O)CC1 Cn1ncc([N+](=O)[O-])c1C(N1CCOC(C)(CNC(=O)C=CCO)C1)=O N1(C(C2C(NC(c3c(C)nn[nH]3)=O)CCO2)=O)CCCC(C)(C)C1 C1(N(C(c2n(CC)nnc2)=O)C)CCCC(NC(c2cnc(=N)[nH]c2)=O)C1 C=C(Cl)C(C)(C)C(=O)NC1CCN(C(=O)CCc2ccccc2O)C1C Cc1cc2[nH]c(=O)c(C(=O)NC3CCC(C)N(C(=O)C4=CC(C)(C)C4)C3)cn2n1 C1(C)(C(N2CCCC(COC)(NC(c3ccc(C)s3)=O)C2)=O)CCCCNC1=O C(C)(C(C(=O)NCC1CC12CC2(F)F)NC(C1CN2CCC1C2)=O)OC c1(C(=O)NC(C(C)NC(c2cc(C)ncc2)=O)C)cnc2[nH]c(=N)sc2c1 C1(OC)CCC2(C(=O)NCC3CN(C(=O)CS)CC3C)CCC12.c1ncc[nH]1 C1(C)(CC)C=C(C(=O)N2CC(O)(C(F)C(=O)NCCCCCC(=O)NC)C2)C1 CC1(C)CCC(CC(N2CCN(CC3=NOCC3)CC2)=O)NC1 c1(C(=O)NC(C)CCN(C)C(C2(F)CCC2)=O)cc2ccc(Cl)c(F)c2o1 C=C(C)CCCC(=O)N1CC(NC(=O)CCC2C(=O)NN=C2C)C2(CC2)C1 N1(C(C(C)SC)=O)CCN(C(=O)CCc2cnccn2)C2CCC12 c1(C(=O)NCC(CNC(c2ncc(F)cn2)=O)F)ccc2cccnc2c1O N1(C(COC(CC)(C)C)=O)CC(OC)CC1(C)C(N1CCC(OC)CC1)=O N1(C(C(C(C)C)n2cncn2)=O)CC2CC(C1)CN(C(C1CCCC13CC3)=O)C2 c1(C(=O)OC(CC(C)C)C(=O)NC(N)=O)ccc([Si](C)(C)C)s1.CC(C)C.S CC1c2ccc(Cl)c(F)c2CCN1C(C1C2CCC12c1ccccc1)=O C12(C(=O)N)CCCCC1C2(F)F.C1(CC=C)(C(=O)N(CCC)CC)CCOCC1 N1(C(c2nccc(C)n2)=O)CCOCC(C)(CNC(c2cccc(CO)n2)=O)C1 C=CC1(C(N2CCCC2CNC(c2cnn(C(C)C)c2)=O)=O)CCOCC1 N1(C(C2(N(C)C)CCC2)=O)CCC(C)(CC(=O)NCC2CCSC2)C1 CCC(C)C(C(=O)N(C)CC1CCN(C(C2(SC)CC2)=O)C1)NC(=O)OC n1(CC(=O)NCCC2(C)CC2)cc(F)ccc1=O.C12(C(=O)N)CCCC1C2 N1(C(c2c(C)c(=O)cc[nH]2)=O)CC(C)(C(=O)N)CC1(C)C.C(C(F)(F)F)C1CC1 C(CC(CC)C(=O)N1CCN(C)C(CNC(=O)C(F)=CCC)C1)=CC c1(OC)cccc(C(=O)N(CCCNC(C2CCC3CC2CO3)=O)C)c1[N+](=O)[O-] C1(C(=O)Nc2ncc(OC)nc2)C2CCCC1CN(Cc1c(C)nn(C)c1C)C2 N#Cc1ccc(CNC(=O)C(N)Cc2cc(Br)ccn2)cn1 Cc1nn(C)c2c(NCC(C)(C)C(C)(C)C)nc(=NCCc3sccc3Br)[nH]c12 c1(C(=O)NC2CC(NC(c3c(SCC)cccc3)=O)C2)cccc2nonc12 C(=O)(N=S(C)(=O)c1ccccc1)c1cc(C)c([N+](=O)[O-])cc1 N1(C(C(=O)NC(C)C)=O)CC2CCN(C(c3ccnc(C(F)F)c3)=O)C2C1 Cc1cc(C)sc1C(=O)NC1CCOC(CNC(=O)CCSC(F)(F)F)C1 c1(C(=O)N)cc(C)c(C)cc1N.c1(OC)ccc(F)cc1C(=O)NC(C)CCO C(c1cccnc1C)=CC(N1CC(NC(c2c(SC)cccc2)=O)C2C1C2)=O Cc1ccn2cc(C(N3CCCC4C(NC(c5cn(C)nn5)=O)C34)=O)nc2c1 N1(C(C(CC#C)O)=O)CC2CCCC(NC(=O)C(C)(C)COC)C2C1 C(=O)(C(C(CC)C(C)C)N1CCC(C(F)(F)F)C(F)(F)C1)NCCC CCCCCC(C)(C)C(=O)NCC1CC1NC(=O)C(=CC1CCCCC1)F C1(C(=O)NC2CCC(NC(C3(C4CCCO4)CC3)=O)CC2)CCC2CC2CC1 CCCC(C(=O)N(C1CCCN(C(c2cccc(N(C)C)n2)=O)C1)C)NC(N)=O N(C1CCCc2ccccc21)(CC(=O)Nc1ccc(S(=O)(=O)N(O)CO)cc1)C1CC1 N1(C(c2cc(C)on2)=O)CC2CN(C(=O)Cc3cccc(O)c3)CC(C1)O2 C(c1cc2ccccc2o1)=CC(N1CCCC(CC(=O)Nc2cccnc2Cl)C1)=O Cc1cccc(CN2CCC(CNC(C3CCOCC3)=O)C2)n1 C1(NC(C2C(C)CC2)=O)COC2(CCN(C(=O)CN3CCS(=O)CC3)CC2)C1 c1(C(=O)OC)cccc(C(=O)NCC(CNC(C2CCC2(F)F)=O)CO)c1O C(CC(C(=O)N1CCC(c2ccco2)C1)NC(=O)CC1CCOC1C)SC c1(CCCC)ccc(C(C)C(=O)NCCOCC)cc1.C1(C(=O)N)CCCCC1 c1(-c2nc(-c3c(C)cco3)nn2C2CCOC2)cnn2cnnc2c1 Cn1cc(C(N2CCCC(CC(=O)NC3CNC(=O)OC3)CC2)=O)ccc1=O c1(C(=O)NC2CN(C(c3c(C)nc(CO)s3)=O)C(C)C2)ccn2cncc2c1 N1(C(COC(CC)C)=O)CCN(C(c2cc(N)ccc2F)=O)CC1COC c1(C(N2C(C)CC(NC(CN(C)CC)=O)C2)=O)ccc(N)c([N+](=O)[O-])c1 Cc1oc(C)c(C(N2CC3CC3(NC(=O)C(c3cncnc3)C)C2)=O)c1Br N1(C(C2C(C(C)C)C2)=O)CC(NC(=O)CC(C2CCC2)C2CCC2)CC(O)C1 Cc1nc(C(=O)NC2CCC(C)(C)C2)n2c1CCC2 c1(NCC(C)OC)cc(=NCc2csc(C(F)(F)F)n2)[nH]c(C(C)C)n1 Cc1ccc(OC(C)C=O)c(C)c1.C(C)C(C)(C)C.C1(C=O)CNC(=O)N1.N c1(N(C)C)cccc(C(C(=O)NCc2cnn(CC3CC3)c2)N(C)C)c1 C1(C#N)(C(N(C)CC2N(C(CC(C)SC)=O)CCC2)=O)CC(C)C1 Cc1cc(C(=O)NCCC2CCN(C(=O)COc3ccsn3)C2)cc(C)c1 Cc1cnc(C(=O)NCC2CC(O)CN2C(c2ccc(C(F)(F)F)[nH]2)=O)cn1 C(C1c2ccsc2CCN1C(=O)CCN1CCOCC1)NC(C1OCCCO1)=O c1(C(N2C(C)CCC(CNC(c3c(C)snc3)=O)C2)=O)ccc2c(C)noc2c1 C1(CCNC(c2c(C)[nH]cc2)=O)CCCN(C(C2CC(=O)N(C)C2)=O)C1 C12(CNC(=O)C3=CCOC3)CCC(CC1)N2C(=O)C(c1ccccc1Br)(F)F C=CCC(C)(CNC(=O)C(O)CCCNC(=O)CCn1cnnn1)CO C1(NC(C(CSC)OC)=O)CN(C(c2nn[nH]c2Cl)=O)Cc2nccn2C1 c1(CC)ccc(C(=O)NCC2(C(N)=O)CN(C(C3CCNC3=O)=O)C2)s1 C12(NC(C3N(C(c4cncc(C)n4)=O)C4C(C3)C4)=O)CC3CC(CC1C3)C2 Cc1cc(C)c(CNC(c2conc2C)=O)cn1.C1(C=O)CCCC2(CC2)C1 c1(C(CC2N(C(C(=C)Cc3ccccc3)=O)CCC2)=O)sc(C)nc1C c1(C(N2C(C(N3CC(NC(C)=O)C(O)C3)=O)CCC2)=O)cc(F)cc(F)c1 CC(C(=O)N1CCCC(CCNC(=O)C(C)(F)F)C1)S(N)(=O)=O N1(C(c2ccon2)=O)CC2CN(C(c3ccccc3Br)=O)CCC2(CO)C1 C(C(=O)N(C(C)CN(C(=O)CN(C)C(C)=O)C)C)=CCC N1(C(COCCCC)=O)CCN(C(C2CCCCC23CC3)=O)C(C2CC2)C1 C(=O)(C(C)P(C)(C)=O)N(Cc1c(OC)cccc1)Cc1csc(Br)c1 CCC(C)C(C(=O)N1CCCC1C1CCOCC1)c1ccccc1 c1(OC)cc(CC(N2CC3CC(NC(C4CCCNC4=O)=O)C2C3)=O)ccc1O C(=O)(CCCCc1ccc(C)cc1)N(CCCCN(C(CCOC(C)=O)=O)C)C Cc1cc(C2CC2)ncc1C(=O)NC12CCN(C(=O)CCS(C)(=O)=O)CC1C2 C1(NC(CCOCc2n(C)ccn2)=O)COCCN(C(=O)CCC2CC2)C1 CCC1=NOC(C(=O)NCC2CC(O)CN2C(C23CC2CNC3=O)=O)C1 c1(CN(C(c2ccc(SC)s2)C(=O)NCC=C)C)cccc(C(=O)OC)c1 c1(N2CC(NC(CCC=C(C)C)=O)C(C)(C)C2)ncnc2c(F)c(F)ccc12 C1(NC(=O)NCCCNC(CC(C)C)=O)CCN(S(=O)(=O)N(C)C)CC1 c1(C(N2CCCC(NC(c3cc(C)ncn3)=O)(CO)C2)=O)c(C)nc(O)nc1S C(c1ccccc1F)=CC(=O)NCCN(CC(C)O)C(C1CCOC1(C)C)=O Cc1cn(C)nc1C(N1CC2CC2(CNC(=O)COc2ccccc2)C1)=O O=C(C1COc2ccc(Cl)cc21)NCC1CCCC1NC(C1CC(F)C1)=O CC(C)C#CC(=O)NCCCN(C1CCCC1)C(=O)Cc1ccccc1Cl c1(C(CN(C(CNC(C)=O)C(F)(F)F)C)=O)cc(C)n(C2CCCOC2)c1C CC1CC(NC(=O)CP(C)(C)=O)CN(C(=O)CC2CCCN(C)C2)C1 C12(C(N3C(CN(C(=O)Cn4cnnn4)C)COCC3)=O)CC3CC1C2C3O C1(C(N(C(c2csc(N(C)C)n2)C(=O)N)CC(C)C)C)CCOCC1.CC(F)F CCCC(CNC(C1CN2CCC1C2)=O)C(=O)NCc1ccc(Cl)nc1 C1(CNC(c2csc3cncn23)=O)CN(C(C2CCCOCC2)=O)CCC1(F)F c1(OC)ccc(CNC(C2CC3CC3N2C(=O)CCc2ncccc2C)=O)cc1 N1(C(c2cn(C)nc2)=O)CC(NC(C2(C)CCCNC2=O)=O)CC(O)C1 CC1(C(=O)NCC2(F)CC(NC(=O)C3=CCCOC3)C2)COc2ccccc2O1 Cc1cnc(C(=O)NCc2nc(C(N3CCC(C)C(CO)C3)=O)co2)c(F)c1 C(=O)(Nn1cnc2ccccc12)c1c(CNC(C(C)NC(=O)OC)=O)cco1 c1(CC(=O)NCC2N(C(C3=C(C)CCC3)=O)CC3(CC3)C2)cn2ccccc2n1 Cc1cc(NC(C)CN(C)C)nc(N2CCC(C(c3ccccc3)C#N)CC2)n1 C1(C=O)OCCN(C)C1=O.N1(C(C(CC)NC(C)=O)=O)CCC(CCOC)C1.N N1(C(c2ncoc2C2CCCO2)=O)CCCC(C2CC2NC(C2(O)COC2)=O)C1 CN1CCC(C)(CNC(=O)NCc2ccccc2)C1.C(C)(C)C.C=O.N C1(CC)CN(C(=O)C)CCN1C(=O)C(C)N1CC(C)C1.c1(C=O)ccccc1.N C1(C(N2CC(C(N)=O)(CNC(C(C)=C3CCCC3)=O)C2)=O)CCCC(O)C1 Cc1ccc2ncc(C(N3CCCCCC(NC(=O)C(O)C(F)F)C3)=O)cc2c1 N1(C(c2c(CC)nc(C)o2)=O)CCCCC(C(=O)NC2COCC2N=[N+]=[N-])C1 N=c1[nH]nc(C(N2CC(CNC(=O)CCN3CCCC3)C2)=O)[nH]1 c1(OC)cc(C(=O)NCC2CCCC2)cc(Cl)c1O.C(=O)(CC)N.C(N)=O c1(C(=O)NCCC2N(C(C3OCCN(C)C3)=O)CCC2)ccc2nnn(C)c2n1 C1(CC(=O)NC(CC)C(C)O)CCCN(c2cc(-c3ccccc3)ncn2)C1 C12(CNC(CSCCC)=O)CN(C(C3CCC3)=O)CC1CS(=O)(=O)C2.C Cc1[nH]nc2cc(C(=O)NCC(C)NC(C3CCC4(CCC4)CC3)=O)ccc12 CC(CCCCNC(=O)CCOCc1ccccc1)NC(C1CC1(F)F)=O c1(CC(=O)NCCCNC(c2cc(OC)no2)=O)c(F)cccc1F C1(NC(CCC2(NC(C(C3CC3)SC)=O)CCCC2)=O)(CO)CC2CCCC12 O=C(C1=Cc2ccccc2OC1)N1CCC2CCN(C(C3CCCC3)=O)CC2C1 C1(C(=O)Nc2cccc(SC)c2)CC1C1CN(C(=O)Cc2ccns2)C1 Cc1cccc(F)c1CC(N1CCC(CCC(N2CCCCCC2)=O)C1)=O C(=O)(C(O)CC(C)C)NC(CC=CC)C(=O)N1CCOC(CO)C1 CC1(C)CN(C(c2ccsc2C#N)=O)CCC1NC(c1ncc2ccccn12)=O C1(C)(C(=O)NCc2nc(C(=O)Nc3cc(C)sc3)c(C)o2)CCC2CC2C1 C(=O)(C(C)CC(F)F)NCC1N(C(c2cccc(OC(C)C)c2)=O)CC1 NS(=O)(=O)c1cc(C(=O)NCCC(O)CNC(c2cnns2)=O)cc(F)c1 CCS(=O)CC(=O)N(CC(=O)NCc1nc(C(C)C)n[nH]1)C N1(C(CN(C2CCC2)C)=O)CCCC(CC(N2C3COCC2C3)=O)C1 C1(C2CCN(C(=O)CN3CCCS3(=O)=O)C2)CC1.c1(C=O)coc(C2CC2)n1 CC(CF)CC(=O)N(C)CC1CCCCN1C(C1CC(C)(C)C1)=O N1(C(C(C=CCCC)O)=O)CC2(CC(NC(c3cn(C)nc3OC)=O)CO2)C1 c1(CC(=O)NCC2(NC(CC(CC)OC)=O)CCCCC2)cc(C)ccc1O c1(C(N(C(C)C)CC)=O)ccc2ocnc2c1.c1(CC=O)cc(C2CC2)no1.N C1(NC(CC=CCC)=O)CCC2(CCCN(C(=O)C(C3CCC3)C3CCC3)C2)C1 N1(C(C)=O)CCC(CC(=O)NC2CCCC(NC(=O)CC3(C)CC3)C2)CC1 CCC(C(=O)NCC(CC)(CC)NC(c1cc(C(C)(C)C)oc1C)=O)C(C)O C1(CNC(C(C)=C2CCCC2)=O)CC2CCC(C1)N2C(c1ccncc1F)=O N1(C(CCC(C)(F)F)=O)CCC2(CCCCC2NC(=O)C2=C(Cl)CCC2)C1 C1(CC)CCCC(c2nnnn2C)(NCCC(=O)N(CC)Cc2ccccc2)C1 CCS(=O)(=O)CC(=O)NCC(C)CC(=O)NCc1cnc(C)cc1C C1(C(=O)NC(CCN(CC)CC)C)COC(CNC(c2ccsc2)=O)C1 C12(COC)CC(CN1C(C1CC(N(C)C)C1)=O)C2.c1(CC=O)cnc[nH]1 C1(NCc2n(C(C)(C)C)ncn2)CC2CC1C(O)C2O C1(C(N2CCC(CNC(C(C)OCCCC)=O)C2)=O)Oc2ccccc2OC1C C(=O)(CC(O)CC)NCC1CC(OC)C1.C(=O)(C)N.C(=O)CN(C)C C1(CCNC(C(C)CN(C(=O)C(C)(C)F)C)=O)CC2C=CC1C2 c1(C(=O)NC2CC(NC(CC(CCC)O)=O)C2)cc(C)nc(Cl)c1N Cc1nnc2n1CC(C(=O)NCCNC(c1sc3ccccc3c1Cl)=O)N(C)C2 N1(C(C2CC(OC)(OC)C2)=O)CCC(C2CC2)CC1.C(=O)CS(=O)(=O)C1CC1 c1(CNc2c(C)c(N(C)Cc3cncnc3)ncn2)ccnc2ccccc12 c1(C(N2C(CNC(c3c(C)nc(CCC)s3)=O)CC2)=O)cc(Cl)cc(F)c1F C1(C(=O)NC2CC3CN(C(CC=C=C)=O)C(C2)C3)Cc2cccc(F)c2O1 c1(OC)cnnc(C(N2CC(C(C)NC(=O)C(c3cnn(C)c3)C)C2)=O)c1 c1(OCC=C)cc(OC)ccc1C=O.C(C)CC.C1(CCC=O)CC1.N CCCCCCCC(=O)NC(C(=O)N1CCC(CCCO)C1)C(C)C C1(CC)CCCN1C(=O)C(=O)N(CCNC(=O)Cc1cccn1C)CC n1(CCC(N2C(CNC(C3CC34CCOCC4)=O)CC2)=O)ccc2cccnc12 N1(CC)CCCCC1C(N1CCC(CC(=O)N(CCCN2CCCC2)C)CC1)=O CC(C)C(F)C(=O)NCc1ccc(C(=O)N(C(CO)C2CC2)C)cc1 C1(C)(C(N2CC(C(C)NC(C3CCCN3C)=O)C2)=O)CNC(=O)C1 O=C(CC1=CCCC1)NCCNC(C1CCC12CCCO2)=O S(=O)(=O)(c1ccc(N2CCC(C3CCCC3)C2)c(F)c1)N(CC(C)CO)C N1(C(CN(C(C)C)C)=O)CCCC(C(=O)NCC2CC23CC3)CC1 N1(C(CCc2onc(CC)n2)=O)CC(n2cc(-c3cccs3)nn2)CCC1(C)C c1(CNC(c2ccc(OC)c(F)c2)C)ccc2cn(C)nc2c1 N1(C(C(C)S(N)(=O)=O)=O)CCC2(CCCCC2NC(=O)COC(F)F)C1 c1(C(N(C(C)CNC(c2cn(C)cn2)=O)C)=O)cc(C(F)(F)F)cs1 N1(C(C(COC)(C)C)=O)Cc2ccccc2C(NC(=O)Cc2c(C)n[nH]c2C)C1 c1(CC(N2C3CC(CN(C(C4CC4C4CC4)=O)C3)C2)=O)ccc2ccccc2c1 Cc1ccc(C=CC(=O)NC23CCCN(C(=O)C4=NNC(=O)CC4)C2C3)cc1Cl C=C1CC2CC1CC2(c1nnnn1C(C)C(=O)OC)NC1CCC(C2CC2)CC1 CCCC(C(=O)NCC=CCNC(=O)C(C(C)C)n1ccc(C)c1)OC c1(C=O)ccc(C2CC2)cn1.c1(C(N(CC(O)C)C)=O)cnc(N(C)C)cn1.N C1(CNC(C(c2cccnc2)NC(CC=C)=O)=O)CCCCNC1=O CCC(C)C(=O)N(CC(CC)NC(=O)Cc1n[nH]cc1Br)CC c1(C(=O)NCC2CC(C)N(C(=O)CSC(F)(F)F)C2)cc(Cl)cnc1O c1(C(=O)NC(CCCNC(c2scc(C)c2C)=O)C)cc(C)c2ncccc2c1 Cc1ccc(NCC2CCCC2NC(=O)Cc2cnccc2C)c([N+](=O)[O-])c1 C=C(C)CC(C)C(=O)N1CC(F)(F)CC1CCNC(=O)C.c1n[nH]c(O)n1.S Cc1cc(C(=O)N)n(C(F)F)n1.C1CCN1C(C1(C(C)(F)F)CCC1)=O.C C1CCN=C(NC2CCCSC2)NC1.c1(OCC)ccc(-c2ncccn2)cc1 C1(NC(c2cc3[nH]ccc3s2)=O)CCCCN(C(=O)CC2CCCCC2(F)F)C1 C1(NC(C(C)OCC(F)(F)F)=O)CC(F)(C)C1.N1(CC(=O)N)CCC1C N1(CC)CCCC(C(=O)NCC(CC(=O)NCc2scnc2C)OC)C1 C1(C(=O)NCC(C)CN(C)C(c2cc(-c3cnn(C)c3)[nH]n2)=O)COCCO1 C1(NC(C2CCS2(=O)=O)=O)CCC2(CC1)CN(C(=O)CCc1ccc[nH]1)CCO2 c1(C(N2CCC(NC(C3(CO)CCCO3)=O)CC2)=O)cc(Cl)sc1Cl C1(C(NNC(C2Cn3c(nc(C)n3)CC2)=O)=O)CC(=O)C12CCCCC2 C(C#Cc1cccc(Cl)c1)Nc1c(C)ccc(Cl)c1 O=C(CCS(=O)(=O)Cc1nc(-c2cccc(Br)c2)no1)NCC(F)(F)F N1(C(C=CC)=O)CC(NC(C2CC2c2ccc(F)cc2F)=O)CCC1C Cn1ncc2ncnc(Nc3ccc(-c4ccc5c(c4)CC(=O)N5)s3)c12 C12CCC(CC1)N2C(c1c[nH]c(C(N)=O)c1)=O.c1(C(C)C)nocc1C(=O)N C1(CC)CN(C(c2cc(C)cc(O)n2)=O)CCN1C(=O)CC1CCCC1 C1(Br)(C(=O)NC(CC)CNC(c2cnn(C(C)C)c2)=O)CC12CCC2 C1(NC(CS(CC)(=O)=O)=O)CCC2(CCCN(C(=O)CSC(C)C)C2)C1 C#CCCCC(C)C(=O)NC(C1CCN(C(C2CCCCN2CC)=O)CC1)(C)C C(=O)(C(C)(O)C1CCC1)NCC(CC)NC(=O)CCN(c1ccccc1)C Cn1ncc([N+](=O)[O-])c1C(=O)NC(CNC(C1CCCCC1O)=O)CO c1(N2CC(CC(=O)OC)OC(C)C2)nc(C(C)(C)C)nc(C)c1C CCC(CC(=O)NCC1CCCC(CNC(=O)C#CC2(CC)COC2)C1)C(C)C c1(C=O)coc2cc(C)ccc12.C1(NC(CCSCCC)=O)CCC(C)(C)C1.N CCC(C)C(C)N=c1nc(N(C)CCOCCN(C)C)c2[nH]ccc2[nH]1 C1(NC(C(SC)SC)=O)CCC(C)(NC(c2ocnc2C2CC2)=O)CC1 c1(CC)cccc(C(=O)NCCC)c1.C(=O)(CC)N.CCN(C)C.C1CC1 c1(C(=O)NCC(CN(C(c2cc(C)ns2)=O)C)O)ccc2nc(S)oc2c1 C(=O)(C(C(C)C)n1cc(CCCOCCO)nn1)Nc1ncc(C)s1 c1(-c2nc(C(C3CC3)OC)nn2C2CCC(C)(C)C2)cc(C)cc2cccnc12 C#CCCCC(C)C(=O)NCC1CCC2(CN(C(c3ccc(CC)o3)=O)C2)O1 N1(C(c2c(CCC)[nH]cc2)=O)CC(C2(NC(=O)CCCC(C)=O)CC2)C1 Cn1cnc(CC(O)C(=O)NC(C)(C)CCNC(=O)CN2CCNC2=O)c1 C#CCCCCCC(=O)NCC1COCC1NC(=O)C(C)NC(=O)C(C)(C)C Cc1cc(Br)ccc1CC(=O)NC1CN(C(=O)C(F)CC2CC2)CC1O c1(CNc2c(N)n(-c3cc(F)c(Br)cc3O)nc2)ccc2c(c1)CCOC2 S(=O)(=O)(c1cccc(=NCC(C)c2c(Cl)cccc2Cl)[nH]1)N(CC(C)C#N)C c1(CN2C(C(N3CCOC(C(F)(F)F)C3)=O)CC3CC32)cc(F)cc(Cl)c1O c1(C(=O)NCC(C)NC(=O)CSC)ccc2c(O)n[nH]c2c1.C1CCCCO1 C1(NC(=O)CC2CCC(C3CC3)O2)CCCN(C(c2cnoc2C2CC2)=O)CC1 C=CCC(C)(O)C(=O)NCc1cccc(NC(=O)C(C)C(C)(C)C)c1 C1(CSCC)CCNCCC1(F)F.C12(CCS(=O)(=O)C1)CC(=O)N2 N1(C(C(C(COC)C)C)=O)CCCC2(CCN(Cc3ccc(C)c(C)c3)C2)C1 C1(C(=O)NC2CCC(NC(c3c(OC)n(C)nc3)=O)C2)CCCCC1(F)F C1(CC)CCC(CNC(C2COCCN2C(c2c[nH][nH]c2=N)=O)=O)CC1 C(N=c1[nH]c2c(c(=NC(C)CCC(C)(C)C)[nH]1)COC2)c1c(C(C)(C)C)[nH]nn1 c1(-c2cn(CCCC(=O)N(C)Cc3csc(C4(C)CC4)n3)nn2)ccc(N)cn1 C1(COC)(C)CCN(C(c2cnc(S)n2C)=O)CC1.c1(C(=O)N)ccc(C)[nH]1 C1(C(=O)NCCCC(=O)NC)CC(NC(=O)C=Cc2nccs2)CCO1 C1(NC(C(F)=CCC)=O)CN(C(=O)Cn2ncc(Br)n2)CC(C)(C)C1 C(C(=O)N1CCCC1C=CC(=O)N(C)Cc1ncco1)(C(C)C)OC C(C1=NOC2CN(C(c3ccc(Cl)c(F)c3)=O)CC12)NC(C=COCC)=O c1(C(=O)NC(CNC(CCC=C=C)=O)(C)C(C)C)ccc2c(c1)nc(CO)n2C C1(NC(CCC(=O)OC)=O)CN(C(=O)C(C)N)CC2(CCC2)C1.[SH](C)(=O)=O N1(C(Cc2cc(C)nn2C)=O)CCCC(C)(NC(C2C(C)CC2C)=O)C1 c1(-n2cc(C(C)NC(C3CCC3C(F)F)=O)nn2)ccccc1CO c1(CN(C)C(c2ncoc2CNC(=O)CCCF)=O)nnnn1C C1(CC(=O)NC2C(NC(c3n(CC)cc(Br)c3)=O)C2)CC(C=O)=NO1 C(=O)(C1=C(Cl)CCOC1)NCC1C(NC(c2cc(C(C)(C)C)on2)=O)CC1 c1(CC)cc(C(=O)NC2COCCN(C(C3(F)CC=CC3)=O)C2)c(C)nn1 n1(CCC(N2C(CNC(C(n3ccc(C)n3)C)=O)C=CC2)=O)cccnc1=O C(CC1=CCCCC1)N(C)C(C1CCCC1CNC(=O)CCCN=[N+]=[N-])=O c1(C(=O)NCc2cc(C(N3C(C)(CC)CC3)=O)on2)c(C)noc1C c1(C(N2CCCC(C(C(=O)N(CCC)CCC)C)C2)=O)c(F)cccc1F C1(CC#C)(C(=O)NC(C2CCN(C(C3(Br)CC3)=O)C2)C)CCCCO1 C1(NC(COCc2ncc(C)o2)=O)CCN(C(=O)Cn2cccnc2=O)C1(C)C Cc1ccc(C(=O)NC2CCN(C(=O)CC3CC4CC4C3)C(C)C2)cc1F C(=O)(C(F)(F)C(C)(C)O)NC1CCCN(C(CN2CC(C)(OC)C2)=O)C1 c1(CN(S(CC)(=O)=O)C2COC2)cn(CC(=O)NC)nn1 c1(C(=O)Nc2cc(C)cc(Cl)c2)ccnc2c1nnn2C c1(OC)ccnc(OC)c1C(=O)NCCC.c1(C(=O)N)nc(C(C)C)ncc1Cl c1(CNCc2cccc(OCC)c2Br)ccc(C#N)cc1OCCOC N1(C(CCOCC)=O)CCC(CNC(=O)Cn2ccc(C)n2)C(C)C1 CCC(C(=O)N1CCN(C(c2cc(Cl)ncc2N)=O)CC1CO)C(C)(F)F N1(C(C(CCC)N(C)C)=O)CCCN(C(c2cc(C3(C)CC3)on2)=O)C(CO)C1 c1(C(N2CCC(CNC(C3CCC(CCC)CC3)=O)C2)=O)ccc(N)c(O)c1 N1(CCC)CCCC(C(=O)N)C1.CCCCC1CN(C(=O)CCN(C)C(C)=O)C1 c1(N2C3C(NC(c4n(C)ncc4)=O)CC(CC3)C2)nc(O)c2cnn(C)c2n1 Cc1oc(Cl)nc1C(N1CC=CC1(C)C(=O)NCC1(C)C=CCCC1)=O Cc1cc(C(N2CC(F)(C(=O)Nc3nc(C)co3)C2)=O)nc(C)c1 c1(C(N2C(c3cn(CC=C)nn3)CC2)=O)cnc2n1CCC2 C1(C(C)C)C(NC(c2sccc2F)=O)CCN1C(=O)CC1CCCN1C C(CCCCCC(=O)NC1CC(CC)(CC)C1)NC(C(C(CC)C)O)=O C1(C=O)CCC2(CCC2)C1.C1(C(N2CC(OC)(C)C2)=O)CCC(F)(F)CC1.N Cc1ccc(C(=O)Nc2cccc(NC(c3ccn(C(F)(F)F)c3)=O)c2)cc1 c1(NC(C(CC2CC2)NC(=O)OCC)=O)cccc(C(=O)OC)c1 Cc1nccc(C(=O)NCC2(C(=O)NCC3CCCOCC3)CCCO2)c1C c1(OC)ccc(CCCNC(C2CCC(=O)N2C(C)C)=O)cn1 C=C=C(C)CC(=O)NC(CN(C)C)C(=O)NCC(=O)N(C)O c1(C(=O)NC(CCNC(C(CCC)OC)=O)C(C)C)ccc(OCC)c(F)c1F c1(C(=O)NC2CCCN(C(c3cc(C)c(F)nc3)=O)CC2)ccc2nccn2c1 c1(CC)cccnc1C(N1CCC(C2CCCN2C(c2ccc(CO)s2)=O)C1)=O c1(NC2CC(CNC(C(CCCC)(C)F)=O)C2)ncnc2c1nnn2CC(=O)OC C1(C(C(=O)NCCN(C(=O)CC2CC(CF)C2)C(C)C)C)CCOCC1 Cc1cccc2[nH]cc(CC(N3CC(C)(NC(=O)CSc4ccccn4)C3)=O)c12 C12(CNC(N3CC4(CN(C(C(C)C)=O)C4)C3)=O)CCCCN1CCC2 c1(C(=O)Nc2c(C)ccnc2C#N)cc(O)c2ccc(C3=COCC3)cc2c1 c1(C=O)cn2c(n1)CCC(C)C2.c1(C(N(CCC)CC)=O)cc(=N)[nH]c(Cl)n1 C1(O)(CNC(CC(C)(C)C)=O)CCCN(C(C2(C)CC2(Cl)Cl)=O)CC1 C1(C(N2CCC(CNC(C3(CCC)CC3)=O)CC2)=O)CCC2(CC1)OCCO2 CC(C)(C)C.c1(C=O)ccon1.C(=O)(CC1(C=O)CC1)OC.N(C)C.N C=CC1OCCCC1C(=O)NC1CC(O)CN(C(C2(c3cc[nH]n3)CCC2)=O)C1 C#CC1CC2(CC2)CN1C(c1cn(C)cn1)C(=O)NCC(F)F C1(NC(c2nn(CC)nc2C)=O)CCCC(C(=O)N)CC1.C1CC(C)CC(C)C1 Cc1ocnc1C(=O)NCc1n[nH]cc1C(N1CC(C)(N(C)C)C1)=O c1(CC(N2C(C(=O)NC(CC)C)CC(C)C2)=O)ccc(Br)cc1OC C1(C(=O)NCCC2CCC(C)(C)O2)CCCCCC1NC(=O)CSC1CC1 C1(C(N2CC(N(C)C)C2)=O)CCN(C(=O)CC2CCN(C)C2=O)C12CCC2 c12occc1CNC2=O.C(=O)(C(C)CO)N1CC(OC(CC)=O)C1 c1(C(N2CC(O)CC2c2ccccc2)=O)cnn2ccsc12 C(N=c1ccc2ncc[nH]c-2n1)C1(CCNC(=O)CC2CCCS(=O)(=O)C2)CC1 C1(C(C)NC(C2(O)CC2)=O)CCCN1C(=O)CCc1ccncc1 CCCC(C(O)C(=O)NCC1=C(C)CCOC1)NC(c1conc1CC)=O C1(CNC(=O)NC(CC)Cc2ccc(Br)cc2)CCCC(F)(F)CC1 c1(CCC)cc(C(=O)N(C2CCCN(C(C3(C)CC(F)(F)C3)=O)C2)C)n(C)n1 C(=O)(C1=C(Cl)CCC(C)C1)NC1CC(NC(CCN2CCN(C(C)C)CC2)=O)C1 N1(C(CC2C(CC)C2)=O)CCCC(CCNC(c2ccn(CC)n2)=O)C1 N1(C(=O)Cc2coc(C(F)F)n2)CCC(NC(C2(O)CCCCCC2)=O)C(F)C1 CC1CN(C(c2cc[nH]c(=N)c2)=O)CCN1C(=O)CN(c1cnccn1)C N1(C(COCCOC)=O)CCCC(C2CCN(C(=O)CC(C)P(C)(C)=O)CC2)C1 C1(C(C)NC(C2(N3CCCC3)CC2)=O)CCCN1C(=O)C=CC1CCOC1 c1(C(N2C(CCNC(C3C(C(N)=O)C3)=O)CCC2)=O)cc([N+](=O)[O-])n[nH]1 N1(C(Cc2cn(CC)nc2)=O)CCC2(CCCN(C(=O)CC(F)(F)Cl)C2)C1 c1(C(N2CC(NC(c3c(SC)cnn3C)=O)C(C)C2)=O)cccc(N)c1O c1(C(=O)NC2(CN=c3nc(C)[nH]s3)CCCCC2C)cccc2c1CCC2 S(=O)(=O)(CCC=O)NC(C)=O.C1CCN(C(=O)C(=O)N(C)C)CC1O.CC.N C(=O)(CC(C)CC(C)(C)C)N.COC=CC(=O)NC(C)(C)C(=O)NCC(C)C C1(NC(c2n[nH]c(C)c2Cl)=O)CCS(=O)(=O)C12CN(C(C1COC(C)C1)=O)C2 c1(OC)ccc(N(C)C)cc1-c1cscc1C(=O)N(c1nccc(OC)n1)C Cc1cc(Br)nc(Cl)c1NC(c1nc(NCc2ncco2)cn1C)=O c1(C(=O)NCC(C)N(C(C2CCN(C(C)=O)CC2)=O)C)cccc2c1nnn2C N1(Cc2cccc(C)c2)CCC(C(=O)Nc2ccc(CC#N)cc2)C(O)C1 c1(C(=O)NC(CNC(C(CC)OC)=O)(C)C(C)C)cc(OC)c2ccccc2n1 C(=O)(CCCC(=O)NCCOCCN(C)C(c1cc([N+](=O)[O-])c[nH]1)=O)NC Cc1cc(C)c(C(N2CCC(OCC(=O)N(C3CCOC3)C)C2)=O)cn1 N1(C(c2n(C)ccn2)=O)CC2(C1)CN(C(=O)CCOCC(F)(F)F)C2 c1(C(N2CC3C(C2)N3c2nccc(Br)n2)=O)ccc(F)c(Br)c1F C1(NC(CC(CC)CN(C)C)=O)C2CC(CN(C(c3cc(Cl)c[nH]3)=O)C2)C1CO N1(C(c2nccs2)=O)CCC(O)C2(CCN(C(c3cnc(O)nc3O)=O)CC2)C1 c1(C(=O)O)ccc(O)c(CN2CCC(CNC(c3ccc(Cl)[nH]3)=O)CC2)c1 C(=O)(C1=Cc2ccccc2OC1)N1CC2C(CNC(=O)CC3CCCO3)C2C1 c1(C(=O)NC2CC(N(C(=O)CCC3CCCC(O)C3)C)C2)cc(O)cc(F)c1F C(CC(C)C)(C(=O)NC1(C)CC1)OC.c1(C2(C=O)CC2)cccc(Cl)n1.N N1(C(C(CNC(C2C(OCC)CC2)=O)(C)CC)=O)CC2(CNC(=O)N2C)C1 C1(C(N2CCC(NC(=O)CCNC(c3ccccc3)=O)C2)=O)CCN2CCC1C2 c1(C(=O)NC(C)(C)CCNC(C2CCCC2O)=O)ccc2ccccc2c1O C(=O)(CS(=O)(=O)C1CC1)N1CC2CC(NC(C3N(C)C(=O)CCC3)=O)C2C1 c1(C(C(=O)N(CC(C)N(C(=O)Cn2cnnc2O)C)C)O)ccc(Cl)cc1 C1(NC(=O)C2=NOCC2)CS(=O)(=O)CC1.c1(C=O)ccc(C(F)(F)F)cn1.N C#Cc1cn(C)nc1C(N1CC(O)(C)C1)=O.C1(C=O)CCCN(C(N)=O)C1.N C1(C(N2CC(CC)OCC2)=O)CCC2CN(C(=O)CC(C)(C)C(=O)OC)CC12 c1(CC)ccc(C(=O)NC2CC3(C2)CCC3)c(C)n1.C1(C=O)CC2CC2C1.C C1(CNC(CN(C)C(C2(C)CSC2)=O)=O)CCC(=O)CC1 Cc1cccc2oc(C(N3CCN(C(=O)CC4CCN(C)C4=O)C(C)C3)=O)cc12 Cc1[nH]c(C(=O)NC2(CO)CCCN(C(=O)C(C)C3CC3)C2)c(C)c1[N+](=O)[O-] c1(C(N(CC(CC)NC(C2C3CC4C(C3=O)C24)=O)C)=O)nc2ccccn2c1F C1(CNCCCc2cccc(OC)c2)CNCC(C)(C)O1.C(C)(C)C.C=O.C C(=O)(C(CC(C)C)OC)N(CCC(=O)NC1C=CC(CO)C1)CC=C c1(C(N2C(C)CC(CNC(c3c(CC)nc(C)[nH]3)=O)C2)=O)cc(C)ccc1O N1(C(c2ccc(CC)cc2)=O)CCC(C)N(C(C2CCC3(CC3)C2)=O)CC1 CNS(=O)(=O)NCC(=O)NC1CC(F)(CNC(=O)CCc2cnc[nH]2)C1 C(CC(O)CNC(=O)C)NC(C(c1ccccc1)C)=O.N1(C(C)=O)CCOCC1.S S(=O)(=O)(c1ccc2c(c1)CCN2C(C12CCCC1CS(=O)(=O)C2)=O)N(C)C Cc1ccc(=O)n(CC(=O)NC(C2CCOC2)CNC(=O)C=CC(C)C)n1 C1(O)(C(=O)OC)CCCC1NC(=O)NCc1cc(CC2CC2)nn1C N1(C(C2(CCC=C)CN(C(=O)C(CC)CC=C)C2)=O)CCCCCCC1C C1(C(=O)NCCC2(CNC(c3c(N)nccn3)=O)CC2)CCCCC12CC2 C1(CNC(CC(CC)OC)=O)(CO)CCCN(C(c2ccc(C)s2)=O)C1 c1(OC)ccc(C(=O)N)cc1C(F)(F)F.C1CCCN1C(C1CNC(=O)N1)=O N1(C(C2(CC)CN(C(C3CCCC(C#N)C3)=O)C2)=O)CCCC2C(O)CC12 c1(OC)cc(C)c(C(N2CCC(C)C2)=O)c(F)c1.C(c1ccco1)=CC=O.C c1(NCC(CN(C(=O)CC2CCC(F)(F)C2)C)O)cc2c(cn1)C(=O)CCC2 C1(NC(C2(C)CC3CC3C2)=O)CC2(C1)CN(C(c1cnn(CC(F)F)c1)=O)C2 C1(C(N(CCN(C(C(C)SC)=O)C)C)=O)CCn2c(C)cnc2C1 N1(C(C2C(C)N(C(c3cc(Cl)n[nH]3)=O)CC2)=O)Cc2cnn(C)c2C1 Cc1ncc(Cl)c(C(N2CCC(NC(c3cc4n(c3)CCC4)=O)C(CO)C2)=O)n1 c1(C(=O)NCC(C)C)ccnc2nccnc12.c1(C(=O)N)ccsc1C(F)(F)F Cc1cnc(C(N2CC(NC(=O)Cc3ccccc3)C(C)C2)=O)cn1 C(=O)(CCCC(F)(F)F)NC(CC(=C)C)C(=O)NCCCC1CCOC1 N1(C(CCCC#C)=O)CC(N=[N+]=[N-])CC1C(=O)NC1CC2C=CC1C2 c1(C(=O)NCC(C(=O)NCC2N(C)CC(O)C2)N(C)C)ccc2[nH]ccc2n1 C1(NC(c2c(CC)nn(C)c2)=O)CC(O)CN(C(c2c(Br)n[nH]c2C)=O)C1 Cc1c(C(N2CCC(CNC(C3(C#N)CC(C)C3)=O)CC2)=O)[nH]c2ccccc12 C1CCC(C)(C)CN1C(=O)C=C(C)C.c1(CSC)ccc(C(=O)N)cc1 C1(C(N2CCCC2)=O)CC12CC(F)(F)C2.C1(C(=O)NC(C)C=O)CCCCC1.N C1(NC(c2c(SC)cccc2)=O)CC2CN(C(C3CCOCC3(C)C)=O)CC2C1 C(=O)(C(C)(C)C(=O)N(C(C)C)C)O.c1(C=O)ccccn1.C(=O)CC.CC C1(N2CCC(CNCc3cc(C)ncn3)CC2)CC2CCC(C1)N2C c1(CNC2CN(CC)C(=O)C2)c(Cl)ccc(Cl)c1F c1(CCC)cnnc(C(N2CCCCC2CCNC(C2CC(C)(C)CO2)=O)=O)c1 c1(C(N2CCC(NC(C3CC(OCC)C3)=O)C2(C)C)=O)cc(Cl)c(F)cc1C C(CCCC(=O)NCC1(CNC(=O)CCC2CC2C)CC1)OC C1(NC(C(CC(=C)Br)(C)C)=O)CC2CCC1CN(C(=O)C=CC)C2 N1(C(c2ccnc(OC(C)C)c2F)=O)CC(NC(=O)C)CC(F)(F)C1.C(C)C c1(C(N2CC(=O)NCC2)C(=O)NC2CCOC2)cn2cc(Br)ccc2n1 CCC(CC)C(C(=O)NC(C(=O)NCCCCC(F)(F)F)C1CCC1)OC C1(CC)CC(F)(F)CN1C(=O)CCC(C)C.C1(C(=O)N)(COC)C=CCC1 N1(c2c(C(=O)NC)cccn2)CCC(C(=O)Nc2ccc(C#N)cc2)C(O)C1 Cc1c[nH]cc(C(=O)NC2CC3C2CCN3C(=O)Cc2c(F)cccc2Cl)c1=O c1(C(N(CCCN(C(c2cc(OCC)n[nH]2)=O)C)C)=O)c(C(C)C)n[nH]c1C C(=O)(CC1=CCCC1)N1C(C)CC(CNC(C2(C)CCC2)=O)C1 c1(C(=O)NC2CN(C(C(COCC)C)=O)C(C)(C)C2)cc(F)c(C)cc1N CN1CCCCC1CCC(=O)NCC1(F)CN(C(=O)CCc2ccc(O)cc2)C1 C1(CC)COC(C)(C)CN1C(C1CCC(C)(C)N(C(=O)C(C)c2cc[nH]n2)C1)=O N1(C(C(C)CN(C)C)=O)CCC2(CC1)CN(c1ncc(C#N)cc1Br)CCO2 C1(NC(c2c(C)con2)=O)CN(C(=O)C2=CS(=O)CCC2)CC2CCCC12 C1(C(C)NC(=O)C(C)C2CCOC2)CCCCN1C(c1ccccn1)=O C1(C(=O)NCC2(NC(=O)Cc3nc[nH]n3)CCC2)CCCCO1 Cc1ccc(C)c(C(=O)NC(C)C(C)NC(=O)Cc2ccc(C)c(F)c2)c1N C(=O)(C1CCCc2nc[nH]c21)NC1CC(C)(NC(c2cnc(S)nc2)=O)C1 C(CCC(C)(C)C(=O)N1CCC(NC)C1)NC(CSCC)=O c1(OCC)ccc(F)c(C(=O)NC)c1F.c1(C(N2CCC2)=O)c(C)coc1C CC1CCN(C(=O)C=CCF)CCN1C(C1C=CCS1)=O C1(N(C(CCN2CCN(C)CC2)=O)C)CC(C)(C)OC1=O C1(O)(CNC(CCC2(C)CC2(F)F)=O)CCN(C(c2ccc(Cl)[nH]2)=O)CC1 N(C(=NCCc1cccc(Br)c1C)NCC1(C#N)CCC1)C(CC)C C1(NC(c2n(C)ncc2Br)=O)CCCCCC1NC(C12CC(C)(C1)C2)=O N1(C(C(c2cncnc2)C)=O)CC2CC(C1)N(C(c1ccc3c(c1)COC3)=O)C2 Cc1cc(F)c(C(=O)NC2CC3CC2N(C(c2ccoc2Cl)=O)C3)cc1F Cc1ccc2occ(C(=O)NC3COCCN(C(=O)CN(C)C4CC4)C3)c2c1 c1(C(N(CC(C)NC(=O)CC2CC3(CC3)C2)CC)=O)nnn2c1CCC2 n1(CC)ccc(C(=O)NCC2CCCC2NC(=O)CC2CCOC2)cc1=O C1(NC(Cc2c(C)nc[nH]2)=O)CC2CN(C(c3ncsc3S(N)(=O)=O)=O)CC2C1 C(=O)(C1=C(SC)CCCC1)N1CCCN(C(COCCOCCOC)=O)CC1C c1(C(C)C)cccc(C(N2CCCC(CO)(NC(=O)C(C)C(C)(F)F)C2)=O)c1N C(c1c[nH]cn1)=C(C(=O)N(C1CCOCC1)CC(=O)OCC)F c1(CC(=O)NC2C(CNC(CCC#C)=O)C2)ccc(C)c(N2CCOCC2)c1 N1(C(c2[nH]cc(CC)c2)=O)CCCN(C(=O)Cn2nnc3ccccc23)CC1C c1(SC2C(O)CCCC2)ccc(Cl)nc1C(F)(F)F C1(CNC(CN(C2CCC2)C(C2CC(SC)C2)=O)=O)CC12CC2(F)F C(C(C)(C)C(C)(C)C)NC(CCOCCN(C)C(C1(F)CCOCC1)=O)=O c1ccc2c(c1)COC2.c1(OC)cc(C(=O)NCCCNCCOC)n(C)n1 N1(C(C(CCC)(C)O)=O)CC=C(C(=O)N(C2CCOCC2)C2CC2)CC1 C1(CC)CCN(C(c2cnc(C)s2)=O)C1CNC(=O)COCC(=O)N c1(C(=O)NC(CC(C)NC(=O)CC2CC2(Cl)Cl)C)ccc(Cl)nc1 CC1(C(=O)N2CCC(CNC(=O)C(O)P(C)(C)=O)CC2)CCCc2ccccc21 N1(C(C2CCN(S(C(CC)C)(=O)=O)CC2O)=O)CCC2(CCCCC2)CC1 C(CC1=CCN(C(=O)CCC#N)CC1)NC(c1ccc(SCCC)cc1)=O C=CC(O)(C(=O)N1CCC(CNC(C2(C(=O)NC)CC2)=O)C1)C(F)(F)F N1(C(CC2N(C(C=C(C)C3CC3)=O)CC2)=O)CC2(CCNC2=O)C1 C1(C(N(CCC(C(C)C)NC(c2csc(=N)[nH]2)=O)C)=O)CC2OC1C1CC21 N1(C(c2snc(C)c2N)=O)CC2=C(C1)CN(C(=O)CC(CN(C)C)C(F)F)C2 C1(C)CN(C(=O)CC2CC3(CC3)CO2)CCO1.Cn1ncc(Cl)c1CC(=O)N.C C1(OC)CC(NC(=O)NC2CCC3(COC3)C2)CC(O)C1O C1(C(=O)NC(C(C)NC(CCCNC(C)=O)=O)CO)CCCOC1c1ccccc1 CC(O)CCCC(=O)NCC(C)(C)Cn1cc(C2CCCC2(F)F)nn1 C12(CC(N3CC(NC(C(C(C)C)O)=O)C(F)CC3)=O)CCC(CC1)C2(C)C c1(NCCc2nccn2-c2ccccc2)cc(OC)nc(CO)n1 CCCC(O)CC(=O)NCCC1(O)CN(C(c2cncc(C(=O)OC)c2)=O)C1 Cc1cc(Br)cnc1C(=O)NCC1CCN(C(C2(n3cnnn3)CC2)=O)C1 CP(C)(=O)c1cc(C(N2CCCC2C)=O)ccn1.C1(O)(C=O)CC(F)(F)C1.N N1(C(C2(NC(C(C)C3(O)CCC3)=O)CC(F)(F)C2)=O)CCC2(CCO2)C1 C1(NC(c2c(CC)ocn2)=O)CCCCC12CCCN(C(=O)C(C)CCOC)C2 c1(CN2C(C)CC(F)C2)coc2cc(F)cc(F)c12 c1(C(c2nnnn2C)NC2(CCOC)CC2)coc2ccccc12 n1(C(C)C)cc(C(N2CC(C)(NC(C3CC(O)CN3C)=O)C2)=O)c(O)nc1=O CCCC(C#N)C(=O)N1CC(NC(=O)CC=Cc2ccc(F)cc2)C(SC)C1 N1(C(C(CSC)C)=O)CCC(C)(C)C1CNC(=O)C.c1ccc(F)cc1F.O c1(NC(=O)CC2COCCN2C(c2cc(Cl)cnc2O)=O)ncnc2occc12 Cc1ccc(C=CC=O)nc1.c1(C(C(=O)N(CC(C)C)C)C)cccc(F)c1.N Cc1csc(C(=O)NCCN(C)C(C2CC3(CSC3)C2)=O)c1C c1(C(N2C(C)(C(=O)OC)C=CC2)=O)cc(OC)cc(OC)c1Cl C1(CC)CCC(C)N1C(=O)C(C)C(N)c1ccccc1 c1(OC)ccc(Cl)c(C(=O)NC(C)CC(C)C)c1F.C(=O)(C1=C(C)OCCC1)N N1(C(Cc2c(C)nc(C)s2)=O)CCC2(NC(=O)CC3CCC(=O)NC3)CCCC12 c1(C(=O)NC(C)Cc2cn(C)nn2)cc([N+](=O)[O-])cc2c1NCC2 c1(CC)n[nH]c(=NC2CC23CC(NC(c2c(C(F)F)cnn2C)=O)C3)s1 c1(C(N2CC(CCOC)N(C(=O)C(C)O)CC2)=O)cn2cc(C)sc2n1 C1(CNC(=O)COCC2CCCC2)CCCN(C(c2ccsc2)=O)CC1 c1(C(=O)NC2CCC(C(=O)NC(C(CCC)O)CO)C2)ccc2occc2c1 N1(C(c2c(C)cnnc2)=O)CCC(NC(=O)C(C)(F)C(F)(F)F)CC(O)C1 c1(C(N2CC3CCC(C(N4CCCC(CF)C4)=O)(C3)C2)=O)n[nH]c2ccccc12 CC(C(=O)NC1CC(CNC(c2ccc(C3CC3)nc2)=O)C1)S(C)(=O)=O C1(N(C(c2c(C)cn(C)c2)=O)C)CN(C(C2CC2(Cl)Cl)=O)CCC1C CC1CN(C(c2cc(-c3ccc(Cl)cc3)ns2)=O)Cc2c[nH]nc21 C1(c2cn(CC(COC)O)nn2)CCCCN1C(c1ccnn1CC1CC1)=O C(=O)(CCCC(=O)NC1CCCC1C(=O)NCc1nc(CC)no1)OCC N1(C(C(CC=C)OC)=O)CCN(C)CC1C(=O)NC(CC)C(=O)NCC c1(C(N2C(CN(C(C3C(CC)C3)=O)C)CCC2)=O)ccc2oc(C)nc2c1 C(C1CCN(C(=O)CNC=O)CC1)=CC(=O)NC(CC(C)C)C Cc1cc2ncc(C(N3CCN(C(=O)C(C)C#N)CC3C)=O)cc2[nH]1 c1(C(N2CC(O)(C(C)NC(c3ccc(F)o3)=O)C2)=O)ccc2n[nH]cc2n1 C1(C(=O)N)CCCC1S(C)(=O)=O.c1(CCC)ccc(CC(=O)NC2CCC2)cc1 C=C1CC2CC1CC2(c1nnnn1C)NC(C)COCC(F)(F)F N=c1ccc(C(=O)NC23CC(C2)N(C(=O)Cc2ccc(Cl)nc2)C3)c(Cl)[nH]1 c1(CNC(=O)CSCCNC(C23CCCCC2C3)=O)cc(O)ccc1F CC(c1cccs1)=CC(=O)N(C1CN(C(=O)CN(C(C)C)C2CC2)C1)C CC1CCC(C(=O)NCC=O)CN1C(c1cc(N2CCCC2)ccn1)=O.C1CC1 c1(C(N2C(C)CCC(C)C2)=O)coc(S(N)(=O)=O)c1.C(=O)(C)N.CC(N)=O Cc1nc(C)c(C(N2CCCC(N(C(=O)CC3=NNC(=O)C3)C)C2)=O)nc1C c1(C(=O)O)ccccc1.C(C(N)=O)N(C(=O)CNC)CCC.C(N)=O.N C1(CNC(c2cc(CC)no2)=O)CN(C(=O)C(C)N=[N+]=[N-])CCC1C c1(CC(=O)N(C(C)C)CC)cc(O)ccc1Cl.c1(C=O)cncn1C1CC1 N1(C(COCCCCC)=O)CCC(CO)(C)CC1.C1(C)(C=O)CC2(CCC2)C1.N C(CC(F)F)(C(=O)N(C)Cc1ncc[nH]1)NC(c1cc(OCC)no1)=O Cc1c(C(=O)NC2CCC2NC(c2nc(C(F)(F)F)ccc2F)=O)cccc1N Cc1cc(-n2ncc(C(=O)NCCC(C)N(C)C(c3cncs3)=O)n2)cc(C)c1 O=S(=O)(c1ccc(-c2ccc(Cl)c(Cl)c2)s1)NC1CONC1=O c1(C(N(C2CCN(C(=O)CN(C3CCSC3)C)CC2)CC)=O)cc(C)ncn1 C1(NC(CCC(N)=O)=O)CCCCN(C(C2CS(=O)(=O)CC(=O)N2)=O)CC1 c1(C(=O)NC2CC(F)(CNC(C3C(C)CCCC3)=O)C2)cc2ccccn2c1 C1(CCO)(NC(C2CC2C2CC2)=O)CN(C(=O)CCOc2ccccc2)C1 C=CCC(C(=O)N1CCC1CC(=O)NC(C(C)C)C1CCC1)NC(C)=O Cc1c(C(=O)NCC2CC2)[nH]c2c1CCCC2.C(=O)(C(O)C(C)(C)C)NC.C N1(C(c2cc3ccccn3n2)=O)CCCC2CCCCC12 Cc1cccc2nc(CCC(N3CCC4(CCCN4C(=O)CC4CC4)C3)=O)[nH]c12 C1(CNC(C(CCC)O)=O)CN(C(C2CCC(SCC)CC2)=O)CC1(C)C C1(OC)CCC(N(CCC(=O)N(c2ccccc2)Cc2ccccc2)C)C1 c1(C(N2CCCC2C(C)C)C(=O)NCc2c(NC)cccc2)ccc(C)cc1Br C(=O)(C(CNC(=O)CCn1cccc1)N(C)C)N(C)CC1CCCO1 N1(C(c2nc(C)nc(O)c2)=O)CCN(C(=O)C(F)(F)C(C)O)CC(CO)C1 c1(OC)cc2c(cc1O)CCN(N1CCOC3(CCSC3)CC1)C2 c1(CC(=O)NC2(CNC(C(C)OCC#C)=O)CCC2)cc(C)ccc1 c1(OC)cc(OC)cc(CC(=O)NC(C)CCNC(=O)C2=CC(C)(C)C2)c1 C1(NC(CCCNS(C)(=O)=O)=O)CC2CC1N(C(=O)C(c1cccc(C)c1)O)C2 C1(NC(N(CC(C)(C)C)CCO)=O)CCC2(CCOCC2)CC1 c1(C(=O)N)cc2nc(C)sc2[nH]1.C1(NC(Cn2ccc(C)n2)=O)CC(C)C1(C)C C(=O)(C1=COCCO1)N(C1CN(C(C2CCCC(C)(C)O2)=O)CC12CC2)C Cc1ccc(C(=O)N(CC(=O)NC(C)C(=O)NC2CC2)C2CCC2)cc1F CCCCCC(F)C(=O)NC(C)CCC(=O)NCC1CCCC12CCC2 Cc1cc(C(=O)NC2C(C)CN(C(=O)C(F)(F)CO)CC2C)nc2[nH]nc(O)c12 CC1=C(c2ccccc2)CN(Cc2nc3ccccc3s2)CC1 CC(O)CCCN=C(NCc1ccccc1)NCC(Cl)C(F)(F)F CCCC(O)C(=O)NCC=CCC(=O)N(C)CCOC.C(=O)C(C)C Cn1cccc1CC(=O)NC1CCCC1NC(=O)Cc1ccccn1 C1(C(NOCC(CSC2CNC2)(F)F)=O)CCCC1.N1CCC1 n1(C(C)C)c(O)nc(N2CC(CN(C)C(C3CCc4nncn4C3)=O)C2)cc1=O C(=O)(CC(C)(O)COC)NC(C(C)NC(c1cc(CC)oc1C)=O)CO N1(C(C(C)SCC)=O)CCOCC1.C1(C(NC)=O)CCN(C(=O)C2CC2)CC1 c1(C(=O)NC(CC=C)CNC(c2cc(C)no2)=O)cnc2c(Br)cccn12 N1(C(Cc2c(C(=O)OC)cccc2)=O)CC2CN(C(c3cc(C)ns3)=O)CC2C1 C1(C(=O)O)CCC(C(N2CCCC2c2cc(Br)cs2)=O)C1 N1(C(CCSCCC)=O)CC2(CC2)CC1C(=O)NCC1(O)CCCOC1 C1(NC(C(c2cccs2)NC(C2C(CC)N(C)CC2)=O)=O)CCC(C)(C)CC1 N1(C(c2n(CC=C)ccc2)=O)CCC(CO)C1.c1(C(=O)N)cnc(N(C)C)cn1 c1(SC)nc(NC(C)CCNC(c2cnn(CCC3CC3)c2)=O)ncc1C c1(NC2CN(CC)C(=O)C2)ccc(S(=O)(=O)NCCC(=O)N)cc1Cl.C1CC1 C(C(=O)N1CCC1C(N1CC(c2ccon2)C1)=O)(C1CCC1)OCC n1(CC(=O)NCc2cc(C3CC3)no2)cc(CNC2CCCC2)nn1 C1(C)(C(N2CCN(C(C=COCC)=O)CC2C)=O)CCC(C)C1(C)C CCC(CC)(CCNC(=O)C(C)(Cl)Cl)NC(c1cc(C(N)=O)cc(F)c1)=O N1(C(c2cc(N)ncn2)=O)CCCCC(NC(=O)CC2CC3CC3C2)C1 N1(C(c2cn(CC)nc2C)=O)CCC2CCN(C(=O)CC(=O)N)CC12.C1CC1.C Cc1cc2[nH]c(C(N3CC4(CCCN4C(C4CC4(F)Cl)=O)C3)=O)cc2s1 C1(CC(=O)NCC(C)C2CC2)CCS(=O)(=O)C1.c1nc[nH]n1.C(=O)C.N N1(C(CCC(=C)C)=O)CC(C)CCC1CNC(C1C2CCC1(c1cscn1)C2)=O c1(C(=O)N)cc(Cl)c2ccncc2n1.C1(=CC(=O)NCC2CCC2)CCOCC1 N1(C(c2c(C)noc2)=O)CC2(C1)CN(C(C1CC3C=CC1C3)=O)C2 N1(C(C2CC(CC)C2)=O)CC2(CNC(c3cnn(C)c3OC)=O)CC1CO2 c1(CC)cc(C(=O)NC(CNC(=O)CN(C2CCCC2)C)CC)nn1C CC(N=[N+]=[N-])C(=O)N1CCC(O)(C(C)NC(c2ccccc2)=O)C1 CC1CCOC(C(=O)NCCN(C(=O)C(C)Cn2cccn2)C2CCCCC2)C1 CCCC(C#N)C(=O)N(C)CC1CCCN1C(c1cc(C(N)=O)ccc1OC)=O Cn1cc(Cl)c(C(=O)NC2CCC(C(=O)NCCCC3(O)CCC3)CC2)n1 N1(C(C2(C=C)CCN(C(=O)C(F)CCC)C2)=O)CCC(C)(C2CC2)C1 C12(COCC)CCOC1CN(C(=O)C(=O)NC1(C)CC3CCC(C1)S3)C2 N1(C(c2cc(C(=O)OC)[nH]c2)=O)CC(NC(c2ccsc2)=O)C(C2CC2)C1 N1(C(c2c(CC)nc(C)[nH]2)=O)CCC(C2CCN(C(=O)COCCS)C2)CC1 Cc1ccc2c(c1)CCC2C(=O)NC(CNC(c1ccc(Cl)cc1)=O)C1CCC1 c1(C(N(C)CC2CCCN(C(c3ccc(=O)oc3)=O)C2)=O)cc(O)ccc1F O=S(=O)(c1ccc(NC2CCCn3ncnc32)c(F)c1)NC1CC2CC2C1 C1(C(=O)NCCN2CC=CCC2)CC(NC(C2CCCC2F)=O)C12CCC2 Oc1ncnc2ccc(CSc3nc4cccc(Cl)c4s3)cc12 C#Cc1ccc(OCC(=O)N(CCNC(=O)CCc2cc(C)no2)CC)cc1 C(C(C)(O)CC(=O)NCCCN(CCCNC(=O)CCCCCF)C)OC c1(N2CC(C(C)NC(=O)CC3CCCCC3C)C2)ncnc(Cl)c1Br c1(CN(C(=O)Nc2cccc(OC)c2F)C)cc2c(cc1Br)OCO2 c1(N2CCC(N(C(=O)C=Cc3cocn3)C)C2)nc2c(cc1C#N)CCCC2 C(CC(C)C)(C(=O)NCC1(CSC)CC1)NC(C(CC#C)C1CC1)=O CC(C)C(C)CCNC(=O)CCNC(=O)C(C)c1ccsc1 C(N=c1nc(N2CCC3(CCC(O)C3)C2)c2c([nH]1)COC2)C1CCN(C)CC1 c1(C(=O)NCC(CC(C)C)NC(=O)C(C)(C)n2cnnn2)ccc(Cl)c(O)c1 C1(CNC(CC2(CC)CCC2)=O)CN(C(c2cc(F)ncc2OC)=O)CCC1C N1(C(C2C(C)OCC2)=O)CCCCCC1CNC(=O)CC=Cc1ccccc1F N1(C(c2cc(OC)ns2)=O)CC2CC(C1)C2NC(=O)C1=COCC1 Cn1ccc(C(=O)NCCCC(O)C(=O)N2CC(F)C(F)C2)cc1=O C=C(CC(=O)NC1(C)CCS(=O)(=O)C1)C(=O)OC C(=O)(C1CCc2cc(F)ccc21)N(CC1CNCC2(O1)CCC2)Cc1ccccc1 C1(C(=O)Nc2ccc(CCC(=O)OC)cc2)CCC2(CC1)OCCO2 C1(CN(C)C)CC(NCc2ccnc(C(=O)OC(C)(C)C)c2)CCS1 C1(O)(CCNC(COC2(C)CCCC2)=O)CCCN(C(c2ccc[n+]([O-])c2)=O)C1 N1(C(c2c(CC)n[nH]c2)=O)CC2(CCC2)CC1C(=O)N(CC(C)C)C c1(SC)ncc(C(=O)NC2CN(C(c3ncncc3F)=O)CC2(C)C)c(O)n1 N1(C(C=CCOCCOC)=O)CCC2C(C(=O)NC)C2C1.c1nnc(C)s1 C1(CNC(CCCC)=O)CCCC12CCN(C(C1CCC(C)O1)=O)CC2 c1(CC=O)c(C)nn(C)c1Cl.c1(OCC)cc(NC(C)C2CCC2)ncn1.N CC(c1ccccc1F)=CC(=O)NC(C)C(C)NC(c1ccncc1)=O c1(CC(=O)NC2CCC(F)(CNC(C3OCCO3)=O)C2)ccncc1Cl c1(C(N(C(C(=O)NCC2CCC(C)N2C)(C)C2CC2)C)=O)n[nH]c2c1COC2 C1(C(N(CCOC)CC2CCOC2)=O)CN(C(=O)Cc2ccsc2)CCC1O n1(CCC)ncc(C(=O)NCC2CN(CC3CCCN3C)CCO2)c1C1CC1 C#CC1(C(=O)NCCC=CCCC)CCN(C(C2C(C#N)C2(C)C)=O)C1 Cc1cc(C(N2CCCC(C(C)C(=O)NCCN(C)C)C2)=O)nc(C)n1 C1(C(N2CCC(NC(C(CC)OC)=O)(COC)CC2)=O)CCC(N=[N+]=[N-])CC1 N1(CC(c2c(C)noc2C)C)CCC(=O)N(CC2CC2C2CCC2)C1=O CC1CN(C(=O)CCN2CCOCC2)CCCN1C(c1nncn1C1CC1)=O CC(C)CC(C(=O)NC1CCCC(NC(c2nn(C)c(Cl)c2Cl)=O)C1)N(C)C Cn1cnc(I)c1C(N1CCC(c2cccc(Cl)c2)C1)C(=O)N(CC)CC1CC1 C1CCC2(CN(C(=O)CC3CCC4CC34)C2)O1.c1(C(=O)NC)cnnc(Cl)c1 C(CC(C(=O)NCC1C=CCCC1)NC(=O)CC1CCCC12CC2)SC N1(C(C2(OC)CCSC2)=O)CC2CCCC(CNC(C3CSCCS3)=O)C2C1 N1(C(C(C)N(C)C)=O)CC(NC(C2(C#N)CC2C(F)(F)F)=O)CCC1C Cc1nc(C)c(CNCC2CC(n3ccnc3)C2)nc1C Clc1ccc(C2CCCC2NCc2cnc(C3CCOCC3)nc2)cc1 C=C1Cn2c(C(N3CC(NC(=O)C(C)CCC)C(C)(C)C3)=O)nnc2S1 C1(N(C)C)C2CN(C(=O)C(C)(C)NC(=O)CC3CC=CCN3C)CC12 c1(OC)ccc2oc(C(N3CCC(C)(F)CC3)C(=O)NCC3CCCO3)cc2c1 c1(C(N(CC=O)CC)=O)nsc2ccccc12.c1sc2c(c1C(N)=O)CCC2.N CC1(C)COC(C(=O)NCC2C(C(=O)NC3CC(F)(F)C3)C2(C)C)C1 N1(C(C(C)C(C)(C)C)=O)Cc2ccc(CNC(C3CC3C3CC3)=O)cc2C1 C(=O)(CS(=O)(=O)CCOC)NC1(C)CCN(C(C(CC)COC)=O)C1 c1(SC)ccccc1C(=O)N(C1CCCCC1N(C)C(C1CCC(=O)N1C)=O)C C1(C(=O)NCC(CCC)OC)CCN(C(=O)C=C(C)C(F)F)O1 C(CC(C)C(=O)N1CCC(CCC(=O)N(C)Cc2nnc(CC)o2)C1)=CC c1(CNC(C(n2cc(C3CC3c3ccccc3)nn2)C)=O)nc(Br)n(C)n1 N1(C(C(CNC(c2c(CC)ncnc2)=O)(C)CC)=O)CCCC(C)(O)CC1 N1(C(CC2C=CC(NC(c3c(CC)non3)=O)C2)=O)CCn2nccc21 CCC(CC)CCCC(=O)NCC(CC(=O)N(CC(=O)NC(C)(C)C)C)OC c1(C2C(NC(C(=O)NC3CC(=O)NCC3)=O)C2)ccc2ccccc2c1 CC1=NN(CCC(C)C)C(=O)C1CC(=O)NCCN(C(=O)C)C.CCC#N.S C1(C(N(CCCC)CC)=O)CCC2CCC1N2C(=O)CC12CCCC1C2 C1(C=O)(CC)CC1(F)F.N1(C(C(=O)N(CC)C2CC2)=O)CCC(C)C1.N C1(C(N(C2C3C=CC(C3)C2N)Cc2n(CC)cnc2)=O)CC2(C1)OCCO2 S(=O)(=O)(c1ccc(=NCc2cn(C3CC3)c(=O)nc2O)[nH]c1)NC(CC)(C)CO C(=O)(C(C)CC(C)(C)C)N(CCC)CC.c1(C=O)csc(CC(F)(F)F)n1.N c1(CC)onc(C(=O)NC2(C)CCN(C(C3(F)C4CCCC34)=O)C2)c1C N1(C(c2cc(C)n(C)n2)=O)CCN(C(c2ncc(N)cc2Cl)=O)CC1CO C1(NC(c2cnc(COC)s2)=O)CCSC12CN(C(c1[nH]cnc1C)=O)C2 C1(CC(=O)NC2(C)CCC2)C2CN(C(=O)CC3C=CCCC3)CC12 c1(C(N2CC3(CN(c4nc(C(C)C)cc(C)n4)C3)C2)=O)ccc2ccnn2c1 C=C(C)CC(C)C(=O)NC1CC(N(C)C(c2ccnn2CCF)=O)C1 N1(C(CC(CC)(F)F)=O)CCCC2(NC(c3ccno3)=O)CC2C1 CC1CCN(C(c2cc(CF)on2)=O)C(C)C1.C1(C=O)CCC(C(C)(C)C)O1.N c1(C(N(C2CCCN(C(c3n[nH]c(C)c3O)=O)CC2)C)=O)ccnc2ncnn12 c1(CC)ccsc1C(=O)NC1CCOC1C(=O)NCC1CCOC1C C(=O)(C1CCOc2ccccc21)N(CCCN=c1cc(C)[nH]c(SC)n1)CC C1(C(N(CC)CC2CCC2)=O)CC2CCCC2N1C(c1ncccc1O)=O C(=O)(CCCCCCNC(C1(C)CC=CC1)=O)N1CCN(CCC)CC1 C1(CNC(CN(C(C)C)C(C2CC3(CCO2)CC3)=O)=O)CC(C)(C)CCO1 CON=C(C(=O)NC1CCC(Nc2cc(SC)nc(SC)n2)CC1)c1ccco1 N1(C(c2cncc(N)c2)=O)C2CCCC1CN(C(=O)CCc1cn[nH]c1)C2 Cc1cc(C(=O)NCC(C)(F)CNC(=O)Cc2cccnc2O)nn1C(F)F N1(C(C=CC)=O)CCCC2(CCCN2C(c2[nH]c3ccc(F)cc3c2Cl)=O)C1 N1(C(CSCCC(C)C)=O)CC(NC(C2CC3CCC3C2)=O)CC(O)C1 c1(C=O)ccc(NC=O)cc1.CC(C(=O)NC1CC1)NC(c1ccoc1)=O.N N1(C(C(C=C)(C)O)=O)CC2CCC2(CNC(=O)C)C1.c1(C(=O)N)cscn1 c1(C(=O)NCC(C)(C)NC(c2cccc3sccc23)=O)c[nH]c2ccc(O)cc12 c1(C(=O)NC(CNC(CSCCCC)=O)C)cc(F)c2ccccc2c1 N1(c2cccc(C)n2)CCCC(C)(C(=O)NC(c2nncn2C)C)C1 C1(NC(CCC2N(C(c3c(CC)cno3)=O)CCCC2)=O)C(=O)OC2CCCC12 c1(CC)nn(C)c(C(=O)NC2CCCCN(C(=O)CCC3CC3(F)F)C2)c1Cl C1(C(N2CCCC(CCNC(=O)CC3COC4CC3C4)C2)=O)CN2CCN1CC2 C(C(CC(C)C)C(=O)N1CC(c2cc(O)no2)C1)NC(c1ccc(C#C)cn1)=O N1(C(c2ccc(C)nc2)=O)CCCC(O)(c2ccccc2)CC1 c1cccc(C)c1.N1(C(C2(SCC)CC2)=O)CC(O)(C)C1.C(=O)(CC)N N1(C(CC)C(=O)NCCN(C(=O)CCN2CCC(F)C2)C)C(=O)CCC1=O C=C(C)C(CC(=O)NC(CNC(=O)CCn1c(C)csc1=O)CC)OCC C(=O)(CC(F)(F)F)N(C1CC2(C1)CC2)C.c1(CC(=O)C(=O)N)nc[nH]n1 CC(C)CC(C)(C)C(=O)NCCCN(C(C1CCOC(C)C1)=O)C1CC1 CC1CC=CCC1C(=O)NC1CCC1C(=O)NC1(c2ccsc2)CC1 CCC(C)C(CN=c1cccc(S(=O)(=O)N2CCN(C)CCN(C)CC2)[nH]1)OC C1(CNC(CC2CC(=O)NCCC2)=O)CN(C(=O)C2=CCCCC2)CCC1(F)F CCC(CC)CCCC(=O)N1CC(OC)CC1(C)CNC(c1cnc(OC)s1)=O C(=O)(C1=C(CC(C)C)N(c2ccc(F)c(F)c2)C(=S)NC1c1c[nH]c(Br)c1)OC n1(C(C)C)ccc(C(=O)NC)n1.C1CCN1C(=O)CC1(c2ccon2)CCC1 c1(N2C3C(COCC)CC(CC3)C2)nc2c(c(=NCC#CCCO)[nH]1)CCCC2 C1(OCC)CN(C(c2ccc(CO)cc2)=O)CC1.c1(CC=O)n[nH]c(C)n1.C CC(C)C(C(=O)N1CCC1CNC(c1ccc(NC2CC2)nc1)=O)C(C)C CC1c2c[nH]nc2CCC1C(=O)NCC(C(C)(C)C)NC(=O)CCc1nccs1 CC1CC(C(=O)NCC2CC(O)(CNC(C3CC(O)C3)=O)C2)=NO1 C1(NC(c2nc(N(C)C)oc2)=O)CCCCC1.C1(S(C)(=O)=O)(C(=O)N)CC1 C1(C(C)NC(=O)CCSC(F)(F)F)CCN(C(C2CCCOC2)=O)C1 c1(C(=O)NC(C(CC)CCO)C)ccc(C)c(Cl)c1F CC1C(NC(c2ccnc(Cl)c2)=O)CCN1C(c1cnco1)=O C1(C(N(CC(F)(F)F)C(C)C)=O)COCCN(C2CCCNC2)C1 C1(NC(N(C(c2cc(F)cc(F)c2)CN)C)=O)CC2CCC(C1)S2(=O)=O Cc1cccc(Br)c1C(=O)NC12CCC1CN(C(=O)NC(=O)C(Cl)(Cl)Cl)C2 C1(C(=O)NCC(c2ccccc2)OCC)CCc2c(ncn2C)C1 C(CC(C(=O)NCC#CC(F)(F)F)NC(C1CC2(CC2)CO1)=O)N(C)C Cc1cc(C)c(-n2nnnc2C(C2CCOCC2)NCC2C3COCC23)c(C)c1 N1(C(C(c2cn(CC)nc2)=O)=O)CCCC(C)C1.C1(C(=O)N)CC2CCC(C1)O2 c1(NC2C(OC)COC2)nccc(N2CCC(N3CCC(O)CC3)C2)n1 c1(C(c2nnnn2CCCF)NC(C)CCc2ccco2)cc(Cl)c(Cl)c(Cl)c1 c1(C(N2C(CC)CN(C(=O)C(O)P(C)(C)=O)CC2)=O)noc2ccc(F)cc12 c1(C(N2CCC(N(C(=O)CCC(C)(F)F)CCC)C2)=O)cccc2ccn(C)c12 C(=O)(C1CCCc2ncnn21)N1CCC(CNC(c2ncn(C)c2)=O)C12CCC2 Nc1cc(C(N2CCC(CNC(c3c[nH]nc3F)=O)C23CC3)=O)ncc1Cl CC(CC(=O)N)P(C)(C)=O.C1(F)(C=O)C(C)(C)C1(C)C.C1CC12CCC2.C N1(C(C2CC3(CN(C(C)=O)C3)OC2)=O)CC2CCC(C1)C2C#N.C(=O)(C)OC.O C1(OC)CN(C(=O)C2=C(Cl)CC2)CC1NC(C1C(c2ccccc2)C1(F)F)=O CCCCCC(C)(C)C(=O)NCC(C)C(F)C(=O)NCCN(C(C)C)CC CC1CC(NC(C2(C)CC2)=O)CCN1C(c1cnoc1C1CC1)=O.C1CCC1 c1(CCC)n[nH]cc1C(=O)NC(CNC(c1occc1CO)=O)C(C)C C1(NC(C2CC(CCC)C2)=O)CCCCCN(C(c2ccc(CC)s2)=O)C1 CC1COCC(CC(=O)N(CC(N2CC(F)C2)=O)C2CC2)O1 CCCCC(O)C(=O)N1CCC(CNC(=O)CCc2ccc(O)nn2)C12CC2 Cc1nc(Cl)ccc1CN1CC2C(C(=O)NC3CCC(=O)NC3=O)C2C1 CC(CC(C)(F)F)C(=O)NCC(C)(C)CNC(=O)CC1CCC(F)(F)CC1 C(CC)(CCCC(=O)NCC1(SC)CCC1)NC(C(CCCC)C)=O C(=O)(C(CC#N)c1ccccc1)NCCC1CCC(NC(CSC(C)C)=O)C1 c1(NC(C2CN(S(C)(=O)=O)C2)=O)ccc(C(=O)Nc2ccccc2)c(Cl)c1 N1(C(C(C=CC)O)=O)CCCC(CC(N2CCC3CCC23)=O)C1 C(=O)(CC(CC)CC(F)(F)F)NC12CN(C(C(C(C=C)C)C)=O)C(CC1)CC2 c1(C(=O)NC2C(OC)CN(C(CC=C)=O)C2)cc(-c2ccncc2)ccc1C C1(C)(CNC(CCN(C(C)=O)C)=O)CCCN1C(C1CC(C)(C)CO1)=O c1(C(=O)NC2(CO)CN(C(Cc3cc(C)sc3)=O)C2)cnc2ccoc2c1 S(=O)(=O)(CC(=O)NC1CC(C(=O)NC2(CO)CC(F)C2)C1)NCC CC1C(C(=O)NC2CC(CNC(=O)CCCCCF)C2)C(O)C(=O)N1C N1(C(c2cccc(N)c2N)=O)CCC2CCN(C(C3CCSC3)=O)CC2C1 c1(C=O)c(C)cc(C)cc1O.c1(C(N(CCC)CC)=O)ccc(C)n1C1CC1 c1(C(N2CC(O)(C(C)NC(C(C)OCCC=C)=O)C2)=O)ccn(CC)c1C N1(C(C(C)OCCN(C)C)=O)CCC2(CCC2)C1.c1(C(=O)N)cc(Cl)nnc1O N1(C(CCCOC(C)C)=O)CCN(C(C2(C#N)CC=CC2)=O)CC(C)C1 CC1(C)CCN(C(=O)Cc2cncs2)CC1NC(=O)C(c1ccc(F)cc1)F c1(OC)cc(N2CCCC(CNC(c3cncc(F)c3)=O)CC2)nc(OC)n1 Cc1ncccc1CC(N1CC(C)(NC(=O)C(C)Cc2ccccc2Cl)C1)=O c1(NC(CC(CC)c2ccc(OC)cc2)=O)cc(S(N)(=O)=O)ccc1OC(C)C C1(C(N2CC(CN(C(C3CCN(CCC)CC3)=O)C)C2)=O)CCc2n[nH]cc2C1 c1(C(N2C(CC(=O)N(CCC3CC3)C)COCC2)=O)cc(C)cc(C#N)c1.C CC(c1cnn(C)c1)=CC(=O)NC1C2CC1N(C(=O)CC1CNC(=O)C1)C2 c1(CN(C(=O)NC2C(C)COCC2)CCO)ccc(Cl)cc1Cl N1(C(c2cnoc2)=O)CCCN(C(C2CC(C(C)C)C2)=O)C(C(C)C)C1.CO.C C(=O)(C(C)(C)C)NC.C1(CC=O)CCCCC1.c1(C=O)cc(C(N)=O)c[nH]1 N#CC1CN(C(c2ncc(Cl)cc2Br)=O)CCN1C(c1nccs1)=O C(=O)(C1=C(Cl)CCCC1)NC1C=CC(C(=O)NC2(C(C)C)CCC2)C1 C1(C(=O)NCc2ccc(OCC)cc2)CCCN(C(C2CC(C)C2)=O)CC1 c1(C=O)ccc2c(c1)CNC2=O.c1(COC)cc(C(=O)NC)n[nH]1.C1CC1 c1cc(C)nn1C.c1(CC)ccc(C(=O)NCc2nc(C(=O)NC)co2)[nH]1.C c1(C(=O)NC(CCC(=O)Nc2c(OC)cc(C)cc2)(C)C)ccc2occc2c1 C1(C)(CNC(CCC(C)SC)=O)CCCN(C(=O)C(=O)NCC2CC2)C1 c1(OC)nn(C)cc1C(=O)NC(C(=O)NCCc1ncc(C)o1)C1CCC1 N1(C(CC2CCCN(C(CCC3(C)CC3)=O)C2)=O)CCCC(C#N)C1 C1(CC)CN(c2cc(NC(c3ccncc3F)C)ncn2)CCO1 CC(C)C(O)C(C)(C)C(=O)NCCC1CCN(C(C2(C)CCNC(=O)C2)=O)CC1 N1(C(C(C)NC(CC)=O)=O)CCCC(CO)(NC(c2csc(C3CC3)n2)=O)C1 N1(C(CC(n2c(CC)ncc2)C)=O)CCOCC(F)(C)C1.C(=O)C=C(C)Cl.N C1CN(C(c2cnc(C(N)=O)s2)=O)CC2CC12.C(C(=O)N)N(C1CC1)CC Cc1cc(C(=O)NCC2(CCNC(c3cccs3)=O)CC2)ncn1 N1(C(C(C2CC2)OCC)=O)CC2CCCC(C1)N2C(c1cncc2[nH]ccc12)=O C1(C(N2C(C(N3CC(CO)C(O)C3)=O)C=CC2)=O)OCC2CCCC12 C1(CC(=O)NCC2(OC)CCOC2)CN(C(=O)C(C#N)C(C)C)CC12CC2 c1(NC(=O)NCCN=[N+]=[N-])cc2c(Br)cncc2s1 c1(-c2n(C(COC)C)nc(C3CN(C)CCO3)n2)nnc2ccc(OC)nn12 c1cc2c(cc1Cl)OCO2.C(C(C=O)NC(=O)CNCC1CN(C)C1)OC C1(C(N(CC(CC)NC(c2cc(Cl)ccc2F)=O)CC)=O)CC2(CCCC2)C1 Cc1cccc2oc(=NC(C)CCNC(C3CCCC4C3C4(F)F)=O)[nH]c12 C=CC(CCC)CC(=O)NC(CC)CCC(=O)NC1C=CCCC1 CCCC(CCC)NC(C1CCN(C(=O)CC2CC3(CCC3)C2)C1C)=O Cn1cnc2cc(C(N3CC4(C3)CN(C(C3CCC3C(F)F)=O)C4)=O)ccc12 N1(C(CCC(=O)NC)=O)CC(C)OC2(CCN(C(C34CC5CC3C4C5O)=O)C2)C1 N1(C(c2cc(C(C)=O)on2)=O)CC(CNC(C2CCOC2C)=O)OC(C)(C)C1 C#CCCCC(C)C(=O)N1CCC(C(=O)NC(c2n[nH]c(C)n2)C)CC1C Cc1ccc(C)c(C(N2CCOCC(NC(=O)CC3CC(C4CC4)C3)C2)=O)n1 c1(NC(C)=O)ccsc1C(=O)NCC1CCN1C(c1nnnn1C)C c1(C=O)cc(F)c(O)c(F)c1.C(CNC(=O)CC)(C)OC.C(=O)(CO)N CCC(C)(C)C(=O)NCC1CC(F)C1.c1(C=O)cnn(CCN(C)C)c1.C n1(CCCNC(C2C(OC)CNCC2)=O)nc(O)c2c1CCCC2 N1(C(c2cnc(CC)s2)=O)CCC(C2(O)CN(C(C3CCO3)=O)C2)CC1 CC(CC(=O)NC(C)(C)CN(C(=O)C=Cc1ncco1)C)CC(C)(C)C CC1=C(C(=O)N2CC(C(N)=O)(CNC(c3nc(O)sc3C)=O)C2)CCCC1 c1(C(=O)NCC(CC(C)C)NC(c2ccc(C)s2)=O)cccc2oc(O)nc12 c1(OC)cnc(C(N2CC(CC(=O)NC(C)CO)C2)=O)c(C)c1 c1(C(=O)NCCC(C)NC(C(CC)NC(C)=O)=O)cccc(OC)n1 CC1CN(C(c2cccc(F)c2C(F)(F)F)=O)CCN1C(=O)CC1CCCOC1 c1(C(C#N)N(C2CCN(C(c3csnc3Cl)=O)C2)C)ccc(C(F)(F)F)c(C)c1 C12(NC(N(C(C)CS(C)(=O)=O)C)=O)CCC(CC1)C2(C)C C1(C)(C(=O)NCc2c(C)nc[nH]2)CCN(C(=O)CCC2CCCN2C)C1 Cc1ccc(C(C)OC(c2cnn(-c3c(F)cccc3F)c2)=O)cc1[N+](=O)[O-] C1(NC(N2CCC(N3CCCCC3)C2)=O)C2Cc3ccc(Br)cc3C12 Cc1nc(C)c(CNC(=O)Nc2ncccc2Cl)c(C)n1 C1(C(=O)NCCN(C2CCCCCC2)C(CN(C)C)=O)CN2CCC1C2 C(=O)(C1CC(=O)Nc2cc(F)ccc21)NCC(C)(C)C.c1(CC=O)ccco1.N Cc1cc(Br)cc(C)c1C(=O)NCC1CCN1C(=O)CC1CCOC1 Cc1cccc(C)c1OCC(C)NC(c1cc(Br)ccc1O)C CCCCC(O)C(=O)OCC1CCC(=C2CCC2)CC1 C1(NC(c2cncc(OC)n2)=O)C2COCC1CN(C(=O)CC1CC(OC)C1)C2 c1(C(C(=O)NC(C2(O)CN(C(CCOCC#C)=O)C2)C)C)ccc(F)cc1F c1(NC(C(=O)N(C)C)=O)ccccc1.CC(C)(C)CN(C)C=O.C(C)(C)C c1(C(C(N2CCCC(NC(c3ccno3)=O)C2)=O)O)ccc(F)cc1Br CC1(C)CC(C(=O)NCC2CN(C(=O)COC3CCOC3)CC2(F)C)=NO1 c12ccc(F)cc1NC(=O)C2.n1(CC(C)=O)cc(C(=O)O)nn1 N1(C(c2cc(C)n(C(F)F)n2)=O)CC2CCN(C(C3(CO)CCCC3)=O)CC2C1 c1(C(=O)NC2CCC(NC(CC(COC)(C)O)=O)C2)cccn2cncc12 C1(C(=O)NCC2(C(F)(F)F)CCCC2)CCCCN1Cc1cccc(F)c1 C1CCCCN1C(=O)C(C)C1(O)CCC1.c1(C(C)OCC)ncc(C(=O)N)s1 N1(C(C(C=C)(C)O)=O)CC(NC(c2cn(CC)cn2)=O)C2(CCC2)C1 CC(=O)CCCC(C)C(=O)N(CCC(=O)N(C)Cc1nc(=O)o[nH]1)C1CC1 c1(N2CC(C=O)C2)ncc(F)cn1.CCCC.C1(C=O)(C(=O)N(C)C)CC1.N C1(NC(CC(C)(F)F)=O)CC2CC(C1)N(C(=O)CC1C=CS(=O)(=O)C1)C2 C(=O)(CCCCC(=O)N1CCC1CNC(=O)Cc1csc(C(C)C)n1)NC c1(C(=O)NCC(CO)Nc2ncc(C(C)=O)cc2C)cc2c(nc1O)CCCC2 C1(CC(=O)NC(CNC(C(COC)COC)=O)C(C)C)CCCCC1(F)F c1(CC(=O)NCC2(NC(=O)CC3OCCO3)CCCCC2)ccc(O)c(Br)c1 c1(C(N2CCC(C(C)NC(COCC)=O)C2)=O)c(C)nn2c(C)cccc12 c1(CNC2CCC(C(=O)NC(c3cccc(O)c3)CO)C2)ccn2ccnc2c1 N1(C(c2ccc(C)[nH]2)=O)CCCC2(CCN(C(=O)C(CO)C(C)C)C2)C1 c1(C(=O)NCCCCCNC(C2C(C)=CCS2)=O)cnc2cc[nH]c2c1 N1(C(c2cccc(CC=C)c2)=O)CCC(C(N2CCC23CCC3)=O)C(O)C1 C=C1CCN(C(=O)CCC2CCC(=O)C2)C(C(N2CC(N=[N+]=[N-])C2)=O)C1 CN1CCC(C(=O)NCCCN(C(=O)C(O)CF)CCO)CC1=O c1(C(N2CC(O)CC(NC(=O)CCCC3CCC3)C2)=O)cnc2ccccn12 C(=O)(C(F)CCC(C)C)NC1CN(C(C(C(CC)O)C)=O)C1 N1(C(CN(CCOC)C(c2cnncc2C)=O)=O)CC2(CC(C)CO2)C1 n1(CCC)ccc(=NC(=O)C2(NC(=O)C(C)OCCOCC)CCCC2C)[nH]1 N1(C(C(OC)OC)=O)CCC(C(C)C(=O)NC2CC(OC)C(OC)C2)CC1 C1(C(=O)Nc2ccc(CC)cc2)CC(F)CN(C(=O)N)C1.c1cccc(F)c1.C c1(C(=O)NC2CCCN(C(CC(C)(C)O)=O)C2)ccc(C(F)(F)F)nc1O C(=O)(C1=C(CF)N(CCC2CC2)C(=S)NC1c1nc(C)c(C)nc1C)OC CC1(C)CCOC(C(=O)NC(C2(O)CCCCC2)C(N2CC3(CC3)C2)=O)C1 C(CCCC(=O)NCC(C)(CNC(=O)C=CC(C)(C)C)OC)OC C(=O)(C(CC(C)C)NC(N)=O)N(CCOCCNC(CC=C=C)=O)C c1(CCC)cc(C(=O)NCCCCCN(C)C(C2CC23CCCC3)=O)ccc1Cl C(CC(=O)NCC1CC12CCOCC2)(C(C)(C)C)NC(c1c(C)ccs1)=O CC(C)CN=C(NCc1cn(C)nc1C(C)C)NC1CCOc2ccc(F)cc21 C1(C(C)C)CCCCC1NC(=O)CCCN(C)C(c1ccc(N)cn1)=O N1(C(CCCOCC)=O)CC2CC(NC(c3conc3-c3ccccc3)=O)C1C2 c1(C(C)C)ccc(C(N2CCOC(CN(C(=O)CC3CC(CF)C3)C)C2)=O)cn1 c1(C(=O)NC)cc(C(F)(F)F)ccc1[N+](=O)[O-].C1CC2CC2N1.C1CC(O)C1 CC1CCCC=C1C(=O)NCCCC1CCN(C(C2C(C#N)C2(C)C)=O)CC1 c1(COC)cc(N2CCC2CNC(=O)C(n2cc(C)cn2)C)ncn1 c1(C(N2C(CNC(C(c3ccccc3Cl)N(C)C)=O)C=CC2)=O)cccnc1S C1(C(=O)NCC2C(C(=O)NCC3(C)CSC3)CC2)CCCC(C#N)C1 c1(C(N2CC(N(C)C(c3ncc(F)cn3)=O)C2)=O)ccc(C(F)(F)F)c(Br)c1 CC(C)CS(=O)(=O)CCC(=O)N1CCN(C(C2(C)CCCOC2)=O)CCC1C C1(C(=O)NCc2cc(OCC)ncc2)COCCN(C(=O)O)C1.C(C)(C)C C1(C(N(C2CCCN(C(c3csc(CO)n3)=O)CC2)C)=O)COC2CCCCC12 C1(CC(=O)N(C(C)(C)C(=O)NCC2(N3CCOCC3)CC2)C)CCCOCC1 N1(C(c2c[nH]c(=NC)o2)=O)CCC(C2CC2)C1CNC(=O)CC(F)(F)Cl C1(O)(C(=O)OC)CCCN(C(C(=O)NC2CCC2)c2ccns2)C1 C1(F)(OCC)CCN(C(C2CC(C(=O)OC)(CC)C2)=O)CC1 C1(CCCNC(CCNC(=O)CO)=O)CN(C(c2c[nH]c(Br)c2)=O)CCO1 C1(C(=O)NC2CCN(Cc3cn(C(CC)C)nn3)C2)C2Cc3ccccc3C12 N1(C(C(C)OC(C)(C)C)=O)CCC(CC(=O)NCCCC2(O)CCC2)C1 c1(CCC)ccc(C(=O)NCC=CC)s1.c1(C(=O)N)cnn(CC(F)F)n1 C1(C(=O)NCCO)CCc2nc[nH]c2C1.C1(C(N2CCC2)=O)CC(=O)N(O)C1 n1(CC=C)nnnc1C(CC1CCCCC1)NCCCSC(F)F c1(C(C)OC)nc(-c2ccc(CN3CCCC3)cc2)n(CCCCO)n1 C(=O)(C1=C(C)NC(=O)NC1C)OCC.c1(C=O)cnn(C)c1CCC(F)(F)F c1(C(C)C)nc(NCCCCC2CC2C)cc(=NCC2(CF)CC2)[nH]1 N1(C(c2csc3nnsc23)=O)CCCCC2(CCN(C(C3CCC(F)C3)=O)C2)C1 CC(C(CO)NC(=O)C)NC(=O)COCc1ccccn1.CC.CCO.O n1(CC(N2CC(F)CC(NC(CC(C)CF)=O)C2)=O)c(O)nc2ccccc12 C12(C(=O)NCCC3(C)CCN(C(=O)Cc4cnc[nH]4)C3)CCN(CC1)CC2 c1(C(=O)NCCC(C)NC(c2c(Cl)cccc2Cl)=O)ccc(O)cc1F c1(C(C=O)=O)ccc(F)c(F)c1F.Cn1nccc1CC(=O)NCC1CCC1.N c1ccc(C#N)cc1.CC1CC(CNC(C2CC3(CCC3)C2)=O)CN1C(=O)C N1(C(C2C(C(C)C)CCC2)=O)C(C(=O)NCC2=CCCC2)CCC12CC2 C(=O)(C(C)CC(N)=O)NCC(CCC)NC(c1cc(C)c(C)cn1)=O C(=O)(C(C)(C)C=O)OCC.C1(S(N)(=O)=O)(c2cn(C3CC3)nn2)CCC1 C1(NC(c2c(CC)[nH]cc2)=O)CCN(C(=O)Cn2nccc2C)CC1C(C)C C(=O)(C(C)(C)CC(=O)NCCOCC(=O)N(C1CCC1)C1CC1)OC C1(C(N2C(CCC)COCC2)=O)CCN(C(=O)CCC(=C)C)O1 C1(NC(Cc2ncc(COC)[nH]2)=O)CCCC(OC(C)(C)C)C1 C1(CC)(NC(=O)CCC=CC(C)C)CCCN(C(=O)CC(=O)N)C1.C1CC1 c1(CCC(=O)NC2CC2NC(c2cscc2C(F)F)=O)cccc2cnccc12 C1(CCC)(NC(=O)CS(C)(=O)=O)CCCN(C(=O)C2=CCOCC2)C1 Cc1oc(CNC(=O)C(C)N=[N+]=[N-])nc1C(=O)NC(C)CN=[N+]=[N-] N1(C(c2cc(SC)oc2C)=O)CCOC2(C1)CN(C(C1(C)CCCNC1=O)=O)C2 CC1CCCC=C1C(=O)NCC=CCNC(c1ccnc2[nH]nnc12)=O C1(NC(COCC=C)=O)CN(C(C2CN(C3CCC3)C2)=O)CC1OC Cc1ccc(C(=O)NCC2C=CCN2C(=O)C#CC(C)(C)C)cc1S(C)(=O)=O Cc1[nH]c(=N)sc1C(=O)NCC1CCCN1C(=O)COc1cccnc1 c1(C(N2CC(N3CCN(Cc4ccc(C)cc4)CC3)C2)=O)cnn2c1CCCC2 CC1(NC(=O)C(C2CCCCC2)F)CC(O)C1 N1(C(CCOCC(C)C)=O)CC2N(C(=O)CSCC(F)F)CCC2(C)C1 c1(C(N(CCNC(c2c(C)nc(C)o2)=O)C2CC2)=O)coc2c1C(O)CCC2 CCCCCCC(C)CC(=O)NC1CN(CCNC(C)=O)C1 N1(CCCOCc2nc(C)on2)CCN(Cc2cccc(C(F)(F)F)n2)CC1 c1(C(N2C(C)CCC(NC(c3cnn(C)c3F)=O)C2)=O)cn(C)c2ncccc12 C1(CC(=O)NCCC(CNC(C2CN(C)C2)=O)O)CCCCC12CC2 N1(C(=O)CCC2CCC2)CCC2CCCC12C(=O)NC1CCCC1(F)F C1(CCCNC(=O)CC2CCSCC2)CN(C(c2cncnc2)=O)CCO1 c1(C(N2C(C(N(C(CC(=O)OC)C)C)=O)CC2C)=O)cccc2[nH]ccc12 C1(COC(c2c(C)nc(C(C)(C)OC)s2)=O)C2CC3CC(C2)CC1C3 N1(C(C(F)=CC)=O)CCC(NC(=O)C=C2CN3CCC2CC3)CC1C C1(O)(CNC(C2CCN(C(C3(CC)CNC(=O)C3)=O)C2)=O)CCN(C)CC1 C(=O)(C1=C(Cl)CCCC1)N1C(CNC(C2Cc3nnsc3S2)=O)CC(F)C1 C12(NC(=O)CN3CCCNC3=O)CCN(C(c3cccnc3C3CC3)=O)CC1C2 Cc1ccc2sc(C(=O)NCC(C)NC(c3cnc(C(F)F)nc3)=O)cc2c1 C1(CC(=O)N(CCCNC(c2c(CC)csc2)=O)CC)CCC(=O)NC1=O n1(CC(=O)OCC)cc(C2CCCN2C(C2(C)CC2)=O)nn1 C(CS(=O)c1cc(Cl)ccc1Cl)C1N(c2c(C)ccc(Cl)c2F)CCOC1 C1(NC(CC2N(C(C(C)n3cnnn3)=O)CC(F)C2)=O)CCn2cncc2C1 c1(SC)ccc(CCCC(=O)NC(C2CCCN(C(=O)CP(C)(C)=O)C2)C)cc1 C=CC1CN(C(C2CC23CCCC3)=O)CC1NC(c1ccn(CCF)n1)=O CC1(C)CCCC1CCNC(=O)COC1CCCC1 C(=O)(C(C)(C)C)N.C1(CCC)(C(=O)NC(C)C(C)NC(=O)C)CCC1 N1(C(C2(C)CSC2)=O)CCC2(CC1)OCCCC2NC(C1CCNC(=O)C1)=O C1(NC(=O)C(Cc2cccnc2)C2CCCC2)CN(C(=O)C(F)F)CC1O C1(CNC(COCCC)=O)CC2(CCC2)CN1C(=O)CCNC(=O)C N(C1CCCc2ccccc21)c1cc(NC(c2nccc(=N)[nH]2)C)ncn1 C1(C(=O)NCc2ncc(C(N3CC(CC)(CO)C3)=O)cn2)OCCCC1(C)C CCCCC(C)C(=O)NCC1(C)CN(C(c2cc(C(F)F)cc(F)c2)=O)C1.O c1(N(C)C)cc(-c2ncsc2C(=O)Nc2ccn3nccc3c2)ccc1[N+](=O)[O-] CC(C)(CCC#N)C(=O)N1CC2CCC1CN2C(=O)C#CC1(C)CC1 c1(NC)cnc(C(=O)NCC2(OC)CCN(C(=O)CSC(F)F)C2)cn1 c1(C(=O)NCCCC(C)NC(Cn2cc(C(C)=O)nn2)=O)ccc(C)c(F)c1F c1(CC)ccc(F)cc1.C(CC)(C(=O)N)OCC.c1(C=O)ccsc1C(F)F c1(CC)nocc1C(=O)NCCC1CCCC1.C(=O)(C(O)Cn1cncn1)N N1(C(c2c(Cl)cccc2Cl)=O)CC2(CCCC2Nc2ccc(C(F)(F)F)cn2)C1 C(=O)(C1=CC2CC(C1)CC2O)N1CCN(C(C(COC)N(C)C)=O)CC1C Cc1cc(Cl)c(C(=O)NC2CCCCN(C(=O)Cc3[nH]cnc3C)C2)cc1N Cc1cc(Br)c(C(=O)NC2C3CCN(C(c4ncccc4O)=O)C23)cc1Cl N1(C(C(C)OCC(C)C)=O)CCN(C(c2c[nH]c(=O)cn2)=O)CC1c1cn[nH]c1 N1(C(c2n(CCCC)ncc2)=O)CCCC(N(C(=O)C(Cl)=CCl)CCF)C1 CCC(C(=O)N1CC(C(C)NC(=O)Cc2ncccc2C)C1)C(C)O N1(C(COCCOCC#C)=O)CC2CCC1CN2C(c1cc(C)c(C)cn1)=O c1(C(=O)NC2C(CC=C)C(OC(C)(C)C)C2)cccc(C2CCCC2)c1 CCC(C)(C(=O)NCC(CC(C)C)NC(c1ccc(C(F)(F)F)s1)=O)OC c1(N(C2CCC(NC(C(CCCC)NC(N)=O)=O)CC2)C)cc(C#N)nc(C)n1 Cc1ccc(C(O)CNC(c2cccc(N)c2)=O)cc1 CCC(C#N)(CC)C(=O)NC1CS(=O)(=O)CC1NC(=O)CC=O.C1CC1.N N1(c2c(C(=O)OC)nccn2)CCC(NC(=O)CC2OCCC2C)C(F)C1 C1(c2n(-c3cnc(C)s3)nc(Cc3cccnc3)n2)CCCCN(C)C1=O C(c1ccc(F)cc1)=CC(=O)N(C(c1ccc(F)cc1)CC(=O)O)C1COC1 C1(C(=O)NCCOCCCNC(c2cnc(SC)s2)=O)CCC2CC1CO2 Cc1cc(C(=O)NC2CCOCC2NC(C2CC23CCC3)=O)ncc1S(N)(=O)=O Cc1nnc2n1CC(C(=O)N(C)CCN(C)Cc1nnc(-c3ccccc3)s1)CC2 c1(NC(CNC(C(COC)O)=O)(C)Cn2cccn2)ncc(Br)c(C)n1 C1(C(=O)NC(C2CN(C(COCCCOC)=O)C2)C)CCC(=O)CC1(C)C CCCCCCC(C)NC(=O)Nn1ncc(C(C2CC2)C2CC2)c1 c1(N(C2CCC(SC)C2)C)[nH]c(=NCc2nccn2C(C)C)nc2scnc12 c1(C(=O)NC(C(=O)NC(C#C)C2CC2)c2ccoc2)cc(C)[nH]n1 C(=O)(CCCCC(N)=O)NC(C)C(C)NC(=O)CCCCCC#N [SH](=O)(=O)c1cc([N+](=O)[O-])c(C)c([N+](=O)[O-])c1C.c1(C(COC)N)cnn(C)c1 c1(SC)nc(C)cc(=NC2CN(C(c3cc(C4CC4)nn3C)=O)CC23CCC3)[nH]1 CC1CN(C)C(=O)CN1C(=O)CC1CCCC1NC(c1ccon1)=O c1(C=O)cccc(P(C)(C)=O)n1.C(C(C)(C)C)NC(CNC(=O)OC)=O c1(C(=O)NCCOCCNC(c2ccsc2)=O)c[nH]nc1OCCF Cc1ccc(F)c(O)c1C(N1CC(C(C)NC(=O)CN2CCC(C)C2)C1)=O C#Cc1ccc(C(=O)NCC2CN(C(=O)C=Cc3cn[nH]c3)CC2O)c(F)c1Cl CCCCC(C)CCC(=O)N1CCOC(CNC(c2cc(F)c(C)c(F)c2)=O)C1 C12(C(N(CCC)CC)=O)CC3CC(CC1C3)C2.c1(C=O)cc2n(n1)CCO2.N C1(NC(CC2(C)CC2(Cl)Cl)=O)CN(C(c2ccc(N)cc2Cl)=O)CC2(CCC2)C1 C(c1cccc([N+](=O)[O-])c1)=CC(N1CC2N(C(CC3CC(C)C3)=O)C(CC2)C1)=O C(=O)(CCCCC(=O)N1CC2CC1C2C(=O)Nc1ccnc(C)n1)OC C#CCC(C)(C(=O)NCC1(SCC)CC1)NC(c1cc(C)cc(O)n1)=O c1(C(N(C2CCN(C(CCCOCCC)=O)CC2)C)=O)cc(C)cc(Cl)c1 c1(C(=O)NCC(C)N(C(c2c(CC)con2)=O)CC)cccc(Cl)c1 c1(C(=O)NCC2CCN(C(c3cccnc3Cl)=O)C2)cnc2ccc(F)cn12 N1(C(C2C(C)C2)=O)C(CNC(C2CCC3C(C2)C3(F)F)=O)CC2COCC12 C#CC12CCCC1(F)CN(CCNC(N1CCn3nc(C4CC4)cc3C1)=O)C2 C1(C)(CNC(CC2COCC(C)O2)=O)CCN(C(C2(c3cccs3)CC2)=O)CC1 c1(SCCC)ccc(C(=O)NCCCCC(C)NC(c2ccc(F)cc2)=O)cc1 CN1CCC2CCN(C(=O)NC3CCCC(OCCN(C)C)C3)C2C1 N1(C(=O)CCCc2cccnc2)CCC2CCN(C(c3ccc(O)cn3)=O)C2C1 N1(C(COCC)=O)CC23CCCC2(C1)CN(C(c1cc2n(n1)CCCCO2)=O)C3 Cc1nc(CC(=O)NCC2CC(F)CN2C(c2ccc(C3CC3)o2)=O)c(C)s1 c1(C=O)coc(C#N)c1.c1(CC)ccc(F)cc1.C1(CCOC)(C=O)CC1.N c1(C(N2CCC(N(C(c3cc(Cl)nc(=N)[nH]3)=O)CC)C2)=O)cccc2cnnn12 CN1CCN(C(=O)COC2CCOCC2)C(C)C1.c1(CC(=O)N)cccc(Cl)c1 C1(CC)(NC(c2cc([N+](=O)[O-])c[nH]2)=O)CCN(C(=O)CC2CCOC2C)CC1 c1(C(=O)NCC(CC)NC(=O)C)ccc(S(C)(=O)=O)c(C)c1.C(C)C.O CCCCCC=CCC(=O)N(CC(CC)NC(C1(C(N)=O)CC1)=O)CC N1(C(c2c(OC)ccnc2)=O)CCN(C(=O)C(c2ccccc2)F)CC(C)C1 CCC(C)(O)C(=O)N1CCN(CCNC(c2cn(C)nc2C(=O)OC)=O)CC1 Cc1c(F)cccc1S(=O)(=O)N1CCC2C1CCCN2C(c1ccc(S)cc1)=O C(C(CC(C)C)C(=O)N1CCOCC1CCO)NC(C1(OC)CCCOC1)=O Cc1cccc(C)c1CC(=O)NC12COC(CNC(C3(Cl)CC3)=O)(C1)C2 c1(C(N(CC(C2CC2)OC)C)=O)cn(CCCCN)nn1 c1(C(N2CC(CO)C(c3cncn3C)C2)C(=O)NC)ccnc(Br)c1 C(=O)(C(C)(C)CC(F)(F)F)NCC1N(C(c2nn(C)c(F)c2)=O)CC(F)C1 C=CCCCC(=O)NC(CO)C(=O)NCC1COCC(C)O1 C1(CC(=O)NCC(C)(F)CNC(C2CC23CC3)=O)CCCCCCC1 CCCCCC(CC)C(=O)NCCCC(C)NC(=O)Cc1c(OC)cccc1Cl CC(C(=O)NCc1ccc(C(C)NC(c2cncnc2)=O)cc1)C(F)(F)F N(C(=NCC(=O)NC1CCCCC1)NCC)CC1(CC)CCCC1.C1(C)CCCC1 c1(C(=O)NCC2CC2c2cncs2)ccc(=O)n2c1CCCC2 CCCC(C(=O)OC)C(=O)N1CCC(F)(C(N2CC(C(=O)N(C)C)C2)=O)C1 n1(CC(N2CC(CC(C)NC(CC(=C)Br)=O)C2)=O)nc(C)nc1C C1(C(=O)OC)C(C)CCCN1C(c1cn(C)cn1)C(=O)NC(C)(C)C CCCCCCC(CC)C(=O)N1CC(NC(c2n[nH]c(C)c2Cl)=O)C(SC)C1 Cc1ccc(C2CCCN2Cc2cnnn2-c2ccccc2)cc1 C1(C(N2CCC3(CCC3)C2)=O)COc2ccc(F)cc2C1.CS(=O)(=O)SCC=O.N c1(NC)nc(C)ccc1C(N1CCC2(CC2NC(C2CC(C)CO2)=O)C1)=O c1(C(=O)NCC2N(C(C3CN(C(N)=O)C3)=O)CC2)c(F)cccc1Cl CC1CCC(C(N)=O)CN1C(=O)C(=O)NC1CCN(Cc2ccccn2)CC1C Cc1ccc(C(=O)N(C)CC2CCCN2C(=O)C(O)CCC(C)C)c([N+](=O)[O-])c1 c1(C(N2CC3(C(C(=O)Nc4c(CC)cccc4Br)C3)C2)=O)cc(Cl)c(Br)cc1Cl N1(C(C2CCCN(CCC)C2)=O)CCC(CNC(c2cnn(CC)c2)=O)C(C)C1 n1(CCC(=O)N)nc(O)c2c1CCCC2.CC(C(=O)NC1CC(C)C1)C1CCC1 C1(C=O)C(O)CCN1C=O.CN1CC(C(=O)N(C2CCC2)C)C1.C(C)(C)C CC1=C(C)CC(C)(C(=O)NC2CCN(C(c3ccc(N)c(Br)n3)=O)C2)CC1 C1(C)(C=O)CCC(=O)N(C)C1.CCCCCCNC(=O)CSc1ccccc1.N c1(C(=O)N)ccc2nn(C)cc2c1.c1(CC)cccnc1C(=O)NCC1CC1 c1(N(CC(C)NC(c2c(CC)c[nH]c2)=O)C)ncnc2sccc12 C=Cc1cncc(C(N2CCCC2c2nc(C)co2)=O)c1 C1(C)(NC(C=Cc2ncc(C)[nH]2)=O)CCCN(C(C2CC2C(F)(F)F)=O)C1 C1(CNC(C(C)OC2CCOC2)=O)CN(C(C2CCCO2)=O)CC12CCC2 n1(COC)ncc(C)c1C(c1nnnn1C1CC1)NC1(C)CC2CCC1C2 c1(C=O)ccc(S(N)(=O)=O)cc1.c1ncc(C(=O)N(CC)C(C)C)[nH]1.CC c1(CN(C(=O)NC(C#C)CC(C)C)C)nc(O)c2ccccc2n1 c1(C(=O)NCCCC)conc1CNC(C1CCCO1)=O C1(NC(C(=O)N(CC(C(C)C)OC)C)=O)CCOC2(CCSC2)C1 c1(C(C2CCN(C(c3ccc(F)cc3)=O)C2)=O)ccc(Cl)cc1 C1(C)(CCNC(C(c2ccn(C)c2)C)=O)CCN(C(c2ccnn2C)=O)C1 Cc1cccc(F)c1.c1(CNC(COCCN=[N+]=[N-])=O)ncoc1C1CN(C)C1 C=C(F)C1(CC(N2CCN(CCNC(c3c[nH]nc3Br)=O)CC2)=O)CCC1 C=CCC(F)(F)C(=O)NCc1csc(C(=O)NC(C)CC(N)=O)c1 C=C1CCN(C(=O)NCCCC(=O)N(C)C)C(C(=O)OC)C1 c1(CC(=O)NC(C)CN(C)C(C2CC23CCOCC3)=O)ccc2ccccc2c1 c1(CN(C)Cc2cc(Br)c[nH]c2=N)ccc(F)cc1Cl c1(CNC(N(C2CCCSC2)C)=O)ccc(O)c(Br)c1 c1(C(=O)N(c2ncncc2Br)c2cnn(C3CNC3)c2)ccc(O)c(O)c1O C1(COC)CCOCC1.N1(C(CN(C(=O)CC2CC2)CCN)=O)CCC1 CC(C(C)C(=O)NC1(CNC(c2cc(Br)n(C)c2)=O)CC1)C1CCCCC1 c1(C(=O)N)nn(C)cc1S(N)(=O)=O.C1(NC(C(CC=C)C)=O)CC(F)(F)CC1 S(=O)(=O)(c1ccccc1N)OCC(=O)NC(c1ccc(CC)cc1)(C)C N1(C(COC(CC)C)=O)CC(C(=O)NCC23CC(CO2)C3)C(C)(C)C1.C N1(C(CN(CCC)C)=O)CCC(CO)(NC(=O)C(F)n2ccnc2)C1 C1(C(N2CCCC(C(C)(C)O)C2)=O)C2CCCC2CN1C(C1CC=CC(O)C1)=O C1(NC(c2nc(OCC)sn2)=O)CC(C)CN(C(c2c(C)csc2Cl)=O)C1 C1(NC(C(NOC)=O)=O)CC2CCC1(C(N1CC(C)(C)C1C(=O)OC)=O)C2 N1(CC)CCCOC(CNC(=O)CNC(=O)Cc2cnn(C)n2)C1 Cc1cnoc1C(=O)NCC(C1CCCN1C(=O)C)(C)C.C(C)(C)C.C=O N1(C(C2(C)CC2)=O)CCOC2(CCC(NC(=O)Cn3ncc(O)nc3=O)CC2)C1 CC(CC(C)(C)C)C(=O)NC(CO)C(=O)NC(CO)CCCO C1(CCNC(c2nc(C(C)C)oc2)=O)COCCN1C(c1cnn[nH]1)=O CCCCC(CNc1nccc(OCC)n1)NC(c1cncnc1)=O C(=O)(CC(C)(C)CNC(=O)C(F)CC1CCOC1)NC(C1CCCCC1)CC CC1CCC=C1C(=O)NCC1CCC(NC(c2cccc(CCO)c2)=O)C1 C(=O)(C(CCNC1C(C)C1(C)C)c1ncco1)OCC C(=O)(C(C)(O)C(C)C)NCC(CC)(CC)NC(=O)C=Cc1ccc(Br)o1 CCCCCCN(C(=O)CC1(C)CC1)CCC.C(C(C)(C)C)NC(=O)CO.S C1(C(=O)NC(C(C)NC(c2cnc(C(F)F)s2)=O)(C)C)CC2(CC2)CN1C CC1CCC(C(=O)NC2CC(O)C(F)C2)N1C(=O)C(=C1CCCCC1)F c1(C(N2C(CNC(C(C)(C)C3CC3)=O)CCC2)=O)ccc([N+](=O)[O-])cc1Cl C12(C(=O)NC(C(N3CC(CCC#C)C3)=O)c3ccoc3)CC(C#N)(C1)C2 CCN=c1[nH]c(C(=O)NCC2CC2C)cs1.c1c(F)cccc1F.C(=O)C.N N1(C(c2c(C)ccs2)=O)CCCC(C2(NC(c3ccc(Cl)nn3)=O)CC2)C1 CC(O)CCNC(=O)CSCCNC(=O)N(C)C C(CNC(=O)CCC1CCCN1C)(CC(F)(F)F)NC(CCn1ncc(C)c1)=O O=C(N1CC(n2cc(C3CC3)nn2)CO1)c1cc(-c2ccncc2)nnc1O C1(NC(C2CC3(CCC3)CO2)=O)CC2CC1CN(C(c1ccc(Cl)s1)=O)C2 c1(NC(C2N(C(CCc3cccc(OC)c3)=O)CC(C)C2)=O)nc(Br)cnc1Cl C(=O)(CCCCN=[N+]=[N-])N1C2(C(=O)NC(CSC)C)CC2CC1 N1(CCOCCOC)CCCCCC1NCC1=CCOCC1 N1(CCC(C)C)C(=S)NC(c2ccnc(Cl)c2Br)C2=C1CC(C)(C)CNC2=O c1(CC)ncc(C(=O)NCCC2CCC(NC(=O)C3=CCC3)C2)s1 C1(C)(CC)C=C(C(=O)NCC(C)(O)CNC(=O)C)C1.c1ccccc1Cl.N c1(C(=O)OCC)ccc(C(=O)NCC(C)NC(=O)C(CC)SC)nc1 C1(C(=O)NC2C(CNC(=O)CCc3ccoc3)CCC2)CC2OC1C1CC21 CC1(C)CCCC(CC(=O)NC2(CCNC(=O)C(F)(F)CO)CC2)O1 C(=O)(CCC(=O)NCCCNC(C1C2CC(=O)CC12)=O)NC C1CC2(CC2)CN1C(C1CC1(F)F)=O.c1(C(C)C)noc(CCCC(=O)NC)n1 c1(SC)cc(C(=O)NC2CCC(Cn3cc(CC(CO)CO)nn3)C2)ccn1 N1(C(CSCCCC)=O)CCC2(CNC(c3nocc3CC)=O)CCCCC12 n1(CCC)nc(C)c(C(=O)NCCC2CCCC2)c1C.C(=O)C(C)C1CCC1.N c1(C(=O)Nc2c(C(=O)OC)cc(CN)s2)c(-c2ccccc2)nc2n1CCCC2 Cc1ncc(NC(=O)C(c2ccoc2)NC(c2cc(Cl)cs2)=O)c(C)n1 N1(C(CCC=C=C)=O)CCN(C(c2cc(OC)cc(F)c2)=O)CC1CC Cn1nc(C(=O)NCC(C)(CO)NC(=O)CCC(C)(F)F)c(Cl)c1Cl c1(C(=O)Nc2cc(C(=O)OC)c(Br)cc2F)c(O)nc(C)c([N+](=O)[O-])c1C C(=O)(CCOC)NC1CC(CCNC(C(C)OCCOCC)=O)C1 c1(-c2c(Cl)ccc(OCC(=O)OC)c2)cc(N=c2cc[nH]c(C#N)n2)ccc1C c1(CC(N2C(CNC(C(COC)(C)O)=O)CC(O)C2)=O)csc2ccccc12 c1(C(=O)OCC)c(Cl)cc(NC(c2ccc(Cl)c(C(F)(F)F)c2)=O)cc1Cl c1(C(N2CCN(C(c3c(C)cccc3Cl)=O)CC2)=O)sc2ncccc2c1N Cc1cc(CNC(=O)CC2CCC(NC(C3CC3C)=O)CC2)ccc1F N1(C(C23CC(OC)C2C3)=O)CC=CC(NC(=O)CP(C)(C)=O)C1 C(=O)(C(C)C(O)C(C)C)NCC(CNC(c1cc(N)cnc1C)=O)OC c1(C(c2cn(C(C)C(=O)NCc3ccccn3)nn2)O)ccccc1OC(F)F N1(C(COCCNC(C2(CC=C)CCCC2)=O)=O)CCCC2CC12 C=C=CCCC(=O)NCC(CC)NC(c1cn(C(C)C)cc1C)=O O=C(C=C(Cl)Cl)N1CCC(N(C(=O)CCCC2CCCO2)CC2CC2)C1 c1(C(=O)NC2CN(C(C3(CC4CC4)CCCO3)=O)CC2O)cc2n(n1)CCO2 O=C(CC(C(F)F)NC(=O)CN1CCOC1=O)NCC(O)CCO n1(CC(=O)NCC2C(NC(C(CC)O)=O)C2)cnc2c1CCCC2 c1(C(N2C(C)CN(C(C3CCCO3)=O)CC2)=O)c(N)c(F)cc(F)c1F CC(C)(CC(=O)N1CCCCC1C1(NC(=O)COCP(C)(C)=O)CC1)CC(F)F C=CCC(C(=O)NCC(c1ccc(C)cc1)NC(c1n[nH]c(C)n1)=O)C(C)C C1C2CC1N(C(c1n[nH]c(C)c1C(F)(F)F)=O)C2.n1(CC)ncnc1C=O.N C(=O)CCc1cnc[nH]1.CC(C=CC(=O)NCC)OC.C(C)(C)C.C=O c1(CC(N2CCN(C(c3ncn(C)c3)=O)CC2CCO)=O)ccc2c(c1)CCO2 c1(CC)cc(C(N2CC(C)C(C)C2)=O)oc1.C1(CC=O)C(C)(C)C1(C)C C1(CNC(C2(C)CC2)=O)CCCN(C(c2[nH]nnc2C(F)F)=O)C1 c1(CNC(C(=O)NCC(C2CCOC2)N)=O)cnc(C2OCCO2)s1 C#CC1(C(=O)NC(CN(C)C)CCO)CN(C(C2CC2(C)C(C)C)=O)C1 N1(C(c2c(C)noc2C2CC2)=O)CC2CN(C(=O)C=C3CCCCC3)CC2C1 c1(N2CCN(c3c(C(=O)OCC)cc(Cl)nn3)CC2)nc2c(cc1C#N)CCC2 N1(C(c2c(C)nns2)=O)CCC(CCN(C2CCCNC2=O)C)CC1 N1(C(C(=O)Nc2ccc(Cl)cc2F)c2ncco2)CCCC(C2CCCC2)C1 C1(NC(CN(C(C2CCO2)=O)CC)=O)CCC(F)(F)C1 Cc1c(NCc2ccc(C3CCC3)cc2)ccnc1F c1(C(=O)NC2CN(C(C3(C)CCCS3)=O)CC(O)C2)cc2c(s1)CCSC2 N1(C(C(CC)C)=O)CCC(CCC2CCCN(C(=O)CCCc3cc[nH]n3)C2)CC1 N1(C(C2(CCOCC)CCC2)=O)CC(O)(C)C1.C1(C)(C=O)CC(F)C1 C1(NC(C(CC)n2cccn2)=O)CC2(C1)CC2NC(c1nc(Cl)cs1)=O CC1CCC(CC(=O)NCc2cccc(C(=O)NC)n2)CC1.C1C(C)C1(F)F C1(NC(C2(C)CC(NC(c3n[nH]c(C)c3C)=O)C2)=O)CCCCC1N=[N+]=[N-] c1(CN(C)CC2CN(C(c3ccc(NC)cc3)=O)C2)ccc(Cl)nc1C Cc1cc(CC(N2CCN(C(C3CCCOC3)=O)CC2C2CC2)=O)ccc1Cl N1(C(c2ccc(CC)cn2)=O)C2CCC1CC(NC(c1ncc(CC)s1)=O)C2 N1(C(c2c(C)nc[nH]2)=O)CC2CCN(C(=O)CC(C)(C)O)C2C1 C1(NC(=O)CC2CCC2)CC(F)CN(C(=O)CCCCN2CCCC2)C1 N1(C(c2cc(C)sc2)=O)CC(C2CCCN(C(C3CCn4ncnc4C3)=O)C2)C1 CCC(C)C(O)C(C)C(=O)NC1CCN(C(=O)C(C)CC2CC2)C12CC2 Cc1ccc(Cl)c(Br)c1CN1CC2CC3CC2C1C3 C(c1ccccc1)=CC(=O)NCC=CCNC(C1CC1(F)Cl)=O N1(C(C=CSC)=O)CC2CCC1C(CNC(=O)CC(O)C(C)C)C2 N1(C(=O)NC(c2ccsc2)C)CCN(c2ccnc(O)c2)CC1 C1(CC)CCCCC1C(N1CC(NC(c2cnccc2C)=O)C(CO)C1)=O C#CC1(CNC(c2ccc(CNC(c3sc(F)cc3C)=O)o2)=O)CCOCC1 N1(C(C(CC=C)(C)C)=O)CC2CCC(C1)C2N(C)C1CC1 c1(NC(C2(O)CCN(C(c3ccc(F)cc3)=O)C2)=O)nc(Cl)cc(Cl)c1[N+](=O)[O-] C(C1=CCSC1)(c1n(CC)nnn1)NCC1(Cl)CC1(F)F N(C(=NCCSC)NCCN(S(=O)(=O)c1cccs1)C)CC(COC)(C)O c1(NC(C2CC(F)CN(C(=O)CN3CCCCC3)C2)=O)cnc2c(c1)CCCC2 C1(CC)CCN(C(=O)C2=CCCCO2)C(C)C1.c1(C(=O)OC)cc(C(=O)N)cs1 c1(C(=O)NCC#CCNC(C2(O)CCC(CC)C2)=O)ccnc2[nH]c(O)nc12 c1(C(=O)NCC2N(C(c3ccc(OC)s3)=O)CC=C2)ccc2ccoc2c1 N1(C(C(C)(C)N=[N+]=[N-])=O)CCC2(CC1)COC(CNC(=O)C(F)(F)CO)C2 Cc1ccnc(C(=O)NCC2CCN(C(C3(Cc4cnn[nH]4)CCC3)=O)C2)c1N CC(C)(C)CC(=O)NCC(F)CNC(c1ccc(C2CCCOC2)cc1)=O c1(NC(C2(SC)CC(=O)C2)=O)ccc(OC(C)(C)C)nc1 N1(C(c2c(CC)onc2)=O)CCN(C(=O)C(C)CC2CC2)CC2(C)CCCC12 n1(CC)cnc(C(=O)N(C2CN(C(c3csc(-c4ccccc4)n3)=O)C2)C)c1 c1(C(=O)NCCCOCCN(C)C(C2CCCN2C=O)=O)ccc(C#N)cc1F Cc1cc(C(=O)N(C)CC2CCN(C(=O)CC3(O)CCCOC3)C2)cc(O)n1 C1(C=O)CCCCCN1C.CC1CCCCN1C(=O)CSCCOCCO Cc1cc(C(=O)N(C2CC(C(=O)N(C3CC4CC4C3)C)C2)C)nn1C C1(O)(C=O)Cc2ccccc2C1.C1(CNC(C2CC=CC2)=O)CC(F)(C)C1 c1(C(N(CC(CO)(CO)NC(C(CCOC)OC)=O)C)=O)c(N)cccc1Cl N1(C(C2C(C=C(C)C)C2(C)C)=O)CCCC(C2CC2)C1.C(=O)C(F)=CC1CC1 C(=O)(C(C)CS(C)(=O)=O)NCC1(OC)CN(C(=O)CCC(C)C)C1 C(=O)(CCCC(=O)OC(C)(C)C)NC1CC(NC(C2C(=C)C2)=O)C1 N1(C(c2c(C)cc(F)cc2)=O)CCC2(CCC2NC(=O)Cc2cscn2)CC1 N1(C(=O)COCc2nc(-c3ccccc3)no2)CCCC(CS)C1.C1CC1(F)F C1(CNC(CCC(C)C)=O)CC2CCC1N(C(=O)CNS(N)(=O)=O)C2 C(C(C)S(C)(=O)=O)NC(C1(C)CC1(F)F)=O.C1(C(=O)N)CC(F)(F)CS1 c1(C(N(CC(CNC(C2C(CCOC)C2)=O)O)C)=O)cccc2c1CCO2 C(=O)(C(C)C=O)N.CC(C)CC.C(=O)C(C)(C)N(C)C.C(C)(C)C.C=O C1(NC(CCSCCC)=O)CC(NC(c2cc[nH]c(=N)c2)=O)C12CCC2 C(C(O)CC(F)(F)F)NC(C1N(C(C2(CSC)CC2)=O)CCC1)=O C1(F)(CNC(CNS(C)(=O)=O)=O)CN(C(=O)C(F)(F)C2CC2)C1 c1(C(N2CCN(C(CC=C)=O)C(C)C2)=O)nc2nc(C)ccn2n1 C(=O)(CCCCNC(=O)C(CNC(C1CC1(Cl)Cl)=O)N(C)C)OC C=C(Cl)C(C)(C)C(=O)N1CCC(O)(CN(C)C(C2CCC(C)(C)C2)=O)C1 c1(CC(=O)NC)cn(C)nc1C(F)(F)F.C(C)C=O.C1CC1.C#CCO C=CCC(CN(CC(CO)OCC)CC1CCC1)C(=O)OCC O=C1C=C2CN(C(C3CN(C(c4cc(Br)cnc4O)=O)CCS3)=O)CCC2S1 C(=O)(C(O)CC(F)(F)F)NCC(C)NC(c1cnoc1-c1ccoc1)=O C(=O)(C(CC)C(=O)NC12CC1CN(C(c1ccc(O)c(Cl)c1)=O)C2)OCC C(C(C)CC(=O)N1CCC(C)(C(=O)NCCNC(=O)C2CC2)C1)OC CC(CCNC(C)(C)C)C(=O)N(C(C)C(=O)N(C)Cc1ccccc1Br)C C12(NC(c3nn(C)nc3Br)c3nnnn3C3COC3)CC1COC2(C)C Cn1cc(C(=O)NC2CCC2)c(C(F)F)n1.C1(C=O)(CCNC=O)CC1.C CCC(C(=O)NC1(C(=O)NCC2(O)CC(O)C2)CC1C)C(C)C N1(CCNC(C(CC)OCC)=O)CCC(NC(c2[nH]ccc2C)=O)CC1 CCC(C)C(C)C(=O)NCC1CN(C(c2nccnc2SC)=O)CCO1 C1(C=O)CN2CCC1CC2.C1(NC(C2(C)CC2C(F)(F)F)=O)CCC(C)CC1 C=CCC(C(=O)N(C)CCOCCC=O)NC(C)=O.C1(CCO)CC=CCC1.N CCCCCC(F)C(=O)NCC1(C)CCCN(C(C2NC(=O)OC2(C)C)=O)C1 c1(OC)cc(OC)c(C(N2CCCCC2C(C)CO)C(=O)NC2CCOC2)cn1 C1(O)(C(=O)NCCN(CCC)C(c2ccc(CO)cc2)=O)CC(C)(C)C1 C(=O)(C1Cc2ccccc21)C(CC1N(C(C2CC(CC(=O)OC)C2)=O)CC1)=O c1(OC(C)C)ccc(C(C)CNC(=O)Nc2ccc(-c3ccccn3)cc2)cc1 C(=O)(CC(C)C)NC(CC)CN(C(C)=O)CC.C(=O)CCCc1ncco1.N C1(CN2CCN(C(C3CN(C(C)=O)C3)=O)CC2)CCC2(C1)NC(=O)NC2=O C(CCC(C)C(=O)NCC1CCCCN(C(=O)Cn2nc(O)ccc2=O)C1)OC N1(C(C(n2c(C)ccn2)C)=O)CC=C(CCNC(=O)CC2CCCOCC2)CC1 c1(C(=O)NC(C)CCN(C)C(C2CCC(=O)O2)=O)cc(F)cc(F)c1 C1(C(=O)NCC2(O)CC(NC(Cc3ncc(C)o3)=O)C2)CCCCC1O c1(C(N2CCN(C(C3C(OCC)C3C)=O)C(C)C2)=O)cnn2ccn(C)c12 CC1=C(C)CC(C)(NC(=O)CC(C)(C)NC(c2cc3occc3[nH]2)=O)CC1 c1(-c2cccc(C(C)=O)c2)ncc(Cl)cc1C(=O)Nc1cc(Br)cnc1C(F)F C1(NC(CC(CC)C2CC2)=O)CCN(C(c2cn(C)c(C)cc2=O)=O)CC1(C)C c1(C(=O)Nc2c(N(C)C)cccc2F)c(Cl)ccc(CO)c1Cl C1(C(N2CCC(CO)C(O)C2)=O)CCN(C(=O)CCc2ccsc2)C12CC2 CC1CCC(C)(C(=O)NOCCO)CC1.n1(CCNC=O)cncc1.C(C)C CC1CN(C(c2ccn(C(F)F)n2)=O)CCC1NC(=O)C.c1(CC)cccs1.O N1(C(c2c(C)csc2)=O)C2COCC1CC(NC(c1cc(C)c(F)cc1F)=O)C2 Cn1cc(C=CC(=O)NC2C=CCN(C(c3n[nH]c(C(C)(C)C)n3)=O)C2)nn1 c1(CC)cnc(C(=O)NC)nc1.C12(CC)CCC(CC1)C2.C1(C=O)CCCO1 Cc1cc(CN(CC(C)C)Cc2nn[nH]c2-c2ccnn2C)ccc1Br C1(CC(N2CCC3(CCC3)C2)=O)C2CCCC2N1C(C1CCC2CC12)=O C(c1cccc(O)c1)=CC(N1C(C(=O)Nc2cccc(C(C)=O)c2)CC1)=O C12(CC(=O)NC(C(C)(C)C)CNC(c3cccnc3)=O)CCCCC1C2(F)F Cc1cc(C(=O)N(C(C(N2CCC(n3ccnc3)C2)=O)C2CC2)C)[nH]c1C c1(C=O)c[nH]nc1C1CCOC1.c1(OCC(=O)NCC(=O)N)ccsc1.CC C12(OC)CCC(C(=O)NC3(C)CCCCC3C)(CC1)C2.c1(C=O)cnn(C)c1 N1(CC)CCCC(C(N2CCSCC2C(=O)NOC(c2ccccn2)C)=O)C1 Cc1nc2c(CCC(=O)NCCN3CCN(C(=O)C(C)C#N)CC3)cccc2o1 C(=O)(C(F)(F)C(C)O)N1CC2C(CNC(CSc3c(C)n[nH]c3C)=O)(C2)C1 C(=O)(C1=CC(O)C(NC(=O)CC(C)n2ccnc2)C1)NCCOCC c1(C(N2CCC(Br)C2)=O)nc2ccc(-c3cnn(CC4OCCO4)c3)cc2s1 c1(C(=O)NC2CN(C(C3N(C(C)C)CCC3)=O)C2)cc(Cl)ncc1N C(=O)(CCN(C(C(=O)NCC1CCOC1)c1ccsn1)C)OCC C1(NC(c2n(C)ccc2)=O)CN(C(c2cn[nH]c2)=O)CC1c1ccccc1 CC1CCCN(C(=O)CN2CCCNC2=O)C1CNC(c1ccnn1CC#N)=O Cc1ccc2c(C(N3CC4CC(C3)N(C(=O)Cc3ccnn3C)C4)=O)coc2c1 c1(C(=O)NC2CCN(C(=O)CCc3cc[nH]n3)C23CC3)cc2nccn2c(O)n1 N1(C(c2n(C)ccn2)=O)CCC(C)(C)C(CNC(c2cc3n(n2)CCCC3)=O)C1 C(=O)(CC(C)CC(C)(C)C)N(CC(CC)NC(c1cc(C#N)no1)=O)CC CCC(CC(=O)N1CCN(CC(O)COc2ccc(C)cc2)CC1C)C(C)C C=CCC(C)(C)C(=O)NC1CC(NC(=O)C(C)(C)c2cnsc2)C1 c1(C(=O)NC2C(C)(C)CN(C(C3CCCOCC3)=O)C2)nc2c(s1)COCC2 C1(NC(C(CCOC)OC)=O)C(C(=O)OC)C2CCCCC12 C(C#Cc1cnn(C)c1)NC(C1CCN(C(c2c(C)nc(C)o2)=O)C1C(C)C)=O C1(n2cc(C3(OC)COC3)nn2)COC2(CCC2)C1OC(C)C N1(C(CSCC)=O)CCCCC1C1CCCN1C(c1ccsc1C#N)=O C=CC1(C=C)COCCN1C(c1ccc(Cl)c(Cl)c1C)C(=O)NC(C)CC c1(C(N2CC3CC(NC(=O)CCc4cccs4)C3C2)=O)ccc2cc[nH]c2n1 c1(CC(=O)NC(C)CNC(=O)CC(C)N2CCCC2=O)c[nH]c2cc(Cl)ccc12 C1(C(N(CCN(C)C(C2CC2(F)Cl)=O)C)=O)(NC(N)=O)CCCCC1 c1(C(=O)NC2CCC(N(C(c3noc(CC)c3C)=O)C)C2)cnn2c1CCC2 C1(C(=O)NCCCN(CCO)C(C2CC(F)C(=O)N2)=O)CC12CCCCCC2 C(=O)(C(C)(O)CNC(C1CCCCC1)=O)OC.C1(C=O)CN(C(N)=O)C1 c1(C(=O)NCC(CCCC)NC(c2ccoc2)=O)ccc(F)cc1F C(=O)(CN=c1ccc(C#N)c[nH]1)NCCCC(C)NC(C1(C)CCC1)=O N1(C(CCC(CC)=O)=O)CCOC2CN(C(=O)CCN(C)CCO)CC12 c1(OC)cccc(C2(C(=O)NCCCCCNC(C3CCOC3)=O)CCCC2)c1 CCCC(C)(CC)C(=O)NCC1C2CN(C(c3ccnn3C)=O)CC12 c1(C(N2CC(C)C(NC(=O)Cc3ccon3)C(C)C2)=O)oc2ccccc2c1Cl C=CCC(C)(C(=O)N1CCN(C(=O)Cc2csnn2)C(CCO)C1)N(C)C C(=O)(C(C)C(O)CC(C)C)NC(CC(=C)Cl)C(=O)NCc1c(C)cnn1C CC1CCC(C(N2CCCC2CN(C)Cc2sccc2Br)=O)CC1C CCCC(C)CCCC(=O)N1CCN(C(C2CC(N(C)C)C2)=O)C(CC)C1 C12(NC(CN(C)CC)=O)CC1CN(C(c1cnccc1Br)=O)C2 Cc1csc(CCC(=O)N2CCC2CNC(=O)C=CC(C)C)c1 c1(NC(c2ccc(C3CC3)cc2)C)cc(OCC(F)(F)F)ncn1 C1(C)(CC)C=C(C(=O)NCC2(C)CN(C(c3cn(C)nn3)=O)CC2C)C1 n1(CC(=O)Nc2scc(C(N)=O)n2)c(=O)cnc2ccccc12 c1(C(=O)N)ccnnc1.c1(CCC(=O)NCC(C)OC)cccnc1.C1CC1 c1(-c2c(C#N)scc2)nc2c(s1)CC(C(=O)NCc1cc(Br)cnc1F)CC2 c1(C(N2C(CNC(C(c3ccccc3Cl)C)=O)CCC2)=O)nccc(Cl)c1F c1(CCC(=O)N(C)CCNC(=O)Cc2cnccn2)ccccc1Br C#CC(C)(C)C(=O)NC1CCCC(NC(C2COCCN2CC)=O)C1 C1(NC(COCCC=C)=O)CN(C(c2cc(N3CCCC3)ccn2)=O)CC1C C1(CCNC(C(C)N(C)C)=O)CCCN(C(c2cc(C3CCC3)[nH]n2)=O)C1 n1(-c2c(C)ccs2)nc(C(N2CC3C(Br)C3C2)=O)c(O)cc1=O C#Cc1c[nH]nc1C(=O)NCc1ocnc1C(=O)NC(c1cccnc1)C c1(C(C)C)ccc(C(CNC(=O)C=C(Cl)Cl)NC(=O)CC(F)(F)Cl)cc1 Cc1ccc2c(C(=O)NCC3CN(C(=O)C(C)(O)C(F)(F)F)C3)csc2c1 c1(C(C(=O)NC2CC(F)(F)C2)N(CC(C)C#N)C)cc(F)cc(I)c1 c1(C(N(CC(=O)NC(C)CCSCC)CCC)=O)cncn1C1CC1 c1(C(N2C(CNC(C(C(C(C)C)O)C)=O)CC2)=O)cc(F)c(F)c(F)c1N CC1CC(C(=O)NCCOC2CCCC2)CN(C(=O)CC2CCCC(=O)C2)C1 c1(OC)cc(C(C)NC(=O)NCC2CCCC2)ccc1SC C(=O)(CCCCC(=O)NCC1CCCN(C(=O)CCc2cnoc2)C1)NC Cc1sc(C(=O)NC(C2CN(C(c3cscn3)=O)CCO2)C)cc1Br c1(-c2scc(C(N3C(c4n(C)cnn4)CCC3)=O)n2)ccc(Cl)cc1Cl Cc1cnc(C(=O)NC2CCCC2NC(c2occc2C2CC2)=O)c(C)c1 C(=O)(C(C)(C)C(=O)N1CCCC1(C)C(=O)NCC1(C)CNC(=O)O1)NC C1(N(C(CCC#C)=O)C)CCCCN(C(c2ccc(O)c(C(C)=O)c2)=O)C1 c1(C(N2C3CN(C(C(C=C)(C)O)=O)CC2CC3)=O)ccc2c(=O)ccoc2c1 Cc1coc(C)c1C(=O)NC1CCC(NC(C2CCCC(CF)C2)=O)CC1 C1(CNC(CCC)=O)CCCN1N(C)Cc1ccc(OC)cc1 n1(CC(C)NC(=O)N(C2CCCCC2)c2ccco2)cnnc1O CC(C)CC(C)C(=O)N1CCC(C)(CNC(c2ccnc(Cl)c2)=O)C1 c1(C(=O)NC2CC(C)CN(C(=O)C(C)(C)N(C)C)C2)cc2c(s1)CCOC2 c1(C(=O)NC2CCN(C(C3CC(CC)(CC)C3)=O)C2)cccc(F)c1Br Cn1ncc2c(C(N3CC4(CC4)CC3C(=O)NC3CC3)=O)cccc12 c1(C(=O)NC2C=CCN(C(C3(C)CC3)=O)C2)csc2c(O)ccnc12 C(C1CCCN1C(=O)C=CC1CCCC1)=CC(=O)N.CC(C)CCOCC c1(CC)oc(C(=O)NC2CC(NC(=O)C(C)Cc3cnc[nH]3)C(O)C2)cc1C C1(NC(c2c(C)nn[nH]2)=O)CCOCC1NC(c1ccc(F)cn1)=O C#CCC(C(=O)NCc1ccccc1CC)NC(=O)CC(C)C1CC1 N1(C(c2ccc(OC)c(F)c2)C(=O)NCC(=C)C)CCC2(CCC(O)CC2)C1 C(C(O)C(=O)N1CC(CC(C)NC(c2conc2C2CCCC2)=O)C1)=CC Cc1[nH]c2ncccc2c1C(=O)NCC1CCC(NC(=O)CCc2cnco2)C1 C1(CNC(C2(OC)CCSC2)=O)CCCCC1NC(c1cccnc1CO)=O c1(C(=O)NCC2(F)CC(NC(C34CC(C)(C3)C4)=O)C2)ccccc1F c1(CN2CC3N(C(C(C)(C)Cc4ccccc4)=O)C3C2)cc(Br)ncc1F C1(CNC(=O)Cc2cnoc2)CN(C(=O)CCCCF)CCC12CCOC2 C1(OC)CC2CC(C(C(=O)NC(C)C)N(C)Cc3ccccc3Cl)CC12 C1(N(C(COC(C)C)=O)C)CCCN(C(c2cccc(C3(C)CC3)c2)=O)C1 N1(C(c2cc(C)no2)=O)CCCC2C1CCN2C(=O)Cc1nc2ncccn2n1 c1(C(=O)NCC(CNC(C(C)c2ncco2)=O)O)cn(CCCF)nn1 c1(C(CCCNC2C(C)(CN)CCCC2)=O)ccc2c(c1)CCC(=O)N2 C1(CCC)CN(C(C2CC(O)C2)=O)CCN1C(=O)C(Cc1ccccc1)C1CC1 N1(C(Cc2c(CC)cccc2)=O)CC2CN(C(=O)C(COC)N(C)C)CC2(C)C1 c1(C(N2CCC(C(C(C)C)NC(=O)CCC3CC3)CC2)=O)cc2ccccn2n1 C(=O)(C1=CC2CCCC12)N1C(C)CC(NC(c2cncnc2C2CC2)=O)C1 c1(C(C)C)ccc(C#N)c(NC(C)CO)n1.c1(CC=O)ccc(C(N)=O)nc1.N C1(NC(C2CCC(C(C)C)CC2)=O)CC2CC1N(C(c1ccoc1C1CC1)=O)C2 C(CC(=O)NCC(C)CNC(=O)Cc1ccc(O)nc1)(C(C)C)OCC Cc1cc(Cl)c(C(N2CCCC(CNC(c3cscn3)=O)CC2)=O)cc1F Cn1cc(F)c(C2CN(C(=O)N(C3CCCC3)Cc3ccco3)C2)n1 N1(C(C(C2CCN(C(c3cncc(CC)c3)=O)CC2)C)=O)CCC(O)C(F)(F)C1 C1(NC(C(CN(C(C(C(C)C)C)=O)C)(C)C)=O)CCC(C2CC2)C1 C(=O)(CCCCCCCCC1CC1)NCC1C2N(C(CCCOC)=O)C(CC2)C1 N1(C(Cn2c(C)ccc2C)=O)CCOCC(NC(=O)C=CCn2cncn2)C1 c1(N(CCNC(C2CCOC2)=O)CC)c(C#N)cccc1[N+](=O)[O-].C(C)C.O c1(C(N(CC(C)(C)CNC(=O)CC2CC=CC2)C)=O)cc2cccn2cn1 C1(N(C)C(C2CCCC2CNC(=O)CCCn2cccc2)=O)CCCOC1 C1(N(C(=O)NC2C(c3c(C)ccs3)C2)CC2CC2)Cc2ccc(F)cc2C1 C1(NC(=O)C=CCc2cccs2)COC2(CCN(Cc3n[nH]cc3Cl)CC2)C1 N1(C(c2c(C(C)C)cco2)=O)CC2(C=C(C(=O)NC)CO2)C1.c1nccc(O)n1 Cc1ccc(SCC(=O)NC(C2CCN(C(c3ccnnc3S)=O)C2)C)cc1C c1(C(=O)NCC2C(NC(=O)CSc3cccs3)CCC2)cccc2nncn12 C(CCC(CCC)NC(C1CCC(C)(C)CO1)=O)NC(CC=C)=O N1(C(c2cscc2F)=O)CCC2(CCCN2C(c2cc(C3CC3)ncn2)=O)CC1 C1(NC(CN(C(=O)OCC)C)=O)CCOCC1NC(=O)C(C)C1CCC1 C(=O)(C(F)(F)C(F)(F)C(F)F)N1CCN(C=O)CC12CCC2.C1(C2CC2)CCC1 c1(C(=O)N)cccc(C)c1[N+](=O)[O-].N1(C(COCC=C)=O)CCCC(O)(CC)C1 Cc1cc(=O)c(C(=O)N(CC(C)NC(c2c[nH][nH]c2=N)=O)C)cn1C C12(NC(CC=CC=C)=O)CCCCC1N(C(c1cc(N(C)C)nc(Cl)c1)=O)CC2 Cc1ccc(CN2CCC2(C)C(=O)N(CC#N)CC#N)c([N+](=O)[O-])c1 c1nc2ccccc2cc1F.c1(CN(C2CCC2)C(=O)OC(C)(C)C)ccsc1.N c1(C(CN(CCC)CCNC(=O)C(C)Nc2cccs2)=O)cc(C)ncn1 C(=O)(CCN=c1[nH]c2ccccc2s1)NC(C)C(CO)NC(C1CCNC1=O)=O c1(C(C)=O)c[nH]c(C(N2CC(O)(C(F)C(N3CCC(C(F)(F)F)C3)=O)C2)=O)c1 C1(CC(=O)N(C)CCc2cnc[nH]2)CCN(C(C2CC2C(C)(F)F)=O)CC1 c1(CC(N2CCOCCC2C2CC2)=O)ncc2ccc(Br)cn12 Cc1ccc2c(C(=O)NCC(C)(C)CN(C(=O)CCCC3CC3C)C)n[nH]c2c1 C(=O)(C(C)(C)C(C)C)N1CC(CCNC(=O)CN(C2CCC2)C)(OC)C1 c1(C(=O)NC(CNC(c2c(CCC)[nH]cc2)=O)C)cccc2c1C(=O)NC2 c1(C(=O)NCCC2(NC(=O)CC(=O)NC3CC3)CCCC2)ccc(F)cc1 C(=O)(C1=CS(=O)CCC1)N1CCC(CCNC(C=COCC)=O)C1 C1(NC(c2[nH]cc(CC(C)C)c2)=O)CC2(C1)CC2N=c1[nH]c2ncc(Cl)cc2s1 c1(CNC(C(c2c(CC)noc2)N(CC(C)C)C2CC2)=O)cccc(Cl)c1 Cc1nccc(C(=O)NCc2cn(CC(N3CC4CC(C)C4C3)=O)nn2)c1C CC1(C)CCC(C(=O)N2CCC(CCCO)C2)c2ccccc21 N#Cc1ccc(C(=O)NCC2CCCN(C(=O)Cc3ccno3)C2)cc1O n1(CC(=O)N(CC(=O)NC(COCC)(C)C)CC(C)C)cc(Cl)cn1 C1(C(=O)NC2C(NC(C=C3CCN(C)CC3)=O)COCC2)CCS(=O)(=O)N1C C(=O)(CCCC)NC(C12CC(C1)C2)=O.C=C(CC=O)CC#N.C(C)(C)C C(=O)(C1=CC2(CCOCC2)C1)N1CC2(OCCN(C(C3C(C)(C(C)C)C3)=O)C2)C1 c1(C(C)(F)C(=O)NCCCCNC(c2cn(CC3CC3)nn2)=O)ccccc1F c1(C(c2n(C(CC)C)nnn2)Nc2ccc(F)cc2)cc(Br)cc(F)c1F CC1CCC(Cl)=C(C(=O)NC2CC3CC2CN3C(=O)CN2CC(C)(C)C2)C1 C1(CC)CC(O)CN1C(C1CCOC1CNC(=O)CCCn1ccnn1)=O C(=O)(C(CC(F)F)NC(=O)CCOCC(C)C)NCCCOC C#Cc1cccc(CC(=O)NCC(C)(F)CNC(c2cccc(F)c2)=O)c1 c1(C(c2nnnn2C2CCOCC2)NCc2cc(C)sc2)cc(Br)ncc1F CCCCC(CN=c1nc(CC)[nH]s1)NC(c1c(C)oc(C)c1C)=O CC(C)CCCC(=O)NCC1C(C)CCCN1C(=O)Cc1ccn(C)n1 CN1CC=C(CC(=O)N2CC3CC(NC(=O)CC(C)(C)CC(F)F)C(C3)C2)CC1 C1(C(C(=O)NC)C)CCCN(C(c2ccc(C(=O)OC)o2)=O)C1 C(=O)(C1=CCCC(C)(C)C1)NCC1CC(NC(CC(=C=C)C)=O)C1(C)C N1(C(CCC=C(C)C)=O)CCN(C(c2cccc(Cl)c2C)=O)C(CF)C1 C(CCCNC(C1CN(C(C)C)C1)=O)OC.C1(C=O)CC1C(C)(C)C.N c1(N(C(c2cccc(C3CC3)c2)=O)CC2CCCNC2)ncnc2c(Br)c[nH]c12 C=CC1CN(C(=O)C(CNC(C2CCCN2CCC)=O)CC2CC2)CC1O c1(C(=O)NC2CN(C(C3CC3C(F)F)=O)CC23CC3)cncc2ccc(F)cc12 c1(C(N(CC(=O)N(CC)CC)CCOC)=O)cc2ncccc2[nH]1 N1(C(COC(C)=O)=O)CCCC(C(=O)N(CCCN=[N+]=[N-])C(C)C)C1 CC1CCN(C(C2CCC(C)(C)CC2)=O)CC1NC(=O)C1=CCOCC1 C1(NC(CSCCC)=O)CCN(C(c2sc(C3CC3)nc2C)=O)CC1(C)C C1(NC(c2cc(F)c(F)cc2O)=O)CN(C(=O)Cn2ccnn2)CC(F)(F)C1 C=CCCCC(C)(C)C(=O)NCCSCC(=O)N(C1CC(C(N)=O)C1)C C(=O)(CCCCCCCC(=O)OC)NCCC(C)NC(C(CCC)NC(C)=O)=O n1(CC(=O)NCC(C)(CO)NC(=O)CCc2ccc(Br)cc2)ccccc1=O C1(N(C)C(C2CC3CCC2C3)=O)CC2CCC(C1)N2C(=O)CCc1nncn1C c1(NC(C(CC)Oc2ccc(Br)cn2)=O)c([N+](=O)[O-])c(C)nn1C C1(C=O)CN(C(c2cncc(C)c2)=O)CC1C(C)C.C(=O)C(C)C1CC1.CO C12(NC(CC(C)(C)F)=O)CCCC1N(C(c1cc(Cl)c(Cl)cc1N)=O)CCC2 c1(NC(C(CNC(=NCCOC)NCCOC)(C)C)=O)ccc2c(c1)CC(C)O2 n1(CC(=O)N(CC(C)NC(C2(CF)CCC2)=O)C)ccc(C(F)(F)F)n1 c1(CC(=O)NCCC(=C)CNC(C2CC23CC(O)C3)=O)ccc(O)cn1 c1(CC)cc(C(N2CCC(C)(C)C2)=O)ccc1C.C(=O)(C(CC(C)C)N(C)C)N c1(C(=O)N)cc(Cl)ccc1-n1ccnc1.C(CC(C)(C)C)NC(C1CC(C)C1)=O c1(CC)ccccc1C(=O)NC(C)(C)C1CC1.C1(CC(=O)N)CCOCC1 CC1CC(C)N(C(c2cccn3cnnc23)=O)CCN1C(=O)CC1(C)CCCC1 C=CC1(CC(=O)NC2CC(C)OC2=O)CN(C(C2(CC)CCC2)=O)C1 C12(CNC(C(CSC)(C)C)=O)CCCC1N(C(c1cc(Cl)ccc1F)=O)CCC2 C(=O)(CC(C)NC(=O)C=CCNC(C1CC1[N+](=O)[O-])=O)OCC Cc1cc(C(=O)NCC(C)CC(=O)NCCC2(O)CCOC2)ncn1 C1(NC(c2c(C)cnc(F)c2)=O)CCC2(CC1)CN(C(C1(C)COC1)=O)CCO2 c1(-c2c(OC(C)C)cc(C(F)(F)F)cc2)nc(CO)n2ccccc12 C(CCCCCN(C(=O)CCc1ncc(F)cn1)C)NC(CC1CC(=C)C1)=O C12(CNC(C=CSC)=O)CCCCC1N(C(=O)Cc1ccccn1)CC2 CC(C)CC(C(=O)NCCNC(c1ncn(C)n1)=O)N(C)C.c1ccccc1.C S(=O)(=O)(c1ccc(NCC(N2CCOCC2)=O)cc1)NC(c1nc(O)n[nH]1)C c1(CC(=O)N(C(C)CNC(C2CCC(=O)N2)=O)CC)cc2ccccc2s1 c1(C(C(N2CCC(CNC(C3CS(=O)C3)=O)C2)=O)O)cccc2c1OCC2 Cc1n[nH]c(C)c1CC(=O)NCC1CC(O)CN1C(c1nc(Cl)cs1)=O Cc1cc(C(=O)NC2CN(C(=O)Cc3cnoc3)C3(CCC3)C2)c(N)c(Cl)c1 c1(C(C)=O)oc2cccnc2c1NC(C1CC(NCc2c[nH]ccc2=N)C1)=O CCC(CNC(C1CCC1)=O)(CC)C(=O)NC1CCCOC1 C(=O)(CC(CC)NC(C1CCOC1)=O)N(CCC1CC1)CC C#Cc1cccc(CC(=O)NCCCC(C)(C)NC(C2CCC2(OC)OC)=O)c1 CCCC(C#N)C(=O)N1CCCC1C1(C(=O)N(C)Cc2ccc(C)nc2)CC1 C(=O)(C1=C(CC)OCCS1)NC1(CCC)CCCN(C(C2(C)CCCN2C)=O)C1 C1(C)(C(=O)NC2C(NC(c3cncc(C)c3)=O)CCCC2)CCC12CCC2 N1(C(CCC(=C)C)=O)CC(OC)CC1(C)CNC(c1cnc(COC)[nH]c1=N)=O N1(C(C(c2ccc(O)cc2)C)=O)CCOC(C(=O)NC(CO)C(F)(F)F)C1 N1(C(CN(CC)CC)=O)CC2CCN(C(=O)Cc3cnn(C)c3)CC12 C1(CNC(C(C2CC=CCC2)NC(=O)CC2CCC2)=O)CC2(CC2)C1 CC1CC(NC(c2nc[nH]c2C(C)(C)C)=O)CN(C(=O)Cn2ncccc2=O)C1 C1(N(C(COC(c2noc(-c3ccccc3)n2)C)=O)CCO)CCCC(C)C1 N1(C(C(C)(C)C)=O)CC(NC(=O)CN2CCCCS2(=O)=O)C(C2CC2)C1 N1(C(CC2CC2)=O)CCN(C(=O)CC2CCC2C(F)(F)F)C(C2CC2)C1.C C1(C(=O)NCC2COCCO2)CC2(CCN(Cc3nc(Br)ccc3F)CC2)C1 C1(NC(c2ocnc2C(F)F)=O)CC12CCCCC2.C(=O)(C(F)C(F)(F)F)N Cc1cc([N+](=O)[O-])cnc1C(=O)NC(C)CCCNC(=O)C1=CCCC1C CC1CN(C(c2cncn2C)=O)CC(C)C1NC(c1cnn(CCO)c1N)=O c1(C(N(CC(CN(C(c2n(CC=C)ccc2)=O)C)O)C)=O)n[nH]cc1[N+](=O)[O-] N1(C(C)C(=O)N2CC(CNC(=O)CC3CC3)C2)C(=O)CCC1=O O=C1OCCC1CNC(C1(F)CN(C(C2CS(=O)C2)=O)C1)=O N1(CCC)CCC(C(N2CCC(C)(N(C(=O)C)CC)C2)=O)CC1.CC(C)(C)C c1(C(N2CCC(C(CC)C)CC2)=O)cc(C(=O)O)cc(C(F)F)c1 c1(OCC(=O)NCC(C)CNC(c2cc[nH]n2)=O)ccccc1 Cc1cc(C(=O)N(C)CC2COCCN2C(=O)CCCF)cc2nn[nH]c12 n1(CC)cnc2nc(=NCC=C(Cl)Cl)[nH]c(NCC3CCOC(C)(C)C3)c12 N1(CC(=O)NCC(CNC(C=C2CCC(C)C2)=O)(C)C)CCC(C)(O)C1 CC1COc2ccccc2CN1C(n1c(OC(C)(C)C)ncc1)=O c1(C=O)c(F)cc(N)cc1F.CN1CCC(C(=O)NCCC2(C)CC2)C1=O.N Cc1nc(O)ccc1C(=O)NC1CN(C(c2ccns2)=O)C2CC12 C1(CNC(CCCc2ccc(C)cc2)=O)CN(C(=O)C=CC2CC2)C2(CCC2)C1 CC#CCC(CO)NC(C1(C)CN(C(=O)Cc2cncnc2O)C1)=O c1(C=O)ccc(C)cc1F.C1(C)(C(=O)NCCC(=C)C)CC(OC)(OC)C1.N c1ccn(C)n1.CC(CNCCn1cccn1)C1CC1.C(C)(C)C.C=O.N C(CCCCC(=O)N(CC(CC)NC(=O)C(C)NS(=O)(=O)CCCC)C)=CC N1(C(C(C2(C)CC2)NC(=O)Cn2cccnc2=O)=O)CCC([N+](=O)[O-])CC1 c1(CN(C(=O)CC2CCCCC2O)C)ccc(C)cc1.c1(C=O)cc(Cl)ns1.N N1(C(Cc2cc(C)on2)=O)CCN(Cc2cc(C#N)ccn2)C2CC12 c1(C(=O)NCCN(CC(C)O)C(C2CCOC2)=O)ccc(O)c(Br)c1 c1(C(=O)NCC2(C)CN(C(=O)Cn3ccnc3)C2)cc(Cl)c2cc[nH]c2c1 c1(C=O)c(C)c[nH]c1CC(N)=O.C(C=CC(=O)NC(C)C)(CC)=CC c1(CCC)c(C(=O)NC2CC2NC(C2COCCO2)=O)cnn1C C1(NC(c2ccc(C#C)cc2F)=O)CCC2(CC1)CC(NC(c1ccsc1)=O)C2 c1(CCOCC)ccc(NCc2nnnn2Cc2nncn2C)cc1.CC#N N1(C(C(C=C)(F)F)=O)CCCC(N(C)C(c2cc(C)c(C)o2)=O)CC1 CC1(C)OCC(C(O)CNC(c2ccc(Cn3cc(Cl)cn3)s2)=O)O1 c1(C(=O)NCC(CCCC)NC(c2cccnc2CO)=O)cc2c(s1)CCC2 C1(CC(=O)NCCc2c(C)nc[nH]2)CC(C)N(C(C2CC3CC3C2)=O)C1 N1(C(C(C2CCC2)OCC)=O)CCCC(C)(C(N2CC(CC)C2)=O)C1 c1(C(=O)Nc2cn(CS(C)(=O)=O)nc2)cnn2c(C(F)(F)F)cccc12 CN=c1ccc(C(=O)NCC(C)(C)C(=O)NC(C2CC(C)C23CCC3)=O)c[nH]1 N1(C(CCc2c(C)ncs2)=O)CCN(C(c2cc[nH]n2)=O)CC1C(C)C c1(NC(c2cc(C)on2)C(F)(F)F)cccc(OC(N2CCCCC2C)=O)c1 Cc1ccc(-c2cn(CC(C)NC(c3ccc(=O)n(C)c3)=O)nn2)c([N+](=O)[O-])c1 C#CCCCCC(=O)NC1CCN(CCCC(C)(C)C)CC1C Cc1cc(C(=O)NC2CN(C(=O)CC3SC(=N)NC3=O)CC2C)c(O)nn1 C1(CCN(C)CC2CCCN2C(c2csc(C(F)F)c2)=O)CCOCC1 N12CC(=O)NC(C1)C2=O.N1(C(C(=O)OCC)=O)CC=CC1C(=O)NC C(CN=C(NC1CCC1)N1CCCC(OC(F)F)C1)OCCOCC O=C(C1=CS(=O)CCC1)NCCCCCNC(=O)C(c1ccc(F)c(F)c1)O Nc1cc(F)cc(F)c1C(N1CCCOC(CNC(c2cccs2)=O)C1)=O N1(C(C2N(CCC)CCC2)=O)CCCC(N(C)C(c2ccc(CSC)s2)=O)C1 CC1(C)CCCOC1CC(=O)NC1CCN(C(=O)CSCC(F)F)CC1 C=CCCCCC(=O)N1CCC2CC12C(=O)Nc1cccc(Cl)c1 C1(C(N2CC(=C)C2)=O)CC(CC)CCN1C(c1csc(CO)n1)=O c1(C(=O)NC2CC3(CC(C(N4C(CC)C(O)CC4)=O)C3)C2)cccc2[nH]ncc12 c1(-c2c(C)n[nH]c2)ccc(F)c(C(=O)NC2CN(C(=O)CC3C=CCCC3)C2)c1 C1(NC(C(c2ccc(C)cc2)OC)=O)CCS(=O)(=O)C12CN(C(=O)CC)C2.O c1(C(=O)NC(C2CCCN2C(c2ccnn2CC#N)=O)C)cn(C)c(=O)n1C C(=O)(C1=C(C)OCC1)N1CCCC(N(C(=O)Cc2cn(C)nn2)CC)C1 N1(C(CCN(C(C)=O)C)=O)CC(C)OC2(CCN(C(=O)CC3CSC3)C2)C1 CC(C)C(CC(=O)NCCOCCNC(=O)CCCn1ccnn1)C(C)C Cn1ncc(Br)c1CC(=O)NCCC1(O)CN(C(c2cncc(N)c2)=O)C1 C(C(F)(F)C(=O)N1CCC(N2CCC(NC(c3cc[nH]n3)=O)CC2)C1)N(C)C C1(NC(c2scc(OC)c2)=O)CC2(C1)CC(C)C2.c1(CC=O)ccccc1F n1(CC)nc(C(=O)COC(c2ccc(C3CCCC3)cc2)=O)c(C)n1 c1ccc(C=O)cc1F.C12CC(C1)C2.C(=O)C.C(=O)CN(C)C.COC Cc1c(NC(c2cc(F)ccc2F)C)ncnc1N1CCCC(OC(F)F)C1 c1(NC(C2(OC)CCN(C(CCC(C)OC)=O)C2)=O)ccc(C)c(CO)c1 C(=O)(CCS(=O)(=O)C1CCCC1)NCC(C)N(C(=O)C=C(Cl)Cl)CC N1(C(c2ccnc(OC)n2)C(=O)NCCSC)CCOc2ccc(C)cc2C1 c1(C(N2CCC(C)C2C(=O)NC2CCCC2N(C)C)=O)ccc([N+](=O)[O-])[nH]1 c1(CC(N2C(C(CNC(CCC#C)=O)(C)C)CCC2)=O)ccc(O)cn1 Cc1nc(NC(C2CC(F)CN(C(=O)COCC3CCCC3)C2)=O)ccc1O c1(C(=O)NCCN(C)C(C2CC2(C)Br)=O)c[nH]nc1C1CCC1 C(=O)(C(CC)C(C)C)NCc1ccc(CC)cn1.C1(CC=O)CC2(CC2)C1 c1(N2CC(O)(CCNC(=O)COc3ccc(O)cc3)C2)c(Cl)cccc1[N+](=O)[O-] c1(CC(=O)NC(CC)(CNC(c2ccnc(O)c2)=O)CC)c(C)cccc1F Cc1cc(C(N2CC(C)C2)=O)c(-n2cccc2)s1.N1(CC(=O)N)CCCC(C)C1 CN1CCCCCC1C(=O)NC1CCC(n2cc(-c3ccc(Cl)nc3)nn2)CC1 n1(CCCC)cc(C(N2CC(CCNC(=O)Cc3ccoc3C)C2)=O)nn1 C1(C)(CNC(CCc2n(C)cnc2)=O)CCN(C(=O)CSc2cn[nH]c2)CC1 C(=O)(C1CCCc2cncn21)NCCNC(=O)CCOc1cc(Cl)ccc1Cl c1(C(N2C(CC(=O)NCC3CNC(=O)C3)CC(C)(C)C2)=O)ccc2[nH]ccc2c1 C(=O)C(C)(C)CC(F)(F)F.C(CCC(C)(C)C)N(C(c1cn(CC)nc1)=O)C.N C1(C(=O)Nc2c(CC)cccc2)CCCC(NC(C2C3CCC(C3)C2C)=O)CC1 N1(C(c2ccc(C#C)o2)=O)CCCC(C)(NC(c2cnc(CC(C)(C)C)s2)=O)C1 N1(C(C(CC)(CC)OC)=O)CCC2(CCCN2C(C2CC(F)C(=O)N2)=O)C1 C=CC(CC)CC(=O)NCC1(OC)CCN(C(c2c(C)nn(C)c2OC)=O)C1 N1(C(c2ccc(C)nc2O)=O)CC(NC(c2cn(C)[nH]c2=N)=O)C2CCCC2C1 CC1CCN(C(=O)CCC2(C)CC2)C1CNC(=O)CCc1ccncc1 N1(C(c2ccn(CCC)n2)=O)CCN(C(c2cc(C)nc(C)c2)=O)C2COCC12 C1(NC(c2ccc(=NC)[nH]c2)=O)CN(C(=O)CC2(C)CCOCC2)CC1C1CC1 c1(C(=O)NCC2N(C(c3c(COC)ncs3)=O)CC2)cc(N)cnc1Cl C(C#Cc1cccnc1)NC(CCC1N(C(c2nc(CC)oc2)=O)CCC1)=O c1(C(=O)NCC2N(C(C3C(OCC)C3)=O)CCC2)cc[nH]c(=N)c1 C1(CCNC(COCCCOC)=O)CCN(C(c2ccc(Cl)o2)=O)CC1(F)F CC(C)C(C)CC(=O)N1CC2CC1C2NC(C1CCN(c2ncccn2)C1)=O C1(CC(=O)NCC2CCCC2C(=O)NCC2CCC2(F)F)CCOCC1 N1(C(C2CCCC(NC(CC(C)(C)OC)=O)C2)=O)Cc2cccc(C)c2C1 c1(C(=O)OCC)cc(NC(C2(CNc3ccccc3)CC2C)=O)ccc1Cl N1(C(C(C)C2CC2)=O)CCC(c2ccccc2)C(NC(C2CCC(=O)N2)=O)C1 c1(C(=O)Nc2ccc(NC(CN(C(C)=O)C)=O)cc2C)cc2ccsc2c(O)n1 c1(C(=O)NC2C(NC(C3(OC)CCCCC3)=O)CC2)cccc(C)c1O Cc1cc(N)c(C(=O)NCC2CC(O)CN2C(=O)Cc2cnnn2C)cc1F c1(OC)ncc(C(=O)N(C)CC=CC(=O)N(C2CC2C)C)s1 CCC(C)CCCCC(=O)NCC1CN(C)CCN1C(=O)Cc1ccc(Cl)cn1 CCCCC(CC)CC(=O)NC(C)C(=O)Nc1cnc2ncnn2c1 C1(C(NCP(C)(C)=O)=O)(NC(C=C(COC)C)=O)CCCC1C C1(C(N2CC(CC)C2)=O)CC12CC(NC(=O)Cc1ccoc1)C2 C1(NC(CC2(C)CCCCC2)=O)COC2(CCN(C(C3(CO)CCC3)=O)C2)C1 N1(C(COC2CCC(C)CC2)=O)CCCC12CCN(C(C1(CO)CCCO1)=O)C2 c1(C(=O)NC(c2cn(C)nn2)C(=O)NC(C)Cc2cnccn2)c[nH]ccc1=O C1(C(=O)NCc2c(F)ncc(C)c2)N(C(=O)C(F)CCC(C)C)CC12CCCC2 c1(NC(C2CC(F)CN2C(=O)Cc2cc(Br)cs2)=O)ccnc(C2CC2)c1 C1(NC(=O)COC2CCCOC2)CCCCN(C(=O)CCc2ccc(Cl)s2)C1 C1(C(=O)OC)CCC(NC(=O)C(C2CCN(C(=O)CCc3csnn3)C2)F)C1 C(CCCCCN=C(NCCn1cnc(C#N)n1)NC(C)C(C1CC1)OC)SC CC(Cn1ccnc1)N=c1ccnc(N2CCC(N3CCCC3)C2)[nH]1 n1(C(CC)C)nnnc1C(c1ccncc1)NC1(C)CC=CC1 c1(NC2CCN(S(N)(=O)=O)C2)nc2ccccc2n1-c1ccccc1F c1(C(N2CC(F)CC(NC(C(C)=C(CC)C)=O)C2)=O)c[nH]nc1S(N)(=O)=O Cc1ccc(C2(C(=O)NC(=O)N(C3CCOC3C)C3CC3)CCOCC2)cc1 C(=O)(C1CCc2cc(F)ccc21)NCC(CC)NC(=O)C(C)(C)c1nncn1C c1(C(C)C)[nH]nc2cncc(C(=O)NC3CC(C)C3)c12.S(C(F)(F)F)CC=O C1(C)(CNC(C(CSC)OC)=O)CN(C(=O)CCC2CCCCC2)CC1C N1(C(COCP(C)(C)=O)=O)CCC2CCCN(C(=O)CS(N)(=O)=O)C2C1 c1(N(CCCN(C(C2(O)CCC(C)CC2)=O)C)C)cnc2cc(F)c(F)cc2n1 c1(C=O)cnn(C2CCC2)c1.c1(C(N(CC(C)O)CC)=O)cc(CN)no1 C(=O)C(C)(O)C(C)C.c1(CCN(CCC)CCC)ccc(N2CCC2)nc1 C12(NC(CCN(C)CC)=O)CC(CNC(C3(SC)CC3)=O)(C1)OC2C C1(CC)C(C(=O)NCCCN(CC(C)C)C)CCN1C(C1CC(C)(O)C1)=O C=CCC(CC=C)C(=O)NC1CCC(C(=O)NC(=O)C=C)C1.CC=CCC.C C1(OC)CN(C(=O)CC2C=CCCC2)CC1C(=O)NC1COC(C(F)F)C1 C1(C(N(C(c2ccccc2)C(=O)NCC)C)=O)C2CCC(C2)C1C(=O)O C1(CNC(C2N(C(C)C)CCC2)=O)CCCCCN1C(c1cc(F)n[nH]1)=O C(=O)(CC(C)(C)C#N)N1C(C(C(=O)NC2C(C(C)C)C2)(C)C)CCC1 C1(NC(N2Cc3c(ccc(C(C)=O)c3)C2)=O)CCc2cc(O)ccc2C1 Cc1cc(Cl)c(C(N2CCC(C)(CNC(=O)CC(=O)N(C)C)C2)=O)cc1C c1(C(=O)OC)ccc2c(c1)CN(C(c1ccnc(F)c1OC)=O)C2 c1(C(N(C2CCN(C(C=CCC)=O)C2)CCO)=O)sc2cc(F)ccc2c1C CC1(C)CC(NC(C2C3CN(C(C4(O)CCOC4(C)C)=O)CC23)=O)CCO1 C1(C(=O)NC2(C#C)CC2)CCN(C(=O)CCc2cnoc2)CCO1 c1(CN2CC3C(C(N4C(C(=O)OCC)CCC4)=O)C3C2)cccc(OC)c1 C(CC(O)CC(=O)N1CC2(CC2)CC1CNC(c1occ2c1CCC2)=O)SC C1(C(=O)NC2(C)CN(C(=O)CCc3nnc(C(F)F)o3)C2)C2CCN1CC2 Cc1c(NCCCCCC2CC2)ncnc1N1CCC(C(C)C)C1 C(=O)(C(C)C1=CCCC1)N1C(CNC(COCC(=O)NC)=O)CCC1.O c1(CCC(=O)NC(C)CCCNC(=O)Cc2nnc(O)s2)ccc2[nH]ccc2c1 C1(NC(COC(CC)C)=O)CN(C(c2c(C)ncn2C)=O)CC1c1ccccc1 C(=O)(CC(C)(C)C(=O)NC(C)CN(C(c1cnccn1)=O)CC)OCC CCC(C(C)C)(c1nnnn1CC(F)F)NCC1CC1(Br)Br CC1(C2CCCCN2C(=O)Nc2nnc(COCc3ccccc3)s2)CCCO1 C(C)(C(=O)NNC(=O)C(C)Oc1cccc(Cl)c1)(c1ccccc1F)OC c1(NC(c2nc(C(=O)NC(C)C)sc2)=O)ccnnc1Nc1ccccc1 c1(C(=O)OC(c2nnc(-c3ccccc3)s2)C)ccc2[nH]nc(Br)c2n1 c1(CCC(=O)NC2CN(C(C3COCCO3)=O)C2)ccc(Cl)cc1O Cc1ccc2c(C(N3CCCC3C(C)NC(=O)C(C)c3cccs3)=O)coc2c1 c1(CNC(C(=O)NCC2C(C)CNCC2)=O)cccc2c1OCO2 c1(C(=O)NCC(C)N(C(=O)COC2CCC2)CC)c(C)coc1C c1(NC(C2(F)CN(C(C3CCCCO3)=O)C2)=O)cnc2c(O)cccc2c1 c1(OC)cncc(C(=O)NC2CCCC(NC(c3c[nH]cc3C)=O)C2)c1 C1(CNC(c2c(C)cc[nH]2)=O)CC(C)CCN1C(=O)CCC1CCCN1C S(=O)(=O)(c1cccnc1NCC1CC1)NC1(CC)CCOC1 O=NN1CCCCC1C(=O)NCC1CCCCN1C(C1CCS(=O)(=O)N1)=O c1(OC)cc(C#N)ccc1C(=O)NC1CC1C(=O)N.c1cc(F)cc(C)c1O C1(F)(CC)CN(C(=O)NCCn2cnc(I)c2)C1 N1(C(C(CCC)C)=O)Cc2ccc(CNC(=O)C(O)CCC(C)C)cc2C1 CC1(C)CCC(CNC(=O)CC2(C)CCN2C(C2CCO2)=O)OC1 C1(C(=O)NCC2N(C(c3cnc(CC)s3)=O)CCCC2)CCC2CC2CC1 C1(NC(=O)C=Cc2ccsc2)(CNC(=O)CC2CCCO2)CC2CCC1CC2 C1(CCC(N2CC(C)(CC=C)C2)=O)CCCCN1C(=O)C(C1CCCCC1)F Cc1nn(C(C)C)c(C)c1CC(=O)NCCCc1nc(-c2ccoc2)no1 CCC(CC(C)C)C(=O)NCC1=CCCN(C(=O)Cc2ccc(O)c(F)c2)C1 CN=c1[nH]cc(C(N2CC(F)CC2C(N2CC(C)C2(C)C)=O)=O)o1 c1(C(C)C)nc(NCCc2ccc3ccccc3n2)cc(=NC2CCCSC2)[nH]1 Cc1ccc(F)cc1S(=O)(=O)NCC1(F)CCCN(C(c2cc(C)n(C)c2)=O)C1 Cc1nn(C)c(C)c1C(N1CC(OCC)C1)=O.C1(C=O)CC(N(C)C)C1.N C1C2CCC(C2)N1C(c1ccnc(OC(F)F)c1)=O.C(C(C)=CC(=O)N)OC C1(NC(=O)C=Cc2nccs2)CCCC12CN(C(c1nc3cnccc3s1)=O)C2 C(=O)(C1=CNC2=NCCC2=C1)N1CC(C=C)CC1.C(=O)C(F)C(F)(F)C(F)(F)F.N c1(C(N2CCN(C(=O)Cc3ccc(F)cc3F)CC2)=O)c(Br)cc(F)c(Cl)c1F c1(CC(=O)OC(c2ccc(F)cc2F)C)ccc2c(c1)CCCS2 c1(C(=O)NC2C(CNC(=O)CCc3cscn3)CCC2)cnc2[nH]nnc2c1 c1(C(N2CCC(OCC3CCOCC3)C2)=O)ccc(C#CC2CC2)cc1 C(C(C)(C)CNC(c1cnoc1)=O)OCC.C1(C=O)CC1CC=O.C c1(C(N2CCN(Cc3ccccn3)CC2)C)cc(-c2ccncc2)nn1C c1(N2CC3C(C(N4CCN(C=O)CC4)=O)(C3)C2)ncnc2c1oc1ccccc21 C1(O)CCCN(C(=O)Cc2ccco2)C1.c1(CC(=O)N(C)C)ccc(C#N)nc1 N1(C(C(CSC)O)=O)CCN(C(c2ccc(C(F)(F)F)o2)=O)CC1C1CC1 c1(CC(N2C(CNC(CCC=C)=O)C=CC2)=O)cc(Cl)c2c(c1)OCCO2 c1(CNC2C(C(=O)O)CCC2)ccc(CCc2ccccc2)c(F)c1 Cc1ccn(CC(=O)NC(c2ccnn2C)C(=O)N(CC(=O)N(C)C)C)n1 C(C)(C1CCCCC1)=CC(=O)N(C(C)C)C.C(C)(C=O)NC(C)=O.C(C)C CC1(C)CCC(C(=O)NCC(CNC(c2n[nH]cc2Br)=O)CO)O1 C1(C(N2CC(OCCNC(c3cnn(CC(F)F)c3)=O)C2)=O)CCCCC1O C1CCN(C(=O)Cc2cc(C)nn2C)C(C)C1.C1(O)(CC#C)CC(C(=O)N)C1 C(=O)(C(CCN(C)C)NC(=O)Cn1ccnc1C)NCC(CC)(C)OC c1(C(=O)Nc2cc(C(=O)OC)c(Br)cc2F)ccc2sc(=N)[nH]c2c1 CC1=CCC(C(=O)NC(C)CCCCNC(=O)C(N)=O)CC1 N1(C(C(CC)C(C)(F)F)=O)CCCC12CCN(C(=O)CCN1CCC(O)CC1)C2 C1(c2n(CCOCC)nnn2)(NC2CCC2C(=O)N)CCCCC1.C1CC1 C1(C(=O)NCC(C)=CC(=O)NCC(C)S(N)(=O)=O)CCC2(CCC2)C1 c1(CN2CCN(C3CCC(OCC)CC3)CC2)c(Br)ccc2c1OCO2 Cc1cnncc1C(=O)NCC(C)CNC(c1csc(O)n1)=O c1(C(=O)NCC2(CCNC(C3CCCN3C3CC3)=O)CC2)n[nH]cc1Br C(=O)(C(F)(F)C1=CCOCC1)N1CCC(C2CC2)C1.C1(C(N)=O)CC1C(=O)N C12(NC(C(CC#C)C3CC3)=O)CCC1CN(C(=O)Cc1cccc(OCC)c1)C2 C(CNC(C1(O)CC(C)(C)C1)=O)(CC(F)(F)F)NC(c1cccc(C)c1)=O Cc1cc(C)c2nc(N3CCCC4(CNC(C5(C)COC5)=O)CCCC34)sc2c1 c1(NCc2c(CC)nccn2)ncccc1S(=O)(=O)N(C)CC1(F)CCC1 C1(NC(c2cc(C#N)ccn2)C(C)C)CNCC1C1CCCC1 Cc1ccc(C(C)C(=O)NCC2(CCNC(C3CCC3(F)F)=O)CC2)s1 CCCCS(=O)(=O)CC(=O)NCC1CC2CCC1C2.c1(C=O)cc(C)n(C)n1.N c1(OCC[Si](C)(C)C)noc2ncc(OC3CCC(C)(C)CC3)cc12 C1(C(C)C)CCC(NC(=NCC2CCCO2)NCC(C)(C)CC#N)CC1 C1(C=O)CCCN(C(C2(N(C)C)CC2)=O)CC1.c1(OC)cccc(C(O)C)c1.N N1(CCC)CCCC(C(=O)NCC2COCCN2C(=O)CCCNC=O)C1.O n1(CCC)ccnc1CNC(=O)CC1CCC1.C(=O)CCCN(C)C(C)C c1(CC(N2C(C)CC(CNC(=O)CC)C2)=O)ccc2nn[nH]c2c1.C(N)(=O)N S(=O)(=O)(c1c(Br)ccc(OC(F)(F)F)c1Br)NCCN=S(C)(C)=O C(=O)(CC(C)C(F)(F)F)NCCCC(C)NC(c1cc(OC)c(O)cc1)=O c1(C(=O)NC2CCN(C(C(C)(C)C3CC3)=O)CC(O)C2)c[nH]c2ccc(F)cc12 C(C(=O)NCCC1CCN(C)C1=O)(C(C)O)NC(c1c(CC)nco1)=O CCC(CC)CCCC(=O)N1CCCC(C2CCCCN2C(=O)C=NOC)C1 C1(C(=O)NCCC(C)F)CCCN(C(=O)Cn2ccnn2)CC1 N1(CC)CC(C(=O)N)CCC1=O.c1(C=O)cc(C)n(C2CC2)n1.C(C)C(C)C N1(C(C(C=C)O)=O)CCCC(CN(C(=O)C(c2ccc(OC)cc2)(F)F)C)C1 C(CCCCCN=c1ccnc(CO)[nH]1)NC(=O)C(C1CCCO1)C1CC1 C1(C(=O)NC2CCCN(C(c3c[nH]cc(Br)c3=O)=O)C2)Cc2ccccc2O1 N1(C(C=Cc2cc(C)no2)=O)CCCCCC1C(=O)NCC(C)(C)F C=CCCOCC(=O)NC(C)C=CC(=O)N(C)CC1(N(C)C)CC1 c1(C(=O)N)ccc2c(c1)nc(O)n2C.CCC(CNC(=O)C=CC(C)C)CC c1(C(=O)NCC2C(NC(c3c(C)csc3)=O)C2)cccc2ccoc12 c1(C(=O)NC(C(=O)NC(C)C)C)cccnc1.C(=O)C(O)CCN(C)C.C CCCCC(C(=O)NCc1cnn(CC)c1C)NC(c1ccc(OC)nn1)=O n1(CC)cc(S(=O)(=O)NC2CC2(c2ccccc2)C)c(C2CC2)n1 c1(N(C(c2ccccn2)C)C)cccc(C(C)(C)O)n1 CN(C)S(=O)(=O)NC(C1CC1(C)C1CNC1)=O c1(C(=O)OCC)cn2c(n1)C(NC(c1cc(Br)cc(C)c1F)=O)CCC2 c1(CC)c(C(=O)NC2CN(C(C3CC3c3ccccc3Cl)=O)CC2C)cnn1C c1(C(N2CC(NC(CCC(C)SC)=O)C(C)C2)=O)cnc2[nH]nc(O)c2c1 c1(C(=O)NC(C)C(C)NC(c2ccc3c(c2)CC3)=O)coc2c1C(=O)NCCC2 CC1CC(NC(=O)C(=O)N(C)C)CN(C(c2ncoc2-c2ccccc2)=O)C1 N1(C(C2C(=C)C2)=O)CCC2(CC1)OCCC2NC(c1csc(COC)n1)=O c1(C(N2CC(OC)CC2(C)CNC(=O)CCS)=O)cnn2c(=O)cc[nH]c12 C(=O)(CC1=CCOCC1)N1CCN(CCNC(C2C(C)CCS2)=O)CC1 c1(C(N(CCC(=O)N(CCCOCC)C)CC#C)=O)cnc(C)cn1 c1(C(=O)NC(C2CN(C(C3C(SC)CCC3)=O)C2)C)cnn(C)c1C(F)F C(C(=O)N1CCCO1)NC(c1cnc(CNC(C2C3CN(C)CC32)=O)nc1)=O C(=O)(C(C)CC(N)=O)N1C(C2(NC(C3(CC=C)CC=CC3)=O)CC2)CCC1 n1(CC(=O)NCCC(CNC(CSS(C)(=O)=O)=O)O)cnccc1=O [N-]=[N+]=NC1CN(C(=O)C(O)c2ccsc2)CC1NC(c1ccnc(O)c1)=O C=CC(C)(O)CC(=O)N1CCC(c2ccccc2)(NC(=O)C(C)CC=C)CC1 C1(C(N(C2CCCC2)CCCNC(c2ccsn2)=O)=O)CC2(CCC2O)C1 N1(C(=O)NCC(CCC)C)CCCC(N(S(C)(=O)=O)C)C1 N1(C(CCC2N(C)CCC2)=O)CC2CCC(NC(=O)CCc3ccccn3)C2C1 c1(N(C(C2CCCC(NC(c3n(CC)ccn3)=O)C2)=O)C)cc(F)ccc1C N1(C(CNC(CCC)=O)=O)CCCC(C(C)C(=O)NCC(F)(F)C(C)C)C1 C1(F)(CNC(C=CCCC=C(C)C)=O)CCN(C(C2CCOC2C)=O)CC1 c1(OCC(CN(CC(F)C(=O)O)CCOCC)O)ccc(F)cc1 N(C1CC2(CN(C(=O)CC3C=CCC3)C2)n2ccnc21)C(c1cc(C)sc1C)=O C(=O)(CCC=O)N(CCNC(C=C(CCC)C)=O)CC.c1(CC)ccccc1.N N1(C(COCCCC#C)=O)CCCC(N(C(=O)C(CC)NC(N)=O)CCO)C1 N1(C(CC(C)C(F)F)=O)CC2(CCN(C(c3ccc(C4CCOC4)cc3)=O)C2)C1 Cc1ccc(C(=O)NC2CC(CNC(C3COCC(C)O3)=O)C2)c(O)c1 C#CCC(CC(=O)N(CC#CC)CC)NC(c1cc(C)c(F)cn1)=O c1(C(=O)NC(c2ccccc2)CC#C)coc(COC)n1 CCC(C(=O)NC1CC(CNC(=O)CS)C1)C(C)C.c1ccc(C)cc1.C c1(C(=O)NC2CCC(NC(c3ncc(Cl)cc3F)=O)CC2)scc2c1CCCC2 C1(CC)CN(C(c2nccnc2C)=O)CCC1NC(=O)C(c1c(C)n[nH]c1C)C c1(C(=O)NC2C(CNC(CC(OCC)O)=O)C2)cc(C#N)cn1C.C c1(C(=O)NCC(CN(C(c2cnc(SC)s2)=O)C)C)cn(C)c2ccccc12 CCCCC(C)NC(=O)C(O)CNC(=O)CNC(=O)CCC Cc1cc(F)ncc1-c1ncsc1C(=O)Nc1cnc(C)c(C)n1 N1(C(COC)=O)CCCC2CN(Cc3nc(-c4cccs4)oc3C)CC12 CCCCS(=O)(=O)NCC(=O)N(C1CCCCC1N(C(=O)Cc1nc[nH]n1)C)C N1(C(C=C)=O)CC2(CCC(CNC(C3CN(C)CC3C(F)(F)F)=O)O2)C1 Cc1cc(C(=O)NC2CC3(C2)CCC3)cc(C)n1.C1(C)(C=O)CCC12CCC2.N c1(C(N2CCN(C(C(CCSC)NC(C)=O)=O)C(C)C2)=O)ccc([N+](=O)[O-])cc1 c1(OC)ccc(N2CCN(CC3CC(=O)N(C(C4CCCSC4)=O)C3)CC2)cc1 C(C(=O)N=c1cc(C(C)(C)C)o[nH]1)N1CCC(C)C1 C(=O)(CCCCCCC)NCC1CC(NC(C(F)=CCC)=O)C1(C)C CC(CCN=c1nc[nH]s1)NC(c1ccc(F)c(C(F)F)c1)=O C1(C(N2C(CNC(CNC(=O)NC)=O)CCC2)=O)CC2CCC1CC2 c1(CN2CCC(C#N)(NC(c3cccc(OC)c3F)=O)C2)cc(F)c(Cl)c(F)c1 CCC(C(=O)NC1CC1NC(=O)CCCOC)N1CCCC1=O C1(C(=O)NCCOc2ccn(C)n2)N(C(=O)CC2CSC2)CCCC1(C)C C1(C2CCCN(C(=O)COCC(F)F)C2)(NC(c2ccc(C)nc2)=O)CC1 N1(C(COC(CC)C)=O)C2CCC1C(NC(c1ccc(O)c(Br)c1)=O)C2 C1(CNC(CC2C(C)C2)=O)CC2CCC(C1)N2C(=O)C(C)(C)n1ccnn1 C12(CNC(=O)Nc3c(C)oc(-c4ccc(C(F)(F)F)cc4)n3)CNCC1CCO2 CC1(CNC(=O)C(c2cccc(Br)c2)O)CCCN(C(c2cnco2)=O)C1 C(N=c1[nH]c(=NCc2ccc(F)cc2F)c2c(F)cccc2[nH]1)c1ccn(C)n1 c1(C(N(C2(C(=O)O)CCSC2)CC)=O)ccc(OCC)cc1.C(C)(C)C C(=O)(C(O)CC(F)F)N1CCN(C(C2(CC(=O)OCC)CCCC2)=O)CC1 CC1C(NC(C2CC(=C(F)F)C2)=O)CCN1C(=O)CN1CCNC(=O)C1 C(C(C(=O)NCC(c1ccccc1)C)C(C)C)NC(c1c(CC)ccs1)=O C(=O)(CCCCCNC(=O)CC1CC(F)(F)C1)NC(C#C)CC1CCC1 c1(CNc2c(C)nc(-c3cccc(C)c3O)s2)c(Cl)cc(Br)cc1Cl C1(NC(C(F)(F)C2(OC)CCC2)=O)CCN(C(c2ccc(C)n2C)=O)CC1C N1(C(C(C)OCC=C)=O)CCC2(C1)CN(C(c1cc(Cl)ccc1O)=O)C2 C(C(C)(C)CN=c1ccc(Br)c(S(=O)(=O)N2CCCC2c2nncs2)[nH]1)OCC Cc1ccc(C(C)(C)C(=O)NCC2CCCC(C)C2)cc1.C(=O)C1=CCSC1.N N1(CC(=O)NCCn2cc(C(N3CCOC3=O)C)nn2)CCCNC1=O c1(C(=O)NCC(=C)CCNC(=O)CCC2CCCCC2)ccc2nn[nH]c2c1 N1(C(c2ccc(C(C)C)nc2)=O)CCCC2(NC(=O)C(C)C(C)(C)C)CC12 C1(NC(C=CCOC)=O)CCN(C(c2cc[nH]c2)=O)CCC1CO C1(C(=O)NC2(C3N(C(Cc4nnc(C)o4)=O)CCC3)CC2)CCc2ccnn2C1 C(C1=CCCN(C(C2CCCN(C(C)C)C2)=O)C1)NC(c1cc(C)sn1)=O c1(CC(=O)NC2(C)CCN(C(c3ccc(F)cc3Cl)=O)C2)cc(F)c(N)cc1F C(=O)(CC(C)(C)CNC(c1cccc(=O)n1C)=O)NC(C(=O)OC)C(C)O c1(OC)ccnc(OC)c1C(=O)NCCC1CCCN1C(c1cocc1C)=O C(CCCCC(=O)N1CC(C(N)=O)(CNC(C2CC23CCCOC3)=O)C1)SC C(=O)(CC(C)C(F)(F)F)NCCN1CCCN(C(C(C=C)(C)CC)=O)CC1 c1(OC)c(C(C(=O)Nc2ccc(F)cc2)N(C2(C)CC2)C)ccnc1F C(N=c1ccnc(NCc2noc3c2CCCC3)[nH]1)C1(CO)CCN(C)CC1 N1(C(C2N=C(C)SC2)=O)CCC(C2CCN(C(=O)CC3SC(=N)NC3=O)CC2)C1 c1(OC)cccc(O)c1NC(c1ccc(-c2cccc(C(C)(C)C#N)c2)cc1)C C(=O)(CCCCC(N)=O)NC1CC(C)(NC(c2ccc(CC)c(OC)c2)=O)C1 c1(NC(C2(O)CCCC(C(F)(F)F)C2)CC)c(C)cc(Cl)nc1Cl N1(C(c2cc(Br)cs2)C(=O)NC2CC(C(=O)OC)C2)CC(C)SC(C)C1 Nc1cccc(-c2cn(C3CCN(C(C4(CCO)CC4)=O)C3)nn2)n1 Cc1c(C(=O)OCCCc2cccc(F)c2)cc(C2CCCCC2)n1C N1(C(c2c(C(=O)OC)c(C)[nH]n2)=O)CCCN(C(=O)C#CC(=O)N(C)C)C(C)C1 C1(CC)CCN(C(=O)CCC(C)(F)F)C(C(=O)NCc2cnn(C)c2C)C1 C(=O)(CCC(=O)NC1(C)CCN(C(c2cccc(C(N)=O)n2)=O)C1)NCC C1(CC(=O)Nc2ccc(Cl)c(O)c2)CC2(C1)CN(Cc1c(I)ccnc1Cl)C2 Cc1ccc(C)c(C=O)c1.N1(C(C=CC(C)C)=O)CC(C(N)=O)C2(CC2)C1 CCN=c1ccc(C(=O)NCC2C3CN(C(=O)C(C)(C)C(F)F)CC23)c[nH]1 c1(C(=O)N)cccc2c1OCC2.N1(C(C)=O)CCCC(C(=O)NCC2CCC2)C1 N1(CC(CC)F)CCC2(C1)NC(=O)N(C(C)C)C2=O CC(C)CN=C(NCc1cccc(S(N)(=O)=O)c1)N1CCC(C(C)O)C1 C1(C(=O)NC2CC(c3ccccc3)C2)(NC(C(C)c2cncs2)=O)CCCCC1 c1(CSC)cccnc1C(=O)NC1CC(C)C1.C(C=C(Cl)Cl)=CC=O.N N1(C(c2ccoc2C)=O)CCCCC(O)C1.C(=O)C(C)(C)CN(C)C.COC C(=O)(C1CCc2c[nH]nc21)N(CC(C)C(N1CCC2CCCC2C1)=O)C CCCC(CC)CC(=O)N1CCCCC1C1CCN(C(c2c(C)nsc2C)=O)C1 N1(C(c2n(CC)ccn2)=O)CC(NC(=O)C=CCOC)C2(CC2)C1 c1(C(=O)NCC2CCN(C(C=CCCC)=O)CC2)cc(=O)c2cc(F)ccc2o1 C1(N(C)C(C2CCCN2C)=O)C2CN(C(C3CNC(=O)C3)=O)CC12 C1(C(=O)N)CC(C2CCCC2)C1.C1(C(N(CCC)CC)=O)CCN(C=O)CC1 Cc1ccc(C(N2CC3CC3(CNC(=O)CCCC(F)F)C2)=O)cc1C(F)(F)F C1(C(N(C)CC=CC(=O)NC(C2CCOC2)(C)C)=O)COCOC1 Cc1c(C(=O)NCCc2ccc(CNC(C3CC3C)=O)cc2)cccc1C#N N1(C(CC(CC)(C)C)=O)CCC2(C1)CN(C(=O)CCc1cccc(F)c1)C2 N1(C(C2C(CC)C2)=O)CCC(O)(C2CC2)CC1.C1(O)(C(=O)N)CCOC1(C)C N#Cc1ccc(C2(C(=O)NC3CCC3NC(C3CCSCC3)=O)CC2)cc1 CC1=C(C)CN(C(=O)C(c2ccoc2)NC(c2n[nH]c(C)c2Cl)=O)CC1 c1(C=O)c(C)c(-c2ccccc2)nn1C.C1(C(=O)NC2CC2)(CC)CCC1.C N1(C(c2c(C)noc2C)=O)CC2(CC(C)C2)C1.C1(C(=O)N)COC(C)(C)CO1 c1(OC)nc(Cl)ccc1C(=O)NC1CCC(C)N(C(=O)CS)C1.C1CCCO1 Cc1c(C(N2CC3CC2(CNC(=O)CCc2cn[nH]c2)C3)=O)oc2ccccc12 C1(Cn2cc(COC)nn2)CCCCN1C(c1ccc(-n2ccnc2)cn1)=O C=C(Cl)C(C)(C)C(=O)NC1CCCC(NC(=O)CNS(=O)(=O)CC)CC1 CC(C)C(C)(C)C(=O)Nc1cccc(NC(=O)C(C)C(F)F)c1 C1(CNC(CC2CC(=C)C2)=O)CCN(C(C2(OC)CCCOC2)=O)CC1 N1(C(c2c(NC)cc(Cl)cc2)=O)CCC2CC1CN(C(=O)C=CC1CCC1)C2 C1(C(N(C2CCC(CC)CC2)C)=O)COC2(C1)CN(C(c1ccc(C)cn1)=O)C2 C1(CNC(c2c(NC)cncc2)=O)CCN(C(=O)CC2(C)CCC2)C(C)C1 N1(C(C(C)NC(CC)=O)=O)CC(NC(=O)CC2CC2CC)CC12CCC2 N1(C(c2cn(CC=C)nn2)=O)CCC2(CCCC2NC(c2nonc2CC)=O)C1 CC(C)C(C(=O)NCC(CO)N(C)C)C(C)NC(C12COCC1C2)=O N1(C(C(c2ccc(C)cc2)(C)C)=O)CCN(C(C2C3CCC(=O)C23)=O)CC1C CCCCC(COC)N=c1nc2c(ncn2C)c(N2CC3CSCC(C3)C2)[nH]1 C1(C(N2CC(NC(C(F)=CC)=O)(COC)C2)=O)CCCCN1C(C)C Cc1ccc(NC(=O)C(=O)NCC(C)CNC(=O)C(C)C#N)cc1 c1(OC)ncc(C(C)NC(=O)NC2CC(CC)C2)cn1.C(C)(C)C.C=O c1(C(=O)NC2CC3CN(C(CS(CC)=O)=O)CC32)cccc2ncoc12 N1(C(C2(CCNC(Cc3nc(C)sc3)=O)CC2)=O)CC(O)C(C)(C)C1 S(=O)(=O)(c1cc(Br)c(C)cc1Br)NCc1cc(C)nn1C c1(C(N2CC(C(C)NC(C3(F)CCOC3C)=O)C2)=O)ccc2[nH]c(=N)[nH]c2c1 N1(C(C(CCC)=CCC)=O)CCC2(CCCC(CNC(=O)C(C)C)O2)CC1 c1(OCC)ccccc1C=CC(=O)N.c1(C=O)ccc(C2CC2)cc1.C1CC1 C1(NC(C2(CC)CC2(F)F)=O)CN(C(c2ccsc2C)=O)CC1SC C(C(C)(O)CC(=O)N)OC.C1(CC(N)=O)CCN(C(=O)C=Cc2cc[nH]n2)CC1 c1(CCC(=O)NCC(C2CCC2)NC(c2cnc(C)s2)=O)ccc2[nH]ccc2c1 C=CC(C)(CC)C(=O)N1CC(NC(c2csc(CCC)n2)=O)C(C(F)(F)F)C1 C(C(C)(C)C#N)N(C(=O)CCC1(C)CN(C(C2CC2)=O)C1)C.N(C)(C)C C1(N(C)C(c2coc(O)n2)=O)CCCC(N(C)C(c2cncs2)=O)C1 c1(OCC)c(C(=O)NC2C=CCN(C(=O)CCc3cc(C)on3)C2)cccc1F N(C(=NCC(=O)NC(C)C)N1CCN(c2cccc(Cl)c2)CC1)C1C(OCC)C1 c1(SC)cc(C(=O)N)ccc1N.c1(C(N(CCC)C)=O)cc(C(C)(C)C)n[nH]1 Cc1cc2c(cc1C)C(C(=O)NCCOCCCN(C(=O)CCC(N)=O)C)CO2 CC1(C)CCN(C(C2CCCS2)=O)CC1C(=O)NC(CO)C1CC1 c1(OC)c(C(=O)NCC(C)CNC(C2(OC)CCCCC2)=O)csc1C C(CC(C)C)(C(=O)NC(C)(C)CNC(=O)CCC1CCCN1C)OC CC(N=[N+]=[N-])C(=O)N1CCCC(CCC(=O)NC(c2cccc(O)c2)C)C1 c1(C(N2CCC(NC(CCC=C)=O)C(CO)CC2)=O)c(F)ccc2n[nH]cc12 C1(C)(CC)CC(NC(C2SCC=C2C)=O)CN1C(=O)CCCCCOC N1(C(c2ncc(Cl)cn2)=O)CCC2(CC1)CC2c1cn(-c2ccncc2)nn1 C(=O)(CC1=CCN(C(c2ccc3[nH]ccc3n2)=O)CC1)NCC(CN(C)C)(C)O N1(C(C(C(=C)C)(C)C)=O)CCC2CC(C1)CN(C(c1ccccc1OC)=O)C2 c1(C(=O)NCC(CNC(CCCCC)=O)(C)O)cnn2c1NCC(C)C2 CCCC(O)CC(=O)N1CC(F)CC1CNC(=O)Cc1ccccc1C(F)(F)F C(CNC(=O)CCCn1ccnc1)(C(=O)NCC1(OC)CC1)OC N1(C(=O)C=Cc2nccs2)CCC2(CC1)CN(C(C1CC=CCC1)=O)CC2CO N1(C(CCc2nc(C)sc2)=O)CC(F)CC1CNC(C1CCC(=O)N1)=O c1(OC)ncnc(OC)c1NC(C1CCCN1C(=O)C=CCBr)=O C1(C#N)(C(=O)NCC(CNC(c2ccnc(C)c2C)=O)(C)F)CC2CCC1C2 N1(C(CN(C(COC)=O)C)=O)CCC(C(C)NC(C2(CF)CC2)=O)C1 N1(C(C2CCCN(CC)C2)=O)CC2(C)CC1(C(=O)NC(CCO)C(C)(C)C)C2 C12(C(N3CC4C(NC(C(N5CCCC(O)C5)C)=O)C4C3)=O)CC(C)(CCO1)C2 CC(C)C(=O)C(=O)N(C1CCCCC1N(C(=O)C(C)Cn1ccnc1)C)C C1(CC)CCN(C(=O)C(C)CSCC)CC1.C(=O)CCCC=O.C(C)(C)C C(=O)CC(C)(C)C.C1(NC(C(C)NC(CC)(C)C)=O)CCN(C(=O)C)C1.N Cc1oc(CO)cc1C(=O)NCCN1CCN(C(=O)C(c2cnn(C)c2)=O)CC1 N1(C(C(CCC)OC)=O)CCN(C(c2cnc(COC)nc2O)=O)CC(O)C1 N1(C(C(C)=C2CCCC2)=O)CC(C)C(C)(C(N2CC(C)(CSC)C2)=O)C1 Nc1c(C(N2CC=CC2CNC(=O)CCC(F)F)=O)nc2c(Cl)cc(Cl)cn12 c1(NCC2CCN(CC)CC2)ccc(S(=O)(=O)NCCF)cc1C#N N1(C(c2cncc(CC)c2)=O)CCN(C(=O)Cc2cnc(C)s2)CC1C1CCC1 N1(C(C)=O)CCCCC1CC(=O)N(CCC)CC.C(=O)C(C)(C)CN(C)C C(=O)(C1=CCCCC1)N1CCC(C)(CNC(C(c2ccc(F)cc2)C)=O)C1 C(c1cc[nH]n1)=CC(=O)NC1CN(C(=O)CCc2ccncc2)C1 C(C)(C)(CC(=O)NCC1C(C)(C)C1(F)F)NC(Cc1n(C)ccn1)=O c1(SC)nc(Cl)c(SC)c(=NCCc2csc3cc(Br)ccc23)[nH]1 C1(C(C)NC(COC(CC)C)=O)CCCN1C(c1ccc(C(N)=O)o1)=O CC#CCC(C(=O)NC(C)COC(C)C)NC(c1cccc(O)c1)=O Cc1occc(=O)c1OCC=O.C1(N(CCC)C(C)C)CCC(C(C)C)CC1.N C1(CC(=O)NC(c2ncc(C)[nH]2)(C)C)CCN(C(c2sccc2F)=O)CC1 c1(-c2cn(CC3OCCN(C(C(=O)N4CCCC4)=O)C3)nn2)cnc2ccccc2c1 c1(C(N2CCN(C(C(C)NC(=O)OC)=O)CC2)=O)cccc2ncc(Br)n12 N1(C(CC(CC#C)NC(c2c[nH]c3cnccc23)=O)=O)CC2CCCCCC2C1 c1(C(N(C)CCNC(=O)C(C2CCOCC2)O)=O)cccc2nccn12 N1(C(c2cc(C)oc2)=O)CC(NC(c2cn(-c3ccccc3)nc2C)=O)C(O)C1 c1(CC)sc(C(=O)NCCC2CCN(C(C3CC3C(C)(C)C)=O)C2)cc1C N1(C(c2nc(C)c(Br)cc2)=O)CCN(C(C2CC2Cl)=O)CC12CCC2 c1(NC(CN(C)C)CCO)ccc(-c2ccsc2)cc1[N+](=O)[O-] CCC(CC)(CCNC(=O)C(F)C1CCC1)NC(c1cn(C)nn1)=O C(CC(C(C)C)NC(=O)CC1CC(C)(C)C1)N(C(Cn1c(C)nnn1)=O)C CCCC(C(=O)N1CC(NC(=O)C(F)=C(C)C)C(n2cccn2)C1)OCC C1(C=O)CC12CCOC2.C(CCO)NC(=O)OC(C)(C)C.C1(C=O)CC1.N N1(C(COCC(=O)NC)=O)CCCC(F)(F)CC1.C1(C(=O)N)CCCC(F)C1 C(N=c1cc(C)nc(NC2CCCC2C#N)[nH]1)C1(OC)CCC(C)(C)CC1 c1(OCC)ccc(C2CCCN2C(=O)NC2CC(CC3CCC3)C2)cc1 c1(C(=O)NC(CC)CNC(=O)CSC(C)C)ncnn1CC C(CCSC#N)(C=O)N(CCCNC=O)C.C1CCC2(CC2)C1.C(C)(C)C C12(CNC(CN(CC)CC)=O)CC1CN(C(=O)CO)C2.c1ccccc1C c1(CC(N2CC(C3(NC(C4CCCCCC4)=O)CC3)C2)=O)ccc2c(c1)COC2 CC1CCCC1(C(=O)NCCCc1cn[nH]c1)NC(=O)CC1CC1CN c1(SC)ccc(C)c(C(=O)NCC2CN(c3nnc(O)s3)CCO2)c1 n1(CC)cnc2c(NCc3cccnc3Cl)[nH]c(=NC3CN(S(C)(=O)=O)C3)nc12 C(C(=O)N1CCC(C)C1)(C(C)C)NC(=O)OCC.c1(C(=O)N)ccsc1 Cc1ncc(C(=O)NC2CC(CO)N(C(=O)C(F)C3CCC3)C2)cn1 c1(C(=O)NCC2(OC)CN(C(C3CCCC(F)C3)=O)C2)ccn2c1CCCC2 C#CC1CC2(CC2)CN1C(C1CCN(C(c2ccc(C(C)=O)o2)=O)C12CC2)=O Cc1cc(CCNC(C2(C3CCCN3C(c3cc(F)c[nH]3)=O)CC2)=O)n[nH]1 c1(CC)cc(C(=O)NCCC(O)CNC(=O)Cc2ccnn2C)ccc1F Cc1cc(CC(N2CCN(C(CNC(=O)C(C)O)C(F)F)CC2)=O)ccc1F C(=O)(CC(C)(C)CC)NC(CNC(C1(C)CC(=C)C1)=O)Cc1ccccc1 C1(C(=O)NC2(C3CCCO3)CC2)CCN(C(=O)CCCC2CCCO2)C12CC2 CC1(C)CC(C)(C)CN1C(=O)C=CC1CCOC1.c1(C(=O)N)ccc(F)cc1 c1(C(N2CC(N(C(=O)Cc3coc(C(F)F)n3)C)C2)=O)cnc2n1CCC2 c1(NC(C2CCCCN(C(c3c(CC)con3)=O)C2)=O)cccc2c1OCC2 CC1CCC(NC(c2cccc(C(N)=O)n2)=O)CN1CC(O)Cn1cccn1 c1(OC)ccc(C(=O)NCC2CCC(NC(c3cnc(Cl)[nH]3)=O)C2)cn1 c1(CN2C(C(=O)NC(COC)(C)C)CNCC2)ccc(OC)c2ccccc12 N1(C(C(CC)n2cncn2)=O)CCC2CCN(C(=O)CCC(C)SC)C2C1 N1(C(C2CCC(=O)O2)=O)CCC(C(F)CNC(=O)Cc2ncc(Cl)s2)CC1 O=C(O)CC(CC(=O)O)NCc1cn(C2COCC2O)nn1 N1(C(C2(COC)CC2)=O)CCN(C2CN(C(=O)C(C)c3ccsn3)C2)CC1 C(c1cccc(C)c1)=CC(=O)NC1CN(C(C(CC)N(C)C)=O)CC1CC c1(C2(C(=O)NC3C(NC(C=CC)=O)CCOC3)CC2)ccc(F)c(Cl)c1 c1(CC(N2CC(NC(c3c(C(C)C)ocn3)=O)C2)=O)cc(O)nnc1O Cc1cc(CCC(N2CC3C(NC(=O)CC4CCC(=O)N4C)C3C2)=O)cc(C)c1 C(CCC(=O)NCCNC(c1ccc(C(F)F)s1)=O)N(C(C)=O)C.C1CC1 c1(N(C(=O)CCc2ccccc2)CC)ccc2c(c1)CCC2.C(C)(C(C)(C)C)N C12(CC=O)CCC(CC1)OC2.C1CCCC1.c1(CC=O)cnc(C(F)(F)F)s1.N c1(CC)cc(C(=O)NCC(C2CCCCN2C(=O)C(O)C(C)C)(C)C)cc(F)c1 C1(CC=C)(NC(c2nc(Cl)cs2)=O)CCN(C(C2CCC(=O)O2)=O)C1 c1(CCC(=O)NCC2CCC(NC(C3CC3(F)F)=O)C2)ccccc1 Cc1cc(C#N)cc(C(=O)NCC(c2ccccc2)NC(=O)Cc2nc[nH]n2)n1 CC#CCCCC(=O)NCC1CC1NC(=O)CNC(c1ccco1)=O Cc1cc(C(N2CCC2(C)CC(N2CC(F)(F)C2C2CC2)=O)=O)ncc1N c1(SC)c(C(=O)NCC2CCN(C(C3CCC3(C)C)=O)C2)cccc1F Cc1c(CC(=O)NCC(C2CCOC2)NC(C2COC2)=O)cccc1[N+](=O)[O-] C1(C(=O)Nc2cccc(NC(C#CC3(C)CC3)=O)c2)CCC2(CC1)CC(OC)C2 C1(C(N2C(CNC(=O)CCc3nc[nH]n3)COCC2)=O)Cc2ccc(F)cc2C1 c1(CNC(C2N(C(CCC)=O)CCCC2)=O)nn(C)c(=O)n(C)c1=O c1(CCOC)nc(=NC2(CNC(c3n[nH]c(C)c3[N+](=O)[O-])=O)CC2)s[nH]1 c1(C(N2CCN(C(C3C(C)C3C)=O)CC2CCO)=O)cnc2ccccn2c1=O CC1(C2CC2C(=O)NC2CCCCC2CC(N2CC(F)C2)=O)COC1 C(CCS(=O)(=O)CC)NC(CCC)(CC)c1nnnn1CC(F)F c1(C(=O)NC(c2nn[nH]n2)C2CC2)cc2c(s1)CCNC2 c1(C(N2CC(CNC(c3c(COC)nn[nH]3)=O)OCC2)=O)cc2ncccc2[nH]1 c1(NC(C2C=CC(NC(c3cc(C)no3)=O)C2)=O)cccc(C#N)c1.C(C)C N1(C(C(COC)C)=O)CCN(C(=O)C(C)(C)COC(C)C)CC1C1CCC1 C1(CNC(COC)=O)CCN(C(c2cccs2)=O)C1.C(=O)CN(C)C.C c1(C(=O)NCC2(F)CN(C(C(CCCC)C)=O)C2)cnc(O)c2ccsc12 c1(C(N2CCC(CC=C)C2)=O)c(N)cc(OC)cc1F N1(C(C(C)Oc2ccc(C)cc2)=O)CCC(NC(=O)CC(=O)N(C)C)C12CC2 c1(C(=O)NC2(CNC(C3(CC)CC3)=O)CCOC2)ccc(C)cc1F C1(c2[nH]nc(-c3c(F)cccc3)n2)CC(C2CCN(Cc3ccccc3)C2)C1 Cc1ncn(O)c1C(=O)NCC1CC(NC(=O)Cc2ccns2)C1 c1(C(=O)N)cc(F)cnc1O.C1(C)(CNC(c2c(CC)nc[nH]2)=O)CCCC1 Cc1nc(O)ccc1C(=O)NC1CC(NC(C2CCCCS2)=O)C1 c1(C(N2CCC(N(C)C(C3CC4(CCC4)CO3)=O)CC2)=O)ccc(F)cc1C#N CCC(C(=O)NCC1(CCNC(=O)C=C(Cl)Cl)CCCC1)NC(N)=O c1(C(=O)NCCCCC(C)(C)NC(C2CCC(CC)O2)=O)onc2c1CCCC2 C1(CNC(CCC=C)=O)CC2(CC2)CN1C(C1CC1c1cccs1)=O N1(C(c2ccc(OC)s2)=O)CCC(C(F)F)(CNC(=O)CC(C)CF)C1 c1(N2CCN(c3n(C)ccn3)CC2)nc(=NCC(F)CO)[nH]c2ccsc12 C=C(Cl)CC(C(=O)NCCc1cccs1)NC(=O)CS(=O)(=O)CC N1(CC)CCCC(CN)C1.c1(C(N(C(CC2CC2)=O)C)=O)nc[nH]c1C=O Cc1cc(N2CCC(C)C(CNC(=O)C3=COCCO3)C2)ncc1[N+](=O)[O-] C(=O)(C(O)CN1CCOCC1)N(CC(CC)NC(=O)CC(=O)OC)C O=C(C(F)(F)C(O)C1CC1)N1CCN(Cc2ccc(Br)c(F)c2)CC1 c1(C(=O)NCC(C2CCC(F)(F)CC2)OC)cc([N+](=O)[O-])ccc1C c1(C(=O)NCCOCCCNC(=O)CC2CCCOC2)cc2c(nn1)CCCC2 c1(C(C=O)(C)C)ccc(F)c(Cl)c1.c1(CC(=O)NC(C)CC)ccc(O)cn1.N c1(CNC(C(c2ccc(OCC(F)(F)F)cc2)C)=O)cc(F)ccc1I c1(C(=O)NCCC2CCC(NC(c3n(C)ccn3)=O)C2)ccc(Br)c(O)n1 c1(N(C(C(CNC(=O)Cc2cc[nH]c2)OC)=O)C)cc(C)cc(F)c1 C1(OC)CCC12CCN(C(=O)CC(F)F)CC2.C(c1nc(C)c(C)[nH]1)=CC(=O)N C1(C(=O)NCC(n2cc(CN3CC4CC4C3)nn2)C)CCN(S(N)(=O)=O)CC1 c1(COC)cc(=NCCCNC(=O)C(=O)C(C)(C)C)[nH]c(C)n1 CC1(C)CN(C(C2CC=CCC2)=O)CCC1NC(=O)C(F)(F)C1CC1 c1(COC)nc(=NC2CC(NC(c3ccc4nn[nH]c4n3)=O)C2(C)C)s[nH]1 O=C1NC(=O)C2(CN(C(C3CC4(CCC4)CN3C(=O)C)=O)C2)N1.C(=O)C C1(C(=O)NC2CCC(CCC(=O)NCC3C4CCCCC34)C2)CC2C=CC1C2 c1(C(c2nnnn2C)NC(c2c(C)c(Br)ccc2)C)c(F)ccc(Cl)c1F c1(C(=O)NCc2ccc(C(C)NC3CCNC3)cc2)c(Cl)ccc(Br)c1F C1(CNC(C2N(C(C)=O)CCCC2)=O)CCCCN(C(c2cc(CO)on2)=O)C1 C#Cc1ccc(C(N2CC(NC(c3cc(OC)ccc3C)=O)CC2C)=O)cc1Cl c1(C(=O)NCC2CC3CC3N2C(c2cc(Br)no2)=O)cnn2cnnc2c1 C(=O)(CS(=O)(=O)Cc1cccs1)N1CC(N(C(=O)CN2CCOC2=O)C)C1 CC(C)C(C)(CNC(C1CCCCO1)=O)NC(=O)Cn1ncn(C)c1=O CCCCC(O)C(C)C(=O)NCC(CO)NC(C1CCCN1C=O)=O C1(N(C(CN(C(C)C)C)=O)C)CCN(C(=O)CCc2ncccn2)CC12CC2 C1(C(N(CCCC)C)=O)CC2(CCOCC2)C1.c1(OCC)cccnc1C=O.N C1(C(=O)NC(c2ccccc2C)C(=O)OC)CC(O)CN1c1cc(C)ncn1 C1(CNC(c2ccc(O)cn2)=O)CC2CCC(C1)N2C(c1ccnc(F)c1F)=O Cc1[nH]c(-c2ccco2)nc(=S)c1C(=O)NCC1CC(C(N)=O)=NO1 C1(C=O)CC2CSCC(C1)C2.C(C(=O)NC1CC(F)(C)C1)(C(C)(C)C)SC C1(C(=O)NCCC2ON=C(C)C2)CN(C(C2CCC(C)(C)C2)=O)CC1F C1(CNC(C(CSC)C)=O)CCCCN(C(c2cc3sccc3cn2)=O)CC1 C(N=c1[nH]c(=NC2CC(CC#N)C2)[nH]c2c1CSC2)c1scc(CN(C)C)n1 N1(C(Cc2ccc(C)o2)=O)CC2CC3CC2C1C3NC(=O)C(O)Cn1cncn1 c1(NCC2CN(C(c3cnn(C)c3C(F)(F)F)=O)C2)ncnn2cccc12 Cc1cc(NC(=O)CC2CCC(NC(c3cc(C(C)C)on3)=O)C2)ccc1O Cc1ccc(OCC(=O)NC2CCC2)c(F)c1.N1(CC=O)CC(=O)NC1=O.C CCC(CC(=O)NC(C)(C)CNC(C12CCOC1CC(=O)NC2)=O)CC(F)(F)F C(=O)(C(CC)CCCC)N1C(CNC(c2cn(CCCC)nc2C)=O)COCC1 N1(C(C2CC(OCC)C2)=O)CC2CCCC(N=c3[nH]c(SC)nc(Cl)c3C)C2C1 C1(NC(=O)CC2CCCC23CC3)CN(C(C2(C3CC3)CC2)=O)CCC12CCC2 N1(C(CCNC(=O)C=CCl)=O)CCCC(N2CCN(C(=O)C=CCO)CC2)C1 c1(CNC(=O)CC2CCN(C(=O)COCC3CCCC3)C2)ccccc1.C N1(C(CCc2cncc(C)c2)=O)CC2(C1)CN(C(c1n[nH]c(C)c1N)=O)CCO2 c1(C(=O)NC(C(C)C)CCNC(c2n[nH]cc2Cl)=O)ccc(O)c(CO)c1 C(N=c1ccc2nccc(Cl)c2[nH]1)(c1ccc(Cl)cc1)c1ccccc1 C(N=c1ccnc(C2CCCC2)[nH]1)C1CC(NC(c2cc3n(n2)CCCC3)=O)C1 c1nccc(S(C)(=O)=O)n1.CC(C)C(C(=O)NC12COC(C1)C2)n1cccc1.C CN1CCC(O)(CONC(C2CCN(C3CCSCC3)CC2)=O)CC1 N#Cc1cc(N2CC3(CCN(C(c4ccc(F)cc4)=O)C3)C2)c([N+](=O)[O-])cc1F C1(C)(C(N(CCCCN(C(C(CCOC)OC)=O)C)C)=O)CCN(C)C1=O Cc1cc(C(=O)NC(CC2CCCC2)C(=O)NC)cc(C#N)c1.C1CC12CC2 C1(C(=O)NCC2N(C(C(C)c3ccn[nH]3)=O)CC2)CC(C#N)C1 C1(N)(C(N(C(c2cn(-c3ccc(C(C)(C)C)cc3)nn2)C)C)=O)CCCCCC1 c1(CN2CCC(CC(=O)N(c3nnc(C)s3)CC)C2)ccc(OCC)cc1 Cc1cc(C(=O)NCC2CCCCO2)cc(C)c1O.C1(CC(=O)N)CC2CC2C1 c1(NC(c2cccc(NC(CC(CC)O)=O)c2)=O)cc(Br)cc(O)n1.C1CC1.C N1(C(COCC(C)C)=O)CCC2CCN(C(c3ccc(O)cc3Cl)=O)C2C1 CCC(C(C)(F)F)NC(=O)CC(CNC(C1(O)CCCC1)=O)C1CCC1 C(=O)(C1=CCCC(C)(C)C1)N1CC(CC)C(NC(=O)C(C)C2CC2)CC1 c1(OC)nn(C)cc1CNC1CCC(CC(=O)O)C1 C(=O)(C(O)C(C)C)NCCn1ncc(C(=O)NC2CCN(CC)C2)c1 C1(NC(C2CC(=C)C2)=O)CN(C(=O)CCOC(C)CC(C)C)CC1C1CC1 c1(OC)ccc(C(=O)NCC2CC2NC(=O)C(C)SC)cc1[N+](=O)[O-] c1ccc(Cl)cc1.C(CC(=O)NCC1CCC1)NC(=O)NC.C(=O)CC.N N1(C(=O)CC2CCOC2)CC2CCN(C(c3sc([N+](=O)[O-])cc3Cl)=O)C2C1 C=C(CNC(=O)C(O)CSC)CCNC(c1cc(C2(C)CC2)n[nH]1)=O c1(C(=O)NCCN(CCCCCC)CCC)cc(OC)c(C)c(OC)c1 N1(C(c2cccc(SC)c2)=O)CCN(C(=O)Cc2csc(C)n2)C2CC12 c1(SC)nc(Cl)cc(=NCC2CCCCN(C(C3(C)CC(F)(F)C3)=O)C2)[nH]1 C(=O)(C(=O)C(C)CC)NC(CC(=O)NC(CCC=C)C1CC1)CC C(CNC(=O)COC(C)C)(CC(=O)NCCC12CCCC1C2)OC c1(C(N(C(C)C(=O)NCc2cn(CC)cn2)CCC)=O)ccc(C#N)s1 CC(C)C(C)(O)C(=O)N1CCC(C(=O)NCCC2CCOC2(C)C)C1 C(C(C(=O)NCC(=O)CC)n1cc(C2(c3ccccc3)CC2)nn1)OCC CCC(CC)(CC)C(=O)NCC1CCCC1NC(C1(P(C)(C)=O)CC1)=O C1(C(=O)NCC2CCN(c3nc(OC)c(F)cn3)CC2)CCCCC12CC2(F)F C(C(CO)C(C)C)NC(c1n(CCOC)nnn1)(C)CSCCF CCC(F)(F)C(=O)NCC(CC(C)C)NC(C1C2CNC(=O)C12)=O C1(C(N(C2CCC(NC(C(F)=CC)=O)CC2)C)=O)CCS(=O)(=O)C1(C)C C1(NC(C2C(C)(C)C2(C)C)=O)CCCN(C(=O)CC2COC(=O)C2)CC1 C1(=CC(=O)NC(CNC(C(C2CCC2)OC)=O)(C)C2CC2)CCCCC1 N1(C(c2ccnn2Cc2ccc(F)cc2)C(=O)NCC=C)CCS(=O)CCC1C N1(C(C)=O)CC2(C(=O)NOC(C3(C)CC3)C)CCC1CC2.C1COCCC1C c1(CC)nc(N2CC(C(C)NC(C3CCOC(CC)C3)=O)C2)c(CC)c(Cl)n1 c1(CNC(=O)NC2CC(CO)C(O)C2O)c(F)ccc(F)c1Cl CN1CC2OCCN(C(=O)NCC3(n4cc5ccccc5n4)CCCC3)C2C1 C(C1C(C(N2CCC(C(C)NC(c3ccc(F)o3)=O)CC2)=O)C1(C)C)=C(C)C C1CCCCN(C(=O)Cn2ncc(O)nc2=O)CC1.C(C)(C(=O)NC)NC(C)=O C(=O)(CCC(C)C)N(C1CCN(C(C2CCC(=O)N2C)=O)C1)CC c1(NCC2N(C(C(C)C3CCCC3)=O)CCC2)nnccc1C#N c1(OC)ccc(OC)c(S(=O)(=O)N2CCCC2(C)C(=O)NC2COCC2O)c1 Cc1nn(C(C)C)c(C)c1CC(=O)NCC1CC1.c1(C=O)ccc(Cl)cc1F c1(CNC(C(C(C)C)C)=O)ccccc1F.C12(C=O)CCCC1(C(N)=O)C2.C C1(C(C)C)C(C(=O)N(C)CCC2CC2)CCN1C(C1SCCS1)=O c1(C(=O)NCC2(OCCO)CCCC2)nc(Br)cnc1Br c1(CC(C)C(=O)NC2CC(CNC(C3CCCCC3O)=O)C2)ccc(O)cc1 c1(C(=O)OC)nc(NC(=O)Nc2ccc(-n3cccc3)cc2)sc1C c1(C(=O)NC2C(OC)CN(C(CC(CC)(C)C)=O)C2)cc2c(s1)CCC(C)C2 C1(C(=O)OC)N(C(c2cc(C(C)(C)C)on2)C(=O)NC2CCCC2)CC1(C)C C1(C(N(CCCNC(c2[nH]cc(CC)n2)=O)C)=O)CCCCC1CC S(=O)(=O)(c1ccncc1)N1CCC2(C(C(=O)NC(c3cc(F)cc(Br)c3)C)C2)C1 c1(C(N2CCC(O)C2)=O)nccc2ccsc12.c1(SC)cn(C)nc1C(=O)NC CC(C)CC(C(=O)NCCCOC1CCC1)ONC(c1cnnn1C1CC1)=O C#Cc1ccc(NC(C2C3CC2N(C(C2(C)CC4C=CC2C4)=O)C3)=O)c(C)c1 C(=O)(C(CO)C(F)(F)F)N(C(CC)C(=O)NCC1CN(C(C)C)C1)C C1(C(=O)NC(c2nncs2)C)C(CNC(=O)CCc2cnn[nH]2)C1(C)C C(C)(C)(C(=O)NC1CC(C)C1)N(C)C.c1(C(=O)N)c[nH]cc1-c1ccccc1 c1(CC(=O)OC)occc1C(=O)NCC1C=CCN1C(c1ccsc1)=O CC1COCCC1CNC(=O)CCC1(NC(=O)C(C2CCOCC2)=O)CCC1 N1(C(CCOCCC)=O)CCC(C2CC(NC(=O)Cc3cccc(Cl)c3Cl)C2)C1 C1(C(=O)NCc2n(C(C)C)ncn2)CCN(C(=O)CSc2cn[nH]c2)C1C N1(C(CC2(CNC(c3n(C=C)ncc3)=O)CC2)=O)CC(CO)C2(CCC2)C1 c1(OC)ccccc1.C1(C#N)(C(N(C2(C=O)CCC2)C2CC2)=O)CCCO1.N CC(C)(CCCNC(=O)CC1CC(O)C1(C)C)C(=O)NC1CC12CCCCC2 Cn1ncc2cc(C(N3CC4CC(NC(=O)Cn5cccnc5=O)C4C3)=O)sc12 N1(C(=O)NCC(CC)C#N)CCN(Cc2ccc(C)cc2)C(=O)C1 c1(C(=O)NCC2C(NC(CN(C(=O)OC)C)=O)CCC2)c(C)ncnc1O C#CCCN=C(NCC1(C)CCCCCCC1)N(C)Cc1ncc(C)s1 N1(C(c2c(CC=C)cccc2)=O)CCC2CN(C(C3CCCC(CF)C3)=O)CC12 N1(C(C23OCC(C(C)C)(C2)C3)=O)CCC(C)C(C)C1.C1(C=O)COC(=O)N1C c1(C(N2CCC(CCNC(C(CCCC)O)=O)C2)=O)cnc2c(c1)CCC(=O)N2 Cc1ccc(C=CC(N2CCC(CO)C(NC(=O)C(O)C3CCC3)C2)=O)cc1 C(=O)(C(C)CN=C(NC(c1cccs1)C)N1CCN(CC(F)(F)F)C(=O)C1)OC C1(O)(CCNC(CC(=O)OC)=O)CCN(C(c2ccc(Cl)c(C)c2)=O)CC1 CC(N=c1[nH]c(=NC2CCC(F)(F)C2)[nH]c2c1CSC2)c1ncc(F)cc1F C(=O)(CC(C(C)OC)NC(=O)C(F)C1CCC1)N(CC(=O)OC)C C(=O)(C(CNC(C1CC1Cl)=O)C(C)(C)C)NC(C)(C)CCCF N1(C(c2ccc(C)n2C)=O)CCC2CC2(C(N2CCN(C(C)(C)C)CC2)=O)CC1 CCC(CC(C)C)C(=O)NC(C)CCCNC(c1sc(F)cc1Cl)=O C1(C#N)(CNC(CC2(C)CCN(C(C3CSC3)=O)C2)=O)CCCCC1 CC1CCCCC1C.C(c1cn(C)cn1)=CC(=O)N.C1(=CC=O)CCSCC1 Cc1ccc(S(=O)(=O)N(CC(=O)NCC(C)(C)c2cnc[nH]2)C)cc1 c1(CCC)n[nH]c(=NCC2CCCCN2C(=O)C(c2c(C)noc2C)C)s1 C1(C(N2CC(C(=O)NCC(N3CCOCC3)=O)(CC)C2)=O)C2CCC(F)C12 N1(C(CN(C(C)=O)C)=O)CCN(C2CCN(C(=O)CCc3ccc(Cl)s3)C2)CC1 CCCCCC(F)C(=O)NCCCCCNC(=O)C=CCN(CC)CC N1(C(=O)CN2CCCC2)CC2CC(C1)N2C(c1ccc(Br)cc1Cl)=O Cc1cc(CNCC2CCC2)ccc1O C(C)(C(C(C)C)NC(c1nn(C)cc1Br)=O)NC(C(C)(C)OC)=O n1(C(C)C)cnc2c(N3CC(C)C(F)(F)C3)nc(N3CCC(CC(F)F)C3)nc12 N1(CC(=O)NC2CCN(C(C3C(C)OC(=O)N3)=O)C2)C(=O)CCCC1=O c1ccc(F)c(Br)c1.CC(C)(C)C(O)c1cn(CC2C=CCN2C(=O)C)nn1.O c1(OC)cc(C(=O)NC(C2CC=CCC2)C(=O)NCC(C)CC(C)C)ccn1 C1(OC)C2CC3CN(C(c4n[nH]c(C)c4Br)C(=O)NCC4CCCO4)C1C3C2 c1(C(C)=O)csc(C(=O)NC2C=CC(N)C2)c1 c1(C(=O)NC2CCCN(Cc3noc(C4CC4)n3)C2)cc2c(s1)CCOC2 c1(NC(C2CCC(=O)N(CC(F)(F)F)C2)=O)ccc2c(c1)CCC(=O)N2 O=C1CCc2cc(C(=O)NOCC(C3CC4CC4C3)=O)c(F)cc2N1 C(=O)(CC(C)(C)C)NC1CCN(C(C2C(c3ccc(C)s3)C2)=O)CC1.C(C)=O C=CCCCCCCCCC(=O)NCC1CCC(N(C(=O)C(C)O)C)CC1 C(COC)(CC(=O)NCC1CCCSC1)NC(CCN(C)CC)=O CC1CN(C(=O)CN2C(=O)CCC2=O)CC1CCNC(C1C=CCCC1)=O C1(C(=O)NCC2CCN(C(=O)Nc3ccc(C)s3)C2)CC12CCc1ccccc12 c1(NC(N2CCC(C(C(=O)OC)(C)C)C2)=O)ccccc1Cl c1(OC)n[nH]c(=Nc2cccc(C(C(=O)O)N(C)C)c2C)s1 C(=O)(C(CCOC)NC(=O)C(F)=CC1CC1)NC(CN(CC)CC)C c1(C(=O)NC(C)CNC(=O)CCc2cccc(C(F)F)c2)ccc2ncccn12 C1(CCC(=O)N(CCCC)CCO)CCN(C(C2CCCOC2)=O)CC1 Cn1ccc(C2CC2C(=O)NCC(O)CC)n1.c1(CC)ccoc1.C(=O)(C)N c1(OC(C)C)ncccc1C(=O)NC.C1CCCC1.c1(CC=O)cn(C)nn1 Cc1cc(C#N)cnc1C(=O)NCC1CCCC1C(=O)NC1COCCOC1 C(=O)(CC(O)C(C)(C)C)NCCCCCCNC(c1c(O)ccc(C)c1)=O N1(C2CCC(NC(c3cc(CC)on3)=O)C2)CCN(C(=O)CC2CC2)CC1.O C1(NC(c2c(CC)nc(C)[nH]2)=O)COCCN(C(=O)CCC(F)(F)F)C1 C1CN(C(=O)C(F)=CC2CC2)CCC1(C)C.C1(CC)C(CC(=O)N)C1(F)F.C C1(CN(C(c2c(C)ncs2)=O)C)CCCN(C(=O)CCF)C1 CCC(C)C(C)CNC(c1nnnn1C1(C)CC1)COc1ccccc1 N1(C(c2c(C)cno2)=O)CC2(CCCN(C(c3cnn(C)c3N)=O)C2)C1 c1(NC(C(C(C)OC)O)=O)cc(Br)cc2ccccc12 C12(CNC(C)=O)CC(CO1)N(C(C1C3CC(=O)CC13)=O)C2 N1(C(c2c(C)nc(C)[nH]2)=O)CCCC(C)C1CNC(=O)CC(C)C CN1CCN(C(C2CC2(C)C)=O)C(C(=O)NC2(C(O)CO)CC2)C1 c1cc(O)nc(Cl)c1.C1(C(=O)OC)CC(C(=O)NCCSCC(=O)N)C1 C1(NC(CCC=C)=O)CC12CC(NC(c1c(C3CCCOC3)noc1CC)=O)C2 N1(C(CN=c2scc(C)[nH]2)=O)CCC2(CCCC2NC(=O)CC2CC2C)CC1 O=C1CCC(C(=O)NCCC2CCN(C(=O)CC3CC=CCC3)CC2(F)F)=NN1 c1(C(=O)NCC2(CNC(=O)Cc3cscn3)CCCCC2)ccc2cc[nH]c2c1 c1(C(=O)NC(C)CCCO)ccc(C2COCCN2C(C2CN(C)C2)=O)n1C N1(C(CCC)=O)CC23CCCC2(C1)CN(C(c1cc([N+](=O)[O-])oc1C)=O)C3 C1(C(N(CCO)CC)=O)CN(C(C2CC3CCC2CC3)=O)CC12CC2 C1(CNC(C2C(CC)C2)=O)CN(C(=O)Cc2n[nH]cc2Br)CC12CCC2 N1(C(C2CC3CC(OC)C3C2)=O)C2CCC1CN(C(=O)CC(=O)N(C)C)C2 N1(C(CCn2ncc(C)c2)=O)CCC(C(=O)NC2CN(C(C)C)C2)C1(C)C N1(C(c2ccc(C(=O)OC)n2C)=O)CCCOC(CNC(=O)CC(C)SC)C1 Cc1nc(C(=O)NC2CCC(C)CC2)cn1C(F)F.C1(CC=O)CC2CC2C1 CC1(C(=O)NCC(F)C)CC(F)(F)C1.C1(C(=O)N)CCC(=O)N1C1CC1 C1(NC(N(C)Cc2cc(C)nn2C)=O)CC(S(=O)(=O)c2ccccc2)C1 N1(C(C=NOC)=O)CCOCC(NC(=O)C(c2ccc(C(F)(F)F)cc2)F)C1 Cc1cc(C(=O)NCC2(C)CCN(C(=O)C3=CCCS3)C2)n(C2CC2)n1 C12(C=O)CCC(CC1)N(C(=O)Cc1cnc[nH]1)C2.C1(C(=O)N)CC1.C#CC c1(C(C(C)NC(c2sccc2)=O)NC(CCOCCOC)=O)ccccc1.O N1(C(C(c2scc(C)n2)C)=O)CC2(CC2)CC1C.C(=O)C(O)Cc1cnc[nH]1.N c1(OC)ccc(C)cc1CC(=O)NC(C1CCCN1C(=O)Cc1scnc1C)C C1(C(CNC(C(COC)O)=O)F)CCN(C(c2coc(CO)c2)=O)CC1 C1(NC(c2cnn3ccsc23)=O)CN(C(C2CCCOCC2)=O)C2(CCC2)C1 N1(C(CC2CC(=C)C2)=O)CC2CCCCC2(NC(c2ccc(NC)cc2)=O)C1 C1(C(N2C(C)CCC(C(=O)O)C2)=O)COC2CCCCC12 c1(C(=O)NC2C(NC(C3C(=C)CC3)=O)CCCC2)ccc2scnc2c1 C1(CCC)CN(C(C2(O)CCC2)=O)C1.C1CC1C=O.C(C)(C)C.CC.O CC(C)C(CCN(C(=O)Cn1ncnn1)C)NC(=O)CC.C1(C=O)CCC1.N c1(C(=O)Nc2n(CCCC)ncc2)cc(C2CC2)n(C)c1 Cc1cc(C(=O)NCC2CN(C(c3cc(CO)ccc3Cl)=O)CCO2)nc(C)c1 Cc1cccc2c(CCC(=O)NCCCCNC(=O)C(C)C(C)(C)C)c[nH]c12 CC1CCN(CC(=O)NCC2(O)CN(C(C3(CC4CC4)CC3)=O)C2)C1 c1(-n2cc(CCN(C)C(C3(CO)CCCO3)=O)nn2)cccnc1C(=O)O CCCC(O)(CCC)CC(=O)N1CCN(C(C2CC(F)C(=O)N2)=O)CC1CC N1(C(C(C)NS(CC)(=O)=O)=O)CCCCC1.C1(CC=O)CCC1.C(C)=O.C c1(C(=O)NCC(CNC(C2(CC=C)COC2)=O)F)cc(C)c(CC)o1 C#Cc1cccc(C(=O)N(CC(O)CNC(=O)CSCC(C)C)C)c1F c1(C(=O)NC(CCN(C)C)C(=O)NC2CCC2)coc2c1COC2 N1(C(C)=O)CCC(CC=O)CC1.C1(CC(=O)NC2CC2)CCCC1.C1CC1.N N1(C(C2CCCC(C)O2)=O)CCC(C)(CNC(c2cncnc2)=O)CC1 CCC(C)(CO)C(=O)NCCCCC(C)NC(=O)Cc1ccc(C)c(OC)c1 c1(NC(C2CCCN(C(c3ccn(CCC)n3)=O)C2)C)ncc(Cl)c(O)n1 n1(CC(=O)N(C2CC(NC(c3cnn(CCO)c3)=O)C2)C)nc(Cl)ccc1=O C(=O)(C(O)C(F)(F)F)N1C(CN(C(=O)CCC2CCCN2C)C)CCCC1 c1(-c2nc(-c3cn(C(C)(C)C)c(=O)nc3O)on2)cccc2c1CCCC2 Cc1cc(C(=O)NC(C(=O)NC2CCC(=O)NC2)C2CCC2)c(C)cn1 C(C)(CCC(=O)N(CCCN(C)C(c1ccc(Br)o1)=O)C)OCC c1(C(N2CCN(CCC)CC2)=O)ccc(Br)cc1C(F)(F)F.CC(C)C(O)C(=O)N C1(C(=O)NCCN(C(=O)Cc2ccc(Cl)c(Cl)c2)C)CCN(C)S1(=O)=O Cc1nn(C)cc1C(O)C(=O)NCC1CCN(C(C2(C)COC2)=O)CC1 c1(NC(CC)CC#N)ccc(S(=O)(=O)NCC(CC2CCCCC2)OC)cc1Cl C1(C(c2nc(Br)cs2)=O)CCN(Cc2cccn2Cc2cccs2)CC1 N1(C(c2n(C(CC)CC)ncc2)=O)C2CCC1CN(C(C1(C)CCCC1O)=O)C2 C1(CC(C)NC(C2(C=C)CC2)=O)CCN(C(=O)CC2CC3CCC2C3)CC1 C12(NC(CN(C)CC)=O)CCC(CN(C(c3cc4n(n3)CC(F)C4)=O)C1)C2 c1(NC(C2(CN)CCNC2)=O)cc(Cl)ccn1 C1(C(=O)NC(c2ccnn2C)C(=O)NC(C)CN2CCOCC2)CCCC(O)C1 CC(C(=O)NCC1CC1C(=O)NC(c1cnsc1)C)=C1CC1 N1(C(C2(CC=C)CC2)=O)CCN(C(=O)CCCC2CCCC(=O)N2)C(CC)C1 C1(CNC(=O)C(F)=CCCF)CN(C(c2ccc[nH]2)=O)CCCO1 C1(CNC(COCC)=O)CN(C)CCN1C(C1CC(C)(C)O1)=O C1(C(=O)NC2(CCCNC(C3(C#C)CCCC3)=O)CC2)CC(=O)NC1(C)C C(CC(C(=O)NOC1CCN(C)CC1)NC(c1ccc(C)o1)=O)SC N1(C(c2sccc2Cl)C(=O)NCc2cccs2)CCN(CC2CCOC2)CC1 N1(C(c2[nH]cc(CC)c2)=O)CCC(C2CN(C(C3CC3c3cccs3)=O)C2)CC1 C=CCC(C(=O)OC)NC(C1COCC1NC(c1cc(O)cs1)=O)=O CCCC(C#N)C(=O)NCCCC(C)NC(c1ccc(C2CC2)s1)=O N1(C(Cc2c(C)nc(S)s2)=O)CC2(CNC(=O)C(C)n3ccnc3)CCC1C2 C1(O)(CNC(c2n[nH]cc2C2CC2)=O)CN(C(=O)C(O)C2CCCC2)C1 c1(C(N(CC(C)NC(=O)C(C)(C)O)C)=O)ccc(-c2cn[nH]c2)cn1 N1(C(CCC(=O)N(C)C)=O)CCC2(C1)CN(C(=O)CC(F)(F)F)CCO2 N1(C(c2ccn(CC)n2)=O)CCC2(CCCN(C(=O)Cc3nonc3C)C2)C1 C1(CN(C(C2(OCC)CC2)=O)C)COCCN1C(=O)CSCCC(C)C C(CCCCCC(=O)N1CC(NC(=O)C(C)n2cncn2)CC1(C)C)SC CCC(C)C(O)C(C)C(=O)N1CC=CC1(C(=O)NCC=CCl)COC N1(C(COc2ccc(C)c(C)c2)=O)C2CCC1CN(C(C1CC3CCC3C1)=O)C2 Cc1cc(C)c(C(N2CCC(C)(NC(=O)Cc3ncn4c3CCC4)C2)=O)c(C)n1 C=CCCC(C(=O)NCC1(O)CCC(C)CC1)NC(=O)CCNC(=O)NC O=S(=O)(c1ccc(NCC2(F)CC(C)C2)c(Cl)c1)NCC1CCC(F)C1 n1(CCC(=O)NC(CNC(c2c(CC)ccs2)=O)C)ccc2cc(C)ccc12 CC(C)C(F)C(=O)NC(C1CCN(C(=O)C=CC(=O)N(C)C)CC1)C C1(C(N2CC(F)CC(NC(Cn3nnc(C)n3)=O)C2)=O)CCc2ccnn2C1 c1(C(=O)N)cc2cc(Cl)sc2[nH]1.N1(C(C(C)(C)OCC)=O)CCC(CCC)CC1 CC(C)CC(CNC(=O)Cn1cnc(C(N)=O)n1)NC(c1cc(F)cs1)=O c1(C(N(CC(CC)NC(=O)CCC2(C)CC2)C)=O)ccc(N(C)CC)cc1 C1(CCCC)CN(CC)CCN1CC1CC(C)CC(C)C1 c1(NC(C(CCC)NC(c2cccnc2NC)=O)=O)cccc(N=[N+]=[N-])c1 N1(C(CNS(CC)(=O)=O)=O)CCC(C)(CNC(=O)C(C)SC)C1 C1(C(=O)NC2CC(CCNC(CSCC)=O)C2)(CO)CC1(F)F C(c1ccc(OCC(N2CCC2CC(C)C)=O)cc1)=CC(=O)NCC#C CCC(F)(F)C(=O)NCC1CC2CC2N1C(c1ncn(-c2ccccc2)n1)=O C1(CC(=O)NCC(=O)N)CN(C(=O)COCC(F)F)CC12CC2.C1CC1 c1(NC)snc(C)c1C(=O)NCCCOCC.C(=O)(C(C)C1CCCO1)N O=C1OCc2ccc(C(N3CCC4CC3CN4C(=O)C(F)F)=O)cc21 CC1CC=C(C(=O)NC2CCN(C(=O)CCCc3ccccn3)CC2(C)C)CC1 C1(NC(C2C(C)(C)C2)=O)CN(C(c2ccc3c(c2)NCC3)=O)CC2(CC2)C1 CC1C(NC(C2CC2CC(C)(C)C)=O)CCCN1C(c1cc(Br)c[nH]1)=O N1(C(c2c(-n3cc(CC(C)OC)nn3)cccc2)=O)CCCC(C(=O)OC)CC1 C(CCCC(=O)NCC(C)CN(C)C)NC(C(C)OCCC=C)=O CC1C(NC(=O)C=Cc2ccncn2)CCCN1C(=O)CCc1ccn(C)n1 C(C)(C(=O)NOCC1CCOCC1)(N(C(CC1CCC(C)C1)=O)C)C1CC1 c1(C(=O)NCC(CC)NC(C2(SC)CCC2)=O)cnc2nccnc2c1 N1(C(C(C(C)C)OCC)=O)CCCC(C(N)=O)C1.c1(C(=O)N)cncc(N)n1 C=C(F)C1(CC(N2CCCC(NC(C3CC3C(C)(F)F)=O)C2)=O)CCOCC1 c1(CC(=O)NC2(C)CCN(C(CCC(C)O)=O)C2)ccc(C(=O)OC)cc1F C1(CNC(c2cc(CC)ncc2)=O)CCCN(C(=O)CN2CCCC2CO)CC1 C1(CNC(=O)NCCOCC)CCCN(C(=O)C(F)=C(C)C)C1 N1(C(C(CSC)C)=O)CCN(C(c2nc(Cl)oc2C)=O)C(c2nccn2C)C1 C(=O)(CCC(=O)NC1CCC(NC(=O)Cc2cncnc2O)C1)NC C1CC(N2CC3CCCC3C2)CN(Cn2ccc(N3CCCCC3)n2)C1 C=CC(O)(C(=O)NC1CC(NC(=O)C=CBr)C1)C(F)(F)F C(=O)(CC1=CCOCC1)NC1(C(N2CCCC(C(C)C)C2)=O)CC(F)C1 N1(C(C(CC(C)C)O)=O)CCC(NC(C2CCN(C3CC3)CC2)=O)C12CCC2 C12(NC(c3ccc(CC)s3)=O)CCN(C(c3c(C)ccnc3O)=O)CC1C2 CC1(C)CCC(C(N2CCCC(CNC(=O)C=Cc3ccncn3)CC2)=O)CO1 Cc1ccc(C=CC(=O)NCCC2CN(C(c3n[nH]c(C)c3F)=O)C2)s1 c1(C(N2CC(C(N)=O)OCC2)=O)coc2c1C(O)CCC2 C1(C(=O)OCC)CN(C(=O)Cc2sccc2-c2ccccc2)CC12CC2 C1(NC(CCC2CC(OC)C2)=O)CC2CCC(C1F)N2C(=O)CC1(O)COC1 C1(C(=O)NC2(CNC(=O)CC3CCCCCO3)CC2)CCC2(CCOCC2)O1 C1(NC(CNC(C(CC)C)=O)=O)CC12CCC(NC(c1c[nH]nc1O)=O)CC2 C1(NC(C(C=CCCC)O)=O)CCC2CN(C(=O)C(F)C3=CCCCC3)CC2C1 C1(NC(CCSC)=O)CCN(C(C2CC3CC3C2)=O)C(c2ccccc2)C1 c1(CCC)ccc(-n2cc(-c3cc(C4CC4)ccn3)nn2)cc1Cl N(C1c2ccccc2C2CCC1C2)C(C1CCN(CC(=O)NC2CC2)CC1)=O C1(C(=O)NCC(C=C)O)CC(O)C(O)CC1CNC(=O)CCn1ccnn1 CCC(CC)(CN=c1[nH]cncc1Br)NC(=O)CC(C)C(C)C Cc1cc(N2CC(C)C(F)(F)C2)nc(=NCCCCOc2ccc(F)cc2)[nH]1 N1(CC)CCCCC1C(=O)NC1CCN(c2cnc(C3CCCC3)nc2)C1 C1(CNC(C(CC)CCc2ccccc2)=O)CCC2(CN(Cc3csc(C)c3)C2)O1 Nc1c(C(N2CC(CNC(C3CC3c3ccco3)=O)C(O)C2)=O)ccnc1F CCC(C)C(O)CC(=O)N1CC2CC(C1)C2NC(C1CCC2(C1)CC2(F)F)=O Cc1cnn(C)c1CC(=O)NCCCCC(C)NC(c1cccnc1C1CC1)=O N1(C(C2C(CCC)CCC2)=O)CCCC(C2CCCCO2)C1 N1(C(C2(CCCC)CCC2)=O)CC2C(NC(=O)C(C)OCCOC)C2C1 c1(OC)nc(C)c(Br)cc1C(=O)NCC1CCCN(C(C2(C)CC2)=O)C1 C(C)(CC1CCC1)(C(=O)NC1CC2(C1)CC2)OC.c1(CC=O)nocc1C C1(n2cc(CC(C)(C)OC)nn2)CN(C(C2CCN(C3COC3)C2)=O)CC1C C1(CNC(COCCOC)=O)CCC12CN(C(=O)CCc1ccccc1)C2 C12(C(N(C3CCC(NC(=O)CCc4ncc[nH]4)C3)C)=O)CCC(CC1)OC2 N1(C(C(CSC)O)=O)CC(NC(c2ccc(Cn3cccc3)cc2)=O)C(C)C1 CC1CN(C(c2[nH]nc3ncccc23)=O)C(C)CN1C(=O)Cc1ncc(Cl)s1 C1(NC(c2nc(C)c(C)[nH]2)=O)CCC2CN(C(C3CCCCC3)=O)CCC2C1 c1(C2N(C(=O)NCC3(c4ccccn4)CCC3)CCC2)ccc(Br)cn1 C1(NC(C(C)SC)=O)CCCCC1C(=O)NCCC(C)C C(=O)(C(C)CCc1ccccc1F)NCC(CNC(CCNC(C)=O)=O)(C)C CC(C)(C)C1=NOC(C)(C(N2CCCC(C)(NC(=O)Cc3ccsc3Cl)C2)=O)C1 c1(OC)ccc(CNC2CC2C(=O)Nc2cnnn2C)cc1C c1(OC)c(C(N2CCC(C(=O)NCC(N)=O)C(O)C2)=O)cccc1Br C=CC(C)(O)CC(=O)N(C)CCOCCC(=O)NCCN1CCCC1 CCC(C)CCC(=O)N1CCC(CN(C(=O)COCC2CC2)C2CC2)CC1 c1(NC(N2CCN(C(=O)NC3CCCC3)CC2)=O)cc(F)c(Cl)cc1F Cc1cc(C(N2CCCC2C(C)NC(=O)C(F)CC2CC2)=O)sc1Cl CN(C)NC(=O)CCC(=O)NCC(C)(C)NC(C1CC1C1CC1)=O c1(OC)ncc(C(=O)Nc2c(Br)cnn2C)cc1-c1ccc(-c2ccccc2)s1 c1(C(=O)NCC2(OC)CCN(C(=O)CCC(C)O)C2)ccn2ccccc12 N1(C(CCc2n(C)ncc2)=O)CC2CC(NC(c3cc(C4CC4)no3)=O)CC1C2 c1(C(N2CC(NC(C(CCOC)C)=O)C(OC)C2)=O)ccc(OC(C)C)nc1C CC(C)C(=O)C(=O)NCC1CC(NC(=O)Cn2cnnc2O)C1(C)C CC(=O)CCCC(=O)N1CCN(CC(C)NC(=O)CCc2c(C)noc2Cl)CC1 N1(C(C2(OC)CCSC2)=O)CC2CC2(NC(=O)C(F)(F)c2nccn2C)C1 CC1CC(NC(c2cc3ccsc3s2)=O)CN(C(=O)CC23COC(CF)(C2)C3)C1 Cn1ccc(C(=O)NC(C(=O)N2CCC2CC2CCCC2)C2(O)CCC2)n1 N1(C(CCC=CCC=C)=O)CC(CNC(C2(C(C)(C)O)CC2)=O)CCC1C C1(CNC(C(=O)NCC)=O)CCOC1.C(=O)CC.c1(C=O)cccs1.N Cn1cc(C(N2CCC(CO)(NC(=O)C(C3CCCCCC3)O)C2)=O)nc1O c1(C(=O)NCC(CCNC(c2cc(F)cc(F)c2)=O)O)c[nH]cc(Cl)c1=O C1(NC(Cc2scc(C)n2)=O)CCC(C)N(C(c2cnco2)=O)C1 C(=O)(C(CC(N)=O)NC(c1ccc(CO)o1)=O)NC(C(C)F)C C(=O)(C(C)(C)CCC#N)NCc1cc(C(N(C(C=C)C)C)=O)sc1 c1(CC)nc(C)c(C(N2CCOC(CCCNC(C3CC4CC4C3)=O)C2)=O)o1 C(CCCCC(=O)NCC1(C2CC2)CCCO1)NC(=O)Cn1cccc1 C1(CC)CN(C(c2cc(Cl)ccn2)=O)CCN1C(c1ccc(CC(C)C)cc1)=O c1(C(N(CC(C(C)C)c2ccccc2)C)C)ccc(F)cc1Cl c1(C(N(C)CC2(CNC(C(CN(C)C)O)=O)CC2)=O)cn2ccsc2n1 C1(CC)(CNC(=O)C(O)CNC(c2cccc(=O)o2)=O)CC12CCC2 Cc1occ(C(F)(F)F)c1C(N1CCCC1C(=O)Nc1cnc(Cl)cn1)=O C1(NC(c2nc(CC)sc2)=O)CC(C)(C)C1C(F)(F)F.C1(CC)CCCN1 N1(C(C=NOC)=O)CC(CNC(C2(N(C)C)CCCSC2)=O)C2(CC2)C1 c1(C(N2CC(CNC(C(C)C3CCCC3)=O)OCC2)=O)ccc(O)c(N=[N+]=[N-])c1 N1(C(c2n(CC)cnc2)C(=O)Nc2ccccc2)CC2CCC(O)CC2C1 C1(C=O)CCC(C)(C)C1.C1(C(=O)NCCSCC(C)C)COC(C)C1.N C1(C(N(C(C)CN(C)C(c2cnn(C3COC3)c2)=O)C)=O)CCn2cnnc2C1 CC(CC(C)NC(c1nonc1N)=O)NC(=O)C=CCN1CCCC1 c1(OCC)nccc(C)c1C(=O)NC(C)Cn1cc(CN2CCOCC2)nn1 CC(CC(N)=O)C(=O)NC1CC(C(=O)NCC2(F)CC(O)C2)CC1O CC1(CNC(=O)CCC2CCC2)CCN(C(=O)CC2CCCC2)C1 O=C1Cc2cc(NC(N3Cc4[nH][nH]c(=N)c4C3)=O)c(Cl)cc2N1 Cc1nccn1C(C)C(N1CCCC1C(C)NC(c1ccoc1)=O)=O C1(C(=O)NCC(CNC(c2cc(C(C)C)n(C)n2)=O)C)CCCCCC(=O)C1 Cc1occc1C(=O)NC(CCN(C(=O)C(C)(C)F)C)c1cccs1 c1(CC(=O)NC2C3CN(C(CCC(C)(C)OCC)=O)CC32)c(C)cc(C)cc1O c1(NC(=O)C(F)OC(F)(F)F)ncc(-c2ccccc2)[nH]1 C1CN(C(=O)C(F)=CCCF)CC(C)(C)O1.C1(COC)(C)CC1C=O.O c1(NC(c2ncc(C)nc2)=O)ccc2c(c1)CCN(C)C2 C(=O)(C(C)(C)C1=CCN(C(=O)CC=C(Cl)Cl)C1)N1CCC(OCC(C)C)C1 C(c1ccc([N+](=O)[O-])cc1)=CC(=O)N(C(C)CNC(=O)CCC1CCC1)C c1(OC)ccc(C(=O)NCCC2CCCN(C(c3ccc(CO)o3)=O)C2)c(F)n1 CCCC(CC)CC(=O)NCC1CCCCN1C(=O)C(c1ccccc1)O CC(C)C(CCNC(c1ccnc(-n2cccn2)c1)=O)NC(=O)C1=NOCC1 C1(C)(C(=O)OC)CCCN(C(C2C=CC(NC(C3CC(OC)C3)=O)C2)=O)C1 C1(C(=O)Nc2cccc(C(=O)OCC)c2)CC2(C1)CN(Cc1cc[nH]n1)C2 c1(CC)ccc(C(=O)NC2CC(C)C2)c(F)c1.c1(C=O)cc([N+](=O)[O-])sn1 CC1CN(C(=O)CCN2CCCC2=O)CCC1CNC(c1ccccc1CO)=O C=Cc1cc(C(=O)NCC(C)(C)OCCNC(=O)C(F)(F)CC)cc(F)c1 N1(C(C2(CC=C)CCOCC2)=O)CCN(C(C2CCN2CC)=O)CC12CCC2 c1(CN(CC(COCC=C)(C)C)CC)nc(CCCC)[nH]c1Cl C(CN=c1cc[nH]cc1S(=O)(=O)N1CCCC2(CC1)CC2(F)F)c1cc(C)ns1 c1(C(=O)NC2(C3CN(C(C4(CCCC)CCC4)=O)C3)CC2)cc2n(c1)CCSC2 Cc1cc(C)c2cc(C(=O)NCCNC(=O)CCNS(C)(=O)=O)[nH]c2c1 N1(CC)CCC(N(C)CC2CCN(C(c3cc(OC)ccn3)=O)C2)C1=O C1(C(=O)OC)CCCCC1CNC(=O)NC(CC)(CC)CC c1(CC)cncc(C(=O)N(C2CCC2)C)c1.C1(C(=O)N)CC(C(F)(F)F)C1 c1(NC(C(C)C(C)(C)C)c2n(CCOC)nnn2)ccc(S(C)(=O)=O)cc1.O C(=O)(CCC(F)(F)F)N1C(CN(C)C(c2c(C(F)(F)F)ncn2O)=O)CCC1 C12(C(=O)NC3(C)CCCC3O)CC(C)(CN1C(C1CCC(F)(F)C1)=O)C2 C(=O)(C(C(C)(C)CC)OC)NCC(CC)NC(c1cc(C)c(C)cc1C)=O c1(CC)cccc2c1CCN(c1cc(NCC(C)(CO)OC)ncn1)C2 C(CCCC(=O)OC)(c1nnnn1CCCOC(C)(C)C)NC(CCSCC)C c1(C(N2CCC(Nc3c(C#N)ccnn3)C2)=O)ncn2ccccc12 Cc1cc(C(N2CCC(C(=O)Nc3ccc(O)c(F)c3F)C2)=O)ccc1[N+](=O)[O-] c1(C(=O)NCC(CNC(COCC#C)=O)O)ccc(F)cc1C(F)F Cc1cc(C(=O)N(CC(N2CCCC3CC23)=O)C)ncc1N Cc1ccc(C=CC(=O)NC2(C)CCC2)cc1Cl.C1(C=O)C2CCC(F)(F)C12 C12(NC(COCCOC)=O)CCCN(C(=O)COCCC(C)C)CC1C2 c1(C(N2CC(NC(c3nc(C4CC4)cs3)=O)C3C2C3)=O)noc2c1CCCC2 Cc1nc2ccc(C(N3CCCC(C)C3CNC(=O)C(=O)C(C)(C)C)=O)cc2[nH]1 C12CN(C(c3cnc(Cl)c(N)c3)=O)CC(F)(C1)C2.Cc1ccncc1C(=O)N.C C(=O)(N=S1(=O)CCN(C(c2cc(Cl)nn2C)C(=O)NCC2CCCO2)CC1)OC CC1CN(C(C2(c3cccs3)CCCC2)=O)CC1NC(=O)CCC1CC1(F)F c1(C(=O)NC2CC(F)(CNC(CC(COC)C)=O)C2)ccnc(OC)c1F C=CCC(C)(O)C(=O)NC(CC)CCC(=O)N1CCCC(C(C)C)CC1 CN=C(NCCOCC1CCOC1)NC1CCC(C(=O)OC)C1 c1(CC(=O)NCC2CCN(C(C3(CCC)CC3)=O)C2)nn(C)cc1Br N1(C(CCC#CC)=O)CCC(C2CCN(C(c3cccn3C3CC3)=O)C2)C1 c1(CCCC)nc(-c2ccc(COC)s2)n(Cc2csc(Cl)c2)n1 c1(CC)cccc(C(=O)NCCOC(C)(C)C)n1.C1(C#N)(C=O)CCC1 c1(C(=O)NCC2N(C(C=C(C)C)=O)CCCC2)noc2c1COCC2 c1(C(N2CC(C)C(NC(c3cn(C)nc3Br)=O)CC2)=O)ccc(C#N)c(O)c1 N1(C(c2c(OCC)ccs2)=O)CCC(NC(c2cc(C)on2)=O)C(CO)CC1 CC1C(=O)CCC1CC(=O)NC1CC(CC(=O)NCC(O)C2CC2)C1 C(=O)(CC(F)(F)CS(C)(=O)=O)NCCCN(C(CCc1nc(C)sc1)=O)CCO N1(C(c2c(C)nn(CC)c2C)=O)CCC(C2CCN(C(=O)CNC=O)C2)C1.N c1(C(N2C3(CNC(C(CC)OC)=O)CCC3CC2)=O)nn(CC)c2c1COCC2 [N-]=[N+]=NC1CN(C(c2ncoc2CNC(=O)CC2CC(=O)C2)=O)CC1O N1(C(c2c(C)ncnc2O)=O)C2CCC1CN(C(=O)CCCc1cnccn1)C2 N1(C(c2cc(C)c(C)s2)=O)CCC(F)C(NC(=O)CCSCC(N)=O)C1 C1(C(=O)N)CN2CC3CC2(CO1)C3.C1CCCCN1C(=O)C=Cc1cscn1.C C1(C(N2C(C(=O)NC3C(CN=[N+]=[N-])CCC3)CSC2)=O)CC2(CCC2O)C1 C(CCC)(CCCNC(c1ccsc1OC)=O)NC(C(CC#C)C1CC1)=O Cc1cccc(C2CC2C(N2CCCC2)=O)c1.C(=O)(C(C)(C)O)NC1CC1.C c1(CN2CCCC(NC(c3n(C)ncn3)=O)CC2)c[nH]c2nccc(Cl)c12 CCC(CC)C(C(=O)NCC(C)C(F)C(=O)NCC(C)(C)CCOC)OC C#CCCC(=O)N(CC(C)(C)CNC(c1ccc(CN2CCCC2)o1)=O)C C(C(=O)NCC1CCN(C2CC2)C1)(C(C)(C)C)NC(CCn1ccc(C)n1)=O Cc1[nH]nc(C#N)c1C(=O)NCC1CCC12CCCO2 CN(C)S(=O)(=O)NCC1CC1.c1(C(C=O)O)cccc(OC(F)(F)F)c1.C C1CC(C(=O)O)C1(C)C.C1(N(C)C)CC(O)C1CC=O.C1CCCC1C(=O)N c1(NC(C2CC2C(N2CCCC(Br)C2)=O)=O)ccc(I)cc1Cl c1(C(=O)NCC2(OC)CN(C(C3CCCS3)=O)C2)cc(Cl)cc(C)c1C c1ccc2c(c1)CCC2.Cc1cc(C(=O)NC2CC2CNC(=O)C)nnc1C CCC1=C(C(=O)NC2CCN(C(c3cncc(N)c3)=O)CC2(C)C)SCCO1 c1(C(=O)NC2CCN(C(C3CCN(C)C(=O)C3)=O)C2)cccc2sncc12 c1(C(=O)NCC2OCCN(C(Cc3cncc(C)c3)=O)C2)cccc(Br)c1N c1(C(N2CCN(C3CCC(C)CC3)CC2)C(=O)NCC=C)ccc(C#N)o1 c1(CC(=O)NCCC(C)NC(=O)CC23CCC(CC2)CC3)c(F)cccc1F N1(C(c2c(OC)nccc2)=O)CC2CCCC2(C(=O)N(C(CO)C2CC2)C)C1 c1(CC(N2CC(CC(C)NC(C3CC3c3ccsc3)=O)C2)=O)ccc(O)nn1 CCC(CCC(=O)N1CCC(CC(C)NC(=O)Cc2sccc2Cl)CC1)OC Cc1cnc(C(N2CCC(NC(=O)C(O)C(C)C)C(O)C2)=O)cc1C#N C1(CNC(c2n(C(C)C)nnc2)=O)CC2(CC2)CN1C(=O)CC(C)(C)C#N C1(CNC(C2N(C(N)=O)CCC2)=O)C2CC1N(C(C1CCC3CC3C1)=O)C2 N1(C(C(CCCCC)O)=O)CCC2(CCC(NC(C3(C)CCCOC3)=O)C2)C1 C1(C2CCC2)(C(=O)NC(CC2CN(C(C(CC#C)C3CC3)=O)C2)C)CCC1 CC(C)CC(CNC(c1ccn(C)n1)=O)C(=O)N1CCOC(CCF)C1 CC#CCC(C(=O)NCCCCC1CC1)NC(c1ccc(C#N)cc1)=O C(=O)(CCCCCCBr)NC1C(C#N)CN(Cc2cnc(Cl)c(F)c2)C1 C1(CNC(c2ccc(CSC)o2)=O)CN(C(=O)Cc2cnccc2Cl)CC1C CC(C)C(C)CC(=O)NC(C(=O)NCCC1CCCOC1)C(C)(C)C Cc1cc(NC(=O)CSCCNC(=O)COC2CCCCC2)cc(O)c1 N1(C(C2COC(C)(C)O2)=O)CC2(CCN(C(=O)C(c3ccccc3Cl)O)C2)C1 n1(C(C=O)(C)C)cc([N+](=O)[O-])cn1.C1(C=O)CN2CCC1C2.C1(CC)CC1.N c1(C=O)ccccc1.C=CC1(C(=O)NCC(C)C2CC2)CCC1.[SH](C)(=O)=O N1(C(Cc2ccc(OC)cc2)=O)CCC(NC(=O)CCc2ccoc2)CC1C N1(Cc2cn(C(C)C)nn2)CCCCC(C)(C)C1.C1(C)(C(=O)N)CCCS1(=O)=O C(=O)(C1Cc2ccccc21)NCC1(C(=O)NCC(CC)CO)CCC1 Cc1cc(N)c(C(N2CCC2CNC(C23CC(CCO2)C3)=O)=O)c(F)c1 CCCCC#CC(C)(C)NC(C1CN(C(c2ccccc2O)=O)CCN1C)=O CCC(C#N)(CC)C(=O)NCCN(CC)C(c1cnoc1C(C)C)=O.CCO C(=O)(C(C)C(O)C(C)C)N1CCCC(C(=O)NCCC(C(C)C)N(C)C)C1C C1(C(=O)N)CC2(C1)CC(C)(C)C2.C(CCC)OC.C1(C=O)CC1.C(C)=O N1(C(C2=NOC(C)C2)=O)CCC(NC(=O)Cn2nc(O)ccc2=O)CC(O)C1 N1(C(Cc2nnc(C)o2)=O)CC(CCNC(C2(CO)CCCC2)=O)C(C)C1 C(=O)(CC(O)CNC(=O)N(C)Cc1ccc(O)cc1)N(C)C c1(OC)ccc(F)cc1C(C)NC(=O)C(N1CCC(F)(C(=O)O)CC1)=O C12(NC(c3cc(C)nc(C)n3)=O)CCCN(C(=O)CCC3CCCCC3)CC1C2 Cc1ccc(O)c(C(N2CCCCC(N(C)C(c3nocc3Br)=O)C2)=O)c1 C(=O)(C1=CCCN(C(C2(O)CCSC2)=O)C1)NCc1n(C(C)C)ccn1 c1(NC(CC)=O)cccc(CC(=O)NC(CO)C(C)Nc2ccc(OC)cc2)c1 CC1(C2CC2C(=O)NCC23CC2CN(C(=O)CC)C3)CCOCC1.C(=O)CO C=CC(CC)CC(=O)NC1CN(C(C2(OCC)CCCCC2)=O)CC2CC12 N1(C(C(COC)(C)C)=O)CCCC(C2CN(C(C3CC=CC3)=O)C2)C1 C1=CC(=O)NS(=O)(=O)c2ccc1cc2.CC12CC1(c1ncc[nH]1)C2 C(c1c(F)cccc1F)=CC(N1CCCCC1)=O.C1(SC)CC(C(=O)N(C)C)C1 C(CN=c1[nH]c(=N)[nH]c(=N)[nH]1)(c1c(SC)cccc1)C1CCC1 N1(C(C(CC2CCC2)OC)=O)CC(O)CC1(C)C(=O)NCC(O)C(C)(C)O N1(C(C(CNC(c2cc(CCC)on2)=O)O)=O)CCCC12CCNC2=O C(=O)(C#CC1CCC1)N(CCC(C(C)C)NC(c1cccc(C(F)F)c1F)=O)C Cc1cccc(C(=O)NCCC2CCC(NC(=O)CCc3ccsc3)C2)n1 c1(N2CC(CCOC)OCC2)nc(C2CCCCC2)nc2sc3c(c12)CCC3 CC(C)C(C)(C)C(=O)N1CC2(NC(=O)CC3CCCCC(=O)N3)CC1C2 c1(OC)ccc(F)c(C(=O)NC(CNC(C2CCC2)=O)C2CCC2)c1F.O N1(CC(=O)NC(CC)C)CCCOC(CNC(c2ccccc2C2CC2)=O)C1 O=S(=O)(c1ccc(=NCC2CCOCC2)[nH]c1)NCC1(CO)CCCO1 C#CCCC(C(=O)NC(C)Cc1cc(C)[nH]n1)NC(=O)C(C(C)C)OC C1(C(=O)NCc2c(C)scn2)CC(NC(=O)C#CC(C)C)C1(C)C N1(C(c2c(CC)occ2)=O)CC2C3CCC(C2C1)N(C(C1CCSC(C)C1)=O)C3 c1(C(N2CC(NC(C3CC(F)(CO)C3)=O)CCC(O)C2)=O)cc(F)c(F)cc1Cl C1(C(=O)NCC(C(C)C)N2CCCC2)(OCC)CCCCCC1 c1(CC)noc2ncc(C(=O)NCC3CC(C)CO3)cc12 C1(OC)(CNC(=O)Cc2occc2C)CCN(C(=O)C(c2cccs2)S)C1 C1(CNC(=O)C=C2CCCC2)CN(C(=O)CSC(F)F)CCO1 CC(C)CCCNC(=O)C(c1cnccn1)C.c1(C(=O)N)n[nH]c(C(C)(C)C)n1 Cc1cc(C(=O)NC2CN(Cc3cc4n(n3)CCC4)CCC2C)c(F)cc1F c1(C(=O)NCC(n2cc(-c3ncccc3Cl)nn2)C)cnc2ccc(F)cc2c1 N1(C(C2CN(C(C)=O)C2)=O)CC2CC(C1)C2.c1(C=O)ccc(C(C)(C)C)nc1 c1c(F)cccc1F.CC(C)(CF)C(=O)NCCOCCNC(=O)C(=O)N c1(C(=O)NC2C(C)CN(C(=O)Cc3ccc(Cl)s3)CC2)ccc2c(c1)OCCO2 c1(CCNC(C2C(CNC(C3C(C)CC3)=O)C2)=O)ncccc1F C(CC(=O)N1CCSCC1C)(C(F)F)NC(c1c(OC)n(C)nc1)=O C12(NC(c3cc(F)cc(F)c3)=O)CCN(C(c3cc(Br)cs3)=O)CC1C2 C1(CC)C(C(=O)NC(Cc2ccco2)C(=O)NCCCC(N)=O)CCN1C C1(N(C(=O)CCc2cccs2)C)CCN(C(c2ccsn2)=O)CC12CC2 N1(C(C(Cc2cnc[nH]2)NC(c2ccnc(C)n2)=O)=O)CCC(O)CC(C)C1 c1(OC(C)C)cc(NC(=O)CC2CNCC(C)(C)O2)ccc1C(N)=O n1(CC)c(CNC2CCCC2C)cnc1C c1(C(=O)NCC(C2CCOC2)NC(Cn2c(=N)nc[nH]2)=O)cccc2cncn12 c1(C(=O)NCCNCCO)cc2c(-c3c(O)cccc3F)cccc2s1 C(=O)(C(C)(C)C(C)C)NC(CCNC(c1scc(C)c1)=O)C C1(C)CCN(C(c2n[nH]c(C)c2Cl)=O)C1.C(C(C(=O)NC)NC(C)=O)OC c1(CNC(=O)CCc2ccc3c(c2)OCCO3)nc2c(C(=O)O)cccc2s1 c1(C(=O)NCC(CO)NC(C2(C)CCC23CCC3)=O)ccc2ccccc2c1O c1(OC)cc(F)ccc1C(=O)NCC1CN(Cc2cnn(C3CC3)c2)C1 C1(NC(Cc2ccn(C)n2)=O)CC2CCC1CN(C(=O)CCC1(C)CC1)C2 CC(C)CC(C)CC(=O)N1CCCCC1CCNC(c1cc(N(C)C)ccn1)=O C(=O)(C(C)C(CC)CC)N1CCC(NC(C(C(=C)Cl)(C)C)=O)C1 C1(CNC(c2cc(C3CC3)ncn2)=O)C2CCC(C2)N1C(=O)C(F)F N1(CCCNC(C(=O)NCC(c2ccccc2)N(C)C)=O)CCNCC1 CC(C)(O)CCCN=C(NCC1CC1)N1CCCC2(C=C2)C1 C1(Cn2cc(CCC(C)(C)O)nn2)CCCN(C(=O)CCc2ccoc2)C1 c1(CNC(c2cccc(C(N)=O)c2)c2n(C(CC)C)nnn2)c(C)cnn1C C1(C(N2CC(NC(C(C(=O)OCC)F)=O)C2)=O)COC(C)(C)CO1 N1(C(CC(CC)OC)=O)CCN(C(c2ccc3c(c2)CC3)=O)C(CF)C1 O=C1CC(C(=O)NC2(CC)CC2)NC(=O)N1.C1(C(=O)N)CC2CCC(C1)S2 C1CN(C(c2cccc(Cl)c2)=O)CC(C)(C)C1.C1(C(=O)N)(OCC)CCSCC1 c1(C(=O)NCC23C(CN(C(Cc4cc(C)no4)=O)C2)C3)c(Cl)ccc2c1OCO2 CN1CCN(C(=O)C=Cc2cscn2)C(CNC(c2csc(C#N)c2)=O)C1 CC1CC(NC(=O)CCOCC2CCC2)CCN1C(=O)CCO.C1CCCC1 Cc1cc(C(=O)NCC2CCCC2C(=O)NC2(C(O)CO)CC2)oc1C c1(C(=O)NC2(CO)CN(C(C(COC)(C)OC)=O)C2)cn(C)c(C)cc1=O c1(C(N2CCC(CNC(C(C)OC3CCCC3)=O)C2)=O)cnn2c(=N)[nH]cnc12 Cc1c(C(=O)NC2CC(F)(C)C2)sc2ccc(Cl)cc12.C(=O)CC1CC1.N Cc1cc(=O)c(C(=O)NCCCCC(=O)NC2CC(C)(O)C2)c[nH]1 CC(C)C(F)(F)CCNC(=O)C(c1cccs1)NC(C1CC12CC2)=O C#Cc1cn(C)nc1C(=O)N(C(C(=O)N1CC(O)C(O)C1)C(C)CC)C c1(C(=O)NC2C(C)N(C(=O)CS)CC2)cnc(Cl)c(C2CC2)c1.c1ccccc1 c1(C(=O)NCC2(CNC(c3c(C)coc3C)=O)CC2)nc(Cl)ccc1N N1(C(C(c2cnccn2)C)=O)CCC(OCCNC(=O)CSc2nccn2C)C1 C(C#Cc1ccc(I)cc1)NC1CCN(c2cccc(C)n2)CC1 C(=O)(CC(C)(C)CN(C)C)N1CCC(C(=O)N)(CC)C1.C1CC[Si](C)(C)C1 c1(OC)cc(C(=O)N(CCCCN(C(=O)C(c2cccnc2)C)C)C)ccn1 C=C1CCC(C(=O)NC2CCOCC2NC(=O)C=CC(=O)N(C)C)CC1 c1cccc(F)c1.N1(CC(C)C)CCCC1C(N1CC(C(C)NC(=O)C)C1)=O C1(C)(C(=O)NCCCC2N(Cc3onc(CCCC)n3)CCC2)CCNC1=O N1(C(CCOCC#C)=O)CC2(NC(c3cc(CC)cc(F)c3)=O)CCC1CC2 C=CCN(OC)C(=O)C1(COC)CN(C(=O)CC2COCCO2)C1 c1(N2CC(C(C)NC(=O)C3=CCCCC3)C2)cc(=O)n2cc(Cl)ccc2n1 CCC(C)C(O)CC(=O)N1CCC(N(C(=O)CC2CCC2)CCO)CC1 N1(C(C(c2ccccc2)OCC)=O)CCC(CN(C(=O)C(C)C)CC)C1.S C1(OC)(CNC(=O)CC2CCOCC2)CCN(C(=O)Cc2cncnc2)C1 c1(CN(CCCN(C)C)C(CC2CC2)C2CC2)ccccc1 Cn1nc([N+](=O)[O-])cc1C(=O)N(CC)C1CC1.C(=O)(CC(C)(C)C(F)F)N CCC(COC)C(=O)N(C(C)CN(C(=O)CCC(=O)Nc1nnc(C)s1)C)C CCC(C)C(C)C(=O)N(CCCCC(=O)N(CC(C)(F)F)C)C CCC(C)(C)CCCC(=O)N1CCCCCC1CNC(C1CCCN1C)=O N1(C(c2c(C)cccc2O)=O)CCC2CN(C(c3cc(Br)no3)=O)C2C1 C1(C)(NC(C(C)Cc2ccccc2)=O)CCCC1NC(=O)C=Cc1cnc[nH]1 c1(C(N2CC3CC3C2)=O)cc(F)cc(F)c1.C(=O)(C(C)(C)C=O)OCC.N c1(C(=O)OC)nc(C(=O)NCC(C)CNC(=O)CCc2nccn2C)co1 c1(C(=O)NC2CC3CN(C(CCc4cc(C)on4)=O)C2C3)csc(S(N)(=O)=O)c1 c1(SC)cc(C(=O)NCC2CC(O)CN2C(c2cnsc2C)=O)oc1C Cc1cc(C2CC2)ccc1C(=O)NC.C1(C(NC)=O)CC2CCC1C2.C1CC1 c1(N2CC(CC=C)(NC(c3cc(C(F)(F)F)cs3)=O)C2)nc(C)ncc1F Cc1cc(=O)c(NC(C2CCCN(C(c3ccc([N+](=O)[O-])o3)=O)C2)=O)c(C)[nH]1 C12(NC(C3CN(C(C)C)C3)=O)CCC(C(N3CCC(C#N)C3)=O)(CC1)C2 c1(C(=O)OC)cc(C)c(NC(c2cn(CC3CCCN3)nn2)=O)nc1OC c1(C(=O)NC2C(CNC(=O)CCCc3cnccn3)C2)ccc2nnnn2c1 C(CC(C)CC)(C(=O)NCCCC(C)(C)O)NC(C(C=C)OC)=O O=C(CCC(F)(F)F)NC1CCCC1NC(=O)Cc1c[nH]ccc1=O N1(C(c2cccc(OC)c2C)=O)CC2CN(C(C3CC(O)CN3C)=O)CCC12 N1(CCC)CCC(NC(=O)CC2CC(C)N(C(c3[nH]ccc3C)=O)C2)CC1 C(CNC(=O)C(Cc1cccc(C)c1)CC)(CC(F)(F)F)NC(C=CC)=O N1(Cc2cnc(SC)nc2Cl)CCC2C1CCCN2c1cc(N(C)C)ncn1 Cc1cc2occ(C(=O)NC(C)CNC(c3cc4n(n3)CCCO4)=O)c2cc1C C12(NC(c3cn(C)c(Br)c3)=O)COC(C1)C(NC(C1CNC(=O)N1)=O)C2 C1(CC)CCCCN1C(=O)C(=O)C1CCCC1.c1(COC)nc(CC(=O)N)cs1 C1(NC(C(CC)=CCCC)=O)(CO)CCCN(C(c2oncc2CC)=O)C1 CCCC(C)CC(=O)N1CCC(C)C1CNC(c1c(C)nsc1NC1CC1)=O C(=O)(CCCCCC=C)NC1CCC(CCC(=O)NCCC=C=C)C1 N1(C(C(n2cc(C3(n4ccnn4)CC3)nn2)C)=O)CCS(=O)C2(CCC2)C1 Cc1cc(C(=O)NC2CC23CCN(C(C24CCC2C4)=O)CC3)cc2cccnc12 N1(C(C(C(CC)C)O)=O)CCn2nc(CNC(c3cnc(C(C)C)[nH]3)=O)cc2C1 C1(N(C(c2cc(CC)no2)=O)C)CCC(NC(c2ccc(C)cc2)=O)CC1 c1(CC)c(Br)c(C(N2CC(C)(CC(=O)Nc3ncc(I)cc3I)C2)=O)nn1C N1(C(CCC(C)CN(C)C)=O)CCC(N=[N+]=[N-])(C(=O)NCCCc2cnn[nH]2)C1 c1(N(c2ccccc2)C2C(C)C2)[nH]c(=NC2CCCC2)nc2c1ncn2C O=S(=O)(c1ccc(N2CC3CC(O)CC3C2)c2cnccc12)N1CCCCC1 N1(C(=O)CC2(O)CCCCC2)CC2CC1CN(C(=O)C(=CC1CCCCC1)F)C2 c1(C(c2nnnn2-c2ccccc2Cl)NC(C)CCC2CC2)cccnc1O CCCCC(O)C(=O)NCCCC(C)NC(=O)Cc1ccc(Cl)c(OC)c1 Cc1ccc2nsnc2c1S(=O)(=O)Oc1cccc(OCC(=O)O)c1 N1(C(c2cc(C(C)C)[nH]n2)=O)CCCCC1CNC(=O)C(C)c1cc[nH]n1 Cc1ncnc(C)c1C(N1CCC(O)C(NC(=O)C(c2ccc(Cl)cc2)C)C1)=O c1(C(=O)N)c(C)nn(C2CCCCO2)c1C.CCCC(=O)NCC(=O)NC1CC1 c1(N(CC(C)C)CC)ccc(-c2nccn2C(CO)CO)cc1-c1cnsc1 CCCCCC(C)CC(=O)NCCOCCN(C)C(c1cccc(F)c1)=O C(c1cccc(O)c1)=CC(=O)NC1CN(C(C2(C)N(C)CCC2)=O)CC1C(F)F N1(C(c2cnoc2)=O)CCCC(C2CCN(C(C3(O)CCSC3)=O)CC2)C1 CC1Cc2cc(CC(=O)N(CC(C)O)CCNC(C3(F)CCC3)=O)ccc2O1 c1(C(=O)NCC(CNC(C(c2scc(C)n2)(F)F)=O)C)c(C)cc(Cl)cc1N C1(C(F)F)CC(=O)N1.C(C1CCCC1)=C(C)C(=O)OCc1nc(C(C)C)no1 c1(C(N2C(C(=O)N(CCCO)C)(CC)CCC2)=O)cc(C)cc(F)c1 c1(C(C(=O)NC(CC)(C)C)N(CC(C)OC)CC(F)F)cc(SC)nn1C N1(C(C(C)OCCOC)=O)CCC2(CCC(N(C)C(C3CCCCS3)=O)CC2)C1 C1(CNC(c2c(C)noc2)=O)CCCCC1N=c1nn[nH]n1C N1(C(C2C(NC)CCO2)=O)CCN(CC)CC1.c12cn(nn1)CC(C)NC(=O)C2 Cc1ccc(Cl)c(C(=O)NC2CN(C(c3cnccc3Cl)=O)CCC2F)c1O CONC(=O)C(=O)NCc1ncccc1C(=O)NCC12CCN(CC1)C2 N1(c2cc(C)nc(-c3ccc4oc(=N)[nH]c4c3)n2)CCOC2(CCCSC2)C1 Cc1cnc(NCc2ccc(F)cn2)c(S(=O)(=O)N(C)Cc2cc(Br)no2)c1 C1(CC(N2CC(C)(NC(=O)CC3COC(=O)N3)C2)=O)CCCCC(=O)N1 C1(C(=O)NCC#CCNC(C2CN(S(CC)(=O)=O)C2)=O)CCCC(C#N)C1 N1(C(C(C2CCCCC2)OC)=O)CC2CC1CN(C(c1ccc(C)n1C)=O)C2 C1(CC(=O)NC(C)Cn2cc(CCO)nn2)Cc2ccc(Br)cc2C1=O Cc1ccc(C)c(N(C(=O)CC2CN(C(=O)C3=NNC(=O)C3)CC2C)C)c1 Cc1ncc(C(=O)NC23CC(C(=O)NCCCc4cc[nH]n4)(C2)C3)s1 N1(C(C2CC(C3CC3)C2)=O)CCC2(C(=O)NC3CC4CCCC4C3)CCCC12 Nc1cnc(C(=O)NCCc2nc(-c3ccccc3)n[nH]2)cn1 c1(-c2n(CC(C)CO)nc(C3CCC3)n2)ccnc2[nH]cnc12 c1(C(N(CC(O)CNC(=O)CN2CC3CC3C2)C)=O)ccccc1.C1CCC1 N1(C(C)=O)CC(NC(C2(CC(=O)NC(C3CCCC3)=O)CCCC2)=O)CC1C Cc1ccc2[nH]nc(C(=O)NC(C)C3CC3)c2c1.c1(CC(=O)N)ccc(F)cn1 C1(CNc2n(-c3ccccc3)cnc2)CCC2(CCCOC2)O1.C12COCC1O2 c1(CC)ncncc1C(N1CCC(F)(C(=O)NCC23CCC(CC2)C3)C1)=O N1(C(c2c(=N)[nH][nH]c2)=O)CCCCC(NC(=O)CC2CN3CCC2CC3)C1 Cc1cccc2c(C(=O)NC3CCC(C)N(C(c4n[nH]cc4Cl)=O)C3)n[nH]c12 Cc1cc(C(N2CCC(NC(C34CCC(CC3)C4)=O)C2)=O)c2ccccc2n1 N1(C(C2N(C(C)=O)CSC2)=O)Cc2ccnn2CC(NC(=O)C(=O)N(C)C)C1 N1(C(C)=O)CCCC(C(N2CC(O)(C(C)NC(c3oncc3C)=O)C2)=O)C1 Nc1ncc(C(=O)NCC2(NC(C3CC3C(F)(F)F)=O)CCCC2)cc1 C(CCO)(C(=O)NCCCC1CN(C(=O)Cn2cccc2)CCO1)N(C)C Cc1ccc2cc(C(N3CCC(NC(C4CCCNS4(=O)=O)=O)C3)=O)ccc2c1 c1(C=O)cc(=O)cc(Cl)[nH]1.C1(C)(C(N(C)CC)=O)C(C)(C)C1(C)C.CC c1(C(=O)NCCCNC(c2nc(OCC)oc2)=O)ccc2c(c1)CNC2=O Cc1cn2c(C(=O)NC(C)C(C)NC(c3cnc(C4CC4)nc3C)=O)cnc2s1 C(=O)(CC(O)C)NC1C=CC(C(=O)NC)C1.c1(CC(=O)N)c(C)noc1C C1CCS(=O)(=O)C12CN(C(C1(C)CC(=O)C1)=O)C2.Cc1cnc(C=O)c(C)c1 c1(SC)cn(C)nc1C(N1CCC(C)C1)=O.c1(C(=O)N)ccc(N(C)C)nc1 CC(C)(CC(=O)NC1(C(F)F)CC(NC(c2ccoc2)=O)C1)c1ccccc1 N(C(=NCCCc1ccc(Cl)c(Cl)c1)NCc1cccs1)C(COC)C N(C1CCc2cc(Br)ccc21)C(c1c(C)sc(CN)n1)=O N1(C(C(c2ccccc2)SC)=O)CCC(O)(CO)CC1.c12cnn(c1)CC(=O)N2 N1(C(Cc2c(C)nc(S)s2)=O)CCC12CN(C(C1CC3CCC1O3)=O)C2 c1(C(N2C3CC(CNC(C(C(CC)C)O)=O)C(C3)C2)=O)cc(=O)c(OC)cn1C CCCC(C)CCCC(=O)NCCCC(C)NC(=O)COc1ccc(F)c(C)c1 C1(C)(C(N(CC(C)(C)CNC(=O)C(F)C(F)(F)F)C)=O)Cc2ccccc2C1 c1(C(N(CCC)CCNC(=O)CCC2CC2C)=O)cccc2nsnc12 Cc1cc(C(N2CC3CC(NC(=O)Cn4cnnn4)C2C3)=O)cnc1C(F)(F)F N1(C(C(CCCC)NC(=O)Cc2cccc(C)c2)=O)CC2CC(O)CC1C2 C(C)(CO)(C(=O)NCC(C)(O)CNC(c1cccc(C)n1)=O)OC C1(NC(CC2(C)CCN(C(c3c(C)ccn3C)=O)C2)=O)CC(C)(C)OC1=O CC(C)(C)CCC(=O)C(=O)NCCC1CCN(C(c2cc(Br)co2)=O)CC1 C1(OC)CC(CO)N(C(=O)C#CCNC(c2cc[nH]c2)=O)C1 Cc1ccnc2c(C(=O)NCC(C)(O)CNC(=O)C)cnn12.CC(F)(F)F.S C1(CNC(C2(SC)CC(O)C2)=O)CCC(C)CN1C(c1ccc(C)cn1)=O C1(C(N(CCC(=O)NC(c2ccnn2C)C)C2CC2)=O)OCC2CCCC12 c1(C(N(CC(O)CN(C)C(c2cn(C)cn2)=O)C)=O)nccn2cnnc12 c1(C(=O)NC2(CNC(C(C)OCOC)=O)CC2)ccc2ncc(=O)[nH]c2c1 C(C)(C)(CC(=O)NCC1CC(O)(C)C1)SC.C1(F)(C(=O)N)CCCOC1 Cc1c(Cl)cnn1CC(N1CCCC1CN(C)C(c1ccncn1)=O)=O C#Cc1ccc(C(=O)NC2CCCCC2NC(C2(c3ccc(C)nc3)CC2)=O)o1 N1(C(c2cccc(Br)n2)C(=O)NCCSC)CCCC2(CCCC2)CC1 c1(C(=O)NCCC(CNC(CCC=CC)=O)OC)c(C)ccn1C N1(C(c2c(C)c(Cl)ccn2)=O)CC(C)N(C(c2cccn3ccnc23)=O)CC1C Cc1cc(F)c(NC(C2(NC(=O)CC3C=CCCC3)CSC2)=O)cc1F Cc1cc(C(=O)NC2CN(C(C3(C)CC=CC3)=O)CC23CC3)c(O)c(C)c1 Cc1nc(C)n(CC(=O)NCCC2CCCN(C(C3(n4cccn4)CC3)=O)C2)n1 C1(NC(c2cc(F)n[nH]2)=O)CCN(C(c2c[nH]cc2Cc2ccccc2)=O)C1 C1CCC(F)(F)C1.c1(CNC(C2CC(CC)C2)=O)cc(C(=O)N)n[nH]1.C C1(N(C2CCC2)C(=O)N)CCCN(C(c2ncccc2F)=O)C1.O=CC.C1CC1 C1(C#N)(C(=O)NC2CC(CNC(C3CCCC(C)O3)=O)C2)CCSCC1 C(=O)(C1CC(=O)Nc2ccc(Br)cc21)NCC1C(C(C)C)OCC1 c1(NC(=O)NCC2(O)CS(=O)(=O)C2)cccc2ccncc12 N1(C(CN(C)CCO)=O)CCN(C(=O)COCC(F)(F)F)C2CCCCC12 C1(CC)CC(C(=O)NCc2cn(C3CCC3)nn2)CCO1.C12CC1CNC2=O.N N1(C(C2(SC)CC2)=O)CC(CNC(=O)CC2CCCCO2)CC(C)(C)C1 C(CC(CC)C(=O)NC1C=CCN(C(c2c(NC(C)=O)c[nH]c2C)=O)C1)=CC N1(C(c2cnc(CC)[nH]2)=O)CC2CCC1C(CNC(=O)C(O)CSC)C2 C(=O)(CC(C)P(C)(C)=O)N1C(CN(C(c2c(C)nn[nH]2)=O)C)CCCC1 Cc1cnn(C)c1NC(N1CCC(CC2CC2)C1C)=O C(C(CO)C(C)C)N(CCCC=CC)N(c1ccncn1)Cc1ccnnc1C N1(C(C(CNC(C(CC#C)O)=O)O)=O)CCC(C)CC1C CC(C)(CNC(C1CCCC1NC(C1(Cc2ccccc2)CC1)=O)=O)CO c1(C(c2nnnn2C2CC2)NCCCS(C)=O)ccc(S(N)(=O)=O)cc1 CC(CC(=O)N1CCNC(C(N2CCC(F)(CO)C2)=O)C1)CC(C)(C)C N1(C(c2n(CC#C)ccc2)=O)CCC(CO)(NC(c2csc(C)c2OC)=O)C1 c1(C(=O)N)cc2c(s1)CCOC2.C1(CNC(CC2C(C)C2)=O)CCC(C)CC1 c1(C(C(=O)N(CCN(C(C2C(CC)OCC2)=O)C)C(C)C)C)ccccc1C CN1CC(C)(C)CC1C(=O)NC1(C)CCN(C(c2ncc(N)cc2Cl)=O)C1 c1(C(=O)NCC2(CNC(CC=C)=O)CC23CCC3)ccc2occ(C)c2c1 C1(NC(COC(CC)(C)C)=O)CCCC(C(=O)N)C1.C1CCC2(C(C)C)CC12 N1(c2snc(C)n2)CCC2CCN(C(c3cc(CN(C)C)c[nH]3)=O)CC2C1 C1(C(=O)OC)CCCCCCN1C(=O)C(=O)NCc1ccc(CSC)o1 Cc1cc(CCC(=O)NC2COCCN(C(C3(C)COC3)=O)C2)ccc1Br c1(C(N2CC(Nc3nccc(C)n3)C3(C2)CC3)=O)ccc2nc(O)[nH]c2n1 C(=O)(CCCC(F)(F)CO)N(C1CCN(C(C=Cc2c(C)n[nH]c2)=O)C1)C CCC(CC)C(CCN1C(=O)CC(c2cccc(Br)c2)NC1=O)OC C(CC(F)CN=[N+]=[N-])NC(C1C=CC(NC(C2C(C)(C)C(=O)C2)=O)C1)=O C(=O)(C#CC1CCCO1)N1CCC(N(C(C(C)(F)F)=O)CCO)CC1 C1(NC(=O)C2=CCC2)CCCCC12CCN(C(=O)CCc1ccc(CO)cc1)C2 c1(CC(=O)NCC2CN(C(CCCC(C)C)=O)CC2C)cnn2c1CCCC2 C1(C(N2CC(C)(CCC(=O)NC(CO)CCC3CC3)C2)=O)CCOC1(C)C c1(C(N2C(C)(c3cn(CCC(=O)OC)nn3)COCC2)=O)c(C)cc(F)cc1C N1(C(C2CCCO2)=O)CCC(C)(C)C1.c1(C=O)nc(C(F)(F)F)cs1.CO.C CCC(C(=O)NCCCC1CCCN1c1nc(Cl)ncc1OC)C(C)C O=C(C1CCCn2ccnc21)NC1COC2(CCN(C(c3cc[nH]n3)=O)CC2)C1 Cc1cc(N)cnc1C(N1CCN(C(c2ccccc2OCC(N)=O)=O)CC1)=O CN1C(=O)CC(C(=O)NC(C)(C)CNC(C2CCCC2)=O)C1c1cccs1 c1(C(N2CCC(NC(C3(C)CCCC3)=O)C2C2CC2)=O)cnc2c(Cl)cccn12 c1(C(N2CCCCC(NC(CCC3(C)CC3)=O)C2)=O)ccn2[nH]c(=N)nc2c1 c1(NC(=O)NCc2cc(C(F)F)c(Cl)cn2)cc(Br)cc(C(F)(F)F)c1O O=C(C1=CS(=O)(=O)CCC1)NC1COC2(C1)CN(C(=O)CC1CSCCS1)C2 c1(NC(c2cc(O)ccc2Cl)=O)cccc(F)c1.[SH](=O)(=O)CCc1ccccc1.N CC1CCC(C(=O)NCCC2CSCCN2C(=O)Cc2ccc(F)cc2)CC1 C1(C(N(CC(COCC)O)C)=O)C(C)CCN1C(=O)Cc1ccsc1C C1(C(=O)NCC(c2ccccc2)N(C(C=CSC)=O)C)CCCCN1C(C)=O CCCCC(O)C(C)C(=O)N(C(CNC(=O)CC(C)(C)C1CC1)CC)C C1C2CC1CN(C(c1ccc(=O)n(C)n1)=O)C2.c1(OC)nsc(OC)c1C=O.N c1(C(=O)NCCCC(C)NC(C2(CO)CCCC2)=O)c(F)ccc2[nH]ccc12 c1(OC)ccc2[nH]c(CN3CCC3(C)C(=O)Nc3cccnc3CO)cc2n1 C12(NC(c3c(C)nn(CC)c3)=O)CCCC1CN(C(C1CC1c1cn[nH]c1)=O)C2 C(CC(C)(C)NC(c1csc(-c2ccc(Cl)s2)n1)=O)NC(C1C(C)C1)=O c1(CCCC)ncc(C(N2CC=CC2CNC(=O)C(C)(C)N2CCCCC2)=O)s1 c1(OC)ccc(C)nc1C(N1CCCC1C1CCN(C(=O)CCC(C)OC)CC1)=O CC(C)(CCC(=O)N1CCC(CNC(c2nonc2N)=O)CC1)[N+](=O)[O-] c1(C(=O)Nc2cc(C)c(F)nc2)nc2cc(-c3cccnc3F)ccc2[nH]1 N1(C(C(COCC)(C)C)=O)CCOCC(NC(=O)NC(C)(C)C)C1 c1(CNC(CC2C(CC)C2)=O)ccc(C)cc1.C1(C(C=O)F)CCCCC1.N Cc1ncc(C(=O)NC(C(=O)NC(C(N)=O)C2CC2)c2cccs2)cn1 N1(C(Cc2c(C)nsc2)=O)CC(C)CCC1C(=O)NCCC(C)c1cn[nH]c1 Cn1nc2cc1C(=O)N2.C1(C)(C(=O)NCCC23CC(C2)C3)CC2CC2C1 c1(CC(N2CC3C(NC(C(COC)OC)=O)C3C2)=O)ccc(C)c(C)c1 c1(C(=O)NC2CC(C(=O)NCCNC)C2)cccc(O)n1.c1ccccc1.C C(C(=O)N(CC(=O)N(C)C)C)(C(C)O)NC(CNC(CC)=O)=O c1(C(=O)NC(CC)CNC(c2cnc(Cl)[nH]2)=O)cc(C)cc(C)c1Br C(CCCN=c1ccnc(N(C)Cc2cccnn2)[nH]1)N(C)C C1(O)(c2cn(C3CC(C(N(C4CS(=O)(=O)C4)C)=O)C3)nn2)CN2CCC1CC2 c1(NC(CCN(C(c2ccn(COC)n2)=O)CCO)=O)cnc(Cl)c(C)c1 C(=O)(C(C)CC1CCCC1)NC1(CC)CC1.c1(C(C(=O)N)C)ccc(C)o1 CC1(C)CC(C(=O)NCC2CCCC(NC(=O)C(N)=O)C2)CCO1 Cn1nc(C(N2CC(CNC(=O)CC3OCCC3(C)C)C(O)C2)=O)cc1CO CCS(=O)c1ccccc1C(=O)NCCCCOC.C(=O)C(F)=C(C)C1CC1.N c1(CCC(=O)N(C)CC2(O)CCN(C(C3CCC(O)C3)=O)C2)c(F)cccc1F N1(C(c2n(CC)ccc2)=O)CCCC2(CCN(c3nc(Cl)ncc3Cl)C2)C1 c1(SC)ccc(C(=O)CCC(=O)N2CCC(CF)(NC(=O)C(N)=O)C2)cc1 N1(C(c2cn(C)c(O)n2)=O)CCCC2(CCN(C(C3CC3CC(C)(C)C)=O)C2)C1 C1(n2cc(C3CCN(C)C3)nn2)(NC(C(c2scc(C)n2)C)=O)CCOCC1 C1(C)(NC(C(C)OCC2CC2)=O)CCN(C(c2cc(Cl)ccc2Br)=O)CC1 N1(C(C2C(C(C)NC(=O)CCc3cn(C)cn3)C2)=O)C2CSCC1C2 C=CC(F)(F)C(=O)NCC(C)N(C(=O)CC1CCC12CCC2)C c1(C(=O)NC23CCC(CN)(CC2)OC3)cc(=O)c2c(O)cccc2o1 c1(C=O)cc(C(C)(C)C)oc1C.C(C(=O)NC1CC1)(c1cccs1)OCC c1(C(=O)OC)cc(NCc2ccc(-n3cc(Cl)cn3)cc2C)cc([N+](=O)[O-])c1 C1(CNC(c2c(C)nco2)=O)(NC(C2CCC2F)=O)CCCCC1 c1ccc(F)cc1.C1(CCC(=O)NCCNC(CNCC)=O)CCC(C)O1 c1(C(=O)NC2C(NC(c3nc(CC)oc3)=O)CCC2)sc2ccc(Cl)cc2c1C c1(CN(C)C(C2CCN2C(c2cscc2Cl)=O)=O)cnn(C)c1 N1(C(C2(OC(C)=O)CC2)=O)CC(C)(CC(=O)NCCn2cccn2)C1 N1(C(COC2(C#C)COC2)=O)CCC(C(=O)NCc2ncc(CC)s2)C(O)C1 C1(C(N(C2CCN(C(=O)CC3CCCCC3O)CC2)CCO)=O)CC1C1CCCC1 C=CCC(CC(F)F)C(=O)NCC1(C)CCCN1C(C1CC(O)C1)=O S(=O)(=O)(C1CCC2(CC1)CC2(F)F)NCC(C(C)C)OC C1(CNC(c2cc(OC)no2)=O)CC2(CCN(C(C3CC3Cl)=O)CC2)C1 C1(CNC(c2cnn(CCC)c2C)=O)CCC2(CN(C(=O)C(O)CF)C2)O1 C(=O)(C(C(C)C)C(C)C)NC1CC(OC)CN(C(CC(CC)SC)=O)C1 c1(C(N2CCSC(C)C2C)C(=O)NC)cc(C)cc([N+](=O)[O-])c1 C1(CCNC(CSCC)=O)CN(C(=O)Cc2ccc(F)cc2)CCS1(=O)=O CS(=O)(=O)c1cc(Br)ccc1C(N1CCN(C(c2ccc(Cl)o2)=O)C2CC12)=O C1(NC(CC2CC(C)C2)=O)C2CC(O)C1N(C(=O)CN(CC(C)(C)C)C)C2 C1CN(C(C2(C(=O)C3CC3)CC2)=O)CC12CCC2.C1(CC(=O)N)CCC(O)C1 c1(NCCCCC#C)ccc(-c2ccc(OCC)cc2)cc1F C1(C(=O)NCc2c(C(N(C(COC)C)C)=O)con2)CCCC(=O)CC1 C1(CNC(C(=O)NC(C)C)=O)CCOCC1.N1(CC=O)CCC1C.CC.O C12(NC(c3cnc4cccnn34)=O)CCCC1N(C(c1n[nH]cc1Cl)=O)CCC2 Cc1cc(Cl)c(C(N2CCCC(CCNC(c3cc4ccsc4[nH]3)=O)C2)=O)cn1 CC1(C)CC(NC(c2cccs2)=O)CN1C(=O)Cc1coc(C(F)F)n1 C(=O)(C(C(C)(C)C)NC(C1CCN1C(C)(C)C)=O)N1CCCC(CCC#C)C1 C1(C(=O)NCCC(C)N2CCC2)CCCN(C(C2CC2c2ccco2)=O)C1 C=C(C)CCCC(=O)N1CCN(C(C2CCC(COC)C2)=O)C(C(C)C)C1 C(=O)(C(CNC(c1cocc1C)=O)C(C)(C)C)NCc1nccc(C)c1 CN1CCOC2CN(C(C3N(C(C4CNC(=O)O4)=O)CCC3(C)C)=O)CC12 Cc1ccc(CC(CNC2(Oc3cccc(Br)c3)CC2)C(=O)O)cc1 c1(C(N2CCCCC(NC(=O)CC3CC4(CC4)CO3)C2)=O)cccc2c1NCC2 CC(CC(=O)NCCC1CC2CCC(C1)N2C(c1ccc(C#N)o1)=O)C(F)(F)F C(=O)(C(O)CC(F)(F)F)N1CCCCC(CNC(C2(CSC)CC2)=O)C1 c1(CCCNC(c2cc(F)c(Br)cc2F)C)nnc2n1CCCCC2 C1(CC)(NC(c2cnc(Br)s2)=O)CCCN(C(c2ncccc2N)=O)C1 c1(C(N(C2C3CN(C(C(CC)C)=O)CC32)C)=O)ccc2c(c1)NC(=O)CN2CC c1(NC2(CNC(=O)C=CCF)CC2)ccc(O)nc1Cl N1(CCC(N2CCC(CCC)(CO)C2)=O)C(=O)c2cccc([N+](=O)[O-])c2C1=O c1(C(=O)NCCN(C(C)C)C(c2nccn3ccnc23)=O)cc2cccnc2o1 c1(-c2n(CCCC)ccn2)ccc(F)c(-c2ccc(F)cc2OCC)c1 c1(OC)ncnc(N(C(=O)CCc2cccc(C)c2)CC2(C)CNC2)c1C c1(C(N(CCC(N2CC(N=[N+]=[N-])C2)=O)CCCO)=O)cc(O)ccc1F c1(OC)cccc(C(O)CN(C(=O)CCc2ccc(N(C)C)cc2)C(C)C)c1 C(CCCCCC(=O)OC(C)(C)C)CC1C(C)CCN1Cc1nccc(Br)c1C C#Cc1cccc(CC(=O)N(C2(C(=O)NC3(C)CCOC3C)CC2)C)c1 c1(NC(C(C2CCCOC2)N)=O)ccc(Cl)cc1CO c1(CNC(C(c2[nH]nc(CC)n2)N2CCCC2CC)=O)ccc(OC)cc1 N1(c2n(CC=C)c(COc3ccc(F)cc3)nn2)CCCC2(CCOC2)C1 c1(C(=O)NCC2CCN(C(Cc3c(Cl)cn(C)n3)=O)C2)cnc2ccoc2c1 N1(C(C(C)(C)N(C)C)=O)CCCC(O)(CNC(=O)CCc2ncc[nH]2)CC1 C1(C(=O)NCC(C)(O)CNC(=O)CCC2CCOCC2)CC12CCOCC2 C1(CC)(NC(=O)CN(C2CCSC2)C)CCN(C(c2cc(F)c[nH]2)=O)CC1 c1(N2CC3OCCN(S(CCCC)(=O)=O)C3C2)ncnc2cc(C)ccc12 c1(CNC(C2SCCN(C(c3scc(C)n3)=O)C2)=O)ccc(F)cc1F c1(OCCCOC)cc(CN2CCOCC2C(=O)NC)ccc1.C(=O)CC(C)O C1(C(=O)NC(C2CCC2)C)(C(F)F)CCCC1.N1(CCC(=O)N)CCOCC1 c1ccc(CC)cc1.C(=O)C(C1CCCO1)C1CC1.c1(C(=O)NC)cc[nH]n1 C1(F)(C(=O)NCCC(N)=O)CCCN(C(c2scnc2Cl)=O)C1 C1(=O)CC(C(F)F)CN1.c1(OCC(=O)OC)cc(F)cc(F)c1 c1(C(N(CCCNC(c2ccc(C)nc2C)=O)C)=O)ccc2[nH]c(=N)n(C)c2c1 CC1=C(C(=O)NCC2CCCCN(C(=O)C(C)(O)c3ccccc3)C2)CCC1 C1(F)(C(=O)NC2CCC(C)CC2)CCN(C(=O)C(C)C2(O)CCC2)CC1 c1(C(=O)NC2(CNC(C(CCC)CC)=O)CCCC2)n[nH]c2ccc(Cl)cc12 C1(N(C(C(CC)O)=O)C)CN(C(c2cn(-c3cccc(Cl)c3)nn2)=O)CC1O CC(C)CC(C(=O)N1CC(CNC(=O)C(CCO)N(C)C)C(F)(F)C1)N(C)C N1(CC)CCCCC1C(N1CC(OC)C(NC(c2sccc2C2CC2)=O)C1)=O c1(NC(N(CC=C)CC=C)=O)nc(C)cnc1C#N c1(C(N2CC(NC(C3C(C)C3C)=O)CC(C)C2)=O)ncc2ccccn12 c1(SCC)ccccc1C(N1CCC(NC(=O)C(C)C2(O)CCC2)CC1)=O.C C(=O)(CCCCCCNC(=O)CC1COC(=O)C1)N(C(C)C)CC1CC1 C1(C(N2CC(C3N(C(c4cc(C)sc4)=O)CCC3)(O)C2)=O)CCCC(C)(C)CC1 N1(C(=O)C=Cc2ccoc2)CCC2(CO)CN(C(=O)CC3=CCCCC3)CC2C1 Cn1cccc(C(N2C(C(=O)NC3CC(c4ccccc4)C3)CC3CC23)=O)c1=O CCCCC(=O)C(=O)N1CC(C(=O)NCC(c2ccco2)O)(CC)C1 C(=O)(C(C)S(=O)(=O)C(C)C)N1CCCCCC1.C(CC(=O)NC)SCC(C)C c1(C=O)ccc(CC#N)cc1.c1(C(C)OCC)ncc(C(=O)NC2CC2)s1 C1(C(=O)NCC2C3CN(C(CCOC(C)C)=O)C(C3)C2)CCCCC12OCCO2 CC1CC(CNC(=O)Cn2nccn2)CN(C(=O)CC2CC(=O)C2)C1 c1(C(N2C(CN(C(c3oncc3C)=O)CC)CCCC2)=O)ccc(CO)c(F)c1 C=C=C(C)CC(=O)NC1CC(C(=O)NCCc2nncs2)C1(C)C C1(C(N2C(C)CC3(CC3)C2)=O)CCCCCCN1C(C1CC(=C2CC2)C1)=O c1(C(=O)NCC2CC(C)N(C(c3cn(C)c(O)n3)=O)CC2)cc(C#N)ccc1Cl C(=O)(C(Cc1ccco1)NC(=O)CCC1CC1)NCCC1CC(OC)C1 c1(C(=O)NCC(CC=C)NC(=O)CCCC(C)C)ccc2c(c1)[nH]c(=N)n2C N1(C(C2C(F)(C(=O)OC)C2)=O)CCCC(C)C1.C1(C)(C=O)CCNC1=O.N CCCCCCOC(C)C(=O)NCC=CCNC(c1ccnn1CCF)=O c1(CC)cccnc1NC1CN(C(=O)C(c2ccccc2)SC)CC1C c1(NC(CN(C(=O)CN2CCCCCC2)CC#C)=O)cnc2n1CCCC2 CC1CCCN(C(=O)CCCc2csc(=N)[nH]2)C1CNC(=O)CCc1cncs1 Cc1c(NC(C2CC2C(=O)NCC2(C)CCC2)=O)cccc1Cl C1(CCNC(c2c(C(C)C)n[nH]c2)=O)CN(C(=O)CC(C)F)CCS1(=O)=O C1(CC)CN(C(c2n[nH]c(C(C)(C)C)n2)=O)CCS1(=O)=O.C=CC(C=O)OC.N c1(C(N2C(CNC(c3cc(F)n[nH]3)=O)CC(F)(F)C2)=O)cccc2ccccc12 C(N=c1[nH]c(=N)[nH]c(=NCC2CC(CC(S)C)CCO2)[nH]1)c1ccc(SCC)o1 C12(CNC(COCCC#C)=O)CCC1CCN2C(c1sccc1F)=O c1(NC(CNC(c2ccccc2OC(F)F)CC)=O)ccc(O)c(C)c1 C=C(C)CN=C(NCc1csc(C(F)(F)F)n1)NCC1(C#N)CCOCC1 CC(CC1CCCCC1)C(=O)NCC1CCN(C(C2CC2C)=O)C1 N1(C(C(CSC)(C)NC(c2ccc(CO)nc2)=O)=O)CC(O)C(C2CC2)C1 CC(C(=O)N1CCC(c2nnnn2C)CC1)C(N)c1ccccc1 C1(C(=O)NC2CC3(C(NC(c4ccns4)=O)C3)C2)CCCC2(CCCCC2)C1 c1(C=O)ccc([N+](=O)[O-])o1.N1(C(CSCCN(C)C)=O)CCCC1C1CC1.N CC1(C)CC(C(=O)N)CC(C)(C)C1.C12CN(C(=O)C=C3CCC3)CC1CCO2 C(N=c1nc2sccc2c(NCCSC(F)(F)F)[nH]1)C1(OCC)CN(C)C1 N1(C(C(CNC(c2c(C)noc2C)=O)O)=O)CC23CCC2(COC3)C1 N1(C(c2c(OC)nsc2)=O)CCN(C(c2cccc(C)c2)=O)CC1C(F)F C1(c2nnnn2C)(NC(CC(C)C)CO)CCN(C2CCOC2)CC1 C(C)(CCC(=O)NCCC1CCSC1)NC(c1c(CCC)n[nH]c1)=O c1(C(N)=O)nc(Cl)cnc1NC(C1CNCCN1Cc1ccnn1C1CC1)=O N1(C(c2c(C)cc(CNC(=O)CNc3ccccn3)o2)=O)CC2CCC2(C)C1 c1cnccc1Cl.C=C1CC(C(=O)N)(CNC(=O)CCC2CCC(C)O2)C1.C N1(C(CC(=C)C)=O)CCCC2CN(C(c3ccn(CC4CC4)c3C)=O)CCC12 C1(COC(C2CN(C(=O)CCCC3CCCC3)C2)=O)CCCC2(CCOCC2)O1 N1(CC2OCCN(Cc3c(C)cccc3)C2)CCS(=N)(=O)C2(CCC2)C1 c1(CC)cc(CC(=O)NCC2(C(=O)NC(c3ccoc3)C)CCC2)on1 Cc1ccc(C=CC(N2CC(F)CC2CN(C(=O)CO)C)=O)nc1 C1(NC(c2[nH]cc(C(C)=O)c2)=O)(CO)CCCN(C(c2nccnc2N)=O)C1 C1(N(C(C=CCN(C)C(c2ccc[nH]2)=O)=O)C)CCCOC1 Cc1c(CC(=O)NC2(c3cccnc3)CCCC2)c(O)nc2ccccc12 Cc1cccc(F)c1C(=O)N.C12CC(CO1)N(C(=O)C=CCN1CCCC1)C2 N1(C(CCCOCCC)=O)CC2(CCCC2)C1C(=O)NCC(C)CCCC(C)C c1(C(=O)NCCC(C)NC(C(CCC)OC)=O)cc(O)nc2c(F)cc(C)cc12 C1(NC(=O)NCC2(CSC)CC2)CC2CC1C1CC21.C1CCCN(C)C1 CC(C)(F)C(C)(F)CNC(C1CCN(C(=O)CSC(F)(F)F)C12CC2)=O CCC(CC(=O)NC1(CNC(C2CCC(c3cc[nH]n3)O2)=O)CCC1)OC c1(C(=O)NC2C(NC(CS(CC)(=O)=O)=O)CCC2)cc([N+](=O)[O-])cn1C N1(C(C(CC)N(C)C)=O)CC2(CCCC2NC(c2cnc(C)nc2C2CC2)=O)C1 c1(OC)ccc(Br)cc1NC(c1conc1C1CCNCC1)=O C1(C(N(C(C)CNC(=O)Cc2ccc(O)cc2)C)=O)C2Cc3cc(Cl)ccc3C12 c1(C(C(N2CCC(NC(C(C)CN(C)C)=O)CC2)=O)(C)C)cccc(Cl)c1F c1(C(N(C2CC(NC(=O)CO)C2)C)=O)nccc2ncccc12.C1CCCO1.C c1(C(=O)NC2CCC(C(N(C(C)C3CC3)CC)=O)C2)coc2c1COC2 c1(CC(=O)NC2CN(C(C3CN(C)C3)=O)CC3(C2)CC3)ccc(F)cc1[N+](=O)[O-] c1(C(=O)NC2C(NC(c3ccc(C)nc3)=O)CC2)cc(F)c(Cl)c([N+](=O)[O-])c1 n1(CC=O)c(C)nc2cc(F)c(F)cc12.C(S(=O)(=O)CC)c1cn(CC)nn1.N CC1CCCC=C1C(=O)N1CC(CC(=O)NCc2ccnc(F)c2)CC1C C(C1=CCCCC1)NC(C1(C(C)NC(=O)Cc2cn[nH]c2)CC1)=O N1(C(c2n(COC)ncc2)=O)CC2CCC1CN2C(c1c[nH]c(=O)cn1)=O Cc1oc(CO)cc1C(=O)NCC1CCCC1NC(c1ccccn1)=O C#CC1(C(N2CC(C)(CSC)C2)=O)CCN(C(=O)Cc2n[nH]c(C)n2)C1 CC1CC(C(=O)NCCCCCNC(=O)C(C)(C)c2cc[nH]n2)CO1 N1(C(CCN(C(C(CC)C)=O)C2CC2)=O)CCCC2(CCOC2)C1 C1(NC(C2(COC)C=CCC2)=O)CN(C(c2ccc(OC)s2)=O)CC1O C(=O)(C(C)C1=CCCC1)N1C(CNC(Cc2cc(CC)nn2C)=O)CCC1 C=CCC(C)(C)CC(=O)NCC1(CO)CCN(C(c2ccncc2)=O)CC1 C1(C(=O)NC(C2CN(c3ncccc3[N+](=O)[O-])C2)C)CCc2nc(O)[nH]c2C1 C1(C=O)CCCC(=O)N1.n1(CCCC)nccc1C(=O)NCC1CC1C.N c1(C(=O)NC(C2CCCN2C(c2ccsn2)=O)C)coc(C(F)(F)F)n1 c1(OCCCC)ccc(NCCCC2CCCC(C)(C)C2)cc1OCC C1(C(=O)O)CN(C(=O)COCCNCc2ccc(O)nc2Cl)CC12CC2 Cc1cc(N2CCOC(C(C)NC(=O)CCc3cnc[nH]3)C2)nc(C(C)C)n1 CC1(C)COC(CC(=O)NCC(C)(C2CC2)NC(c2ccccn2)=O)CO1 C1(C(=O)NCCN(C(c2ccnn2C2CC2)=O)CC)C2COCC12 N1(C(CC2CC(=O)OC2)=O)CC2CC(C1)N(C(c1cc(Cl)cc(Cl)c1)=O)C2 c1(CNC(Cc2cn(C)nc2)=O)n[nH]c2c1CN(C(C1CCC=CCC1)=O)CC2 O=C(C1=CCCN(C(C2C3CCCCCC23)=O)C1)N1CC(F)(CF)C1 C1(CNC(c2cnccn2)=O)COC(C(F)(F)F)CN1C(c1cocn1)=O C1(C(N2CCN(CC(C)O)CC2)=O)CN(C)CCN1C(=O)CSCCC#N N1(CCCC(=O)N(C2CC(C)CC(C)C2)C)C(=O)c2ccccc2C1=O c1(CC)ccc(C(=O)N)cc1F.C1CN(C(=O)Cc2cc(C3CC3)no2)C2CC12 C(=O)(C#CC(C)(C)C)N1CCC(O)(C(CNC(CCc2c(C)cccn2)=O)C)C1 N1(CC(=O)N(C(CN(C(C2(CCCC)CCC2)=O)C)C)C)CCSCC1 c1(OC)cc(Cl)c(-c2cn(Cc3occc3C(=O)O)nn2)cc1Cl.C(C)CO CC(CCC(=O)NC1CC(CCC(=O)N(C2CCN(C)C2)C)C1)N(C)C c1(CC)cnoc1C(N1CC(CNC(=O)C(C2CCC2)C2CCC2)C1)=O N12CCC(CC1)NC(=O)C2.c1(Cn2cc(CCC(CC)O)nn2)ccccc1Cl N1(C(CCC)=O)CCN(C(C2C(C(=O)OC)C2(C)C)=O)CC1c1cn[nH]c1 C1(CCNC(C2(C(=O)NC)CC2)=O)CN(C(C2(O)CC2)=O)CC(C)O1 Cc1cc(C(N2CC3(CC(CC(N4CC(O)CC4C)=O)C3)C2)=O)c(F)cc1Br N1(C(C(=O)Nc2cc(C)on2)C)CC(CO)C(c2cnn(C)c2)C1 C=C(C)CCC(=O)NCC1CN(C(=O)Cc2csc(C)c2)CC1C(F)(F)F N1(C(c2n[nH]c(C)c2Br)C(=O)NCCCSCC)CCOC2(CCOC2)C1 c1(CC(=O)N(CC(C)(C)CNC(=O)C(F)C2CCOC2)C)c(F)cncc1Cl c1(C(=O)OC)ccc(C=CC(=O)NC2CCCC2)o1.c1(C=O)cnc(O)o1 N1(C(c2cnc(S)nc2)=O)CCCC(C2CN(C(C3CCCO3)=O)C2)C1 C1(C(=O)Nc2nnc(C)s2)CCC(OCCCc2ccccc2)CC1 CCC(C)C(O)C(C)C(=O)NCC1CN(C(=O)CCCC(F)(F)F)CCO1 C(=O)(CCC(F)(F)C(F)F)N1C(CCC)CN(C(C2CCCN2C=O)=O)CC1 N1(C(C2CC=CC2)=O)CC2(C1)CN(C(=O)C(c1ccc(Cl)cc1F)O)CC2CO c1(C(=O)NCCCCCCNC(C2(C)CCCC2O)=O)cnc2sccc2c1 C1(CC=C)(NC(C2CC(C)CO2)=O)CCCN(c2cc(C(C)C)nc(CC)n2)C1 Cc1cc(S(C)(=O)=O)cc(NC(=O)C(O)CC(O)CO)c1C N1(C(c2cc(CC)nnc2C)=O)CCCN(C(C2(C)CCCC2(F)F)=O)CC1C C1(CC)C(=O)N(C)CCN1Cc1cccc(-c2cccc(C(C)N(C)C)c2)n1 C1(NC(C(C)Oc2cc(C)c(C(C)C)cc2)=O)CC2CC1CN(C(=O)CO)C2 CCC(CC)C(=O)N(CCC(N1CCC2CC2C1)=O)CCCO c1(C(=O)NCC2(NC(C(CC=C)CC)=O)CCOC2)cc([N+](=O)[O-])ccc1N c1(N2CCCC(NC(=O)NC)C2)nc(=NCP(C)(C)=O)[nH]c2c1CCCCC2 C=CC(C)C(C)C(=O)N(C)CCO.c1(C(N(CC)C)=O)cnc(C2CC2)nc1O C1CC(O)CN(C(=O)CCC2CCC2)C1.c1(CSCCC(=O)N)cccc(Cl)c1 C1(C(N2CC(CC(C)NC(=O)CCCC(F)F)C2)=O)CC(=O)NC(=O)C1 N1(C(c2nc(C(C)(C)C)co2)C(=O)NCCCCCC)CCC(C(N)=O)C(O)C1 C1(NC(CCOCC)=O)C2CN(Cc3nccnc3C)CC12 CC(C)(C)CC(=O)N1CC(CNC(C2CC3CCC2O3)=O)C(c2ccccc2)C1 c1(OCC(=O)Nc2ncsc2-c2ccc(F)c(F)c2)cccc2cccnc12 C(=O)(CCC(F)(F)F)NC1C(CNC(CCC(=C)Br)=O)C1 CCC(CC)C(C)C(=O)N(C1CN(C(=O)C(c2ccc(C)cc2)F)CC1(C)C)C N1(C(C=C(C)C2CC2)=O)CC(O)CCC1C(=O)NCC1CC1[N+](=O)[O-] C1(C(=O)NC(CC)(C)CC)CC2CN(C(=O)CC(C)C(F)F)CC2C1 c1(NC(C2N(Cc3scc(C)c3)CC(C)C2)=O)ccc(C#N)cc1F N1(C(C=CC(C)C)=O)CCC(C2CC2)(CNC(=O)Cn2nccn2)C1 c1(C(N2CCN(C(c3cc(OCC)ncc3)=O)CC2)=O)cc(C)c(F)c(C)c1 CCCN=C(NCCC(c1ccccc1)O)NCC1C(C)(C)C1(C)C c1(C(N(CCC2N(C(COCCC)=O)CCCC2)C)=O)cncc2c1CCCC2 C1(NC(Cc2ncc(C)o2)=O)CC2(C1)CC(NC(=O)CCc1cnn[nH]1)C2 Cc1nn(C)c(C)c1CNC(=O)CC(C)(C)N(C(=O)C(=O)C1CCCC1)C c1(C=O)ccccc1Cl.C(C(C)C)NC(C1(OC(C)=O)CC1)=O.C1CC1.N CC(C)CC(C)NCc1ccc(-c2ccccn2)s1 CC1(C(=O)NC(c2ncc[nH]2)CO)CCCN(C(c2ccccc2Cl)=O)C1 c1(C2(C(=O)NCC3CC(C)C3)CC2)ccccc1.C(=O)CC.C1CCCC1 CS(=O)CCN=c1[nH]c(=NCC2(OCCO)CCOCC2)[nH]c2c1SCC2 c1(NCCCOC(C)(C)C)cc(N2CCC(OCCO)CC2)ncn1.C1CCCC1 C(=O)(C1=NOC(C)C1C)N1CC(N(C(C(C(C)OC)N(C)C)=O)C)C(C)CC1 Cc1ccc(Cl)c(F)c1C(=O)NCC(CC(C)C)NC(c1ccc(O)nc1)=O C(=O)(C(O)CC(C)C)N(CCNC(c1c(C)[nH][nH]c1=N)=O)C(C)C CC(CCC(=O)NCC1CCCCS1)NC(c1cc(C#N)cs1)=O c1(C(N2CCN(C(CCCC#C)=O)C3(C2)CCC3)=O)n[nH]c2c1CC(F)(F)CC2 CC#CCCCC(=O)N1CC(C)C(C)(CNC(=O)CC2CCOC2C)C1 N1(C(CCCC#C)=O)CCCCC(CNC(=O)CC2(OC)CCCC2)C1 C1(O)(CN(C(C(C)C)=O)C)CCCN(C(=O)CN(C)C(C)C)C1 S(=O)(=O)(c1ccc(I)cc1)NC1C(F)CCN(c2c(C#N)cnc(SC)n2)C1 c1(COC)n[nH]c(=NC2CCOC3(CCN(C(c4ccc(F)nc4)=O)CC3)C2)s1 C(c1cccc(O)c1)=CC(N1CCCC1)=O.CC(C)(C)OC1CC1C(=O)N c1(OC)ccc(C(N2CCC(NC(=O)CCOC3CCCOC3)CC2)=O)c(F)n1 c1(OCc2cn(CC)nn2)cccc(C(=O)NO)n1 Cc1cc(C)c(C(=O)NCC2CCCN(C(=O)CCC=CC(C)C)CC2)c(C)n1 N1(CC=O)CCc2sccc2C1.c1(CC(C)C)oncc1C(=O)NCC1CC1 Cn1cc2cccc(C(N3CCC4(CC4C(=O)NCCn4ccnc4)C3)=O)c2n1 C12(NC(=O)C=Cc3ccc(Br)o3)CCN(C(C3(F)CC3)=O)CCC1C2 n1(CC)ncc([N+](=O)[O-])c1C(=O)NC(C)CCCNC(=O)CCCN=[N+]=[N-] C1(c2n(CCCCCC)nnn2)(NC2CC2)CCCC1CCF c1(OC)cc(Cl)ccc1NC(=O)Nc1cc[nH]c1C c1(OC)ccc(SCC(=O)NC(C2CCCC2)CNC(=O)C(O)C)cc1.S c1(NC(C(C(C)(C)C)NC(=O)CCS(C)(=O)=O)=O)ccccc1N=[N+]=[N-] C1(NC(c2nc(C)c(C)[nH]2)=O)CCSC12CN(C(=O)CN1CCCNC1=O)C2 n1(CCC(=O)NCc2cc(O)nc(O)n2)sc2ccccc2c1=O N1(C(C2C(NC(CN3C(=O)NCCC3)=O)CCC2)=O)CCC2(C1)CC2(F)F C(=O)(C1=CCC2CCC1N2C(C1CC1CC(C)(C)C)=O)NC(CC)CC CC1(C)CC(C(=O)NC2CCCN(C(c3cnns3)=O)C2)=NO1 C=CCCCC(=O)N1CCSCC1C(=O)NC1CCOC1=O N1(C(Cc2nc(C)oc2)=O)CCC2(CC1)CCN(C(C1COCCC1C)=O)CC2 C(=O)(C(=O)N=S(C)(C)=O)N1CC(CC)CC1.C1(C(=O)N)OCCC1C(C)C C=CCCC(F)(F)C(=O)NCC1CC12CCN(C(=O)C(C)C1CCC1)CC2 Cc1cc(CNC2(C)CN(CC3CC3)C2)ccc1C=Cc1ccoc1 c1(SC)ccc(C)c(C(=O)N(C2CN(C(c3csc(=N)[nH]3)=O)CC2O)C)c1 Cn1ccnc1SCCNC(N1CCC(C(=O)Nc2ccccc2)C1)=O Cc1cc(C(=O)NC2(CC)CC2)n(CC(F)F)n1.c1(C(=O)N)cn(C)cc1C c1(C(C)C)ccc2c(Cl)c(C(=O)NC(C)CC)sc2c1.C1(C(=O)N)CCC(C)O1 c1(C(CC(=O)NCC2(CC)CC2)O)cccc(F)c1.C(=O)CCc1ccoc1.N c1(C(=O)N)ccc(C)c(C(F)(F)F)c1.Cc1cc(CC(=O)N(CC(O)C)C)no1 C1(NC(CCC(=O)NC)=O)CC(O)CN(C(c2cnc(C(N)=O)cn2)=O)C1 N1(CC2CN(Cc3cn(-c4cccc(OCC)c4)nn3)C2)CCc2ccccc21 S(=O)(=O)(c1ccc(NC2Cc3cscc3C2)c(Br)c1)NC(COC)CCO c1(C(=O)N)cc2nc(Cl)ccc2s1.c1(C(N(CC)CC)=O)conc1C1CC1 C12(CNC(C(C3CCCOC3)OC)=O)CCC(CN(C(=O)CCC(C)SC)C1)C2 c1(C(N2C(C3(NC(C(CC=CC)C)=O)CC3)CCC2)=O)ccc2c(c1)CCCO2 CC(C)C(C)C(C)CC(=O)N1CCCC2(C1)CN(C(=O)C(=O)N=S(C)(C)=O)C2 N1(C(C(C2CC2)SC)=O)CCC(C(=O)Nc2cc(C)c(C)c(C)c2)=C(F)C1 c1(C(=O)NC2CN(C(CC(C=C)CC)=O)CC2C)c(F)cc(C)cc1Cl C(=O)(C(C(C)OC)N(C)C)NCC(C(=O)NC(C(=O)OCC)CC)O C12(C(=O)NC(COC)C(C)C)CCCC1CCN2C(=O)CN1CC2CC2C1 C1(NC(CC2C(CNC(c3nc(C)oc3C)=O)C2)=O)CC2CCC(C1)N2C N1(C(Cc2ccc(OCC)cn2)=O)CC=C(CNC(c2cnc[nH]2)=O)CC1 c1cccc(F)c1.C1(C(=O)N)CCCO1.C1(NC(C2(O)CC2)=O)CC1C CCCCCCCCOCCC(C)(C)Cn1cc(C#N)nn1.C(=O)C(CC)C(C)C C1(C(N2CCCC(NC(c3c[nH]c(=N)o3)=O)CC2)=O)CC1C1CCOCC1 N1(C(C(C)c2cc[nH]n2)=O)CC=CC1(C)C(=O)N(C1CSC1)C C1(O)(CC(C)C)CCN(C(C2CC2CNC(=O)C=Cc2cncs2)=O)C1 c1(C(=O)NCC(C2CCC2)NC(c2cn(C)[nH]c2=N)=O)ccc2ncccc2c1 c1(C(=O)NC2C(CNC(CC=C=C)=O)CCC2)ccc(C(F)(F)F)nc1C c1(C(N2C(C(=O)Nc3ccc(F)c(Cl)c3)CC3CC32)=O)cccc2nccnc12 C1(NC(CSCCN(C)C)=O)CS(=O)(=O)CC1.c1(CC(=O)N)cc[nH]n1 C1(NC(COCCOC)=O)CCN(C(c2cn(C)nc2Cl)=O)C1c1ccccc1 c1(OCC=C)ccc(C(=O)NC2CCN(C(C3CC3C)=O)C2CC)cc1 C(=O)(C(F)C(C)CNC(C1(C)CCCCCC1)=O)NC(c1cn[nH]c1)C Cc1cc(OCCC(=O)NCCCCCCNC(=O)C(O)C2CCC2)cc(C)c1 c1(CC(=O)N(C2CCCN(C(c3n(CC)c(O)nc3)=O)C2)C)cc(C)cc(F)c1 C1(CNC(C=NOC)=O)CN(C(c2ccc(OC3CCC3)cc2)=O)CCC1C Cc1cccc(C(N2CCC(O)(CNC(=O)CC(C)CN(C)C)CC2)=O)c1Cl c1(CNC(=O)CSCCNC(=O)CCOCC(F)F)cc(Cl)ccn1 CCN=c1[nH]cc(C(=O)NC(C2CCN(C(=O)CC(O)CC)C2)(C)C)s1 c1(C(=O)NCC2CN(C(CC3CCC(=O)N3)=O)CC2(F)F)cccn2nnnc12 C1(N(C(=O)CN(C)CCO)CC)CCN(C(c2ccoc2C2CC2)=O)C1 C(CCCCC(=O)NC1CCN(C(C2CCC2)=O)C1(C)C)OC c1(OC)ccc(F)cc1C(N1CCC(NC(c2ccc(=O)oc2)=O)C12CC2)=O C1(CC(=O)NC(C2(O)CN(C(=O)CC(C)(C)O)C2)C)CN2CCN1CC2 c1(OC)cc(C(c2nnnn2C2COC2)NC2(C)CCC(C)C2)c(F)cc1Cl c1(NC(C2(C)CC(O)CN2C(=O)CCc2ccc[nH]2)=O)ccccc1N=[N+]=[N-] c1(C(=O)NC2CC(NC(c3ccc(CCC)s3)=O)C2)ncccc1C(F)F C1(C(=O)NC2CC3CC2CN3C(c2c[nH]c(=N)o2)=O)(OC)CCC(F)(F)CC1 c1(OCC)ccc(C(C)C(N2CCC(NC(=O)C(O)C3CCCC3)C2)=O)cc1 C(CC(=O)NCC12CCC(CC1O)C2)(C(F)(F)F)NC(c1cc(C)ns1)=O C1(CNC(c2cccc(Br)c2)C(C)C)CNCC(C2CC2)O1 C1(CCC)CCCN(C(C2CCCN2C(=O)CCc2csnn2)=O)C1 CCC(C)CCCC(=O)N1CC(CCNC(C2(C(F)F)CCN(C)CC2)=O)C1 c1(C(C(N2C(CNC(C3(C(C)=O)CC3)=O)CC2)=O)C)c(C)nn(C)c1C C1(C(N2CCN(CCC)CC2)=O)(OC)CCN(Cc2ncnn2C(C)C)CC1 C(=O)(CC(C)(C)C(C)=O)N1C(C(=O)N)(COC)C=CC1.c1cncc(O)c1 C1(C(N2C(CCC#C)CCC2)=O)CC2(CCN(C(=O)C(C)CC(C)C)C2)C1 C1(CC=C)CCCCN1C(C1CCC(C)SC1)=O N1(C(CCOCC#C)=O)CCN(C(=O)C(=O)NCC)CC(O)C1 CCCCCCC(=O)N1CCC1CNC(c1ccc(Nc2nccs2)cc1F)=O c1(OC2CCN(CC3C(N4CC(C)(C)C4)CNC3)C2)ccc(C#N)cn1 C(=O)(C1=CCCOC1)NC1CCC(CNC(C(C(C)O)NC(N)=O)=O)CC1 CCC(CC)C(=O)NC1COCC1C(=O)NC1(c2nccn2C)CC1 N1(C(c2c(C)ccc(OC)c2)C(=O)NC(C)(C)C)CCC(OC)C12CCC2 C(=O)(C1=CCN(C(c2ccns2)=O)CC1)N(C(c1nccs1)C)C C(N=c1[nH]c(=NCCCCSC)[nH]c2cccc(F)c12)c1ncc(CC)[nH]1 C1(C)(CC)CC(NC(=O)CN2C(=O)CCCC2=O)CN1C(=O)C1=COCCC1 c1(CNC2CCC(C(=O)NCC3CCOCC3)C2)ccc(F)c(Br)c1 C1(CCC)CN(C(C2CCC(=O)N(CC)C2)=O)CCN1C(=O)CC1(OC)CCC1 C1(CNC(c2cnn(CCC)c2C)=O)CN(C(=O)C(F)C(C)(C)O)CC12CC2 N1(c2nc3ccc(C)nc3s2)CCC2(CCCC2NC(=O)C(O)C(C)(C)C)CC1 c1(C(N2CCCC2c2ccncn2)C(=O)NCCSC)ccc(C)cc1 c1(C(=O)NCC2(CNC(CN3C(C)CC3)=O)CCC2)c[nH]cc(Cl)c1=O c1(C(C(=O)NCC(CN(C(CSCC#C)=O)C)(C)C)(C)O)cccc(F)c1 C(=O)(C(O)C=C)NCCC1(C(N(CC#C)CCF)=O)CCC1 C1(C(=O)NC2(C(C)=O)CC=CC2)CCOCC1NC(=O)CC(C)c1ccco1 N1(C(CCCNC(C(C)OCCOC)=O)=O)CC(=O)NC(C)C1 c1(CCC(=O)N(CCN(C)C)C)c[nH]c2ccc(C)cc12.c1(COC)ccco1 C(=O)(C(C)(O)C1CC1)NCC1CC(NC(COCCCC)=O)C1 C(O)(CN=C(NC1CC1)NC1CC12CC2)c1cn(C)nc1 c1(C(=O)NC2COC3(C2)CN(C(c2coc(Br)c2)=O)C3)ccc2ccccc2n1 c1(C(N2C(C)(C)C(CNC(c3cccc(O)n3)=O)CC2)=O)cccc2cncn12 CC1(C)Cc2cccc(NCC(=O)NC3CC(O)C3CN)c2O1 C1(N(C)C(C23CC(c4ccccc4)(C2)C3)=O)CCCCC1.C(=O)(C)N.CC#N c1(CC(N2CCC3C2C3)=O)coc2ccc(F)cc12.C(C=O)N(S(C)(=O)=O)C C(=O)(C(C)(C)C1=CCN(C(=O)Cn2ccccc2=O)C1)NCC=CC C1(CNC(C2CCCC2(F)F)=O)(CO)CCCN(C(c2ccc(Cl)s2)=O)C1 CC1CCC(F)(C(N2CCC(C)(CNC(c3cc4n(n3)CCC4)=O)CC2)=O)CC1 C1CS(=O)(=O)N(C)C12CCN(C(=O)C(O)C(F)F)CC2.C(C=O)N(CC)CC c1(C(N2CCC(N(C(=O)CC3CCCC3(F)F)C)C2)=O)cnc2c[nH]nc2c1 N1(C(c2scc(C(=O)NCCc3ccc(OC)cc3)n2)=O)CCCCC(F)(F)C1 CCC(F)(F)CN(C(=O)CCCNC(c1ncsc1NC)=O)C C1(C(C(C)C)NC(CC=C)=O)CCN(C(=O)C(F)(F)CC)CC1 N1(C(C(C)(CO)NC(C2CCN(C)C2)=O)=O)CCC2(CCOC2)CC1 c1(NC(C2CCC(NC(C3C(C)(C)OCC3)=O)CC2)=O)ccc2nn[nH]c2c1 C1(CNC(CN2C(C)CCC2)=O)CCN(C(=O)CCCC2CC2)C12CC2 C1(C(=O)NC2C(C(=O)NCc3nnc(C)s3)CC=CC2)CC2CCCC2C1 c1ccccc1CC.c1(C=O)ccc(Cl)[nH]1.C(=O)CN(C)C(C)=O.COC c1(C(N(CC(C)O)CCNC(C(CCCC)O)=O)=O)ccn2nnnc2c1 Cc1ccc(C(N2CCCC2CCC(=O)NCC23CCC(F)(CC2)C3)=O)c(F)c1 C1(NC(C2(CC=C)CCCCC2)=O)CCN(C(=O)CCn2cccn2)CC1F c1(OC)cc(C(=O)NC2CN(C(C3(C)CC4CC4C3)=O)CC2C)ccc1Br Cc1cc(C(=O)NCC2CCCC2O)c(C)n1C1CC1.c1(C=O)ccsc1Cl.N N1(C(Cc2ncc(C)o2)=O)CCCC(NC(c2cc(Cl)c(Cl)n2C)=O)C1C C1(NC(C(=Cc2ccccn2)C)=O)CCSC12CN(C(=O)CN1CCC(C)(C)C1)C2 c1(C(N2CCC(NC(c3ncn(CC)c3)=O)C23CC3)=O)cc(F)c(Cl)c(N)c1Cl Cn1ccc2[nH]c(C(=O)NC3CC4(C3)CCC4)cc12.C1(C)(C(=O)N)C=CCCC1 N1(C(c2ccc(OC)nc2C)=O)CCCN(C(=O)C(C)CO)CCC1 CC(CCC(C)(C)C)C(=O)NC(C)(CNC(c1c[nH]cc1Br)=O)C1CC1 N1(CCNC(CNC(CNC(c2c(C)noc2)=O)=O)=O)CCOCC1C c1(C(=O)NCC(CN2CC(C)OCC2)O)cc2c(n1C)=C1C(=C(SC)N=C1)C=2O C1(NC(=O)COC(F)(F)F)CN(C(=O)Cc2cccc(O)c2)C2(CCOCC2)C1 O=S(=O)(c1cc2ccccc2s1)Nc1ccc(-c2cccn3ccnc23)c(F)c1 Cc1cc(NC(C2C3CCC(C3)C2)=O)cc(Cl)c1.c1(C=O)cc2n(n1)CCO2.N c1(C(N2CC(n3cc(CC(=O)OCC)nn3)C(O)C2)=O)cc(OC)cc(C)c1 c1(CC(=O)NC(CCCNC(c2c(CC)ccs2)=O)C)ccc(C)c(OC)c1 c1(C(=O)NC(C)CC(C)NC(C2CC3(CC3)C2)=O)cnc(O)c(F)c1 C(=O)(C(CCN(C)C)NC(C1CCC(F)(F)C1)=O)N1CC(C(CC)C)C1 N1(C(COCCC#C)=O)CCC(C)C1C(=O)NCC(=O)OC(C)C C1(NC(C(C)S(C)(=O)=O)=O)CC2CC1CN(C(c1ncc3ccccn13)=O)C2 c1(NC(=O)CSc2cncc(OC(F)(F)F)c2)ccc2c(c1)CCC2 c1(C=O)c[nH]c(=N)nc1C(F)(F)F.N1(C(C(=O)NCC)=O)CCC(C)C1 N1(C(C2C(C)(C)CCC2)=O)CC2(CC2)CC1C.C(c1ccc(F)cc1)=CC=O Cc1ccc(O)cc1C(N1CCSCC1CCNC(c1ncc[nH]c1=O)=O)=O c1(C(=O)NCC2(NC(CSc3nc(C)[nH]n3)=O)CCOC2)cccc(CO)c1 CC1(C)C2CC(C(=O)NCCc3cc(C(=O)N)no3)CC12.N1(CC)CCCC1 C1(C(=O)N)(COC)CCN(C(=O)CC2CC(O)C23CCC3)CC1.C1CC=CC1 C(=O)(C(CNC(=O)CCC1CC1C)C(C)C)NCC(COC)C C(=O)(C1=CNC2=NCCC2=C1)NCC1N(C(C2N(C)CCOC2)=O)CC(F)C1 C12(CC(=O)NC(c3ccc(OC)cc3)CCCC)COCC(c3cccs3)(C1)C2 C1(NC(C2CC(CC)(CC)C2)=O)CN(C(=O)CCO)C(C)C1.C1CCCC1 CCC(C(=O)NCC(O)CN(C(=O)COCCF)C)C(C)(C)CC C(CCC(C(=O)NCC1CC2(CC2)C(=O)O1)NC(c1ccccc1)=O)OC CC1=C(C(=O)N2CCCCC2CC(=O)NCC(O)CC2CCC2)COCC1 Nc1ccc(F)c(C(N2CCC(CF)(NC(=O)COc3ccsn3)C2)=O)c1F c1(OC)ccncc1C(=O)NCCCCNC(c1nocc1C1CC1)=O C1(C(=O)NC(C)CC(C)NC(=O)C(c2ccc(N)cn2)C)CCC2(C1)CC2(F)F Cc1nc(C(=O)NC(CCF)C(=O)NCCC2OCCC2C)c(C)s1 c1(C(N(CCOCCC(=O)NC(CC=CC)CO)C)=O)ccc2cc[nH]c2n1 c1(C(N2CCC(CCNC(c3ncc(N(C)C)nc3)=O)C2)=O)ccc(=N)[nH]c1Cl Cc1ccc(C=CC(=O)NCC2CC(NC(c3c[nH]nc3C)=O)C2)s1 N1(C(C(=O)NC)=O)CC(NC(c2ccc(O)c(CCC(F)F)c2)=O)CCC1C CCC(C)C(N)C(=O)N1CCC(C(=O)NCC2CC(=O)N(C)C2)(OC)CC1 c1(C(=O)NCC2CC(NC(CSCC=C)=O)C2(C)C)cc[nH]c(=N)c1Cl c1(C(=O)NCC(CC(=O)N2CCC(CC(N)=O)C2)OC)cc(C)cc(C)c1 C1(C)(C(=O)NCC(C)=CC(=O)NCc2cc(=O)cc[nH]2)CCOC(C)C1 C1(C)C(=O)N1.C1(C(N(CC(=C)C)C)=O)C=CC1C(=O)OCC C12(C(=O)NC3CCN(C(c4nc(C)nn4C)=O)C(C)C3)CC=CCN1CCC2 c1(C(=O)N)cc(C)c(F)cc1F.n1(CC)ccnc1C(=O)NC1(CCC)CC1 O=C1NC(CN2CCCCC2)C(=O)N1CC1(n2cc(Br)cn2)CC1 Cc1ncc(C(C(=O)NCC)N(C)CCN(C2CC2)C)[nH]1.C(C)(C)C.CCO C1(C)(CC)CC(C(=O)NC(C)(C)CNC(c2ccc(CO)cn2)=O)CCO1 N1(C(c2c(CC)nnc(C)c2)=O)CCC(NC(=O)C2=CCSC2)C(CO)CC1 N1(C(C(CC)(C)C)=O)CC(NC(=O)CCNC(=O)C=CCl)CC(O)C1 c1(OC)ccc(NC(=O)C(N2CCC(SC)CC2)C2C3CCCC23)c(OC)c1 C1(C(N2CC(NC(c3cc4sccc4[nH]3)=O)C(F)CC2)=O)CCn2cnnc2C1 C1(C(=O)OC)C(NC(=O)Cc2ccc(C(C)C)c(F)c2)C2CCCC12 c1(C(=O)NCCN(C(C2CC2(F)F)=O)C2CC2)cc2cc(Br)sc2[nH]1 Cn1nc(-c2ccccc2)cc1NC(c1nc(Nc2cscc2Br)cn1C)=O C(=O)(CC1=NNC(=O)C1)N1CC(NC(C2C(CC)CCO2)=O)C(C)C1 S(=O)(=O)(c1ccc(C#N)cc1)N1CC(CC(=O)Nc2cc(C)c(C#N)c(C)c2)C1 N1(C(C(COC)O)=O)CCC2CN(C(=O)CCc3nc(C(C)C)no3)CC2C1 C12(C(N3CCC(CNC(=O)CC4CC5CC5C4)C3)=O)CCCN1CCC2 c1(OC)ccc(N)c(C(=O)NC2CN(C(c3cc(S)oc3C)=O)C(C)(C)C2)c1 C1(NC(c2ccc(C(=O)OC)nc2)=O)CC2(C1)CN(C(C1CC1F)=O)C2 N1(C(c2c(NC)scn2)=O)CCCC(CC(=O)NCCN2CCCC(O)C2)CC1 N1(C(C(Cn2ccc(C)n2)C)=O)CCCCC(NC(=O)CN2CCC(O)CC2)C1 C#CCC(CC(=O)OC)NC(=O)CC1CN(C(=O)C(CO)OC)CC12CC2 c1(C(=O)NCCC(C)NC(C(CSC)O)=O)ccc(OCC(F)F)nc1 C(CCC(C)(C)C(=O)N(CCNC(=O)C(C#N)CC1CC1)C1CC1)OC c1(CC(=O)N(CCN(C(CC2CCC2)=O)C)C(C)C)cc(Cl)ccc1F.CO c1(C(N2C(CNC(c3cc4cn[nH]c4cn3)=O)CCC2)=O)ccc(F)c(Cl)c1F c1(CNCCNC(c2[nH]c3c(C)cc(C)cc3c2)=O)cc2cc(C)c(C)cc2o1 c1(OC)cc(Br)ccc1CN1CCOCC1CC(N1CC2CCCC2C1)=O N1(C(C2(CC)CCC2)=O)CC2CCC2(CNC(C2CCOC2C2CC2)=O)C1 N1(CC(c2cc(O)ccn2)=O)CCC(F)(Cc2ccccc2)C1 Cc1cn(C)nc1CNC(c1ccnc(CNC(=O)C(F)C2CCC2)c1)=O N1(C(C2(NC(=O)CSCC(F)F)C(C)CCC2)=O)CCC(O)C(C)C1 c1(C(N2CCC(N(C(=O)CCCC(F)(F)F)CCO)C2)=O)cc2n(c1)CCOC2 CCC(C)(CNC(=O)Cc1csnc1C)C(=O)NC1(CF)CCC1 C1(CN(C(C(=Cc2cccs2)C)=O)C)CCN(C(C2CC(F)(F)C2)=O)CC1 CCCC(C)(C)CC(=O)NCC1CCC(NC(=O)CCCN=[N+]=[N-])CC1 C1(c2nc(-c3n(CC)ncc3)on2)CCC2(CC1)CNC2 CCC(CNCC)C(=O)N1CCC1C(=O)NCC1CCCN1C(C)=O Cc1cc(C#N)ccc1CN1CC(C(=O)Nc2c(I)cccc2C#N)CC(F)C1 CC(C(=O)N1CC(F)(CNC(C2(C3CCCCO3)CC2)=O)C1)S(C)(=O)=O c1(C(=O)NCCC(C)NC(C(N2C(=O)CCC2=O)CC)=O)ccnnc1O Cc1ccc(C(=O)NCC2CCC(CNC(C3CC3F)=O)CC2)cc1Br c1(-c2cc(C)[nH]n2)nc2c(s1)CC(C(=O)Nc1cc(Br)nc(Br)c1)CC2 Cc1cc(CCC(=O)N(CC2CC2)CC2CN(C)CCN2C)ccc1Br c1(OCCOC)cccc(CC(=O)NC2(C)CC2)c1.C1(O)(C=O)CCC1 c1(C(=O)NCC(C)NC(C(C=C)O)=O)ccc(F)c2ccccc12 C1(N(C(C(C)C)=O)C)CC2CCC(C1)N2C(c1cnc(O)c(F)c1)=O CCCCC(CC)C(=O)N1CC(C)(C)CC1CNC(c1cocc1C(=O)OC)=O c1(C(C)=O)c(CCC(=O)NCC(CO)NC(C2CN(C)C(=O)N2)=O)c[nH]c1C C1(NC(CCC(=C)Cl)=O)CN(C(=O)CCCOc2cccnc2)C2(CCCC2)C1 C(=O)(C(CC(C)C)N(C(=O)C=Cc1cc(C)no1)C)NCC#C C1(C(=O)NC(C)CCCNC(=O)C(C)C(C)(F)F)CC2(C1)CC(F)(F)C2 O=Cc1ccc(N2CCC(n3cc(C(=O)O)nn3)C2)nc1 C1(NC(CCN(CCCO)C(c2n(CC)nnc2)=O)=O)CC2CCC1N(C)C2 Cc1c(C(=O)NC2COCC2NC(c2cc(F)cs2)=O)oc2cc(Cl)ccc12 C1(CCCCNC(C(C)(C)O)=O)CCCN(C(=O)Cc2c[nH]nc2O)C1 c1(C(N2C(C)C(O)CCC2)=O)cn2ccc(-c3cnn(CC4CC4)c3)cc2n1 C12(NC(COC3C(CC)CCCC3)=O)CCCN(C(c3ccc(Br)o3)=O)CC1C2 Cc1cc2[nH]c(C(N3CC4CCN(C(=O)Cc5conc5C)C4C3)=O)cc2s1 N1(C(c2ccc(C(N)=O)cn2)=O)CC(NC(c2csc(Cl)c2)=O)CC(O)C1 N1(C(c2c(C)nsc2)=O)CC(NC(c2cc3n(n2)CCOC3)=O)CC12CCC2 C1(Cn2cc(C(=O)NOC34CC5CC3C4C5)nn2)CCC(=O)N(C2CC2)C1 N1(C(CCCCNC(C2(CC#C)CCOC2)=O)=O)CC2(CCCC2)CC1C CC(C(=O)N1CCCC1C(C)NC(=O)C(C)(C)c1ccsc1)C(F)(F)C(F)F C1(Nc2nccc(=NCc3ccn(C)n3)[nH]2)CCCCCCCC1 C(=O)(C1=CS(=O)(=O)CCC1)N(C(C)C)CCN(C(=O)C(C)c1ccsc1)C C1(CCC)(NC(=O)COCCCN=[N+]=[N-])CCOC1.C12CCC1C(=O)N2 c1(C(=O)N)ccc2cccc(C)c2n1.C(C)(C(C)(C)C)NC(C1ON=C(C)C1)=O c1(C(N2CCN(CCNC(=O)C(F)CC3CC3)CC2)=O)ccc2nccnc2n1 Cc1cc(Cl)ncc1C(N1CC2C(C(=O)N(CCCO)CCCO)C2C1)=O C1(NC(C(C)N(C(=O)CC2CC=CCC2)C)=O)CNC(=O)C12CC2 c1(C=O)ncc(F)cn1.c1(CC)csc(-n2cc(C(=O)NC(C)CO)cn2)n1.N C12(C(=O)N)C3CC(CC13)C2(F)F.N1(C(COCC(C)C)=O)CC(C)CC1C N1(C(Cc2nc(C)sc2C)=O)CCN(C(=O)Cc2cccc(Cl)c2)CC1CF c1(C(C(=O)OCC2CCCOC2)O)cccc(Br)c1 N1(C(c2c(C)nc3sccn32)=O)CCC(NC(C2CC(C#N)C2)=O)C2(CCC2)C1 C(=O)(CC1=NN(C)C(=O)C1)N(CCCC(=O)NCC(C(CC)C)O)C C1(CC=C)(NC(c2nsnc2O)=O)CCCN(C(C2(OC)CCSC2)=O)C1 C(C)(CNC(=O)CC1C(=O)ON=C1C)(CC(C)C)NC(CCC(=C)Br)=O Cc1ccc(SC(F)C(=O)NC(c2ccccc2)CN(C)C)cc1 C(C1=CCN(C)CC1)NC(C(C1CCC1)NC(C=C(CC)CC)=O)=O CCC(C)(C(=O)N1CCOCC1)OC.C(=O)(C(F)CN(C)CC=C(C)C)NC C=CC(C(F)(F)F)NC(C1(CF)CCN(C(=O)CC2C(=O)NN=C2C)C1)=O c1(C(N2C(C)CC(NC(C(C)NC(C)=O)=O)C2)=O)ccc2c(c1)C(=O)NC2 C1(C(=O)NCC(C(=O)OCC)C)CCN(C(=O)Cc2scnc2C)CC1 C(=O)(C1=CCCCC1C)NCC(=C)CCNC(c1nc(O)sc1C)=O N1(C(C(C(C)C)NC(N)=O)=O)CCN(C(c2nccnc2C(N)=O)=O)CC(O)C1 N=c1ncn(CC(=O)NC(C2CCOC2)CNC(=O)Cc2cnns2)[nH]1 c1(C(N(CCC(C)NC(C2ON=C(C)C2C)=O)C)=O)cc2ccccc2nc1O Cn1ncc(C(=O)NC2CC(NC(c3cnc(O)o3)=O)C2)c1S(N)(=O)=O Cc1cc(C(C)(C)C)ccc1NC(=O)NCC1CCCCC1(C)C c1(C(=O)NC(C)(C)C(N)=O)ccc(CNC(=O)CC2CCC3CC23)nc1 c1(CCC(N2CCC(C)(c3cn(C4CC4)nn3)CC2)=O)cccc2c1OCCO2 N1(C(c2c(C)nn(C)c2Br)=O)CC(NC(=O)C(C)(C)C)C(C2CC2)C1 c1(OC)cccc(C2(C(=O)NCC3C4CN(C(=O)C(C)OC)CC34)CC2)c1 c1(NCc2c(C)cnc(F)c2)cc2c(cc1C(=O)O)CCCC2 N1(C(c2c(C)c(Cl)c(Cl)cc2)=O)CCC2CN(C(=O)CC(C)F)CC2C1 C#CC1CCC(CNC(=O)C(c2ccco2)NC(C2CCS(=O)CC2)=O)CC1 CC(C)C(F)C(=O)N(CCCCCNC(c1ccncc1-n1cccn1)=O)C Cc1cc2n[nH]cc2cc1C(=O)NCC(C)CNC(=O)C=Cc1nccs1 C12(CC(=O)NCC(C(=O)N3CCC(CC(F)F)C3)N(C)C)CCC(CC1)C2 C1(C(=O)NCC2CC(SC)C2)(NC(c2ccnn2C)=O)CC1(C)C C1(NC(CCCCCCC)=O)CN(C(=O)CN2CC3CC3C2)C2(CCCOC2)C1 C(=O)(C(C)(C)N1CCOCC1)NCC(C)NC(=O)CC1(C)CC1(Cl)Cl c1(C(=O)NC(CC2CN(C(C3(CC)CCC3)=O)C2)C)ncnc2sccc12 C1CCS(=O)(=O)C12CN(C(C1C3CCC(=O)C13)=O)C2.Cn1cnnc1C(=O)N c1(C(=O)NC(C(=O)N(CCOC)CC)C2CCC2)ccc(O)nc1 C1(NC(c2ccnc(C)n2)=O)CN(C(=O)CCCN(C)C)CCC1(C)C c1(NC(CNC(C2C(C#N)CC2)=O)=O)ccc2cc[nH]c2c1 c1(OC)ccc(Br)c2[nH]c(C(=O)NCC3CC3NC(=O)C(C)(C)C)cc12 Cc1cc(C(=O)NCc2cc(C=O)on2)n(C)n1.C1(C(=O)N(C)C)CC1 c1(C(N(C(CN(C2CCSCC2)C)=O)C2CC2)=O)cccc(-n2cncn2)c1 C(=O)(CCCC(=O)NC1CN(C(=O)C#CC2CC2)CC1O)N(CCC)CCC CC1CCN(C(=O)Nc2cc(F)ncc2Cl)CC1CNC(=O)OC(C)(C)C N1(c2c(OC)cncn2)CCC(O)(C(=O)NOCc2cccs2)CC1 C1(NC(=O)CC2CCOCC2)CCSC12CN(C(=O)COc1cncc(Cl)n1)C2 N1(C(C2N(C(C)=O)CCOC2)=O)CCC2(CC2)C1.c1(C(=O)N)cc(C)nc(C)n1 N#Cc1cc(C(N2CCCC3(CCN3S(=O)(=O)CCCl)C2)=O)cc2[nH]ccc12 c1(C=O)cnn2c1CCC2.CC1(C)CC(C)(CNC(=O)C(F)C2CCC2)C1.N C1(NC(CSS(C)(=O)=O)=O)CN(CCC2CC2)CC2(CCOCC2)C1 C1(NC(c2nc(CCC)oc2)=O)CC(C(=O)NCC(O)C(C)O)CC1O Cc1ccc(F)c(C(C)N(CCCC(=O)OC(C)(C)C)C(c2ccccc2)=O)c1F C1(CC)(CC)CN(C(=O)CC2CCC(NC(c3cnns3)=O)C2)CCO1 CCC(CCC(=O)N(C1CCC(CNC(C2CCC(O)C2)=O)CC1)C)OC C(=O)(CCC(C)(C)F)N1C(CN(C(c2coc(C(C)O)n2)=O)CC)CCC1 c1(C(=O)NC2CCN(C(C(CC)C)=O)C2(C)C)cc(S(=O)(=O)NC)c[nH]1 c1(C(=O)NC2CCN(C(C3NC(=O)OCC3)=O)CC2F)ccc([N+](=O)[O-])cn1 Cc1cc(O)nc(C)c1C(=O)NC1CN(C(C2CN(C3CCOC3)C2)=O)CC1C C1(OC)CC2CC1N(c1ccc(CC(=O)N(C)C)cn1)C2 C1CS(=O)(=O)CC1.c1(CCC=O)ccc(N(C)C)cc1.C#CC1(C=O)CC1.N C=Cc1cncc(C(=O)NCC2CCCC(NC(C34CCCC3C4)=O)C2)c1 c1(C(N2CCC(C(=O)Nc3scc(C(=O)OC)n3)C2)=O)c(F)cccc1F C1(C(C)NC(=O)CCc2ccn(C)n2)CCCN(C(c2cnc(C#N)s2)=O)C1 c1(C(N)=O)cc(C(=O)NCC(O)CNC(=O)C(F)(F)C2CCOCC2)n[nH]1 N1(C(c2cnc(C)nc2)=O)CCC2(CCCN(Cc3c(F)cc(O)cc3F)C2)C1 Cc1ccc(F)cc1C(=O)NC(CCC1CCC1)C(=O)NCCCCC(C)(F)F N1(C(CCOC)=O)CCCOC(CNC(C2(C#N)CC3CC3C2)=O)C1 c1cncc(Cl)n1.C1(N(C)C)CCC(C(=O)N)C1.C(=O)C.CC=CC.C=O c1(NC(c2ncc(C)o2)C)cccc(N2CCN(C)C2=O)c1 C1(N2C(C(=O)NCC)CCC2)CCCC12CN(C(c1nccc(=N)[nH]1)=O)C2 Cc1scc(C(N2CCCC(N(C(=O)C=CCn3cncn3)C)C2)=O)c1N CCCCCCC(C)C(=O)NC1CCCCCCC1NC(=O)Cc1scnc1C c1(C(N2CCCC(C)C2CNC(c2coc(Cl)c2)=O)=O)cc2n(n1)CCCCO2 C(=O)(C1=Cc2ccccc2OC=C1)NCCC1CN(C(CCCS(C)(=O)=O)=O)C1 C12(NC(C3C(CC)C3)=O)CCCC1N(C(C1(OC)CC(C)C1)=O)CC2 C1(NC(CC=CC)=O)CCCCC12CCN(C(=O)COCCN(C)C)C2 Cc1nc(NC(C2(C)CCN2C(=O)CCc2ccc(O)c(O)c2)=O)ccc1Br C=CCCCC(C(=O)NC1CCCC(C2CC2)C1)NC(=O)CSC1CC1 C12(CNC(C(C)(C3CC3)OC)=O)CC(CO1)N(C(C1CC3CC3C1)=O)C2 C(=O)(N1CC(C)(O)CO1)C1CC(O)(CNC(c2cn(CCC)nn2)=O)C1 C(C)(CC1CCC1)(C(=O)NCCC1CC1)OC.n1(CC=O)ccnn1.C CC(F)(F)C(C(=O)N1CCCC(C)(c2nn[nH]n2)C1)c1ccccc1 N1(C(CC(C(=O)OC)C)=O)CCOc2nc(C)ccc21 C1(CNC(=O)COCC2CC2)CN(C(c2nscc2Br)=O)CCC1(F)F C(=O)(C(F)CC(C)(C)C)NC(CC#CC)C(=O)NCCNC(c1ccoc1)=O Cc1c(C(N2CCCC2C)=O)noc1C1CC1.C1(C=O)CC(O)CN1C(N)=O.N N1(C(CSCC#C)=O)CC(NC(=O)C=C2CCC(C)CC2)CC1(C)CO C=CCC(C)C(=O)NC1CC(NC(c2cncc(NC)c2)=O)CC1O c1(OCCOC)ncccc1C(N1CCCC(C)C1)=O.C1(C(=O)N)C=CCC1 c1(CC(N2CCN(C(C3C(C=C)C3)=O)C(C)C2)=O)ccc2oc(C)nc2c1 c1(C(=O)NC2CCC(NC(C3C=C(C)CS3)=O)C2)c(C(C)C)n[nH]c1C c1(OC)ccc(Br)c(C(N2CC(O)CC2C(=O)Nc2ccns2)=O)c1F CCC(C)CC(C(=O)NCCCC(C)(F)F)NC(C1COCCC1C)=O Cc1cc(=NCCC(C)NC(=O)C2CCCc3sccc32)[nH]cc1[N+](=O)[O-] c1(OC)ccc(Cl)c(Cl)c1C(=O)N.C1(CCC=O)C(=O)NN=C1C.C(C)CO c1(NC(CC(CNC(CC(COC)C)=O)C2CCC2)=O)cc(O)ccc1F C(=O)(C1COCc2ccccc21)N1CCCC(O)(CNC(c2cscc2Cl)=O)C1 C#CCC(C)(C)C(=O)NCCC1CN(C(C2(C)CC(=C)C2)=O)CCCO1 c1(CNC(C(C=C)OC)=O)ncc(C(=O)NCCCCCF)cn1 c1(CC(C)C(=O)NCC(CO)NC(=O)C(c2ccccc2)=O)cccc(Cl)c1 c1(OC)cccc(C(=O)N)c1.c1(CCC(N2CC(O)(CC)C2)=O)c(C)noc1C C(C(C)(C)C(=O)NCC12CC1CN(C(=O)C(n1cnc(C#N)n1)C)C2)OC C(=O)(C(C)(C)C(C)N)N1CCC(c2c(CC)cccc2)C1 CCN=c1[nH]c(C(=O)NC23CCC(CN=c4[nH]nc(C(F)(F)F)s4)(C2)OC3)cs1 C1(COC)(NC(=O)C(C(C)C)NC(C2CC=C(C)CC2)=O)CC=CCC1 Cc1cccc(-c2nnc(C(C)Cc3cccc(Cl)c3)o2)c1 c1(OCOC)ccc(CN2CC3C(C2)N3C(c2ccc(C)o2)=O)cc1 C1(NC(CCC=C(C)C)=O)CCN(C(=O)CCc2c[nH]c(=N)[nH]2)CC1O c1(NC(NCC(O)C(F)(F)F)=NCCF)ccc2c(c1)OCCCO2 N1(C(c2cc(C)ns2)=O)CCCC(C(C)(O)C)C1.C(c1ccc(C)o1)=CC=O.N Cc1onc(C(=O)NCCCNC(C2CC(=O)N(C(C)(C)C)C2)=O)c1Br Cc1cc(Cl)ccc1C(=O)NCCCOCCN(C(=O)CCC1CCOCC1)C C1(CC=C)(NC(=O)COc2ccccc2F)CCCN(C(c2nc(C)cs2)=O)C1 N1(C(C2(C)CC(C)(C)C2)=O)CCC2(CCC2)C(O)C1.C(=O)CCC1CCCO1.N c1(OC)ccc(Cl)c(C(N2CCC(C(=O)Nc3cncc(Cl)n3)C(O)C2)=O)c1F C1CCCCC1.c1(C(C(N2CC(C(=O)NCC)(C)C2)=O)(F)F)ncc(F)cn1 c1(OC)nccc(C)c1NC(=O)C(N1CCC(c2cccc(F)c2)C1(C)C)=O C1(NC(=O)Cn2ccc(Br)n2)C2CC1CN(C(=O)CC1CC13CC3)C2 C1(NC(=O)CCCn2cncn2)CC(F)CN(C(C23COCC(C2)C3)=O)C1 C=C1CC2(C1)CC(C(=O)Nc1cccc(CNC(C3CCC3)=O)c1)C2.C N1(c2cc(NC(C3CCCCCC3)CCO)ncn2)CC=C(c2cncs2)CC1 C1(CC(=O)N)CCCC(C)(C)C1.n1(CC=O)cnc([N+](=O)[O-])c1.CCC(C)C CCCC(C(=O)NCc1ccc(C(N2CCCC2(C)CC(C)C)=O)s1)OCC c1(C(N2CCN(C(C(CC)(C)OC)=O)CC2C2CC2)=O)ccc(F)c2ccoc12 Cc1cnc(CCNC(C2CC(O)CN2Cc2c[nH]c(Br)c2)=O)nc1 N1(C(C2C(OC)C2)=O)CCCCC1Cn1ccnn1.c1(C=O)coc(Cl)n1.C Cn1nc(CNC(=O)O)cc1C=O.c1ccc(C=O)cc1.C=O.C1CC1 N(C1CCCc2c(F)cc(Cl)cc21)C(C1(CC#C)CCOCC1)=O c1(NCC2(CC)CC2)ccc(S(=O)(=O)N2CCN(C(C)(C)C)CC2)c(Cl)c1 C1(NC(C(COC)COC)=O)CCCCCC1NC(=O)C(c1cn(C)nc1C)C C1(C(C)C)N(C(=O)Cc2nccn2C)CC12CCN(C(=O)COC1COC1)CC2 N1(C(COC(C)C)=O)CC2(CNC(C3CCC(O)C3)=O)CC1CCO2 Cc1cc(C=O)c(C)s1.c1(C(N(CCCN(C)C)CC)=O)ccnn1CC C1(C(=O)NCC(=O)NCCC)CCCCCCN1C(=O)CCc1cncn1C C1(NC(c2ccc(C(C)(C)C)s2)=O)CCCC1(C)C.C(=O)(C=O)N.C1CC1 C1(NC(c2ccc(CC3CC3)s2)=O)CC2CCC1N2C(=O)C=C(Cl)Cl Cc1ccc(CC(=O)NCCCN(C2CCCC2)C(C2CCC(=O)C2)=O)cc1Cl C1(NC(=O)CCc2cscn2)CC(C(=O)N2CCC(c3nn[nH]n3)C2)=CC1O CC(C)(C(=O)NC(C1CCCCC1)CNC(=O)Cc1cccc(Cl)c1)C(F)F Cc1cc(C(=O)NCC(=O)NC2CCCC2)cc(C)c1.c1(C=O)ncc(C)cn1 c1(C=O)cccc(F)c1Cl.c1(C(=O)OC)ccc(C(=O)NC2(CC)CC2)cc1 c1(OC)cc(Br)cc(F)c1C(=O)NC1CC(C(=O)N)C1.c1cccc2ncsc12 c1(C(N(c2cccc(NC(C3CC(F)C(=O)N3)=O)c2)C)=O)nn(C)cc1Cl CCCCS(=O)(=O)CC(=O)N1CCC(CN(C)C(c2cccc(O)c2C)=O)CC1 c1(C(=O)NCC(CO)NC(C2CC=C(C)CC2)=O)cnc(N)c(N)c1 CC(C)(C)C(CNC(c1ccncc1F)=O)C(=O)N1CCC(F)(CO)CC1 Cc1ccn(CCC(=O)N2CC(CN(C)C(c3sccc3-n3cnnn3)=O)C2)n1 n1(CC(=O)NC(CNC(c2cccnc2S)=O)C2CC2)nc(O)ccc1=O Cc1c(C(N2CC3C(NC(=O)C(c4cccnc4)C)C3C2)=O)cnc2ccnn12 CC(C)CC(C)(C)C(=O)NC1CN(C(c2c(O)cccc2Cl)=O)CCC1CO C(=O)(CC(C)(O)C(F)(F)F)NC12CC(CNC(CCCC)=O)(OCC1)C2 C#CCC(C)(CC)C(=O)N1CCOC(c2ccsc2)C1 c1(CC)nc(N2CCCC(CNC(=O)C=CC3CC3)C2)c(C#N)cc1C C(=O)(CCCCCNC(=O)Cc1ccc(C)o1)NC(COC)(C)C1CC1 C(=O)(C(Cc1ccoc1)NC(=O)CC(C)c1ccco1)N1CC(CC(C#C)C)C1 C1(C(=O)NCCCNC(C2(N(C)C)CCC2)=O)CCCCO1 n1(CC(N2CCCC3(C2)CN(C(C24CCC2C4)=O)C3)=O)sc2ccccc2c1=O c1(C(=O)NC(C=CC(=O)NC2CN(CCC)C2)C)c(C)noc1N Cc1cc(Cl)c(F)cc1C(=O)NC1C2CN(Cc3ccc4n[nH]cc4c3)CC12 CC1CN(C(c2ncc(C(F)F)s2)=O)CC2(CCN(C(=O)CC3CC3(Cl)Cl)C2)O1 C(=O)(CCCCCC(C)C)NC(CCC)C(O)C(=O)NC(c1ccc(F)cc1)C N1(CC(=O)N(CCC(=O)OCC)C)CC(C)=CC(C)C1 N1(C(CC(=O)NCC#C)=O)CC=CC(NC(=O)C(O)C(C)C)C1 n1(CC)cccc(NC(C2CCN2C(=O)CC(C)c2ccco2)=O)c1=O Cn1cc(C(=O)NC23CC2CN(C(C2(C)CCCOC2)=O)C3)c2cc(F)ccc12 Cn1c(NCC(O)C(F)(F)F)nnc1C1CC(n2cncn2)C1 c1(CCCC)ccc(CC(=O)N(C)CCOCCCN(C)C(=O)C2CC2)cc1 N1(C(C2(C(CC)=O)CC2)=O)CC2=C(C1)CN(C(c1cc(Cl)cnc1C)=O)C2 c1(C(C)N(c2nnc(C(=O)N(C)C)n2Cc2cccs2)C)ncc(Br)cn1 N(C1CCCc2c(F)cc(F)cc21)C(=O)NCC1(COC)CCOC1 Cc1cccc(C(C)(C)C(=O)NCCCCNC(C2(C)CC2)=O)c1.C1CCC1 N1(C(CCc2cnc(C)s2)=O)CCC(NC(C2(C)CCCN2C)=O)C12CC2 C1(NC(c2cc(C)[nH]n2)=O)CC(C(=O)NC(C2CCOC2)CO)CC1O c1(OC)ccccc1C(C)(C)C(=O)NC1CCC1NC(=O)C.C1CCC1.O C1(NC(C(c2c(C)cccc2)C)=O)CCC2(CC1)CC2.C1(C=O)CS(=O)(=O)C1 C1(C=O)CC12CCOCC2.C1(CC(=O)N)CCCCC1.C1(COC)(C)CCC1 N1(C(C2C(C=O)C2)=O)CCCC12CCC2.c1(C=O)cccn1C1CC1.CC.O N1(C(C(=O)NCCCSC)c2ccoc2)CCC2(CC1)CC(=O)NC(=O)C2 Cc1[nH]nc2ccc(C(=O)NC3CN(C(C45CC(CO4)C5)=O)CCC3C)cc12 c1(C(C=O)C)cc(F)cc(F)c1.C1CC2(C1)CC2.C(C(=O)N)OCCOC N1(C(CC(C)(C)O)=O)CCC2C(C1)CN2C(=O)CCCOC(=O)N.c1ccsc1 c1(C(c2nnnn2CC2CCOC2)NC(CC=C)(C)C)cccc2c1CCO2 C1(C)(CC)C=C(C(=O)N(CC(C)N(C)C(c2onc(Br)c2C)=O)C)C1 c1ccc([N+](=O)[O-])c(O)n1.c1(C(C(=O)NCC2COC2)OC)cnn(C)c1.N Cc1cc(OC(F)(F)F)ccc1NCC1CCC(C)O1 C(=O)(C(C)(CC)CCCCC)NC1CN(C(C(CC=C)(C)O)=O)CC(F)(F)C1 C(C(CC(=O)NCC12CCC(CC1)O2)NC(C1C(C)C1C)=O)OC C(=O)(C(C#N)C(C)(C)C)N1CC(C(N(C)Cc2ncn(C)n2)=O)OCC1 c1(OC)c(F)ccc(F)c1C(N1CC(NC(=O)C(O)CC(C)C)C(F)C1)=O N(C(=NCCc1nc(-c2ccnc(C)n2)no1)NC(C)CCSC)C(CC)C Cc1noc(C(C)C)c1C(=O)NC(C1CCCCN1C(=O)C)C.c1cccs1.S C(=O)(C(C)C(F)(F)C(F)F)N1CCCN(CCNC(CS(CC)(=O)=O)=O)CC1 CCC(O)C(F)(F)C(=O)N1CCC(NC(c2[nH]c(C)nc2C)=O)C(C)C1 CCC(C)(C)C(O)C(=O)NCCN(C1CCCC1)C(c1cc(C)cc(C)c1)=O C1(C(=O)NC(C(C)C)CCN(C)C(C2CC2(F)F)=O)CCC(C2CCC2)CC1 C12(NC(COCCCCCC)=O)CC1CN(C(=O)C(C)OCCOCC)C2 c1(C(=O)NCC(CN(C(c2cnc(C)s2)=O)C)O)ccc(S(N)(=O)=O)cn1 C1(C(=O)NC(CC)C(=O)N2CCC(COC(C)=O)C2)CC=CC(O)C1 C(=O)(CS(=O)(=O)CCO)N1CCN(C(c2cc(OC)cc(O)c2)=O)CC1C(C)C N1(C(C2(C=C)CCC2)=O)CCC(NC(C2(C)CC2)=O)C(c2ccccc2)CC1 C1(C(=O)NC2CC(CNC(c3cc(C)ncn3)=O)C2)CCCC(C(N)=O)CC1 c1(C(=O)NCCN(C(=O)C)CC)c[nH]c2c(C)cc(F)cc2c1=O.CCF.O c1(CC(CN(C)C(=O)C2CC2)NC(CC=CCC)=O)ccccc1 C1(CC(=O)NCCNc2ccccc2)CNC2(CC2)CO1 C(CSC)(C(=O)N1CCCC1CNC(=O)CC(C)F)OC c1(C2C(CC)C2)c(C)[nH]c(C(=O)NCCCC)c1C.C(=O)(C)N.C(C)=O Nc1cnc(C(N2CCC(O)(CNC(=O)CC(O)CC3CC3)C2)=O)cn1 c1(CC(N2CC(C)N(C(c3nc(Cl)ccc3F)=O)CC2)=O)cc2ccccc2o1 C=C(C)CC(C(=O)N1CC(O)(CC)C1)NC(C)=O.c1nccn1C.C(=O)C.N N1(C(CC(=O)OCC)=O)CCC(C)(CNC(=O)CCC2CCC2)C1 C1(NC(=O)CC2CCCC23CC3)C2CC3C1C3C2C(=O)NCC.C1CC1.O C1(CC(=O)NC(CN(C(=O)CCc2cnoc2)CC)C)CC2CCC1CC2 C(=O)(CC(C(F)(F)F)NC(c1ncccc1Cl)=O)N1C(CC=C)CCCC1 c1(C(=O)NC(CNC(Cc2c(C)nccc2)=O)(C)C2CC2)cc2n(c1)CCOC2 C(c1ccc(C)cc1)=CC=O.c1(SCC)nc(C)c(CC=O)s1.C1CCC1.N c1(C=O)ccc(S(C)(=O)=O)o1.Cc1oc(C#N)cc1C(=O)N.C1(F)CCC1 CCC(CC)CC(=O)NC(CCSC)C(=O)NC(C)CCNC(C)=O N1(C(C(C)N(CC)CC)=O)CCCC2C1CCN2C(=O)CCSC CCCCC(CNC(c1cn(C(C)C)nn1)=O)NC(C1CCC1(C)C)=O c1(C(N(C)CCN(C(=O)C(O)CC(F)F)C)=O)ccnc(S(N)(=O)=O)c1 c1(OCC(N2CC(C)CCC2)=O)ccc([N+](=O)[O-])cc1.C(=O)(CCCN(C)C)N O=C(C1=CC2CCCC12)NCC12CCCC1CN(C(c1cc3sccc3[nH]1)=O)C2 C(C(C)(C)CN=c1[nH]c(N(C)CC2CCCN2C)nc2c1COC2)OCC C(CC(CC)(CC)NC(c1coc(C2CC2)n1)=O)NC(C1C(=C)C1)=O c1(C(=O)NCC(C(C)C)N)ccc(NCCF)cc1 C1(C(=O)NC2(COC)CN(C(=O)C3=C(Cl)CC3)C2)CCCC2(CC2)C1 C1(CCC=O)(N(C)C)CCCCC1.C1(NC(CC2(C)CCC2)=O)(C)CCCC1.N N1(C(CCCCN(C(C)=O)C)=O)CC2CCN(C(C3CCCCN3C)=O)CC2C1 c1(C(N2CCN(C)CC2CNC(=O)CN2CC=CC2)=O)ccc2n[nH]cc2c1Cl CN1CC(=O)N(CCC(=O)NCCCN(C(C2CCCCS2)=O)C2CC2)C1=O c1(NC2CCN(c3cn(C)nc3)C2=O)ccnc(Br)c1[N+](=O)[O-] N1(C(c2ccc(CC)s2)=O)CCC2(NC(c3cn(CC)nc3C)=O)CC2C1 c1(C(=O)N)cc(F)cc2cnccc12.c1(SC)ccc(O)c(C(=O)NC(C)C)c1 N1(C(C(CC(F)F)NC(CCC(=O)NC)=O)=O)CCC12CCSCC2 C1(NC2CC(c3c(OC)ccc(OC)c3)C2)C(=O)OC2CCCC12 c1(NC(CN(C(=O)C(C)C(C)C)CC)=O)cc(C)c(F)cc1C c1(CCCC=O)ccc2c(c1)CC(=O)N2.C1(C)(C(N(C)CC)=O)COC(=O)C1 CCCCC(C)CCC(=O)N(C1CCN(C(=O)CCNS(C)(=O)=O)CC1)C c1(OC)cccc(F)c1C(C)NC(=O)NC(c1ccc(Br)c(F)c1)C CCC(CC(=O)NC1CC(N(C(=O)C2=CCOC2)C)C1)Sc1ccc(C)cc1 N1(C(C=CCC(C)(C)NC(c2c(C#C)cn(C)n2)=O)=O)CCC2CCC(O)C1C2 N1(C(CC(C)C2CC2)=O)CCC2(C1)CN(C(=O)CN1CCN(C)C(=O)C1)CCO2 c1(OC)cccc(CC(=O)NC2CN(C(=O)Cn3ccnn3)C3CC23)c1 C1(C(CNC(=O)CC2CC2C(F)F)=O)CCC2CC2C1 N1(C(CC(C)C)=O)CCc2nn(C)c(C(=O)Nc3ccns3)c2C1 C1(NC(c2c(COC)cccc2)=O)CCC(O)CN(C(c2cnc(=N)[nH]c2)=O)C1 N1(C(CCCC(OC)OC)=O)CCCc2ccc(C)nc21 C1(C=O)CC2(C1)CS(=O)(=O)C2.Cc1sc(O)nc1C(=O)NC(C)C(C)C CC(CC(=O)N(C1CC1)CC1CCCN1C(=O)Cc1cccs1)N(C)C C1(CNC(C(CNC(C(CSC)O)=O)CC2CCCC2)=O)CCCC(C)(C)C1 C1(C2CCOCC2)(C(=O)NC2CC3CN(C(C4(C)CCCS4(=O)=O)=O)CC32)CC1 c1(C(=O)NC2CCN(C(CCC(C)C)=O)C23CC3)cc2cc(Cl)cc(Cl)c2[nH]1 N1(C(c2cc(C)sc2)=O)CC(C(=O)NCC2CC23CCOC3)CCC1C c1(C(=O)NCC2(C)CCN(C(c3nc(C)n(C)n3)=O)C2)cccc2nc(Cl)cn12 N1(C(C2CCCOC2)C(=O)Nc2c(OC)cccc2)CCCCC(SC)C1 C12(C(=O)NCCN(CCCC)C)CC1CCN2C(=O)C(C)OCCOC C(=O)(C1CCCc2cccnc21)NCCCNC(=O)CC1(C(F)F)CC1 C1(NC(c2cn(CCNC(c3ccc(CC)s3)=O)nc2)=O)CN(C)CC1.O C1(C(=O)OC)CC(C(=O)NCCCNC(=O)CCc2nccs2)C12CCC2 C1(C(=O)NCC(C)N(C)CCF)CSCCN1C(=O)CCCCN(C)C C1(CNCc2c(C)ccnc2Cl)CCc2cc(F)ccc2O1 C(=O)(C(F)C(=O)NCCCN(CCCCNC(=O)C(F)CC)C)OCC C1(NC(C(C)N2CCC2)=O)CCC12CN(C(=O)CC1C(C)(C)C1(C)C)C2 c1(C(=O)NCC(CC=C)NC(=O)CCCC(=C)C)ccc2n[nH]c(CCC)c2c1 c1(CN2CC(NC(C(C(C)C)NC(C)=O)=O)(CO)C2)cc(C)ccc1C c1(NC(c2nc(-c3cccc4ncnn34)cs2)=O)ccc2cc[nH]c2c1 Cc1cccc(NC(=O)CCN(C(=O)CNC(=O)C(C)(C)C)C)c1C CCC(C)(C)C(O)C(=O)N(C1CCCCN(C(=O)C(C)(C)C(=O)OC)C1)C c1(C(=O)NC2(CO)CN(C(c3c(C)oc(Cl)n3)=O)C2)cc2c(nc1O)CCOC2 c1(N(C)C)nccc(=NC(=O)C2CCN(C(C3CCCCO3)=O)CC2O)[nH]1 C#CC1(NC(=O)C(CCOC)NC(=O)C(=O)NC2CC2)CC2CCCC12 C1(NC(c2occ3c2CCC3)=O)CC2COCC(C1)N2C(C1CCCC(F)C1)=O N1(C(c2c(NCC)scn2)=O)C(C)CC2CN(C(C3(C)CC=CCO3)=O)CC12 c1(C=O)ccc(C)c(C(F)(F)F)c1.C(CO)(C(=O)NC(C1CCCC1)C)OC c1(C(=O)NC(CNC(C(CC#C)O)=O)(C)C(C)C)nc(OC)cc(OC)n1 N1(C(c2c(C)ncc(C)c2)=O)CC2(CCN(C(C3CCC4CC34)=O)CC2)CC1C O=C(C1=NNC(C(F)(F)F)C1)NCC1CCC1NC(c1ccccc1Br)=O CC1(C)CC(C(=O)N2CCCC2(C)C(N2CCC(CC3CC3)C2)=O)=NO1 c1(NC(C2CCC(NC(CC(OCC)OCC)=O)CC2)=O)ncc(C)nc1Br C1(NC(CN(C)C(=O)C2CC2)=O)CCC(NC(C23CCCCC2C3)=O)CC1 N1(C(c2c(C)nsc2)=O)CCC(C2(NC(=O)CSC(F)(F)F)CC2)C1 N1(C(C(COC(C)=O)C)=O)CC=C(C(C)(C)C(=O)NCCc2c[nH]nc2C)C1 c1(C(=O)NCCOCC#C)cccc(NC(=O)CCc2cnoc2)c1 O=C(C(F)C(F)(F)F)NC1CCC(NC(c2ccc(-n3cncn3)nc2)=O)C1 C(=O)(C(C)CCO)NCc1occ(C(N(C)CC2N(CC)CCC2)=O)c1 Cc1cccc2c1OC(C(=O)NC(C)(C)CNC(=O)C1=C(C#N)CCC1)C2 c1(C(=O)NCC(C)(CO)NC(C2C=CCC2)=O)cc(=O)c2cc(F)ccc2o1 C=Cc1ccc(C(N2CC(C(=O)NC3CC34CCCC4)(CC)C2)=O)cc1 N1(C(C2(NC(Cc3cc(C)[nH]n3)=O)CCC2)=O)Cc2c[nH]nc2C1 C1(C(=O)NCC(C2CCN(C(c3ccns3)=O)CC2)C)CCC(O)CC1 c1(OC)ccc(CC(=O)NC2CCC(NC(C3CCCCC3C)=O)CC2)cc1 N1(C(C(n2ncc(C)c2)C)=O)CC2CCCC(C1)N2C(c1cnc(N(C)C)s1)=O Cc1cc(C(N2CCOC(Cc3cn(-c4ccc(Cl)cn4)nn3)C2)=O)ncc1Cl c1(C(=O)NC2CC(CCNC(C(F)=CC)=O)C2)ccc(OC)cc1OC CC1CCCC(CNC(=O)N(c2c(Br)cnn2-c2ncccn2)CC(F)F)O1 c1(C(N(CC(C)NC(C23CSC(C2)C3)=O)C)=O)cnc(-c2ccccc2)o1 N1(C(CC2CN(C)CC2O)=O)CCN(C(C2CS(=O)(=O)C2)=O)C(C2CC2)C1 c1(C(C(=O)NC)N(C)Cc2ccn(CC)c2)ccc2c(C)[nH]nc2c1 C(CN=c1[nH]ncs1)(C1CCCC1)OC.C1(CC(=O)N)CCCN(C(C)C)C1 Cn1nc(C(=O)NCC(CO)NC(=O)CCOc2cccc(F)c2)cc1Br CCCCCCCCC(C)C(=O)N1CCC(O)(c2ccccc2Br)C1 C1(CC#C)(C(=O)NC(C)(C)CCCF)CCN(C(=O)CCCCN(C)C)C1 C1(C)CN(C2CCN(C(C3CN(C)C(=O)N3)=O)CC2)C1=O.C#CCCC(=O)NC Cc1[nH]cc(C(=O)NCCCCNC(C2CCN(C)C(C)C2)=O)c(=O)c1Br N1(C(CCC(C)C)=O)CCC(C)(NC(c2cnc(CC3CC3)s2)=O)CC1 c1(N2C(CNC(C34C(C)OC(C)(C3)C4)=O)CC3(CC3)C2)ncnc2sccc12 S(=O)(=O)(c1ccc(NCCc2cccc(F)c2)c(F)c1)NCC(CC)N(C)C CC(CCC(C)(C)C)C(=O)N1CCC(O)C1C(=O)NC(CCO)C(F)(F)F C1(NC(c2ccc(COC)nc2)=O)CN(C(c2sc(OC)nc2C)=O)CC1S C12(C(=O)NC3C(NC(=O)C=CC(F)(F)F)C3)CC(CC(F)F)(C1)C2 c1(N2CCN(C(C3C(C=O)C3)=O)C(C)(C)C2)ncc2ccc(F)cc2n1.CC(C)C.O N1(C(C2C(CC)N(C(=O)C(CCOC)OC)CCC2)=O)CC(C)OCC(C)(C)C1 C(=O)(C1=C(Cl)CCOC1)NCC(C1CCOC1)NC(C(F)=CCC)=O C(CC(C(=O)NCCCN1CCC1)NC(c1c(Cl)cnn1C)=O)OCC CCC(C)CCCC(=O)NC(Cn1ccnn1)C(=O)N(C(C)CC(N)=O)C C(C(C(=O)NC1CC2CC(OC)C2C1)C(C)C)NC(c1c(NC)cncc1)=O c1(NC(C2N(C(c3ccc(C(C)O)cc3)=O)CCOC2)=O)ccc(I)cc1F CC1CC(NC(C2(NC(=O)C)CC2(C)C)=O)C(=O)O1.C(=O)C(C)(C)C c1(OC)ccc(CN2CCNCC2C(=O)NCC(C)(F)F)c(C(F)(F)F)c1 c1(C(N(CCC)C(C)C)=O)cnc2n1CCOC2.C1(COC)CC1C(=O)N C1(C=O)CNC(=O)C(C)(C)C1.C(CCCC)N(C(CC1(NC(C)=O)CC1)=O)C C1(NC(=O)Cn2nccn2)CCN(C(c2cc(C(F)F)ncn2)=O)CCC1CO CCCCC(C(=O)N1CCN(C(c2ccoc2C)=O)C(CC)C1)N(C)C CCCCCCCC(F)C(=O)N1CCC2CN(C(=O)C(C)CO)CC2CC1 C(=O)(CC1=CCCCC1)N1CCC(C(CNc2ncc(C)cn2)(C)C)CC1 N1(C(CCC=C)=O)CC2CS(=O)(=O)CC2(NC(=O)Cc2cn3ccccc3n2)C1 c1(C(=O)NCCCCCCN(C(C2N(CC)CCCC2)=O)C)ccc(C)cc1N C1(c2nc(COCC)nn2-c2cncc(Br)c2)CC2(CC(C)=NO2)C1 C(=O)(C(CO)NC(=O)CC(C)O)NCCC(C)c1cn[nH]c1 c1(C(=O)N)cccc2c1CCC2.C1(COC)C2CCN(C(C3CC3(C)C)=O)CC12 CCC(F)(F)CC(=O)NC(C)(C)CCC(=O)NCCc1[nH]cnc1C N1(C(Cc2nc(CC)sc2)=O)CCOC(CN(C(=O)C(C)n2ccnn2)C)C1 C#Cc1ccc(Cl)c(C(N2CCC(C)N(C(=O)C(CCC)N(C)C)CC2)=O)c1 N1(C(=O)OC)CCC(NC(=S)NCc2ccsc2)CC1 N1(C(C(C)C2CCC2)=O)CC(C)(C)CC(C)(C)C1.c1(C=O)cc([N+](=O)[O-])c[nH]1.N Cn1cc2ccc(C(N3CC4CC(CNC(c5cscn5)=O)CC3C4)=O)cc2n1 c1(C(N2CC(C)(C)C(NC(=O)Cc3cnoc3)C2)=O)c(F)ccc(Cl)c1[N+](=O)[O-] C1(CNC(c2ccc(F)cc2F)=O)CN(C(=O)C2=COCC2)CC1(F)F c1(C(N(CCN(C(CC(=O)NCC#C)=O)C)C)=O)cc(CC)cc2c1OCC2 c1(C(N2CCCC(C)C2CNC(=O)CC2=NNC(=O)C2)=O)nccc2ccsc12 c1(C(C)=O)cc([N+](=O)[O-])c(NC(C2CC3CC3N2C(C2(Br)CC2)=O)=O)s1 C#Cc1cccc(C(N2CCC(C)C2CNC(c2cccn2C(C)C)=O)=O)c1F C1(CN(C)C(C2(N(C)C)CCC2)=O)CN(C(=O)CO)CCO1.C1CCCOC1 C(=O)(C(C)C(CC)CC)NC(CC#C)(C)C(=O)NCCC1CCCC1 c1(C(N(C2CCN(Cc3cc(C)c(Cl)c(C)c3)C2)C)=O)c[nH]c2cccc(C)c12 Cc1nccc(=NCC2CN(C(c3cccc(N4CC=CC4)c3)=O)CCC2C)[nH]1 C1(CC(=O)N(C)CC2(CO)CC2)CCN1C(C1CC=CC1)=O C1(CC)CCC(C)CN1C(C1(F)CCN(C(C2CC3CCC(C2)O3)=O)C1)=O CC1CCC2(CCN(C(=O)Cn3cc(-c4cccc(Cl)c4)nn3)C2)C1 c1(C(=O)NCC#CCNC(C(CC)SC)=O)cc2c(Cl)ccnc2s1 N1(C(Cc2cn(CC)nn2)=O)CCCC2(NC(=O)CN3CCNC3=O)CCCC12 c1(CC)nc(C)ncc1C(=O)NCCCCCN(C(=O)CCCCCSC)C n1(CC)cnc2c(NC3CC=CCC3)[nH]c(=NC3C=CCC3)nc12 N1(C(C(=O)NCCCC)CC2CCCCO2)CCc2ccc(Cl)c(Cl)c2C1 C1(NC(CC(C)(C)C)=O)CCCCC12CCN(C(=O)COc1cccc(O)c1)C2 c1(N2CCC(CN(CC)CC)C2)nc2c(c(=NCC(F)CO)[nH]1)CSC2 N1(C(C(C(C)C)F)=O)CCC2(CC1)CN(C(=O)CC1CCC(C)C1)C2 CCC(CC(=O)N(CCC(=O)N1CCOCC(O)C1)OC)SC C1(c2cn(C)nc2)CS(=O)(=O)CCN1C(=O)OCCCCC(=O)O c1(N2CCC3(N(C)CCC3)CC2)nc2c(c(=NC3CC(NC4CC4)C3)[nH]1)COCC2 Cc1ccc(-n2cnnc2SCC(O)CC2CC2)cc1 c1(NC)ccc(F)cc1C(=O)NC1CCC1NC(=O)C(C)(O)C(C)C C1(CNC(C2C(=C)C2)=O)(NC(c2cccnc2CC)=O)CCCCCC1 c1(SC)cccc(F)c1C(=O)NCC1CCCCC1NC(c1ccnnc1C)=O C#CC1(CO)CCN(C(=O)CCCC2CCCC2)CC1.C12CCN(C1)C(=O)CO2 CC1CN(C(=O)CC2(C)CCCC2)CCN1C(=O)Cc1ccc(Br)cc1F N1(C(CC)=O)CC(C=O)C2(CCC2)C1.C1(O)CCC(C)(C)C1.C(=O)(NC)N C(=O)(C1=NOC(CNC(C2CCC3(CCC3)O2)=O)C1)NCCC(N)=O n1(CC)ccc(=NC(=O)C2=CC(O)C(NC(=O)C(C)(C)CCOC)C2)[nH]1 Cn1ncc([N+](=O)[O-])c1NC1CCCCC1CNC(=O)Cc1cccc(F)c1 C#CC1(C(=O)NCCCC=C)CN(C(C2CC(=O)CS2)=O)C1 C1(N(C(c2occ(C)c2C)=O)C)CCCN(C(c2cccc[n+]2[O-])=O)CC1 C(=O)(C1CCc2nccn21)N1CC(C(C)C)N(C(=O)CC2CC=CC2)CC1 N1(CC(N=c2ccn(-c3c(C)cccc3)[nH]2)=O)CCC2(CC1)CC(O)CCO2 Cc1cc(C(F)(F)F)cc(S(=O)(=O)Oc2ccc3cc[nH]c3c2)c1 CC1=C(C(=O)NCC23CN(C(C4(N(C)C)CCC4)=O)CC2CCO3)CCCC1 N1(C(C2C(C)C2)=O)CC(O)CC1CNC(=O)Cc1cccc(F)c1 N1(C(C2NC(=O)OCC2)=O)C2CCC1CN(C(=O)CCC1CCC1)C2 N1(C(C2C(NC(C3OCC(C)(C)C3)=O)COCC2)=O)CCCCC(CO)C1 c1(Cc2ncc(C)cc2Br)ccc2c(c1)CN(S(=O)(=O)c1cccnc1OC)C2 N1(C(C2N(C(C)=O)CSC2)=O)CCCC(C)(NC(c2c(Br)noc2C)=O)C1 c1(C(N(CC(=O)NCC2CCOC2C)CCOC)=O)cccc(F)c1C C12(C=O)CCC(CC1)C2(C)C.C(C)(C)(CCC)NC(c1c(OC)scc1)=O.N C1(N(C)C)CCCN(C(=O)C=CCNC(C2C=CCC2)=O)CC1 C1(C(=O)NCc2n(CCCC)nnn2)Cc2ccccc2C(=O)O1.C(C)C N1(C(c2c(SC)ccc(N)c2)=O)CCCC1C1CCCCN1C(C1CCC1)=O c1(C(=O)OC)ncoc1CNC(=O)C=O.C1CCCN1C(=O)C(C)(C)C C(CC(C(C)(C)C)NC(=O)CCc1ccccc1)N(C(=O)CCc1nncs1)C c1(C(C)OC(CSCCCC)=O)c(Br)c(C(F)(F)F)nn1C Cc1cccc2c1OC(C(=O)NC(CO)C(C)NC(=O)Cc1cc[nH]n1)C2 C1(C(=O)NCCC(C)NC(c2ccc(Br)cc2)=O)Cc2cccnc2C1 C(CN=c1[nH]ccc(=NCCNS(C)(=O)=O)[nH]1)C1CC(C)CC(C)(C)C1 CC(C)CCC(=O)NCCCNC(=O)CCCNC(=O)Cc1scnc1C C(=O)(CCC(C)NC(=O)C(=O)NC(C)C)N1C(C)(C(=O)NC)CC1 N1(CCCNC(CCSCCCC)=O)CCN(C(=O)COCCC)CC1 n1(CCC(N2C(CNC(=O)CCc3cnc[nH]3)C=CC2)=O)cnc2ccccc12 c1(C(=O)NC(C)CCNC(=O)C(O)C2CCC2)ccnn1C1CCOCC1 C1(C(F)(F)F)(C=O)CCCCO1.C1(C(N(CCC)C)=O)CCC(=O)N1.CC.O c1(CCN(C(C(=O)NC(C(=O)OC)C)C2CC2)C)ncc(Br)cn1 c12ccc(c(C)n1)-c1cn(nn1)C2.N1(C(C)=O)CCC(c2cnc(Cl)s2)C1 C1CN(C(=O)CCN(C2CCCCC2)C)CC1(C)C.C(C)(C(=O)N)(C1CC1)OC CC(C)C(CNC(C1COCC1C(N)=O)=O)C(=O)N(C1COC(C)(C)C1)C C12(NC(=O)C3=COCCC3)CCCCC1N(C(=O)Cc1ccc(Cl)cn1)CC2 C1(C(N(CCNC(c2cccc(C3CC3)c2)=O)C2CC2)=O)CCCCC1O c1(N2CCCC(NC(c3c(C)nsc3)=O)CC2)ncnc2c1cnn2C C1(NC(C=CCC)=O)CC2(CCCN(C(=O)CCC3CCC(=O)NC3)C2)C1 Cc1cccc(C)c1OCC(N1CCC(C)C1)=O.c1(C(=O)N)ccc(F)c(Cl)c1 N1(C(C=CC)=O)CCOC2(CCN(C(c3cc(C)c(C(F)F)cn3)=O)C2)C1 CC(CCCC(=O)NCC1(C(F)(F)F)CC1)NC(c1cc(Cl)cs1)=O CC1CC2CCC(C(=O)NC3(C4CCN(C(=O)CC5C=CCC5)C4)CC3)CN2C1 C1(CNC(c2cc(C)n(C(C)(C)C)n2)=O)CCN(C(c2cncs2)=O)CC1C CC(C)CC(O)CC(=O)N1CC(C)N(C(=O)CC2CCCNC(=O)C2)CC1C CC1CC(NC(c2cncc(C3CC3)c2)=O)CN1C(c1sccc1Cl)=O C(=O)(CCCCCS(N)(=O)=O)N1CCCCC(NC(CC(C)c2ccco2)=O)C1 Cc1cc(OC(F)(F)F)ccc1C(=O)NC1CCN(C(C2CSCCS2)=O)CC1 CC(C)(F)CCC(=O)N1CCC(NC(C2CCCOCC2)=O)C(F)C1 N1(C(C=C(C)C)=O)CCCC(C2CCN(C(=O)CC(C)C(F)F)CC2)C1 N1(C(C2(C)CCN(C(c3c(C)ccs3)=O)C2)=O)CCn2c(O)nnc2C1 c1(C(=O)Nc2cn(C(C)C)nc2)cnc2ncc(-c3cnn(C)c3)cn12 c1(C(=O)NCC2N(C)CCN(C(C=C(C)C)=O)C2)ccc2ccncc2c1 Cc1ccc(C)c(NC(N2CCCN(C(c3sccc3I)=O)CC2)=O)c1 c1(N2CCC(NC(Cc3ccc(CC)cc3)=O)CC2C)ncc2c(n1)CCCC2 N1(C(C(CC#C)C2CC2)=O)CCN(C(c2ccccc2NC(N)=O)=O)C2(CC2)C1 C(CCC(F)(F)F)NC(c1ccccc1NCCn1cc(CCCO)nn1)=O C(=O)(CC(C)(C)CC(F)F)N1CC(CCC)C(NC(C2CCCN2C)=O)C1 N1(C(c2n(C)cc(F)c2)=O)CCC(C(=O)NC2CCCCC2F)C2OCCC12 c1(C(=O)NC2C3CCN(C(c4ncn(C)n4)=O)CCC32)cncc2ccccc12 c1(NC(COC)COC)nc(N(CC(C2CCCCC2)C)C)nc2c1cnn2C CCCC(CCC)C(=O)NC1CN(C(c2cnn(C)c2C#N)=O)CC1SC c1(C(=O)N)sc(-c2c(C)noc2C)nc1C.C1(OC)CC(C(=O)NC2CC2)C1 CCC(CC)(CO)C(=O)NCCNC(C1CCCN(C(=O)C(C)N(C)C)C1)=O c1(C(N2CC(NC(c3cnc(C(C)C)[nH]3)=O)C3C2C3)=O)cc(F)c(F)c(F)c1F CC1=C(C(=O)NCCCNC(=O)C2CCCc3ccnn32)Cn2nnnc2N1C C(=O)(C1=CNC2=NCCCN12)NCCCCNC(C1(C)CCC(=O)NC1)=O Cc1cc(N)ccc1C(N1CC(CNC(C2CCCCN2C)=O)CC(C)C1)=O CC(F)(CNC(C1CC(CC(F)F)C1)=O)CNC(C1CC=CCO1)=O C#Cc1ccc(N(C(=O)C(C)(C)CC2CC2)C(C)=O)cc1.n12cc(cn1)C2 N1(CC(=O)NCCC)CCC(O)(CO)C1.C(=O)(C(F)(F)c1cnn(C)c1)N C1(NC(=O)CC2(O)CC2)CCC2(CC1)CCN(C(=O)Cc1cn[nH]c1)CC2 N1(C(CC=C=C)=O)CC(CNC(=O)CCc2ccccc2OC)C(COC)C1 C=CCCCCCCCC(=O)N1CC2OCCN(C(=O)C=Cc3ncc[nH]3)C2C1 C1(NC(C2CCC(NCc3n[nH]c(O)n3)C2)=O)CCCC(F)C1 C(CCCC(=O)N1CC(O)(C(C)NC(c2cccc(NC(N)=O)c2)=O)C1)SC C(C)(N=c1nc(N2CCC(C)(F)CC2)c2cc(F)cc(F)c2[nH]1)c1nc(CC)sc1 C(=O)(C(CNC(c1cc(C)co1)=O)CC1CCCC1)OC C1(CCC)(NC(=O)CO)CCN(C(=O)C(C)(C#N)CC)CC1.c1cc(C)no1 C1(C(=O)NC2CC(OCC(=O)N(C(C)CCO)C)C2)CCC(F)C1 C1(NC(C(C2CN(C(C3CCCC34CC4)=O)C2)OC)=O)CC(C)(OC)C1(C)C C1(C(N(C(CC)CC)C)=O)OCCC1CNC(=O)C(O)c1ccsc1 N1(C(c2cn(C)nc2O)=O)CCC2(CC(NC(=O)Cn3cnccc3=O)CO2)C1 C(=O)(CC1CN(C)c2ccccc21)NCCC(C)N(C(c1c(C)occ1)=O)C C(C1OCc2ccccc21)c1onc(C2C(F)(F)C23CC3)n1 C#CCCC1=C(C(=O)OCC)C(c2ccc(C)cc2Cl)NC(=O)N1CCF N1(C(c2nc(OC)nc(O)c2)=O)CCC2C(C1)CN2C(=O)C(C)n1ccnc1 C1(NC(C2CCCCO2)=O)CC2(C1)CC(NC(=O)C(O)C(F)(F)F)C2 c1(CNCCc2cc(C)ns2)c[nH]c2ccc([N+](=O)[O-])cc12 c1(C(=O)N)cc(C)cnc1Cl.c1(CSCC)cc(C(=O)N(C(C)C)C)no1 Cc1cc(Br)ccc1C(N1CCC(C(=O)Nc2cnccn2)C(O)C1)=O c1(NC(C2(C)N(C(CC3(COC)CC3)=O)CC=C2)=O)ccc(Cl)cc1C Cc1cc(C(=O)NC2CCN(C(=O)CSCC=O)C2)c(O)nn1.C(C)(C)C CN1CCC2(CC1)CN(C(=O)CC(C1CC1)NC(c1cccn1C)=O)C2 C=CC(C)(CC)C(=O)N1CCOC(CNC(=O)CCCC2CCCO2)C1 C1(NC(C=C2CCN(Cc3cccc(C(=O)OC)c3)CC2)=O)CCCCC1(F)F N1(C(C2C3CCC(C3)N2C(=O)CSc2cccc(Cl)c2)=O)CC2CCCCC2C1 Cc1c(C(N2CC(O)(C(C)NC(=O)Cn3cc(Br)cn3)C2)=O)cccc1N C1(C(C)NC(C2=NOCC2)c2nnnn2-c2ccccc2Cl)CCC2(CC1)COC2 N1(C(C(C2CC2)OCC)=O)CC(NC(=O)Cn2nc(C)nc2C)C(O)C1 N1(C(c2cc(C)sn2)=O)CCC2(C1)CN(C(c1csnn1)=O)CC(C)O2 C(=O)(C1=COCCC1)NC(c1cn(C)nc1)C(=O)NC1CCC(CO)C1 C1(NC(C2CN(C)C2)=O)CCC12CCN(C(c1cnc3c(c1)CCOC3)=O)CC2 c1(C(=O)NC(CC=C)CNC(c2cc(OCC)no2)=O)nc2ccccc2[nH]1.O N1(C(C2(C)CCCC2)=O)CCC2(C1)CN(C(C1COC(=O)N1)=O)CCO2 CCCC(C)(O)C(=O)NCCN(C(=O)CCCC(=O)OC)C1CCCC1 C(=O)(C1=NOC(C)(CNc2cccc(CC(=O)OC)n2)C1)OC C1(NC(C2CCCC2C(F)(F)F)=O)(CO)CCN(C(c2coc(Cl)n2)=O)CC1 C(C)(CC(=O)NCC(C)(C)NC(=O)CCc1cc(C)[nH]n1)OC c1(C(N2CC(CC(=O)NCc3nccs3)C2)=O)ccc(I)c(F)c1F C1(NC(=O)C(F)=C2CCC2)CCC(NC(c2cnc(-c3cccnc3)s2)=O)CC1 c1(C(=O)NC2(CNC(CCN(C)CC)=O)CC2)ncnc2sccc12 C1(C(N2CCCC(C(C)NC(CCn3c(C)ncc3)=O)C2)=O)C2CC3C(C2=O)C13 N1(C(=O)NC(C)CCC(C)(C)C)CCSc2ccc(Cl)cc21 n1(CCC)cc(C(N2CC(C)(CCC(=O)NCC(C)CC)C2)=O)nn1 c1(C=O)ccc(Cl)cc1.C1C=CCC1.C(C)(C(=O)NC)OCCOCC c1(C(=O)OC)cnc(C)nc1N(C1CCCN(C(c2cnc(C(C)C)[nH]2)=O)C1)C C=CCC(CNC(=O)CC(C)(C)CNC(=O)C(F)C1CCOC1)CC(C)C C1(NC(Cn2ccc(C)n2)=O)CC2CC1N(C(=O)Cc1cc(C)[nH]n1)C2 S(=O)(=O)(c1ncccc1Cl)NC(c1ccc(F)c(F)c1)C C(c1cnc(C(C)(C)C)s1)=CC=O.CC(C)CO.CC=O.[SH](C)(=O)=O.CN C1(C(C)NC(c2nc(NC(C)=O)sc2)=O)CCCCN1C(=O)C1=CCC1 N1(C(C2=CCC(NC(=O)C(F)F)C2)=O)CCc2nccnc2C1 c1(C(=O)OCC2(C(=O)OC)CC3C=CC2C3)ccc(Cl)c2c1OCCO2 C1(C(N(C(CCNC(c2c(C)c[nH]c2)=O)C)C)=O)C2(CCC2)C12CCC2 N1(C(c2c(Br)cn(C)n2)=O)CCCC(O)(CNC(C2CCC(O)C2)=O)C1 c1(CC)cccc(OCC2CC2)c1.c1(C=O)ccccn1.C1(C(=O)N)CC1 c1(C(=O)NC2CN(Cc3c(C)ccc(OC)c3)CC2F)cc2cc(Br)ccc2s1 c1(CN2CCC(CC(=O)NCc3cc(C)no3)C2)ccc(O)c(C)c1 N1(C(C(c2c(C)noc2C)(C)C)=O)CCN(C(C2C3CC4C(C3)C24)=O)C(C)C1 c1(C=O)cnn(CCC)c1C.n1(CCC=C)cc(C(=O)NC2CCC2C)nn1.N N1(C(c2c(CC)n[nH]c2)=O)CC(C2CC2(F)F)C1.C1(C(=O)N)CC2(CCC2)C1 N1(C(CC2(CSC)CC2)=O)CCCC(NC(C2(C)C=CCCC2)=O)C1 CCCCCC(C)(C)C(=O)N(CCCNC(=O)C(c1cccc(F)c1)O)C1CC1 c1(N(C2CCN(C(C3CCC4(CC3)CC4)=O)C2)C)cncc(C#N)n1 N1(C(C2CCC(NC(=O)C(F)C3CCC3)C2)=O)C2CCC1CC(F)C2 Cc1cc(C#N)ccc1C(=O)NC.C1(CC(N2CCCC2)=O)CCC(=O)NC1=O C(CCNC(C1CCCCC1)=O)(C(=O)NC(C)CCSC)OC C1(C2CC2)(OC)CN(C(C)=O)C1.C12CC(C1CC(=O)O)N2 n1(CCC(N2CCC(c3cn(-c4ncc(C)s4)nn3)C2)=O)ncc2c1CCCC2 c1(C(N(C2CCN(C(C3C=CCCC3)=O)C2)CC)=O)ccc2c(=O)ccoc2c1 c1(C(=O)NC2CC(C(N3C(C#C)CCC3)=O)CC2O)c(C)cccc1C C1(CC(N2CCC(NC(c3c(CC)cco3)=O)CC2)=O)CC2(CCC2)CO1 c1(CN(C(C=CCCC)=O)C)cnn2c1CN(C(C1C3CCCC13)=O)CC2 CCN=c1ccc(C(=O)OCC(N2CCC(C)C2)=O)c[nH]1 C#Cc1ccc(OC)c(C(N2CCCC2CCNC(C2CC(F)(C)C2)=O)=O)c1 C1(C(C)C)CCC(C(N2CCC(C(C)NC(=O)CC3CCN(C)C3)CC2)=O)CC1 C1(C(=O)NCCCN(C)C(c2cnc(C(C)(C)C)[nH]2)=O)COCCN1C Nc1ccc(C(=O)NC2CCCC2NC(=O)CN2CCCS2(=O)=O)c(F)c1 CC(C)(C)CC(O)CC(=O)NCC(O)CNC(=O)CCc1cccs1 c1(CN(C(=O)COCN)C)cccc(CNC(=O)CO)c1 CN1CCC(CC(=O)NCCCCNC(=O)CC2(O)CCOC2)CC1 CCCCCS(=O)(=O)CC(=O)NCC(C)(CO)NC(c1scc2c1CCCC2)=O N1(C(C(C)NC(C)=O)=O)CCC(CC(N2CC(c3ncc[nH]3)C2)=O)C1 N1(C(C(=O)NCCNC(C)=O)=O)C2CCCC1CCC2.c1(C=O)ccccn1.N c1(CC(=O)NCC2CCCN2C(=O)Cn2cnnc2O)ccc2nsnc2c1 Cc1nc(C)n(CC(N2CC(NC(c3n[nH]cc3Cl)=O)C(CC(C)(C)C)C2)=O)n1 C(=O)(C(C)(C)CO)N1CC(CC(=O)NCC(=O)Nc2ccccc2)(OC)C1 CC1(C(N2CCC2c2cn(-c3ccc(Cl)cn3)nn2)=O)CCCCCC1 N1(C(C(C)(C)OCC)=O)CCC12CN(C(=O)CCCC(=O)OC)C2 O=C(CCS(=O)(=O)Cc1ccccc1)N(C(C1CCC(OC(F)F)C1)=O)C1CC1 C(=O)(C(O)CCCNC(=O)Cn1nccn1)NCC(c1ccncc1)C C1(NC(c2c(SCC)cccc2)=O)CC(C)CN(C(=O)Cc2ccccc2F)C1 c1(C=O)ccc(OC(F)(F)F)cc1.c1(C(=O)OC)cc(C=O)c[nH]1.C(C)C.N S(=O)(=O)(c1cc(C(F)(F)F)ccc1)NCC1(S(C)=O)CCC1.CC(C)C.N c1(OCCC)ccc(-c2cc(NC(C3CC(O)C3)=O)ccn2)cn1 C1(O)(C(=O)NCCNC(c2c(OCC=C)cccn2)=O)CC2CCC1C2 N1(C(C(CCC)NC(N)=O)=O)CC2CN(C(=O)CCc3cc(C)nn3C)CCC12 c1(NC2(CNC(C3CC3C3CCCC3)=O)COC2)ccnc2ncnn12 C1CN(C(C2(C=O)CC2)=O)CCC1(C)C.C(C(=O)N)N(C)CC.C(C)(C)C Cc1ccc(F)c(C(N2CC=CC2C(N2CCOC(=O)C2)=O)=O)c1F N1(c2scc(-c3ccc(CC)cc3)n2)CC2CCCC(O)C2C1 C(=O)(CC(C)CC(C)C)N1C(CNC(=O)C2=CCCC2C)CC(OC)C1 c1(NC(C2N(Cc3c(C)ccc(F)c3)C3CCC2C3)=O)nc(Br)c(Br)cc1Br CC(=O)CCCC(=O)N(C)CCN(C)C(C1CS(=O)(=O)CCO1)=O C1(C(=O)NCC(C(C)C)(C)O)CCCCN(C(c2cccc(O)n2)=O)C1 c1(C(C)C)ccc(NC(=O)C(C2(O)CCC2)NC(=O)C(C)n2ccnn2)cc1 C(=O)(C(C(C)C)n1cccc1)N1C(C2CCN(C(C=CC=CC)=O)C2)CCC1 N#CC1(C(=O)NCCN2CCN(C(C3(Br)CC3(F)F)=O)CC2)CCOC1 C1(C(=O)NCC(C)NC(C23CC(CO2)C3)=O)CCS1(=O)=O Cc1cc(C(N2CC3C(CNC(c4cc(Cl)cc(Cl)n4)=O)C3C2)=O)cc(C)c1 c1(C(=O)NC2CCC(=O)NCC2)cccn2nncc12 c1(C(=O)NCCCC(c2ccccc2)NC(C=CC)=O)cccc(N)c1F CC1=C(C(=O)NC2CC3CCC2(C(=O)N(C2CCCC2C)C)C3)CCO1 n1(CC)nc(C(C)C)cc1C(=O)NC1CCC1NC(c1cncs1)=O.C C=C(Br)CC(C)(C)C(=O)NCC1CN(C(C2CC(C)C2)=O)CCCO1 c1(C(C)C)ccc(C(N2CCC(C)(CNC(=O)CCN3CCC3)C2)=O)cn1 c1(C(N(c2ccsc2O)Cc2ccc(C3C(C)C3)o2)=O)ccc(N)cc1.C1CC1 C=CCCCCC(=O)NC1CN(C(c2cc(OC)ccc2C)=O)CC1C N1(C(C(C)OC(C)C)=O)CCc2cc(-c3ccc4occc4c3)ccc2C1 n1(CCOC)c(N2CCC(Nc3ccccc3)CC2)nnc1C(c1ccco1)C C(CC(F)F)(C(=O)NCC1(C)CC1(C)C)NC(c1n(C=C)nnc1)=O C(=O)C(C)CCC(C)(C)C.C1(CC=CC=O)CCC1.C(=O)(C)OC.CC Cc1c(Br)noc1C(=O)NC(C)CC1CCN(C(C2CC2C2CC2)=O)CC1 c1(NC(=O)NCCN2CCN(C)CC2)cnc(Cl)c(C(=O)O)c1 C1(C2CCS(=O)(=O)CC2)(C(=O)NC(c2cnn(C)c2)C(C)C)CCC1 C(=O)(CC(C)(C)C)NCC(=O)NC1CC(C)(NC(C(CSC)O)=O)C1 c1(OCC)ccc(C(N2CC3CC3(NC(C3CCC(C)O3)=O)C2)=O)cc1Cl.O C1(C(=O)NCCCOC(C)C)CN(C(=O)CC2(O)CCC2)CC12CCC2 C1(NC(C(C)=CC)=O)COC2CCOC12.c1(C(=O)N)cc(C2CCOCC2)no1 C1(C(=O)NC2CCN(c3c(CC)nc(=N)[nH]c3)C2)COc2c(F)cc(F)cc2C1 c1(NC(N2CCN(CC(=O)OC)CC2)=O)ccc2oc(N(C)C)nc2c1 C(=O)(CCC1=NNC(=O)CC1)NC1CCN(C(CCCOCCOC)=O)C(C)C1 C1(N(C(c2cnc(SC)s2)=O)C)CN(C(c2cc(C3CC3)no2)=O)CC1O c1(OCC(=O)NC(C)CN(C(=O)C(C)(C)c2cnsc2)C)cncc(Cl)n1 Cc1cccc(CC(=O)NC2CCC(F)(CNC(c3cc(C)no3)=O)C2)c1 Cc1cc(C(N2CC3CN(Cc4c(C(F)(F)F)cccc4F)C3C2)=O)ccc1Br c1(C(=O)NC(C(C)NC(c2n(COC)ncc2)=O)C)cccc(CCO)c1 Cc1ncc(Br)cc1C(N1CCCC1CNC(=O)C(F)C(C)C)=O C(=O)(C(C)CCCOC)NC(C1CCN(C(CC(=C=C)C)=O)C1)(C)C Cc1oc(Br)cc1C(N1CCCC1CN(C(=O)Cc1cc[nH]c(=N)c1)C)=O c1(C(=O)NC(CNC(c2cnc(CC(C)C)[nH]2)=O)C)cc2ncccc2o1 N1(C(c2nn(CC)c(O)c2)=O)CCCN(C(c2cc(N)ccn2)=O)CC1C(C)C C1(C(=O)NCC2(C)CCCN2C(c2ncccc2F)=O)CCC2(CCC2)CC1 C1(CC=O)CCN(C(=O)Cc2ccnc(O)c2)C1(C)C.Cc1nn(C)cc1C.N C1(C(=O)NC(C)CC(C)NC(=O)CC2CCC(=O)C2)CCC(C)(C)CC1 C1(C=C)(C(=O)NCCC(CCC#C)O)CCN(C(C2CN(C(C)=O)C2)=O)CC1 C(=O)(C(C)CCC(C)(C)C)N1CCC(C)(NC(c2c(OC)cc(Cl)cc2)=O)C1 CC(C)C(CNC(C1CC(=O)CS1)=O)C(=O)NCC1CCC2(CC1)CC2 n1(CC(N2CC3C(CNC(CN(C)CC)=O)C3C2)=O)ncc2cc(C)cnc12 N1(C(CC(C)OCC)=O)CCOC(C2CN(C(c3ccn(C)c3C)=O)C2)C1 C1(CNC(C2CC(OC(F)F)C2)=O)CN2CCC1CC2 C1(NC(C2CCN(CC)C2)=O)CN(C(=O)CSCC(N)=O)CC1(C)C C1(N(C)C(C2CC=CCC2)=O)CCCN(Cc2nnnn2C2CC2)CC1 c1(OC)ccc(C(=O)NC2CCC(CNC(=O)CC3CCSCC3)C2)cc1 Cc1cc(Cl)c(C(N2CC3CC3(NC(=O)CCCCN3CCCCC3)C2)=O)cn1 CC1CN(C(c2cnc(O)c(F)c2)=O)CCC1CNC(C1(C)CC1)=O CN1CCC(NC(c2cnc(S)nc2)=O)C12CCCN(C(=O)C(C)(C)C(N)=O)C2 N1(C(C2C(=C)C2)=O)CCN(C(C2CC(OC(F)(F)F)C2)=O)CC1CO C(=O)(C1=C(Cl)CCC1)NCC(C(=O)NC(C(=O)NC)C)CC1CCCC1 C#Cc1cccc(CC(=O)N(C2CCCN(C(=O)CC3COC4CC3C4)C2)C)c1 C1(C)(CC(=O)NC(C)CCN(C)C)CCN1C(=O)COCCF C1(CC#C)CNCCN1C(=O)NCc1ccccc1.C(=O)OCC c1(NC(=O)CC2CCCN(C(c3ccns3)=O)C2)cc(Cl)c(Cl)cc1I NC(=O)C(=O)NCC=CC(=O)NCCC(O)C1CCCC1 c1(C(=O)NCCC(=C)C)c(C#N)cnn1C.n1(CC=O)cnc([N+](=O)[O-])n1.N CC1(C)CC(C(=O)NCC2COC(C)C2)CO1.c1nccc(C(C)(C)C)n1.N c1(C(N(CC(C)C)C)=O)nn(C)c(C)c1Cl.Cc1c(C(=O)N)cnn1C1CCC1 C(=O)(C1CCCCc2ccccc21)N1C(CNC(c2cccc(N)n2)=O)CC1 c1(C(=O)NC2C(CNC(CCC(C)(C)F)=O)CCC2)ccc(S(N)(=O)=O)o1 c1(CC(N2CCCC(C)C2)=O)csc2cc(C)sc12.CC(C1CC1)=CC(=O)N.C CC(C)(CCF)C(=O)N1CCOC(CCNC(c2ccc(C3CC3)s2)=O)C1 Cc1nc(CC(C)C)sc1C(=O)NC1CCC1NC(=O)CCN1CCCC1 C1(CCC(=O)N(C2CCN(C(=O)C(C(C)O)N(C)C)CC2)CC)CCCCN1C c1(OC)c(F)ccc(C(=O)NCC(C)CN(C)C(C2CC2)=O)c1F.C1CC1 C1(CC(N2C(CNC(c3c(N)non3)=O)CC(O)C2)=O)SC2=NCCN2C1=O C1(O)(CNC(C(CC)Cc2ccccc2)=O)CCN(C(=O)C(=O)CC(C)C)CC1 CCN=c1[nH]cc(C(=O)NCCN(CC(C)O)C(c2ncsc2C)=O)s1 CC1(C)CC(NC(C2CCCC(F)(F)CC2)=O)CN(C(=O)C=CI)C1 c1(C(N(CCCNC(c2nccn2C)=O)C)=O)c(C2CC2)cccc1F N1(C(C2C(C)CC(=O)N2)=O)CCCC(C)(NC(C2CCCNS2(=O)=O)=O)C1 c1(C(=O)NC2CC(CNC(Cn3c(C)ccn3)=O)C2)ccc2[nH]nc(O)c2c1 Cc1ccc(C(=O)N(CC(c2nn[nH]n2)C)C)cc1S(=O)(=O)N1CCCCCC1 C(=O)(C(F)CC(C)(C)C)NCC(CCC)C(=O)N(C(C)C(=O)NC)CC c1(C(=O)OCC(N2CCN(c3ccc(CC)cc3)CC2)=O)ccc(Cl)cc1I C1(C(N2CCC(CC(=O)NC)C2)=O)CN(C(c2cncc(O)c2)=O)CCN1C N1(C(c2cccn3nncc23)=O)CCC2(CCCN2C(=O)Cc2nnc(O)s2)C1 CC1(C)CCCN(C(=O)CCS(C)(=O)=O)C1C(=O)NCC1CCC2(CC2)C1 C1(C(=O)NCc2ccccc2C)CCN(C(C2(OC(C)=O)CCC2)=O)CC1 C(=O)(C1CCNc2cc(F)ccc21)NC(C)CCNC(c1cc(O)cc(O)n1)=O c1(NC(=O)NC(c2csc(C(C)C)n2)C)ccc(S(C)(=O)=O)cc1 N1(C(CCCC(N)=O)=O)CCC2CCCC(C1)N2C(C1CC1Br)=O C1(C(N2CCC(N(C)CC)C2)=O)CNC(=O)CN1C(c1ccc(NC)cc1)=O C1(C)CCN(C(C2CCCN2C(N)=O)=O)CC1.CC1CC(C)OC1C(=O)NC Cc1c(C(N2CCCC(CNC(=O)CC3CCC3(F)F)C2)=O)nn2ccccc12 CC1CC(c2ccccc2)CCN1C(c1cnc(-n2cccn2)cn1)=O Cc1ncc(Cl)c(C(=O)NC2CCN(C(=O)C(O)CN3CCCC3)C2C)n1 c1(C=O)ccnc(S(N)(=O)=O)c1.CC1(C)CC(CC(=O)NC(C)CO)CCO1.N c1(C(N2CC(C3(Nc4c(F)cnc(C)n4)CC3)C2)=O)cccc2nc(O)ccc12 Cc1cc(Cl)cc(Br)c1NC(=O)COc1ccc(Cl)c(Cl)c1 C1(CC)CN(Cc2ccc(OC(F)(F)F)c(F)c2)CCN1C(=O)C(O)C(C)C O=S(=O)(c1cccc2ccsc12)N1CC(O)C(F)C1 C1(N(C(=O)CC(C)C)CC)CCCN(C(C23CC(C2)C3)=O)C1.C(C)(=O)O CP(C)(=O)CN1CCC(C(=O)NCCCn2cc(C3(F)COC3)nn2)CC1 N1(C(C2CC3N(C(C4CC4[N+](=O)[O-])=O)C(CC3)C2)=O)CCC(F)(F)C(O)C1 C#Cc1c[nH]nc1C(=O)NC1(C(=O)NCCC(C)(O)CC)CCN(C)C1 c1(N2CC3CCC(N(C)C)CC3C2)nc(Cl)nc2c1CS(=O)(=O)C2 Cc1coc(C(=O)NC2CC(N(C)C(c3cnc(NC4CC4)s3)=O)C2)c1 Cc1cc(C(N2CC(F)(CNC(=O)C(c3ccnn3C)C)C2)=O)sn1 N1(C(CC(C)C)=O)CCOCC1C(=O)NCC1CC1c1ccccc1Cl Cc1cc(O)c(Cl)cc1C(N1CC(NC(=O)C(C)(C)F)C1)=O N1(C(c2cc(SC)oc2C)=O)CC(NC(=O)CCc2ccc(O)cc2)CC1(C)C N1(C(c2nccc(CNC(C3CCC(OC)C3)=O)c2)=O)CCN(C)C2(CC2)C1 CC12CCCC(C(N3CCN(c4nc5cncnc5[nH]4)CC3)=O)(CO1)C2 N1(C(Cc2nc(C)[nH]n2)=O)CCC2CCCC12CNC(=O)CCNC(=O)OC n1(CC)nc(C(N2CC(CCCCNC(c3ncccc3C)=O)C2)=O)c(Br)n1 Cc1ccc([N+](=O)[O-])c(C(=O)NC(C)CCNC(=O)C2=CCCS2)c1C c1(C(=O)NC2(CC=C)CCN(C(=O)C(F)OC)C2)cnc2ccc(C)cc2c1 C12(NC(COCCOC)=O)CCC(CN(C(C3CN(C)CC(C)O3)=O)C1)C2 C1(C(N2CCC(N(C(C(C)OCOC)=O)CCO)C2)=O)CCc2nn[nH]c2C1 CC(CC(=O)NC(CC(F)F)C(=O)NC1C(O)C2CCOC12)C(F)(F)F C(=O)C(C)(O)CCN(C)C.c1(C=O)c[nH]nc1CC.C(C)(C1CC1)SC.N C1(C(N2C(C)C(NC(=O)CC3(C)CCOC3)CC2)=O)CCCCCN1C C(CCCCCNC(c1nn(-c2ccccc2)cc1C)=O)NC(CNC(C)=O)=O C(CCCC(=O)NCC1CC1CC(=O)NCC1(CCCO)CC1)OCC C(C(=O)NC1CCCCC1CC(=O)NCc1ccccc1)(C(C)C)SC Cc1c(C(=O)NC23COC(C2)C(NC(C2SCCCS2)=O)C3)c[nH]c1C#N Cc1ccc(F)cc1NC(C1CC12CCN(C(=O)Cc1ccc(Br)cc1I)C2)=O c1(OCC(N2CC(NC(c3n(C)cc(Cl)c3)=O)C(O)C2)=O)ccccc1C#N C(=O)(CCCCC(F)(F)F)NC1CCC(NC(CCCOC(C)C)=O)CC1 CC1(C)CN(C(=O)CNC(=O)C2CC2)CCO1.C1(C=O)CC(F)(F)CS1.C Cc1ccc(C(=O)N(C2CC(NC(c3cc(SC(F)(F)F)c[nH]3)=O)C2)C)nn1 CC(C)(C)C(O)C(=O)N1CCSC(C(=O)Nc2cc(O)nc(Cl)c2)C1 c1(C(=O)NCCCC(C)NC(=O)C2=CCCS2)cc(Cl)c2c(c1)OCCCO2 C1(C(N2CCN(CCNC(C(CC)F)=O)CC2)=O)CCC2(CCC2)OC1 C(=O)(C(C)(C)C(=O)NCCOC1CCN(C(C2C3CCCC23)=O)CC1)NC c1(OC)ccc(CNC2(c3nnnn3C3COC3)CC(SC)C2)cc1Cl Cc1cc(N)ccc1C(=O)NC1C2CN(C(=O)Cc3ccsn3)CC12 Cc1ccc2c(n1)OCCN(c1nc(=N)[nH]c(=NC(C)c3ccc(Br)o3)[nH]1)C2 C=CC(CCC)CC(=O)N1CCCCC1CNC(=O)CC1(OC)CCCC1 Cc1cccc(Br)c1C(C(N1CCC(C)(F)C1)=O)NC(C1CC12CCCCC2)=O CC1CCCC(C(=O)N(c2cccnc2)C)N1 N1(C(C2CC=C(C)CC2)=O)CCN(C(c2nc(C)ncc2Cl)=O)CC12CC2 CC(C)(CCCC(=O)NCC1CCC=CCCC1)NC(=O)C=Cc1ccco1 CC1CN(C(C2CC3(CCC3=O)C2)=O)C(C)CN1C(C1CCCN1C1CC1)=O c1(CC)oncc1C(=O)NCC1CC(O)(CNC(c2cncs2)=O)C1 C1(OCC)CCC(C(=O)NC2CC(C)N(C(c3ccco3)=O)C2)CC1 C1(OCC(=O)NCc2cn[nH]c2)CCN(C(c2cn(C3CC3)cn2)=O)C1 C(N=c1cc[nH]c2cnccc12)c1cc(C(=O)OCC)sc1C Cc1cnc(F)c(NC(=O)NCCC2CC2C2CC2)c1 c1(C(N2C3CCC2CC3)=O)[nH]c2cc(F)ccc2c1C.C(CC)(C(=O)N)=CC.C c1(C(=O)N)[nH]ccc1.N1(C=O)CC(C(=O)NCC=CC)C1.CCO C=CC1(O)CCN(C(=O)CC2(NC(c3cnc(OC)s3)=O)CC2)C1 N1(C(c2ccc(OCC)c(O)c2)=O)CCC2(CC1)CN(C(=O)C=C(C)Cl)C2 C1c2ccccc2N=C(O)N1CC(=O)NCC(CO)NC(C1(CF)CCC1)=O N1(C(C(C)OCCCC)=O)CC2(CC(CNC(c3[nH]nnc3C)=O)C2)C1 N1(C(C(COC)NC(C)=O)=O)CCCC(C(=O)NC(c2cccnc2)C)C1 c1(C(N(C(C)CNC(C2CC2(C)C)=O)CC)=O)cccn2c(C)nnc12 CCCCC(C)C.C1(CC=O)C(C)(C)C1(C)C.CC(C=O)OCCN(C)C.N N1(C(CN(C(COC)=O)C)=O)CCN(C(C2(CN(C)C)CCCC2)=O)CC1C Cc1cc(Br)cc(NC(N2CCCC(C(=O)Nc3nccs3)C2)=O)c1Cl C1(NC(CSCCNC(C2C(C(N)=O)COC2)=O)=O)CCOCC1F c1(OCC)cccc(C(C2CCCCN2C(C)=O)O)c1.N12CC(C1)C2 C1(C(N2C(CC)CN(C)C(=O)C2)=O)CCCN1NC(=O)C1CCCSC1C c1(NC(COCC)C)nc(N2CCS(=O)(=O)CC2)nc2c(C)nn(C)c12 C(=O)(CCCCCCS(N)(=O)=O)NC(C)CNC(C1CCN(C)C1=O)=O C(CCCCC(=O)Nc1ccc(Cl)cc1)NC(C1(C)CCN(C)C1)=O c1(OC)cnccc1C(=O)NC1CCOCC1NC(C1CC1c1nccn1C)=O O=C(C1=CCc2ccccc21)NCCC1CN(C(=O)C=CCO)CCO1 CCCC(CCCNC(c1occ2c1CCC2)=O)NC(=O)C(O)CC Cc1nnc(NC2CCCN(C3CCC=CCCC3)C2)nc1C c1(C(C)C)cccc(F)c1C(N1CCCC(N(C)C(C2CCC2)=O)C1)=O c1(OCC)nccc(C(N2CC(CNC(=O)C(O)CS)CC2(C)C)=O)c1F c1(C(N(CCCCNC(c2c(CC)csc2)=O)C)=O)csc(N=S(C)(C)=O)n1 C1(CC=C)(NC(=O)COC2CCC2)CCN(C(c2ncccc2Cl)=O)CC1 C1(C(C)NC(c2cc(OC)no2)=O)CCN(C(=O)C(C#N)=CC2CC2)CC1 c1(C(N(CCNC(Cc2c(C)noc2C)=O)C2CC2)=O)csc2cccnc12 c1(C(=O)NC2C(NC(COCC)=O)C2)c(-n2cccc2)sc2c1CCSC2 C1(N(C(=O)CSc2nnnn2C)C)CCCCN(C(C2CC(C)(O)C2)=O)C1 C1(CC)(CC)CC(C(=O)NCc2c[nH]nc2C(=O)Nc2cnsc2)C1 Cc1cc(S(C)(=O)=O)ccc1NC(c1ccccc1F)=O.C1(C=O)CC1(F)F.N N1(C(C2(CC(C)C)CC2)=O)CC(F)(CNC(=O)C(F)(F)c2cscn2)C1 Cc1cn2c(=O)c(C(N3CCC(C)C(NC(c4ccc(Cl)[nH]4)=O)C3)=O)cnc2s1 c1(C=O)cc(F)cc(S(N)(=O)=O)c1.N1(C(C(CC)NC(C)=O)=O)CC=CCC1 CCCC(CCC)Nc1cccc(CN2CCOCC2)c1 CCCC(C)(C)CC(=O)N1CCCC(CC)(NC(c2ncsc2C)=O)C1 C12(C(=O)NCC3CCN(c4nc(C)nc(=N)[nH]4)C3)CCC(C(F)F)(CC1)CC2 C1(NC(c2c(C)oc(C(C)C)c2)=O)CN(C(C2(C(N)=O)CC2)=O)CCC1O c1(-c2cn(CC(CCNC(C(CCC)F)=O)(F)F)nn2)cc(Cl)ccc1Cl N1(C(=O)NC(C)(C)Cn2cccn2)CCC(CN)(CO)CC1 c1(CC)cc(C(=O)NCc2ccc(C(=O)N(C(C)C(=O)O)C)cn2)ccn1 C(c1ccccc1)=CC=O.c1(COC)nn[nH]c1C(=O)N(CCC)C(C)C C1(C(=O)NC2CN(CC)C2)CC(C)N1C(c1cnnn1CC)=O C1(NC(=O)CCCCBr)CCCN(C(c2ccc(C(F)(F)F)[nH]2)=O)CC1 C1(O)(CCNC(C=CSC)=O)CCCN(C(=O)C(F)C(C)(C)O)C1 c1(OC(C)=O)ccc(-c2ccc(NC(=O)COc3ccc(F)cc3)s2)cc1 c1(C(C(=O)NC(C)CN(C(=O)C(C)c2cncs2)C)=O)ccc(F)cc1 N1(C(C(C)N2CCC2)=O)CCC(NC(c2coc(CN(C)C)n2)=O)C1 C1(CCC)CN(C(=O)C(C)SCC)CCN1C(c1ccc(-n2cnnn2)cc1)=O C(=O)(C1=C(C)OCCS1)N(C1CCCN(C(C(CC)(F)F)=O)C1)CCF C1(NC(C(C)C)=O)CC2CCC(C1)N2C(=O)CC1CC12CC2 C1(C(=O)NC2CC(=C)C2)CN(C(=O)C=CC2(C)COC2)CC1(F)F N1(C(c2cc(OCC)n[nH]2)=O)CC2CCC(C1)N2C(=O)C(n1nc(C)cc1C)C c1(CC)nscc1CNC(C12CC(C=O)(C1)C2)=O.C1(C(N)=O)CC1 C(CO)CC(C)(C)C.n1(CC)ncc(C)c1C(=O)NCC1CC(C=O)C1.N Cc1cc(C(=O)NCCCN(C(=O)CCn2ccnn2)C)n2ncc(Br)c2n1 CC(C)C(C)C(C)CC(=O)N1CCOC(CNC(C2(C(N)=O)CCC2)=O)C1 N1(C(=O)COc2ccccc2)CC2CCCCC2(CNC(c2ccco2)=O)C1 C=CCC(CC)C(=O)NCC1COCCN(C(c2c[nH]nc2CC)=O)C1 c1(NCC(CC)(C)CC)ccc(S(=O)(=O)N2CCOC(C(=O)NC)C2)cc1C#N C1(OCC)CN(C(C2(CC)CCCCC2)=O)CC1C.C(=O)(C)N.C(N)=O c1(C(N2CC=CCC2)=O)cn2c(n1)SCC2.C(=O)(CCC(=O)N)NCCCOC C1(C(=O)NC(C)C(CO)NC(c2ccc(=O)n(C)n2)=O)CC2CCCN2C(=O)N1 N1(C(CCOCCCOC)=O)CCC(C2CC2NC(c2ccc[n+]([O-])c2)=O)CC1 C1(NC(c2cn(CC=C)nc2)=O)CCN(C(c2ccc(NC)cc2Cl)=O)C1(C)C C(=O)(CCCS(N)(=O)=O)NC1C2(CN(C(C(C)(C)c3cccs3)=O)C2)CC1 C(CC(C(C)C)NC(c1nnnn1-c1ccccc1)CCC1(C)CC1)OC(C)C c1(C(N2CCCCC2c2ncc[nH]2)=O)cc2cc(F)ccc2s1 c1(C(=O)NCC(c2ccccc2)N(C(C2C(C)C2C)=O)C)cccc2cncn12 Cc1ccc(C=CC(=O)NCC2C(C)CCN2C(=O)CCCN(C)C)cc1Cl CCCC(C)(O)CNC(c1c[nH]nc1CNC(=O)C(C)CC1CC1)=O C1(C(N2CCCC2)=O)CCCC2(CC2)C1.C12(C(=O)N)CC(C(F)F)(CO1)C2 C(=O)(C(C)(C)C(=O)NC)N1CC2C(CN(C(C3CCN(CC)C3)=O)C)C2C1 N(C(=NCCc1ccc(Cl)cc1Cl)NC1CCC(C(=O)OC)C1)CC(=C)C C1(NC(C(CCNC(C(CC)NC(N)=O)=O)O)=O)CCN(C)CC1C#N c1(C(C)CC(=O)NC2CC(CNC(=O)CCC3CC3(C)C)C2)ccc(F)cc1 C(=O)(C1=C(CC)OCCC1)NCC(=C)CCNC(C1CCC(=O)N(C)C1)=O C#Cc1ccc(C(=O)NC(C)C(C)C(=O)N2CC(F)(C#N)C2)c(C)c1 N1(C(CCCCCC)=O)CC2(C=C(C(=O)NC(CO)CC(C)C)CO2)C1 N1(C(CSCCNC(Cc2c(C)nn(C)c2)=O)=O)CCOCC(F)(F)C1 N1(C(C(C)NC(=O)OC)=O)CC=CC(NC(C2CCOC(C(C)C)C2)=O)C1 O=C1CCCC(C(=O)NC2CCCCC2CNC(c2cccc(F)c2)=O)C1 O=C(N=c1[nH]n(-c2ccccc2)c2c1CCC2)c1ccc(NC(=O)C2CC2)cc1 Cc1ccc(C=CC(N2CCC(C)(C)C2)=O)cn1.c1(C=O)cc[nH]c1C1CC1.N c1(C(C)NC(C(CC)C#N)=O)cc(F)cc(Cl)c1.c1(CCC(=O)N)ccn(C)n1 c1(C(CCC)C)nc(-c2ccncc2)n(C(C)C2CC2)n1 N1(C(C(C)NC(C=CCC(C)(C)NC(C)=O)=O)=O)CCOCC1CO C12(NC(c3c(C)oc(Cl)n3)=O)CCCC1N(C(=O)Cn1ccnn1)CCC2 N1(C(C2(COC)CC(=O)C2)=O)CC(C(=O)NC(C2CSC2)C)C(C)C1 N1(C(c2c(C)n[nH]c2)=O)CC(NC(C2(F)CCCOC2)=O)CC12CCCCC2 CCC(C(=O)NC(C1(C(=O)NCC(C)(CC)CO)CC1)C)C(C)(C)CC C1(NC(CCc2ccc(C)nc2)=O)C2CCN(C(C3CCCCC34CC4)=O)CC12 CC1c2cc(O)ccc2CCN1C(=O)Cc1cc(C2CC2)on1 N1(C(C(CCSC)N(C)C)=O)CCCC(C)(NC(c2cnn(CCF)c2)=O)C1 Cc1noc(C)c1C(=O)NC(C1CN(C(=O)Cc2ccc(CO)cc2)CCO1)C N1(C(Cc2cnc(C)s2)=O)CCOC(C(C)NC(=O)C(N2CCN(C)CC2)C)C1 Cc1ccc(-n2cc(CCCCNC(=O)C(=O)CC3CCCO3)nn2)cc1Cl C12(C(=O)NC3C(CNC(C(N4CCCCCC4)C)=O)CCC3)COCC(C1)C2 C12(C(=O)NCCCCC)CCN(CC1)S(=O)(=O)C2.c1(C(=O)N)cncc(F)c1 C(CCN=C(NCc1cnccc1Cl)N1CCc2c(Br)cccc2C1)OC N1(C(CSC(C)C)=O)CCN(C(C2C3CC4C(C3=O)C24)=O)C(c2cccnc2)C1 CCCC(CC(C)C)C(=O)N1CC(NC(c2oc(CO)cc2C)=O)C(SC)C1 Cn1cncc1C(=O)NCC(C)(CO)NC(C1CCOC1)=O c1(OCC)ncccc1C(N1CCC(C)(C(=O)N)C1)=O.N1(C(C)=O)CCOCC1 N1(C(C(=Cc2ccncc2)C)=O)CCC(O)C(NC(C2CC(C)=NO2)=O)C1 CN1CC2CCCC(C1)N2C(C12CC1CCN2C(=O)C(O)CN1CCCC1)=O c1(C(=O)NC(C)CNC(c2ccccc2OC(F)F)=O)cccc2nccn12 c1(N(C(=O)C(Cc2ccncc2)NC(C2CC2N)=O)C(C)C)nc2sccc2s1 CC1(C)CCCN(C(=O)CNS(C)(=O)=O)C1C(=O)NCCC1CC1 c1(C(N2CCN(C(C34CC(C)(C3)C4)=O)C(CO)C2)=O)ccc2c(n1)NCCO2 c1(OCC(C)C)ccc(C(=O)NC(c2ccnn2C)C(=O)N)cc1.C(C)(C)C c1(CC(=O)N(CC(CC)NC(=O)C(C)(C)N(C)C)CC)cccc2c1OCO2 c1(C(N2CCC3CN(C(C4CCC(C)(C)C4)=O)CC32)=O)ccc2c(c1)COCC2 c1(C(C)C)conc1C(=O)NCC1CC1CC(N1CCCC1C(O)CO)=O N1(C(c2cn(CCC(C)C)nn2)=O)CCN(C(C2(CO)CCCCC2)=O)CC1 CCC(CC)(CC)C(=O)N1CC(NC(=O)CC(O)CC(C)C)C1 C1(C(N(C(C2CCC2)C)CC)=O)CCN(C(C2CNC(=O)N2)=O)CCO1 c1(CC(C)C)ccc(C(=O)NCCNC(C(C)CF)=O)cn1 Cc1nc(C(=O)NCCCCCN(C)C(C2COC(C)C2)=O)c2ccccn12 C(c1cccc(F)c1F)=CC(N1CC(NC(CCCC#C)=O)C(O)CC1)=O N1(C(C(CCOC)C)=O)CCCC2CN(C(=O)CN3CCOCC3)CC12 c1(CC(N2CC=C(C)CC2)=O)cccnc1C.C(C(=O)OCCOCC)=CC N1(Cc2ccc(C#C)s2)CCC2(CCCC2C(N2CCC(CCCO)CC2)=O)C1 c1(OC)cc([N+](=O)[O-])ccc1S(=O)(=O)N1C2CN(C(c3ncc(C)s3)=O)CC12 C(=O)(C1CCCc2cccnc21)NCC1CC(C)(C)N(C(=O)CCC(N)=O)C1 C1(C#N)(CNC)C(C#N)C1(C)C.c1(CC=O)csc(C2CC2)n1.C1CC1 n1(CC(N2CCN(C(=O)CC3(O)CC3)CC2)=O)ccc(O)nc1=O CC1(C)CC(NC(=O)CC=C(Cl)Cl)CCN(C(C2Cc3cccnc3C2)=O)C1 C1(CC)CN(C(=O)C2=CCCCO2)CCN1C(=O)Cc1cc(OC)n(C)n1 N1(C(CC(C)SC)=O)CCCC(F)(C)C1.c1(C(=O)N)[nH]c(C)c(C(C)=O)c1C C(C1CCCN1C(=O)C(C1CCOCC1)F)=CC(NOCC(=O)OC)=O C=CCCCCCC(=O)N1CCN(C)CC1C(=O)NC1C2CCC1CC2 c1(CNC2C(C(=O)Nc3ccc(C)nc3F)C2)ccc(F)c(C)c1Cl C1(C(N(C)CC2CCN(C(=O)C(F)n3ccnc3)CC2)=O)CN2CCN1CC2 N1(C(CC2CCC(C)C2)=O)CC2(C1)CN(C(=O)CO)CCO2 n1(CC=C)cc(C(=O)NC(C)(C)C)nn1.n1(CC=O)cc(Cl)cn1.CCC c1(CC)c(C(=O)NCC#CCNC(=O)C(c2cscc2Br)=O)cccc1F N1(C(CCC)=O)CC2CC(NC(c3csc(C4CC4)n3)=O)C2C1 CC(C)CC(C(=O)N1CCCC(C(C)NC(=O)C(C)(C)O)C1)C(C)C C12CCC(CC1)N(C(=O)CC1CC1C(F)(F)F)C2.CC(C(=O)N)c1ccco1 c1(C(=O)NCC2CCN(C(c3ccc(C(C)=O)o3)=O)C2)cnn2c1CCCC2C C(C(C)(O)CCN=C(NCCN1CCC(C)CC1)NC(c1cccs1)C)OC CC1CC2(CCN(C(=O)C=CC(F)F)CC2)CN1C(=O)C(=O)NCC(F)F N1(C(c2cnc(Br)o2)=O)CCOc2nccc(Cl)c2C1 CCC(C(=O)N1CCCN(C(c2[nH]c(C)cc2C)=O)C(CO)C1)C(C)(F)F CCC(C)C(C(=O)NC1CC2CCC1N2C(=O)CSC(C)C)OC Cc1cccc(NC(C2CC(NC(C3(CO)CCCO3)=O)C2)=O)c1C C12(C(=O)NC3CCN(C(c4ccc(CC(N)=O)cc4)=O)C3)CC1CCC2(F)F C(=O)(NNc1ccc(F)c(F)c1)NC(CCCCC(=O)OC)C(F)(F)F Cc1c(NC(C2CCCN(C(c3ccccc3)C)C2)=O)cnn1CC(C)C C1(NC2C(C)N(C(=O)OC(C)(C)C)CC2)C2(C)CCC(C2)C1(C)C C1(CN(C)C(c2scnc2Cl)=O)CN(C(C2CCC(=O)NC2)=O)CCO1 C(=O)(C1CCc2ccccc21)NC(CNC(c1c(C)c(Br)cnc1)=O)CO C1(CC(N2CCOC(F)(F)C2)=O)CC(F)(F)CN1C(=O)OCc1ccccc1 C1(CC=O)CN(C(=O)CN2CC=CC2)CCN1C(=O)C=CC.[nH]1cncn1 c1cccc(F)c1.N(S(N)(=O)=O)CC(=O)NCCN(C(=O)CC)C(C)C c1(-c2ccc(-c3n(CC4C(C)(C)C4)ccn3)cn2)ccccc1[N+](=O)[O-] N1(C(c2ccnc(C)n2)=O)CC(NC(c2cccc(Br)c2)=O)C2(CCC2)C1 N1(C(c2cc(C)c(C)s2)=O)CC2CC(N(C)C(c3cnn(CCF)c3)=O)C1C2 C#CC1CCCN1C(=O)C(=O)NCC1(c2ccc(C(=O)NC)cc2)CC1 C(=O)(C(CC(C)C)n1nnnc1C(C)(COC)Nc1cc(F)ccc1C)OC CCCCCC(=O)NCCCNC(c1c(-c2ccccc2)nnn1C)=O c1(C(=O)NC2CC(NC(CC3(OC)CCCC3)=O)CC2O)cnc2n1CCC2 Cc1cncc(CC(=O)NCCN(C(=O)CC2CCC(C)C2)C)c1 N1(C(C=CS(C)=O)=O)CCOCC(NC(=O)C(F)=C2CCC2)C1 c1(-c2scc(CC(=O)NC(C3CCN(C(C=NOC)=O)C3)C)n2)ccc(C)cc1 C(=O)(CC(F)(F)C(C)(F)F)NCCCNC(c1ccc(C(C)C)c(F)c1)=O C(=O)(C1=CS(=O)(=O)CCC1)NCC(CC(C)C)Cc1ccccc1 C1(C(N2C(CNC(Cc3cn(CC)nc3)=O)CC2)=O)CCCC12CC2 C(CCCCCNC(=O)C(C)CSC(F)(F)F)NC(C(c1cncnc1)C)=O c1(-c2nc(CCCC)nn2C(C2CCCCC2)C)ccc(C)cc1-n1cnnn1 C(=O)(CC(=O)N(C(C(=O)NC1CC(CC(=O)OC)C1)C1CC1)C)NCC C=CCC(CC(C)C)C(=O)NCC12CC1CN(C(c1cccc(C)c1Cl)=O)C2 c1(CC(=O)NC2CN(Cc3nccc(OC)c3)C2)noc2ccccc12 c1(COC)ccccc1CNC(=O)Cn1cc(C2CCCOC2)nn1 C1(CNC(c2cc(Br)no2)=O)CN(C(=O)C=CCF)CCC12CCOC2 C=C=CC(C)C(=O)N1CCOC(CC(N2CCC(CC(=O)NC)C2)=O)C1 C(=O)(CCCCCF)N(CC(C)(C)CNC(c1cc(C(N)=O)cs1)=O)C C(=O)(CC1CCc2ccccc21)NC(CNC(c1c(C(C)C)ncs1)=O)CO C(C)(CO)(C(=O)NCC1CCN(C(=O)CN2CCC(C)(C)C2)C1)OC C1(C(N2CCN(C(=O)Cc3cccc(F)c3Cl)CC2)=O)OCC2CCCCC12 C1(C(=O)NCCC2N(C(c3c(N)non3)=O)CCCC2)CC2CCCCN2C1 c1(CC(=O)N(c2cccc(C(=O)OCC)c2)C)c[nH]c2ccc(O)cc12 N1(C(C2(C)CCC(OC)CC2)=O)CCC(NC(c2cc(F)n[nH]2)=O)C2(CCC2)C1 c1(OC)ccc(C)cc1C(=O)NC1CC2CC(NC(=O)Cc3cscn3)CC12 c1(C(=O)NCCC2OCCCN(C(C3C(C)C3)=O)C2)cc2c(nc1O)CCSC2 C(=O)(C(F)CC(C)(C)C)N(C1CCCC(NC(=O)CN2C(=O)CCC2=O)C1)C C(=O)(CCCc1cnccn1)N(CC(C)NC(=O)CC1CC1)C.C1CCCC1.S N1(C(CCC2CCN(C(c3c(C)nncc3)=O)C2)=O)CCC(CO)C1(C)C C#Cc1c[nH]nc1C(=O)N(CC(CC)NC(c1cc(C)ccn1)=O)C C(=O)(C1=NOC2(CCC2)C1)NCC12CCN(C(C3(C)COC3)=O)C1CCC2 c1(CC)cn2c(n1)CC(C(=O)N(CCC)C)CC2.C(=O)(C(C)CC)N(CC)C.O N1(C(CSCC=C)=O)CCCCCC(NC(=O)C(C)N(C)C(C)=O)C1 N1(C(CCSCCCC)=O)CCN(C)CC1CNC(=O)C(C)N1CCC1 O=S(=O)(c1ccccc1)Nc1ccc(C2(SCCCCC3CNC3)N=N2)cc1 CCCCCC(O)C(=O)NC(C1(CNC(c2noc3c2CCCC3)=O)CC1)C C(=O)(CN1C(=O)Cc2ccccc21)NCCCOCCCNC(CC(C)C)=O Cc1c(C(=O)NC2CCC(C)N(C(=O)CSC3CC3)C2)sc2ccccc12 c1(-n2c(CCCSC)nc(COC(C)(C)C)n2)ccc2ccsc2c1 N1(C(C2(CC)COC2)=O)CCC(NC(c2ccccc2)=O)C(F)C1.C1CCC1.O C1(CCC)(NC(=O)Cc2ccco2)CCN(C(=O)CCC2CCCCN2C)CC1 CC1Oc2ccc(C(N3CC(C4(NC(=O)CCCCCF)CC4)C3)=O)cc2C1C C(c1cnc2ccccc2n1)=CC=O.CC1(C)C=C(C(=O)NC23CC(C2)C3)C1 c1(C(N2CCC(N(CCC)C(C3(Cl)CC3(C)C)=O)C2)=O)ccn(CCO)n1.C C#CCCCCCC(=O)NCC1(F)CCN(C(c2cc[nH]c2CCC)=O)C1 CCC(C)CCCCC(=O)NC1(CCOC)CCN(c2nnc(C)s2)C1 Cc1ccc(C(C)NCC2NC(=O)CC2(C)C)cc1C#N N1(C(c2cc(C(C)C)on2)C(=O)Nc2ccccc2)CC2C(C1)C2(C)C Cc1cc(N)c(C(=O)NCC(CC(C)C)NC(c2sccc2F)=O)c(F)c1 C(=O)(C(C)(C)C(=O)OC)NCC=CCNC(C(C)OCOC)=O C(=O)(CCC(=O)N(CC(C)NC(c1ccc(-c2ccsc2)cc1)=O)C)NC c1(C(=O)NC2CCN(C(c3cnn(C)n3)=O)C2)cc2n(n1)CCCC2 c1(C(=O)NC2(C)CCN(C(c3cc(Cl)ccc3Cl)=O)C2)ccc(O)c(N)n1 CC1CN(C(c2occ3c2CCOC3)=O)CC(C)C1(O)c1ccccc1 S(=O)(=O)(c1cnc(NCC2(C)CC(C)C2)c(Cl)c1)NC1(CCC)CCOC1 CC1CCCN(C(=O)CCOCCNC(c2ncccn2)=O)C1C n1(CCOCC=C)c(N2CCC(OCC=C)C2)nnc1-c1nccs1 Cc1cnc(C(N2CCCC2(C)CNC(=O)C(C)(O)c2ccccn2)=O)c(C)c1 C(CCC(C)(C)C(=O)NC(c1cccnc1)CO)NC(CCC(C)CN(C)C)=O N1(C(CC(C)C2CCCCC2)=O)CCC2CCC(NC(c3cnc(Cl)[nH]3)=O)C1C2 c1(C(C(=O)NCCSC)N(C)CC2CN(C)CCO2)cccc(Br)c1F N1(C(c2nc(C)sc2)=O)CC2CCN(C(c3ccc4c(c3)OCC4)=O)CC12 c1(C(N2CCC(C)(CCNC(C3(C)C(C)(C)C3)=O)C2)=O)ccc(O)cc1Cl c1(OC)ccc(C=NOCC(=O)NC2CC(C(C)NC(=O)C(C)CO)C2)cc1 C1(CNC2(OC)CC(C(F)F)C2)CCCCCC1C(C)C Cc1c(C(N2CCC(C)C(CNC(C3(C#N)CCC3)=O)C2)=O)c[nH]c2nccc1-2 C=C=CC(C)C(=O)N1CCC(C(=O)NCC(C)C(=O)NC)C1CC S(=O)(=O)(c1ccc2c(c1)CCC2)N(C(CC1(C)CCNC1)=O)CCO c1(C(N(C2C3CN(C(c4c(CCC)[nH]cc4)=O)CC32)C)=O)cc(C)nc(C)n1 C1(NC(CCC(=O)OC(C)(C)C)=O)CC2(CCCCN2C(C2(Cl)CC2)=O)C1 c1(C(N2CC(OC)C2)=O)ccc2c(c1)COCC2.C(=O)C(C)(C)CC1CC1.C CCCCC(O)CNC(C1(COC)C=CCN1C(C1CCOCC1)=O)=O CCCCCCC(CC)C(=O)NC(CNC(c1cn(C)nn1)=O)C1CC1 CCC(C(c1nnnn1C)Nc1ccc(-c2nnc(C(C)C)o2)nc1)C(C)C CC1CC(NC(c2ccc(CCC(N)=O)cc2)=O)CN1C(c1cnc(S)[nH]1)=O Cc1cc(F)ccc1C(=O)NCC1CC(O)CN1C(=O)C(CO)c1ccccc1 CCC(C)C(O)C(C)C(=O)N1C2CCC(C(=O)NC3CNC(=O)C3(C)C)C1CC2 N1(C(C2=C(C)OCC2)=O)C2CCCC1CN(C(c1cnc3n1CCCC3)=O)C2 N1(C(C(C)OCCOC)=O)CCOC(CNC(=O)C=CCO)C1 Cc1nc(C(=O)NCC(C)CCc2ccccc2)c2ccnc-2[nH]1 Cc1nc2c(o1)CCN(C(C1CC(C)(C)CCN1C(=O)CC1CC(F)C1)=O)C2 Cc1cn2c(C(N3CCC(F)(CNC(c4cnnn4C)=O)CC3)=O)c(C)nc2s1 N1(C(Cc2ccn(C)n2)=O)CC(C(=O)NCC2CC3CCC3C2)C(O)C1 Cc1cc(CCC(=O)NCC(F)CNC(=O)CC2COC(C)(C)C2)cc(C)c1 CC1CC(NC(=O)CCc2cn[nH]c2)CN(C(=O)CCC2CC2(Cl)Cl)C1 c1(-c2cc(C(=O)NCc3n[nH]cc3Cl)no2)ccccc1F CN1CCN(C(=O)C(C)(F)c2ccon2)CC1C(=O)NC1CC2CC(O)C1C2 c1(CN2CCC=C(C(=O)N3CCC(O)C(O)C3)C2)ccc(F)c2ccoc12 N1(C(c2c(Cl)c(C)n(C)n2)=O)CC2CCCC(C1)N2C(C1CCOCC1(C)C)=O c1(C(=O)NCCN(C(c2c(COC)cccn2)=O)C)cc(OC)nc(C)c1 N1(C(CC2CC(C)C2)=O)CC(C)OC(C)(C)C1.c1(C(=O)N)ccc(C(C)C)cn1 C1(C(N2CCC(C#C)C2)=O)CC(C)(C)CCN1C(c1cc(C)cs1)=O c1(NC2CCN(C(c3ccnc(C)n3)=O)C2)ncc(C(C)(C)C)cc1C#N C1(NC(C2C(C)(C)C(NC(=O)C#CC3CC3)C2)=O)CCC(C2CC2)C1 CCCCC(C)(F)C(=O)N1CC(CC(N2CCC(F)(C(N)=O)C2)=O)C(C)C1 C(=O)(C(C)(O)C(F)(F)F)N1CCC(C(C(=O)NCC(C#C)C(C)C)C)CC1 C(c1cccc(F)c1)=CC(=O)NC1C(NC(Cc2nc(C(C)C)sc2)=O)CC1 C(=O)(CS(=O)(=O)C(C)(C)C)NC1CCCCN(C(CSc2n(C)ccn2)=O)C1 CN1CCCC(NC(C2(CCNC(=O)C=Cc3ccn(C)c3)CCCC2)=O)C1 Cc1ccc(CC(=O)NCCOCCN(C)CCCC(F)(F)F)s1 c1(NC(N2CCC(O)(C(CC)C)C2)=O)ccc2c(c1)OC(C)(C)O2 c1(OC)ccc2[nH]cc(CC(N3C4CCC3C(NC(=O)C(C)N(C)C)C4)=O)c2c1 N1(C(C(C)C#N)=O)CCN(C(c2cc(=O)n(-c3ccc(Cl)cc3)[nH]2)=O)C(CO)C1 c1(C=O)ccc(F)c(C)c1O.C(CC(C)CC)NC(C1(C(C)(C)OC)CC1)=O CCCC(C(=O)OC)C(=O)N1CC(CNC(c2ccc(Cl)o2)=O)CC(C)C1 Cc1ccc(CN2CC(O)(CNC(c3ccnn3CC(F)F)=O)C2)cn1 N1(C(C(CC(=O)OC)C)=O)CC=C(C(C)(C)C(=O)NCC(C)CCCC(C)C)C1 c1(C(=O)NC2COCCN(C(c3cc(C)nnc3O)=O)C2)cc2cnn(C)c2s1 N1(C(C2(C)CCC2)=O)CC(C2CN(C(=O)CCOCC3CCCO3)C2)C1 C(=O)(CCCCCF)OCc1cn(CCOC)nn1 c1(CNC(c2cc(C)ncc2)=O)nn(C)c2c1CN(C(=O)C(C)(Cl)Cl)CC2 CC1(C(N2CCN(C(C3CC4CCC3C4)=O)CC2)=O)CCC2(CC1)OCCO2 Cc1ncnc(C)c1C(=O)NCC1(F)CCN(C(c2cc(Br)ncc2F)=O)CC1 C(=O)(C1SCCc2sccc21)N1CC(CC=C)(NC(c2ccn(C)c(=O)c2)=O)C1 C1(CNC(C2CCC(CC)O2)=O)CCCC(CNC(c2cocc2C)=O)C1 c1(OC)cc(Br)c(C(N2CCN(c3ccnc(C4CC4)n3)C3CC23)=O)cc1OC NCCCCC(N)C(=O)N1CCC(C(N2CCCC(C(N)=O)C2)=O)(C(F)F)CC1 C(C(=O)NCCCN(Cc1cccnc1)CC)(C(C)C)OC.C(=O)C(F)F C=CC(CC)CC(=O)N1CCC(CCOC)(NC(=O)Cc2ccsn2)C1 C12(C(=O)NCC3(NC(CC(C)C4CCCCC4)=O)CCC3)CC1COC2(C)C c1(OC)ccc(C(N2CC3C(C2)N3c2nccc(N3CCCC3)n2)=O)cc1Cl Cc1cc(C(=O)NC2CC3(C2)CC3NC(=O)COC2CC=CC2)cnc1C c1(C(=O)NCC2(F)CCN(C(c3cc[nH]c3)=O)C2)ccc2nc(O)nc(O)c2c1 c1(C(=O)NC2(CC(N3C(C#C)CCC3)=O)CC2)cc(N)cc(F)c1 C(=O)(CCCCC(C)=O)N1CCC(C(CNC(CC(C)OC)=O)O)CC1 C1(CC=O)CCC(F)(F)CC1.c1(C(N(CCC)CC)=O)cc(C=O)on1.N CC1CN(C(C2CCN(C(=O)N(C)C)CC2)=O)CCC1.C1(CC(=O)N)CC=CC1 c1(C(N2C(C(CNC(C(CC)(C)C)=O)(C)C)CCC2)=O)ccc2c(c1)COC2=O C(=O)C#CC1CCCOC1.C(C(=O)N(CCCOCC)C)(C(C)C)OCC(C)C Cc1ccc(C(=O)NC2(CCNC(C3CCCCN3C)=O)CCC2)cc1O C1CN(C(=O)C(C)Cc2c(C)nn(C)c2C)CCC1C.C1(CC=C)(C(=O)N)CC1 c1(OCCCCC)cc(C)ccc1CNC(=O)C(c1ncccc1F)(F)F N1(C(=O)OC(C)(C)C)CCCCC(F)(F)C1.c12ccc(s1)C(=O)N1CC2C1 N1(C(C(=O)Nc2ncc[nH]2)=O)CCN(C(c2c[nH]nc2F)=O)CC2CCCCC12 CC(C(F)(C(=O)O)C(=O)O)NC(c1c(Cl)cncc1Br)=O C1(NC(c2csnn2)=O)CCC(NC(C2(n3cccn3)CCOCC2)=O)CC1 Cc1cc(C(N2CCC(C(=O)Nc3cc(F)ccc3C)C(O)C2)=O)cc(C)c1 CC1CC(=O)NC(C(=O)NC(C(=O)NC2CCC(C)(C)C2)C(C)(C)O)C1 CC1(C(=O)NCC2CCCCN(C(C3(C#N)CC3)=O)C2)COc2ccccc2O1 Cc1cc(C(=O)N(C2CCC2)C(C)C)n(C2CCOC2)n1 N1(C(CCSCCC)=O)CCCC2CCN(C(=O)C3=CCSC3)CC12 n1(C(CSC)C)cc(C(C)O)nn1.C1(c2cccs2)C(=O)N1 C(=O)(CCCCCCNC(c1c2c(nn1C)CCC2)=O)NC1CC(OC(C)C)C1 C(=O)(CC1COc2ccccc21)N(C(C)CCNC(c1ccc(C(N)=O)o1)=O)C c1(CNC(C(C)CCN(C)C)=O)nn(C)c2c1CN(C(=O)C(O)C1CCC1)CC2 N1(C(C(=O)NC)=O)CCCC(C(C)NC(=O)C(C)n2cccn2)C1 N1(C(CCc2n(C)cnc2)=O)CCN(C(c2cnnc(O)c2)=O)CC1CO c1(CNC2CCC(C(=O)Nc3cccc(OC)c3Br)CC2)cccc(Cl)c1C#N C(=O)(C#CC1CCOC1)NC(C(C(=O)NC1C(OCC)CCC1)(C)C)C c1(C(=O)NCC2CN(C(C3CC=CC3)=O)CC2(F)F)ccn2nncc2c1 C1(NC(C2ON=C(CC)C2)=O)CN(C(c2cc(C#N)ccc2C)=O)CC1N=[N+]=[N-] c1(OC)ccc(C(=O)NC2C3CC2N(C(=O)C(c2cnn(C)c2)=O)C3)nc1Br Cc1ccn2nc(C(N3CC(NC(=O)CC(C)F)C(C)(C)C3)=O)nc2n1 CC(=O)C(C)CC(C)C(=O)N1CCCC(N(C(=O)CC(C)N(C)C)C)CC1 CCC(CC(=O)NCc1ccccc1C(N)=O)OC C1(CNC(C(C)CCO)=O)CN(C)CCN1C(=O)CC1CC(=O)NC1=O c1(CC2OCCN(C(Cn3cc(CC(C(=O)OC)C)nn3)=O)C2)cnc(C)cc1Cl c1(-c2n(-c3ccc(C(=O)NC)cc3)nc(C3CCCO3)n2)cc2cnccc2o1 c1(C(=O)NC23C(CN(C(C4(C)CCC45CCC5)=O)C2)C3)ccc2cnccc2c1 c1(C(=O)NC(CC)CN(C(=O)C=Cc2ncco2)C)ccc(F)c(C)c1N c1(C(=O)NC2COCC2NC(c2coc(C(F)(F)F)c2)=O)cncc(O)c1 N1(C(C2(CC(C)C)CC2)=O)CCCC(O)(C)C1.C1(C=O)C(C)(C)OC1(C)C N1(C(C2C=CC(=O)N=N2)=O)CC(C(=O)Nc2cncc(F)c2)CC(F)(F)C1 c1(OC)nc(Br)ccc1C(N1CC2CN(Cc3ccnc(Cl)c3)C2C1)=O c1(C(=O)NCC2CN(C(CCCSC)=O)C(C)C2)ccc2c(c1)nc(O)n2C c1(CNC2CC(CC(N3CCCC(C(=O)OC)C3)=O)C2)c(O)cccc1Cl CC1(C)CC(C(=O)NCC2(O)CCC2)O1.c1(C=O)ocnc1C(F)F.C C1(C(=O)NCC(CCOC)O)CCCCCN1C(c1ccoc1C)=O c1(OC)ccc(C)c(C(N2CCC(C(=O)NCCO)CC2)C(=O)NCCCF)c1 c1(C(N2CCN(C(=O)CCc3ccc(F)c(Br)c3)C(C)C2)C)ccc(F)cc1F c1(C(N2C(CNC(=O)CC3CCC4CC4C3)CC(F)C2)=O)cc([N+](=O)[O-])n[nH]1 C#CCC(C)(C)NC(=O)CCOCCN(C)C(C1(COC)C=CCC1)=O C(c1ccc([N+](=O)[O-])cc1)=CC(=O)NC1(CO)CCCN(C(=O)C=CI)C1 N1(C(CSCC=C)=O)CCN(C)CC1C(=O)NC(C)Cc1cc(C)[nH]n1 CC1(NC(=O)CCCCCn2cc(C3CC3)nn2)CCCCC1(F)F c1(C(=O)NC(CNC(C(CCC)C)=O)(C)CO)ccc2occ(C)c2c1 C1(CC(=O)NCC(C)NC(C=CCCC)=O)COC(=O)N1 N1(C(CC=C(C)C)=O)CCCC2(CC(NC(c3nnn4c3CSCC4)=O)CO2)C1 C(=O)(C(F)(CNC(C1(O)CCCOC1)=O)C(C)C)N(CC=C)CCOC N1(C(C(C)CCCc2ccccc2)=O)CCn2c(C#N)ccc2C1C CS(=O)c1ccc(CNCc2nc(-c3cc(Br)cc(Br)c3)no2)cc1 C1(CNC(c2c(F)cccc2F)=O)CCCN(C(=O)CCCC2CC2)CC1 C1(NC(c2ccc(N)cn2)=O)CC(NC(=O)CC2CCSCC2)C12CCOCC2 c1(C(c2nnnn2C2CC2)NC(CCCC=C)C)c(Cl)nc2ccccn12 c1(C(=O)OCC)cc(Br)c(OC)cc1Oc1cccc(C#N)c1 n1(CCC(=O)NC2CC(NC(C(CSC)C)=O)C2)cc(Br)c(C)n1 n1(C(C)C)nnc2c(N3CCC(C)C(NC(=O)CC4CCCC4C)C3)ncnc12 N1(C(c2cc(OC)ncc2)=O)CCN(C(C2CC3CC2C3)=O)CC1CO c1(C(=O)OC)cccc(NC(=O)C(c2csc(Br)c2)NC)c1.C1CCOCC1.C CCCCC(CC(=O)NOCCC(C)C)NC(c1ccsc1Cl)=O N1(C(c2ccc(OC)cc2O)=O)CCC2CCC(NC(C3CSC(C)=N3)=O)C1C2 C1(CNC(C(Cn2ccnn2)NC(C(C(C)C)=O)=O)=O)CCCCC1(C)C N1(C(CC(C)n2cccc2)=O)CCC(N=[N+]=[N-])(C(=O)N(C2CCC(O)CC2)C)C1 C1(C=O)Cc2ccccc2N(C)C1=O.CC(F)CC(=O)NCC1(F)CC(C)C1.N C#CC12CC1CN(C(=O)C(=O)NC1CCCC1C(C)(C)C)C2 c1(C(N(C(C)CNC(=O)Cc2nc(C3CC3)cs2)C)=O)ccncc1O c1(C(=O)NCC2CN(C(C3=CC(C)(C)C3)=O)CC23CC3)n[nH]c2c1CCCC2 CSC=CC(=O)NC(C1CCCC1)CNC(c1sccc1-n1cnnn1)=O c1(C(=O)NC(C)C(C)NC(c2cccc(=O)n2C)=O)cc2nc(Cl)ccc2s1 c1(OC)c(C(=O)NC)ncnc1C.C1(C)CCCN(C(C2CC2C(C)C)=O)C1 N1(C(CCCC(C)=O)=O)CCC2CCCC(C1)N2C(=O)CC(=O)OC(C)(C)C n1(CCOC)cc(C(=O)N(CCC(C)NC(=O)Cc2ccon2)C)cn1 C1(CC=C)CCCCN1C(=O)CC1(NC(=O)CCC2CCCOC2)CCCCC1 Cc1ccc(C(=O)NCCCC(C)NC(c2ncncc2Cl)=O)c(Br)c1 Cc1cc(C(=O)NC(C)(C)C2CC2)cc2nc[nH]c12.C1(C(=O)N)CCC12CCC2 c1(C(N2CC(N(C(=O)CC3(O)CCC3)C)C(F)C2)=O)cc(F)cc(Br)c1O C#CCC(C)(C(=O)NC1(CC)CC1)NC(=O)C(C)CCCC c1(C(C(=O)NCC(CC)NC(=O)CN2C(C)CCC2C)O)cc(F)cc(F)c1 CCC(C)C=CC(=O)N(CC(=O)NCC(C)OCC1CC1)C CC1CN(C(C2CCN(C)CC2)=O)CCCN1C(C1CC1Br)=O N1(C(c2cc(OC)ncc2)=O)CC2(CC(NC(=O)C(C)(C)C3CCCO3)CO2)C1 N1(C(CCC)=O)CC2CC2(CNC(=O)Cc2c(CC)noc2CC)C1 c1(NC(c2ccc(C)cc2C)C)nccc(=NC2COCC2CO)[nH]1 CCCCC(CNC(c1cn(CC)nc1C)=O)NC(=O)CC(=O)N(C)C C1(C(N2CC(CC)(OC)C2)=O)CC2CCC(C1)C2.C1(CC(=O)N)COCCOC1 Cc1ccc(C(=O)NC2CC3CC(NC(=O)CN4CC=CC4)C2C3)c(N)c1 N1(C(c2c(C)c(O)ccc2)=O)CCC2(CCC2NC(c2cnn(C)c2Cl)=O)CC1 n1(CC(CO)F)c(-c2c[nH]c3nc(Cl)ccc23)csc1=Nc1ccccc1F O(C=C(C#N)C(=O)NCCOC1CCN(C(c2cnc(C)nc2)=O)C1)CC.C C(CN=C(NCCOC)N1CCC(C2CCOC2)C1)c1nc(CC)c(C)s1 CC1CCCN(C(c2nc(Cl)ccc2F)=O)C1CNC(C1SCCS1)=O c1(C(N2CCC(NC(c3n[nH]cc3F)=O)CC2)=O)ncnc(O)c1Br C1(C(=O)NCCCNC(N)=O)CC2CCC1N2C(=O)CC1CCC(=O)NC1 CC1CN(C(C2(C(F)F)CC(=O)C2)=O)CCC1.C1CC(F)(F)C1.C(=O)(C)N C1(NC(C(C)(F)F)=O)CCN(C(c2coc(C(N)=O)c2)=O)CC1(C)C N1(C(CC(=O)NCC)=O)CC2CCCCC2(NC(=O)C2=CCCCCC2)C1 c1(SC)ccc(OCc2nc(-c3cc(Cl)cs3)n(-c3cccnc3)n2)cc1 c1(C(=O)NCCCC)c(OC)ccc2[nH]ccc12.N1(CC(=O)N)CCCS1(=O)=O C1(NC(C(CN(CC)CC)F)=O)CCN(C(c2nc(O)c(C)s2)=O)C(C)C1 CCC(CC(=O)N1CC=C(CNC(C2CCCOC2C)=O)CC1)C(C)C Cc1ccc2sc(NC(=O)NCC(c3ccc(F)cc3)(F)F)nc2c1C c12ccc(cc1)C(=O)N1CCOC(C1)C2.C1(N(C)C)CCCCC1 C1(NC(c2cc(C(F)F)no2)=O)C2CC1N(C(=O)C(c1ccc(F)cc1)O)C2 N1(C(CNC=O)=O)CC(NC(=O)CCCNC(c2ccsc2)=O)CC12CCOC2 C#CCCCCCC(=O)NC(C1CCN(C(=O)Cn2cc(C(C)O)nn2)CC1)C C(=O)(C(F)(F)C1CC1)NC(C1CCN(C(=O)COC2CCCOC2)C1)C C1(C(N(CCC)CCC)=O)(NC(=O)CC2CC=CC2)CCc2cc(Br)ccc2C1 c1(C(=O)NCC(CCOC)NC(=O)Cc2cscn2)nc2cnccc2s1 c1(C(C)C(N2CC(O)(CNC(=O)CC3OCCCO3)C2)=O)ccc(Cl)cc1 N1(C(c2c(C)occ2)=O)CCCC2(C1)CN(C(=O)C(F)(F)C1CCCC1)C2 c1(N2CCCC(c3ccc(CC)cc3)C2)nc2nc(C)cc(=O)n2[nH]1 C(N=c1[nH]c(=NCCC#CBr)[nH]c2c1SCC2)C12OCC(C(F)F)(C1)C2 CC1CCc2cc(C#N)c(NCc3ccc4ncccc4c3)nc2C1 CC#CCC(CO)NC(C1CC2CC2N1C(=O)CCCCC1CC1)=O Cn1nnc2cc(C(N3CC(NC(=O)C(O)C(F)F)CC(C)(C)C3)=O)ccc12 C(C(C)S(C)(=O)=O)NC(Cc1ccn(C)n1)=O.C1(C(=O)N)CCC(C2CC2)C1 N1(C(c2c(CC)ccs2)C(=O)NC2CC(F)(F)C2)CCC2C(O)CC12 n1(CC)cnnc1C(=O)N(CCC(C)NC(=O)CCOC1CCOCC1)C C1(NC(C=C(C)C(F)F)=O)CN(C(C2CCCC(=O)N2C)=O)CCC1O C1(CC)CCCC(NC(C2(C)CCCCC2)=O)C1.C(C)(C(F)F)=CC=O.N C=CCC(C)(O)C(=O)N1CCC(NC(=O)CC2(C)CCCCC2)C(CO)C1 Cc1nocc1C(=O)NCCC(O)CNC(=O)CCN(CC(C)C(C)C)C c1(NC(CC(C)C)=O)ccc2oc(=O)n(C)c2c1.C12CCN(C1)CCO2 C1(NC(=O)OC(C)(C)C)CCC1C(=O)NC1CC1.C1(C=O)CCOC1 C1(N(C(c2ncc(Cl)n2C)C(=O)NC)CCC)CC(=O)NC1=O.C(C)C C1(F)CCCN(C(=O)CC2(C)CC2(F)Cl)C1.Cc1cc(C)n(CC(=O)NC)n1 C1(F)(CNC(c2n[nH]c(C)c2F)=O)CCCN(C(C2(C(C)(F)F)CCC2)=O)C1 N1(C(C(=O)NCCCF)C2CCSC2)CCOCC1CC1CCC1 C1(NC(C=CC=CCC)=O)C2CCN(C(c3cc(C(N)=O)co3)=O)C12 N1(C(COC)=O)CCC(NC(=O)CCCn2ccnc2C)C(CO)CC1 c1(C(=O)NCC2C(NC(CC(=C)C)=O)C2)cc(C#N)ccc1O N(C(=NCCC1OCCC1C)NCc1ccccc1)C(c1ccccc1)C#C Cc1nnc(C(=O)NCC(C)(C)CN(C(=O)CCOc2ccccc2)C)s1 C1(C=O)CC2C(C1)C2(C)C.C1CCC1.c1(C(N(CC(=O)N)C)=O)cccs1 N1(C(c2c(C)nncc2)=O)CC(NC(=O)C(C)(C)C)CC(F)C1 c1(N2C3C(NC(C(C(C)C)OC)=O)CC(CC3)C2)nc(Cl)nc2c1CCOC2 c1(C=O)ccn2c(O)nnc2c1.n1(CC)cccc1C(=O)NC1CC(O)(C)C1 N1(CC2CCC(C)CC2)CCC(=O)N(CC(C)(C)C2CC2)C1=O C=CC1COCC1NC(=O)CC1CCCC(NC(C2(CC)CCC2)=O)C1 CC(C)C(C)(F)CNC(C1CCCN(C(C2CC(=O)C2)=O)C1)=O c1(OC)ccc(C(=O)NC2CCC2CNC(=O)C2=COCC2)c(Br)c1 N1(C(C(C)O)=O)CCc2sccc2C1CNC(=O)C=Cc1ccc(N(C)C)cc1 c1(C(=O)NC2CC(NC(C3CCC(=O)NC3)=O)C2)cnc(-c2nccs2)nc1O C(C1=CCN(C(c2cc(C)ccc2CC)=O)CC1)NC(CC1CC(=C)C1)=O Cc1nc(CC(C)C)sc1C(=O)NC1CCN(C(c2ccnc(O)c2)=O)C1 N1(C(C)C)CC(C(=O)NCC2(C)CCCN(C(=O)Cn3ccnn3)C2)CCC1=O C1(C=O)CCC(C)=C(C)C1.N1(S(CC)(=O)=O)CCCC1C(N1CCC(C)C1)=O C1(C(=O)NCC(O)CNC(c2ncoc2Br)=O)(COC)CCOCC1 c1(CNC(=O)NC(C(C)(C)O)Cc2ccc(F)cc2)ccc2c(c1)CCCS2 n1(CCC)nc(C)c(C(=O)NC2C3CN(C(=O)C(=C4CCCCC4)F)CC23)c1C C1(NC(C(CC)SC)=O)CN(C(c2c(C)ccnc2O)=O)CC(C)(C)C1 CC(CC(=O)N(C1CCC(CNC(=O)CCc2ccnn2C)CC1)C)C(F)F c1(C(=O)NC2CC(NC(CC3CC(=O)NC(=O)C3)=O)C2)cc2c(cn1)CCCC2 C(CN=c1[nH]c(=NCc2cccc3ccnn23)[nH]c2ccsc12)SCC C12(C(=O)N)CC(CO1)N(C(C1(C)CCC3CC3C1)=O)C2.CC(C)S(N)(=O)=O C=CCCC(CC(C)C)C(=O)N1CCC(CC)(NC(c2ncccc2F)=O)CC1 c1(CC=O)cc(S(=O)(=O)N(C)C)c(C)o1.c1(C(=O)OC)cccc(C)c1.C CC1CC(C(=O)NC2C=CC(C)(C)CC2)CN(C(=O)C(O)CN(C)C)C1 N1(C(C2C(C=C)OCC2)=O)CCCC(C(=O)N(C2CC(CO)C2)C)CC1 N1(C(CCCSC)=O)CCCN(C(=O)C(C)NC(C2CCCC2)=O)CC1 c1(C(=O)NCC(C)N(C(=O)C=Cc2ccco2)C)cc2n(n1)CCC2 O=C(CCC(=O)N1CCC2C(NC(=O)CC3CC=CC3)C12)c1ccc[nH]1 C12(CNC(=O)CCC3CCCN3)CC(C1)C(C(F)(F)F)N2 N1(C(C(CC)(C)C#N)=O)CC2C3CCC(C2C1)N(C(c1c(Cl)cnn1C)=O)C3 N1(C(c2cnn(C(C)C)c2Cl)=O)CC2C(C1C(=O)NC)C2(C)C.c1ccccn1 CC1(O)CCN(C(=O)CSCCNC(C2(C)CCC3CC3C2)=O)CC1O C(C(=O)NCC(C1CC1)N(C(=O)CO)C)(C1CCOC1)OC.c1nc[nH]n1 N1(C(C)=O)CC2CCCC(NC(c3ccnc4[nH]nnc34)=O)(C2)C1 c1(C(=O)NCCN(C)C(c2cc3ccsc3n2C)=O)cc([N+](=O)[O-])cn1C C(=O)(CCCCC(=O)OC)NCC(CC)(CC)NC(=O)CS(C)(=O)=O C1(OC(C)(C)C)CCCCC1NC(=O)NC1(CC)CC(F)(F)C1.CCO.O N1(C(c2c(Cl)nc(OC)s2)=O)CC(NC(c2[nH]c(C)nc2C)=O)C2(CC2)C1 C1(NC(c2c(C(C)(C)C)n[nH]c2)=O)CCCC2CN(C(=O)Cn3cccc3)CC12 c1(C(N)=O)cc(NC2CCCC(NC(=O)CCC3CCCC3)C2)ncn1 C=CC1CN(C(c2ccc(Cl)cn2)=O)CC1NC(=O)Cn1nccn1 c1(C(=O)NC(CSC)(C)C(=O)N)ccc(=O)n(C)c1.c1cccc(C(C)C)c1 c1(CC(=O)NC(CN2CCCC(C=C)C2)=O)ccc(S(N)(=O)=O)s1.C1CCCO1 c1(OCCCNC(=O)Nc2cnn(CC3CCOC3)c2)ccc(F)c(F)c1 C(=O)(C1=CCCCC1C)N1C(CNC(c2ccc(C)c(C)c2)=O)CC(C)(C)C1 N1(C(Cc2c(Cl)ccc(OC)c2)=O)CC(C2CN(C(c3nnn(C)c3N)=O)C2)C1 N1(C(c2cc(OC)ncc2)=O)CC2(C1)CN(C(=O)CCC(C)OC)C2 c1(NC(c2ccc(OCCCCCC)cc2)=O)c(Cl)ccnc1Cl CC1CN2CCN1C(C(N1CCC(N(C(=O)Cc3nncn3C)C)C1)=O)C2 C1(NC(CN2CC(C)(OC)C2)=O)CCN(C(c2ccsc2)=O)C(C)C1 c1(OCC)ccccc1-n1cc(CNC(=O)CC2CCC(=O)C2)nn1 CC1(C)CCC(C(=O)NCCCc2ccccc2)O1.C1(C(=O)N)CC(C2CC2)C1 C1(CC=C)(NC(=O)OC(C)(C)C)CC(C(=O)O)C1.c1cccc(Cl)c1.N CCCCC(O)CC(=O)N1CCN(C(c2cc(Cl)cnc2C)=O)C(C)C1 CCC(C(=O)OC)C(=O)N(CC(O)CN(C)C(c1ccc(C(C)(F)F)nc1)=O)C c1(C(=O)NCC(CC)NC(=O)CC2SC(=N)NC2=O)cc(COC)oc1C CC1CCN(C(=O)CC2CCCSC2)CCN1C(C1CC2(CSC2)C1)=O CC1(C)CCN(C(=O)C(F)(F)C2CC2)CC1CNC(c1ccc(CF)cc1)=O CCC(N=c1[nH]c(=NC(C)c2nnc3n2CCC3)c2sccc2[nH]1)C1CCCC1 Cc1cc(=NCCCC(C)(C)NC(c2ccn(C)c2)=O)[nH]cc1[N+](=O)[O-] C=CCCCC(C(=O)NCc1ncn(C)n1)NC(=O)C(C)n1ccnn1 C1(C=O)CC(CC)=NO1.C12CC(C1)C2.C1(CC(=O)N)(OCC)CCC1.C N1(C(C2(CF)CCN(C(C(COCC)N=[N+]=[N-])=O)C2)=O)CCC2(CCOC2=O)C1 c1(C(=O)NCC(CO)NC(c2cn(CCC=C)nn2)=O)cn2cccc(C)c2n1 C#Cc1cnn(C)c1C(N1CC(N2CCN(C(C3CC34CC4)=O)CC2)C1)=O N1(C(C(c2scc(C)n2)C)=O)CCC(N(C(=O)Cn2ccnn2)C)C2(CC2)C1 C1(NC(C2(CC=C)CCN(C(=O)CCCCCF)C2)=O)CCCCC1C#N c1(CC)ccc(C(=O)NC2CCC2NC(c2sc(C(C)C)nc2C)=O)nc1 C1(C(=O)OCC)OCCNCC1N(C1CCC(F)C1)C(c1cccn1C)=O C1(NC(CC(C)c2ccco2)=O)CCC2CCN(C(C3CC(O)C3)=O)C1C2 CC1CCN(C(=O)CC2(O)CCOCC2)C1CNC(c1cnc(N(C)C)s1)=O c1(C(=O)NCC(CO)Nc2nccc(CC#N)n2)ccc2[nH]ccc2n1 CCCS(=O)(=O)C1CCCC1NCC1OC2(C)CC1(CO)C2 C1(C(N(CC=C)C)=O)CCN(C(C2(Cl)CCCCC2)=O)CC1 Cc1cc(Cl)ncc1C(N1CC(O)CC1C(N1CC2CC2C1C#N)=O)=O CC1(C)CCOC1CC(N1CC=CC1(C)C(=O)NCCF)=O c1(C(N2CC3CCC2CN3C(C2(F)CCOC2)=O)=O)n[nH]c2c1CC1CC21 C1(C(N2CCC2C(C)C)=O)(COC)C=CCN1C(=O)CC1CCC(O)C1 c1(C(N2CCCC2)=O)cc(C)cc(C)c1N.C(=O)(C(C)N1CCCC1)N(CC)C c1(C(N2CCCC(O)(CC)C2)=O)cccc(S(=O)(=O)NCCCc2nn[nH]n2)c1 C1(C(N2CCC(C)(C)C2)=O)Cc2ccccc2O1.c1(CC)cnoc1C(=O)NC c1(C(=O)NC(C2CCCN2C(C2CC=CCO2)=O)C)cc(C(F)F)ccn1 c1(C(=O)NC2CCCN(C(c3cccc(O)c3Cl)=O)C2)cc2cc(F)ccc2s1 C(=O)(C1=CCCOC1)NCCC(C)NC(c1ncnc(O)c1Br)=O c1(C(=O)NC2CC3CN(C(CC(CC)CC)=O)CC2C3)cc([N+](=O)[O-])cnc1C Cc1c[nH]c(C(=O)NCc2cc(C(=O)Nc3cscc3C3CC3)n[nH]2)c1 c1(C(C(=O)N)=O)cc(F)cc(Cl)c1.Cc1ccn(CC(=O)NCCC2CC2)n1 N1(C(C(C(C=C)C)C)=O)CCn2nc(CNC(c3cnn[nH]3)=O)cc2C1 C(C(C)(C)S(C)(=O)=O)c1nnnn1C1CCOC1.c1(COC)nc(C)cs1.N C#Cc1ccc(C(N2CC(NC(=O)CC=C=C)C(O)C2)=O)cn1 c1(C(=O)N)ccc(N)cc1F.Cc1c(C(=O)NC2(C)CCC2)cnn1CC(F)F Cc1cc(C(=O)NCC(O)CN(C)C(C2(C(C)C)CCC2)=O)c(Cl)cc1N C1(N(C(C(CSC)C)=O)CC2CC2)CCN(C(C2C3CC3C3CC23)=O)CC1 c1(C(N(CC(CNC(c2c(SC)csc2)=O)O)C)=O)cc(C2CC2)ccn1 C(=O)(C(F)C(C)CNC(=O)C(=O)NC(C)C)NC(c1c(C)nns1)C CCCC(C(O)C(=O)N1CCCOC(CNC(=O)COC)C1)NC(C)=O C(=O)(C(C)(O)C(F)(F)F)NCC(CC)NC(CCC(=C)Cl)=O C1(C(=O)NCCC2(O)CN(C(C(C(C)(C)C)=O)=O)C2)Cc2ccncc2C1 Nc1c(O)ccc(Cl)c1C(N1CCC(NC(C2(CF)CCOCC2)=O)C(O)C1)=O C(=O)(C#CC1(CC)COC1)NC1C(CC(=O)NC(C=C)C)CCC1 N(C1CCc2cccnc21)C(C=CC(C)NC(C=C(C)C1CC1)=O)=O C1(NC(CCn2ncc(C)c2)=O)CCC(C)(CNC(C2CCC2(F)F)=O)CC1 CC1(C)CC(C(=O)NCC2CCC(NC(=O)C#CC3CCC3)C2)=NO1 C1(CNC(CCNC(CC=CC(C)(C)C)=O)=O)CC12CC2(F)F Cc1nscc1CC(=O)NCCC(C)NC(c1snnc1C(C)C)=O c1(NCC(c2cccnc2)C)nc(N2CC3CSCC3(C)C2)nc2ncn(C)c12 C1(C)(CNC(CC(CC)C)=O)CCN(Cc2ncc(C(C)(C)C)o2)CC1 C(=O)(C#CC1CCCCO1)NC1(C2N(C(C(CC)N(C)C)=O)CCC2)CC1 CC1CN(C(C2CC(=O)N(C)C2)=O)CCC1.c1(C(=O)N)ccc(N(C)C)c(Cl)c1 N1(C(C(CO)OC)=O)CCOC(C(=O)NCC2(CN(C)C)CCC2)CC1 c1(C(=O)NC(C(=O)NC2CC(COC)C2)C(C)C)cccc2ccoc12 N1(C(c2c(OC)cccc2)=O)CCC(F)(C(=O)N(C2CCC(CO)CC2)C)CC1 C=CCC(CC(C)C)C(=O)N1CC(C)(C)CC1C(=O)NCCCn1ccnn1 CCCS(=O)(=O)CC(=O)N1CC(NC(=O)C(C)CSC)CC2(CC2)C1 C1(NC(c2scc(COC)c2)=O)CN(C(=O)CCC(C)(C)C)CC12CCOCC2 Cc1oc2cc(C(=O)N(C3C4CN(C(=O)CC(=O)N(C)C)CC34)C)[nH]c2c1C c1(C(N2CC3CN(C(c4onc(C)n4)C)CC3C2)=O)cc2ccccc2nc1O Cc1c[nH]c(C(=O)NCC(C)CNC(c2cc(F)cnc2O)=O)cc1=O C1(c2cc(CNC(c3ccc(OC)s3)=O)on2)CCN(C(=O)C(C)C)CC1.O [N-]=[N+]=Nc1cccc(CNC(=O)CC2(CSc3ccccc3)CC2)c1 c1(CC)nnc(COC2CCN(C(=O)NC(C)C)C2)o1 N1(C(c2c(C)cc(F)s2)=O)CC(C)(C)CC1CNC(=O)CC1CC(=O)C1 N1(C(CSCC=C)=O)CC(OC)CC1CCNC(c1ccoc1C)=O c1(C(=O)NCC2(F)CCN(C(C(C)C3CCCC3)=O)C2)cc2ccncc2[nH]1 c1(C(N2CCN(C(CS(=O)(=O)N(C)C)=O)C3C2C3)=O)noc2c1COCC2 c1(C(=O)NC(CNC(C2N(CCCC)CCCC2)=O)(C)CC)nn(C)c(N)c1C c1(NC(C2N(C(C3(COC)CC3)=O)C3CCC2C3)=O)ccc2nsnc2c1 N1(C(C(C)(C2CC2)OC)=O)CC(NC(=O)CC)C2(CC2)C1.c1cccnc1.O N1(C(c2n(C=C)nnc2)=O)CC2CCCC(C1)N2C(c1cnc(C2CCC2)s1)=O Cc1cc(NC(=O)C(C2CCN(C(=O)Cc3csnc3C)C2)C)cnc1F c1(OC)cnnc(C(=O)NC2(CCNC(=O)Cc3ccc(O)nc3)CC2)c1 C1(CNC(C(CC)OCC)=O)COCCN1C(=O)CCC(=O)NCCC c1(OC)cc(C(N2CCC(C(=O)NCC(C)(O)C3CCCC3)(CF)C2)=O)ncn1 C1(C(=O)NCC2CCC(NC(=O)Cn3cccnc3=O)C2)SC2C=CC1CC2 C1(C)(CCNC(C2(CSC)CC2)=O)CCN(C(C2COC(=O)N2)=O)CC1 c1(CNC(c2c[nH]nc2-c2ccccn2)=O)ccc2c(c1)CCNCC2 Cc1cc(C(=O)N(CC(C)C)C)ccc1C(F)F.c1(C(=O)N)ccc2c(c1)CC2 C1(C(N2C(C3CCN(C(c4cocn4)=O)C3)CCC2)=O)C(F)(F)C12CCC2 C1(NC(CC=C=C)=O)CCCC(NC(=O)C(C2CCC2)OC)C1 CP1(=O)CCN(CC(=O)NC2COC3(C)CC2C3)CC1.C(=O)(CCC1CC1)N N1(C(C(=Cc2ccccn2)C)=O)CC(=O)N(C)CC1C Cc1cc(C(=O)N)c(C)o1.C(=O)CC=C(Cl)Cl.C1(N(C(C)=O)CCO)CCCC1 N1(C(C23OC(C)(C)C(C2)C3)=O)CC2(CCC(CNC(=O)C(F)(F)F)O2)C1 C1(CNC(CNS(CCCC)(=O)=O)=O)CC2CCC1N2C(=O)C(O)CCC C1(C(=O)NCCC2CCN(C(C(C(C)(C)C)O)=O)C2)CCCCCC(=O)C1 C12(C(=O)NCc3ncc(C)o3)CC(CO1)N(C(c1cc(C#N)n(C)n1)=O)C2 C1(OC)CC(C(=O)NCC(CNC(=O)Cn2nccn2)CO)CC1OC Cc1cc(C(=O)NC2C3CC2N(C(=O)C(C)C(C)(C)O)C3)c(C)cc1Br c1(C(N2C(CNC(C3COC(C)(C)C3)=O)CC(C)(C)C2)=O)cnn2ccccc12 c1(C(=O)NCC(CNC(C(CC)SC)=O)CO)cccc(O)c1C N1(C(c2c(C)ocn2)=O)CC2(NC(c3cc4n(n3)CCC4)=O)CCC1CC2 C1(NC(C(C)CF)=O)CC2CC(C1)N(C(=O)C(C)(C)C1CCC1)C2 CC1=NOC(=O)C1CCC(=O)NCC#CC.C(=O)(C(C)(O)Cc1ccccc1)N C(=O)(CC(F)(F)F)NCC(Cn1cc(CC(CC)(C)O)nn1)(C)C N1(CCNC(Cn2ccc(C)n2)=O)CCN(C(c2coc(Cl)n2)=O)CC1 c1(SC)cccc(CC(=O)N(CC(O)CNC(c2cc[nH]c(=N)c2)=O)C)c1 C(=O)(CN=S(C)(C)=O)N(CCCNC(c1c(C)nccn1)=O)CC1CCCC1 Cc1cc(C)c(C(N2CC3(CCN(C(=O)Cc4csc5nccn45)C3)C2)=O)c(O)n1 C=C(Cl)CCC(=O)NCC1CCN(C(C2(C(F)(F)CC)CC2)=O)CC1 Cc1cc(C(=O)N(C2CCN(C(c3cccc(C4CC4)n3)=O)C2)C)cc(F)c1C C(=O)(C1=CCN(C(C2CNC(=O)C2)=O)C1)N(CCCCOC)C C1(CC(=O)N(CCCOCCC)C)CCCC(O)C1.C(=O)(CC)N.C(N)=O CCC(CC(C)C)C(=O)N1CCC(N(C)C(c2ccc(C#N)n2C)=O)C1 C#CCC(C)C(=O)NCCOC1CCN(C(=O)Cn2cnc(C#N)n2)C1 CC1CCC(=CC(N2CCOCC2CNC(c2csnn2)=O)=O)CC1 C(=O)(C(C)C(CC)CC)NCC(=C)CCNC(c1ccn(-c2ccccc2)n1)=O c1(C(=O)NCC2CCN(C(CC3(CSC)CC3)=O)C2)cnc(O)n1C C(=O)(C(C)C(C)(C)C)N.n1(CC)nnnc1C.C1(CC(C)C)(C=O)CCC1 CCCCCC(O)CC(=O)NCC(C)NC(C1(COCC)CC1)=O C1(C(F)(F)F)(OC)CN(N2CC(CC(F)F)C2)C1 C1(C(=O)N)CC2CS(=O)(=O)CC2C1.C1(NC(c2cnc(S)[nH]2)=O)CCCCC1 N1(C(C2(CCOC)CC2)=O)CCC(C(C)NC(=O)Cc2cc(C)on2)C1 C(C)(CO)(C(=O)N1CCC(N(C(=O)CCCCC)Cc2ccccn2)CC1)OC c1(C(=O)NCC2C(CNC(CC(C)O)=O)C2)cc(Br)c(F)c(F)c1F C1(C(N(C2(C(=O)Nc3c(COC)nccc3)CC2)C)=O)CCCC(C#N)C1 c1(C(=O)NCCC(C)N(C(C(c2c(C)n[nH]c2C)C)=O)C)cnc2nccn2c1 N1(C(C(CNC(=O)Cn2ccnc2)OC)=O)CCOCC1CC(C)C c1(C(=O)NC(CN(C(=O)CC(C)OC)CC)C)ccc(F)c(F)c1N c1(C(=O)NCC2(C)CCN(C(CC(C=C)C)=O)C2)nc2cc(F)ccc2s1 C1(C(C)C)CN(C(c2cc(=O)cc[nH]2)=O)CCC1NC(=O)Cn1ncn(C)c1=O C1(CN(C(=O)CCNC(=O)CO)C)CCCN(C(=O)Cc2ccn(C)c2)C1 [N-]=[N+]=NCCCC(=O)NCC1CN(C(=O)COCP(=O)(O)O)C1 C1(N(C)C(C2(O)CCCC2)=O)CC2CC1N(C(C1CCC(C(N)=O)C1)=O)C2 C1(C)(CNC(CCC(=C)C)=O)COCCN(C(c2cc(Br)c(C)o2)=O)C1 C1(C(N(C(C)C(=O)NC(C)C(N)=O)CC)=O)CC(F)(CF)C1 c1(C=O)cccc2c1OCO2.C1(C(=O)NCC(C)C2CCC2)CC(F)(CO)C1.N c1(C(N(C)CCn2cc(C(C)(C)O)nn2)=O)cc2n(n1)CCN(C)C2=O CCCCCCCCC(=O)NC1CCCCCN(C(=O)CC(C)CF)C1 c1(C(N(C2CCC(NC(CCCCCC)=O)C2)C)=O)ccc2nccnc2c1 c1(C(=O)NC(CN(C(C2(C(=O)OCC)CCC2)=O)C)C)n[nH]cc1CC C1(O)(CNC(c2cccc(Br)c2F)=O)CCCN(Cc2c(F)cncc2F)C1 C(=O)(C1=C(C#N)CCC1)NCC(C(N1C(C)C(O)CC1)=O)N(C)C C(=O)(CCCCCn1cc(-c2cnccn2)nn1)N(C1CCCC(O)C1)C CC1CN(C(=O)Cc2nnc(S)n2C)CCC1CNC(=O)COC1CC1 N1(C(COC23CN(C(=O)OC(C)(C)C)C(CC2)C3)=O)CCC(O)C(F)C(F)C1 C(=O)(C1CCCc2nccn21)N1C(CCN(C)C(c2cnsn2)=O)CCCC1 C1(CNC(c2c(OCC)ccs2)=O)CN(C(c2ccc(Cl)cc2)=O)CC1C C1(NC(c2c(COC)cco2)=O)COC2(CCN(C(C3CC3(Cl)Cl)=O)CC2)C1 C1(C(=O)OC(C)Cc2cccs2)CCN(C(=O)OCc2ccccc2)CC1 Cc1ccc(-n2ccnc2)c(C(N2CCC(C)C(CON)C2)=O)c1 c1(OC)ccc(C(=O)NC2CC(CCNC(C3CCO3)=O)C2)c(Br)c1 C1(NC(CCSC)=O)CCCC12CCN(C(=O)Cc1cnc3c(C)cccn13)C2 Cc1ccc2c(cc(C(=O)NCCCc3ncn(C)n3)n2CC(F)(F)F)n1 C1(C(=O)NCC(CCCC)NC(c2ccc(C=C)cc2)=O)CC2(CCCC2)CO1 Cc1cc(C(N2CCC(C(=O)N(CCCCO)C)(CO)C2)=O)nnc1C c1(C(=O)NC(c2ccccc2CC)CNC(CCCC#C)=O)ccc(N)cc1C C1(N(C(=O)C(c2ccccc2)NC(=O)C)C)CCC(=O)NC1.C1CCOCC1.O CC1(C)CC(C(=O)N2CC=C(C(=O)NC3CCCC(F)(F)C3)CC2)=NO1 N1(CC(=O)NCCC2(OC)CCC2)CCC(CC2CC2)C1 Cc1cc(CC(=O)NCC2OCCC2C(=O)NCC2(CO)CC2)nn1C O=S(=O)(c1c(Cl)cc(F)cc1Br)Nc1ccc(-n2nc3ccccn3c2=O)cc1 C=CCCCCC(=O)NC1CCN(C(C23CCC(OC)C2CC3)=O)CC1CO C(=O)(C(CCF)NC(=O)CSC(F)F)Nc1c(CC)nsc1 c1(C(N2CC(C)CC2)=O)nn(C)cc1S(C)(=O)=O.C1(C(C)(F)F)(C=O)CCC1 N(C1COc2cc(Br)ccc21)C(=O)CN1CCN(Cc2ccccc2)CC1 c1(CC)cc(CC(=O)NCCN(C(=O)CC2CCC(O)C2)CC)n(C)n1 c1(NC(CC2C3CN(C(c4c(C)n(C)cn4)=O)CC32)=O)cccn2ccnc12 c1(CNC(c2cc(OC)nc(C)c2)=O)cc(OC)c(OC)c(Cl)c1 C#Cc1cccc(CNC(=O)CCC2CC2)c1.c1(C(C(=O)N)O)cnn(C)c1 n1(CC(=O)NCC2N(C(C3(OC)CCOC3)=O)CC2)nc(O)ccc1=O c1(C(=O)N)oc2ccccc2c1C.C1(OC)(C)CCN(C(=O)C(F)(F)C2CC2)C1 CC(C(=O)NC1CCCCN(C(=O)CC2COC(=O)C2)C1)C(C)(F)F CCCCCC(O)CC(=O)NCCCNC(c1cnnc(O)c1)=O C1(CC(=O)N)CCCC12CC2.c1(C(N(C)CCOCCC)=O)cnnc(O)c1 C1(CC)CN(C(c2cnc(C)c(C)c2)=O)CCN1C(c1nocc1Br)=O C=CCC(CNC(=O)C(O)c1ccsc1)NC(=O)CC.C1(CC=O)CCCC1 C(=O)C(C)(C)C(=O)NC.C1(CC(N2CC(O)C2)=O)CCS(=O)(=O)C1.CO C=CC1CCCN1C(=O)C=CCC1(NC(C2CC(C#N)(O)C2)=O)CCC1 c1(OC)cc(C(=O)NCCOCCC)ccc1C.C1(C(=O)N)CCC2CC1CO2 C1(C(N2C(CNC(C)=O)CCC2)=O)CC=CCN1C(=O)CCc1cnc(C)o1 CCC(C#N)C(=O)N(CCCNC(c1cc(-c2ccccc2)cn1C)=O)C(C)C N1(C(C2CC(SC)C2)=O)CC(O)(C2CCCN2C(c2ccc(CO)o2)=O)C1 c1(NC(C2C3CC2N(Cc2cccc(O)n2)C3)=O)ccc2c(c1)NCCC2 C#Cc1cccc(C(N2CC(CC)(NC(=O)CS(=O)CC)C2)=O)c1F C(C(CO)C(F)(F)F)NC(C1N(C(CN(C(C)=O)C)=O)CCCC1)=O N1(C(c2nc(OC)oc2)=O)CC(NC(C2CC=CCC2)=O)C2(CCC2)C1 N1(C(C(C)=C2CCC2)=O)CCC(C)C(CNC(=O)C(c2ccc(F)cc2)C)C1 c1(CONC(C2C(C)CN2C(=O)C(C)O)=O)cncnc1O CC1(C)CC=C(C(=O)NC2(C(N3CCCC(CF)C3)=O)CC2(C)C)CC1 C1(NC(=O)Nc2cccc(OCC=C)c2)CCCN(c2ccnn2C)C1=O C(C(=O)NC1CC(C)OC1=O)(C(C)(C)C)NC(c1n(CC)ccn1)=O C1(C(N2CCC(C(C(=O)NCC(F)(F)C(F)F)F)C2)=O)CC(=O)C12CCC2 CCCCCCOCC(=O)N(CCNC(C1CSCCS1)=O)CC1CC1 C(C(C)(C)C#CC(=O)NC1CCN(C)C1C)NC(c1ncc(NC)nc1)=O c1(-c2cn(CC(CCNC(C(CC)N(C)C)=O)F)nn2)cccc(Cl)c1F C(=O)(C(C)(C)CCCO)NC(C)CNC(C1CC(O)(CCC(C)(C)C)C1)=O c1(CNC(C(C)N(C(COCCCC)=O)C2CC2)=O)cc(C2CC2)on1 N1(C(C2N(C(C)=O)CSC2)=O)CCCN(C(c2cc3scc(C)c3[nH]2)=O)CCC1 c1(C(N(C23CCC(C)(C2)OC3)C)=O)ccc(Br)cc1N.C1(F)(C(=O)N)CC1 c1(C(=O)NC2CC(C)(NC(C(CC)=CC)=O)C2)cc(O)c2ccccc2c1 c1(NC2CCCN(C(CC(CC)CC)=O)C2)nc(C)nc2[nH]ccc12 Cc1csc(C(N2CC(O)CC2C(=O)Nc2nccnc2C(N)=O)=O)c1C C1(CNC(C(CC)N(C(=O)Cc2cccnc2F)C)=O)CCCC12CCC2 C1(C(N(C)CC2CCN(C(c3c(C(C)C)n[nH]c3)=O)C2)=O)CC2C=CC1C21CC1 C(C=CC(=O)N(CC(C)NC(=O)C=CC(=O)O)CC)(CC)=CC N1(C(Cc2cc(CC)no2)=O)CCCC(C(C)(C)C(=O)NC(C)(C)CF)C1 C1(C)(C(N2CC(NC(C(C)n3ccnc3)=O)C2)=O)CCc2ccccc2C1 Nc1cc(F)c(Br)cc1C(=O)NCC1CC2CCC1N(C(C1CC1F)=O)C2 CCC(C)C(O)CC(=O)N1CC2CCC1C(NC(=O)C(C)CC(F)(F)F)C2 c1cccc(F)c1.Cc1n[nH]cc1CC(=O)NCC1CCCC1NC(=O)CC.O CC(C)(CC(F)C(=O)NCC1CCC(=O)N1)NC(C1CCOC1)=O Cc1cc(=NCC(C2CCCCC2)NC(=O)C2=COCCO2)c(C#N)c[nH]1 C(C(F)(F)C(F)(F)F)n1c(-c2cc(Br)cs2)nc(CCSC)n1 C#Cc1ccc(C(=O)N(CC(CO)(CO)NC(=O)CCc2ccn(C)n2)C)cc1 C1(n2c(-c3c(CCC)csc3)ncc2)C2C3CCC(C3)C12 C1(OC(C2(CO)CCCO2)=O)CC2(C(=O)OCc3ccccc3)COC1C2 c1(C(N2CC(NC(C(C)SCc3ccccc3)=O)C2)=O)ccc2c(n1)CCC2 c1(C(=O)NCC(C(C(C)C)C)N)ccc(S(C)(=O)=O)o1 Cn1cc(CCC(N2CC(C)(CC(=O)NCCOC3CCOCC3)C2)=O)cn1 C1(C(=O)NC(C2CC2)C2CC2)CCN1C(=O)CCc1nncs1 N1(C(C(CCC2CCC2)NC(C(C=C=C)C)=O)=O)CCC2(CCOCC2)C1 C12(C(N(C)CC3COCCN3C(C3CC=CCO3)=O)=O)CC=CC(C1)OC2 C1(CC)C(NC(c2cnc(N(C)C)nc2)=O)CCCN1C(=O)CCC1CCCO1 C1(CNC(=O)CCn2cc(COC3COC3)nn2)COCCC1(F)F c1(SC)nc2ncn(CC(=O)N(C(C)(C)C)C)c(=O)c2s1 C(=O)(CC(C)C(C)(C)NC(=O)CC1CC(F)(F)C1)NCCC(C)OC CCC(O)(CC(=O)NCCCOCCNC(=O)CSC(F)F)c1ccco1 C1(CNC(c2c(CC)noc2)=O)CN(C(C2(CO)C=CCC2)=O)CCC1C N1(C(CNC(CNC(C)=O)=O)=O)CCCC(C)C1.n1(CC=O)cnc(=N)[nH]1 C1(NC(C(n2cc(Br)cn2)C)=O)(CO)CCCN(C(=O)C(C)CC(N)=O)C1 c1(NC(C2(C)N(C(CCOCC)=O)CCC2)=O)ccc([N+](=O)[O-])c(C)c1 C(=O)(C1=C(C#N)CCC1)N(C(C)C(N1CC(=O)NC(C(C)C)C1)=O)CC N1(C(c2nc(OC)c(C)s2)=O)CCC2(NC(=O)C(=Cc3ccccc3)C)CC2C1 CC(C)S(=O)(=O)C(C)C(=O)N1CCCCC(NC(=O)CCCC(F)F)C1 Cc1cc(Oc2ccc(NC(=O)C(C)Oc3cccc(O)c3)cn2)ccc1Br N1(C(c2c(C)nsc2)=O)C2CCC1CC(O)(CNC(C1(CF)CCOCC1)=O)C2 c1(C(N(CCNC(C2C(C)C2(F)F)=O)CC)=O)cc2c(C)n[nH]c2s1.C C(CNC(=O)C=Cc1cc[nH]n1)(CC(C)C)NC(C(CC)c1ccccc1)=O CN1C(=O)c2ccc(C(N3CC4(CCC4NC(=O)CCCF)C3)=O)cc2S1(=O)=O c1(C(=O)NC(CNC(c2c(C)con2)=O)C2CCC2)ccc2c(c1)OCO2 O=S1(=O)CC2CN(c3nc(NC4CCOCC4)c4ncsc4n3)CC2C1 N1(C(C2(OCC)CC2)=O)CC2(CC(NC(=O)C(C)C(C)O)C2)C1 C=CC1(CC(N2CCN(C(=O)C(O)CCC)CC2CCOCC)=O)CCOCC1 C1(NC(c2n(C)ccn2)=O)CN(C(C2SCCCS2)=O)CC2(CC2)C1 n1(CCCN(C(C(C)SC(F)(F)F)=O)C2CC2)cc(CN2CCNC2=O)nn1 c1(CC(=O)NCC2(C)CCN(C(C(F)OC)=O)C2)ccc2ncsc2c1 Cc1ccc(SCC(=O)NC(C)(C)C(C)C)cc1.c1(C=O)cnc(C(C)C)s1 c1(C(C(=O)NC2(C)CCN(C(c3nc(OC)oc3)=O)C2)C)cc2ccccc2s1 c1(N2CC(CC)N(C)CC2)nc(N(C)Cc2cc(Br)cs2)nc2cc(C)ccc12 N1(C(CCNC(N2CCC(NC(C)=O)C2)=NC)=O)CCCc2ccccc21 c1(C(N2CC(NC(C=C(CC)C)=O)C(C)C2)=O)ccc(Br)c(SC)c1 C1(NC(CCc2cc(C)on2)=O)CCN(C(=O)CN2CCN(C)CC2)C(C)C1 c1(C(=O)NCC2C(C(=O)NC(C)Cc3cccs3)C2)ccn(C2CC2)n1 C1(NC(COCC)=O)CN(C(c2c(F)ccc(F)c2F)=O)CC2(CCOCC2)C1 C(c1ccc(F)cc1)=CCC=O.Cc1nc(C)c(C(=O)NCCC(C)(C)C)o1.N C#CCC(C)(CC)C(=O)NCC1(CNC(C2(OC)CCOC2)=O)CCCC1 N1(C(C2C(OCC)C2)=O)CC(n2cc(-c3ccn(CC(F)F)n3)nn2)C(C)C1 C1(NC(c2c(C(C)=O)cn(C)n2)=O)CN(C(=O)C(C)O)C2(CCC2)C1 N#Cc1ccc(C(N2CCCC2CCCNC(c2ncccc2Cl)=O)=O)cc1Cl c1(CC)cnc(C=O)cn1.N1(C(C(=O)N(CC(C)O)C)C2CC2)CCOCC1.N CC(C)C(C)(O)C(=O)NC1CC(CCNC(c2c[nH]nc2C2CCOC2)=O)C1 CN(C)S(=O)(=O)NCC(N1CCCC(n2cc(C3CCCC(=O)C3)nn2)C1)=O c1(C(N2CC(NC(Cc3scc(C)c3)=O)C(C)C2)=O)ccnc2ccc(N)cc12 C1(CC)CN(C(=O)CCN(C)C(C)=O)CCN1C(=O)CC(C)c1ccccc1 N1(C(C2(N(C)C)CC2)=O)CCOC(CCCNC(=O)CSC(F)(F)F)C1 C1(C(N2CC3CC(C=O)(C3)C2)=O)CC2(C1)CC2(F)F.C1(CC)CCCCCC1.N C(CC(O)CC(=O)NCC(O)CN(C)C(C1(C(N)=O)CC1)=O)SC n1(CC)nc(C)c(C(N2CCC(O)(CNC(=O)C)C2)=O)c1C(F)(F)F C12(C(=O)OC)CCC(CC1Nc1cc(F)ccc1OC(C)C)C2 C1(NC(c2c(Cl)cnc(CC)n2)=O)CC12CCC(NC(=O)C(F)(F)CO)CC2 c1(C(=O)NCCN(C(=O)C(C)OCOC)CCC)ccc(-n2cncn2)cn1 c1(CCC(=O)NCC(CNC(C2CC(CC)C2)=O)(C)F)cncc(C)c1 Cc1cc(O)nc2cc(NC(=O)CC3CCC3)ccc12 Cc1cnc(C(=O)NC2CCCC2)c(C(F)(F)F)c1.C(=O)(C(C)C(F)(F)F)N Cc1ccn(CC(=O)NCC2CCC(C(=O)N(C)CCN(C)C)O2)c1 C(C)(C)(CC(C)N=c1[nH]c(N(CCC(C)C)C)nc(=N)[nH]1)OC C(CC(=O)N(C)CC1(CNC(C2(C)CCC2)=O)CC1)NC(=O)NC C1(NC(c2cnn(-c3ccncc3)c2)=O)CCC12CN(C(c1cnc(S)[nH]1)=O)C2 N1(C(C2C(=C)C2C(=O)O)=O)CC2(C1)SCCC2.n1(CCC=O)cc(Cl)cn1 c1(CNC(CCNC(C)=O)=O)cccc(C)c1.c1(CCC(=O)N)ccncc1 c1(C(N2C(CNC(C(N)=O)=O)C=CC2)=O)cc(C(F)F)ccc1F c1(CC(C)C(=O)NC2CC2C)cccc(Cl)c1.C1(C(=O)N)CC1.C1CC1 C(=O)(C(CNC(=O)CC(OCC)OCC)OC)NCCCC=C CC1(CO)CCN(C(C2C3CC4C(C3)C24)=O)CC1.C(=O)C(C)(C)n1ccnn1.N C(=O)(C(c1ccccc1)C(F)(F)F)NCC(CC)NC(C1(C(F)F)CCC1)=O C1(C(=O)NCCn2cc(CN3CCCC3)nn2)CCCOCC1 C1(C#N)CCCC1.C1(NC(C(C)OCCCC)=O)C(C(=O)NC)C1(C)C c1(C(N(C(C)C(=O)NC2CN(C3CCC3)C2)CCC)=O)ocnc1C c1(C(=O)NC(C2CCCCC2)CNC(C2(F)C(C)OCC2)=O)cnc2n1CCC2 c1(C(=O)NCC(CO)NC(C2C(OC(C)=O)C2)=O)ccc2nn[nH]c2n1 C1(CNC(c2nnc(C)s2)=O)CCC(C)N(C(C2CCOCC2)=O)C1 c1(C(=O)NCCCN(C(Cc2c(C)scc2)=O)C(C)C)ccc(NC=O)cc1 C(C1CCN(C(=O)C(C)CO)CC1)=CC(=O)NC(COC)(C)CCO CC(C)C(C)(C)C(=O)NC1CCCCN(C(c2nc(C3CC3)ncc2Cl)=O)C1 CCCC(C(O)C(=O)N(C)Cc1ccn(C)n1)NC(=O)C=Cc1cnn(C)c1 c12ccc(c(N)c1)C(=O)C2=O.C1(=O)CCCCN1.C(C(C)C)SC.CCO C1(NC(c2c(C)[nH]cc2)=O)CN(C(C2C3COCC23)=O)CC12CCS(=O)(=O)CC2 c1(CC(=O)NCC(F)CNC(C2CC2c2ccccc2)=O)ccccn1 c1(NC(C2SCCN(Cc3cccc(C)c3C)C2)=O)cc(Cl)c([N+](=O)[O-])cn1 C(=O)(C#CC1CCCCC1)N1CCC(NC(C(C)OCCOC)=O)CC(O)C1 c1(C2N(CCC)CCC2)nc(-c2cc(OC)ccn2)nn1CCc1ccccc1 N1(C(Cc2nc(C)sc2C)=O)CCC2(CC(NC(=O)CC(F)(F)C(C)C)CO2)C1 C12(C(=O)NCCC(C)NC(CCc3cncc(C)c3)=O)CC1CCC2(F)F c1(C(N2CCCC(C(C)NC(C3CC(F)(F)C3)=O)C2)=O)c(N)ccc(F)c1F C1(C(NOCCCCC)=O)COCCC1NC(=O)Cc1cccc(C)c1 C(=O)(CC(CC)CC(F)(F)F)N(CC(C)N(C(CCOCC#C)=O)C)C c1(C(N2C(C(CNC(COCC)=O)(C)C)CCC2)=O)cc2n(n1)CCCC2O c1(CN2CCC(CC(=O)NC(C(C)C)CCO)C2)c(F)c(F)c(F)c(F)c1F C1(CC)CN(C(C2(CC)CC2(F)F)=O)CCN1C(c1cncc(OC(F)F)c1)=O N1(C(C(C)(C)C)=O)CC2CC(NC(=O)C(C#N)CC3CC3)C(C2)C1 C1(C(C#C)C)CCN(C(=O)CCOCCNC(c2cc(OC)no2)=O)CC1 C(C(C)C)OC.C1(SC2CC2)CCCO1.C1C(OCCOC)CN1.O N1(C(C(CC#C)C)=O)CCC(C2CCN(C(=O)Cc3cc(C4CC4)on3)CC2)C1 c1(C(N(C2CCN(Cc3cc(F)cnc3Cl)CC2)C)=O)ccnc(F)c1F Cc1ccc(F)c(OCC(=O)NCC2CCCCN2C(c2[nH]c(C)nc2C)=O)c1 c1(CNC(c2c(Br)cc(C)s2)c2nnnn2C2(C)CC2)ccc2nc[nH]c2c1 c1(CC)ccc(C(=O)CCC=O)cc1.C1(CC)CN(C(=O)C(F)=CC2CC2)C1.N c1(C(N2CCN(C(=O)CCCCCO)C3(CC3)C2)=O)ccc2sccc2c1 C#CCC(C)(C(=O)N(C1CCNC1=O)C)NC(C1CCCN1CC)=O c1(C(=O)NC(CNC(C2(C)CC(C)C2)=O)(C)CO)cc(O)cnc1Cl CC1(C)CC(C)(NC(C2CCN(S(=O)(=O)c3cccnc3)CC2)=O)C(=O)O1 N1(C(C(CC)n2ccnc2)=O)CCOC(C)(CNC(c2cc(Cl)cn2CC)=O)C1 C=CC1COCCN1C(C1CCC(NC(=O)Cc2sccc2C)CC1)=O C1(C=O)CCC(S(C)(=O)=O)CC1.C(c1cnccn1)=CC(=O)NCCC.CC C1(C(=O)NC(CCC)C(=O)NCC(CO)OC)CCCC12CCC2 C1(NC(C2(C(=O)NC)CCC2)=O)CS(=O)(=O)CC1.c1(C=O)cnn[nH]1.N N1(C(c2n(CC)cc(Cl)c2)=O)CCCN(C(=O)CC2CN3CCC2CC3)C(C)C1 C1(C(NOCC)=O)(NC(=O)Cc2ccn(CC)n2)CCCCC1 N1(C(CC(CC)C)=O)CCN(C(c2ccc(Cl)c(N)c2)=O)CC(CO)C1 c1(OCC=C)ccc(Cl)c(C(=O)N)n1.C1(O)CCN(C(c2ncn(C)n2)=O)C1 c1(-c2cn(C(C3CCCCC3)C)nn2)ccc(C(NCP(C)(C)=O)=O)cc1 C(=O)(N=c1cc(-c2ccncc2)[nH][nH]1)c1ccc(C=O)s1 C(=O)(C(O)CC(F)F)N1CCC(C(C)(C)NC(CCC(=O)NCCC)=O)C1 c1(C(=O)NC2CN(C(CC(=O)OC)=O)C3C2C3)ccc(F)cc1C C(c1cccc(F)c1Cl)=CC(N1CC(NC(Cc2ccn(C)n2)=O)(CO)C1)=O C(=O)(CCC(F)(F)F)N(CC(CNC(C1N(CCC(C)C)CCC1)=O)O)C c1(C(=O)OC(C(C)OC)C(=O)OC)nc2c(C)cc(C)cc2s1 N1(C(C2C(C)C2C)=O)CCCC(C2CC2NC(c2ccc3n[nH]cc3c2)=O)C1 c1ncnn2c(Br)ccc12.c1(CC(=O)NCC=CC)ccc2c(c1)NC(=O)C2.N c1(CCC(N2CCC(F)C2)=O)ccc(F)c(F)c1.C1(CC)CC(C(=O)N)C1.C c1ccccc1S(C)(=O)=O.c1(OC)cc(NC(C2CC2C=O)=O)cc(Cl)n1.N c1(-c2onc(CN(C(c3cccc(C(F)(F)F)c3)C)C)n2)cc(F)ccc1F CCC(c1ccccc1)=CC(=O)NC1CC1NC(c1ccc(C)cc1O)=O n1(CCC(=O)N)cc(C#N)c(O)nc1=O.C1(C(N(C(C)C)C)=O)CC(CCO)C1 Cc1ncc(Cl)cc1C(=O)NC(C)CN(C(=O)C(C)Cc1cccc(F)c1)C c1(C(N2CCOC(C(C)C)C2)C(=O)NCCCSC)cnc2c(c1)CCC2 CC(O)CCC(=O)NCC1CCC(NC(=O)C(C)(C)O)C1 C=CC(C)(CC)C(=O)NCC1C=CCN1C(c1ccc(C)nc1OC)=O CC1CC(NC(c2ncccc2C(F)F)=O)CCN1C(C1CCNC1=O)=O C1(C)(C(=O)NCCCNc2cc(C(C)=O)ncc2)CCC(C)CC1 C1(NC(=O)CCc2ccc(Br)cc2)CC2CC1CN2C(C1(O)CC1)=O c1(-c2cn(C(CN(c3nnc(Br)n3C)C(c3c(C)nn[nH]3)=O)C)nn2)cncc(N)c1 c1(C(=O)NC(CCCC)CNC(=O)CC2CC(CC)C2)c(F)ccc2ccoc12 N1(C(C2CCC(N(C)C)CC2)=O)CC(C(=O)N(C)C)Cc2ccccc21 c1(C(=O)N)cc2c(cn1)COCC2.Cc1[nH]nc(Cl)c1C(=O)NCCOCC N1(C(c2cnc(C)s2)=O)CCCC12CCN(C(=O)CC(C1CC1)C1CC1)C2 S(=O)(=O)(C1CCCCC1)N1CCC(F)(C(N2CCCC(C(=O)OCC)C2)=O)C1 O=C1CC(Cc2nc(-c3nccn3Cc3ccccc3CO)cs2)C(=O)N1 Cc1ccc(C(=O)NC2CCC(Cn3cc(C4(O)CCC4)nn3)C2)cc1C N1(C(c2ccn(C(C)C)n2)=O)CCC2CCC(NC(=O)Cn3cc[n+](C)c3)C1C2 N1(C(C(n2ccc(C)n2)(C)C)=O)CCOCC1(C)CNC(=O)OC(C)(C)C N1(C(c2n(C)ncc2)=O)CCN(C(=O)Cc2cccc(O)c2)C(CF)C1 C1(N(C(C(COC)N(C)C)=O)C)CCCN(C(=O)CNC(c2ccco2)=O)C1 c1(C(=O)NCCCCCC)cnc2cccc(C)n12.C(=O)C=CC(=O)N(C)C.N c1(OC)ccc(CC(=O)NC2CCC(c3ccnn3C)C2)cn1 C1(C(NNC(C2CCOC2(C)C)=O)=O)CCCN2CCSCC12.CO c1(C(C)C)ccc(C(=O)NC(C2(O)CCN(C(=O)C(C)N(C)C)CC2)C)cc1F c1(C=O)cc(F)c(F)c(C#N)c1.CC(C)(C(=O)NCCC1CC1)c1ccns1 CN1CC(O)CCC1C(N1CCCC(N2CCOC2=O)C1)=O C(=O)(C(CCC1CC(F)(F)C1)N1CCCC1C(C)C)NC(CC)C C(CNC(c1ccccc1)=O)(C(C)(C)C)NC(C1CC(C)(F)C1)=O.CC#N CC1(CCC(=O)NCC=CBr)CCCN1C(C1CCC2(CC2)C1)=O CN(C)S(=O)(=O)N(C)CC(N1CC(NC(=O)C(C)(O)C2CCC2)CC1(C)C)=O N1(CCCN(C)C[Si](C)(C)C)CCC(F)(F)C(c2nn[nH]n2)C1 C1(C=O)CN2CCCC1CC2.C1(CC=C)(C(=O)NCC2(CC)CC2)CCCC1 c1(C(N(CCCCN(C)C)C)=O)nn(-c2ccon2)ccc1=O c1(N2CCN(CC(CC)O)CC2)cccc(S(=O)(=O)NCCCOC)n1 N=c1[nH]ccc(C(N2CC3CCOCC3(NC(=O)C3=CCSC3)C2)=O)c1[N+](=O)[O-] CN1CCOC(C(N2CCC(CCCNC(c3nocc3Br)=O)CC2)=O)C1 C1(CCCCNC(COCCC)=O)CCN(C(=O)CCNC2CCCC2)CC1 C12(NC(C3CCC3)=O)CCN(C(c3cccn4nncc34)=O)CCC1C2 C(=O)(C#CC1CCCC1)N(C1CCCCN(C(C(C)OCCOC)=O)C1)C C12(CNC(CC#N)=O)CCCC1CN(C(=O)C=CC(=O)NC1CC1)C2 c1(C(=O)N)cc2cc(F)ccc2cn1.C12(CNC(C(C=C)O)=O)CCC(CO1)C2 c1(C(=O)NC23C(CN(C(C4CCC(C)(C)O4)=O)C2)CC3)cc2ccncc2[nH]1 N1(C(C2=C(C)OCCS2)=O)CCc2ccc(C(=O)Nc3cnc(Cl)nc3)nc2C1 C(=O)(CC(COC)NC(c1cccnc1C)=O)N1CCC(CN(C)CC)C1 c1(CN(C)N2CCCNCC2)cccc2ccccc12 Cc1c(S(=O)(=O)N2CCC(O)C(C)C2)sc(C(=O)O)c1Cl CN1CC(C(N2CCCC(C)(CNC(=O)CCCC3CCC3)C2)=O)CCC1=O c1(C(N(CC)C2CC2)=O)oc(C(C)C)nc1C.c1(CC=O)ccc(Cl)cc1.C c1(SC)nc(C)c(CC(=O)NCC23CC2CN(C(=O)CC=C(Cl)Cl)C3)s1 C(=O)(CCCN=[N+]=[N-])N1CCC(C(C)CNC(C2CCS(=O)(=O)N2)=O)CC1 CCC(CC(=O)NC(C(=O)NC1(c2nocc2C)CC1)c1ccco1)SC N1(C(c2c(C(C)NC(=O)CCc3ccn(C)c3)noc2)=O)CCSC2CCC12 c1(CC(=O)NC2CCCC2NC(C2CC2(F)F)=O)ccc(CO)cc1 C1(CNC(C2ON=C(CC)C2)=O)CN(C(=O)CN2C(=O)CCC2=O)CC1(C)C C1(C)(C=O)CC2CCC(C1)S2.Cn1nc(CC(=O)NC(C)C(C)(C)C)cc1Cl.N C(C(COC)CC(=O)N1CC(NC(=O)Cc2n[nH]cc2Br)C(O)C1)OC C12(NC(=O)CCF)CCCCC1N(C(c1cc(-c3cccc(F)c3)no1)=O)CC2 O(N(CC)C(=O)C1(C(C)C)CCN(C(c2cc(C(N)=O)co2)=O)C1)CC c1(CCC(=O)NC2C=CC(CNC(c3cc(Cl)cs3)=O)C2)cccnc1F C=CC(C)(C)CC(=O)N1CCCC(CN(C)C(c2cc(COC)[nH]n2)=O)C1 O=C(CCCCc1ccccc1)NCCOCCCNC(C1CCCS1)=O Cc1nc(NC2CC(n3cncn3)C2)cc(N2CCOCC(C)C2)n1 Cc1nc(N(C)C)sc1C(=O)N(CC(C)N(C)C(c1cnn(CCF)c1)=O)C N1(C(C(CCC)=CCC)=O)CC(C(N2CCCC2CC2CCC2)=O)CC(C)C1 c1(C(=O)NCC(C2CCCCC2)NC(C2(C)C(C)C2)=O)c(Cl)cncc1Cl C12(C(N3C4CC(CNC(C(CC)(C)C)=O)C3CC4)=O)CCCCN1CCC2 c1(C(N2CC(C)N(C(=O)CP(C)(C)=O)CCC2)=O)cnc2ccc(F)cn12 C1(CCNC(c2nn(C)c(O)c2)=O)CCCN(C(C2(CO)COC2)=O)CC1 c1(C(N2CC(NC(C=Cc3c(C)ncs3)=O)C(F)C2)=O)cccc(S(N)(=O)=O)c1 N1(C(CCOCC)=O)CCC(CO)(NC(C23CCCC(C2)OC3)=O)CC1 Nc1c(F)ccc(C(=O)NCC2CCCN2C(C2(c3ccno3)CCC2)=O)c1F C1(NC(C2C(C(N)=O)COC2)=O)CCCCCN(C(c2n[nH]c3c2CCC3)=O)C1 N1(C(C2(NC(C3CC(C4CC4)=NO3)=O)CCCC2)=O)Cc2ccncc2C1 C#CC1(C(=O)NCC(CC2CC2)C(=O)NC)CCCC1 N1(C(CC(CC)CC)=O)CC2(CCCCN2C(=O)C(C2CCOCC2)OC)C1 C#Cc1cncc(C(C(=O)NCC(C)C)N(C)CC2CC2C)c1 c1(C(N2CC(CCn3cc(COc4ncccn4)nn3)C2)=O)ccc2c(c1)CC2 C(=O)(C1=C(Cl)CCCC1)N1C2C(NC(CCC(=O)NC)=O)CC(C2)C1 CC1CCCCC1C(=O)NCC(C1CCCC1)NC(=O)COCC(F)(F)F C1(C(=O)NCCCCC#C)CCN(C(=O)NC(c2ccccc2)C2CC2)CC1 c1(C(=O)NC2C3CN(C(CCc4ccc(C)cn4)=O)CC32)cc(Br)ncc1N(C)C C1(CC=C)(NC(=O)CC2(O)CCC2)CCN(C(c2sc(=N)[nH]c2C)=O)C1 Cc1cc(C)c(C(=O)NC2CCCCCN(C(C3CC3CF)=O)C2)cc1N c1(C(N2CCN(C(CCC(C)=O)=O)C(C#N)C2)=O)cc(S(=O)(=O)O)ccc1O c1(OCC)ccc(Br)cc1CN1CCN(C(c2ccn(C(F)F)n2)=O)CC1C C(=O)(C1=C(C)CCC1)N1CC(CC=C)(NC(=O)CC2CC(C=O)C2)C1.N C1(O)CC=CC1.c1(C(=O)NCC(C)(C)OCC(=O)N)cocc1C(N)=O c1(CNc2ccc(C(=O)NCCCC#C)nc2)c(Br)ccc(OC)c1F C1(C)CC(F)(F)CN1C(=O)CCn1nc(C)cc1C.C1(CCC)CC1C(=O)N Cc1nn(C)c(C)c1S(=O)(=O)N1CCC(CNC(c2cccc(F)c2O)=O)C1 N1(C(CC=CC=C)=O)CC2CCOC2(CNC(=O)CCc2cc(F)ccc2F)C1 C1(C(N2CCC(CC(=O)N(CC(F)Cl)C)CC2)=O)CCCC1C1CC1 C1(CNC(C2(N)CC2)C)CC12CCC(F)(F)CC2 c1(CC(N2CCN(c3ccccc3)C3=CS2=CC=C3)=O)ccc2cccnc2c1 C1(C(=O)NCC2CCC(C)N2C)CC(F)(F)CN1C(C1CCSCC1)=O CCCCCCC(C)C(=O)NC(C1CCCN1c1cc(C)ncn1)(C)C C1(NC(c2ccc(C(C)C)cc2)=O)CCCC(NC(=O)C(=O)NC(C)C)CC1 C#Cc1cc(F)c(C(=O)NCC(F)Cl)cc1F N1(C(CCC(=O)NCCC)=O)CCN(C(C2CC=C(C)CC2)=O)CC1CF c1(C(=O)NC2CCC(CCNC(CC=C(C)C)=O)C2)cnc2cnc(Cl)cc2c1 Cc1cc([N+](=O)[O-])cnc1C(=O)NC1CCCC1NC(C1CNC(=O)N1)=O N1(C(Cc2n[nH]c(=NC)s2)=O)CC(CNC(c2ccc[nH]2)=O)CC1(C)C N1(C(CCCOC)=O)CCN(C(c2cc(O)cc(N)c2C)=O)C2CCCC12 CC1(NC(=O)C(O)C2CCCC2)CN(C(=O)CC2(c3ccccc3)CCCO2)C1 C1(C2CN(C(=O)CC3CC4COCC34)C2)(NC(Cc2nc(C)oc2)=O)CC1 C(=O)(CC(O)C(C)C)NCCN(C(=O)CC(=O)N(C)C)CC C1(OC(c2c(C)cc(C3CC3)cc2)=O)CCC2(CCCC2)C1 c1(C(=O)NCCOCCNC(C(C)OCC2CC2)=O)cncc(O)c1 C1(CCCN(C2CCC(c3ccccc3)C2)C(C)C)COC(C)(C)O1 CC1CCN(C(C2CCCCC2)=O)C1C(=O)N1CCCO1 c1(C(C)C)cnc(CN(C2CCN(C(=O)C(N3CCSCC3)C)C2)C)o1 C1(NC(CCC=C(C)C)=O)CCCC12CN(C(=O)CS)C2.c1nnnn1C1CC1 C(=O)(C(F)CCC(C)C)N1CC(C(=O)NC(C2CC3(CCC3)C2)C)(CC)C1 N(C1CCCc2cc(C)ccc21)C(CSCC)=O.C1(S(C)(=O)=O)(C=O)CC1.N Cc1c(C(N2CCC(NC(=O)CCC3CC3)C(O)C2)=O)cccc1C(F)(F)F C=CC(F)(F)C(=O)NCC(C)CNC(C1C2CCCOC12)=O n1(CC(=O)NCc2cc(Br)cs2)c(=O)oc2ccccc12 CC1(C)CN(C(c2c[nH]ccc2=N)=O)C(CNC(C2CCOC2(C)C)=O)CO1 c1cc2ccccc2cc1C(=O)N(C(C1CC(C)(C)C1C(F)(F)F)=O)CC N1(C(C2C(C)CC(C)O2)=O)CC2CC1CCC2NC(=O)Cc1cnn(C)n1 c1(CCN2CCC(C(=O)NC3CCCC(O)C3)C2)nc2ncccn2n1 n1(CCOC)cccc(C(=O)N(C)CC2COCCN2C(=O)CC(F)F)c1=O Cc1ncsc1CNC(=O)C1=CCC1.C1(O)CN(C(C2COC(=O)C2)=O)C1 C1(CC=C)(C(N2CCC(N(C(=O)C=CC(F)(F)F)C)C2)=O)CCCCC1 CCC(C(=O)NC12CC1CN(C(=O)Cn1ccc(Br)n1)C2)C(C)(F)F S(=O)(=O)(CC(=O)NCCNC(c1ccccc1-n1cccn1)=O)N(C)C C(C(C)(C)CNC(c1cnns1)=O)N(C(c1cnc(S)[nH]1)=O)CC C(=O)(C(C)(CSC)NC(=O)Cc1nnc(-c2ccccc2OC)n1C)OC C(CS(=O)(=O)CC(=O)NC1(CC)CC1)OC.c1(C=O)cn(C2CCOC2)nn1 C1(NC(CONC(C(C)OC)=O)=O)CCCCCC1CO N1(C(C(F)OC)=O)CC(CO)C2(C1)CN(C(=O)Cc1cc(F)ccc1C)C2 C1(C2(NC(c3c(C(=O)OCc4ccccc4)scc3)=O)CC2)CCCCO1 C1C2CC1CN(C(C1C3C4CCC(C4)C13)=O)C2.C(C=O)(C(C)C)NC(C)=O.N c1(C(=O)NC(CC#C)C(=O)NC(C2CCCC2)CO)cc(C#N)ccc1N c1(C(=O)Nc2ccc(NC(C(CC)OCC)=O)c(C)c2)c(O)nnc2c1CCC2 S(=O)(=O)(c1cc(Cl)ccc1F)N1CC(C#N)C(NC(C2C3COCC23)=O)C1 C1(NC(Cc2cn(C)nc2)=O)CCC(O)CN(C(c2ccnc3c2CCC3)=O)C1 c1(C(N2CCC(CCNC(C3(OC)CC3)=O)CC2)=O)cc(Cl)c2ccncc2n1 c1(C(=O)NC(CNC(C2CN(C(C)C)C2)=O)C)c(F)ccc(Br)c1Cl c1(CC)cccc2c(CC(=O)N(C)CCN(C)C(C3CC(F)(CO)C3)=O)c[nH]c12 C1CC12CCN(C(=O)C=Cc1ccc(Cl)cc1)CC2.O=C1CC(C(=O)NC)CN1 N1(CC(=O)NC2CC(NC(COCCN(C)C)=O)C2)CCSC2CCCCC12 c1(SC)cccc(CCC2CCN(CC(=O)Nc3cncc(F)c3)CC2)c1 C1(CC)CN(C(c2ccc(C(F)F)cn2)C=O)CC(C)S1(=O)=O.CCC1CC1.N N1(c2cc(CCC)nc(Cl)n2)CCC2(CC1)CN(C(=O)C=CC1CCOCC1)C2 C12(C(=O)NC(C)CS(C)(=O)=O)CCC(CN(C(=O)CCCC3CC3C)C1)C2 c1(CC)c(C=O)cccc1F.c1(C(N(CC(C)C)C)=O)cccc(C2CC2)c1.N CC(C)(CCC(=O)NC(CO)C1(C)CC1)NC(=O)CCC1CCOC1 C1(NC(c2ccnc(CO)c2)=O)CC2CC(C1)CN(C(=O)CC1OCCCO1)C2 c1(C(N2C(C(=O)Nc3cc(OC)n[nH]3)CCCC2)=O)ccc(C#N)c(Cl)c1 c1(CC(=O)N(CCOCCNC(C(=O)NC)=O)C)ccccc1Cl.CC N1(C(COCc2ccc(C)cc2)=O)CCC2CCCC12C.C1(C=O)CN(C)C1.N CCCC(C(=O)N1CCOC(CC(=O)N(C(C)CC(N)=O)C)C1)NC(C)=O CCC(C)C(C(=O)NC1C=CCCCC1)N(C)C(c1cnc(NC)cn1)=O C(=O)(CCCC(C)(C)NC(c1ccc(C)n1C)=O)NCCC(COC)O N1(C(c2ccc3nc(OCCCC)sc3c2)=O)CC2(C1)OC1(CN)CC2(NC)C1 C(=O)(CC(C)(C)CCOC)N(CCC(=O)NC(CCC=C)C1CC1)C1CC1 N1(C(CN(c2ccc(C#N)cc2)C)=O)CC2CCN(C(=O)C(C)(C)C)C2C1.CO c1(OC)ccc(C(=O)C=O)cc1.C1CC12CCC2.C1(C)(C=O)CC(F)(F)C1.N c1(CC(=O)N(C(CNC(c2cncc(C(C)=O)c2)=O)C)C)c[nH]c2cccnc12 O=C1CCC(CC(N2CCC(C)C2)=O)(C(F)(F)F)CN1.C12(C=O)CC(CO1)C2 N(C)(C1CCc2c(OC)cccc21)C(c1nc(Cl)ccc1Cl)C(=O)NC(CC)C c1(C(=O)NCC(C)(C)C)cnc2c(c1)CCCO2.C1(C#N)(C(=O)N)CCCCC1 N1(C(C(=O)NCCC)c2cn[nH]c2)CCCCC1c1nccs1 CC1CCN(C(=O)CCC2CCN(C(=O)CCc3cnccn3)C2)CC1(C)C C(C)(C(=O)NC)(C1CCC1)NC(CC1CC(=C)C1)=O.C1CCCC1.C1CC1 CC1CN(C(c2sccc2C(C)(C)C)=O)CCC1NC(c1ccc(F)cc1N)=O C1(NC(C=Cc2n(CC)ccn2)=O)CCCC(NC(=O)CCS(C)(=O)=O)CC1 C(c1cccnc1C)=CC=O.c1(N2CC(OC)(C)C2)cc(C)nc(C(C)C)n1.N N1(C(C=CS(C)(=O)=O)=O)C2CCC1CC(NC(=O)C(O)Cc1ccccc1)C2 C(CNC(c1snnc1C1CC1)=O)(CCOC)NC(C(F)=CC)=O CCCC(O)CC(=O)NCCC1(NC(=O)C)CCC1.c1ccccc1C(C)C.O Cc1cc(C(=O)N(C2CC3CC2N(C(C2(O)CCC(C)CC2)=O)C3)C)ccc1Cl C1(NC(COc2ccc(C)cc2)=O)CCC(C)(C)CC1C.C12(C=O)CCC1C2 c1(NC(C2N(Cc3ccc(OC)c(C)c3)CCOC2)=O)cc(F)c(F)c(F)c1Br N1(C(c2c(CC)ocn2)=O)CC2(CC(CC(=O)NC(c3cc[nH]n3)C)C2)C1 C1(NC(C)COCc2ccccc2)CCC(C(=O)O)C(C)(C)C1 O=C(C1CCc2cccnc21)NC1(C2CCN(C(C3(O)CCC3)=O)C2)CC1 c1(CC)cccc(C(N2CC(NC(c3ccc(C)s3)=O)CC(C)C2)=O)c1N C(=O)(C(CO)C(F)(F)F)NC1(CC=C)CCN(C(c2ccc(=O)oc2)=O)C1 N1(C(c2ncncc2-c2ccc3c(c2)CCO3)=O)CCn2c(Br)nnc2C1 C1(O)CCOCC1.N1(C(C#N)CC2CC(NC(=O)C(=O)N3CCC3)C2)CCOCC1 c1(CCC(N2CC3(C2)OCC(O)C3O)=O)nc2cc(Cl)ccc2s1 C(=O)(CC(O)CNC(c1ccc(C)cc1)=O)NCC1CC(CC)C1 C(=O)(C(CCC1CC(F)(F)C1)N(C)Cc1nc(Br)cs1)NCCC C1(C(N2CCN(C(=O)Cc3ccoc3)C3C2C3)=O)CCC2(CCCC2)CC1 C#Cc1cncc(C(N2CCCC(CNC(=O)CN3CC4CC4C3)C2)=O)c1 c1(C(=O)NC(c2c(C)nccn2)C)cc2cnn(C)c2nc1Cl c1(C(=O)NCC2(NC(C3C(CC)C3)=O)CC2)ccc2c(c1)CCC2=O N1(C(C(C(C)C)OCC)=O)CCCCCCC1C(=O)NCCC1(O)CCC1 c1(CC(=O)NCC2C(CNC(CCCN(C)C)=O)C2)cccc(F)c1Cl c1(C(=O)NCC(CCCC)NC(c2sccc2F)=O)c(C#N)ncn1C C1(C(=O)OC)CCC(C)(C)N1C(c1ccccc1-n1ccnn1)=O C12(C(N(CCC)CC)=O)CC3CC(C(=O)N1)C2C3.C(=O)(C1=C(Cl)CC1)N C#Cc1ccc(CC(N2CCCC(NC(c3sccc3C(C)C)=O)C2)=O)cc1 N1(C(CNC(CC)=O)=O)C2CCC1CN(C(c1sc(C)c(C)c1C)=O)C2 N1(C2CN(C(=O)OC(C)(C)C)C2)CCC2(CCOCC2)C(NC(N(C)C)=O)C1 N1(C(C2CCCC(F)(F)C2)=O)CC2CCC(C1CO)N2C(=O)C=CBr CN1CC(O)CCC1C(N1CCOCC(NC(c2ccc(C(F)F)o2)=O)C1)=O c1(C(=O)OC)cc2c(nc1N1CCOC(C)C1)CCC2.C1(C(=O)N)CC2CC2C1 C(N=c1[nH]c(=N)[nH]c(=NC2CCn3nnnc3C2)[nH]1)c1cc(COC)on1 c1(C(N(CCCCC(=O)N2CCOCC2CC(N)=O)C)=O)cnn2c1OCC2 N1(CC)CCOC(C(N2CCCC(C(C)(C)C(=O)N(C(C)CCO)C)C2)=O)C1 CC1(NC(C2CCN(c3ccc(Cl)nn3)CC2)=O)CCCN(C(C2CC2F)=O)C1 C=C(C)CCCC(=O)NCC1(C)CCCN(C(C2CC(C)CO2)=O)C1 C(CC1=CCN(C(c2cnc(C(C)(F)F)s2)=O)CC1)NC(c1cc(C)no1)=O C1(CNC(=O)Cn2cncn2)CCCCN1C(=O)CCc1cnccn1 c1(OC)cc(C)ccc1C(C)NC(c1cc(Cl)sc1C)c1nnnn1C(C)C c1(N2CCCC(CC#C)C2)ccc(C)c(C(C)=O)c1 c1ncc(Cl)nc1C(N)=O.c1(C(=O)OC)cc(N2CCC(F)(C=O)C2)ncn1.N c1(C(CO)NCc2c(F)cccc2F)cccc(OC(F)(F)F)c1O CC1(CNC(=O)CCC2CCC(=O)NC2)CCCCC1.C(=O)(COC(F)F)N c1(C(N(CC(CC)NC(=O)C)C)=O)ccc(C2CCC(=O)N2)cc1.C(C)C.O N1(c2nc(C)cc(C(=O)NC)n2)CCCC2(NC(=O)C(C)CCOC)CCCC12 C(=O)(C1=CC2(CCN(C(c3ccn(CC#N)n3)=O)CC2)OC1)OC C(CC)(C(=O)O)NC(c1nc(COC)sc1)=O.c1cn(C2CCCC2O)nn1.C c1(C(N2C(CNC(CC)=O)CC(F)(F)C2)=O)c(Br)ccc(Cl)c1F c1(N2CCC(OC)(CO)C2)cccc(S(=O)(=O)NC2CCN(C)CC2(C)C)n1 CC1CN(C(c2cnc(S)[nH]2)=O)CC1CNC(C1(CN(C)C)CCCC1)=O c1(C(N2C(C(N(C)Cc3cn(C)nn3)=O)CCC2)=O)cnc[nH]c1=N CCCCC(C)CCC(=O)NCCCN(C(=O)C(C)CC1CC1)CCC C(N=c1[nH]c(=NCc2csc(C(F)F)c2)[nH]c2cc[nH]c12)c1c(C)cc(Br)nc1 C(=O)(CC(C)(C)C)N1CCC1.c1ccsn1.C(=O)(C)NC(C)C.CCO c1(NC(C(C2CN(C(=O)OC(C)(C)C)C2)OC)=O)cnc(Br)c(C)c1 N1(C(c2ccsc2OC)C(=O)NC)CCC(SCC)CC1C C1(NC(C(CC)F)=O)Cc2ccccc2C1NC(c1cnc(=N)[nH]c1)=O C(=O)(C1CCCc2scnc21)NC(CC(C)C)CNC(=O)C(C)C c1(CN2CCC(C(=O)Nc3cnc(C)nc3)CC2)cc(Br)c(O)c(Br)c1 C1(C2=CCCCCC2)(C(N2CCCC(C(C)NC(c3ccc(Cl)[nH]3)=O)C2)=O)CC1 N1(C(c2n(C)c(O)nc2)=O)CC(NC(=O)N)C2(COC2)C1.c1cnn(C2CC2)c1 c1(C(=O)NC(Cc2cn(CCOC)nn2)C(=O)OC)cc(=O)cc[nH]1 c1(C(=O)NC2CC(NC(CCC(C)OC)=O)C2)cc2c(C)ccc(Cl)c2[nH]1 C1(NC(CC=CC)=O)CN(C(=O)C[SH](=O)=O)CC2(CCC2)C1.C(C)(C)C.N C12(C(=O)NCCCNC(=O)NC)COC(C1)C(NC(=O)CCCC)C2.S C1(N(C)C)CC(C(=O)NC2CC(CCC(=O)NCCc3ncon3)C2)C1 c1(C(N(CCN(C)C(c2cnn(-c3nccs3)c2)=O)C)=O)cnn(C)c1Cl C1(NC(c2[nH]cc(CC)c2)=O)CCN(C(c2cscc2OC)=O)CC1F n1(CC)cc(C(F)(F)C(=O)NCC2(F)CC(C)C2)cn1.C(=O)CC(C)O CC(C)(O)C#CC(C)(C)NC(c1cc(C(=O)C(F)(F)F)c[nH]1)=O N1(CC(=O)NC2CC2)CCn2ccnc2C1.c1(C2C(C(=O)N)C2)ccc(Cl)cc1 c1(SCC)ccccc1C(N1CCCC1)=O.c1(C(=O)N)cc(C(F)(F)F)c[nH]1 C1(C(=O)NCC(C(C)C)NC(C2CCS2(=O)=O)=O)CCC(=O)NC1 N1(C(C(Cn2ccnn2)NC(C2CNC(=O)O2)=O)=O)CCC2(CCOC2=O)C1 C(c1ccc(F)cc1)=CCC(=O)NCC1N(C(C(N2CCCC2=O)C)=O)CC1 c1(CN2CCC(N)(CC)C2)ccc2c(c1)CCC(C)(C)O2 N1(C(C(CC)COC)=O)CCC2C(C1)CN2C(=O)CN(C)C(=O)C1CC1 CC1CN(C(c2ccc(-c3ccc(Cl)s3)cn2)=O)CC1NC(C1CCC(=O)O1)=O Cc1ccc2ncc(C(=O)NCC=CCNC(=O)CCn3cc(Cl)cn3)n2c1 C(c1ccoc1)=CC(=O)N(CCC)CCO.CC1CC1(c1cccs1)C(=O)N N1(C(c2c(CC)nccn2)=O)CC(F)(F)CC1C(=O)NC1CC1CC C1(CCOC)CCN(C(=O)CC)CC1.C1(CC(=O)N)CCCC1(F)F.C1COC1 CC1C(NC(c2cc(C3CC3)no2)=O)CC2CCC1N2C(=O)CCO.C1CC1 C#Cc1ccc(C(=O)NC2(CCOC)CCN(C(C3CC3F)=O)C2)o1 C(=O)(CCC1=CCCCC1)N(C1CCN(C(CCOCCOC)=O)CC1C)C Cc1cc(O)c(C(N2CC3(CCCC3NC(C3CC=CC3)=O)C2)=O)cc1Br N1(C(c2ccc(C)cc2Br)C(=O)NCCOC)CCCN(CC(=O)OC)C(=O)C1 c1(C(N2C(C)CC(NC(C3CC(=O)N3)=O)C2)=O)cnn2ccn(C)c12 c1(OC)cc(S(=O)(=O)NC(C)C)ccc1NC(C)CCc1ccc(Br)cc1 N1(C(c2cc(C(C)=O)c(C)o2)=O)CC(NC(C2CC23CCCC3)=O)CCC(O)C1 c1(C(=O)NC(CN(C(CC(=C=C)C)=O)C)C)ccc(F)c(C2(C)CC2)c1 c1(C(=O)NCC(C(C)(C)C)NC(=O)CN2CCCC2CO)cc(N)ccc1F c1(C(=O)NCC2CCN(C(C3(C=C)CCOCC3)=O)CC2)cc2cnn(C)c2s1 C(=O)(C1=CC(O)CC1)N1C(C)(C(=O)OC)CCC1.C(=O)CN(C)C(N)=O n1(CC)nc(C(F)(F)F)cc1C=O.CC(C)(O)C.C1(C=O)COC(=O)C1.N C12(NC(C(COC)(C)OC)=O)CCC(C=O)(CC1)C2.C1(CC)CCCC12CC2 C1(C(=O)NCCC(C)NC(=O)CC23CCC(CC2)C3)CCc2ccccc2C1 c1(C(N2CC(NCc3nc(COC)sc3)C2)=O)c(C)cc(F)cc1C C1(CC(=O)NCCNC(c2cnc(O)o2)=O)CS(=O)(=O)c2ccccc2O1 c1(C(=O)OC)cccc(-c2cn(CC3(O)CCN(C(=O)CCSC)C3)nn2)c1 c1(C(c2ccccc2F)NC(=O)NCc2sccc2Br)ccc([N+](=O)[O-])cc1 C1(C)CN(C(=O)CN2CCS(=O)(=O)CC2)CCO1.C(C)(C=O)N(C(C)=O)C.N CC1CCN(C(c2csc(O)n2)=O)CCN1C(=O)CCc1cc[nH]n1 N1(C(C(C)OC)=O)CC(CNC(c2sc(Br)nc2C)=O)C2(CC2)C1 N1(C(c2cc(COC)on2)=O)CC2CC(CNC(C3CCC4CC34)=O)C2C1 c1(C(=O)NCCC(C)N(C(CC(CC)O)=O)C)cc2c(cc1OC)OCO2 C1(C(N)=O)CCC(OC(=O)C2CC2)C1.N1(C(C)=O)CC2CC2C1 c1(C(N2CCC(NC(C(CCCCC)O)=O)CC2C)=O)ccc2c(c1)ncn2C C1(NC(c2cccc(Cl)c2Br)=O)C2(CCC2)C12CCC2 C1(CNC(C(CC)CC)=O)CCN(C(C2CCC(=O)O2)=O)C1(C)C C1(C(=O)OC)CN(C(C2COCCN(C(=O)OC(C)(C)C)C2)=O)CC(=O)N1 N1(C(Cc2nc(C)[nH]n2)=O)CC=C(C(=O)N(C)CC2CCCOC2)CC1 c1(C(=O)NCC(CC)(CC)NC(c2csc(Br)n2)=O)cnc(O)c(F)c1 c1(C(C(=O)NCCNC(C(C2CCOCC2)OC)=O)O)cnn(C)c1 C1(NC(c2sccc2Cl)=O)CCN(C(=O)CN2CCCNC2=O)CC1CO c1(C(=O)NCC(C2CCC2)NC(C2CCSCC2)=O)csc2ccc(F)cc12 C1(C(N2C(CC)CCCC2)=O)C2CC3C(C2NC(=O)CC2CCCC2)C13.O C1(C(=O)OC)CC(C(=O)NC2(CNC(=O)CC)CC2)C1.C1CCOC1 CC(C)(CC(=O)NCC1(C)CCCN1C(=O)C(F)=CC1CC1)C(F)F c1(OC)ccc(-n2cc(-c3csc(-c4nccn4C)n3)nn2)cc1OC CC(O)CCC(=O)N1CCOCC1CN(C(=O)CSc1ccccn1)C CCCC(CC)C(=O)NC1CN(C(c2ccc(Br)cc2OC(C)C)=O)C1 N1(C(c2c(C)ccnc2O)=O)CCC2(CCN(C(=O)C=CC3CCOC3)C2)C1 C1(C(=O)NC(CC)CNC(=O)CCCN(C)C)CCCC(C(=O)OC)C1 c1(C(=O)NC(CCNC(C(CCOC)C)=O)C(C)C)ccc(F)c(Br)c1 C1(C2(O)CN(C(C3(C)CCOC3C)=O)C2)CC1.c1(COC)cc(C=O)on1.N N1(C(C2CC3C(C2)C3(F)F)C(=O)NC(CC)C)CCC(O)CC12CC2 N1(C(C)=O)CCOC(C(=O)NCC2CC2NC(=O)CCCn2cccc2)C1 N1(C(c2c(CC)cc(F)cc2)=O)CCC2CN(C(C3CC4(CC4)C3)=O)CCC2C1 N1(CCOC)CC(NC(c2ncccc2OC)=O)CCC1C c1(C(=O)NC2(CN(C(=O)CC3CCCOC3)C)CC2)c(N)cc(Cl)nc1Cl c1(C(=O)NCCN(C(=O)CS)CC)ccc(C)c(OC)c1F.c1ncc[nH]1 CCC(C)(COC)C(=O)NCCSCC(=O)NCC1CCC(=O)NC1 C1(C(N2CC(NC(=O)OCC)C2)=O)CCC12CCC2.C(=O)CC1CC1 c1(SCC)c(C(=O)NC(C)CNC(=O)C(C(C)C)OC)sc2ccccc12 c1(C(N2C(CC)CCC2)=O)ccc(S(C)(=O)=O)s1.c1(CC=O)ccc(F)cc1 S(=O)(=O)(c1cc(F)ccc1C)NCCC(=O)Nc1ccc(C)nc1CC1CC1 C1(C(=O)NCC(C)NC(C2CC(O)CN2C)=O)C2CCC1(c1ccco1)C2 C(=O)C=CS(C)(=O)=O.c1(CN(C(C)C)C)cn(CC2C(C)C2(F)F)nn1 N1(C(C=CSC)=O)CCCC(O)(CCNC(c2sccc2C(F)F)=O)C1 c1(N(CC(=C)C)C)cc(Br)ccc1S(=O)(=O)N(C)C(c1cnn(C)c1)C Cc1cnoc1C1(C(=O)NCC(C)N(C(=O)Cn2cccc2)C)CC1 C1(NC(CN2CCN(C(C3=C(C)OCC3)=O)CC2)=O)C2CCCC1COC2 c1(OC)c(C(N2CCCC(CC(N3CCCC(O)C3C)=O)C2)=O)cccc1Br c1(C(N2C3CN(C(C(=O)C4CC4)=O)C(C3)C2)=O)ccc2c(n1)OCCO2 Cn1cnc2nc(=NCCOC3CCS(=O)(=O)C3)[nH]c(NCCO)c12.C1CC1 c1(OC)cc(C(N2CCCC2CCNC(C2CC2C2CCC2)=O)=O)ccc1Cl c1(CC)ncc(-c2noc(-c3cnc(OC(C)C)cn3)n2)c(=N)[nH]1 c1(C(=O)NCC(C)OC)cc2c(nn1)CCC2.C1(C=O)CC(N2CCCC2)C1 c1(C(=O)NC2C=CCN(C(c3cc(O)ccc3Cl)=O)C2)c[nH]c2nc(Cl)ccc12 N1(CC(=O)N(C2CCCCC2O)C)CCN(C(C2CCC(C)(C)C2)=O)CC1 CC1(C(=O)O)CC(O)CN1C(=O)CCn1cc(CC2(O)COC2)nn1 CC(C)(C)C(CNC(C1CCC2(CC2)C1)=O)NC(C1(CCF)CC1)=O c1(SCC)cnc(O)c(C(=O)N)c1.c1(C(N2CCC2)=O)sccc1C(C)=O C(C(=O)NC1CC(C)CCC1O)(C(C)(C)O)NC(c1c(C)cc(CC)o1)=O C(C)(C)(CC(=O)NC(C(N)=O)C1CCCC1)NC(CSCCOC)=O Cc1cc(C)c(C(=O)NCC2C=CC(NC(=O)CN3CCCNC3=O)C2)cn1 C12(C(N(C3CCN(Cc4ccc(F)cc4)CC3)CCC)=O)CC=CCN1CCC2 c1(NC2CN(C(C(c3ccccc3Cl)OC)=O)C(C)C2)cccc(F)c1[N+](=O)[O-] CC1(C)CCCN(C(C2Cc3ccccc3C2)=O)C1C(=O)NCCn1cccn1 C1(NC(C(c2ccccc2Cl)N(C)C)=O)CC2CC(NC(=O)C3=CCSC3)CC12 O=C(C(C1=CCSC1)N1CCCC2(CCC2)C1)NCSc1ccccc1 Cc1c(C(N2CC3C(C(=O)O)C3C2)=O)[nH]c2ccc(NCCCS(C)(=O)=O)cc12 C1(NC(CNC(=O)NC)=O)CCC(N(C(=O)CCn2cc(Cl)cn2)C)CC1 CC1CCCn2c(CC(=O)N(C)CCOCC)cnc21.C1(C(=O)N)CCC(=O)C1 C1(C(N(CCNC(c2c(C#C)c[nH]n2)=O)CCC)=O)CC1C1CCCC1 c1(CCCC(=O)OC)n[nH]c(=NC(=O)NC2CC(=O)N(c3ccc(Cl)cc3)C2)s1 C(=O)(C1=CCN(C)C1)NCC(CN(C(C=C=C(C)C)=O)C)(C)C CS(=O)(=O)c1ccc(Sc2ncc(C3CC3)c(O)n2)s1 c1(OC(C)C)ccc(Cl)cc1C(=O)NC.C(=O)(CCCC(F)F)N1C(C)CCC1 c1(OC)ccc(C(=O)NCC(C)C2CCC2)c(C)n1.C(=O)CCc1ccoc1.N Cc1onc(C(N2CCC(N(C)C(C3CC3c3cnc[nH]3)=O)CC2)=O)c1[N+](=O)[O-] c1(C(=O)NC2(CC(=O)Nc3nccs3)CCC2)n[nH]c2cccnc12 Cc1nnc2ccc(C(=O)NCC(C)(CO)NC(=O)C(F)CC3CC3)cn12 Cc1cccc(CC(=O)NC2CCCCC2Nc2nccc(C(C)(C)C)n2)c1 N1(C(COC)=O)CCn2cc(C(=O)NCC(Cc3cccs3)CO)nc2C1 c1(CC)sc(=N)[nH]c1C(=O)NCCC1CCCCN1C(c1ccncc1F)=O N1(C(c2cnc(C)nc2C)=O)CCC2CC(C(=O)NCCN3CCOCC3)C2C1 CC(C)(C)CC(=O)NC1CCC(NC(C2(Oc3ccc(F)cc3)CC2)=O)C1 c1(N2CC(C)NC(=O)C2)nc2c(c(=NCC(=O)NCCON)[nH]1)CCCCCC2 c1(C(=O)NCCN(CCC)C(c2ccnc(C)c2)=O)n[nH]c(C)c1C C(=O)(C(C)(C)CF)NCC(C)CNC(=O)C(CO)NC(N)=O C1(C2CC2)(CNC(=O)NC2(c3ccc(O)nc3)CC2)CCOC1 C1(C(=O)NCC2C(CC(=O)NCCC(C)O)C2)CC2(CCCO2)C1 C1(CC=C)(NC(c2cn[nH]c2)=O)CCCN(C(c2sc(OC)nc2Cl)=O)C1 N1(C(C2(C(N)=O)CC2)=O)CC(NC(C2CC(=O)N(C3CC3)C2)=O)C(O)C1 c1(C(=O)NCC(CCCC)NC(=O)C(C)(C)CN(C)C)ccn2ccnc2n1 c1(CC)nn(C)cc1NC(c1csc(C(F)F)n1)=O N1(C(C(C)SCc2ccccc2)=O)CCN(C(=O)CC2=CCCC2)C(C)C1 C(CC(C)C(=O)NC1(CNC(=O)Cc2ccns2)CCOCC1)=CC c1(C(=O)NC2CC(CCNC(CN(CCC#C)C)=O)C2)cnncc1C C1(C(N2CC(CNC(c3n(C(C)C)cnc3)=O)C(O)C2)=O)Cc2nccn2C1 C(=O)(CC(O)C(C)C)N(C)CC1CCN(C(C(CC=CCC)C)=O)CC1 N1(C(CC2N(C(C(F)=CCC)=O)CCC2)=O)CC(=O)NCC1C c1(C(N2CCC(N(C(c3ncsc3C)=O)CC)CC2)=O)nc2nc(C)ccn2n1 CON1CC(C(N2CCC(CC(C)NC(C3C4CN(C)CC34)=O)CC2)=O)CC1=O C(=O)(CC(C)(C)CC(F)(F)F)NC1CCCN(C(CC(CC)C)=O)CC1 C(=O)(CCC(C)(C)C)NC1(C(=O)Nc2cn(CC(C)C)nc2)CC(F)C1 c1(C(=O)NC(CC)(C)CNC(=O)C(O)C2CCCC2)[nH]cc(C)c1C C1(C2CCCCC2)(C(=O)NC2C(NC(COc3cc(C)on3)=O)CCOC2)CC1 c1(C(N2C(CNC(c3c(O)ncc(CC)c3)=O)C=CC2)=O)ccn2nncc2c1 Cc1cc(N(C)Cc2cccc(Cl)c2)nc(NC2CCN(C3CCOCC3)C2)n1 c1(OC)cnc(C(N2CCC(F)(CNC(C3CC34CCC4)=O)CC2)=O)cn1.O CC(C)(CC(=O)N1CCC(NC(=O)Cc2csc(Cl)n2)C(C)(C)C1)C(F)F C1(C(=O)NCc2c(C)csc2)CN(C(=O)CCC(C)CN(C)C)CC(C)(C)C1 c1(OC)cccc2c1NC(=O)CN2C(c1ccc2ccccc2n1)=O c1(N2CCC(NC(c3ccc4nc[nH]c4n3)=O)CC2)nc(Cl)nc2c1CCC2 c1(CC(=O)NCCNC(C2(F)CC=CCC2)=O)ccc(F)cc1F.C1CC1.C C(CO)(C(=O)NCc1nnc(CO)s1)NC(C(C)C)=O c1(N(CC(CN(C)C(c2coc(C3CCCCC3)n2)=O)O)C)cncc(Cl)n1 C1(NC(c2nc(CC)oc2)=O)(CO)CCCN(C(=O)C(C)C2CCCO2)C1 C1(C(N2C(CN(C)C(c3ocnc3C3CC3)=O)CCC2)=O)C2CCCCC12 CCC(O)CC(=O)N1CC(OC)CC1C(N1CCC1C1CCCC1)=O C1(C(=O)NC(CNC(Cc2ccc(OC)nc2)=O)(C)C)CCC2(CCCC2)CC1 C(CO)(CCCCNC(=O)CN1CCCC1C)NC(c1c(CC=C)cccc1)=O C=CCC(C(=O)NCCC1CN(C(c2cccc(NC)n2)=O)CCO1)NC(C)=O N1(C(=O)CN2CCCCC2)CCC2CCN(C(C3(CC(F)F)CCC3)=O)CC12 C1(C(=O)NCC2(NC(C3C(CC)CCO3)=O)CC2)CC2(CCCCC2)CO1 CCCC(C)C(C)(c1nnnn1C1CCCC1)NC1(c2ncccc2F)CC1 c1(C(=O)OCC)csc(C(C(=O)NCCCF)N(C)Cc2cc(Br)cs2)n1 CC(C)CC(F)C(=O)N(CC(O)CN(C(=O)CSc1cccc(F)c1)C)C c1(C(=O)NCCn2cc(C(=O)NC(C(C)C)(C)C)nc2)c[nH]c2cnccc12 c1(CNC(=O)C(=O)N2CCC2C2CCOC2)nnc2n1CCCCC2 C(=O)(CCC(F)(F)F)NC1CCC(CCNC(c2ccn(CCCC)n2)=O)C1 C(=O)(CC(C)CC(F)(F)F)N1CCN(C(CCSCCC)=O)CC1CC(C)(C)C C=CCC(CNC(=O)OC(C)(C)C)C(=O)NC(c1ccccn1)C(F)F Cc1n[nH]c(C)c1C(C)CC(=O)NCC1CN(C(=O)CC2CC=CC2)CCO1 CCCCC(O)C(=O)N1CCC1CNC(c1cn(Cc2noc(C)n2)nn1)=O c1(N(C)C)nc2cc(C(=O)NC)ccc2o1.C(=O)C(O)C1CC1.C1(CC)CC1 CC(C)CC(C)CC(=O)N1CCN(C(c2cc(C#N)no2)=O)C(CCO)C1 C1(CCC)CN(C(C2(F)CCN(C(c3nonc3N)=O)C2)=O)CCO1 N1(C(c2ccc(SC)cc2)=O)CCC(N(C(=O)Cc2ccsc2)C)C(C)C1 c1(OC)cnc(F)c(C(N2CC(OC)CC(NC(=O)CCC3CCOC3)C2)=O)c1 Cc1cccc(C(=O)C(=O)NC2CC(C)(NC(c3cnn(C)c3F)=O)C2)c1 c1(OCC)ccc2c(c1)C(NC(=NCC(C)C)NCc1cccs1)CCO2 CC1(C)CCOC1CNC(=O)Nc1ccccc1C1CC1 c1(C(=O)NC2CCN(C(c3cn(CC)nc3)=O)C2C)cc2n(n1)CCNC2=O N1(C(c2c(CC)nc[nH]2)=O)CCOCC(CNC(C2CC(SC)C2)=O)C1 CC1CCc2nc(C(N3CC(NC(c4cnn(C(F)F)c4)=O)C3)=O)cn2C1 C1(C(=O)NOC(C)C)(CC=C)CCCN1C(=O)CC1(C)CCOCC1 c1(C(=O)NC(CNC(C2CC(C(C)C)C2)=O)C2CCC2)ccc2nn[nH]c2n1 C(=O)(CCC(F)(F)Cn1cc(CNS(N)(=O)=O)nn1)N(C)CC1CCCC1O C1(CNC(CC=CCC)=O)CN(C(c2cc(CC)cc(Cl)c2)=O)C2COCC2O1 N1(C(c2oc(C(=O)OC)c(C)c2)=O)CC2CCN(C(=O)CC3CCC3)C2C1 Cc1cncc(CCC(=O)NC2CC(NC(=O)COc3ccc(F)cn3)C2)c1 C=Cc1ccc(C(=O)NC2CC(C)N(C(c3cnn(C4CCC4)c3)=O)C2)cc1 Cc1c(C(N2CC(C(=O)Nc3cncnc3)C2)=O)cc(F)cc1Br c1(NC(C2(COC)CN(C(C3CCCC3)=O)C2)=O)cncc(C(N)=O)c1 C1(CNC(C2(CO)CN(C(c3cnc(OC)nc3)=O)C2)=O)CCC=CCCC1 C(CC(C)(O)CNC(C1CC2CCC1O2)=O)OC c1(C(=O)NCCC(C)NC(c2cnsc2)=O)ccc(F)c(N)c1F Cc1nn(-c2ccccc2)cc1C(=O)NC(C(=O)O)C(C)C N1(C(c2cnc(C)s2)=O)CC(C)(C)OCC1CNC(c1cc(N)c(F)cn1)=O C1C=CC(C)(C)CC1.c1(COC)cc(C(=O)NC2CCCC2C(=O)N)n[nH]1 Cc1sc(C(=O)N(C2CCCCC2)CCNC(=O)Cc2ccccc2O)nc1O C(=O)(CCCS(N)(=O)=O)N1CC2C(CNC(c3cnc(CC)[nH]3)=O)(C2)C1 c1(C(N2CCC(C3N(C(c4c(C)scc4)=O)CCC3)C2)=O)cc2ncccn2n1 C1CCC12CCN(C(C1CC1C(C)C)=O)CC2.c1(SC)ncc(C(=O)N)c(C)n1 C1(C(=O)NCC2(C#C)CCC2)CC(O)CN1C(=O)C(O)CN1CCCC1 CC(CCC(C)(C)C)NC(=O)C(CC1CC1)NC(C1CC=CCC1)=O c1(CC(c2ccccc2)=O)ccc(-c2ccc(F)cc2)cn1 C(C(C)(O)CC(=O)NC1CCCCC1NC(C1CCN(OC)CC1)=O)OC CC1(C)CCC(C(=O)NCCC2CCC2)C1.c1(C=O)cccc(C2CCC2)c1.N C1(NC(C(C)(C)F)=O)CCC2CN(C(c3ccc(C#N)s3)=O)CCC2C1 c1(CC(=O)NC2CCN(C(=O)CCc3ccncc3)C3CC23)ccc(Cl)c(F)c1 C1(NC(CCN(C(C2CC(N=[N+]=[N-])C2)=O)CC2CC2)=O)CCn2cncc2C1 c1(OC)ccnc(C(=O)N(C2CCN(C(=O)CC3(C)CCOC3)C2)C)c1O N1(C(C2(SC)CC2)=O)CC2(CCN(C(C3CCCN3c3nccs3)=O)C2)C1 c1(C(N2CCC(NC(=O)Cc3ccc(Cl)c(Cl)c3)C2)=O)cccc2c1CCOC2 Cc1ccc(C(=O)NCC(C(=O)N(C2CC2C)C)N(C)C)c(F)c1 C1(C(=O)NCC(CC=C)NC(C2(c3ncco3)CC2)=O)C(C)(C)C1(F)F c1(CC)cn2c(n1)CC(C(=O)NC1(C)CC1)CC2.c1(C(=O)N)cnccc1 Cc1c(CNC(N2CCOCC(C(=O)N(C(C)C(C)C)C)C2)=O)cccc1F c1(C(=O)NC(c2ccccn2)C(C)C)cccc2c1CN(C(=O)C(O)CCl)CC2 Cc1ccn(C)c(=O)c1NC(=O)NCC.c1nc(Cl)c(Cl)cc1C(F)(F)F C1(C(N2CCC2)=O)CC2(CCC2O)C1.N(C(C(=O)N)=Cc1cccs1)C(C)=O.C C1(NC)CCCCC1C(=O)NCC1CC1.c1(C=O)ccncc1.C(C)=O.C N1(C(Cc2c(OC)cccc2)=O)CC2CCCC(C1)N2C(C1CCCCC1C)=O C12(CNC(CC3(OC)CCC3)=O)CCC1CCN2C(=O)C(F)F c1(C(O)CN2CCOCC2)ccc(C23CNCC2C3)cn1 Cc1cccc2cc(C(N3CC(NC(=O)C(C)N4CCC4)CC(C)(C)C3)=O)[nH]c12 C1(C)(C(=O)NCCC(C)(C)NC(c2nc(C(C)(F)F)cs2)=O)C=CCCC1 c1(CSC(COCC)C)nnc(-c2ccc(Br)o2)o1 C(=O)(C1=CS(=O)CCC1)NC(C)(C)CCNC(c1cnn(CC(F)F)n1)=O c1(C(C)C)ccccc1C(=O)N(CC(O)CN(C)C(c1occc1F)=O)C c1(C(=O)Nc2c(C)cc(-c3c[nH]nc3C(F)(F)F)cn2)nc2cccnc2s1 C(CC)(C(=O)N1CCCC1C(C)(C)C(=O)NCC(C)Cc1cn[nH]c1)=CCCC O=C1CCC(CC(N2CC(CNC(c3cnsn3)=O)C(O)C2)=O)CN1 CCC(C)C(O)CC(=O)N1CC(OCCC(N2CCCC2C(C)(C)C)=O)C1 c1(N(CC(C2CCC2)OC)C)cccc(S(=O)(=O)N(C)Cc2nncn2C)n1 C12(C(=O)NC3CN(C(CCCCSC)=O)CC3O)CCC(C(F)F)(CC1)CC2 C#CC1CN(C(=O)C=C(C)C)CCN1C(=O)CC(C)COC C(N=C(NC1CCCCC1)N1Cc2ccccc2C(F)(F)C1)C1S(=O)(=O)CCC1 C1(OCC)CCCN(C(=O)CCC2(C)CN(C(C3(C)CNC(=O)C3)=O)C2)CC1 c1(CCC)ncc(C(N2CCOCC(NC(=O)OC(C)(C)C)C2)=O)c(C)n1 c1(C(=O)NCCCN(CCCCNC(C2C(C)CCO2)=O)C)cccnc1S C1(NC(C2CCC(C)(C)C2)=O)CC2CCCC(C1)C2NC(C1CC(O)C1)=O C#Cc1cncc(C(=O)NCC2CCN2C(c2ccc(C(N)=O)o2)=O)c1 C(C)(CSC)(C(=O)NC(C)C(=O)NC1CC1)NC(CN(C)CC)=O c1(C(=O)NCCC2CCN(Cc3c(C)noc3)C2)c(Cl)nc2ccccn12 C12(OC)CCC(C(=O)NC3CCC(O)C3)(CC1)C2.c1nncs1.C(=O)C.C c1(C(N2CCC(NC(CCC(=C)Cl)=O)C(C)(C)C2)=O)ccc2c(N)nccc2c1 C1(C(C)C)C(NC(=O)CCC2CCC(=O)NC2)CCN1C(c1cc[nH]n1)=O C(=O)(C(CN=[N+]=[N-])NC(=O)CCc1ccn(C)n1)N1CCN(CCC)CC1 CC(C)C(CNC(=O)C(c1cncn1C)O)C(=O)NCCCc1cncnc1 C1(C(=O)NCC(COC)(F)F)(NC(=O)CSC(F)F)CCCCC1 Cc1cc(C(=O)NC(Cc2ccoc2)C(=O)NCc2ccncc2Cl)nn1C CCC(C)(C(=O)NCCC1CC1)OC.c1(-c2scc(C=O)n2)ccc(O)cc1.N C(CN=C(NCc1cccc(Br)c1C)NCC1CCOC1)c1nnc(C)s1 c1(C(=O)NCc2c(OC)nccc2)ccc2c(c1)CN(C(=O)C(O)C(C)C)C2 C1(NC(c2cc(Cl)cnc2O)=O)CCCN(C(C2(CC(F)F)CCC2)=O)CC1 Cc1cc(C(=O)NCCOCCN(C(=O)CCCc2ccsc2)C)ccc1O C(C)(CSC)(C(=O)N(CC(C)C(C)C)C)NC(C(CC)N(C)C)=O N1(C(c2c(C)noc2)=O)CCC2(CC1)CCN(C(c1cc(C)n(C)c1)=O)CC2C Cc1cc(N2CCN(C)C(C)(C)C2)ncc1S(=O)(=O)N(CCCn1ccnc1)C Cc1cnccc1C(c1nc(-c2cncs2)nn1CC1CCCCO1)C N1(C(C(CSC)O)=O)CC2(CCCC2)C1C(=O)NCc1ccncc1F C(CCC(C)(C)C(=O)NCCCC1CCCCO1)NC(C=CC=CC)=O C1(CC=O)CC2C=CC1CC2.N1(C(C=CCN(CC)CC)=O)CCC(O)C1 C1(C(N2C(C(N3CCC3)=O)C=CCC2)=O)Cc2nccn2C1 C1(C(=O)NCCN(C(=O)COCCc2cccs2)C)(CSC)CCC1 CC(C)(C(=O)N1C2CCC1CN(C(C13CC(C1)C(C)(C)O3)=O)C2)C(F)(F)F Cc1c(-c2ccc(C(=O)NCC3(C)CCN(C)CC3)nc2)cccc1F S(=O)(=O)(c1cccc(C(=O)N)c1)N(CC)CC.C1CN(C(=O)CC)C1.C Cc1c[nH]c(C(N2CC(O)(CNC(C3(C)CCOC3C)=O)C2)=O)cc1=O Cc1cc(=NC(=O)C(=O)NCCN(C(c2sc3nccn3c2C)=O)C(C)C)[nH]o1 CC(C)CCC(=O)NC(C1CCN(C(c2cc(F)c[nH]2)=O)CC1)C C(=O)(C(C)C(O)CC(C)C)NC(CC=C)CC(=O)NC1CCOC12CCCC2 N1(C(c2ccc(C)s2)C(=O)NC2CCOC2)CCC(C2CCCOC2)CC1 CC1CCC(C(=O)NC(CC2CC2)C(=O)NCC2CSCCO2)CC1 C1(C2CCCN(C(=O)C3=CCS(=O)(=O)C3)C2)CC1.c1noc(C=O)n1.COC c1(C(=O)NCC2C(O)C(O)CN2C(=O)C=C(Cl)Cl)oc2ccccc2c1Cl C1(CC(=O)NCC(C)CN(C(=O)CN2CC=CC2)C)CCCN1C c1(C(=O)NCCCN(C(CNC(CCC)=O)=O)C)cc(Br)c(O)nc1C CC1=NOC(C)C1C(N1CC(NC(c2ccccc2)=O)C(C)C1)=O N1(CC)CC(NC(C2CCCN(C(C3CC4(CC4)CO3)=O)C2C)=O)CCC1=O C(=O)(C(O)C(C(C)C)OC)N1C(CC(N2C(CC)CCC(C)C2)=O)CCC1 N1(C(C(C)OC2CCCCC2)=O)CC2(CC(NC(C3CC4(CCC4)CO3)=O)C2)C1 CCC(C)CONC(=O)NCc1cnsn1 C12(C(=O)NCC(C(C)C)NC(c3sccc3CC#N)=O)CCCCC1C2(F)F c1(C(=O)N)noc2ccccc12.CC(C)CCCNC(=O)C(C)OCC(F)(F)F C#CC1CCN(C(c2nc(CNC(C3(C(=O)OC)CC3)=O)oc2C)=O)CC1 C(=O)(C(C)S(N)(=O)=O)N1CCC(OCCCNC(c2n[nH]c(C)c2O)=O)CC1 N1(C(C(C)=C2CC2)=O)CCN(C(C2Cc3nccn3C2)=O)C(c2ccnn2C)C1 N(C=O)(C1c2ccccc2OCC1F)Cc1snc(CC)n1 c1(OC(C)C)cncc(C(=O)NCC(C(C)(C)C)NC(=O)CN(C)C)c1 c1(CC)nc(C)sc1C(=O)NCCN(C(=O)C(CO)N(C)C)CC N1(C(C(COC)C)=O)CC(C)(C(N2CCN(C3CC3)CC2)=O)CC1(C)C C(C(C)S(C)(=O)=O)NC(C(C1CC1)SC)=O.c1(CC=O)n[nH]c(C)n1.N C1(CCC)CN(C(C2CCCS2(=O)=O)=O)CCN1C(=O)CC1(CO)CC1 c1(C(=O)NC2(CNC(C3CCC3C)=O)CC(OC)C2)ccn(C)c1C C(=O)(C#CC1(C)CCCO1)N1CCC(N(C(CCSC)=O)CC2CC2)CC1 C1(C(=O)NC(C)(C)CNC(=O)Cn2ncnn2)CCCC(F)(F)C1 C1(CNC(=O)CC2CCCOC2)CC2CN(C(=O)CCOC3CCC3)CC12 N1(C(C2C(C(=O)OC)C2)=O)CCCC(NC(C2(O)CCCC2)=O)C1C CC(C)CC(C)C(=O)N1CCCCC1c1nnc2n1CCC2 N1(C(c2[nH]n(C)c(=O)n2)=O)CC2CN(c3ccc(C(F)(F)F)cn3)CC2C1 O=C1NCc2ccc(C(=O)NCC3C4CN(C(c5ccc(F)o5)=O)CC34)cc2N1 C1C#CCCCCC1.N1(C(COCCC(C)C)=O)CCOCC1CNC(=O)CO c1(COC)cc(C(=O)NCC2OCCC2C(=O)NCC(C)C)no1 C1(C)(C(N(CCOC)CCNC(C2CC2C(N)=O)=O)=O)CCOC1 N1(C(C(=Cc2cncn2C)S(C)=O)=O)CC2CC2C1.C1(C=O)(CC2CC2)CC1 N1(C(C2(CC#C)CCOCC2)=O)CCC(CO)C(NC(=O)CC2(O)CC2)C1 N1(C(C(=O)NCC(N2CCCC2)C)=O)CC(CCO)OCC12CCC2 c1(OC)cc(C(N2CC3CN(C(C4(F)CCOCC4)=O)CC23)=O)ccc1Br N1(C(C(C(C)C)O)=O)CCOC2(C1)CN(C(c1ccc(Br)nc1)=O)C2 C12(C(=O)NCCCC=C)CC3CC(C1)CC(F)(C3)C2.c1(CC=O)cncs1.N N1(C(C)=O)CCCCC(CCC(=O)O)C1.C(=O)(C(CC(=O)O)CC)NC(C)(C)C Cc1c(C(=O)NC2CCC(NC(c3ccc(O)c(O)c3Cl)=O)C2)cc(Br)cc1F C=CCC(C)(C)C(=O)NCC(CC(C)C)NC(=O)C(F)CC1CCC1 c1(NC(CCC2CCN(C(C(COC)N(C)C)=O)C2)=O)cc(C#N)cnc1C c1(C(N(CC(C)NC(C2(C)CC2(C)C)=O)CC)=O)cc2occ(Br)c2[nH]1 c1(C(N(C(CNC(c2ccncc2N)=O)C2CC2)C)=O)cnn2c1C(=O)NCC2 C=CCN(Cc1ccccc1)N1CCC(N2CCCCC2=O)C1 c1(C(=O)NC2CC2)cc2c(nc1O)CCCC2=O.c1(C=O)scnc1C1CC1.N CC1(NC(=O)CC2CCCC3(CC3)C2)CCC(NC(=O)CCC(N)=O)CC1 C12(C(N3CC(C4(NC(=O)Cn5cnnc5O)CC4)C3)=O)CCCC(=O)N1CCC2 CC1CCCC1CNC(=O)CC1(NC(c2cnns2)=O)CC1 CC1CCN(C(=O)Nc2ccccc2Br)CC1C C1(CC)CN(C(c2cnc(C)s2)=O)CCN1C(=O)CNC=O c1(C(=O)NCC(CC=C)NC(=O)C=CCCC)c(Br)nc2n1CCOC2 CC(CCCCNC(c1n[nH]cc1Br)=O)NC(=O)CCc1ccc(F)nc1 CC1(C)CCC2(CCN2C(=O)CC(=O)NCCc2ccccc2)C1 c1(NC(=O)NCCCCn2cc(C(C)=O)nn2)ccc2scnc2c1Br N1(C(C2C(C#C)C2)=O)CC(CNC(c2ccnc(C3CC3)c2)=O)C(O)C1 C(=O)(C1=C(C)N(C)c2nnnn2C1)N1C2CCC(NC(CC(CC)C)=O)(C2)C1 C1CCN(C(c2cc(C(N)=O)cs2)=O)CC1C.n1(CC)cc(C(=O)C(=O)N)cn1 C(=O)(CCCC(CC)CC)N1C(CNC(CCC=C=C)=O)CC(F)C1 c1(C(=O)Nc2cccc(CO)c2)cc(F)cc(F)c1.C1CC1C(F)(F)F CC1(C)CC(CNC(c2cccc(F)c2)=O)CN1C(=O)Cc1cocn1 C1(CNC(C=CC)=O)CCN(C(=O)C(N2CCOC2=O)C)C1(C)C C1(NC(=O)CCC2CCOCC2)CCN(C(C2COCCOC2)=O)CCC1CO CN1CCC(F)(C(=O)NCC2CC(F)CN2C(c2ccc(C#N)[nH]2)=O)CC1 CC1CCc2nc(C(=O)N)cn2C1.C1(C2(O)CN(C(C3CC(O)C3)=O)C2)CC1.C C(=O)(CC1C(=O)Nc2ccccc21)NC(C)CCN(C(=O)CS(N)(=O)=O)C c1(N(C)CC2C(C)C2)[nH]c(=NC2CC2C)nc2scnc12 CC(C)C(C(=O)N1CC(N(C)C(c2ccc(C#N)s2)=O)C1)c1ccc(Cl)cc1 c1(OC)c(C(=O)NC(C)Cn2cc(C3CCCN3C)nn2)csc1C N1(C(C2(CC=C)CCCC2)=O)CC2(CCCN(C(C3(C#N)CCCC3)=O)C2)C1 c1(C(=O)NC(C)CCNC(=O)Cc2cnn(C(F)F)c2)c(N)ccc(F)c1F O=C(C1CCCc2nn[nH]c21)N1CCOCC(NC(C2CC(O)C2)=O)C1 c1(CC(=O)NC2C(NC(C(CC)C)=O)C2)ccc(SC)cc1Br N1(C(=O)CC2C=CCCC2)CCC(F)(C(=O)NC(c2cscn2)CO)C1 C1(CCC)CN(C(=O)CCSCc2ccccn2)CCN1C(C1CCCO1)=O c1(C(N2CC(CNC(c3cnc(OC)s3)=O)C2)=O)c2c(c[nH]c1=N)CCC2 C(CC)(C(=O)NCC1(CNC(=O)C(C)(C)OC)CC1(F)F)OCC c1(C=O)ccc2c(c1)C(=O)NCC2.c1(CC(=O)NCC2CCC2)ccsc1Cl.N c1(C(=O)NCC=CC)c[nH]nc1CNC(c1sccc1Cl)=O CCC(CNC(=O)C(C)COC)(CC)NC(c1sccc1OC)=O c1(CC2CCN(C(CC3C(C)C(=O)CC3)=O)CC2)ccc2[nH]ccc2c1 N1(C(C2(C)N(C(c3ccc(COC)o3)=O)CC=C2)=O)CC2CC=CC1C2 C12CCCCC1N(c1nc(C#N)c(Cl)s1)CC2.C1(OCC)CC(CC(=O)NC)C1 CCCC(C)(O)CC(=O)NC1CCCCC1NC(c1nccc(Cl)c1C)=O C1(CSC)NC(=O)N(CCc2nc(-c3ccccc3Cl)cs2)C1=O C1(C(=O)NC2CC(NC(c3nc[nH]c3C(C)(C)C)=O)C2)(CC)CCOCC1 CN=C(NCCC1(OCC)CCC1)NC1CCN(S(C)(=O)=O)C1 n1(CC)cnc2c(N(CCCCO)C)nc(N3CCS(=O)C4(CCC4)C3)nc12 Cc1cc(C)c(C(=O)NCCCC(=O)NC(Cc2ccccc2Cl)C(=O)O)c(O)n1 c1(C(C(=O)NCCCSC)N(CCC(=O)NC2CC2)C)nc(F)ccc1Br C1(NC(C(c2ccc(C)cc2)F)=O)CC2CCC1CN2C(=O)Cc1nocc1C c1(NC)ncccc1C(=O)NCC=CCNC(C1(C)CC1(C)C)=O C(=O)(C(C)(C)C(F)(F)F)NCC(C(N1CCC(COCC)CC1)=O)OC C1(NC(C(C)OCC(C)C)=O)CCN(c2cc(C3CCCCC3)ncn2)C1(C)C Cc1cc(C(=O)NCC2CC2NC(=O)Cc2cn[nH]c2)c2cnn(C)c2n1 N1(C(C2ON=C(CC)C2)=O)CC2CC(NC(=O)C#CC3CC3)CC1C2 N1(C(CC2C(C)=NNC2=O)=O)C(CC(N2CCC(O)(CO)C2)=O)C2CCCC12 c1(C(N2CN(C)C(=O)C2C)C(=O)NC(CC)C)c2cc(Br)ccc2nn1C CC1=NNC(=O)C1CC(N1CC2C(NC(=O)CCc3cc[nH]n3)C2C1)=O C1(OC)(OC)CCCN(C(c2cc(C)nn2C)C(=O)NCC2CCCO2)C1 c1(NCC2CN(C(c3c(C)nc(CC)s3)=O)C(C)C2)cc(C)c([N+](=O)[O-])cc1Br C(CCCC(=O)NCCC1CCN(C(C2CCC(COC)C2)=O)CC1)OCC Brc1ccsc1-c1cn(CCC2CCSC2)nn1 C1(CCNC(=O)C(O)C2CC2)(NC(c2nc(Cl)cs2)=O)CCOCC1 C1(NC(C=CSC)=O)CC2CC(NC(=O)CCOc3ccc(F)cc3F)CC2C1 N1(C(C2OCC(C)C2)=O)CCC2CC(NC(C3(C)CC3Br)=O)CCC2C1 c1(C(=O)NCCC2CCO2)ccc2c(c1)CN(C(C1(F)CCOCC1)=O)CC2 C1(CN(C(CC2C(CNC(C(C)C3CC3)=O)C2)=O)C)CCC(=O)N1 CCC(CC(F)(F)F)C(=O)N.C1(C=O)CC2(C1)CC(C)(C)C2.C(C)C(C)(C)C Cc1ccc(C(=O)NC(C2CCN(C(=O)CCc3cccs3)CC2)C(C)C)n1C c1(OC)ccc(C)c(C(=O)NC2CCC(CC(=O)NC(C3CCOC3)C)CC2)c1 CCCC(C)(CC)C(=O)N(C1(C(N2CCCC(N(C)C)C2)=O)CC1)C C(=O)(CCCN1CCCC1)N(N(C(C1(CC2CCN(CCF)C2)C(C)C1)=O)C)C C1(NC(c2c(C)c(N)cnc2)=O)CN(C(=O)Cn2ncccc2=O)CC12CCC2 c1(C(N(C(C)CNC(c2cc(C(C)C)on2)=O)CC)=O)nn(C)nc1Br N1(C(C(CC)NC(C)=O)=O)CC(NC(c2ccccc2F)=O)C2(CCC2)C1 c1(N2CC(C)(C)C(c3ccccc3)C2)cccc(S(=O)(=O)NCCO)n1 c1(-c2nc(C3CC(C(=O)OCC)OC3)on2)ccc(CS(N)(=O)=O)c(F)c1 C1(C(=O)NCCc2nc(C)sc2)CN(C(C2OCC3CCCC23)=O)CC1C1CC1 C1(CC#N)(NC(=O)CCC2CCCN2C(c2cnccn2)=O)CCCC1 N1(C(Cn2c(C)ccn2)=O)CC2(CCCC2)C1C(=O)N(CCC(C)(C)C)C C(=O)(C(C)(F)C(=O)OC)N1CC(OCCC(=O)NC(C=C)(C)C)C1 C1C2CN(C(c3cscc3C3CC3)=O)CC12.CC(Cc1cnc[nH]1)C(=O)N(C)C CC1(OCC(=O)NC2C(NC(=O)CC)C2)CCC1.C1(C(=O)N)CCCC1 C1(NC(c2c(C)cc(C)nc2)=O)CC12CCN(C(=O)Cc1csnc1C)CC2 C1(F)(CNC(C(F)OC)=O)CCC(NC(=O)C(F)=C(C)C)C1 c1(CN(C(=O)C(C)NC(C2C(C)C2C)=O)CC)ccncc1 C(=O)(C(CC)C(=O)OC)N1CC(OCCC(=O)NC(C=C)(C)CC)C1 N=c1nc(C(=O)NCc2ncc(C(=O)NCc3cnccn3)cn2)cc[nH]1 c1(C(=O)NC(CC)CNC(=O)CC(C)NC(N)=O)cc2c([nH]1)CCCC2=O C(=O)(N=c1nc(-c2cccnc2Cl)[nH]s1)Nc1cc(C)nnc1O N1(C(c2c(SCC)cccc2)=O)CCC2CN(C(=O)C=CC(C)CC)CC12 c1(C(N2CCCC2CCCOCC2CC(F)(F)C2)=O)c(Cl)cncc1Cl N1(C(C2(C)CC(=C)C2)=O)CC(C2CN(C(=O)Cc3ccc(Br)c(C)c3)C2)C1 C1(CC(=O)NC)CN(C(=O)CCC2CCCC2)CCO1.c1c[nH]c(C(F)(F)F)c1 C1(C(N(CCCCOC)C)=O)CCN(C(C2(OC)CCC(C)C2)=O)CCO1 N#CC1(c2ccccn2)CCCN(C(=O)Nc2ncc(CC3CCCO3)s2)C1 C=CCC(Cc1ccccc1)C(=O)N(CC)Cc1cn(C2CC(C(=O)O)C2)nn1 C(CCCCN(C(=O)CC(C)N(C)C)C)NCCNC(C1C(C=C)C1)=O C#CCC(CC(=O)NCc1ccc(Cl)o1)NC(=O)CN1CCCC1C N1(C(CN(C2CC(C#N)C2)C(Cn2c(C)ncc2)=O)=O)CC(C)CCCC1C C1(CNC(Cc2cc(C)on2)=O)C(C)CCN1C(=O)C(C)Oc1ccccc1F Cc1ccnc(NCCC(C)NC(C2(O)CCSC2)=O)n1 C(=O)(C(=O)NNc1nc(C)c(C)s1)N1C(c2ccc(OC)cc2)CC(C)C1 C1(NC(C(F)=CCC)=O)CC(O)CN(C(=O)CCNC(=O)C=CCl)C1 N1(C(c2cc(C)ns2)=O)CCC(N(C(C2CC2C#N)=O)CC2CC2)CC1 C1(F)COCCN(C(=O)CCC=O)C1.n1(CC)nncc1C(=O)N.C(C)(C)C.C c1(C(N2CC=CC(NC(=O)C(F)CC3CCCC3)C2)=O)ccc([N+](=O)[O-])cc1 O=C1NC(CC(N2CC(C(O)C(F)(F)F)C2)=O)CO1 c1(C(=O)NC2CC(NCc3ccc(Br)nc3)C2)nccc2ccccc12 N1(C(c2c(C)cno2)=O)CCC(C(CO)NC(=O)CC(C)N(C)C)CC1 C(=O)(C(C)CC(N)=O)NCC1N(C(c2ccc(CCC)[nH]2)=O)CC=C1 C1(C(N2CCC(CCNC(CC(CC)C)=O)CC2C)=O)CCC2CC1C2(C)C C(CCCC(=O)NCC(F)CNC(C1CC1c1cncn1C)=O)OC C(C#Cc1cccnc1)NC(C1(C2CC2)CN(C(CCC(C)OC)=O)C1)=O c1(OC)cccc(Br)c1CN1CC2(CC(CC(=O)NCCCS(N)(=O)=O)C2)C1 C1(C#CC(=O)NCC(CCOC)NC(c2cc(C)nc(O)c2)=O)(CC)CC1 c1(C(N(C)CC2CN(C(c3ccc(F)cn3)=O)CCO2)=O)cnc2nccn2c1 C1(N2CCSCC2)(NC(=O)NCC(C)(OCC)OCC)CCCC1 n1(CC)ccc(C(=O)N(C(C)C(=O)NCCN2CCC2)C2CC2)n1 N1(C(Cc2cnc(OC)s2)=O)CC(C)CN(C(c2ccccc2C#N)=O)C(C)C1 N1(C(C(N2CCC(CC(N)=O)C2)=O)=O)CCN(c2cccc(Cl)c2)C(=O)C1 C1(Nc2nc(SC)c(F)cn2)COC2(CCN(C(=O)Cc3csc(C)n3)CC2)C1 N1(C(C(=O)NCC(c2ccc(-n3c(C)ncc3)cc2)C)=O)CC(C)C(C)(C)C1 C1(C=O)CC(C(C)C)=NO1.C(=O)(CCCN(C)C)N(C(C)C)CC1CCC1 C1(C2CCOCC2)(CNC(=O)NCC(=C)C(F)(F)F)CC1 CC1OCCC1C(=O)NCC1(C(N2CCC(OCCO)C2)=O)CCCO1 C(=O)(CC(CCN)C(F)(F)F)N1CCN(C(C)(C)CF)CC1 Cc1scnc1C(=O)NCCCC1CCCN1C(=O)COCC1CCOCC1 c1(OC)ccc(-c2nc(CSc3ccccn3)n(Cc3cnn(C)c3)n2)c(Cl)c1 c1(OC)c(C(N2CC(CO)C2)=O)cc(Cl)cc1C.C1(C(=O)N)CC(C)CC(C)C1 N1(C(CCOCC#C)=O)CCC(N2CCN(Cc3cccnc3OC)CC2)CC1 N1(C(C2CC2)=O)CCN(C(N2CCN(C(=O)CNS(N)(=O)=O)CC2)=O)CC1 c1(CN2CC3C(NC(=O)CCCCCCCBr)C3C2)cc([N+](=O)[O-])cc(O)c1O C1(NC(CSC)=O)CCN(C(=O)CC2(N(C)C)CCCC2)C1c1ccccc1 N1(C(C(CCC)C)=O)CCN(C(C2(CC(C)C)CCC2)=O)CC1C c1(C(=O)OC)cc(OC)ccc1Cl.c12ccc(nc1)c1ccc(cc1)[nH]c2=O C1(CC(N2C(C(C)C)C(C)(C)C2)=O)CC2(CC2)CN1C(c1ccsn1)=O C(=O)(C1=C(Cl)CCCC1)NCCC1CC(NC(c2ccc(C)cc2F)=O)C1 c1(NC(=O)NC2CCN(C(=O)NC(C)C)C2)ccc(C#N)c(Br)c1 c1(SCC(=O)NCC2N(C(Cc3cnc(C)o3)=O)CC2)ccc(O)cc1 Cc1cccc(OCC(=O)NCC(O)CC)c1.C(=O)C(F)(F)c1csc(=N)[nH]1.N CCC(C)C(C)C(=O)NC1CC2(C1)CC(NC(C1CC3CC1C3)=O)C2 c1(CC)noc(C)c1C(=O)NCC1CC1NC(c1cscc1OC)=O N1(C(C(C)(C)C#N)=O)CC2(C1)CN(C(=O)C(F)(F)C1CCCCC1)C2 C12(OC)CCCCC(C(N3CCC(F)C3)=O)(C1)C2.C1(C(=O)N)(C(C)C)CC1 C1(NC(N(C(C)CCN)C)=O)CC2(C1)CC1(CCC1)C2 c1(C(=O)NCC2CN(C(C(c3ccc(C)cc3)=O)=O)C2)sc2cccnc2c1Cl N1(C(C=CC=CCC)=O)CCCC(N(C(=O)C=C=C(C)C)C)C1 C#Cc1cccc(C(=O)NC23CC(NC(=O)CC(CC)CCC)(C2)C3)c1F c1(C(=O)NCC2C=CC(NC(C3CCN(C)CC3)=O)C2)ccc2nnc(O)n2c1 c1(CC)cc(C(=O)NC2(C)CC(NC(=O)CC(C)N3CCCC3=O)C2)n[nH]1 C(=O)(CCC(C(C)C)NC(C1CC(C)(F)C1)=O)NCC(C(CC)C)CO c1(C=O)cnn(CC(F)(F)F)c1.c1(C(C(=O)NC2CC2)N(C)C)cccnc1.N N1(C(C2CC=C(C)CC2)=O)CCC2(CCN(C(c3coc(Cl)c3)=O)C2)C1 N1(C(C2C(C)OCCC2)=O)CCC2(CC1)CC2CNC(=O)CCc1ccsc1 Cc1ccc(C(=O)NCCC2(NC(C3CCCCC3)=O)CCC2)n1C.C(N)=O c1(C(N2CCC2)=O)ccn2nccc2c1.c1(SCC=C)ccccc1C(=O)NC N1(C(COC(C)(C)C)=O)CC2CC(NC(=O)C(C)(C)c3cscc3Cl)CC1C2 C1(C(=O)NCC2(NC(c3cc(C)on3)=O)CCCCC2)CC(F)(F)C1(F)F C1(C(=O)NC(C)CCO)CC(C)CN1C(c1cc(Cl)n(C)n1)=O c1(OC)nc(C(N2CCCC(C(=O)Nc3snc(C)c3C#N)C2)=O)ccc1Br C1(CC(=O)N)CCC2(CCCC2)CC1.N1(C(C2(C#C)CC2)=O)CCOC(C)(C)C1 c1(CC(=O)NC2CC(NC(C=CC=CC)=O)C2)ccccc1.CCCCC CCCC(O)CC(=O)N1CCN(C(=O)C(C)NC=O)C(COC)C1 c1(N(C(N(C2CC2)CC2CC(OC)CN2C)=O)C)cc(N(C)C)ccc1F c1(COC)c(OC)cccc1C(N1CCN(C(C2CC2C(N)=O)=O)CC1)=O c1(C(NC(C)C)=O)ccc(C(C)=O)c(C)c1.c1(C=O)nccc(Cl)c1F.CC C(=O)CCCCN(C)C.c1(C(N(C(C)C)CC)=O)nccn1C(C)(C)C.N CC1(F)CCCCN(C(C2CCCN(Cc3ccc(Br)[nH]3)C2)=O)C1 c1(NC(C2N(C(c3n(C(C)C)ncc3)=O)CCCC2)=O)ccc2c(O)n[nH]c2c1 C1(C(=O)NCC2CCN2C(c2cnccn2)=O)COc2ccc(F)cc2C1 C#Cc1ccc(Cl)c(C(N2CC3CCC(C2)N3C(c2cc(C#N)n(C)n2)=O)=O)c1 c1(C(=O)NCC2(O)CN(C(c3ccc(S)cc3)=O)C2)[nH]cc2c1CCC2 C1(NC(c2scc(C)c2)=O)CCN(C(c2ccc(Br)cc2F)=O)CC1C C(C(C)(C)CC(=O)N1CC(N2CCN(C(=O)C(C)(C)OC)CC2)C1)OC CC1(C)CC(CNC(=O)CC(F)(F)F)N(C(=O)C=Cc2ccccc2)C1 C(N=c1[nH]c(NC2CCC2)nc2c1CCC2)C1(N(C)C(=O)OC(C)(C)C)CC1 Cc1[nH]nc2ccc(C(N3CCN(C(C4CCCCC4)=O)CC34CCC4)=O)cc12 C1(CNC(C2(C#C)CN(C(C3(COC)CC3)=O)C2)=O)CNC(=O)CC1C S(=O)(=O)(c1ccc2nc(N3CCC(C)(F)C3)ccc2c1)N1CC(C)C(F)(F)CC1 CC(C)C(F)C(=O)NC(C)Cn1cc(CNc2cccc(Cl)c2)nn1 N1(C(C=C(CC)CC)=O)CC(CNC(C2(C3(O)CCC3)CC2)=O)C(C)(C)C1 C=CC1CC1CNC(C)(C)C.C1CCCS1 C=C(CN=C(NCC1CC(O)CCO1)NCCc1ccccn1)C1CCOCC1 C1(C(N2C(C#C)CC2)=O)CN(C(c2cc3n(n2)CCC3)=O)CC12CC2 N1(C(COCCNC(c2n(C(C)C)ccc2)=O)=O)CCC12CCC(O)CC2 C(=O)(C(CCC1CCC1)NC(=O)C)NC(CN(C(C)C)C)C.C1CCCC1.O C#CCCCC(C)C(=O)N1CCCC(O)(CN(C(=O)C(O)C=C)C)C1 C1(CCNC(=O)CCC2CCC(O)CC2)CN(C(c2ccccc2)=O)CCCO1 N1(C(c2c(CC)nn[nH]2)=O)CCC(C)C(C)C1.n1(C2(C(=O)N)CC2)cnnn1 C(=O)(C1CCCn2ccnc21)N1CCCC(O)(CNC(c2cc(C)n(C)c2)=O)C1 O=C1CC(C(=O)NCCCOCC)CC(=O)N1.C1(Cl)(C(=O)N)CC1(F)F N1(C(=O)NCCC[Si](C)(C)C2CC2)CC(S(=O)(=O)c2cccc(F)c2)C1 Cc1nnc(N2CCN(CCNC(c3cccnc3C3CC3)=O)CC2)nc1C C(=O)(CCCC(CC)NC(C1CC(C)(CC)C1)=O)NCCOCC#C C1(C(=O)NC(C2CCCN2C(=O)C=Cc2cscn2)C)C(F)(F)C12CCC2 Cc1ccc(C(C)N(C)C(=O)OCC2OCCC2(C)C)cc1 C1(C(=O)NCC)CN(C(=O)NC(C)CN(C)C)c2ccccc2O1 C1(C(N(C2CCN(C(CCC#C)=O)C2)CCO)=O)OCCOC1(C)C c1(C(N2CC(CNC(CNC(C)=O)=O)C3(C2)CCC3)=O)coc2cc(C)ccc12 N1(C(CC2(NC(C(CC(C)C)OC)=O)CC2)=O)CCC2(CNC(=O)O2)C1 Cc1ccc(C(N2CCOC(C)(CNC(=O)C)C2)=O)c(F)c1F.C1(F)CC1.O N1(C(C=CCCC)=O)CCCC12CCN(C(C1CCC(C)(C)O1)=O)C2 C1(CCOC)(NC(C2CCOC(C)C2)=O)CCN(C(C2(O)CCCCC2)=O)C1 C(CCCCC(=O)NC1COCC1CO)NC(c1n[nH]c(C)c1Cl)=O C(CC(C)C)(C(=O)NCc1cccc(O)c1F)NC(C(C)OC(C)=O)=O C1(CC(=O)NCc2cc(C(C)C)no2)(NC(c2nccs2)=O)CCOCC1 O=C(Cc1cc(C(F)F)on1)N(O)Cc1cn(C2CCCC2(F)F)nn1 CC(C)C(C)(CNC(=O)CC(O)C1CCCC1)NC(c1sccc1CO)=O c1(C(=O)NCC2C3CN(C(c4cccc(C#N)n4)=O)CC32)ccn2cncc2c1 N1(C(c2cn(CCC)nn2)=O)CC(NC(=O)C(O)CCSC)C(C2CC2)C1 C1(CNC(=O)Nc2nnc(O)o2)CCCN(c2ccc(Cl)cc2)C1 C1CN(C(=O)CN(C)C(=O)C2CC2)CCC1C.c1nc(C)c(C=O)s1.CS.C c1(-c2ccc(C(N3CCN(C(COC)=O)CC3)=O)cc2)c(OC)cc(C)cc1C Cc1ccc(C(=O)N(CC(O)CN(C)C(c2n[nH]cc2C2CC2)=O)C)c(C)n1 C1(NC(C2SCCS2)=O)CC2CC1N(C(c1ccncc1F)=O)C2 Cc1c(Br)ccc(NC(C2CC(C)CN2Cc2ccc(Br)cn2)=O)c1C c1(CC(=O)N(C2CCC2)C)cc(C2CC2)on1.C1(N2CCCC2)(C=O)CCC1 c1(CN2CC(C(N(C)CCO)=O)CC(F)(F)C2)cc2c(Br)cccc2s1 N1(C(C2C(C)(CC)C2)=O)CCCC(NC(=O)COC)C1 c1(NC(CC2(NCc3cc(OC)c(Br)cc3)CCC2)=O)cc(F)c(C)c(F)c1 c1(CC=O)ccc(Cl)nc1.C(=O)(CC(=O)NC1CCCC1)OCCC(C)C.C c1(Nc2ccn(C)n2)ccc(NC(=O)C=Cc2cncn2C)cc1 c1(CC)nn(C)c(CC(=O)NCC(CNC(C2CN(CC)CCO2)=O)O)c1Cl N1(C(c2c(C)c(Cl)cnc2)=O)CC2CCC(C1)N2C(=O)C(C)Sc1ccccc1 N1(C(c2c(C)nn[nH]2)=O)CC2CC(NC(=O)CCc3cncnc3)CC2C1 c1(C=O)ccc2c(c1)OCCN2.C1(C(C)C)CC(C(=O)NCC2CC2)CCO1.N C(=O)(C(CNC(c1ccn(CC)c1C)=O)CCC)NC(C#C)C(C)(C)C C1(CC=C)CCCCC1(c1nnnn1CC)NCc1nccn1CC(F)F C(=O)(CCC(C)C)N(C1CCN(C(C2C(Cl)(Cl)C23CC3)=O)CC1)CC#C c1(C(=O)NC2CC(CNC(C3C(CCC)C3)=O)C2)csc2c(F)cccc12 CC(CF)CC(=O)N(CC(C)N(C)C(c1csc(C(F)(F)F)n1)=O)C C1(C2CCC2)(C(=O)NCCCN(C(C(C2CCC2)OCC)=O)C)CC1(F)F c1(C(N(CCCN(C(c2n(CC)nnc2C)=O)C)C)=O)cc(F)ccc1C C1(C(N(CC(=O)NCC)CC)=O)CCN(C(c2ccn(C)n2)=O)C1 C1(C(=O)NCCN(C(=O)CO)C)CC12CCc1ccccc12.c1cncc(Cl)n1 CC(CCCCNC(=O)CC1CCNC(=O)C1)NC(=O)C.c1(C=O)ccoc1 C#CC1(C(=O)NCC2(C)CCCN(C(=O)C3=C(C)OCC3)C2)CCOCC1 c1ccc(N=S(C)(C)=O)s1.C(=O)(CC(C)C)NCC(=O)OC.CC(C)C.C C1(C(N2C(CN(C(C(c3ccc(F)cc3)C)=O)C)CCC2)=O)CCC2CC2C1 C(=O)(CC(C)(C)C=O)N.c1(C(=O)NCC(=O)NCCC)occc1C C(=O)(C(O)CC(F)(F)F)N(CCC(=O)NC)CCNC(COC)=O Cc1cc(C#N)cnc1C(N1CCC(CNC(C2CCC(=O)N2)=O)C1(C)C)=O C1(C)(OC)CC(NC(=O)C(CC(C)C)NC(C2CC(O)C2)=O)C1(C)C C(=O)(C1=CC(O)C(NC(=O)C2=C(C)CCC2)C1)Nc1cc(OC)cc(F)c1 N1(C(C(C)OCC(C)C)=O)CCCCC12CCC2.C1(C(=O)N)CC(C(C)C)=NO1 C1(C(C)NC(c2nnc(C)s2)=O)CCCN(C(c2c(Cl)noc2C)=O)C1 N1(C(C)=O)CCC(C(C)(C)C)(NC(=O)C(O)C2CCCC2)C1 c1(CC)nc(C)n(C)c1C(=O)NC1CCN(C(c2cc(O)nc(O)c2)=O)CC1 C1(C(N2CC(NC(=O)CNC(C3CCOCC3)=O)C2)=O)CC(=O)C12CCC2 C1(CC(=O)NCCOCCNC(C2C(=C)C2)=O)C(CC)C1(F)F c1(CC(N2C(C(=O)Nc3cnsc3)CC(OC)C2)=O)ccc(C#N)cc1 C1(C(C)NC(=O)C(n2cc(Cl)cn2)C)CN(C(C2(CO)COC2)=O)CCO1 CC(O)C(C(=O)NC1CCN(C(C2(c3cnccn3)CC2)=O)CC1)NC(N)=O N1(CC)CCC(NC(C2CCC(NC(C3CN(C)CCN3C)=O)C2)=O)CC1C C1CN(C(=O)CC2CCC(C(=O)O)CC2)C(C)(C)C1.CC1=CCC(C=O)CC1.N C1(NC(=O)CC2CCCC2NC(C2(O)CC(CF)C2)=O)CCC(F)(F)C1 CC1OCCOC1C(=O)NC(C1CCCN1C(=O)COc1ccc(F)nc1)C C1(C(=O)NC(CC2CCN(C(CCCOCC)=O)CC2)C)Cc2nc(C)cn2C1 c1(C(=O)NC2CC(=O)OC2)ncn2cc(-c3cccc(F)c3CO)sc12 C(=O)(CCN=C(NCC(F)F)NCCNC=O)NC(C)C.c1csc(Cl)c1.N CC1CN(C(C2CCCCS2)=O)CC2(CCN(C(=O)CC34COC(C)(C3)C4)C2)O1 C1(NC(c2c(OC)n[nH]c2)=O)CCCCC1CNC(c1cc(C)[nH]n1)=O Cn1cccc(C(N2CCC23CN(C(=O)CC2CC2(Cl)Cl)C3)=O)c1=O c1(C(N2CC(C)C(NC(=O)C(=O)N(C)C)C2)=O)c[nH]c2nc(Cl)ccc12 C(=O)(C(CC)CC(C)C)NCCNC(C1CCN(C(CC)=O)C1)=O.C1CC1.C Cc1cc(=O)n(Cc2cc(F)ccc2C)c(=O)n1-c1ccccc1 C1(C(N2CC(C(=O)NC)C2)=O)CCN(C(=O)CCCNC(=O)OC)C1 c1(C(C)=O)cncc(C(=O)NCCCN(C)C(C2(C)CCCC2O)=O)c1 C1(NC(C(C(C)C)O)=O)CCC2(CC1)CC(NC(=O)C1=CC(O)CCC1)C2 CC(C)CC(O)C(C)C(=O)NC1CCCC(C(N2C(CO)CC2C)=O)C1 C1(NC(C=Cc2cn(C)nn2)=O)CN(C(c2cnc(N)cn2)=O)C(C)(C)C1 C1(CNC(=O)CCn2cccn2)CN(C(c2ccsc2)=O)CCCO1 N1(C(CC2(C=C)CC2)=O)CC(N(C)C(c2ccn(C3CC3)n2)=O)C(O)C1 C1(C(=O)NCC(C)(C)CN(C(=O)C)C)(OC)CCCOC1.c1ccccc1Cl.N N(C(=NCCc1ccc(SC)cc1)NC1CSC1(C)C)C(COC)C c1(C(N2CC(CNC(=O)CC=C(Cl)Cl)C2)=O)cc2cc(Br)ccc2[nH]1 c1(NC(C2CCC(C)O2)=O)cccc(C(F)F)c1 Cc1nn(CC(=O)N(C2CCCN(C(=O)C(C)(O)C(C)C)C2)C)c(C)c1Cl C(=O)(C1=NN(C2CC2)C(=O)CC1)N(C1CCN(C(c2cn(C)nc2)=O)C1)CCO CN=c1[nH]c(=NCC2CCC(C)(C)O2)[nH]c(=NCCCc2ncccc2C)[nH]1 C#Cc1ccc(C(=O)N(C)CC2CCN(C(c3cc(Br)co3)=O)CC2)cc1C CC(C)(C)C(=O)C(=O)OCC(=O)Nc1nc(-c2cncc(F)c2)cs1 N1(C(C(CNC(c2c(OC)scc2)=O)C(C)C)=O)CCC(C2CCCC2)C1 c1(OCC(=O)N(CCOCCNC(C=C(C)Cl)=O)C)ccc(C)cc1Br C1(NC(=O)C=Cc2cnccn2)COC2(C1)CN(C(C1CC3(CCC3)C1)=O)C2 C=C(C)CC(C(=O)OC)NC(C1CCCC1NC(=O)Cc1ccoc1)=O c1(NC(c2c(CNC(C(CC)OCC)=O)cc[nH]2)=O)cncc(Cl)c1 N1(C(COCCC=C)=O)CCN(C(C2(C)CCCC2C)=O)C2(CCC2)C1 CC(C)CC(C(=O)N(C(C)CCNC(=O)CC1CCC1)C)N1CCCCCC1 C1(C(NC)=O)CCC(CC(F)(F)F)CC1.N1(C(CNC(=O)OC)=O)CCCC1 C1(N(C)C(C2(N(C(C3CC(F)C3)=O)C3CC3)CCC2)=O)CCCCC1O O=C1CCCC(CCCC(=O)NCCCN(C(C2CC2C2CCC2)=O)C2CC2)N1 c1(NC(CN(C(CC2C(OCC)COCC2)=O)C)C)nccc(C#N)n1 C(=O)(C(C)(C)CO)NC(CC)C(=O)N1CCC1(C)CCO c1(-c2onc(-c3c(C)ccc(OC)c3)n2)ccc(S(=O)(=O)N(C2CCCC2)C)o1 C(CCCCCC(=O)NC1CNC(=O)C12CC2)NC(C(C)NC(N)=O)=O C(CNC(=O)C#CCNC(=O)CN(C)C)(CC(C)C)OC Cc1cc(F)ccc1C(N1CCC(CC2CC3CC3C2)C1)C(=O)NC1CCC1 C#Cc1cccc(OCC(=O)NCC(C)CNC(=O)CC2CC(CC)C2)c1 Cc1nnc(CCCC(=O)NC(C)(CNC(c2ccoc2)=O)C(C)C)n1C Cc1cc(Br)cc(C(=O)N(C2CSCCN2S(=O)(=O)CCCCl)C(C)C)c1C C(=O)(CC(O)CNC(c1n[nH]c(C)c1O)=O)NC(CSCC)CO N1(C(CCCOC(C)=O)=O)CC(C)CN(C(=O)C(c2ccc(F)cc2)F)C(C)C1 C1(NC(C(n2ccc(C)n2)C)=O)CC2CCC1N(C(c1cc(Cl)cc(Cl)c1)=O)C2 CCCCC(O)C(=O)NCCCCN(C)C(C1(c2ccc(C)cc2)CCCC1)=O Cc1nccn1CC(=O)NC1CC(CNC(c2ccc(CO)o2)=O)C1 c1(C(C(=O)NCC(C(OCC)OCC)O)O)ccccc1C(F)(F)F c1(C(N2CC3(C(NC(C(CC)F)=O)CC3)C2)=O)cc(Br)c(O)nc1C C1(=CCNC(c2c(C)scn2)=O)CCN(C(=O)Cc2cscn2)CC1 C(C(C)(C)C#CC(=O)N1CC(OC(=N)O)C1)NC(CC1C(CC)C1)=O c1(SCC)ccccc1CC(=O)NCC(C)C(C)C.C1(C(=O)N)CC2CC2C1 Cc1nc(N2CCOCC(NC(c3cccc4nncn34)=O)C2)c(C)c(O)n1 N1(C(C(C)C#N)=O)CCC2CN(C(c3cn4ccnc4s3)=O)CCC12 C1(CC=O)C(=O)NN=C1C.C1(C)(C(=O)OC)CC(C(=O)N(CCCC)C)C1 N1(C(C(c2cc(C)c(N)cc2)(F)F)=O)CC(C2CN(C(=O)OC(C)(C)C)C2)C1 C1(CCNC(c2n(CCOCC)nnn2)(C)C(C)C)CC2(CCO1)CC2 C(=O)(CC(F)(F)C(C)C)NCC1CN(C(C(Cc2c(C)cccc2)C)=O)CC1C C(CCCCC(=O)NCC(C)(CO)NC(c1cnc(-n2cccn2)cn1)=O)=CC C1(NC(C=CC(C)NC(C2(C)CCCCCC2)=O)=O)CCCCCC1(C)C N(C1C(=O)N(C)CCc2ccccc21)C(c1ccc(C(=O)NC)cc1)=O Nc1cncc(-c2cccc(CN3CCC3c3cccc(Br)c3)c2)n1 C1(C2(O)CCOCC2)(C(N2C(CNC(C3CC3C3CCOCC3)=O)CC2)=O)CC1 c1(NC(=O)NC2(C(=O)OC)CC23CCC3)cc(F)c(N)cc1OC c1(C(=O)NCCC2(C(=O)NCCc3ccn(C)n3)CCCC2)ccccc1C C1(NC(c2c(CNC(C3N(C)C(=O)OC3)=O)cco2)=O)CCNC(=O)CC1 CC(C)CC(O)CC(=O)NC12CCN(C(=O)Cc3nc[nH]n3)CC1C2 C(CC(F)F)(C(=O)NCCN1C(=O)CCC1=O)NC(c1c(C)noc1)=O C1(NC(c2n(CC)ncc2)=O)CCCCCN(C(c2cn(CCO)nn2)=O)C1 Clc1cccc2[nH]c(=NCc3cnn4c3CCCC4)nc(N3CC4CC4C3)c12 C12(CNC(C(C(C)C)C)=O)CCCC(CN1C(c1ccc(OC(F)F)nc1)=O)C2 CCC(CC)C(=O)N1CC2CC1C2CNC(c1cncc(N2CCCC2)n1)=O N1(C(C2(CCOC)CC2)=O)CCn2ncc(CNC(C3C(C)C3C)=O)c2C1 C1(CNC(CCC=C)=O)(Cn2cc(-c3cnn(CCC)c3)nn2)CC12CCC2 c1(C(N2C(CNC(C(CC)=CC)=O)COCC2)=O)ccc(O)nc1Cl C1(COC)(C)CCCN1C1(CC=O)CC1.c1(C=O)ccc(C(N)=O)[nH]1 c1(C(=O)NCC2CC(NC(c3n[nH]cc3Br)=O)C2)cc2n(n1)CCC2 Cc1nn[nH]c1C(N1CCC(CN=[N+]=[N-])C1)C(=O)NC1CC1 N1(C(c2cc(CC)nn2C)C(=O)NCCCC)CC(C)(C)C12CCOCC2 c1(N(C(C2Cc3ccc(F)cc3O2)=O)C(=O)C2CC2)cc2c(cc1Cl)OCO2 c1(C(=O)NC2CN(C(Cn3ncc(C#C)c3)=O)CC2C)cnc2ccccn12 N1(C(C(=O)NC(C)C)=O)CCCN(C(c2cccc(Cl)c2Br)=O)CC1C Cc1noc(C(C)C)c1C(=O)N.C1(O)(C(C)C)CCN(C(c2cnc(Cl)s2)=O)C1 N1(C(c2scc(C)c2)=O)CCOCCC1C(=O)NCC1CC(=C2CC2)C1 N1(C(CCc2c(C)n(C)nc2)=O)CC2=C(C1)CN(C(c1ccc(Cl)cc1N)=O)C2 C1(C(=O)NCCNC(C2(CC)CC(F)(F)C2)=O)CCn2cc(C)nc2C1 C=CCC(CC)C(=O)N1CCCC(n2cc(Cn3ccnc3C)nn2)C1 Cc1[nH]nc2cc(C(=O)NCC3CC4CN(C(c5cncnc5)=O)CC34)ccc12 C1(CNC(c2nc(CC)oc2C)=O)CCC(C)N(C(c2ccccn2)=O)C1.O CC1(C)CNCCC1NC(=O)CCc1cccc(N)c1 c1(C(OCC)(OCC)OCC)cn(CC(=O)NC2COC(=O)C2)nn1 CN(C)S(=O)(=O)NCC(=O)Nc1cccc(NC(c2ccc(O)cc2)=O)c1 CCCCC(CNC(=O)C(C)OC1COC1)NC(c1csc(CCCC)n1)=O c1(C(=O)NCCC2N(C(CC(C)c3ccco3)=O)CCC2)csc(S(C)(=O)=O)c1 CC1C(NC(c2cncc(Cl)c2Cl)=O)CCCN1c1ccnc(C2CC2)n1 Cc1ccc(CNC(C2(NC(c3cscc3C)=O)CCN(C)C2)=O)cc1C C(=O)(C(F)C(C)CNC(=O)C=C(CC)CC)N(C1CCC1)CCC N1(C(C(CC)C)=O)CCn2nc(C(=O)NC3C4Sc5ccccc5C34)cc2C1 c1(C(=O)NCC2(CO)CN(C(C3ON=C(CC)C3)=O)C2)csc2cccnc12 N1(C(C(C)=C2CC2)=O)CCCCC(CNC(c2ccn(C3CC3)c2C)=O)C1 C1(NC(C2(CSC)CC2)=O)C=CCN(C(=O)CCC2CC2(Cl)Cl)C1 Cc1ccc(C(N2CCOCC(CNC(=O)C#CC(C)C)C2)=O)c(C)c1 c1(C(=O)NCC(C2CC2)NC(Cc2c(C)ccs2)=O)c(Br)ncn1C N1(C(COCC(=C)C)=O)CCCC1C1CCCN1C(C12CCC(C1)C2)=O C1(OCC)COCCC1CC(N1CCN(C(c2cccc(Cl)c2)C)CC1)=O C1(CC)CC2(CCN2C(=O)C(F)C(C)CNC(=O)C=CC)C1.CC.O C12(NC(CCCN(C)C)=O)CCC(C(N3CCOCC3CCO)=O)(CC1)C2 CCCCCCNC(C1(C)CC(C)(C)C1)=O.c1(C=O)n[nH]c(C(C)(C)C)n1.N CC1C(O)CCN1C(=O)C(CCC1CC1)NC(=O)C(C1CCCCC1)=O C1(NC(c2ccc(C)s2)=O)C2CCN(C(C34COCC3C4)=O)C12 C1(CC)CC(CC(N2CC(CO)C(c3cccc(F)c3)C2)=O)CCO1 c1(CCCOC)nc(-c2sc(Cl)nc2C)n(C2CCCOC2)n1 N1(C(C(F)OC)=O)CCN(C(=O)CCC(C)C)CC1c1ccncc1 CC(C)(C)C(CO)C(=O)N(C1(C)CCNC1=O)C(C1CN(C(N)=O)C1)=O C1(CC(=O)NCC2(CO)CCCO2)CCC(NC(c2c[nH]nc2Cl)=O)C1 CCC(CNC(=O)CNC(c1cc(F)c[nH]1)=O)C(C)(F)F CC1CN(C(C2(O)CCSC2)=O)CCN1C(=O)C1=COCCC1 C1(CNC(C(C)=C2CC2)=O)(CO)CCCN(C(=O)CC(C)(C)C)C1 C1(c2nc(C)on2)CCCN(C(C2CN(C(C3CC3C3CC3)=O)CCS2)=O)C1 C(=O)(C(CO)C(C)(C)C)NCC(CNC(CCc1n(CC)ccn1)=O)F c1(C2(NC(C(C)C3CC3)=O)CN(C(=O)C(C)(C)C(F)F)C2)cc(F)cc(F)c1 c1(C(N2CCC(CCC)(NC(c3cc(O)cs3)=O)CC2)=O)c(C)nc(C)nc1C c1(C(C)C)ccsc1C(=O)NC1CCC(NC(=O)CCNC(=O)CO)C1 N1(C(C(C)OCCOC)=O)CCC(F)(F)C(C)C1.C(=O)(C(C)(C)CC)N c1(OC)ccc(CC(=O)NC2CCC(C)(C)C2)c(C)c1.c1(CC=O)cocn1 C1(C(=O)NC(c2ncon2)C)CC12CCN(C1CCC(CO)C1)CC2 CC(CC(N)=O)C(=O)NC1CCN(CCNC(c2nnn(C)n2)=O)CC1 Cc1nn(-c2ccc(Br)cc2)c(NC(=O)C(=O)NC2CC(O)C2(C)C)c1C N1(C(CC2(C)CC2)=O)CCc2c(CNC(=O)CN3CCC3)cccc2C1 C1(N(C(C2CN(C)C(=O)C2)=O)C)CCCC2CN(C(c3csc(C#N)c3)=O)CC12 Cc1cnc(NC(C2(C)CCN2C(C2CC2C)=O)=O)s1 N1(C(CCC(C)OCC)=O)CCCOC(CCNC(=O)CN2CC=CC2)C1 c1(CC)cc(C(N2CCC(CNC(=O)Cc3cccc(Cl)c3)C2)=O)ncn1 Cc1ncn(O)c1C(=O)NCC1(F)CCN(C(c2snnc2C2CC2)=O)C1 c1(CC(CC(=O)O)NCc2ccc(Cl)cc2O)ccc(Cl)cc1Cl O=C(N=c1[nH]oc2cnccc12)C1CC12CCN(C(c1ccc(O)nc1)=O)CC2 C(=O)(CCCC(C)O)NC12CC(NC(c3cccc(C(=O)NC)c3)=O)(C1)C2 C(C1CN(C(c2cnc(C)n2C)=O)CC1C(N1CC(n2ccnc2)C1)=O)=CC N1(C(C(CC)F)=O)CC(NC(=O)C(n2nnnc2C(C)(C)C)C)CC(C)(C)C1 c1(COCC(=O)N(CC(CC)NC(CC)=O)CC)ccnc(OC)c1 C1(C#N)(C=O)CC2CC2C1.C(C)(C(=O)NCC1(CC)CC1)SCC.N Cc1ccc(O)c(C(=O)NC(C)CNC(C23CC(F)C2C3)=O)c1 C(CCCC(=O)N1CCCC1CCCO)NC(=O)Cc1ccsn1 c1(CCCC(N2CC(O)(CC)C2)=O)ccc(C2CC2)cc1.C(C(C)C(=O)N)SC C=CC(CC)C(=O)NC1CCCCC1C(=O)NC1(C(C)C)CC1 O=C(CCOc1ccc(F)cc1)NNC(=O)NCC1(c2cccc(I)c2)CC1 C(CN=C(NCc1ccnc(SC)c1)N1CCCC2(CCOC2)C1)OCC C1(C(N(C(C(=O)NCC2CC(OC)C2)C)C)=O)CC(C(C)C)=NO1 Cc1cccc(C(N2CCC(CCNC(C3(CC(C)C)CC3)=O)CC2C)=O)c1O C(=O)(CCCC(=O)OC)N1CCCC(N(C(C(F)=CC)=O)Cc2ccccc2)C1 O=S(=O)(c1cccnc1NCCOC1CCC1)NCCC1CCCCC1O C=C(Cl)CC(C(=O)NCC1(C)CCCCO1)NC(c1cnnc(C)c1C)=O CC1(C(N2CCC(CNC(=O)CS(N)(=O)=O)C2)=O)CCOCC1 N1(C(CCn2ncc(C)c2)=O)CC2CCC1CN(C(c1ccc(C3CC3)o1)=O)C2 CCCC(C(=O)N1CCCC1(C)C)NC(=O)CNC(=O)C(C)CCC Cc1csc(=O)n1CCC(=O)N(CCCN(C(=O)CC1CC1)C)C C(=O)(CCCN(C)N=O)N1C(CN(C)C(c2ccc(Cl)c(N)c2Cl)=O)CCCC1 C1(C=O)CC2(C1)CC2(F)F.c1(CCC(=O)N(CCCCO)CC)ccccc1Br.N C#Cc1ccc(F)c(C(=O)NC2CC2CNC(C2CC2)=O)c1.C=O.N n1(C(CC)C)nc(C(=O)NCCCCNC(C2COCCN2C)=O)cc1C C1(CC(=O)NC(CNC(C(C)NC(C)=O)=O)(C)CO)CCCCCC1 C1(CNC(C(C)SCCCC)=O)COCCN1C(=O)CC1(C)CC1 N1(C(c2c(C)csc2)=O)CC(C)C(NC(c2ccc(N(C)C)c(F)c2)=O)C(C)C1 c1(COC)c(C(N2CCN(C)C(CCF)C2)=O)[nH]c2ccccc12 C(=O)(CCP(C)(C)=O)N(CC(=O)NCC(=O)NCCC1CCC1)CCC c1(-c2ccc(N(CC(C(CC)C)C)C(C)C)cc2)c(C)nn(CC(F)(F)F)c1Cl N1(C(C2N(C(c3ccsc3Cl)=O)CC(=O)NC2)=O)CCC12CCCCC2 c1(C(=O)OC(c2ccc(F)c(Cl)c2)C(=O)OC)cc(=O)n2ccccc2n1 c1(C(N2CC(NC(=O)C(F)=C3CCC3)C(CO)CC2)=O)cnn2c1NCCC2 Cc1cc(C(N2C3CCC2C(CNC(C2CCCCO2)=O)C3)=O)c(C)c(C)c1 N1(CC#C)CCN(C(=O)C2=CCN(C(C3(C)CCCC3O)=O)C2)CC1=O Cc1ncc(C(=O)NC2CCCC2(C)CNC(c2cccc(O)n2)=O)cc1N C(=O)(CC(C)(C)C(F)F)NCc1c(C(=O)NCC(C)C(F)F)nco1 c1(C(=O)NC2C3CN(C(C(=O)NCCOC)=O)CC32)nnn2c1CCCC2 Cc1ccc(S(=O)(=O)NC2CCC(NC(c3cccc4cc[nH]c34)=O)C2)c(C)c1 c1(C(N(CC=CC(=O)N)C)=O)cncc2[nH]ccc12.c1(CC)cc(CC)on1 C=Cn1nncc1C(N1CCCC(CN(C(=O)Cc2cscn2)CC)C1)=O C12CC(C1)C(C)(C)O2.c1(C=O)cc(C)nn1C.C(C(=O)NCC=O)OC.N c1(C(N2CC(CNC(C(C)C)=O)C2)=O)cn(CCN2CCOCC2)cn1 C(=O)(C1=CC(O)CCC1)N1CCCC(NC(c2cnc(C(C)=O)s2)=O)CC1 Cc1cc(F)cc2c1N(C(C1CC3CCCC(C1)C3N)=O)CC2 C(C)(C(=O)NCC1CN(C(=O)CC2(CO)CC2)CCO1)(C(C)C)OC C1(C(=O)NCc2cn(CC=C)nn2)(CO)CCN(C(=O)C)C1.CC(C)C.S c1(CNC(CC2C(C)(C)C2)=O)ccc(C)c(F)c1.c1(C=O)cnn2c1CCC2 Cc1c(C(N2CCCC2CCN(C(=O)C(F)(F)CC(C)C)C)=O)sc2ccsc12 C1(C(N2CCC(C(NOCCCC)=O)(CC)C2)=O)CC(=O)NC1(C)C C(CCCCNC(=O)Cc1cncs1)N(C(=O)C(c1cccnc1)O)C N1(C(C(CC)F)=O)CC(C2CCN(C(=O)Cc3ccc4c[nH]nc4c3)CC2)C1 C(CC(=O)NCCCC1CC1)N(C(=O)CNC(N)=O)C N1(C(C(C)OCC(F)(F)F)=O)CCOCC1CCNC(C12CC1CNC2=O)=O Cc1cc(Cl)ccc1C(N1CCC(C)(NC(=O)CC2CCC(C)CO2)C1)=O N1(C(C2(CC)COC2)=O)CC2(CCCCN2C(C2CCC(C(F)(F)F)CC2)=O)C1 C1(NC(C(C)C#N)=O)CCCCCN(C(c2cc3cccnc3o2)=O)C1 C1(NC(C2C(C=C)OCC2)=O)CC2CCC1(NC(=O)Cc1ccnc(Cl)c1F)C2 c1(C(N2CC(F)(CNC(C3(Cl)C(C)(C)C3)=O)C2)=O)ccnc(-n2cccn2)c1 C(C(C(C)(C)C)NC(c1csc(C)c1)=O)NC(C1C(CC)C1)=O C12(C(=O)NC(C(C)C)C)COC(C1)C(NC(=O)C(C)(C)O)C2 C1(CNC(c2c(C)cno2)=O)CCCCC1.c1(C(=O)N)cc(C(C)(C)C)c[nH]1 Cc1c(CCc2nc(CCc3ccccc3)nn2-c2ccn(C)n2)cccc1Cl C1(CC(N2CCN(C(=O)CN(C)C)CC2)C(=O)NCCC)CCC(F)(F)CC1 c1(C(=O)OC)cn2c(CN3CCC4CCCC4C3)cnc2s1 C1(O)(C(C)NC(C(C2CC2)OC)=O)CCN(C(=O)CNc2ncccn2)C1 N1(C(CONC(c2n(C)ncc2Cl)=O)=O)CCC2C(C(N)=O)C2C1 N1(C(c2ccn(CC)n2)=O)CCN(C(c2cnn(C)c2Cl)=O)C(COC)C1 C(C(C)(C)CCNC(c1ccon1)=O)NC(CNC(c1c(C)onc1)=O)=O C1(CNC(c2coc(Br)c2)=O)C2CN(C(=O)C=C3CCCCC3)CC12 CC1(C)CCC(CC(N2CC=CC2C(=O)NCC(CO)C(F)F)=O)C1 C1(NC(c2scc(C#N)c2)=O)CC(NC(c2cc(Cl)cs2)=O)C12CCOCC2 C1(NC(CCn2cc(CN3CCN(C)CC3)nn2)=O)CCC(F)(F)CC1(C)C c1(C(N2CCCC(N(C(=O)CCC3CC3)C)C2)=O)c(F)cccc1Cl C1(NC(C(CC)(C)OC)=O)CCN(C(=O)C(CC(F)F)c2ccccc2)CC1F N1(C(C(C(C(C)C)O)C)=O)CCC2CCN(C(=O)CCc3cnc(O)[nH]3)CC12 C1(C(=O)NCCCC2(NC(C3C(C)(C(F)F)C3)=O)CC2)(CO)CCCC1 c1(CC)ccc(C(=O)NCC2CCC2)cc1N.c1(CCC(=O)N)cnc(O)[nH]1 N1(C(COCCCC)=O)CC(OC)C(c2cn(C3CC3)nn2)C1 C(CCCCCNC(=O)Cc1nccn1C)NC(C(c1cccnc1)N(C)C)=O C(=O)(C(CNC(=O)CO)N(C)C)N(C1(COC)CC1)C.c1ccsc1 C1CC2(CCC2)CN1C(=O)C=CC1CC1.CC(O)(CC(=O)N)c1ccccc1.C N=c1ccc(C(=O)NC2CCCC2NC(=O)C2=CCCOC2)c(Cl)[nH]1 c1(C(=O)NC2CCN(C(CCC#C)=O)CC2O)cc(C)nc2ccnn12 N1(C(CC(C(F)(F)F)NC(C(C(CC)O)(F)F)=O)=O)CC2OCCN(C)C2C1 O=C1CCCCC(C(=O)NC(CC2CC2)C(=O)NC2C3CCCCCC23)N1 N1(CC=C)C(=O)NC(c2cc(F)cnc2Br)C(C(=O)OCC)=C1C1CCC1 c1(C(=O)NCC2CCN(C(C(CCCC)O)=O)C2)c(F)ccc2cnn(C)c12 N1(C(CCC(=O)OC)=O)CC23CCCCC2(C1)CN(C(c1ncccc1F)=O)C3 Cc1conc1CNC(=O)NCC(F)(F)CO Cc1sc(C(N2CCC(NC(C3(C)CCCOC3)=O)CC2)=O)cc1CS(C)(=O)=O C1(CN(C(=O)CCOCC(F)F)CC)CCN(C(=O)Cn2ccnc2)CC1 Cc1nn(C)c(Cl)c1C(=O)NCC(C)NC(c1c[nH]nc1-c1ccoc1)=O C12(NC(c3cccc(CC)c3)=O)CCCC1CN(C(=O)C)C2.C(=O)C(C)CC.N C1(C2CC2)CCN(C(c2cc(=O)cc(Cl)[nH]2)=O)C1.C1(CC(=O)N)CCC(=O)N1 N1(C(C2N(CC)CCOC2)=O)Cc2cccc(CNC(c3ccns3)=O)c2C1 Cc1cc(C)n(-c2ccc(C(=O)N(C)CCN(C)C(c3oncc3C)=O)cc2)n1 C1(C(N2CC(OC)C(NC(=O)C(=O)N(C)C)C2)=O)(OC)CCCCCC1 c1(C(=O)OC)ccc(C(=O)NC2CCC(CC)C2)nc1.C(=O)C.C1CC1.N c1(C(N(C(CN(C(c2cc(CC)oc2C)=O)C)C)C)=O)cccc(F)c1F CCCC(C(O)C(=O)N1CC(c2ccccc2)C1)NC(=O)Cc1cc(C)nn1C C(=O)(C(C(C)(C)C)OC)N1CC(CC=C)(C(N2CCC(SC)C2)=O)C1 N1(C(c2n[nH]c(=N)[nH]2)=O)CCCC2(NC(=O)CCC3CC(F)(F)C3)CC2C1 N1(C(CC=C)=O)CCN(C(C2(C(F)F)CC2)=O)CC1C1CC1 C1(CNC(C2CCC(CC)CC2)=O)CN(C(=O)CSc2nncn2C)CCCO1 C(=O)(CCC(C)(C)C#N)NC(CCC)CNC(C1(O)CC2CCC1C2)=O c1(C(N2C(C)(COC)CC(NC(=O)C(C)(C)C#N)C2)=O)nc2cccnc2s1 c1(C(=O)OC)ccc(C(=O)NC2COCC2)cn1.c1(CC=O)cc(C)cs1.N C(=O)(C1=CCC(C)CC1)N1C(CC(=O)Nc2cnc(CC)nc2)CCCC1 C1(NC(c2n[nH]cc2Cl)=O)CC2CC(C1)CN(C(=O)C(F)(F)CO)C2 N1(C(CC(C=C)CC)=O)CC(NC(=O)Cc2csc3sc(C)cc23)C(N=[N+]=[N-])C1 c1(C=O)ccc(F)c(S(C)(=O)=O)c1.CC(C(=O)N)C1CCCC1.C(C)C1CC1 N1(C(c2cc(CC)c(F)cc2)=O)CCC2CN(C(c3ncc(CC)s3)=O)CC12 C1(C(=O)NCC2N(C(C(=Cc3cnc[nH]3)C)=O)CC2)CCCCN1C1CCCC1 C1(CNC(C(CC)CC)=O)CC2(CC(NC(=O)Cc3cncc(Br)c3)C2)C1 Cc1nc(C=CC(=O)NC2CC2)[nH]c1C.C1(C=O)CCCC(C(C)(C)C)C1.C c1(OCCC(=O)NC2(C)CN(C(C(CC)n3ccnc3)=O)C2)ccc(F)c(F)c1 C1(NC(CCN(C(c2nc(CC)sc2)=O)C2CC2)=O)CCN2CCCCC12 c1(C(=O)N)ccnc2c1ncn2C.c1(CC(C)C)ncc(C(=O)NC(C)(C)C)s1 C(=O)(C(CC)C(C)(F)F)Nc1cnn(CCC)c1C C#Cc1cccc(C(=O)NCC2CCN(C(=O)C=Cc3csc(C)n3)CC2C)c1 Cc1oncc1C(=O)NCC(=O)NC.c1(C(C(N2CCC2)=O)=O)cccn1C N1(C(c2csc(C)c2C2CC2)=O)CC2CCN(C(=O)CCC(F)(F)F)C(C2)C1 N1(C(CCn2ccc(C)n2)=O)CCN(C(C2C=CCS2)=O)CC1CCO N1(C(C(c2cn(C)nn2)NC(C(CO)OC)=O)=O)CC2(CCC(=O)O2)C1 C(C(C(F)(F)F)N1CCN(C(C2CC(F)(F)C2)=O)CC1)NC(CC1CC(C)C1)=O C1(C(C)C)OCCC1C(N1CC(O)(CCc2cn(-c3ccccc3)nn2)C1)=O N#Cc1ccccc1C(=O)NC1(C(=O)NCCC2(O)CCC2)CCSC1 C1(C(C(=O)NCCNC(CC)=O)C)CCN(C(=O)CCc2ccsc2)CC1 C(=O)(C(F)(F)C(F)F)N1CC(CCNC(=O)CN2CCCCC2CO)C1 c1(C(N2CC(CC(=O)O)OCC2)=O)ccc(O)c(F)c1 N1(C(C2CC(C)(C)O2)=O)CC(O)(C2CCN(C(=O)CCCN=[N+]=[N-])CC2)C1 CC(C)C(C)C(=O)N1CCN(CCCNC(=O)C2=C(Cl)CC2)CC1 c1(NC2CC(NC(C3(C)CC3)=O)C23CCC3)c(F)cc([N+](=O)[O-])cc1F c1(C(N2CC3(COC)CC2(C(=O)OC)C3)=O)ccc2c(c1)CCN2 Cc1oc(C(=O)NCC2CC(F)CN2C(=O)CCC2CCC2)cc1Br c1(OC(C)C)ccc(-c2ncccc2C(=O)NC2CCN(C(=O)CO)C2)cc1 CCCC(CC(C)C)C(=O)NCCC1(O)CCN(C(c2cc(O)n(C)n2)=O)CC1 c1(CN2CC3N(C(c4c(Br)cnc(C)n4)=O)C3C2)cccc2cc[nH]c12 c1(CCC)cccc(C(=O)NC(C)Cn2cc(C)nn2)c1.C(=O)(C(C)CF)N c1(OC)ccc(CC(=O)NCC2CC2)cc1.C1(C)(C(NC)=O)CCCO1.C C1(C(=O)NCC2CC(C#N)C2)CCC2CCC1N2C(=O)C(C1CCCCC1)O Cc1ccc(NC(=O)COC2CCC(=O)NC2=O)c(C=O)c1 N1(C(C2N(CC)CCC2)=O)CCCCC(C(=O)NCCC2CC=CC2)C1 Cc1csc2ncc(C(N3C4CCC3CN(C(C3(CO)CCCO3)=O)C4)=O)n12 C1(F)(CN(C(CC(=C)C)=O)CC)CCN(C(=O)C(CC)Sc2ccccc2)C1 C1(NC(Cc2cccc(C)c2Cl)=O)CCC(=O)N(C2CC2)C1=O c1(C(=O)NCCN(CCC)C(c2cnns2)=O)nn(C(C)(C)C)cc1Cl C#CCC(C)(C)C(=O)NCCCCCC(=O)N1CC2CCC1C2 C12(C(=O)NC(C)C=CC(=O)NCC3CNC(=O)O3)CCCC(CO1)C2 C(C)(C(F)(F)F)OCCNC(C(=O)NC(C)C(F)F)=O C1(CNC(C(N2CCOCC2)C)=O)CC2(CCN(C(c3csc(O)n3)=O)C2)CO1 C(CS(=O)(=O)c1ccc(Cl)cc1)NC(NC(C#C)C(C)(C)C)=NCCC(C)C c1(OC)ncccc1CN(C)C(c1coc(-c2nn[nH]n2)c1)=O C1(OCC)CC2CN(C(C3(C)CCCN3C(=O)C(C)COC)=O)CC12 C12(C(=O)NC(c3ccccn3)C)CCC(NCc3cccc(I)c3O)(CC1)CC2 C(C)(C)(C(C)NC(=O)CCN(C)C(c1ccnn1C)=O)OC N=S(=O)(CCNC(=O)CC1CC1(F)Cl)c1cccc(Br)c1 c1(CC)nc(C(=O)NC2CCOC2COC)c(N)s1 CCCC(CC)C(=O)NC1CN(C(=O)CCCn2ccnc2C)CC12CC2 c1(OCC)cnc(=NCC2CC2C(=O)Nc2ccc(Cl)c([N+](=O)[O-])c2)[nH]c1 N1(C(CC2CCN(C(C(C=C)(C)CC)=O)CC2)=O)CCC(C)(C2CC2)C1 CC1(NC(=O)Cc2ccc(F)c(Br)c2)CCCN(C(=O)CC#N)C1 c1(C(N(CC)C)=O)ccn(C)c(=O)c1.C(C(=O)N(C)CCO)(C(C)C)OC N1(Cc2c(C)nsc2C)CCC(NC(=O)CCCC2CCCC2)C(O)C1 c1(C(N2C(CCCNC(C(=O)NCC)=O)CCC2)=O)ccc(Cl)c(OC)c1F c1(NC(c2ccn(CCN(C)C)n2)=O)cc(Cl)c(F)cc1Cl C1(NC(CC2(CNC(CC(C=C)C)=O)CC2)=O)CN(C)CCN(C)C1 c1(C(=O)N)nccc2ncncc12.C1(OCC)CC(C(=O)NC2CC2C)C1 c1(C(=O)NC(CC=CC)C(=O)NC(C)C(C)C(=O)OC)ccc2cc[nH]c2c1 CC1CN2CCN1CC2C(N1CCC(NC(=O)CCCC2CC2)CC1C)=O C1(CNC(C(C)NC(C)=O)=O)CC(C)(C)CN1C(=O)C.c1nccs1.N C=CC(CCC)CC(=O)N(C)Cc1cccc(CNC(=O)CS(=O)(=O)NC)c1 N1(C(C2CC(C)N(C)CC2)=O)CCC2(CC1)CC(NC(=O)CC(=O)N(C)C)C2 C=CCCCC(=O)NC(C)(C)CNC(C1(C)CC1C)=O c1(C(N2CC3C4CCC(C4)C23)C(=O)NC)ccc(C#N)cc1F N1(C(c2scc(C)c2C)=O)CC(CO)C2(C1)CN(C(=O)CSCC(F)(F)F)C2 CC1CC(C(N2CCC(C(F)C(=O)N(C3CCOC3)C3CC3)C2)=O)CC(=O)N1 c1(OC(C)C)c(C(=O)NC2CCCCN(C(C3(Cl)CC3(C)C)=O)C2)cccc1N c1(-c2cn(CCC(=O)N(C3CCCCC3C)CC)nn2)ccc2cccnc2c1 C1(C(N2CCC(C(C)NC(=O)C=Cc3ccncn3)CC2)=O)CCCCC1(F)F CC(C)CC(O)C(C)C(=O)NC1CC2C(NC(C3C4CN(C)CC34)=O)C2C1 N1(C(CCCCOC)=O)CCC(C2CC2)(NC(c2cnc(F)c(C)c2)=O)C1 c1(C(=O)NC2C(NC(CCCC)=O)C2)oc2ccccc2c1Cl C1(CC(N2CCN(C(C(CC)NC(N)=O)=O)C(C)C2)=O)CCc2ccccc2N1 c1(CNC(CNC(=O)CCC2OCCO2)=O)ncc[nH]c1=O C1(NC(c2cc(Cl)ns2)=O)Cc2ccccc2C1NC(C1CC2CCC(C1)O2)=O N1(C(C2(CC)CC2)=O)CC2CC1C2NC(C1CC1CC(C)C)=O C1(NC(c2cc(C)nn2C)=O)CCCN(C(c2c(F)cccc2Br)=O)CC1 N1(C(c2c(COC)ncs2)=O)CCN(C(c2cn3ccnc3s2)=O)C2(CCC2)C1 Cn1cc(CC(N2CCC(C(F)CNC(C3CCC(O)CC3)=O)CC2)=O)c(Cl)n1 C1(C(=O)NC2(C)CCSCC2)CCCCCN1C(C1CC(=O)CCO1)=O c1(C(=O)NCCN(C(=O)C(O)Cc2ccccn2)C)cc(N)cc(O)c1F CC1CCC(C(N2CCC2C(=O)NCC=C2CCSCC2)=O)O1 N1(C(CN(C(C)=O)C)=O)CCCN(C(c2cocc2Br)=O)C(C(C)C)C1 c1(C(N(C(CCC(C)C)C)C)=O)cc2c(=O)n(C)c(=O)n(C)c2n1C C1(Cn2c(C)ncc2)COCCN1C(=O)C(C)NC(C1CCCCC1)=O C1(C(=O)NCC2CCC2C(=O)NCCOC(C)=O)(CC)CCC1 C1(C(N2CC=CC(NC(C(CC)(C)CC)=O)C2)=O)CCCC2(C1)CC2(F)F C(CC(C)(C)C)(C(=O)N1CCN(C)C(C#N)C1)NC1CC=C(C)CC1 c1(CC(N2C3CCC2C(O)CCC3O)=O)noc2ccc(F)cc12 c1(C(=O)OC)ccc(C(=O)NC(C)C(C)NC(c2ccc(C)cn2)=O)nc1 Cc1n[nH]cc1C=CC(=O)NC(C)CNC(C1CCCN(C)C1)=O c1(C(=O)NC2CCCN(C(C(C)CC(N)=O)=O)CC2)ccc2c(=N)[nH]cnc2c1 c1(C(=O)OC)nc(=NCCCCNC(=O)CNC(c2ccccn2)=O)cc[nH]1 CC(C)(CC(=O)NC(C)(C)CNC(=O)CCC(=O)c1cccs1)CC(F)F c1(C(N2CC(NC(C(CCCC)C)=O)C(O)CC2)=O)ccc2c(c1)nnn2C c1(C(C)C)cncc(C(=O)NC2CCC(NC(C3(C(C)C)CCCO3)=O)C2)c1 c1(C(=O)NC(C)C(C)C)ccnc(OC2CCOC2)c1.c1(CC=O)ccco1.N N1(C(CCCCN(C)C)=O)CCC(CNC(C2(O)CC(C)(C)C2)=O)C12CC2 CCCCCC(O)CC(=O)NC(C1CN(C(=O)CC2(N(C)C)CC2)C1)C C1CC2(CCC2)CN1C(=O)C.CC1=NOC(=O)C1CCC(=O)NC.CC(F)F Cc1cc(F)ccc1NC(=O)C(N1C(C)CCCC1C)=O c1(C(=O)NC(CNC(CCC=C=C)=O)C2CCC2)ccc2cc(O)ccc2c1 C1(C(N2CC(COC)OCC2)=O)CN(C(c2cc(F)cc(Cl)c2Cl)=O)CCC1(F)F N1(C(C(C)=C(CC)C)=O)CC(NC(C2CC2OC(C)=O)=O)CCC(O)C1 NS(=O)(=O)C(C(=O)NC)c1ccccc1.C1(C(N2CCC2)=O)CCCS1(=O)=O c1(N2CC(CC)OCCC2)[nH]c(=NC2CCOCC2)nc2sccc12 CC1C(NC(=O)C(CNC(=O)CC2OCCO2)N(C)C)CCCN1C c1(C(=O)NCC(CC)NC(c2coc(C)c2)=O)cnn2c1OCC(O)C2 C(CC1=CCN(CCn2cc(Cl)cn2)CC1)NC(CC1CCCC(C)C1)=O C(=O)(C#CC1CCOCC1)N1CCCC(CNC(C(C)n2ccnc2)=O)C1 c1(C(N2CCCC(N(C(c3cc(C)c[nH]3)=O)CC)C2)=O)ccnc2c1CCC2 S(=O)(=O)(c1ccc(NC2(c3ccc(F)cc3)CC2)nc1)NC1CN(C)C(=O)CC1 N1(C(CCCC)=O)CC2C3CCC(C2C1)N(C(c1oc(C2CC2)nc1C)=O)C3 N1(C(CCSCC)=O)CC2CC2(NC(C2CC=C(C)CC2)=O)C1 CCC(C(=O)N=c1cc2n([nH]1)CCCC2)N(C)C(c1cccn2cncc12)=O N1(C(C2(CC)CCCO2)=O)CC2(CCN2C(=O)C(C)C(=O)O)C1.C(C)(C)C N1(C(CC2CCN(C(C(C)OCCOC)=O)C2)=O)CCCC(N2CCCC2)C1 C(=O)(C1=CCCSC1)N(CCNC(c1nc(-c2cccc(C)n2)sc1)=O)C(C)C C(=O)(C1=NOC(CN)C1)OC(CC)C(=O)c1ccccc1 C1(NC(=O)CCc2ccccn2)CC2(C1)CC2C(N1CCCC1c1ncc[nH]1)=O CC(C)CC(F)C(=O)NCC1(C)CCN(C(C2(CF)CC3(CCC3)C2)=O)C1 C1(NC(c2ccc(Br)o2)=O)CCC2CN(C(=O)CCn3ccnc3)CCC2C1 N1(C(CCc2cn(CCN(CC)CC)nn2)=O)CC(O)C(O)CC(C)(C)C1 C(=O)(C1CCCc2nncn21)N(CCN(C(C1(CC)CCC1)=O)C)C(C)C O=NN1CCCC1C(=O)NC1CC(NC(=O)Cc2cccc(Cl)c2)C(O)C1 C1(C(=O)NCC2C(C(=O)NCCn3c(CC)ncc3)C=C2)CCCCC1 Cc1cc(=O)n(C)cc1C(=O)NC1CCCC1NC(=O)C(C)CC(C)(C)C C(=O)(CCCN(C)C(C1CC=CC1)=O)NC(C(=O)N(C)CC)C.CC c1(CCC(=O)NC2CC2C)ccccc1Cl.c1(C=O)cnn(C(C)(C)C)c1Cl.N N1(C(CNC(=O)Nc2c(C)nn(C)c2Cl)=O)CCc2sccc2C1 N1(C(COCC=C)=O)CCN(C(C2C3CCC2CC3)=O)C(C2CCCC2)C1 c1(C(=O)NCC(C)N(C(=O)CCC(=O)c2ccc[nH]2)C)cc2cnc(Cl)cc2s1 N1(C(C2C(C)N(C)CC2)=O)CC2(CC(NC(=O)CC3CCN(C)C3)C2)C1 C1(NC(C(n2ccc(C)n2)(C)C)=O)CCCN(C(c2cnc[nH]2)=O)CC1F N1(C(C(F)=C(C)C)=O)CC(CNC(=O)CCO)CC1C.C(C)(C)C.CC N1(C(C2CC(SC)C2)=O)CCN(C(=O)C(O)C(F)(F)F)CC1CC(F)(F)F C1(C=O)CCCCC(F)(F)C1.c1(C(=O)NCC2CCC2)ccncc1C1CC1 C1(NC(=O)CCN2C(=O)CCC2=O)CC2(CCN(C(C3CC4CCC3O4)=O)C2)C1 c1(CC(=O)N)cn2cc(C)sc2n1.C1(NC(c2cc(OC)n[nH]2)=O)CCCCC1 c1(C(N2CCN(C(C(CC)OC)=O)C(C)CC2)=O)cnn2cccc(OC)c12 c1(C(=O)NCC2C(C(N3CC(NC(N)=O)C3)=O)CCO2)ccn2cncc2c1 c1(OC(C)C)ccccc1C(=O)NC.C1CCN(C(C23CC(C)C2C3)=O)CC1.C C(=O)(CC1=CCCCC1)NC(C)C(=O)NC1CCN(C(c2cn[nH]c2)=O)C1 N1(C(CCC=C(C)C)=O)CCC(C)C(NC(c2cnn(C(C)C)c2C)=O)C1 C(=O)(C1=CCCC1P(C)(C)=O)N1C2C(C(=O)OC)(CCC2)CCC1 Cc1c(F)ccc(C(=O)N(CCCN(C(=O)CC(C)(C)C(F)F)C)C)c1O N1(C(C(C2CCC(C)CC2)CC)=O)CCC2CCC(C1)N2C(=O)C(C)C(C)C N1(C(C2CC(CN(C)C)C2)=O)CCC2(CCC2NC(=O)COCCF)CC1 Cc1cnc2n1CCC(C(N1CC3(CCC(CNC(C4CCC4)=O)O3)C1)=O)C2 N1(C(COCCSC)=O)CCCC(NC(=O)CNS(C)(=O)=O)CC1 c1(C(C)C)sc(Cl)nc1C(=O)N.C1(O)(CC)CCN(C(=O)CCC)C1.C(N)=O CC(C)CC(C(=O)N1CC(CO)C2(C1)CN(C(C1(C)CCC(C)C1)=O)C2)C(C)C c1(C(=O)NC(C(C)NC(=O)Cc2cn[nH]c2)CO)cc(Br)cn1C C1(NC(CCOCC)=O)(C)CCC(F)(F)CC1.c1(C=O)nc(C)n(C)n1.N CCCC(C(O)C(=O)NC(c1ccccc1O)C)NC(C1CCC(C)O1)=O Cn1cc(C(=O)NCC2CCCN2CCC2CCOC2)c(C(F)(F)F)n1 c1(NC(C2CC(F)CN2C(c2nccnc2Br)=O)=O)cccc(CO)c1F c1(CC)nc(C)oc1C(=O)NC1CCOC1C(=O)NCC(N1CCCC1)=O c1(N)ccccc1.c1(N2CC(COC)(NC(=O)CSC)C2)ccnc(OC)n1 N1(C(C(C)SC)=O)CCCCC1CNC(=O)CNC(C1CCC1)=O N1(C(c2ccn(CCC)n2)=O)CCC(C2CC2)(NC(=O)Cc2ccc(C)cc2)C1 C(C(CC(C)C)C(=O)Nc1cn(C2CC(N)C2)nn1)OC c1(C(=O)NCC(C2CC2)NC(c2cc(C)no2)=O)ccnc(-n2ccnc2C)c1 c1(OC)cc(CNC(C2CN(C(c3cncc(O)c3)=O)CCN2)=O)n(C)n1 c1(C(C(C)NC(c2cccc(OC(C)=O)c2)C(=O)O)O)c(F)cccc1Cl N1(C(c2cc(C(C)=O)on2)=O)CCN(C(=O)Cn2ncnn2)C2(CC2)C1 C(=O)(C(O)CC(F)(F)F)NCC1C(OCC)CN(C(CS(CC)=O)=O)C1 C1(C(=O)NC(CNC(c2ccc(CCC)s2)=O)(C)CC)Cc2cncn2C(=O)N1 N1(C(C(C(C)C)OC)=O)CCC2C(CCN2C(c2cccc(Cl)c2)=O)C1 N1(C(CN(C2CCC2)C)=O)CC2(CNC(=O)C=CC3CCC3)CCC1CC2 c1(C(c2nnnn2CC(F)F)NCCS(C)=O)ccc(F)c(Cl)c1 N1(C(CN(C)CC)=O)CCN(C)CC1C(=O)NC(c1nccc(C)n1)C N1(C(C(COC)O)=O)CCN(C(CNC(c2cccs2)=O)C(F)(F)F)CC1 N1(C(C2C(OC)C2)=O)CCOC2(C1)CN(C(c1ccc(N(C)C)nc1)=O)C2 C1(CNC(c2n(CC#C)cnn2)=O)CN(C(C2C3CCCC23)=O)CCN1C N1(C(=O)C=Cc2cccc(O)c2)CC2CC(NC(C34CCC(CC3O)C4)=O)C1C2 CC(C#N)CCC(=O)NC1(CNC(=O)CCS(C)(=O)=O)CCOC1 N1(C(C(CC)=CCCC)=O)CCC(NC(c2cc(C)cc(F)c2)=O)C(CO)C1 N1(C(CC=CC=C)=O)CC(NC(c2ncc(C)cc2Br)=O)CC(O)C1 c1(C(=O)NCC2C(NC(C3CCC(CC)O3)=O)CC2)cc(Br)nn1C Cc1ccc(NCC(=O)NCC2CC2NC(c2cnsn2)=O)cc1 CCC(C(N)=O)NC(=O)CC1CC1CNC(c1ncccn1)=O N1(C(c2cnc(C(C)=O)s2)=O)CC2(NC(c3cnsc3)=O)CCC1CC2 C(C)(CCC(=O)NC(CN(C)C)C(=O)N(C)Cc1cccc(C)n1)OCC C1(NC(c2cc(C(F)(F)F)n[nH]2)=O)CCN(C(=O)C(F)CC2CC2)C1 c1(CN(C(=O)CCOCCCNC(c2cccnn2)=O)C)cccnc1 c1(CC(N2CC(NC(C3COCCO3)=O)C(F)C2)=O)cc(O)cc(Br)c1 c1(C(N2C(CN(C(COCCCCC)=O)C)CCC2)=O)cc(C)cc(C)n1 C=CCN=C(NCc1cnn(CC(C)C)c1)NCC1CCCOC1C(C)C c1(C(N2CCC(NC(c3nc(C#C)sc3)=O)C(O)C2)=O)cc(OC)c(Cl)cc1Cl CC1(C)CC(CNC(=O)CCCCO)N(C(=O)CC2(C)CC2(F)Cl)C1 CC(C)(C)C(C(=O)NCc1cc(F)ccc1OC(F)(F)F)C(=O)O c1(C(=O)NC2(CNC(c3cc[nH]c3)=O)CCC2)ncccc1F CCC(F)(F)CC(=O)NC1C2CC(NC(c3cc(C4CCC4)no3)=O)CC12 Cc1ccc(C)c(SCC(=O)NC2CCN(C(c3ncc(Br)cn3)C)CC2O)c1 Cc1cc(=O)c(C(=O)NC2CN(C(=O)CCOC3CCOC3)CC23CC3)cn1C C12(C(=O)NC(CCN(C)C(C3CCCCC3(C)C)=O)(C)C)CCC(N=[N+]=[N-])C1C2 C1(NC(c2c(C)ccc(C(F)F)c2)=O)CC=C(C(C)C)CC1 c1(C(=O)NCC(C)NC(=O)CSC(F)F)n[nH]cc1-c1ccncc1 N1(C(C2CC3CCC2N3C(c2cccc(O)n2)=O)=O)CCc2ccccc2CC1 c1(C(=O)NCCN(C(C(C=C)C)=O)C2CC2)ccc(C)cc1N Cc1cccc(C)c1CNCCNC(=O)CC(=O)N.C1CCC(=O)NC1C.C C1(CNC(C(CC)SC)=O)CCCN(C(C2CCN(S(C)(=O)=O)CC2)=O)CC1 CC1(C2(C(=O)NCc3nocc3C(=O)NC3CCOCC3F)CC2)CC1 Cn1ncc([N+](=O)[O-])c1CNCC1CCC(c2ccccc2)C1 C=C(C)CCCC(=O)NCC1CN(C(c2cn(C)nc2Cl)=O)CCC1C C1(C(=O)OCC)N(C(C2CCCN(CC(=O)O)C2)=O)CC1(C)C N1(C(C(C)OCCC#C)=O)CC2C(CNC(c3cc(CCC)on3)=O)C2C1 C(=O)(C(C)C1CC1)N(C1CC(C#N)C1)CCOC.n1(CC=O)ccnn1 Cc1cc(CNC(=O)C(=O)Nc2nc(C3CCC3)cs2)nc(Cl)c1Br C#Cc1cncc(C(N2CC3CC3(NC(C3CS(=O)(=O)C3)=O)C2)=O)c1 C(CNC(=O)CCOCC1CCCO1)(N=c1nc[nH]s1)c1c(OC)cccc1 N1(C(C2C(CC)C2)=O)CC2CC(NC(c3occc3C)=O)CC2C1 Cc1nc2cc(C(N3CCC(C(C)NC(c4c(C)nsc4C)=O)C3)=O)cnc2[nH]1 c1(C(N2CCC2)=O)cc(Cl)nnc1O.c1(C(N(CC(=O)NC)C)=O)ccccc1 N1(C(C(C(C)C)C#N)=O)CCC2CC2(C(=O)NCC2(O)CCCCC2)CC1 c1(CNC(c2c(F)cc(Br)cc2Cl)=O)ccc(F)c(F)c1Br c1(CN2CCCC(CC(N3CCCC(C#N)C3)=O)C2)ccc([N+](=O)[O-])cc1O CC1(C)CC(C(=O)N2CC3(CC(NC(c4coc(O)n4)=O)CO3)C2)=NO1 S(=O)(=O)(c1ccn(C)n1)NCC1CN(Cc2cc(C)c(F)cc2)C1 C1(C(=O)NCCn2cccnc2=O)CC12CCN(C(C1CN3CCC1C3)=O)CC2 c1(OC)ccc(C(=O)NC2CN(C(=O)Cn3cccn3)CC2OC)c(F)c1 Cc1c(C(=O)NC2CCCCN(C(=O)C=CSc3ccccc3)C2)nn(C)c1N Nc1cccc(Cl)c1C(N1CC2(NC(=O)CN3CCC(O)CC3)CC1C2)=O C1(CC=C)(C(=O)NC(c2cnsc2)C)CCN(C(c2ncn(CC)n2)=O)C1 CC1(C)CCC(C(=O)NCCOCCCNC(c2sccc2Cl)=O)O1 C1(NC(C(C)NC(c2n(CCC)ccc2)=O)=O)CCCN(CCO)C1 c1(N2CC(CNC(=O)C(=O)NC3CC3)CC(C)(C)C2)nc2ccc(Br)cc2o1 C(C(=O)N1CCCO1)NC(C=CC(C)NC(=O)CN1CC2CC2C1)=O Cc1cc(C)c(C(=O)NC2CC(NC(=O)CN3CCC(C)C3)C2)c(C)c1 c1(C(=O)NCC(CCCC)NC(c2cncs2)=O)cc2c(C)nn(CC)c2s1 C1(CNC(C2CC(OCC)C2)=O)CCN(C(=O)C2=CCCCO2)C1(C)C C1(NC(CC2C(CC)C2)=O)CC12CCN(C(c1ccc(O)c(F)c1)=O)C2 N1(C(C(CC)N2CCCC2=O)=O)CC(NC(c2ccnn2C)=O)C2CCCC2C1 Cc1cc(C(=O)NC(C)(C)COc2ccccc2-n2cccn2)ccc1[N+](=O)[O-] Cc1cc(C(N2CC(CO)(NC(C3CC4CC3C3CC43)=O)C2)=O)c(C)cn1 Cc1cc(C(=O)NCc2ccc(C(N3CCC(O)C(O)C3)=O)s2)cc(O)n1 N1(C(c2cc[nH]n2)=O)CC(F)(F)C1C1CC1.CC(C)(C(=O)N)n1cncn1.C N1(C(COCCC=C)=O)CC2CC1CCC2NC(=O)C(c1cnn(C)c1)C C1(F)CCN(C(c2nnn(C)c2C(F)F)=O)C1.C(C(=O)N)(C1CC1)SC.C c1(OC)ccc2[nH]c(=NC(C)C)[nH]c(=NCC(C)c3cccs3)c2c1 N1(C(c2c(C)n[nH]c2)=O)CCC(C2CCN(C(C3CC(CF)C3)=O)CC2)C1 C1(NC(CC(=C)C)=O)CCCN(CCC(=O)NCc2ccc(CC#N)cc2)C1 C1(NC(CC(C)(C)OC)=O)CN(C(c2conc2C)=O)CCC1C(F)(F)F C(C1CCCc2nccn21)N1C(c2ccc(COC)o2)CCC1 CON(CCO)C(=O)c1conc1C(C)NC(c1n[nH]cc1Cl)=O n1(CCS(C)(=O)=O)nc(-c2ccc(SCC(F)(F)F)cn2)nc1C.C1CCOCC1 c1(C(N2C(c3ccc(OC)c(O)c3)SCC2)=O)nc2cc(Br)ccc2n1C c1(C2C(C(N3CCCC(O)(Cc4onc(C)n4)C3)=O)C2)cc(Br)cc(Br)c1N c1(C(N(C(CCNC(C(CC)(C)OC)=O)C)C)=O)nccc(Cl)c1F c1(C(C(=O)NCCO)N(C2C(C)CCC2)CC(C)(C)CO)cccc(F)c1I Cc1c[nH]c(C#N)nc1=NCC1(C)CCCN(C(c2cccc(Cl)c2)=O)C1 N1(C(c2ccc(I)cc2Cl)=O)CC2(CCN(C(c3cc(Cl)cnc3F)=O)C2)C1 Cc1c(C(=O)NC2CC23CC(NC(c2cnc(O)s2)=O)C3)cnc2ncnn12 Cc1nnccc1C(N1CCCCC1Cn1cc(C(O)C2CC2)nn1)=O C1(CC)C(C)CCN1C(C1CC(NC(c2ccns2)=O)C1)=O c1(C(N2CC(C(N3C(C(=O)OC)C3)=O)C(O)CC2)=O)c(C)ccc2ccccc12 N1(C(CCC(=O)NCC)=O)CC2CCC1C(C(=O)Nc1ccc(Cl)nc1)C2 c1(C(=O)NC(C(C)NC(=O)CN(CC(C)(C)C)C)CO)cc2n(c1)CCCC2 Cc1nc(C(C)C)sc1C(N1CC=CC(NC(=O)CC2CCOCC2)C1)=O N1(C(=O)C=CCO)CC(C2CCCN(C(c3cc(CCCO)on3)=O)C2)C1 C1(CNC(=O)CCCC2CC2)CCC2(CN(C(c3cc(Br)sn3)=O)C2)O1 CCCCCN(C(=O)CCN(C(=O)CCC1CCOC1)C1CC1)C C1(C(N2CCC(Br)CC2)=O)CNCCN1Cc1sc(Br)nc1Br C(C)(N=c1cc[nH]cc1S(=O)(=O)NCC1CCC=CO1)c1nc(C)sc1 C(C(C)(CC)NC(C1C=CCC1)=O)NC(C(=O)NCC)=O N1(C(CCS(C)(=O)=O)=O)C2CCC1CC(NC(=O)Cc1ccnc(Br)c1)C2 c1(NC(C2N(c3c(OC)cnc(SC)n3)CCC2)=O)ncnn2cccc12 C1(CNC(C(COC)C)=O)(NC(=O)C(C)SC(C)C)CCCCCC1 C1(C(=O)NC(CC)C(=O)NC2(CSC)CC(F)(F)C2)CCCCC1(C)C N1(C(CC2CC(CC)C2)=O)CC(N(C)C(c2csc(C(N)=O)n2)=O)C(O)C1 C(=O)(C#CC1CCCOC1)NCCC1(NC(=O)Cc2cc[nH]c2)CC1 C1(Nc2ncc(C)cn2)CCN(C(=O)CCCOC2CCOCC2)CC1C CC(c1ccco1)=CC(=O)NC(Cn1cncn1)C(=O)N.C1COCC1N(C)C c1(C(N)=O)cc([N+](=O)[O-])cnc1N1CC=CC(NC(=O)CN2CCC2)C1 c1(C(=O)NCCCNC(Cn2c(CCC)ncc2)=O)oc(CO)cc1C C(=O)(C(CC(C)C)C(C)C)N.N1(C(C(=Cc2cnc[nH]2)C)=O)CC(C)C(C)(C)C1 C1CCCN(C(=O)C(=O)NCCC2SCCS2)C1.C(C(=O)NC)=CC=CC Cc1cccc(C(F)(F)C(=O)NCC=CC)c1.C(c1cncn1C)=CC=O.N c1(CCC)cc(C(=O)NCC2CC2)nn1C.C1(C=O)CC(OC(F)(F)F)C1 C12(C(=O)NCC3CC(NC(=O)CC4CCCOC4)C3)CCCC(CO1)C2 C(=O)(CC1OCCc2sccc21)N1CCC(CNC(c2c(CC)onc2C)=O)C1 CN1Cc2cc(NCc3cnn(CC4CC4)c3)ccc2NC1=O N1(C(CCCC)=O)CC(NC(C2CC2C2CCC2)=O)CC2(CCOCC2)C1 c1(NC(CC)=O)nc(C)c(S(=O)(=O)NC(=O)C(N)C(C)SC)s1 CC(CN=c1[nH]c(N2CCC(=NO)CC2)nc2c1SCC2)Oc1cccc(F)c1 c1(C(N2CCC(C(=O)Nc3ccc(C(C)(C)C)nc3)C2)=O)cc(O)c(O)c(Cl)c1 N(C1c2cc(Br)ccc2CC1(C)C)C(CC(C#C)c1ccccc1)=O c1(C(=O)NCC(CN(C(C=Cc2nc(C)sc2)=O)C)O)cc2ccc(Cl)cc2o1 c1(C(N(C2CN(C(C3(C4CCC4)CCC3)=O)C2)C)=O)ccccc1S(C)=O N1(C(Cc2cccc(CC)c2)=O)CC2CCC(N(C(=O)C3=C(C)OCC3)C)C2C1 CCCC(C(=O)N1CCC(C)(NC(C2CC3(C2)CC3F)=O)CC1)S(N)(=O)=O c1(SC)ncc(C(=O)NC(C2CC(NC(C34COCC3C4)=O)C2)C)s1 c1(SC)cc(C(N2CCC(O)(Cn3cc(C4CCC4)nn3)CC2)=O)ccc1O C1(CC(=O)NCC#CCNC(CCCSC)=O)CCOC(C)(C)C1 C1(C=O)COC2CCCCC12.CC(C)C(C(=O)NCC1(C)CC1)n1cnnc1.N c1(C(=O)NC2CC(NC(C(C)(c3cccs3)N(C)C)=O)C2)ccc(Cl)cc1 c1ccc(C(=O)C(=O)N(C)CCN(C(=O)C)C(C)C)s1.c1ccon1.CC c1(CNC(C=C(C)C)=O)cc(C(=O)NC(C)C(C)n2cncn2)n(C)n1 C1(OC)CN(C(c2ccccc2-c2ncn(C)n2)=O)CC1NC(=O)CCCF C12(NC(COC)=O)CCN(C(c3cc(-c4ccccc4)c[nH]3)=O)CCC1C2 c1(CC)cn2c(C(=O)NCC3CCCN(c4nnc(CO)s4)CC3)cccc2n1 c1(C(=O)NCC2(COC)CCCN2C(C2CC2C)=O)cc2c[nH]nc2s1 C(CSC)(C(=O)N)NC(CNC(=O)OCC=C)=O.C1(CCC=C)CC1 c1(CN2C(C(=O)Nc3ccnn3C)CC(OC)C2)ccc([N+](=O)[O-])c(F)c1 CC1CC(C(=O)NC2CCN(C(c3sccc3C(F)F)=O)C2)CC(C)C1 CCC(C(=O)NC1(CSC)CN(C)C1)NC(=O)CCc1cscn1 Cn1cc2c(n1)CC(Cn1c(N3CCN4CCOCC4C3)nnc1CO)NC2=O n1(CC(N2CCC(C)(CNC(CCC(CC)C)=O)C2)=O)cc(C#N)c(O)nc1=O C1(CCC)CN(C(C2COCC2(C)C)=O)CCN1C(c1cnn(CCC)c1)=O c1(C(N2CCC(CC)C2CNC(c2cc(CO)on2)=O)=O)cnc(C)cc1C CC1CC(NC(=O)C=Cc2ccccc2)CCN1C(c1cc(Br)n(C)n1)=O Cc1ccc(=O)n(CC(=O)NCC2CN(C(c3ncncc3C)=O)CC2C)n1 C(=O)(CCCCC(N)=O)N1CC(CC(N2C(CC)CCOCC2)=O)C(C)C1 C1(NC(Cc2cccc(C(C)C)c2)=O)CN(C(c2csc(O)n2)=O)CC(C)(C)C1 N(C(=NCCc1ccccc1)NCc1nnn(C)n1)C(C)Cc1cccc(F)c1 N1(C(C(C)SCC)=O)CCC(C(O)CNC(=O)CN(C2CCC2)C)CC1 CCCC(CCCO)C(=O)NC(C1CCCN1C(c1cnn(C)n1)=O)(C)C c1(C(=O)NC2CC(NC(C3(C)CCCCC3)=O)C2)csc(N=S(C)(C)=O)n1 CC(C)C(C)CNC(=O)CCC1(NC(=O)C(C)CO)CCC1 c1(C(N(C(CNC(C(C2CCCC2)OCC)=O)C)CC)=O)ccncc1F.O Cc1ocnc1C(=O)NC(C)CCCNC(=O)CCc1cnc(C2CCC2)o1 CC1CCC(NC(c2ccnc(C3CC3)n2)=O)CN1C(=O)C=CC(F)F C1(C(=O)NCCCN(C(=O)CCc2cccc(O)n2)C(C)C)CN2CCC1CC2 CCC(C(=O)NC1CN(C(c2cnc(C3CC3)[nH]c2=N)=O)C(C)(C)C1)C(C)C N1(C(C(C)CBr)=O)CC2CCC(C1)N(C(=O)CCCc1ccccc1)C2 C(c1ccc(Cl)cc1)=CC(N1CC(NC(CCOCC(C)C)=O)C1)=O C#Cc1ccc(OC)c(C(=O)N(C2CCCC(NC(=O)C(F)=CC3CC3)C2)C)c1 c1(CC(=O)NCC2N(S(CC)(=O)=O)CCOC2)c[nH]c2ncccc12 C1(OC)CC(C(=O)NCCCCCNC(c2nonc2N)=O)C12CCC2 c1(C(N2CC(O)(CNC(c3cn(CCC=C)nn3)=O)C2)=O)ccn2ccsc12 C1(C(=O)N(C)OCC(F)(F)F)(CC)CCN(C(c2ncnc(O)c2F)=O)CC1 C1(CNC(c2cc(CC)co2)=O)CCC(C)CN1C(c1ccc(C)nn1)=O.C c1(NC(C2C(Nc3c(C(=O)OC)nsc3)C2)=O)cc(I)cnc1Cl c1(C(N2C(C)(C)CC(NC(C3CC3C(F)F)=O)C2)=O)ccc2cnccc2c1 N1(C(CSS(C)(=O)=O)=O)CCN(C(c2sccc2C(F)F)=O)CC1CCO c1(OC)ccc(C(N2CCCC2)CNCC2CCCN2C2CCCCC2)cc1 c1(C(CC)NC(=O)CC2CCCN2C(c2cnn(C(C)C)c2)=O)ccccc1Cl CC1CC=C(C(=O)NCC2CC3CCC2N3C(c2ccc(F)o2)=O)CC1 c1(C(C)OC(C2CC2c2cccc(Cl)c2)=O)ccc(C(F)(F)F)cc1 CCCCC#CC(C)(C)NC(C1C(C)CCN1C(=O)C=C1CCOCC1)=O C1(C(=O)NC(CC)CCCO)C2CCC(C2)N1C(C1(C(=O)N(C)C)CC1)=O c1(N(CCS(CC)(=O)=O)C)ccc(S(=O)(=O)N(CC(C)SC)C)c2ccncc12 N1(c2cncc(C#N)n2)CCC2(CCCN(C(=O)COC3CCOCC3)C2)C1 c1(NC(C2CCN(C(c3cnc(Cl)c(Cl)c3)=O)CC2O)=O)ncc(CO)cc1Br n1(CC)ccc2nc(NC34CCC(NC(c5cc(C)[nH]n5)=O)(CC3)C4)ncc12 C1(C(=O)N)CC2CCC1CC2.CC1(C)C(C(N2CCC(c3ccon3)C2)=O)C1C N1(C(c2c(CC)nc(C)nc2)=O)CCCN(C(=O)COC2CCCCC2)C(C)C1 C=CC(CC)CC(=O)NCC(c1ccc(C)cc1)NC(=O)CC(F)(F)Br C1(C)(CNC(COCCNC(COC(CC)CC)=O)=O)CCC(=O)N1C C1(C(=O)NCC2C(NC(c3cnc(Cl)s3)=O)CCCC2)CC2CCC(C1)C2 C1(C(N2CCC(CCC)C2)=O)CCCN(Cc2cnn(CC(F)(F)F)c2)C1 Cc1cc(C(=O)NCC#CC(=O)NOCc2ccc(O)cc2)ccc1C#N N1(C(C(C)(O)C2CC2)=O)CCC(NC(c2ccc(CO)c(F)c2)=O)C2(CCC2)C1 C1(C(N2C(C(C)(C)C)CCC2)=O)CC2(CCCC2)CO1.C(=O)(C1=CCCOC1)NC c1(CC(=O)NC(C(C)(C)C)CNC(c2cnco2)=O)ccc(Br)cc1C#N C=CC1CCN1C(C1CC(C)(NC(=O)CC(C)=C(C)C)C1)=O C1(C2CCN(C(=O)CCC3CCCCO3)C2)CCCCN1C(C1CC1(Cl)Cl)=O CC1CC(C(=O)NCCOc2ccccn2)N(C(=O)CC2CC(F)C2)C1 CC1(C#CC(=O)NC2CN(C(c3csc(-c4ncccc4Cl)n3)=O)C2)CC1 c1(C(=O)OC)cc(OC)ccc1NC(=O)CC1CN(C)C1.C1C=CCC=C1C c1(OC)ccnc(C(=O)NCC2CC(C)N(C(c3cnn4ccsc34)=O)C2)c1N C(=O)(C1=C(C#N)CCC1)N1CC(NC(C23CC(C)(CO2)C3)=O)CC(C)C1 Cc1nc2ccnn2c(C)c1C(=O)NC1(C)CN(C(=O)C(C)c2cc[nH]n2)C1 C(=O)(C(C)C(=O)N=c1[nH]n(CCCl)cc1C#N)c1ccc(C(C)C)cc1 C(=O)(C(CC)CCC)NCC1C(NC(CNC(=O)OCC=C)=O)C1 C(=O)(C(C)C1=CCCC1)NC1(CO)CN(C(Cc2cc(C)sc2)=O)C1 c1(OC(C(=O)NCCC)C)ccc(C)cc1.C1(=O)C(C)O1 N1(C(COCCCCC)=O)CCN(C(=O)C(c2ccncc2C)C)CC1COC C1(CCNC(C(F)OC)=O)CCN(C(c2c[nH]c(-c3ccc(Cl)cc3)n2)=O)CC1 C#CC(C)CN=C(NCc1cccs1)NCc1nccc(OC)n1 c1(C(C)(C)C)cccc(C(=O)NC2CN(C(=O)C(C)(F)c3ccccc3)C2)c1N C(C)(CN=c1[nH]c(C2CC2)nc2ccccc12)NC(C1(COC)CCOCC1)=O N1(C(c2c(CNC(C(C)C#N)=O)nnn2C)=O)CC(O)CC(C)(C)C1 C1(C(N(CCOCC)C)=O)CN(C(C2CC(C)N(C)C2)=O)CC1CC c1(CC)cnccc1C(=O)NC(CNC(=O)C(O)C(F)F)C(C)(C)C N1(CCNC(C23OC(C)C(C2)C3)=O)CCCN(C(=O)C(C)(C)CC#N)CC1 C1(CC)CCCCC1.C(CC=O)OCCCN(C(C1C(C(=O)OC)C1)=O)C.N C1(CC(=O)NCC2CC(C)N(C(c3cc(Cl)ccc3O)=O)C2)CCCC(C)(C)O1 c1(C(=O)NC2CCCC(C(N(CCCO)C(C)C)=O)C2)cnc2snnc2c1 c1(OCCC)ccc2c(OC3CC(Cn4ccnn4)C3)ccnc2c1 C1(C(=O)NC(C)C(C)Oc2ccccc2)CCN(Cc2cccs2)CC1 N1(C(c2c(CC)noc2C)=O)CC2(COC(C)C2)C1.c1(CC=O)cscn1.N CCC(C)(C)C(O)C(=O)NCCCN1CCC(NC(c2cnn3c2SCC3)=O)C1 N1(C(Cn2c(C(C)C)ncc2)=O)CCN(C(=O)C=CC2CC2)C(CCO)C1 c1(CC(C(=O)N(CCNC(CC(C)C)=O)C)C)cccc(Br)c1 C12(NC(c3cscn3)=O)CCC(C)(CC1)OC2.C1(C(=O)N)OCCOC12CCC2 c1(CN(C(=O)COc2ccc(F)cc2)CCOC)cccc(C)c1Br CCC(C)C(C)C(=O)NC1CCCC1CN(C)C(c1nc(C(C)C)oc1C)=O Cc1ccc(C(=O)N(C2CCN(C(c3cc(C(C)(C)C)nn3C)=O)C2)C)c(F)c1 C1(C(N(C2CCCN(C(c3cnc(O)o3)=O)C2)CCO)=O)CC12CC(F)(F)C2 c1(-c2cc(C(=O)Nc3c(C#N)n[nH]c3)c(F)nc2)ccc2occc2c1 c1(C(=O)NCC(F)C(=O)O)ccc2ccncc2n1 c1(C(N2CC3CN(C(=O)CN4CCCCC4)C3C2)=O)[nH]cc2c1CCC2 c1(C2C(NC(N3CCCC3Cc3csnn3)=O)C2)c(F)cccc1Br C1(NC(C(CC2CC2)NC(=O)COCC2CCCC2)=O)CC12CCOCC2 C12(CNC(CC(=O)OCC)=O)CCCC1CN(C(=O)CCC=CC(C)C)C2 Cc1ccnc(C(N2CCC(CNC(c3cc(I)c[nH]3)=O)C2)=O)n1 Cc1nc2c(O)cc(C(N3CC4=C(C3)CN(C(=O)CC=C(Cl)Cl)C4)=O)cc2n1C CC1(C(=O)NCC2(C)CCCC2)C=CCCC1.C1(C#N)(CC(=O)N)CC1 CS(=O)(=O)C1(C(=O)NC2CCOCC2NC(=O)CCc2cncs2)CCCCC1 O=C(C1=CCNC1)NC1CCC(NC(=O)CC2CC23CC3)C1.c1ccccc1.C c1(OCC#C)ccc(C(=O)OC(c2noc(CCC)n2)C)c(Br)c1 n1(CC)nc(C(N2CC(F)(C(=O)Nc3ccccc3F)C2)=O)c(C)n1 CC(C)CC(C(=O)NC(C)CCCCNC(C1CC(OC2CC2)C1)=O)C(C)C C(=O)(C#CC(C)(C)C)NC(C)C(C)C.c1(CC(=O)N)cc(C(F)(F)F)n[nH]1 C(=O)(CCCCNC(C1CC2(CC2)C1)=O)N(C(C1CCC1)C)C C1(C(=O)NCCC(=O)NCc2c(OC)nsc2)CC1C1CCCC1 c1(NC)cccc(C(=O)NCC2CCN(C(c3cnn(CC(F)F)n3)=O)CC2)n1 Cn1c(NC(=O)CNC(N2CCCC2)=O)nc2c(Cl)cccc12 c1(CCC)cnn(C)c1.N1(CC(=CC=O)C)CCCC1.C(=O)C=CC.N c1(OC)ccc(CNCC2CC(=O)N(C3CCCC3)C2)cc1OC1CC1 C1(C(N2C(C)C(C)(C)CC2)=O)CCN(C(=O)C(F)F)O1 c1(-c2cccc(SC)c2)cc2c(C(N3CCOCC3)=O)coc2cc1N C1(C(N(CC)C)=O)CC(C)=C(C)C1.C(C(=O)N(CCC)C)N(CC)C.CC c1(CC)c(C(=O)NC2CCCC2CNC(c2conc2C)=O)cnn1CC CC(C)C(F)(F)CC(=O)N1CCOC(CNC(=O)CCC)C1.C(=O)(C1CC1)N N1(C(C2CCCN(C(CN3CCN(C)CC3)=O)C2)=O)CCC2(CCOCC2)CC1 C=CC1CCN(C(c2cc(Cl)ccc2O)=O)CC1.N12CCCC(C1)C2=O C(=O)(CCS(=O)(=O)N(C)C)N(C)CC1N(C(C2C(CC)OCC2)=O)CCC1 Cc1cc(F)cnc1C(=O)N(CC(C)C(=O)Nc1ccc(O)cc1)C C(=O)(C(Cn1nnnc1C1(NC2CC2(C)C)CCC=CCC1)C(C)C)OCC CC1CCCC(C(N2CCOC(c3nc[nH]n3)C2)C(=O)NC2CCCC2)C1 c1(CN(c2nccc(C#N)n2)C2CCCNC2)cc(Br)cc([N+](=O)[O-])c1 N1(C(CC=C(C)C)=O)C(C(=O)NC(CC2CC2)CO)CC2CC12 C(=O)(C(C#N)C(C)C)N1C(C(N2CC(CC)(OC)C2)=O)CC=CC1 C1CCN(C(C2CCC(=O)N2C2CC2)=O)CC1.C(=O)(C(C)(Cl)Cl)NCC.C CCCC(CNC(=O)CCc1nc(O)n[nH]1)C(=O)NCCC(O)C1CCC1 c1(OC)cncc(C=CC(N2CC=C(C)CC2)=O)c1.C1(C(=O)N)CC12CCOC2 c1(C(C)C)cccc(C(N2CC3C(NC(=O)C(O)CCN(C)C)C3C2)=O)c1F c1(C(N2CCCC(CN(C(C3OCC(C)C3)=O)C)C2)=O)ccc2c(c1)CCC2=O C1(C)(C(=O)NCC2CN(C(C(C)C3CCCC3)=O)C2)CC(F)C1 C12(CN(C(CCC)=O)C)CC(CN1C(=O)CC(c1ccccc1)C1CCCO1)C2 c1(OC)ccc(F)c(S(=O)(=O)NC2C3CN(C(c4ccc(Cl)cc4)=O)CC23)c1 c1(NC(C2C=CC(NCc3c(C)cc(C)[nH]3)C2)=O)cnc(Cl)c(Br)c1C N1(C(Cc2cc(C)no2)=O)CC(=O)NCC1C(=O)NC1CNC(=O)C1 C(=O)(C(COC)CC(C)C)NC1CCCN(C(Cc2cc(COC)no2)=O)CC1 c1(OC)cc(C(=O)NC2CN(C(C3(Cl)CC34CCC4)=O)CC23CC3)ccc1C#N CC(CC#N)C(=O)NC1COCCC1NC(c1cccn1C)=O C[Si](C)(C)c1cccc(C(N2CCC(c3nnc4n3CCNC4)CC2)=O)c1 C1(N(C(CC(C)CN(C)C)=O)C)CN(C(=O)Cc2cnc[nH]2)CCC1O C1(C(=O)NCC2(C(N3C(CCC#C)CCC3)=O)CCC2)CCC(NC)CC1 C(=O)(CC1=CCN(C)CC1)NC(CCOC)CNC(c1nccnc1N)=O n1(CC(=O)NC2C(NC(COCC(C)C)=O)C2)cc(CO)nn1 C1(NC(c2cc(C)sc2C)=O)CCCN(C(=O)C(=O)Nc2ccccc2)CC1F c1(C(=O)NC2CN(C(c3ccnc(F)c3Br)=O)C2)cccc2nscc12 c1(NC(=O)NC(c2nnns2)C)cnccc1C(F)(F)F C(C)(C(CC(=O)NCc1cc(=O)cc[nH]1)NC(=O)CNC=O)OC.O CCC1c2ccsc2CCN1CC(=O)NCc1sc(C(F)(F)F)cc1C N1(Cc2n(C)cnc2)CC(C(=O)NCCc2ccco2)CC(F)C1 c1cc(C=O)ncn1.C(=O)C(C1CC1)C1CC1.CC(C)C.CCNCC c1(C=O)cc(C(C)=O)c[nH]1.C1(CC=O)CCN1C(=O)CCC1CCC1.CN c1(CC)nc(C(=O)NCc2cn(C3CCCN(C(=O)C(C)O)C3)nn2)c(Br)s1 c1(N2c3c(cc(OC)c(F)c3)CC2)[nH]c(=NC2CCC(C)(C)C2)nc2c1ncn2C c1(NC(C2C3(CCN(C(CCSC)=O)CC3)C2)=O)cc(S(N)(=O)=O)ccc1C CC(O)C(C)(C)C(=O)N1CC(C(C)(C)O)(CNC(=O)CC(F)(F)F)C1 C1(CC=C)(NC(C2CCC(CC)O2)=O)CCCN(C(=O)CCC(C)OC)C1 c1(NC(C(F)=C(C)C)=O)cccc(NC(c2coc(C(F)F)n2)=O)c1 c1(C(N2CCCC(C(C)NC(=O)C(F)=CCCF)C2)=O)cc2n(n1)CCCO2 S(=O)(=O)(c1ccc(C2(C(F)(F)F)CC2)cc1)NCc1cn(C(C)C)nn1 C(=O)(C1CCOc2ccccc21)N(C(CNC(c1cccc(OC)c1C)=O)C)C c1cccc(F)c1.C1(COC)(NC(=O)C(F)=CC2CC2)CN(C(=O)C)C1 C=CC(C)(CCOC)C(=O)N1CC2(CC(NC(c3cnn(C)c3F)=O)CO2)C1 C#Cc1ccc(C(=O)NC2CC3CC(NC(=O)C4CC4)CC23)nc1 c1(NC(C2N(Cc3c(C)nc(C)[nH]3)CC(C)C2)=O)cc(Cl)cc2[nH]ccc12 c1(OCC(=O)OC)cccc(C(=O)Nc2ccccc2)c1.C(=O)C(C)C.N CCC(C)CC(C(=O)NC(C)CC(C)(C)OC)NC(c1csnc1C)=O c1(C(=O)OC)cc(C)c2c(c1C)CCCN2C(=O)NCC1OCCC1(C)C c1(CCC)[nH]ccc1C(=O)NCc1csc(C(=O)NC(CO)C(C)O)c1 C=CC1COCC1NC(C1CN(C(c2cc(C)sc2C)=O)CC1CC)=O c1(OC)ccc(SC(C)C(=O)NC2CCCC2)cc1.C(=O)(C(C)N1CCC1)N N#Cc1cccc2c(C(=O)NCC3CN(C(C4CC5CCC4CC5)=O)C3)c[nH]c12 Cc1ccc2cnc(C(=O)NCC3(CCCNC(=O)C(N)=O)CCCC3)cc2c1 c1(NC(C2C(NC(c3cc(C)ncc3)=O)CCC2)=O)ccc(C)c(Br)n1 c1(CC)ccc(C(=O)NCCC(C)(C)C)cc1Cl.C(=O)CCCN(C)C(C)C.N C(=O)(C1=CCCC1C)NCCC(C(C)C)NC(=O)Cc1ccccc1.C(C#N)O C1(NC(=O)C2=CCSC2)CCN(C(=O)C(F)OC(F)(F)F)C12CCCC2 CCCC(F)(F)C(=O)N1CCC(C)(CC(=O)NCc2conc2C)C1 C1(SCCC)CCCC1.CCC=O.C(=O)CN(C=O)C1CC1.C(C)(C)C C1(C(N(C)C)=O)CCC(C(=O)N(C)C)CC1.C1CCN(C(=O)Cc2cn[nH]c2)C1 CCC(CC)(C(=O)NCCC(O)C(=O)N1CCC(CCO)C1)C(C)C c1(-c2nc(C)sc2)ccc2c(c1)CCN2C(=O)C(=O)NCC1CC1CF Clc1ccc2nc(CN3CCCCC3c3n[nH]cc3C(Cl)(Cl)Cl)[nH]c2c1 N1(C(C(c2cnn(C)c2)NC(C=CCCC)=O)=O)CC(C(N)=O)(N(C)C)C1 C(=O)(C(CCCc1ccccc1)N1CCC(F)C1)Nc1cccc(OC)c1 N1(C(C23CC(NC(c4nc(C)sc4)=O)(C2)C3)=O)CC2C(C)C2C1 c1(OC)c(Cl)ccc(C(=O)N)c1N.C1(CC)CCN(C(C2CC2)=O)C1.N(C)C C1(C(N(CCCNC(=O)CC2CC(F)(F)C2)C)=O)OCCCC1(C)C CC1(C)CCCOC1CC(N1CCCC1CCNC(=O)C(F)=CCCF)=O c1(C(N2CCC(O)(CNC(C(C=CC)O)=O)C2)=O)ccc(N)c2ncccc12 CN1CCCCC1C(=O)NCC1CC1C(=O)NCC(O)C1(Cl)CC1 C=CCC(CC(=O)NC(C)(CC)CCC)NC(c1ccc(CO)s1)=O c1(C(N2CCC(NC(C(C)O)=O)CC2)=O)ccc(F)c(O)c1 N1(C(C2(C(=O)NC)CCC2)=O)CC2(CC(NC(C3CC(OC)C3)=O)C2)C1 N1(C(C(CCCCC)O)=O)CCC(C2(O)CCN(C(c3ncccn3)=O)C2)CC1 C1(C(=O)NC(C=C)C2CCC2)CC(NC(=O)CCO)C1(C)C.C1CCCC1 N1(C(CC(C)C2CC2)=O)CC2CC(NC(=O)CCc3ccnc(Cl)c3)CC2C1 N1(CC)CCC(N=c2cc(C)[nH]c(=NCCC(C)(C)CC)[nH]2)CC1C Cc1ccc(C(N2CCC(Nc3nccc(-n4ccnc4)n3)C(C)C2)=O)nc1C N1(C(c2ccnc(C)n2)=O)CCC(CNC(c2coc(C3CCC3)n2)=O)C(C)C1 c1(-c2cccc(C(=O)NC3CN4CCC3CC4)n2)ccc(C(F)(F)F)cc1CO c1(C(=O)NCC(C)NC(=O)CCc2cccn2C)nnc2ccccc2n1 Cc1ncc2n1CCC(C(=O)NCC1CC1NC(=O)CC1CCN(C)CC1)C2 C1(O)(CCNC(C2(OC)CCCC2)=O)CCN(C(C2CC3(CCC3)C2)=O)CC1 C1(CC)CN(C(c2cc(C)nn2C(F)F)=O)CCC1.C1(CC=O)CC1(C)C.C c1(NC(C2CC(NC(c3csnn3)=O)C2)=O)cc(F)c(F)cc1I c1(C(=O)NC(C(=O)N(CC(C)CNC(=O)C=CBr)C)CO)cccc(F)c1 C1CN(C(c2nc(=O)n(C)[nH]2)=O)CC1CC(C)(C)C.C(C=O)(N(C)C)C1CC1 c1(COC(C(=O)NC(CNC(CCCC)=O)C2CCC2)C)ccc(C)cc1 C1(C(=O)NC(CC(C)NC(C(C=CCCC)O)=O)C)CCC(N=[N+]=[N-])CC1 Cc1ccc(O)c2c1C(C)CC2NCc1cccnc1Br Cc1cncc(C(N2CCC(CN(C(=O)C(=C3CCCCC3)F)C)C2)=O)c1C c1(C(N(C2CN(C(=O)Cc3ccn[nH]3)C2)C)=O)cccnc1 Cc1c(Cl)cnn1CC(N1CCCC(C(C)NC(C2(C3CC3)CCC2)=O)C1)=O N1(C(C(=O)NC)C2CC(OC)C2)CC(C(N)=O)CC(C)C1.C1CCO1 C(C)C(C)(C)CO.C(C(C(=O)N)n1cc(CCS(=O)(=O)N(C)C)nn1)OCC c1(C(=O)N)cnc(C(F)(F)F)c(F)c1.CCCC.C1(C=O)CC1C(F)(F)F Cc1cn2c(C)c(C(N3CC4CC(NC(=O)C5CC5)CC3C4)=O)nc2s1 N1(C(C(CCC)OC)=O)CC2CC(O)C1C2NC(c1cc(C(C)C)ccc1C)=O C(C)(CN=C(NCC(C)(C)C)NCC(c1cccc(C(C)(C)C)c1)O)OCC N1(C(C2C(CCC)C2)=O)CC2(COC(CNC(C3(C)CC=CC3)=O)C2)C1 c1(C(=O)NC2C(NC(CSCC)=O)C2)cccc2sncc12 c1(C(=O)OCCCOCCc2ccccc2)ccc2c(c1)S(=O)(=O)CCC2 CC1CCC(CCC(=O)NCC(C)(C)NC(c2ccnn2C2CCC2)=O)O1 N1(C(C(C(C)C)NS(CCCC)(=O)=O)=O)CCC2(CC1)CC2(CO)C.C(C)=O c1(N(C(c2ccc(C)nc2)=O)CC)cc(Cl)c(-c2cn(CC(=O)O)nn2)cc1Cl c1(N(CCCN(C(c2ccc(OCC)cn2)=O)C)C)nc2ccc(C)nc2s1 C(=O)(C(C(C)(C)C)NC(C1CCCN1C(N)=O)=O)NCCCCN=[N+]=[N-] CC1CCC(NC(c2cccn2C2CC2)=O)CN1C(c1cnccc1Br)=O c1(CCCC(N2CCCc3ccccc32)=O)ccc2c(c1)OCCCO2 Cc1ccn2ncc(C(=O)NCC(CNC(=O)CCC(C)(C)F)CO)c2c1 C1(NC(CC(C)N(C)C)=O)C2CC3C1C3C2C(=O)NC1CC1.N(C)(C)C CS(=O)(=O)c1cc(C(=O)NCCC2CCCN2C(C2CCC(=O)C2)=O)cs1 c1(C=O)ccc(C(=O)N(C)C)nc1.C1(CC(=O)NCC)COC(C)(C)C1 C(=O)(CCCCCC#N)N1CC(C)C(C(=O)NC2CCN3CCCC23)C1 C1(N(C(=O)CCC#N)CC)CCCN(C(=O)C(C)c2ccsc2)C1 c12cc3c(cccc3s1)[nH]c2=O.CC(C)CC(C)(CN(C)C)NC(=O)CC(C)F c1(OCC=C(C)C)cc(-c2ccc(N)c(OCC(=O)O)c2)cc(F)c1 CCCC(C(O)C(=O)N1CC(n2cnnn2)C1)NC(=O)C(C)(C)C(F)(F)F c1(C(=O)NC2C(CC)N(C(c3cscc3C)=O)CC2)[nH]cc2c1CCCC2 Cc1ccc(O)c(C(N2CCC(C)C2C(N2CCC(OC(C)C)CC2)=O)=O)c1 Cc1cc(C#N)cnc1C(N1CC2C(CC(=O)NC3CC(=O)N(O)C3)C2C1)=O CC1=C(C(=O)NC2CCN(C(=O)OC(C)(C)C)C23CCC3)CCCC1 C1(NC(c2ccc[nH]2)=O)CN(C(=O)CCc2cnc(O)[nH]2)CCC1C(F)(F)F Cn1cnc2cc(C(=O)NC3CCCCCN(C(C4CC=CCO4)=O)C3)ccc12 CCCC(C)(C)C(=O)N(C)CC1CN(C(C2CC(C)CO2)=O)CCO1 Cc1cc(Br)c(F)cc1CN1CCC(C(=O)OC(C)(C)C)CC1C N1(C(C(CCC)CNC(=O)CC2CCCOC2)=O)CCC(N=[N+]=[N-])CC1 C(CCCCCCC(=O)N1CC(O)(CNC(c2nn(C(F)F)cc2Cl)=O)C1)SC N1(CC)C2CCC1CN(C(=O)C(C)=CCNC(=O)CC1CCN(C)C1=O)C2 Cc1ccnc(CCNC(=O)C=CCN(C)C(C2(F)CCOCC2)=O)n1 c1(C(N2C(C)CC(NC(Cc3c(C)occ3)=O)C2)=O)cc(S(C)(=O)=O)cs1 CC(C)(C#N)CC(=O)NC1CCCC1NC(C1(c2ccc(Cl)cc2Cl)CC1)=O C(=O)(C(CO)C(F)(F)F)N(C(C(=O)NC1(CC)CCCCCC1)(C)C1CC1)C C1(CNC(CC(CC)C2CC2)=O)CN(C(c2ccc(Cl)cc2O)=O)C(C)(C)C1 n1(C(C(=O)NCC#CCNC(C2(COC)COC2)=O)C)cc2ccccc2n1 c1(C(=O)NC2CC(NC(CC3(NC(C)=O)CC3)=O)C2)cc(C)cc(Cl)n1 c1(N2CC(C)(NC(C3CCC(N=[N+]=[N-])C3)=O)C2)ncc2ccsc2n1 C(N=c1[nH]c2ccccc2s1)C1CN(C(c2cc(C3CC3)[nH]n2)=O)C1 c1(C(=O)NC2(CO)CCN(C(C(C)n3cncn3)=O)C2)ccc(C(F)F)cc1F CC(CCC(=O)NCC1CCC(NC(=O)C(C)(Cl)Cl)C1)N(C)C C(C(C)(C)C#CC(=O)NCc1ccc(C)s1)NC(c1c(CC)occ1)=O c1(Nc2ccc(-c3c(F)nc(C(F)(F)F)cc3)cc2)ncnc2c1CCC2 n1(C(C)C(=O)N2CC(N(C)C(C3Cc4nncn4C3)=O)C2)cnc2ccccc12 CC(C)CCC.C1(=CC=O)CCC(C)CC1.C1(C=O)CN(S(C)(=O)=O)C1.N c1(C(=O)NCC2C(C)C2C)cnc(CNC(=O)CC2CCCCN2C)nc1 Cn1c(O)nc(NCC(C2CC2)NC(c2ccon2)=O)c([N+](=O)[O-])c1=O N1(C(C2N(C(c3nc(OCC)oc3)=O)CCSC2)=O)CC2C(C1)C2(C)C c1cccc(Cl)c1.C=CC1(CC(=O)NC(C)CCN(C(=O)COC)C)CC1 CCCCCCCCC(=O)NC(C1CCN(C(C2(OCC)CCOCC2)=O)C1)C Cc1ccc(CNC(=O)C(CC2CC2)NC(=O)Cc2ccccc2F)c(C)c1 Cc1noc(C(N2CCN(C(=O)C(n3cc(Cl)cn3)C)CC2)=O)c1C C1(C(=O)NCCN(C)C(c2ccnc(C(F)(F)F)c2)=O)CCC2(CC2)C1 C1(CS(C)=O)CCN(C(=NCCC2CCSC2)NCCN2CCCC2)CC1 c1(OC(C)(C)C)cc(C(N2CCC(n3nccn3)CC2)=O)cc(Br)c1 O=C(CCc1ccc[nH]1)NN1CCCC1C(N1Cc2ccc(O)cc2C1)=O c1(NC2(C(F)(F)F)CC(F)(F)C2)cnc(N2CCOCC2)c(Br)c1 CCC(C)(CC)C(=O)N(C1CC(NC(C2(C)CCCOC2)=O)C1)C c1(NCCCN(C)C)ccc(S(=O)(=O)N)cc1Br.C1CCS(=O)(=O)C2(CCC2)C1 N1(C(c2scnc2C(F)(F)F)=O)CCc2ccccc2C1.[SH](=O)(=O)C(F)(F)F.N Cc1cc(OCC(O)CN2CCNC(=O)C2c2cccc(C)c2)cc(F)c1 N1(C(CSc2n(C(C)C)cnn2)=O)CCCC12CCN(C(=O)Cn1cccc1)C2 c1(CC(N2CC(C(C)C)C(NC(C3CC=CC3)=O)CC2)=O)nsc2ccccc12 N1(CC(=O)NC(CCNC(C(c2n(C)ccc2)=O)=O)(C)C)CCCCC1=O N1(C(CS(CC)(=O)=O)=O)CCC(C2CC(NC(c3c(Cl)cccc3Cl)=O)C2)C1 Cc1ccncc1C(=O)NCCC1CN(C(C2CNC(=O)C2)=O)CCO1 c1(C(N2CCCC(C)(c3nn[nH]n3)C2)C)ccc(C(F)(F)F)c(Cl)c1Cl CCCC(C(=O)N1CCN(CCNC(c2oc(Br)nc2C)=O)CC1)N(C)C C(CN=c1nc(N2CCC3(CC3)C2)c2ncccc2[nH]1)C1C2C=CC(O2)C1 O=[N+]([O-])c1cccc(S(=O)(=O)Nc2ccc3cc[nH]c3c2)c1 C(=O)(C(C(C)(C)C)NC(c1cc(=O)n(C)cn1)=O)NC(C)C(C)(C)C#N Cn1nc(C(N2CCCC2CNC(c2cccnc2SC(F)(F)F)=O)=O)cc1O C1(O)(CN(C)C)CCN(C(C(=O)NC2CC2)c2cnsc2)C1 C(=O)(C1CCSc2ccccc21)NCC(C)NC(c1ccc(F)c(F)c1)=O C1(C(N2C(C)(C(=O)NC)COCC2)=O)C2CCC(C2)C1.C(C)(C)C.C=O.N C1(C(N2CCC(C(C)C(=O)N(C(C)CO)CC3CCC3)C2)=O)CC(O)CN1C O=S(=O)(c1ccc2oncc2c1)NCC1CCCC1CF N1(C(CC2C(CC)C2)=O)CCC2CCCC12C(=O)Nc1ccc(SC)cc1 Cc1cccc(C(N2CCC(CCC(N3CC(C#N)C3)=O)CC2)=O)c1N Cc1cc(C(=O)NC2CN(C(c3csc(O)n3)=O)CC2C)cnc1C(F)(F)F CN1CC(C(=O)NCC(C2CC2)NC(=O)C(F)C2CCCC2)CC1=O C1(N(C(C(c2ccccc2)OC)=O)C)CN(C(=O)C=Cc2ccoc2)CC12CC2 N1(C(C2N(CC)CCC2)=O)CC(CO)C2(C1)CN(C(=O)Cn1[nH]cnc1=N)C2 CCCC(CNC(c1ncn(C)c1C)=O)C(=O)N1CC(O)(COC)C1 C(=O)(CS(=O)(=O)c1ccc(Cl)cc1)NCCNC(C1(C)Cc2ccccc2N1)=O C=CCCN=C(NCc1csc(N(C)C)n1)NCC(CC)C(C)(F)F C1(N(C)C)CCCN(CC(=O)NCC2(NC(c3cncnc3)=O)CC2)C1 CCC1=C(C(=O)N(C)CC2CCCN2C(C2C(C(C)=O)C2(C)C)=O)CCCO1 C1(O)(CCNC(C=CCC)=O)CCCN(C(=O)C2CC2)C1 Nc1cc(F)c(Br)cc1C(=O)NC1(CNC(C2CCNC(=O)C2)=O)CC1 C(=O)(CC(F)F)NC1C(NC(C2(C)CC2)=O)CC1 c1(C(N(CCNC(=O)C(c2ccc(F)cc2F)C)CC)=O)ccc2nnnn2c1 C(=O)(C(O)C(C(C)C)OC)N(CCN(C(C(CC)C1CCC(=O)N1)=O)C)C N1(C(C2ON=C(CC)C2)=O)CCC2C(NC(=O)C(C)Cn3ccnc3)C2C1 C1(CCNC(CC(C)SC)=O)CN(C(c2scc(C)c2C)=O)CCS1(=O)=O Cc1c(C(N2CCC3(NC(c4cnsn4)=O)CC3C2)=O)sc2nccn12 CC1SCCCC1C(N1CCC1Cn1cc(-c2cccs2)nn1)=O CC(C)CC(C(=O)NCC1(O)CN(C(=O)C(F)(F)c2cnnn2C)C1)C(N)=O Cc1cccnc1CC(=O)NC(C)(CNC(C1(C)CCNC1=O)=O)C1CC1 C1(NC(CC2CC(=C)C2)=O)CN(C(C2CC(F)(F)CS2)=O)CC1C1CC1 C12CCC(CN(C(=O)CC3CC=CCC3)C1)C2.C(C)(C(=O)N)N(CC)CC C=CCC(CNC(C1CCCC1C(F)F)=O)NC(C1CC(N(C)C)C1)=O C12(NC(c3cc(C#N)sc3)=O)CCC(C(=O)Nc3cnnc(Cl)c3Cl)(CC1)CC2 N1(C(Cc2cc(C)on2)=O)CC(C)(C)CC1CC(=O)NCC1CCOC1 C1(C)(OC)CN(CC(N2CCC(CCNC(=O)Cc3n[nH]cc3Br)C2)=O)C1 C(=O)(C(C)(O)CCN(C)C)N1CCC(F)(C(=O)NC(CC)COC)C1 c1(C(C)CC(=O)NCCN(C)C(C2CC(C3CC3)=NO2)=O)c[nH]c2ccccc12 c1(C(N2CCC3(NC(Cc4c(C)cccn4)=O)C(C2)C3)=O)cc(Cl)cc(Cl)c1N C1(C(=O)NC2CC2NC(=O)CCc2ccc(Br)cn2)(CC)CCNC1=O c1(CN2CCOCC(NC(c3ccccc3C3CC3)=O)C2)cc(Br)cc(Cl)c1O c1(C(N2CCN(C(CC)=O)CC2C)=O)cc(C#N)c(F)cc1F C1(C(N2C(CCNC(c3c(C)csc3)=O)CSCC2)=O)CCC2(CC1)CC2(F)F N1(C(CCC(=C)Cl)=O)CCCC(CO)(NC(c2ccnn2CCF)=O)C1 C1(CC)(NC(=O)CCCC2CCCC2)CCCN(C(=O)Cc2cc[nH]c(=N)c2)C1 Cn1ncc2c(NC3CSC3)[nH]c(=NC3CSC3)nc12 c1(C(N2CC(C)(C)OCC2)=O)cnc2c(c1)CCN(c1ccn3nccc3n1)C2 c1(C(=O)NC(c2c(C(=O)NC(c3nncs3)C)con2)C)ncn2ccccc12 Cc1cnoc1C1(C(=O)NCC2(NC(C3(C)CC3)=O)CCCC2)CC1 Cc1c(NC(=O)CC2CN(C(=O)C(C)C3CC3)C(C)(C)C2)cccc1C#N C1(C(N2CCC(C3N(C(c4c(C)onc4)=O)CCC3)C2)=O)CCCC2CC12 C12(NC(c3cn(CC(C)C)nc3)=O)CCCN(C(=O)Cn3cnnn3)CC1C2 c1(C=O)noc2c1CC(F)(F)CC2.c1(CC)c(C(=O)N(CC)CC)csc1C.N O=C(C(CO)C1CC1)NCC(F)CNC(=O)C(F)F c1(C(=O)NC2CN(C(C(COC)OC)=O)CC(C)C2)nc2cnccc2s1 c1(CNC(c2ccns2)C)ccc(C(=O)O)c([N+](=O)[O-])c1 C(=O)(CCCC(C(=O)NCCSC)N(C)Cc1cc(Cl)n(C)n1)OCC CCC(CC)CCC(=O)N(CC(C)NC(=O)C(F)CC1CCC1)C Cc1[nH]c2ccc(C(=O)NCC3CCN3C(c3cc(C#N)cs3)=O)cc2c1C C#Cc1cncc(C(=O)NC2(CC=C)CCN(C(=O)C(C)(C)N(C)C)C2)c1 N1(C(=O)NCCCOCC)CC2CCC1C(C)C2.C1(CC(=O)N)CCOC1 c1(C(N2CCC(N(C(COCC#C)=O)C)CC2)=O)cnc2ncnn2c1CC c1(C(=O)NC(CNC(c2cnn(C(C)C)c2Br)=O)(C)C)cc(F)ccc1F C1(NC(=O)CCn2cnccc2=O)CN(C(=O)C(O)C(F)F)C2(CCOCC2)C1 O=S(=O)(Cc1ccccc1)CCc1nnc(-c2ccc(O)nc2)n1C1CC1 c1(NC2CN(C(C3CC(C)C3)=O)CC2C)ccccc1[N+](=O)[O-] c1(N2CCC(P(C)(C)=O)C2)[nH]c(=NCC(F)CO)nc2scnc12 Cc1cccc(C)c1C(=O)N(C(C)C(=O)NCC1CC(F)C1)C1CC1.C C1(C(C)NC(c2occc2Br)=O)CCCCN1C(=O)CC1COC2CC1C2 N1(C(C2CC(OC)C2)=O)CCC(CNC(c2nn[nH]c2C(F)(F)F)=O)C1 CC1CC(C(=O)NCC(F)F)CCN1C(C1CCSCC1)=O CCCCC(O)C(C)C(=O)N1CC2CN(C(=O)CC(C)(C)C)CCC12 n1(CC(=O)OC(c2c(SC)cccc2)C)c(C)nc2ccccc2c1=O c1(OC)ccc(Cl)c(C(N2CCC(CN(C)C(c3coc(SC)c3)=O)C2)=O)n1 N1(C(c2n(CC)nnc2)=O)CC2CC(C1)CN(C(=O)C(C#N)CC1CC1)C2 C1(CNC(c2ccc(I)cc2F)=O)CCCC2(CNC2)O1 N1(C(C=CC(C)(C)C)=O)CCCC2(CCCCC2NC(=O)CN2CCSCC2)C1 C1(C(=O)NCc2cccc(CO)c2)CC12CCN(C(c1n[nH]c(O)n1)=O)C2 C(=O)(C(F)(F)c1cnn(C)c1)NC(CC)CN(C(=O)C(C)N1CCC1)C c1(C(N(C2CN(C(c3ccc(C)nc3C)=O)CC2F)C)=O)cc2c(ncn2C)[nH]1 C(=O)(C1CCCc2ccnn21)N1CC(CNC(=O)C2=CCOCC2)OCC1 N1(C(CC(C)(C)F)=O)CCC2(CCCN(C(C3CCCCC(=O)N3)=O)C2)C1 N1(CC)CCN(C(c2cc(C(C)C)on2)=O)CC1.CC(C)CCOC(C)C=O.N C1(NC(CN(CCOC)C(c2cncs2)=O)=O)CC(C)(C)C12CCC2 c1(C(=O)OC)oc(S(=O)(=O)N2CCC(N3CCCC3C)CC2)cc1C CC1(NC(=O)CNc2ncccn2)CC=CCC1 C1(NC(C(Br)=C(C)C)=O)CN(C(c2ccnc3ccccc23)=O)C2CCCCC12 C1CCC(C)(C)CN1C(c1cccc(C#N)c1)=O.C1(C(=O)N)(OC)CCOC1.C C(=O)(CC(C)C(C)(C)C)N1CC(CNC(c2ccc(C)nc2C)=O)C(C)C1 N1(C(=O)C=CC2CC2)CCC2CN(C(C3CCC(C(F)(F)F)O3)=O)CC2C1 C1(CC(N2CCCC(CC)(NC(c3ccc(Cl)o3)=O)C2)=O)CC2(CCCC2)CO1 N1(C(C2N(C(CC)=O)CSC2)=O)CC2CCC(C1)N2C(=O)C(O)C1CCCC1.O c1(C(=O)NC(C(C)NC(C2(C(C)C)CC2)=O)C(C)C)ncc(N)cc1Cl C1(C(=O)NCc2c(C)n(C)nc2)CC2CC1CN(C(c1csnn1)=O)C2 N1(C(CCCCC(=O)NC)=O)CCN(C(C2CCN(C)C2=O)=O)CC(C)(F)C1 c1(N2CCCN(C(CC(C)Oc3ccccc3)=O)CC2)ncc2c(ccn2C)n1 Cc1cccc(C(=O)NC(C)(C)CNC(=O)CC2OCCO2)c1Br CC(CC(C)NC(c1csc(C(C)(C)C)n1)=O)NC(=O)COc1ccon1 C1(NC(CSCC#C)=O)(CF)CCN(C(c2cc(OCC)n[nH]2)=O)C1 N1(C(c2ncc(C)nc2)=O)CC(CNC(=O)C(C)Cc2ccncc2)CC1(C)C C1(NC(C(C(C)C)OC)=O)CC2CC(C1)N(C(C1CCCC13CC3)=O)C2 C12(C(=O)NC(C)CNC(=O)CCN3CCCC3)CCCC1C2(F)F N1(C(c2c(C)oc(C)c2C)=O)CCC2C(CCCN2C(C23CC(C)(CO2)C3)=O)C1 C1(OCCOC)CCN(C(C(=O)N2CC(Oc3ccccc3)C2)c2ccsn2)C1 c1(OC)ccc(C(=O)NC2(C)CCOC2)cc1N.C1(C=O)CC(N(C)C)C1.N N1(C(Cc2c(C)noc2)=O)CCC(NC(c2ccc3c(c2)COC3)=O)C(C)(C)C1 C(CCCC(C)(C)C(=O)NNC(=O)CCC1OCCC1C)NC(CC)=O CC1CN(C(=O)C(O)CC2CCCCC2)CCN1C(c1csc([N+](=O)[O-])c1)=O c1(C(=O)N)ccc(P(C)(C)=O)nc1.c1(C(=O)NCCCC)cn(C)c(=O)n1C c1(C(N(C2(CC(=O)NC(c3cnn(C)c3)CC)CC2)C)=O)cc(F)c[nH]1 C1(NC(C(CC)COC)=O)CN(C(=O)CCCCc2cnc[nH]2)CC2(CCC2)C1 C1(OC)(CNS(=O)(=O)CC2CC(C(F)(F)F)C2)CCS(=O)(=O)C1 c1(COC)nc(NC2(C)CCCC2)cc(O)n1.c1(C=O)cc(C(F)F)ncn1 Cc1cc(C(=O)NCC(C)(CC(C)C)NC(c2cccn(C)c2=O)=O)ccc1O C1(C(=O)NCC(CCN(C)C)OC)(C(=O)N)CCCOC1.C1CCN(C)C1C C1(C(=O)NC2CCN(C(c3cc(C)n(C4CC4)n3)=O)C2)CCc2c(nnn2C)C1 c1(C(=O)NC(CNC(C(CC)N(C)C)=O)C(C)C)cc(N)cc2c1OCCO2 c1(C(=O)NC2C(CNC(C3(C)CCC3)=O)CCCC2)sc2ccccc2c1Cl c1(C(N2CCC(C)(CCNC(C3C(C)OCC3)=O)C2)=O)c(F)ccc(F)c1N C1(NC(CN2C(C)CCC2C)=O)CCC2CN(C(=O)CCCC3CC3)CC2C1 C(C(=O)N1CCC(C(=O)NCCc2noc(=O)n2C)O1)=C1CCC(C)C1 C(=O)(C#CC1CCCCC1)N1CC(C)C(CNC(c2nnc(O)cc2O)=O)CC1 N1(C(=O)NCc2n(-c3ccc(C)cc3)nc(C)c2)CCc2c(C)ccnc21 CC(C)(C#N)CCC(=O)N1CSCC1C(N1CCC(CCCO)CC1)=O C=CCC(C)(C)CC(=O)N1CCN(C(c2cnc(C(F)(F)F)s2)=O)CC1 N1(C(CC)CC)CCC(C(=O)N(c2ocnc2C)CCN2CCOCC2)CC1 C(CCCCC(=O)N1CC(N(C)C(c2cc(CC)nc(O)c2)=O)C2(CC2)C1)=CC c1(C(=O)NC(CNC(c2[nH]cc(C(C)=O)c2)=O)C)nc(O)[nH]c(=O)n1 S(=O)(=O)(c1cc(Br)cnc1Cl)NC(CC)C(C)C N1(C(C(C)=CC)=O)CCOC2CN(C(c3ccc(C(C)CC)cc3)=O)CC12 C(=O)(C1=CC2CCCCCC12)N1CC(CNC(c2ccc(SC)cc2Cl)=O)C1 C(=O)(CCC(C)(C)C#N)N1CCC(CNC(Cc2cc(C)sc2)=O)CC1 N1(C(CCc2n(C)cnc2)=O)CCC(N=[N+]=[N-])(C(=O)Nc2cc(O)cc(F)c2)C1 C1(C(=O)NCC2COCC2)CCC(F)CC1.C1(C=O)CCC(C(F)(F)F)CC1 C(=O)(N1CCC(C(N2C3CSCC2C3)=O)O1)C1(CC(C)C)CC1 N1(C(C(CC)N(C)C)=O)CCCC(C)(NC(c2cc(=O)c(OC)co2)=O)C1 c1(C(=O)NCC(C(C)C)(C)NC(=O)CN2CCCCC2)ccc2oc(S)nc2c1 C(N=c1nc2sccc2c(NC2CC2CC(C)C)[nH]1)c1ccc(SC)nc1 Clc1sccc1Cc1noc(CCc2nc(-c3cccnc3)no2)n1 C1(C(=O)NCCC(C)NC(c2ccccc2-c2ccncc2)=O)CCOC(=O)N1 C1(NC(C=Cc2scc(C)n2)=O)CC(NC(=O)CCc2cncnc2)C12CCC2 Cc1c(C(=O)N(C2CN(C(=O)C3=CCOC3)CC2O)C)noc1C1CC1 c1(OCCC)ccc(C(=O)NC)cc1.C1CCN(C(c2cnn(CCF)c2)=O)C1 c1(CN2C(C(=O)NCCc3ccccn3)C3CCC2C3)c[nH]c2ncc(Br)nc12 CC(c1ccccc1)=CC(=O)NC1CCC1NC(C1(C)CCC(=O)C1)=O NS(=O)(=O)c1c[nH]c(C(N2CCOCC(F)(CNC(=O)C3=CCOC3)C2)=O)c1 CCC(C)(C)C(O)C(=O)N1CCC(O)(CNC(=O)Cc2ccc(C)cc2F)C1 C1(C(N2CCC3CCN(C(C45CC(CO4)C5)=O)CC23)=O)CCOC2(CCCCC2)C1 C1(OC)CCC(C(=O)N(CCCNC(=O)CC)C2CC2)C1.c1ccccn1.S C1(n2cnnn2)(CNC(C2(Br)C(C(=O)O)C2)=O)CCCCC1 c1(C(=O)NCC(CC=C)NC(=O)C(c2ccccc2Br)O)cc[n+]([O-])cc1 N1(S(CC(C)C)(=O)=O)CCCC(O)(CNC(C2(Br)CCC2)=O)C1 C1(NC(=O)C=Cc2cncs2)CN(C(c2cn(C3COC3)nn2)=O)CC12CCC2 CCCC(CCCNC(=O)CC1CC(C)=NO1)NC(=O)CCC(F)(F)F c1(CC)ncc(Cl)c(C(=O)NCC(C2CCOC2)NC(c2cnccc2Cl)=O)n1 C(=O)(C(C)(C(C)C)OC)NCC(c1ccc(F)cc1)NC(C(C)=CC)=O c1(C(N2CCC(CC(=O)NCC=C)C2)=O)ccc(O)cc1 Cc1nc2n(n1)CC(NC1(c3nnnn3C)CCCCC1CNC=O)CC2 CC(C)(CC1CC1)C(=O)NCC1CCC(C(=O)NC(c2ncc[nH]2)CO)C1 C1(NC(CCC=C)=O)CN(C(C2(COC)CC=CCC2)=O)CC1C C(=O)(CCC(C)(C)C)N.c1(C(=O)NC(COC)C2(C)CC2)coc(C)c1 N1(C(COCCOC)=O)CCN(C(C2OCCCC2(C)C)=O)C(CO)C1 C(CNC(c1cscc1C)=O)(CCNC(C1CCOC1C)=O)OC C12CC(O)C1CC(=O)N1CCC(C1)C(=O)N2.C(COC(C)=O)=CC N1(C(c2cc(SC)c(N)cc2)=O)CCCC(NC(c2cnoc2C)=O)C(F)C1 C1(NC(COC)=O)CCSC12CN(C(=O)C(n1cnc3ccccc13)C)C2 C1(C(=O)NCCN2CCN(C(CC3(C)CCCC3)=O)CC2)Cc2cccnc2C1 N1(C(c2c(CC)n[nH]c2)=O)CC2CN(C(=O)CC3CCCN(C)C3)CC2C1 Cc1cc(=O)n(C)nc1C(N1CCC2C(C1)CN2C(c1cc(F)ccc1F)=O)=O c1(C(=O)NCCCC2CCCN2C(C2(F)CCCC2)=O)coc2c(Cl)cccc12 CCCC(C(=O)NC1(CCNC(C2CC3CC23)=O)CCC1)N(C)C N1(C(c2n(C)cnc2)=O)CCN(C(=O)COCCF)C(CC(F)F)C1 C1(C)(N(CCC)C)CCN(C(C2C(CC)CCN2C(=O)C(CC)CC)=O)C1 Cc1cc(C=CC(=O)NC2CC(C)N(C(c3oncc3C)=O)C2)ccc1F C(CCCCCNC(=O)CSCCC#N)N(C)C(c1coc(C2CCCC2)n1)=O C1(C(=O)NCC2C(NC(c3c(C)n(C)cc3)=O)CCC2)CCc2ncc(C)n2C1 c1(C(N2CC(N)CC(C)C2)=O)cc(Br)c(F)cc1Cl c1(C(N2CC(NC(=O)C=CSc3ccccc3)C(O)C2)=O)cc2c(o1)CCCC2 N(C1CCCn2ccnc21)C(C1C=CC(NC(CSCCOC)=O)C1)=O C=CCC(CC)C(=O)NCC1(C(=O)NC2CCN(C)CC2C)CCC1 c1(NC(CC(COC)NC(CC=CCC)=O)=O)ccc(O)c(=O)cc1 C(=O)(C(C)(C)CC(C)C)N(CCC)C.CCCC(C=O)NC(=O)O.C(C)(C)C c1(C(C)=O)c(C)cc(NC(=O)C(N2CCC(Sc3ccc(Br)cc3)C2)=O)cc1C N1(C(c2cnc(O)[nH]2)=O)CC2CCC(C1)N(C(=O)CC1Cc3ccccc3C1)C2 C(=O)(C(F)CCC(C)C)NCC1(F)CN(C(c2ccc(CCCCCC)s2)=O)C1 Cc1nn(C)c(C)c1OCC(N1CCCC(C(N2CC3C(C2)C3(F)F)=O)CC1)=O C1(NC(C(C)CC(F)F)=O)CCCCCN(C(c2cnnc(O)c2)=O)C1 c1(C(N(C(CNC(C(C2CCOC2)OCC)=O)C)C)=O)cc2cc(N)ccc2s1 c1(C(=O)NC2C(NC(CC(C=C)CC)=O)CCC2)ccc2cnn(C)c2c1 c1(C(N2CC(C)CC(NC(CNC(=O)NC)=O)C2)=O)cc2ccncc2s1 C1(C(N2C(CCNC(=O)CCC3CC3(Cl)Cl)CCC2)=O)CC2(CCOCC2)CO1 C(=O)(CCC(C)(C)[N+](=O)[O-])N(CC(CNC(C(n1ccc(C)n1)C)=O)(C)C)C C1(CNC(c2cccc(S(=NC)(C)=O)c2)=O)CCC2(CCCCCCC2)O1 C1(C(=O)NCC(C)NC(c2cc(C)n(C)n2)=O)(OC)CCC12CCC2 c1(CC(=O)NC(CCN(C(c2c(C)cc(C)o2)=O)C)C)cc(F)cc(Br)c1 C(CCCC(=O)NC1(C)CC1C)N(C(C(C)=CC=C)=O)C Cc1nsc(C(N2CCSCC2C(=O)NCCN2CCCCC2=O)=O)c1N c1(C(=O)NCCCN(C)C(c2ccc(-c3cnc[nH]3)cc2)=O)csc([N+](=O)[O-])c1 N1(C(C(CN(C)C)O)=O)CC(CNC(=O)CC2(O)CCC2)C(F)(F)C1 C1(C(N2CCC(CCNC(C3C(C)C3C)=O)C2)=O)Cc2cscc2C1 C1(NC(Cc2c(C)n(C)cn2)=O)CCN(C(=O)C(C)C(C)C)CCC1(F)F N1(C(c2c(C(C)C)ncnc2)=O)CC2CCN(C(=O)Cc3nn(C)cc3Cl)C2C1 Cc1nn(C)c(C(=O)NCC23CCC2CCN3C(c2ccc(N)c(F)c2)=O)c1Cl c1(C(N2C(C(N)=O)CC(O)CC2)=O)ccc(Cl)c2c1CNCC2 c1(C(=O)N)cc(Cl)cc(Cl)c1Cl.c1(OC(C)C(=O)NCC2CC2)ccccc1 c1(C(C)C)nc(N2CCC(CNC(=O)C(c3cccc(F)c3)C)CC2)cc(Cl)n1 c1(CC(=O)N(C2CCCN(C(C3C(C)C3C)=O)C2)C)cc(F)c(F)cc1F c1(CC=O)cc(C)cc(C)c1.N1(CC(=O)N(CCC)CC)CCC(C)(O)C1 CC(C)(O)C(C)(C)CNC(=O)CC1(C)CC1.C1(C(=O)N)CCC(O)C1 c1(C(N(CC(C)C(=O)O)CCOC)=O)cccc(-n2cccn2)n1 N1(C(CC=CCC)=O)CCc2cc(C)ccc2C1.C1(F)(C=O)CCS(=O)(=O)C1.N N1(C(c2n[nH]cc2Cl)=O)CC2C3CCC(C2C1)N(C(c1ccc(Cl)cn1)=O)C3 C#CC1CCCC1NC(C1CCOC1CNC(C1SCC=C1C)=O)=O CC(=O)CCCCC(=O)NC(CCF)C(=O)NC1CC2CC1C(O)C2O C1(NC(C2N(C(C)=O)CCOC2)=O)CC2CC1N(C(c1cnc3sccn13)=O)C2 c1(C(N)=O)csc(C(=O)NCC#CCNC(=O)C(O)C2CCCC2)c1 C=C(C)CN=C(NCC1(SC)CCN(C)CC1)NC(C1CCOC1)C N1(C(C2C(NC(C3(C)CC(C)(C)C3)=O)CCO2)=O)CCC2(CC1)CC2 c1(C(=O)NC2C3CC(NC(=O)CC4CCCOCC4)CC32)cc([N+](=O)[O-])c[nH]1 C1(NC(COCCC)=O)CCCC2CN(C(c3ccnc4[nH]cnc34)=O)CC12 C1(CNC(C2N(C(C)C)C(=O)CC2)=O)N(C(C2CCCSC2)=O)CCCC1(C)C Cc1cc(Br)cc(C)c1CNC(=O)C(c1c(Cl)cccc1Cl)C C1(N(C(C2CCCS2)=O)CC)CCCN(C(c2cc(-c3ccsc3)on2)=O)C1 C1(C(N2CCC(NC(c3c(C)nn(C)c3F)=O)CC2)=O)OCCOC12CCC2 CCC(C)CC(C(=O)NC1CN(C(N)=O)C1)NC(c1ccc(F)cc1F)=O N1(C(CCSCC)=O)CC(F)CC1CN(C)C(c1cc(COC)cs1)=O N1(C(c2csc3nccn23)=O)CCC2(CC1)CN(C(C1C(F)(F)C13CC3)=O)C2 N1(C(CSCC#C)=O)CC2=C(C1)CN(C(c1ccc(C(N)=O)o1)=O)C2 c1(NC(C(C)C)CNC(c2ccc(C3CC3)o2)=O)cc2c(cn1)C(=O)CCC2 N1(C(c2cc(=NC)[nH]cc2)=O)CCCC12CCN(C(=O)CC1CC1(C)C)CC2 C1(OCC)COCCC1CC(=O)NCC1CN(C(=O)C)CCO1.C(C)=O.O C(=O)(C(O)CCc1ccccc1)NC(C)CCN(C(=O)COC1CCCC1)C C1(CNC(=O)Cn2nccn2)C2CCC(C2)N1C(c1ccoc1Cl)=O CC(C)C(CC(=O)N1CCC(F)(F)CC1)NC(=O)C(O)CC(C)C c1(C(=O)NC(C)(CNC(C2(C3CC3)CCCO2)=O)C2CC2)ccsc1C#N c1(C(=O)NC2CCC(N(C(c3ccc(C)s3)=O)C)C2)ccc2c(c1)CCOC2 c1(SC)ncc(C(=O)NCCCOCCNC(C2(O)CC2(C)C)=O)s1 C12CCCC1CN(C(=O)C=Cc1cnccn1)C2.O=C(COCC1CCC1)N N1(C(C)=O)CS(=O)(=O)CC1C(=O)NC1CCC1NC(=O)C1=CCOC1 N1(C(C23C(CN(C(C4(C(C)C)CCC4)=O)C2)C3)=O)CCCC2OCCC12 N1(C(C(CN(C)C)NC(c2ncn(CC)n2)=O)=O)CC(OC)C(NC)C1 c1(CC(=O)NCC2CCC(NC(Cc3cnc(C)[nH]3)=O)C2)n[nH]c2c1CCCC2 C1(CC)CCCCC1C(=O)NCC(=O)NCC(=O)NCC1(C#N)CC1 c1(OC)ccnc(C(=O)NCC2CC(O)CN2C(c2cnc(S)n2C)=O)c1C c1(NC(C2C3CN(C(CSc4ccc(C)cc4)=O)C2C3)=O)cnc(O)nc1O N1(C(c2ccn(C)n2)=O)CCC(NC(c2ccncc2F)=O)C(O)C1 C(=O)(CS(=O)(=O)C1CC1)NCCNC(c1c(Br)nc(C)s1)=O N1(C(c2cc(CC)no2)=O)CCC(CNC(=O)C(C)CC2CC2)C12CCC2 N1(C(=O)NC2C(C)CCOC2)CCCC2CCNC(=O)C12 c1(OC)cc(SC)ccc1C=O.C1(O)(CC)CCN(C(C2CC(F)C2)=O)CC1.N S(=O)(=O)(CCC(=O)NC1CCCCC1NC(=O)C(Cc1ccccc1)O)NC N1(C(c2c(OC)n[nH]c2)=O)CCCC2C1CCN2C(c1ncsc1C)=O c1(C(N2CCN(C(C(=O)N)=O)C(C3CC3)C2)=O)c(Cl)c([N+](=O)[O-])nn1C.CC N1(C(c2c(CC)nc[nH]2)=O)CC=C(CNC(c2ccc(C)n2C)=O)CC1 C(=O)(C1CCOc2c(F)cccc21)NCC(C)NC(C1(NC(C)C)CC1)=O c1(C(N2C(CNC(=O)Cc3cccnc3Br)CCC2)=O)ccc2c(c1)NCC2 N1(C(CC(C)SC)=O)CC2(CCOCC2)CC1CNC(=O)CC.CCN(C)C Cc1ccc(Br)c(C(N2CC(NC(=O)C(C)(C)CCl)C(F)C2)=O)c1F O=S(=O)(c1cccc(=NCC=C2CCSCC2)[nH]1)N1Cc2ccncc2C1 c1(OC)cc(C)cc(C(N2CC3CC2CN3C(C2(CO)CC(F)(F)C2)=O)=O)c1N C1(OC)CCC2(C(=O)NC3C4CN(C(C5OCCC5(C)C)=O)CC34)CC12 c1(C(=O)NC2C3CN(C(c4c(C)nn[nH]4)=O)C(C3)C2)cc2ccccc2[nH]1 c1(C(N(C2CCC(NC(c3cccc(C)n3)=O)C2)C)=O)cc(C2CC2)cc(F)c1 c1(OC)ncccc1S(=O)(=O)N1CCCC1(C)C(N1CCN(C(=O)C(C)C)CC1)=O Cc1ccc(C(CNC(=O)C(C)CC2CC2)NC(c2ccc(F)cc2)=O)cc1 C(=O)(CC(C(F)(F)F)NC(=O)CC(C)CC)NC(CCCCC)C1CC1 C1CCCN(C(=O)CC2CCC(C)(C)C2)C1C(=O)NC.C1(O)CN(C)C1.CC N1(C(Cn2cc(CNC(CCc3ccn(C)n3)=O)nn2)=O)CC2CSCC2C1 N1(C(COCC=C)=O)CC2(CCCC2NC(c2cc(C)[nH]n2)=O)C1 C1(C)(C(=O)Nc2c(CC)n(C)nc2)CCN(C(c2ncoc2C(C)C)=O)CC1 c1(OC)ccc(CC(N2CCC(C)(NC(=O)CCCCCSC)C2)=O)c(Cl)c1 n1(CC(=O)NC23C(CN(C(CC4C=NN(C)C4=O)=O)C2)C3)cnc2c1CCCC2 N1(C(CC(=O)N)=O)CCC2(CC1)CC(NC(c1nc(Cl)cs1)=O)C2.CC(F)(F)F c1(C(C)C)ncncc1C(=O)NCC(C)CNC(C1CCCN1C)=O CCCCCCC(C)CC(=O)NCCN(C(c1ccc(F)c(C)c1)=O)CC1CC1 c1(-c2n(CCC)nc(C)c2)ccc(C(=O)NCC2CCC(F)C2)c(C)c1F c1(C(=O)NC2(COC)CN(C(=O)C(C)C)C2)sc(C(F)(F)F)cc1C.S c1(OC)ccc(C(=O)NC(C)(CNC(c2nnsc2)=O)CC(C)C)c(C)n1 C1(C(C)(F)F)(C=O)CCOCC1.c1(C(N2C(CC)CCC2)=O)cc(CN)c[nH]1 Cc1cnc(C(=O)NC2CCC(NC(=O)C=Cc3ccoc3)C2)cc1C C12(C(=O)NC3C(NC(c4c(C)occ4)=O)CC3)CCCCC1C2Br CCCC(C(=O)N1CC2CC2(CNC(=O)CCC2CCCCCC2)C1)OCC C1(C(=O)NC(C)CNC(=O)Cc2ccon2)CCCN2CCCC12 N1(C(c2c(CNC(C(F)=CCC)=O)noc2)=O)CCC2CC2C1 C1(CC#C)(C(N2CCC(C)(C)C2)=O)CCN(C(=O)C=Cc2cn(C)cn2)C1 C1(CC)CN(C)C(=O)CN1C(C1(CC)CC1)=O.c1(C=O)[nH]ccc(=O)c1C.N C1(C(=O)NC(C)(C)CNC(=O)CN2CCC(=O)NC2=O)CSc2ccccc2O1 C#CC1(NC(C2CCN(C(=O)CCOC3CCC3)C2CC)=O)CC2CCCC12 N1(C(c2c(C)ccnn2)=O)CC(NC(c2scnc2C2CCCC2)=O)CC1(C)C N1(C(c2cnc(C)[nH]2)=O)CCCC(N(C(=O)C(c2cccn2C)=O)C)CC1 C1(C2(NC(c3coc(O)n3)=O)CC2)CCCCN1C(=O)COC1CCCOC1 C1(C)(NC(CC(C(C)C)NC(c2ccc(C(C)C)o2)=O)=O)CCC(=O)N(C)C1 c1(C(=O)NC2C(C)N(C(C3CC4CCC3CC4)=O)CC2)cc2c(nn1)CCOC2 C1(CC=C)(C(=O)N(CCNC(C2CC3CCC2O3)=O)C2CC2)CCOCC1 c1(OC)cc(C)[nH]c(=NCC(C2CCCCC2)NC(=O)C(=O)C(C)(C)C)n1 c1(C(=O)NC2C3(CC(NC(C(C)C(F)(F)F)=O)C3)C2)cc2ccc(Cl)cc2[nH]1 c1(C(=O)NC(CC)CN(C(=O)Cc2ccc(C)cc2)C)cc2ncc(C)cn2n1 CC(N=c1[nH]nc(C(C)(C)C)o1)C1CCN(C(=O)CC2CCCC2C)C1 CC(CO)(CO)C(=O)N1CC(CC(=O)Nc2ccc(Br)c(I)c2)C1 CC(CC(F)(F)F)C(=O)N1CC2C(C(=O)NCc3ccn(C)n3)C2C1 c1(C(=O)NCC2N(C(c3c(C)cc[nH]3)=O)CC(F)C2)ccc2c(n1)CCO2 C1(NC(c2n[nH]c(C)c2O)=O)CN(C(C2CCCC2O)=O)C2CCCCC12 N1(C(c2nccc(CNC(Cc3c(C)n[nH]c3C)=O)c2)=O)CCC(O)C(F)(F)C1 C1(CNC(=O)CCC2CC2(Cl)Cl)CN(C(c2occ3c2CCC3)=O)CCCO1 N1(C(C(C(C)C)OCC)=O)CC2CCC(C2)C1.c1(C=O)cnc(C2CC2)o1.C Cc1cc(C(N2CCN(C)C(C(=O)NCCOCC(C)(C)O)C2)=O)c(C)nn1 C1(NC(c2cnn(CC)c2C)=O)CN(C(C23CC(C)(C2)OC3C)=O)CCC1C C1(CNC(c2c(CC)scn2)=O)CCCN(C(c2ccnnc2Cl)=O)C1 C(=O)(C1=CCCOC1)N1C(C(CNC(CC2C(C)(C)C(O)C2)=O)(C)C)CCC1 CN1CCCC(N2CCN(C(c3ccc(F)cc3)C(=O)O)CC2)C1 C1(NC(c2n(C)cc(Br)c2)=O)COC2(C1)CN(C(=O)CCF)C2 C#CC1(F)CCN(C(=O)C(CC(=C)C)NC(=O)C(C)n2cccn2)CC1 CCCC(O)C(=O)NCC1CC(C(=O)NOCC(C)C)CO1 C1(CC(N2CCC(C)(NC(c3c(C)ocn3)=O)C2)=O)CC2CCC1CC2 C(=O)C1CCc2nccn21.C1(C(=O)NCC(=O)OCC=C)CCC12CCC2.N C1(CCNC(C(C)Cc2cnc[nH]2)=O)CN(C(c2cnnn2C)=O)CC1C N1(CCNC(CC=CC=C)=O)CCC(NC(=O)CC2CC3CC3C2)CC1 C(=O)(C1=Cc2ccccc2C1O)NCC1(NC(C(CC)CC(F)(F)F)=O)CCC1 Cc1nn2c(c1C(=O)NCCC1CCN(C(c3cn(C)c(O)n3)=O)C1)CCCC2 c1(OC)cc(C(N2CC(NC(C3CCOC3C3CC3)=O)C(C)C2)=O)cc(C)c1 C1(C)(C(=O)NCC(C(C)C)NC(C2(C(F)F)CCC2)=O)CCCC1C Cc1ncc(S(N)(=O)=O)cc1C(=O)N.c1(C(N2CC(O)C2)=O)nccnc1C.C Cc1ccc(C2CN(CCC3(C(=O)O)CCOC3)CCO2)cc1 c1(C(=O)NC2CN(C(C(CC)C(=O)OC)=O)CC2C)c(C)c(C)c(C)c(C)c1C c1(-c2ccc(C(=O)NC(C(C)NC(C3CC(C)C3)=O)CO)s2)ccccc1F C1(C(=O)NC2(CC#C)CC2)(COC)C=CCN1C(c1cccc(C)c1)=O Cc1c(C)c(C)c(S(=O)(=O)N2CCC(CNC(=O)CO)C2)c(C)c1C C1(C(N(CCN(C)C)CCO)=O)CC(O)(CNC(C2CCCCO2)=O)C1 N1(C(C2(N(C)C)CCC2)=O)CC(NC(C2CCCC(C)(C)O2)=O)C(C2CC2)C1 C1(NC(CN(c2cccc(Cl)c2C)C(CCC(C)OC)=O)=O)CN2CCC1CC2 C1(CCO)CCC(N=c2[nH]c3c(c(=NC4C5COCC45)[nH]2)CCCCC3)CC1 C1(C(=O)NCCC2CN(C(C(C=CC)O)=O)C2)CCOC(=O)N1 C1(NC(C(C=C)(C)CCOC)=O)C2CCCC1CC(NC(=O)CC(C)(C)O)C2 CC1CCCCC1NC(=O)CNC(c1cccc[n+]1[O-])=O C1(NC(C(=Cc2ccco2)C)=O)CCCC2CN(C(c3cnc(Cl)[nH]3)=O)CC12 C12(C(=O)NC(C(C)C)CNC(=O)C(C)(C)C3CCCC3)CC(C)(CCO1)C2 N1(C(=O)CN2CCCC2)CCCC(C2CCCN(C(=O)C(Cl)Cl)C2)C1 CC(CC(C)NC(=O)C=Cc1ccccc1F)N=c1[nH]c(Cl)nc2c1CCC2 c1(C(C(=O)NC(CC)(CNC(=O)CCNC(C)=O)CC)=O)ccccc1 C1CCN(C(C2CCS(=O)(=O)C2)=O)CC1F.c1(C(=O)N)coc(C(F)(F)F)n1 c1(CCC(N2CC(N(C(=O)CCS)CC=C)C2)=O)ccccc1C(F)(F)F C1(CC(=O)NCC=CCNC(C2(CC(C)C)CC2)=O)CCC(=O)C1 C(=O)(C(F)C(C)(F)F)NC(C1CCCN(C(c2cc(C(F)F)no2)=O)C1)C CC1(C(=O)NCC2CC2CNC(c2cc(Br)no2)=O)CCOC1 C(C(C)C=O)N1C(C(=O)NC(C)(C)C)CC1.n1(CC)ccc(=N)[nH]1 CC(C)C(C)C(=O)N1CCC(OCCNC(=O)CCCC2OCCO2)C1 CCCCCC(CCCCC)C(=O)NC(C)CNC(C1CCCOC1)=O N1(C(C(COC)O)=O)CCCC2(C1)CN(C(=O)CC1CCC(=O)NC1=O)CCO2 C1(C(=O)N)CC(F)CCN1C(C1CC2CC(=O)C1C2)=O.CC(C)CCOCC C1(O)(COC)CCCN(Cc2ccc(C(=O)O)c(F)c2)CC1 N1(C(C(=C(C)C2CC2)F)=O)CCC2CN(C(C3CNC(=O)N3)=O)CC12 c1(C(=O)NCCN(C(CCOCC#C)=O)C)c[nH]nc1C1CCCCC1 Cc1cccc(C(N2CCOCC2C(=O)Nc2ccnc(C3CC3)n2)=O)c1C C1(NC(N(C(c2ccncc2)CC)C)=O)CCC(S(C)(=O)=O)C1 CC1(CNC(c2cc(CNC(=O)C(C3CCOCC3)F)no2)=O)CCOC1 c1(NC(c2ccc(O)cc2)=O)cccc(NC(C2CC2Br)=O)c1 CC1OC2(C(N3CCN(C(=O)CC4CCCOC4)CC3)=O)CCC1CC2 c1(C(N(C(C)CCNC(=O)COC2CCOC2)C)=O)[nH]cnc1C#N Cc1cc(C(=O)NC(C)(C)CNC(C2(N(C)C)CC2)=O)ccc1O C1(NC(=O)NC2CCC(O)(C(F)(F)F)CC2)CCCC2C1C2(F)F O=C(CC1CC1CNC(c1ccc([N+](=O)[O-])o1)=O)N=c1ccn(CCCO)[nH]1 C1(NC(c2n(C)ncc2Br)=O)CN(Cc2c(F)ccc(Br)c2Cl)CC(F)(F)C1 CC(C(=O)N1CCC(C)(NC(=O)C=CC(N2CCOCC2)=O)C1)C(C)(F)F CCCC(C)(O)C(=O)NCc1occc1C(=O)NC1CN(C)NC1=O C(=O)(C1CCCc2nn[nH]c21)N(CCC(C(C)C)NC(c1cccc(C)n1)=O)C N1(C(C(CCC)N(C)C)=O)CCN(C(=O)Cc2cccc(F)c2F)C(C)C1C C1(n2cc(CN(C(C3(CCCC)CC(=O)C3)=O)C)nn2)CCCC(C)C1 C1(O)(CNC(C2CCCOC23CCC3)=O)CCCN(Cc2ccccc2)CC1 C1(C(N2CCC(COC(C)=O)C2)=O)CC12CCN(C(c1cnn3c1CCC3)=O)C2 N1(Cc2cc(OCC)ncc2Br)CC2CN(C(c3ccccc3I)=O)CC2C1 C(CC)(C(=O)N)OCC.C12CC(C1)C2.C1(C=O)CCCN1S(C)(=O)=O Cc1cc(C(N2CC(NC(c3cccc(C(=O)C4CC4)c3)=O)C2)=O)oc1C N1(C(C(N2CC(C)(C)C(O)CC2)=O)=O)CCOc2c(F)cc(Br)cc2C1 C(N=c1[nH]c(=NCCCCCN2CCCCC2)c2sccc2[nH]1)C1(C(C)C)CC1 C1(C2N(C(c3n(CC)ncc3)=O)CCC2)CCN(C(C2CC2(F)F)=O)CC1 N1(C(c2ccc(C)nc2)=O)C2CCC1(CNC(=O)C=CS(C)=O)CC2 C12(NC(c3cnc(C)s3)=O)CCCC(CN(C(=O)Cn3cccn3)C1)C2 C1(NC(C2CCN(C(COCCCCC)=O)C(CC)C2)=O)CC=C(C(C)C)CC1 C1(C(=O)NC2CCN(C3CCN(C(C4CCCO4)=O)C3)CC2)(OC)CCCCCC1 N1(C(C(C)NC(C)=O)=O)CCSCC1C.c1(C(=O)N)ccccc1-n1cccn1 C1(NC(Cc2c(F)cc(C)c(F)c2)=O)CCCC2CN(C(=O)C(C)(C)C)CC12 CC(C)C(C(=O)N1CC(O)CC1CNC(=O)CCCC#N)n1cc(Br)cn1 N1(C(C=CC=CCC)=O)CC(OC)C(OCC)C1.C(=O)(C)NCC.O C1(OC)COCCC1NC(c1ncc(C2CC2)[nH]1)c1nnnn1CCCSC N1(C(C(Br)=C(C)C)=O)CCCC(NC(C2CC(N3CCCC3)C2)=O)C1C Cc1c(C(C)OC(c2nc(Cl)ccc2O)=O)sc2ccccc12 c1(-c2nc(CC(C)OC)nn2-c2nc(C)nn2C)cc2c(Br)ccc(F)c2[nH]1 CC1(C)C(O)C2CCN(c3nnnn3C(c3cccc(O)c3)C3CC3)C12 CC1CCC(C)CN1C(C1(F)CCCC1)=O.c1(C(=O)N)cnccc1C(C)(C)C C(=O)(CCCC(C)(C)C)NCC1C(NC(c2cc(C(C)C)no2)=O)CCC1 c1(N2CCCC(NC(c3n(C)cc(Cl)c3)=O)C2)ncnc(Cl)c1C#N C1(N(C(c2cc(C)c(C)nn2)=O)CC)CCCN(C(=O)C(C(C)(C)C)SC)CC1 C=C=C(C)CC(=O)N(C1CCN(C(c2ccccc2)=O)C1)CC.C(C(F)(F)F)O c1(C(N2CC(NC(C(CC)COC)=O)C(C)C2)=O)ccc2ccc(OC)cc2c1 C1(OCC(=O)NCC2CN(C(c3cscn3)=O)C2)C#CCCCCC1 C1(c2n(C(CC)(C)C)nnn2)(NCCC(C)(C)F)CCC(C)(CO)CC1 Cc1cc(C(=O)NC(CNC(=O)CCn2cccn2)C2CC2)c(C)cc1Cl N(C1CCCn2ccnc21)C(C1(CNC(c2ccc(C)nc2)=O)CC(=C)C1)=O c1(C(N2C(CCNC(CC3(C=C)CC3)=O)COCC2)=O)ccc2c(c1)CNC2=O N1(CC(=Cc2ccccn2)C)CC2(C)CN(C(c3csnn3)C)CC2(C)C1 C1(CNC(C(n2ccc(C)n2)C)=O)CCC2(CN(C(c3ccc(O)nn3)=O)C2)O1 CC1CN(C(c2ccnc(N3CCCC3)c2)=O)CC(C)C1N=c1[nH]nc(O)s1 Cc1cc2c(cc1Cl)N(C(c1cn(C)nc1OCC(F)F)=O)CC2 N1(C(c2ccn(CC)n2)=O)CC2CC(C)N(C(=O)CC3CCC(O)C3)C2C1 c1(C(N2CCCC2)=O)ccc(C(N)=O)c(Cl)c1.N1(CC)CCCC1C(=O)N.C CC1CCCCC1(CO)NC(=O)C(c1cccs1)NC(C1CC2(CC2)C1)=O c1(CN(C(c2ccc(Cl)c(F)c2)C(=O)NC2COC2)C)nnc2n1CCCCC2 N1(C(c2cc(C)cc(C)n2)=O)CC(C(=O)NC(C)CC(N)=O)CCC1(C)C c1(C(F)(F)F)cc(Br)ccc1-n1cnnn1.c12cn(-c3ccccc3)nc1CS2 CC1(NC(=O)CC2CC(F)C2)CCN(C(=O)CCC23CCC(CC2)C3)C1 c1(C(C)(C)C)ccc(CN2CCCC2CC(=O)NCCn2ccnc2)c(Br)c1 C1CCN(C)C(=O)C1.N1(C(CNC(C2C(C)C2)=O)=O)CCC(C)(CC=O)C1.N C=CCC(C)(O)C(=O)N(CCC(C(C)(C)C)NC(=O)CCCN(C)C(C)C)C Cc1cc(=NCCC23CCC(CC2)CC3)[nH]c(N2CCC(c3cnn[nH]3)C2)n1 C(C)(C)(CCCC(=O)NCC(O)C1CCC1)NC(C(C)C1CCC1)=O C1(NC(C=C(C)C)=O)CN(C(c2ccnnc2)=O)C2(CCC2)C1 c1(OC)cccc2c(C(N3CC(CNc4ncnc(O)c4Br)CC3C)=O)cnn12 C1(CC(=O)OCC2C=CCOC2)Cn2c(nc3ccccc23)NC1=O Cc1cc(NC(=O)C(O)CCNC(C2CC(=O)CS2)=O)cc(C)c1C Cc1cc(C(=O)NC2(C(=O)NOCC(F)F)CCSC2)nnc1O C(CCC)(C(=O)NCc1ncoc1CCNC(=O)C(C)N=[N+]=[N-])=CCC Cc1nc(C2CCC2)oc1C(N1CC(CC(C)NC(C2CCCOCC2)=O)C1)=O C=CC1CCN(C(=O)C=CC(C)(C)NC(c2cc(O)n(C)n2)=O)C1 c1(CC)cccc(CC)c1NC(=O)C(C1CC1)(C1CC1)OCC C(=O)(CCCCCC(=O)N1CCC(NC(c2cccc(C3CC3)c2C)=O)C1)OC N1(C(C(C)OC)=O)Cc2cccc(CNC(c3cc(Cl)ns3)=O)c2C1 N1(C(c2cnnc(C3CC3)c2)=O)CC2CN(C(C3CC34CC(F)(F)C4)=O)CC2C1 C1(C(N2CC(C(C)(C)O)C2)=O)CCOC(C(F)(F)F)C1.C1(O)(C=O)CC1.C c1(C(N2CC(CC)C2)=O)cnn2c(C)cccc12.c1(CC)nn(C)cc1C(=O)N C1(NC(c2ccsn2)=O)CN(C(=O)C=CSc2ccccc2)Cc2ccnn2C1 c1(C(=O)NCCCCn2cc(CCCC)nn2)c(SC)cnn1C N1(C(C(CC)OC)=O)CC2(CCCCN(C(c3ccc(NC(C)=O)c(Cl)c3)=O)C2)C1 N1(C(c2cc(-c3ccc(C)s3)[nH]n2)=O)CCCN(CCc2cccs2)CC1 C(=O)(CCC(CC)NC(=O)C(CC)OC)N1CC(O)(CC=C)C1 Cc1ccc(NC(C2CC(=O)N(c3nc4ccccc4[nH]3)C2)=O)c(Cl)c1Cl N1(C(c2c(CC)nc(C)[nH]2)=O)CCC2(CCN(C(C3CCCC4CC34)=O)CC2)C1 CCC(CNc1nccc(OCC(F)F)n1)(CC)NC(=O)CC1(C)CC1F CN1CCN(C(c2cccc(=O)o2)=O)CC1CNC(C1(C(F)F)CCCO1)=O c1(C(=O)NC2CC(CNC(CCC(C)OC)=O)OCC2)cnc2ncccc2c1 CC1CC(NC(=O)CCOC2CC2)CN1C(c1cccnc1NC1CC1)=O C1(CC(=O)NCCCC#C)CN(C(=O)Cc2c(C)noc2C)CCO1 CCC(C)(O)CCNC(=O)C(O)CCNC(=O)C(C(=O)OC)OC C1(NC(COCCNC(CCOCC(C)C)=O)=O)CCCCCC1O C1(N(C(C=CSC)=O)C)C2CN(C(=O)Cc3ccc(C(C)=O)s3)CC12 CON=Cc1ccc(C(=O)NC(C2CN(C(c3ccon3)=O)CCO2)C)cc1 C(=O)(C1=Cc2cc(C)ccc2OC1)NC1C2N(C(=O)OC)CC(CC2)C1 Clc1ccc2c(c1)N(Cc1c(Cl)cc(Br)cc1Cl)CC21CC1 c1(C(=O)NCC(=O)NCC(=O)N(CC#C)CC)cccc2[nH]ccc12.C c1(C(N2C(C)(C(=O)Nc3scc(C)c3C#N)CC2)=O)cccc2ncccc12 c1(NC(C2C(CC)N(C(C3CN(C(N)=O)C3)=O)CC2)=O)ccc(C)c(O)c1 N1(C(C2(C)CC2c2ccccc2)=O)C2CCC1CN(C(C1CCCC13CC3)=O)C2 O=C(NNc1ccc(F)cc1F)c1nc(-c2ccccc2)cs1 C(=O)(CN=c1cc[nH]cc1)N1CC2CC(C(=O)NCCCC(F)F)CC2C1 N1(C(C=Cc2ncc(C)[nH]2)=O)CC2CCC2(NC(C2CCS(=O)(=O)C2)=O)C1 c1(C(=O)N)ccc2[nH]ccc2n1.C1(OCC)CCCC1NC(C1CC1(C)C)=O C1(CNC(CCCCC)=O)CCN(C(c2c(C)ccnc2Cl)=O)CC1C Cc1nc2cc(NC(C3CCCN3Cc3ncccc3C)=O)cnc2[nH]1 C(C(C)(C)CC(=O)NC1CCOCC1C)NC(c1nc(CCC)oc1)=O N1(C(C2CCN(CC)CC2)=O)CC(C2CN(C(C3(C(C)(F)F)CC3)=O)C2)C1 C1(C(=O)NCCC2C(=O)NC(=O)N2)CC12CCN(C(=O)Cn1cnnc1)C2 C1(C(=O)NCC(C)N(C)C(c2cncc(N)n2)=O)CCN(C2CC2)CC1 C1(NC(c2c(C)cc(C)o2)=O)CN(C(=O)C(F)CC2CCCCC2)CCC1F CS(=O)(=O)CCC(=O)NC1CC1C(=O)Nc1ccc(Cl)cc1OC(F)(F)F Cc1cccc(OCCCC(=O)NC2(CO)CC(C(=O)O)C2)c1 N1(C(C=CCN(C)C)=O)C2CCCC1CC(Nc1cc3nncn3cn1)C2 CCCCC(F)C(=O)NC(C1(O)CCCCC1)C(=O)NC(CC)C(C)CN(C)C C#CC1CCCC(NC(C2(CC)CCN(C(=O)C(C)C(F)(F)F)C2)=O)C1 N1(C(c2c(C)occ2)=O)CCCC(F)(CNC(C2(C)CC2(C)C)=O)CC1 C1(NC(C2C=CCN(C(C3(C(C)(F)F)CC3)=O)C2)=O)CCOC12CCCC2 C1(CCCC)CN(C(C2CCCN2C)=O)CCN1C(c1ccc(C)cn1)=O Cc1ccc(C(N2CCC(C(=O)NCC(C)(C)F)C2C(C)C)=O)cn1 c1(C(=O)NCCCC(C)(C)NC(CC(C=C)CCC)=O)ccc2ccccc2n1 C1(CC=C)(NC(=O)C(C)C(F)F)CC2CCC(C1)N2C(C1CCOCC1)=O C=C(F)C1(CC(=O)NC(C2(CNC(C34CCCC3C4)=O)CC2)C)CCC1 C(=O)(C(COC)CC(C)C)NC1C(NC(Cc2cccc(CC)c2)=O)COC1 Cc1sc(O)nc1C(=O)NCC1(F)CC(C)C1.c1(CC(=O)N)cncs1 c1(C(N(C(C)C2CC2)C)=O)cnn(C)c1C(F)(F)F.C(=O)CC=C(Cl)Cl.N c1(C(N2CCCC(CNC(c3cccc(C)c3C)=O)C2)=O)cccc2c1CCC2 c1(CC)onc(CSCC(C2CC=CCC2)=O)c1C CCC(CC)(C(=O)N(CC(=O)NOCC1CC1)C)C(C)C CC1CC(CNC(=O)Cc2cnccc2Cl)CCN1C(c1cnc(S)n1C)=O C=CCCC(O)CNC(C1C=CCN(C(=O)C=CC(F)F)C1)=O n1(CC)nnc(C(N2CCCC(CCNC(C3CCCC3(F)F)=O)C2)=O)c1C CCC(CC)CC(=O)N(C)CCOCCCN(C)C(C1(C)CC=CCO1)=O C=C(CNC(C12CCC(CC1)C2)=O)C1CCOCC1.C(=O)(C(C)c1cccs1)N N1(C(C2(CCCC)CC2)=O)CCC(O)(CCNC(=O)C(c2ccncc2C)C)C1 c1(OC)ccnc(C(=O)NC2CCC(NC(C34CC(C)C3C4)=O)CC2)c1Br C1(C(=O)NCC=CCNC(CCCNS(C)(=O)=O)=O)CCCCC12CCC2 C1(C)(C(N(CCCN(C(C2C(CC)OCC2)=O)C)C)=O)CCN(C)C1 c1(NC2CCn3c(C)nnc3C2)[nH]c(=NC2CCOC(C)C2)nc2sccc12 n1(CC(N2CCC(NC(c3ccc(C#N)cc3)=O)C2)=O)cc2ncccc2n1 c1(C(N2C(CNC(=O)Cc3cnns3)CC2)=O)ccc2n[nH]cc2n1 N1(C(C(=O)N(C)Cc2nc(C)sc2)=O)CCC(C(C)(C)F)CC1 c1(C(=O)N)nc(C)nn1C.C(CC(=O)NCCOC(C)(C)C)N(CCC)C Cc1cncc(C(=O)NCc2cnc(C(=O)N)s2)n1.C1CN(C(N)=O)CCO1 c1(CN=C(NCc2c(C)cco2)NC2CCCC2)cccc(F)c1F N1(C(C(C)(C)C#N)=O)CCC2(CCOCC2)C(CNC(c2ccnc(S)c2)=O)C1 C1(CNC(C(CC#C)NC(C2CC(OC3CC3)C2)=O)=O)CCCN(C)C1=O C(=O)(C(C)C(O)C(C)C)N.C1(C(N2CCC(COC(C)=O)C2)=O)CCOCC1 C1(OCC(=O)NCCN(C2CCCCC2)C(C2CNC(=O)C2)=O)CCCOC1 C(c1ccccc1[N+](=O)[O-])=CC(=O)NCC(CNC(CCC(C)=O)=O)C Cc1ccc(Sc2ccccc2OCN2CCCC2C(=O)O)cc1 C1(C#N)(C(=O)NCCC(C)NC(=O)C(C2CCC(=O)N2)C)CCOC1 CCC(C#N)C(=O)N1CC(F)CC1C(=O)NCC1CCN(C2CC2)C1 c1(CNC(C=C(C)CNC(=O)C(F)n2ccnc2)=O)ncccc1C C1(CC(=O)N(CC(C)NC(C=C(C)Cl)=O)C)CCCO1 N1(C(c2c(C)cnnc2)=O)CCCC(C2(NC(c3cc(Cl)nnc3O)=O)CC2)C1 C(c1ccccc1)=CC(C)C(=O)N.C1(C(N2CC(O)(CC)C2)=O)CC2C=CC1O2 N1(C(C(=O)NCCCC)COCc2ccccc2)CCC(O)C(CO)C1 Cc1cc(C)n(C(C)CC(=O)N(C)CC2CCCCN2C(=O)CC2CC2(C)C)n1 CCC(C)CC(C)NC(N1CCCC1COc1ccccc1F)=O Cc1cnccc1CCNC(=O)C(C1CCCN(C(c2ncccc2N)=O)C1)C C(=O)(CC(C)(C)CN(C)C)N.c1ccc(F)cc1.CC(C)CN(C(=O)CC)C c1(C(N2CCCC(C(=O)NCc3cnc(C)s3)C2)=O)ccnc(O)c1F C(=O)C(C)C(C)C.C1(C(=O)NCC2CCC2)(OC)CCOC1.C(C)=O.N C12(C(=O)NC(CC)CN(C)C(c3nn(C)c(C)c3Cl)=O)CCCC1CC(=O)C2 c1(N2C(C)CCC(NC(=O)CN3CCCC3=O)C2)nc(O)c2ccccc2n1 c1(C(N2C3CC(NC(C(C(C)(C)O)F)=O)CC2CC3)=O)cccc2nccnc12 CN1CC=CCC1CC(N1CCCCC1CNC(c1csnn1)=O)=O C(C)(C)(C(=O)N)NC(=O)OC.C1(C=O)CCN(c2ncccn2)C1.C(C)C N1(C(c2cc(C)no2)=O)CCC(C(F)(F)F)C(NC(=O)CCC#N)C1 CC1(CCCC(=O)NC2CCC(NC(C3COCCOC3)=O)C2)NC(=O)NC1=O Cc1ccnc(C(=O)NCC2CC(C(=O)NC(c3cn(C)nn3)C)=NO2)c1F C1(NC(C2CCCCO2)=O)CN(C(c2cc(O)ccc2Cl)=O)C2CCCCC12 N1(C(c2ccn(C)n2)=O)CC(C)C2CC12.c1(C(=O)N)cn(C)nc1-c1ccco1 N1(C(CCCC(=O)NCC)=O)CC2CCN(C(=O)C3=CC4CCC3C4)C2C1 c1(N(C2CCC(N)C2)C(c2nccc3nc[nH]c23)=O)ccn2nccc2n1 N#Cc1ccc2c(CN3CCC(F)(C(=O)NCc4cc[nH]n4)C3)c[nH]c2c1 S(=O)(=O)(CCCCS(=O)(=O)N1CCCC1c1nonc1C)Nc1nc(C)c(C)s1 C=CCCCCCC(=O)NCC12CC1CN(C(=O)CC1CC(=O)C1)C2 c1(C(=O)NCCCN(CCC)C(C2CCC(=O)N2)=O)ccc([N+](=O)[O-])s1 Cc1c(CC(=O)NC2CN(C(=O)C(C(C)C)n3cnnn3)C2)sc2ccccc12 Cc1cccc(C(=O)NC2(CNC(c3cccc(CCO)c3)=O)CC2)c1F Cc1cccc(C)c1CCNC(=O)N(CCC1=CCCCC1)C CC(C)CCCNC(C12CCCC1(C(N)=O)C2)=O.C(c1ccccc1)=CC=O N1(C(CC2N(C)CCCC2)=O)CCC(C)(C)C(NC(=O)Cc2cnc[nH]2)C1 c1(C(=O)NCCN(C2CCCCCC2)C(CSC)=O)cn2c(n1)SCC2 C1(NC(=O)CCCc2ccccn2)CCCC(NC(=O)CC2CSC2)C1 C1(O)(CNC(C2CC(CCO)C2)=O)CCCN(C(=O)CC(F)(F)C(F)F)CC1 C1(NC(C2CC23CC(O)C3)=O)C=CCN(C(c2coc(C(F)(F)F)c2)=O)C1 CN1CC(O)CCC1C(=O)NC(CNC(C1CCCC2(CC2)C1)=O)CO n1(CC(=O)NCC(O)CNC(=O)CC2CCCNC2=O)nnc2ccccc12 Cc1nc(CNC(=O)C(=O)NC2CC23CCC3)n[nH]1 Cc1cccc(C(N2CC(CNC(=O)C(C)(CO)CO)C2)=O)c1F C1(CC(=O)NCCN(C)C(C2CCN(C)S2(=O)=O)=O)CCCC(C)(C)O1 c1(C(=O)NCCC2CCN(C(C(CC)(C)COC)=O)C2)cc(C)nc(C)c1O CCCC(C)(C)CC(=O)NC(C)C(=O)N(CCC(=O)NC)C c1(CC)cc(C(N2CCC(NC(=O)C=CCOC)C2C)=O)cc(F)c1 C(=O)(CCCCCC(=O)NC1CN(CCOC(C)(C)C)C12CCC2)OC C1(C(N2CCC3(CC(NC(C(C(CC)O)C)=O)C3)C2)=O)CCC2(CC1)CC2(F)F Cc1cc(C#N)nc(N2CC3CC(NC(C4(F)CCOC4C)=O)CC2C3)n1 C(N=c1cc(C)nc(CO)[nH]1)C1(C)CCCN(C(c2c(CC)nccn2)=O)C1 CC1(NC(=O)COC(F)F)CN(C(=O)C(c2ccccc2)C2CC2)C1 N1(Cc2cc(C)n(C)n2)CCc2cc(NC(=O)CCC(N)=O)ccc2C1 C#CC1(C(=O)NC2CC3(C2)CC3C(=O)NC(C)CCCC)CC(=O)C1 N1(C(c2c(N)snn2)=O)CC2(C1)CN(C(=O)CN1CC(F)(F)C1)CCO2 C1(NC(C=Cc2n(C)cnc2)=O)(CNC(=O)CC(C)(F)F)CC2CCC1CC2 c1(OC)ccc(N(C)C(c2cnn(C)c2C2CNC2)=O)c(F)c1 N1(C(c2cc(C)nn2CC(F)F)=O)CCCC(C2COC2)C1 C(=O)(C=CS(C)=O)NCC#CCNC(C(c1ccccc1F)(C)NC(C)=O)=O C1(C)(C(N2CC(F)(CNC(Cc3c(C)occ3)=O)C2)=O)CCC(=O)N1 CCCCC(CC)CC(=O)N1C2CCC1CN(C(=O)C(CCC(N)=O)N(C)C)C2 CC(C(CO)NC(=O)C(n1ccc(C2CC2)n1)C)NC(c1ccccn1)=O Cc1ncsc1C=CC(=O)NCC1CCC1(C)C.C(=O)(CCCn1cccn1)N N1(C(C2CC(=C)C2)=O)CCCC(CCOC2CCN(C(=O)CSC)C2)C1 c1(NCC)scnc1C(=O)N(C)C.C1(O)CN(C(=O)CC2CC2(Cl)Cl)C1 C1(CCCC)CCCN(C(C2(N(C(=O)CCCN(C)C)C)CC2)=O)C1 C1(OCCC)CCCN(C(C2(C)CCN(C(=O)CC3CCCCN3C)C2)=O)C1 c1(C(N2CCCC2)=O)cnc2[nH]cnc2c1.C1(C(=O)OCC)(C(=O)N)CCCC1 C1(C(=O)NCCCN(C(C2C(CCC)CCC2)=O)CC)CCc2cncn2C1 C1(CCN(C)C(c2csc(C)c2)=O)CCCCC1.C1(C=O)CC1(C)C(F)F.N CC(CNC(=O)Cc1cccs1)C(F)C(=O)NCC(C)(C)n1cccn1 CC1CCN(C(=O)CC2CC3(C2)CN(C(C2CCC(=O)C2)=O)C3)C1(C)C N1(C(c2ccc(C)c(F)n2)=O)CCN(C(c2cc(C3CC3)on2)=O)C2(CCC2)C1 C1(NC(c2c(CC)csc2)=O)CCC2CN(C(c3cnc(N)c(Cl)c3)=O)CC2C1 N1(C(c2cc(C)no2)=O)CCCCC1CC(=O)N(C)Cc1ncc[nH]1 C1(NC(CCNC(=O)NC)=O)CCC(C)CC1.n1(CC=O)ncccc1=O.N C(=O)(CC(C=C)CCC)NC(C(=O)NCCC=CC=C)CC1CCCC1 C12(NC(C3C(CCC)C3)=O)CCC(CC1)OC2.c1(C=O)cc(C)c(C)s1.C C1(CNC(CCCc2ccc(C)s2)=O)CCN(C(c2cc(C)c(C)s2)=O)C12CC2 Cc1ncc(C=CC(=O)NCCNC(c2nn(C)nc2Br)=O)c(O)n1 N1(C(C(C)N(C(=O)CC2CC(OCC)C2)CCC)=O)CCc2cccnc2C1 c1(C(C(=O)NC(CC)(C)C)N(CCC(C)C)C)cc(C(F)(F)F)cc(C)c1.O c1(C(C(=O)NC(C(=O)NCCSC(C)C)C2CCC2)C)cnn(C)c1 C(=O)(C(C)C(O)C(C)CC)N(C1CCCN(C(c2c(C)cc(CC)o2)=O)C1)C c1(C(=O)OC)csc(C(N2CCC(C(C)NC(=O)C)C2)=O)c1.c1ncccn1 N1(C(c2cc(COC)[nH]n2)=O)CC2CN(C(C3CCOCC3)=O)CC12 C(=O)(N=c1[nH]sc2ncccc12)C12C(CN(Cc3c(F)ccc(C)c3Br)C1)C2 c1(NC(CC)CNC(c2cncc3nc[nH]c23)=O)ccc(C(=O)OC)cc1[N+](=O)[O-] c1(-c2scc(C)n2)nc(C(F)C(F)(F)F)n(-c2ccc(Br)cc2)n1 C1(CNC(=O)CCC2CCCCO2)CCCCN1C(=O)C(C1CCCO1)C1CC1 c1(OCC(=O)OCC)cnccc1.N1(C(C=O)=O)CCC(C(F)(F)F)CC1 C=C(C)CC(C(=O)NC(C(=O)NCCC1(O)CCOC1)C(C)O)OC CC(C)C(CNC(=O)C(F)=CC1CC1)NC(c1cnc(N(C)C)s1)=O c1(C(N2CCC(NC(C)=O)C2)=O)cnn2c1CN(C(c1ccc(Br)cn1)=O)CC2 C1(C(=O)NCCOCCC)(OC)CCC12CCC2.c1(CC(=O)N)ccon1 CC1CN(C(=O)C(C)(C)CCl)CCN1C(c1ccc(F)c(NS(C)(=O)=O)c1)=O C(=O)(C1CCc2nccn21)N1CCC(CC)C1CNC(=O)CP(C)(C)=O C(=O)(C1=CC2C=CC1C2)N1C2C(NC(c3c(C)coc3)=O)C(C2)C1 Cc1cc(C)c(C(=O)NCC2CCC(C)CC2)c(C)c1.c1(C=O)ccccn1.N n1(CCNC(C2CN(C(COC)=O)C2)=O)nc(C)nc1C c1(C(=O)N)cccs1.C(=O)C(O)CN1CCCC1.C1(C(=O)OC)CCC1C c1(C(N2CCCCC2)=O)coc(=O)c2ccccc12.O=C(CCNC(=O)CO)N.C C1(CC=O)C(=O)NN=C1C.c1(CCC(=O)N(CCC)CCC)cnc(O)[nH]1.N c1(C(=O)NC2CCC2CO)cc2c(s1)CCC2=O c1(CN2C(C(=O)NCCCOC=C)CC(C)C2)cccc(I)c1O C1(C(N(C(C)C(F)F)C)=O)C(O)CCN1C(=O)CC1CCC(C)(C)O1 C1(OC)CCCN(C(C2CCN2C(=O)CC(C)F)=O)C1 c1(C(C)C)n[nH]c(=NC2CC(NC(c3ccc(-n4cccn4)cc3)=O)C2(C)C)o1 c1(SC)nn(C)cc1C(=O)NCCC1CCN(C(=O)CO)CC1.C1CCOC1 C1(CNC(C(C(C)OC)NC(=O)Cn2cnnc2O)=O)CC(C2CC2)=NO1 c1(OC)cccc(S(=O)(=O)N2CCCC2c2cnco2)c1 c1(C(=O)NCC(C2CC2)NC(Cc2ccc(C)s2)=O)cnn2c1NCC(C)C2 C(CCC(=O)NCc1ccc(C(=O)NCC2CC23CC3)o1)N(C)C C1(NC(=O)CC2CCN2C(C2CNC(=O)O2)=O)CC2CCCC2C1 N1(C(C)C)CCC(CNC(=O)C=CCN(C(=O)CCc2cnn[nH]2)C)C1 N1(C(c2c(CC)c[nH]n2)=O)C(C)CC2CN(C(=O)C=CS(C)=O)CC12 C(c1ccc2occc2c1)=CC(=O)NC1(CO)CCCN(C(=O)C(F)C2CC2)C1 Cc1cc(C(N2CCCC2C(C)(C)C)=O)c(C)o1.C(=O)(C(F)=C1CCCC1)N C1(NC(C(C)n2cncn2)=O)COCC1NC(c1cc(Cn2cccn2)on1)=O C(=O)(C1=CCC(NC(C2CCCCN2C)=O)C1)NCc1cc(C)oc1 Cc1nn(C)c(-n2cccn2)c1C(=O)NC(C)C(C(C)C)NC(=O)C(F)F N1(C(C(c2ccc3c(c2)OCCO3)C)=O)CCCC2CCNC(=O)C12 C(=O)(C(O)C1=CCCCC1)N1CCCC(CCNC(C(C)(C)OC(C)=O)=O)C1 N1(C(c2ccn(CCC)n2)=O)CCN(C(=O)C(O)CC)CC(C)C1 Cc1cccn2ncc(C(=O)NCCN(C)C(C3(C)CCC(=O)C3)=O)c12 C1(C(=O)NC(c2ncc(C)o2)C)CN(C(=O)CNC(=O)C2CC2)CC1C O=C(C1=CCCS1)NCCC1CCCCN1C(c1ccncc1Cl)=O C1(CC)C(C(=O)NCC2CC(OC)C2)CCN1C(=O)COc1ccsc1 c1(NC2CCN(NC(CSCCOC)=O)C2)ncnc2sc3c(c12)CCC(C)C3 N#Cc1ccccc1C=CC(N1CC2C(CNC(C3CCCC3(F)F)=O)C2C1)=O C12(CC)CC(C(=O)NCCCNC3CC3)(C1)C2 Cc1cc([N+](=O)[O-])cc(C(=O)NC(C)C(C)C)c1Cl.C(=O)(C(F)n1cccn1)N C1(C)(N(C(C)(COc2ccccc2)C=O)C(C)=O)CC=C(C)CC1.C1CNC1 N1(C(CCOCC#C)=O)CC=C(CC(=O)NC2CCC(C)(C)C2)CC1 C1(CC(N2CCCC(NC(c3ccc(CC)nc3)=O)C2)=O)CCCC(F)(F)C1 c1(C(=O)NC2(CC)CN(C(=O)C(C)CO)C2)ccc(F)cc1C#N C1(CCC=C)(C(=O)NCC(O)C(=O)NC)CN(C(=O)Cc2cc[nH]c2)C1 N1(C(=O)Cc2cncs2)CCCC2(CCN(C(C34CCCC3C4)=O)C2)C1 c1(C(=O)NCC23CN(C(CCCCC)=O)C(CC2)C3)nn(C)c2c(=O)[nH]cnc12 N1(C(C(C)Sc2ncccn2)=O)CCCC(NC(C2CC(OC(F)F)C2)=O)C1C CN1CCCC12CCCN(C(=O)CC(c1ccc(O)cc1)C1CC1)C2 c1(OC)nccc(C(=O)OCC(C2(C#N)CCCNC2)O)c1Br c1(OC)cncc(NC(c2csc(C(C)(C)C)c2)c2nnnn2C2CCOC2)c1 C=CCCCCN=c1cc(C)[nH]c(=NCC(C2CCCOC2)OC)[nH]1 c1(C(N2C3CC(N4CC5C(C(=O)O)C5C4)C(C3)C2)=O)cnc2ccccc2c1 Cc1cc(NC(=O)CNC(CCO)C(C)C)n(-c2ccccc2F)n1 N1(C(C2N(C(C)=O)CSC2)=O)CCN(C)C(CNC(C2CCCN2C)=O)C1 C1(OCCC)CCCN(C(C2CCCC2NC(c2ccc(C(C)C)o2)=O)=O)C1 CN1CCC(C2CCN(C(=O)Nc3cc(F)cnc3Br)C2)C1 N1(C(c2c3cc(CNCCCC)[nH]c3ccc2)=O)CCC(C2CC(COC)C2)C1 CCCC(F)(F)C(=O)N1CCC(C(=O)NCCCOCCOC)CC1 C(=O)(CCC(C)(C)C)N1C(C2CCN(C(COCCCOC)=O)CC2)CCC1 C1(C(=O)NC2CC2c2ccccc2)Cc2nccnc2CN1C(=O)C(F)F C(=O)(CC1=CCOCC1)NCCOC1CN(C(C2C(C)C2)=O)C1 Cc1cc(Br)c(CNC(Cc2cccnc2Cl)CO)cc1Cl C(=O)(C(F)(CNC(=O)Cc1sccc1C)C(C)C)NC(COC(C)=O)CO Cc1cc(C)c(C(=O)NC2CCC2C)c(C)c1.C1(C#N)(C=O)CCN(C)CC1 N1(C(=O)Cn2ccnn2)CCCCC12CN(C(C1CCCC(C(F)(F)F)O1)=O)C2 Cc1cc(CC(=O)NCC(C)CN(C(=O)C(C)C#N)C)no1 C1(C(N2C(CC=C)CCCC2)=O)CCN(C(=O)c2cccc(O)c2C)O1 C1(OC)CCCCC1CCCN(CCO)C(C1CCCOC1c1cn[nH]c1)=O C=CC(C)(CC)C(=O)N1CC(CO)(NC(=O)C=Cc2cnccn2)C1 C=CCC(F)(F)C(=O)N1CCCC(C2CCCN2C(=O)COCC2CCC2)C1 CC(C)C(N=[N+]=[N-])C(=O)N1CCN(C)C(C(=O)N(C)Cc2cccc(O)n2)C1 C(=O)(C1=CSCCO1)NCC.c12cccc(c1)O2.C1(=O)CO1 CCCC(O)C(CO)NC(C1CC(C)(NC(=O)CC2(C)CCCCC2)C1)=O C1(C(N2CCC3(C(NC(CCC(C)(C)F)=O)C3)C2)=O)CCc2c[nH]nc2C1 C(=O)(CCNC(c1cnn[nH]1)=O)NCC(c1ccsc1)C CCC(C)(O)C(=O)NC(C)CNC(c1ncc(OC)cn1)=O CCC(CNC(=O)C=CC(c1ccc(Cl)cc1)=O)CC.c1(C=O)cccn1C.N c1(CC)ccc(F)c(C(=O)NCCC2(C)CC2)c1.c1(C=O)cccnc1S.N N1(C(C2CC(=C)C2)=O)CCOC(C2CN(C(C3CC(O)C3)=O)C2)C1 C(=O)(CC(C)C(C)(C)NC(=O)C(C)CC(C)(C)C)NCCCn1ncc(C)c1 c1(C(=O)NCc2c(SC)ccc(F)c2)cc(F)cc2ccoc12 N1(CC)N=C(C(=O)NC2CN(C(=O)Cc3ccc(F)cn3)CC2C)CCC1=O C1(c2cn(CC(=O)NC(c3cnn[nH]3)C)nn2)CCCCCC1 c1(CNC(C(C)NC(CC)=O)=O)nc(C(=O)NC(C2CCOC2)CO)co1 C1(OCCOC)COCCC1NC(=O)NC1CCCOC1c1ccnn1C c1(CC)oc2ccccc2c1CN1CC(C(=O)OC(C)(C)C)C(C)C1 c1(N(CCCN(C)C)CC)ncc2ncnc-2[nH]1.C1(CC=C)(C=O)CC=CC1.N CN1CCC(C(=O)NCC2CN(C3CC3)C2)(NC(=O)Cc2ncnn2C)C1 N1(C(C2(CC)CCCN(C(=O)CCCC(F)(F)F)C2)=O)CC(=O)N2CCCC2C1 CC(C)C(C)CCNC(=O)CSc1cn[nH]c1.C1(C(=O)N)CC1.N(C)C c1(OC)cc(F)c(C(=O)NCC2CCOC2)c(F)c1.c1(C(=O)N)nocc1C C(=O)(C(O)CCCC)NCCCCC(=O)NC(C#C)CC1CCCC1 Cc1[nH][nH]c(=N)c1C(N1CC(NC(C2CCC2(C)C)=O)C(F)C1)=O c1(C(=O)NC2C(NC(CNC(CCC)=O)=O)COC2)cccc(N)c1.C(C)C c1(OC)cc(OC)nc(C(=O)C(N2CC(S(C)(=O)=O)(C=O)C2)=O)c1.CC c1(-c2cc(C(=O)NC(CNC(C(COC)C)=O)C)n[nH]2)ccc2c(c1)OCCO2 C1(O)(CN(C(Cc2ccc(C)s2)=O)C)CCCN(C(c2nc(=O)n(C)[nH]2)=O)C1 N1(C(C(CCC=C)(F)F)=O)CCC2CCN(C(c3cc(C(N)=O)cs3)=O)CC2C1 N1(C(C2N(C(c3c(CC)cco3)=O)CCCC2)=O)CCC2CCCC12 C(=O)(C1=CC2(CN(C(=O)COCC)C2)OC1)N1CCC(OCC=C)C1 C(C(=O)NC1CCSC1)(C(C)CC)NC(C(C(=O)OCC)OC)=O C(=O)(C(C)C(C)S(C)(=O)=O)NC(CC(C)NC(c1c(C)c(Cl)ccc1)=O)C C1(CC)CN(C(=O)C2=NOC(C(C)(C)C)C2)CCC1NC(=O)C(OC)OC S(=O)(=O)(c1c(Br)ccc(C)c1F)NCC(COC)(C)O CC(C)C(C(=O)N1CC2(CCOCC2)C1)C(C)NC(c1ccncc1N)=O C(=O)(C(F)C(F)(F)C(F)(F)F)NC1C(NC(c2snc(C)c2N)=O)CCC1 N1(C(c2cc(OC)n[nH]2)=O)CCN(C(c2ncsc2S(N)(=O)=O)=O)CC2(CC2)C1 N1(CC(=O)NC2C(NC(=O)CCC3CCC3)CC2)CCOCC1 C(=O)(C#CC(C)(C)C)N1CC2C(C(N(CCC(C)C)CCO)=O)C2C1 N1(CC(=O)NC(CCC)C)CC2C=CC1C2.c1(C=O)cnn(C)c1C(F)(F)F c1(OC)cccc(CNC(=O)CC(c2ccc(N)cc2)C)c1-n1cccn1 N1(C(c2c(CC)csc2)=O)CCCC2(CCC2)C1.c1(C(=O)N)ccn(C(C)C)n1 c1(N(C)C)ccccc1CCCNC(c1ccc(C2COCCN2)n1C)=O c1(C(N2CCCC(N(C)C(C34CSC(C3)C4)=O)CC2)=O)cnc2ncnn2c1N C1(NC(c2c(C)nc[nH]2)=O)CC2(C1)CC1(CC(C(=O)ON)C1)C2 CC(CC(F)(F)F)NC(=O)CN(C(c1cccc(CO)c1)=O)CC1CC1 C(=O)(C1=CCCOCC1)N1CCC(C)(CC(N2CCN(C(CC)C)CC2)=O)C1 C1(C(N(CC(CNC(C(CC)F)=O)C)C)=O)CC(=O)N(C2CCCC2)C1 C12(NC(c3cnn(C)c3Br)=O)CCC1CN(C(c1cc(Cl)cs1)=O)C2 N1(C(c2ccc(C)[nH]2)=O)CC2(C)CN(C(=O)CCC3CCCCO3)CC2(C)C1 C1(F)CCNC1.C12CC(C(F)(F)F)(CO1)C2.O=CC=CC(=O)N1CCC1.C C1(C(=O)NC2CC3CC2N(C(=O)C2=COCCC2)C3)Cc2ccccc2O1 C#CCCCCC(=O)NC(C)CCCNC(c1c(C)nn(C)c1Br)=O N1(C(c2cc(C)n(C)c2)=O)CC(C)CN(C(c2cn(C)c(=O)cn2)=O)C(C)C1 c1(SCC(=O)NC2CC(C)(NC(CSCC#C)=O)C2)ccc(Br)cc1 c1(C(=O)OC(c2ccc(C)c(C)c2)C)cnc2c(C)nsc2c1 c1(SC)ccc(OC(C)C(=O)N(CCC)C)cc1.C1(CC=O)CCOC1(C)C.N N1(C(=O)OC(C)(C)C)CCC(NC(c2nccc(N)c2Cl)=O)CC1C1CC1 CC1CCC(NC(c2cc(O)nc(O)n2)=O)CN1C(c1ccc(N)c(F)n1)=O C(=O)(C1CC(=O)Nc2ncn(C)c21)NC12C(CN(C(CC(C)C)=O)C1)CC2 N1(C(c2cccc(N(C)C)c2)=O)CCOC2CCN(C(c3cccn3C)=O)CC12 c1(C(N2CC(O)(CNC(=O)CCc3cncs3)C2)=O)c(F)cncc1Cl C(CCNC(C1CCOC1C(C)C)=O)(C(=O)Nc1ccc([IH]C)nc1)OC C(=O)(C1CSc2ccccc21)NC(CCNC(COCCCC)=O)C C(=O)(C1=CC2(CN(C(=O)C(F)C(C)(C)O)C2)OC1)NCC(CC)CO C(=O)(CC1=CCOCC1)NC(CCSC)C(=O)NCC1(S(C)=O)CC1 Cc1cc(F)ccc1C1(C(=O)NC)CC1.C1C2CC2CN1C(C1CCCCO1)=O Cc1cc(C(=O)NCC2CCCN2C(=O)COc2ccccc2F)ncc1Cl N1(C(c2c(CC)ccs2)=O)CCC2CCC(NC(=O)CCCCF)C1C2 CC1(C(N2CCC(NC(=O)CCCc3ncco3)C2)=O)CCC(=O)NC1 c1(CCC(=O)NC2C(CNC(Cc3ccc(C)s3)=O)CCC2)cc(F)ccc1F c1(OCC(CN(C(CC2C(C)CCO2)=O)C)O)ccc(C=O)cc1.N(C)C C1(C(N2CC(CC(C(=O)NCCCO)F)C2)=O)CN2CCC1C2 C#CC1(F)CCN(C(=O)CC2(NC(C3CCC(F)(F)C3)=O)CCC2)CC1 c1(NC(C2CC(O)CN2C(C2CCCO2)=O)=O)cc(N2CCCC2)ccn1 N1(C(C)=O)CCC(CNC(=O)Cc2cccc(C)c2)C(C)C1 CCC(C)CC(=O)C(=O)NCCN(C1CCCC1)C(=O)C=Cc1nccs1 N1(C(C)=O)CCC(CNC(C23CSCC2C3)=O)C1 c1(C(=O)NCC2N(C(CCC3CCC(C)O3)=O)CCC2)cc(C#N)cs1 C1(C(C)(C)C)CCN(C(=O)C=CC2CCCCC2)C1.C1(CC=O)CCNC1=O.C CCCC(C)(CC)C(=O)N1CC2CCC(N(C(=O)CS(N)(=O)=O)C)C2C1 c1(OC)cccc(C=CCN2CCc3ncsc3C2)c1OC C(C(=O)NCC1CCCN(C(c2cccnc2NC)=O)C1)(C(C)C)OCC N#Cc1c(C(=O)NCCC2CCCCN2C(=O)CO)cccc1Br Cn1cc(NC(=O)CN2CCC(C(=O)O)CC2)c(-c2cccnc2)n1 C(C)(CN=c1[nH]c(Cl)ncc1Cl)NC(C(COC)C)=O N1(C(C2(NC(=O)CCCC(=O)N(C)C)C(C)C2)=O)CCC12CCN(C)C2 c1(NC(N(C2CCN(C)C2)CC(=O)OC)=O)cccc(C(C)F)c1 c1(Nc2ncc(-c3ccc(NCC)nc3)cc2C)cc(C)c(OCOC)c(C)c1 C(=O)(C1=CCCC1(C)C)NCC1CC(OC)CN1C(c1ccn2c1CCCC2)=O C1(CN(C(=O)C(C)Cn2nc(C)cc2C)CCC(=O)OC)C2CCC1CNC2 c1(C=O)cc(F)c(Cl)c([N+](=O)[O-])c1.N=c1[nH]nc(SCC(=O)NCC#CC)s1 N1(C(C(C)C2CCCO2)=O)CC(F)(F)CC1CNC(C1CCCC2(CC2)C1)=O C(CC(C(=O)O)NC(=O)Cn1nnnc1C)(C1CC1)OC C1(OC)(OC)CC(C(=O)NCCOCC(=O)N(C)C)C1.C1(F)CCCC1 O=C1OCCC1CCNCc1cn(CCNC2CCCC2)nn1 c1(C(=O)NC(CC)CNC(=O)C(C(C)CC)OC)ccc2cc(F)c(F)cc2n1 CC1(C)CCC(C(=O)NC)(NC(=O)CCC2CCCCC2)C1.c1cncc(Cl)c1 C1(CNC(C2(CC)CN(C(=O)C(N)=O)C2)=O)CCCC(OC)C1 c1(NC(=O)NCc2cc(OC)nc(C)c2)nc2c(s1)CCCC2 Cc1oc(C)c(C(N2CCC(NC(=O)C(Cl)=CCl)C2C(C)C)=O)c1C C1(C(=O)NC(c2ccccc2)CNC(C2(O)CCC2)=O)(CC)CC1(F)F c1(CSCC(=O)NC2(C)CN(C(CCc3n(C)ccc3)=O)C2)cccc(Cl)c1 N1(C(c2c(OC)ccc(OC)c2)=O)CCC2(CCCN(S(=O)(=O)CCBr)C2)CC1 N1(C(CNC(C(CC)C)=O)=O)CCCCC1CNC(c1sc(C)nc1C)=O.O CCCC(C)CN=c1[nH]c(=NCc2ccc(CO)c(F)c2)c2c(F)cccc2[nH]1 C1(NC(c2oc(C)c(CO)c2)=O)C2CCC(C2)C1C(=O)NCC(O)C(C)O c1(C(=O)NC2C=CCN(C(CCOC(CC(C)C)C)=O)C2)ccc2c(c1)COC2 N1(C(C(=O)NC(C)C)C)CCC(F)(F)C(C)C1.c1cccc(F)c1.C(=O)C.N c1(C(N2CC=CC(NC(c3c(C)noc3)=O)C2)=O)oc2c(Cl)cccc2c1C c1(NC(C2(C)CN(Cc3nc4ccccc4[nH]3)C2)=O)cc(Br)cnc1C#N C1(C(N2C(C)(CNC(CNC(C)=O)=O)CCC2)=O)C2C3CCC(C3)C12 N1(CCNC(=O)NCCCO)CCOCC1c1nc(C(F)(F)F)n[nH]1 c1(C(=O)NCCC(O)CNC(=O)C(C2(O)CCOCC2)F)cn2cccnc2n1 C(C)(CCC(=O)NCC(c1ccccc1)CNC(=O)CNC(C)=O)OC S(=O)(=O)(c1cccc(Cl)c1F)N1CC(CC(=O)Nc2ccnc(Cl)c2I)OCC1 c1(OCC)cccc2[nH]c(C(N3CC(C)C(O)C3)=O)cc12.C(=O)C1=CSCS1.N c1(OC(CCC2(C)CC2(F)F)=O)ccc2cccnc2c1 C1(CNC(C2N(S(C)(=O)=O)CC2)=O)CCOC1.C(c1ccoc1)=CC=O CCC1=NOC(CNC(C2C3CC2N(C(C2(C(C)C)COC2)=O)C3)=O)C1 c1(OC)ccc(C(=O)N(C(C)C)C)nc1.c1(C(C=O)N(C)C)cccc(Cl)c1 C(C(C(C)C(C)C)NC(=O)CCCCC1CCCCC1)NC(COCC#C)=O c1(C(N(C2CCCN(C(C3(C)C=CCC3)=O)C2)C)=O)ccc(Br)c(F)c1N C(C(C)(C)C#CC(=O)N1CCOC(C)(C)C1C)NC(C(F)=C(C)C)=O C(=O)(C1=CC2(CCNC2)C1)N1C(CC)CCCC1C N1(C(C)C)C(=O)COCC1C(=O)N.c1(CC(=O)N(CCC)CCO)cncnc1 Cc1ccc(N)cc1C(N1CC(NC(c2cc(C(F)(F)F)n[nH]2)=O)CC(C)C1)=O C1(N(C(c2c(C(C)C)ocn2)=O)C)CCCN(C(C2CCC(N(C)C)CC2)=O)C1 C1(C(N(CC(=O)NCc2snc(C)n2)C)=O)CC2(CCO1)CC2.C1CS1 c1(C=O)ccc(-n2cncn2)c(N)c1.C(=O)(CCC1CCCO1)N(C)C.C1CC1 CC(C)CC(C(=O)N1CC2CC(C(=O)NCC(O)(CO)CO)CC2C1)C(C)C N1(C(c2c(C)nc(Cl)cc2)=O)CCCN(C(=O)C(F)C(F)(F)F)C(CO)C1 N(C(=NCCCC(C)O)NC(C)C)Cc1ccc(OC)c(OC(C)C)c1C C1(C(N(C2(CC(=O)NC(C(C3CC3)OC)C)CC2)C)=O)CC2CCC1CC2 c1(NC(C2(F)CN(C(c3c(SCC)cccc3)=O)C2)=O)c(F)ccc(Cl)c1F Cc1ccc([N+](=O)[O-])c(C(c2nnnn2C2(C)CC2)NCC2CCC=CCC2)c1 C1(C(N2CCC(C(C(=O)NC3(CC)CCOC3)C)C2)=O)CC2(CCO1)CC2 Cc1c(C(=O)N(CC(N2CC(N(CC(F)F)C)C2)=O)C2CC2)cncc1F S(=O)(=O)(c1ccc(C)cc1C)N1CC(CC(=O)Nc2ccc(OC)cc2Cl)C1 C=CC(C)(C)CC(=O)NC1CC2CN(C(c3csc(C4CC4)n3)=O)CC12 CCC(CCCC(=O)N1CC2CSCC2(C)C1)NC(c1nc(=N)cc[nH]1)=O c1(C(N2CC(N(c3ccncn3)C)C2)=O)ccc2oc(=O)oc2c1 CCCCC(CCCC)NC(=O)C(c1ccco1)NC(=O)Cc1cnccc1C C(CC(C)CC)(C(=O)NCC1CC(C)(O)C1)NC(c1ccc(CC)cc1)=O CC1(C)CC(C(=O)NC2CCCCC2(C)C)CN(C(=O)C=Cc2ccncc2)C1 C1(NC(CCCC)=O)COC2(C1)CN(Cc1ccc(C(C)(C)CC)cc1)C2 CC1=C(C(=O)NCC2(CO)CCCN(C(c3cccc(O)c3F)=O)C2)CCO1 N1(C(c2nccc(N)c2)=O)CCCC2(CCCCC2NC(=O)Cc2cccs2)C1 Fc1cc2[nH]c(CNc3ccc(Cl)c(C(F)F)c3)nc2cc1Cl CCC(Cc1ccccc1)C(=O)NC1CCC1NC(c1nc(C)oc1C)=O Cc1c(C=CC(N2CCC(CNC(C3OCC3(C)C)=O)C2)=O)cnn1C c1(C(=O)NCCC(C)NC(c2cn[nH]c2)=O)cccc(C(F)(F)F)c1F C(c1cncnc1O)=CC(=O)N(C(C)CCNC(C1(CC(F)F)CC1)=O)C c1(C=O)ccc(C)c2c1CCC2.C12(C(=O)NCCCC)CCN(C1)S(=O)(=O)C2 c1(C(C)C)ncc(C(=O)NC2CCCCC2NC(c2ccncc2O)=O)cn1 C(CNC(c1csc(C(C)C)n1)=O)(CCNC(=O)Cn1cnnc1O)OC C1(C(=O)Nc2scc(C(C)=O)n2)CC12CCN(Cc1scnc1C)C2 CC1(C)CC(C(F)(F)F)(C(=O)N)C1.N1(C=O)CCCC1.C1CC1.C(=O)C C1(NC(C(COC)(C)O)=O)CN(C(c2ccc(C3CC3)cc2)=O)C2(CCC2)C1 n1(CC(=C)C)nnnc1C(C)(CC1CCCO1)NCC1COC(=O)N1 C=C1CC(C)(C(=O)NCC(C)(CO)NC(=O)CC)C1.c1(C=O)ccco1.N C(C(=O)NCC1CC(NC(c2cc[n+]([O-])cc2)=O)CC1O)(C(C)(C)C)OC C1(NC(C=C(COC)C)=O)CC2CC(NC(C3(Br)CC3)=O)CC2C1 C#Cc1ccc(F)c(C(=O)NCCC2(C)CCN(C(=O)CCCN=[N+]=[N-])C2)c1 CCCC(C)CC(=O)NC1CC2(C1)CN(C(c1ccccc1Cl)=O)C2 C1(CC(=O)N)CN(C(C2CCC2)=O)CC12CC2.C(CCC(N)=O)OC.C(C)C c1(C(=O)NC2(C(=O)NCCCC=C)CSC2)cccc(F)c1N Cc1nccc(Cl)c1C(=O)NC(C)CNC(=O)CC.CC(F)(F)C(F)(F)F C(C(CNC(C1CC(F)CN1C)=O)C(F)(F)F)NC(c1cnc(C)o1)=O n1(CC)ncc(C(N2CC(CNC(C3CC(C)=NO3)=O)C2)=O)c1Br c1(C(N(CCN(C(=O)CC(C)S)CC)CC)=O)cc(C(F)(F)F)n[nH]1 n1(CCNC(C(N2CCN(CCCN(C)C)CC2)=O)=O)cnc2ccccc12 C1(NC(CCc2ccc(C)s2)=O)CCN(C(=O)CCSc2nccn2C)CC1 N1(C(CCOC(C)C)=O)C2CCC(C(N3CC4CC3(C=O)C4)=O)C1CC2.CCO.O c1(CNC(C(CC)NCC)=O)nnc2n1CCN(C(C1(C)CC1(C)C)=O)C2.C c1(C(=O)NC(CCN(C(CC=CCCCCC)=O)C)C(C)C)cnn2ccsc12 Cc1cccc(CCC(=O)NC2CCC(CCNC(=O)Cc3cncn3C)C2)c1 N1(C(C2CN(C)C2)=O)CCCC(C2CCN(C(=O)COC3(C)CCC3)CC2)C1 C(=O)(C1=CC(C)(C)C1)NCC1C(C(=O)NCCC2CC(C)C2)CCC1 c1(OC)cc(NC2CCN(C(c3cc(O)nn3C)=O)C2)c(F)cc1[N+](=O)[O-] C1(CC)CN(C(=O)CC2CC3(C2)CN(C(=O)CC2CCC(=O)NC2)C3)CCCO1 C1(C)(CCC(=O)Nc2ccc(CC)[nH]2)CCCN1C(c1ccc(C)nc1)=O.O c1cccc(O)c1C.C(C(C(=O)O)NC(C1CC(n2cc(C)nn2)C1)=O)SC.O C1(CC)CN(Cc2ccc(C)nc2)CCN1C(c1cccc(OC)c1O)=O c1(SCC(=O)NC2CN(C(C(CC#C)C)=O)C(CO)C2)nc2ccccc2o1 S(=O)(=O)(C1CCCN(C(c2ccccc2)=O)C1)NC(c1ccccc1F)CC S(=O)(=O)(c1csc(C(=O)N)c1)NC.c1(C=O)c(N)ccc(C)c1F.C1CCC1 N1(C(c2ccc(CO)o2)=O)CC2(CCCCN2C(C23CCCC2CC3)=O)C1 C1(CN(C(C=C(C)Cl)=O)C)CCCN1C(C1(C(C)(C)C)CCCC1)=O N1(C(CN=[N+]=[N-])=O)CC2(C(=O)Nc3cc(CO)cc(F)c3)CC1CCO2 C1(C(=O)NCCn2c(=N)nc[nH]2)CCCC(CC(F)(F)F)N1 N1(C(CC(CNC(C2C(C)SCCC2)=O)O)=O)CCC12CCC(O)CC2 C(CCC(C(=O)N1CC(OCCO)C1)NC(C1CC=CC1)=O)OC c1(NC2CN(C(Cc3c(C)nn(C)c3)=O)C2)ccc(Br)cc1[N+](=O)[O-] C1(NC(C2C(=C)C2)=O)CN(C(C2(C)CCCC2CC)=O)CC1C C1(C(=O)NCC(C)N(CC(=O)N(C)C)C)CC12CCOC2.c12ccccc1S2 N1(C(c2cn(C)c(=O)n2C)=O)CCCC(C2CN(c3nc(Cl)ncc3Br)C2)C1 C(=O)(CCC(=O)N1CCCC1CNC(C)=O)NCCC.C(c1cncs1)=C C1(NC(c2cc(C)nnc2)=O)CCCC(C(N2CCC2(CO)CO)=O)CC1 n1(CC(=O)NC2C(CNC(C(C)(C)C3CCC3)=O)C2)cc2ncccc2n1 N1(CC(=O)NC(C2CC3CCC2C3)CC)CCN(C)CC1 C1(C(N2CCCC2c2ccc(Cl)nc2)=O)CC(F)(F)CCN1 c1cnn(C)c1.C(=O)CCc1ccoc1.C(CC)N(C(=O)C=CC)CC.N O=S(=O)(c1ccc(NCC2OCCO2)c(Cl)c1)NCC1CC2C(C1)C2(F)F C1(C(=O)Nc2cn(CCC)nc2)CCCN1NC(=O)C1CCCC(O)C1 C=C(C)CCC(C(=O)NCC)N(C(C)COC(C)=O)C C1(NC(C(CC)OC)=O)CC1C1CCN(C(=O)C=Cc2cccc(O)c2)CC1 c1(CCCC)ccc(N(C)C)c(C(=O)COC(=O)CN2CC3(COC3)C2)c1 C1(CC=C)(NC(=O)C=Cc2nc(C)co2)CCN(C(c2cnsn2)=O)CC1 N1(CC)CC2CC1CN2C(c1ccc(CN2CCN(C(=O)CO)CC2)cc1)=O C1(NC(C2CCC2(F)F)=O)CCCCC1.c1(C(C(=O)N)O)ccc(C2CC2)cc1 N1(C(C2OCC(C)(C)C2)=O)C2CCC1CC(NC(c1csnn1)=O)C2 c1ncc2c(n1)CCCC2N=c1[nH]c(=NCC2COCCO2)[nH]c2c1CCC2 C(C)(C)(CC(F)C(=O)Nc1csc(C)c1)NC(c1ncn(CC)n1)=O C(c1cccnc1)=CC(=O)NCC(C)C1CC1.C(=O)C(O)Cc1cnc[nH]1.N C1(CC(N2C(CNC(CC(=C)C)=O)CCC2)=O)CC2(CCOCC2)CO1 N1(C(C2C(=C)C2)=O)CC(NC(C2CCC(C)(CC)O2)=O)C(C)C1 N1(C(C2CC(CCC)C2)=O)CCN(C(=O)C(C2CCCC2)C2CCCC2)CC1C C1(C(=O)NCC2(OC)CN(C(C3(F)CCC3)=O)C2)CCN(OC)CC1 N1(C(COC)=O)CCN(C(c2ccc(-c3ncc[nH]3)cc2)=O)C(C2CC2)C1 CC(C(=O)NC(C1CCCC1)CNC(=O)C=CI)C1CCCO1 N1(C(CC=C)=O)CCOCC(F)(CNC(c2cc(C)cc(Br)c2F)=O)C1 C(=O)(CC(C(F)F)n1ccnc1)NCC(C1CCC1)NC(C(C=C)(C)C)=O CC(C)C(CCNC(C1(C#N)CC1)=O)NC(C1(CO)CCCO1)=O Cc1ccccc1C(=O)NC1CCC(CC(=O)NCc2csnn2)C1 C(=O)(C1=NNC(=O)C1)N1C(C)CC(CNC(c2c(C)[nH]cc2)=O)C1 Cc1csc(C(C)C(=O)N(CC(C)NC(c2ccn(C)n2)=O)C)n1 C(CCC(=O)NCC(C)(Cn1cccn1)NC(C1SCC=C1C)=O)=CCC=C CC#Cc1nnc(N(C)C(C2CCN(C(=O)OC(C)(C)C)CC2)C)n1CC c1(NC(C)CN(C)C(c2ccc[n+]([O-])c2)=O)nc[nH]c2ncc(C(N)=O)c1-2 c1(SCCC)ccc(C(=O)NC2CCOC(CNC(C3CC3C)=O)C2)cc1 n1(CC)nc(C)cc1C(=O)NCC1CN(C(C2CC2C(C)C)=O)C1.C N1(C(C2C(C)OCCC2)=O)CCC(Nc2ncc3ccnc-3[nH]2)C2(CCC2)C1 N1(c2cccc(OC)c2OC)CCC2(CCCN(C(=O)C(C)n3cncn3)C2)C1 c1(C(N2C(C)(CC)CC(NC(c3cc(C)on3)=O)C2)=O)ccc(N=[N+]=[N-])cc1 N1(C(C(C=C)O)=O)CCCCC1C(C)(C)CNC(c1cc(Br)n(C)c1)=O N1(C(c2on(C)c(=O)c2)=O)CCC2CN(C(c3ncccc3S(C)(=O)=O)=O)CC12 Cc1ccc(C(=O)NCC(C)(CC(C)C)NC(C2CC23CCCC3)=O)cc1C#N C1(NC(c2c(C)csn2)=O)CCN(C(=O)CN=S(C)(C)=O)C(C2CC2)C1 C1(C(=O)NCC(COC)O)CN(C(c2cc(=O)cc[nH]2)=O)CC(C)(C)C1 N1(C(COCCC)=O)CCCC(C2CCCN(C(=O)CCc3ccnn3C)C2)C1 CCCCCC(C)CC(=O)N1CC(O)CC1CNC(C1CCC2(CC2)C1)=O C1(NC(CCC#CC)=O)CCN(C(c2cc(Cl)cc(C(F)(F)F)n2)=O)C(C)C1 N1(C(c2c(COCC)nc(C)nc2)=O)CCCC(CO)CCC1 N1(C(C(C)N(C(C)=O)C)=O)CCC2(CCCN2C(=O)Cn2ncn(C)c2=O)C1 C1(CNC(Cc2c(C)cccc2)=O)CN(C(=O)CCP(C)(C)=O)CC2(CCC2)O1 C(=O)(N=c1ccn(CC(=O)N(C)C)[nH]1)NC1C(c2c(C)n(C)nc2)N(C)C(=O)C1 O=C(CCOC1COC1)NC1CCC1NC(=O)CC1CCCO1 C#CCCC(O)CCNC(=O)C(C(C)C)NC(=O)C(C)(C)n1ccnn1 Cc1cc(NC(=O)C(C)(C)C)c[nH]c1=NCc1cc2sccc2s1 C(=O)(C1COc2ccc(F)cc21)N1C2CCC(NC(C(C(C)C)C#N)=O)(CC2)C1 O=C1NC(=O)N2CCN(C(c3cnc(-c4ccccc4)cn3)=O)CC12 c1(OC)cccc(COCC(=O)NCC(C)C)c1.c1(C=O)cnc(O)n1C.N C(=O)(C(C)(C)C1CCCC1)N(C1(C=O)CC1)C1CC1.CCC.C(C)=O.N c1(C(N2CC(COC)N(C(=O)CCN(C)CCO)CC2)=O)noc2c1COCC2 c1(C(C(=O)NCCCC2(NC(C(C)c3ccco3)=O)CC2)O)ccccc1Cl C1(NC(C2CCCC(NC(c3cc(Cl)no3)=O)C2)=O)CC2(CCC2)C1O CC1(NC(c2csc(F)c2)=O)CCCCC1C(=O)Nc1cncc(CO)c1 C1(C(=O)NCC(C2CCN(CC)CC2)C)CCN(C(=O)C2CC2Cl)O1 c1(C(N2C(C)CC(NC(=O)CCn3ccnn3)C2)=O)cccc2ncoc12 C(C(C(=O)NC(C)CN=[N+]=[N-])NC(=O)C(=C1CCCCC1)F)SCC C1(O)(C(CNC(CCCOCCOC)=O)C)CCN(C(c2cnc(C)cn2)=O)C1 c1(C=O)ccc(S(N)(=O)=O)cc1F.N1(C(C(C)OCC)=O)CCC(CO)C1.N c1(CNC(CCC(=C)C)=O)nnc2n1CCN(C(c1cnn(CC3CC3)c1)=O)C2 N1(C(CCCC(CC)(C)C)=O)CCCCC(C2CN(C(c3csnc3C)=O)C2)C1 Cc1nc2ccc(NC(C3(C(F)F)CC(N)C3)=O)cn2c1Br N1(C(CCCOC(C)C)=O)CCN(C(=O)CSCC(N)=O)CC1CF CCC(CC)(CC)C(=O)NCC1CN(C(=O)C(C)(C)C(N)=O)CCC1(F)F N1(C(C2CCC(CCCC)CC2)=O)CCOC2CN(C(C3(C#N)CC3)=O)CC12 N1(C(Cn2ncc(C)c2)=O)CCC(NC(=O)C(c2c(F)cccc2F)C)C(F)C1 c1(CC(=O)NC2(CNC(C(CCC)OC)=O)CCOCC2)cnn2c1OCCC2 Cc1ccccc1C1(C(=O)NCC2CCCN(C(C3(CCO)CC3)=O)C2)CC1 c1(N2CCCC(NC(=O)Cc3coc(C(F)F)n3)C2)nc(Cl)nc2[nH]c(O)nc12 C(CO)(C(=O)NC12CC(C(N3CC(CO)C3)=O)(C1)C2)N(C)C c1(C(N(C(C(=O)OCC)C)C)=O)cc(C)on1.C12(CC=O)CCCC1C2 CCCCCCNC(c1sccc1OC)=O.C1(C=O)CCN(S(C)(=O)=O)C1 C=CCCCCCC(=O)NCC1CCC(N(C)C(c2ccc(NC)cc2)=O)CC1 O=C1NC2(CCSC2)C(=O)N1CCCOCc1cccc2ccccc12 c1(C(N2CC(O)CC(NC(C3N(C)CCC3)=O)C2)=O)c(Cl)ccc(Cl)c1Cl C1(NC(=O)CSc2ccncc2)CC2CCC1(CNC(=O)C1=COCCC1)C2 S(=O)(=O)(c1c[nH]ccc1=NC(C)c1ccncc1Cl)NCc1c(CC)nco1 N1(C(c2c(SC)csc2)=O)CC2CN(C(C3CCS(=O)(=O)N3)=O)CC(C1)O2 N1(C(CCOC)=O)CCC(F)C(NC(c2ccncc2)=O)C1 N1(C(CCC)=O)CCC(c2ccccc2)(NC(=O)C(C)OCCN(C)C)C1 C(CCSC)(C(=O)NCC1CC[Si](C)(C)C1)SCC C#Cc1ccc(C(N2CCCC(O)(CNC(=O)C(C)=C(C)CC)C2)=O)nc1 c1(C(N(CCN(C)C)C)=O)ccc(C)cn1.C1CC=CC1.CCCF.C(=O)(C)N N1(C(C2(C)C(C)OC(C)(C)O2)=O)CC2CCC(C1)C(NC(c1csc(Cl)c1)=O)C2 C(CCC(=O)NC(c1cc[nH]n1)C)N(C(C(C)SCC)=O)C c1(C(=O)NCC(C)NC(c2scnc2Cl)=O)ccc(CN(C)C)o1 N1(C(C2CC2F)=O)CCC2(CCCN2C(C2CCC(n3cccc3)CC2)=O)CC1 c1ccc2c(c1)CCC2.N1(C(c2c(C)nsc2)=O)CCCC1(C)CNC(=O)CO c1(OC)cc(N)c(F)cc1C(=O)NC1CCC1NC(c1cnccc1C)=O Cc1c(C(=O)NCC(C(C)C)NC(=O)C(c2cccc(N)c2)O)cccc1Cl c1(C(N2CCC(C)C2)=O)ccc(S(N)(=O)=O)c(F)c1.C1(CC)OCCC1C=O.N C(=O)(C(=O)CCC(C)(C)C)NCC(CC(F)(F)F)NC(=O)OC(C)(C)C N1(C(=O)Cc2cnsc2)CCCN(CCc2cn(-c3ccccc3O)nn2)CC1 N1(C(c2c(C)ccc(F)c2)=O)CC(C)CN(C(=O)C)C(C)C1.C(=O)C(C)(C)C.N C1(CNC(c2c(CC(C)C)onc2)=O)CN(C(C2CCC2)=O)CCC1(F)F.C c1(CC(=O)NCC2N(C(CCN(c3ccccc3)C)=O)CCC2)ccc(F)cc1 CC1=CCSC1C(=O)N(C)CC1(C)CC1.c1(C2(C(=O)N)CC2)ccno1 c1(NC(=O)NC2CCC(CNc3nccc(OC)n3)CC2)ccc(F)c(Cl)c1 N1(C(C2CC(N(C)C)C2)=O)CCCC(C)(C)C1.C1(n2cccn2)(C=O)CCC1.N c1(SCCNC(C2C(c3scc(C)n3)C2(C)C)=O)ccccc1.C(=O)C(C)O CC1(C)CCCC(C(=O)NC2(C3CN(C(C4(C#N)CC4(C)C)=O)C3)CC2)CC1 c1(CC(N2C(C)(CNC(CC3N(C)CCC3)=O)CCC2)=O)ccc(F)c(Cl)c1F N1(C(c2cocc2)=O)CC(C2CC2)C1C1CC1.S(C(F)(F)F)CC(=O)NC C1(NC(C(CC)NC(=O)C(C)C(=O)OC)=O)CCCCC1(C)C Cc1cc(C(=O)N(CC(C)CNC(=O)C(C)CC2CCCC2)C)c(C)cn1 C1(C(=O)NC2C(NC(c3c(C)nc(C4CC4)[nH]3)=O)COCC2)COCCC1(F)F C1(C(C(N2CC(C(=O)O)CC(CC)C2)=O)N)C2CC3CC(C2)CC1C3 C1(C(=O)NC(CC)CO)(NC(c2[nH]ccc2C)=O)CCCC1 C1(CNC(CC=C(C)C)=O)CC2CCC(C1)N2C(c1cnc(N)c(N)c1)=O N1(C(C=C(C)C2CC2)=O)CC(C(=O)NCC2COCC2(C)C)CC1(C)C Cc1ccc2c(c1)SC(C(N1CCC1CNC(C1(CCF)CC1)=O)=O)C2 N(C1COc2ccccc21)C(C1CC2(CCN1C(=O)CC1(O)CCC1)CC2)=O Cc1cn2c(CC(=O)NC(C)C(C(=O)NCC3CCCC3)C(C)C)csc2n1 C1(CNC(c2ccn(C(C)C)n2)=O)COCCN(C(=O)CC2(O)CCOC2)C1 C1(NC(=O)CCCF)CC(CNC(=O)CCc2cnc(O)[nH]2)CC1O C12(CC(=O)OCC)CCC(CC1)N(C(=O)CCc1nc(CC)n(C)n1)C2 C=CCC(CNC(=O)Cc1cc(COC)no1)NC(c1ccoc1)=O N1(C(C(c2cccc(C)c2)C)=O)CCC2CN(C(=O)C#CC3CCCC3)C2C1 c1(NCC(C)NC(=O)C(C)(C)C(F)c2ccccc2)c(C#N)nnc2ccccc12 c1(COCC)cn(CC2CC(NC(=O)CCc3ccncc3)C2)nn1 c1(Sc2ccc(C(=O)NC3C(CNC(=O)CCF)C3)cc2)c(F)cccc1F c1(C(=O)NC(CCCC)CNC(=O)CN(C)CCOC)nc(OC)ccc1F CCCC(C(=O)NOCC1CCOC1)NC(=O)CC(C)(C)O N1(C(C2C(C)C2)=O)CCC(NC(=O)Cc2cc(C(C)C)no2)C12CC2 CC(C)(C)CC(=O)NCCC1CCCN1C(c1ccc(CC(C)(C)O)s1)=O CCC(C(F)(F)F)NC(C1(COC)C=CCN1C(=O)C=C(C)C)=O.O Cc1ccn(C(C)CC(=O)NCC(C)CNC(=O)COC)n1.c1ccnn1C Cc1ccc(C=CC(N2CC(NC(=O)CCc3cc(C)[nH]n3)CC2(C)C)=O)nc1 C1(C(=O)NCCC(C)N(C(=O)CS)C)CNC(=O)C(C)(C)C1.C(C)(C)C N1(c2c(C)ccc(F)c2)C(=S)NC(c2cnc(O)c(C)c2)C2=C1C(C)(C)NC2=O CC1CN(C(c2cc(-c3ccccc3)no2)=O)CC1NC(C1CN(C(N)=O)C1)=O C1(C(=O)OC(C)(C)C)(C(=O)NC2CC2NC(=O)C2CC2)CCCCO1 c1(CC)cc(-c2nc(-c3ccnc(Cl)c3)nn2CC2CC2C)c(C)nn1 c1(C(N2C(C(N3C(C(C)C)CC(O)C3)=O)CCC23CC3)=O)ccc2nccn2c1 c1(OC)nc(Cl)c(C(N2CC(CC(C)NC(=O)C(O)Cn3cncn3)C2)=O)s1 C(CC(F)F)(C(=O)N1CC(C(C)(C)C#N)C1)N(C(C(C)SC)=O)C c1(C(=O)NCC(CNC(CCC(C)N(C)C)=O)(C)O)c(F)ccc2ccncc12 C(C)(CC(C)(C)C)(c1n(CCC)nnn1)NC(c1cc(C)cnc1F)C C(C)(CCC(=O)N1CCC(O)(C(C)NC(c2cnn(C3CCCC3)c2)=O)C1)OC C12(C(=O)N)COCC1CN(C(C1CC(=O)N(C)C1)=O)C2.Cc1cc(C)cc(C)c1 N1(CC=O)C(=O)NC2(CCCC2)C1=O.C(=O)(C(C)C=O)N1CCC1.COC C1(NC(C=Cc2n(C)cnc2)=O)CCN(C(c2cccc(Cl)c2F)=O)CC1O C1(NC(C2(C)CCCCO2)=O)CCCN(C(c2cnc(N)c(Cl)c2)=O)CC1 C=CCC(C(=O)N(C1CCN(C(c2ccc(F)s2)=O)C1)CCC)C(C)C N1(C(c2cc(OC)ncc2)=O)CC2(C1)CN(C(=O)CCC13CCC(CC1)C3)C2 N1(C(c2cnc(C)[nH]2)=O)CC(NC(c2nnn(C)c2C)=O)C2(CC2)C1 N1(C(Cn2cc(C(C3CCCO3)C)nn2)=O)CCCC(c2nccs2)C1 c1(C(C)C(=O)NCC2CCCN2C(C2CC2C)=O)cccc(F)c1 c1(C(N2C(C)CCC(NC(C(CC)(C)CC)=O)C2)=O)nc2c(s1)CN(C)CC2 C1(C(N(C)Cc2nnc(C)o2)=O)C2CCC(C2)N1C(C1CC2CCC2C1)=O C(=O)(C1=CC2C=CC1C2)N1CC(CC(=O)N)CC1(C)C.C=C(C)C(F)(F)F c1(C(=O)Nc2ccc(NC(C(C=C)O)=O)c(C)c2)cc2ncccc2[nH]1 Cc1[nH]nc2cc(C(=O)NCC3C(C)CCN3C(=O)CCC(C)(F)F)ccc12 c1(NC)ccc(C(=O)NCC(O)CCNC(=O)COC(F)(F)F)c(C)c1 CC(C)C(C)CNC(=O)CCCN1CCCCC1.C1(CC=O)CCC(C)(C)O1.N Cc1cc(C)c(C(=O)NC(C)CCCCNC(c2cc[nH]n2)=O)c(C)n1 Cc1cccc(C2(C(c3nnnn3CC3CC3)Nn3ccnc3)CC2)c1[N+](=O)[O-] c1(C(N(CCCOCCN(C(C(C)=C2CCCC2)=O)C)C)=O)c(C)cncc1C Cc1cc(C(=O)N(C2CCCN(C(c3coc(C)c3)=O)C2)CCF)c(C)cn1 N1(C(C(C)n2cccc2)=O)CCCC(O)(CCNC(=O)C=Cc2ccnn2C)C1 N1(C(CSCCOC)=O)CCc2cc(C(=O)NC(c3ccsc3)C)ccc2C1 CC1(C)CC2(CC(C(=O)NCCCCCNC(=O)CC(O)C(C)(C)C)C2)C1 c1(C(=O)Nc2c(C(N3CC(C#N)OCC3)=O)nccc2)c(O)cccc1[N+](=O)[O-] C(=O)(C(CC(C)C)NC(=O)CC1(C)CCN1C(=O)CCCC1CC1C)NC C1(CNC(C=CCOC)=O)CCN(C(C2CC3COCC3C2)=O)CC1C1CC1 CCC(CCCC(=O)N1CCC(OC)C12CCC2)NC(=O)C(SC)SC CC(C)CCCCNC(c1ccc(NC(C)=O)nc1)c1nnnn1CCCF C1(CNC(CCCOC(C)=O)=O)CC(NC(C2CC(F)(F)C2)=O)C1(C)C c1(C(=O)NCCCNC(=O)CCC2CCOC2)csc(Br)n1 C(=O)(C(C)(C)C1CC1)NCC(C)N(C(=O)C(c1cscc1Br)=O)C N1(C(CCC#C)=O)CCCC(CCNC(C2(CSC)CCC2)=O)C1 c1(C(=O)NCCN(C(=O)Cc2cccc(F)c2)C)nn2cccnc2c1Br C1(C(=O)OCC)CCC(C)N(C(c2cscc2Cl)=O)C1C C1(C(N2CCC(C(=O)NC(CC)COC)(CC)C2)=O)CC(=O)OC1(C)C C=CCC(CNC(=O)CCC(CC)OC)C(=O)N1CC(=O)NC(CC)C1 C1(C(N(C(C#C)C)C)=O)CN(C(C2Cc3nccn3C2)=O)CCN1C c1(C(=O)OC)nccc2cc(NC(N3CCC(COC(C)=O)C3)=O)ccc12 S(=O)(=O)(c1sc(O)nc1C)NCCNC(c1ccc(OCC)c(Cl)c1Cl)=O c1(C(N(C2CCN(C(=O)C=C(Cl)Cl)C2)CCC)=O)ccc(O)nc1C Cc1cccc(CC(N2CCC(NC(=O)C(C)CN(C)C)CC2C)=O)c1F C1(CCNC(c2ccc(OC)o2)=O)CN(C(=O)CC2CCCOC2)CCO1 N1(C(C(C(C)C)F)=O)CCN(C(=O)C=CCN2CCC2)C(CCO)C1 CCC(C)C(C(=O)NCc1cn[nH]c1)N(C)C(c1cnc(C)c(C)c1)=O C1(CC(=O)NC(CC)CSC)CCCN(C(c2cnc(Cl)s2)=O)CC1 C1(CNC(CC(C=C)C)=O)CN(C(c2c(C)nn(C)c2OC)=O)CC12CCC2 N1(C(C2CCC(=O)NC2)=O)CCC2(CCCN(C(=O)C=CSc3nc[nH]n3)C2)C1 C(=O)(C(C)CC(C)C)N(CCN(C(C(CCC)=CCC)=O)C1CCCCCC1)C Cc1nc2c([nH]1)CC(C(N1C3CCC1(CNC(=O)CCC(F)(F)F)CC3)=O)CC2 C1CCN(C(=O)C=CC2CCCC2)CC1.CC(CC(=O)NC1CC1)C1CCCO1.C c1(C(=O)OC)ccc(F)c(NC(C2CC3CC3N2C(=O)C(C)(C)OC)=O)c1 N1(C(c2n[nH]c(C)c2O)=O)CC(C)(C(N2CCC(CN(C)C)C2)=O)CC1(C)C C1(NC(=O)Cc2ccc(Cl)cn2)CN(C(c2cnnc(O)c2)=O)CC1C1CC1 c1(CCC(=O)NC2(C)CC(NC(=O)CCCCc3cnn[nH]3)C2)ccnc(Cl)c1 c1(C(=O)N)cn2cc(C)nc2s1.N1(C(C2(CC#C)CC2)=O)CCC(C)C(C)C1 C(=O)(C(C)(O)COC)N1CC(NC(C(C2CCCC2)OCC)=O)(CO)C1 c1(C(N2CC3(C2)CN(C(C2CC(F)C2)=O)C3)=O)cc2cc(Cl)c(Cl)cc2[nH]1 C(C)(C)(CN=c1[nH]cnc(=N)[nH]1)NC(C1N2CC(C)N(CC2)C1)=O c1(-c2cn(CC(C)NC(C(CC(=O)OC)C)=O)nn2)ccc(C#N)cc1F c1(CN2C(C(=O)Nc3ccc(Br)cc3CO)COCC2)n[nH]c2ccc(F)cc12 c1(OC)ccn2ncc(C(N3CCC4(NC(=O)C=CC(C)C)CC4C3)=O)c2c1 c1(C(=O)NC(CC#CC)C(=O)NCC(O)C2CC2)cc(C#N)ccc1C N1(C(=O)Cc2cnc(O)nc2O)CCC2C(CCN2C(c2cnncc2O)=O)C1 c1(C(=O)NC2CCN(C(C3CCCC3)=O)CC(O)C2)ccc2c(c1)CCCO2 C1(C(N(C2CCN(C(C(=O)N(C)C)=O)C2)C)=O)CC2CCC(C1)S2 CC1CCCn2c(C(=O)NOCC3(c4cccc(Br)c4)CCCC3)cnc21 C(=O)(CC1=NNC(=O)C1)NC1(C)CCCN(C(CCn2ncc(C)c2)=O)C1 Cc1cccc(F)c1C(N1CC2CC2(C(=O)NCCn2cnnc2C)C1)=O C1(NC(c2cncnc2C2CC2)=O)CC2CCCC12.c1(C(=O)N)cc(Cl)ccn1 N1(C(=O)C=C2CC2)CC(C2CCCCN(C(=O)C(O)CC3CCCCC3)C2)C1 NS(=O)(=O)c1coc(C=O)c1.C1CN(C(=O)C=CCN2CCCC2)CCC1F.N C=C(CN=C(NCC(C)C)NC1CCSC1)c1ccccc1 n1(CC(C)C)cc(CNC(=O)NCC2(C(F)F)CCCC2)cn1 C1(C(C)C)CN(C(=O)C(C)P(C)(C)=O)CCN1C(c1csc2nnsc12)=O C(CCN=C(NCc1c(OC)cccc1F)NC1COC(C)C1)OC CC1(CNC(C2(C)CCC(=O)N2)=O)CCN(C(=O)CNC=O)CC1 C1(C(N(CC(C2CCCC2)O)C)=O)CCC2CCC1N2C(=O)C#CC(C)(C)C C(=O)(CCCC(N)=O)N(CC(C)CNC(=O)CCc1ccc(F)nc1)C c1(CNC(=O)CCOCCCO)cc(Br)c(O)cc1F N1(C(C2CCC(=O)N2)=O)CCC2CN(C(=O)Cc3cc(F)cc(Cl)c3)CC12 C1(O)(CN(C(C(C)OCCC(C)C)=O)C)CCN(C(C2OCCO2)=O)CC1 Cc1nc(C(N2CCC(C)C2C)=O)cc(O)n1.N1(CC=O)CCS(=O)(=O)CC1 Cc1n[nH]c(C)c1S(=O)(=O)NCCc1csc(-c2ccncc2)n1 Cc1cccc(OCCCN2CCCCC2Cc2ccccc2)c1 N=c1ncc(C(=O)NC2CCN(CC)CC2)c[nH]1.C1(C(=O)N)CCOC1C1CC1 c1(C(N(CCCCCNC(c2c(C)n[nH]c2)=O)C(C)C)=O)cc2c(s1)CCC2 c1(CC=O)ccc(-c2nnco2)cc1.C(C)(C(=O)N)OCCOC.C1CCC1 CC(C)C(C(=O)N(CCCCN(C(=O)CCn1cccc1)C)C)C(C)C N1(C(CCN(C)C(C2CC3(CCC3O)C2)=O)=O)CCc2nccnc2C1 C=CCCCCCCC(=O)N1CC(COC)(NC(=O)CC2CCC(C)O2)C1 c1(CC)cc([N+](=O)[O-])ccc1NC(CNC(=O)CC1CC1)C1CCC1.C c1(CCC(=O)N(C2CN(C(C3(C#N)CCCO3)=O)CC2F)C)ccc(Cl)cc1 CCC(C)(C)C(O)C(=O)NCc1ccsc1C(=O)NC1CC1C1CCCCC1 Cc1ccc(N2CCN(CC(=O)Nc3ncc(Br)n3C)CC2)cc1 C1(CNC(c2cc(C(C)(C)C)[nH]c2)=O)CCC(C(N2CCOC(O)C2)=O)CC1 C(=O)(CS(=O)(=O)c1ccccc1Cl)NC1C(C)CN(C(C2C3(CC3)C23CC3)=O)C1 Cc1cc(N)ccc1C(N1CCC(NC(c2ccccc2OC(F)(F)F)=O)C1)=O CCC(C(=O)N(C)CCN(C(=O)C(CCSC)SC)C(C)C)C(C)C c1(C(C)C)nn(C)c(Cl)c1C(=O)NC(C)C(CO)NC(=O)CCc1nccs1 Cc1cc(C(N2CCCC2(C)CNC(C2(F)CC2)=O)=O)ccc1-n1cncn1 c1(C(=O)NC2C(NC(CN=S(C)(C)=O)=O)CCOC2)ccc(C#N)cc1O C12(CNC(C(CC#C)NC(=O)CC3CCSC3)=O)CCCC1CCO2 c1(C(=O)NC2CC3CCC(C2)N3S(=O)(=O)C2CC2)cncc2nc(O)[nH]c12 C12(NC(c3cc(OC)n[nH]3)=O)CC3CCC(C1C2)N3C(c1c(C)cncc1C)=O C1(C(N2CCC3CCN(C(c4sccc4Cl)=O)C3C2)=O)CCc2nc(O)[nH]c2C1 c1(OC)cc2nn[nH]c2cc1C(=O)N.C1(C)(CC=O)CC(F)(F)C1.C(C)CC N1(C(=O)OC(C)(C)C)CCCC2C(CCCN2C(C2CC3CSCC(C2)C3)=O)C1 Cc1cc(CC(N2CCC(C)C(NC(C3CC(F)(CO)C3)=O)C2)=O)ccc1Cl Cc1c(S(=O)(=O)N2CCC3(CC2)CC3C(=O)NC2CCN(C)C(C)C2)ncn1C Cc1nc(O)ccc1C(=O)NC(C(=O)NCCc1noc(=O)n1C)C1CC1 C(=O)(CC(C(F)(F)F)NC(=O)C(CO)OC)N1CC2C(C(=O)OC)C2C1 c1(CC)c[nH]nc1C(=O)NC1CC(CNC(c2n[nH]c(C)n2)=O)C1 N1(C(c2cc(C)no2)=O)CC(NC(=O)COC(C)(C)C)C(C)C1 N1(CCNC(C=CCNC(C(=Cc2ccco2)C)=O)=O)CCCOCC1 Cc1ccc(F)c(N)c1C(=O)NC1CC(C)CN(C(=O)COC2CC2)C1 C=CC(C)(CCOC)C(=O)NCC(C)CNC(c1c(C)ccn1C)=O N1(C(C(CC)=CCCC)=O)CCCCC1c1cn(CCOCC)nn1 Cc1cc(N2CCC(=CCNC(C3CCC(=O)N3C)=O)CC2)ncn1 c1(C(=O)NCCCOCCNC(C(CC)=CC)=O)cncc(F)c1Cl C=CCCC(C(=O)N1CCC(C(C)(C)C)C1)NC(=O)COC(C)(C)C C(=O)(C1COc2ccc(Cl)cc21)N(CC(C)NC(=O)CCOC)CC N1(C(C2CCC(C)S2)=O)CCN(C(=O)COc2ccsn2)C2(CCC2)C1 c1(N(C(CC=C)=O)C(c2cnc(N3CCCC3)s2)=O)ccc(S(C)(=O)=O)c(Br)c1 C=C=CCCC(=O)N1CC(C(=O)NC(C)(C)CC2CCOC2)C(CC)C1 N1(C(C2C(C)C2)=O)CCN(C(=O)CCCCN(C)C)C2CCCC2(C)C1 N1(C(C(C)(C)c2ncco2)=O)CCC2(NC(=O)Cc3ccccc3NC)CC2C1 O=C1NCC2(CCN(S(=O)(=O)Cc3cc(Cl)cc(Cl)c3)C2)O1 C#Cc1cccc(C(N2CC(CN(C(=O)C(O)C(C)(C)C)C)C3(CC3)C2)=O)c1C N1(C(C(c2ccncc2)C)=O)CC(C)OC2(CCN(C(C3CC4CC4C3)=O)C2)C1 S(=O)(=O)(c1ccc(C#N)cc1)NC1CN(C(CCc2c(C)cccn2)=O)CC1O N1(C(c2c(COC)cco2)=O)CCCCC1C(=O)NCC(C)(C)C1CCC1 N1(C(Cn2c(C)cc(=O)cc2)=O)CCCC(C2(NC(=O)CO)CC2)C1.C1CCC1 C1(CNC(=O)CC2C=CCC2)CC2CCC(C1)N2C(=O)CN1CCC(F)CC1 C1(C(=O)NC2C(NC(c3cncc(SC)c3)=O)CCCC2)Cc2nnc(C)n2C1 CC1(C)CC(CNC(C2CSCCN2C(=O)CCc2ccsc2)=O)CO1 c1(C(=O)NCC23CC(CC2CO)C3)cc2c(nn1)CCCO2 c1(C(=O)OCC)c[nH]nc1C1CCN(C(C)C(=O)N(c2ccccc2)C)C1 CON1CCC(NC(C2CC23CCN(C(C2CC(C)=NO2)=O)C3)=O)CC1 c1(C(c2nnnn2CCC2CC2)NCC2C(CO)C2)cccc(Br)c1 C(c1cncn1C)=CC(=O)NC1(c2ccccc2)CN(C(C=C(CC)CC)=O)C1 c1(C(N(C(C)C2CC2)C)=O)cncc(Cl)c1.C(C=O)(C1CCC1)OCC.N N1(S(C)(=O)=O)CCOC(CCC(=O)OCCSc2nccn2CC(F)F)C1 C(=O)(C#CC1CCCOC1)NCCC1CCCN(C(c2c(C)nn(C)c2)=O)CC1 c1(OC)ncc(Br)c(C)c1.C1(C(=O)N)CSCCN1C(c1ccn(C(F)F)n1)=O Cc1ccc(S(=O)(=O)CC2CC(O)CN2CC(=O)NCC(c2ccccc2)=O)cc1 c1(C=O)cccn(C2CC2)c1=O.Cc1ccc(C(=O)NC2CC(O)(C)C2)s1.N N1(C(C(C)(C)NC(C2CCCC(O)C2)=O)=O)CC2C3CCC(O3)C2C1 c1(C(C)C(N2CCC(COC)(NC(c3cnn(C)n3)=O)C2)=O)ccc(C#N)cc1 C1(C(=O)NCCC2NC(=O)NC2=O)(CC)CCCN1C(=O)C.C(C)=O.O C1(CC(=O)NCCCC)COCC(C)(C)O1.C(C(C)(C)C)N(CC=O)C.C CC1(C=CC(=O)NC2(C)CCC2)COC1.C1(C=O)CC(C(F)(F)F)CO1 c1(OCC)ccc(C(=O)NC(C2CCN(C(=O)C(C)(Cl)Cl)C2)C)cc1Cl N1(C(CSCC)=O)CCN(C(c2cc3ncsc3[nH]2)=O)C(CC#N)C1 n1(CC(N2CCCC(NC(CC(CCC)O)=O)(CC)C2)=O)cnc2c1CCCC2 C(=O)(C1=CCCN(C(c2cccn(C)c2=O)=O)C1)N1CCC(N(C)CC)C1 O=C1CCN2NC(NS(=O)(=O)CC3(F)CCCC3)=NC2=N1 Cc1ccc2c(c1)C(=O)N(C(C)C(N1CCOCC1CCC(F)(F)F)=O)C2=O C1(CCC)CC1C(=O)N(C1(CC(=O)N(CC(C)OC)C)CC1)C c1(CC)cc(C(=O)NCC2CC(OC)CN2C(c2ccsn2)=O)oc1CC C(CCCC(C)(C)C(=O)NNC(=O)C(C)(F)F)NC(c1c(OC)cc(F)cc1)=O N1(C(c2n(C)cnc2)=O)CCOCC1CCNC(c1coc(C(F)F)n1)=O S1(=O)(=O)c2ccc(cc2)C2(CC2)N1.c1(-c2n(C=C)ccn2)cccc([N+](=O)[O-])c1 Cc1cc(O)nnc1C(=O)NCCNC(=O)C(CO)NC(=O)C(C)C C1(CC(=O)NC(CC)CC(=O)OC)CC2(C1)CN(C(c1oc(C)nc1C)=O)C2 C(=O)(C(C)S(C)(=O)=O)N(C1CCN(C(c2cnc(C)nc2C)=O)CC1)CC C1(C)(C(=O)NCCC2(OC)CN(C(C3CCC3(F)F)=O)C2)CCN(C)CC1 C(=O)(C#CC1CCCC1)N1CCCC(NC(c2n[nH]c(CC)c2Cl)=O)C1C c1(C(N2C3C(NC(CCCC)=O)C(C3)C2)=O)ccc2c(c1)COC(=O)N2 c1(C(=O)NC2C(C)(C)C(C(=O)NC3CCC(F)(F)CC3)C2)ccc2cncn2c1 [SH](=O)(=O)c1cccnc1.C(C(COC)CC(=O)NCCNC(=O)C)OC.N CC(F)CC(=O)N1CCC(C(=O)NC2(CO)CC=CC2)O1 C#CC1(C(N2CC(=O)NC(C)C2)=O)CCN(C(=O)C(C)C(C)C)CC1 CC1(C)COC(CC(=O)NCCC(F)(F)Cl)C1.C12CCCC1C(=O)NC2 C(=O)(C1CSc2ccccc21)N1CC2(OCCN(C(C(C(=O)OC)OC)=O)C2)C1 c1(C(N2CC(NC(c3cc(C)c(O)nc3)=O)C3C2C3)=O)cccc2c1COCC2 CC1CCCN1C(c1cnccc1)=O.C(=O)(C=CC)N.C(C)(C)C.N(C)C C1(CC)CCC(C(N2CCCC2CNC(=O)C(F)=C(C)C)=O)O1 c1(N(C)Cc2c(OC)nsc2)cc[nH]c(=NCCC2CC3CCC2O3)n1 C1(C(C(=O)NCCO)NC(C2CC(CC)C2)=O)CCCCC1.C1(C)CCC1 Cc1cc(F)cc(C)c1C(N1CCCC(NC(c2cccc(C(N)=O)n2)=O)C1)=O C1(CC)C(C(=O)NC(CN(C)C)C(C)(C)C)CCN1C(=O)CCC1CC1 c1(CCNC(=O)NC(CC(=O)OC)C)cc2ccccc2o1 CCCC(CC1CCCC1)C(=O)N1CC(CNC(=O)CC2CC2C)(OC)C1 Cc1cnc(C(=O)N)c(F)c1.N1(CC)CCN(C(C2(S(C)(=O)=O)CC2)=O)CC1 N1(C(c2c(C(C)C)c[nH]n2)=O)C2CCC1CN(C(c1cn(CC(N)=O)nn1)=O)C2 C(=O)(C(C#N)C(C)(C)C)NC1C(C)CN(C(c2csc3nnsc23)=O)C1 C(CC(C)C(=O)NCC1CCCC1C(=O)NCc1nncn1C)=CC C1(CNC(Cc2c(C)noc2C)=O)CC2(CCN(C(C3CCC3)=O)C2)CO1 C1(N2CCN(C(COC)=O)CC2)CCCCC1OC1CCC(F)CC1 c1(C(N2CC(CCC)C2)=O)cc(C(F)(F)F)sn1.C1(C)(CC=O)CC1(Cl)Cl Cc1cc(C=O)cc(O)n1.c1(CC(=O)N(CCC)C2CC2)csc(C2CC2)n1 c1(NC)cncc(C(=O)NCCc2n[nH]cc2C(=O)N(CC(C)C#N)C)c1 C1(NC(C2(OC)CCCC2)=O)CCCCC1N(C)C(c1cc(C#N)c[nH]1)=O c1(OC)ccc2c(N3CCC(Nc4nc(C)ncc4Br)C(F)C3)ncnc2c1 C(CC(C(=O)NC1CC(C(C)O)C1)NC(=O)Cn1[nH]cnc1=N)OC C1(N(C(CC(=C=C)C)=O)C)CN(C(=O)CC2CC3(CC3)C2)CC1(C)C C=CCCC(F)(F)C(=O)NCC(CCNC(=O)Cc1ccsc1)OC C12(CNC(C(C3CCOCC3)OC)=O)CCC1CN(C(=O)CCc1nncs1)C2 N1(C(c2ccc(N(C(C)=O)CC)nc2)C(=O)N)CCOC(C)(C(F)(F)F)CC1 N1(C(CSCC=C)=O)CCCC(NC(=O)C(F)(F)c2nccs2)C(F)C1 C1(C(=O)OC)CCN(C(c2cc(C#N)c[nH]2)=O)CC1.C12(C=O)CC(C1)C2.N c1(CCC)nc2cc(C(=O)NC(C)CNC(=O)C(CC)(CC)CC)cc(C)c2[nH]1 CS(C)(=O)=Nc1nc(C(=O)NCCc2cn(C)nn2)cs1.c1ccc(Cl)cc1.S c1(NC(C(C2CCCCC2)NC(CCC)=O)C)nc(CC(C)C)ccc1C#N N1(C(CCOc2cccc(C)c2)=O)CCOCC(CNC(=O)Cc2ccon2)C1 C12(CC)CN(C(=O)Cc3cn[nH]c3)C(C)(C1)C2.C(=O)CCN(C)CCO.N C(=O)(C(C)CCC(C)(C)C)NC1C(C(F)(F)F)CCN(C(COCCC)=O)C1 Cc1nc(C)n(O)c1C(=O)NC1CCN(C(C2CC(C(C)C)=NO2)=O)C(C)C1 C(=O)(C(C)(O)C(C)(C)C)N1CCC(O)(CC)CC1.C1(CC=O)CC2CC2C1.N c1(N(C(=O)CSCC)CC)cn(C)nn1.C1(=O)CN1.CCN(C)C CC(c1ccccc1F)=CC(=O)NCC12CCCC1N(C(=O)CS)CC2.C(C)C N1(c2cc(C(C)C)ncn2)CCC2(NC(=O)CC3CCCCC3)CCCC12 O=C(C1=CCC(NC(c2ccccc2F)=O)C1)NC1CC(CF)C1 c1(OCC(=O)NC2(CF)CCN(C(c3cnc(Cl)s3)=O)C2)cc(F)cc(Cl)c1 N1(C(C(c2ccc(Cl)cc2)N(C)C)=O)CCCCC(O)C1 c12cc(C#N)ccc1OCC(=O)N2.c1(C(C)=O)[nH]c(O)nc1C.C1(C=O)CC1 C1(CC)CCC(C(=O)NC2(CF)CN(C(c3cn(C(C)C)cc3C)=O)C2)CC1 N1(C(C(CCC)OC)=O)CCCC(COC)(NC(c2cc(C)nn2CC)=O)C1 C1(C(N2CCCC(C3(C)COC(=O)N3)C2)C(=O)NCCOC)CC12CCOC2 N1(C(C(CC)(C)C)=O)CCN(C(C2CSCCS2)=O)C(C(C)C)C1 c1(NC(=O)NC(C2CCCC(C)C2)C)cnn(S(C)(=O)=O)c1 CCCC(CC)CC(=O)N1C2CCC1CC(CNC(=O)CCCC(=O)NCC)C2 Cc1ccc(C=CC(=O)NC(C)CCO)c(C)c1.N1(CCC(=O)N)CCOC1=O Cc1cccc(C(C)C(=O)N(C)CCN(C)C(c2cnc(C(C)O)s2)=O)c1 C(=O)(C(O)CC(C)(C)C)N1CCCC(NC(C2(CC)CC2)=O)C1 c1(CC(=O)NCC(C)NC(c2c(CC)oc(C)c2)=O)csc2nccn12 C1(NC(c2cnn(CC)c2Cl)=O)CN(C(=O)C(C)N(C)C)CCC1(C)C C1(C(=O)N)CCC(C(N)=O)CC1.Cc1sncc1C(=O)NC1CC(F)(C)C1 C1CC2(CC2)CN1C(=O)CN1CCCCS1(=O)=O.C1(CC=C)(C(=O)N)CC1 n1(CC(=O)NCC(CCNC(=O)C=Cc2cnc[nH]2)O)ncc(O)nc1=O Cc1ccc(F)c(C(=O)NC2CCOCC2C(=O)N(C)CC2CCCC2)n1 N1(C(C2CCC(=C)CC2)=O)CC2CCC1CC2NC(C1(C)CCN(C)C1)=O Cc1onc(-c2ccsc2)c1C(=O)NC.C1(C=O)CCC(C)O1.C1(CC)CC1 c1(NC)ncccc1C(=O)NCC1C(C)CCN1C(=O)CNc1nccs1 c1(C(=O)Nc2ccc(OC)c(N3CCOC3=O)c2)ccc2cccc(F)c2n1 C(=O)(C(F)C(C)CNC(C1CCN(C(c2ccccn2)=O)C1)=O)OCC.C n1(CC(=O)NNC(=O)C2CCCS2)c(=O)oc2cc(Br)ccc12 C1(CC(N2CCC(C)(CC)C2)=O)CCN(C(=O)CC2(C)CCOC2)C1(C)C n1(CC)ncc2c(N3CCCCC3CCNC(=O)C=CC(C)(C)SC)ncnc12 C(=O)(C(O)CCCNC(C1CS(=O)(=O)C1)=O)NC1(CCC)CCC1 C1(NC(C2CC(C)(O)C2)=O)CCN(C(C2CCN(C3CCSC3)CC2)=O)CC1 N1(C(COC(C)C)=O)CC(CNC(c2cc(-n3cnnc3)ccn2)=O)CCC1C c1(OC)ccc(C(=O)C(=O)N2CC(NC(c3ccnc(O)c3)=O)C2)cc1OC c1(C(CNC(N2CC(C)SC2)=O)(F)F)ccc(F)cc1F C=C(CNC(C1CC1(C)C(F)F)=O)CCNC(c1ccc(C(C)C)o1)=O C1(C)CN(C(=O)CSC(F)F)C(C)(C)C1.CC(C)(C)C(C(=O)N)c1cc[nH]n1 Cc1cc(Cl)ncc1S(=O)(=O)N1CCN(C(c2ccc(Br)cc2O)=O)C(CO)C1 C1(N(C(C(=O)N)=O)C)CCCCN(C(C2CC3(C2)CC(O)C3)=O)C1.C(C)OC c1(C(=O)NC2C3CCN(C(c4ccc(C)nc4N)=O)C32)ccn2nccc2c1 CS(=O)(=O)C1(C(=O)NC2CCCCC2)CC1.C1(C=O)CN(CC(F)(F)F)C1 C1(CC(N2CC(CC(=O)Nc3cccnc3OC(F)F)C2)=O)CCCCC1(F)F c1(C(=O)NC(C(=O)NCC)C2CC2)ccncc1.C1(C=O)CCSC1.C c1(C(=O)NC(CNC(CCCCC#C)=O)C2CCC2)c(Cl)cccc1[N+](=O)[O-] Cc1ccnc(C(=O)NC(C)(CNC(=O)COC2(C)CCOCC2)CO)c1 Cc1cc(C(=O)NC2CC(C)C2)ncc1C(N)=O.c1(C=O)ccc(C#N)o1.N C12(CNC(=O)CCC(F)(F)F)CCC(CN(C(=O)CCCn3ccnc3)C1)C2 c1(C(N)=O)coc(C(=O)NC2CCC2C(=O)NC2CCCOC2)c1 C1(C(NOCCC(C)C)=O)CC2C=CC1N(C(c1ccon1)=O)C2 C1(CC#C)(C(=O)NC2CCN(C(=O)CCNc3ccccc3)C2C)CC=CCC1 N(C1CCCc2c1cnn2C1CCCC1)C(N1CCC(CCC(=O)OCC)CC1)=O N1(C(C(CSC)C)=O)CCN(C(c2ncc(Cl)cc2F)=O)CC1c1nccn1C C1(OC)CCCN(C(=O)CCN(CCCO)C(C2(CC(C)=O)CC2)=O)C1C O=C(CCC(=O)Nc1nccs1)NCC(C1CC1)NC(C1CCCCC1)=O N1(C(CN2C(C)CCC2)=O)CCN(CCCNC(c2cnc(N(C)C)s2)=O)CC1 C(=O)(C(C)CCCC(C)=O)N(CC(=O)N(CC(COCC)O)C)C1CCC1 c1(C(=O)NCCCNC(c2ccns2)=O)cnc2c(c1)COC2 CCCCC(O)CC(=O)NC1(CF)CCN(C(=O)Cn2cc(Br)c(=N)[nH]2)C1 C1(NC(C(C)CC2CCC2)=O)(CF)CCN(C(=O)CC2CCC(=O)N2)C1 Cc1ccc(C(N2CCC(O)(CCNC(=O)C(C)(C)CO)CC2)=O)nc1C N1(C(CCSC)=O)CCCC(CN(C)C(C2CCCN(C(=O)C(C)C)C2)=O)C1 C1(CC)CN(C(c2cccnn2)=O)CC1C(=O)N(CCCC(F)(F)F)C CC1COCCCN1C(=O)CC(C)NC(=O)C=Cc1cn(C)nn1 CCCC(C)CC(=O)NCC(CCC)NC(=O)CNC(=O)OC C1(C=O)CCCN(S(N)(=O)=O)C1.C(C)(C)(C=O)NC(=O)OC.CC(C)C c1(C(N2C(CNC(C(CC=C)C)=O)CC2)=O)c(C)ccc2c1CCCN2 C1(C(=O)NC2CCN(C(C)=O)CC2)CCN(C(=O)Cc2csc(C)n2)CC1O C1(NC(=O)Cc2ccon2)CCC(CNC(C2(F)CCC2)=O)C1 C1(CNC(c2cncc(C)c2)=O)CN(C)CCN1C(=O)Cc1cnccc1C N=c1[nH]c2c(s1)CC(NC(=O)Nc1ccc3nc(O)oc3c1)CC2 CC1CCN(C(=O)Nc2ccc(C(N)=O)cc2)CC1.C12CCCN1C(=O)CN2 c1(NC(C2(CO)CC(C)C2)=O)ccnc2c1cnn2C N1(C(c2n(C)ncc2Cl)=O)CCC2CCN(C(c3cccc(N)c3F)=O)CC12 c1(C(N2CCC(O)(C(C)CNC(=O)CCC3CCCC3)C2)=O)nnc(O)nc1O c1(C(CN(C(=O)NC2CC(O)(C(F)(F)F)C2)CC)OC)ccccc1Br N1(C(c2c(CC)nn[nH]2)=O)CCC(C(=O)NCCN2CC=CC2)CC1C C1(NC(c2ccn(CC)n2)=O)CC(NC(c2cccc(C)c2C)=O)C12CCC2 c1(NC(CCC)=O)ccc(C2(C)CC2(F)F)cc1 C1(CC(C(=O)NCCOCC)N2CCC(C(C)(C)O)C2)CCCC(C)(C)C1 N1(C(C2CN(C(C3CCCN3)=O)CCC2O)=O)CCc2ccc(Br)cc2C1 CCC(C)C(O)CC(=O)NC(CNC(=O)C(F)(F)c1ccccn1)(CC)CC N1(C(C2OCCN(C(C3CCCC(C#N)C3)=O)CC2)=O)CC(O)CC12CCOC2 c1(OC)ccc(S(=O)(=O)NC2CN(C(=O)C3=COCCC3)C2)cc1 CCC(C)C(C)C(=O)NCc1cc(C(=O)NC(c2cccnc2F)C)n[nH]1 c1(CC)c(C(=O)NCCC(C)NC(c2ncc(OC)cn2)=O)sc2ccccc12 N1(C(c2c[nH]cc(C)c2=O)=O)CCCC2(NC(=O)CSC(C)(C)C)CC2C1 O=S1(=O)CC=C(c2ccc3c(c2)CCN(Cc2ccc(C(=O)O)cc2Br)C3)CC1 CC1Oc2cc(Br)ccc2C1NCc1ccc(N2CCOCC2)cc1 C1(NC(C2(F)C(C)OCC2)=O)CC2CCC(C1C)N2c1nnnn1-c1ccccc1 c1(NC(=O)NC(c2c(C(C)C)cccc2)C)ccc2c(S(N)(=O)=O)cccc2c1 C(=O)(C(F)(F)CC(C)C)N1CC(NC(c2c(NC)ccc(F)c2)=O)C(F)CC1 c1(CC)cccc2c(F)c(C(=O)NC(C)(C)C)[nH]c12.C(=O)CC.CC(C)C.N N1(C(c2cnc(C)nc2)C(=O)NC(C(=O)OC)C)CCN(C)C(C)C1 c1(CC)cccc2nc(C(=O)NC(C)(C)CC(=O)OC(C)(C)C)ccc12 c1(C(N2CCC(NC(C(CC(C)C)OC)=O)C2C)=O)cccc2oc(C)cc12 c1(OC)ccc(C=CC(=O)N(CC(C)(C)NC(=O)CP(C)(C)=O)C)cc1Cl c1(C(N2CC(NC(C(CCCOC)C)=O)(CO)C2)=O)cnn(C)c1S(N)(=O)=O N1(C(c2n[nH]cc2F)=O)CCC(O)(Cn2cc(C3CCCS(=O)(=O)C3)nn2)CC1 N1(C(C(N)=O)=O)CC(NC(c2ccsc2)=O)C2(CCC2)C1 c1(C(CNC(c2ncn(C(C)(C)C)n2)=O)NC(C=NOC)=O)ccc(O)cc1 O=C1NCc2ccc(NC(=O)CC3CN(C(=O)Cc4cc(Br)ccc4O)C3)cc21 N1(C(C(F)OC)=O)CCCC(C2(NC(c3n[nH]c4ccccc34)=O)CC2)C1 C(=O)(CCC(=O)NC1CN(C(c2cn(C(C)C)nc2C)=O)CC1O)NCC C(C(C)(C)CCNC(=O)CC(C)(C)O)NC(Cn1c(C(=O)OC)cnc1)=O CCCCCCN(C(=O)CC)CCNC(=O)CCCNC(C)=O.CCCC.C c1(CC(=O)OC)cccc(NC(C2CCN2C(=O)C=CC(C)C)=O)c1 C1(C(=O)NCCc2ccc(F)cc2)CCN(Cc2cc(Cl)ccc2Cl)C(=O)C1 N1(C(CC2CC(C)(C)OC2)=O)CCCC2CN(C(=O)CCc3cnoc3)CC12 C1(O)(CC)CCCN(C(c2cnnn2-c2ccccc2)C)C1 C1(NC(C(CC)n2ccnc2)=O)CCN(C(=O)CCN2CCCS2(=O)=O)CC1(C)C c1(NC(C2CCN(C)C2)=O)c(F)cc(Br)cc1Br.c1cc(C(F)(F)F)cc(Br)c1 c1(C(=O)NCCC(CNC(CC=CC)=O)O)ccc2c(c1)NC(=O)C2(C)C N1(C(C(CC)N(C)C)=O)CC(CNC(=O)C(C)C)CC1(C)C N1(C(C2C(NC(c3ccc(O)cc3)=O)CCC2)=O)CC2CCC1CC2 n1(CC(=O)NC2C=CC(CNC(C(C)N3CCCC3)=O)C2)cc(C#N)cn1 C(c1cccc(Br)c1)=CC(=O)NC1CCN(C(C(CCC)NC(N)=O)=O)C1 C1(COC)CN(C(C2CCCC2)=O)CCN1C(C1CCCC1(F)F)=O C12(NC(C34CC(OC)C3C4)=O)CCCC1N(C(c1scnc1C)=O)CC2 c1(C(=O)NC2C(C)CN(C(=O)C(C)(C)CN(C)C)CC2)ccc2nn[nH]c2c1 N1(C(c2cccc(I)c2)=O)CCN(C(c2ccc(C(F)(F)F)nc2)=O)C2CC12 C(N(C)N1CCN(CC(O)CN(C)C)CC1)c1nccc(OC)c1 C1(C(N(CC(C)CNC(C2CSC2)=O)C)=O)CCCCCCC1 c1(C(=O)NC(C)C(CO)NC(C2CCC=CCC2)=O)cc2nccc(Cl)c2s1 c1(CCNC(C(N2CCC(c3cccc(Cl)c3)(C)C2)=O)=O)c(F)cccc1F c1(C(=O)NC2(CNC(C3C(c4ccc(C)s4)C3)=O)CC2)cccc(Cl)c1 C#CCC(C(=O)OC)NC(=O)CC1CCN1C(C1CCNC(=O)C1)=O C1(CC)CN(C(c2coc(Br)n2)=O)CCN1C(=O)Cn1ccnn1 Cc1cc(=NCCCNC(c2ccnc(OCCO)c2)=O)[nH]cc1[N+](=O)[O-] N1(C(CC(CC)OC)=O)CCCC2(NC(c3cc(O)n(C)n3)=O)CCCC12 CCC(C)(CNC(=O)CCN(C(c1cn(C(C)C)nn1)=O)C(C)C)CO C1(NC(=O)NC)CN(C(C2CC(F)CN2C(=O)Nc2ccccn2)=O)CCO1 N1(C(c2csc(-c3cn[nH]c3)n2)=O)CC2CC(NC(C3CC(O)C3)=O)C2C1 N1(C(C(CCC)C#N)=O)CC2(CCN(C(c3cnc(C4CCOC4)s3)=O)CC2)C1 C(=O)(C(CC)CC(C)C)NCC1(O)CCN(C(CCCOCC)=O)C1 Cc1nc(C2CCCO2)sc1C(N1CC(C)(NC(=O)CC(C)F)C1)=O C(N=c1ccnc(NC(c2cc3cnccc3o2)C)[nH]1)c1c(CC)c[nH]n1 c1(C(=O)NCC2N(C(CC(C)(C)C#N)=O)CCC2)ccc2n[nH]cc2n1 c1(OC)ccc(CN(C)Cc2ccc(Br)cc2N2CCOCC2)c2ccccc12 N1(C(c2c(COC)n(C)nc2)=O)CCC(O)C(N(C)C(c2ccnn2C)=O)C1 Cn1ncc(-c2nn[nH]n2)c1CNC(=O)N.C1CC(=O)N(c2ccc(Cl)cc2)C1 c1(C(N2CC(C)(NC(=O)CCN3CCC(O)CC3)C2)=O)ccc(F)c(C2CC2)c1 CC12CN(C(c3ccc(Cl)c(C(F)(F)F)c3)=O)CC1CN(C(=O)C1CC1)C2 C1(CCC)CN(C(c2ncn(C(C)C)n2)=O)CCN1C(c1cc(O)nc(Cl)c1)=O C(CC(O)C(=O)N1CC(n2ccnn2)C1)NC(C1(OCC)CCCC1)=O C1(C(N(C(C)CCNC(=O)C(F)(F)c2cnccn2)C)=O)CC2C=CCC(C1)C2 Cc1ccncc1CC(=O)NC1CCN(C(c2cn(C)[nH]c2=N)=O)CC1 C1(CNC(Cc2c(C)non2)=O)(CNC(=O)CN(C)C)CC2CCCC2C1 C1(C(=O)NCC(=O)NCC(=O)Nc2cnc(Cl)[nH]2)(CC)CCCCO1 C12(CC(=O)N(C)Cc3cnnn3C)CCC1CN(C(C1(CO)CC1)=O)C2 CC#CCC(C(=O)NC1CCS(=O)(=O)C1)NC(C1CC=CCC1C)=O C(C)(C)(C(=O)NCC(C(C)C)NC(=O)C(F)C1CCOC1)OC C1(C(=O)NC(C=C)CO)C=CCN1C(c1cnnn1CC)=O C12(C(=O)NC(CCC)CCCNC(=O)CC(C)CN(C)C)CCC(CC1)OC2.C C1CCC(C)(C)CO1.N1(C(=O)OC(C)(C)C)CCCC1C1(O)CN(C=O)C1.N N1(C(C2=CCN(C(C3(CC)CCCC3)=O)C2)=O)CCSC2CCCC12 c1(CC=O)ccnc(Cl)c1F.C1(CNC(CN(C(=O)OC)C)=O)CCC1.C N1(C(C(CO)N(C)C)=O)CC2(CC2)CC1CNC(c1ccc(Cl)nc1O)=O C1(C2CCN(C(=O)CC3OCCCC3(C)C)C2)(NC(Cc2c(C)n[nH]c2)=O)CC1 C1(c2ccc(CC)cc2)CN(C(=O)CSCC)CCN1C(=O)C(C)C1CC1.O C1CC2(CCN(C(=O)C(F)CC3CCCC3)CC2)CO1.C1(C(=O)NC)C=CCC1 c1(OC)ccc(CC(=O)NC(C2CCN(C(c3csc(C#N)c3)=O)CC2)C)cc1 CN1CCN(C(=O)COC2CCC2)CC1CNC(c1cc(Br)nn1C)=O c1(CN(C(C(n2cc(C(C)(C)C)nn2)C)=O)C)nncn1C C1(c2ccccc2)CN(c2nnnn2C2CC3(CSC3)C2)C2(CCOCC2)C1 CC1=C(C(=O)N2CCCCC2CC)CCS1(=O)=O.c1(C(=O)N)ccc(=O)n(C)n1 S(=O)(=O)(c1ncc(Cl)s1)NCc1ccc(N(C)C)c(F)c1 CC(=O)C(C)CC(C)C(=O)NCCCNC(c1cnn(C2CC2)c1)=O c1(OC)ccc2oc(C(N3CCC(NC(=O)CC4(C)CC4)C34CCC4)=O)cc2c1 N1(C(C2ON=C(C)C2)=O)CC(CNC(=O)COC2CCC2)OC2CCCC12 c1(-c2nc(C(C)O)nn2-c2ccc(C(=O)O)cc2)cccc(N=S(C)(C)=O)c1 N1(C(CC(CC)C)=O)CCC(CNC(c2cc(Cl)cs2)=O)C(C2CC2)C1 N1(C(C(CCC)C)=O)CCOCC(NC(=O)C(F)(F)c2ccccc2)C1 C(=O)(N=c1cc(Cl)c(C#N)c[nH]1)C1CCC(C)N1c1ccnc(S(C)(=O)=O)n1 C1(CN(C)C)CN(CCC(C(=O)O)c2ccccc2)CCO1 N1(C(=O)NCC2(C(C)C)CCCO2)CCCN(C(C)(C)C)CC1 C1CCCC(C)(C)O1.N1(C(C=CC(C)(C)SC)=O)CCN(CC(=O)N)CC1.C c1(C=O)ccccc1.C12(CCO)CC(C1)C2.C(C)(C=O)N(CC)CC.C C1(CNC(c2cnc(CC)s2)=O)C(CC)CCN1C(c1scnc1Cl)=O N1(C(CCNC(C)=O)=O)CCCC(NC(c2ccc(CO)c(F)c2)=O)C1C Cc1cnc(C(=O)NC(C)C(C)NC(c2cnccc2Br)=O)c(C)c1 C1(C(N2CC3C(CNC(C(C(C)C)N(C)C)=O)C3C2)=O)CCC(C)(C)CC1 C1(NC(COCCC)=O)CCCCC12CCCN(C(c1ccc(OC)s1)=O)C2 C#CC1(NC(=O)C(C2(O)CCC2)NC(=O)CC)CC1.C(=O)C1CC1.N N1(C(c2cncc(C)c2)=O)CC(C(=O)NCC2CC2C2CCC2)CC12CCC2 C(=O)(C(CO)C(C)(C)C)NC(C)CN1CCN(C(=O)C(C)(C)Br)CC1 C1(C(N(CC=C)C)=O)CC2CCN(C(C3(N4CCOCC4)CC3)=O)CC12 c1(C(N2C(C)CN(C(c3[nH]nnc3C3CC3)=O)CC2)=O)noc2c1CCCCC2 O=C(C1=CCCOCC1)NCCC1CN(C(C2CC2c2cccs2)=O)C1 N1(C(C2(COC)CCCC2)=O)CC(C(=O)N)C(F)(F)C1.C1(CC)C=CCC1 CC1=C(C(=O)N2CCC(CCNC(C3CC(S(N)(=O)=O)C3)=O)C2)CCO1 C1(NC(CC2CC(=O)OC2)=O)CCCC12CN(C(C1(CO)COC1)=O)C2 C1(F)CCCC1.C1(C(=O)N)(NC(=O)OC)CCCC1.C1(F)(C=O)CCC1 N1(C(C2(CC)CCN(C(=O)CC(C)(C)OC)C2)=O)CCNC(=O)C1C C1(C2CCC2)(C(=O)NC2CN(C(C3(c4cccc(C)c4)CC3)=O)C2)CC1(F)F C1(C(N(CC(C)C)Cc2c(C)ocn2)=O)NCCC12CC2(F)F CCCCC(C)CCC(=O)NCC1(NC(=O)CCNC(C)=O)CCOCC1 N1(C(CCCNC(c2cccc(CC)n2)=O)=O)CC(C2CCCC2)C1 C1(NC(c2ccnnc2O)=O)(CF)CCN(C(=O)C(c2cccc(F)c2)F)C1 c1(CCNCC(c2cc(Cl)ccc2Cl)O)ccc(Br)c(C(F)(F)F)c1 C1(C(=O)NC(c2ncc(C)s2)C)C=CCN(C(C2(CCCF)CC2)=O)C1 CC1(O)CC2CC1CC2NC(=O)COCCNC(c1c[nH]c(=O)cn1)=O C12(NC(C3(C4N(C(CC5C(C)OCC5)=O)CCC4)CC3)=O)CC=CC(C1)OC2 Cc1cc(NC(=O)CCCCNC(=O)Cc2cc[nH]c2)c(C)c(C)c1 C=CCC(C(=O)N1CCN(C(=O)C2=CCCCO2)CC(O)C1)C(C)(C)C c1(NC(C(C)NC(C(C=C)(C)CC)=O)C(C)C)ncnc2c([N+](=O)[O-])cccc12 c1(C(=O)NC2C(C)CN(C(c3ccon3)=O)C2)ccc(O)c(Cl)n1 Cc1ccccc1C(C(C)C)NCC(c1ccncc1)(C)C Cc1cc(N)cnc1C(=O)NCC=CCNC(=O)CC1CCC(F)(F)C1 c1(C(=O)NC(C(C)NC(c2c(Br)c(C)n(C)n2)=O)C)ccc2cnoc2c1 C1CC(F)(F)CN1C(c1cccn(C)c1=O)=O.C(C(=O)N(CC(=O)N)C)OC C1(C)(C(=O)NCc2cc(C(=O)OCC)no2)CC2(CCC2)C1 Cc1ccc(N2CC3CN(C(C4CCC(C)O4)=O)CC3C2)c([N+](=O)[O-])c1 Cc1ncc(NC(=O)C=C2CCN(C(c3ccc(Cl)cc3F)=O)CC2)cc1F c1(C(N2CCC(N(C(C(C)OC)=O)C)C2)=O)cccc([N+](=O)[O-])c1F N1(C(=O)CCN2CCCCC2)CC2OCCN(C(c3cccnc3S)=O)C2C1 C1(CC)OCCC1C(N1CCC1CNC(C1(CCOC)CCCC1)=O)=O C#CC1(C(=O)NCCC2CCCN(C)C2)CCN(C(c2cncn2C)=O)C1 N1(C(CCNC(=O)OC)=O)CCN(C(c2cc(Cl)n[nH]2)=O)CC1CO c1(CN2CC3C(C(=O)Nc4onc(C)c4C)(C3)C2)ccc2nn(C)cc2c1 C1(NC(CCc2ncn(C)c2)=O)CN(C(=O)CC2CCC(F)(F)CC2)CC1(C)C Cc1ccc(C(=O)NCC(C)NC(c2ccsc2)=O)cc1F c1(C(N2CC(OC)(C)C2)=O)cccc(F)c1Cl.c1(C=O)cnn(C2CCC2)c1.N C(C(C)NC(c1cc(C(F)(F)F)ccn1)=O)(C(C)C)NC(c1nnc(C)s1)=O c1(CC(N2C(CNC(C(CC)O)=O)CC(O)C2)=O)c(F)cccc1Br N1(C(CSCC)=O)CCC(C(C)C(=O)N(c2ccccc2O)C(C)=O)CC1 Cc1ccncc1CNC(C1CCCN(C(=O)Cc2cccc(Cl)c2)C1)=O N1(C(c2c(C)coc2)=O)CCC(NC(C2(CF)CCC2)=O)CC1C CC(C(=O)NC1CCN(C(=O)CCCc2ccc(C(F)(F)F)cc2)C1)C(F)(F)F Fc1cc2c(c(F)c1Cl)CCCC2NCc1ccccc1C1CNC1 C1(C(=O)NC2(C(NOCC(C)(C)O)=O)CC(F)(F)C2)CC2(CCC2O)C1 Cc1ccc(OCC(=O)N(CC(C)NC(=O)Cc2nncn2C)C)c(F)c1 CC(C)CCC(C(=O)N1CCC(C)(N(C)C)CC1)NC(c1cccc(Cl)c1)=O N1(C(COCCC=C)=O)CCCC(C2CN(C(C3(S(C)(=O)=O)CCC3)=O)C2)C1 C1(C(=O)NCC#C)CCCN(C(=O)C(O)C(C)C)CC1 N1(C(C(C(=O)OC)OC)=O)CC(CNC(=O)C#CC2CC2)C2(CCOCC2)C1 c1(C(N2CCC2)=O)ccccc1C(C)(F)F.CC(C(=O)N)OC(C)(C)C.C c1(C(=O)N)cnc2sccc2c1.c1(C(=O)NCCC2CC2)c(O)cc(Cl)cc1F N1(C(CN(CC#C)C(c2cnsn2)=O)=O)CC2(CCOCC2)C1 Cc1nccc(C(=O)NC(Cc2cn[nH]c2)C(=O)N2CCCC2CN(C)C)c1C N1(CC(=O)OC)CCN(C(C2CCCN2c2ncc(OC)cc2F)=O)CC1=O CCCC(C)CC(=O)N(C)CC1(NC(c2cnc(C3CC3)[nH]2)=O)CC1 C(CC(CC)C(=O)NC(Cn1cc(-c2ncccc2C)nn1)CC(C)C)=CC CCC(CCOC)C(=O)NC(c1cccnc1)C(=O)N(C1CC2CC2C1)C O=C1NC2(CO1)CC(C(N1CCCC(NC(C3(CCO)CC3)=O)CC1)=O)C2 C=Cc1cc(C(=O)NCC2CCN(C(=O)C=CCO)C23CCC3)cc(F)c1 N1(C(C(c2cn(CC)nc2)=O)=O)CCC2CN(C(c3nn(C)cc3C)=O)CC2C1 c1(C(=O)NCCC2N(C(c3cn(CC)nc3)=O)CCCC2)ccn2nncc2c1 O=C(C1Cc2ccccc21)NCC1CC(Cn2cc(CCC3CCOC3)nn2)C1 Cc1cccn2ncc(-c3nc(C(F)F)nn3CC(F)(F)F)c12 c1(CC(=O)NCC2C(NC(C(C)N(C)C)=O)CCC2)ccc(Cl)c(Cl)c1 Cc1ccc(C=CC(=O)NCCC(O)CNC(=O)C(C)(F)c2ccon2)o1 C1(NC(c2nn(C)c(=O)cc2)=O)CCN(C(C2(C)CCCC2)=O)CC12CCC2 N1(Cc2cncc(OC)n2)CCCN(C(C)(C)C)CC1 Cc1cnc(N2CCCCC(NC(=O)C(F)CC3CC3)C2)nc1SC(C)C n1(C2CCN(C(=O)NCc3ccc(Br)cc3OC(F)F)C2)cnc2ccccc12 c1(C(=O)NC2C3CN(C(c4cc(CC)nn4C)=O)C2C3)cccc2[nH]ncc12 C1(COC)(C)CCCN1C(=O)Cc1csc(C)c1.c1(C=O)coc(Cl)n1.N C(CF)(C(F)(F)F)NC(CC1CC(NC(CCSCCCC)=O)C1)=O c1(C(=O)NC2C(NC(=O)C3=C(Cl)CCCC3)CC2)cc2c([nH]1)CCCC2=O CC1CN(C)CC(C(=O)NCC2CCN(C(=O)C(c3ccc(O)cc3)(C)C)C2)O1 C1(CNC(C2(CCNC(CNC(CCC)=O)=O)CCC2)=O)C2CCCC12 c1(N(C)CCC2CCN(C(=O)CNC(=O)C3CC3)CC2)cncc(C#N)n1 C1(NC(c2n(CC)c(O)nc2)=O)COC2CN(C(=O)CN3CCCOC3=O)CC12 N1(C(c2cscc2Cl)=O)CCN(C(=O)Cc2cn3c(n2)CCCC3)CC(CO)C1 CC1CCN(C(C2(O)CCOCC2)=O)CC1CC(=O)NC1(C)CC1 C(C)(CCC(=O)NOCCN(C)C)NC(c1c(CC)noc1C)=O N1(C(C2(C)ON=C(C)C2)=O)CCN(C(=O)C(C)=C2CC2)C(c2cccnc2)C1 C(=O)(C1=CC(C)(C)C1)N.c1(CN(C(=O)CC2CCCO2)C)cccc(F)c1 c1(C(=O)NC2CC(F)(CNC(=O)CC3CCCC3)C2)cc2c(nn1)CCOC2 N1(C(CCCC)=O)CC(O)CC1CC(=O)NCC1CC(C)(O)C1 N1(C(c2nc(C)c(C)[nH]2)=O)CCC(C2CC2)(CNC(=O)CC2CC=CCN2C)C1 c1(C(=O)NC(CC)CNC(=O)Cc2cccnc2)cc2cc(Cl)ncc2[nH]1 CN=c1cc(C(=O)NCC(C)N(C)C(c2nccc(OC)c2F)=O)cc[nH]1 C(=O)(C(C)(C)C)NCC.C1(C=O)C=CCCN1C(C1CC=C(C)CC1)=O.N N1(C(c2c(C)scn2)=O)CCC2(CCCCC2NC(C2CCCCC2O)=O)C1 C1(CC)CN(C(c2ccsn2)=O)CC1NC(c1ccc(OC(C)C)nc1)=O C(=O)(C(CCC1CC1)NC(C1CC2(CC2)C1)=O)NC(c1ccsc1)C CC1CN(C(C23CC(CC(F)F)(C2)C3)=O)CCCN1C(c1ncncc1F)=O c1(C(C)NC(C(CNC(c2scc(C)c2)=O)O)=O)nccc(O)n1 c1(C(N2C(C(N3CCN(CC(F)F)CC3)=O)CCCC2)=O)cc(Br)cc(Cl)c1F N1(C(C(C)N(C)C(C2CCN(C)C2)=O)=O)CCOC(CF)C1 N1(C(c2cc(C(=O)O)nn2C)=O)CC2(C1)CN(C(C1CC1F)=O)CC2.CC c1(C=O)coc2c1C(=O)CCC2.N1(CC(=O)NCC2CCCC2)CC2CC2C1.N c1(C(C)C)ncncc1C(N1CC(CC(C)NC(c2cc(Cl)cn2C)=O)C1)=O Cc1ccn(C(C)C(=O)NCC2CC(CNC(=O)Cc3cnoc3)C2)n1 c1(C(=O)NC2CCC(CNC(c3c[nH]cc(Cl)c3=O)=O)C2)ccc2[nH]ccc2n1 c1(C(=O)NC2CCN(C(=O)COCCCF)CC2F)ccc2ncncc2c1 C1(CCC)(NC(C2CCC3CC23)=O)CCCN(C(c2cc(CC(C)C)c[nH]2)=O)C1 C(=O)(C(C)(CCC(F)(F)F)c1ccccc1)N(C)C.C1CC1.C1(O)(C=O)CC1 CC1CN(C(c2ccc(=O)oc2)=O)CC(C)N1C(=O)CCCCCN(C)C C1(OC)(CNC(=O)C(O)CN(C)C)CCN(C(=O)CC2CCOC2=O)CC1 C1CN(C(c2ccc(-c3cccs3)o2)=O)CC(C)(C)C1.C(C)(C=O)NC(C)=O.N C1(CC)C(C(=O)NC2(CCNC(=O)CC=C(C)C)CCC2)CCN1C N1(C(C2CN(C(C)=O)C2)=O)CC(NC(c2cnc(O)c(C)c2)=O)CC12CCOC2 C(=O)(C(CO)C(F)(F)F)NC(COC(C)C)C(N1C2CCC(C2)C1CO)=O N1(C(=O)NC(C)C)CCCC(C(N2CCC2C(=O)N(CCO)C2CC2)=O)C1 N1(C(c2cccc(OC(C)C)c2Cl)=O)CCC2(CCN(C(=O)C(C)S)C2)C1 c1(C(=O)NC2(C(=O)NC(c3scc(C)n3)C)CCC2)ncc2ccccn12 C1(C(=O)OC)C2CC2CN1N1CCCC(c2ccccc2)CC1 C#CCCCCCC(=O)NC(C)CC1CCN(C(=O)C#CC2(C)COC2)CC1 c1(C(N2CCN(C(C=CC(=O)OCC)=O)C(C)CC2)=O)cc2cccc(Cl)c2o1 C1(C(=O)Nc2cnn(C)c2)(CNC(Cn2nnc(C)n2)=O)CCCCC1 O=C(O)CCC(c1ccccc1)NCCc1ccoc1 c1(C(=O)NC2C(C)N(Cc3ncc(Br)s3)CCC2)ccc2nnc(O)n2c1 C1(C(=O)N)CC1C1CCCC1.c1(CC)n[nH]cc1C(=O)NCCCN(CCC)C Cc1ccc(CC(=O)NC2CCCC(NC(c3cnn(C(F)F)c3)=O)C2)cc1 C(C(=O)NCCNc1cc(O)ncn1)(C(C)C)SCC.c1cccc(Cl)c1.C N1(C(Cc2n(C)cnc2)=O)CC(NC(=O)C(O)CC(C)(C)C)C2(CCC2)C1 c1ccc(Br)c(F)c1.c1(COC)nnc(CN(CC)C(C)C)s1.C(=O)N C=CC1OCCC1C(N1CCOC(CCNC(=O)C(C)(C)CSC)C1)=O N1(C(c2c(OC)n[nH]c2)=O)CC(CNC(=O)C(C)(C)CCSC)CCC1C C1(C(N2CC(CC(C)NC(=O)CCC(=O)N(C)C)C2)=O)CCc2[nH]nc(O)c2C1 N1(C(CC(C(C)C)NC(C2(C(C)C)CC2)=O)=O)CCC(F)(F)CC1C c1(C(=O)NC23C(CN(C(C(OC)OC)=O)C2)CCC3)ccc2cccc(F)c2n1 c1(C(C)N(C)C)cn(CC2CCCN2C(=O)Cc2n[nH]cc2Br)nn1 N1(C(COCCC=C)=O)CCN(C)CC1C.C1(CC(=O)N)CCOC(C)(C)C1 C1=C(CN=c2nc(N3Cc4ncsc4C3)c3c([nH]2)CCCCC3)CCCCC1 N1(C(=O)C2CC2)CC2C3CCC(C2C1)N(C(=O)C=Cc1ccccc1)C3 N1(C(C2CC(=C)C2)=O)CC(C)(C)OC2(C1)CN(C(C1(OC)CCOCC1)=O)C2 C=CC1CCCN(C(C(=O)Nc2ccc(Cl)cc2F)C2CC2c2ccco2)C1 n1(CCNC(=O)NCc2ccnc(Cl)c2F)cnc2ccccc12 c1(C(C)NC(N(CC(CCC)C)C)=O)ccc(N(C)C)cc1 C1(C)(CNC(COC)=O)CC(F)(F)CN1C(c1cc(-c2ccccn2)[nH]n1)=O N1(C(c2c(OC)ccs2)=O)CC2CCC1C1CN(C(c3cc(C)c(C)[nH]3)=O)CC21 C1(C(=O)NCCC(=O)N(CC(C)C)C(C)CO)CCCN1C(=O)C(C)C C1(C(N2CC(NC(CCC=C)=O)CC3(C2)CC3)=O)C2Cc3ccccc3C12 c1cccc(Cl)c1C.c1(C(=O)OC)ccc(CNC(C2(NC)CC2)=O)cc1 Cc1cc(N2CCC(NC(C3(Br)CC34CCC4)=O)CC2)nc(C)n1 C1CC2CC1N(C(=O)CC1(C)CC(F)(F)C1)C2.N1(CC)CCOC(C(=O)N)C1 N1(C(c2cc(C)on2)=O)CCN(CCCNC(=O)CCCn2cncn2)CC1 C#CCCCC(C)C(=O)NC1CCOCC1C(=O)NCC(C)(C)C(=O)NC Cc1csc2c(C(N3CCC(NC(=O)Cn4ncnn4)C(C)C3)=O)cccc12 C=CCCC(C)C(C(=O)NCCC)N1CCC(Cl)=C(Cl)C1 N1(CCOCC(C)(C)C)CCN(c2ccccc2)CC1 Cc1oc([N+](=O)[O-])cc1C(=O)NC(C)CCNC(=O)Cn1ccc(Br)n1 Cc1cc2ncc(C(N3CCN(C(C45CCC4C5)=O)CC3C(C)C)=O)cn2n1 CC1(C)CC(C(=O)NC2CC3(NC(=O)CCN4CCC4)COC2C3)CCO1 N1(CC(=O)NC2C(CNC(CC(COC)C)=O)CC2)CCCCS1(=O)=O n1(CC)ncc([N+](=O)[O-])c1C(=O)NC1CC(C)C1.c1(C=O)nccnc1O.C CC1CCN(C(c2ccc(C(C)(C)C)cn2)=O)CC1CNC(C1CCSC1)=O CC(CC(C)(C)O)NC(=O)CC1(C)CCN1C(c1coc(CO)c1)=O C(C)(C)(CC(C)NC(=O)CC=CCNC(=O)CNC(=O)O)OC N1(CC(=O)N)CCCOC1=O.C1(N(C(c2ccon2)=O)C2CC2)CCCCCC1.C C1(CC)(NC(C2(NC(=O)CC3CCCSC3)CCCC2C)=O)CC(C)(C)C1 Cc1cc(C)c(C(=O)N(CCCCN(c2ccnc(C3CCCC3)n2)C)C)o1 c1(C(=O)NC2C(NC(C(C)OCCC#C)=O)COC2)cc2nccnc2cc1F C1(CNC(C(C(CC)C)O)=O)CC2(CCC2)CN1C(C1CCC(C)(O)CC1)=O N1(C(c2c(CC)nns2)=O)CC2(C1)CN(C(=O)C(c1ccccc1Cl)C)CCO2 Cn1cc(C(=O)NCCC(O)CNC(C2(Cl)CC2(C)C)=O)c(C(F)F)n1 c1(C=O)cncc(S(N)(=O)=O)c1.Cn1ncc(Cl)c1CC(=O)NC1CCCC1.N c1(C(=O)N)cccc(F)c1F.C1(CNC(c2coc(C3CC3)n2)=O)CCCC1 c1(CC(C(=O)OCC)NCC(C=C)C)ccc2c(c1)OCO2 C1(CC)CCN(C(=O)CCn2ccnn2)C1CNC(c1ccoc1)=O N1(C(C(C)C(F)F)=O)CCC(C(=O)NCC2(O)CCCC2(C)C)CC1(C)C C1(C(N2CC3C(C)C3C2)=O)CC2(C1)CC(O)C2.C1(C=O)CCCO1.C1CC1 C(=O)(C(C(O)C(C)(C)C)c1ccccc1)N1CCN(c2nccn(C)c2=O)CC1 N1(c2c(S(=O)(=O)NCCC=CC)cc(C)cn2)CCc2ncc([N+](=O)[O-])cc2C1 C1CC(O)CN1C(=O)CCc1nc[nH]n1.c1(C(=O)OCC)cc(C=O)on1.N CC(CCc1cn[nH]c1)N=c1[nH]c(N2CCC(OC(F)F)CC2)nc2cc[nH]c12 C1(CNC(C(C)N(C(=O)CC2CSCCO2)CCC)=O)CCCOC1(C)C CN1C(=O)c2ccc(C(=O)N)cc2S1(=O)=O.C1(C=O)CC(F)C1.CC=CC CN=c1[nH]c(C(N2CCOC(CCCNC(=O)CCc3nc(C)no3)C2)=O)cs1 c1(C(=O)NCCC2CCN(C(c3c(CC)ccs3)=O)C2)c(C)nn2cccnc12 C1(C(F)(F)F)(OC)CCN(C(=O)NC(C)CC2CCCCC2)CC1 N1(C(C2C(=C)C2C(=O)OC)=O)CCC2C(NC(c3ccc[nH]3)=O)C2C1 N1(C(C(C)N(C(C(C)=CC(C)(C)C)=O)C2CC2)=O)CCC(C)C1CO c1(NC(c2cccc(C)n2)=O)ccc2c(c1)CCN(Cc1ccc(O)cc1Cl)C2 N1(CCOC)CC(C(=O)NCC(C)(C)CNC(c2nocc2Br)=O)CC1=O Cc1ccc(F)c(C(=O)NCCOCCC(=O)NCC2(C)CC2)c1 CCCCC(O)C(=O)NCCC(C)N(C(=O)C=CC(c1cnn(C)c1)=O)C C1(CC(=O)N(C)CC2N(C(CC(C)OC)=O)CCOC2)COCC(C)(C)O1 c1(CC(=O)NCC2CC(C)N(C(=O)Cc3ccc(F)cc3)C2)ccc(O)cc1Cl C#Cc1ccc(C(N2CC3C(C(=O)NC(COC)C(C)C)C3C2)=O)o1 C(C(C)C(C)C(=O)NCC1CN(C(=O)C(C)Cc2cccc(F)c2)CCO1)OC C(=O)(C(C(=O)N1CCCC1CCCNC(C1(C)CCCCC1)=O)OC)OC CC1CCCC(N(C(=O)CN(C2CCC2)C(C2C3CC4C(C3)C24)=O)C)C1 N1(C(c2cc(Br)ccc2I)=O)CCC2C(CCN2Cc2cccnc2O)C1 c1(C(=O)NC(CCC)C(N2CC(F)(F)CC2C#N)=O)c(C)nc2ccc(F)cn12 c1(C(N2CCC(F)(C(=O)OC(C)(C)C)C2)C(=O)NC(C)C)ccccc1I C1(NC(C2CC(F)(F)CS2)=O)CN(C(C2CC23CCOCC3)=O)CC12CCCC2 CC(C)(O)C(F)C(=O)NCC(O)C(=O)NC1CCC(C)(O)CC1 N1(C(CCNC(COC)=O)=O)CCN(C(=O)C2=NOC(C3(O)COC3)C2)C(C)C1 N1(C(c2c(C)cno2)=O)CC2CCC1C(NC(=O)CCC(=O)O)C2.C(C)(C)C.C C1(CCC(N2CC(CO)C(O)C2)=O)CCCCN1C(=O)CCCCn1ccnn1 c1(NCC2C(NC(C3C(=C)CC3)=O)CCCC2)ccc([N+](=O)[O-])c(C)c1 C1(C=O)CC2(C1)CC1(CC1)C2.N1(C(c2cnn(C)c2)=O)CCC(C)(C)C1.C c1(C(=O)NCCC(C)N(C(=O)C(=O)NCC(F)F)C)cc2c(=O)cc[nH]c2s1 N1(C(C2CCC(C)O2)=O)CCCC2(CCN(C(=O)CC(C)(C)C)CC2)C1 Cc1ncsc1C(=O)N(C1CCN(C(c2sccc2C(F)F)=O)C1)C.C1CC1.N N1(C(c2c(OC)csc2)=O)CC(NC(=O)CC(C)c2ccco2)CC(C)C1 C(=O)(C(C)(C)CC(=O)N1CCN(C(c2ccoc2C)=O)CC1C(F)(F)F)OC N1(C(c2c(C)csc2Cl)=O)CC(C)CN(C(=O)CN2CCCNC2=O)C(C)C1 C1(NC(=O)CO)CN(C(C2(N3CCCC3)CC2)=O)CC1c1ccc(F)cc1 CCCCC(C(=O)NCCCC1(CNC(=O)CCN2CCC2)CCCC1)N(C)C N1(C(c2cnc(C(F)F)s2)C(=O)NCC(=C)C)CCC2(CCCCO2)C1 Nc1ccnc2c(C(=O)NCC3CCCCN3C(c3cc(=O)cc[nH]3)=O)cnn12 N1(C(Cc2ncc(C)s2)=O)CCC(CNC(c2cc(C)oc2C)=O)C(C)C1 S(=O)(=O)(c1ccc(C(=O)NC2CCN(C(=O)CS)CC2F)o1)NC.C1CC1 c1(C(=O)NC(C2CN(C(=O)CC3CCCC3)CCO2)C)ccc(Cl)cc1N c1(C(N(C2CCC(NC(C34COC(C)(C3)C4)=O)CC2)C)=O)csc2nccn12 N1(Cc2cn(CCC(N3CCC(CC(C)C)C3)=O)nn2)CCNC(=O)C1 c1(CC2CN(C(=O)CN(c3ccc(Cl)s3)CC3CC3)C2)c[nH]c2ccccc12 c1(C(=O)NCC2C3CC2N(C(c2cc4ccsc4s2)=O)C3)ccnc2cc[nH]c12 c1(SCC)cnccc1C(=O)NC(C)CC(C)NC(=O)CCCCSC Cc1sc(-c2ccco2)nc1C(=O)N(C)CCNC(c1cc(C(F)F)ccn1)=O C1(OC)C(NC(=O)CCC2(NC(=O)C)CCC2)CC1(C)C.c1nc[nH]n1.S c1(C(=O)NCCc2cn(Cc3cc(C)c(Br)cc3)nn2)cc(Br)cc([N+](=O)[O-])c1 c1(CCC(=O)NC2C(NC(C(C)OCCOC)=O)C2)ccccn1 C1(NC(=O)CC2(O)CCC2)CN(C(C2CC3CCCCC23)=O)CC12CC2 C12(C=O)C=CC(CC1)C2.C1(CNC(C2COC(C)C2)=O)CCC1(F)F.N C1(C)CCCN(C(C2CC(S(C)(=O)=O)C2)=O)C1.C1(OC)CC2(C=O)CC12.N N1(C(c2cn(C)c(=O)cc2)=O)CCC2(CC1)CCN(C(C13CCC1C3)=O)C2 C(c1cccs1)=CC(=O)NCC1CC1CNC(=O)CC1CCCCO1 C(=O)(C1CCCc2scnc21)N1CC(CC=C)(NC(c2cscc2C)=O)C1 C1(C(=O)NCCC2(NC(C(c3cccc(Cl)c3)C)=O)CC2)CC2CCC1C2 CCC(CC)C(=O)NC(CNC(c1ccc(C=O)cc1)=O)C1CCC1.C(C)C Cn1nc(C(N2CCC(c3nc[nH]n3)CC2)C(=O)NC2(C)CC2)c(Br)c1Cl c1(C(=O)OCC(=O)Nc2c(CCC)cccc2)ccc(C(C)=O)c(C)c1 CCCCCCC(C)C(=O)N1CC(F)(CNC(=O)C(F)(F)c2csc(C)c2)C1 CC(CC(=O)NCCCCC1CN(C(c2ccc(N)c(N)c2)=O)C1)C(F)F C1(CC)CC12CCN(Cc1ccn(-c3ccccc3)n1)CC2 C=C=C(C)CC(=O)NC(CNC(=O)CC1(CSC)CC1)(CC)CC CC(C)CC(C)C(=O)N1CCCCC1CCNC(=O)CCNc1n[nH]c(=N)[nH]1 CC(C)CCC(C(=O)NCC1CCCCS1)NC(=O)OC(C)(C)C C#CCC(C(=O)NOCCOCC)NC(C1C=CCS1)=O c1(NC(c2ccc(N(C)C)cc2)C)cc(N2CCCC(CO)C2)ncn1 C#CCC(CC(=O)OC)NC(=O)NCCCC.C1(=O)C(C)OCCO1 CCCC(C(=O)N(CCCNC(=O)CNC)CC1CCCC1)NC(C)=O N1(C(c2c(C)[nH]cc2)=O)CCN(C(c2ccc(F)c(C)c2Cl)=O)CC(C)(F)C1 c1(C(N2CCC(N(C(C3(C#C)CCC3)=O)C)CC2)=O)ccc(Cl)cc1Br c1(OC)cc(C(=O)NC(C)(C)CN(C(=O)C(F)C2CC2)C)c2ccccc2n1 Cc1cccc(C(=O)NC(CNC(=O)Cc2coc(C)n2)C(C)C)n1 C1(NC(C2CC(C)NC(=O)C2)=O)CCC2(CC1)CN(C(=O)C(C)c1ccco1)C2 Cc1ccc(Cl)c(C(=O)NCC2CCN(C(=O)CN(C)CCO)CC2C)c1N CCCC(C(=O)N1CC(CC(C)(C)CNC(=O)Cn2ncnn2)C1)S(N)(=O)=O CCCCC(CNC(c1cncc(F)c1)=O)NC(=O)C(C)Sc1nncn1C c1cc(Br)cc2c1OCC2.c1(C(C(=O)NCCOC)N(C)C)cnn(CCO)c1 C(=O)C(C)(C)CS(C)(=O)=O.c1(OC)cc(Cl)ccc1C(N1CC2CC2C1)=O.C Cc1ccc(C(=O)NC2COCCC2)cc1S(N)(=O)=O.C(=O)(C(O)C(C)(C)C)N C(=O)(C1CCCCc2ccccc21)NCCNC(C1N(C)Cc2ccccc2C1)=O C1(C(C)(C)CNC(=O)CC2CCCC23CC3)CCN(c2ccncn2)CC1 C12(NC(C3CC4CCC3O4)=O)CCCCC1CN(C(C1(C3CC3)CC1)=O)C2 Cc1ccccc1C(C)CC(N1CCCCC1CN(C(=O)COC(C)C)C)=O c1(C(N2C(CC)CC2)=O)ccn(CC)c1C.N12CCCC1C2=O c1(C=O)cc(F)cc(Cl)c1O.C1(NC(c2ccc(OC)s2)=O)(C)CCCCC1.N N1(C(c2cc(C)cc(F)c2)=O)CCC(C2CC2)CC1.C1(C(=O)N)C(F)(F)C12CC2 C(c1ccncc1)=C(C)C(=O)NCCC1CN(C(C2(O)CCSCC2)=O)CCO1 CCC1=NOC(CC(=O)NC2CCC(F)(C)C2)C1.c1(CC=O)cc(C)sc1C.N CCC(COC)C(=O)N1CC(F)CC1CNC(=O)COC1CC(F)(F)C1 c1(C(=O)NC2C3CN(C(C4C(C)N(C)CC4)=O)CC32)cc(O)nc(O)c1 c1(C(=O)N)ccc2nn(C)cc2c1.Cc1cn(C)nc1C(=O)N(CC(C)O)CC N1(C(C2CC(C)N(C)C2)=O)CC2(CCC2)CC1CNC(c1cnns1)=O C(c1ccccc1)=C(OC)C(=O)NCC(C)(O)CNC(=O)CCC1CC1(C)C c1(-n2ccc(C)n2)ccc(C(=O)NCC(O)CNC(c2cnncc2O)=O)cc1 C1(NC(CC2(C=C)CN(C(=O)C(=O)C3CCCC3)C2)=O)CN(C)CC1(C)C N1(C(Cc2n(C)ccn2)=O)CCC(C(=O)OCCO)CC1=O N1(C(C(C=C)O)=O)CCC(NC(c2cnc(CC3CC3)s2)=O)C(F)C1 Cc1cn2c(CC(N3CC(NC(c4csc(C)c4)=O)C4CC34)=O)csc2n1 N1(C(CC(CC)C2CCC2)=O)CC2CCN(C(=O)CCc3cnc(O)[nH]3)C2C1 S(=O)(=O)(CCC(=O)NC1CC1NC(=O)COc1ccccc1C#N)N(C)C C1(CC)CCCCC1C(N1CCOC(C2CN(C(c3cc(O)ncn3)=O)C2)C1)=O C1(C=O)C2CC1N(C(=O)CC1CC1)C2.c1(C(c2cnsn2)=O)ccccc1.C c1(NC2CN(C(CCc3cccc(OC)n3)=O)C(C)C2)ncnc2c1COC2 Cc1cc(N2CCCC(C)(C)C2)nc(=NCC(F)C2CCC2)[nH]1 N1(C(CC#N)=O)CC(O)CC1C(=O)Nc1ccccc1CCO C12(CNC(CC(CNC(CCC=CC(C)C)=O)O)=O)CCC(C1)C(=O)N2 C1(NC(C(CO)NC(c2c(=N)[nH][nH]c2)=O)=O)CC12CCOCC2 Cc1cc([N+](=O)[O-])cc(C(=O)NCC23CCC2CCN3C(c2cnc[nH]2)=O)n1 O=C(N=c1[nH][nH]c2c1CCCC2)C1CN(S(=O)(=O)c2ccc([N+](=O)[O-])cc2)C1 CCS(=O)(=O)C=CC(=O)NC1(C2CCN(C(c3cnc(Cl)c(Cl)c3)=O)C2)CC1 c1(CNC(CN(C(C)=O)CC#N)=O)ncc(CN(C)C)o1 CON1CC(C(=O)NCC2CC(C(=O)N)CO2)CC1=O.C(C)C(C)n1cccn1 c1(COC)cc(C(=O)N(C)CC2CCCN2C(=O)C(C2CCC2)O)n[nH]1 C(CC(C)CCNC(=O)CO)NC(c1c(C)ncs1)=O.c1(C=O)ccccc1C C(CCCC(=O)NC1CN(C(C23CC4CC2C3C4)=O)CC12CC2)(OC)OC N(C1CCc2c(F)cc(Br)cc21)S(CC1(OCC)CCCC1)(=O)=O CC1CCCC(C(=O)NCC(C)(C)C(=O)N(CCS(N)(=O)=O)C)C1 CC1CC(C(N2CCC(OCC(N)=O)C2)C(=O)NCCC2CC2)CCO1 N1(C(Cn2ccc(C)n2)=O)CC2CC(O)C1C2NC(=O)C(C)O c1ccc(F)c(C(=O)O)c1.CC(Cn1cccn1)C(=O)NC(C1CCNC1)=O.C N1(C(C)=O)CCNCC1.C1(NC2CCCCC2)CC12CN(C(=O)CC#N)C2 N1(C(c2cc(C(C)C)no2)=O)CCN(C(=O)CC(C)c2ccncc2)C(C)C1 c1(C(=O)NCCN(C(C2(F)C(C)OCC2)=O)C)c(F)cncc1Cl C1(CC)C(NC(c2ncncc2Br)=O)CCN1C(=O)C=Cc1ccoc1 c1(OC)ccc(NC(=O)C(C2CCC2)NC(c2coc(C)n2)=O)cc1 CC1CN(C(c2cc(N)c(Cl)c(O)c2)=O)C(C)CN1C(=O)C=CC=O.CCC C1(C(=O)NC2CC(CNC(CCc3c(C)ncs3)=O)C2)CCN(C)CC1 N1(C(CC(C)OC)=O)CC(C)(C)CC1C.c1ccc(C(C)C)cc1.C(=O)C.N c1(C(=O)NCC(CNC(CC(C=C)C)=O)(C)F)ccc(OC)c(F)c1 Cc1ccc(-c2csc(NC(=O)Nc3ccc(C4(C#N)CCCC4)cc3)n2)cc1 C1(NC(c2cnc(CC)[nH]2)=O)CCCC12CN(C(C1CCCC1C)=O)C2 c1(C(N2C(C)CCC(NC(=O)C(C)(C)N(C)C)C2)=O)ccc([N+](=O)[O-])c(O)c1 C(C)(C)(C(C)(C)F)NC(C(C)CC1CCOCC1)c1nnnn1C1CCCCC1 c1(OC)ccc(C(=O)NCC)cc1[N+](=O)[O-].c1(C(=O)N)csc(C2CCCO2)n1 C12(CNC(c3ccc(Cl)cc3F)=O)CCCC1CCN2C(=O)COC(F)F C1(CNC(c2conc2C2CC2)=O)CN(C(=O)CCCc2cccs2)C2CC12 C1(C(=O)NC(C(=O)OC)C2CCCC2)CC2CCN(C(=O)C(C)SC)CC12 Cn1cnc2sc(C(=O)NC3CC4CC3N(C(C3(C#N)CC35CCC5)=O)C4)cc12 C(N=S(C)(=O)N(C)C)c1ccccc1.c1(CC(=O)OC)occ(C)c1C(=O)N Cn1ncc(CC(=O)NC(C2CCCN2C(c2nncs2)=O)(C)C)n1 Cc1csc2c(C(=O)NC3COCC3NC(=O)C(N3CCC(C)C3)=O)cccc12 C1(OCC)CC2(C1)CC2.N1(C2(C(=O)N)CC2)CCCC1.C(=O)C.CC N1(C(CC(C=C)CC)=O)CC2(CCN(C(=O)C(C)Cc3cnc[nH]3)CC2)CC1C N1(S(CC)(=O)=O)CCCC(CNC(C2CCOC2C2CCNCC2)=O)C1 N1(C(N=c2c(C)cn(C(C)C)[nH]2)=O)CC(c2ccccc2)Cc2ccccc21 Cc1ccc2c(c1)C(C(=O)NC1CCC(O)CN(C(c3cc(C)nn3C)=O)C1)C2 N1(C(C(COC)(C)OC)=O)CCS(=O)(=O)C(CCNC(c2ncoc2C)=O)C1 C(CN=C(NCC1CC1)NC1CC=CC1)N1CCCC(C)C1 c1(N(CC(CCC)C)C)nc(=NCCN2CCC(C)C2)[nH]c2c1CCCC2 c1(C(=O)NC(C(C)NC(=O)C=CC(F)(F)F)C)ccccc1-c1cncnc1 C1(O)(CNC(CCn2c(C)ncc2)=O)CC2CCC(C1)N2C(=O)CC.C(N)=O C(=O)(CCCCC(=O)OC)NCC1(C)CN(C(C=CC=CCCCCC)=O)C1 c1(C(c2c[nH]nc2-c2cccc(C#N)c2)Nc2c(C)ncs2)ccc(C#N)cc1 C(=O)(C(F)CC(C)(C)NC(c1cncc(F)c1)=O)NC(C(CCC)C)C c1(C(=O)NC(CN(C(C(c2n(CCC)ccn2)(F)F)=O)C)(C)C)c[nH]ccc1=O c1(C(N2CCC(C#CC)C2)=O)ccc2c(n1)CN(C(=O)C(Cl)Cl)CC2 CCCC(CN=C(NC1CCOCC1)NC1C(C)C1C)OC C#Cc1ccc(C(N2CCN(C(=O)C(CC=C)OC)C(C(C)C)C2)=O)cc1C C(N=c1cc(C)[nH]c(=NCC2(CO)CCCO2)[nH]1)C1(C=C)CCC1 CC1C(NC(C2CC(=O)CO2)=O)CCN1C(=O)CCc1ncc[nH]1 C1(NC(C(C=C=C)C)=O)CCC2(CC1)CC2NC(=O)Cc1cc(C)cc(C)c1 C1(N(C(c2c(C)cnc(OC)c2Cl)=O)C)Cc2ccc(C(=O)O)cc2C1 Cc1ccc(C(=O)N(C(C)CCNC(C2CCC(c3ccccc3)C2)=O)C)s1 CC(C)CC(C)OCCC(=O)NCc1noc(CC(C)(C)C)n1 N1(C(CCc2ccnc(C)n2)=O)CCC(C)C(NC(c2sc(C)cc2Cl)=O)C1 C(=O)(C1=CS(=O)CCC1)NCC1N(C(C(C)OCC#C)=O)CC(F)(F)C1 C#CC1CCCN(C(=O)NCC2(CC(C)C)CCC2)C1 C1(CNC(c2cc(CCC)nn2C)=O)CN(C(c2csc(O)n2)=O)CCCO1 Cc1ccc(-c2csc(C(=O)Nc3ccc(CO)c(C)c3)c2)c(O)c1 N1(C(c2scc(C#N)c2)=O)CCC(NC(=O)CCc2cc(F)ccc2F)C(O)C1 c1(NC)ccccc1C(=O)NCC1(F)CN(C(C2CN(C)CCO2)=O)C1 CC(F)CC(=O)NC(Cc1ccoc1)C(=O)N1CC(C(C)(C)O)C1 CC(C)(CCS(C)(=O)=O)C(=O)N1CCCCC(CNC(c2cncs2)=O)C1 C1(NC(C2CCCC23OCCO3)=O)CC12CCN(C(c1scnc1Cl)=O)CC2 N1(C(C2CCC(C)O2)=O)CCN(C)CC1CNC(C1CCS(=O)CC1)=O c1(CN2C(C(=O)Nc3ncc(Br)nn3)CC(F)C2)nccc2ccccc12 O=C(CCN(C(=O)C(O)C1CCC1)CC1CC1)NC1CCC1.C1CC1.C C(C)(CCCCNC(=O)CC(c1ccc(Cl)cc1)NC(=O)OC)NC(CC)=O C1(C(=O)NCCCNC(C(CC)N2CCCC2=O)=O)COCC2(CCC2)O1 C(CC(=O)NC1(COC)CN(C(C2(SC)CCC2)=O)C1)(OCC)O.C C(C(C(=O)NCCC(C)(C)NC(C1CC(O)C1)=O)c1ccccc1)OCC=C CC1N(C(C(=O)NCC2CCCCC2)c2ccsn2)CCCC12CCC2 CN1C(C(=O)NC2CC(NC(=O)Cc3cccnc3O)C2)CCS1(=O)=O c1(CC(=O)NCC2CN(C(=O)CC3CC4CC4C3)C2)ccc(Br)cn1 C1(C(N2CCC(C)C(F)(F)C2)=O)CC2OCCC2N(C(c2cc[nH]n2)=O)C1 CN1CCCC1(C)C(=O)NCC1(CO)CCN(C(=O)CCc2ccc(F)cc2)C1 c1(C(=O)NC2CC(F)C2)ccc(F)c(C(F)(F)F)c1.C1(C=O)CCCO1.C C12(C(N(C3CCCC3(C)O)C)=O)CC(CN(C(=O)COC(C)(C)C)C1)C2 c1(C(N2CCCC(C(=O)NCC(CCC=C)O)C2)=O)cnn2c1CCC2 CC1=NOC(C(=O)NCC=CC)C1C.C1(C=O)CCCC1c1nc(S)n[nH]1.N c1(Nc2c(-c3ccc(OCC)nc3)c[nH]n2)c(OCC)ncnc1Cl N1(C(C2CC(CN(C)C)C2)=O)CCCC2(CCC(NC(c3cnsc3)=O)C2)C1 C1(C(=O)N)CNCCS1.c1ccccc1C(F)(F)F.C1(C(=O)OCC)CCC1 C1C2CCC(C2)N1C(=O)CC(C(F)F)n1ccnc1.C12(C=O)CC(F)(C1)C2.N CCS(=O)(=O)CC(=O)N1CC(n2cc(CNC(c3c[nH]c(=O)cn3)=O)nn2)C1 N1(C(c2c(C(C)C)scn2)=O)CCC2(CC(C(F)F)=NO2)C1 C(=O)(C1CCCc2nnn(C)c21)N1CCCC(CN(C(C(=O)NCC)=O)C)C1 CC(C(=O)N1CCCC(CNC(C2(F)C(C)(C)C2(C)C)=O)CC1)P(C)(C)=O N1(C(CCCC)=O)CCC(C)CC1C(=O)N(CC(C)O)C N=c1[nH]c2ncc(C(=O)NCC#CCNC(C3CCC=CCCC3)=O)cc2s1 C1(C(N2CC(CC)C(C(=O)N(C)Cc3nc(C)ns3)C2)=O)CC(C)(C)CCO1 Cc1cc(CC(=O)NCC2CCCN2C(=O)Cn2ccnc2C)cc(Cl)c1 C1(C(=O)NC(COC)(C)C)CCC2(CC1)CC(NC(=O)CCC(C)C)C2 C1(C(N2C(CNC(C3CC3F)=O)CC(O)C2)=O)CCc2nc[nH]c2C1 C1(NC(=O)Cc2cccnc2)CCC2CN(c3ccc([N+](=O)[O-])c(O)n3)CC2C1 c1(C(N2CC3C(NC(=O)C(F)F)C3C2)=O)ccc2nc(Br)nn2c1 c1(C(=O)NC2CCC(C)N(C(=O)C(F)=CCCF)C2)cc2scc(Cl)c2[nH]1 C1(CC(=O)OC)CN(N(CCO)CCC(C)C)CC(C)O1 N1(C(=O)Nc2c(C)ccc(C)c2)CC2CCCC(C1)N2Cc1ccc(O)c(F)c1 C1(NC(C2(C)CCCOC2)=O)CCC2(CC1)CC2NC(c1ccc(F)cc1N)=O N1(C(COC(C)=O)=O)CCOCC1CN(C)C(c1ccc(N(C)C)cc1)=O C#CCC(C)(C(=O)N1CCSC(C)(C)C1)NC(=O)CC(C)=C=C C#Cc1ccc(C(N2CCN(C(=O)C(F)F)CCC2C)=O)c(F)c1 N1(CC=C)C(=O)C(CC(N2CCC3(CC3NC(=O)C3CC3)C2)=O)NC1=S c1(C(=O)NCC2C(NC(c3c(C)nc(CCC)s3)=O)C2)ccc(F)cc1 N1(CC)CCCC1C(=O)N(CCCNC(C1CN(S(C)(=O)=O)C1)=O)C N1(C(=O)CCOC2CCC2)CCC2(C1)CN(C(C13CCOCC1C3)=O)C2 C1(NC(c2cncn(C)c2=O)=O)CN(C(C2COCOC2)=O)CCC12CCC2 C1CCC(N(C(=O)C=Cc2nnn(C)n2)C)CC1.C(C(=O)N)(C1CCCC1)OC N1(C(c2cncc(SC)c2)=O)CC2CN(C(=O)C3=CCC(C)CC3)CC2C1 CCC(CC)C(F)C(=O)N1CC(C)C(F)(F)C1.C1(CC(=O)N)CS(=O)(=O)C1 N1(C(C(c2cccc(C)c2)O)=O)CCC2CN(C(=O)CN3CCCCCC3)C2C1 C1(C(N(C2CCC(NC(=O)Cn3cc(Cl)cn3)CC2)CC)=O)COCCN1C=O c1(CC)c(C)sc(OC(F)F)c1C(=O)Nc1ccc(C)c(F)c1.C1C(=O)N1 Cc1cc(C(=O)NC2(C)CCOC2)c(C)c(C)c1.c1(C=O)scnc1C1CC1 CC1(C)CC(c2ccccc2)(CNCCc2ncccn2)C1 C(C(C(=O)NOCCCC(=O)NC)NC(c1ccccc1F)=O)OCC C1(O)(CCNC(Cc2n(C)ncc2)=O)CCCN(C(C2(O)CCSC2)=O)C1 CCCC(CNC(c1cc(C)ccc1F)c1nnnn1CCOC)CCO N1(CC(=O)NCC2OCC(=O)NC2)Cc2ccccc2C1 N1(C(CC(C)(C)OC)=O)CCN(C(=O)COCc2cccc(Cl)c2)C(C)CC1C CC(CC(=O)NC1CCC1NC(=O)CS)c1cccnc1.c1csc(=N)[nH]1.C C(=O)(CCCCCCCCCO)NCC1OCCCN(C(C(CC)(C)C)=O)C1 C(=O)(CC(F)(F)CS(C)(=O)=O)N1CCCC(C)(CNC(C2CCCCS2)=O)C1 n1(CCNC(=O)CC2C(NC(=O)CSC(F)(F)F)CC2O)ccc(=O)cc1 C(=O)(C(C)C(=O)NCCC1(C(N2CC(O)CC2C)=O)CCC1)OC C=C1CCC(C(=O)NC2C3CC2N(C(=O)C(C2CCCC2)OCC)C3)CC1 c1(-n2ncc(C(=O)N)c2)ccccc1Cl.C(C(=O)N(CCC)C)(C1CC1)OCC c1(COC)cc(C(=O)NC(c2ccccc2)CC)no1.c1(C(=O)N)ccnn1C c1(C(N(C2CCN(C(C(C)c3ccco3)=O)CC2)C)=O)cc(Br)cnc1N CC1=NNC(=O)C1CC(N1CCCCC1CC(=O)NCC(C)(C)CN(C)C)=O c1(C(=O)NCC2CCN(C(c3ccc(C)cc3C)=O)C2)c(C)cc(C)cc1C Cc1ccc2c(c1)CC(C(=O)NCC1CCCCN1c1ccc(C#N)c(C)n1)S2 N1(CCN(C(=O)CCC2CCC2)C)CCC(O)CC1.C(=O)(C=O)N.CC(F)F N1(C(C(C)N(C(c2ncncc2OC)=O)CC)=O)CCC(F)(F)CC1C C1(C(=O)NCC(C)NC(c2c[nH]nc2C2CCC2)=O)CCCN1C c1(-c2nc(CC3COC(C)(C)O3)on2)ccc(O)c(O)c1 Cc1nc(C(=O)NCC2(NC(=O)Cc3nnc(C)s3)CC2)c2ccnc-2[nH]1 c1(CC(C(=O)N)O)cccc(Cl)c1.C1(CC(=O)NCCC2CC2)C=CCCC1 c1(C(=O)NC2CN(C(=O)C=CCBr)CC2O)ccc(I)c([N+](=O)[O-])c1 C(=O)(CCC1=CCCCC1)N1CC(OC)C(NC(c2c[nH]nc2C(C)(C)C)=O)C1 C1(C(=O)NCc2nn(C)c(=O)o2)CCC(C)(C)N(C(C2CCCO2)=O)C1 c1(CCC)nnc(S)n1CC(N1CCCC1(C)CNC(C1CCOC1(C)C)=O)=O c1(COC)nc(N2CCC(NC(c3cncc(OC)n3)=O)C(C)C2)cc(O)n1 c1(OC)cnc(C(F)(F)F)cc1C(=O)NC1CC1.c1(C=O)cnn2c1CCC2 C1(NC(c2c(C)c[nH]c2)=O)(CNC(C2(F)CCCC2)=O)CCCCC1 c1(CC)c(C(N2CCCC2C(C)NC(=O)CC(=O)N(C)C)=O)sc2ccccc12 c1(C(=O)N)cc2c(cn1)OCCO2.c1(CC)nn(C)cc1C(=O)N(C(C)CC)C N1(Cc2n(C)nnc2)CCC(C(N2CC(c3cccnc3)C2)=O)CC1 N1(C(C2C=CC(=O)N=N2)=O)CC(C(=O)Nc2cncc(Br)c2Cl)CC(F)C1 c1(OC)ccc(C=CC(=O)N)nc1.C1CCN(C(c2cnc[nH]2)=O)C(C2CC2)C1 c1(C(N2CC3CN(C(C4C(C)(CC)C4)=O)CC3C2)=O)cnc2ccccc2n1 Cc1cc(NC(C2CCN(C(c3ccnn3C(C)C)=O)C2)C)n2ncnc2n1 N1(C(C2(NC(C3C(C)(C(F)F)C3)=O)CCCC2)=O)CC2C(C1)C2(F)F C(=O)(C(CC)CCOC)NC(CC#C)C(=O)NCCC1CCCCC1 C12(NC(c3c(C)nc(CC)s3)=O)CCCN(C(=O)CCOC(C)C)C1C2 N1(C(c2c(C)coc2)=O)CC(CNC(C23CCC(CC2)CC3)=O)OC2CCCC12 c1(N2CCC(CCC)(CO)C2)nc(=NCc2nccc(O)n2)[nH]c2cccnc12 c1(C(=O)NCC(C2CCCC2)NC(CC2(C=C)CC2)=O)noc(C)c1Br CCCC(C(O)C(=O)N1CCC(CC(C)(C)C)C1)NC(c1cc(Cl)no1)=O C(=O)(C(C(C)(C)C)OC)NC(COCC)C(=O)NCC1CCCOCC1 C(=O)(CCC(=O)NC1(C)CCN(C(C2CCCN(CC(F)F)C2)=O)C1)NCCC C1(C(N2C(C)(C(=O)NC)CC2)=O)CC2(CC2)CN1C(=O)Cc1ccccc1C C1CC2CCC(C1)N2C(C1(C(F)F)CCCC1)=O.CC12CCOC(C=O)(C1)C2.N CC1(C(=O)NCC2CCCCN2C(c2occc2F)=O)CCCOC1 C1(C(=O)OC)CCC(C)(C)N(C(=O)C(=O)N(C2CCCOC2)C)C1 Cc1cc(C(=O)NCC2CCCN(C(=O)CCc3csc(=N)[nH]3)CC2)nnc1C N1(C2(C(=O)NC(C)CCN(C)C(C3(C)CC3C)=O)CC2)CCCCC1=O C1(C(N2CC3OCC(CNC(CSCC)=O)C3C2)=O)Cc2ccccc2CO1 N(C1CCC(NC(c2cc3c[nH]nc3s2)=O)c2ccccc21)C(C=CC=CC)=O CC(C)C(C(C)NC=O)NC(=O)CCCCN(C)C.S(C(F)(F)F)CC=O Cn1c(C(N2CCCC2(C)CNC(=O)C(c2csc(=N)[nH]2)=O)=O)cnc1O c1(C(CC(=O)N(CC)CC)C)c(C)noc1C.C1(N(CC=O)C)CCCC1O.N C(=O)(CC(CC)C(C)(C)C)N1CC(O)(CNC(C(CC)CC2CCCCC2)=O)C1 Cn1cc(C(c2nnnn2C)NCC(c2ccc(Cl)cc2)C2CC2)c(C#N)n1 c1(CNC(C2(C)CCCN(CC(C)C(F)(F)F)C2)=O)ccc(N=NC(N)=O)cc1 c1(OCCCCC)cc(C)ccc1C(N(C[Si](C)(C)C)Cc1cccs1)=O c1(OC)ccncc1CNC(=NCc1ccccc1)NC1CCOC(C2CC2)C1 C(C(C(=O)NCC1(C#N)CC1)NC(=O)COCC1CCCO1)OC c1(C(=O)NC2CCCN(C(C(c3cncnc3)C)=O)C2)nn(C)c2c1COCC2 c1(CN(C(CC)C)Cc2sc(Cl)cc2Cl)ccc(S(N)(=O)=O)cc1 N1(C(CSC)=O)CC(NC(=O)COC2CC2)C(c2ccc(F)cc2)C1 Cc1ccc(CNCC(C)(C)CC(F)(F)F)c(O)c1Br C(C(CNC(=O)CCN)CO)NC(C)=O.c1(CC)cc(CCCCC)no1 c1(C(N2CCC(N3CC=C(C)CC3)CC2)=O)ccc(=O)n(C)n1 O=C(C1=CCCOCC1)NCC1CN(C(c2ccc(-c3cccnc3)cc2)=O)C1 c1(C(=O)NC(C2OCCN(C(CCCCC=C)=O)C2)C)ccc(F)c2ccsc12 CC(C)C(CO)N(C)Cc1cn(C(C)C(=O)N2CCCC2)nn1 Cn1c(CCOC2CC2)nnc1-c1nc(C2CCCO2)ns1 C1(C)(C=O)CC2(C1)CC(F)(F)C2.CC1=C(C=O)CCO1.C(C)(C)CC(C)C.N C(C)(C)(CC(=O)NCC1CCOC1)N(C(CNC(C(CC)C)=O)=O)C c1(-c2n(CCCOC)nc(-c3ccc(C(F)F)cc3)n2)cccc2c1CCCC2 N1(C(C(C)(C)C#N)=O)Cc2ccnn2CC(NC(=O)CC2CC3C=CC2CC3)C1 N1(C(CCc2ccc(C#N)cc2)=O)CC2CCC(C1)N2C(C1CCOCC1)=O C(=O)(CC(C)(C)CC(=O)NCCCNC(c1csc(C)c1)=O)OCC.O c1(C(=O)NC)cc2ccc(F)cc2s1.C1(C=O)CC1C1CCC1.C12CC(C1)C2 Cn1cc(Br)cc1C(=O)NCCC1CCCCN1C(C1CC12CCC2)=O c1(SC)ccc(CC(=O)NC2CC(C)(NC(C3CC4C=CC3C4)=O)C2)cc1 c1(NC(C(N2CC(CC)N(CC(C)O)CC2)=O)=O)ccc(OC)c(Br)c1OC c1(C(N2C3CN(C(C(C)(C)c4ccsc4)=O)C(C3)C2)=O)cc(S(N)(=O)=O)co1 C1(NC(c2c(C)occ2)=O)CCCC(CN(C(=O)Cc2nnc(O)s2)C)C1 c1(C(N2C(CNC(C)=O)CN(C)CC2)=O)ccc2c(c1)C(=O)C(=O)N2 c1(C(N(C(C)C(=O)NCC(O)C2(Cl)CC2)CCC)=O)cc[nH]n1 C(C(C(=O)NC1CC(n2cccn2)C1)C(C)C)NC(C1C(OCC)CC1)=O CN(C(=NC1CCC1)NC1CC(C)N(C2CC2)C1)C(c1ccc(Cl)c(F)c1)CCC c1(C(=O)N)cc(F)c(F)cc1Br.C(=O)(CC1(O)CC1)N(C)CCOCC N1(C(C2C(CC)OCC2)=O)CCCC(C2CCCN(c3ncc(C)c(O)n3)C2)C1 Cc1cn2c(n1)CC(C(N1CCC3(CCC3)C(CNC(=O)C(C)O)C1)=O)CC2 c1(C2(C(=O)NCCCCCNC(C(COC)C)=O)CC2)cccc(Cl)n1 n1(CC(=O)N(C2(CC(=O)NCC(C)(C)C3CC3)CC2)C)cccc1 CC(C)(CC(F)(F)F)C(=O)NCC1CCCCN1C(=O)CCP(C)(C)=O C1(NC(Cc2c(C)n(C)nc2)=O)Cc2ccccc2N(C(=O)CCC(C)(C)F)C1 N1(C(c2nc(C)oc2)=O)CCC(CCC(=O)Nc2cnn(C)c2C(N)=O)CC1 C=CCC(C(=O)N(C)CP(C)(C)=O)NC(c1ccccc1COC)=O c1(CCCC(=O)NCCCN(C(=O)CC2CC=CCN2C)CC)ccc(F)cc1 c1(C(N(CC)CC2CCN(C(=O)OC(C)(C)C)CC2)=O)cnc(Cl)cc1I c1(COC)nc(C(=O)N(C2CCNCC2)C2CC2)c2n1CCCC2 c1(OC)cccc(C(=O)NCC2CCCCC2NC(c2cn(C)nc2O)=O)c1F CCCCS(=O)(=O)NCC(=O)NCCCN(C(=O)CCCC1CCCC1)C C1(NC(C(CC)CC(C)C)=O)COC2(CCN(C(c3ncn(C)n3)=O)CC2)C1 c1(C(=O)NCC2(C(C)NC(C=C(CCC)C)=O)CC2)ccc(NC)cn1 c1(C(=O)NCC2C(C)CCN2C(=O)C(C)(C)F)cc2c(=O)[nH]ccn2n1 c1(NCc2cnc(C)s2)cccc(C(=O)NC=O)c1.c1ccc(F)nc1 N1(C(c2cnc(OC)c(Cl)c2)=O)CCN(C(=O)CCC2CC(OC)C2)CC(O)C1 CC1CCC(C(=O)NCc2cnsc2)N(C(C2CCOC2C2CC2)=O)C1 c1(C(N(CC)CC2CCCCN2C(c2cccs2)=O)=O)c2c(nn1C)CCC2 C1(C(=O)Nc2c(C)ncc(C)c2)CC2OCCC2N(C(=O)C#CC2CC2)C1 N1(C(c2c(CC)[nH]cc2)=O)CCC(F)(CNC(=O)CC)C1.CC(F)(F)F.O c1(C(N2C3CN(C(Cc4cc(C)on4)=O)C(C3)CC2)=O)cc2c(s1)CCC(C)C2 CCCCC(O)C(=O)NC1CN(Cc2cc(C)ccc2F)CC1F C1(C#N)(C=O)CC12CCCC2.c1ccccc1.C1(COC)CC1C(=O)NC C(CCCCC(=O)NC1CCOCC1C)N(C(CC1C(CC)C1)=O)C CC1(OC2(C(N3CC(C)C3)=O)CSC2)CCC1.C12CC(C1)C2.C1C(=O)N1 N1(C(C(C)C)=O)CC(C)OC2(CCN(C(=O)Cc3nncn3C(C)C)CC2)C1 C1(CN(C(c2cc(C)[nH]n2)C(=O)NCCC)C)CCN(C)CC1 C=C(C)CC(C(=O)N1CCN(C(=O)CC(O)CC)CC1C(C)C)NC(C)=O CCCCC(O)C(=O)NC1COCCN(Cc2cccc(CC)c2O)C1 c1(-n2ccnn2)c(F)cc(Cl)cc1F.C1(C(N(C(C)C)C)=O)C=CC1C(=O)O N1(C(C(CSC)O)=O)CCC2C(NC(=O)CN(C)S(N)(=O)=O)C2C1 N1(C(CC(=O)NCC#C)=O)CCN(C(C2C=CCC2)=O)CC(C)(F)C1 C(=O)(CC(C)(C)CNC(C1CN(C2COC2)C1)=O)NCC1C(C)OCC1 CCCC(CC)C(=O)NC1(CCC(=O)NC2CC(CCF)C2)CCC1 O=C(C1=CCCC1)N1CCOCC1CCNC(C1CN(C2CCC2)C1)=O N1(C(c2c(C)scn2)=O)CC2CCN(C(C3CC4(C3)CC(C)(C)C4)=O)C2C1 C1(NC(COCCCC#C)=O)CCC(C)(NC(=O)CO)CC1.CC.CC#C C(=O)(CC(=O)N)OCCC(C)C.C(C)CCC.c1(C=O)cc(C(C)(C)C)n[nH]1 N1(C(C(C)CNC=O)=O)CCC(C2CC2)C1.C(C)(C)C.C(=O)CN(C)C C1(NC(C(COC(C)C)NC(c2ccc(C3CC3)o2)=O)=O)CCC(=O)NC1 CC1CC2CN(C(=O)C(C3CCCC3)NC(C3CC4C(C3)C4(F)F)=O)CC12 c1(C(=O)NC(CC)(CNC(=O)CC(C)n2cccn2)CC)sc(C#N)cc1C N1(C(c2c(C)noc2N)=O)CCC(C)(C)C(C(N2CC(C(F)(F)F)C2)=O)C1 N1(C(C(CC)N(C(=O)CC2CCOC2(C)C)C)=O)CCC(O)(C(=O)OC)CC1 c1(C(N(CC)CC)=O)cnn2c1OCC(F)C2.C1(C=O)(C(N)=O)CC1.CO NS(=O)(=O)c1n[nH]cc1C(=O)NC1COC2CCOC12.c1(CC=O)nc[nH]n1.N c1(C(=O)N)c(C(F)(F)F)cccc1O.C1(CC#C)(C(=O)NCC)CC=CCC1 CCCCCC(CC)C(=O)NC1CC(CCNC(C2(C(F)(F)F)CCO2)=O)C1 N(C1CCCc2c[nH]nc21)C(C=O)=O.C1(NC(=O)OC(C)(C)C)CC(O)C1.C N12CCN(C(C)C1)C(=O)CC1(CC1)C(=O)NC1(CC1)C2=O.CNCC Cc1cccc2sc(C(=O)N(C)CC3(NC(=O)Cc4cc[nH]n4)CC3)c(Cl)c12 c1(C(N2CCN(C(=O)C=C3CCCCC3)C(CCO)C2)=O)cc2c(nn1)CCC2 N1(C(CCC2(C)CN(C(Cn3ccc(C)c3)=O)C2)=O)CC2CCCC12 Cn1nc(C(=O)NCC2COCCN2C(=O)C2=COCC2)c2c1CCOC2 C1(C(=O)N(C2CC(F)(F)C2)C)(CC)CCCN(C(C2CC2(Cl)Cl)=O)C1 CCC(C)(CC)C(=O)NCC1(O)CC(C(=O)Nc2cc(CO)cc(F)c2)C1 CC1CCC=C1C(=O)N1CCN(C(C23CC(F)(C2)C3)=O)C(C2CC2)C1 c1(CC)ccc(F)cc1C(=O)NC1CCN(C(C2(C)CCCC2)=O)CC1O c12ccc(cc1C)o2.C1(C(=O)NCC)CCCN1C(c1sccc1OC)=O C(=O)(C(CC(C)C)N(C(c1cc(C#N)n(C)c1)C(=O)NC1CCCCC1)C)OC C1(NC(C2CCN(C(C3CC(=C4CC4)C3)=O)CCO2)=O)CCc2n[nH]cc2C1 N1(C(C(C(C)NC(=O)CCc2nc(=N)[nH][nH]2)(C)C)=O)CC2(CCC(=O)O2)C1 c1(C(C)NC(C=CCOC)=O)csc(C(C)OC(C)=O)n1 N1(C(CC2(CC=C)CCCC2)=O)CCN(C(=O)C(C)(O)C2CCC2)CC1 C(C(O)C(=O)NCCc1cnc(C)s1)NC(CC1CC(OCC)C1)=O CC(C)CC(O)C(=O)N=c1ccn(CC(=O)Nc2c(O)ncnc2O)c(O)n1 C1(c2ccc(F)cc2)CCOCC1.C1(CNC(=O)N)CCCN1Cc1ccsc1 c1(C(N2CC3CCN(S(=O)(=O)c4cccs4)C3C2)=O)coc2ccccc12 C(=O)(CC(C)CC(=O)N1CCCC(O)(CNC(=O)C(CO)OC)CC1)OC CCC(CN=c1[nH]c(=NCCCCCCN(C)C)c2cc(Cl)ccc2[nH]1)N(C)C N1(C(c2c(C)occ2)=O)CCSCC1CCNC(C12CC(C1)C2)=O N1(C(c2cc(C(=O)OC)c(Cl)cc2)=O)CCC2CCC(O)CC2C1 N#CC1CN(C(N2CC(Cc3ccncc3)C2)=O)CCN1C1CC1 C(=O)(CCCN=[N+]=[N-])NC(CCCC)CNC(=O)CCc1c(N)cnn1C N1(C(c2cccc(NC)n2)=O)CCN(C(=O)C(C2CCC2)OC)CC(CO)C1 C1(C(N(C(C)C)CCN(C)C(c2cc([N+](=O)[O-])n[nH]2)=O)=O)OCCOC12CCC2 c1(C(N2CC3C(CNC(c4c(C)ncn4C)=O)(CC3)C2)=O)cnc2[nH]cnc2c1 c1(CSC)cc(-c2nc(C(C)OC(C)(C)C)nn2CC2CCC2)ccc1Br C(=O)(C(C)(C)C(N)=O)NC(CC)CN(C)C(c1nccn1C)=O c1(C(N(C2CCN(C(CC(CC)O)=O)C2)CCO)=O)cnc(S(C)(=O)=O)s1 c1(SC)ccc(C(=O)N(C2CCC(NC(c3sc(N(C)C)nc3C)=O)C2)C)cc1 N1(C(C2(C(C)=O)CC2)=O)CCC=C(C(=O)N(C2CCC2C)C)C1 C(=O)(C1=CCCOCC1)NC(c1ccccc1)CNC(C(c1ccnn1C)C)=O Cc1cc(=NC(=O)C2COC3(C2)CN(C(c2c(Cl)cncc2Cl)=O)C3)cc[nH]1 c1(CNC(C(C)(C)SC)c2nnnn2-c2ccccc2)cccnc1S(C)(=O)=O c1(C(=O)NCC(CO)NC(=O)CC2CC2C(F)(F)F)cnc2ccnn2c1 C(=O)(CC1=NNC(=O)C1)NC.c1(C(=O)OC)ccn(CC(N2CCCC2)=O)n1.C C1(NC(C(C2CCCN(C(C3CCC=CCC3)=O)C2)(C)C)=O)CC12CC(O)C2 Cc1cc(C(N2CC3CC(C2)N3C(=O)C(C)(F)c2ccccc2)=O)nc(C)c1 C(CCN=c1[nH]c2cc(Cl)c(S(=O)(=O)NCCOCCO)cc2s1)N1C(C)CCC1 CCC(CCCC(F)(F)F)OC(C1CC2(C1)CN(C(=O)OC(C)(C)C)C2)=O N1(C(CCCOC)=O)CC2(NC(c3ccn(Cc4ccccc4)n3)=O)CCC1C2 CN1CCCCC(CNC(C2CCCN(C(C3C4CC(=O)CC34)=O)CC2)=O)C1 C1(OC)CC2C1CCN2C(=O)C(CNC(=O)C(C)(O)C(C)C)CC1CC1 c1(CC(=O)NCC(CNC(c2cc(C)no2)=O)(C)C)ccc2ncsc2c1 C(c1cc(Cl)ccc1Br)=CC(=O)NCCC1(CC(=O)OC)CC1(F)F O=C(CCC(=O)N1CCCC1)NCCN(C(=O)CCc1ncc[nH]1)C1CCCC1 C(=O)(C1CCCn2cnnc21)N1C(COC)CN(C(=O)C2=CCCCC2)CC1 CCCCCC(C)CC(=O)NC1(C)CN(C(c2c(C)nc(C)n2O)=O)C1 Nc1ccc(C(N2CC3(CCN3C(=O)CSCCc3ccccc3)C2)=O)c(F)c1 c1(C(N2CCC(O)(C(C)NC(Cc3nnc(C)s3)=O)C2)=O)ccc(S(C)=O)cc1 CC1CCC2(CCN(C(c3csc(CNC(c4ccnn4CCF)=O)c3)=O)C2)C1 C#CCC(C)C(=O)N1CCC1CNC(c1cc(CC)no1)=O C1(CNC(c2cc(CC(C)C)on2)=O)CCC(C)CN1C(c1n[nH]cc1Cl)=O c1(C(N2C(CC(=O)Nc3nc(Br)cnc3Cl)CCC2)=O)cc(O)c(O)c(O)c1 C(CC(CO)NC(=O)C(CN(C)C)NC(=O)CC(C)F)OC c1(NC(C2SCCN(CC)C2)=O)cc(F)ccc1C(=O)Nc1c[nH]nc1C#N c1(N2CC(NC(c3c(C)ccs3)=O)C(O)C2)nc(C(C)C)ncc1Br c1(C(=O)NC(COC)C)cc(-c2ccc3c(c2)CCC3)cc2[nH]ncc12 C1(C(N2C(C)C(NC(c3cncnc3)=O)CCC2)=O)CCS(=O)(=O)C12CCC2 n1(CC=C)ncc2c(O)nc(N3CCCC(NC(=O)C=C4CC4)C3C)nc12 C1(C(N2CC(n3ccnn3)C2)=O)(NC(C(C)OCCOC)=O)CCCC1C C(=O)(C(F)(F)C(F)(F)C(F)(F)F)NC1CN(C(Cn2ccc(C)n2)=O)C2C1C2 N1(C(CNC(CCC)=O)=O)CC(NC(c2onc3c2CCCC3)=O)C2CCCC12 C(=O)(C(C)(F)C(=O)N1CC(NC(c2ccc(O)nn2)=O)C1)OCC N1(C(Cc2cnn(CCC)c2Cl)=O)C2CCC1CC(CN)C2 c1(C(N2C(CCNC(C3N(CC)CCCC3)=O)CCCC2)=O)ccc2c(c1)CC2 C=CC(CCC)CC(=O)NC(CNC(c1ccc(-c2ccco2)s1)=O)CCCC C(C(=O)NC1CC(N(C(=O)CCc2ccon2)C)C1)(C1CC1)SC C1(CC)CN(C(C2CCS2(=O)=O)=O)CCO1.C(=O)(C=CC(=O)N(C)C)N C1(CC(=O)NC(CC)CNC(C2(CC(C)C)CCC2)=O)CCC(O)C1 N1(C(C(C2CC2)OCC)=O)CCN(C)CC1C(=O)NC1C(=O)OCC1C O=C(N=S(=O)(c1cccc(Br)c1)C1CCOCC1)C1(c2cc(F)ccc2F)CC1 N1(CC(=C)Br)CC2(CC(NC(=O)CCC(C)(C)C)CO2)C1 N#Cc1csc(NC(C2CC(F)CN2Cc2ccc(N3CCCC3)cc2)=O)n1 O=C1CCN(CC(=O)NC2CC3CN(C(=O)CCC4CCCCC4)CC23)C(=O)N1 C1(CCC(N2CC(C(=O)NC)C2)=O)CCN(C(c2scnc2CN)=O)C1 N1(C(CCC(C)NC(=O)COC2(C)CCCC2)=O)CCCC(N=[N+]=[N-])C1 N1(C(CC(C)C)=O)CC2(C1)OC1(CO)CC2(NC(=O)C2=COCCO2)C1 N1(C(C(CCC)OC)=O)CC2(CCCC2NC(c2cc(Cl)cc(Cl)n2)=O)C1 N1(C(C(CCOC)OC)=O)CCCC(C)(NC(=O)CC2(N(C)C)CC2)C1 C1(CC(=O)N(CCCNC(=O)C)CCC)C(=O)NN=C1C.C1CCCO1.O c1(OC)cc(C)c(C=O)c(C)c1.C(=O)C(O)CC1CC1.C1(CC)CCCC1.N N1(C(CC(C=C)(C)C)=O)CCCC2(NC(C3CSCCS3)=O)CCCC12 C#CCC(C)(C(=O)NC(C=C)C(F)(F)F)NC(c1cccc(C#N)c1)=O c1(C(=O)Nc2cc(C)nc(-c3ccccc3)n2)cc(Br)cc([N+](=O)[O-])c1C c1(C(N2CC3CN(C(c4ncccn4)=O)CC3C2)=O)ccc(F)cc1[N+](=O)[O-] c1(C(=O)NC2CC(O)CN(C(C3(F)CCCCC3)=O)C2)cc2c(Cl)nccc2o1 c1(C(N2CCC(CCCCNC(C(C)OCC)=O)CC2)=O)cnc2ncccn12 C1(CN(C(=O)C=C(Cl)Cl)C)CC(F)CN1C(c1coc(-c2ccccc2Cl)n1)=O C(=O)(C(C(=O)N1CCC(CF)(NC(c2ccc(C)o2)=O)C1)OC)OCC CC1(C)CN(C(=O)C(C2(O)CN(C(c3cnc4n3CCC4)=O)C2)F)CCS1 C1(NC(c2ccc(C3(C)CC3)cc2)=O)CC2CC(C1)N(Cc1cn(C)nc1Cl)C2 N1(C(C2CC(NC(c3c(C)ccnn3)=O)C(O)C2)=O)CCC2CN(C)CCC12 c1(-c2cc(C(=O)NCc3ccc(C)cc3C)ncc2)cc(F)cc(F)c1CO N1(CC2N(C(C(C(C(C)C)C)N)=O)CCC2)Cc2ccccc2C1=O Cc1nc(CCCC(=O)NC(CNC(=O)C(C)(O)C2CCOCC2)CO)cs1 CC1(C)OCC2CC12NC(c1cc2sccc2s1)c1nnnn1C1(C)CC1 O=C(CCCCN1CCOCC1)NC1C=CC(CNC(c2cnn[nH]2)=O)C1 C#CC1(C(=O)NC2CCCSCC2)CN(C(=O)CC23CCCC2C3)C1 c1(C(=O)OCC)cncc(C(N2CCN(C(C3CC34CCOC4)=O)CC2)=O)c1 N1(C(CC(=C)C)=O)C2CCC1CC(NC(=O)C(C)Oc1ccc(C)cc1)C2 C(=O)(C(Cn1cccn1)NC(c1cncs1)=O)N(CC#C)Cc1ccco1 C#Cc1cccc(C(=O)NCCc2cc(C(=O)N(C(C)CO)C)no2)c1C c1(C(=O)NCCC2CN(C(CCSC)=O)C2)cc2c(F)c(F)ccc2s1 N1(C(CC=CC=C)=O)CCCC(O)(CCNC(=O)CCC2CCOCC2)C1 Cc1nnc2n1CC(C(=O)NC(C)CC1CCN(C(C3C(C)C3C)=O)CC1)CC2 C=CCCN=C(NCC1CC(=O)N(C)C1c1cnn(C)c1)NCC(C(C)C)OC c1(C(N2C(c3cn(CCC(=O)NC)nn3)CCCC2)=O)ccc2nncn2n1 C=CC(C)(O)C(=O)N1CC(CC(C)NC(c2cnc[nH]2)=O)C1 N1(C(C2C(CCC)CN(C(C3CC3(Cl)Cl)=O)C2)=O)C2CCCC1CC2 c1(NC(C2CC(O)CN2C(c2c(Cl)cncc2Cl)=O)=O)ccc2c(c1)C(=O)NC2 C12(C(=O)N)CCCC1N(C(c1cccn3ccnc13)=O)CC2.C(=O)(C)OCC=C C1(CC)(CC)CCCN1c1nc(C=O)c(C)s1.C1(C(=O)N)CN(C)C(=O)N1 Cc1cccc(C(=O)NC2CCCCC2NC(c2ccccc2)=O)c1F.C(C)(C)S C(=O)(CCC(C)S(C)(=O)=O)N(CCCCCNC(c1cccc(C)c1Cl)=O)C O=C(CCC(CF)CF)NCC12CC(NC(=O)Cc3ccc(Cl)nc3)(C1)C2 N1(C(C2C(CCC)C2)=O)CCCC(O)C1.c1(C(=O)N)ccc(-c2csc(C)n2)s1 C1(C)(C(N2CCN(C(CC(C)CF)=O)C3(C2)CC3)=O)Cc2ccccc2NC1=O N1(C(C=Cc2cn(C)nc2)=O)CC(NC(=O)CN2CCCC2)CC12CCCC2 Cc1[nH]c(C(=O)NCC(C)(C2CC2)NC(=O)C)c(C)c1C.C1CCCCCC1.O Cc1cc(CC(=O)NCC2CCCC2NC(c2sccc2CO)=O)cs1 C(=O)(C(C)CC(F)(F)F)NC(CCCNC(c1c(C)n(C)cn1)=O)(C)C c1(CC(C)C(=O)OCC(=O)NC2CCCC2)ccc(Cl)cc1.C(=O)N(C)C.C c1(Cc2onc(C(c3ccccc3F)OC)n2)ccc2nc(O)oc2c1 C1(C)(CC)CC(C(N2CC(CNC(c3cc(C)cc(O)n3)=O)C2)=O)CCO1 N1(C(c2cnc3n2CCC3)C(=O)NCC)CC2CC1CN2C(C)=O c1(C(=O)NC(C2(CNC(COC)=O)CC2)C)ccnc(C(C)(C)C)c1 C1(C(N2CCCC2)=O)Cc2cncn2C(=O)N1.c1(C(=O)N)cn(C2CC2)nn1.C N1(C(C(c2cnccn2)C)=O)CC2CC(NC(=O)C(C3CCCCC3)OC)C2C1 c1(C(N2CC=C(CCNC(CC3(C=C)CC3)=O)CC2)=O)ccc2cncn2c1C C1(C(N(CCCCNC(c2c(Br)cnn2C)=O)C)=O)CCc2nn[nH]c2C1 c1(C(=O)NC(C(C)NC(c2coc(CO)c2)=O)CO)c(S(C)(=O)=O)cnn1C Cc1c(C(=O)NCC(CNC(c2ccc(C(C)C)[nH]2)=O)CO)cncc1Br Cc1nc(C=CC(=O)N(C2CC(NC(C3CCOC3)=O)C2)C)[nH]c1C N1(C(c2ccn(C)n2)=O)CCOC2CN(C(=O)C=Cc3cc[nH]n3)CC12 c1(OC)c(C(N2CC(NC(=O)COC(C)C)CC(C)C2)=O)ccnc1Cl N1(C(c2cnc(CCCC)s2)=O)CC2CC1CC2NC(c1nccc(C)n1)=O c1(COC2CCCN(C(c3c(C)coc3)=O)C2)ccc([N+](=O)[O-])cc1 c1(CNC(CCOC)=O)cccc(CNC(=O)C(C)(F)CC2CCCC2)c1 n1(CC)cnc2c1NC1=NCC3(CO)S(=O)CCN(C2=N1)C3.CC Cn1c(CC(=O)NC(CNC(C2CC=CCC2C(F)(F)F)=O)CO)nnc1S S(=O)(=O)(c1ccc2c(c1)CCC2)N1CCN(C(c2cc(OC)c(Br)cc2)=O)CC1 Cn1nc(C(N2CCCC(F)(C(=O)NCCc3ccco3)C2)=O)cc1C#N Cc1cccc([N+](=O)[O-])c1C(=O)Nc1cccc(F)c1.c1(C(=O)N)ccn(C)c1 CC(N=c1ccc2nnnn2[nH]1)C1CCCCN1C(c1cc2cccn2cn1)=O C1(CC(=O)OC)CN(C(=O)NCCCN2CCN(C)CC2)CC(=O)N1 c1(NC)cncc(C(=O)NCC2(C=O)CC23CCC3)c1.C(C)CC1CC1 N1(C(c2cccc(CC)n2)=O)CCN(C(c2sc(C)cc2C)=O)C(C)C1C Cc1cc(C(N2CCN(C)C(CNC(=O)CC3CCCC3)C2)=O)cc(O)c1 CCCC(C)C(=O)NCCCC1CCCCN1C(=O)CC1CC1 C(=O)(C(C)(C)CC(F)F)N1CCCC(C)(CNC(C(c2ccc(F)cc2)C)=O)C1 N1(C(C2CC(CC)C2)=O)CCCC(CC)CC1.n1(C2(CC=O)CC2)cncn1.N C1(C(=O)NCC2CN(C(C3CNC(=O)O3)=O)CC23CC3)CC2CCCC(C1)C2 C1(NC(=O)CSC(F)F)COCCN(C(c2ccc(-c3cccnc3)cn2)=O)C1 N1(C(c2c(C)nns2)C(=O)NCCCF)CCCCC12CCN(C)C2 C1(F)(CNC(C(C=C=C)C)=O)CCCN(C(=O)Cc2ccc(O)cc2)C1 N1(CC)CC(C(N2CC(CO)(NC(C3CC(F)C3)=O)C2)=O)CCC1=O c1(CCC(=O)NCC(C2CC2)NC(CCCC(C)=O)=O)n[nH]c2c1CCCC2 CCCCC(CC(=O)N1CCC(CO)CC1)NC(c1n[nH]c(C)c1C)=O N1(C(C2(F)CCN(C(C(CC)OC)=O)C2)=O)CCCC(C#N)C1 C1(C)(NC(CCSc2ccc(C)cc2)=O)CCCN(C(=O)CN(C)CCO)C1 N1(CC=C(C(=O)OC)F)CCOC2(CCC2)C1CO c1(C(=O)NCC2C3CN(C(C(CCC)F)=O)CC32)c(C(F)(F)F)nc(C)n1O c1(CC)cc(C)c(C(=O)NCC(C)(CO)NC(=O)CCO)o1.C1CCCO1 Cc1cc(C)c(C(=O)NC2CN(C(c3ccn(C)c3)=O)CC2O)s1 C12(CNC(C3CN4CCN3CC4)=O)CCC1CN(C(=O)Cc1cnsc1)C2 N1(C(CC(C)n2cccn2)=O)CCN(C(c2cnc(N)c(Cl)c2)=O)CC1C1CC1 C(C)(C(C)(C)C(=O)N(C)OC1CCCC1)NC(CCCCC(C)=O)=O Cc1cc(NC(C2CC(C(C)(C)O)C2)=O)n(CC2CCC2)n1 c1(C(N2CC(NC(C)=O)C(C)C2)=O)cc2cc(F)ccc2[nH]1 c1(CC)ccccc1OC.c12c(cnn1-c1ccccc1C)NC2c1nnnn1C N(C1CN(C(=O)CNC=O)CCc2ccccc21)C(c1nn(C(F)F)cc1Cl)=O c1(CC)cc(C(=O)OC)nn1C.C12CC(C1)C(F)C(=O)O2 c1(C(C)O)cn(CC(=O)NCC2CC(NC(C3(C)CCCO3)=O)C2)nn1 C1(NC(c2c(CC)cno2)=O)CN(C(c2ccccc2COC)=O)CC12CCC2 C1(CCN(C(C(C)N(CC)CC)=O)C)CCN(C(=O)Cc2ccsc2C)CC1 N1(C(CSCCOC)=O)CC(C)C(NC(c2cc(Cl)cc(Cl)n2)=O)C(C)C1 C(CC(O)C(=O)NCC(O)CNC(C1(C(N)=O)CCC1)=O)SC CCC(CC)CC(=O)N1CCC(C)(CNC(c2cc(SC)c(C)o2)=O)CC1 C1(NC(CN(C(C(C)C)=O)C)=O)CC=CCC1C(=O)NCC[Si](C)(C)C C1(C(C)NC(CC=CC=C)=O)CCCN1C(=O)C(COC)N(C)C O=S(=O)(C1Cc2ccccc2C1)NCCc1cccnc1Cl N1(C(c2ccc(OCC)nc2)=O)CC(C(F)(F)F)OC(C)C1.C(=O)(CCF)N C1(C(N2C(Cn3cc(CNC(=O)CO)nn3)CCC2)=O)CCCN2CCCCC12 C(C(C(=O)N1CC(N(C)C)C(C)C1)C(C)C)NC(CSC(C)C)=O c1(C2N(Cc3nc(OC)c(C)s3)CCC2)cn(C)c2ccccc12 N1(C(C(COC)C)=O)CCCC2CN(C(c3cnn(-c4ccccc4)c3)=O)CC12 c1(CC(=O)N)ccc2c[nH]nc2c1.Cc1cccc(C(=O)NC2CC(F)(C)C2)c1 N1(C(CC(=O)NCC#C)=O)CCC(CC=C)(Nc2ccncn2)C1.C(C)(C)O Cc1nc(O)ccc1C(=O)NCC1CCN(C(C2CC2(C)C(F)F)=O)CC1 C(CC)(C(=O)NC1(C)CN(C(=O)Cn2cc(-c3ccccc3)nn2)C1)=CCCC c1(NC(=O)C(=O)Nc2ncc(C(=O)O)[nH]2)ccc2c(c1)CN(c1ccncn1)C2 N1(CC(=O)NCC(CC)NC(=O)CCc2cnc(O)[nH]2)CSCC1=O N1(c2ccc(C)cc2)C(=S)NC(c2ccc([N+](=O)[O-])o2)C2=C1CC(C)(C)NC2=O N1(C(c2c(C)ccs2)=O)CCC2(CC1)CC(C(=O)NC1CC(C)C1)C2 CCC(C(=O)OC)C(=O)N1CC(CO)(NC(c2ncnc(OC)c2F)=O)C1 N1(C(C(COC(C)=O)C)=O)C2CCC(C(=O)NC3CC(O)C(O)C3)C1CC2 CCCCCCCCOCC(=O)NCC1CCCN1C(C1(SC)CCOCC1)=O N1(C(c2ccc(CC)o2)=O)CC(C)OC(C)(C)C1.c1(C(=O)N)cn2ccnc2s1 C1C(O)C2CCOC12.C1(CC=C)(C=O)CCCN1C(=O)CN(C(=O)C)C.N C(c1c(Cl)cccc1Cl)=CC(=O)NC1CCCCN(C(C2CCCN2N=O)=O)C1 C1(COCC)CCN(C(c2ncccc2C)C(=O)NC2CC2)CC1 c1(CC2N(C(C3C(Cl)(C(=O)OC)C3)=O)CCCC2)cccc(S(N)(=O)=O)c1 c1(C(=O)N)ccc(=O)n(C)c1.CC1OC(=O)NC1C(N1CCC(=CC)CC1)=O C(CCCC(=O)NCC1CC(F)CN1C(=O)C(C)c1cccs1)OC CC(F)(F)CCC(=O)N(CCCNC(c1c(F)cncc1Cl)=O)CCO C(=O)(C1=NN(C)C(=O)CC1)N(C(C)C)CC.c1(CC=O)nc2c([nH]1)CCCC2 Cc1cc(C)c(C=CC(N2CCC(N(C(=O)CCc3cscn3)C)C2)=O)cc1C N1(C(C2C(C)C2C)=O)CC(NC(=O)C=Cc2cnc[nH]2)CC1C C1(CC(=O)NC)CN(C(c2ccsc2C#N)=O)CCN1C(c1ncsc1C)=O N1(C(c2ccc(I)cc2O)=O)CC2CCC(C1)N(C(c1cc(O)ccc1Br)=O)C2 C(C(=O)NCCCF)(C1=NOC2COCC12)N1CC(C#N)C(F)(F)CC1 C(=O)(CC(C)(C)C(=O)NCCCNC(C1CCCC(C(N)=O)CC1)=O)OC N1(C(C2C(CNC(C3CC4(CSC4)C3)=O)CCO2)=O)CC(C2CC2(F)F)C1 C1(NC(CC2CCCC(OC)C2)=O)CC2CCC(C1C)N2C(=O)C=CSC CCCC(C(=O)OC)C(=O)NC(C)(C)C(C)NC(=O)CCCc1ccc(F)cc1 c1(NC(N2CC(c3ccnc(O)c3)C2)=O)nccc2c[nH]nc12 C1(CC)CN(C(c2nc(C)ccc2C)=O)CCC1NC(c1c(C)noc1N)=O C(=O)(CC(O)C(C)C)N1C(C(=O)NC(C(=O)NCC)CC)CC1 C(CCCC(=O)NC1CN(C(c2nc(C(C)C)oc2C)=O)CC1SC)OCC CC1(C)OCCC1CCNC(=O)NCCS(=O)(=O)CC1CC1 c1(NC(COC2CN(C(CNC(C3C(C)C3)=O)=O)C2)=O)ccc(CO)s1 C1(NC(CC=CC)=O)CC2CCC(C1)N2C(=O)CC1C(=O)ON=C1C CC(C)CC(CNC(=O)CC1CC2CCC1O2)NC(c1cc(C#N)cs1)=O c1(OC)ccc(OC)c(C(N2CCC(N(C)C(C3CC3C)=O)CC2)=O)c1 C1(CCC(N2CC(c3ccccc3)(NC(C3C(C)C3)=O)C2)=O)NC(=O)NC1=O CCC(CN(C)C)CC(=O)NC1CC(C(=O)NCC2CC3(CC3)CO2)C1 c1(C=O)ccc(N(C)C)cn1.C1(CNC(CC2CC(SC)C2)=O)CCCC1.N N1(C(CC(=C=C)C)=O)CC2CC1CCC2NC(=O)CCCCN(C)C N1(C(C2(C)CCC(C)C2)=O)C2CCCC1CC(CNC(=O)CCC1CC1(F)F)C2 C(=O)(CC(C)c1cccnc1)NC1CC(NC(C(C2CC2)OCC)=O)C1 N1(C(CCC(C)OCC)=O)CC2(CCN(C(=O)CC3=CCOCC3)C2)C1 C1CN(C(c2c(C)noc2C(F)F)=O)CCCO1.n1(CC)cnnc1C(=O)N.C C1(CC(=O)N2CCC2C=O)CC=CCC1.C1(CC(=O)OC)CCC1C=O.N C1(C(N2CC(C)C2)=O)CCc2cnc(C)n2C1.C(C=O)(C(C)C)NC(=O)OC c1(C(N2CCC(NC(C(CC)COC)=O)C(C)(C)C2)=O)cccn2cc(C)nc12 N1(C(CN(C2CC2)CC)=O)CC(C)CN(C(=O)CC2CC(O)C23CCC3)CC1C O=C1CCC(CC(N2CCCC2CNC(c2ccc(C3CCCCC3)s2)=O)=O)C1 Cc1nc(N)cnc1C(N1CCCC(N(C(=O)CN2CCCCCC2)C)CC1)=O N1(C(c2nc(C(C)NC(C3CCOC3=O)=O)oc2)=O)CC(S(C)=O)C1 C(=O)(C1=CCCSC1)NC(C(N1CCC(OCC)CC1)=O)Cn1cncn1 N1(C(CCOC(C)=O)=O)CCCC1C(C)NC(=O)CN1CCCC1 C1(CC(=O)NCCC(C)NC(c2occ(C)c2)=O)CCCC(C#N)C1 C1(C)(N(C)C)CN(C(C2C(NC(=O)CCc3cncs3)C2(C)C)=O)C1 c1(Cn2cc(C(C3CCCCC3)OC)nn2)cc(C(C)C)nn1C N(C1CCCc2ccoc21)C(CC1N(C(c2ccn(C(C)(C)C)n2)=O)CCC1)=O C1(NC(C2(CC)CCC2)=O)CCC(CCNC(=O)Cc2csc(S)n2)C1 c1(C(=O)NCC(C)CNC(=O)CC(C)O)cc2c(N(C)C)ncnc2n1C C(=O)CS(=O)(=O)C(C)C.c1(OCCOC)cc(C=O)ccn1.CC=CC c1(OC)ncc(NC(=O)C(C2CCC2)NC(c2cccs2)=O)cc1C C1(C(N2CC3(CC(NC(=O)CCc4cc[nH]n4)C3)C2)=O)CCC2C(C1)C2(F)F c1(C(N2C(C)CCCC2C)=O)c(Nc2cc(F)ncn2)sc2c1CCC2 N1(C(C(CC)Cc2ccccc2)=O)CCN(C)CC1CNC(C1CC(F)C1)=O c1(-c2cc(C(N3CCC(NC(C4CC4CF)=O)C3)=O)n[nH]2)ccccc1O Cc1cncc2nc(CC(=O)NCC3(NC(c4csc(=N)[nH]4)=O)CCCC3)cn12 C1(C)(CC)NC(=O)N(CC(=O)NCC(CC)CC)C1=O.C(=O)CC1CC1.N c1(C(N2CCCC(C(=O)Nc3cccc(O)c3Cl)C2)=O)cccc2c1CCCO2 CCC(CNC(N1CCC(OCC2CC2)CC1)=O)CCC1CCCC1 c1(C(N(CCN(C(=O)CC(C)CF)C(C)C)C)=O)cnc(O)cc1O Cc1c(F)cc(CNC2C3CN(C(c4ccc(Br)cc4C(C)C)=O)CC23)cc1Br c1(NCc2ccc(C)cc2Br)nc2ccccc2nc1N1CCSC(C)(C)CC1 CC1(C)C(CNC(=O)CC2COC(=O)C2)CCN1C(=O)Cc1nccs1 Cc1cc(C(N2CC3(CO)CC2(C(N2CCC2(C)CF)=O)C3)=O)ncc1F CCC(C(=O)NC(COC)C(=O)O)NC(N)=O C(=O)(C(C)C(O)C(C)CC)N1C(C(=O)NC(C=C)C(F)(F)F)(CC)CCC1 N1(C(C(C)n2cccn2)=O)CC2CCC(C1CO)N2C(=O)CCC(C)(C)C CCC1=C(C(=O)NCCOCCN(C(=O)C(O)Cc2ccccn2)C)CCCO1 Cc1cc(CN2CCC(O)C(C(=O)NC3CN(C)C(=O)C34CC4)C2)c(C)cc1O c1(NC(C=C(C)CNC(C2CC(F)C2)=O)=O)cccc(C)c1 CCC(C)C(C(=O)NC(C)C(=O)OC)N(C(=O)C(OC)OC)C N1(C(c2cc(CNC(C3CCN(C)C3)=O)oc2)=O)CC2(CCOCC2)C1 C1(NC(c2nccc(C)c2)=O)(C)CCC(C)(C)CC1.c1(C(=O)N)ccc(F)cn1 CC1=C(C)CC(C)(C(=O)NCC2(O)CCN(C(=O)CC)C2)CC1.C1CCCC1 N1(C(C=CC=CC)=O)CC(C(=O)N(C(C)CC(N)=O)C)C2(CCC2)C1 c1(C(C(N2CCC(=CCNC(c3occ(C)c3)=O)CC2)=O)=O)ccc(Cl)cc1O C1(C(N(C)Cc2cn(C)cn2)=O)CC2(CC2)CN1C(=O)Cc1cccnc1 C(=O)(CCCn1nnnc1C(c1cnc[nH]1)NC(c1ccccc1)C)OCC c1(C(N2CC(C(=O)NCc3cncc(O)c3)(CC)C2)=O)cc(C)c(F)cn1 N1(C(=O)CCF)CCC(C2CCN(C(c3ccc(-c4ccco4)nc3)=O)C2)C1 C1(C(N2CC(OC)(CNC(=O)CC=C(Cl)Cl)C2)=O)C2CCC(C2)C1C C1(C(=O)NC2C(CC(C)C)C2)CC1(C)C.C(=O)(CC=CC(C)(C)C)N C(=O)(C1CCOc2c(F)cccc21)N1CC(C)(OC(F)(F)F)C1 C1(CC)(CNC(=O)CC2CCCN(C(=O)Cc3cncs3)C2)CCCCC1 C(c1sc2ccccc2c1Cl)=CC(N1CC(NC(C=C(C)C)=O)C(C2CC2)C1)=O N1(C(C2CCCN(C(C3(OC)CCC(C)C3)=O)CC2)=O)CC(C)(C)OC(C)(C)C1 Nc1ccc(F)c(C(=O)NCC2(F)CCC2)c1.C1(C=O)(C(F)F)CCOCC1 C=CCCCCC(c1nnnn1C(C)(C)C)NC(C1CCCCC1)CC C1(NC(C(c2c(F)cccc2F)OC)=O)CCC2CCN(C(c3ccon3)=O)C12 CCC(C)(C)CC(=O)N1CCCC1C1(NC(c2cnc(OC)cc2C)=O)CC1 c1(C(N(C2CCCC(Nc3ccncn3)C2)C)=O)cccc(-c2cc[nH]n2)c1 C(=O)(CCCCN1CCCCC1)N1C(CN(C(c2c(CC)noc2)=O)C)CCC1 CC1OC2(CO)CC1(C(=O)NC(C)(C)CC)C2.c1(CC=O)cccc(F)c1.N N1(C(C(CCC)(C)O)=O)CCn2c(CNC(=O)C(n3cc(C)cn3)C)nnc2C1 C(CCN=c1nc(N2CCOC(C3CC3)C2)c2c([nH]1)CCCC2)c1n(C)ncc1 C=CCCCCC(=O)NC(C1CN(C(C2(CCF)CCOCC2)=O)C1)C C=CCCCCC(=O)NCC1CCN1C(c1sc(NC2CC2)nc1C)=O c1c(C(F)(F)F)cccc1F.C(c1ccccc1)=CCNC(C1CCCCN1C)=O c1(CNC(CC2N(C(C(F)=CCC)=O)CC2)=O)ccc(C)c(F)c1 C1(C=O)CCOC(=O)CC1.C(CNC(C1(CC)CC1)=O)(N(C)C)C1CC1.N NS(=O)(=O)CCCNC(=O)C(CC1CCCC1)NC(c1ccc(=N)[nH]n1)=O C(=O)(CCCCC(N)=O)NC(CCNC(Cc1c(C)n[nH]c1)=O)C Cc1cc2c(cc1Br)N(C(c1cc3ccsc3n1C)C(=O)NCC1CC1)CCC2 C(CC(C)C)(CS(C)(=O)=O)NC(N1C(c2ccc(C)o2)CS(=O)CC1)=O C1(C(N(CCN(C(c2c(C)csc2)=O)C(C)C)C)=O)COC(=O)N1C C1(C(N2C(CC(=O)NC(c3ccccc3O)C)CC2)=O)CC2CCC(C1)C2 c1(C(N2C(C(N(C)Cc3nnc(O)o3)=O)CCCC2)=O)cnn2ccccc12 c1(OC)cc(CNC(=O)CCCOc2cccc(Br)c2)c(Cl)cc1Cl N1(C(C2C(C)CCC2)=O)CCC(CNC(=O)Cn2[nH]cnc2=N)C(CO)C1 CCC(CCCC(=O)NCc1n[nH]c(C)n1)NC(=O)CCCCNC(N)=O c1(-n2cc(-c3ccc(CO)cn3)nn2)cccc2c1CCN2 C(=O)(CC(C)CC(C)(C)C)NC(CN(C(CCCN(C(C)=O)C)=O)C)(CO)CO C(CC1=CCN(CC2CC2)CC1)NC(CCCCC#C)=O c1(C(N2CC(C)(NC(COCCC#C)=O)C2)=O)cc(CC)ccn1 Cc1cc(C(=O)NC2CCCCC2NC(=O)C(c2ccc(Cl)cc2)C)cc(F)c1 C1(NC(c2cn(C(C)C)nn2)=O)CCC(NC(=O)CCC2CCCC2)CC1 CC(CCNC(=O)C(c1ccco1)NC(C12CC1CNC2=O)=O)C(F)F CCC(CC(=O)NOCCCC(=O)OC)NC(c1cnc(OC)s1)=O N1(C(c2c(OC)cccn2)=O)CCC2(CC1)CN(Cc1cc(Cl)ccc1Cl)C2 c1(CC)nn(C2CC2)cc1C(=O)NCC(C)N(C(=O)C(O)C1CC1)CC C(=O)(C(C)CC(F)F)NCC1(C(=O)NC2(C#C)CCOC2)CC12CCC2 C1(C)(CC)CC(N=c2[nH]c(=NCCOC(F)F)[nH]c3c2CC(C)CC3)C1 C1(C#N)(C(=O)NC(C2CCCN2C(=O)CCCc2cccnc2)C)CCCCC1 C1(CNC(C(CC#C)CC#C)=O)CN(C(C2CC2F)=O)CC12CCOCC2 C=CCCC(F)(F)C(=O)NCC(CC(F)(F)F)NC(C1CC(O)C1)=O CC1CCN(C(C23CC2CCN3C(c2c[nH]c(=S)cn2)=O)=O)CCO1 C=CCC(Cc1ccccc1)C(=O)N1CCN(C(c2ccsc2)=O)CC1C C1(NC(C2CC(SC)C2)=O)CC(F)(CNC(C2CC=CCC2)=O)C1 CC1(C(N2CC(O)CC2C(=O)NCC23CCCC2C3)=O)CC2CCC1O2 N1(C(C2CCN(C(C)=O)CC2)=O)CC(NC(c2scnc2C)=O)C(C)(C)C1 c1(N2CCCC(NC(c3nn(CC)c(C)c3)=O)C2)cc(C#N)ccc1[N+](=O)[O-] C1(NC(C(=O)NC(C#C)C)=O)CN(C)C2(CCOCC2)C1 C1(C(=O)NCCN2CCC(NC(C3C4COCC34)=O)CC2)COC2COCC12 c1(NC(c2nc(NC(C)C#N)sc2)=O)cnc(C(F)(F)F)cn1 c1(C(=O)NC2(CN(C)C(C3(N(C)C)CCCC3)=O)CC2)cc(N)cnc1Cl Cc1c(-c2ccccc2)o[nH]c1=NC(=O)N(c1nn(C)cc1Br)C C1(C(=O)NCC2CCCC(NC(C3(F)CC=CC3)=O)C2)CN2CCC1CC2 C(=O)(CCCCCn1cnnn1)NCCC(C)CCNC(C1(C2CCCO2)CC1)=O c1(C(=O)NC(C2CN(C(=O)Cc3cncc(F)c3)C2)C)cnn2c1OCC(O)C2 c1(OC)ccc2cc(C(=O)NCC3CC3)[nH]c2n1.C1(C=O)CCCCC1(C)C.N c1(C(N2CC(CNC(c3cc(OC)n(C)n3)=O)C3C2C3)=O)cc(Cl)ccc1C c1(N(CCNC(=O)C(C2CCC2)C2CCC2)CC)ccc(C(=O)N)cn1 C(C(C)(C(=O)N1CC(c2cc(O)no2)C1)NC(=O)CCC1CCOCC1)SC C(=O)(CC1OCCc2sccc21)NCC(CN(C(=O)Cc1cnn(C)c1)C)(C)C C1(n2c(C(c3cc(Cl)c(Cl)s3)NCCCC3(C)CC3)nnn2)CCC(F)(F)CC1 C1(SC(C)C)NCC1(C)C.c1(CC=O)cccc(C(=O)O)c1.c12cn(nn1)C2 c1(C(=O)NC2CC(NC(C3CCCN3C3CC3)=O)C(O)C2)ccc(Cl)cc1F C#CC1C(C(=O)NCC2CC(NC(C3CCCS3)=O)C2)C1(C)C N1(C(C#CC(C)(C)CNC(c2cc(O)ncc2F)=O)=O)CC2(CNC(=O)OC2)C1 C(C)(C(C(=O)N(C1CCN(OC)CC1)C)C(C)C)NC(c1nc(CCC)oc1)=O C1(NC(CC(c2ccc(OC)cc2)C)=O)CCCCCC1NC(c1ccon1)=O c1(CC)cc(C(=O)NCC2CC2CNC(=O)CCCOC)nn1C.CC N1(C(COCC#C)=O)CCC(C)(NC(=O)Cc2csc(-c3ccsc3)n2)C1 C1(C(F)F)(CNC(c2sccc2F)=O)CCN(C(=O)C#CC2CC2)C1 C(CCC(C)C)NC(Cc1cc(OC)no1)=O.c1(C=O)cc(C(F)(F)F)on1.N c1(C(=O)NCCC(C)NC(C(CC)F)=O)cnc(OC)cn1 C1(NS(C)(=O)=O)CCN(C(=O)NCC2CCCN2C(N)=O)C1 C1CCN(C(C2CCCC2)=O)CC1.CC(C(=O)NCC(F)(F)F)NC(N)=O.C N1(C(c2c(CC)nc[nH]2)=O)CC2C(NC(=O)C=Cc3ccc(C)s3)C2C1 Cc1oc([N+](=O)[O-])cc1C(=O)NC(CNC(=O)C(C)c1ncco1)CC(C)C c1(C(=O)OC)cc2cc(NC(c3cccnc3C(=O)OC)=O)ccc2[nH]1 c1(-c2n(CCCOC)nc(Cc3cccnc3)n2)ccc(C(C)CC)nc1O c1cc(O)cc(F)c1.c1(CNCC2(C(=O)NCC=O)CC2)cn[nH]c1.N c1(C(=O)NC2C(NC(c3cccnc3O)=O)CCC2)cccc2ccccc12 C1(NC(C2N(CCC)CCCC2)=O)CN(C(c2c[nH]cc(C)c2=O)=O)CCC1O C1(CC(=O)N)CN2CCN1CC2.CC1(C)CCN(C(C2C(F)(F)C23CC3)=O)C1 C=C(C)C1OCCC1C(N1CCN(CC2CC2)CC1)=O.C(=O)C#CC1(C)CC1.N C1(c2n(CCC)nnn2)(NC2(C)CC=CC2)CC2CCCC(Br)(C2)C1 n1(CC(=O)NCCC(C)C)cc([N+](=O)[O-])cn1.C1(C)(C=O)CNC(=O)C1.N CC1CN(Cc2cnc(Br)s2)CCC1NC(c1ccc(F)cc1)=O C1(C(=O)NC2C(NC(c3nc(C4CC4)cs3)=O)CC2)CC2(CCCCC2)C1 C1(O)(C(N2CC(CN(C)C)C2)=O)CCN(C(c2cc[nH]n2)=O)C1 C(=O)(CCC(=O)NN(C)C)NC1C(C)CN(C(C2(CF)CC3(CCC3)C2)=O)CC1 N1(C(=O)CN2CC=CC2)CCCC1C1CCCCN1C(=O)COc1cccnc1 C1(C(=O)NCCCCCN(C(C2C(OC)C2)=O)C)CCCCC12CCC2 C(=O)(CCC(=O)N1CCC(CCCNC(C2(CC)CCCCC2)=O)CC1)OCC C1(NC(C2CC(F)CCN2C(c2ccccc2)=O)=O)CC12CCOCC2 O=C(C#CC1CCCO1)NCC1(O)CC(NC(c2ccc(Br)c(F)c2)=O)C1 c1(C(=O)NCCC(C)NC(C2N(CC)CCCC2)=O)cc(OC)cc(Cl)c1F N1(C(CC=C)=O)CCN(C(=O)CCCOc2ccccc2Cl)CC1CF Cc1ccc(F)cc1C(=O)NC1CCN(C(c2coc3c2COC3)=O)C12CC2 C1(C(=O)OC(C)C)CCCCC1NC(=O)NCC1CC1c1cncs1 CC1CC(C(=O)NC(C)(CNC(C2CCC2)=O)C2CC2)C1 C#CCC(C)(CC)C(=O)NCCC(O)CNC(c1ccc(Br)o1)=O C1(CNC(c2cc(CNC(C(C)C#N)=O)[nH]n2)=O)CC12CCOCC2 C1(CNC(c2ncnc(C)c2C)=O)CN(C(C2C=CCS2)=O)CCC12CCC2 C1(NC(Cc2nc(C)sc2)=O)CC12CCN(C(c1ncc(Cl)cc1Br)=O)CC2 C1(O)(C(=O)NCC(CNC(c2cc(CC(C)C)[nH]n2)=O)C)CN2CCC1CC2 C(=O)(C1CCCc2scnc21)NC(C(CO)NC(c1c(CC)occ1)=O)C C(=O)(C(CO)C(F)(F)F)NC(c1cn(C)nc1)C(=O)NC1CCC(N=[N+]=[N-])CC1 C1(C)(C(C)C)CN(C(C2CC23CCC3)=O)CCO1.C1(CC(=O)N)CCC(=O)NC1 C1(CC(N2CCC(=CCNC(C3CCCN(C)C3)=O)CC2)=O)COCC(C)(C)O1 c1(OC)cc(Br)ccc1S(=O)(=O)N1CCSC1c1cc(F)ccc1F C1(CNC(c2cc(CCC)on2)=O)CC(O)CN1C(=O)C(c1ccncc1C)C N1(C2CCN(C(=O)Cn3ccc4ccccc34)CC2)CCc2c(O)cccc2C1 c1(C=O)cc(N)c(F)cn1.CC(C(=O)NCCOCC)C(C)C1CCCCC1.N N1(C(c2ccc(C#C)o2)=O)CCCCC(CNC(c2cc(CC(C)C)on2)=O)C1 S(=O)(=O)(c1ccccc1F)NCCC(N1CCN(c2ccc(Cl)nc2I)CC1)=O c1(C(CC(=O)NCCN(C2CCCC2)C(c2nc(C)oc2)=O)C)c(C)noc1C C=CC(CCC)CC(=O)NC1CC2(C1)CC(NC(c1n[nH]c3c1CCC3)=O)C2 CCC(C)(CCC(C)C)C(=O)N1C(C(=O)Nc2ccc(C(F)F)nc2)CC2CC12 Cc1ncnc(C)c1OCC(=O)NC(c1ccc(Cl)nc1)C N1(C(C)C)CCN(C(=O)C(CCN(C)C)NC(=O)C=C2CCCCC2)CC1=O C1(C(N2CCC2)=O)CCc2nc(=N)[nH]cc2C1.C1(CC#C)(C(=O)NC)CCCO1 N1(C(c2ncc(Cl)s2)=O)CCCC(C(N2CCC(c3ccc(F)cc3)C2)=O)CC1 N1(C(C2(COC)CCCO2)=O)CC(CC=O)C2(CC2)C1.c1(CC)ncc(C)o1 C1(C(N(CCC(=O)NCC(F)Br)C)=O)COCC1(C)C C(=O)(C(CO)C(C)(C)C)NC1C(NC(c2cnn(CCCC)c2C)=O)CCCC1 C12(C(=O)NC(c3ncccc3F)C)CC(CCO1)N(C(c1ccsn1)=O)C2 C1(NC(c2ccc(C(=O)NC)cc2)=O)CCN(C)C(C)C1.c1ccc(F)c(F)c1 C(=O)(C1=C(Cl)CCCC1)NC1CC(C(=O)NCc2cn(C)nn2)C1 C1(NC(C2CCN3CCOCC23)=O)CCCC12CN(C(c1cnc(Cl)cn1)=O)C2 c1(OC)ccccc1C(O)C(=O)NC1CCC(NC(c2cc(C)cs2)=O)C1 C(CN=[N+]=[N-])(C(=O)NC(C)CCN1CCCC1)NC(CNC(C(CC)C)=O)=O N1(C(CCCOC)C(=O)Nc2ccccc2)CCCCC12CCS(=O)(=O)CC2 N1(CC)CC2CN(C(C3CCN(C(=O)CC(C)C(C)C)CCO3)=O)CC2C1 C(=O)(C(F)(C)C(C)C)N1C(C)(CC(C)C)CCC1.C(=O)C(C)C1(O)CCC1.N C12(C(N3CC(O)(CC)C3)=O)OCCCC1C2(F)F.c1(C=O)sc(N(C)C)nc1Cl N1(C(c2c(C)nc(C)[nH]2)=O)CCN(C)CC1CNC(C1C(Cl)(Cl)C12CC2)=O C(=O)(C1=CCOCC1)N(C(CCNC(c1n(C(CC)CC)ncc1)=O)C)C Cc1oc(C)c(NC(=O)C(=O)NCc2cn(-c3ccccc3)nn2)c1C C1(O)(CC(=O)NC(C(=O)N(CCCO)CC)CC2CC2)CCCOC1 C1(CNC(c2cnc(OC)s2)=O)CN(C(=O)Cn2ncc(C#N)c2N)CCC1C C(=O)(C(CC)C(C)O)NC1(C)CN(c2nnc(CC)o2)C1 C1(CC=O)CCC12CCC2.c1(C(C)NC(C2(CO)CC2)=O)ccc(C)cc1 N1(C(CCC)=O)CCCCCC1CNC(c1ccc(C)nc1C(C)C)=O N1(C(C(C(C)C)OCC(C)C)=O)CCC(C(=O)O)C(Cc2nnsc2Cl)C1 C1(NC(Cn2c(C)cnc2)=O)CCC(C)N(C(C2CCCN2N=O)=O)C1 c1(C(=O)OC)scc(C)c1NC(=O)NC(c1cccc(OC)c1)C C1(N(C(CN2CCC(CC)CC2)=O)C)CCCN(C(=O)CC2CCCO2)CC1 C1(NC(C=C(C)Cl)=O)CCC(O)CN(C(=O)C(C)(O)c2ccccc2)C1 N1(C(c2cc(CC)n(C)n2)=O)CCN(C(c2cc(OC)nc(C)c2)=O)CCC1C N1(C(COC(CC)(C)C)=O)CCC2CCCC12.C(C1CC1)(C1CC1)=CC=O.C N1(C(C2(C(C)C)CC2)=O)CC=CC(NC(=O)C(N2CCCC(O)C2)C)C1 CC1(C)CCOC1CC(=O)Nc1ccccc1NS(C)(=O)=O N1(C(C(CCOC)OC)=O)CC(CNC(c2cccc[n+]2[O-])=O)OC(C)(C)C1 Cc1nc(N)cnc1C(N1CCCC1C(C)C)=O.C1(C=O)CCS(=O)(=O)CC1.N CC1CCC(CNC(c2ccc(F)cc2I)=O)N(C(=O)C(N)=O)C1 C1(NC(C(CC)=CC)=O)CC(NC(=O)CCC(C)C)C12CCOCC2 CCC(C)C(O)C(C)C(=O)NCCCOCC(C)(C)NC(c1cncnc1)=O c1(C(=O)NC2(C)CN(C(C(C)Cc3ccccc3)=O)C2)ccc([N+](=O)[O-])n1C Cc1cc([N+](=O)[O-])cnc1NC(C1CCCN(C(c2cc([N+](=O)[O-])c[nH]2)=O)C1)C c1(C(=O)NC2CC2NC(C2(F)CC2)=O)ccc(=NCC2CC2)[nH]c1 C(C(=O)N(CC(=O)NCC1(C)CC(C)=NO1)C)(C(C)C)OCC N1(C(C2CC(C)(CC)C2)=O)CCCCC1C1(NC(c2nccnc2N)=O)CC1 Cn1cc2cc(C(=O)NC3(CNC(=O)CC4(C)CCOCC4)CC3)ccc2n1 N1(C(c2ccc(CC)[nH]2)=O)CC2(NC(c3cnc(C)nc3C)=O)CCC1C2 c1(C(N(C2(C(=O)OCCOC)CC2)C)=O)cc(C)c(OC)c(C)c1 C=CCCCCCCCCC(=O)NCC1CCCN(C(c2nccn2C)=O)CC1 c1(CC(N2C(CC(=O)N)CC2)=O)ccccc1F.C1(CC2CC2)CC1C1CCC1 Cc1cnc(NCC2CC(NC(=O)CC)C2)nc1S(C)(=O)=O.[SH](C)(=O)=O C(=O)(CC1C(=O)Nc2ccc(C)cc21)N1CC2CC(CC(NC(CCC)=O)C2)C1 N1(C(COC)=O)CC2CC1C2NC(C1(c2cccc(Br)c2)CC1)=O CCCCC(CC)CC(=O)N1CCC(F)C(NC(c2cnn(CCC)c2)=O)C1 Cc1coc(C)c1C(=O)NC1CN(C(C2CCCCC2C(N)=O)=O)CC1O Cc1nnc2n1CC(C(N1CCCC(F)(C)C1)=O)C2.n1(CC(=O)N)nnc(=O)[nH]1 C1(CC=C)(C(=O)N)CCOCC1.C(C)C(C)(C)C.c1(C2C(C=O)C2)ccco1 N1(C(CC(C)SC)=O)CCC2(CC1)CC2c1cn(CC2CC(F)(F)C2)nn1 c1(C(N2CCN(C(C=C(COC)C)=O)CC2)=O)cc(OCC(C)C)nc(Cl)c1 c1(C(=O)NC2CCCC(NC(COCCC(C)C)=O)C2)ccc2nnc(S)n2c1 C(C(CC(C)C)C(=O)NCCC(C)(C)C(=O)NC(C1CCOC1)C)OC c1(NC(C2CN(Cc3sc(Cl)nc3Cl)CCS2)=O)ccc(F)cc1CO CC1OCCCC1C(N1CCC(N(C(=O)CC2(C)OCCO2)C)C1)=O CCCCCCC(O)CCC(=O)N1CCC(Cn2cc(COC(=N)O)nn2)CC1 CCCC(CNC(=O)C(c1cccn1C)=O)C(=O)N(C(C)CC(=O)OC)C c1(C(N2CCCN(C(CCC=C=C)=O)CC2CO)=O)ccc2c(c1)NC(=O)C2 CC1=C(C(=O)NC2(CNC(=O)C(C)O)CCC(C)(C)CC2)Cc2ccccc2O1 C1(CCN(C(=O)C(C)(C)c2ccn(C)n2)C)CCN(C(=O)CCC2CCC2)CC1 c1(OC)cc(C(=O)NCCC2CC2)c(F)cc1N.C1(C=O)Cc2nncn2C1.N c1(C(=O)NCC(C(C)(C)C)NC(CC2N(C)CC=CC2)=O)c(F)cccc1Cl N1(C(C2CN(C)C(=O)N2)=O)CCC2CN(C(c3c[nH]c4nccc-4c3)=O)CCC12 C1(NC(CCC(=O)NCC)=O)CC2CCCC(C1)N2C(c1cnn(CC)n1)=O c1(C(=O)NC2(CNC(C(C)OCOC)=O)CC2)nc(O)c(C)s1 Cc1ccc(CC(=O)NC(C)(C)CNC(=O)CCc2ccc(O)cc2)cc1C C1(CNC(C2C(C)C2)=O)CCC(N(C(=O)CN(C)C2CC2)C)CC1 c1(CN2CC(NS(=O)(=O)c3nccs3)C(F)(F)C2)c(F)c(F)c(F)c(F)c1F CC(C)CC(F)(F)C(=O)NC1CCC(NC(C2CC2(c2ccccc2)C)=O)CC1 c1(CC(=O)N)cnc(O)nc1O.CC(Cc1ccccn1)C(=O)NCCC1CC1 C1(NS(C)(=O)=O)CN(CC(=O)NCC)CCO1.c1ccccc1C(F)(F)F.O C1(c2cn(CCN(C(C(C)C3CCOC3)=O)C)nn2)CCCC(=O)C1 c1(CC)cccc2ccc(CN(c3nnc(-c4ccccc4OC)n3C)C)nc12 CCCC(C(=O)NCc1cccc(C(N2CCOC(C)(C3CC3)C2)=O)n1)C(C)C N1(C(c2cn3cccnc3n2)=O)CCCC2(C1)CN(C(C1CCC1)=O)CCO2 CN1CCCCC1CCc1cn(CCC2CN(C(=O)C(F)OC(F)(F)F)C2)nn1 C(CC(CC)CC)NC(C=CC(CC)=CC)=O.N1(CC=O)CC2CCC1C2.N C(=O)(C#CC1CCOCC1)NC1(C)CN(C(CCOc2ccc(C)c(C)c2)=O)C1 c1(C(=O)NCC(C2CC2)NC(C2(CC#C)CCCO2)=O)ccc(Br)cc1N CN=c1[nH]nc(CC(N2CC(NC(=O)C(F)(F)CO)C(n3cccn3)C2)=O)s1 N1(C(C2(SC)CN(C(C3CCC(F)(F)C3)=O)C2)=O)CC(C)OCCC1C C1(NC(C(C)SC(C)C)=O)C=CCCC1C(N1CC(S(C)=O)C1)=O c1(CNC2CC(C(=O)NC(C=C)CO)C2)[nH]c(C)c(C(=O)OC)c1C C1CCC(C)CC1.N1(C(COCC(=O)OC(C)(C)C)=O)CC2CC1C2.C=O N1(C(C(C(C)C)NC(N)=O)=O)CCN(C(c2cc(C(F)F)cs2)=O)CC1C c1(C(c2nnnn2C(C)(C)CC)NCC(CC)C)cc(C)nn1CCC Cc1cc(O)cc(=O)n1CC(=O)N(C(C)CNC(=O)C(F)CC1CC1)C C=CC(C)(CCOC)C(=O)N(CCCCCC(=O)NCC(=O)OCC)C CC1(C)CC(NC(C2CC(C)(C)C2)=O)CCN(C(C2CC2c2ccccc2)=O)C1 N1(CC(=O)N(C2CCCCN(C(=O)CCCCCF)C2)C)CCc2sccc2C1 N1(C(c2c(C)c(F)ccc2)=O)CC2CCOC2(CNC(=O)C(O)CC(F)F)C1 C1(N)(CC)CCN(CC(CBr)C2CCC2)CC1 Cc1coc(C)c1C=CC(=O)NCC1C2CCC(C2)N1C(c1ccon1)=O c1(C(N2CCC(CNC(C3CCC(C)O3)=O)C23CC3)=O)cc([N+](=O)[O-])ccc1O c1(C(N2C(CNC(c3c(C)ncs3)=O)CN(C)CC2)=O)cn2cccc(C)c2n1 C1(CNC(C(CC)=CC)=O)CC2CC(C1)N(C(=O)CCSC(F)(F)F)C2 Cc1nc2c(s1)CCCC2C(=O)NCC#CCNC(=O)C(C#N)(C(C)C)C(C)C Cc1c(C(=O)NC2(C)CN(C(C3(F)CC=CCC3)=O)C2)cnc2ccnn12 C(=O)(C(C(C)C)N(C)C)NCC(C1CCCCC1)NC(C(C)=C1CC1)=O Cc1c(C(=O)NC2CC(NC(=O)CCC3CC3(Cl)Cl)C2)nnn1C(C)C N1(C(C(c2ccc(C)s2)C)=O)CCC2CCC(C1)N2C(=O)Cn1nccn1 c1(NCC(=O)NCC2N(C(c3ccc(C=C)cc3)=O)CC2)nc2ccccc2s1 c1(C(N2CC(NC(C(C)Sc3nncn3C)=O)C(C)C2)=O)cc2c(s1)CCC2 N1(C(C2(C=C)CC2)=O)CC2(CC(NC(=O)C(F)C3CCOC3)C2)C1 c1(C(=O)NCC(C)(C(C)C)NC(C2C(OC)CC2)=O)ccn2ccnc2n1 c1(C(N(CCCNC(c2cncnc2)=O)C)=O)ccc(N=S(C)(C)=O)cc1 N1(C(C(Br)=C(C)C)=O)CCN(C)CC1CNC(=O)CCC1OCCO1 N1(C(CCSC)=O)CCC2(CC1)CN(C(=O)CN1CCC(C)CC1)C2 N1(C(C(C(C)C)(C)O)=O)CC(C)(C)OC2(C1)CN(C(c1c(N)cccc1Cl)=O)C2 CC1(C)CC(C)CN1C(c1coc(C(N)=O)c1)=O.c1(C(=O)N)cncc(N)n1 CCCC(C)CC(=O)N(CC(=O)NC1CC1C1CCCC1)C1CCC1 C1(C(=O)OCCCC)C2CCN(CC2)S1(=O)=O c1(N(CCCNC(c2c[nH]c(=O)cn2)=O)C2CC2)nc2c(F)cccc2o1 c1(C(N2CCC3(CCCN3C(=O)C(O)C(F)(F)F)C2)=O)cc(Cl)cc2c1OCC2 C1(C(N2CCC(N(C(Cn3nc(C)oc3=O)=O)C)CC2)=O)CC2(C1)OCCO2 c1(N2C3CN(C(CC4C(C)CCC4)=O)C(C3)C2)ncc2ccccc2n1 c1(OC)cc(C)c(CN2CCSCC2C(=O)NC(C)CN(C)C)c(C)c1 c1(NC(CCCOC(C(C)C)=O)=O)ccc(S(=O)(=O)NC(C)(C)C)cc1 Cc1ccc(C(N2CCC3(CC(NC(C4CC4C(F)F)=O)C3)C2)=O)c(=O)n1C CC1(C(=O)NC2CCCN(C(=O)C(C)(C)C3CCCCC3)C2)CC(C#N)C1 c1(C(=O)NC2CN(C(c3cnc(C)o3)=O)CC(C)C2)cn2ccn(C)c(=O)c2n1 C#CCC(C)(C(=O)NCc1ccnc(OC)n1)NC(=O)CC1CCC(=O)NC1 C(=O)(C1Cc2c(Cl)cccc21)N.N1(C(c2n(CC)cnn2)=O)CCC(COC)C1 C1(CCNC(C2CCC3(CC3)C2)=O)CCCCN1C(=O)C=Cc1cscn1 C1(NC(=O)CN2CC3CC3C2)CC(C2CCN(C(=O)CCc3ccco3)CC2)C1 c1(C(=O)NCC(=O)OCC=C)cc(Br)ccc1.C1(CC=O)CCC2CC12 C1(CCCC)CN(C(=O)CC2=CCCC2)CCN1C(c1cc(C)n(C)n1)=O Cc1cc(NOCC(F)(F)F)ccc1OCC1OCCC1(C)C c1(C(N2CC(C(C)NC(=O)COCC3CC3)C2)=O)ccc(N)c(F)c1 c1(OC(C(=O)NC(CC#C)C(N)=O)C)cccc(C#N)c1 C1(C(N2C(CN=[N+]=[N-])CC2)=O)CCC2(CC2)N1C(=O)CC1CC=CCC1 c1(Cn2cc(CN(C)C)nn2)cncc(C(=O)N(O)Cc2ccccc2)c1 C1(C(=O)NC(C)CCNC(=O)CC(O)c2ccccc2)CCC=CCC1 C#Cc1ccc2c(c1)CN(CC(=O)Nc1sccc1SCC(F)(F)F)CC2 N1(C(C=CCC)=O)CCN(C(=O)C(C)(C)c2cc[nH]n2)CC1c1ccncc1 N1(C(CCS(C)(=O)=O)=O)CC2CC1CN(C(=O)Cc1ccc(O)c(Cl)c1)C2 C(=O)(CC(C)(C)O)NCCC1CC(NC(C(C)O)=O)C1 c1(C(=O)NC2C(NC(C3C(=C)C3)=O)COC2)csc(C)c1OC N#Cc1ccc(C(=O)O)cc1.c1(C=O)ccc[nH]1.C1C(=O)NC2C(C2)CO1 C(=O)(C(CC)CCOC)NCCCC1(NC(C(CC=C)c2ccccc2)=O)CC1 C(=O)(C1COc2ccc(F)cc21)NC(CCNC(CC(=O)NCC)=O)(C)C C1(C(N(CC(C)NC(CC2CC(SC)C2)=O)C)=O)CCN(C)C(=O)C1 c1(NC2CCCC(NC)C2)nc2ccccc2nc1NCc1nn[nH]c1C1CC1 C(C(CC(F)(F)F)NC(c1cccn(C)c1=O)=O)NC(Cc1cnc(C)[nH]1)=O Cc1nc(=NC(=O)C2CC(NC(c3cc(C4CCCN4C)[nH]n3)=O)C2)s[nH]1 c1(OCCOC)cccc([SH](=O)=O)c1.C1(C(=O)O)CCCO1.c1ccccc1.N C1(C(=O)NCC(O)CCNC(c2ccon2)=O)(CC)CCCO1.N(C)(C)C Cc1cn2cc(C(=O)NC3(CNC(C4CCOC(C)(C)C4)=O)CCC3)sc2n1 C(=O)(C1CCc2scnc21)NCC1C(NC(c2oc(C)c(CO)c2)=O)COC1 C(CCC)(C(O)C(=O)N1CC2(C)CCC2(C)C1)NC(C1(CCCC)CC1)=O C(C(C)C(=O)N(C(C)CCNC(=O)C(C)Cc1cnco1)C)OC(C)=O C1(C)(CC)NC(=O)C2=C1N(CC(F)F)C(=S)NC2c1cccc2ccncc12 c1(C(N2C(c3cn(C)nc3C(=O)O)CCC2)=O)ccn2ncc(Br)c2n1 C1(NC(CCCOCC=C)=O)CN(C(=O)CC(C)(C)C)CC1OC C(=O)(CC(C)C(F)F)N1CCN(CCN(C(C(CCOC)OC)=O)C)CC1 c1(C(=O)NCC(c2ccsc2)C)cc(CNC(=O)CC2CC=CCC2)no1 C1(C(=O)NC2CCCC(NC(c3ccc(F)o3)=O)C2)(COC)CCOCC1 N1(C(C2ON=C(C)C2C)=O)CC2(CCN(C(=O)CCc3cncc(Br)c3)C2)C1 C1(NC(CC=C)=O)CCN(C(c2noc(Cc3ccc(Cl)cc3)n2)=O)C(C)C1 C(CN=C(NCC(c1ccc(F)cc1)(F)F)NCC1CCOC1)c1scc(C)n1 N1(C(C(C)n2cncn2)=O)CCC(C)(C)C(NC(c2scnc2Cl)=O)C1 N1(CCC)CC(NCC(C)(C)CSC)CC1=O N1(c2cc(C)nc(CO)n2)CC2(C1)SCCC2NC(=O)CC1CCOCC1 c1(CC(=O)NCC(CO)NC(CCSCCCC)=O)ccc(Cl)c(F)c1 c1(OC)cc(F)ccc1-n1cc(CS(=O)(=O)CC)nn1.C1(O)(C=O)CCCOC1.N c1(SC)ccc(NC(=O)CC2CC(NC(C3CCC4(CC4)C3)=O)CCO2)cc1 C(=O)(CC(F)(F)C(F)F)N1CCC2(C(C(N(c3c(C)nsc3)C)=O)C2)C1 C1(NC(c2c(C(C)C)con2)=O)CCC2CCN(C(=O)C=C3CCC3)C12 c1(C(N2C3CC(CNC(CN4C(C)CCC4)=O)(OC3)C2)=O)ccc2nnnn2c1 C(=O)(CC(C)CC(C)C)N(CC(CN(C(c1ccc(C)nn1)=O)C)O)C Cc1ccc(C(N2CC3CCC(CNC(C45CSCC4C5)=O)C3C2)=O)c(=O)n1C O=C(C(F)(F)CCn1cc(-c2ncc(F)cn2)nn1)NCC(=C1CCSCC1)F N1(C(COCC=C)=O)CCCC2(CCCN2C(=O)C(CC)CCCCC)C1 c1(-n2ncc(CNCC(c3c[nH]c(=N)s3)N3CCCC3)c2)ccc(Cl)cc1Cl c1(C(N2C(C)CC(NC(Cn3c(C)csc3=O)=O)C2)=O)ccc2c(c1)COCC2 C1(C(=O)NC)C2CN(C(=O)CC3CCCN(C(c4ccn(C)c4)=O)C3)CC12 N1(C(C(C)NC(c2cn(CCS)nn2)=O)=O)CCS(=O)(=O)CC1.c1ccccc1 C1(C(=O)NC(CN(C(c2ccccc2)=O)CC)C)OCCC1(C)C.N(C)C.C n1(CCCC(=O)OC(C)C(=O)N(C)C)ccccc1=O C(=O)(C1=CCCC1C)N1CC(NC(c2cncc(C)n2)=O)C(CC(C)(C)C)C1 C1(NC(C=CCC)=O)CCC(C)N(C(c2csc(Br)c2)=O)C1 C1(NC(Cc2ccc(C)c(Cl)c2)=O)C2CC3CN(C(=O)C=CC4CC4)C1C3C2 Nc1cnc(C(=O)NC2CCCC2NC(c2cc(-n3cnnc3)ccn2)=O)cn1 Cc1ccc(C(N2CCCC(CNC(=O)CC3(C4CC4)CC3)CC2)=O)c(F)c1 C1CCCN1C(=O)CC1CCC(C(F)(F)F)O1.C(CC(=O)NC)OCC#C c1(C(=O)NCC23CC(NC(C(CC)O)=O)(C2)C3)cnc2n1CCOC2 N1(C(C2CCN(C(=O)CCN3CCCC3)C2)=O)CCN(c2cc(Br)ccn2)CC1 C1C2CC1N(C(C13CCCC1(C(N)=O)C3)=O)C2.c1(OC(C)C=O)cccnc1.N N1(C(c2cc(C3(C)CC3)n[nH]2)=O)CCC(F)(CNC(C2CCC23CCC3)=O)C1 C(=O)(CCCCCCN=[N+]=[N-])NC1C(NC(c2n(C)cnc2C#N)=O)CC1 c1(C(N2CCC(NC(CC(C)(C)O)=O)C2(C)C)=O)ccnc2ncnn12 c1(C(N(C)CC)=O)cnc2nc(NC(c3n[nH]c4ccc(C)cc34)=O)ccc2c1 C(C1CN(C(c2cc(C)[nH]n2)=O)CC1C(N1CCOCC1C)=O)=CC C1(C(N(C)CCNC(=O)CSC(F)F)=O)Cc2cccc(OC(F)F)c2O1 c1(C(C)NC(C(F)=C(C)C)=O)ccncc1 c1(C(=O)NC(C(C)NC(c2cc(C)c(C)[nH]2)=O)CO)c(O)cc(Br)cc1F c1(C2CCN(C(CN(C(C)C)Cc3nn[nH]n3)=O)C2)ccc(C(F)(F)F)nc1Cl c1(C(=O)NC2(CCCNC(C(F)OC)=O)CC2)cccn1C C1(CC)(NC(c2ccc(C)cn2)=O)CCCN(C(C2(C(=O)NC)CCC2)=O)C1 C(=O)(CCCC(=O)N1CC(NC(=O)C2=COCC2)CC1C)N(CC)CC C1(C(N2CC3C(NC(C4CC5CC4CC5O)=O)C3C2)=O)C2CCCCCC12 CCCC(C(=O)NC1CC1CNC(=O)CSCc1ccccc1)C(C)C N1(C(c2c(OCC#C)nccc2)=O)CC2OCCN(C(=O)CCOC3CC3)C2C1 c1(COC)ccnc(C(=O)NCC(O)CN2CCOC(C)C2)c1 C#CC1CCN(C(=O)C(=O)N2CCC2CNC2CC2)CC1 n1(CCOC)cc(C(=O)N(C2CN(C(C3CC34CCC4)=O)CC2O)C)c(C)n1 C1(C)(NC(Cc2cn(CC)nc2)=O)CCCN(C(=O)CCCc2nncn2C)C1 N1(C(CCC(C)OC)=O)CC(C)(C)OCC1CNC(=O)Cc1ccc(O)nc1 C1(C(N2CC3CCC2CC3)C(=O)Nc2ccccc2Cl)CCC2(CCCC2)CC1 c1(C(=O)NC(C2CCN(C(C(C)C(C)(F)F)=O)C2)(C)C)cnc2n(c1=O)CCS2 C1(CN(C(=O)C=O)C)COCCN1C(=O)CSCC(F)(F)F.C1CC1.N C1CCCN(C(c2ccccc2C(F)F)=O)CC1F.C(=O)(COCC(=O)N)NC Cc1ccc(Cl)cc1C(=O)NC1CC(CO)N(C(c2ccc([N+](=O)[O-])[nH]2)=O)C1 N1(C(C(CC)C2CC2)=O)CCCC(C2CN(C(C3(O)CC3)=O)C2)C1 C1(C(N(CCCCN(C)C(C2CCC(=O)N2)=O)C)=O)CCCC1S(C)(=O)=O C(CC(C)(C)NC(C1CCCC1CNC(C1(C(C)C)CC1)=O)=O)OC CC1CC2CCC(C1)N2C(C1COCCN(C(C2(C3(O)CCC3)CC2)=O)C1)=O O=C(N=c1[nH][nH]c2c(Cl)cccc12)C1CC1NCc1ccc(O)c(F)c1F N1(C(CCn2ncc(C)c2)=O)CCC(CNC(=O)C=Cc2ccsc2)CC1C C(=O)(CC(C)(C)C(=O)OC)N1CCCCC(CNC(c2ccn(CC)n2)=O)C1 NC1C2CC3CC(C2)CC1(NS(=O)(=O)c1cccc(N2CCOC2=O)c1)C3 N1(C(C(C2CN(C(=O)C(O)CC(C)C)C2)OC)=O)CCC2(CCCOC2)C1 c1(CC=C)cc(CNCc2nnc(C(C)(C)C)s2)cc(OC)c1OC c1(C(N2CCC(COC)(CNC(=O)CCC)CC2)=O)nc(Cl)cc(N)c1Cl.O C1(C(N(CC=C)CC)=O)CN(C(C2C=CCS2)=O)CC1OC C1(C(=O)NCC(CCC)NC(=O)C(F)(F)CC)CCCN1N=O c1(C(N2C(C)CC(NC(=O)C(C)(C)C)CC2)=O)cc(O)cc(N)c1Cl C1(NC(CCCC#C)=O)COCCN(C(c2ccc(C)cc2SC)=O)C1 c1(C(N2CCC(CC3CC3)C2)=O)csc(-c2cc(Br)cs2)n1 C(CCN=c1ccc(C)c[nH]1)NC(C(=O)NCc1c(OC)nn(C)c1)=O C(=O)(C1=CC2(CN(C(C3CCC3C)=O)C2)OC1)N1C(C)C(C)(C)CC1 c1(OCC=C)ccc(Cl)nc1C(=O)N.C12CC1CN(C(c1cn[nH]c1)=O)C2.C C1(C(=O)NOCC2CCOC2)CC(F)(F)CN1C(c1occ2c1CCC2)=O N1(C(C2(CCC)CCNC2=O)=O)CCN(C(c2coc(C(C)=O)c2)=O)C(CF)C1 Cc1cc(C(=O)NC(C2(CNC(=O)C)CC2)C)nc(O)n1.c1cccnc1 C1(NC(CCNC(=O)C=CCl)=O)CN(C(=O)C(F)=C2CCC2)CC1C(F)F C1(C(N(C2(C(=O)N)CCC2)C2CC2)=O)C2CCCC12.CCCCC1CCCO1 c1(C(N2CC(C(C)NC(C3CN(C(C)C)C3)=O)OCC2)=O)ccc(CO)cc1F C(CCO)(C(=O)N1CCCCC1C1(NC(C2CNC(=O)N2)=O)CC1)N(C)C c1(C=O)ccc2nn[nH]c2c1.C12(NC(C(C)OCCC(C)C)=O)CC(C1)C2.C c1(NC(C2NCC(C)C2)=O)cccn(Cc2ccccc2)c1=O C(CS(=O)(=O)CC(=O)N1CC2CN(C(C3CC(C)CC(=O)N3)=O)CCC12)OC CN1CC(O)CC1C(=O)NC1CC(C(=O)NCCCc2nncs2)C1 C1(c2n(CCC)nnn2)(NCC2(C)CSCCO2)CCCC(C)(C)C1 N1(C(C=CC)=O)CC2CC(C1)CN(C(=O)C(F)(F)c1nccs1)C2 C1C2=CCN(CC2)CCN1.c1(C2C(C(=O)Nc3csc(O)n3)C2)ccccc1F c1(SC)nccc(=NC2CN(C(c3nccnc3N)=O)CC2C)[nH]1 c1(N(CC(C)C#N)C)nc(N2CCCCC(N3CCOCC3)C2)c2[nH]ccc2n1 C#Cc1cc(NC(=O)CC2(C)CC2)cc(F)c1.n1(CC=O)cc(C)cn1.N C1(C(N2CC(N(C(=O)CSc3cn[nH]c3)C)C2)=O)CCc2nncn2C1 C(=O)(CCCNC(=O)C=CC1CCC1)NCCN(C)C1CC1 C=C(C)C(CC(=O)NCC(C(C)C)NC(=O)Cc1ccns1)OCC N1(C(C2(C#C)CC2)=O)CCC(CCOC)(NC(c2cnc(N(C)C)nc2)=O)C1 N1(C(C2(CC=C)CCC2)=O)CCCCC1C(=O)NCC(c1ccc(O)cc1)O C1(NC(CCCCC#N)=O)CN(C(c2cnc(Cl)s2)=O)C2(CCCCCC2)C1 Nc1cnn(CC(=O)NCCC(F)(F)F)c1.C1C(=O)N1 Cc1cc(CN2CC(NC(c3ocnc3C)=O)CC(C)C2)cc(O)c1 c1(OCC)ccc(C(N2CC(CCNC(C3(C=O)CCC3)=O)C2)=O)cn1 Cn1cnc2cc(C(N3C4CN(C(c5ccc(O)c(Br)c5)=O)CC34)=O)ccc12 Cc1cc(C(N2CC3CCC3(NC(c3ncncc3F)=O)C2)=O)c(C)n1C Cc1c(C(=O)Nc2ccc(C3CC3CO)cc2)cc(C(C)(C)C)n1C N1(C(CCS(C)=O)=O)CCC2(C1)CN(C(C1CC(O)CN1C(N)=O)=O)C2 n1(CC(=O)Nc2c(OC)c(C(N)=O)ccc2)ccc2c(C)cccc12 CC1CN(C(c2cc(C(N)=O)[nH]n2)=O)CC(CC)O1.C1(C(=O)N)(CCF)CCC1 C=CCC(C)(CC=C)NC(=O)C(O)CCCNC(=O)CC1CCN(C)C1=O c1(C(=O)NCC(C)C)cc2c(s1)CCSC2.c1(C=O)coc(C(F)(F)F)n1.N C(=O)CC(C)CC(C)(C)C.C(=O)(C(C(C)(C)C)NC(C1CC=CCC1)=O)NC N1(CC(C)(C)NC(=O)CC2CC=CC2)CCCC1=O CC1CCN(CC(=O)NC2(CNC(=O)CCOC(C)CC(C)C)CCC2)C1 CC1CN(C(c2ccc(=O)n(C)n2)=O)CCC1NC(c1cc(Br)sn1)=O n1(CCC)cc(C(=O)NC(C2CN(C(C3CCOC3C)=O)C2)C)nn1 n1(CC(=O)NC2C(NC(CC3C(CC)C3)=O)COC2)cccc(N)c1=O C(=O)(N=c1[nH]onc1C(N)=O)C1N(C(c2cc(OC)c(O)cc2)=O)CC(O)C1 c1(CCCC)cc(C)c(NC(=O)NC2(Cc3ccccc3)CCC2)cn1 C#CC1CCC(NC(=O)Nc2ccncc2C)C1 C(=O)(CC(O)CC(C)C)N1CCC(NC(C2C3(CC(OCC)C3)C2)=O)C(O)C1 C12(CNC(C(c3cn(CC)nc3)=O)=O)CC1CN(C(C1CCCOC1C)=O)C2 c1(NC)cnc(Cl)cc1C(=O)NC1CCCN(C(=O)COCCOC)CC1 C1(C(N(C(C)C=O)CCC)=O)CC(=O)CC(=O)N1.c1(CC)ccc(F)cc1.N N1(CCC)CCCC(C(=O)NC(C2CCCN2C(=O)C)(C)C)C1.C(C)(=O)N CC1(C)C2CC(C(=O)NC3C4CC5C(C4)C35C=O)CC12.N1(CC)CCCC1 C1(NC(CCn2cc(-c3ccc(OC)nc3OC)nn2)=O)CC2CCCCN2C1 CC(C1CCCCC1)=CC(=O)NCC1CCCC1NC(=O)CC1CC12CC2 N1(C(CC2(C)CCOCC2)=O)CCCC2(CC(NC(=O)CC3=NNC(=O)C3)C2)C1 C1(CNC(=O)CCOCC(F)F)CCCC1.c1(C=O)ccn[nH]1.C1CC1.C CCCCCCC(F)C(=O)NC(c1ccccc1)CNC(=O)CC1(OC)CC1 N1(C(c2cc(C)ns2)=O)C2CCC1CN(C(C1(C)CCCC1C)=O)C2 Cc1ncc(NC(c2nnn(C)n2)c2nnnn2C2(C)CC2)cc1C1CC1 O=C(CS(=O)(=O)c1ccccc1)NC1CCCN(Cc2ccc(F)c(F)c2Br)C1 Cc1ccc(CC(=O)NC23CC(NC(=O)CCC4CCOC4)(C2)C3)c(Br)c1 N1(C(CCC=C(C)C)=O)CCC(C)(C(N2CCCC2c2ccccc2F)=O)C1 C1(O)(CN(C(=O)COC2CN(C(=O)CC3CC=CC3)C2)C)CN(C)C1 c1(CNC(C2(CCNC(C(C)SC)=O)CC2)=O)nc(C(N)=O)co1 Cn1nc(Br)cc1C(=O)NC1(C)CC1.c1(C=O)ccn(C2CC2(F)F)n1.N CC(C)CS(=O)(=O)CC(=O)NCC1CCCN1C1CCN(c2ccccc2)C1=O c1(CC(=O)NC(C2CN(C(c3ccc(CC)o3)=O)C2)C)c(C)nc(O)nc1O C1(NC(COCCCC#C)=O)CN(C(c2ccnn(C)c2=O)=O)CC12CCC2 c1(C(=O)NC2CC3CCC2(NC(C2CC24CCC4)=O)C3)cnn2ccccc12 C(=O)(CCCC(=O)c1ccccc1)NC(CC(C)NC(c1n(CC)nnc1)=O)C c1(C(=O)NC2CCN(C(c3ncc(N)cc3Cl)=O)C2)c[nH]c2ccncc2c1=O C12(C(=O)NCc3c(C)ccc(C)c3)CCCC1CN(C(=O)C=C1CCC1)C2 C1(SC)CCCN(C(=O)C(C2CCCCC2)NC(=O)C2=CCSC2)C1 n1(CCCC)nc(C)c(C(=O)NCC(C)C)c1Cl.c1(C(=O)N)cc(N)cc(O)c1 C1(C(NOCCOC)=O)CCOC(=O)N1 c1(-c2n(CCC(C)C)nc(CCOC(C)C)n2)noc2ccc(F)cc12 c1(OC)ccc(Cl)c(CC(N2CCC(NC(C3(O)CCSC3)=O)CC2C)=O)c1 C(=O)(C(C(C)OC(C)(C)C)N(C)C)NC(CNC(C(CC)N(C)C)=O)CO c1(C(N2CCCC(CCNC(c3ccc(C#N)s3)=O)C2)=O)c(O)ccc(F)c1F C1(CNC(CC=C)=O)CN(C(C2CC(CN(C)C)C2)=O)CC1(C)C CCC(CC)C(=O)NC1C=CCN(C(C2CC2C)=O)C1 N1(C(CSC)=O)CC2(CCNC(c3ccnc(C(F)(F)F)c3)=O)CCC1CC2 N1(C(=O)NCC2(N(C)C)CCC2)C(CC2CCCCC2)CC2CCCC12 C1(C(=O)NCCCN(C(C)=O)C)CSCCN1C(=O)C(c1ccn(C)c1)C C(CCC)(C(=O)N1CCOCC1CC1CC1)NC(CSCC)=O C=CC(CC(=O)N(C)CC1CCCN1C(C1(C)CC1C)=O)c1ccc(OC)cc1 c1(OCc2cn(C3CC(C(=O)NC4CCOC4)C3)nn2)ccc2c(c1)OCO2 Cc1c(F)ccc(C(N2CCC(N(C(=O)C(CO)C(C)(C)C)C)CC2)=O)c1Cl C=CCC(C(=O)N1CC2CCCC2C1C(N1CCC(O)CC1)=O)C(C)C c1(OC)ncccc1CC(=O)N(CCC(C)NC(C1(C2CCCO2)CCC1)=O)C N1(CC(=O)N(C23CCCC2CCO3)c2c(C)onc2)CCCC(C)(C)C1C c1(CCC(=O)N)cncc(F)c1.n1(C(CC)C)nccc1C(=O)NCC(C)(C)C Cc1cc(C(F)(F)F)ncc1C(=O)N(CC)C1CC1.c1(C=O)n[nH]c(C)c1Cl Nc1ccc(CNC(C2(c3ccc(F)cn3)CCC2)=O)nc1F C(=O)(C(C(C)(C)C)NC(C1CCC1C)=O)NC.C(=O)C(O)CC(N)=O.N c1(CCNC(c2cccc(OCCc3ccc(F)cc3)c2)=O)ccc(Cl)c(F)c1 C1(C)CC(F)(F)CN1C(=O)CCCC1(C)N=N1.c1(OC)nccc(C=O)n1.N N1(C(C(C2CCOC2)NC(c2ccc[nH]2)=O)=O)Cc2ccc([N+](=O)[O-])cc2C1 C1CCC2(CN(C(=O)C=Cc3ccoc3)C2)O1.C1(C(=O)N)(COC)CC1 CC1(C)CC(C(=O)NCC2(O)CC3CCC2C3)N(C(c2ccc(Cl)s2)=O)C1 N1(C(CN2C(C)CCC2C)=O)CCCC(NC(C2CCN(CCF)CC2)=O)CC1 c1(C(N2CCN(C(CC3C(C)CCC3)=O)CC2)=O)nccc(F)c1Cl C(=O)(CCC(CC)CCC)N1CC(CC(=O)NC(CCCC)CCC)(OC)C1 C(c1ccc(C(F)F)o1)=CC(N1C(C(C)NC(C2CC2F)=O)CCC1)=O Cc1[nH]nc(CNC(C2CN(C(c3cncnc3)=O)CC2C)=O)c1C CC1=C(C(=O)N2CC(CC(=O)NCC(C)(O)C3(C)CC3)C(C)C2)COCC1 c1(C(=O)NCCc2cnc(Nc3ccn4nccc4n3)s2)ccc2ncoc2c1 N1(C(c2cnc(SC)n2C)=O)CCCN(C(C2CC(F)C2)=O)CC1 N1(C(Cc2c(CC)noc2CC)=O)CCCC2(NC(=O)C(O)C3CC3)CCCC12 C1(C(=O)NCc2c(C)c(F)ccc2)N(C(=O)C2=CCCSC2)CC12CCCC2 Cc1noc(N)c1C(=O)NC(C)C1CCC1.c1ccncc1.C1(C(=O)N)CC1 CC1(C)CC(C(N2CCC2CN=[N+]=[N-])=O)CN(C(=O)C2=CCSC2)C1 CC1c2ccc(F)cc2CCN1C(=O)Nc1ccn2ccnc2n1 C1(C(N2CCOCC(NC(=O)CN3CC=CC3)C2)=O)CC12CCCCCC2 c1(C=O)ccc2ccnc(O)c2n1.N1(C(C2CN(C(N)=O)C2)=O)CC(F)(C)C1.N C(=O)(C(C(C)C)NC(N)=O)N1CC(N(C(c2c(C)con2)=O)C)C1 C1(C(=O)NCCC2(O)CN(C(Cc3ccc(C)o3)=O)C2)CCC2CCCCC2C1 N1(C(CC2=NNC(=O)C2)=O)CC2ON=C(CNC(c3cccc(Cl)c3Cl)=O)C2C1 c1(C(=O)NCC2CCCCC2NC(=O)C(F)F)cc([N+](=O)[O-])ccn1 Cc1cc(S(=O)(=O)NC2CCCN(Cc3ccc(Br)cc3Br)CC2)c(F)cc1Cl C1(C(N(CCCC)CCO)=O)C=CCN1C(=O)CCc1ccn(C)n1 N1(C(CC2CC3(CN(C(COCC(=C)C)=O)C3)C2)=O)CC(CO)C2(CCC2)C1 c1(OC)ncc(Cl)c(=NC2CCCCC2CNC(C2(C)CC(F)(F)C2)=O)[nH]1 C1(CNC(=O)NC(C)CC(O)c2ccco2)CCN(C2CCCC2)CC1 N1(C(C2(C(=O)NC)CC2)=O)CCOC(CCCNC(=O)C)C1.C1CCCCO1 c1(C(N2CCCC3C(C2)C3)=O)c[nH]c2nccc(Cl)c12.C1(C(=O)N)(SCC)CC1 C1(C(N2CC(CC)OCC2)=O)C2CCC1CN(C(c1ccc(C)cc1C)=O)C2 c1(C(=O)NC(CCCNC(C=Cc2c(C)cccc2)=O)C)ncc2[nH]ncc2n1 c1(NC2C(CNC(C=COCC)=O)CCC2)ncc(C(C)(C)O)cn1 C(=O)(C(=O)NC1(CNC(=O)C(C)O)CCC1)NCC c1(C(=O)NC(C2CCN(C(C(CC)C)=O)CC2)C)c(C)c(Cl)cc(C)c1N C(CCN(C)C(C1CCCCC1O)=O)(C(C)(C)C)NC(c1c(C)ccnn1)=O c1(CN2C(C(=O)NC(c3ccc(Br)cc3)CO)COCC2)cc(Cl)cc(Br)c1O n1(COC)ccc(C(=O)NCC2(NC(=O)C(Cl)=CCl)CCOC2)n1 C(CC(=O)N1CCCC(CCNC(C2C3CCC2CC3)=O)C1)(C(C)C)OCC CC(N)(CC(=O)N1CCCC(N2CCOCC2)CC1)C(F)F c1(C(=O)NC2C(NC(=O)CCCCn3ccnn3)CC2)ccc2cccnn12 c1(OCC)cncc(N2CCC(C(=O)OC)(C(F)F)C2)n1 C1(NC(c2ccc(=NC)[nH]c2)=O)C(C)(C)C(NC(c2cnn[nH]2)=O)C1(C)C c1(CNC(C2(SC)CN(C(COC(CC)C)=O)C2)=O)cc2ccccc2[nH]1 c1(NC(C)CC(C)(C)C)ccc(S(=O)(=O)N(C2CSC2)C)cc1C#N N1(C(Cc2cc(CC)no2)=O)CC(NC(=O)C=Cc2ccnn2C)C2(CCC2)C1 Cc1cc(Cl)c(C(=O)NCCCOCC)cc1F.C1(CC=O)CCCC(C)C1.N N1(CC(F)F)CCCCC1Cc1ncc(Br)cn1 C(=O)(C1CCc2scnc21)N1CCN(C(C2CCCC2O)=O)CC1 c1(OC)ccc(C(N2CC3CC3(NC(=O)C=Cc3cnc[nH]3)C2)=O)cn1 CC1(C)CCCCN(C(=O)C=CCNC(C2C3CCC(=O)C23)=O)C1 N1(C(c2ccc(O)nc2)=O)CCC2C(CCN2Cc2cc(Cl)cc(Br)c2)C1 CC(C)CC(O)CC(=O)NCCN(C)C(c1cc2c([nH]1)CCCC2)=O c1(C(N2C(CNC(c3cnc(SC)s3)=O)CC2)=O)c(F)cc(O)cc1F N1(C(Cn2ncc(C)c2)=O)CC(C2CN(C(=O)CN=S(C)(C)=O)C2)C1 c1(NC(C(C2CCN(Cc3cscn3)CC2)C)=O)c(Cl)ccc2c1OCO2 N1(C(C2C(CC)CCCC2)=O)CCC2(CCC(NC(C3(F)CC3)=O)C2)C1 C1(O)(C(=O)OCC(C(C)(C)C#N)=O)CCc2ccccc2C1 c1(C2C(N(C(C=C(CCC)CCC)=O)CC)C2)ccc2c(c1)OCCO2 c1(C(N(CC(C)NC(=O)CCn2cnc(=N)[nH]2)C)=O)ncncc1Cl C1(NC(C(CCC#C)O)=O)CN(C(c2cccc(OC)c2C)=O)C2(CCC2)C1 N1(C(CC2C(C)CCN(C(c3cccc(O)n3)=O)C2)=O)CC2CC(C1)N(C)C2 N1(C(CCN(C)CCO)=O)CCC(CN(C)C(C23COC(CF)(C2)C3)=O)CC1 C1(CC=O)CCOCC1(C)C.c1(N(C)C)ccnc(C(=O)NCC2CCC2)c1.N N1(C(CCCNC(c2c(C#C)c[nH]n2)=O)=O)CC2CCC1C(O)C2O C#Cc1ccc(C(N2CC3(CC3)CC2CNC(=O)Cc2ccsc2)=O)cc1.O N1(C(CC=CC)=O)CC(OC)CC(NC(=O)COCCCC(C)C)C1 C1(C#N)(C(=O)Nc2[nH]nc(CC)n2)CC12CCC2 N1(C(Cc2c(C(C)C)con2)=O)CC2C(C)C2C1.C(c1ccnn1C)=CC(=O)N C1(C)(CNC(C2(CC#C)CCC2)=O)CCN(C(=O)CCC(C)C)C1 c1(C(=O)OC)ccoc1C(=O)NCCCC1CCCN1C(c1ccco1)=O.C C1(CC(=O)NCc2nc3ccccn3n2)CCCC12CN(C(=O)CO)C2 c1(C(C(=O)NCCN(C(c2ccc(C#C)o2)=O)C)C)ccc(S(C)(=O)=O)cc1 O=C1CC(C(=O)NC2CC2NC(c2ccc(-c3ccccc3)s2)=O)CCN1 c1(OCC(=O)NCC2(CNC(C(C=C)O)=O)CC2)ccc(F)cn1 c1(C(=O)OCC)nc(=NC(C)c2ccc(Br)cc2Br)[nH]o1 C1(C(=O)OC)CCN(C(=O)CCn2c(C(=O)OC)nnc2)C1C(=O)OC c1(NC(C2CCN(C(C(C=C)O)=O)C2)C)[nH]c(=O)n(C)c(=O)c1C#N C(=O)(C(C)CC(N)=O)N(C(C)C)CCNC(=O)CCN1CCCCC1 N1(C(C2(CC)CC2(F)F)=O)CC=C(CCNC(=O)CNc2nccs2)CC1 c1(N2CC(C)(C)C(NC(=O)CN3CCCCC3)CC2)ncc2cc(Br)ccc2n1 Cc1ccc(-n2nc(C3CCOC3)nc2COCc2ccncc2)c(C)c1 c1(C(=O)Nc2n(CC)ncc2)cccc2[nH]nc(C3=CCC(C(F)(F)F)CC3)c12 c1(Cc2n(-c3cc(C)ncc3)nc(CC(F)(F)F)n2)cnc2sc(C)c(C)n12 CCCC(O)C(=O)NC1CCC1NC(c1csc(-c2ccoc2)n1)=O C1(NC(C=C(C)C(C)C)=O)CS(=O)(=O)CC1NC(C1(F)CCCC1)=O CC(C)C(O)(C(=O)N1CCCC(C)C1)C(F)(F)F.C(=O)C(C)C.[SH](C)(=O)=O c1(C(=O)NC(C(N2CC(F)(COC)C2)=O)C2CC2)cnc2c(Br)cccn12 C1(NC(c2ccc(O)cc2)=O)CC2CCC1N(CCNC(=O)C1CC1)C2 C1(c2nnnn2C(C)C(=O)OC)(NCCSCC=C)CCC(C)(O)CC1 N1(C(C23CC(C(=O)C4CC4)(C2)C3)=O)CCCC(C)C1.C(=O)CC.CC.N c1(-c2scc(C(=O)NC(C)CNC(c3csnc3Cl)=O)n2)ccc(O)cc1 C1(C(=O)NCc2c(OCC)cccc2)CC2(CCC2OC)C1 CC1(C(=O)NCC2CN(C(c3cccc(Cl)c3)=O)CC2O)CCNC(=O)C1 C(CCCC(=O)N(C)CC1(O)CCN(C(c2cnc(C(N)=O)cn2)=O)C1)N(C)C C=CCC(CC(C)C)C(=O)N1CCC(C)C(CNC(=O)CCC(C)N(C)C)C1 C1COCCN1C(c1ccccn1)=O.C(=O)(C(F)=C1CCC1)N(C)C.C(N)=O N1(C(C2(CC(C)=O)CC2)=O)CCCC(CC(=O)NC23CCC(CC2)C3)CC1 N1(C(c2c(OCC)ccs2)=O)CCN(C(C2CCCCN2C(=O)CCF)=O)CC1 CCCCC(O)CC(=O)N(CCCCN(C)C(c1ccc(OC)cc1OC)=O)C n1(CC)c(C)cc(C(=O)NCC2COCC2)c1C.c1(CCC=O)cnc(O)[nH]1 n1(CC)cc(C(N2CC(C(=O)NC(C)C(F)F)C(C(C)C)C2)=O)c(C)n1 c1(C(=O)NC2CN(C(C3(C)CC(F)C3)=O)CC2C(F)F)ccc(F)cc1N S(=O)(=O)(c1cccnc1NCC1(CCO)CCCC1)NC(c1ccccc1)C c1(C(N(C2CC2)C)=O)ccc2c(c1)CNC(=O)N2.N1(C(CSC)=O)CCCC1 C(C(C(C)C(C)C)NC(=O)CCc1ccccc1F)NC(CC1CC(=C)C1)=O N1(C(Cn2nnc(C)n2)=O)CC(CNC(C2(F)CCCN(C)C2)=O)CC12CCC2 N1(C(c2n(CCC)ccn2)C(=O)NC2CC2)CCCC(c2noc(C(C)C)n2)C1 c1(C(=O)N)cccc(C#CCO)c1.C1(CNC(C2C(OC)CC2)=O)CCCCC1 C1(NC(C2C3CC4C(C3)C24)=O)CN(C(C2(C(F)(F)F)CCC2)=O)CCC1 c1(C(C=O)C)cccc(Cl)c1.C1(C(=O)N)(COC)CCCC1.C(C)C1CCC1 c1(OC(C)C)cccc(CC(=O)N(CCC)C)c1.C(=O)(C[SH](=O)=O)N.C1CC1 N1(C(C2Cc3n(cc(C)n3)C2)=O)CC2CCCN(C(=O)COc3ccon3)C2C1 c1(CC(=O)NC2CCCC2)ccccc1C(C)C.C(=O)(C)NCCOC CC(C)C(O)CC(=O)N1CCC(C)(CNC(=O)C)C1.c1(C=O)cccc(O)c1 CC1CC(NC(c2c(Br)cnn2C)=O)CN(C(=O)CC2C(C)(C)C2(C)C)C1 N1(C(C2(CCCC)CC2)=O)CC2(CNC(=O)Cc3cc(C)no3)CC1CO2 C1(Cc2cn(-c3nccc(NC(=O)CC4CCCC4)c3)nn2)CC2CCC1CC2 Cc1cc(NC(=O)CC2C(NC(=O)C(C(C)C)C3CCC3)CC2O)cnc1C C(C)(CCCN=c1[nH]c(Cl)ncc1[N+](=O)[O-])NC(C1(C=C)CCC1)=O C=CCC(CC=C)NC(c1cc(-c2ccccc2)nn1C)c1nnnn1CC Cc1cccc(CNC(C2(F)CN(C(=O)C(=O)NC3CC3)C2)=O)c1 c1(CC=O)ccc(C#N)cc1.Cc1coc(C(C)C)c1C(=O)NC1CC(C)C1 C1(C(=O)NC(C)(C)CCCNC(=O)Cc2cnccn2)CCCC(F)(F)C1 c1(NC(C2(NC(=O)COC(F)(F)F)CCC2)=O)cc(O)nc(O)n1 CC1CC(C)(C(=O)NCC(C)(O)CNC(=O)CC2CCSC2)CCO1 C1(CCNC(c2cc(F)n[nH]2)=O)(OC)CN(C(C2CCS2(=O)=O)=O)C1 Cc1nc(C)c(C)c(=NCCCN(C)C(C2(S(C)(=O)=O)CCCC2)=O)[nH]1 C1(N(C(CC)CO)Cc2cc(Cl)ccc2Cl)CCCN(C)C1=O C1CCCCCN1C(=O)CC1CC1.c1(OC)ccccc1C1(C(=O)N)CCC1.C C=CC(C)(CC)C(=O)NCCn1cc(C(=O)NC2CC(n3cccn3)C2)cn1 c1(C(N2CCC(CC=C)(NC(c3ccoc3)=O)C2)=O)cc2cc(N)ccc2o1 CC(O)C(C)C(=O)NCC1CCCN(C(c2ccc(CO)nc2)=O)C1 CCCC(C)(C)CC(=O)N(C(C)C(=O)NCCCCCCO)C CC1CCC(O)CN1C(C1(CNC(=O)C=CC2(C)COC2)CCC1)=O c1ccc(F)c(Cl)c1.C1(N(C(=O)CC)C)CCCN(C(=O)C=CC2CC2)CC1.O c1(COC)cccnc1C(=O)NC(C1CN(C(c2c[nH]c(=N)s2)=O)CCO1)C N1(C(C)=O)CCOCC1C(=O)NC1CC(C)C1.C(=O)C(C)(C)C1CCOC1.N N1(C(C(N2CC(C)C2)C)=O)Cc2[nH]nc(C(=O)NCCN3CCNC3=O)c2C1 c1(C(N2C(CNC(C(C)(C)c3ccccc3)=O)CCCC2)=O)cc(O)ccc1F C1(C=O)C(C)(C)C1(C)C.c1(C(NC(C)C)=O)ccc(C2CCOC2)s1.CC N1(C(CN(C(C)=O)C)=O)CC2CCC1C1CN(c3ccc(S(C)(=O)=O)cn3)CC21 CCCC(C)(CCC)C(=O)NCC(C(C)C)NC(c1ccncc1OC)=O n1(CC)ncc(C(=O)N(C(C)CN(C)C(c2ccnn2CC(F)F)=O)C)n1 C1(C(=O)NCC2C(CNC(C3(C#C)CC3)=O)C2)CCCNS1(=O)=O c1(C(=O)NC2CC(NC(c3cc(C)nn3C(F)F)=O)C2)cccc(N)c1Br c1(C(N2C(CC=O)CCC2)=O)ccc(O)c(F)c1.c1(C(=O)O)ccc[nH]1.CC C1(CNC(=O)C#CC2CC2)CC(NC(=O)CCCN2CCOCC2)C12CCC2 c1(C(=O)NCCNC(c2cc(C(=O)OC)nn2C)=O)cc2cccnc2[nH]1 C1(NC(CCC(=O)OC)=O)CCCC2CN(C(=O)C(F)C(C)C)CC12 c1(C=O)cc(C)n(C(C)(C)C)n1.C(C)(C(=O)NC)OCCCC.C1CC1 c1(C(=O)NC(CC(C)NC(COC(C)=O)=O)C)cnn2c(C)ccnc12 c1(C(N(C)CC2(NC(c3cc(C(CC)C)no3)=O)CC2)=O)c(C)cnn1C C1(C(=O)NC(CC)CCOC)COCCN(C(=O)Cc2ccc(F)cc2Cl)C1 Cc1cn(C)cc1C(N1CCC(CCO)CC1)=O.C(=O)(C(C)C)N(CC=O)C.N CCC(CNC(c1cc(C)ccc1C)=O)(CC)C(=O)NCC.C1(N)CC1(F)F CCCCCCC(C)CC(=O)NC(C)CCCNC(C1(C)CC(O)CN1C)=O C(c1ncc[nH]1)=CC(=O)N(CCC)CC.c1(C(=O)N)cnc(C(F)F)nc1 c1(C(=O)NC2CN(C(C3N(C)C(=O)NC3)=O)C(CO)C2)c(Cl)oc2ccccc12 Cc1ccc(F)c(C(=O)NC2CC2NC(=O)CCc2c(C)nc(O)nc2O)c1F C(C(C(C)(C)C)NC(=O)Cc1c[nH]ccc1=O)NC(CCOC(CC(C)C)C)=O S(=O)(=O)(CC(=O)NCC(F)(F)Cn1cc(C=O)nn1)NC.c1ccccc1.N C1(CNC(c2c(OC)scc2)=O)C(C)CCN1C(=O)CCS.c1nnnn1C C1CCN(C(=O)CN(C)C(N)=O)CC1.C1(C(=O)NCC(N)=O)CCCO1.C C1(C(=O)NCCCC(C)NC(=O)CC2CC(OC)C2)(OCC)CCCC1 c1(OC)ccc(OCC(=O)NC(c2ncc(Cl)cc2Cl)C)cc1C N1(C(C(C)=C(CC)C)=O)CC2(C=C(C(=O)N(C3(c4cc[nH]n4)CC3)C)CO2)C1 C1(CNC(c2c(Br)n[nH]c2Br)c2n(CCCOC)nnn2)CCCCCCC1 N1(C(c2ncn(C)c2)=O)CC2CN(C(=O)COCC3CC3)CC2(C)C1 Cc1cc(O)nc(C)c1C(N1CCCC(C)CC1)=O.C1(C=O)C(F)(F)C12CC2.N N1(C(C(COC)C)=O)CC2CCC1C2NC(c1ccc(C(C)C)c(Cl)c1)=O C1(C(=O)NCCCCCNC(c2scc(OC)c2)=O)CCC(=O)CC1(C)C C(=O)(C(C)CC(C)C)N1C(CC)C(C(=O)N(CC(C)(C)N(C)C)C)CC1 N1(C(CC(CNC(=O)CN2CCNC2=O)OC)=O)CC2CC(OCCO)C2C1 C1(C2=CCCCCC2)C(=O)NCSC2CCCN12.n1(CC)cc(C(=O)O)c(C)n1 c1(C(N2CC(C)N(C(=O)C=C3CC3)CC2)=O)c(F)ccc(OC(F)(F)F)c1N C12(CNC(c3ncn(C)c3)=O)CC1CN(C(c1ccc(-n3cncn3)nc1)=O)C2 C1(NC(C2C(C#N)C2)=O)CCCN(C(C2(CC(F)F)CCOCC2)=O)CC1 Cn1cnc(C(N2CC3CCC3(CC(N3CCOCC3C(N)=O)=O)C2)=O)cc1=O n1(CC)nc(C(=O)N)cc1O.c1(C(N2CC(O)C2)=O)cc(C(C)=O)cn1C.C N1(C(C2(O)CCC(CC)C2)=O)CC[Si]2(CCCC2)CC1 C1(CNC(C2C(C)OCC2)=O)CN(C(=O)C=Cc2cncs2)CCCO1 C(CCC(C)(C)C)NC(c1cc(C)[nH]n1)=O.c1(C(=O)N)sc(C)cc1OC(F)F C1(C(N2CCN(CCN(C)C)CC2)=O)COCCN(CCN2CCCCC2)C1 CCC(CC(=O)NCCOCCOCC)C(C)C.C(=O)C1=NNC(=O)C1.N C1(C(CN2C(NC(C(=O)N(CC(F)F)C)=O)CCCC2)=O)CC2(CCOCC2)C1 N1(C(c2c(OC)nc(C)cc2)=O)CCC2(CCN(Cc3cn(C)cn3)C2)C1 C#CCC(O)C(=O)N(CCC(=O)N1CC(NC(=O)NC)C1)C c1(NC(COC2CCN(C(C3CC(C#N)(OC)C3)=O)C2)=O)c[nH]c2cccnc12 CCCCC(O)C(C)C(=O)N1CCCC1CC(=O)N(CC(=O)N(C)C)C C(=O)(C1=NOC(C)(C)C1)N1C(C)CCC1.Cc1noc(C)c1C(C)C(=O)NC c1(C(=O)NCC(CCC)NC(c2cscn2)=O)cnc2ncccn12 Cc1nccc(CCC(=O)NCC(CO)NC(c2ccccc2NC(N)=O)=O)n1 C1(NC(NCC(C)(C)SC)=NCC2CCCCC2)Cc2ccccc2C1 c1(C(=O)NCC23C(CN(C(C=C(C)C)=O)C2)C3)cnc2cnc(Cl)cc2c1 N1(C(C2CNC(=O)O2)=O)CCCN(CCc2cn(CCO)nn2)CC1 N1(C(CCSCCCC)=O)C2CCC1CC(N(C(=O)C(F)CC)C)C2 C1(C(=O)NC(C(NOCC(N)=O)=O)c2ccccc2)CC(=O)C12CCC2 C(C(C(C)C(C)C)NC(=O)Cc1ccsn1)NC(Cn1c(C)csc1=O)=O c1(C(=O)NC2CCCCCCC2)ccc2cncc(Br)c2n1 N1(C(Cc2nc(C)[nH]n2)=O)CCCCC(N(C(=O)C(c2ccc(F)cc2)C)C)C1 C1(CC)OCCC1N=c1cccc(S(=O)(=O)N2CC(O)CC2C2CCCCC2)[nH]1 N1(C(C2CN(C(CCC3C(C)(C)C3)=O)CC2(F)F)=O)CCC(O)C(C)(O)C1 C1(NC(c2cc(C(CC)C)no2)=O)COC2(C1)CN(C(=O)CC1(C)CCC1)C2 c1(C(N2CCC(O)C2)=O)cccc([N+](=O)[O-])c1.C=C1CC1C(=O)N.C(C)C N1(C(C(C=CCCC)O)=O)CCc2sccc2C1CNC(=O)CSC N1(C(C(C)N(C)C)=O)CCN(C(c2ncccc2O)=O)CC1C1CCC1 C1(C)(C(=O)NC2CCN(CCC)C2)C=CCN1C(=O)Cc1sccc1C C1(C)(OC)CC2CC1CC2NC1CCOC(C2CC2)C1 c1(C(=O)NC2C(CC)CN(C(=O)C(F)(F)C(F)F)CC2)ccc(OC)c(F)c1F c1(C(=O)NCCCN(C)C(C2CCCC2)=O)cc(C(N)=O)cs1.N1CCCC1 Cc1cc(-n2cc(C(=O)NC3CCN(C(C4CCCC4)=O)CC3)nn2)cc(=O)o1 CCCCC(C(=O)NCC1CC(C)CCN1C(=O)C)C(C)C.[SH](=O)(=O)C1CC1 N1(C(c2c(C)noc2N)=O)CCC2(CC1)CC2NC(c1cnn(C)c1C)=O CC1(C)CC(O)(CC(N2CC(OCCNC(=O)CC)C2)=O)CO1.C(=O)CO C1(CN(C)C(c2cn[nH]c2)=O)CCN(C(C2(O)CCC2)=O)CC1.C1CCOC1.C CC(C)C(C)C(=O)N1CCCC1CN(C)C(c1c[nH]nn1)=O N1(C(C(C(C)C)F)=O)CCC2CCC(NC(=O)C=Cc3cn(C)cn3)C1C2 N1(C(C=CSC)=O)CCCC(CO)(NC(=O)CC2SC(=N)NC2=O)C1 c1(OC)ccc2c(c1)C(NS(=O)(=O)c1ccc(F)cc1CN(C)C)C(=O)N2 N1(C(c2scc(CC)n2)=O)CC2CN(C(c3csc(C)c3C)=O)CC12 C1(NC(Cc2cccc(CC)c2)=O)CC(O)CN(C(c2cccc(=O)n2C)=O)C1 Cc1cccc(Cn2nc(Cn3cccn3)nc2-c2coc(-c3ccccc3)n2)n1 N1(C(C(CC(=C)Cl)NC(C2COCC2(C)C)=O)=O)CCC(C2CCC2)C1 CC1CCOC(C(=O)NCCC2(O)CCN(C(C3(CF)CCC3)=O)C2)C1 Cc1c(NC2CCCCC2)ncnc1N1CCCC(N2CCCC2)CC1 c1(C(=O)NC2CCC(NC(C(CC)C#N)=O)CC2)cc(S(N)(=O)=O)sc1C N1(C(c2c(OC)csc2)=O)CC(C)(C)CC1C.C12(C=O)CC(C)(C1)OC2C C(C(=O)NC1(C(=O)NC2CON(CC)C2=O)CC1(C)C)(C(C)C)OCC CCC(C)(C(=O)NC1CC1NC(c1cc(Cl)ccc1OC)=O)C(N)=O c1(C(=O)NCC(CCNC(CCc2n(C)cnc2)=O)O)cnncc1C(F)(F)F N1(CCCCNC(CCOCC#C)=O)CCCN(C(=O)C=CC(C)(C)C)CC1 C1(NC(CC2(CNC(CC3(OC)CCC3)=O)CC2)=O)CC2CCC1O2 C1(NC(CC2C(C)CCO2)=O)CCCC2CN(C(C3CCCC(C)C3)=O)CC12 Cc1ncc(C#N)c(N2CCC23CN(C(c2c[nH]cc2C)=O)C3)n1 C1(COC)CN(C(C23CCC(C2)C3(C)C)=O)CCN1C(=O)CC.CC(C)C.O c1(C(=O)NC(CNC(C2(C)CCN(C)C2=O)=O)(C)CO)cc2cc(O)ccc2[nH]1 c1(C(C)O)ncc(C(=O)NC2CCC(C)C2)s1.C12(C(=O)N)CC(F)(C1)C2 Cc1cccc([N+](=O)[O-])c1C(N1CC=CC1C(=O)Nc1cccc(Br)c1O)=O C1(NC(C2CC(=C3CCC3)C2)=O)CN(C(c2n[nH]cc2Cl)=O)CC1C1CC1 N1(C(=O)OC)CCC(NC(=NCC2CC(SC)C2)NCC2CCOC2)CC1 Cc1cc(C)c(C(=O)NC2CC(NC(=O)Cc3ncccc3C)CC2O)cn1 Cc1cc(C(=O)NCCC(C)N(C(=O)CC2COCC2O)C)cc(N)c1O N(C(=NCCC(C)=O)NCC1CCCN(C)C1c1cnn(C)c1)CC(F)=C(C)C c1(C(N2CC3CC(NC(=O)C=C4CCCC4)CC3C2)=O)ccc2ccncc2c1 c1(C(=O)NC2CC(C)(NC(=O)Cc3cccs3)C2)n[nH]c2ccc(Cl)cc12 C1(C(=O)NC)(CN2CCCCC2)CCN(S(=O)(=O)N2CCCC(C)C2)C1 C(C)(CC(C)NC(c1[nH]nnc1C)=O)NC(C1C(C)(CC)C1)=O c1(C(=O)NCC(CNC(C(C)OC(C)(C)C)=O)F)ccnc(N(C)C)c1 Cc1c(Cl)ccnc1C(N1CCC(NC(=O)CSS(C)(=O)=O)C1C1CC1)=O Cc1cccc(C(=O)NC(CCF)C(=O)NC(C)CC2CCC2)n1 c1(NC2CN(CC)C2)cc(N2CCCC(C(C)O)C2)nc(C)n1 C=C(F)C1(CC(=O)NCC2CCCN2C(=O)C(c2ccccc2)F)CCC1 N1(C(c2cc(C)oc2)=O)CCCC2C1CCCN2C(c1cnc2cc[nH]c2c1)=O C1(NC(c2c(CC)ncs2)=O)CCCCC1C(=O)NCC1CC2CCC1O2 C(=O)(C(C)CC(C)CC)NCCOCCCNC(C1CCC(CCCC)CC1)=O C1(C(=O)NCC2(CC)CC2)CCN(C=O)C12COC2.C(C)(C)C.CS C(=O)(NNc1ccc(Cl)c(Br)c1)Nc1c(CN2C3CN(C)C(C3)C2)cccc1 c1(C(=O)NCC(CSc2c(OC)cccc2)C)ccn2nnnc2c1 C(C1=NOC2COCC12)(c1n(CCC)nnn1)Nc1ccc2nc(CC)sc2c1 C1(C(N(CC(CC)OC)C)=O)CC(F)CCN1C(=O)C=Cc1ccc(C)o1 N1(C(C23CC4CC2C3C4)=O)CCC(O)CC(C)(C)C1.n1(CC)nccc1C=O c1(NC(C2N(Cc3ccc(C#N)s3)CCNC2)=O)ccc(Br)cc1C(N)=O N1(C(=O)OC(C)(C)C)CC2(CC(NCc3ncc(Cl)cc3F)c3nccn32)C1 N1(C(C(C)=CC2CC2)=O)CCc2ccccc2C1CNC(C1CCCO1)=O CC1CC=C(C(=O)N2C3CCC2CN(C(C24CCCC(CO2)C4)=O)C3)CC1 c1(CC)ncc(C(=O)N(CCCNC(=O)C(c2nc(C)cs2)C)CCO)[nH]1 C=CC1(C(=O)NCC2CCN(C(c3cc(=N)[nH]n3C)=O)CC2C)CCOCC1 c1(C(C)C)n[nH]cc1C(c1nnnn1C1(C)CC1)NC1(C)CC(F)C1 N1(C(Cc2cccc(OC)c2)=O)CC(NC(c2cccc(O)c2C)=O)CC(O)C1 C1(CNC(CSC)=O)CN(C(=O)C(c2cccnc2)O)CCC1(C)C C(=O)C1=C(Cl)CCC1.N1(CC=CC(=O)NC(C2CC2)C)CCCCC1.C c1(C(N(CC(C)NC(=O)CC)CC)=O)ccc2cc(Br)ccc2n1.C(N)=O.N C#Cc1ccnc(C(=O)NCCOCCC(=O)NCCCN(C)OC)c1 N1(C(c2cc(CC)no2)=O)CC(CNC(c2ccc(OC)o2)=O)C(C)(C)C1 C#CCC(C)(CC)C(=O)NCC1(O)CCCN(C(C2(CC)CCCCC2)=O)C1 c1(NS(C)(=O)=O)ccc(C=O)c(Cl)c1.C1(C)(C(N2CCC2)=O)CC2CC2C1 c1(CN(C(=O)C(O)C2CN(C(C3CC(N(C)C)C3)=O)C2)C)ccncc1 N1(c2nccc(C(=O)OC)n2)CCC(NC(=O)CC2CC=CCC2)C(O)C1 C12(C(=O)NC3CC4CC(N)C4C3)CC1COC21CCC1 C=CCC(CC)C(=O)NCC1C=CCN1C(=O)CS(=O)(=O)NCC C(C(C)(C)CC(=O)NCc1noc(C2CC2)n1)NC(C(c1ccc(C)o1)C)=O c1(SC)nn(C)cc1C(=O)Nc1ccnc(-c2ccc(Br)cn2)n1 C(=O)C(=O)C(C)(C)C.C(C)(CC(C)C)NC(COCc1onc(C)n1)=O.N N1(C(C2(C(C)(C)C)CCC2)=O)CCC(CC)CC1.c1(C=O)cc(C(F)F)on1.N Cc1cc(C(=O)N(CC(O)CNC(=O)Cn2nnc(-c3cccs3)n2)C)cn1C c1(NC)cnccc1C(=O)NC1CN(C(c2ccnc(OC)c2)=O)C1 C=C1CCN(C(c2ccc(F)c(C)c2)=O)C(C(=O)NCCn2ccccc2=O)C1 c1(C(=O)NCCN(C(C2(CC)CCCO2)=O)C)ccc(C)c(F)c1 n1(C(C)C)nnc(C=O)c1C(F)(F)F.c1(C(N2CC(CC)C2)=O)cn(C)nn1 C1(NC(c2ccc(S(C)(=O)=O)[nH]2)=O)CCN(c2ccnc(C3CC3)n2)C12CCCC2 c1(OC)ccccc1C(C)C.C1(CCNC(=O)CC(C)F)CO1 C(C(C)C(=O)N1CCCC1C(C)NC(=O)CSCCC(C)C)OC N#Cc1ccc(C(N2CCCC2)CNC(C2COCCN2)=O)nc1 N1(C(c2c(-c3onc(C)n3)cccc2)=O)CCc2cc(C(F)(F)F)ccc21 C1(C(=O)O)C2CCN(C(=O)CN3CCC(O)CC3)CC12 CC1C(C)N(C(c2cnc(Br)s2)=O)CCN1C(=O)Cn1nnc(=O)[nH]1 c1(C(=O)Nc2nccc(C)c2C#N)cccc2c1NC(=O)CC2 Cc1cc(C(=O)NCCC(C)CCNC(C2CC3(CCC3)C2)=O)ccn1 N#CC1CCC(C(N2CCC2Cn2cc(-c3ccc(C(F)(F)F)cc3)nn2)=O)C1 C=CCN=c1[nH]c(C(=O)OCc2ccc(C#N)cn2)cs1 N1(C(C2(C#N)CC2)=O)CC23CCCCC2(C1)CN(C(=O)CC1CCC=CCC1)C3 c1(C=O)cc(S(N)(=O)=O)c[nH]1.C(C(=O)NC)(C(C)C)SC.C1(O)CCC1 N1(C(c2ccc(CCF)cc2)=O)CC2(CCN2C(c2ccc(F)c(F)c2)=O)C1 S(=O)(=O)(c1ccc2nc(N3CCC4(CCCCO4)C3)sc2c1)N(C(CSC)C)C C(=O)(C(F)(F)C(F)(F)C(F)F)N(C)CC.C(=O)(C#CC1(C)COC1)NCC C1(NC(C(C)=C2CC2)=O)CC2CCC(C1F)N2C(=O)C(C)(Cl)Cl c1(C(=O)NC)ccc(O)cc1.C1(C=O)CC(=O)N(c2cn[nH]c2)C1.C1CCC1 CCC(CC)CCCC(=O)N1CCC2CC12C(=O)NC(c1cncc(F)c1)C C1(CC=C)(C(=O)NCCOCCC(=O)NC(CO)CCC)CCCC1 c1(C(=O)NC(C)COCC2CCC2)ccccc1CCC(F)F CCC(CC(=O)NC1(COC)CN(C(=O)CN(C2CCC2)C)C1)C1CCC1 Cc1cccc(C(=O)NC(C)CCCCNc2cnc(C#N)cn2)c1F CC(C(=O)NC1CCN(C(=O)COC(F)F)CC1)S(=O)(=O)c1ccc(F)cc1 c1(C(N(C2CC3CCC(C2)N3C(=O)C(C)(O)C2CC2)C)=O)occ2c1CCOC2 C1(N(CC(CC)C)C)CCN(C(c2cc(-c3cccs3)cs2)C(=O)NC(C)C)C1 C(CCC)(C(=O)N1CCC(CCC(=O)N(CC)CC2(O)CCC2)C1)=CCC Cc1cc(F)ccc1CC(=O)NCC1CN(C(=O)CCC(F)(F)F)C2CC12 c1(OC)cc(NC(C2CC23CN(C)C3)=O)cc(C#N)c1.c1ccc(N(C)C)cc1 C(C)(C(=O)N=c1[nH][nH]c2c1CN(Cc1ncc[nH]1)C2)c1c(C)n[nH]c1C C1(F)(CNC(c2c(C)ncnc2)=O)CC2CCC(C1)N2C(=O)C#CC1(C)COC1 c1(C(N2CCCC(C(C)(F)F)C2)C(=O)NC2(C)CC2)ccc(O)c(F)c1 c1(CC(=O)NC(CNC(CC2CC(C(=O)OC)C2)=O)CO)ccc(Cl)s1 N1(C(C(Cc2cnc[nH]2)NC(c2ccc(=N)[nH]n2)=O)=O)CC(=O)N2CCCC2C1 O=C1Cc2c(C(N3CCCC3C3(NC(C4CC4[N+](=O)[O-])=O)CC3)=O)cccc2N1 n1(CC)ccc(C(N2CCC(CCC(=O)NCC3CC34CC4(F)F)C2)=O)c1C N1(C(C)C)CC(C(N2CC3(CC3C(=O)NC3CSC3)C2)=O)CC1=O C(=O)(C(O)C(C)(C)CC)N1CCC(CNC(CCCCOCC)=O)C(C)C1 O=C(CCCCCF)NC1C2CCN(C(=O)CCOc3cccc(Br)c3)C12 C=CCC(C)(C)CC(=O)N(C1CCN(C(c2cc(N)cc(F)c2)=O)CC1)CC Cc1c([N+](=O)[O-])c(C(N2CCC(NC(=O)CCO)C(C)C2)=O)nn1C.CC(C)C Cc1nc2c(-c3nc(C(F)F)nn3-c3ccc(F)c(Cl)c3)ccnc2[nH]1 C(C(C)C(C)C(=O)N1CCN(C(=O)CN(C(=O)C)C)CC1)OC.c1cccs1.S C(C)(CC(=O)N1CC2C(N(C)C(c3ccsn3)=O)C2C1)(C(F)F)N(C)C C(=O)(C(F)CC(C)(C)C)N(C1CN(C(CCC(CC)C)=O)CC1(C)C)C Cc1cnn(C)c1C(N1CCC(CCC(=O)N(CC(F)F)CC(C)O)CC1)=O c1(C(N2CC3C(NC(C(C)c4ccco4)=O)(C3)C2)=O)coc(S(N)(=O)=O)c1 C(=O)(C(C(C)(C)O)NC(=O)C(n1cc(C)cn1)C)NC1C(C=C)COC1 c1ccc(C(c2cn(CCC(C)(C)C)nn2)(C)C)cc1.C(C)(C)(C)N(C(C)C)C c1(C(=O)NC(CCNC(c2c(CC)nc[nH]2)=O)C)cc2cc(Cl)ccc2s1 c1(NC(c2c(C)nns2)C)cc(S(=O)(=O)NC)ccc1C#N.C1(C2CC2)CCC1 C=CC(C)C(=O)NCCCC(=O)NC(C(C)C)C1CCC1 C1(CC=O)COC(C)(C)CO1.c1(CC)occc1C(=O)NC.C1CC(F)C1 N1(c2ccc(C)cc2)CCCC(c2nn[nH]n2)C1=O.N12CCN(CC1)CCCC2 CCC(CC)CC(=O)N1CCC(CCNC(=O)C(C)C2CCCC2)C1 C12(NC(=O)CC3CC4(CC4)C3)CCC(CC1n1cc(CO)nn1)C2 C1(C)(C=O)CCC(C)=C(C)C1.C1(C(=O)NC2CCCCC2)(OC)CCCCC1.N C(=O)(CC(F)(F)C(F)(F)F)N1C(CCNC(c2c[nH]cc(C)c2=O)=O)CSCC1 C1(OC)CN(C(C2CCCN(C(=O)CSC(F)F)C2)=O)CC12CC2 C(=O)(NN1CCCC1C(=O)NCCCC(=O)OC)c1c(CC)cccc1 CCN=c1[nH]c(C(=O)N(CC(C)NC(c2ccc(OC3CC3)cc2)=O)C)cs1 C1(C(C)NC(C(=C(C)C2CC2)F)=O)CN(C(c2ccnc(C)n2)=O)CCO1 c1(CC(=O)NCCC(C)N(C(C2N(CC)CCC2)=O)C)ccccc1C N1(C(c2c(SC)cccc2)=O)CC(CNC(c2cccn(C)c2=O)=O)CCC1C C(=O)(CC(C)C(=O)N1CCN(CCNC(c2c(OC)ccnc2F)=O)CC1)OC C1(NC(Cc2nc(C)[nH]n2)=O)CC2CCCC(C1)N2C(C1CCC2CC2CC1)=O c1(C(=O)N)cnc2c([N+](=O)[O-])cnn2c1.N1(C(C(C)OCC)=O)CCCC12CC2 C1(CNC(CCOCC#C)=O)CCN(C(C2CC2(C)Br)=O)CC1 Cc1scc(C(=O)NCC2(F)CN(C(C3CCCN3C(C)C)=O)C2)c1C C1(NC(=O)NCc2ccc(C(=O)OCC)o2)CC(C)(OC)C1(C)C CC1=C(C(=O)N2CC(NC(=O)CC3(O)CCCCCC3)C(C)C2)SCCO1 N(C1CN(C(C2CC2C2CC2)=O)CCc2ccccc21)C(c1cc(C)nn1C)=O CCCCCS(=O)(=O)CC(=O)N1CC=C(CNC(=O)C(C)(C)COCC)CC1 c1(C=O)ccc2nnn(O)c2c1.N1(C(C=C(C)C(C)(C)C)=O)CC2CC2C1C.N CC(C)CCC(C)N(C(=O)CC1CC(F)CN1C(=O)CCc1ccncn1)C C1(CNC(C2C(C)=CCC=C2)=O)CCN(C(c2ccc(F)nc2F)=O)CC1(F)F N1(C2C(NC(c3c(C)ncs3)=O)CCC2)CCN(C(=O)Cc2scnc2C)CC1 C1(NC(C(CC(C)C)OC)=O)CCC2CN(C(=O)C=CSC)CCC2C1 C(C)(CN=c1[nH]cnc2ccc(Cl)cc12)N(C(Cc1cc(C)no1)=O)C N1(C(C(C)CO)=O)CCC(CCCNC(C2CC(=C3CCC3)C2)=O)CC1 Cc1cc(Cl)nc(N)c1C(=O)NC1CN(C(c2ccnc(C(C)(F)F)c2)=O)C1 c1(NC(C(CC#C)(C)NC(c2cc(C)n(C)c2C)=O)=O)cccc2ccccc12 CCCC(C(O)C(=O)N(CCOCCO)CC)NC(C1C=CCS1)=O C1(C(N2CC(OCC(=O)Nc3scc(C)c3)C2)=O)CCCCC1.C(N)(=O)O N1(C(c2c(C)nc(C)s2)=O)CC(NC(C2(C)CCCO2)=O)CC12CCCCCC2 C1(C(=O)NC2C(NC(C(CC#C)(C)C)=O)CCOC2)CNC(=O)CC1(C)C CC(CC(=O)NCC1(NC(=O)C(Cl)=CCl)CC2CCC1C2)C(F)F N1(C(CC2(C=C)CCC2)=O)CCN(C(c2c[nH]nc2C2CC2)=O)CCC1C c1(OC)nc(C)sc1C(=O)NC1CN(C(C2COCCN2C)=O)CC1C(F)F N1(C(C=CC=CCC)=O)CC2(CC2)CC1CNC(C1CCC2CC2C1)=O c1(CNC(C(C(C)OC)NC(=O)C(O)CCN(C)C)=O)ccc(C#N)cn1 N1(C(Cn2c(C)cnc2)=O)CC(CNC(=O)C(c2ccccc2F)C)CC1(C)C C1(CC(=O)NCCOCC=C)CC(C)N(C(c2ncn(CC)n2)=O)C1 N1(C(C2(CSC)CC2)=O)CC2CCC1CC2.C1(CC(=O)N)SC(=N)NC1=O C(=O)(C1=CS(=O)(=O)CCC1)N1C2CN(C(c3cc(OC)cc(C)c3)=O)C(C2)C1 C1(NC(C=CC)=O)CC(NC(=O)Cc2ccc(OC(F)F)cc2)C12CCC2 C1(C)(C(=O)NC(CNC(c2cncc(C(C)=O)c2)=O)C)CCCS1(=O)=O c1(CN2CCC(C(c3ccccc3)C(=O)N(CC)CC)CC2)cnc(Cl)cc1C C1(CC(N2CCC(CN=[N+]=[N-])C2)=O)CC2(C1)CN(C(=O)C(F)OC(F)(F)F)C2 CN1CCC(C(=O)NC2CC(CO)N(C(=O)C(=C3CCCCC3)F)C2)CC1 Cn1cc(CNC2(c3nnnn3C3CCC3)CCC2)ccc1=O.N1(C)CCCCC1 c1(CCC(=O)NCC(C(C)(C)C)OC)c(-c2ccccc2)[nH]c2ccc(F)cc12 n1(CC(C(N2C(CCNC(C=CC(C)C)=O)CCC2)=O)C)ncc2c1CCCC2 N1(C(C(C)C(=O)N2CCOCC2)=O)CCN(C(=O)OC(C)(C)C)C2CCC12 C1(C(=O)NCC2CN(C(c3c(CC)cc[nH]3)=O)C2)CCN(C)CC1 Cc1ccc(NC(C2(F)CCN(C(C3C4CC5C(C4)C35)=O)C2)=O)cc1CO N1(C(C)=O)CCC(N=[N+]=[N-])(C(=O)N(C2CC(C)C2)C)C1 C1(C(=O)NCCN(C(c2cc(CCO)on2)=O)CC)Cc2cc(C)ccc2O1 C1(O)(NCc2snc(C)c2N)CCN(C(=O)C(F)(F)CCn2ccnn2)CC1 c1(C(N2CC(NC(c3ccccc3)=O)C(F)C2)=O)cc(Cl)c(F)cc1O Cn1cc2ccc(NC(C3(C)CN(C(=O)C#Cc4ccccc4)C3)=O)cc2n1 N1(C(C(CCC)N(C)C)=O)CC2CCCC(CNC(c3ncnn3CC)=O)(C2)C1 C1(C(N(C2CC(OC)C2)C)=O)CC2CC2N1C(c1ns[nH]c1=O)=O C1(F)(CNC(C(C)OCC(F)(F)F)=O)CCCC1.C1(C=O)CC2(CC2)C1 C(=O)(C1CCCc2c1ncn2C)NCC(CC)NC(c1nn(C)c(=O)cc1C)=O Cc1[nH]nc(C(F)F)c1C(=O)NC(C)CCCCNC(=O)C(c1cccnc1)O C1(CC)(NC(c2scc(C)c2Cl)=O)CCN(C(=O)C(C)c2ccon2)CC1 c1(C(CNC(=O)CS)NC(CC(CC)C2CC2)=O)cc(F)cc(Cl)c1.CC c1(C(=O)NC2C(NC(C(C)Cc3ccco3)=O)C2)cnn2c1N(C)CC2 CC(O)CCC(=O)N1CCCC1C(C)(C)NC(c1cnn(C)n1)=O c1(OC)cc(C(=O)NC2CC(F)(F)CC2)cc(F)c1F.C(=O)C(F)C(F)(F)F C(=O)(C1CCCc2nc[nH]c21)NC(CC(C)C)CNC(c1cc(Cl)cnc1O)=O C1(CC(=O)NC)CCN(C(c2ccccc2OC2CC2)=O)CC1.C1(F)CCC1 Cc1ccc(C)c(C(N2CCC(c3ccc(O)cc3)C2)=O)c1O c1(C(N2CCCCC(CNC(C)=O)C2)=O)cccc2c1SCCC2 N(C(=NCC(C)C)NCc1ccnc(OC)n1)C(C#C)C(C)(C)OC C1(C(=O)NC2C(C)C2(C)C)CCC(C)CC1N(C)C C1(CC(N2C(CNC(C=CCCC)=O)CCC2)=O)Cc2ccccc2O1 C=CCCCC(C)(C)C(=O)NCC1CCN(C(=O)C=Cc2cccnc2)CC1 c1(CC)nc(C(C)C(c2ccc(Cl)cc2)C)n(-c2cccc(Cl)c2)n1 N1(C(Cc2nnc(C)o2)=O)CC(NC(=O)CCOCC2CCC2)CC(F)C1 n1(CC(=O)NCC(C)C2CC2)c(O)nnc1O.c1(CCC=O)ccc(Cl)s1.N N1(C(C2CC(C)N(C)C2)=O)CCOCC(CNC(c2ccoc2Cl)=O)C1 N1(C(c2c(C)nc(CC(C)C)s2)=O)CCC2(CC1)CCN(C(C1CSC1)=O)CC2 C1(NC(c2c(CC)cncc2)=O)(C)CCCCC1C.c1(C(=O)N)cc(C#N)on1 c1(C(=O)N)cccc(N2CCOC2=O)c1.c1(CC)cc(C(=O)NCC(C)C)on1 C12(NC(c3c(CC)noc3)=O)COC(C1)C(NC(C1(C)CCCCO1)=O)C2 c1(C(=O)NCCCN(C(C(C(C)n2cccn2)C)=O)C)ccn2c1CCCC2 C12(CCNC(CSCCCC)=O)CCC(C1)N(C(C1CCOC1)=O)C2 C#Cc1cn(C)nc1C(=O)NCC(CCC)C(=O)NC(C1CCCCO1)(C)C N1(C(c2cc(C(C)=O)oc2C)=O)CCC2(CC1)CC(C)N(C(=O)C1=CCCC1)C2 c1(CNC(C(N2CCC(CC#C)C2)=O)=O)ccc(CCCN)cc1 C1(C(F)F)(CNC(C(N2CCC(N3C(C)COCC3)CC2)=O)=O)CC2(CCC2)C1 Cc1cc(C(N2CCC(N(c3nc(C4CC4)ns3)CCO)CC2)=O)c(C)cn1 c1(C(=O)NC(c2ccc(C)cc2)CC)ccc2nccnc2n1 C1(C(C)C)(C(=O)NCC(C2CC2)N(C(=O)CCc2nncs2)C)COC1 c1(-c2cc(C(=O)Nc3cc(O)nc(O)n3)sc2)cccc2c([N+](=O)[O-])cccc12 Cc1ccc([N+](=O)[O-])c(CNC2CCCN(c3ccc(F)cc3C)C2=O)c1 C(=O)(C(COC)CC(C)C)N1CC(NC(Cn2c(CCC)ncc2)=O)C(C)C1 C1(C(C)NC(=O)C(c2ccccc2)=O)CCCN(C(=O)Cc2cccc(C)c2)C1 c1(C(=O)NC2C(NC(C(CC=CC)C)=O)CCC2)cnc2c(Cl)cccn12 c1(C(N2CC(F)C2)=O)nn(C)c2c1CSCC2.n1(C(C)C)ccc(C(=O)NC)n1 N1(C(C(C)=C2CC2)=O)CCOC(C2CN(C(C3(C4CC4)CC3)=O)C2)C1 C1(NS(C)(=O)=O)CCN(C(C2CC3CC3N2Cc2sccc2Br)=O)CC1 c1(C(N2CCN(C(=O)C(F)F)CC2C(F)(F)F)=O)c(Cl)ccc(Br)c1F CC1(C)CCC(C(N2CCCC2C2(C(N3CC(F)CC3C(N)=O)=O)CC2)=O)C1 c1(C(N)=O)ccc2ncc(Br)c(OS(=O)(=O)C(F)F)c2c1 c1(-c2c(C)occ2)nc(C2CC2Cl)n(-c2ccn(C)n2)n1 c1(C(N(C)CC2N(C(C3C(OCC)C3)=O)CCOC2)=O)cnn2c1OCCC2 CN1CCN(C(=O)C=CC2CCOCC2)C(CNC(=O)CC2CCCOC2)C1 N1(C(C2(OCC)CCC2)=O)CCC2(CCCO2)CC1.C(=O)C(C)C(C)(C)C.C Cc1cc(C#N)ccc1C(=O)NC(CC(F)F)C(=O)NC1CC1 C1(NC(c2c(C)coc2)=O)COC2(CCN(C(=O)C(N)=O)C2)C1 c1(C(=O)NCC(CNC(c2[nH]c(=NCC)sc2)=O)C)ccn2c1CSCC2 N1(C(C=Cc2ccc(C)cn2)=O)CCC2(CCCN(C(=O)CCP(C)(C)=O)C2)C1 C1(C(=O)NC(COC)C(=O)N(C)Cc2nnc(O)o2)OC2CCC1C2 C1(C)(C(=O)NCCC(C)NC(=O)C(c2ccccc2)F)CCCS1 c1(C(N2CC(NC(C3(CCCC)CCC3)=O)C(O)C2)=O)ccc(F)c(C(F)F)n1 N1(C(C(CCC)OC)=O)C2CCC1CN(C(c1ccccc1C(C)C)=O)CC2 C1(C(=O)NC(c2cnn(C)c2)CC)(C)CCCN1C(=O)Cc1ccccc1.O N1(C(c2cnc(C)[nH]2)=O)CC2(CCC(CNC(=O)CC3(C)CCCCC3)O2)C1 Cc1nc(CNC(c2cnc(Cl)s2)C)sc1Br c1(OC)cc(C(N2CC(CCNC(C3(O)CCOCC3)=O)(OC)C2)=O)nn1C N1(C(c2cc(C(C)=O)c(C)cc2)=O)CC(C2CN(C(C3CCCC3C)=O)C2)C1 N1(C(C(C)(C)OC)=O)CCCC(F)(CNC(c2c(O)noc2C)=O)C1 Cc1nc(-c2cc(C(N3CC(NC(=O)C(C)CC4CCCO4)C3)=O)co2)cs1 c1(C(C(N2C(C)CCC2)=O)C)c(C)nn(C)c1C.CCCC(C(=O)N)NC(N)=O CCCC(CCCNC(c1cc(Cl)no1)=O)NC(c1c(N)cccc1Cl)=O N1(C(c2c(C)c(C(N)=O)ccc2)=O)CCC2(CC(NC(c3ccon3)=O)C2)C1 N1(C(CC2CCC(=O)C2)=O)CCC(C(=O)NC23CCN(CC2)C3)=C(F)C1 C1(C(=O)NC2CN(C(c3cnn(C)n3)=O)CC23CC3)CCOC2(CCC2)C1 CCCCC(CC(=O)NC1CCC2(CCC2)CC1)NC(C1CCCC12CCC2)=O N1(C(C(C=C)C)=O)CCCC(C(C)C(=O)NCc2n[nH]cc2C2CC2)C1 Nc1c(C(=O)NCC2(C)CCCC2)sc2ncccc12.C(=O)C(F)=C1CCC1 c1(C(CC)(C)O)cn(Cc2ccc(C(=O)NC(C(F)(F)F)C3CCCO3)o2)nn1 C(c1cc(F)c(F)c(F)c1)=CC=O.C#CCC(C)C(=O)NCC(C)C1CC1.N C1(C(N)=O)CC(O)CCN1CCCOC1CCOCC1 c1(C(C(=O)NC(c2csc(NC=O)n2)C)C)cncc(F)c1.C(C)(C)C.O C(CNC(C1CCCCCC1)=O)(CC(F)(F)F)NC(c1c(C)scn1)=O c1(OC)c[nH]c(C(=O)NCC(C)C2CC2)cc1=O.c1(C(=O)N)cc(F)cnc1Cl CCC(CN(C(=O)C(F)=CCCF)C)NC(C1CCSC1)=O C1(NC(C(C)Cc2cnc[nH]2)=O)CC(CO)N(C(=O)C=Cc2ccc(Cl)s2)C1 c1(Sc2n(C)nnn2)ccc([N+](=O)[O-])cc1C(N1CCn2cc(C)nc2C1)=O S(=O)(=O)(c1ccc(Cl)cc1)NCc1nccc(C(=O)Nc2cc(C)c(F)cc2)c1 N1(C(C(C(C)C)n2ncc(C)c2)=O)CC(NC(c2sccc2C)=O)CC(C)(C)C1 C1(C)(C(=O)NC(C)CN(C)C(c2ccc(C(N)=O)cc2)=O)CCC12CCC2 Cc1nc2ccccc2cc1C(=O)NCCC(C)NC(=O)COCC1CCOC1 C12(CC(N3CC(CC)OCC3)=O)CCC(CC1)OC2.C1(N(CC=O)C)CCCC1 C=CCC(C)(C)C(=O)N1CC2(CCNC(C3CCN(CC(C)C)C3)=O)CCC1C2 Cc1cc(C(=O)NC2COCCC2NC(=O)CCC2CC2(C)C)cc2nc[nH]c12 c1(C(=O)Nc2c(OC)nccc2C)n[nH]c2c1CN(S(=O)(=O)C(C)C#N)C2 n1(CCCC)cc(C(=O)NCC2CC(NC(=O)CO)C2)c(C)n1 CCCC(CC(C)C)C(=O)N(CCCNC(c1ccc(=NCC)[nH]c1)=O)CCO Cc1ccc(CCCC(=O)NC(C)C(CO)NC(C2CCC(C)CC2)=O)cc1 N#CC1CN(Cc2ccc(Cl)cc2)CC1NC(=O)CNC(N)=O n1(CCOC)cc(C(=O)NC2CC2)c(C)n1.C(c1sccc1C)=CC=O.N CCCCCC(C)(C)C(=O)N1CC(CC(=O)NC(CO)C(C)C)C2(CC2)C1 CC(CC1CCCO1)C(=O)N(CCNC(=O)CNS(N)(=O)=O)CCO CC#CCCCC(=O)N1CCCCC(N(C(=O)C(CCSC)OC)C)C1 C12(C(=O)NCC(CC=C)NC(=O)Cc3ccccc3S)CC(C)(C1)OC2C c1(OC)ncc(C(=O)NC(C2CCCN2C(=O)C=O)(C)C)nc1C.C(C)C.N C(C)(C(C(=O)NCCCCS(C)=O)NC(=O)Cc1ccc(C)o1)OC c1(C(=O)NC2CN(C(C3N(CCC)CCC3)=O)C2)sc(Br)c(C)c1C CC(C(=O)N1CCC(C(=O)NCc2ncc[nH]2)CC1)S(=O)(=O)c1ccc(F)cc1 Cc1csc(Cl)c1C(=O)NCC1CCCN1C(c1ccnc(C2CC2)c1)=O C1(NC(c2c(N)nccc2)=O)CC2(C1)CN(C(=O)CCC1CC1(Cl)Cl)C2 c1(C(N(C2CCN(C(C=C(CC)C)=O)CC2C)C)=O)ncnc2sccc12 C1(C(C)NC(=O)CCc2nccs2)CCCCN1C(=O)CCNC(N)=O C1(NC(c2scc(C)c2)=O)CCCN(C(c2cnc(O)s2)=O)C1C C1(NC(c2n(C(C)C)cnc2)=O)CN(C(=O)C(CC2CCCC2)OC)CCC1C Cc1cc(C)c(NC(=O)C(C2CC2(C)C)N(C)CC2CCCOC2)c(C)c1 c1(OC)ncc(C)cc1NC(C1(NC(=O)Cc2ncoc2C)CCSC1)=O c1(NC(C2CNCCN2Cc2ccc(Br)c(O)c2)=O)cc([N+](=O)[O-])c(F)cc1F CC(C)=C=CC(=O)N1CCCC1C1(C(=O)NC2COC(C)(C)C2)CC1 C1(C(C(F)(F)F)NC(c2ccc(Br)cn2)=O)CCN(C(=O)C(F)F)CC1 N1(C(c2cnc(C(C)OC)s2)=O)CC2CC2(NC(=O)C=Cc2cccs2)C1 CCCC(O)CC(=O)NC1CCC(NC(C2CN(c3nnnn3C)C2)=O)CC1 C1(C)(C(N2C(C)(COC)CC2)=O)CCCN(C(=O)C(O)CSC)C1 N1(C(C(F)=C(C)C)=O)CCCC2(CCN(C(c3cc(Br)ccc3N)=O)C2)C1 Cc1ccc(OCC(=O)NCCC2CC2)cc1.C12(C(=O)N)CC(C)(C1)C2 CC(C)C(CCO)NC(=O)CC1CCCN1C(C1CC(=O)CCO1)=O Cc1cc(-c2cscn2)c(S(=O)(=O)NCc2cnc(C(C)C)s2)cc1C c1(CNc2ccc(NCC3C(OC(C)C)CC3)cc2)ccccc1[N+](=O)[O-] c1(N2CCC(CCOC)(NC(CCC(=C)C)=O)C2)c(C)c(C)nc2ncnn12 c1(CC(N2CC=CCC2)=O)ccsc1[N+](=O)[O-].O=C(CCOCC1CCCO1)N C(C(C)C(F)(F)F)NC(c1[nH]c(=NC)sc1)=O.C1(C(=O)N)C2CC3C(C2)C13 C1(NC(c2cnn(CCF)c2)=O)CN(C(=O)COCc2ccccn2)CCC1F CN=c1ccc(C(=O)NCC(C)N(C)C(c2cc(C)nc(C)c2)=O)c[nH]1 CCC(CNC(=O)C(C)(C(C)C)NC(C)=O)N=c1[nH]c(SC)nc2ccccc12 c1(CC)ncnc(N2CCC(NC(c3cc(=O)c(OC)co3)=O)CC2)c1F C1(NC(c2cccc(CO)c2)=O)CN(C(C2CCCN2C2CCCC2)=O)C2CC12 C1(NC(CCOC)=O)CN(C(=O)C=C2CCC(C)CC2)CC2(CCOCC2)C1 C1(CNC(C2C(C)CCC2)=O)CC2CCC1N2C(C1CC(C)OC1C)=O c1(OC)cc(F)c(NC(C2(C)CC2)=O)c(F)c1.c1ccc(CN=[N+]=[N-])cc1.N C1(CNC(C2CCOC2)=O)CCCN1C1CCc2c(Cl)cccc21 N1(C(C2CC3CCC2C3)=O)CCC(O)(C2CC2)CC1.CC(C=O)NC(N)=O.N Cc1cc(C(=O)N(CCNC(C23CC(F)C2C3)=O)CCOCCO)on1 c1(CC(=O)N(CC(CC)NC(=O)CC(CC)OC)CC)ccc2c(c1)COC2 c1(NC(=O)NCC2CCCC(F)(F)C2)cc(N2CCOCC2)cc(F)c1 C1(C(=O)NCCSC)CCN(C(=O)C(C)(C)CCl)CC1 c1(N2C(CNC(C(C)SCCCC)=O)C(C)CC2)ccnc(C)n1.C(C)C.S c1(C(N(C2CCC(NC(c3cnns3)=O)C2)C)=O)ccncc1Br c1(C(N2C(C(=O)Nc3c(C(C)O)cccc3)CC2)=O)ccc2ccncc2c1 Cc1c(C(=O)NC(C(N2CC(F)CC2C)=O)c2ccco2)cccc1O Cc1ccccc1C(=O)NC1(C)CCN(C(=O)C(O)Cc2[nH]cnc2C)C1 C(=O)(CCCCCF)N1CCC(NC(CC(C=C)C)=O)C1C1CC1 C1(COC)CCN(C(c2cc(C(C)C)[nH]n2)=O)CC1.n1(CC=O)nnc(C)n1 Cc1ccc(C=CC=O)nc1.C1(CC(N2CC(O)(CC)C2)=O)COC(C)(C)C1 c1(C(=O)NCCN(C(=O)CC2CC(=O)C2)C)cc(Br)c2c(c1)OCO2 Cc1nc(C2CC2)oc1C(=O)NC1(C)CCCC1.C(=O)CCC1(C)CC1.N Cc1sc(O)nc1C(N1CC(CCCCNC(=O)C=CCn2cncn2)C1)=O CCS(=O)(=O)c1ccc(C(C)NC(=O)Cc2sncc2Br)cc1 C1(CNC(C2C(NC(=O)CCC3CCOC3)C2)=O)CNC(=O)CO1 c1(CNC(=O)CN2CCCC2CCc2ccccc2)cnc2ccc(F)cc2c1 C(=O)(C(F)C(F)(F)F)NCC(CC)CC.c1(C(=O)N)cccc(C(C)(F)F)n1 C12(C(=O)NCC(C)(CO)NC(C(C)Cn3ccnc3)=O)CCCN(CCC1)C2 C#CCCCCCC(=O)N1CCCCC1CCNC(=O)CC1CCCC(C)(C)C1 n1(CC)nc(C(=O)NCC(CO)NC(=O)C(C)(C)n2cnnn2)c(C)n1 CC1CN(C(=O)C(=O)NC(C2CC2(C)C)CC)CC1C(F)(F)F CCCS(=O)(=O)CC(=O)NC1(CO)CCN(S(=O)(=O)c2ccccc2)CC1 Cn1cc(-c2cn(CC3CC(NC(=O)C(n4cc(Br)cn4)F)C3)nn2)ccc1=O c1(C(=O)NC2CC(C)(C(N3C(CC)CCCC3)=O)C2)cc(C)c(F)cn1 CC(C)C(C)(N)C(=O)NC1CCCN(C(C)(C)C)C1=O N1(C(c2cncc(C)c2)=O)CCN(C(c2ccc(F)c(CO)c2)=O)C(C(F)F)C1 Cc1c(-n2cc(C(C)N(C)C(c3cn4c(n3)CCC4)=O)nn2)cccc1Br C(C(=O)N1OC2CCC1C2)=CC(C)(C)NC(=O)C=Cc1cscn1 c1(CC)c[nH]c2cc(CN3CCN(c4ncnc5[nH]cc(Cl)c45)CC3)ccc12 C(=O)(C1=NOC(C)C1)NC(CCCC)CNC(=O)Cn1cc(CO)nn1 CC1CN(C(C2CN3CCN2CC3)=O)CC1(C)C(=O)NCC(C)(C)CN=[N+]=[N-] C(=O)(C1=CS(=O)CCC1)N1C(C)CN(C(c2ccc(C(C)(C)C#N)cc2)=O)CC1 CC1(NC(c2cn(C(C)(C)C)cn2)=O)CCC(NC(c2ccco2)=O)CC1.C CCC(C(=O)NC1COCC1NC(c1cc(COC)on1)=O)n1nccc1C Cc1[nH]nc(Cl)c1C(=O)NCC1(O)CCN(C(c2ccncc2N(C)C)=O)C1 CCC(C)CC(C)NC(c1ncoc1CNC(c1nc(Cl)cs1)=O)=O c1(C(C)C)ccc(O)c(C(N2CCC(NC(C3NC(=O)C4CC34)=O)C2)=O)c1 CC1(C2CC2)CCCN1C(C1CC(NC(=O)C=Cc2ccncn2)C1)=O C1(CNC(C=CCNC(CCC(=C)Cl)=O)=O)CCCC(C)(C)O1 c1(C=O)ccc(C)c(C)c1Cl.c1(CCNC(C2CC(CC)C2)=O)ccccc1.N C(C(C(=O)NCCCc1cnn[nH]1)n1cc(-c2nc(C)cs2)nn1)OCC C1(CNC(C(C=CC)O)=O)CCC2CN(C(=O)COCCOC)CCC2C1 C#Cc1cnc(NCC(C2CC2)N(C)C(c2c(C)nn(CC)c2C)=O)nc1 N1(C(CN2C(c3c(C)nn(C)c3Cl)CCC2)=O)Cc2ccccc2S(=O)(=O)CC1C C#CCCCCC(=O)NCC1(C)CCN(C(=O)Cc2cccnc2Cl)C1 C(=O)(CCC(C)(C)C(=O)NC1CC(n2ccnn2)C1)OC c1(C(=O)NC(C)(CNC(C2CC2F)=O)CO)ccc(C(F)F)cn1 Cc1cc(NC(C2CCCC(NC(c3ccc(F)c(F)c3)=O)CC2)=O)cc(Cl)c1 C1(C)(CC)CC(C(=O)NC2CC3CC(NC(c4sncc4C)=O)C2C3)CCO1 C1(NC(C2C(C=C)CC2)=O)CC(F)CN(C(c2cccc(CC#N)c2)=O)C1 N1(C(C(C)(C)c2cnsc2)=O)CCC(=CCNC(=O)CO)CC1.C1CCCOC1 CC1(CCNC(C2(CF)CC2(F)F)=O)CCN(C(c2cncs2)=O)C1 Cc1[nH]nc(C(F)F)c1C(=O)N(C)CC1CN(C(C2(F)CCC2)=O)CCO1 c1(C(CC(=O)N)C)cccc(F)c1.C1(CNC(CNC(CC)=O)=O)C=CCC1 C(=O)(CC1=CCOCC1)NC1CCN(C(CCc2n(C)ccc2)=O)CC1 Cc1onc(C2CC2)c1C(=O)NCC1C(C)CCN1C(C1CCCN1C=O)=O c1(OCC(=O)NC(C(=O)OC2C(CCOC)C2)=O)ccc(C)cc1 CC1(C)CCC(C(=O)NCC(O)CNC(c2cnc(O)s2)=O)c2ccccc21 c1(C(=O)NC2CCN(C(c3c(COC)ccs3)=O)CC2F)ccn2nnnc2c1 C12(CCC(C)C=O)CC3CC(CC(C3)C1)C2.C(C(O)CN(C)C)NC(=O)NC CCC(CC(=O)N1CSCC1C(=O)NCCC(C)O)C(F)F C1(C(N(C2CCC(NC(C=CC)=O)CC2)C)=O)CCC2(CCC2)O1 c1(C(=O)NCC(C)N(C)C(C2(C)CCOCC2)=O)c[nH]c2ccccc12 c1(C(n2cc(CN3C(C)CC3(C)C)nn2)C)ccc2c(c1)CCO2 C1(CNC(C2(CC)CCC2)=O)CN(C(=O)C(Br)=C(C)C)CCC1(C)C CC1(C)CN(C(=O)CCC2CCCCO2)CCC1C(=O)NCC1=CCCCC1 C1(CNC(Cc2cccc(C)c2)=O)CC(NC(=O)C)C12CCC2.CC(F)(F)F C1(CNC(C2C(C)CCO2)=O)(NC(C2CN(C3CCOC3)C2)=O)CCCCC1 CC(c1ccco1)=CC(=O)NCCCC(C)NC(C1C2COCC12)=O S(=O)(=O)(c1cccc2cccnc12)NC1CCCN(Cc2ccc(SC)s2)CC1 Cc1c(NC(c2ccc(F)cc2)C)ncnc1N1CCCC(N2CCC2)C1 Cc1nc(C)c(CNC(=O)C(C)(CO)NC(=O)CCCC#N)[nH]1 C1(NC(C2(CC)CCCCO2)=O)CCCCCN(C(=O)CC=C(C)C)C1 c1(-c2nc(C3CC(N)C4C3C4)on2)cc(Cl)c2c(c1)OCO2 C(=O)(CCCC(=O)N1CCCN(C(c2cncn2C)=O)CC1)NCCC C1(NC(C(c2cnn(C)c2)C)=O)CCCN(C(c2ccccn2)=O)CC1 N1(C(=O)CN2CCN(C(c3ncc(F)cc3F)=O)CC2)CC2C(C1)C2(F)F c1(OCC)ccc(C)nc1C(N1CC(NC(C2(C)CC(F)(F)C2)=O)C1)=O CC1(C)CCC(C)N(C(c2cncc(O)c2)=O)C1.c1(C(=O)N)cc([N+](=O)[O-])n[nH]1 C1(N(C(=O)CC2CC2)CCC)CCN(C(c2nncn2C)=O)C1 C1(C(=O)NC2(C)CCN(C(=O)CC3(O)CC3)CC2)CC(=O)c2ccccc2O1 N1(C(C(C=C)(C)C)=O)CCCC(C)(NC(=O)CNC(c2ccoc2C)=O)C1 C(=O)(C1CCCc2nn[nH]c21)NC1(CCNC(CCCC=C)=O)CCCC1 C(CCCCC(=O)NCC(F)(F)C(N)=O)N(C(CCSCC)=O)C C(CC(C(=O)N(CCC(=O)OCC)C)NC(=O)COCC)OCC Cc1cc(C)c(C(N2CCC(C)(C)CC2)=O)c(O)c1.N1(CC(=O)N)CCC(C)C1 c1(C(N2CC(CC)C(c3ccccc3)C2)C(=O)NC(C)C)cc2n(n1)CCC2 C1(N(C(C2C(C(C)C)N(C(=O)C(O)CN(C)C)CC2)=O)C)CCOC(C)(C)C1 N1(C(c2ccc(CNC(c3n(CC)ccc3)=O)nc2)=O)CCC(C)C(F)(F)C1 C1(NC2CCCN(c3c(C)c(Cl)ccc3)C2)CC2(CCOCC2)C1 C(=O)(C1=Cc2ccccc2OC1)NC1CC(F)(CNC(c2n[nH]c(C)c2Cl)=O)C1 C=CC(C)(C)C(=O)NC1CC(NC(c2oc(CC3CC3)nc2C)=O)C(O)C1 C1(N)(C(=O)NC(C)CN)CC2(CCCC2)C1 C#CC1CC2(CC(C(N3CCCC3C)=O)C2)C1.c1(C(=O)N)cc(F)cc(F)c1N C(CC(C)C(=O)N1CC(C(=O)NCC2(O)CC2)(COC)C1)=CC Cc1ccc(C=CC(N2CC(C(O)C(=O)NC(C)(C)C(O)CO)C2)=O)cc1 CS(=O)(=O)c1ccsc1C(N1CCN(C(=O)C(O)C2CCCC2)C(CO)C1)=O N1(C(c2ccc(OC)s2)=O)CCCC2CN(C(=O)CC(CC)C3CC3)CC12 C12(n3cc(CC(COC)O)nn3)CCC(NC(=O)C(C3CC3)OC)(CC1)C2 C(=O)(C(CC(C)C)n1ccnc1)N1CC(COC)(NC(=O)C(C)(C)OC)C1 N1(C(C2CCCC(C)C2)=O)CCN(C(c2cc3[nH]ccc3s2)=O)CC1CO C1(C(=O)NCC2(O)CCN(C(=O)C3=CCCCC3)C2)CCOC2(CCC2)C1 C1(CC)(NC(=O)C(C2CCOCC2)F)CCN(C(c2nn[nH]c2Cl)=O)CC1 N#Cc1ccc(=NC2C3CN(C(c4cc5ccccc5nc4O)=O)CC23)[nH]c1 c1(C(NOCc2cn(-c3cc(C)oc(=O)c3)nn2)=O)ccc2ncccc2c1 CC1(C#CC(=O)N2CC(O)CC2CC(=O)NCC2CC(C3CC3)=NO2)COC1 c1(-n2cc(CCNC(Cc3n(C)ccc3)=O)nn2)ccc(Cl)c(C(F)(F)F)c1 N1(C(c2c(CC)cno2)=O)C2CCC1CN(C(=O)Cn1cnc(=N)[nH]1)CC2 N1(C(CC(=O)OCC)=O)CCCCCC1C.C(=O)(C(C)(F)CC1CCCC1)N C(=O)(C1CCc2ccccc21)NC1C(NC(c2ccc(CF)cc2)=O)CCC1 C12(NC(CCCC(=O)NC(C)C)=O)CCN(C(c3cnncc3O)=O)CCC1C2 N1(C(c2nc(C3OCCO3)cs2)C(=O)NCC)CCC(Cn2ccnn2)CC1 C1(CC(=O)N(C(C)CNC(=O)C(C)COC)CC)CC(C)(C)OC1=O C(N=c1[nH]c(=NCC(C)(C)CN(C)C)[nH]c2cc(C)ccc12)C1N(CC)CC1 C12(CCNC(c3[nH]cc(C)c3)=O)CCC1CN(C(c1cc(C3CC3)ccn1)=O)C2 C1(C(C)C)C(NC(c2cn(C)nn2)=O)CCN1C(=O)CCc1cccs1 CCCCCCC(O)CCC(=O)NCC(C)NC(=O)C(O)Cc1cnc[nH]1 N1(C(CC2OCC(C)(C)C2)=O)CCS(=O)(=O)C(CCNC(c2ccncc2)=O)C1 C(CNC(=O)CCCn1ccccc1=O)(C(C)C(C)C)NC(c1c(C)nns1)=O c1(NC(C(=O)N(CCCC)CCO)=O)nc2cc(F)c(F)cc2s1 CC#CC1CCN(C(C2(N(C(=O)C(C)C3CC3)C)CC2)=O)CC1 c1(C(N2CCC(CC)CC2)=O)nn(C)cc1S(C)(=O)=O.CC(C(=O)N)C(F)(F)F Cc1cc(C(N2CC3CN(C(c4cnc(O)[nH]4)=O)CC23)=O)cc(Br)c1 N1(C(=O)C=Cc2nccs2)CCC(O)(CNC(C2(C(F)(F)F)CC2)=O)C1 c1(C(=O)NCC(N(C)C(c2c[nH]nc2F)=O)C2CC2)cnc(-n2cccn2)cn1 C=C1CCC(C(=O)NCCCN2C(=O)CCC2=O)CC1 N1(C(c2cccc(CCC=C)c2)C(=O)NC)CCS(=O)(=O)C2(CCCC2)C1 C1(OC)CCCCC1C(=O)NC(C1CCCCC1)CNC(=O)C=CCO CCC(F)(F)CC(=O)NC1CCCC1NC(c1ccc(-c2cscn2)nc1)=O CC(C)CCCC(C)C(=O)NC(C(=O)NCc1ncsn1)C1CCOC1 C12(C(=O)OC)CC(C(=O)N)(C1)C2.C1(C=O)CC(C)(C)C1.C1CC1.C C1(C(N2CC(CCCCNC(C(C3CCCCC3)C)=O)C2)=O)CCCC1C1CC1 C1(COC)(NC(C2CC3CC3C2)=O)CCN(C(c2sc(Cl)cc2Cl)=O)CC1 C1(C(=O)NCC(C)C)CC(=O)N(C2CCCC2)C1.C1(O)(C(C=O)F)CCCC1 C=C(C)C1CN(C(=O)CCC(C(C)C)NC(c2cnc(O)c(F)c2)=O)CCO1 C(=O)(C(F)(F)C(C)(C)O)N1CC(CCC(NOCC(=C)Cl)=O)(OC)C1 N1(C(CC2(C)CC2)=O)CC2CCC(CNC(=O)CN3CCCCC3)C2C1 N1(C(C(C)(C)c2ccncc2)=O)CC2CC1CCC2NC(=O)CN1CCOC1=O c1(C(N2C(CN(C)C(C3CCCC(C#N)C3)=O)CCC2)=O)ccc2c(c1)CCC2 C1(NC(=O)CCN2CCCC2)CN(C(c2c(F)cncc2Cl)=O)CCC1O c1(C(N(C)C)=O)ccc(NC(=O)C(c2cncc(Br)c2)F)c(F)c1 N1(C2CN(C(c3n(C(OC)C)ncc3)=O)C2)CC(NC(c2cn[nH]c2)=O)CC1=O N1(C(C(CC=CC)CC)=O)CC2(C1)CCCS2(=O)=O.c1(C(=O)N)sc(F)cc1C O=C1CC(C(=O)NCCCn2cc(-c3ccc(F)cn3)nn2)CCN1 C1(C(N(C2CCN(C(=O)Cn3ccc(CF)n3)C2)C)=O)CCC(=C(F)F)CC1 C(=O)(CC(C)C(C)(C)NC(=O)CC1CC=CC1)NCCC(CC)(F)F C1(NC(CCCC(C)=O)=O)CN(C(=O)C(C(C)(C)C)N(C)C)CC(C)(C)C1 c1(NC(C2N(Cc3c(OC)ccs3)CC(F)C2)=O)cnc2ccc(Br)cc2c1 CCC(C)C(C(=O)NCC(C)(CC)C(=O)N1CC(O)(C(F)(F)F)C1)N(C)C C1(NC(c2c(C)nc(Br)o2)=O)(CNC(C2CC2F)=O)Cc2ccccc2C1 C1(C(N(C2CCN(C(=O)C(c3cnccn3)C)CC2)CC)=O)CC(F)CN1C S(=O)(=O)(c1cnc(NCC)cc1C)N(CC(CCC)O)C.C(F)(F)C(F)(F)F.O C(CCC(C)(C)C)(C(=O)NCc1cccc(Br)c1)N1CCSCC(C)C1 C1(C(N(CC(CC)NC(=O)CN(C2CC2)CC)C)=O)CCCSC1C C#Cc1ccc(NC(=O)C(F)(C)C(C)C)c(C)c1.c1(CC=O)nc(=N)[nH][nH]1.N c1(C(=O)NCC(CC)NC(c2snc(Cl)c2Cl)=O)cnn2c1OCC(O)C2 c1(CCCC)n[nH]c(=NC(=O)NC2CC(OC)C(OC)C2)s1 N1(C(C2(C)CN(C(c3ccc(C(C)(C)C)s3)=O)C2)=O)CCCC(C#N)C1 N1(C(C2(CCC)CCC2)=O)CCN(C(C2CC(CF)C2)=O)CC(O)C1 c1(C(CC)C(=O)N2CC(CC(C)NC(=O)C(=O)NC3CC3)C2)ccc(O)cc1 n1(CC(=O)NCC2CCN(C(CC3(C=C)CC3)=O)CC2C)nnc2c1CCCC2 N1(C(COC(CC)(C)C)=O)CCN(C(c2ccc(C)cc2)=O)CC1CC(F)F N1(C(C(C)=CC=C)=O)CC(C(=O)N(C)Cc2ccc(C)cn2)CC(C)C1 N1(C(C2CNC(=O)N2)=O)CC2CCC1CN2C(=O)C(F)=C1CCCC1 CCS(=O)(=O)CCn1nc(C(C)C)nc1-c1ccnc(COC2CCCCC2)c1 CC(C)C(CCNC(c1ccc[nH]1)=O)NC(=O)CC(C)(C)C C1(N(C(CCC=CC)=O)C)CCCCN(C(C2(C)CC(C)=NO2)=O)C1 CC(C(=O)N1CCC(CCNC(c2cc[nH]c(=N)c2N)=O)CC1)C(C)(F)F c1cccc(C#N)c1.C1(C(=O)NC)(COC)C=CCN1C(=O)C(O)C(C)C c1(C(N2CC(C)C(N(C(=O)C3=C(Cl)CCOC3)C)CC2)=O)ccc2cc[nH]c2n1 C(=O)(C(F)C(F)(F)F)NCCOCCN(C(C1(CC#C)CC1)=O)C c1(NC(CC2CCN(C(C3(CC)CC3)=O)CC2)=O)ccc2cc[nH]c2c1 C1(NC(c2c(C)snn2)=O)CCN(C(=O)C(C)(C)C2CCCO2)CC(C)(C)C1 C1(CCC=C)(NC(CCNC(N)=O)=O)CN(C(=O)CC(C)C2CC2)C1 Cc1cc(C2CC2)ccc1C(=O)NC(C)CNC(=O)Cn1cccnc1=O C1(CNC(C(C)OC)=O)C2CN(C(=O)C=Cc3scnc3C)CC12 Cc1cccnc1C(N1CCOC(CNC(c2ccc(OC(F)F)cn2)=O)C1)=O C(=O)(C(C)CC(C)C)NCC1CN(C(C(CC)(F)F)=O)CC1C(F)(F)F C(=O)(C(C)(C)C(F)(F)F)NC(C1CC(NC(CCCC(C)C)=O)C1)C N1(C(C)=O)CC=CCC1C(=O)NC(C)C(=O)N(C)C1CC1 c1(OC)ccc(C(N2CCC(NC(c3sc(=N)[nH]c3C)=O)CC2C)=O)nc1Cl C1(NC(C(CC2CC2)OC)=O)CN(C(=O)C)CC1F.c1cccc(C(C)C)c1 CCC(CC)(CCNC(=O)CN1CCCCCC1=O)NC(c1ccsc1C#N)=O C(=O)(C(CCC(C)C)NC(=O)CCCN=[N+]=[N-])NCC(C(C)(C)C)OC C(c1ccc(Cl)cc1F)=CC=O.c1(OC)ncncc1.C12(C(=O)N)CC(C1)C2 CON(C)C1CCN(C(C2CCC2CNC(C2COCCO2)=O)=O)CC1 C(=O)(C1CCc2c[nH]nc21)N1CCC(NC(=O)CCc2nncs2)C12CCC2 N1(C(c2[nH]cc(C(C)=O)c2)=O)CC(C)CC(C)(C)C1.C1(CC(=O)N)CCC1 C1(NC(c2ccc(NC)cc2)=O)CCC(C)N(C(c2cn(C3CC3)nc2C)=O)C1 C(C(CC1CC1)C(=O)NC1(C2CCCCO2)CC1)NC(c1ccccc1O)=O C(=O)(CS(N)(=O)=O)N(CCC)C1CC1.C1(C(C)C)(CC)CC1C=O.N c1(C(N2CC(NC(=O)CC3CC3)C(F)(F)CC2)=O)ccc2cncc(Br)c2c1 c1(C(=O)NC2CN(C(C=CC(C)C)=O)C3C2C3)cc2c(s1)-c1ccccc1OC2 c1(CC)ncc(C(=O)NCCCCNC(=O)Cc2cc(C)nn2C)c(C)n1 C1(CNc2ccc(F)cc2C(F)(F)F)CC2CCC(C1)C2F c1(C(N2CCCC(O)(CNC(=O)CC3CC(F)C3)C2)=O)cnn2c(Cl)cccc12 Cc1cccc(C(=O)C(=O)NCCC(C)CCNC(c2csnc2C2CC2)=O)c1 c1(C(=O)NCC(C)(CO)NC(c2cnccc2Br)=O)ccc(C2CC2)nn1 c1(C(N2CC(NC(c3ccc(O)cn3)=O)CC(C)C2)=O)cc(Cl)c(Cl)c(Cl)c1Cl C1(CNC(c2cc(C)[nH]n2)=O)CC(O)CN1C(c1cncs1)=O CC1CN(C2CC2)CC(C)N(c2nc(=N)[nH]c(=NCC34CC(CN3C)C4)[nH]2)C1 CCC(C)C(C(=O)N1CC(CCO)(NC(C2(O)CCCCC2)=O)C1)NC(C)=O C=CC(CC)CC(=O)NC(CNC(C1CCCCC1c1nc[nH]n1)=O)C(C)(C)C N1(C(C(C(C)(F)F)F)=O)CC(N=[N+]=[N-])C(S(C)(=O)=O)C1 N1(C(C=C(C)C(F)F)=O)CC(NC(c2c(C)noc2N)=O)CC12CCOC2 c1(C(=O)NC2(C)CC(NC(c3cc(C(CC)C)no3)=O)C2)cc(C)oc1C Cc1c[nH]cc1C(=O)NCCc1ocnc1CNC(c1nnn(C)n1)=O C(=O)(C(F)(F)C(O)C(C)C)Nc1ccc(Oc2ccc(C)nn2)cc1 c1(CC)ccccc1C.C1(SCC)CCC(CNC(=O)CCn2ccnn2)C1.N C1(c2n(C)c(N3CC4(CCCC4)CC3CO)nn2)Cc2ccccc2C1(C)C Cc1nc(C)c(C(=O)NCC(C)N(C(=O)C(C)OCC2CCCCC2)C)nc1C C(=O)(CC1COc2ccccc21)NC1C(NC(Cc2n(C)ncc2Cl)=O)CCC1 N1(C(C2(C)CNC(=O)N2)=O)CCCC(CC(=O)NC2CC(CCF)C2)CC1 C1(CNC(C(CC)F)=O)CC2CCCC(C1)N2C(=O)C(C(C)C)C1CCC1 N1(C(C(C)OCC)=O)CCC(NC(C2(C)CC(C(F)(F)F)C2)=O)C1 c1(OC)ccc(C=CC(=O)N(C2CN(C(=O)CCC3CCCO3)C2)C)c(O)c1 N1(c2n(CCOCC=C)c(CC)nn2)CC2(CCC2)CCC1C c1(C(=O)NCC(C)(O)CNC(=O)C=CC2CC2)cc2ccc(Br)cn2c1 C1(OC)CCC(C(N2CC(O)(CNC(=O)CC3(O)CCCCC3)C2)=O)CC1 C1(N(C(Cc2c(C)scc2)=O)C)CCCN(C(c2cc(Cl)cn2C)=O)C1 Cc1cnc(COCC(N2CCC(N(C(=O)Cc3cnc[nH]3)C)C2)=O)o1 c1(C(c2n(CC(=C)C)nnn2)NCCn2cncn2)c(-c2ccccc2)cnn1C c1(C=O)ccnc(C2CC2)n1.C(C)(C(=O)N(CC(C)O)CC)SCCCC.N Cc1cc(-c2nc(C3CCOC3)nn2CC2CCCO2)c2nccn2c1 N1(C(Cc2cccc(C)c2)=O)CCC2(CC1)CC(N=c1[nH]nc(C)o1)CO2 C1(N(C)C(c2coc(Br)n2)=O)CN(C(C2CC3(CC3)CO2)=O)CC12CC2 c1(C(N(CC(CCC)O)C)=O)cc(C)c(OCC(=O)OC(C)(C)C)c(C)c1 c1(C(N)=O)ccc(C(=O)NC2CC(CC)C2)cc1.C1(CC(=O)N)CCCOCC1 c1(C(=O)NCCC(C)N(C(C(CCC)N(C)C)=O)C)cc(O)nc2ccccc12 CCC(CC)CC(=O)N(C1CCC(NC(C2(c3ccc(Cl)nc3)CC2)=O)C1)C CC(C)CC(=O)NCC(=O)NC(C)CCCNC(C1CC1c1nccn1C)=O C1(NC(C(C(CC)C)N(C(=O)C=Cc2cncs2)C)=O)CCc2nncn2C1 C(CCN(C(=O)C=Cc1cnn(C)c1)C)(C(C)C)NC(Cn1c(C)cnc1)=O N1(C(C)C(=O)N(C)C)CCCC1C1CCCCN1C(c1cnn(C2CCC2)c1)=O c1(C(=O)NCC(C)N(C(C(CC2CC2)OC)=O)C)c(Cl)ccc2ncccc12 c1(CCC(=O)NCC2(OC)CN(C(CSCC)=O)C2)cnc2n1CCCC2 N1(C(C2C(OC)CN(C(=O)CS(C)(=O)=O)C2)=O)CCCSCC1C C1(NC(c2nccc(C)c2N)=O)CCCC2CN(C(=O)CC3CCCOC3)CC12 C(=O)(C(O)CC(F)(F)F)N1CC(C)(NC(c2sc(F)cc2Cl)=O)C1 CC1(C)OC2(CCN(C(=O)CC(N)C3CCCCC3)CC2)NC1=O c1(OC)n[nH]cc1C(=O)NC1CC(C)(NC(C2CC(SC)C2)=O)C1 C(=O)(C1CCCc2c[nH]nc21)NCC1CC(NC(=O)CCC2CCCC(=O)N2)C1 c1(CC)ccc(C(=O)NCC(O)CNC(C2CCC(C)(C)O2)=O)c(OC)c1 C(C1=NOC2CN(C(=O)CCCCN3CCCCC3)CC12)NC(=O)CC(F)(F)F C(=O)(C(C)(C)CC(F)(F)F)NCCN(C(c1c(C)sc(O)n1)=O)C N1(C(CCc2onc(C)n2)=O)CCN(C(c2cc(C(F)(F)F)on2)=O)C(C)C1C C#CCC(CC(=O)N(C)Cc1ccc(C)nc1)NC(c1nc(Cl)oc1C)=O C=CC1(C2(C(=O)N)CCC2)CCC1.c1(CC(=O)N(CC(C)O)C)ccc(O)nc1 N1(C(C(CC)NC(N)=O)=O)CC2CC(C=O)(C2)C1.C(O)(C(C)C)C1CC1.N Cc1cc(F)ncc1CNC(=O)C1=NOC(C)C1.C1(C=O)C2CCC(C2)C1C NS(=O)(=O)c1ccc(C(=O)N)cc1.C(c1ccncn1)=CC(N1CCCC1)=O.C N1(C(C(CC)(C)C)=O)CCC(CNC(=O)C(F)C2CCCC2)C(O)C1 c1(C(N2CCCC(C)(CNC(C=NOC)=O)C2)=O)cccc(N=[N+]=[N-])c1 c1(C(=O)NCC2CN(C(C3CCCCCC3(F)F)=O)C2)cc2cccn2c(O)n1 c1(OC)ncc(C=CC(=O)NCCNC(=O)C(c2cccc(C)c2)O)cn1 C1(N(CC(COC)O)C)CCCCN1C(=O)Cc1nccn1C Cc1cc(N)c(F)c(C(=O)NCCCCCNC(C2(CC(F)F)CC2)=O)c1F C1(NC(C2CC=CC2)=O)CCN(C(=O)C(C2CCCCC2)F)C1C1CC1 c1(C(C)(F)F)cccc(C(=O)NC2CCCC(c3ccc(Cl)cc3)C2)n1 CS(=O)(=O)C1(C(=O)NCCCO)CC1.c1(C=O)cccnc1.CC(F)(F)F.N c1(C(=O)NC(CC)CNC(C2(F)CC=CCC2)=O)ccc(C)c2ccccc12 C1(C(N2CC(C(C(=O)N(C)CC3(O)CCC3)O)C2)=O)CCC(O)C1 C1(NC(Cc2cn(C)nc2)=O)CCCN(C(c2cc(-c3ccncc3)on2)=O)C1 N1(C(CCN(CC)CC)=O)CC2CCC(N(C(=O)CCCC(F)(F)F)C)C2C1 C1(CC(=O)NCC(C)NC(c2c(CC)non2)=O)CCCC(C)(C)C1.C C=CCC(CC(C)C)C(=O)NC1CC1CNC(c1cnn(CCO)c1)=O N1(C(C2CCCC(OC)C2)=O)CC=C(C(=O)N(C2C3CCCC23)C)CC1 c1(NC(C2N(C(CC(CC)O)=O)CC(C)C2)=O)cnc(CO)nc1C C1(C(N(C)Cc2nc(C)[nH]n2)=O)(CO)CCN(C(=O)CC2CCCCO2)CC1 c1(CC(=O)NC2(C)CCN(C(c3[nH]nnc3C3CC3)=O)C2)ncn2c1CCCC2 c1(OC)ccc2c(c1)OCC(CNC(=O)C(=O)NCC1CC(OC)C1)C2 CC1(C)COC(CNC(=O)C(CNC(c2ccc[nH]2)=O)CC2CC2)C1 Cc1noc(C(C)C)c1C(N1CCC(C(C)NC(c2ccsc2C)=O)C1)=O c1(C(=O)N)c[nH]c(=NC)s1.C(C(C)C(=O)NCC1CCC1)N(CC)CC C1(c2n(C)cnc2)CCCN(C(C2C(CO)C2(F)F)=O)C1 c1(NC(C2(C)CN(C(C3CC3(C)C)=O)C2)=O)cncnc1Cl c1nn(C)cc1.C1CCN(C(C)=O)C1.C(=O)C.C(=O)CN(C)C1CC1.CC CCC(C)C(C(=O)NC(CNC(c1occc1Br)=O)C(C)(C)C)NC(C)=O C1(C(C)C)CN(C(=O)CC2(C)CCN2C(=O)C(C2CCOCC2)O)CC(=O)N1 CCC(Cc1ccccc1C)C(=O)N(CCNC(=O)C(F)=C(C)C)CC C#CCC(CC(F)(F)F)C(=O)NC1CCC(C)(C#N)CC1 c1(NCC2(C(C)(C)C)CCN(C(CS(=O)(=O)NC)=O)C2)nccnc1C#N C1(NC(=O)OC(C)(C)C)CCCN(C(=O)CC2CCCCCC2)CC1F N1(C(C(C2CCCO2)NC(COCC=C)=O)=O)CCC(C(=O)OC)CC1 N1(C(c2c(C)nc(COC)s2)=O)CC2CCC(C1)N2C(c1[nH]cnc1CN)=O CCC(C)C(C(=O)N1CC(O)CC1CNC(C1(C)CC1)=O)NC(N)=O C(=O)(C=C1SCC(=O)N1C)N.CC(C)CC(C(=O)NCC1(F)CCC1)N(C)C C(=O)(C#CC(C)(C)O)NC1CCCC(NC(c2c(C)n(C)cc2)=O)C1.C1CC1 c1(C(=O)NC(C#C)C(C)(C)OC)cc(C)cc(O)c1 C(C)(CCC(=O)NCc1nc(C)cs1)OC.C(=O)(C(C)(C)C1CCCCO1)N CC1=NS(=O)(=O)NC=C1C(=O)N1CCC(C)C1.c1(C(=O)N)nn(C(F)F)cc1Cl Cc1cc(N2CCC(NC(C3(C)CCCCCC3)=O)CC2)ncc1[N+](=O)[O-] c1(OC)ccc(O)c(C(N2CC(F)CC2CNC(c2ccc(Cl)cn2)=O)=O)c1 C1(c2nnnn2CC)(NC2(CC)CC2)CCC(C)SC1 c1(C(N2CCN(C(c3cc(C)sc3C)=O)C(CO)C2)=O)cc(C)c2[nH]cnc2c1 c1(C(=O)NCC2N(C(CC=CC)=O)CC2)cc2cc3c(cc2[nH]1)OCCO3 c1(NC(c2[nH]cc(C)c2C)=O)sc2c(c1C(=O)Nc1ncc(C#N)s1)CCCC2 C=C(Cl)CCC(=O)N1CCC1CNC(c1ccc(N(CC(C)C)C)cc1)=O C1(NC(C2(OC)CC(C)(C)C2)=O)COCCN(C(C2CCCCC2(C)C)=O)C1 C(=O)(CCCCC(C)C)N1C2CC(CNC(Cc3ccc(C)nc3)=O)C1CC2 C1(C(=O)NCCCN(C(CC=CC=C)=O)C)SCCC1C C1(C=O)CCCSC1.C(=O)(C=CC(=O)NC1CC1)NC(C1CC1)C.C c1(C(=O)NCCC2CCCN(C(CC3CC(=O)C3)=O)C2)cc2ccccn2n1 N1(C(C2C(C)(NC(c3cc[nH]n3)=O)CCCC2)=O)CC2C3CCC(C3)C2C1 C1(CCC)(NC(c2ccc(F)cc2)=O)CCN(C(c2cccn2C)=O)CC1 CC(CN(C)C)CCC(=O)NC1CCC(NC(=O)C(C)(O)C2CC2)CC1 c1cccc(F)c1.CCC(C)C(c1nnnn1C1CC1)NCCCn1ccnc1 c1(C(=O)NC(CC(C)NC(c2[nH]nc([N+](=O)[O-])c2Cl)=O)C)cnc2occc2c1 CC1CN(C(c2cnc(Cl)n2C)=O)CC1NC(=O)C(c1cncn1C)N(C)C c1(C(=O)NC2C(CNC(CC(=O)OCC)=O)CCCC2)cnc2ccsc2c1 Cc1cc(N)c(C)nc1C(N1CC(NC(=O)CCn2cccnc2=O)CC1C)=O CCCC(O)CC(=O)N(CCNC(=O)CC(C)n1cc(Br)cn1)C1CC1 n1(CC)nc(-c2ccc(OC(C)C)cc2)nc1C(C1CC1)SC N1(C(C(C)(C)OC)=O)CC2C3CCC(C(NC(=O)CCc4ccon4)C3)C2C1 c1(C(=O)NCC2(C)CCC2)cc2n(n1)CCCC2O.C1(CC(=O)N)CC=CC1 C1(NC(C(C(C)C)CNC(C2CCS2(=O)=O)=O)=O)C2CCC3C(C2)CC13 c1(CN(C(c2sc(Cl)cc2Br)C(=O)NC2CCOC2)C)ccc2ncccc2c1 C1(CCC(=O)NCCN2CCCC2)CCCN1C(=O)CCn1cnnn1 C1(NC(CCCCCC=C)=O)CC1C1CCN(C(c2cc(CO)n(C)n2)=O)CC1 N1(C(C(C(C)C)Oc2ccccc2)=O)CCN(C(c2csc(Cl)c2)=O)C2CCC12 C1(NC(C2ON=C(CC)C2)=O)COCCN(c2nc(C)ns2)C1 N1(C(c2ccc(SC)o2)=O)CCC(C)(NC(c2cnn(CCF)c2)=O)C1 c1(N(C(c2c(NC(C)=O)cccc2Cl)=O)C)nccc2ccccc12 c1(C(N2CCC(CNC(c3ccc(Cl)s3)=O)C2)=O)cc(O)nc(O)c1 O=C1CC2(C(N3CCCC3Cn3cc(C4CCCCO4)nn3)=O)CCC1CC2 C(=O)(C(C)(C)C(=O)N)NC.c1c[nH]nc1C1CCN(C(=O)C)C1.C1CC1.C N1(C(CN(c2cnccn2)C)=O)CCN(C2CCOCC2)C(=O)C1 CCCCC(O)C(C)C(=O)NCC1(O)CCCN(C(c2c(C)cnnc2O)=O)C1 c1(C(=O)NCCC(C)NC(c2n(CC)nnc2)=O)cn2cc(C)c(C)cc2n1 C1(CC(=O)NC2CONC2=O)(NC(C2C(C)=CCS2)=O)CCCCC1 C(=O)(C1c2cc(Br)ccc2CCN1C(=O)Cc1ncccc1C(F)(F)F)OC C1(C#C)(C(=O)NC(C#C)CC(C)C)CCN(C(C2OCCCC2(C)C)=O)C1 C(=O)(C(F)(F)C(C)(C)O)NCc1c(C(=O)NC(CCCC)CCC)con1 c1(C(=O)NC(CC)CNC(=O)CC(CC)C2CCC2)cc(C)nc(C)n1 C(C)(C(C)C(=O)NCCc1ncn(C)n1)NC(CCCOC(C)=O)=O N1(C(C(C=C)(C)C)=O)CCOCC(CNC(c2c(C(F)(F)F)ncn2O)=O)C1 C(CCCNC(=O)C(C)(C)c1nncn1C)OC.c1(C=O)ccn(C(C)C)n1.N CC(CC(=O)N1C(C(=O)N(C)Cc2ccon2)CCC12CC2)C(F)F O(C1CCOc2c(F)cccc21)Cc1cn(CCC(C(C)C)C(C)C)nn1 CC(CN(C)C)CC(=O)N1CCCC(C(=O)N(CC(F)(F)F)CCO)C1 C#CCCC(O)C(=O)NCCCN(C(c1onc(OC)c1Br)=O)C1CC1 N1(C(N(C)C)=O)CCCC(C(=O)N(CC(O)C)C)C1.c1(C(=O)N)ccc(Cl)nn1 N1(C(CNC(=O)NC)=O)CCC(C)(C)C1.c1(C(=O)N)ccccc1.CCCO C(C)(CNC(=O)CCC1CCOC1)(CC(C)C)NC(c1n(CC)ccn1)=O c1(CN(C(=O)CC2CCN(C3COC3)C2)C(C)=O)[nH]cnc1C#N C1(NC(C(COC)O)=O)CN(c2nnnn2Cc2ccccc2)CC(C)(C)C1 c1(CC(=O)NCC(CC)NC(c2cncc(C(=O)N)c2)=O)cc(F)ccc1C C1(NC(C(CNC(C)=O)(C)C)=O)CS(=O)(=O)CC1.c1(N)nccc(C#N)n1 C1(CC)CCN(C(=O)Cc2ccc(C(C)C)cc2)CC1.C=C1CC(C)(C=O)C1.N c1(C(NCCNC(C2CCC(C(N)=O)C2)=O)=O)cc(O)nc(C)n1.CC C(C(C)(CC)CO)NC(c1n(C(CC)(C)C)nnn1)c1occc1C1CC1 C1(CC)CC(O)CN1C(c1oc(CNC(=O)C(C)N2CCCC2)nc1C)=O Cc1ccc(C(C)NC(=O)C(Cc2ccco2)NC(C2C3CCCC23)=O)s1 c1(C(N2CCC(CN(C)C(C3CC=CCC3)=O)C2)=O)cc2c(s1)CCOC2 C(=O)(NNC(=O)C(F)c1ccc(Br)cc1)c1c(C)ncn1C N1(C(c2n(CC)ccn2)=O)CC2(C(=O)N)CCC1CC2.c1cnn(C(C)C)c1.C C1(NC(c2cnc3ccccn23)=O)CN(Cc2cnc(C3CC3)s2)CCC1(F)F C1(C(=O)NCC2N(C(C(OC)OC)=O)CCC2)Cc2ccncc2C1 CC1CC(NC(c2ccc(C(F)F)cn2)=O)CN1C(c1cccnc1C(F)F)=O [SH](=O)(=O)c1ccc(C#N)c(N2CCOC(C)(C(F)F)C2)c1.CC(C)(C)C(N)=O.N C12(CNC(=O)Cc3csnn3)CCCCC1N(C(=O)C=Cc1ccncc1)CC2 C(=O)(C(C)(C)C(N)=O)N(CCNC(c1c(C)nc(CCC)o1)=O)CC N1(C(CCCc2nc(C)sc2)=O)CCCCCC(NC(c2ccnnc2O)=O)C1 c1(C(=O)NC2CC(NC(CCSC)=O)C2)cc(CC(C)C)nc(O)c1 N1(C(C(CC)C(C)O)=O)CC2CCCC1C2CNC(c1ccc(O)nc1C)=O c1(OCC(c2nnnn2CC)(C)NC2CCC(CCC)CC2)ccc(C)cc1O n1(C(CC)C)ncc(C(CN2CCCC(NC=O)C2)=O)c1C1CC1.C(C)(C)C.O c1(CC(=O)NC2CCC(N(C)C(c3cnn(CCO)n3)=O)C2)ccc(Cl)nc1 c1(C(=O)NCC(CNC(C=C(C)C)=O)C)ccc2c(=O)cc[nH]c2c1 N1(C(CSC)=O)CCN(C(c2ccc(Br)c(F)c2C)=O)CC(CO)C1 N1(C(CN(C)CC)=O)CCCC2(CCN(C(=O)COC3CCCCC3C)C2)C1 n1(CC(=O)NC2C(NC(CCCc3ccc(C)cc3)=O)C2)c(C)cc(C)nc1=O c1(OC)cc(C(N2CCC(NC(=O)C3=NNC(=O)C3)CC2C)=O)c(N)cc1F C1(OC)CCCCC1C.c1(C=O)ncoc1C(C)(C)C.C12CC(C1)C(=O)N2.C C(=O)(CC(C=C)CCC)N(CCC(=O)NCCCC(C=C)(C)C)C CC(C)CC(CCc1ccccc1)C(=O)NCCN(C)C(C1(F)CCOC1)=O Cc1csc(CC(=O)NCc2ccc(C(=O)NC(CC3CC3)CO)s2)c1 c1(C(=O)OC)cc(CCCNC(=O)NCC2CCOCC2OC)oc1C C(=O)(C1=COCCO1)N1CCCC(C(C)NC(c2ccnc(C(C)(C)C)c2)=O)C1 C(C(C)(C)CNC(=O)C(CC)n1cccn1)N(CCC)C(c1scnc1)=O.C CC1(CNC(=O)Cc2ccccc2F)CCCN1C(C12CCC1C2)=O CCC(C(=O)NCC1CCCN(C(=O)CSCCC(C)C)CC1)C(C)O CCC(CC)(CO)C(=O)NC1CCOCC1NC(C12CCC(F)(CC1)C2)=O C1(NC(C)=O)CCOC(C(=O)NC(C2CCN(C(=O)NC3CC3)CC2)C)C1 C1(C(N(CCN(C(c2cc(CCC)c(C)s2)=O)C(C)C)C)=O)CCC2CC2CC1 C(c1ccc(OC)cc1C)=CC(N1CCN(C(CC(CC)SC)=O)C(CC)C1)=O C1(C=O)CCCC(=O)N1C.c1(CC)ccccc1CCNC(=O)C.C1CC1.O C1(CC(=O)N(CC(CNC(COCC(C)C)=O)O)C)COC(C)(C)C1 c1(C(=O)NC2C(C)CCN(C(=O)C3=COCCO3)C2)ccn2ncccc12 c1(C(=O)OCC)coc(C=CC(N2CCCC2CC(C2CCCCC2)=O)=O)c1 CCCC(C(O)C(=O)NCC(=O)NC1CC1)NC(c1ccnc(C)c1C)=O N1(C(C2C(CC)N(C(C3CC4(CC4)C3)=O)CC2)=O)CC2CCC2(C)C1 C1(C(=O)NCCCOCCN(C(=O)Cn2ncnn2)C)CCc2nccn2CC1 c1(C(N(C2CCN(C(CN(CCC)C)=O)CC2)CCOC)=O)nc(Cl)ccc1N Cc1cccc2cccc(C(=O)N(CCCCN(C)C(C3CC4CC4C3)=O)C)c12 N1(C(CC2(C)CC2(F)F)=O)CCCC(NC(=O)CCC2(C)CC2(F)F)CC1 C(N=c1[nH]cnc(=N)[nH]1)C1(C)CCN(C(C(CC)N(C)C)=O)C1 c1(C(C(=O)NCC(C=C)O)NC(=O)CCSC)cnn(C)c1 N1(C(=O)C(Cl)=CCl)CC2(CCN(C(C3C4(CC4)C34CC4)=O)C2)C1 N1(C(CCC#C)=O)CCCN(c2ncc3c(n2)CCC3)CC1C CC1CN(C(=O)Cc2cccn2C)CC(C)N(C(=O)CO)C1 C#Cc1cccc(C(=O)N(CCN(C(=O)C(C)(C=C)CCO)C)C(C)C)c1F C1(NC(c2c(CC)n(C)nn2)=O)CCC2(CCCN2C(=O)C2=CCCCO2)CC1 C(CCN=C(NCC1CCCSC1)NC1CCC1)NC(=O)OC(C)C c1(C(N2CC(O)CC(NC(=O)C=Cc3cc[nH]n3)C2)=O)nn2c(c1Br)CCC2 CC1(NC(=O)CCc2cscc2Br)CC(NC(c2cnsn2)=O)C1 c1(CC(COCC(=O)OCC(=O)NC(C)(C)C)C2CCC2)ccccc1 CCC(C)CCCCC(=O)N(C1CCN(C(=O)C=Cc2cn(C)nn2)C1)CC C1(CNC(CC(=C)C)=O)CCCCN1c1ccncc1C(=O)OC C(=O)(CCCCC#N)NC1CCCC(NC(C(C)(C)N(C)C)=O)C1 C(CC(C)C)(C(=O)NC)NC(=O)OC.C1(O)CN(C(c2cc(C)c[nH]2)=O)C1 C(=O)(C(F)C(CC)CC)N1CC(CC(C)NC(c2c(OCC)nccc2)=O)C1 N1(C(C(c2ccco2)NC(=O)COC2CCCC2)=O)CCN2CCCCC1C2 C1(NC(CC2(C)CC2(F)Cl)=O)CC2CCC1CN(C(c1ccco1)=O)C2 CC#CC1CCN(C(C2CC(NC(=O)C(=Cc3ccco3)C)C2(C)C)=O)C1 C(=O)(C(O)CNC(=O)CCC1CC(NC(C2SCC=C2C)=O)C1)NC c1(OC(C)(C)C(=O)NCCC2CSCCN2C(=O)C(O)CF)ccc(Cl)cc1 c1(CN(C(=O)C=Cc2ccc(I)o2)CCC)ccccc1Br c1(CNC(C=NOC)=O)ncc(C(=O)N(CCC(C)C)C)cn1 c1(C(=O)NCCN(CCC)Cc2cnc(C)o2)cc(OCC)cs1 Cc1cccc(C)c1NC(=O)CN1CCC(NC(=O)CN2CCCC2=O)C1 CC1CCCN1CC(N1CC(F)(C(=O)N(C)Cc2cccnn2)C1)=O Cc1cc(=O)oc2cc(Nc3nccc(N4CCC(O)C(C)(C)C4)n3)ccc12 c1(C(N2CC3CC2CS3)=O)n[nH]c2c1CN(C(=O)C1=CC3C=CC1C3)C2 C1(C(=O)NC2(CN(C(CC)=O)C)CC2)CCC2CC1C2(C)C c1(C(=O)NCC2CCC(NC(C=CCCC)=O)C2)sc(Br)c(C)c1C C(=O)(C1=C(Cl)CCOC1)NC1(CNC(C(C)(C)CO)=O)CCCCC1 CC1CCN(C(=O)CC(F)(F)c2ccccc2)CC1NC(c1ccccc1)=O c1(N(C)Cc2c(C)cnn2C)cccc(S(=O)(=O)N2CCOCC2CO)n1 O=C(C(O)C1=CCCCC1)NC1C2CC1N(C(=O)C(F)(F)CC1CCCO1)C2 c1(CCC=O)nc(-c2cccnc2)no1.CCS(=O)(=O)NCC(=O)NCCC.N c1(C(N(C2CCN(C(=O)CC3COC(C)(C)CO3)C2)C)=O)cc2ccncc2[nH]1 c1(CC)c(C(=O)NC)cccc1F.C(=O)(C(C(C)CC)N(C)C)N1CCC(F)C1 c1(OCC)cc(C(N2CCC(C)(CC#N)C2)C(=O)NCCCOC)ccc1F c1(CN2CCC(O)(CC(=O)Nc3cnc(C)c(C)n3)CC2)nc2ccccc2[nH]1 c1(OC)c(-c2cncc(NC(c3ccnnc3)=O)c2)cccc1O C=CC1COCC1NC(=O)Cn1cc(CNC(=O)C(COC)CO)nn1 CC1C(NC(=O)NC2CC(OC(C)(C)C)C2(C)C)CCS1(=O)=O C(C1(C)CCOCC1)=CC(=O)NC1C(NC(CSc2n(C)nnn2)=O)CC1 Cc1cnc(C)c(C(=O)N(C)CC2CCN(C(=O)Cc3csc4nccn34)C2)c1 c1(CC(=O)NC2CCN(C(CCOCCC)=O)C23CC3)cccc2nonc12 N1(C(=O)NC(C)C)CCCC(C(=O)NCC(F)C)C1.C(=O)(CC(C)(F)F)N c1(C(=O)OCCC2(C(=O)O)CC2)occc1-c1ccccc1 c1(C(N2C(C3CCN(C(CNC(=O)NC)=O)C3)CCC2)=O)cccc(F)c1Cl N1(C(c2c(C(C)C)occ2)=O)CC2C(NC(=O)C(O)CN(C)C)C2C1 N1(C(C(CC)c2ccccc2)=O)CC(O)CC1C(=O)Nc1ccccc1N(C)C Cc1[nH]ccc1C(=O)NC(C(=O)NC1CCCC1CCN(C)C)C1CC1 Cc1ccc(C(N2CC(CCNC(=O)C(C)C(C)O)C2)=O)cc1OC(F)F CC(O)CC(C)(C)CN=c1nc2ncn(C)c2c(NCc2ccc([N+](=O)[O-])o2)[nH]1 Cc1nc(O)nc(C)c1CC(=O)NC1CCN(c2nc(C(C)C)ccc2C#N)C1 C1(C)(NC(CCC2(C)CN(C(C3C(C)CC3)=O)C2)=O)CCCC1(F)F N1(C(c2scc(C)c2)=O)CC(C2CC2)(C(=O)NCC2CC(COC)CO2)C1 c1(NC(C(CCF)NC(C2CC3C=CC2C3)=O)=O)ccc(CO)cc1O c1(C(=O)NC23CCN(C(=O)C)CC2C3)csc2ccccc12.C(=O)(C1CC1)N c1(-c2nc(NC(c3cccc(C)c3Cl)=O)sc2)cc2ccccc2s1 CS(=O)c1ccc(C(N2CC3(CCC3)C2)=O)cc1.C1(C=O)CCC(C(N)=O)C1.N C1(O)(c2cn(C(CNC(c3cnc(COC)s3)=O)C)nn2)CCOCC1 c1(N(C(=O)NCCCC(=O)OC)CC)ccc(Cl)c(Cl)c1C C(=O)(CC(C)(C)C(F)F)N1CC(C(N2CC(O)(CC=C)C2)=O)N(C)CC1 CCC(C)(C(=O)NC1CCC(CCC(N2CC(CO)C2(C)C)=O)C1)OC Cc1cc2[nH]c(C(=O)NCCC3(O)CN(C(C4CC4(C)Br)=O)C3)cc2o1 C1(CN2CCC(c3ccc(C(=O)OC)o3)CC2)CC2CCCCC2N1 C1(C(=O)NCC2C(C(=O)OC)CC2)CN(C(c2cc(C#N)c[nH]2)=O)CCO1 c1(C(N2C(C)CC(NC(=O)Cc3cnc[nH]3)C2)=O)ccc2c(c1)CC(=O)N2 C(C1OCc2ccccc21)N(c1c(C)c(N2CC3CCCC3C2)ncn1)C O=C1COC(C2(CNC(=O)Cc3nnc(S)n3Cc3ccccc3)CC2)CN1 C(=O)(CC(C)C(F)(F)F)N1CC(NC(c2cnn(CCC)c2C)=O)C(OC)C1 c1(CNC(COCC#C)=O)nc(C)c(C(N2CC(CO)C(O)C2)=O)o1 C(CCC1CCC1)(C(=O)NCCC1CCCCC1)NC(=O)CCN1CCOCC1 C(C(C(=O)NC1CCCCC1CC(=O)OC)C(F)(F)F)c1ccc(OC)cc1 c1(NC(C)=O)ccc(C(=O)N(C2CN(C(=O)CCCN(C)C)CC2O)C)cc1 Cc1[nH]cc(C(=O)NC2(C)CCC2)c(=O)c1Cl.C1(C=O)CN=C2N=CNN2C1.N O=C(CCCCCCNC(=O)C(F)OC(F)(F)F)NCC1CC(O)C12CCC2 c1(CC(=O)NCCC(CNC(C(CC)C)=O)O)ccc(Cl)c(F)c1 c1(C(=O)NC2(CO)CN(C(CCOCCOC)=O)C2)ccc(C2CC2)nc1O N1(C(C(=Cc2ccccc2)OC)=O)CCC(C)N(C(=O)CCC(C)(C)O)CC1 C1(CNC(COCC)=O)CN(C(=O)C(C)=O)CCC12CCC2 N(C(=NCCCN1CCP(C)(=O)CC1)NC1CCN(C(C)C)CC1)C(C=C)C C1(c2onc(C(C(C)C)N)n2)COCC1(C)C N1(C(c2c(OC)ccc(Cl)c2)=O)CCCC1C1CCCN1C(=O)COC1CCC1 c1(C(N2C(C)CCCC2)=O)ccnc2ccc(-c3ccc4c(O)n[nH]c4c3)cc12 C1(C(=O)NCCCC(C)(C)OC)CC2C=CC1N(C(c1ccco1)=O)C2 C1(NC(c2noc(CC)c2C)=O)CC2CC(C1)N(C(c1ccc(F)c(N)c1)=O)C2 c1(C(N2CCC(C)(NC(CCCOC)=O)C2)=O)nn(C)c(C2CC2)c1C Cc1onc(C2CC2)c1C(=O)NC(C)CCO.C(C1CCCCC1)=C(C(=O)N)F CC1(C(N2CCC(OCCNC(=O)CC3CCSCC3)C2)=O)CCC(=O)C1 C(=O)C1=NN(C)C(=O)CC1.N1(C(C2(OC)CC(C(F)F)C2)=O)CCC(C)C1 C(=O)(C1CCCc2ncnn21)N1C(C)CCC(NC(C2CCCS(=O)(=O)C2)=O)C1 N1(C(Cc2cccc(CC)c2)=O)CCN(C(=O)C(C)(C2CC2)OC)CC1COC c1(CN(C(=O)CSCC(N)=O)C)ncnn1C.c1(C(=O)N)cc(C)on1 C1(NC(C2(CC=C)CCN(C(=O)CC3CCOCC3)C2)=O)CCN(C)C1(C)C c1(C(N2CC(CCCC)C2)=O)ccc(S(N)(=O)=O)nc1.CC1(C=O)CC1(F)F.N C1(NC(C(C)SCC2CC2)=O)CC2CCC(C1)N2CCn1ccnn1 c1(OCC(=O)NC)cccc(Cl)c1.c1(C=O)cc(=O)cc[nH]1.C1(CC)CC1 c1(C(c2n(Cc3ccc(OC)cc3)nnn2)NC(C)C)c(F)ccc(C)c1F C1(C(=O)NCC(CN(C(CCc2cc(C)on2)=O)C)O)CCc2nnc(C)n2C1 C(=O)(C(CC(C)(C)C)OC)N(C(CC)C(=O)NCCn1ccnc1C)C c1(SC)cccc(F)c1C(=O)NCC1(C)CN(C(C2(C)CCC2)=O)CC1C N1(C(CCCOC(C)C)=O)CC(C)CN(C(C2(C)CC2Br)=O)CC1C N1(C(C2CCCOCC2)=O)CCC2CCN(C(=O)COc3ccccc3F)C2C1 C(CCN=C(NCc1cc(C(F)(F)F)n(C)n1)N1CCCC(S(C)(=O)=O)C1)OC c1(C(=O)NC(CNC(C2N(CC)CCCC2)=O)CCOC)nnn2c1CSCC2 c1(C(=O)NCC2CC2NC(c2nc(Cl)sc2Cl)=O)cn2ccnc2s1 N1(C(Cn2c(C)nnn2)=O)CC(C)(C)OCC1CNC(=O)CCC=CC(C)C c1(CC(C(N2CC(NC(C(C)=CC)=O)(COC)C2)=O)O)ccc(O)cc1 C1(NC(c2c(COC)ccs2)=O)CCN(Cc2cccnc2)CC1 N1(C(C=CC(C)C)=O)CCN(C(=O)C(F)n2ccnc2)CC(C)(F)C1 C(C1=CCCN(C(c2ccnc(F)c2O)=O)C1)NC(c1c(C(C)C)onc1)=O C1(C(=O)OC)(NC(c2ncc(Cl)cn2)=O)CC(O)C12CCC2 N1(C(C(c2ccccc2)SC)=O)CCN(CCN(C(=O)CN2CCC2C)C)CC1 Cn1ccc2cc(C(=O)NCC3CCC3)cnc12.c1(C(=O)N)cc(O)nc(O)n1 c1(C(=O)NCC2CCCC(CNC(CCC#C)=O)C2)ccc(C)cc1SC Cc1nc(C)c(C(=O)N(C)CC2(C)CC2)c(C)n1.c1(C=O)nc(Cl)ccc1N N1(C(C2CC(OC)C2)=O)CC2(CC(C(=O)N(C)CCN3CCCCC3)CO2)C1 c1(C(N(C)Cc2ccc(C)cc2)=O)c(O)cnc2cc(F)ccc12 c1(NC(C(CO)SC)C)ncnc(NCc2cc(C)ccc2OC(F)F)c1C C1(COC(C2C(C(=O)OC)C=C2)=O)CCC(CC(F)(F)F)CC1 c1(C(N2CCC(NC(C(C)NC(=O)C3CC3)=O)C2)=O)ccc(O)c(F)c1.C C1(NCC(=O)Nc2cc(F)ccc2Oc2cccc(Cl)c2)Cc2nccnc2C1 C1(C(=O)NCCC(C)C)CN2CCCC2CO1.C1(S(C)(=O)=O)(C=O)CCCC1.N c1(C=O)nc(C)n(C2CC2)c1C.C(=O)CC1CN(C=O)C1.C(C)(C)C.C C=CCC(C(=O)NCc1nnn(C)c1C(=O)NOCCC(C)O)OC c1(C(=O)NC(C2N(C(c3c(C)scn3)=O)CCCC2)C)nnc2ccccc2n1 C(=O)(C1=CC2CCCC12)NCC(C)(C)NC(c1ccn(CCCC)n1)=O N1(C(c2c(CC)noc2)=O)CCC(CCNC(=O)CCn2ccccc2=O)CC1 c1(OCCCC(=O)NC2C(NC(C(C)C)=O)C2)cccc(Br)c1 CC1CN(C(C2CCOC2C)=O)CC(C)N(C(=O)C(O)C2CCC2)C1 c1(CC(C)C(=O)NC2CC2NC(=O)C(F)=C2CCCC2)ccc(Cl)cc1 C=CC(CCC)CC(=O)N1C2CCC1C(C(=O)NC(COC(C)=O)CO)C2 c1(CCC(=O)N(C2CCCC2)C)ccc(F)nc1.c1(C(=O)N)cc(C(F)F)no1 N1(C(c2n(CC)ccc2)=O)CC(CC(=O)NCC2CCC=CO2)CC1(C)C c1(NC(Cc2c(C)noc2C)C)ccc(S(=O)(=O)N)cc1Cl.C1(C)CC1(C)C.C C1(OC)CCC(CC(=O)N(CCCNC(C2(c3ccccc3F)CC2)=O)C)CC1 C1(CCNc2c(C)ncs2)CCN(C(c2ccc(Cl)cc2)C)CC1 C=CC1COCCN1C(=O)C(F)C(C)CNC(=O)COCCC C1(C)(CNC(C(CCC)OC)=O)CN(c2nnc(C(F)F)s2)CCO1 Cc1cccc(C(N2CCC(CCNC(c3cc([N+](=O)[O-])n[nH]3)=O)C2)=O)c1C#N C(=O)(C1=C(Cl)CCOC1)NC(c1cn(C)nn1)C(=O)NCCC(C(C)C)C CC1(C(=O)NC2CCN(C3CCN(C(=O)C4CC4)C3)CC2)CCCOC1 n1(CC2CCCN(CC(c3c(OC)cccc3)=O)C2)cnc2ccccc12 c1(N(C(=O)CC(N2CC(O)C(O)C2)=O)C2CCC2)cc2cnccc2[nH]1 C(=O)(C(C(CC)C(C)C)N1CC(F)(F)CC1CC(=O)OC)NCCOCC C=CC(C)(C)CC(=O)NC1CCCCC1CNC(=O)C(C)N=[N+]=[N-] C1(C(=O)NCCC(C)N(C(C2C(CCOC)C2)=O)C)CCC2(CC1)CC2 N1(CCc2nnn(C(C)(C)C)n2)CC2C(NC(c3nocc3C3CC3)=O)C2C1 c1cccc(Cl)c1.CN(S(N)(=O)=O)CC(=O)NCC1CCCC1.C(=O)(C)N C(C)(CC(=O)NCC(C1CCCC1)NC(c1cnoc1-c1ccco1)=O)SC c1(C(=O)OC2CCC(CCC(=O)OC)C2)cn2cc(C)c(C)cc2n1 c1(C(=O)NCC2C(C)CCN(C(=O)C3=CCC3)C2)ccc2nncn2c1 N1(C(c2ccc(CNC(C3(C#C)CC3)=O)cn2)=O)CCC(O)(CC)CC1 C(=O)(C1CCCc2scnc21)N(CCNC(C1CCC(CCC)CC1)=O)C1CC1 c1(OC)cnc[nH]c1=NCC1(F)CC(NC(=O)Cc2cc(O)nc(O)n2)C1 c1(C2CN(C(c3cccc(C)c3I)=O)C2)cn(C2CCc3cc(Cl)ccc32)nn1 C(=O)(C(C)(C)CC(=O)N1CCCCC1CCNC(c1scnc1Cl)=O)OC Cn1nc2c(c1C(=O)NCC1CC1)CN(C(c1ccnc(Cl)n1)=O)CC2 C1(CNC(c2nc(CCC)oc2)=O)CCN(C(c2cc([N+](=O)[O-])c[nH]2)=O)CC1C c1(N2CCCCC(CO)C2)nc(N2CCS(=O)C3(CCC3)C2)nc2c1CCCC2 c1(NC(=O)NC2(CC(NOC(C(C)C)CO)=O)CC2)cn(C)ccc1=O c1(C(N2CC(O)C2)=O)cc(C)nc2c(C)cccc12.C(C)(C)(C(=O)NC)OC.C C(=O)(CC(C)CC(C)C)N.C1(NC(C2C(C(C)=O)C2(C)C)=O)CCCC1(C)C C1(NC(CC=CC=C)=O)CCCC(NC(=O)C(c2ccccc2F)(F)F)C1 C1(C)(C=O)CCS(=O)(=O)CC1.C(C)(CC(C)C)NC(c1nc(CC)sc1)=O CC1(C)CCC=C(C(=O)N2CC3CC(NC(=O)CC4CC5(CC5)C4)C3C2)C1 N1(C(CN(CCC#C)C)=O)CCN(C(C2CCCS2(=O)=O)=O)C(CCO)C1 C1(C=O)(NC(C(C)Cn2ccnc2)=O)CC(F)(F)C1.C(O)(C(C)C)C1CC1 C1(NC(C(CCC)F)=O)CCC(C)(CNC(=O)C(=O)NC(C)C)CC1 C1(CCNC(c2cscn2)C)CCOC1(C)C N1(CC)CCCC1NC(C(=O)NCC(N)CCc1ccccc1)=O c1(C(N2CCC(C(=O)NCCCC=C)CC2)=O)ccc(F)c(C)c1 C(=O)(CC(C)CNC(C1(OC)CCN(C(=O)CC(C)SC)C1)=O)NC C(=O)(C1=CC2(CCOC2)C1)NCCC1(O)CCN(C(C=Cc2n(C)ccc2)=O)C1 c1(CNC(CN(C(C=CC(C)C)=O)C)=O)ccc(=O)n(C)c1 c1(C(C=O)N(C2CCCC2)CC(C)C)ccc(O)cc1.C(=O)C.C(C)=O.CO N1(C(C2N(C(C(C(C)C)OC)=O)CCOC2C)=O)CC2CCC(C1)C2O N1(C(c2c(C)nc(C(C)C)o2)=O)CCCC2(C)CCCC12.C(=O)C=CC(N)=O CC(F)(F)CCCC(=O)NC1(C)CCCN(C(=O)COC2CCC2)C1 C1(n2cccn2)(C(N(C)CC)=O)CCN(CC2(C)COC(=O)N2)CC1.C1CC1 CCC(C)C(O)C(C)C(=O)NCC(=O)NC1CCC(C(=O)OC)CC1 C1(CNC(C2(C(C)C)CCC2)=O)CCN(C(=O)CCC2CCCN2C)C(C)C1 N(C(=NCCc1cnn(C)c1)NCc1ccco1)Cc1csc(C)c1C CC(C)CCCCC(=O)NCC1CCC2CN(C(=O)C=Cc3cocn3)CC12 C1(NC(C(CCC)OCC)=O)CN(C(c2cccnc2S)=O)C(C)(C)C1 N1(C(CCCC(=O)N(C)C)=O)CC2CCC(C1)N2C(=O)C(c1ccc(O)cc1)=O Cc1ccc(COC(C)C(=O)NC2CC(N(C)C(c3cncnc3C)=O)C2)cc1 CCC(C(=O)N1CC(NC(c2cscc2S(C)(=O)=O)=O)C(O)C1)C(C)(C)CC c1(C(=O)NC2CN(C(c3cc(OC)no3)=O)CC2C)ccc(OC)c(OC)c1C CC1CCN(C(=O)CC2CC3(CC3)C2)C1C.c1(C(=O)N)c[nH]nc1C(F)F C(CC(C)(C)CC(=O)NCCCN(C(=O)C(C)Oc1ccc(OC)cc1)C)OC c1(-c2nnc(N(c3nnc(C(F)F)s3)C)s2)ccc(C2(O)COC2)cc1 N1(C(C2(OC)CCOC2)=O)CCC(O)C(NC(c2ccc(CCO)cc2)=O)C1 C1(CC)(NC(=O)CC2CSC2)CCN(C(=O)C(c2ccc(F)cc2F)(F)F)CC1 c1(C(=O)NCC2(O)CN(C(C3C(C(C)C)OCC3)=O)C2)ccn2nccc2n1 Cc1cc(Br)cc(F)c1C(=O)NCC1(C(=O)Nc2cc(Cl)ncn2)CC1 CCCCC(CC(=O)NCC(=O)OC)NC(=O)CC1CCOC1 Cc1cc(CNC(=NCCNS(C)(=O)=O)NCC2CC2(Cl)Cl)cc(C)c1 c1(CC)ccc(C(=O)NCCC2CN(C(C3CC3C3CC3)=O)CCO2)cc1OC C1(NC(CCS(=O)(=O)NC)=O)CCC2(CC1)CC2NC(c1cc[nH]n1)=O.C Cc1cccc2sc(NNC(=O)c3ccc(OC(C)C)c(Cl)c3)nc12 C1(CNC(C(C)C(F)F)=O)CC12CCN(C(=O)C=C1CN3CCC1CC3)CC2 c1(OC)cc(C(N2CC=CC(NC(=O)C(C)Cc3ccco3)C2)=O)ccc1Br c1(C(N2CC3C(C(=O)NC(C)CCO)(C3)C2)=O)ccc2ncsc2c1 c1(CSC2CC(=O)N(C(C3CCCCO3)=O)C2)cn2cc(Cl)cnc2n1 C=C1COCCN(C(=O)CC2CCCN2C(c2cc(C)nc(C)c2)=O)C1 c1(CC(=O)NCCCCNC(CC(COC)COC)=O)nsc2ccccc12 CCCC(CNC(C1CN(CC)CCO1)=O)C(=O)N(C1CCC1)C C1(NC(CCC2CCN(C(C(CC=CCC)C)=O)CC2)=O)CC2(CCCCC2)C1 CCCCCC(F)C(=O)N1CCC(CC(=O)Nc2cccc(O)c2)C1(C)C C(=O)(CC(C(F)(F)F)NC(=O)C(C)NC=O)NC(COC)(C)COC C1(C(=O)NC(CNC(c2c(C)ncc(C)c2)=O)C)CC1C1CCCCC1 CCC(CNC(C1CCCCCC1)=O)(CC)C(N)=O.C(=O)(C#CC(=O)N(C)C)N C1(C2(O)CN(C(=O)C3=NOC(C)C3C)C2)(CNC(C2C(C)C2)=O)CC1 C(=O)(C1=C(Cl)CC1)N(C1CC(C#N)C1)CC=O.C1(OC(C)C)CCC1.C C1(NC(C(CC#C)(C)NC(=O)C2=C(C)CC2)=O)CCn2cnnc2C1 c1(C=O)cc([SH](=O)=O)oc1C.C1(C2CC2)(CC(=O)N(CCC)CC)CC1 C#CCCCCCC(=O)NC1CC2CC(NC(c3cc(C(=O)CC)c[nH]3)=O)C2C1 Cc1cnoc1C(N1CC(CCO)(NC(=O)C(CO)c2ccccc2)C1)=O c1(CNC(C2C(CNC(C=C(C)C3CC3)=O)CC2)=O)conc1C C(=O)(CCCC(C)=O)N1C2C(NC(C3(C(=O)NC)CCC3)=O)C(C2)C1 N1(C(C=CCOC)=O)CCC(C2CC2)C1.C(=O)CN(C)C(=O)C1CC1.N C1(CC)C(C(=O)NCCCCCN(C)C(c2scc(C)c2Cl)=O)CCN1C CCCCCCCC(=O)NC(CC(=O)NCCS(=O)(=O)CC)C1CC1 c1cccc(Cl)c1.c1(C2(C(=O)OC)CC2)cn(C)nn1.C1C=CCN1C(=O)C c1(C(=O)NCC2CN(C(C3CC(CC)C3)=O)C2)cc(Cl)c(Br)[nH]1 c1(NCCC(C)OC)ccc(S(=O)(=O)N2CCC3(CC2)CNC(=O)C3)cc1F C1(CC)C(NC(C2CCN2C2CCCC2)=O)CCCN1C(c1ccccc1)=O CC(C)C(F)C(=O)NC1(C)CN(C(C2CC(=O)N(c3ccc(Cl)cc3)C2)=O)C1 C(=O)(C1CCCc2ncccc21)N1CCN(C(CCCCOC)=O)C2C1COC2 C(=O)(C1COCc2ccccc21)NC(CCNC(CCC#C)=O)C N1(C(C=C(CCC)CCC)=O)CCCN(C(c2ccc(CC)s2)=O)CC1 C1(CNC(C2CSC2)=O)CCCN(C(=O)CCCc2cnn[nH]2)CC1 N1(C(c2c(C)scn2)C(=O)N(C)C)CCC(O)(c2cn(C3CCOCC3)nn2)CC1 N1(C(CC2C(C)C2)=O)CC(NC(C2(F)CC2)=O)CC1C C(CC(F)(F)C(=O)N1CCC(C(C)(C)C)C1)n1ccnn1.C(=O)(CO)OC.C c1(NC(C(=O)NCCC)CO)cccc(C(F)(F)F)c1.C(=O)(C1=CSCS1)N c1(C(=O)NC(C(=O)NC2(CC)CCCCCC2)CC)cnn2ccc(Cl)c(F)c12 N1(C(C2CCC(C(C)C)CC2)C(=O)Nc2ccc(F)cc2)CC2CC(F)CC2C1 N1(C(C2CCS(=O)(=O)C2)=O)CC2CCC(C1)N2Cc1ccon1 C(=O)(N=c1cc(C)n(C)[nH]1)c1cn2c(n1)CN(C(c1c(C)cc(F)cc1)=O)CC2 c1(CN2CC(C(N(C(C)C)C)=O)SCC2)cc(F)c(Cl)cc1Cl Cc1cc(C(=O)N(CCCCN(C)C(c2c(Cl)nn(C)c2C)=O)C)nc(C)c1 c1(C(=O)NCC(CNC(Cc2c(C)non2)=O)C)cnn(C)c1N c1(CN2CCCC(CNC(C(CCCCC)C)=O)C2)ccc(F)cc1[N+](=O)[O-] c1(C(=O)NC2CCN(C(Cc3c(C)n[nH]c3C)=O)C2)ccc2c(c1)N(C)CCO2 N1(c2c(C)c(NCC(C)OCCO)ncn2)CCn2c(CCN(C)C)nnc2C1 C(=O)(C1=CCCN(C(c2ccc(C)nn2)=O)C1)N1CC(C(=O)OCC)C1 C(CC(=O)NC(C)C(C)(C)C#N)(C(F)F)NC(C1OCCN(CC)C1)=O c1(C(=O)NC(C(C)NC(Cc2ccc(C)cc2)=O)CO)cc(C#N)c(N)cc1O c1(C(N2C(C(CC)C)CCC2)C(=O)NC2(C)CC2)cc(S(N)(=O)=O)cs1 c1(C=O)cnc2c(c1)CNC(=O)N2.N1(CC)CCCC(C(N2CCC2C)=O)C1.N CC1(CNC(C2COC2)=O)CCN(C(c2ccc(OCC(F)F)cc2)=O)C1 C1(C(N(C)CC2N(C(C(C)CN(C)C)=O)CCC2)=O)CC(=O)C12CCC2 c1(OC)ccn2c(C(=O)OCC3CNCC3c3cncn3C)cnc2c1 N1(C(C(C)NC(COC)=O)=O)CC(NC(=O)Cc2cnco2)CC(C)(C)C1 C1(CNC(C2(SCC)CC2)=O)C(O)C(O)CN1C(C1CCCCC1)=O N1(C(c2n(C)nc(CC)c2Cl)=O)CCC2(CCN(C(c3nc(Cl)cs3)=O)C2)C1 c1(C(N2CCOC(OCC)C(N3CCOCC3)C2)=O)cc(P(C)(C)=O)ccn1 c1(C(N2CCCCC(N(C(C)=O)C)C2)=O)cc(Cl)c2[nH]c(O)nc2c1 C1(C#N)(CC)CCN(C(=O)NC(c2ccc(O)cc2C)C)CC1 N1(C(C(CC(C)C)(C)C)=O)CCCC(C2CCN(C(=O)Cn3[nH]cnc3=N)C2)C1 C1(NC(C(C)CSc2ccccc2)=O)CCCCC1.C12(C(=O)N)CC3CC1C2C3 C=CCCC(C)(C)C(=O)NCC1CCCCN1C(c1cc(C)sc1C)=O c1(NC(C(C)(CSC)NC(CSCC=C)=O)=O)cnc(O)c(F)c1 C1(NC(C(C)(N(C(C(CC=C)C)=O)C)C2CC2)=O)CCCC(C2CC2)C1 C(N=c1cc[nH]c(C#N)n1)C1(NC(c2cnc(C(C)(C)C)[nH]2)=O)CCCC1 Cc1cc(O)nnc1C(N1CC(NC(c2cnc(Cl)s2)=O)C(C)C1)=O c1(CCOC)n[nH]c(=NCC2CC(NC(=O)CC3(C)CCCC3)C2)s1 C(=O)(C(CC)C(C)(F)F)NCC(=C)CCNC(c1cncc(C(F)F)c1)=O C#CC(C(=O)N(C(C)CSC)C)C(C)C C1(CCOC)(NC(C2CC2CF)=O)CCN(C(=O)CC(=O)N(C)C)CC1 Cc1nc2cc(C(=O)NC3CCC(NC(C4(O)CCC(C)CC4)=O)CC3)[nH]c2s1 C(c1cc(Br)ccc1F)=CC(=O)NCC1N(C(C2C(OC)CC2)=O)CC1 c1(C(=O)NC2C(NC(Cc3nc(CC)sc3)=O)C2)ccc([N+](=O)[O-])cc1.O Cc1ccc(C(C)C)c(C(=O)NCCNC(c2cc(F)n[nH]2)=O)c1.C1CC1 Cc1nnc(N2CC(NC(c3nn(C)cc3Cl)=O)C3(CCC3)C2)c(C#N)c1C c1(N2C(CNC(C3ON=C(CC)C3)=O)CCCC2)ncnc2[nH]ccc12 c1(C(N(CC(C)(C)C)C)=O)cn(C)nc1-c1ccoc1.C(C=O)OC(C)=O.N c1(OCC(=O)NC2CCCCC2C(=O)NC2(CO)CCOCC2)cccc(F)c1 c1(C(N2CC(CNC(c3c(C)csc3C)=O)N(C)CC2)=O)cnn2ccncc12 c1(C=O)ccnc2nccnc12.CC1(C(=O)NCC2(C)CC2)CCCS1(=O)=O C1(CC=O)CC2(CCC2)CCO1.C1(F)(CNC(C2C(C#N)C2)=O)CCC1.C N1(C(C2N(C(C)(C)C)CC2)=O)CCC(N=[N+]=[N-])(C(=O)NC)C1.c1ncccc1F C1(NC(c2c(C)con2)=O)(CF)CCN(C(C2CCN(C)CC2)=O)C1 C=C(C)c1ccccc1NC(C1CC(CNC(=O)C(C)CN(C)C)C1)=O C(=O)(C1=NN(C)C(=O)CC1)NCC1N(C(C2C(OC)CC2)=O)CC1 C1(C(=O)NCCC(N)=O)CCCCN1C(=O)C(c1ccc(F)cc1)O CCC(CC)CC(=O)NCC(C)(C1CC1)NC(=O)C(C)NC(C)=O CON1CCC(CC(N2CCC(NC(=O)C(c3cncnc3)C)C(F)C2)=O)CC1 C(=O)(C1=CCCC1C)NCCN(C(=O)C(c1ccc(F)c(Cl)c1)O)CC CCCCCC(O)CC(=O)NC1CC(NC(=O)Cc2csnn2)C(O)C1 c1(C(=O)NC2CN(C3CN(CCC=CCC)C3)C(=O)C2)cc2cnccc2o1 N1(C(CN(C)CC)=O)CC(NC(c2ccn(C)c2C)=O)CC(F)C1 C#Cc1ccc(CC(=O)NC2CC3CC2N(C(=O)CCCS(N)(=O)=O)C3)c(F)c1 C(=O)(CCC(=O)NC(C(=O)N(C)CCC1CCCN1C)C1CCCC1)N(C)C n1(CCC(=O)N)cnc([N+](=O)[O-])c1.CC(CC)NC(=O)CSC(C)(C)C N1(C(C2(CCOC)CC2)=O)CCCCCC(NC(c2cn(C)nc2C)=O)C1 Cc1nc(C(N2CC=CCC2C(N2CC(CC(C)(C)C)C2)=O)=O)cn1C C1(C=O)CC(C)(C)CCN1C=O.C(C(=O)NC(C)C)OC.C(C)(C)C.N O=C(C#CC1CCCCO1)NC1(CNC(C2C=CCCC2)=O)CCCCC1 C(=O)(C1CCCn2c(C)nnc21)N(C1CN(C(CC2(C=C)CC2)=O)C1)C N1(C(C=CC=CC)=O)CCC(NC(=O)Cc2ccc(C)o2)C(C(C)C)C1 c1(C=O)n[nH]c2ccc(O)cc12.C1(C(=O)N)(OCC)CCC1.CCCC1CC1 N1(C(c2cc(C)c(C3CC3)cc2)=O)CC2(CCN(C(=O)C(C)CC3CCC3)C2)C1 CCC1=NOC(CC(=O)N(C)CC2CCN(C(=O)CCN3C(=O)CCC3=O)C2)C1 c1(OC(C)C)ccccc1C(=O)NCC1CC(O)C1.c1(CC=O)ccns1 Cc1cc(F)ccc1CNC(=NCc1ccco1)NCC1(C)CCCCO1 C=CCC(CC=C)C(=O)N1CC(=O)NCC1C(N1CCC(N(C)C)CC1)=O C#CCCC(C(=O)NC(C)CCC)NC(=O)CC(CC)OC C1(CC(=O)NC(c2ccccc2)CNC(CSCCC)=O)CC2CC2C1 C1(C(=O)NCCCN(C(=O)CC2(C)CCC2)C)CCc2ccc(F)cc2C1 C1(CN(C(CC)=O)CCCO)C2CCC1CN(C(=O)Cc1ccc(Cl)cc1)C2 c1(CN(C2CCC(N3CCN(CC=C)CC3)C2)CC)cc(=O)n(C)cn1.CC.O CC1(NC(=O)C=CC2CCCCC2)CCCCC1C(N1CC(O)(C(F)F)C1)=O C1(C)(C(N2CCN(CC#CC)CC2)=O)CCN(C(C2CC(C)C2)=O)CC1 C1(CC)CN(C(=O)C(CCC2CC2)NC(=O)C(C)=CC(C)(C)C)CCCO1 CC#CCC(C(=O)N1CC2(C1)CN(C(=O)C(F)(F)F)C2)c1ccccc1 CCC(C)CCCC(=O)NC1CCCC(CC(N2CCC(C(C)C#N)CC2)=O)C1 C(=O)(C(Cc1ccccc1)C(F)(F)F)N1CCN(C(CC2(C)CC2)=O)CC1 C(C(=O)NC1CC1CC(=O)NCC1(OC)CCCC1)(C(C)(C)C)OC c1(CC(=O)NCC#CCNC(CC(C)N(C)C)=O)ccc(O)c(Br)c1 CC1CC2C(=O)N(CCN(C3CCCCC3)C)C(=O)N12 C(=O)(CCCCCn1cc(CC(O)C2CC2)nn1)Nc1ccc(C)cn1 C=C(C)CC(C(=O)NC(C1(O)CCCCC1)C(=O)NC1CCCSCC1)OC CCCCC(CNC(=O)CSC)NC(=O)C=Cc1cn[nH]c1 Cc1ccc(C(N2CC3CC3(CNC(=O)C3=COCCO3)C2)=O)c(Cl)c1 CCC(CC(C)C)C(=O)NCc1ncoc1C1CN(C(C2CC(SC)C2)=O)C1 c1(C(C(N2CC(O)(CNC(c3ccc(=O)oc3)=O)C2)=O)O)ccc(Cl)cc1Cl C#Cc1cncc(C(N2CCOC(C(C)NC(=O)Cc3cc(C)on3)C2)=O)c1 c1(C=O)cccc(C)c1C.S(=O)(=O)(CC(=O)N1CC(O)CC1)N(CC)CC.C c1(NC(=O)NCC(=O)NC(C2CCCCC2)CNC(C)=O)ccccc1F C1(OC)CCN(CC(N)C2(C)CC2)C(C)(C)C1 Cc1ccc(C(N2CCC(C)CC2CNC(c2nccnc2N)=O)=O)c(F)c1C C=C1Cn2c(C(=O)NC(C)C(CO)NC(c3cnc(C)o3)=O)nnc2S1 C1(C(=O)Nc2cnsc2)CSCCN1C(c1cc(Br)ccn1)=O C=CCCCC(C(=O)NCCCNC(C)=O)NC(c1cc(COC)on1)=O c1(C(=O)NC2CCN(C(CC3CCCN(C)C3)=O)CC2F)cc(Cl)cc(Cl)c1F C(CCC(=O)NCC1(C)CC1(F)F)OCCC.C1(C=O)(CC)COC1.N N1(C(C=CC(=O)OCC)=O)CC2CN(Cc3ccc(OC)c(C)c3)C2C1 C1(C(=O)NCCC(C)(C)Nc2ncnc(C)c2Br)CCOC2(CCC2)C1 C#CC1CN(C(c2cc(CC)ccn2)=O)CCN1C(=O)CC(C)=C(C)C c1(C(=O)NC2CCCCC2C(N2CC3COCC3C2)=O)n[nH]c2c1CS(=O)(=O)C2 C1(C(=O)NC2C(NC(c3cnc(CC)s3)=O)CCCC2)CC2CCC1C21CC1 CCCC(CNC(=O)COCCNC(c1conc1C)=O)CCO N1(CC(N2CCC(CCN)C2)=O)CCCNC1=O c1(C(=O)NC2C3CCN(C(C=NOC)=O)C32)ccc2cc(Br)ccc2n1 C#CC1CN(C(=O)CC(CC2CC2)NC(C2CC(=O)OC2(C)C)=O)CCO1 c1(C(=O)NC2CN(C(C=C3CCN(C)CC3)=O)CC2(C)C)csc2cccnc12 c1(C(C(=O)NCCCNC(c2cc(N)c(F)cn2)=O)O)cccc2c1OCC2 N1(C(C(CCC)F)=O)CCCCC(NC(=O)C(F)=C(C)C)C1 C1(c2ccccc2)CCN(C(c2cnc(O)s2)=O)C1.C(CC1CC1)(C(=O)N)OC C=C(C)CC(C(=O)N1CCC(C(=O)OC)O1)NC(=O)C(C1CCOCC1)F N1(C(c2c(SC)cnn2C)=O)CCC(NC(c2cccc(F)c2Cl)=O)C(O)C1 c1(OCC)cc(C#N)c(NC(C2CN(Cc3cncs3)CCC2O)=O)cc1OC C12(CNC(C3CC=CC3)=O)CCCC1N(C(C1CC13CCSCC3)=O)CCC2 c1(CC(=O)OCC2(CC(F)F)CCC2)cccc2ccccc12 Clc1cccc2c1C(Nc1nc3ccccc3c(=NCc3ccc[nH]3)[nH]1)CCO2 CC(C)C(C(=O)N1CCC1CNC(c1ccccn1)=O)n1cnnn1 N1(C(c2c(C)nc(F)cc2)=O)CCCC2(CCCN2C(c2ncccc2F)=O)C1 N1(CC(=O)NCC2CCCCO2)CCN(C(=O)CC2CCCOC2)CC1 C1(CNC(C(C)(C)SC)=O)CCN(C(c2cc(C)n(C(C)C)c2)=O)CC1C C1(COC)(NC(=O)Cc2cccnc2)CCN(C(=O)CNC(C)=O)C1 c1(CN2CCC(C#N)(C(=O)OC)CC2)cn(C)c(=O)n(C)c1=O c1(OC)cc(C(N2CCC(O)CC2)=O)c(F)c(Cl)c1.C(=O)CN(C)C1CC1.N C1(N(C(C2(CCCC)CC2)=O)C)CCCN(C(c2cnns2)=O)CC1 N1(C(c2nc(OC)c(C)s2)=O)CC(CNC(c2ccc(Cl)cc2N)=O)CCC1C c1(OC)cc(-c2nc(CSc3ccccc3)nn2C)cn(C)c1=O.C1CCCCC1 O=C(C1=CC2CCCC12)N1CCC(N(C(=O)CCC=CBr)CCO)CC1 C1(OC)CCN(C(C23CC(CO)(CN2C(c2cncnc2C)=O)C3)=O)CC1(C)C C(=O)(C1=C(C)C(C)(C)OC1=O)N1CCC(O)(CC)C1.c1(OC)ccc(C=O)s1 C(CC(F)F)(C(=O)O)N(C(=O)CCc1cn(CC2CCCO2)nn1)C C(C(=O)NCCCCNC(C1CC(O)CN1C(N)=O)=O)(C(C)(C)C)OC C1(OC)CCCC1C(=O)NC(C1CCN(C(=O)C(O)CC2CCCC2)C1)(C)C C(c1ccc(F)cc1F)=CC(N1CC(NC(c2c(C(C)(C)C)ccnc2)=O)C1)=O c1(C(=O)Nc2c(C(=O)OC)sc3ccccc32)ccc2c(c1)C1(CC1)CN2 C(CC(C)C)(C(=O)N)OC.C1(F)CCCC1.c1(C=O)cc(C2CC2)n(C)n1.C C1(CNC(NC2CCS(=O)(=O)C2)=NCC2CC=CC2)C2CC3CC(C2)CC1C3 C1CN(C(=O)CN(C)C(C)C)CC1C(F)(F)F.CCC(C(=O)N)n1ccnc1 N1(C(c2ccc(C)[nH]2)=O)CCOC2(CCCN(C(c3cncc(N)c3)=O)C2)C1 N1(C(CNC(C2C(C)C2)=O)=O)CC(O)CCC1C(=O)NC1CCCCNC1=O C1(CC(=O)NCC)C(NC(=O)COc2cccnc2)C1(C)C N1(C(Cc2c(C)non2)=O)CCN(C(=O)COc2ccc(Cl)c(Cl)c2)C(C)C1C c1ccc2ncc(Cl)n2c1.N1(C(=O)OC(C)(C)C)CCC(NC(=O)N)CC12CC2 C(=O)(C1=C(C)C(C)(C)OC1=O)NC(CNC(C(CC)C)=O)(C)CO C(=O)(CCC(=O)NCC)NCCC1(CNC(C2C(=C)CC2)=O)CC1 c1(C(=O)NC(CCNC(c2c(C(C)C)cccc2)=O)C)c(O)cc(F)cc1F N1(CC(C)NC(=O)C2=CCCC2)CCN(C(=O)C(=Cc2cccnc2)F)CC1 c1(N(C(=O)NCCS(=O)(=O)N(CC)CC)C)cc([N+](=O)[O-])ccc1Cl C(=O)(C(O)CNC(=O)CC1CCC(=O)C1)N(C)CCOCCCO c1(C(=O)NCCCC(C)NC(C=COCC)=O)c(OC)cccc1Cl.C1CC1 CCC(CCC(=O)N1CC(CO)C(C)C1)NC(=O)COCCC(C)C C(=O)(C(C)CS(C)(=O)=O)NCCC1N(C(C(C)=C2CCCC2)=O)CCCC1 C1(C=O)CCS(=O)(=O)C1(C)C.C(C)(C(=O)N(C)CC)(C(C)C)NC(C)=O C12(CNC(C(CCC)CC)=O)CN(C(c3ncn(CC)n3)=O)CC1CCO2 C(=O)(C1CCOc2ccccc21)NC(CC)CNC(=O)CCCC1CCCCC1 c1(C(=O)NC2CCN(C(CC3(C#N)CCC3)=O)C2)cncc(F)c1C(F)(F)F C1(OCC)(CNC(=NCCc2cnccn2)NCC(F)F)CCCS(=O)(=O)C1 C1(CC(=O)NC(CNC(Cc2cn(CC)nn2)=O)COC)OCCC1(C)C N1(c2cc(C)ncn2)CCCC(O)(CNC(c2ccccc2-c2cnco2)=O)C1 CCN=c1[nH]c(C(=O)N(C2CCCCN(C(C3(COC)C=CCC3)=O)C2)C)cs1 C(=O)(C(CCOCC)NC(c1cc(CC)ncn1)=O)NCC(CCC)O N1(C(Cc2c(C)ccs2)=O)CCC(O)(CN(C)C(c2cc(CO)n(C)n2)=O)C1 C(=O)(CC(C(F)(F)F)NC(=O)C(F)C(C)(C)O)NC12C(C)OC(CC1)C2 N1(C(c2ccc(OCF)cn2)C(=O)NCCSC)CCC2CCCCC12 C#CCCC(C(=O)NCC1(C=C)CCOCC1)NC(C1CCCC1O)=O S(=O)(=O)(c1cc(Cl)sc1C(=O)O)N1C2(CN(S(CCC)(=O)=O)C2)CCC1 C1(NC(Cc2ccn(CC)n2)=O)CC(CO)N(C(=O)CCOC2CCC2)C1 c1(C(N2CC(F)(CNC(CCCOCC)=O)C2)=O)ccnc(S)c1 N1(CC=C)CCCN(C(c2coc(CNC(=O)C(C)SC)n2)=O)CC1 C(N=c1[nH]c(Cl)nc(C2CC2)c1F)C1C(C)CN(C(=O)C(C)O)C1 Cc1noc(Cl)c1CCC(=O)NC1CC(C)N(C(=O)COC2CCC2)C1 N1(C(C(C(C)C)C)=O)CC2CC1CN2C(c1cc(-c2cc(F)ccc2F)on1)=O CC(C)(C)C(C)(O)C(=O)N1CC2(COC(C)C2)C1.C1(CCC(=O)N)CCOCC1 c1(C(=O)NCCCC(CO)NC(C2(SC)CCC2)=O)cccn(C)c1=O c1(C(C)C)cc(C(=O)NC2CN(C(=O)CCC3CCC3)CC2C)cc(O)n1 C(=O)(CCC(=O)N1CCC1CNC(=O)C(C)(C)Nc1ccccn1)OC C1COCCN(C(=O)C(C)(C)CC)C1.c1(OCC)ccc(NCC(=O)N)cc1.C c1(CCC(N2C3CN(C(CN(C)C)=O)C(C3)C2)=O)nc(O)c2cnn(C)c2n1 CC1(C)C2CCC1(C)C2C(N1CCN(C(C2(C=O)CC2)=O)CC1CCO)=O.N N1(C(c2n(CC)ncc2)=O)C2CCC1C(CO)N(C(C1CCCN1C)=O)C2 C1(NC(c2cc(OC)cc(Br)c2)=O)CC2CN(Cc3cccnc3C)CC2C1 C#Cc1c(NC(N2CCC(O)(c3ccccc3F)CC2)=O)c(C)nn1C c1(OC)ccccc1C1CCN(C(=O)NCC2CCC(OC(F)(F)F)CC2)C1 CC(C)C(C(=O)N1CC(CCNC(C2(C(C)(C)O)CC2)=O)C1)C(C)C c1(CNC(C(C2CN(C(=O)Cc3cncn3CC)C2)OC)=O)ccnc(O)c1 CN=c1ccc(C(=O)NCCC(C)(C)C(=O)NCC23CCCC2CCC3)c[nH]1 N1(CCC)CCCC(C(N2CCOCC2CN(C(=O)Cc2c[nH]nc2C)C)=O)C1 c1(C(N2C(CNC(C3CCCCS3(=O)=O)=O)C=CC2)=O)cccc2c1NCCC2 N1(C(=O)Cc2csc(-c3ccccc3)n2)CCNCC1c1ccc(F)cc1 c1(OC)ncccc1S(=O)(=O)N1CC(NC(=O)CCc2cccs2)C(C)C1 c1(C(=O)NC(C2N(C(C(C)NS(CC)(=O)=O)=O)CCC2)C)cccc(O)n1 N1(C(CC(C)C2CC2)=O)CCC(C2CCCN(C(C3(C)COC3)=O)CC2)CC1 Cc1nn(-c2ccc(F)cc2)c(C)c1C=CC(=O)N(C)Cc1nnc(O)o1 C1(CCNC(C2(C(C)NC(c3cccs3)=O)CC2)=O)NC(=O)NC1=O N1(C(c2ccc(OCC)nc2)=O)CC2CCC(NC(=O)CN3CCOCC3)C2C1 c1(NCC2C(CC)C2)cc(N2CCC(C(O)C(N)=O)CC2)ncn1 C12(C(N(CCC(=O)Nc3cc(CC)ncn3)CC#C)=O)CC(C)(CCO1)C2 C(=O)(C(C)(C)CC#N)NCC1CN(C(c2c(C(C)C)noc2)=O)CC1O N1(C(C(C)(C)O)=O)CCCC(C)(NC(=O)CC2CCN(CC(F)(F)F)C2)C1 N1(C(=O)NCCCn2cnnn2)CCC2(C1)CC(F)(F)C2 C1(C(N2CC(NC(CCCC)=O)CC3(C2)CC3)=O)CN2CCCCC2CO1 c1(CN(C(=O)C(O)C2CN(C(c3cncc(O)c3)=O)C2)C)ccc(O)nc1 C1(NC(=O)CCc2cn[nH]c2)CCCN(C(=O)Cc2cnc(C(F)(F)F)s2)CC1 c1(C(N2C(CCNC(C3CCCCS3(=O)=O)=O)CSCC2)=O)ncn2c1CCC2 C=C(C)C(C)(O)C(=O)N1CCC(O)(CNC(C2CC(n3ccnn3)C2)=O)C1 Cc1noc(C)c1CC(=O)NCC1COCCN1C(c1ccc(C(N)=O)o1)=O c1(C(=O)NC(CCNC(C(C(=O)OC)(C)F)=O)C)c(C)[nH]c2ccccc12 O(C1CCc2c1cccc2[N+](=O)[O-])C(c1sc2ccc(OC)cc2c1C)=O C1(NC(C(C)c2ccon2)=O)CCN(C(c2cncc(Br)c2)=O)CC1O c1(CNC(C(c2ccoc2)NC(C(CC)N(CC)CC)=O)=O)ccncc1Cl C1(C(=O)NCC(C)CN(C)C(c2cc(CC3CC3)on2)=O)CCC2CC12 c1(C2N(C(=O)Nc3cc(Cl)c(Cl)cc3F)CCCC2)nc2ccc(Cl)cc2[nH]1 c1(C(N2CCC2)=O)cn2c(n1)CCC2.C1(C(=O)NC)CCCN1C1CCOCC1 N(C1CN(C(=O)C(O)c2ccsc2)Cc2ccccc21)C(CCCCC(C)C)=O N1(C(c2ccn(CCCC)n2)=O)CC(NC(c2cc3n(c2)CCC3)=O)CC1(C)C CCC(CC)C(C)NC1(C)CCC1 C1(N(C(=O)CSc2ccccn2)C)CCCCN(C(=O)C(F)(F)c2nccs2)C1 N1(C(c2nc(C)on2)C)C2CCC1CC(NC(c1cnc3[nH]nnc3c1)=O)C2 N1(C(c2c(C)ccc(OC)n2)=O)CC2CCC1CC2NC(C1C=CCC1)=O c1(C(=O)NCC(C(=O)N(CC(=O)OC)CC#C)O)cnnc(C)c1C C(=O)(C1CCc2snnc21)NC(C(C)NC(C(C(C)C)OCC)=O)CO C12(CNC(CCC(=C)C)=O)CCC(Nc3ccnc(SC)n3)(CO1)C2 C1(NC(C(CC#C)C)=O)CN(C(c2ccccc2)=O)CC1(C)C.C(=O)(N(C)C)N c12ccc(cc1Cl)c(=O)[nH]2.c1(C(CC(C2CCOC2)=O)=O)ccccc1 c1(N2CC(CN(C(=O)C=CI)C)C2)nc(Cl)nc2c1SCC2 C1(NC(c2cn(CC=C)nc2)=O)CCOC(C(N2CC(SC)C2)=O)C1 CCC(C=O)NC(N)=O.C12(C(NCCCC)=O)CC(C1)C2.C1CC1.N c1(C(=O)NCC(CC)NC(c2cc(C)co2)=O)c(C)nn(C2CCCCO2)c1C N1(C(Cc2cc(C)[nH]n2)=O)CCCCC1CN(C(=O)C(C(C)O)N(C)C)C CCC(CNC(=O)CC(C)(C)C)(CC)C(=O)NCC1(n2cccn2)CC1 C1(C(N2CC(CCC#C)C2)=O)CN(C(c2cocc2C)=O)CC1CC c1(C(=O)NCC(CNC(COCC)=O)O)cn(-c2ccn(C)n2)cn1 C(C)(C(=O)N)(C1CCC1)NC(CN(C(COC)=O)C)=O.C1(O)CCSC1.C c1(CCCC(=O)NCCCCNC(=O)C(c2ccccc2)O)ccccc1Br O=C(C1=CCS(=O)(=O)C1)N1CC2(C1)CN(C(c1coc3ccccc13)=O)C2 Cc1cn(CC(F)(F)F)[nH]c1=NC(=O)C1CCCC(O)(c2nccn2C)C1 Cc1ccc(NC(=O)NCC(=O)NC(C)C)cc1.c1(C(=O)N)ccncc1Br n1(CC)nc(C(=O)N(C(C)(C(=O)N2CC(C)(CF)C2)C2CC2)C)cc1C C#CCC(C)C(=O)NC(CNC(=O)CSC(C)C)C(C)(C)C C1(C=O)CCC2(CC2)N1C(=O)CC1(C(=C)F)CCC1.C=CCC1CCC1.N N1(CC(C(=O)NC2CCOCC2)N(CCCCC)CC)C(=O)c2ccccc2C1=O CCC(C(=O)NC1CCCC1NC(=O)C(Cc1ccccc1)N(C)C)N(C)C CCC(c1ccccc1)=CC(=O)NCC1CC2CC2N1C(c1cncc(Cl)c1)=O CN1C2c3ccccc3CC12.C1(C)(C(CC=O)=O)CCCCC1 c1(CC(C(N2CCC(N(C(C(COC)OC)=O)C)CC2)=O)C)c(C)nn(C)c1C N1(C(c2ccc(=NC)[nH]c2)=O)CC(NC(c2cc(F)ccc2C)=O)CC(C)(C)C1 N1(C(c2nccc(C)c2N)=O)CCCN(C(=O)Cn2nnnc2C2CC2)C(C)C1 c1(C(N2CC(NC(c3ccc(F)cc3F)=O)C(F)C2)=O)ccc(Br)c(Cl)c1F C1(NC(c2c(C)cc(=N)[nH]c2)=O)CN(C(c2cc(Br)ccn2)=O)CC1C1CC1 c1(C(=O)NC2CC(N(C(c3c(COC)cco3)=O)C)C2)cnncc1OC C1(C(N2CC(C)C(NC(c3c(Cl)nn(C)c3Cl)=O)C2)=O)CCC2(CC1)CC2(F)F N1(C(c2n(CC)ncn2)=O)CC2CCC2(CCNC(=O)COC2CCC2)C1 CC(C)C1=NOC(C(N2CC3CC(C2)C3)=O)C1.C12(C(=O)N)CC(C#N)(C1)C2 C1(NC(=O)NC2CCCCC2OC(F)(F)F)CC2CCCCCCC12 C1(C(N)=O)CCCN(C(C2CCC(NC(c3ncccc3Br)=O)CO2)=O)C1 c1(CNC(C(=O)NC)(C)C)c(C)cc(OC)cc1O C(=O)CC1=NN(C)C(=O)C1.c1(CC)c(C(=O)NCC)[nH]c(C)c1C(N)=O c1(C(=O)NCC2C(C)CN(C(c3cnn(C)c3Cl)=O)C2)c(F)cc(F)c(F)c1F C(=O)C1=CCC(C)(C)CC1.S(=O)(=O)(CC(=O)NCCC1CCC1)NCC C1(N(C(=O)C(=O)NC2CC=CC2)C)CCN(c2ccccc2Cl)C1=O c1(C(=O)NCC(CNC(C(CC)OC)=O)F)nccc(Cl)c1F N1(C(C(C(C)C)(C)O)=O)CCC(C)C(F)(F)C1.c1(C=O)cc(C(C)(C)C)n[nH]1 N1(C(c2cc(C(C)C)n[nH]2)C(=O)NC2COC2)CCC(CO)CC1C c1(C2(NC(=O)NCCCC3C(C)C3)CC(O)C2)ccccc1Cl C1(F)(CNC(c2scc(C)c2)=O)CCC(NC(c2n[nH]cc2C2CC2)=O)C1 CC1CN2CCN1C(C(=O)NC(C)(C)CCNC(=O)CCc1ccccc1C#N)C2 C1(NC(c2nc(CCCCC)sc2)=O)CN(C(c2occc2F)=O)CC1O C(=O)(C1CCCc2scnc21)N(CCN(C)C(c1cc(S(N)(=O)=O)c[nH]1)=O)C c1(N2CCCC(CC=C)(NC(=O)C3=COCCC3)C2)cc(C)ncc1C#N c1(CN(CCOC)C)cccc(CNC(=O)NC2CC3C=CC2C3)c1 C=CC(CC(=O)N1CCC(CO)(NC(c2cc(C)[nH]n2)=O)C1)c1ccccc1 N1(C(c2n(C(C)C)cnc2)=O)CCCC2CN(C(C34CCC(C3)C4)=O)CCC12 C1(C(=O)Nc2ccc(C)c(I)c2)C2CCCC1CN(C(c1cccnc1O)=O)C2 c1(C(=O)OC)ccc(C(=O)NC)cn1.c1ccc(C=O)cc1.C1(CC)CCC1 C12(CNC(CCC3N(C)CCC3)=O)CC(CN1C(=O)Cc1cccc(Br)c1)C2 c1(C(N2CCC(NC(c3cc4c[nH]nc4s3)=O)C2)=O)cc2cccnc2[nH]1 C(=O)C(F)(F)CC(C)C.c1(C(N2CC(OC)C2)=O)c(C(F)(F)F)cnn1C.C C(C(=O)NCCCN(CC(=O)N1CCC1)CCO)(C1CCCC1)OC C=CC1(CC(=O)NCC(C)CC2CCC2)CN(C(C2CC23CCCC3)=O)C1 N1(C(C=Cc2ccc(CC)o2)=O)CC(C)N(C(c2cnc(O)c(Cl)c2)=O)CC1C c1(OC)ccc(F)cc1CC(=O)NCC(C)(C)NC(C12CCCC1C2Br)=O C1(NC(CSCC=C)=O)CCC2(CCN(C(c3cn(C)nc3C)=O)CC2)C1 C(C)(C(=O)N1CCC(C(=O)NC(CO)CC=CC)O1)OCCC=C C(CS(=O)(=O)NC(N1CCC(n2cc(CO)nn2)C1)=O)C1(OC)CCC1 C1(NC(c2nc(CC)sc2)=O)C(C)CCN(C(c2ccc(C)cc2)=O)C1C c1(C(=O)NC2CC(n3cc(C(=O)OC)nn3)C2)ccnc(OC)c1Br CC1=NNC(=O)C1CC(N1CCC(C(=O)N(C2CCC3CC23)C)(CF)C1)=O C1(NC(c2c(CC)scc2)=O)CCC(NC(=O)COC2CCC2)CC1 C(CCC)(C(=O)N1CC(NC(C2(C)CC2)=O)C2CC12)=CCC CC(C)C(F)(CNC(=O)CC(C)(C)OC)C(=O)N1CCC(F)(C#N)C1 c1(C(C)=O)cnc(Cl)nc1N1CCC(N(C)C(C2(OC(C)C)CCC2)=O)C1 C1(C)(C(N(C2CCN(C(c3ccc[nH]3)=O)C2)C)=O)CCN(C(C)=O)C1.CO.C C12(NC(CCCC=C)=O)CCCCC1N(C(c1ncc3[nH]ncc3n1)=O)CC2 c1(CC(=O)NC2(CCNC(C=CC)=O)CCCC2)ccc(O)cn1 CN1CC(C(=O)NCC2CC(NC(=O)OC(C)(C)C)C2(C)C)NC1=O c1(C(=O)NCCCOCCNC(=O)Cn2cc(Br)cn2)cccc(F)c1 C1(OC)CC(CC)N(C(=O)CC2CSCCO2)C1.C(=O)(CC(C)C)N.C(C)=O N1(C(C2CCC(=C)CC2)=O)CCC(F)C(NC(=O)CC=CCC)C1 C1(NC(c2cncc(SC)c2)=O)CC(C)CN(C(c2cccc(O)c2C)=O)C1 N1(C(C=NOC)=O)CCCC1(C)C(=O)N(C1CC(O)C1)C c1(C(NC(C)C)=O)cnc(C2CC2)o1.C(=O)C(C)(C)C.C(=O)CC.CC c1(NC(CCC=C)(C)c2nnnn2-c2ccccc2C)ccc(Br)c(OC)c1 C1(C(=O)Nc2cn(CC#C)nc2)CCCCN(C(c2cnn(CCF)c2)=O)C1 c1(C(=O)OCC)cc(=NC(=O)C2(C)CCN(Cc3cnc(F)c(C)c3)C2)[nH][nH]1 C#CCC(CC(=O)NC1CCN(CC)CC1C)NC(C1CCN(C)CC1)=O CC1(C(=O)NC2CN(C(=O)C=Cc3ccc[nH]3)CC2O)CCC2(CC1)CC2 c1(C(=O)NC(CNC(CC2(C)CC2(Cl)Cl)=O)(C)CO)ccc(N)c(Cl)n1 C1(NCC(=O)NCCCCC2(NC(=O)COC(F)F)CC2)CCCCC1O C1(CNC(C(C(C=C)C)C)=O)CCCC(F)(F)CC1 c1(N2CC(OCCNC(c3nn(C)c(F)c3)=O)C2)cc2nncn2cn1 C1(C(C)NC(CC2C(C)CC2)=O)CCN(C(=O)Cn2cnnc2O)C1 C(=O)(C1=C(Cl)CCCC1)NCCC1(O)CCCN(C(CC2CC(=O)NC2)=O)C1 N1(C(CC(C=C)C)=O)CCC2(CCC(N(C)C(c3cnc(CC)s3)=O)CC2)C1 C(N=c1[nH]c2cccc(C)c2s1)C1CN(C(CC)=O)CC1(C)C C1(C(=O)NC(c2ccc(OC)cc2F)C(=O)OCC)Cc2nnc(C)n2C1.O CC1CSCCN(C(c2coc(CNC(=O)CC3CC(=O)C3)n2)=O)C1 c1(N(CCN(C)C(=O)N(C2CCCCC2)Cc2cncn2C)C)ccccn1 CC1=C(C(=O)N2CCC(C)C(CNC(=O)COCC3CC3)C2)CCC1 C=CC1(CC(N2CC(Cn3ccnn3)C2)=O)CN(C(C2(C)CNC(=O)C2)=O)C1 C1(COCC)(C)CCCN1C(=O)CC(C)F.c1(C=O)ccc(C2CC2)cc1 C1(C(N2CC3(CN(C(=O)Cc4ncc(Cl)s4)C3)C2)=O)CC(c2ccccc2)=NO1 C1(C=O)CC2(CCC2)CN1C(c1ccc(C#N)[nH]1)=O.c1(OC)cccc(C)c1.N c1(CC)cccc(C)c1C(=O)NCC(C)(C)NC(=O)C.c1c(Cl)cccc1Cl C(CCC(N)=O)(C(=O)NC1CC1)n1cc(-c2c(C)nc(F)cc2)nn1 C1(F)(C(=O)OCC)CN(C(=O)NCC2CCN(CC(F)F)CC2)CC12CC2 C1(C(N2C(COCC)CCC2)=O)C(O)CCN1C(c1ccc(Cl)cc1)=O n1(CCOC)nc(C)cc1C(=O)Nc1cncc(C(=O)O)c1 C1(NC(c2ncc(CC)cn2)=O)CCCC12CCN(C(C1CCCCS1)=O)CC2 C1(OC)C(OC)CN(C(C2CC=CCO2)=O)C1CNC(=O)C=C(C)Cl Cc1c(C(N2CCCC(P(C)(C)=O)C2)=O)cc(S(C)(=O)=O)cc1Br Cc1nn(CC(N2CCC2CC(=O)NCCC2CCN(C)C2)=O)c(=O)o1 c1(OC)ccc(C(=O)NCC2CC(O)CN2C(c2cnc(C)s2)=O)c(O)c1 C1(C)(C(N(C(C)C(=O)O)C)=O)CCCN(CC2CC(=O)N(c3ccccc3)C2)C1 C1(CC(=O)NC2C(C)CN(C(=O)C(=O)NCC(F)F)C2)CCCCC1(C)C c1(C(=O)NCC2C(C)(Br)C2)cccc(C2CCNCC2)c1 N1(C(CC2(NC(C(C)OCCN(C)C)=O)CC2)=O)CCC(C2=NOCC2)C1 C1(NC(Cc2ccc(CCC)cc2)=O)CC2CC1N(C(c1cc(C)on1)=O)C2 N1(C(CCSCCC)=O)CC(NC(c2nn(C)cc2Br)=O)CCC1C c1(OCCC)ccc(Br)cc1S(=O)(=O)NC(c1ccc(S(C)(=O)=O)cc1)C C1(NC(c2ccc(Br)o2)=O)CC2(C1)CC2NC(c1ncccc1Cl)=O N1(C(C(C)(C)SC)=O)CCC(NC(=O)C(C)(C)C(C)(F)F)C(CO)CC1 CP(C)(=O)CN(c1ccccc1)C(C1(CS(N)(=O)=O)CC1)=O C(C(C)(C(=O)N)NC(c1ccn(CC)c1C)=O)SC.C1(CC)CCC(C)(C)C1 C1(CNC(COC2(C)CCCC2)=O)CN(c2ccnc(CO)n2)CCC1(F)F N1(C(CCC(C)N(C)C)=O)CCC(F)(CNC(=O)C#CC(C)(C)C)CC1 C(C)(N=c1[nH]nc(C2CC2)s1)C1N(C(c2c(C)nc(CC3CC3)s2)=O)CCCC1 C1(CC(=O)NC2CC3N(C(C(CC)(C)O)=O)C(CC3)C2)C2CC3CC(C2)CC1C3 N1(C(C(CC)NC(C)=O)=O)CCOC2(CCN(C(=O)CCc3nc[nH]n3)C2)C1 N1(C(CC(CC)CC(C)C)=O)Cc2ccnn2CC(NC(=O)C(C)CO)C1 C(=O)(C1SCCc2ccccc21)N1CC(CCNC(c2cc(C)nnc2)=O)C1 C1(C(=O)NCC2CN(CC)C(=O)O2)CCN(C(c2csnn2)=O)C(C)(C)C1 N1(C(C(C(C)C)F)=O)CCCN(C(=O)CN2CCCNS2(=O)=O)CC1C C=CCCCC(C(=O)NC1CC(CC)C1)NC(c1c[nH]c(C#N)c1)=O C1(CCC(=O)N(C(C)CO)CC)CCCCN(C(c2cc3n(n2)CCC3)=O)C1 CC1CCCC(CN)N1C(=O)C(=O)NCC(C)(C)C(C)(C)O C1(NC(C2(NC(c3c(CC)[nH]cc3)=O)CC(F)C2)=O)C=CC(C)(C)CC1 c1(OCC)ccc(Cl)c(C(=O)N)n1.c1(CC=O)ccc(C#N)cc1.C(C)CC N1(C(c2cnc(C)nc2)=O)CCC2C1CCCN2C(c1coc(Cl)n1)=O C1(F)(CNC(C(C2CCCC2)OCC)=O)CN(C(C2CC(C)CO2)=O)C1 C1(NC(Cc2c(C)cc(Cl)cc2)=O)COC2(C1)CN(C(=O)COC1CC1)C2 N1(C(c2ccc(SC)o2)=O)CCCCCCC1C(=O)NOCCC(C)O C1(OC)CCCCC1C(=O)NC(C1CCN(C(c2nocc2C)=O)CC1)C c1(SC)cc(NNC(=O)CNC(=O)CCn2c(C)nc3ccccc23)ncn1 C(=O)(C(C)(F)C(=O)NCCC1CCN(C(=O)Cc2ccsc2C)C1)OC Cc1nonc1CC(=O)NCc1c(C(N(CC(CN(C)C)O)C)=O)[nH]cc1 n1(CC(=O)NC2C(CC)N(C(=O)C(O)C3CC3)CC2)ccc2ccc(F)cc12 Cc1cnc(C(=O)NCC2(CNC(C3CCCN3C(C)C)=O)CC2)nc1 c1(-c2n(CCOC)nc(-c3ccc(Cl)cc3)n2)cnc(OC)c(Br)c1 C1(C(=O)N)CCOCC12CCC2.C=C1CC2(C1)CC(C(=O)NCC1CCC1)C2 c1(CNC(CCc2c(C)cc(Br)cc2)=O)c(F)ccc2cccnc12 c1(C(C(=O)NC2CCOC2)N(C(C)C=O)CC)ccccc1.CC(F)(F)F.O c1(C(N2CC(C(N3CCC3CO)=O)C2)=O)cnc(Cl)c(F)c1 C1(C)(CNC(C2CC(C)OC2C)=O)CCN(CC(N2CCOC(C)C2)=O)CC1 C1(NC(C=CSC)=O)CC2CN(C(C3CCC(C(C)(C)O)CC3)=O)CC12 C(CN=c1[nH]c(=NCc2cnsc2)c2cccc(F)c2[nH]1)=CCCOC C1(C(NC)=O)CNC(=O)C(C)(C)C1.N1(CC(N2CCCC2)=O)CCOCC1=O.C C(=O)(C1c2c[nH]nc2CN1C(=O)Cn1ccnn1)NC(c1ncccn1)C S(=O)(=O)(CC(=O)N(C1C2CN(C(c3sc(F)cc3Cl)=O)CC12)C)NC C1(CC)CC(CC(=O)NC(C2CCN(C(c3ccnn3C)=O)C2)C)CCO1 C1(C)(C(=O)NCC(CCOC)(C)C)CC(O)CN1C(=O)CC1(O)CCCC1 C1(CN(C(CCCc2onc(C)n2)=O)C)CC(F)CN1C(=O)CC=C(Cl)Cl Cc1c(N)ccc(C(=O)NCCC(C)NC(c2cscc2F)=O)c1F c1(C(=O)NCCCCN(C(C(C)Oc2ccccn2)=O)C)cn(C)nc1C(F)F Cc1scc(CNC(C2(CCNC(C3(C)CCCS3)=O)CC2)=O)c1C.C N1(C(=O)NCC(COC)C)CCC2(CCC2C)CC1.C(C)(C)C.C(=O)N c1(-n2cc(CCNC(c3cccc(C(F)(F)F)c3)=O)nn2)ccc([N+](=O)[O-])cn1 C1(=O)n2cnc3c(ncnc23)N(C)CCCN1.N1(C(=O)C2CC2)CCCC1 c1(C(N(C2CCN(C(c3nccc(OC)c3)=O)C2)C)=O)cccc(C)c1C N1(C(c2scc(C)c2C)C(=O)NCCCOC)CCN(C(C)C)C(=O)C1 C(c1cnn(C)c1C)=CC(N(CCNC(C=NOC)=O)CCOCCO)=O c1(C(=O)NC(CC)CNC(=O)C(F)(F)COC)nc2ccc(Br)cn2n1 c1(C(=O)NC(CCCCNC(C2(OC)CC(C(F)F)C2)=O)C)cnc(C)cc1Cl C(=O)(C#CC1(C)CCCO1)NC1CCCN(C(c2cccc(C)c2O)=O)C1 n1(CC)nc(C)cc1C(=O)NC1CC(CNC(=O)C(=O)N(C)C)C1 C#Cc1ccc(C(=O)NC(CC2CC2)C(=O)N2CCCC2CC)cn1 CC(C)CC(O)C(C)C(=O)N(CCCC(=O)N(C1CCCCCC1)C)C C1(NC(COC2(C#C)COC2)=O)CCOCC1.C(c1cnc(C)s1)=CC(=O)N N1(C(C(C(CC)C)O)=O)CCC2CCN(C(c3cn4cccc(C)c4n3)=O)C2C1 c1(CN2CCC(C)(CC(=O)N(CC(=O)O)C)C2)nc(O)c2sccc2n1 C1(C(C#C)C)CCN(C(=O)NCCOCCC2CCOCC2)CC1 CCC(C)(O)C(=O)NC1(CC(N2CCC(OC(N)=O)CC2)=O)CC1 C1(OC)CN(C(C2(C)CC(C#N)C2)=O)CC1.c1ccccc1.C1(C(=O)N)CC1 C=C(C)C(C)(C)C(=O)NCC12CC1CN(C(c1cn(C)nc1Br)=O)C2 C(=O)(C1=C(C#N)CCC1)N1CC(CC(=O)N(C(CCC(C)C)C)C)C(C)C1 c1(C(=O)NCC2N(C(c3ccc(C(C)(C)C)[nH]3)=O)CCC2)nnc(O)cc1O CC(C)C(O)C(F)(F)C(=O)N1CCC1C.c1(C=O)nn(CC(F)(F)F)cc1Cl.N c1(C(c2nnnn2CCCC)NCCCC=C)cc(C)on1 C1(CNC(C2(CCC=C)CC2)=O)CN(C(=O)C(C)(C)n2cnnn2)CCN1C c1(CC=O)cccc(Br)c1F.c1(CC)onc(C)c1C(=O)NCC1CC1.N C1C(C)CCN1C(=O)CC1CCCS1(=O)=O.C1(OC)CCCC1C(=O)NC C(=O)(C(O)C(C)(C)C)NC1CC(NC(c2oc(C)c(CO)c2)=O)C1 C(C)(C(=O)NC1CCCC1C)(C1CC1)OC.C(=O)C(F)(F)c1cncs1.N c1(C(=O)NCC(CNC(C(C(C)C)O)=O)O)cc2c(s1)CCC2 CC(C)C(C)(O)C(=O)NCC(C)(F)CNC(c1cc(CN(C)C)on1)=O c1(C(=O)NCC2N(C(COC(CC)C)=O)CC(F)C2)cc2c(nn1)CCCO2 Cc1cc(OC(C)C(=O)N(CC(C)NC(=O)Cc2c(C)noc2Cl)C)ccc1Cl N1(C(C(F)=CCC)=O)CC2(C1)OC1(CO)CC2C1.c1(C(=O)N)c(C)noc1C Cc1ccccc1-c1nsc(NC2CCN(C(=O)CCN3CCC(F)C3)CC2)n1 CC1CCN(C(C2(C#N)CC2)=O)CC1NC(c1ccc(CO)nc1)=O C#CC1(NC(=O)C(C)(C)CC)CCC(C)(C)C1.c1(CC(=O)N)ccc(F)cc1 c1(C(=O)N)ccc2c(c1)CCCN2.C1(NC(c2n(C)nnc2)=O)CC(C)C1(C)C c1(C(N2CC(F)(C(=O)Nc3cn(CC)nn3)C2)=O)ccc2c[nH]nc2c1 CCC(C)C(C)CNC(C1CCC(NC(C2CC(C)(C)C2)=O)C1)=O C1(NC(C(N2C(=O)CCC2=O)C)=O)CCN(C(=O)Cc2cccc(F)c2)C1(C)C c1(NC(CC(CC=C)NC(C2CCC(F)CC2)=O)=O)ccc2nncn2c1 c1(CC)cncc(C(N2CCC(C(=O)NCCS(=O)(=O)NC)(CO)C2)=O)c1 C1(NC(CCC(=O)NC)=O)CC=C(C(=O)NOCC(F)(F)F)C1 c1(C(N2CC(NC(c3ccc(OC)cc3)=O)C(O)C2)=O)cc(O)cc(Cl)c1Cl C(=O)(C(F)C(C)C)NCCOCCNC(C(CC)NC(N)=O)=O S(=O)(=O)(c1ccc(CNC(=O)NCc2cccc3c2OCC3)cc1)NC C12(NC(=O)CC3CC3(Cl)Cl)CCC(CN(C(C3CC(=C4CCC4)C3)=O)C1)C2 O=C(CS(=O)C(F)(F)F)NCC1(O)CCCN(C(C2CC=CC2)=O)CC1 C(CC(CNC(c1c[nH]nc1C1CCCCC1)=O)NC(c1nn[nH]c1Cl)=O)OC C(c1ncc(C)[nH]1)=CC=O.c1(OC)cc(C(=O)NC2CCN(CCC)C2)sn1 CC1C(CO)CCCN1C(c1cc(N(C)C)ccc1F)=O N1(C(C(CN(CC)CC)F)=O)CC2CCC1CN2C(c1cc(CO)c(C)o1)=O N1(C(CC)=O)CC2(CC(NC(=O)CC3CCCC3)C2)C1.C(C)(C)C.C=O.N c1(C(=O)NC2CC(CCNC(C(C)(C)C(F)F)=O)C2)cc2cncn2c(O)n1 c1(C(=O)NCC2(O)CC(NC(C(F)OC)=O)C2)cccnc1-n1ccnc1 C1(C(N(C)CC2OCCN(C)C2)=O)CCCCN(C(=O)C(C)(C)CCF)C1 CC1CCCCC1CC(=O)NC1(CNC(C2CC2(F)F)=O)CCC1 c1(OCC)cccc(C(=O)NC2CCN(C(=O)C(C)N(C)C)C2)c1O c1(OC)ccc(NC(C2C3CC2N(C(C2(C(C)C)CCC2)=O)C3)=O)nc1C c1(C(=O)Nc2cnc(C)s2)nc(NCc2ccc(C(F)(F)F)cn2)cn1C c1(N2CC3CN(C(C(CC)OC)=O)CC3C2)nc(C)nc2scc(C)c12 c1(C(N2CC(C(C(=O)NCCCOCC(C)C)O)C2)=O)ccncc1Cl C(C(F)(F)C(=O)NCC1CCCN1C(C1(N(C)C)CCCOC1)=O)OC C(=O)(C(C)(O)CC(F)F)NCCN(C(C1(C)CNC(=O)C1)=O)CC c1(C(=O)NC(CC=C)CNC(=O)C(c2cccc(C)c2)=O)ccc(C)c(C)c1Cl C1(C(=O)Nc2ccccc2)CCN(S(=O)(=O)N2CC3CCNCC3C2)CC1 N1(C(CCCC#CC)=O)CC2(CC(NC(c3ccnn3CCOC)=O)CO2)C1 O=C1COC(CNCc2cn(CC(F)(F)F)nn2)CN1 C1(CNC(c2cc3ccccn3n2)=O)CN(C(c2cc(Cl)c[nH]2)=O)CCC1(F)F C12(NC(C(C)NC(N)=O)=O)CCCC1N(C(c1cocn1)=O)CC2 c1(NC(c2scc(C)c2)=O)ccc(C)c(Cl)c1F C1(NC(=O)C=Cc2ncco2)C2CN(C(C3(CO)COC3)=O)CC12 C1(C(=O)NCC2N(C(C(Cc3cn(C)nc3)O)=O)CC2)CCN(C2CC2)CC1 c1(CNCCN2CCN(C(C3CCC(=C)CC3)=O)CC2)cc(F)cc(Br)c1 N1(C(CC(C)O)=O)CCC2(CCCN2C(c2ccc(C(N)=O)o2)=O)C1 C1(N(C(C2CC(C=O)C2)=O)CCO)CCCN(C(=O)Cc2ccnc(O)c2)C1 Cc1cnn(C)c1C(=O)NC1(CNC(=O)Cn2cnnc2)CC(F)(F)C1 Cc1cc(C(N2CCN(C(C3OCCC3C)=O)C3CCC23)=O)c2ncccc2c1 C(CC1=CCN(C(=O)Cc2ccccn2)CC1)NC(C(C)Cc1ccncc1)=O c1(OCC(=O)NCc2c(C(=O)OC)n[nH]c2)ccc(CC(N)=O)cc1 CC1(C)CCCC1C(=O)NCC1CCCC1NC(c1ncoc1Br)=O CCCCC(O)CC(=O)N1CC=C(C(=O)NCC2(CC)CCCCC2)C1 c1(OC)c(Br)ccc(F)c1C(=O)NC(C)C.c1(C(=O)N)cc[nH]c1C=O C12(NC(CCOCC)=O)CCC(C1)N(C(=O)C(c1ccccc1)N(C)C)C2 N1(C(COCC(C)(C)C)=O)CC2CC1CN2C(C1(c2ccc(F)cc2)CCC1)=O C(=O)(C(C(=O)N)OC)OCC.C1(C(F)(F)F)(C=O)CCCC1.C1CCC1 C12CC(C1)C(C)(C)O2.CC(COc1ccccc1)C=O.C(=O)C=CCO.N c1(C(=O)NC(CNC(c2ccsc2)=O)C2CC2)cc(-c2ccccc2)no1 O=S(=O)(c1ccc(Cl)cc1F)NC1CCC(NCc2cc(Cl)cnc2F)C1 c1(CNC(CN2CCC(C)C2)=O)nnn(C)c1C(=O)Nc1cnn(C)c1 Cc1cc(C(=O)NC(C2CCCN2C(C2CSC2)=O)C)n(C(C)(C)C)n1 CC1SCCCC1C(=O)N(CC(C)(C)NC(c1ncn(-c2ccccc2)n1)=O)C c1(C(N2CCC(N(C)C(c3csc(Br)c3)=O)C2)=O)cc([N+](=O)[O-])cs1 C12(C(N(CCCNC(C3CCN(CC(F)(F)F)C3)=O)C)=O)CCCC(C1)OC2 C1(NC(CC)C(C)C)CCN(C(=O)OCCO)CC1 C(=O)(C#CC1CCOC1)N1CC(C)(NC(C(C)c2cc[nH]n2)=O)C1 C(CCC(C(=O)NCC1CC(C)(C)CO1)NC(=O)Cc1nccn1C)OC N1(C(CCCc2nc(C)sc2)=O)CCC(NC(=O)C=C(Cl)Cl)C1C C(=O)(C#CC1CCCC1)NC(CNC(c1c(CC)[nH]cc1)=O)CC c1(C(COC(c2ccc(I)c(C)c2Cl)=O)=O)cccc2c1ccn2C(C)C N1(C(C(CNC(CC2C(C)CCCC2)=O)(C)C)=O)CC(C)(C)C12CCC2 C1(NC(C(C)OC)=O)CCOC12CCN(c1cc(Cl)nc(C(C)C)n1)CC2 Cc1ccc2sc(N3CCN(C(C4CC5C=CC4C5)=O)CC(C)(F)C3)nc2c1C CC(C)C(C(=O)N1CC(N(C(=O)C(N)=O)C)C1)N1CCCC1=O C(=O)(C#CC(C)(C)C)NCC(=O)N(C1CCCCC1(C)C)C C1(c2ccc(Br)cc2)(NC(=O)NC2COCC2n2cc(Br)cn2)CCCOC1 CC(C)C(C(=O)NCCN(C)C(C1CCCOC1c1ncc[nH]1)=O)n1ccnc1 CCC(CC)(CC(=O)OC)C(=O)N1CC(NC(C2CC=CCC2)=O)C(C)(C)C1 CN1CCCCC1C(=O)NC1CCOC(CNC(=O)CC2OCCO2)C1 N1(C(c2cnc(C)s2)=O)CC(N(C(=O)C=Cc2ccncc2)C)C2(CC2)C1 C(N=c1nc2ncn(C)c2c(NCCCC2CC2)[nH]1)c1cnc(C(C)C)[nH]1 C(CCC(C)(C)NC(c1ncc[nH]c1=O)=O)NC(CSCCCC)=O C(c1ccco1)=C(C)C(=O)NC(C1CCN(C(=O)C(Cl)=CCl)C1)(C)C c1(C(C)C(=O)NC2CC(NC(=O)CN(C)CCO)C2)cc2ccccc2o1 c1(C(N2CCCC(NC(=O)CSC3CC3)C2)=O)cc2c(=O)[nH]ccn2n1 c1(C(=O)NC2(CC=C)CN(C(c3cc(CC)oc3C)=O)C2)cc2cccnn2n1 CCC(CNC(c1cc(C(C)=O)on1)=O)(CC)C(=O)N1CCN(CC(N)=O)CC1 N1(C(C2(CC)CCCO2)=O)CCCOC(CNC(C2(COC)CCCC2)=O)C1 N1(C(c2cc3cccc(OC)c3o2)=O)CCc2cccc(F)c2C1C c1(C=O)cnc2c(c1)CCS(=O)(=O)C2.O=CCC1CC1C(F)(F)F.CC.N C12(C(=O)NCC(CN(C(Cc3c(C)ccs3)=O)C)O)CCCC(CO1)C2 C1(NC(c2cc(CO)[nH]n2)=O)C2COCC1CN(C(C1CCCO1)=O)C2 CCCC(C)C(=O)NC1CCC1C(=O)NCCc1ccc(F)nc1 c1(CC)cc(=NC(=O)C2COC3CN(C(c4cc(Cl)ccc4F)=O)CC23)[nH][nH]1 CC(C)(C)C(CNC(C1CCCC2CC12)=O)NC(=O)C=C1CCSCC1 CC(C)C(O)C(F)(F)C(=O)N1CCOC(C)C1.N1(CC=O)CCP(C)(=O)CC1.N Cc1cnc(C(N2CCOC(CNC(c3cc(C#N)no3)=O)C2)=O)cc1Br c1(OCC=C)ccc(Cl)c(C(=O)NCC2C=CCN2C(C2CCCC2)=O)n1 C(=O)(C(O)C(C)(C)C)N1CCC1.c1(C(NC)=O)cc(C2(Cl)CC2)n(C)n1.C C(C1CN(c2cc(F)ncn2)Cc2ccccc21)NC(C(C)OCCN(C)C)=O Cn1cc(CN(C=O)CC)nn1.c1(C2C(C=O)C2)nc[nH]n1.C(C)(C)C.N N1(C(=O)NC(C23CCC(CO2)C3)C)CCOCC12CC2 c1(C(=O)NC2CC2(F)F)csc2c1CCN(Cc1ccc(O)c(Br)c1)C2 c1(NC(C)C)ncc[nH]c1=NCC1C(C)C1C c1(C(N2CCCN(Cc3cnc(Cl)cc3F)CC2)=O)ccnc2c1OCO2 C(=O)(CCCC(C)(C)C)N(C)CC1CCCN(C(c2nn[nH]c2Cl)=O)C1 C(=O)(C1=NNC(=O)C1)NC(C)CCCNC(=O)CC1COC(C(F)(F)F)C1 C#CCC(O)C(=O)N(CCCN(C)C)CCNC(C1(C#N)CC(C)C1)=O c1(C(=O)NCC(=C)CCNC(=O)CCC2OCCO2)nnn(C)c1CC C1(NC(NC2CCn3nncc32)=O)CCC2C3CCC(C3)C12 C(CCCCCNC(C1CC(O)C1)=O)N(C)C(C1CN(C)C(=O)N1)=O N1(C(C(c2ccc(F)cc2)OC)=O)CCC(CNC(=O)C2=CCOC2)C12CCC2 C(=O)(C1=C(Cl)CCC1)N1CC(C)C(CCNC(=O)CN(C)C2CC2)C1 c1(C(=O)NCCN(C(=O)C(COC)COC)CCC)cc2nccnc2[nH]1 N1(C(C=CCN(C)CC)=O)CC(N(C)C(C2CCCN(C)C2)=O)C(C)(C)C1 C1(NC(c2nc(OC)oc2)=O)CS(=O)(=O)CC1NC(C1SCC=C1C)=O C=CC1(CC(N2CC(CNC(=O)CCS(N)(=O)=O)C3CC23)=O)CCCCC1 C=C(C)CC(C(=O)N)NC(C)=O.CC(C)(O)C.C(=O)CC(C)C.C(=O)CC N1(C(=O)OC(C)(C)C)CCN(C2CCN(C(=O)NC3COC4CC3C4)C2)CC1 C(=O)(CC(C)C(C)(C)C)NC1CCCCN(C(c2cc(C(=O)OC)on2)=O)C1 C1(CC)CN(C(=O)Nc2cnn(-c3ccccc3)c2)CCN1CC(F)F C1(NC(Cc2c(Cl)cn(C)n2)=O)CCN(C(=O)CCSc2ccccn2)CC1F C1(NC(CCCC=C)=O)CN(C(=O)CCCc2cccc(Cl)n2)C2(CCC2)C1 C1(C(=O)NC2CCCCN(C(=O)C=CC3CCCO3)C2)CCC(=C(F)F)CC1 c1(C(=O)N)cc2c(C)cc(Br)cc2[nH]1.N1(C(COC(C)=O)=O)CCC(O)(C)C1 C(CCC(C)(C)C(=O)Nc1cncc(C#N)c1)NC(C(C)C1CCC1)=O c1(CC=O)cc(Cl)sc1Cl.C(C)(C)(C=O)NC(=O)OC.CCC1CC1.N c1(CCNC(C)=O)cn(C)nn1.C1C=CCN1C(=O)C(F)(F)c1csc(C)c1 C(=O)(C(C)(C)C(=O)O)N1CCC(CC=C)(NC(C23CC(F)(C2)C3)=O)C1 S(=O)(=O)(c1cccc(F)c1)N1CC2(C(C(=O)Nc3c(C#N)nc[nH]3)C2)C1 C12(CNC(C(C)OC)=O)CCCC(CN(C(=O)C(C)(C)C(C)(F)F)C1)C2 Cc1cc(NC(C2CCN2C(c2ccc(Br)nc2C)=O)=O)ccc1O C(CCC(C(=O)NCC1COCC1CO)NC(=O)C(F)C(C)(F)F)OC C1(C(=O)NCCC(C)NC(C2CC(CC(C)(C)C)C2)=O)CN2CCN1CC2C C1(C(=O)NCC(C(=O)O)c2ccccc2)CCCCN1Cc1ccncc1 C(=O)(C1=Cc2cc(F)ccc2OC1)N1C(C)(CNC(CNC(CC)=O)=O)CCC1 C1(C)(NC(C=C(CC)C)=O)CCC(NC(=O)Cn2ccc(C)n2)CC1 C1(n2cc(C(C=C)(C)O)nn2)CCOC2(CCN(Cc3cncc(C)c3)CC2)C1 c1(CNC23CCC(NC(C#C)=O)(CC2)C3)cccc2c1OCC2 C1(Nc2cc(NCc3ccc(SC)nc3)ncn2)CCOCC12CCC2 c1(CNC(C(CO)NC(c2cc(C(C)=O)[nH]n2)=O)=O)ccc(Cl)cc1 c1(NC(CC2N(C(C3C(C)C3)=O)CCC2)=O)c(C(F)(F)F)cc(F)cc1Br Cc1ccc(C(N2CC(CNC(=O)C=CC3CCCCCC3)CC2C)=O)c(C)c1 c1(C=O)cnc(C2CC2)nc1O.Cn1nnc(C=CC(=O)NCCC2CC2)n1 S(=O)(=O)(c1ccc2ncsc2c1)N1CC2C(NC(c3ccc(O)c(O)c3)=O)C2C1 c1(-n2c(CN3CCC(C(=O)NCc4cc(Cl)ccn4)C3)ccc2)cccc(F)c1 C1(CNC(CC(=C)I)=O)CC2(CC(NC(=O)C3=COCCC3)C2)C1 C1(CC(=O)NCc2onc(C)n2)CN(C(C2CC(=O)N(C)C2)=O)CC12CC2 [N-]=[N+]=NCCCC(=O)NC1CCCCC1CNC(c1nnn2c1CCC2)=O C1(C(=O)NCC2CNC(=O)O2)CN(Cc2cc[nH]c2)CCC1O C(=O)(CCCS(N)(=O)=O)NC1C(C)N(C(c2ocnc2C2CC2)=O)CCC1 CC(N=c1[nH]c(C(C)C)nc2[nH]ccc12)c1nc2c(s1)CCC2 c1(C(N(C2CN(C(c3c(C)ncnc3)=O)CC2F)C)=O)ccc2c(c1)OCCO2 N#CC1(CNC(=O)NC2CC2(Cl)Cl)CC1 N#CC1(C(=O)NCCC2CCCN(C(C3CCC(F)CC3)=O)C2)CC2CC2C1 C1(N(C(C2C(CC)C2)=O)C)C2CN(C(c3ccc(-c4cccs4)[nH]3)=O)CC12 N1(C(CNC(=O)OC)=O)CCCC1C1(C(=O)N)CC1.C1(C)C=CCC1.C c1(C(c2nnnn2C)NCc2c(C)c(Br)ccc2)cc(Cl)cc(Br)c1F c1(C(C(=O)NC(C(C)(C)C)CNC(=O)C(N)=O)O)ccc(F)c(Br)c1 C1(C(N(C2CN(C(=O)C=Cc3cccc(F)c3)CC2O)C)=O)COC(C)(C)CO1 CCCC(C(O)C(=O)NCC(=O)NC(C)C)NC(C1(CC)CCCCO1)=O C(=O)(C1=CCSC1)N(CCC)CCNC(=O)COCC1CCOC1 N1(C(C2N(C)CC(C)(C)C2)=O)CC2CCCC2(C(=O)N(C2COCC2(C)C)C)C1 C1(C(N2CC3C(NC(C(CCCC)C)=O)C(C3)C2)=O)CC2(C1)NC(=O)NC2=O C1(CCNC(CN(C(=O)OC)C)=O)CN(C(=O)C(C)(C)CO)CC1C C1(C=O)CCC2(CCC2)C1.CC1(C(=O)NCCC2CCCCC2)CCC(=O)N1.N c1(CCNC2(c3n(C4(C)CC4)nnn3)CCC2CC(F)(F)F)ccc[nH]c1=O N1(C(CC(CC)C)=O)CCCC(C)(C(N2CCC(C(N)=O)C2)=O)C1 c1(C(N(C2CCCC2)C)=O)ccc2c(c1)OCC(=O)N2.C1(SC)CC(C=O)C1.N CCC(C#N)C(=O)NC1CC(CCNC(=O)CCc2cc(C)nn2C)C1 N1(C(C=C2CCC(C)CC2)=O)CCCC(C)(CNC(=O)CC2CCCC2)C1 c1(C(=O)NC2C(NC(CC(C)(C)OC)=O)CCC2)ccnc(C)c1C C(=O)(C1=NNC(=O)CC1)N1CCC(C)(NC(=O)CCCC2CCCC(=O)N2)C1 CC(C)S(=O)(=O)CC(=O)NCC12CCCC(CN1C(=O)C1=CCCSC1)C2 CCCCCCC(=O)N1CCOC(CNC(c2ccccc2NC(=O)CC)=O)C1 N1(C(C2C(C)C2C)=O)CC(NC(c2cc(-c3c(Cl)cnn3C)no2)=O)C(O)C1 C(=O)(C(CCSC)NC(c1ccc(F)s1)=O)NCC(CC)N(C)C c1(OC)ncc(F)c(N2CCC23CN(C(C2CC4(CCC4)C2)=O)C3)n1 C1(NC(C(C)O)=O)CCN(C(c2ccc(CF)cc2)=O)C(c2ccccc2)C1 c1(CC)cnc(CNC(=O)CCCNC(C2(C)CCOC2)=O)o1 C1(N(CC(CC)OC)CC)CCCCC1C(N1CCCC1)=O Cc1cnn2cc(C(=O)NC(C)CC(C)NC(=O)C=C3CCSCC3)cnc12 C12(NC(C(CCC)=CCC)=O)CCC(C1)N(C(C1(C#N)CCCO1)=O)C2 N1(C(C(C)OC)=O)CCC2CCN(C(c3csc(C(F)(F)F)c3)=O)CC12 N1(CCC=O)CCP(C)(=O)CC1.N1(C(c2n(CC)nnc2)=O)CC(C)C(C)C1 N1(C(CSCCOC)=O)CCOCC1CC(=O)NC(CO)C1(O)CC1 c1(C(=O)OCC(C(C)OC)=O)sc(Br)c(C)c1C C1(CNC(C(CC)SC)=O)CCN(C(C2(SC)CCSC2)=O)CC1C1CC1 C1(CNC(Cc2cn(C)nc2)=O)C2CN(C(c3cn(C4CC4)nn3)=O)CC12 CC1CC2(CO1)CN(C(C1CN(C(=O)CCc3ccsc3)CC1C)=O)C2 N1(C(C2C(OC)CC2)=O)CCC2(C1)CN(C(c1c(F)ccc(F)c1F)=O)CCO2 CCCC(CC)C(=O)N1CCC(C)C1C(=O)NCCNC(N)=O c1(CNC(Cc2ccc(OCCOC)cc2)=O)cc2ncccc2o1 C(C(C(C)C)C(C)C)(c1n(C(CC)(C)C)nnn1)NC1CC12CC(O)C2 C1(NC(c2c(C)cccn2)=O)C2CC3C1C3C2C(=O)NC.C1(N(C)C)CCC1 C1(CCOC)CCN(C(c2c[nH]c(C#N)c2)=O)CC1.C1(C=O)CCCS1(=O)=O.N C(=O)(C1COc2ccccc21)N1CC(CNC(=O)CCc2cc[nH]n2)OCCC1 C1(C(N2CC(CNC(C3CCN(CCC#C)CC3)=O)C2)=O)CCN2CCOCC12 N(C(=NCC1CCC1)N1CCC2OCCCC2C1)Cc1cc(C)c(O)c(C)c1 n1(CCC)nc(C)cc1C(N1CC2C(C)C2C1)=O.c1n[nH]c(O)n1.C(=O)C.N N1(CC(N2CCCC(C(N(C)CC)=O)C2)=O)CCOCC(NCC2CCC2)C1 c1(OC)cc(C#N)ccc1NC(c1ccc(Cl)cc1NC=O)=O.C(C)=O.N c1(C(N(C)CCNC(C2CC2F)=O)=O)ccc(I)cc1 C1(C(C)C)CCc2nc(O)c(C(N3CC(NC(=O)CCCC4CC4)C3)=O)cc2C1 C1(NC(c2cc(C#N)oc2)=O)CN(C(c2nncs2)=O)C2(CCCCC2)C1 c1(C(=O)OC)cc(S(=O)(=O)N2CCC(CO)C(C)C2)c(F)c(F)c1F Cc1cnc2cc(C(=O)NCCC3CCCC3)ccn12.C1(CC(=O)N)CN(C)C1 c1(C(N2CC(C)C(NC(c3sccc3-n3cnnn3)=O)C2)=O)cn2ccsc2n1 C=CCC(C)(C)CNC(=O)C(=O)NCCNC(=O)OC(C)C N1(C(c2ccc(Br)cc2O)=O)CC2CCC1CN2C(c1c(Cl)ccc(F)c1Cl)=O C1(CC(=O)NC(C)Cn2cc(-c3nccs3)nn2)CCCCC1(F)F c1(C(N2C(C)CCC(NC(C(C(COC)C)C)=O)C2)=O)cc2c(F)cccc2[nH]1 N1(CC(c2ccc(-c3ccc(N4CCOCC4)cc3)cc2)=O)CCC(O)CC1 CCC(C)C(O)C(=O)N1CC(CNC(c2csc(C3CC3)n2)=O)CC1C Cc1cc(C=CC(=O)N)c[nH]c1=N.C1(CC)CN(C(=O)CC)C1.[SH](C)(=O)=O C1(C(=O)NC2C=CC(CNC(c3n(CCC)ccc3)=O)C2)CCC(=O)NC1 CC1COC(C(=O)NC2CCN(C(=O)CP(C)(C)=O)CC2)c2ccccc21 C12CCC1CN(C(=O)Cc1ccc(C)c(C)c1)C2.C1(C(=O)N)(SCC)CC1 c1(C(=O)N)[nH]c(C)cc1C.C1(NC(C(C2CCC2)OCC)=O)COCC1C C1(C(N2CCC(N(C)C(C3(C)CCCC3O)=O)C2)=O)CCC(C(F)(F)F)CC1 CC1(C(=O)NCCC2CSCCN2C(C2CC(n3ccnc3)C2)=O)C=CCCC1 c1(OCC)cccc(C=CC(=O)N)c1.C1(C(N(C(C)C)C)=O)CCC(=O)N1 C1(C(NC)=O)CC(C)CC(C)(C)C1.Cc1nn(C)cc1C(N1CC(F)CC1)=O.C C(C(C)(COC)CNC(c1ccsc1Br)c1nnnn1CCC1CC1)OC N1(C(C(C)=C(CC)C)=O)CCC(NC(c2cc(OC)ccc2N)=O)C(C)C1 c1(CC)cc(C(=O)NCCC2CN(C(=O)C3=COCCC3)CCO2)ccc1F c1(C(N2C3CN(Cc4ncccc4C(F)F)CC23)=O)cc2cc(Br)cc(Cl)c2[nH]1 CN1C(=O)N(CC2=NOC(C)(C)C2)C(=O)C1c1ccccc1 C1(C)(CNC(C2C(C)(CC)C2)=O)CCCN(c2ncncc2C#N)C1 C1(F)(C(=O)NC2CC(NC(c3cnc(C(C)OC)s3)=O)C2)CCOCC1 C1(NC(c2c(CC)ncnc2)=O)CC2CCC(C1)N2C(c1cc2ccsc2[nH]1)=O C#CC1(NC(=O)CC=CCNC(C23CCCCC2C3)=O)CCC(C)(C)C1 CCCCCCCCCC(=O)NCC1CCN1C(c1ccc([N+](=O)[O-])c(O)c1)=O N1(C(c2nn(C)c(O)c2)=O)CC2CCC(C1)C2NC(c1cc(O)c(O)c(O)c1)=O c1(C(C)NC(c2ccc(C)s2)c2n(CCSC)nnn2)ccc(OC(F)F)cc1 N1(C(C2C=CCC2)=O)CCCC(CCC(N2CCC(C3(C)N=N3)C2)=O)C1.COC c1(N(C)C(C2C(c3ccncc3)C2(C)C)=O)cc(Br)ncn1 Cc1cc(Br)ccc1S(=O)(=O)N(c1ncc(Br)c(OC(C)C)n1)C.c1ccccc1 c1(C(=O)NCC2C(C)CN(c3ncccn3)CC2)cc2c(cn1)CCCC2 c1(CNC(=O)Nc2nc(-c3ccccc3)cs2)ccnc(Br)c1O.C(C(F)F)O C12CC(F)(F)CN1C(=O)C(c1cnn(C)c1)NCC2.CCC(=O)OCC N1(CCc2nn(CC)nc2C)CC(=O)N(CC2CCN(C(C)=O)CC2)C1=O C1(NC(C(CC)(C)CO)=O)CCN(C(=O)CC(F)(F)c2ccccc2)CC1(C)C Cc1c(F)ccc(C(N2CCN(C(=O)COc3ccccc3)CC23CC3)=O)c1Cl N#Cc1cccc(OCC(N2CCCCC2c2cn(C3CCC3F)nn2)=O)c1 N1(C(CC(CC)C)=O)C2CCCC1CN(C(C1COC3(CCC3)CO1)=O)C2 C1(CC(=O)NCC2(NC(C(C(C)C)F)=O)CCC2)COCC(C)(C)O1 c1(NC2CCC(NC(CNC(=O)Cn3cccn3)=O)C2)cnc2ncccc2c1 CCN=c1[nH]c(C)c(C(N2CCOC(C)(CNC(=O)C(CO)N(C)C)C2)=O)s1 Cc1cccc(C(C)(O)C(=O)N2CC(c3ccccc3)(CO)C2)n1 CS(=O)(=O)c1cccc(C(N2CC3CCC2C(C)C3)=O)c1.C(=O)(CC(F)(F)F)N C1(NCc2cc(C(=O)OCC)ncc2)CC2(CCCCO2)C1 c1(OC)cnnc(C(=O)NC(CNC(=O)CC)CC(C)C)c1.C(C)CC(C)C C12(NC(C(C)=CC3CC3)=O)COC(C1)C(NC(=O)C(C)(F)F)C2 N#Cc1ccc(C(=O)NCC2CN(C(C3CN(CC(F)F)C3)=O)CCO2)c(O)n1 CC(C)S(=O)(=O)CC(=O)NC1(CO)CN(C(=O)C(C)N(CC(F)(F)F)C)C1 N1(C(COCCCOC)=O)CCC2(CC1)CC2NC(=O)Cc1cccnc1O N1(C(Cc2cn(C)nc2)=O)C2CCC1CN(C(=O)CCN1CCCC1)CC2 c1(C(N2CC3CN(Cc4c(C)c(F)c(F)cc4)C3C2)=O)cccc([N+](=O)[O-])c1Cl NC(=O)CCC(=O)NCc1nc(C)cs1.c1(C(=O)N)ccccc1N1CCCC1 C(=O)(CCCC(=O)NCCOC1CCN(C(=O)CC(C)n2cccn2)C1)OC C1(C(N(C2CCN(C(c3cnc(-c4ccccc4)s3)=O)C2)C)=O)CC=CCO1 C(=O)(C1=COCC1)N(C1CC(NC(=O)C(O)Cc2ccccc2)C1)C c1(C(N)=O)cc(C(=O)NCC2CC2)co1.c1(C=O)ccc(C(F)(F)F)s1 C12CCC(C1)N(C(C1CC1)=O)C2.N1(C(C=O)C2CC2)CCOCC1.C1CC1.N N1(C(C(C)OCC#C)=O)CC2CCCN(C(C3(N4CCOCC4)CC3)=O)C2C1 C(C(=O)N1CC2CCC2(NC(c2cnc(-c3cccs3)s2)=O)C1)(C(C)(C)C)OC N1(C(c2ccc(C(C)=O)cc2)=O)CCN(C(C2(C)CC(O)CN2C)=O)CC(O)C1 c1(CNCC2CCCN(CCOC)C2C)ccccc1S(=O)(=O)N1CCCC1 c1(C2(NC(Cn3cc(CNC(C4(C)CCOC4)=O)nn3)=O)CC2)ccncc1Cl C1(O)(C(N(C(c2ccccc2)CC)C)=O)CCN(c2nnc(C)o2)CC1 Cc1cc(C(=O)NC(C)(CNC(=O)CC2CC3CC3C2)C(C)C)ncn1 CC1C(NC(c2cc(C(C)(C)C)n[nH]2)=O)CCN1C(=O)C=Cc1cnccn1 C1(CC)CNC(=O)CN1C(C1(F)CCN(C(c2cncc(F)c2)=O)CC1)=O C1(N=c2[nH]ccn3nnnc23)(CNC(c2ncc(C)cc2C)=O)CCCCCC1 c1(OC)ccnc(C(N2CCN(CCNC(=O)C(C)CC3CCCC3)CC2)=O)c1 c1(-n2c(Cn3c(=O)cccn3)nc(CC3=CCCCC3)n2)ccc(Cl)c(Cl)c1 N1(C(C(Cn2ccnn2)NC(CNC(C(CC)C)=O)=O)=O)CCc2nocc2C1 C(C)(C(C)(C)NC(c1scnc1Cl)=O)NC(CC=C)=O CCC(O)C(F)(F)C(=O)N1CCC(C(C)(C)NC(=O)Cc2cc(OC)no2)C1 CN=c1[nH]cc(C(=O)NCCC(C)N(C)C(c2cn(C3CCCC3)nn2)=O)s1 C(C)(C)(CC(F)C(=O)NC1(C2CC2)CC1)NC(CCCOCCOC)=O c1(C(=O)NC2C(NC(COC(CC)C)=O)CC2)c[nH]c2cccnc2c1=O C1(NC(C(F)OC)=O)CCCCC12CCN(C(c1ccc([N+](=O)[O-])[nH]1)=O)C2 c1(OC)cc(C)c(C(=O)NC2COCC2NC(c2c(C)csc2Cl)=O)cn1 C12(C(N(C(C3CCCC3)C)C)=O)CC(CCO1)N(C(c1cnn(C)c1N)=O)C2 c1(C(N2C(C)CN(C(=O)C(N)=O)CC2)=O)ccc(S(C)(=O)=O)cc1Cl C1(NC(C(c2scc(C)n2)(F)F)=O)CCN(C(c2c(C)ncn2O)=O)CC1CO CCC(CC(=O)NC(C)(C)CCCNC(=O)C=C(C)C(C)C)c1ccccc1 N1(C(c2cncc(C)n2)=O)CCC(C2CCN(C(c3ccon3)=O)CC2)C1 N1(C(C=CCCC)=O)CCCC(O)(CNC(=O)Cc2ccc(Cl)c(F)c2)C1 C=CCC(CNC(=O)C(CCOC)NC(c1cn(C2CC2)nn1)=O)CC(C)C c1(C(=O)NCC=CCC(=O)NC(C)Cc2ccnn2C)csc(C#N)c1 Cc1csc2cc(C(=O)Nc3cccc(NC(C4CC4C4(C)COC4)=O)c3)[nH]c12 N1(C(C(COC)O)=O)CCC(NC(C2CC(OC)C2)=O)C1C1CC1 c1(NC(C(=O)NC2C(C)(C(=O)OCC)COC2)=O)c(F)cc(F)cc1Cl c1(C(=O)NC(C(C)NC(COCCCC)=O)(C)C)nc2ccccc2nc1C C1(NC(C(CC=C)C)=O)CC2CC(NC(=O)CSCC(N)=O)C1C2 Cn1ncc(C(N2CC3CCC2C3NC(c2cc(O)cs2)=O)=O)c1S(N)(=O)=O C(=O)(C(C)CC(N)=O)N1CCC(N(C)C)C1.c1(COC)ccoc1C(=O)N N1(C(Cc2c(C)non2)=O)CC2(CCCC2)C1C(=O)NCC1COCC1(C)C c1(C(=O)NC(CNC(c2n(CC)cnn2)=O)C)cn2c(n1)SCC2 c1(C(C)(C(=O)NC(C2CCCN2C(c2cscn2)=O)C)OC)ccccc1F c1(OC)cc(N)ccc1C(=O)NCC1CCCCN1C(c1cc(F)cs1)=O CC1c2cccnc2CCN1C(c1cccc(OC(=O)C2CC2)c1)=O c1(-n2c(C3CCC(C)C3)nc(Cc3ccc(F)cc3)n2)ccc2ccsc2c1 NC(=O)CCC(=O)NC1CCCC(NC(C2(c3cccnc3Cl)CC2)=O)C1 c1(OC(C)C)ccc(CNC2CN(C(c3ccc(CO)cc3)=O)CC2C)cc1Cl CC1(C(N2CC(F)(F)C2)=O)CCN(C(c2ccnc(Br)c2)=O)C1 C(=O)(C(F)(C)C(C)C)NC(CC=C)CC(F)F.C(=O)CN(C)C(=O)C1CC1 C1(NC(C2(C(C)C)CCC2)=O)CCN(C(c2sccc2-n2cnnn2)=O)CC1F c1(C(=O)NCC2CCN2C(=O)C#CC2CCCCC2)cc2cnccc2cc1F C(CC(C(=O)N1CC(C)C1(C)C)NC(=O)C(C)C1CCC1)OCC C1(CNC(c2cnns2)=O)CCCC12CCN(C(=O)CC1(O)CCOCC1)CC2 N1(C(C)C)CCN(C(C2CC(C)N2C(C2(F)CCCC2)=O)=O)CC1 c1(CC(=O)NC2CCCC(NC(=O)CC(F)F)CC2)ccc2nc(O)[nH]c2c1 c1(C(=O)NC2C3CN(C(COCCOC)=O)C(C3)CC2)cc2cccc(Cl)c2s1 C(=O)(C(CC(N)=O)NC(C1CC2C=CC1O2)=O)N(CCC(F)(F)F)C N1(C(CSCCC)=O)CC2CC3CC2C1C3NC(c1ncoc1C)=O C12CC1CN(C(C13CC(C)C1C3)=O)C2.C(C=CC(=O)NC)(CC)=CC C(=O)(C(C)(O)CC(F)(F)F)N1CC(C)C(CCNC(=O)C=Cc2ccco2)C1 O=S(=O)(c1ccc(NCC(F)C2CCC2)c(F)c1)NC(c1cccnc1)CO C1(C(CNC(CCOCC)=O)O)CCN(C(=O)CSC2CCCCO2)CC1 C(=O)(C1SCCc2sccc21)NCC1(NC(C(Br)=C(C)C)=O)CC1 N#CC1CCCC(C(N2CCC(F)(C(=O)NC3(CO)CC4CCCC34)C2)=O)C1 C1(C(N(CC(CC)NC(=O)C(C)N(C)C)C)=O)CC(C)(C)CO1 c1(NC2(CNC(CC3CCCC(OC)C3)=O)CCCC2)ncc([N+](=O)[O-])cn1 N1(C(C(=O)NCCCN2CC(C)OCCC2)=O)CCc2ocnc2C1 CCC(C(=O)NCC(C)CNC(=O)C=CBr)C1CCC(=O)N1 c1(C(=O)NC2C(NC(C=C(C)C(C)C)=O)CCCC2)ccc(=N)[nH]c1Cl N1(C(C)=O)CCN(CC(=O)Nc2ncc(Oc3ccccc3)cn2)C(=O)C1 c1(OC(C)C(=O)NC(C2CCN(C(c3cncs3)=O)C2)C)ccc2c(c1)CCC2 c1(CC(=O)NC23CN(C(C(CCCC)O)=O)C(C2)C3)cn2cc(F)ccc2n1 C=CC1(C(=O)N(CC(C)O)CC)CCOCC1.c1(C(=O)N)cnccc1N(C)C N1(C(C2(CNC(C3CC(=O)NC3)=O)CCC2)=O)CC2CCC2(CO)C1 N(C)(C(=NCC(C)C)NCC(C)N(S(=O)(=O)c1cccs1)C)CCCC c1(C(=O)NCCCCCN(C(=O)CC2CCC2)C)ccnc(C(C)(F)F)c1.C C1CCN(C(=O)CN(C)S(N)(=O)=O)CC1.c1(C=O)cnn(CC(F)F)n1.CC C1(CNC(C2(C#C)CCC2)=O)CCC2(CN(C(c3cc(Br)n(C)n3)=O)C2)O1 c1(NC(c2cccc(C#N)c2)=O)cc(Cl)cc(Cl)c1Oc1ccc(CSC)cn1 C1(CCC)CN(C(c2cc(N)ccn2)=O)CCN1C(c1cnn(C(F)(F)F)c1)=O c1(N(C)C)ccc(C#N)cc1CN(C)CC1CCN(C(c2cccnc2F)=O)C1 C1(CNC(C(C)=CC)=O)CC(NC(c2cnoc2-c2ccoc2)=O)CCO1 c1(C(N2C(C)C(=O)N(C)CC2)=O)cn2c(n1)CN(S(=O)(=O)C(Cl)(Cl)Cl)CC2 c1(C(=O)NCCCCCCNC(c2nc(CC)oc2)=O)cc(S(N)(=O)=O)cs1 CCC1=C(C(=O)NCC(CC)NC(c2cc(O)cs2)=O)SCCO1 c1(CC(C(=O)N(C2CN(C(C)=O)C2)C)O)cccc(C(F)(F)F)c1.C=CCO C12(C(N3CC(CC)C(C(=O)NC4CCCC4F)C3)=O)CCCN1CCC2 c1(OCCC(=O)OC)cccc(CNC(=O)N(C)C(c2ccccc2Br)C)c1 C1(CN(CC(F)(F)Br)C)CC2(CCN(C(=O)OC(C)(C)C)CC2)O1 C1(NC(C(c2ccccc2)NC(c2ccsc2)=O)=O)CC2CCCCCC12 C#CC1(O)CCCN(C(=O)C(C)(C2CC2)N(C(=O)Cn2nccc2C)C)C1 C=CCC(CNC(=O)Cc1ccc[nH]1)C(=O)N1CCOCC1CCC c1(OCC)cccc(C(=O)NC(CNC(=O)CCC2CC2C)CC)c1 O(N1CCC(CC(=O)NCC2CCN(C(C3SCCCS3)=O)C2(C)C)CC1)CC c1(C(=O)OCc2c(C)scn2)cc(Br)cc(I)c1C N1(C(=O)CCc2cccs2)CCC(C2CCN(C(C3(CC4CC4)CCC3)=O)C2)C1 N1(S(CCC)(=O)=O)CC2CCN(C(c3cc(O)c(C)c(O)c3)=O)CC2C1 CCS(=O)(=O)c1ccc(CC(=O)NC2CN(C(C3CCC4(CCC4)C3)=O)C2)cc1 c1(CC)c(C(=O)NCC2CC(C)N(C(C3CC(C#N)C3)=O)C2)nn[nH]1.O CC1=NS(=O)(=O)NC(C)=C1CCC(=O)N1CC2CCCC(NC(=O)C3CC3)C2C1 c1(C(N2CCC(C(C)NC(c3ccc(F)s3)=O)CC2)=O)ccc2nn(C)cc2c1 C(=O)(CC(F)(F)C(F)F)N1CCC(C)(CC(=O)NCC(CCC)OC)C1 C1(C)(CNC(CC2(C)CC2)=O)CCCN(C(=O)CC2CCC2)C1.N(C)C.C C(N=c1cc(Cl)c(O)n[nH]1)C1(C(=O)NCCN2CC3CCC2C3)CCC1 c1(NC)cc(=NCC(C)(C)COC)[nH]c(CO)n1 C=CCC(C)C(=O)NCCN(C)C(C1CCCOC1c1cc[nH]n1)=O Cc1cc(C(=O)NCC2CN(C(=O)C(O)CC(C)C)CCO2)c(F)cc1N C(=O)(CCC=CBr)NCC(CN(C(C1(SCC)CC1)=O)C)C N1(C(C(COC)N(C)C)=O)CCOCC1CN(C(=O)Cc1cnns1)C c1(C(=O)NCC2CCC(NC(Cc3nc(C)sc3)=O)C2)cnc(N)c(CO)c1 CC1(C)CC(=O)N(CC(=O)NC2CC(Cc3nn[nH]n3)C3CC23)O1 C12(NC(COCCCC#C)=O)CCC1CN(C(=O)CN1CCN(CC)CC1)C2 N1(C(C2CCC2)=O)CCCC(C2CCN(C(c3cnc(C)s3)=O)C2)C1.CCOC C1(C)(OC)CCN(C(C2CC(NCc3c(C(F)(F)F)coc3C)C2)=O)C1 C(=O)(C(Cc1ccoc1)NC(=O)C(c1cccn1C)=O)N(C)Cc1cnc[nH]1 CC(C)(C)C(=O)CCC(=O)NCc1cc(C(=O)NC2CC23CCCCC3)n[nH]1 C1(C(N2CC(CN(C(=O)Cc3ccc(Cl)cc3)C)C2)=O)CC2(C1)CC21CC1 Cc1cn2c(C(=O)N(C3CCCC3)CCNC(c3onc(C)c3C)=O)cnc2s1 c1(-c2cn(C(C)CNC(=O)CC3CC3(F)F)nn2)cnc2ccccc2n1 CC(C)(C)CC(C)(C)C(=O)NC1CCOC(C(=O)NC2CSC2)C1 c1(C(=O)NC2CN(C(c3cccc(C)n3)=O)CC2C(F)F)cccc2c1CCO2 CC1CC(NC(c2ccc(C(F)(F)F)cc2)=O)CN1C(=O)C=CC1CCCO1 C(C(CC(F)(F)F)NC(c1cnc(Cl)[nH]1)=O)NC(c1onc(CC)c1C)=O Cc1c(C)c(C)c(C(=O)NCCNC(C2(C)CCCCC2)=O)c(C)c1C c1(C(=O)NCCc2ccc(C(=O)O)nc2)ccc2nc(Cl)nn2c1 C1(C(N(CCCC)C)=O)CC2(COC(=O)N2)C1.N1(CCC=O)CCNC(=O)C1.N NS(=O)(=O)c1cc(C(N2CC(NC(c3cscc3Cl)=O)C3CC23)=O)co1 O(N1CCC(CC(=O)NC2CC(N(C(=O)C(C)(C)c3cc[nH]n3)C)C2)CC1)CC c1(C(N2CC(NC(c3cc(CC)[nH]n3)=O)C(O)C2)=O)cnc(N)c([N+](=O)[O-])c1 C(=O)(C1=NOC(C)C1)NCC(CN(C(c1n(C(C)C)ccc1)=O)C)C c1c[nH]c2ncc(Br)nc12.c1(CCC)nc(SC)ncc1NC(C1(CS)CC1)=O C=C(C)CC(C(=O)NC1CCN(C2CC2)C1=O)NC(c1conc1C)=O C(=O)(C#CC(C)(C)CNC(c1csc(O)n1)=O)NC1C(C)(CC)C1 C1(C(N(C)CCc2ccncc2)=O)C2CCN(C(c3ncncc3Cl)=O)CC12 C1(CC)CC(C(=O)NCC(O)C(C)O)CCN1C(c1ccon1)=O Cc1cc(O)nc(C)c1C(=O)NCC1CCCN1C(c1c(C)nc(C)nc1C)=O C(=O)(C(CCSC)NCC1CNCC1(F)F)OC Cc1cc(C)c(C(=O)NC2CCCN(C(=O)C(c3ccc(Cl)s3)=O)C2)c(C)c1 c1(NC(NNC(c2c(C)ncc(Br)c2)=O)=O)nnc2ccccn12 c1(C(=O)NC2CC(NC(=O)C3CC3)C2)ccc(Br)cc1[N+](=O)[O-] C1(C=O)CC(C)(C)CCO1.C1(NC(CCN(S(C)(=O)=O)C)=O)CCOC1.C C1(c2nnnn2C2CCC2)(NCC(CC(=O)OC)C)CC2CS(=O)(=O)CC2C1 C12(C=O)CC(O)C1C2.c1(C(N(CCOC)CC)=O)occc1C1CC1.N N1(C(C2CN(C(COCCCC#C)=O)CC(C)(C)C2)=O)CCN2CC(O)CC2C1 CCCC(CNC(c1nc(C)ccc1F)=O)C(=O)NCC(CO)OC C(C1CCCN1C(=O)C(Cl)Cl)=CC(=O)N(CCC(=O)NC)CC C1(CNC(C=CC(CC)C)=O)CN(C(=O)CCN2CCC(O)CC2)CC1O C1(NC(CCN(CCCCC)CC)=O)(CO)CCCN(C(c2scnc2Cl)=O)C1 c1(C(=O)NC2CC(N(C(=O)CCc3cnc[nH]3)C)C2)cncc(C(F)F)c1 C1(CNC(C(C)(C)c2cc[nH]n2)=O)CCCC(CNC(C2(Br)CC2)=O)C1 N1(CC2(OCCC)CCCCC2)C(=O)CCN(CCN2CCC(C)(C)C2)C1=O C1(CS(N2CC3C(C(=O)O)(C3)C2)(=O)=O)CC2(CCCC2)CO1 n1(CC(C)F)cc(C#N)c(=NC(=O)NCc2cnc3cn(C)nc3c2)[nH]1 N1(C(CCN(CCC)C)=O)C(C(=O)NCC2(C(C)C)CCCC2)CC2CCCC12 C1(NC(c2cc([N+](=O)[O-])n[nH]2)=O)CC2CC1CN(C(=O)CCc1cscn1)C2 CCCC(C(=O)NCC1(C)CCN(C(=O)C=Cc2cocn2)C1)S(N)(=O)=O N1(C(C2=NOC(C)C2C)=O)CC2CCCC(C1)N2C(C1CCOC1)=O c1(C=O)ccc(C)nc1.C(CC(=O)NCC)OCCOCC.C(=O)C.N C=CC(CC(=O)N1CCSCC1CCNC(=O)CNC=O)c1ccc(OC)cc1 c1(CCC(=O)N(C2CCN(C(c3ccc(CC)o3)=O)C2)CC#C)ncnn1C C(=O)(C1=CCCCCC1)N1CCC(C(C(N2CC(C#N)(C#N)C2)=O)(F)F)C1 C1(C(=O)NCC2(OCC)CCC2)CCN(C(=O)CCCOC(C)C)O1 c1(CCC(=O)N(C)CCOCC)ccccc1C#N.C1(C(=O)N)CC2CCC1C2 C(C(C(=O)NC1CCn2nnnc2C1)C(C)(C)C)NC(C1(SC)CCC1)=O C1(F)(C(N(C)Cc2ccn(CC)n2)=O)CCN(C(=O)C(F)=C(C)C)C1 N1(C(C=CC(C)C)=O)CCN(C(C2CCC(=O)O2)=O)C(C2CC2)C1 Cc1cccc(NC(=O)CNC(C2CCC(=O)C2)=O)c1 N1(C(CN(CC)CC)=O)CCC2(CC(C(N3Cc4ccccc4C3)=O)C2)C1 C(C(F)(C(=O)N(CCCCC(C)C)C)C(C)C)NC(c1c(C)scc1)=O C(CCC(=O)NCC1CCCN1C(=O)COc1ccsc1)OCCOC c1(CC(N2C(C(CNC(c3c(C)coc3)=O)(C)C)CCC2)=O)sc(C)nc1C N1(C(c2cnc(OC)nc2)=O)CC(CNC(=O)C(F)C(C)(C)O)C(F)(F)C1 CN1N=C(C(=O)NCC(O)CNC(=O)Cn2cc(Cl)c(O)nc2=O)CCC1=O CCC(C)(C#N)C(=O)NCC1(NC(=O)CN2CCC(C)(C)C2)CCOC1 Cc1noc(C)c1C=CC(=O)NC1CC(NC(C23CCCC2OCC3)=O)C1 C1(NC(=O)Cc2cccnc2)CCN(C(C2CCN(CCO)C(=O)C2)=O)CC1O CC1(C)C(NC(=O)NC(c2ccc(F)cc2F)C2(O)CCC2)C2CCOC12 c1(C(=O)NC)ccc(NC(C2(C)CN(C(=O)CCc3ccoc3)C2)=O)cc1 c1(N2CC(CO)C3(C2)CCC3)nccc2ccc(Cl)cc12 c1(C(N2CC3(N(C(C(C)c4cccs4)=O)CCC3)C2)=O)cccc2c1CNC2=O N1(C(Cc2cc(C)on2)=O)CC2(CC2C(=O)NC(c2cccc(Br)c2)CO)C1 CC1CCC(CNC(c2scnc2Cl)=O)CN1C(C1CC2CCC1CC2)=O C1(C(=O)NCCc2c(CNC(c3c(C)noc3)=O)nco2)CN2CCCC1CC2 C=CC(C)(CCOC)C(=O)NCC(c1ccccc1)CNC(=O)CC(C)(C)C#N C=C(C)CC(C(=O)N1CC(CCNC(C2(F)CCOC2)=O)(OC)C1)OC C1(CC(=O)NCC(CCNC(c2c(CC)cno2)=O)OC)CCCC(=O)C1 N1(C(c2c(C)scc2)=O)CC2(CC(NC(c3cccc(C(C)C)c3N)=O)C2)C1 CCCCCCC(F)C(=O)N1CCC(N(C(=O)C(=CC2CCCCC2)F)C)CC1 C1(NC(CCCCSC)=O)CCN(C(C2CCC3(CC3)C2)=O)CC(C)(C)C1 N1(C(c2cnc(C)nc2C)=O)CC2CCCC2(C(N2CC3(CC3)CC2CO)=O)C1 c1(N2CCC(CC(C)NC(C3CC=CC3)=O)CC2)ncnc2c1ncn2C C1(C(=O)NCCCCCCNC(c2c(OC)c[nH]n2)=O)C(C)(C)CCCC1(C)C c1(C(=O)NC(c2nn[nH]n2)(C)C)nnn(-c2ccc(F)cc2)c1C(F)(F)F C(=O)(CCCCCNC(C1COCC1C(N)=O)=O)NC1CCN(CC)CC1 C1(C(N(CCCOC(C)C)C)=O)CNC(=O)CN1C(c1cccc(=O)o1)=O N1(C(C(C)(C)OCC)=O)CCOC(C(=O)NCC=CBr)C1 C(=O)(CCCC(C)=O)NCC(CC)NC(c1ccc(OC)nc1)=O Cc1cc(Br)c2nc(C(N3CCCCc4ccncc43)=O)cn2c1 C12(NC(C(CC)C#N)=O)CCCC1CN(C(=O)CCNC(C)=O)C2 C1(C)(CC(=O)NCC(c2cnn(C)c2)C)CCCN1C(C1CC(=O)CS1)=O N1(C(C(CCSC)N(C)C)=O)CC(NC(=O)CCCC(C)=O)CC(C)(C)C1 CCC(C)CC(C)C(=O)N1CC(CNC(=O)Cc2cc[nH]c2)C1 C1(CNC(C(COC)O)=O)CC2(CCOCC2)CN1C(C1CC(C)(C)CN1C)=O C1(N(C(CCOCCOCC)=O)C)CCCCN(C(=O)CC2(C#N)CC2)C1 C1(CC)C(NC(c2cc(C(N)=O)co2)=O)CCN1C(=O)C=CC1CCOC1 N1(C(CC2N(C(C(CC)C#N)=O)CC2)=O)CC(=O)NC(C(C)C)C1 C(=O)(C1CCCc2cc(O)ccc21)NC(CNC(c1c(Cl)ccc(C)c1)=O)C C1(C(=O)NCc2c(CC)nco2)CCCCN1c1nnc(C2CC2)s1 C(C(=O)NCC=CC)(C(C)(C)C)SC.c1(C=O)ccc(-c2ccncc2)cc1 N1(C(C2(OC)CC2)=O)CCC2(CCC(NC(c3cncc(F)c3)=O)C2)C1 C12(NC(C3C(NC(C(C)=C4CC4)=O)CC3)=O)CCC(C#N)(CC1)CC2 CC1(C)C(NC(=O)Cc2ccc(F)cc2)CCN1C(c1nccs1)=O Cc1c(C(=O)NC(CNC(c2cnco2)=O)C(C)C)nnn1C(C)C C1(C)CC2CCC1C2.C1(C(=O)N(C)CCOCCC(=O)N)(CC)CCCO1.C c1(CCC(N2C3C(NC(C(CC)C(C)C)=O)C(C3)C2)=O)c(Cl)cccc1[N+](=O)[O-] N1(C(CS(N)(=O)=O)=O)CCC2CN(C(c3nc(O)nc(O)c3F)=O)C2C1 c1(C(=O)NC(COC)C(=O)NC(c2cn(C)cn2)C)ccc(C)cn1 S(=O)(=O)(c1ccc(C)c([N+](=O)[O-])c1)NC1CCN(Cc2ccc(C)c(O)c2)C1 N1(C(c2cc(C(C)=O)sc2)=O)CCC2(CC1)CC2C.C1(C=O)CC2(C1)CC2F c1(C(C)NC(N2CCCC2(CO)CO)=O)ccc2c(c1)n(C)c(=O)n2C C=CC(C)(CC)C(=O)NC1CCOC1C(N1CCCC(O)C1C)=O O=C(CC(O)CNC(c1cc(CO)on1)=O)NC(CC1CCC1)CO C1(C(N(CCCNC(c2c(CC)c[nH]n2)=O)C2CC2)=O)CCCCC1C1CC1 C1(C=O)CCCCC12CCC2.C1(NC(CCNS(C)(=O)=O)=O)(C)CCCCC1.N c1(OC)cc(Br)cnc1C(N1CCC1(C)C(C)C)C(=O)NC1CC(F)(F)C1 N1(C(CC2N(C(c3cccc(OC)c3)=O)CCC2)=O)CC2CC1CC2(F)F C1(OCC)CC(NC(C2CC(C(=O)OC)C2)=O)C12CCCCC2 C(=O)(CCN(OC)C(=O)C(CCCC)CCCCC)N(C)CC.C=CCCC(O)C N1(C(c2c(CCC)n[nH]c2)=O)CC2(CCC2)C1.C1(C(=O)N)CCC(C(C)C)CC1 O=S(=O)(c1c(F)cccc1F)N1CCN(c2ncnc3n[nH]c(Br)c23)CC12CC2 c1(C(N2C(C3CCN(C(c4n(CC)ncn4)=O)C3)CCC2)=O)ccccc1CO CC(C)CC(C)(C(=O)N1CC2(CCC2)C1c1ccco1)NC(=O)O.C(C)(C)C c1(C(=O)NC2(C)CCN(C(c3n(C)ccn3)=O)C2)ccc2c(n1)CCCC2 CCCC(C(O)C(=O)N(C1CCC1)C(C)C)NC(c1cccnc1NC)=O C1(C(N(C2CCCC2)CCNC(Cc2cc(C)sc2)=O)=O)CC2CCC(C1)C2O c1(C(=O)NCC(CC)NC(C2C3CCC23)=O)c(C)cccc1C C(C)(C(=O)NCCC(C)O)N(CCCN(C(COCCC)=O)C)C C1(NC(=O)CCC2CC2(F)F)COCC1NC(c1ccsc1)=O CCC(O)CC(=O)NC(C)CNC(=O)C(C(C)C)c1ccc(F)cc1 c1(OCC)ccccc1C=CC(N1CCCC1CC(=O)Nc1cnccc1C)=O c1(C(=O)NC(CCC)CCCNC(c2ocnc2C)=O)nccc2ccn(C)c12 c1(C(=O)NCC(CNC(C(C)(CO)NC(C)=O)=O)C)cc2c(s1)COCC2 c1(CC(=O)NCC(F)CNC(c2ccc(C(F)(F)F)o2)=O)cccc(F)c1Cl C1(C(N2CC(CCC)C(CO)C2)=O)CC12CCN(C(=O)C=CC(C)C)C2 C12(C(=O)NC(C3CCN(C(c4c(C)occ4)=O)CC3)C)CCCCC1C2(F)F c1(C(=O)NCCCN(C(=O)C(F)C(C)C)CC)nccnc1.c1ccccc1.S C1(NC(C2C3C4CCC(C4)C23)=O)CC2COCC(C1)N2C(c1ccccc1O)=O c1(CCC(=O)NC2C=CCN(c3cc(-n4ccnc4)ncn3)C2)ccccc1Cl Cn1ncc2c(NCCc3cccs3)[nH]c(=NCC3CCOC3)nc12 C1(OCCC(=O)N(C2CCN(Cc3nnn(C)n3)C2)CC)CCOCC1 C1(N2CCCCC(C#C)C2)CC12CCC1(CC2)OCCO1 Cc1nc(C(C)C)sc1C(=O)NC1CC(O)C1.c1(C(C=O)C)cnn(C)c1.C c1(C(=O)NC(c2ccc(-n3cnc4ccccc34)nc2)C)ccc2c(c1)CNC2 C12(CNC(CC(CNC(c3n(CC)nc(C)c3)=O)C)=O)CCN(CC1)CC2 C1(NC(c2c(SC)scc2)=O)C2CN(C(C3CCN(C)CC3)=O)CC12 C1(C(=O)NC2C(OC)CCC2)CCCCN1C(=O)C(C)Cn1cccn1 CCC(CC)CC(=O)NCC(C)(C)CNC(=O)C(C)CC1CCCO1 N1(C(C=COCC)=O)CC(NC(=O)C(F)CN(CC)CC)C2(CCOCC2)C1 C(c1c(Cl)nc2sccn12)=CC=O.N1(C(C2C(=C)CC2)=O)CC2C(C)C2C1.N c1(C(=O)NCC2C(NC(COC)=O)C2)cc(Br)c(F)cc1F N1(C(C(CO)N(C)C)=O)CCCC2(C1)CN(C(=O)CN1C(=O)CCC1=O)C2 C1(CC(=O)NCC(C(=O)N)N(C)C)CC(C)(C)CO1.C1CN(CC(F)F)C1 C1(COC(CC=COC)=O)(NC2CC(C)(C)C2)CCCCC1 C(CCCC(=O)N(CC(C)N(C)C(c1ccc(C2CC2)cn1)=O)C)SC Cc1ccc(CS(=O)CCSc2ccccc2F)cc1F N1(C(C2CCN(C(C)=O)C2)=O)CC2(CCNC(c3sccc3C)=O)CCC1CC2 N1(C(CC=CC(C)(C)C)=O)CC(F)CC1CNC(=O)C=CC(F)(F)F C(=O)(C1=COCC1)N(C)Cc1cnn(C)c1.C12(CCC1)C(=O)NOC2 c1(C(N2CC(F)(CNC(c3n(C)c(S)nn3)=O)C2)=O)nccc2ccncc12 c1(C(=O)NCCCCNC(C2CC(OC)C2)=O)ccc(C)cc1O C#Cc1ccc(CC(=O)NC2CC(NC(=O)C(C)(C)C3CCCC3)C(O)C2)cc1 c1(C(N(C2CCN(C(CSC)=O)CC2)Cc2ccccn2)=O)nccc(Cl)c1O C1(CC(=O)NCCN(CC(C)O)C(=O)Cc2nc[nH]n2)CCCCCC1(F)F C#CCC(C)(CNC(=O)C(CCSC)NC(C1CCN(C)C1)=O)CO c1(CC)ccc(N)c(C(=O)NCC2(C)CCCN2C(=O)C(O)CC(C)C)c1 C(=O)(C1CCCc2sccc21)N1C(C(C)(C)NC(c2n(CC)ccc2)=O)CCC1 c1(CC)nc(C(N2CC3CC2(CNC(C2(F)CC2)=O)C3)=O)c(Br)s1 C=CC(C)(C)CC(=O)N1CCN(C)C(C(=O)NC(C)(C)COCC)C1 C(=O)(C=C(Cl)Cl)NCCOCCNC(=O)C(=C1CCCCC1)F C1(CC(=O)NCCC2(O)CN(C(c3ccc(CC)o3)=O)C2)CCCC(O)C1 N1(C(c2c(C#N)scc2)=O)CC2CCC1C(NC(=O)C(F)(F)CC1CCCO1)C2 C1(NC(c2c(CC)ncs2)=O)CCN(C(=O)CCF)C(c2ccccc2)C1 Cc1ccc(C(F)(F)CNC(C2CCCN2C(N)=O)=O)nc1 C1(OC)CCCCCC1NC(=O)C(Cn1ccnn1)NC(=O)CCn1cccc1 C(=O)(C(C#N)CC)NCC1(C(=O)NC(C=C)COC)CC(=C)C1 c1(C(=O)NC2CCCC(NC(C3CCS(=O)CC3)=O)C2)nccc(F)c1Cl CC1CCCC(C)N1C(=O)COCCNC(=O)CC1CC1.c1ccsn1.C C1(CC)CCN(C(c2ccc(CO)o2)=O)C1C.c1(CCC=O)c(C)n[nH]c1C.N c1(OC)ccc(Cn2c(N(C)CC3CC3(F)F)nnc2-c2cnccn2)cc1 C=CC1(C(=O)NCc2ccsc2C(=O)NCC(C)CC(C)O)CCOCC1 C1(CNC(C(C2CCCCC2)C)=O)CC(C)(C)CCC1NC(=O)CCCF N1(C(c2ccc(CC)c(F)c2)=O)C2CCC1c1c[nH]c(=N)nc1C2 c1(C(N2CC3CN(C(C(F)=CCC)=O)C3CC2)=O)cnc2c(c1)CS(=O)(=O)CC2 N1(S(CC)(=O)=O)CCCC1C(N1CC(CO)C1)=O.c1(C=O)cc(C(C)C)no1 S(=O)(=O)(c1cccc(=NC2CC3CC(C(=O)OC)CC23)[nH]1)NCCCC N1(C(c2ccc(S(C)(=O)=O)o2)=O)CCCC(C2CCN(c3nncs3)C2)C1 c1(C(=O)NCC2N(C(CN3C(=O)CC(C)(C)O3)=O)CC=C2)cccc2nccn12 CCC(CC=O)CC.C1(C=O)CC(O)CN1C=O.C(C)(C)C.C(C)(C)C.N C1(NC(C(C=C)O)=O)CN(C(c2cn(C(C)C)cn2)=O)CCC12CCC2 c1(C(=O)NC2CC(O)(CNC(C3OCC(C)(C)C3)=O)C2)cc(F)ccc1F C(=O)C(F)(F)C1CCCC1.C1(CCNC(C2(C(C)C)COC2)=O)CCCCC1.N c1(C(=O)OC)cc(C(N2CCC(F)C2)=O)n(C)n1.c1(C(=O)N)cn(C)nc1 c1(OC)cc(C(=O)NCC2(OC)CCN(C(=O)C(C(C)C)S)C2)c(F)cn1 c1(CC)cc(=O)n2nc(CN3CCNC(=O)C3C(c3ccccc3)C)sc2n1 Cc1cc(C)n2nc(C(=O)NCC3CCCN(C(=O)CCCF)C3)cc2n1 c1(C(=O)NCC(CCC)NC(=O)C2=NOC(C(C)(C)C)C2)cccc(F)c1C CC1(C)C(C(=O)NCC(=O)NC2CC2)C1C.C1(C(=O)N)CC=CCC1 C1(CC)(NC(=O)CCc2nccs2)CCCN(C(=O)CC2CCC(=O)N2C)C1 N1(C(c2ccc(C)nn2)=O)CCC2(CCN(C(c3csnc3Br)=O)C2)C1 N1(C(C(CNC(c2c(C)nn(C)c2N)=O)O)=O)CC2CSCC(C2)C1 c1(C(=O)NC2CC3CN(C(c4c(CCC)nco4)=O)C2C3)cc2n(n1)CCCC2 CCCC(CCC)CC(=O)N1CCC(O)CC1C(=O)N(C(C)C(=O)N(C)C)C C(=O)(CCCC(F)(F)F)NCC1CN(C(C2(C(C)(F)F)CC2)=O)C1 c1(-c2n(CCc3cc(C)no3)c(N3CCC4CC4C3)nn2)ccc(C)c(Br)c1 N1(CCNC(C(C2CN(C(=O)CCc3ccncc3)C2)OC)=O)CCOCC1=O C(=O)(C1CCCc2cncn21)NCC1(OC)CN(C(c2ccc(C)s2)=O)C1 C(=O)(C1CCCc2n[nH]cc21)NCCC(C)NC(C1CN2CCCC2CO1)=O C1(NC(C=CCC)=O)CCCCC1NC(=O)CCc1cnc[nH]1 N1(C(c2c(C)scn2)=O)CCN(C(=O)C2=NOC(C3(O)COC3)C2)C2(CCC2)C1 N1(C(COCC)=O)CCN(C)CC1CNC(c1cccc(O)n1)=O N1(C(c2ccc(=N)[nH]n2)=O)CC(=O)NCC1C(=O)NCC1CCCS1 C1(NC(C(c2cccc(C)c2)(F)F)=O)CCC12CCC2.C1(O)(CC=O)CCC1.N C(S(=O)(=O)c1ccc2c(c1)NCCC2)C1(C)CCCNC1 N1(C(c2ccn(C)c2)=O)CCC2CN(S(=O)(=O)CC3CC3)CC12 C1(OC)CCOCC1NC(=O)CCC1(C)CN(C(C2(Cl)CC2)=O)C1 C(=O)(C(Cn1cncn1)NC(=O)CCC1CCCC1)NCC(=C)F CC1CCOC(C(=O)N(C)CC2(NC(=O)CC3CCCCC3)CC2)C1 C1(C(=O)N)N(C(=O)C(F)=CC2CC2)CC12CCCC2.N1(CC)CC(C)OC1=O C1(NC(C(CCF)NC(=O)CC=Cc2ccccc2)=O)CCCCC12CC2 c1(OC)cccc(CC(=O)NC2CCC(NC(=O)C(C)(C)c3cncs3)CC2)c1 c1(CC)nc(C(C(=O)NCCCF)N(C2CC2(C)C)C)c(Br)s1 c1ccc(C)cc1.n1(C2CCC2)cc(C(C(=O)NCCSC)NC)nn1.CC.C c1(CC#N)ccccc1C(N1CC(NC(c2cn(CCO)nn2)=O)C1)=O CC(C)C(F)C(=O)NCC1CC(NC(c2ncoc2-c2ccccc2)=O)C1 c1(CNC(=O)CO)ccc2c(c1)CCCC2NC(=O)COCC(F)F.C1CC1 N1(C(c2c(OC)cnnc2)=O)CCC=C(C(=O)NCCOC(C)C)C1 c1(C(=O)NCC(CNC(C2C(C=C)C2)=O)CO)cc(C)c(O)c(C)c1 C(=O)(C(=O)C(C)(C)CC)NC(CC(=C)C)C(=O)NCC(=C)C C1(C(=O)NC(C(=O)NC2CC=C(C)CC2)C(C)C)CCC(C)(O)CC1 C1(NC(C2CC(O)(CC)C2)=O)CCCN(C(c2n[nH]cc2-c2ccncc2)=O)C1 c1(C(N(CCN(C(=O)C(O)C(F)F)CC)CC)=O)cc(=O)c(O)cn1C c1(C(=O)NC2(C)CN(C(Cc3nc(C)[nH]n3)=O)C2)ccn(CC2CC2)c1C N1(C(c2sc(C)c(Br)c2)=O)CCN(Cc2cccc(Cl)c2F)C2CC12 C(=O)C(C)(O)C(C)c1ccccc1.n1(CC=CC(=O)N(C)CC)cncn1.N N1(C(CCC(=O)OC)=O)CCCC2(CCCCC2NC(C)=O)C1 C(=O)(CCCCCN(C(=O)C(C)OCCC(C)C)C)NCCCCC#C C(CC(C)(C)CC(=O)N(CC(C)NC(C1CC2CC2CC1C)=O)C)OC c1(CC)cccc(C(=O)NC2CCCCC2C(=O)NCCN)c1.c1ccccn1 C1(C(N(CC(C)NC(c2nc(C)nn2C)=O)CC)=O)CC12CCSCC2 C1(OC)CC2C1CCN2C(=O)C(n1cc(CCC2CCCCO2)nn1)C c1(C(N(CCCCCNC(c2cc(C3CC3)nn2C)=O)C)=O)cccc(F)c1Cl c1(C(N2CCC(NC(C(C)SCCCC)=O)C2CC)=O)cc(O)ccc1F CCC(O)C(C)C(=O)NCC1CN(C(=O)C(c2ccccc2Cl)C)CCN1C N1(C(C)=O)CCCN(C(c2cnc(C)[nH]2)=O)CC1CO CC1(CNC(=O)CCN2CCCC2=O)C2Cc3ccccc3C12 C1(C(N2CCC(F)(CF)C2)=O)CC12CC(NC(C13CC(F)(C1)C3)=O)C2 c1(C=O)c(C)c(C)nn(C)c1=O.C1(CNC(C2C(=C)CC2)=O)CCOCC1.C C(C(=O)N1CCCO1)NC(C(C1CN(C(c2ccccc2)=O)C1)OC)=O C1(C(N2CCC(CC)C2CNC(c2csnc2C)=O)=O)CCc2cnc(C)n2C1 C(=O)(C1CCCc2nncn21)NC(C(N1CCC(C(=O)NCCO)CC1)=O)CO C(c1cccc(F)c1)=CC=O.N1(CCC)CC(C(=O)N(CC)CC)CC1=O C1(NC(c2cc(-c3ccccc3)no2)=O)CC2CCC1N2C(=O)CCC1CC1 c1(C(=O)NC2COCCN(C(CC(C=C)(C)O)=O)C2)noc2c1COCC2 c1(C(C)C)cccc(C(=O)NC(CN(C(=O)C(F)F)C)(CO)CO)c1 c1(CC(N2C(C(C)NC(=O)C(O)C(F)F)CCC2)=O)csc2ccc(Cl)cc12 Cc1cc(C)c(C(=O)NCC(C)CNC(=O)CN(CC=O)C)s1.C(C)C C1(NC(C2C(CNC(C3(CC)CCCC3O)=O)CCC2)=O)CC12CCCCC2 Cc1cccnc1C(=O)NCC1C=CCN1C(=O)C(C)Cc1ccccc1Cl N1(C(C(COCC)(C)C)=O)CC2(CCCO2)C1.n1(C(C=O)C)ccc(C)n1.C C(=O)(CCCC(=O)NCC(C(C)C)NC(c1cn(CC(F)F)cn1)=O)NCC N1(C(CCSCC(C)C)=O)CCC2(CCC2NC(=O)C=CS(C)=O)CC1 c1(C(N2C(CNC(=O)CCc3ccc[nH]3)CC(OC)C2)=O)cc(Cl)c(C)cn1 N1(C(c2n(CC)ccc2)=O)CCSCC1CCNC(=O)CSC(=N)N Cc1ncc2n1CC(C(=O)NC1CCC1)CC2.c1(C(=O)N)ccn(C(C)(C)C)c1 C#CC1CC2(CC(N(C=O)Cc3cc(F)ccc3Br)C2)C1 Cc1ccc(CC(N2CC3CC3(CNC(C3CN(C4CCC4)C3)=O)C2)=O)cn1 CC1CNc2ccc(C(N3CCC3CNC(=O)CSC3CC3)=O)cc21 CC1CN(C(c2cccs2)=O)CCCN1C(c1cc(-c2ccccc2)ccn1)=O C(=O)(C1CCCn2cncc21)N1CC(OCCC(=O)N(C2CC2)CC2CC2)C1 C#CC1(NC(C2CC(O)CN2C(c2cncnc2C)=O)=O)CCCCCC1 c1(C(=O)NCC(CC)NC(C2(Br)CC2(F)F)=O)n[nH]c2c1CCC2 c1(C(N(C2(C(N3C(C=O)CCC3)=O)CCC2)C2CC2)=O)cc(C)c(C)s1 C1(NC(C(c2scc(C)n2)(F)F)=O)CCCCN(C(c2ccc(C#N)[nH]2)=O)C1 c1(N2CCCC(CNC(C3N(CC)C(=O)CC3)=O)C2)ccnc2ccnn12 Cc1cnn(C)c1CNC(=O)C(C)NC(C1CCC1C)=O CCCC(C(=O)NC(C)CNC(C1CCNCC1)=O)N(C)C.c1csc(C)n1.C C(=O)(C1=CC2C=CC1C2)NCC1(CNC(C(C)N(C)C)=O)CC12CCC2 c1(C(=O)N)cccc2c1OCC2C.COC=CC(=O)NC(C)(C)C(=O)NC(C)C c1(C(=O)NC2C3CN(C(C(C)CC(N)=O)=O)CC32)c(Cl)cccc1S(C)(=O)=O C1(NC(c2c(C)nn(CC(F)F)c2)=O)CC(O)CN(C(=O)C(N)=O)C1 Cc1ccc(C(=O)N(CCCCNC(=O)CCc2nc[nH]n2)C)c(C)n1 N1(C(C(=O)NC(c2c(OC(C)C)cccc2)C)=O)CC2(C)CCC(C2)C1(C)C c1(C(=O)NC2C(CNC(C3(Br)C(C)(C)C3)=O)C2)ccc([N+](=O)[O-])cc1 N(C1CCCOc2c1ccc(Cl)c2Cl)C(=O)CCOc1ccc(Cl)cc1 c1(N2CCC(CC(C)C)C2)nc2c(c(=NC3CCC(CO)CC3)[nH]1)CC(C)CC2 C(c1cn(CC(C)NC(c2coc(C(F)F)c2)=O)nn1)=CC Cc1cc(=NC(=O)C2CC2C(=O)Nc2cc([N+](=O)[O-])ccc2)[nH]n1C.C(C)C.S c1(C(=O)NC2C3CCN(C(CCSCCC)=O)C32)nnc(O)c2c1CCCC2 N1(C(c2n(CC)ncn2)=O)CCC(CNC(C2CCCS2(=O)=O)=O)CC1 N1(C(C(C)(C)NC(C(C2CC2)SC)=O)=O)CCC(O)(C(C)C)C1 Cc1cc(NC(C2(C(F)(F)F)CCO2)=O)ccc1.N1(CCC=O)CCOC1=O.N N1(C(C2C(C(C)C)N(C(C3COCC3C(N)=O)=O)CC2)=O)CC2CCC(C1)C2O C(=O)(C(CCC(C)C)NC(c1cnn(CCF)c1)=O)Nc1cccc(CC)c1 c1(OC)cc(=O)n(C)cc1-c1nc(CC2COCCO2)no1 CCCC(C(=O)OC)C(=O)NC12CC(C1)N(C(=O)CCCCNC(N)=O)C2 c1(NCC2N(C(C3CC(C)(C)OC3)=O)CCC2)c(F)cc(C#N)cc1[N+](=O)[O-] CCCC(C(=O)N1CCCCCO1)NC(=O)C#CC1CC1 N1(C(CN(C(C(C)C)=O)C)=O)CC2CC1CN(C(=O)CC1CCCC(C)C1)C2 Cc1cc(=NCC2CCCC23CC3)[nH]c(=NCc2c(F)cc(Cl)cc2F)[nH]1 Cc1[nH][nH]c(=N)c1C(=O)NCC1(NC(c2csc(Br)c2)=O)CCOC1 N1(C(c2n(CCC)ccc2)=O)CCC2(CC1)CC2C.c1(C(=O)N)ccc(N)cn1 Cc1csc2nc(CC(=O)NCC(C3CCCC3)NC(=O)CC)cn12.C(C)C.O C(=O)(C(CC=C)OC)NC(C(=O)NCCCOC=C)c1ccco1 Cc1cccnc1CCC(=O)NC1(C)CCCCC1.C1(C(=O)N)C(C)(C)C1(F)F N1(C(C(CC(C)C)O)=O)CC(NC(C2CCC(C)CC2)=O)C(S(C)(=O)=O)C1 C12CC3CC(CC(C3)C1)C2.c1(C(=O)NC)ccc[nH]1.C(=O)C(O)C1CCCC1 n1(CCC(N2CCCOC(CCO)C2)=O)c(O)nc2ccccc2c1=O c1(C(N2CCC(C)(NC(CC(CCC)C)=O)C2)=O)ccc2ccc(O)nc2n1 C1(NC(CNS(CC)(=O)=O)=O)CCC2CN(C(=O)C=CBr)CC2C1 CCCCC(O)CC(=O)N1CC(OCCC(N2CCCCCCC2C)=O)C1 N1(C(Cc2ccn(CC)n2)=O)CCCC(NC(=O)CC23CCCC2C3)C1C C1(CN(C)C(C2CC2F)=O)COCCN1C(=O)C.c1cccnc1Cl.C(C)(C)C O=C(C(F)(F)C1CC1)NC1(C2CCCN2C(=O)CCCc2cccnc2)CC1 N1(C(CCn2c(C)ncc2)=O)CCC(C)(NC(=O)C(F)C(C)C)C1 c1(CCC(=O)NCC2(O)CCN(C(CC=CC)=O)C2)nc2ccccc2[nH]1 N1(C(C(Cn2ccnn2)NC(=O)CCC2CC2)=O)CCC2(CNC(=O)O2)C1 C1(NC(c2c(C)noc2C(F)(F)F)=O)CC2(C1)CN(C(c1ncccc1F)=O)C2 Cc1cc(C(N2CC(NC(C3(C(N)=O)CC3)=O)CC(O)C2)=O)ccc1Br c1(C(N2CC(c3cn(CC(F)(F)F)nn3)(N(C)C)C2)=O)ccc2ncn(C)c2n1 c1(NC(CNC(=O)Cc2cc[nH]n2)Cc2ccccc2)ccnc(C2CC2)n1 CCC(C)N=c1[nH]c(=NCCC2CC(C)(C)NC2=O)[nH]c2ccsc12 c1(OC)ccc(C(C)C)cc1C(=O)NC1CC1NC(c1nc[nH]n1)=O C(=O)(C(C)CC(C)C)NC(C(=O)NCC1(C#C)CCC1)CCF C12(CNC(=O)CCCN3CCCCC3)CN(C(c3cc(Cl)c[nH]3)=O)CC1CCO2 C1(NC(=NCCC=C)NCc2ccc(OC)cc2OC)CCOC2(CCSC2)C1 C1(C(=O)NC(c2ccccc2)CNC(c2cc(C#N)no2)=O)CC12CCOCC2 CC1CC(C(N2CCC(C(F)F)(C)C2)=O)CN1C.c1(C=O)sccc1C(F)F.N c1(N2CCN(C(C(C)OCC(F)(F)F)=O)CC2)ccc2c(c1)OCCO2 CC1=C(C(=O)N2CCCCC2CNC(c2cc(N)ccc2O)=O)S(=O)(=O)CCO1 N1(C(C(C2CC2)SC)=O)CCCC(C)(C)C1.C(=O)C(C)(C)C.C(=O)(CC)N c1(C(N2CC3C(Nc4cc(C)nc(C)n4)(CCC3)C2)=O)cc2n(n1)CC1(CC1)C2 Cc1cc(C)c(C(=O)N(C)CCN(C(=O)C2=COCCO2)C(C)C)cn1 c1(CC)ccc(F)c(C(=O)NCC(C)NC(c2cc(F)c(C)cc2Cl)=O)c1F C1(COC)(NC(=O)C(F)CC2CCC2)CCN(C(=O)CC2CCC2)C1 C=CCN=C(NCC(C)(C)COC)N1CCC(C2CCOC2)C1 CC(C(CO)NC(=O)C(C)(F)c1ccccc1)NC(=O)COC(F)F C(C(C)(C)CC(=O)NCC1(C)CCC1)OC.N1(CCC(=O)N)CCCC1=O CC(C)C(CCN(C)C(C1(C(N)=O)CC1)=O)NC(C1COC(=O)C1)=O C1(N(C(=O)CC2CCC2)CCNC(C(C)(C)c2cccs2)=O)CCCCCC1 C1(CC)CN(c2nnc(C3CCCC3)n2Cc2cc(Cl)sc2Cl)CCS1 c1(-c2cn(C)nc2)ccc(C(N2CC(NC(C3CC4(C3)CC4F)=O)C2)=O)cc1 C1(C(NCC#C)=O)CC12CCN(C(=O)C=C(C)C1CC1)CC2.c1ccccc1 c1(C(C(N2CC(O)(CCNC(COC)=O)C2)=O)C)c(F)cccc1F c1(C(=O)NC(CNC(=O)CCC2CCCCO2)CO)ccc(NC2CC2)nc1 c1(C(=O)NC2C(NC(CCOCC#C)=O)C2)cnc(C(C)O)s1 c1(NCC(=O)NC2(C(N3CCC(O)CC3)=O)CCCCC2)ccccc1[N+](=O)[O-] C1(C(N2CC(C)(C#N)C2)=O)CCC(O)CN1C(C1CN2CCC1C2)=O Cc1c(Br)ccc(N2CCC(NC(=O)COc3ccsn3)C(O)C2)c1[N+](=O)[O-] N1(C(CC(C=C)C)=O)CCN(C(=O)C(C)(C)CC2CC2)CC1C CC1CCN(C(=O)C(C)OCc2ccncc2)C(C)C1NC(C1CCOC1C)=O Cc1ccc(C=CC(N2CCC(C)C(NC(C3(F)CCOCC3)=O)C2)=O)c(C)c1 N1(C(C2C(CC)OCC2)=O)CCC(F)(C(=O)NC2CNC(=O)OC2)CC1 C1(C(=O)NC(C2CCN(Cc3cncs3)CC2)C)CCCCN1C N(C(=NCCc1ccc(C)cn1)NCC1CC1)C(C#C)C(C)C c1(CN2C(C(N3CCCC(C)(O)CC3)=O)CNCC2)ccc(O)c([N+](=O)[O-])c1 c1(OC)ncc(C(=O)NCCCN(C)C(c2cnnn2C)=O)cc1Cl N1(C(CC2N(C(CSCCC)=O)CCC2)=O)CC2CCC=CC12 Cc1[nH]nc(C(F)F)c1C(N1CCC(C(F)F)C1)=O.C1(CC=O)C=CCCC1.N N1(C(C2CN(C)C2)=O)CCN(C(c2ccc(N(C)C)nn2)=O)CC1C1CCC1 c1(C(CNC(C)(Cc2ccccc2)C2CC2)OC)ccc(Br)cc1 C1(O)(C(=O)NCCCC(CO)NC(C(CC)NCC)=O)CCC(C)(C)CC1.C Cc1cc2scc(CC(=O)NC3CCC(CNC(C4(CF)CC4)=O)C3)c2s1 C1(C(=O)NC(C)CCCNC(=O)C(N2CCCCCC2)C)CCCC2(CCC2)C1 C1(CC)CN(C)C(=O)CN1C(=O)CCC1CC(NC(=O)C(C)CO)C1 C1(C)(CC)C=C(C(=O)N2CC(N3CCN(C(=O)CCCC4CCCC4)CC3)C2)C1 CCCCC(O)C(C)C(=O)NC(C1CCCCC1)C(=O)NC(C)COC N1(CC(c2ccc(Cl)cc2)C(=O)OC)CC(C)(C)C1(C)C C(=O)(C1=C(C#N)CCC1)N1C(CNC(c2c(C)noc2)=O)C=CC1 C1(CC)CCC(C(N2CCC(NC(=O)COC3CCOCC3)CC2)=O)CC1 N1(C(CCC=CC)=O)CCn2ncc(CNC(C3(CO)CC3(F)F)=O)c2C1 C=CCC(C(=O)NC(C)CC(C)C)C(C)(C)C.c1(C(=O)N)ccc(C#N)c(C)n1 N1(C(=O)NC(c2ccsc2)C)CCc2ccc(C(N)=O)cc2C1 C1(CNC(C(N2CCOCC2)C)=O)(CO)CCN(C(=O)CCC(=O)N(C)C)C1 N1(C(C2(C#C)CCCC2)=O)CCN(C(=O)CSc2ccncc2)CC(C)(C)C1 CC1(C)CC(C(N2CC(F)(C#N)C2)=O)CN1C(c1ccc(C#N)s1)=O c1(C(=O)OCC(c2cc(C)c(F)cc2Cl)=O)ccc(F)c2c1CCC2 N1(C(Cc2cn(C)nc2)=O)CCOC2(CCC(NC(C3CCSC3)=O)CC2)C1 C1(NC(C2CC(C)=C(C)CC2)=O)C2CCC1CN(C(C1COCCN1C)=O)C2 c1(N2CC(CNC(C3(CCC)CC3)=O)(O)C2)c(F)cc(C#N)cc1[N+](=O)[O-] c1(CC)ccccc1C(N1CCC(O)(CNC(C2CC(CC)C2)=O)C1)=O CCCCCCCCC(C)C(=O)NCCOCCNC(C1CCCN1CCC)=O CCS(=O)(=O)C=CC(=O)N1CCCC1C1(NC(=O)Cc2cn[nH]c2)CC1 c1(CC(=O)NC2CC2c2ccccc2C(F)(F)F)ncc(F)cc1F N1(C(CCC(C)C)=O)CCC(c2ccccc2)(NC(c2coc(Cl)c2)=O)CC1 c1(CC(=O)N)cn[nH]c1.C(C)(C)(C1(CNC(=O)C)CC1)NC(C)=O C12(NC(C3CCC(C)C3)=O)CCC(CC1)N(C(=O)C(c1ccnn1C)O)C2 C(C)(CCC(=O)NC1(C(C)O)CC1)NC(C(=O)NC(C)C)=O C1(CNC(c2cnn(CC(F)F)c2)=O)CCN(C(=O)C)C12CC2.c1cn[nH]c1 c1(C(=O)NC(CNC(C2(COC)COC2)=O)CO)ccn(C(F)F)n1 C#CC1CCCN(C(c2cc(Br)c(C)o2)C(=O)NCc2ccccc2OCC)C1 CC1CC(NC(c2cccc(-n3cc(CCC(C)(C)O)nn3)c2)=O)CCC1(C)C N1(C(C(C)NC(=O)OC)=O)CCCC(CC)CC1.c1(C=O)scnc1C1CC1 c1(C(C)(C)NC(=O)NCc2ccc(C(F)F)cn2)nc2ccccc2[nH]1 N1(C(C(CC)OCC)=O)CCC(C(F)(F)F)C1.C(=O)C(C)(C)c1ccno1.N C1(C(=O)OCC)CCCC(CNCC2(C)CCOCC2)C1 Cc1ccccc1CC(=O)NC1CC(F)(C)C1.c1(C=O)cn(C(F)F)c(C)n1 c1(C(N2CCC3C(NC(CCS(C)=O)=O)C32)=O)cc(O)nc(O)n1 C1(CNC(C=C(CC)CC)=O)CCCCN(C(=O)CC2CN(C)C2)CC1 c1(C=O)cc2c(ncn2C)[nH]1.c1(CC)ncccc1C(=O)NC12CC(C1)C2.N c1(C(N2CC(F)CC(NC(C(CC#C)CC#C)=O)C2)=O)ccccc1S(C)(=O)=O N1C2CCCOc3c(cccc32)C1=O.CC(=NO)C1CCC(=O)C1 N1(C(C2C(C=O)C2(C)C)=O)CCC2(CC1)CC(C)N(C(C1CCOC1)=O)C2.CO C1(c2nn[nH]n2)(NC(C2CCCN2CC2(O)CN(C)C2)=O)CCCCC1 Cc1nccn1CCCC(=O)NC(C)CC(C)NC(=O)C(N1CCSCC1)C N1(CC)CCOC(C(=O)NC2CCC2NC(=O)Cc2nonc2C)C1 c1(CNC(=O)NC(Cc2n(C)cnn2)C(N)=O)nc2ccccc2n1C c1(CC(=O)NCC23CC(C2)CCO3)cccc(Cl)c1F.C(=O)(C1=CCCSC1)N C1(CC(=O)NCC2(O)CCN(C(c3c(C)nns3)=O)CC2)Cc2ccccc2O1 Cc1ncccc1C(C)NC(=O)C(CCOCCO)NC(c1ccn(C)c1)=O C#CCCC(C(=O)Nn1ccnn1)NC(=O)C(C)COCC CCCC(C(=O)OC)C(=O)NCCN(c1nc2ccccc2s1)C1CC1 c1(C(c2nnnn2CC(F)F)NC2(C)CSC2)ccc(C(C)(C)C)s1 N1(C(C(=O)NC)C)CCCC2C(NC(c3cc4c(s3)CCOC4)=O)C(C)(C)C12 N1(C(C)=O)CCC(C(C)NC(=O)C(C)NC(=O)NC2CCCC2)CC1 C=CC(CC)CC(=O)N(CC(C)N(C)C(c1occc1CN(C)C)=O)C C1(C(=O)NCC2CCN(C(c3c(C)cccn3)=O)CC2)CCc2c(cnn2C)C1 C(CC(C)CC)NC(Cn1ncc(CC)c1)=O.c1(CC=O)nc(C2CC2)cs1.N C(=O)(C(CC)C(C)C)NCC1(NC(CC(CC)SC)=O)CCC1 C=CC1CCCC(NC(c2nnnn2Cc2nnn(C)n2)CCC)C1 C(=O)C(F)(F)c1cncs1.c1(C(=O)NC2(C)CCC2)scnc1C(F)F.N c1(CC(N2CCC(CNC(C3(C)CC=CCO3)=O)C2)=O)c(F)cccc1F c1(CC)c(C(=O)N(CCCNC(=O)CC2CCCCC2C)C)csc1C c1(C(N2CC(CNC(c3c(OC)cccn3)=O)C2)=O)oc2ccccc2c1CO n1(CC(N2CCN(C(C3CCCCCC3)=O)C(CF)C2)=O)ccc(O)nc1=O c1(OCC#C)cc(F)ccc1NC(c1ccc(C)n1C)=O c1(C(=O)NC2(CCOC)CCC2)[nH]nc2c1CCC2(C)C Cc1ccc(COC(C)C(=O)NC2C3CN(C(c4cocc4)=O)CC23)cc1.C C=CC1(CNC(C2(CNC(=O)C3=CCCC3C)CC2)=O)CCOCC1 C(=O)(C(C)C(F)F)N(CCC(=O)NCCOc1ccccc1)CC C(=O)(CCS(C)(=O)=O)NCCSCC(=O)N(C1(c2cc[nH]n2)CC1)C C1(N(C(C2(CCCC)CC2)=O)C)CCCN(C(c2ccn(C(F)F)n2)=O)CC1 CC1=NNC(=O)C1CC(=O)N(C)CCNC(=O)C(F)C1CCC1 C1(CN(C)C(c2cnc(C3CC3)s2)=O)CC2CCCCN2C1.C1(CC=O)CC1 C1(C(N(CCCOCCNC(c2c(C)ncnc2)=O)C)=O)CN2CCN1C(C)C2 N1(CCC2(C)CC2)CC(=O)N(CC2OCCC2(C)C)C1=O Cc1cccc(OCC(N2CCC2CNC(C2CCC3(C2)N=N3)=O)=O)c1 c1(OC)ccc(-c2cc(C(=O)NCC(C)(C)O)c(C)o2)cc1 C1(OC)CC2C1CCN2C(C1CN(C)CCN1C(=O)CCC(C)CN(C)C)=O c1(-c2ncc(CN(C3CCNC3)CCC)s2)ccc(OCC2CCCO2)cc1 N1(C(Cc2cc(C)ns2)=O)CCC(O)(CN(C)C(C2CCC3(CCC3)C2)=O)CC1 Cc1cnc2n1CCC2NS(=O)(=O)c1ccc(CCl)cc1 C1(NC(C(CN(C)C)(F)F)=O)CCCN(C(=O)CCC2CC2(C)C)CC1 c1(OC)ccc2cc(CNCc3cc(Br)ccc3Br)ccc2c1 CC1CN(C(=O)CONC(C2CC(O)C(F)C2)=O)CC1N(C)C CC(C)C(CO)CCNC(C1CC(C)N1C(=O)CNC(=O)C(C)(C)C)=O c1(OC)ccc2cccc(NC(c3sc(-c4ccccc4)cc3Br)=O)c2n1 c1(NC(=O)C2=CCSC2)cccc(Oc2cccc(F)c2)c1 c1(C(=O)NCC2CC(NC(C3CCC(C)S3)=O)C2)ccc(F)c2ccccc12 C1(C(=O)NC(CCNC(CC=CC=C)=O)C)CC2(CCOCC2)CO1 C1(NC(C2(CC)CCCCC2)=O)CCCC(NC(c2coc(C(F)F)c2)=O)C1 N1(C(C=C(C)C)=O)C2CCC1(CNC(=O)C)CC2.c1ccccc1Cl.CCF.O C12(NC(c3cnn(CCC)c3C)=O)CCCC(C1)C2.C(=O)(CC=C(C)C)N N1(S(C)(=O)=O)CCC(O)(CNC(=O)N)C1.c1(-c2ccno2)ccccc1F.C C1(NC(CC(CC)CN(C)C)=O)CC1C1CCCN(C(C2(C)CCC2)=O)C1 c1(CN2CCC(CC(=O)Nc3n(C)nc(O)c3)CC2)cc(F)cc(Cl)c1 S(=O)(=O)(c1cc(Br)ccc1Cl)N1CC2CN(c3c(F)cnc(OCC)n3)C2C1 c1(C(=O)NCC2CCCN(C(c3sccc3F)=O)CC2)ccc2cccnn12 C#Cc1cccc(C(=O)NC(CC(=O)N(C)CCC2CCCO2)C(F)F)c1 N1(C(C(C)n2cncn2)=O)CCC2(CC1)CC(C(=O)NCCc1ccco1)CO2 c1(C(c2nnnn2C)NCc2cc(C)n(C)n2)ccc(S(N)(=O)=O)cc1F N1(C(c2c(CCC)cccc2)=O)CCCC(C)C1.C1(CC=O)CCS(=O)(=O)C1.N c1(C(=O)NC2CC3N(C(C4(C)CC4)=O)C(CC3)C2)c(Cl)cccc1[N+](=O)[O-] N1(C(CCC)=O)CCC2CC2(C(=O)NCCc2cccnc2F)CC1 Cc1ccc(N)cc1C(=O)NC1CCN(CCNC(C2CCCC(C)C2)=O)CC1 C1(CC(=O)NCCC(=O)NCC(N2CCC(O)CC2)=O)COCCOC1 C1(CC(=O)NCC2CC2)CCC2(CC1)CCC2O.C(=O)(CCCn1cccc1)N C1(C)(C(=O)NC(CC(C)NC(c2nc(CC)sc2)=O)C)CC(F)(F)C1 N1(C(CC(=C)C)=O)CCN(C(c2sccc2SC(F)F)=O)CC1CC(=O)NC CC12CSCC1CN(C(=O)C(c1cccs1)NC(=O)C1=C(Cl)CCCC1)C2 CC1CN(C(c2ccc3cnoc3c2)=O)CC(C)N(C(=O)C(=O)NCC(F)F)C1 C(c1ccc(F)cc1)=CC(=O)NC1(CF)CCN(C(c2c(Cl)cccc2Cl)=O)C1 C(=O)(C1=Cc2ccccc2OC1)NC(CN(C(c1ccn(CCC)n1)=O)C)CC CC(C)C(O)CC(=O)N1CCOC(CN(C)C(C2(C)CCCCO2)=O)C1 CCC1=NOC(CC(N2CCC(C)(C(=O)NCC34CCCC3C4)C2)=O)C1 N1(C(c2ccc(OC)cn2)=O)CCN(C(c2cnncc2O)=O)C(CCO)C1 c1(C(=O)NCC2C(NC(C(COC)O)=O)CCCC2)cnc(OC)c(C)c1 S(=O)(=O)(c1ccn(C)n1)N(C(=O)O)Cc1[nH]nc(OC)c1Cl.C(C)(C)C C1(NC(C(C(C)NC(=O)CC2CC=CCC2)(C)C)=O)CN2CCC1(C)CC2 C1(O)(CC(C)NC(=O)C(C)SCC)CCC1.C1(C(F)(F)F)(C=O)CC1 c1(CC(=O)NCC23N(C(C(C)=CC)=O)CCC2CC3)c[nH]c2cccnc12 CCC(CN(C1(CO)CCC1)C)OC C(=O)(C(C)(C)CCCO)N(C1CCC(NC(=O)CCC(=O)NC2CCCC2)CC1)C N(C(=NCCCN1CCOCC1)NC1CCOc2ccc(Cl)cc21)CC1(C)CC1 c1(-c2cn(C(CC#C)C(=O)O)nn2)cc(Cl)ccc1F CC1C(NC(=O)CN2CCCC2=O)CCCN1C(C1CCCNS1(=O)=O)=O C(=O)(C1=CCC(C)(C)CC1)NC1CN(C(CC(C)OC)=O)CC1F N1(C(COCCCC#C)=O)CCCC1CC(=O)NCC(c1ccsc1)C C(=O)(C(O)CC(C)C)N.c1(OCC#C)ccc(C(=O)NC2CC23CCC3)cc1 Cc1cccc(C(O)C(=O)NC2CC(CCNC(C3CSC3)=O)C2)c1 C(=O)(C(C(C)O)N(C)C)NC(C1CCCCN1C(c1cnc(=N)[nH]c1)=O)C N1(C(c2c(C)scn2)=O)CC2CCC(CNC(c3coc(C(F)F)n3)=O)C2C1 Cc1cc(N)c(C(=O)N(C)CC2CCCN2C(C2CCCC(C)(C)O2)=O)cc1F c1(C(=O)NCC(C2CCC2)NC(c2scc(C)c2Cl)=O)c[nH]c2cccc(F)c12 C#Cc1ccc(C(N2CCCC(NC(=O)COCC)C2CC)=O)c(OC)c1 c1(OC)cc(C(=O)NCC2CCCN2C(C23CC(C)C2C3)=O)ccc1O O=S(=O)(c1ccc(N2CCC3=C(CCCC3)C2)c(F)c1)N1Cc2cccnc2C1 Cc1cnc2n1CCN(C(c1ccnn1CCF)=O)C2 c1(CC)cccc(OCCC(=O)NC(c2n[nH]c(C)n2)C)c1 N1(C(CC2N(C(c3c(C)scn3)=O)CCCC2)=O)CC(C)CCCC1C CCCCC(C)(F)C(=O)NCC1(C(N)=O)CN(C(=O)C(C)(CC)C(N)=O)C1 C1(CNC(C2(CC=C)CC2)=O)CC(C)(C)CN1C(=O)Cc1ccccc1 C1(CCC(N2CC(CN(C)C(c3nsnc3O)=O)C2)=O)CCC(=O)NC1 C1C(C)CCN1C(=O)Cc1ccc(C(N)=O)cc1.c1(SC)ccc(C(=O)N)s1 C1(NC(C=CC(C)(C)SC)=O)CCC12CCN(C(=O)C(c1cncnc1)C)CC2 C(=O)(CC(=O)NC(COCC)C(=O)NC1CSC1)NCC#C C(=O)(CCC(=O)NC)NC1C(NC(CC2(C=C)CC2)=O)CCC1.C1CCCC1 N1(C(c2cc(=N)[nH][nH]2)=O)CC=C(C(=O)NC2CCOCC2F)C1 N1(C(C=CCOC)=O)CC(O)CCC1C(=O)NCCn1cnc(CO)c1 CC1CC(NC(c2c[nH]c(=O)cn2)=O)CN1C(C1CCN(C)C1=O)=O Cc1oc(C)c(S(N)(=O)=O)c1C=O.C1CCC(C)CC1.C(=O)CC1(C)CC1 C(c1ccccc1[N+](=O)[O-])=CC=O.Cn1nccc1C(O)C(=O)NC1CC1C C1(N(C)C(C2COCC2C(N)=O)=O)CN(C(=O)CC(C2CC2)CC)CCC1O CC1(CO)CCN(C(C2(NC(C3CC(=O)NC(=O)C3)=O)CCCC2)=O)CC1 c1(C=O)ccc(S(N)(=O)=O)c(Cl)c1.N1(C(C2(C#N)CC2)=O)CC2(CCCC2)C1 c1(C(N2CC(N(C)C(C3CC3(C)C)=O)C2)=O)cccc2nnn(C)c12 C(C)(C)(CC(=O)N(C1CCN(C2CC2)C1)C)N(C(CCNC(C)=O)=O)C c1(CSCC)ccccc1C(=O)NC.C1CN(C(C2CC2(F)F)=O)CC1C C(=O)(CCCCCN=[N+]=[N-])N1CCC(O)(CCNC(c2cc(OC)ncc2)=O)C1 C#Cc1ccc(CNC(C2(CC=C)CCCN2C(c2oc(C)nc2C)=O)=O)cc1 CC1(C)CCOC(CNC(C2C(NC(c3nccs3)=O)C2(C)C)=O)C1 N(C1CCCc2ccccc21)(CC#C)C(=O)NC1CC(C)CCC1CC C1(CNC(C2CC23CCSCC3)=O)CCCN(C(c2cnn(CCO)c2)=O)CC1 S(=O)(=O)(c1cccnc1NC(c1nnc2n1CCC2)C)NC(C)CCCCO C1(NC(CCNC(=O)OC)=O)CC(CC(N2CC=C(C)CC2)=O)C1(C)C c1(C(N2CCC(C)(CNC(C3(C#N)CCCO3)=O)C2)=O)nn2cccnc2c1Cl O=[N+]([O-])c1cc(-c2cnc(CNS(=O)(=O)c3ccccc3F)nc2)ccc1O C1(N(C(=O)C=C(C)Cl)CC)CCCN(C(c2csnc2-c2ccccc2)=O)C1 N1(C(C2(CC=C)CC2)=O)CCC(CCC)(NC(c2cn(CCCC)nn2)=O)CC1 C1(NC(c2ccccc2)=O)CC2CN(C(=O)COc3ccc(Cl)cc3F)CC2C1 N1(C(CN(CC)CC)=O)CCN(C(C2(C3CCC3)CC2)=O)CC(C)(F)C1 c1(C(=O)NC(CC)(C)CNC(C2(N3CCCC3)CC2)=O)ccc(C)cn1 C1(C(=O)NC2(CN(C)C(C3CCCC3)=O)CC2)CC2CCC1C2 Cn1nnc2c1C(C(=O)NCCCOCCCNC(C1CNC(=O)C1)=O)CCC2 C(C)(C(C)(C)C(=O)N1CCCCO1)NC(CCCN(C(C)C)C)=O C1CCN(C(=O)C(F)OC(F)(F)F)C12CCC2.C(CCS(=O)(=O)NCC=O)OC N1(C(CCSC)=O)CCCC(C)C1.c1(C(=O)N)cccc(C(F)(F)C(F)(F)F)n1 Cc1ccc(CCC(=O)NC2CN(C(=O)Cc3ccc(C)nc3)C3CC23)cc1 CC1=CCC(C(=O)NCCCCCN(C)C(c2cnn(C(C)C)c2C)=O)CC1 N1(C(C(F)OC)=O)CCC(NC(c2cccc(C(C)C)c2)=O)C2(CCC2)C1 c1(OC)ccc(Br)cc1CNC(c1nnnn1C1CCCCC1)(C)CC1CC1 CC(C(C)(C)NC(c1cocn1)=O)NC(c1cn(C(C)(C)C)nn1)=O N1(CCOc2cccc(OC)c2)CCC(C#N)(C2CCCC2)CC1 C12CCC(CO1)C2.c1(C=O)ccc(N)c(Cl)n1.Cn1cc(Cl)c(C(=O)NC)n1 C1(C(=O)NC2(CC(=O)NCC(CC)n3cccn3)CCC2)CCC(=O)C1 c1(CC)cc(C(=O)NCCC2CCC(NC(=O)Cc3ccco3)C2)ccc1Cl C1(CNC(C2CCCCC2)=O)CN(C(c2cc(C3CC3)ccn2)=O)C2CC12 c1(C(=O)NCCNC(C2C(c3n(C)ncc3)OCCC2)=O)cccc([N+](=O)[O-])c1 C(C(=O)N1CC2C(CN)C2C1)(C(C)(C)C)NC(C)=O.c1c(F)cccc1Cl.C N1(C(CCCCN(C)C)=O)CCCCC(NC(c2cc(F)ccc2O)=O)C1 c1(OC)cc(C)c(CNC)cc1O.c1(CCOCC)cnn(C)c1C1CC1 N1(C(C(CSC)OC)=O)CC2CCC1CC2.c1(C(=O)N)cnn(C(C)(C)C)c1C N1(C(C=CC)=O)CCC2CN(C(c3ncncc3Cl)=O)CC2CC1 N1(C(C2(SCC)CC2)=O)CC(C(=O)N)CCC1(C)C.C1(O)CC2C=CC1C2 CC1(NC(Cc2ccccc2C(F)(F)F)Cc2ccccc2)CCC(=O)NC1=O C1(CCC)CN(C(C2CCCC2(F)F)=O)CCN1C(c1ccc(F)o1)=O N1(C(c2ccc(C#N)cc2O)=O)CCC2CN(C(c3cnc[nH]3)=O)CCC2C1 C(CC1=CCCCC1)NC(=O)C(c1ccc(O)cc1)N(CC(O)CO)C1CC1 N1(C(C(C)OCC2CC2)=O)CC(C2CCN(C(=O)CO)CC2)C1.C1CCCOC1 S(=O)(=O)(c1ccc(Br)s1)N1CCCCC1.c1(OC)cc(F)ccc1NC(=O)N CCC(CC)C(C)C(=O)N1CC(CNC(=O)CC2COCCO2)C1 c1(NCC=CCCC)ncc(S(=O)(=O)N2CCC=C(C)C2)cc1Cl C1(C(=O)NCC2C3CN(C(c4c(C)nco4)=O)CC32)CCC2CC2CC1 c1(NC(CC2N(Cc3ccc(C)cc3)CCOC2)=O)c(F)cc(I)cc1[N+](=O)[O-] C#Cc1ccc(C(N2CCC(C)(CC(N3CCC(CCF)CC3)=O)C2)=O)cn1 c1(OC)coc(C(=O)NC(CC)C(C)C)cc1=O.C(=O)CN(C)C(C)=O.N CC1CCC(CNC(c2csnn2)=O)CN1C(c1csc(Br)c1)=O C1(C(=O)NCCC2CCCOC2)(NC(CN(CCC)C)=O)CC(CO)C1 C1(C(=O)NC(C)CC)CCN(S(=O)(=O)N(C)C)CC1.C1(F)(C(=O)N)CCCC1 c1(C(=O)NCCCOCCCNC(C2N(CC)CCC2)=O)cccc(F)c1 CC1(CNC(c2ccc[n+]([O-])c2)=O)CCN(C(C2(C)CCC(=O)N2)=O)C1 CC1C(NC(=O)C=CCO)CCCN1C(C1CCCCO1)=O N1(C2CCN(C(C)=O)CC2)CCCC(C)(C(=O)N(C)Cc2ccc(C)cc2)C1 c1(OC)ccc2cc(C(=O)Nc3ccc4ncnc(O)c4c3)ccc2n1 C1(C(N2CCCC(CCCO)C2)=O)CCCCN1C(=O)Cc1csnn1 c1(CN2C(CC)CC(C(=O)O)CC2)cnn2c1OCC1(COC1)C2 c1(CCNC(=O)CC(c2ccc(Cl)cc2)O)nccc2c(C(F)(F)F)cccc12 C1(NC(Cc2cn(C)nc2)=O)CCCC12CN(c1ncc3c(n1)COC3)C2 O=C(C1=CCCN(C(=O)C=CC(F)(F)F)C1)N1CCC(CCCO)CC1 c1(C(C(=O)NCCOC)N(C)Cc2ccncc2C)cccn(C)c1=O Nc1ccc(C(=O)NCC2CC2NC(c2cccc(C3CCC3)c2)=O)nc1 c1(C=O)ccc(C#N)cc1.Cc1cc(C(N2CC(O)(C)C2)=O)n(C2CCC2)n1.N c1(C(=O)NC2C(NC(c3nc(N(C)C)oc3)=O)CCCC2)ccc2ccnn2c1 C=CCN=C(NCc1ncc(C)s1)NCC1CC12CC2 N1(C(CC2CC(=C)C2)=O)CCC(NC(c2ncc(Br)cc2F)=O)CC1C O=C1CC(c2ccccc2)N(CC2CCOC3(CCSC3)C2)c2ccccc2N1 C1(NC(CC2(C)CCC2)=O)CC(F)(C)C1.c1(C(=O)N)cn(C2CCCC2)nn1 CC(C)CCCC(=O)NCC(C1CC1)N(C(=O)C(C(C)C)c1ccc(Cl)cc1)C Cc1cccc(N(C)C(C2CC2C(=O)N(C2CCC2)C(C)C)=O)c1C C1(NC(c2n[nH]cc2[N+](=O)[O-])=O)COCCN(C(C2(CF)CC2)=O)C1 N1(C(C2(NC(=O)CC3CCCCO3)CC(F)(F)C2)=O)CCCC2(CCC2)C1 C(C)(CN=c1ccnc(Br)[nH]1)C1CCN(C(c2ccc(OC)cc2O)=O)CC1 c1(C(=O)N)n[nH]c(C)c1[N+](=O)[O-].C1(NC(CCC=C(C)C)=O)CCC(F)(C)C1 Cc1cc(CC(N2CC3CCC(C2)N3C(=O)CC#N)=O)ccc1[N+](=O)[O-] CCCC(O)CC(=O)NCC(C)(C1CCC1)NC(c1[nH]c(O)nc1C)=O Cc1cc(C)c(CC(=O)NC2CCN(C(c3nnsc3C)=O)C2)c(C)c1 c1(C(N(C2CN(C(C3(CO)CC3(F)F)=O)CC2O)C)=O)cn2cc(Cl)cnc2n1 C12(C(N3CC(c4ccccc4)(NC(C=CC)=O)C3)=O)CC3CC1(CO)CC3C2 c1(C(N2C(CO)CC(NC(c3c(OC)csc3)=O)C2)=O)cccc2c1NCC2 c1(CCCC(=O)NCC23CNCC(C2)OC3)ccc(Cl)c(Cl)c1 Cc1cc(O)c(C(C)C)cc1.C1(CC(c2nnnn2C(C)C)N)CCC(C)(C)CO1 c1(CC(C(=O)N(CCO)CC)NC(C2CCCCS2)=O)cnn(C)c1O C12(C(N3CC(CC(C)NC(=O)CO)C3)=O)CC(C)(CCO1)C2.C1CCCO1 c1ccccc1.c1(OC)nc(C(=O)NC2CC2C=O)co1.C(=O)C1CC1.N C(=O)C(C)(C)CC(F)F.C1(OC)C(NC(c2cc(C)no2)=O)CC12CCC2.N N1(C(CN2CCC(C)(C)C2)=O)CC(NC(=O)CSc2ccc(F)cc2)CC1(C)C C12(C(=O)NCc3nc(C)cc(C)n3)CCC(CC1)N(C(C1CCCC1)=O)C2 c1(N(C2CCOC2)CCOC)ncc2scc(C)c2n1 CC1(C)CCCN(C(=O)C=CI)C1CNC(c1cc2c(s1)CCOC2)=O C1(C)(CNC(C(C)n2cncn2)=O)CCCN1C(C1CCOC1)=O N1(C(CN(C(C(C)C)=O)C)=O)CCC(NC(c2cc3sccc3[nH]2)=O)C(CO)C1 N1(C(C(CNC(CN(C)CC)=O)OC)=O)CCCC(CN(C)C)C1 c1(OC)cc(C)c(CN2CC(CO)(NC(c3cncn3C)=O)C2)cn1 c1(C=O)c(S(N)(=O)=O)ncn1C.C1(OCC)CC(C(=O)N(CCC)C)C1.N c1(NC(C2C(O)CCN(S(CCCC)(=O)=O)C2)=O)cn2cc(Br)cc(C)c2n1 C(=O)(CC1CCCc2ccccc21)N1CCCC(N(C(CSCC)=O)CC)CC1 C1(C(N(C(CC)CO)C)=O)CCOC1CNC(c1coc(SC)c1)=O CC1(C)c2[nH][nH]c(=NC(=O)C(=O)C3CCCC3)c2CN1C(=O)Cn1cccn1 C1CN(C(c2cc(C(N)=O)n(C)n2)=O)C(C)(C)C1.C(C(=O)N)(C(C)C)OC C#CC(CC(C)C)NC(=O)CCN(C(c1cc(C)[nH]n1)=O)C(C)C c1(OC)ccc(C(N2CC3CC(NC(C4CCCOCC4)=O)C2C3)=O)c(F)n1 CCCCC(C)C(C(=O)NC1COC1)N(C1(C2CC2)CC1)C c1ccccc1.c1(C(N(CCCNC(C2CC2)=O)C)=O)cnc(C(F)F)s1.C N(C1c2ccccc2CC1NC(C1CCSC1)=O)C(C1(C)CC2CCC1C2)=O C1(NC(CN(CCC#C)C)=O)CCN(C(=O)NC2CCCCC2)CC1C N1(C(Cc2c(C)nccc2)=O)CC(NC(=O)C(F)(F)CN(C)C)CC2(CCC2)C1 C#CCC(O)C(=O)NCCCOC1CCN(C(=O)C=C(C)C(C)(C)C)CC1 C#CCC(C)(CC)C(=O)NC1CC(N(C)C(C2CCC(=C)CC2)=O)C1 c1(C(=O)NCC2(O)CC(NC(=O)C=Cc3ccccc3)C2)cnn2c1CCC2 c1(CCC(=O)NC(C(C)C)CNC(C2(CO)CCC2)=O)cccc(Cl)n1 C(C(CC(C)C)C(=O)N1Cc2ccccc2C1)NC(COC(CC)C)=O N1(C(C2N(C(c3scc(C)c3C)=O)C3(CC2)CC3)=O)CCC(C)(C2CC2)C1 Cc1cc(O)nnc1C(=O)NC1(C)CC1.C1(c2ccccc2)(C=O)CCOC1.N n1(C2CC(N)C2)cc(C(=O)Nc2ccnn2C2CCOCC2)nn1 N1(C(COCC(=C)C)=O)C(C(=O)NC2CCOC(C)C2)CCC1C1CC1 c1(OC)cc(C(=O)N(C2CN(C(C3CCCC3)=O)CCC2C)C)c(N)c(C)c1 c1(CNC(c2cc(CC)no2)=O)cccc(C)c1.C1(C=O)CCC(F)(F)C1 C1(c2c(CNC(C)=O)c[nH]n2)CCCN(C(c2c(C)noc2C)=O)C1 c1(NC)ccc(C(=O)NCC=CCC(N2CCCC(CCCO)C2)=O)nc1 c12cc(ncn1)N2.N1(C(=O)OCC)CCC(O)(C(=O)N(C)C2CC2)C1 Cc1cccn2cc(C(N3CC(NC(C4(C)CCCC4)=O)C(C(F)F)C3)=O)nc12 C1(CCC)CN(C(=O)CN2CCCCC2=O)CCN1C(=O)C(O)Cn1cncn1 Cc1cccc2[nH]cc(CC(=O)NCCC3CC(NC(C4(C)CC4C)=O)C3)c12 c1(CNc2c(C(=O)Nc3ccc(SC)o3)n[nH]c2)cccc(Cl)c1[N+](=O)[O-] N1(CCC(=O)N(CC)CC)CCC2CC(F)(F)CCC2C1 C1CC(=O)NCC(NC(=O)CC)C(CCOC)C(=O)CO1.C=O.N C1(C2CCCCO2)(C(N(CCCN(C)C(C2CNC(=O)N2)=O)C)=O)CCOCC1 c1(C(N(CCCNC(C2(C(C)(F)F)CC2)=O)C2CC2)=O)cccc(Br)c1 CCCC(F)C(=O)N1CCC(O)(CCNC(c2cnn(C(C)C)n2)=O)C1 C(=O)(C(C)(C)C(=O)N1CCCCC(N(C)C(C2CCN(C)S2(=O)=O)=O)C1)OC C1(C(=O)NCC2C(NC(c3c(N(C)C)cccn3)=O)CCC2)CC2CCC1CC2 C1(C)(CNC(CCC(=C)C)=O)CCCN(C(c2nc(C(C)C)ncc2Cl)=O)C1 N1(C(C(C(CC)O)C)=O)CC2CCC1C(NC(=O)CCCC(F)(F)F)C2 CCCCC(C)C(=O)N(CCC(=O)NCc1nc(C)cs1)OC c1(CC)cnc(CNC(C2C=CC(NC(=O)OC(C)(C)C)C2)=O)o1 C1(C)(NC(CCC2CC(C)C2)=O)CC(NC(c2sncc2Br)=O)C1 CC(C)(C)CCC(c1nnnn1C1COC1)NCCC1CCC1C(F)(F)F c1(C(C(N2C(CNC(=O)Cc3ccncc3Cl)CC2)=O)=O)cc(F)ccc1F c1(C(=O)NC(C2CCN(C(C3C(C)C3)=O)C2)C)cc2nn[nH]c2cc1F N1(Cc2c(Cl)ncc(C)c2)C2CCC1CC(NC(c1ccnn1C(C)C)=O)C2 C#Cc1cnn(C)c1C(=O)NC1CC2CC(NC(C3C=CCC3)=O)C1C2 C1(CNC(C2N(CCC)C(=O)CC2)=O)CN(C(=O)CC(C)(C)C)CCN1C CC1=C(C(=O)NC2CN(C(=O)C3=C(Cl)CC3)CC23CCC3)Cn2nnnc2N1C c1(C(=O)NC2C(CNC(CC=C(C)C)=O)C2)coc(Br)n1 CC1CCC(C(=O)NCC(C2CCCCC2)NC(=O)COC(F)(F)F)O1 c1(C(C)C)ccc(C(=O)NCCc2ccc(C(=O)NC(C)C(N)=O)cc2)cn1 C#CCCCCCCCC(=O)N1CCCCC1CCNC(C1(C)CC=CCO1)=O O=C1CCC(C(=O)N(C2CCCCCC2)CCNC(c2ccsc2)=O)=NN1 c1(C(N2C(CNC(c3cncc(C)c3)=O)C(C)CC2)=O)cc(C)cc(F)c1N c1(SC(C(=O)N(CCOC)CC)C)ccc2c(c1)OCO2 N#CC1=C(C(=O)NC2CC3CC(C2)N(C(c2cc(C4CC4)on2)=O)C3)CCC1 C1(NC(COC(CC)C)=O)CN(C(=O)CCCC(OC)OC)CC2CCCC12 C(=O)(C1CCCn2ccnc21)NCC(CNC(CCOC(C)=O)=O)(C)F N1(C(CC(C)(C)NC(=O)CCP(C)(C)=O)=O)CCCC(O)CC1 N#Cc1cccc(NC(C2CC=CCN2C(=O)CCCN2CCCC2)=O)c1 c1(C(N(CCNC(C2C(C)(Br)C2)=O)C2CC2)=O)noc2cc(F)ccc12 O=C1CC(C=O)C2(CCC2)C1.C(CCC1CC1)C=O.CC(F)(F)CC1CC1.N N1(C(c2c(C)ccnc2)=O)CCC(C)CC1CNC(c1c(Cl)cnn1C)=O c1(OCCC)ccc(C(=O)NC2CCN(CCC)C2)c(OCC)c1 c1(C(N(CCN(C(=O)C2=CCOC2)CC)CC)=O)cnn2c1CCCC2C c1(OC)cc(CN2CCOCC(NC(c3cnnc(Cl)c3)=O)C2)ccc1I N1(C(c2scc(C#N)c2)=O)CCCC(NC(=O)C(C2(O)CCCC2)F)CC1 c1(CC)ccc2cc(C(=O)NC3CC(CNC(c4ccsn4)=O)C3)ccc2c1 CC1SCCC1NC(C1(C(C)NC(c2cc(C(N)=O)c[nH]2)=O)CC1)=O C1(N(C(Cc2cc(OC)c(C)cc2)=O)C)CC2CCC(C1)N2C(C1CCC1)=O C1(C(=O)N(CC2NCc3ccccc32)CC2CC2)CC2(CCC(F)(F)CC2)CO1 CN1CCC(C(=O)NC2CCN(CCCNC(c3cc(C4CCC4)on3)=O)C2)C1 c1(C(=O)NCC2(OC)CN(C(=O)CCC(C)(F)F)C2)noc2cc(F)ccc12 c12ccc(C(N)=O)c(n1)C2c1n(C(CC)C)nnn1.C(CCCCC1CC1)NC C1CC2(C1)CN(C(=O)C=Cc1ccoc1)C2.C1(CC=O)CCC(C(F)(F)F)O1 C1(C(=O)NCCOCCN(C(C(C(C)C)N(C)C)=O)C)CCCNS1(=O)=O CC1CCC(C)(C(=O)NCCCNC(C2CC(F)(F)C2)=O)C1.c1cccnc1 C1(C(N(C2CCN(CCC)C2)Cc2ccccc2)=O)CNCC(C)(C)C1 n1(CC(N2C(CCNC(C3(C#C)CCC3)=O)CCC2)=O)ccc(Br)cc1=O c1(C(=O)NCC2COCCN2C(=O)C=CCO)ccc2ccncc2n1 C(N=c1[nH]c2c(c(=NCCN3CC4CCC3C4)[nH]1)COCC2)c1cn(C)nc1Br C(C1(C)CCC(C)C1(C)C)=CC(=O)NCCCCCC.c1(C=O)nnc(C)s1.N N1(CC(=O)N)CCC(C(F)(F)F)C(NC(=O)CN2CCCNC2=O)C1.C1CC1 C(=O)C(C)(C)c1ccccc1.C(C)(C)(C)OCCN(C)C(C1CC1)=O.N c1(C(=O)NCC(C)(CNC(=O)C2=COCCO2)OC)cc(C)cc(N)c1 C(=O)(CCC(F)(F)CN=[N+]=[N-])N1CC(CNC(Cc2cccc(C)c2)=O)OCC1 C1(OC)CN(C(C2CN(C(=O)C=Cc3ccco3)CC(C)O2)=O)C(C)(C)C1 c1(COC(=O)CC2C=CCC2)ccc(OCc2nccs2)cc1 Cc1c(CCC(=O)N2CCC2c2ccncc2Br)cnn1C N1(C(C2CC2C(F)F)=O)CC2(C)CC1CO2.N1(C2(C=O)CCC2)CCOCC1 N1(C(c2n(CC)ncn2)=O)CC2CCN(C(c3cc(C)ncc3C)=O)C2C1 C12(C(=O)NCC3(C)CCCN3C(C3CC4(C3)CC4F)=O)COC(CCO1)C2 C1(OC)CC(NC(c2ccc[nH]2)=O)CN(C(c2cc(C)c(N)cn2)=O)C1 CC1CCC(NC(=O)C=Cc2cncn2C)CN1C(c1cc(C(C)(C)C)no1)=O Cn1ccc(C(=O)NCC(=C2CN(C(=O)CN3CCSCC3)C2)F)c1 C1(O)(CC)CCN(C(C2(F)CCC2)=O)CC1.Cc1ccc(SC(C)C(=O)N)cc1 C(=O)(C(O)CCCCC)NC(CNC(C1(C=C)CC1)=O)C1CC1 n1(CC(=O)NCC(CNC(=O)CCn2cncn2)OC)nnc2ccccc12 C1(C)(CNC(c2n(CC)nnn2)c2ccc(C(F)F)o2)CC2(CCC2)C1 C(C(C)C(F)(F)F)NC(c1ccc(C(C)=O)o1)=O.c1(C=O)cn2ccsc2n1.N C1(N(C(CC(COC)C)=O)C)CC2CC1N(C(c1cc(O)cc(Cl)c1)=O)C2 Cc1ccc(-c2noc(-c3cccc(NC(=O)NCC4CC4)c3)n2)c(Br)c1 Cc1cccc(C(N2CCOC(C(=O)NC(CO)CCC(C)C)CC2)=O)c1O CC(CC(C)NC(=O)CC(O)CNC(c1ncn2c1CCC2)=O)C(F)F C(=O)(C(F)(F)C(O)C(C)C)NC1CC(NC(Cc2c(C)nc[nH]2)=O)C(O)C1 c1(CC)ccc(C=CC(=O)NC2COCC2NC(=O)C(Cl)=CCl)cc1 c1(C(N2CC(CC=C)(NC(C3CCCOC3C)=O)C2)=O)cc2ccc(Cl)nc2s1 CCC(C(F)(F)F)NC(=O)CN(C(=O)CC(C)C)C1CC1 Cc1cc(C(=O)NCCNC(=O)CCOc2cc(F)cc(F)c2)cnc1O C(F)(C(=O)N1CC=CCO1)=Cc1c(C)nc(CCCC)s1 N1(C(CCCC)=O)CCC(C(F)(F)F)C(NC(c2cc(N)nc(Cl)c2)=O)C1 c1(C(N(C)CC2CCCN2C(C2CC3C=CC2O3)=O)=O)nsc2ccccc12 Cc1onc(CO)c1C(=O)NC1CCC(N(C(=O)Cn2cnccc2=O)C)C1 C1(C(C)C)C(NC(=O)CC23COC(C)(C2)C3)CCN1C(c1ccns1)=O c1(N2CCN(C(C(CC)C(C)C)=O)CC2CCO)[nH]cnc2nc(Cl)cc1-2 N1(C(CC2(C#N)CC2)=O)CCCC2CN(CC(N3CCCCCC3)=O)CCC12 C(=O)(C1CCCc2ncccc21)N1CCN(c2nnc(CC(C)C)s2)C(C)C1 C(=O)(C1=CCC(NC(c2sccc2C)=O)C1)NC(c1ncc(C)cn1)C c1(OC)cc(C(N2CC(CCCCNC(=O)CCC3(O)CCC3)C2)=O)ccc1F C1(NC(c2ccc(CC)cc2)=O)C(C)CCN(C(c2cc(C#N)oc2C)=O)C1C C(=O)(CC(C(F)(F)F)c1ccccc1)N1C(COC)CN(C(=O)C)CC1.C(C)C N1(C(CCC)=O)CCN(C(=O)CC(F)(F)CC)CC1c1ccccn1 c1(CC(N2C(C)CC(NC(c3ccn(C)c3)=O)C2)=O)ccc2nc(O)[nH]c2c1 c1(CC)ccc(C(=O)N)[nH]1.C1(F)CN(C(c2cc(C(C)(F)F)on2)=O)C1.C C1(c2n(C(C)C)ccn2)CC12NC(=O)N(CCC1CCC(F)(F)CC1)C2=O c1(C(N2CCN(C(C3C4(CC4)C34CC4)=O)C3CC23)=O)ccc(F)c2occc12 C#Cc1cccc(-c2nc(C)c(NCc3cccc(Br)c3F)s2)c1 C1(CNC(c2ccn(C)c2)C)CCCOC1c1nccn1C C(=O)(C#CC1CCOCC1)N(C1CCN(C(c2csc(CO)n2)=O)CC1)CCC CC1CCC1NC(=O)C(=O)NCC1(COC(C)(C)C)CC1 C1(NC(C(N2CCCC(C)C2)=O)=O)CN(C(=O)CC2CCOC2)CC(C)(C)C1 C(=O)(C(CNC(=O)CCc1cncnc1)C(C)(C)C)N1CC(C)(F)C1 C1(CC=C)(C(=O)NCCOCCCC=O)CCCC1.C(=O)C.C1CCC1 Cc1cc(C(=O)N(C)CCN2CCN(C(=O)CCc3ncc[nH]3)CC2)cc(O)n1 C1(c2n(CCOC)nnn2)(NCc2ccnn2C)CCCC2CC12 C(=O)(C(O)CCN(C)C)N(CC(CNC(CCCc1nc(C)sc1)=O)C)C N1(C(C(C)C#N)=O)C2CCC1CC(NC(c1cnn[nH]1)=O)C2 c1(C=O)c([N+](=O)[O-])ccc(F)c1F.CC(C)C(=O)NCC1CC1C1OCCO1 C1(C(=O)NCCCC(=O)NC)CCN(C(C23CC(F)(C2)C3)=O)C12CCC2 c1(C(N(CCN(C(c2cn(CC)nn2)=O)C(C)C)C)=O)nnn(C)c1N C(=O)(CCC(=O)NC)NCCCOC.C12CC(C1)C2.C1(C=O)CCCC1O CON(CCC(=O)N1CCCCC(C)(F)C1)C(=O)C(C)(C)C(C)(C)O c1(C(N2CC3CCN(C(C(CCC)C)=O)C3C2)=O)cc2nccn2c(O)n1 Cc1ccc2c(C(=O)OCc3cnc(C#N)c(C#N)n3)n[nH]c2c1 C1(O)(CCNC(C2(C#N)C(C)(C)C2)=O)CCCN(C(=O)Cc2cc[nH]n2)C1 Cc1csc2c(C(=O)NCCC(C)(C)NC(c3cnc4n3CCC4)=O)ncnc12 c1(C(N2CC(N(C(C(c3ccccc3Cl)C)=O)C)C2)=O)ccc([N+](=O)[O-])cc1F n1(CC)cc(S(=O)(=O)NC2CC(C(=O)Nc3cccc4[nH]ccc34)C2)cn1 c1(COC(C(CC=C)OC)=O)cc(F)c(Cl)cc1[N+](=O)[O-] C1CCN(C(c2ccc(C#N)o2)=O)CC1F.C12(CSC)CC(C(=O)N)(CO1)C2 C(C(C)C)(C(O)C(=O)NC(CNC(C1CCCC1F)=O)C1CC1)OC C1(NC(C(C)Sc2ccccc2)=O)CN(C(C2CNC(=O)N2C)=O)CC1F C1(NC(=O)C=Cc2cnc[nH]2)CC2CC(C1)N(C(=O)CS)C2.c1cscn1.C Cc1[nH]nc(C(=O)NC(C2CC=CCC2)C(=O)NCc2ccsc2C)c1O C1C2CCC(C2)C1C(N1CC(CC(F)F)C1)=O.C(C=O)N(C)C(=O)C1CC1 CCCCC(C(=O)NC1(CF)CCN(C(=O)COCc2ccncc2)C1)N(C)C N1(C(c2nc(C)nc(O)c2)=O)CC2(CCCN(C(=O)Cc3cccnc3N)C2)C1 c1(C(=O)NC2C(F)CCN(C(c3cc(SC)oc3)=O)C2)cnn2c1CC(C)CC2 C(=O)(C(C)(CNC(c1cc(C#N)cs1)=O)CC)NCC(=O)OCCCC C(=O)(C(O)CCNC(C1CC(C=O)C1)=O)N(C1CCCC1)CCOC.O CC1(C)C(C(=O)NC(CO)C2(O)CC2)C1.c1(C=O)ccc(C2CC2)o1.C O=C(O)C1CCN(C(c2cocc2Br)=O)c2ccccc21 C(C#CC(=O)N(OC)C(C)C(=O)OC)NC(C(C1CC1)OC)=O C1(NC(=O)Cc2ccc(F)cc2Cl)CC2CC1CN(C(c1ccc(O)nn1)=O)C2 N1(C(C(C)N2CCC2)=O)C(C)CC2CN(C(C3(C(F)(F)F)CCCC3)=O)CC12 C1(CNC(CN(C2CCC2)C)=O)CCCN1C(C1CN(CCF)C1)=O C(C)(C(F)(F)C(F)(F)F)=CC(=O)N.C(C)C.C1(C=O)CC1.C(C)C c1(C(=O)NC(CC)(C)C(F)(F)F)n[nH]c2c1CN(C(=O)CCC(C)=O)C2 Cc1cccc(CN=C(NCc2cnns2)NC(C2CCCO2)C)n1 c1(OC)c(Cl)cc(C(N2CC(NC(=O)C=C3CCOCC3)C2)=O)cc1Cl C1(n2cc(CCN(C(c3cnc[nH]3)=O)CC)nn2)CCN(CC)CC1 C1(CNC(CN(CCC)C(C2(C#N)CCOC2)=O)=O)CC2CCC1CC2 c1(N2CC(CC(=O)O)(NC(C(CC(CC)C)C)=O)C2)nc2cc(C)ccc2o1 C=CC(CC)CC(=O)N1CCCC(CNC(c2nc(-c3nc[nH]n3)sc2C)=O)C1 CC1(C)C=C(C(=O)NCCCC2(O)CCN(C(C34CCC(CC3)CO4)=O)C2)C1 C1(NC(CCOCC(C)C)=O)C2CCC1N(C(C1(N3CCOCC3=O)CC1)=O)C2 C1(C(=O)NCc2ccc(CC)cc2)CCC(C)CN1C(c1ccc(C#N)cn1)=O C=CCC(C)(C)C(=O)N1CCCC1CN(C1CCN(C)C1=O)C N1(C(C(CC)(C)C)=O)CCC2(CCC2)C(NC(=O)Cc2cccc(F)c2)C1 C#CC1CCC(C(=O)NCC2C=CC(NC(c3cc(C)[nH]n3)=O)C2)CC1.O CC1CN(C(=O)C(CC2CCCC2)NC(=O)C(C)CO)C(C)CO1 CC1Cn2nccc2CN1C(=O)C(F)CC(C)(C)NC(c1csnc1Cl)=O C1(CC#C)CCCN(N2CCC3(CCC3)C(CO)C2)C1 C1(CCC)CCC(O)(C(=O)N(C)CCNC(=O)COC2CCCOC2)CC1 N1(C(C=C(CC)C)=O)CCC(OCCNC(c2cn(CC)nn2)=O)C1 CC(N=c1nc(N2CCCNC(=O)CC2)c2ncn(C)c2[nH]1)c1cc(Br)n(C)n1 CCCCC(CNC(=O)C=C(C)c1ccsc1)NC(=O)Cc1scnc1C C=CCCN=C(NCc1nc(CC)no1)N1CCN(CC)CC1.[SH](C)(=O)=O Cc1cc(N2CC(CN(C(=O)C(C)C3CCC3)C)C2)nc(-c2cccs2)n1 c1(C(=O)NC(CN(C(c2c(OC)c[nH]n2)=O)C)C)c(N)cc(F)cc1Br C1CC2CCC(C1)N2C(C1C2CC3C(C2=O)C13)=O.c1(CC)ccoc1C=O.N C1(NC(c2n[nH]c(C)c2Cl)=O)CC2CC(C1)N(C(c1cnn3ccsc13)=O)C2 C(=O)(C1CCc2c[nH]nc21)N1CC(C)C(C(=O)NC(CO)CCC2CC2)C1 C=C(C)C(CC(=O)NC1CCOCC1NC(=O)C=Cc1cccn1C)OCC C1CCN(C(=O)C=CCN(C)C)CC1(F)F.Cc1nc(N(C)C)sc1C=O.N N1(C(c2c(N)c(O)nc(O)n2)=O)CCCC2(NC(=O)C=CC3CC3)CCCC12 C1(CNC(CCCC)=O)CCC(F)(CNC(C2(CC)CC(C)(C)C2)=O)CC1 C1(C(N(CCOCCCNC(c2cnc(C)[nH]2)=O)C)=O)CCN(C)C1C c1(CN2CC(c3cc(F)ccc3F)(O)C2)ccc2ccc(F)c(Br)c2n1 c1(C(N2C(C)(C)C(CC(=O)NC(CO)CCF)CC2)=O)ccc2cc[nH]c2n1 C=CCCCC(C(=O)N(C(C)C(=O)OC)C1CC1)NC(=O)C(C)N(C)C N1(C(CCCOCC)=O)CCN(C(c2cnn3cccc(Cl)c23)=O)CC(C)(F)C1 C1(NC(CCCSC)c2nnnn2C2CCOCC2)CC(O)C(O)C1O O=S(=O)(c1csc2ccc(Cl)cc12)N1CC2(CO)CC2(C(F)(F)F)C1 N1(C(C(C)OCC)=O)CC(C2CCCCN(C(C3CCCCC3C)=O)C2)C1 CCCCC(C(=O)NC1CCN(C(N)=O)CC1)NC(c1cccc(CC)n1)=O c1(C(=O)NCCC(=C)CNC(=O)C(C)CC)ccc(CC(F)(F)F)cc1 C1(C)(C=O)CC(C(C)(C)C)=NO1.c1(OC)ccc(C=CC=O)cc1.C1CC1 C1(NC(CCN(CCCCC)C)=O)CC(C)CN(C(c2sccc2NC)=O)C1 C1(N(C)C)CCC(N=c2[nH]c3c(c(=NCCc4nc[nH]n4)[nH]2)CSC3)C1 CCC(C)C(C(=O)NCCCCN(C)C(c1sc(C)cc1OC)=O)OC C(=O)(C1=CC2CCCC12)N1CC(O)(CN(C(=O)CCCC2CC2)C)C1 C(=O)(C(C)CCc1ccc(F)cc1)N1CCC(CNC(C2(CCC)CC2)=O)C1 N1(C(C(=O)NCc2ccco2)C2CCSC2)CCCSCC1c1ccccc1 C1(CNC(C(=O)NC(CC=C)CC)=O)CC2CCC1N(C(=O)CC(C)(C)C)C2 C(=O)(CS(=O)(=O)C1CC1)N(C1CCC(CNC(CC2CCC(C)C2)=O)CC1)C C=CC1CCCCN1C(c1ccccc1CCC)C(=O)NCSc1ccccc1 C(C(=O)NOCC(C)C)(C(C)C)SC.C1(CC2CCC2)C(=O)N1 C1(NC(c2c(C)nns2)=O)COCCN(C(c2ccc(CC(C)C)s2)=O)C1 N1(C(Cn2ccc(C)n2)=O)CCOC2CN(C(=O)C3=CCCCO3)CC12 c1(C(=O)NC2(C)CN(C(C3ON=C(C(C)C)C3)=O)C2)ccc2nc(O)[nH]c2c1F n1(CC)ccc(=NC(=O)C(F)C2CCN(C(C3(NC(C)=O)CCCC3)=O)C2)[nH]1 C(C(CO)N=c1ccc2nnnn2[nH]1)NC(=O)Cc1ccc(Cl)c(F)c1 Cc1ncn(O)c1C(=O)NCC(O)CCNC(=O)C(c1ccc(F)cc1)(C)C CC1(O)CCCC1NC(=O)CN(C(=O)Cc1ccco1)CC1CC1 Cc1cc(NC(C2CN(c3ncccn3)C2)=O)ccc1NC(c1cccs1)=O CCC(C)C(C)(O)CNC(C1CC(F)(F)CN1C(=O)CC1CSC1)=O Cc1cc(C(=O)NC(c2nc(=N)[nH][nH]2)C)c(C)cc1O Cn1cc(C(=O)NC(c2ccccc2)C(=O)NC)cn1.C1CN(C(C)(C)C)C1 C(c1cncs1)=CC(=O)NC1(C2CCCN2C(=O)CCC2CCOC2)CC1 C(=O)(CC(C)C(C)C)NC1C=CCN(C(C2(COC)CCCCC2)=O)C1 c1(C(=O)NCC2(CCNC(=O)C3=C(Cl)CC3)CC2)cc(Br)c(F)cc1O C(CC1CCC1)(C(=O)NCCC(Cl)Cl)NC(COC(C)(C)C)=O N1(C(C(C)SCCCC)=O)CC2(C)CN(C(c3cc(N)cc(N)c3)=O)CC2(C)C1 C(=O)(CS(=O)(=O)C(C)C)NC1(CCC)CCCN(C(C2CC(OC)C2)=O)C1 c1(C(N(CC)C)=O)cc(C(F)F)ccc1Cl.Cc1oncc1C(=O)N(C)CCO N1(C(CC(C=C)(C)O)=O)CCC(C(=O)N2CCOCC2C(C)O)=C(F)C1 C1(CNC(c2c(C)ccc(Cl)c2)=O)CC2(CCC2)CN1C(=O)CO.C1CC1 C(C)(C)(CN=c1oc(C2CC2)nc2ccccc12)NC(C(C)(C)C)=O CC1CN(C)C(=O)CN1C(C12CC(NC(=O)CO)(C1)C2)=O.C1CCCC1 c1(C(N2CCC(NC(CCCC#C)=O)CC2C2CC2)=O)cc(S(C)(=O)=O)cs1 CC1(N)CCCCC1C(=O)NC1(c2nn[nH]n2)CCSCC1 C1(NC(C(C=C)(C)O)=O)CC1C1CCCN(C(=O)Cc2ccn(C)n2)C1 c1(N(C)CC2CCC(=O)N2)nc2cccnc2c(=NC2CCCCC2F)[nH]1 N1(C(C(C(CC)C)C)=O)Cc2nccn2CC(NC(c2ocnc2C2CC2)=O)C1 C(Cn1cncn1)(C(=O)NCCc1cn[nH]c1)NC(CC1CC(SC)C1)=O N1(CC)CCOC(C(N2CCN(C(=O)CNC(C3CC(OC)C3)=O)CC2)=O)C1 C12(CNc3c(C(=O)OC)c(C(C)(C)C)cs3)CC(C#N)(CO1)C2 C1(NC(=O)NCC(C)(C)O)CCc2nc(C(F)(F)F)cn2C1 c1(OC)ccc2c(c1)cc(C(N1CCC(N(C(=O)C=CCF)C)C1)=O)n2C c1(SC)cc(C(=O)NC2CCC(F)(CNC(c3snnc3C)=O)C2)oc1C C(=O)(CC1=CCN(C)CC1)N1C(C2CCN(C(C(C)CN(C)C)=O)C2)CCCC1 N1(C(CS(CC)=O)=O)CCC(n2cccn2)(C(=O)N)CC1.C1(C(=O)N(C)C)CC1 CC1CN=C2NC(C(=O)NCC3CCCN3C(C3CC3(C)C)=O)=NN2C1 c1(C(=O)NC(C(C)(C)NC(CCc2cc(OC)no2)=O)C)cc2cccnc2s1 C(=O)(NNS(=O)(=O)CCCC1(c2ccccc2)CCC1)C1C(O)CCN(C)C1 N1(C(C(CC)SC)=O)CC(O)(C2(CNC(=O)COC(F)F)CC2)C1 N1(C(c2cn(CCC)nn2)=O)CCC2CC12C(=O)NCC(C)C(C)O c1(C(=O)NC(CNC(C2CN(C)C2)=O)C(C)(C)C)ccc([N+](=O)[O-])cc1Cl C1(NC(c2n(C)c(O)nc2)=O)(CNC(=O)Cc2ccsn2)CCCCCC1 c1(C=O)ccc2nc(C)cn2c1.Cc1cnc(COCC(=O)NC2CCC2)o1.N C1(NC(C2C(COC)C2)=O)CCC(N=c2[nH]ccnc2C(=O)OC)CC1 C(N=c1ccnc(NCc2cn3ccsc3n2)[nH]1)C1(OC)CCCC1 n1(CCC(=O)N(C2CCCC2)CCC)nnnc1C1CC1.O=CCSC(F)F.N C(=O)CS(=O)(=O)N(C)C.C1(C(N2CC(COC)C2)=O)CCC(=O)N1C.C C1(NC(C(=O)NCC)=O)CCCC(NC(=O)Cc2ccc(OC)cc2C)CC1 C(c1ccc(C)cc1C)=CC(=O)N(CCCCNC(COC)=O)C C1(C)(NC(CC2(C)CC2)=O)CC(C(=O)NCC2(c3cccnc3)CC2)C1 C(CCC)(C(=O)NCCOC1CCN(C(=O)CCc2nncs2)C1)=CCC C1(NC(CCC)(c2nnnn2C(C)C)C2CCCC2)CCc2ncsc2C1 O=C(C#CC1CCCO1)NC(CNC(=O)Cn1cccnc1=O)C1CC1 N1(C(C2(C)CCC2)=O)CC(C2CN(C(c3ccc(Br)c(C(F)F)c3)=O)C2)C1 N1(Cc2sc(C)c(Br)c2)CCC2(CCCC2C(N2CCC(F)(F)CC2)=O)C1 c1(C(N2C3(CCN(C(C(C(C)C)F)=O)C3)CCC2)=O)cc2c(Cl)c(Cl)ccc2[nH]1 Cc1c(C(N2CCN(CC(C)NC(=O)C=C3CC3)CC2)=O)cnn1C1CC1 CC(C)(C#N)C(=O)NCCC1(O)CN(C(=O)CCc2ccc(Cl)cc2)C1 C1(C(N2CCC(CC)(NC(C3CCCOC3C)=O)CC2)=O)CN2CCCN1CC2 N1(C(c2cc(COC)on2)C(=O)NC(C)C(=O)OC)CCCCC(C)C1 C1(CCNC(C(CCSC)O)=O)CN(c2nc(SC)ns2)CCS1(=O)=O C1(NC(=O)Cn2ccc(Br)n2)COCCC1NC(=O)CC=C(Cl)Cl Cc1ccc2nc(N3CCC(NC(=O)C(F)(F)C(F)F)C3C)sc2n1 c1(OC)ccccc1CN(C(=O)Cc1csc(Cl)c1)C N1(C(c2cc(C)ns2)=O)CCN(C(C2CC3(CCC3O)C2)=O)C(C(C)(C)C)C1 O=C(C1=CCCN(C(c2cc(C3CC3)no2)=O)C1)N1CC2CCC2(CO)C1 Cc1ccnc2nc(C(=O)NC(C3CCOC3)CNC(=O)C(F)=CCCF)nn12 C=C1CCN(C(=O)C(C)CO)C(C(=O)NC2CCC(CO)CC2)C1 N1(c2nc(CC)nc(=N)[nH]2)CC2CCCC1C2C.C1(CC(F)F)(C(=O)N)CCC1 C1(CC)CN(C(=O)CS(=O)(=O)N(C)C)CCN1C(c1cccc(NC)n1)=O c1(CC)cc(Cl)ccc1C(=O)N(CCC(C)NC(C12CCC(OC)C1C2)=O)C C1(NC(C2C=CCC2)=O)CC1C1CCN(C(c2csc3cncn23)=O)CC1 N(C(=NCCNS(C)(=O)=O)NC)C1CCN(C(CC)=O)C1.C1CC1C(F)F C(CS(=O)(=O)C1CCN(CCCCN2CC(C)OC(C)C2)CC1)OC C1(C(=O)NC2(C(=O)NC3(C)CSC3)CC(O)C2)CCCN1C=O c1(C(=O)NC2CCC(CNC(CC(=C=C)C)=O)C2)ccnc(C(F)(F)F)c1F CC(C)(C)C#CC(=O)N1CCC(CCCCNC(=O)CC2(CO)CC2)CC1 c1(OC)cccc(C=CCC(=O)NC(CNC(=O)C)CO)c1.CC(F)F.O C1(CC(N2C(CCNC(c3c(C)nccn3)=O)CCCC2)=O)CCCNC(=O)C1 C=CCC(C)(C)CC(=O)NC1(C(=O)NC2CC(O)C2OC)CCOCC1 c1(C(=O)N)ccc(C(=O)C2CC2)cc1.C(C)(C)(C(=O)NC1CCC1)N(C)C N1(C(C(C)(C2CCC2)NC(CCC(=C)Cl)=O)=O)CCC2CCCC2CC1 N1(C(c2nc(OC)oc2)=O)CCC(C)C(CC(=O)NC)C1 c1(C=O)ccc(C#N)c(O)c1.CC1CN(C(=O)CC(C2CC2)C2CC2)CC1C N1(C(c2cc(C(C)=O)oc2)=O)CC(NC(C2CC3CCC3C2)=O)CCC1C O=C1NC2(CCN(C(C3CSCCN3C(c3ccco3)=O)=O)C2)CO1 C1(NC(c2ccc(Cl)o2)=O)CC(O)CN(C(c2cccnc2-n2cncn2)=O)C1 N1(C(C(c2n(C)cnn2)(C)C)=O)CCC2(CCOC2)C1 Cc1[nH]nc2sc(C(N3CCOC(CN(C)C(c4ccccc4)=O)C3)=O)cc12 C1(C(N2CCN(CCNc3ncc(C#N)nc3)CC2)=O)CCOC2(CCC2)C1 c1(C=O)cccc(F)c1C(F)(F)F.C1(CC)CC(O)CN1C(=O)CN.C N1(C(C(CC)(CC)CC)=O)CCC2C(C1)NC(=O)CN2C(=O)C(COC)OC C(Cc1ccccc1)(C(=O)N1CCC1)NC(=O)OC.C(=O)C(C)(Cl)Cl.CC C(CCS(C)(=O)=O)(C(=O)NCC1CCC1)OC.C(=O)C(C)(C)n1cccn1 CCCCCCCC(=O)N1CC(NC(C23CCCC2(C(=O)OC)C3)=O)C1 C12(CCNC(c3csnc3Cl)=O)CCC(CC1)N(C(=O)CCN1CCCCC1)C2 c1(NC2CCN(C(C(CC(=C)C)NC(C)=O)=O)C(C)C2)nc(C)ccc1C#N C12(NC(c3ncc(C)cn3)=O)CCCC1(F)CN(C(C1C(C)(C)C1(F)F)=O)C2 c1(C(=O)NC2(CNC(C(CC)O)=O)COC2)cc(Cl)ccc1I C(=O)(CC(C)(C)C1CC1)NC(C)CCCNC(=O)CC1(CSC)CC1 N1(C(=O)Cc2cnccn2)CCCN(C(c2noc3ncccc23)=O)C(CO)C1 c1(CC(N2CC(N(C(C3C(C)CC(=O)CC3)=O)C)C2)=O)cc2cc(Cl)ccc2[nH]1 C1(NC(C=C(CC)CC)=O)CCN(C(c2cc(CC(C)C)nc(O)c2)=O)CC1O N1(C(C2(C)CCCN2C(=O)NCCCCl)=O)CCC(C(N)=S)CC1 Cc1ccc(OCCC(N2CCC(N(C(=O)CC3CC4COCC34)C)C2)=O)cc1 c1cc(OC2CCN(Cc3csnn3)C2)ccc1CCO Cc1ccc(C=CC(N2CCC(CNC(=O)C=CC3CCOC3)C2)=O)cn1 C1(C(=O)NCC(C(=O)NC(c2nc(C)[nH]n2)C)(C)C)CCC2(CC1)CC2 c1(CC(C=O)C)ccc(O)c(O)c1.C(=O)(CC(=O)N(CC)C)NCC#C CCC(CCC(=O)N1CCCC(C)(O)C1)NC(c1nc(C)c(C)s1)=O C(=O)(C(C)(CSC)NC(C1CCC1C)=O)NC(CC#C)CO C(CNC(c1cnn(C)n1)=O)(C(C)(C)C)NC(C(C)Sc1ccccn1)=O C1(NC(c2cc(C)on2)=O)CCC2(CCN(C(c3cnns3)=O)CC2)C1.C1CC1 N1(C(C)=O)CS(=O)(=O)CC1C(=O)NC1CCCCC1.c1(C=O)ccnc(O)c1 Cc1ccc(NC(=O)NC2C=CCCC2)c(F)c1 C(=O)(NN1CCCC1C(=O)N(C)C)c1c(-c2ccc(C)s2)cccc1 c1(C(N2CC3C(NC(c4cc(C)on4)=O)C3C2)=O)c(F)cc(F)cc1Cl c1(OC)cc(C2CCCN2CCCOc2ccccc2)cc(OC)c1OC Cc1ncnc(C(=O)NC2CCN(C(c3csc(C(F)F)n3)=O)C(C)C2)c1C C(=O)(C(C#N)(CC)CC)N1CC(C2C(C(N(CC)CC)=O)C2)C1 c1(C(N2C(C(N(C(CSC)C)C)=O)CC(=O)C2)=O)cc(O)ccc1C c1(CCNC(=O)NCCC(=O)NC(C)(C)C)ccc(Br)s1 Cc1ccc(F)c(C(N2CC(O)(C(F)C(=O)N3CCC3C3CCC3)C2)=O)c1 C1(C)(CC)C=C(C(=O)N(C2CCCCC2N(C)C(C2C3CCCCC23)=O)C)C1 Cc1cc(C(=O)NC2CCC(C)(C)CC2)c(C)[nH]1.C(=O)CC(C)C.C1CC1.N Cc1cn2c(C(=O)NC(C3CCCN3C(=O)C(C)CC(F)(F)F)C)cnc2s1 CC1(C)CC(CC(=O)NOCCCF)N(C(C2CCCC(=O)CC2)=O)C1 C1(C(=O)NC(C2CC2C(N2CCCCCC2C)=O)C)CCC2(CC1)CC2 C1(CNC(CCC=C)=O)CN(C(=O)CC2(CO)CCCC2)CCCO1 N1(C(C(c2cccc(Cl)c2)C)=O)C2CN(Cc3ccc(Br)o3)CC12 N1(C(c2nc(C)sc2)=O)CCC2(CC1)CC2C(N1CCOC(C)C1)=O Cc1cccnc1CNC(c1ccn(CCNC(=O)Cc2cnoc2)c1)=O Cc1cc(O)nc(C)c1C(=O)N.C1(c2nc[nH]n2)CCN(C(=O)C2=CCC2)CC1.C N1(C(c2ccc(C(C)(F)F)cc2)=O)CCOC2CCN(C(c3ccc[nH]3)=O)CC12 N1(CC(C)N(C)C)CCC(c2ccccc2)(CC(=O)O)CC1 C1(NC(C(C)O)=O)CN(C(C2CCN(c3cccnc3)CC2)=O)CC12CCC2 N1(C(c2c(CC)nc[nH]2)=O)CC(NC(C2CCCC23CCC3)=O)CC(C)(C)C1 CC1CCCN(C(=O)C=Cc2cc[nH]c2)C1CNc1ccc(C(F)(F)F)cn1 C=Cc1ccc(C(=O)N(C(C)CCNC(c2c[nH]nc2C2CC2)=O)C)cc1 c1(CCC)cc(C(=O)N(C2CCN(C(=O)CC3CCC3(F)F)C2)CC)no1 Cc1ccc(CC(=O)NC2(CNC(=O)CSCCN(C)C)CCOC2)s1 O=C1Cc2cccc(C3CCCN3C(c3snc(-c4ccccc4)c3Cl)=O)c2N1 C1(C)(CNC(=O)NC2C(C)CN(Cc3ccccc3)C2)CCC2(CC1)OCCO2 N1(C(C2CCC(C)C2)=O)CCN(C(=O)CNC(=O)C(F)(F)c2ccnn2C)CC1 Cc1cc(C(=O)N(CCCCC)C)nn1C(C)C1CC1.C(=O)C(F)=CC1CC1.N c1(-c2ccc(O)nc2)ncn2c1CN(Cc1c(Cl)ccnc1Br)CC2 C(=O)(CCCCCCCC=C)NC1CC(C)(NC(Cc2cccc(C#C)c2)=O)C1 c1(C(N2C3C(NC(C4CCCOC4)=O)CC(C3)C2)=O)ccc(Cl)c2ccccc12 c1(C(=O)NC2CCCC2NC(C23COCC(C2)C3)=O)cnc2sccn12 C1(CNC(C2(C)CSC2)=O)C(C(N2CCC(CC3CCC3)C2)=O)C1(C)C N1(C(c2cnc(OC)s2)=O)CCC(C2CCCN2C(C2CCCCN2C)=O)CC1 C12(CNC(C(C3CCCO3)NC(c3c[nH]c(=N)o3)=O)=O)CC(C)(CO1)C2 c1(C(=O)NC(C2N(C(C3N(CC)CCC3)=O)CCC2)(C)C)ccccc1SC N1(C(CC2CCN(C)CC2)=O)CC2(C1)CN(C(C1OCCN(C)C1=O)=O)CCO2 CCC(C(=O)NC(CNC(c1ccccc1)=O)C(C)C)n1cccn1 CCC(C)(C)CCCC(=O)NC1CCCCCC1C(N1CCCC1C(O)CO)=O C12(NC(C3CCCSC3)=O)CCCC1CN(C(c1cccc3sccc13)=O)C2 c1(N2CC3C(F)(F)C3C2)nc(NCC2C3COCC23)c2ccsc2n1 c1(C(N2C(CCCNC(c3c(C)n[nH]c3C)=O)CCC2)=O)cnn2c1OCCC2 c1(NCC2(NC(=O)C3CCCc4nn[nH]c43)COC2)cc2nn[nH]c2cc1[N+](=O)[O-] C(=O)(C1=NN(C(C)C)C(=O)CC1)N1C(C)CCC1.n1(CC)c(C=O)cnc1O.N Cc1nc2c(C(=O)NC34CCN(C(=O)CCc5cc[nH]n5)CC3C4)ccnc2[nH]1 c1(C(=O)NCC(CC=C)NC(C23CC(CC)(CO2)C3)=O)ccnc2ccnn12 c1(C(=O)NCC2CN(C(c3c(C)cc(O)nc3)=O)C2)cc2cc(Cl)ccn2n1 N1(C(c2c[nH]cc(C)c2=O)=O)CCCC(C2(NC(=O)CC(C)C(C)C)CC2)C1 C1(N(C(c2c(C)nns2)=O)C)CCCN(C(=O)C(c2ccc(F)c(F)c2)O)CC1 c1cc(F)cc(F)c1.C1(C=O)C2CC3C(C2)C13.C1(N(C(=O)C)C)CCC1.O C(=O)(C(CCC(C)C)NC(=O)Cn1nc(C)nc1C)NCC(CC)OC N1(C(CC(=C=C)C)=O)Cc2nccn2CC(NC(c2cccc(OC)c2)=O)C1 C1(OC)CC(NC(c2coc(Cl)n2)=O)CN(C(=O)CC2(C)CC2(Cl)Cl)C1 c1(C(N2CC(NC(C3(CC#C)CCCO3)=O)C(SC)C2)=O)nnc(O)cc1C c1(OC)cscc1C(=O)NCC(C)(C)OCC.C1(CCC=O)CCC(C)O1 N1(c2c(C#N)cc(Br)cn2)CCC2(CCN(C(c3cn4c(n3)CCCC4)=O)C2)C1 N1(C(c2c(CC)ncnc2)=O)CC(C)N(C(=O)C(CC)SC)CC1C CC(C)CC(F)C(=O)N1CCC(F)(CNC(c2cnc(C(F)(F)F)nc2)=O)C1 c1(CC)c[nH]cc1C(=O)NCCn1ccc(C(=O)NCC2CCOC2=O)c1 C1(NC(c2c(CC)nc(C)[nH]2)=O)CN(C(c2cccc(F)c2C)=O)CC1N=[N+]=[N-] CCCCCCCC(=O)NCC12CCC1CCN2C(=O)Cc1cccc(Cl)c1Cl C(=O)(C#CC1CCOC1)NCCCC1OCCN(C(Cc2c(C)nc(S)s2)=O)C1 c1(C(N2CCC(N(C(c3cncc(C=C)c3)=O)C)C2)=O)c(Cl)ccc(OC)c1N C1(C2CCOCC2)(C(=O)NC2(CN(C(CCCCC)=O)C)CC2)CC1 N1(C(c2cc(C(N)=O)oc2)=O)CC(C2CCCCN(C(=O)C3=CCCCC3)C2)C1 N1(C(CN2C(C)CCC2)=O)CCC(CO)(CNC(=O)CCS(C)(=O)=O)CC1 C(=O)(C(C)(CSC)NC(=O)C(O)CC)NCC1(CCOC)CCC1.S N1(C(Cc2c(C)ccc(C)c2)=O)C2CCC1CC(CNC(C1CCCCO1)=O)C2 C1(C(=O)OC)CCN(C(=O)CC2CC(O)CN2C(=O)CC2(OC)CCC2)O1 C(CN=c1[nH]n(C)cc1[N+](=O)[O-])(C(C)(C)C)NC(CC(CCOC)(C)C)=O c1(C(N2CCC(NC(C3(C)C(C)C3)=O)C2)=O)c(Br)ccc(Cl)c1F Cc1cc(NC(=O)CC2CC(NC(c3nnc(S)n3C)=O)C2(C)C)cc(F)c1 N1(C(C2C(COC)C2)=O)CC(CF)(NC(=O)C(C2CCOCC2)C)C1 C1(NC(COCC#C)=O)CN(C(=O)CC(C)CC)CCC1F N1(C(CCCC#C)C(=O)NCCCF)Cc2nccn2CC(CO)C1 Cc1cc(C)n2ncc(C(N3CC4C(CNC(c5sncc5C)=O)C4C3)=O)c2n1 C1(NC(C(OC)OC)=O)CCCN(Cc2nc(C)no2)C1 c1(N(C2CC3CNC2C3)C(=O)C=Cc2ccccc2)ccc(Cl)c(F)c1 C(=O)(C(c1cccs1)=Cc1ccccc1)NC(CNC(C(C)N1CCC1)=O)C C(C(C)N=c1nc(C(C)C)cc(OC(C)C)[nH]1)(C1CCCCC1)OC C(C(C)CN=c1[nH]c(N2CCN(C(=O)CC(F)(F)F)CC2)nc2c1CSC2)OCC Cc1cc(C(=O)C(=O)NCC2CCN2C(=O)C(C)NC(N)=O)ccc1F N1(C(C(CC)(C)O)=O)CCC2(CC1)CC2C(=O)Nc1cc(C)cnc1O CC1OC(C)C(C(=O)NCC2CCCCN2C(c2coc(Br)c2)=O)C1C c1(C(N(C2CCN(CC3CCS(=O)(=O)C3)CC2)C)=O)cnc2n1CCCCC2 C1(NC(CSCCOC)=O)CCOCC1NC(=O)CCc1ccc(CO)cc1 N1(C(CC(CCC)O)=O)CCC(C2(NC(=O)Cn3ncc(Br)n3)CC2)C1 C(CC(C(C)(C)C)NC(C1(C#N)CCOC1)=O)N(C(c1cc(C)c(Br)o1)=O)C N1(C(c2nc(OC)c(Br)cc2)=O)CCc2cccc(C(F)(F)F)c2C1 C(C(CO)(CO)NC(=O)CC1CC2(CCC2)C1)N(C(C(CC)O)=O)C C1(CN(C(=O)C)CC)CCCN1C(=O)CCOC1CC1.CC(N)=O.S c1(N2CCC(NC(CCN(CCCCOC)C)=O)(CF)C2)nc(C)cc(C)n1 C1(CNC(CCC)=O)CCN(C(c2ccn(C3CC3)n2)=O)C1 c1(C=O)cc(S(C)(=O)=O)cs1.N1(C(CC2N(CC)CCC2)=O)CC2(CCC2)C1 c12cc(cc(F)c1)CNC1CCN(C1)C2=O.Cc1nsc(C)n1.C(C)(C)C.O N1(C(c2ccc(C(=O)OC)cc2)=O)CCC(CO)(NC(=O)CO)CC1.CCF Cc1c(C(c2nnnn2C)NC(C)CC(C)C)cccc1NC(C)C C1(C(=O)NCCCCCNC(c2n(C)nnc2)=O)CC(C)(C)OC1(C)C C1(C(=O)NC(CC#C)CC)CC(F)(F)CN1C(=O)CCC1CCC(=O)C1 CC1CCN(C(=O)C(CNC(c2cncs2)=O)CC2CC2)CCO1 C1(CNC(=O)CC2CC2)C(C2CC2)CCN1C(c1cncc(F)c1Cl)=O c1(N2CCC(C)(CNC(=O)C(Cc3ccsc3)NF)CC2)ccc([N+](=O)[O-])cc1 C(CCC(=O)NCCC1(C(=O)NC(COC)CO)CCCC1)OCC C1(C(N2CCC(CN(C(CSCCC)=O)C)C2)=O)CCC(C(F)F)CC1 c1(C=O)n[nH]c2ccc(C)cc12.C1CCC1.C(C(=O)NCC(=O)N)NC(C)=O N1(C(CCSCC)=O)CCC(CO)(NC(C2CCCCN2C(C)=O)=O)CC1 N1(C(COCCCC)=O)CC(C(C(=O)N(C)C(c2nccs2)C)OC)C1 c1(OC)cc(Cl)c(C)cc1NC(c1cc2c(Br)csc2[nH]1)=O N1(C(Cc2cc(CC)no2)=O)CC(=O)CC1C(=O)NC1CCC1.C(C)(C)O Cc1ccsc1C=CC(=O)NCC(CNC(C1(CF)CC1(F)F)=O)CO C(N=c1ccnc(N2CCCC(c3cc[nH]n3)C2)[nH]1)c1c(C)nc[nH]1 C1(NC(C(C(C)C)C)=O)CCCN(C(=O)CNc2ccc(C#N)cc2)CC1 c1(C(N(C=O)Cc2nncn2C)C)cccc(C(C)(C)C)c1 c1(NC(C2CN(C(c3n(CC)ncc3)=O)C2)=O)ccc(C(C)=O)cc1C#N N1(C(C(c2cnn(C)c2)C)=O)CCC(NC(C2CN3CCN2CC3)=O)C12CCC2 c1(C(N2C(CN(C(=O)CC3(O)CCCC3)C)CCCC2)=O)noc2c1COCC2 C1(CC=C)CCCC1(c1nnnn1CCCF)Nc1ccc(C)cc1 C(=O)(C1=C2CCN=C2NC=C1)N1CCN(CCNC(=O)CCc2nncs2)CC1 N1(C(Cc2ccc(OC)cc2)=O)CCC(C2CCN(C(=O)CC3CSC3)C2)CC1 N1(C(C2N(C(C)C)CCC2)=O)CCCC(F)(CNC(=O)CS(N)(=O)=O)C1 N1(C(CCC=C)=O)CC2CN(C(=O)C=CCOC)C2C1 C1(NC(c2cc(C)nnc2O)=O)CN(C(C2C=CCS2)=O)C2(CCOC2)C1 n1(CCC)nc(C)cc1CN1CCC(OCCN)C1 c1(C(N2CCC(C(=O)NC(c3ccno3)C)C(O)C2)=O)cc(F)c(F)c(O)c1F c1(N2C(CNC(c3ccccc3[N+](=O)[O-])=O)CCCC2)ncc2cccnc2n1 c1(C(N2CC(C(C)NC(CC(C)(C)OC)=O)OCC2)=O)ccncc1Cl.C(C)=O C(=O)(Nn1cnnc1)C1(NC(C(C(C)C)NC(C)=O)=O)CCSC1 C(=O)(C(CNC(=O)CC1CCCOC1)CC=C)N(C(CC#C)C)C S(=O)(=O)(c1cccc(=NCC(c2cccs2)OC(C)C)[nH]1)N(CC(CCC)O)C C1(NC(c2c(C)nns2)=O)CC2(C1)CC(C(=O)N)C2.C12CC(F)(C1)C2.C c1(C(N2CCCC2)=O)ccc(N)c(N)n1.Cc1c(C(=O)NC)cnn1CC(C)C c1(NCCNC(C23CC2Cc2c[nH]nc23)=O)ncnc2c1nnn2CC1CC1 C=C=CC(C)C(=O)NCC1(CC)CC1.c1(CC(C(=O)N)C)c(C)n[nH]c1C c1(C(=O)NC2CC(C)(NC(Cc3c(C)ncs3)=O)C2)ccc(N=[N+]=[N-])cn1 c1(C(=O)NCC2CCN(C(CC(=O)NCC)=O)CC2C)cnc2ncnn2c1C Cn1cnc2c1C(C(=O)NC(C1CCC(F)(F)CC1)CCO)CC(=O)N2 C(=O)(CCC(F)(F)F)N.c1(NC(C)=O)ccc(C(=O)NCCC(C)(C)C)cc1 C1(C(N(C(CC)CO)C)=O)CCCN(C(=O)CCC2CCC(C)O2)CC1 C1(C(N2C(C(=O)NCc3c(OC)cccn3)C3CC3C2)=O)CCC(O)CN1C c1(OC(C(C)C)C(=O)NCC(C)N(C)C(c2ccnnc2)=O)ccc(F)cc1F c1(NCc2nnn(C)n2)[nH]c(=NCC2(C3CC3)CC2)nc2scnc12 N1(C(C(C)P(C)(C)=O)=O)CC(CNC(=O)Cn2cccc2)C2(CCOCC2)C1 O(NC(=O)C(CC(C)C)N(C)C(C1CC(C)CC(=O)N1)=O)CCCC n1(-c2cnc(C)s2)nc(C2CC23CC3)nc1-c1ccc(C2CCOC2)cc1 c1(C(=O)NCc2c(C(N(CC(C)(F)F)C)=O)nco2)occ2c1CCC2 CC#CCCCCN=c1nc(N(C)CCN2CCOCC2)c2cc(Cl)ccc2[nH]1 CCC(CC)C(C)C(=O)N1CC(O)(CCNC(=O)C(c2ccc(Cl)s2)C)C1 c1(CCN(c2csnc2C)C(N(CCC)CC)=O)ccccn1 N1(C(c2c(CCC)nco2)=O)CCCC(C)C1CNC(=O)C.c1ccccn1.N c1(CC(C)C(=O)NCCC2CCC2)ccccc1Cl.C1(C)(C=O)CNC(=O)C1.N c1(C(C(F)(F)F)NCc2ccc(C)[nH]2)c(F)cccc1F CN(C)S(=O)(=O)NCC(=O)OCC1COC(=O)O1 C1(NC(C(C2CCCCC2)OC)=O)CC2(C1)CC2.c1(CC=O)cc(C)on1.N N1(CC)CCN(C(=O)C(=O)N2CCC2C2CCCOC2)CC1 CC(C)(CC(=O)NCC1CC(F)(F)CN1C(=O)CC(C)(C)C)CC(F)F Cc1cc(CNC(=O)Cn2nccn2)oc1C(=O)NCC(C1CCCC1)O CC1(C)CCCCC1(C)NC(=O)CC1CCC(NC(=O)CCc2nc(O)n[nH]2)C1 c1(C(N(CCNC(c2cc(C(N)=O)cc(C)c2)=O)C)=O)c(C)oc2ccccc12 C1(C(N(CC(=O)NCC(=C)F)CC2CC2)=O)CC2C=CC1C2 c1(C(=O)NCC2C(NC(c3c(C)cc(F)cn3)=O)CCC2)cc2cccnn2n1 C(=O)(C(C)(F)C(=O)NCC1CCCCN1C(=O)CCn1cnnn1)OCC Cc1cc(O)nc(C)c1C(=O)NC(C)CNC(=O)CCc1cncnc1 N1(C(C(CN(C)C)O)=O)CC(C)(C)OCC1CNC(=O)Cc1ccsc1Cl C(=O)(C1=CC2CCCCCC12)NC(CNC(Cc1cccc(CC)c1)=O)(C)C c1(CC(=O)NCC#CCNC(Cn2c(CCC)ncc2)=O)ccnc(Br)c1 CC1(C#CC(=O)N2CCC(NC(c3c[nH]nc3[N+](=O)[O-])=O)C(CO)C2)CC1 C(=O)(C(C)(C)Cc1cn(CC(=O)N)nn1)OC.C1CC1.C(C)(C)C.C=O N1(C(C(C(C)C)C)=O)CCC2CN(C(c3csc(-c4cccnc4)n3)=O)CC2C1 O=C(N=c1[nH]c(Cl)ncc1O)c1ccc(NC(c2ccon2)=O)cc1 C12(C(=O)NC(c3cn[nH]c3)C)CC1CN(C(=O)CCN(C)C)C2 C1(C(=O)NCC(CNC(CC2(OCC)CC2)=O)O)CCC(C2CC2)CC1 Cc1cc(C(N2CC3C(C(=O)NCCCc4ccccc4)C3C2)=O)n(C)n1 C(=O)(C(O)CC[S+](C)C)N1CC(n2cc(CNC(c3ccc(C)s3)=O)nn2)C1 c1(N(C2CNCC2C#N)C(c2c(C)ccc(C)c2)=O)ncnc2cnccc12 N1(C(C#CC2(C)CC2)=O)CCC2(CCN(C(c3cc(C#N)no3)=O)C2)C1 C=C(C)CC(C(=O)N1CC2CC2C1C(=O)NCC1CSCCO1)OC c1(N2CCC(CNC(=O)CC34CCC(CC3)OC4)C2)ccc(S(=O)(=O)N)cn1 C(=O)(CC1=CCN(C(=O)C(N)=O)CC1)NCCC(CC=C)(C)C C1(C(=O)NCCN(C(C(CC)SC)=O)CC2CC2)CCCC2(CCC2)O1 CC1CN(C(=O)Cc2ccsc2)CCC1N(C)C(c1cc2n(n1)CCO2)=O CC(c1ccccc1C)=CC(=O)NC1CC(NC(C2CC2C2CCCCC2)=O)C1 Cc1c(C(=O)NC2CCCC2NC(=O)CCC2CC2(Cl)Cl)cccc1O CCCCC(C(=O)NC1C2CCN(C(=O)Cc3csnn3)CC12)NC(N)=O N1(C(C2CC(C)(NC(CCOCC)=O)C2)=O)CCC(O)C1CC c1(OC(C)C)cc(Cl)ccc1Cn1nnnc1N1CC=C(Br)CC1 c1(C(N2CCC3(NC(C4COCCOC4)=O)C(C2)C3)=O)cn2cc(Cl)cnc2n1 c1(C(CC)C(=O)NCCNC(C2(c3ccccc3)CCOC2)=O)ccc(F)cc1 c1(C(=O)OCC)ccc2c(-c3ncc(CN)o3)cn(C)c2c1 CC(F)(F)CCC(=O)NC1CC2CC1CC2C(=O)NCc1nn[nH]c1C1CC1 CCCCCC(CCCCC)C(=O)N(C(C)CN(C(=O)CC(C)C(C)(C)C)C)C C1(NC(CC2OCC(C)(C)C2)=O)CN(C(=O)CC23COC(C2)C3)C(C)(C)C1 Cn1nc(CNC(c2cncnc2)=O)c2c1CCN(C(C1CCC1)=O)C2 Cn1ncc(CN2CCCC2CC(C2CCCCC2)=O)c1Br Cc1cc(C(N2CCC(CC(=O)NCC3CCO3)CC2)=O)ccc1I c1(CN2CCCC(C(=O)Nc3cncc(C)n3)CC2)c[nH]c2cccc(F)c12 C(=O)(CCC(F)(F)F)N(C(C)C(=O)NCc1ncnn1C1CC1)CC c1(OC(C)C(=O)Nc2nnc(-c3c(F)cccc3F)o2)ccc(S(C)(=O)=O)cc1 c1(NC2CCCN(C(CCC3C(C)(C)C3)=O)C2)ccnc2ncnn12 C1(CN(C)C(c2cnc(C(N)=O)cn2)=O)CCCC(NC(=O)CCCF)C1 CC1CC(=O)CCC1C(N1CC(C)(NC(=O)C2=NOC(C)C2)C1)=O N1(C(C(C(CC)C)N(C(=O)CC2(C)CC2)C)=O)CCC2(C=CCO2)C1 c1(C(=O)NCC2(NC(C3CN(C)C3)=O)CCCCC2)cc(Cl)cc(Cl)c1N c1(C(N(CCNC(C2(C#N)CC2)=O)CC)=O)ccc2ncnn2n1 CCCN=C(NCC12CCCC(C1)OC2)NCC1CC1(C)C c1(C(N2CC(NC(Cc3nnc(C)o3)=O)C(C)C2)=O)cc(C)c(Br)cn1 C(C(C)(C)C(=O)NCC(C1(O)CCN(C(C2C(C)(C)C2(C)C)=O)C1)C)OC c1(C(=O)NC(C2CCCCC2)C)cc(C)on1.c1(C=O)ccoc1C1CC1.N C12(NC(CC(=O)NC)=O)CCCN(C(=O)CN3CCC3)CC1C2 Cc1c(Br)sc(C(N2CCN(C(=O)Cc3cncn3C)C(C)C2)=O)c1C C1(CC(=O)NC2C(C)C2C)CC(C)(C)CN1C(=O)CC1CCN(C)C1=O C(=O)(C(F)CCCCCC)N(C1CC(CC2C3COC(C)(C)OCC23)C1)CC=C N1(C(C(C)P(C)(C)=O)=O)Cc2ccnn2CC(NC(c2cnc3sccn23)=O)C1 CCCC(O)C(=O)NC1CC(CNC(=O)C(c2cccc(C)n2)(F)F)C1 c1(OC)ncc(Br)c(=NCC(C)(C2CC2)NC(c2ccnc3ccccc23)=O)[nH]1 N1(C(c2c(C)n[nH]c2)=O)CC2CC(C(=O)NCC(CO)C3CCC3)(C2)C1 C1(N(C(COCC#C)=O)C)CCN(C(c2cc(-c3ccccn3)[nH]n2)=O)CC1C c1(CC(=O)N(C)CC2CCCN2C(=O)Cc2cn[nH]c2)noc2cc(F)ccc12 C1(CNC(c2ccoc2Cl)=O)CN(C(c2ccoc2)=O)CC(C(F)(F)F)O1 CCCC(C)(C)CC(=O)N1CCCC(CC(N2CCC(CF)C2)=O)CC1 C1(C(C(=O)NCCCNC(=O)OC)C)CCN(C(=O)Cc2ccco2)C1 C1(NC(C(C)SC(C)C)=O)CN(C(c2cc([N+](=O)[O-])c[nH]2)=O)Cc2ccnn2C1 c1(C(=O)NCC(C)CN(C(=O)CCC2CC(C)(C)CO2)C)ccc2ccoc2c1 Cc1[nH]nc(-c2nnc(N3CCOC(c4ccsc4)C3)n2CC(C)C)c1Cl c1(C(N2CCCC3CCCCC23)=O)[nH]nc2c(-c3ccc(O)cc3F)cccc12 C1(CN(C)C(c2csc(Br)c2)=O)CN(C(C2CCOC2)=O)CCO1 CC1(C)CCOC1CC(=O)NC1CC(CCNC(c2cncs2)=O)C1 c1(C(N2CCN3C(=O)OCC3C2)C(=O)NCCCSC)cccc2ccccc12 N#CC1(C(=O)NCC2CCCN2C(=O)Cn2cnnc2O)CCOC1 C(=O)(C#CC1(C)CC1)N(CCN(C(c1ccc(CCN(C)C)cc1)=O)C)C C(=O)(CC(C)CC(C)C)N.Cc1cc(C(=O)NCC2(C)CCCCC2)c(O)nn1 c1(C(N2CCC(C)C(NC(CC(=O)NCC)=O)C2C)=O)csc2c(F)cccc12 n1(C(F)(F)F)ncc2c1CCCC2n1cc(CC2CCC(F)(F)CC2)nn1 C(=O)(CCCCCC(C)O)NC1(CC=C)CN(C(c2cccnc2OCC)=O)C1 C(=O)(CC(C)(C)O)NCCOC1CN(C(c2scc(OC)c2)=O)C1 N1(C(C(C)(C)OC)=O)CC(C(=O)Nc2ccc(N3CCCC3)c(Br)c2)CC(F)C1 c1(C(=O)NC2CC(NC(C(C)C(F)F)=O)C2)ccnc2cc[nH]c12 CC(C)C1=CCC(NC(=O)CCC2CCCN(C(c3cc(CO)[nH]n3)=O)C2)CC1 C(=O)(CC(C)P(C)(C)=O)NC1(CF)CN(C(c2c(CC)[nH]nc2Cl)=O)C1 c1(NC(C23CC2CN(Cc2cccnc2O)C3)=O)ccc(C2CC2)cc1F C(=O)(C1CCCn2cnnc21)N1CCN(C(CN(C(CC(C)SC)=O)C)=O)CC1 c1(CNC(CC2(NC(c3n(C)cnc3)=O)CCC2)=O)c(O)cccc1F C#Cc1cc(C(=O)NCC2CN(C(c3ccoc3C(C)C)=O)CCO2)cc(N)c1 C(=O)(C1CCCc2nncn21)N(CC(C)(C)NC(C=CCOC)=O)C CC1(C(N2CCCCC(CCC(=O)NCCc3ccco3)C2)=O)CCCCCC1 C=CCC(CNC(=O)CCc1cc(C)no1)C(=O)NC1CCN(C)CC1C Cc1cccc([N+](=O)[O-])c1C(N1CCC1)=O.C(c1ccc(F)c(Cl)c1)=CC=O.N N1(C(C(C)(C)C)=O)CCN(C(c2ccc(C3OCCO3)cc2)=O)C2CC12 C1(C(=O)NC(C)CCCCNC(c2cc(C(N)=O)[nH]n2)=O)CCC(C2CC2)CC1 c1(C(=O)NCC(CNC(=O)CC2CCOC2)C(F)(F)F)ccc(F)c(F)c1F N1(C(C(C)=O)=O)CC2CC(NC(c3cc([N+](=O)[O-])c[nH]3)=O)C2C1 C(CNC(c1cc[nH]c1-c1ccccc1)=O)(CC(C)C)NC(c1ccc(C)o1)=O C1(CNC(Cc2ccc(C)s2)=O)CN(C(=O)Cc2cnc[nH]2)C2(CCC2)C1 S(=O)(=O)(c1cccc2c(OC)cccc12)NC(CCC(=O)OC)CCC(=O)OC c1(C(N2CC3C(CC(=O)NC4(C)CCOC4=O)C3C2)=O)cncc2[nH]ccc12 N1(C(C2(CC)COC2)=O)CCOCC(NC(c2ccc(C(C)C)c(F)c2)=O)C1 CC1(CC(=O)NC2CCC(CNC(c3ncc(F)cn3)=O)CC2)CC(F)(F)C1 C(=O)(C(F)(F)c1csc(=N)[nH]1)NCC(C)NC(C1(C)CC1(Cl)Cl)=O c1(NC(=O)NCC=C)ccnc2c1nnn2C C1(C(=O)NCCN(CCCC)C)CNC(=O)CN1C(=O)C(C)CC(=O)OC c1(C(=O)NC2CN(C(c3cc(C)ns3)=O)C(C)CC2)cnc(C)c(C#N)c1 CCCC(CC)C(=O)N(C1CCN(C(=O)CC(C)c2ccncc2)CC1)C N1(C(Cn2nnc(C)n2)=O)CCCC1(C)C(=O)N(C)CCOCC1CC1 N1(C(C)=O)CC2(C)CC1(C=O)C2.c1cn(C)nc1C1CC1.C(=O)(C)NC.O CC1CCn2ncc(C(N3CCC(C)S(=O)(=O)CC3)=O)c2C1 C(=O)CS(=O)(=O)C(C)(C)C.CC1CN(C(=O)CC2CC(C(F)F)C2)CC1C C1(CC(=O)N(CC(C)CNC(C2(C(F)F)CCC2)=O)C)CCCCN1C c1(CC)cc(C(N2CCC(NC(C3CCOC3CC)=O)C2)=O)no1 N1(C(C(C=C)(C)C)=O)C2CC=C(C(=O)NCc3nc(CC)ns3)C1CC2 Cc1nn(C)c2nc(C(=O)Nc3ccc(CN4CCS(=O)(=O)CC4)cc3)ccc12 CCC(CC(C)C)C(=O)NC(Cn1cncn1)C(=O)NCc1ccc(Cl)nc1 C(C)(CCC(=O)N1CCC(C(C)(C)C(=O)NC(C)C(O)C(F)F)C1)OCC N1(C(C23CC(C(C)C)(C2)C3)=O)CC(NC(=O)CCc2ccco2)C2(CC2)C1 C(=O)(C1CCCc2nccn21)N1CCC(NC(c2ccc3nccn3n2)=O)CC1 C(C)(C)(C(=O)NCCCO)OCC.C1(C2(C=O)CC2)CCCN1C(C)=O N1(C(c2c(OC)n[nH]c2)=O)CC(N(C(=O)CS(=O)(=O)N(C)C)C)C(F)C1 n1(CC=O)cnc([N+](=O)[O-])c1.C(=O)(CCC(=O)NC(C)CCCC)NCC.N C1(NC(C2(CC=C)CCC2)=O)CC(O)(CNC(c2sccc2)=O)C1.O c1(CCC(=O)NC(C)C(=O)NCC(F)(F)F)cn(CCC2CC2(Cl)Cl)nn1 C(C(=O)N(CCCO)OC)C1N(C(c2c(C)cc(OC)nc2)=O)CCOC1 c1(C(=O)NCC(CN(C(c2c(CC)nccn2)=O)C)C)cc(C)cc(C)c1C c1(C(=O)NCCC2(OC)CN(C(C3CC=CCO3)=O)C2)ccc(F)c(Cl)c1N Cc1nnc2n1CC(C(=O)NC13CC(C)(C1)C3)CC2.C1(C(=O)N)COCCN1C C(=O)(C(C)S(N)(=O)=O)N.C1(C(=O)OC)C2CN(C(=O)CC3CC3)CC12 c1(OC)ccc(CN2CCC(C(=O)Nc3cnc(Cl)c(C)n3)C2)cc1Br c1(N(c2ccc(=N)[nH]c2)C(c2cc[n+]([O-])cc2)=O)ccnc2cc(Br)nn12 N1(C(CC(CC)C)=O)CCN(C(c2cc(O)nc(O)n2)=O)CC(CO)C1 Cc1ccccc1-c1cn(CC(=O)N(C(C)Cc2nn[nH]n2)C)nn1 CC1CC(CNC(=O)C(F)C2CCOC2)CN1C(=O)CSCc1cccs1 c1(OC)c(C(=O)NCC2CC2NC(=O)CN(C)C)cc(Cl)cc1C N1(C(C(C)OCCOC)=O)CCC2CN(C(c3cncc(C4CC4)c3)=O)CC12 S(=O)(=O)(c1ccccc1[N+](=O)[O-])N(C(c1c(F)cc(OC)c(F)c1F)=O)CCO C(=O)(CC(C)C(F)(F)F)NCC(CNC(c1cc(C)on1)=O)(C)C C1(C2CCN(c3cc(C#N)ccc3[N+](=O)[O-])CC2)(NC(COCCOC)=O)CC1 C(=O)(CCc1ccccc1)N(CC)C.c1(C=O)ncc[nH]1.C(C)C.C(C)=O Cc1csc(C(=O)NC(C)(C)CNC(c2c(C(F)(F)F)noc2C)=O)c1Cl C(=O)(C(O)P(C)(C)=O)NC1(C)CCN(C(c2cccc(OC3CC3)c2)=O)C1 C(CCC(C)CC(=O)N1CCC2(NC(=O)CCC3(O)CCC3)CCCC12)=C(C)C CC(C(C)C(=O)N(CCO)C1CC1)NC(=O)CCn1ccnn1 S(=O)(=O)(c1cccc(C(=O)O)c1Br)NC1(C(C)C)CCC1 C(=O)(C(C)(C)C1=CCN(C(=O)C(O)C2=CCCCC2)C1)NCC1N(C)CCCC1 C1(C(N2C(CNC(Cn3ncc(C)c3)=O)C=CC2)=O)CCOCC12CCCCC2 c1(C(=O)OCC)ccc(NC(=O)NC(C2CCOC2)C)o1 c1(OC)nc(=NCC2CCC(CNC(=O)CC3CCCC3)CC2)[nH]c(C)c1F Cc1cc2ccccc2c(C(N2CCN(C(C3CC3C)=O)CC(C)(C)C2)=O)c1C C(=O)(C(=O)NNc1ccc(C(F)(F)F)cc1F)Oc1c(NC(=O)OC)cccc1 Cc1cc(Sc2cccc(-c3n[nH]c4c3CCC4)c2)n2ncnc2n1 Cc1cc(C(N2CC(NC(=O)CCC3CC3)C3(CCC3)C2)=O)c(C)nc1C c1(C(=O)N)ccc(C2CNC(=O)C2)cc1.C(=O)(C1=CCC1)N(C)CC1CC1 C12(NC(c3c(CC)c[nH]c3)=O)CCCCCC1N(C(=O)C(O)C(C)C)CC2 CC1C(NC(=O)CC2CC23CC3)CCN1C(c1ccc(N2CCCC2)nc1)=O N1(C(CNC(C)=O)=O)CCC(O)(CC)C1.c1(C(=O)N)cc(-c2cccnc2)no1 CN1CC2(CCCN(C(C(=O)Nc3ccccc3)c3cnsc3)C2)CC1=O C12(CNC(C(C)C)=O)CCCCC1N(C(C1CC3(C1)CC(C)(C)C3)=O)CC2 n1(CC(=O)NCC2CC(CCO)C2)cc(C(N2CCC(n3ccnn3)C2)=O)cn1 Cc1cc(C(N2CCC(CNC(=O)CCc3ccoc3)CC2)=O)cnc1Cl c1(C(N(C)CCNC(=O)C=CS(C)=O)=O)coc2c1NC(=O)CCC2 C(=O)(C1CCc2ccc(C)cc21)N(CCNC(c1c(CCC)n[nH]c1)=O)CCC c1(C=O)ccc2c(n1)CCC2.C1(NC(c2cc(C3CC3)on2)=O)CCCC1C c1(C(N2CC(NC(C(C)(C)CO)=O)C(O)C2)=O)cc(Cl)ccc1OC1CCCC1 C1(CNC(C2C(C(=O)OC)C2)=O)CN(C(=O)C(O)c2ccco2)CCO1 C1(C(=O)OC)CCn2c(cnc2N2CCCN(C(c3cccc(C)c3)=O)CC2)C1 c1(C=O)n[nH]c2c1CS(=O)(=O)CC2.N1(C(COCCC#C)=O)CCC(C)C1C N#Cc1cc2c(nc1O)CC1CCC2N1C(=O)NCc1cnc(C(F)(F)F)[nH]1 c1(OC)ccc([N+](=O)[O-])c(C(N2CCC(C)(NC(=O)C(C)C3CC3)CC2)=O)c1 c1(CNC(=O)NC2(C)C(C(=O)OC)CCCC2)cccc2cn(C)nc12 C1(CNC(CN(CCC)C)=O)(NC(C2(C)CC2(F)Cl)=O)CCCC1 C1(CC)CC2CCC(C1)N2C(=O)C(O)C(C)C.c1(OC)ncc(F)cc1C=O.N c1ccc(Cl)cc1.C(F)(C(=O)N(CCNC(=O)CCS)CC)OC.CCO c1(C(N(CC)CC2CCCN2C(c2cnc[nH]2)=O)=O)cc2ncccn2n1 c1(CC=O)cccc(Br)c1C.C1(N(CCC)C(C2(CC)CC2)=O)CCC1(C)C CCCCCC(C)NC(c1cc(OC)ncn1)c1nnnn1CCC C1(C(N2CCC(OC(C)=O)CC2)=O)(OC)CCN(C(=O)CCCC2CC2)C1 c1(C(C(=O)N)O)ccc(F)c(F)c1.c1(C(N(CCC)C)=O)cn(CC(F)F)cn1 CC(CNC(c1cc(C(C)(C)C)no1)=O)N=c1[nH]cnc2cnn(C)c12 C1(C(=O)NC(C#C)C(C)C)CN(C(C2(C)CC2)=O)CC1(F)F N1(CC(=O)N(C(C)C2CC2)CC)CCC(C(=O)N)(OC)CC1.C1CCCO1 c1(C(N2CC(CNC(C3CC(C)C3)=O)OCCC2)=O)cccc(C#CC2CC2)c1 N1(C(Cn2c(C)ccn2)=O)CCN(C(c2ccc(F)cc2)=O)CC1CC(F)F C1(C(=O)NCC(O)CN(C)C(C2CC2(C)C)=O)(OCC)CCOCC1 C1(NC(C2(CC#C)CCCCC2)=O)COCCN(C(c2cc([N+](=O)[O-])n[nH]2)=O)C1 C1(NC(C2(CNC(CC3(N(C)C)CCC3)=O)CCC2)=O)CC12CCCC2 C(=O)(C#CC1(C)CCCO1)NC1C(C)N(C(c2ccc(F)c3occc23)=O)CC1 C1CC(O)CN1C=O.c1(C(C=CC(=O)NC)=O)coc(Cl)n1.c1ccccc1 c1(CC)cc(C(=O)NCC2CC(NC(c3ccsn3)=O)C2(C)C)c(C)nn1 C1(N(C(C(CNC(c2c(CC)noc2)=O)O)=O)C)CN2CCC1CC2 C(=O)(C(C)C(O)C(C)C)N(CCCCN(C(C=CC(C)(C)SC)=O)C)C c1(C(N2CCN(C(CCc3cn(C)nc3)=O)C(CO)C2)=O)cc2n(n1)CC(F)C2 c1(NC(N2C(CC(=O)OCC)CCC2)=O)cc2c(nc1O)CCCC2 C1(C)(CCOC)CN(C(C(=O)NCCCF)C2CCCC2)CCO1 c1(NC(N2C(c3c(F)ccc(C)c3F)CCC2)=O)ccc2c(c1)N(C)C(=O)CO2 c1(N2CCC(=CCC)C2)nc(N2CC=CC(OC)C2)nc2c1ncn2C C1(O)(c2c(C(N3C(CNC(C4(C#N)C(C)C4)=O)CC3)=O)cco2)CCOCC1 C1(C(N(CCC(=O)NC2CN(C(C)=O)C2)C(C)C)=O)CCC(F)(F)C1 c1(C(N2CC(F)(C(=O)OC)C(CN)C2)=O)cccc(Br)c1F c1(OC)cnncc1C(=O)NC1(CO)CCN(C(C2(C)CCCO2)=O)C1 CC(C)C#CC(=O)NC1CC(OCC(=O)N(C2CCOC(C)C2)C)C1 C(CCCCNC(=O)CC1CSCCO1)N(C(=O)C(=O)N(C)C)C(C)C C1(CCC)CN(C(=O)CCC2CC2)CCN1C(=O)Cc1c(C(C)=O)cccc1F N1(C(COC(C)C)=O)CCc2ccc(CNC(=O)Cc3cn[nH]c3)cc2CC1 C1(CNC(C(F)OC)=O)(CNC(C2(C)CCCCO2)=O)CCOCC1 C(=O)(C1=C(C)CCC1)NCC1C(OCC)CN(C(c2cnc(O)n2C)=O)C1 CC1OC2(CNC(c3ncccc3N)=O)CC1(NC(=O)CCCc1nccs1)C2 C1CCS(=O)(=O)C2(C1)CCC2.CC(C(=O)N)C(C)(C)C.C(=O)CSC(=N)N c1(C(N(C2CN(C(=O)C3=CC4CCC3C4)C2)C)=O)cc2ccc(Br)cc2[nH]1 Cc1cc(C)c2c(C)c(C(N3CC=CC3(C)C)=O)[nH]c2c1 Cc1[nH]c2ccnn2c(=O)c1CC(=O)NCC1CCN(C(=O)C(C)(F)F)C1(C)C CC1(C)CCOC(CN=C(NC2CCCCC2)NC2CC23CCC3)C1 Fc1cnc(C2CC(NC(=NCc3cncs3)NCC(F)F)C2)nc1 c1(C=O)cc(N)c(Cl)cn1.C1(C(N(CCCN(C)C)CC)=O)CCCC1(F)F.N C1(n2cc(C=CC)nn2)CCCN(C(C2CC(C)(C)CO2)=O)CC1 c1ccc2nc(-c3ccc(CNC4CCNC45CC5)o3)ccc2c1 c1(C(N2CCCC(NC(COC(C)C)=O)C2C)=O)cc2c(F)cccc2[nH]1 CN1CCN(Cc2cn(CC3CCCCN3C(c3cc(O)n(C)n3)=O)nn2)CC1 C(=O)(CCCC=O)NC(C)C.C1(CC)CN(C(C2CCS(=O)(=O)N2)=O)CC1C.N N1(C(CN(C(C)C)C)=O)C(C(=O)NCCN2CCCC(O)C2)CCC12CC2 C1(CC(=O)NC(C2CCCCC2)CNC(c2c(C)occ2)=O)CCCNC(=O)C1 c1(C(=O)NCCCNC(CCc2cn(C)nc2)=O)ncncc1F CCCC(CCC)C(=O)N1CCCC(CCC(=O)NCC2CCC(=O)NC2C)C1 n1(CC)cnc(CNC(=O)C(N)CC2CCC2)n1 CCC(COC)C(=O)N(CCCCN(C(=O)C(C)Sc1ccc(F)cc1)C)C c1(CN(CCC)C(=O)NC(C2CCC(C)CC2)CC)ccccc1F CC1(C)CCC(CNC(=O)CO)N(C(=O)CC2CCOC2)C1.C1(C)CCC1 N1(C(CC=CC=C)=O)CC2CCC1C(NC(c1cnn(C(C)C)c1Cl)=O)C2 CCC(CC(=O)N1CC(C(=O)NCCC(=O)OC)C2(CCC2)C1)C(F)F C1(C)(CC)CCN(C(C2CCN(C(=O)CC3CCCCO3)CC2)=O)C1 CC1CCCC=C1C(=O)NCCCCNC(=O)CC1COCC(C)(C)O1 n1(CC(=O)N(C2CCN(C(C(CC)CCOC)=O)C2)CC)cc([N+](=O)[O-])nc1C C(C(C(=O)NC1(C(=O)NCc2csc(C)c2)CCC1)OC)OC CC1CC(c2cn(CCc3ccccc3)nn2)CCN1C(C1(O)CC(C)(C)C1)=O Cc1ccnc(O)c1C(N1C(C(=O)NCCCS(C)=O)CC1C)=O c1(CC(=O)NCC(C)NC(=O)C(C)P(C)(C)=O)coc2ccc(F)cc12 N1(C(CC(C)F)=O)CCCC(CCc2ccccc2NC(=O)OC2CCCCC2)C1 C1(C(=O)NC2C(OC)CN(C(=O)C=CCF)C2)CCc2ncsc2C1 Cc1ccc2cc(C(=O)NC3CN(C(=O)C(N4CCN(C)CC4)C)C3)ccc2c1 O=C1CC(NC(c2nnnn2C2CCCC2)CCC2CC(F)(F)C2)C(=O)N1 CC(C)C(O)C(C)(C)C(=O)NC(c1nccc(O)n1)C Nc1ncnc2c1ncn2CCNC(=O)C1=CSCS1 c1(C(N2CC3C(NC(c4c(SC(C)C)nccc4)=O)(C3)C2)=O)ccc(N)cc1F c1(OC)ccc(C(C)NC2CC2)cc1.C1(CO)CCC(C(F)(F)F)CC1.O c1(CNC(NCCN2C(C)CCCC2)=NCCF)cccc(S(N)(=O)=O)c1 N1(C(c2n(C=C)nnc2)=O)CC2(CC2)CC1CC(=O)NCCc1cc(CC)no1 C1(C(=O)N)CC(C)(C)CCO1.CC1C(N(C)C)CCN1C(c1c[nH]nc1CC)=O c1(C(N2CCN(C(CC=C)=O)C(C3CC3)C2)=O)ccn2ncc(C)c2n1 C1(C(=O)NCc2cn(C)nc2)CCCC12CCN(C(=O)CCC1CCOC1)C2 CC1CC(C(=O)N)N1C(c1cc(C(N)=O)[nH]n1)=O.C1(C(N)=O)CCCC1.C CC1CN(C(=O)Cc2ccco2)CCN1C(c1coc(CC2CC2)n1)=O c1(C(=O)NC2C(NC(C=C3CCC(C)CC3)=O)CCCC2)cc2ccccn2n1 N1(C(CC(=C=C)C)=O)CCC2C(CCCN2C(=O)CNS(=O)(=O)N(C)C)C1 Nc1c(C(N2CC(F)CC2CNC(=O)C=O)=O)ccc(F)c1Cl.CC(F)(F)F Cc1ccc(C(=O)NCC(C)CN(C(=O)C(C)N(C)C)C)c(C)c1 CCC(C)C(O)C(C)C(=O)NCCCCC(=O)O CC1CN(C(c2cncnc2)=O)CCC12CCN(C(c1ccc(O)cc1)=O)CC2 S(=O)(=O)(c1ccc(Cl)cc1)N1CC2(N(C(c3nccc(OC)c3)=O)CC2)C1 N1(C(CNC(CC)=O)=O)CC(NC(C2Cc3nncn3C2)=O)C2(CC2)C1 C1(C(=O)NCC2(C)CCN(C(C(CC)(C)OC)=O)C2)CCC2(CC1)CC(O)C2 N1(C(C=NOC)=O)CCC(C2(NC(C3CC(C)OC3=O)=O)CC2)CC1 N1(C(C=Cc2ccc(C)o2)=O)CC2CC(NC(=O)C3=CCCCC3)C(C2)C1 C(CCCCCNC(C1(O)CC1(C)C)=O)N(C(C=CCCC)=O)C Cc1n[nH]c(C)c1C(=O)NC1C2CN(C(=O)CCC(=O)c3ccncc3)CC12 CC1CC(NC(c2cncc(-n3ccnc3)n2)=O)CN1C(=O)CN(C)C(N)=O N1(C(C2(C)CCN(C(C(C)C3CCCO3)=O)CC2)=O)CCCCCCC1C N1(C(CC2CCC(NC(c3c(C#C)cnn3C)=O)C2)=O)CCCC(C)(OC)CC1 CC(CC(=O)NC1(C)CCN(C(=O)C2=CCSC2)C1)C(=O)c1cccc(F)c1 Cc1nn(C)cc1C(C)C(N1CC(NC(=O)Cc2cncn2C)C(C)C1)=O C1(CN(C)C(c2c[nH]c(=N)o2)=O)CCCN1C(C1CC1c1cncs1)=O c1(C(N2CC(NC(c3n[nH]c(C)c3C)=O)C3(C2)CC3)=O)nc2c(s1)CN(C)CC2 Cc1ccc(NC(C2CC(NC(=O)C=Cc3ccc(C)o3)CCO2)=O)c(O)n1 C1(NC(CC2CN(C)C2)=O)CC2CC(C1)CN(C(c1cc3ccccn3c1)=O)C2 Cc1ncc([N+](=O)[O-])n1CC(=O)NC1CCCC(N(C(=O)C)C)C1.CC(C)C.O c1(OCC=C)cc(Cl)ccc1C(N1CC(NC(c2ccon2)=O)CCC1C)=O c1(C(=O)OCC2CCCOC2)cccc(OC2CCOCC2)n1 C1(CNC(CCC)=O)CCCCN(C(=O)CNC(c2ccco2)=O)C1 c1(C(N2C(C(=O)Nc3ncc(SC)s3)CCC2)=O)c(F)ccc(I)c1F N1(C(c2cc(Cl)ncc2F)=O)CCC2C(CCCN2C(c2ccsc2Cl)=O)C1 Cc1cc(C(N2CCC(N(C)C(c3ccn(CC(F)(F)F)n3)=O)C2)=O)cc(C)n1 N1(C(C(c2nc(C)sc2)=O)=O)CCCN(C(=O)C=C2CCCC2)CC1C C1(CCC)CN(C(=O)C(O)P(C)(C)=O)CCN1C(c1csc(Br)c1)=O c1(OC)cc(Cl)c(Cl)cc1C(=O)NC1CCN(C(c2cnsn2)=O)CC1F CCC(O)C(C)C(=O)NCC1(CC(=O)NCCCCCN(C)C)CC1 C(=O)(C(CCSC)NC(=O)C=CCN1CCC1)NC1CN(CCC)C1.C C(=O)(CC(F)(F)C(F)(F)F)N.CC1(C)CC(C)CN1C(C1CCC2CC2CC1)=O c1(C(N2CC(O)(CC)C2)=O)ccc(S(N)(=O)=O)s1.C(C=O)C1CCOC1.CO C=CC1CN(C(=O)Cc2ccccc2F)CC1NC(C1CC12CC(F)(F)C2)=O c1(N(CCN(C(C2COC(C)C2)=O)CC)C)ccccc1Br c1(C(N2CC(NCc3cnccn3)CC(C)C2)=O)cc(Br)cc2[nH]ccc12 c1(C(=O)NCC2N(C(c3c(CCC)n[nH]c3)=O)CC=C2)ccc2cnnn2c1 C(=O)(CCCS(N)(=O)=O)N1CCN(C(c2cnc(C(C)(C)C)s2)=O)C(CCO)C1 c1(C(=O)NC2(COC)CN(C(=O)CS)C2)snc2ccccc12.CCC(C)C C1(CC(=O)NCCCC)CC(C)(C)CO1.c1(CC=O)cccc(C(F)F)c1.N c1(C(=O)NCCN(C)C(C2CC2(F)F)=O)cc(C(F)F)nn1C N1(C(C(CC)N(C)C)=O)CCN(C(=O)CC2CCC(C3CC3)O2)C2(CCC2)C1 CC(C)CC(C(=O)N)C(N)=O.C1CCN(C(=O)CCc2n[nH]c(=N)s2)C1C(C)C C(=O)(CCC(=O)N(CC(C)NC(=O)Cn1cnnn1)C)NCC c1(C(N2CC(O)(C(C)NC(COC(C)C)=O)C2)=O)ccc(C(F)F)nc1 c1(C(=O)NCC(CNC(CC(C=C)CCC)=O)CO)ccc2[nH]cc(C#N)c2c1 c1(OC)cccc(C(c2nnnn2Cc2cccs2)Nc2cccc(F)c2)c1Br c1(C(N(CCCNC(c2cn(C3COC3)nn2)=O)C)=O)ccccc1[N+](=O)[O-] CCCC(C)(CCC)C(=O)NC1CCCC1NC(c1ccc2nc[nH]c2c1F)=O n1(CC)nc(C(=O)NC2CC(C(F)F)C2)cc1C.C(=O)CC.[SH](C)(=O)=O O=C(C1=Cc2ccccc2OC=C1)NC1CC(CNC(C2CC3CC2CO3)=O)C1 c1(C(=O)NCC(CC=C)NC(=O)C(C(C)C)SC)cc(F)c(F)c(N)c1Cl C(=O)(CC(C)C(C)(C)C)N1CCCC(C)C1.C(C(=O)N)SCCN(CC)CC N1(C(C(C)(C)OC)=O)CCC(F)(C(=O)NCCCC(C)(F)F)C1 C1(NC(c2c(C)cc(C)o2)=O)CCC12CN(C(=O)C(C)C1(O)CCC1)C2 C1(C)(C(=O)NCC(C(N2CC(F)C(F)C2)=O)OC)CCCN(C)C1 N1(C(C2CC=C(C)CC2)=O)CCC(F)(F)C(C(=O)N)C1.C(C)C=O.C(C)(C)C S(=O)(=O)(c1ccc(NCC(O)C(C)C)cc1Br)NC(COC)(C)CCO N12CCSCC1CONC2=O.c1(C(=O)OC)nc(C(F)(F)F)c(OC)s1 N1(C(CCc2scc(C)c2)=O)CCC(C)(C(=O)Nc2ccccc2C(C)(C)C)C1 c1(C(=O)NC2CCC(NC(c3c(C)ocn3)=O)CC2)cc(C(C)C)ccc1N CC(C)C(F)C(=O)NCCC1CCCCN1C(c1ccc(CN(C)C)o1)=O N1(C(c2nc(C#C)sc2)=O)CCCC(C)C1CCNC(C1(O)CCC1)=O C1(O)(C(=O)NC2CCN(C(c3cc([N+](=O)[O-])n[nH]3)=O)CC2)CN2CCC1CC2 CC(O)C(C(=O)N1CC=CC1(C)CO)NC(=O)COCCN(C)C CC(C)(C)C(CNC(=O)C(=O)NC1CC1)C(=O)NC1CC12CCCC2 CC1(C)C2CCC(C2)C1C(N1CCN(C(c2nnc(O)cc2O)=O)CC1)=O c1(CC)ccc(NC(=O)C(C2CCCN(C(=O)Cc3cnsc3)C2)(C)C)cc1O c1(C(=O)NC2C(CNC(CCSCC)=O)C2)nccc(Cl)c1O c1(OC)cc(C=CC(N2CCC(C3CC3)C2C)=O)ccc1F.C(=O)CNC=O c1(C(=O)NCC2CCC(C(=O)NC(c3ccccc3O)CC)O2)cc(C)oc1C Cc1csc2ncc(C(N3CC4C(CNC(=O)C5=CCCCCC5)C4C3)=O)n12 c1(CC)c(C(N2CC=CC(NC(=O)CCCCNC(N)=O)C2)=O)cccc1C C1(C(N2CCC3C(NC(c4ccc(OC)cc4)=O)C32)=O)CC(=O)NC(=O)C1 Cc1ncnc(C(=O)NCC2(CNC(=O)Cc3cc[nH]n3)CCOCC2)c1C N1(Cc2c(O)ccc(C)c2)CCC2(CN(C(c3nccc4occc34)=O)C2)C1 c1(C(=O)NCCN2C(C)(C)COCC2)cc2c(nc1O)CCCC2O N1(C(c2c(C(C)C)ocn2)=O)CCCC2(CCCN2C(=O)CC2C=CCCC2)C1 N1(C(C(C(=O)OCC)F)=O)CC(NC(C2CCCC23CCC3)=O)C(C)(C)C1 CC1(C)CC(CC(=O)NCC2CCN(C(=O)CCOCC3CC3)C2)CCO1 c1(C(=O)NC2CCC(C)N(C(c3cnco3)=O)C2)cccc2cc(O)ccc12 C1(C(=O)NC2(CCC)CC2)C2CC3C(C2NC(=O)CC(C)OC)C13 c1(C(=O)NCC2CC3(CN(C(C=CSC)=O)C3)C2)cc2nc(C)cc(C)n2n1 c1(CNC(c2cccc(Br)c2)C#N)nc2ccc(Cl)cc2[nH]1 C(=O)(CS(=O)CCC(F)(F)F)N1CCN(C(CSCCOC)=O)C(C(C)C)C1 N1(C(CCC(=O)NC)=O)CC2CCN(C(C3COCC(C)(C)O3)=O)CC(C2)C1 C1(C(=O)NC2CCC(C)C2)(COC)C=CCC1.C1(C=O)CNC(=O)N1.N N1(C(c2n(CC)ncc2)=O)CC2(CC2)CC1C.c1(C=O)sc(C(C)C)nc1C CC(C)C(C)CCNC(c1cc2n(n1)CCC2)=O.c1(C=O)cnc(C(N)=O)s1 c1(CNC(c2cn(C)c(O)n2)=O)nc2c(s1)CN(C(c1ncncc1Cl)=O)CC2 N1(C(C=CCOC)=O)CCC(O)C(NC(c2ccccc2N2CCCC2)=O)C1 N(C(=NCCC1(CO)CCC1)N(C)Cc1ccc(C)c(C)c1)C(CC)C c1(C(N2CCN(C(C(C)CC(N)=O)=O)C(C)C2)=O)cc2ccnc(Cl)c2[nH]1 CCC(C)CCCCC(=O)NCc1ccc(CNC(=O)C(C#N)C(C)C)cc1 Cc1c(NCC2(CO)CCC2)ncnc1NC1CCC(C(N)=O)C1 C(c1ccc(OC)c(F)c1)=C(C(=O)NCC1N(C(CCCC=C)=O)CCC1)C CCCCC(CN(C(=O)C=CC(C)(C)NC(C1CCN(C)C1=O)=O)C)CC c1(OC)ccc(Cl)c(C(=O)NC2CC2C(=O)Nc2[nH]nc3cnccc23)c1F C(=O)(C(C)(F)C(C)(C)F)N1CC(CC(=O)NC2CCCNC2=O)(OC)C1 c1(CC(=O)CN2CC3(CCCCC3)C2)cc2cc(Cl)ccc2o1 CC(F)(F)CN=c1[nH]c2c(c(=NCC3CCOC4(CCC4)C3)[nH]1)COCC2 C(=O)(C1=CC2CCC=CCCC12)NCCCc1cncc(C(=O)NCC(C)C)c1 CCC(C(=O)NC1(C)CC2CCC1CC2)C(F)(F)F.c1(C=O)cc(C)c(C)[nH]1.N S(=O)(=O)(CCC1CCc2ccccc21)NC(C(=O)O)Cc1ccc2ccccc2c1 C1(C(N2CCC(C)C2)=O)CCCCC1NC(=O)C(N1CCOC1=O)C c1(N(C)CC2CC2(C)C)cnc2c(n1)c(I)cn2C n1(CCC)cc(NC(=O)C(CC2CC2)NC(c2csc(O)n2)=O)cn1 CCC(Cc1ccccc1)C(=O)N1CCCC(CN(C(=O)CCOC)C)C1 c1(C(=O)NC2CC(C)(NC(c3c(NC)cnnc3)=O)C2)ccc2sccc2c1 c1(OC)cc(CNC(C2CSCCN2)=O)ccc1OC(C)C c1(C(N2CC(CNC(C(CC)(C)OC)=O)OCC2)=O)ccc(S(N)(=O)=O)cc1N Cc1noc(C)c1Cc1ccc(CN(C(=O)C(CC2CCC2)N(C)C)C)cc1 c1(CC)cnccc1C(=O)NC1CCOC1C(=O)Nc1cn(C)nc1CC C1(NC(C(CCC)(C)CC)=O)CC2COCC(C1)N2C(c1cnn(C)c1CC)=O C1(C(N2CC(O)CC(NC(CNS(NC)(=O)=O)=O)C2)=O)CCc2nnc(C)n2C1 CC1(C)CC(=O)N(CC(=O)NC2CC3CN(C(c4cc(O)nc(O)c4)=O)CC23)O1 N1(C(CC(CC)C)=O)CCCC(C2CN(C(c3cccc4c3CCCN4)=O)C2)C1 CCCCC(C(=O)NC)NC(C1CCC(NC(=O)CCCn2cccn2)C1)=O c1(C(N(C2CN(C(CNC(CC)=O)=O)CC2F)C)=O)cc(S(N)(=O)=O)cs1 c1(-c2ccc(CN(C)CC3(SC)CCCCC3)s2)ccc(=N)[nH]c1C CC(CC(=O)N1CC(NC(c2ccncc2)=O)CC12CCC2)CC(F)(F)F c1(C(C(=O)NC(C)C)N2CCC2c2ccc(Cl)cc2)cccc(OC(F)F)c1 c1(C(=O)NC(CNC(C2CCCSC2)=O)C2CC2)cc(=O)cc[nH]1 C(c1ccccc1C)=CC(=O)N(CCC(=O)NC(CCC)CCO)CC=C Cc1sc(Br)c(C(=O)NC2CN(C(c3cc[nH]n3)=O)CC2C)c1C N1(Cc2c(F)cnc(Cl)c2)CCC2(CCc3ccccc32)C1 c1(C(=O)NCC2C(NC(Cc3ccc(C)s3)=O)CCC2)ccc(CO)cc1 C=CCC(F)(F)CN(C(=O)C(C)(C)NC(=O)C(=C1CCCCC1)F)C N1(C(C(COC)N(C)C)=O)CCC2CCCC12C(=O)NC.C1CC2(CCC2)CO1 C(=O)(CCCC(CC)NC(=O)C(C)(C)COC)N1C(C=C)CCC1 N1(C(c2cnn(C)n2)=O)CCC2(CCN(C(c3ccc(O)c(Br)c3)=O)C2)C1 c1(-n2c(C)cc(C)n2)n[nH]c(=NC(=O)NCCCN(C2CCCCC2)C)s1 Cc1nnn(NC(=O)C2CN(C(=O)Cc3cnsc3)CC(C)O2)c1C C1(NC(CCCSC)=O)CCN(C(C2CCOC2c2cnn(C)c2)=O)C1C C(=O)(CCC(CF)CF)N1CCC(C#C)(C(=O)NOCCCC=C)C1 N#CCCN=c1[nH]c(=NCc2ccc(N)c(Cl)c2)[nH]c2ccccc12 Cc1ccsc1C(=O)N(C)CCN(C(=O)CCc1cnco1)C(C)C C1(C(N2CCN(C(c3n(COC)ncc3)=O)C(C)C2)=O)CCc2nnnn2C1 C(=O)(C(C)(CNC(c1cnn2c1CCC2)=O)CC)N(CCOC)C C1(NC(CC(C)F)=O)C2CC1N(C(c1ccsc1Br)=O)C2C CC(C)CS(=O)(=O)CC(=O)N1CC2CCCC(NC(c3cc(=N)[nH]n3C)=O)C2C1 c1(C(=O)NC2CC(C(=O)NC(C#C)C(C)(C)C)C2(C)C)c[nH]c(C#N)c1C N(C(=NCCN(C)CC)NC(c1ccccc1)CF)C(C#C)C(C)(C)C c1(C(=O)NC2COCC2C)cncc2c(O)nccc12.C1(C=O)CC1[N+](=O)[O-].N C(=O)(C(C(C)(C)C)N(C)C)NCC(CCCC)NC(C(C)OCC#C)=O C1(NC(C=Cc2c(C)ncs2)=O)CC2CC(NC(C3CC(O)CN3C)=O)CC12 N#CC1(O)CC(C(N2CCOC(CNC(C3CCCSC3)=O)C2)=O)C1 C(=O)(C(C)C(C)NC(=O)CCC1(C)CCCN1C(=O)CC1(C)CC1)OC c1(C(=O)NCC(CC)NC(C2CC2C)=O)ccc(-c2nc(C)no2)cc1 c1(CN2CC3(N(C(CC(=O)OCC)=O)CC3)C2)ccc2nc(OC)sc2c1 N1(C(c2nc(CC)sc2)C(=O)NC2CCCC2)CC(c2ccc(F)cc2)CC1C N1(C(C=CSC)=O)CCCC12CCN(C(C1CCCN1C)=O)C2 c1(C(=O)NNC(=O)C2CCN2)cc(Cl)c2ccccc2c1O CC#CCC(C(=O)NCCCC(O)CO)NC(=O)CC(C)C1CC1 C#CCCC(O)CCNC(C1C=CCN(C(c2nccnc2N)=O)C1)=O c1(NC(C2CCN(c3ncc(F)cn3)CC2O)=O)cc(F)c(F)cc1I C1(C(N2CCC(C)(COC)CC2)=O)CC(O)C(O)CC1C.C(=O)C(C)(C)F c1(CC)nc(C(=O)Nc2ccc(C3(N)CCC3)cc2)c(C)s1 N1(C(C(CC(C)C)F)=O)CC2(CCC(CNC(c3cc(Br)n[nH]3)=O)O2)C1 Cn1cc2c(n1)CCCC2C(=O)NC1COC2(C1)CN(C(C1(C)CC=CC1)=O)C2 N1(C(C(C)OCC2CC2)=O)CC2=C(C1)CN(C(c1ccc(C#N)cn1)=O)C2 N1(C(C23CC(C)(C2)C3)=O)CCC2CCN(C(c3ccc4c(c3)NCC4)=O)C2C1 N1(C(c2n[nH]c(C)c2Cl)=O)Cc2[nH]nc(C(=O)NC(C)CCN3CCCC3)c2C1 C1(Nc2ncnc(C)c2Br)CN(C(C2CCCC2)=O)CCC1(F)F C1(C(N2CCC2C(N)=O)=O)(CC)CCN(C(=O)CCc2cn(C)cn2)CC1 CCC(CC)CCC(=O)NCC1CC1CNC(c1ccnc(F)c1N)=O C1(NC(c2c(C)sc(Br)c2)=O)CN(C(C2COC(=O)C2)=O)CC12CC2 C1(C)CC(F)(F)CN1C(c1cc(C=O)co1)=O.C1(CCC)CC1C(=O)N N1(C(c2c(CC)con2)=O)CCCC2C1CCCN2C(c1ccc(F)c(N)c1)=O C(CCC(C)(C)C(=O)NC1(C)CCCC1(F)F)NC(C(C)CC(F)F)=O c1(NC(COC2CN(C(CCOCCOC)=O)C2)=O)ccc(OC)nc1C Cc1ccc(Br)cc1C(N1CCCC1c1sccc1C)C(=O)NC1CCOC1 c1(C(=O)NCCN(C)C(c2ncccc2F)=O)ccn2c(O)nnc2c1 c1(C(=O)NCCC2(OC)CN(C(=O)C(C)(C)C(C)C)C2)ccc2nccn2c1 C1(OCCOC)CCCN(C(=O)C(c2ccccc2)C)CC1 C1(C2(O)CCOCC2)(C(=O)NCC2CC(=O)N(CC)C2c2ccncc2)CC1 c1(CC)nc(NCC(CCO)CC(C)C)c2ccsc2n1 C1(O)(CNC(C(CNC(=O)C(=CC2CCCC2)C)OC)=O)CCOCC1 C1(NC(C2(OC)CCCC2)=O)CCC2(CC1)CN(c1ncnc3sc(C)nc13)C2 C(=O)(CCCC1CC1)NC(C)CCC1CCCC1.C1(C=O)CC(=C2CCC2)C1 C1(OC)CC(O)(CNC(c2cncn2C)=O)C1(C)C.C(C)(C)C.C=O.C n1(CC)nnnc1C(c1ccc(Br)s1)Nc1ccsc1 c1(C(N2CC3CCC2CN3C(c2cc(Br)no2)=O)=O)cccc2sncc12 N1(C(CCCN(C)C)=O)CC2(CCC(CNC(=O)Cc3ccccc3Cl)O2)C1 C1(NC(c2c(C)nc(Br)s2)=O)CCN(C(c2cnns2)=O)CC1O CC1(C(=O)NCCS(N)(=O)=O)C=CCN1C(=O)CC1COCCOC1 c1(C=O)ccc2c(c1)S(=O)(=O)NC2.N1(C(C(CSC)OC)=O)CCCC(C)C1 C1(C)(C(=O)NC)CCN(C(C(=O)NCc2ccco2)c2cncs2)C1 Cc1cnsc1C(=O)NCC(C)(C1CC1)NC(=O)CCc1cn[nH]c1 c1(CN2CCN(C(=O)NC)CC2)cc(C)c(C)nn1 C1(CNC(C=CC)=O)CC2(CCN(C(C3CCC(=O)N(C)C3)=O)C2)CO1 C1(C(=O)NCC(F)CNC(C2(N3CCCC3)CC2)=O)CCCCC1 N1(C(c2cn(CCC=C)nn2)=O)CC(NC(=O)COC(C)(C)CC)C(O)C1 Cc1cc(N2CCCC23CCN(C(=O)C(C)C(C)C)C3)c(F)cc1[N+](=O)[O-] c1(C(N2CCC3(NC(c4cnc(CC)[nH]4)=O)C(C2)C3)=O)ccc(F)c(F)c1N c1(C(=O)NC2CC(C(C)NC(c3ccc(CC)cn3)=O)C2)cc(C#N)[nH]c1C c1(C(N2CC3C(NC(c4nccc(OC)c4)=O)C3C2)=O)cnc2[nH]ccc2n1 C1(N(C(C(CC)OC)=O)C)CN(C(c2ccncc2N)=O)CC1O C1(CC=C)CCN(C(=O)C)CC1.c1(C=O)ccc(C)s1.C(C=O)OCC=C.N c1(OCCC)ccc(CN2CCSC(CC)C2)cc1-c1nc(=O)n(C)[nH]1 CN=c1cc(C(N2CC3(CC3)CC2CC(=O)NC2CCSC2)=O)cc[nH]1 C(=O)(CC(F)(F)C(C)C)N1C(C)(CNC(C=CC(C)C)=O)CCC1 C1(CC(=O)NC(c2cnn[nH]2)C)CN(C(=O)C=CC(C)(C)C)CCC1C N1(C(C2(C)N(C)CCC2)=O)CCCC(F)(CNC(c2ccc(=O)oc2)=O)C1 c1(CN2CCC(CCc3cnccc3)CC2)ccc(N=c2cc[nH]cc2)cc1 N1(C(Cc2ccc(OCC)cc2)=O)CCCN(C(=O)C(CC)NC(C)=O)C(C)C1 C(=O)(C1=C(Cl)CCC(C)(C)C1)N1CCCC(NC(C)C)C1 Cc1cccc(Cl)c1C(=O)N(C1CCC(NC(C2CC3CC3CC2C)=O)CC1)C C(CCC(C)(C)NC(c1sccc1CN(C)C)=O)NC(C(C)=CC)=O C1(CC)CN(C(c2c(Br)cnn2C)C(=O)NCC2CC2)CCS1 Cc1cc(C)c(C)c(C(=O)N(CC(=O)Nc2ccc(C(N)=O)cc2)C)c1C C1(C)(C(=O)NC(C)CCCNC(C2CC3(CCCC3)C2)=O)Cc2ccccc2C1 C(=O)(C(C(CC)CC)OC)NC1(CNC(C(C)OCC)=O)CC1 N1(C(C=CCCC)=O)CCCN(C(=O)C(C)NS(=O)(=O)CC)C(C)C1 c1(C(=O)NCC2N(C(CNC(C(CC)C)=O)=O)CC2)ccc(Br)c2ccccc12 N1(C(C2N(C(C)=O)CSC2)=O)C2CCC1CN(C(=O)C(C)c1ccsc1)C2 C=CCCCCCCCCC(=O)N1CC(NC(=O)C(C)C2CCCC2)C1 c1(C(=O)NC2C(C(N(CC(CCC)O)C)=O)OCC2)cc(C)cc(O)n1 CCC(C)CCC(=O)N1CCC(C(=O)NC2(c3n[nH]cc3C)CC2)C1 N1(C(c2c(C(C)(C)C)ncs2)=O)CC2(CC(C)C2)C1.C1(C=O)CC2C=CC1O2 C1(C(=O)NC2CC3C(NC(C4(CF)CC(=O)C4)=O)C3C2)CCCCC(=O)N1 C1(CNC(=O)NC(c2ccc(F)cc2)c2ccccc2)CC1C1CCOCC1 Cn1ncc2c1CN(C(C1CC3(CC(NC(c4csnn4)=O)C3)C1)=O)C2 C=CC(C)(C)CC(=O)NCCC(C)NC(=O)COc1cccc(Cl)c1Cl C1(C(=O)NC(CNC(c2nc(C)oc2)=O)(C)CC(C)C)CCC12CCOCC2 C12(NC(C3CCC4(CCC4)O3)=O)CCC(C1)N(C(=O)CCc1ccc[nH]1)C2 c1(C(C)(C)C)nc2c(s1)CCC(NC(=O)CC(O)C(Cl)(Cl)Cl)C2 C1(C(=O)NC(CC)(C)C2CC2)C2CCN(C(=O)C=CC(=O)OCC)CC12 C1(C(C)C)CN(C(C2CCOC(C)C2)=O)CCN1C(=O)CCCCc1cnn[nH]1 N1(C(C2(OC)CCS(=O)(=O)C2)=O)CC2(CCN(C(=O)CC(C)CF)C2)C1 C1(C(C)O)CCN(C(C2(F)CCN(C(=O)Cn3cccn3)C2)=O)CC1 C(C(C(C)C(C)C)NC(=O)CC1(C)CCC1)NC(Cc1cc(C)[nH]n1)=O C1(C(=O)NCCCNC(c2c(C(C)C)c[nH]n2)=O)CC2CC1CC2(F)F C12(C(=O)N)CCC(N=[N+]=[N-])(CC1)C2.C(C(C)CC(=O)NCC1CCC1)OC C(=O)(CCCCCS(N)(=O)=O)NC1CC(NC(c2cc(C)no2)=O)C1 c1(-c2ccc(F)cc2)csc(=NCC(F)(F)Oc2ccccc2)[nH]1 N#CC1(Nc2ncc(I)cn2)CCN(Cc2ccc(Cl)cc2Cl)C1 C1(C(=O)NC2C(NC(c3ncccc3F)=O)CCCCC2)CC2(C1)CC21CCC1 c1(CC(N2CC(NC(c3c(OC)ccnc3)=O)C2)=O)ccc([N+](=O)[O-])cc1 N1(C(CC(CC)C)=O)CCCCC(C2CN(C(c3cc(Cl)ncc3O)=O)C2)C1 CCCCCC(O)CC(=O)NCC1CCN1C(c1ccsc1OCC)=O C12(NC(C(C3CCN(C(c4cc(CO)on4)=O)C3)C)=O)CC3CC(CC1C3)C2 Cc1nc(C=CC(N2CCC(N3CCN(C(=O)CSCC(C)C)CC3)C2)=O)cs1 C(CCN=c1nc(C2CC2)c(F)c[nH]1)OCCNC(=O)CCC1CCCC1 C1(C(=O)Nc2ccc(Oc3nccs3)c(F)c2)CC12CCC(F)(F)CC2 Cc1nc(C(=O)NC2CCC(C(=O)Nc3c(I)cnn3C)C2)ccc1Br c1(NCC2(F)CCN(C(C=CCC)=O)CC2)ncc(C#N)cc1F c1(OC)cccc2c1C(C(=O)N1CCC(N(CCO)C(c3ccsn3)=O)C1)CC2 Cc1ccc(C=CC(=O)NC(C2CCCN2C(c2nncs2)=O)(C)C)cc1 C(C(CC(C)C)C(=O)N)NC(CC1(COC)CC1)=O.C1CC(C(N)=O)=NO1 Cc1nc(C(=O)NC(C2CCCCN2C(=O)CN(C)C2CC2)C)ccc1C#N N1(C(C2C(OC)CCCC2)=O)CC=C(CC(=O)NC(C(F)F)C(C)C)CC1 c1(C(N2C(C(=O)NCCN(C)C)CC2)=O)cccn(C)c1=O CC(CNC(C1(F)CCN(C(=O)C=C2CCCCC2)C1)=O)CC(F)(F)F c1nc2c(s1)CCN(C(=O)C(O)C(F)(F)F)C2.C1(C(C)C)CCOC1C(=O)N.C N1(C(C(=O)NCCOC)=O)CC(CO)C2(C1)CN(C(c1cnccn1)=O)C2 c1(C(=O)NC2CCCN(C(CC=C)=O)C2)cc([N+](=O)[O-])cc(C)c1Cl N1(C(C(CC)F)=O)CCC(OC)C(CC)C1.N(C)(S(=O)(=O)N(C)C)C(=O)C C(C(=O)NC1CCOC1)(C(C)CCc1ccccc1)N(CC(C)SC)C CN1CCOC(C(N2CC3CC3(NC(=O)CCCCC3CC3)C2)=O)C1 Cc1c(C(=O)NCC2CCN(C(C3CC3C3CCCC3)=O)C(C)C2)c[nH]c1C#N C(C)(CC(C)N=c1ccnc(CCc2ccccc2)[nH]1)NC(CN(C)CC)=O C(=O)(C1=CS(=O)(=O)CCC1)NC1CC(CNC(CC(CC)(C)C)=O)C1(C)C c1(CC(N2C3CC(OC3)C2)=O)cn(C)c2ccccc12.C(C(Cl)C(=O)N)OC.C Cc1c(Br)c(C(N2CCC23CN(C(=O)CCc2ccc(F)c(Br)c2)C3)=O)nn1C CN1CCN(C(c2ccc(C(C)(C)C)s2)=O)CC1CNC(=O)C1=CCCO1 C1(CNCCOC2CCN(C(=O)OC(C)(C)C)C2)CCCCC(=O)N1 C1(C(C)NC(C2(CC)CC2)=O)CCN(C(=O)CC2(O)CCOC2)CC1 N1(c2n(CCOC)c(-c3ccccc3)nn2)CCC2(C1)CS(=O)(=O)C2 C1(NC(C2N3CC(C)N(CC3)C2)=O)CC2CCC1CN(C(C1CC=CC1)=O)C2 C1(NC(Cc2ncc(CC)[nH]2)=O)CC(O)CN(C(c2oc(C)cc2C)=O)C1 N1(C(C2CC(C(C)(C)C)C2)=O)CC2C(CNC(=O)C(C3CCCCC3)O)C2C1 C(c1ccc(C)o1)=CC(N1CCC(OCCNC(C=C(CC)C)=O)C1)=O S(=O)(=O)(C1CCN(C(=NCCSC)NCc2ncc(C(C)C)s2)C1)NCC CC(CF)CC(=O)NCC(C)NC(c1ccc(N)cn1)=O Nc1ccc(C(=O)NCCC2CCCN(C(=O)Cn3nnc(=O)[nH]3)C2)cc1Cl CCC(C(=O)NCC12CC(NC(=O)CC3C=CCCC3)(CCO1)C2)C(C)C CC(C)(C)C(O)C(=O)NC1CN(C(c2nc(Cl)cs2)=O)CCC1O c1(CCC)cc(NC(=O)NC2CC(=O)N(C3CCOCC3)C2)ccc1Cl N1(C(C)=O)CCC(NC(=O)C(CNC(=O)C(C2CC2)SC)N(C)C)C1 C(=O)(C1CCCc2nccn21)NC1(CF)CN(C(C(CCC(C)C)F)=O)C1 CC1CCC(=CC(=O)NC2CCC2CNC(c2cn[nH]c2)=O)CC1 CCCC(C(=O)OC)C(=O)N1CCCC1CCCNC(=O)CC1CCCCC1 N1(C(c2cn(CCC)nc2)=O)CCC2C(C1)CN2C(C1C(F)(F)C12CCC2)=O Cc1cc(NC(=O)C(F)(F)Sc2cnn(C)c2)c2ncccc2c1 C=CCC(CC(C)C)C(=O)NC(C(N1CC2(CCN(C)CC2)C1)=O)c1ccoc1 NS(=O)(=O)N1CC(C(=O)NC2CCC2)C1.c1(CCCC(=O)N)ccc(Cl)cc1 c1(OC)cc(C(=O)NC23CC(NCc4cc(Br)co4)(C2)C3)ccc1F C(=O)(C(C)(C)C(C)(F)F)NCCn1ccc(C(N(C2CCN(C)C2=O)C)=O)c1 N1(C(=O)C(F)=CC2CC2)CCCC2(CCCCC2NC(C2(F)CCOC2)=O)C1 C(CCNC(=O)CC(C)(C)N(C(=O)C(O)CN1CCCC1)C)(C(C)C)OC c1(OCC)cc(NC(C2CC(NC(C3(C)CC3)=O)C(O)C2)=O)ccc1C N1(C(CC(COC)C)=O)CCC(C(=O)Nc2cnc(O)c(C)c2)(CC)CC1 CC12COCC1CN(C(=O)CCC1CC(NC(C34COCC3C4)=O)C1)C2 Cc1cc(C(C)C(N2CC(NC(c3cc(C)[nH]n3)=O)CC(F)C2)=O)cc(F)c1 CC(C(C)(C)C#N)NC(c1[nH]ccc1C)=O.C1(CC(=O)N)CCC(C#N)C1 C#CC1(C(N2CCC(SC)C2)=O)CCN(C(c2cncc(OC)c2)=O)C1 N1(C(C(C)(N(C(=O)C2=CCSC2)C)C2CC2)=O)CCOC(C2(C)N=N2)C1 C1(C(N2CCC(OCCF)C2)=O)CC(O)CCN1C(=O)CC1CCOC1 c1(-c2c(F)ccc(C(C)C)c2)cccc2sc(C(N3Cc4c[nH]nc4C3)=O)cc12 CC1COC2(CCC2)CN1C(=O)C(C)(C1CC1)N(C)C(c1sccc1Cl)=O c1(C(=O)NCCC(=O)N(C2CSC2)CC#C)[nH]ccc(=O)c1C N1(C(c2csc(C)c2N)=O)CCC(NC(=O)Cn2nnnc2C(C)C)C(F)C1 c1(NC(C)=O)cc(Cl)ccc1NC(c1cn(Cc2cccc(F)c2)nn1)=O N1(C(C(C)=C(C)C)=O)CCCC(NC(=O)C(c2ccc(Cl)s2)C)CC1 c1ccc([N+](=O)[O-])cc1.CC1=CC1C(=O)N(C)CCOCC.C(=O)(C)N C(c1cccnc1)=C(C(N1CCC(CN(C(C(CC)OC)=O)C)C1)=O)C C1(C=O)CCCC12CC2.c1(C(N(CC)CC)=O)cnn(C(C)(C)C)c1C.CO C1(C)(NC(CSCCCC)=O)CCCN(C(=O)CC2(CSC)CC2)C1 c1(C(N2CC(CCNC(CCOC)=O)(OC)C2)=O)cccnc1-c1cnn(C)c1 C(=O)(CC(C)(C)C(F)(F)F)N1CCC2CN(C(C3C(C)(C)COCC3)=O)CC21 Cc1cc(-c2ccc(NC(=O)C(C)C)cc2)c(Cl)cc1Cl CC(CNC(c1coc(C2CC2)n1)=O)CC(=O)NCC12CC(CN1C)C2 Cc1cnc2n1C(C(=O)N1CC(O)(C3CCCN3C(=O)CNC=O)C1)CCC2 CCC(F)(F)CC(=O)N1CCCCC(NC(c2c(C)nsc2NC)=O)C1 c1(C(=O)NCC(C2CCC2)NC(C2CCCO2)=O)cccc(N(F)C)c1 c1(CNC(C(C)(CO)NC(COC(CC)C)=O)=O)cnc2n1CCC2 c1(-c2ccc(CCCC)s2)cc(C(N2CCC(F)C2)=O)cc2[nH]ncc12 C1(C(=O)NCC(C)(C)NC(CC(CC)C2CC2)=O)COc2c(OC)cccc2C1 c1(C(N(CCC)CCNC(=O)Cn2cc(Cl)cn2)=O)csc(C)c1C C1(COC)CN(C(=O)Cc2cnn(-c3ccccc3)n2)C1.c1(C=O)csnn1.N c1(CCCC)ncc(C(=O)NCC2(NC(=O)C(n3nccc3C)C)CC2)s1 N1(C(c2cc(C)n(CC3CCCO3)c2C)=O)CCCC12CCCOC2 c1(C(=O)NCCC(C)(C)NC(c2ccncc2O)=O)cc(F)ccc1Br N1(C(C2CC(C)NC(=O)C2)=O)CC2CCC1CN2C(c1ccc(C(N)=O)s1)=O c1(NC(C2C(NCc3ccc(CN(C)C)cc3)C2)=O)cccc2c(I)n[nH]c12 C#CC1CCCN1C(c1conc1C(C)NC(=O)C(C)SC(C)C)=O Cc1cc2nc(C(N3CCN(C(c4cn(C(C)C)cn4)=O)CC3)=O)cn2cc1C Clc1cc(CNC2CCNC2)ccc1I Cc1cnc(Cl)[nH]c1=NC(=O)C1CC(F)CN(C(=O)COC2CCC2)C1 C(C(=O)N(CC(=O)NCC(CO)C(C)C)C1CCC1)(C(C)C)OCC c1(CC(=O)NCC2CCCN2C(C2CC3CCCC23)=O)cccc(C(F)F)c1 n1(CC(=O)NCC2OCCN(C(C3C=C(C)CS3)=O)C2)cc(F)ccc1=O c1(OC)cc(C(=O)N(C(C)C)C)cc(N)c1.c1(C(C(=O)N)=O)ccc(Cl)s1 C(=O)(C(CC(C)C)C(C)C)N1CCC(NC(c2c(C)ccnc2C)=O)C1 C12(NC(C=CC(C)(C)C)=O)CCCC1N(C(=O)CCc1cncc(F)c1)CCC2 N(C1CCc2ccccc21)(C(C1C2COCC12)C(=O)NCCOCC)CC=C c1(NC(CONC(C(C)n2ccnn2)=O)=O)ccc(F)c(O)c1 c1(C(=O)NC2(CCNC(C(CC=C)C)=O)CC2)cc(C)cc(Br)c1O C1(CNC(=O)Nc2c(C#C)cc(C(F)(F)F)cc2)CNC(=O)CC12CCC2 C1(C=O)CC2(CCC2)C1.c1(CC)noc(CCCC(=O)NC2CCCC2C)n1.N CN1CCN(C(C2CCCC(=O)C2)=O)C(C(N2CCC(O)(C(F)(F)F)C2)=O)C1 C(=O)(CCC(C)(C)[N+](=O)[O-])N1C(CNC(C=C(CCC)C)=O)C(CC)CC1 c1(OC)ccn2c(C(N3CCC4(CC3)CN(C(c3ccc[nH]3)=O)C4)=O)cnc2c1 N1(C(c2c(C)nc(N(C)C)s2)=O)CC2CCC1C(NC(=O)C1=C(Cl)CC1)C2 c1(CC(=O)NC2CCN(C(Cn3ncc(C)c3)=O)CC2)ccc(C#N)cc1F C1(C(=O)NCc2c(C)noc2)CCOCCN1C(=O)C=CCN1CCC1 c1(NC(C2OCCN(C(c3ccc(C)nc3)=O)C2)=O)ccc(CO)c(C)c1 Cc1cc(C(N2CC3CC2C3CNC(=O)C(F)(F)c2nccs2)=O)c(C)s1 CCC(CC)CCCC(=O)NC1CCCCC1C(N1CC2CCCCC2C1C)=O c1(SC)nccnc1C(=O)NC(C)CNC(c1nccnc1Cl)=O C12(CNC(C(CC)OCC)=O)CCCCC1N(C(=O)CS)CC2.c1cscn1 N1(Cc2c(C)c(F)ccc2)CC2CCN(C(=O)Cc3ccc(F)cc3Cl)C2C1 c1(OC)ccc(C(N2CCC(C(N3CC(O)CC3C(N)=O)=O)C2)=O)c(F)c1F c1(NC(=O)NCc2c(N(C(CC)C)C)cccc2)cc(Br)nc(C)n1 C1(C(=O)NC(c2cnn(C)c2)C)CCN(C(=O)CCC2(C)N=N2)C1 N1(C(C2ON=C(C)C2)=O)CCN(C(=O)CC2CSC2)CC1C CC(C)CC(c1ccccc1)NC(=O)C(=O)NC1CCC(c2ccnn2C)C1 C1(CC(=O)N(CC(Cc2ccc(C(F)(F)F)cc2)CO)C)CCNCC1(C)C N1(C(c2cc(CCC)on2)=O)CCC2(CCCC2CNC(c2cc[nH]n2)=O)CC1 C1(C(=O)NCC2(O)CC(NC(C(C=C)C)=O)C2)CC(C)(C)CO1 CC1(C)CCC(C(=O)NCCC2=CCOCC2)CN1C(=O)CC1CCCC1 c1(C(C(=O)NC2CCOC2)N(CCCO)C2CC2)ccc2c(c1)COC2.CCO Cc1ccc2c(NC(C(C)(C)C)C(F)(F)F)ncnc2c1C C1(CNC(c2nnnn2CC)C2(CC)CC2)CCCCC12CCC2.C1CC1.O C1(C=O)CCS(=O)(=O)C(C)C1.c1(CNC(COCCC)=O)cscn1.C C1(CC)(NC(=O)C=CC2CCOCC2)CCCN(C(=O)C2=NOCC2)C1 Cc1cnc2c(c1)N(C(=O)C(CC(F)F)NC(=O)OC(C)(C)C)CCN2C c1(CCC(=O)NC(CC=C)CNC(=O)Cn2cccn2)ccc(F)nc1 N1(C(=O)C=CC2CCOC2)CCC2CN(C(C3(O)CC(F)(F)C3)=O)CC2CC1 Cc1nc(C(=O)NCc2ccccc2)cc(O)n1.C1(C)(C(NC)=O)CC1(C)C C1(NC(C#CCNC(Cc2c(C)occ2)=O)=O)CCCC(C)CC1 C1(C(N2CC(C(=O)NCC(C)SC)C2)=O)C=CCCC1 O=S1(=O)CCC(N=c2cccc(S(=O)(=O)NC3CN4CCC3CC4)[nH]2)C1 C(=O)(C(C#N)C(C)C)NCCC(C)NC(c1cccc(SCCCC)c1)=O CC1CC(CNC(c2cccnn2)=O)CN1C(c1cnc(C(C)(C)C)[nH]1)=O C1(CC(=O)NCC2(O)CCC(C)C2)CCN(C(=O)CC(=O)N(C)C)C1(C)C C1(C(=O)NCCNC(C(P(C)(C)=O)O)=O)CCc2ccc(F)cc2O1.C1CC1 c1(C(N2C(C(=O)Nc3c(Cl)cccc3Br)CC2)=O)c(Cl)cnc(Cl)c1Cl Cc1ncnc(C)c1CC(=O)NC12CC1CN(C(C1CC(CN(C)C)C1)=O)C2 C=CC1CCN(C(=O)C(CSCC)NC(=O)C(C)(O)C2CCC2)C1 C#Cc1ccnc(C(N2CCC(N(C(=O)C3=C(Cl)CCC3)C)C(C)C2)=O)c1 C=CCC(CNC(=O)C(O)C(C)(C)C)C(=O)NCCC(=O)NCC C12(C(=O)NCC(CNC(C=C(CC)CC)=O)C)CCCN1CCC2 C1(CC(=O)NCCOC2CCN(C(C(C)n3cncn3)=O)C2)CCCCC1(C)C c1(N(CC(O)CC2CCC2)C(c2nc(C)c(C)s2)=O)cccc2c(Br)csc12 C1(CN2CCN(CCNS(N(C)C)(=O)=O)CC2)CCC2(CCC2)CO1 n1(CCNC(c2ccn(CCC(F)(F)F)n2)=O)ncc(Br)n1 c1(OCC(=O)N(CCCNC(C2CC(F)C2)=O)C)ccc(Br)c(Cl)c1 c1(C(=O)OC)ccc(F)c(C(=O)N(C)CC2CC2)c1.C1(C=O)CC1Cl.C C1(CNC(C(CC)CO)=O)CCC2(CN(C(c3ncnn3C)=O)C2)O1 C(=O)(CC(C)C(F)(F)F)NC1C(C(=O)Nc2c(C)nc(Cl)cc2)C2CCC1C2 C1(C(=O)NCC2(C)CCC2)CCC(O)CN1C(c1ccoc1C1CC1)=O CCC(C(=O)OC)C(=O)NC1CCC(NC(c2ccc(-c3cccs3)[nH]2)=O)C1 CCCCCC(O)C(=O)NCC1(NC(c2c[nH]c3cccnc23)=O)CCOCC1 c1(CC(=O)NCC(C2N(C(CC(=C)C)=O)CCC2)(C)C)noc(C)c1C#N N1(C(CC=C(C)C)=O)CC(C)C(C)(CNC(C23CCOC(C)(C2)C3)=O)C1 CCCC(C)(C)CC(=O)NCC(O)C(=O)NCCCC(O)CO C1(NC(C(CSC)C)=O)CCC2CCN(C(c3ccc4ncnn4c3)=O)C1C2 Cc1ccc(C(C)N(C(c2cnc(CC3CC3)[nH]2)C(=O)NC2CCOC2)C)cc1 N1(C(C(CC=CC)NC(c2cc(CC)ccn2)=O)=O)CCC2(CCCOC2)C1 c1(C=O)cc(C2CC2)cc(F)c1.c1(C(N(CCC)CC)=O)cn(C)[nH]c1=N.N N1(C(c2ccc(F)cc2Cl)=O)CCC2(CCN(C(C3(CF)CC(F)(F)C3)=O)C2)C1 c1(C=O)cc2ccc(C)cc2o1.C1(CNC(C(COCC)C)=O)CCCCC1.N C(C(O)CC(=O)NCC(O)CNC(c1cnn(C)c1-n1cccc1)=O)N(C)C c1(CNC(C(COC)(C)O)=O)nnc2n1CCN(C(C1CC(N(C)C)C1)=O)C2 c1(C(=O)NCC#CCNC(CCSCC(C)C)=O)ccn2ccsc12 CC1(C)CC(C)(C(=O)NCC2CC23CC3)CN1C(=O)C=Cc1cscn1 Cc1ccncc1C(=O)NC1(CCC(N2CCC(N(C)C)C2)=O)CCCC1 C(N=c1cc(Cl)nc(C(C)(C)C)[nH]1)C1CN(C(CC(C)(C)OC)=O)CC1(C)C C(=O)(C#CC1CCCCC1)N1CCC(C)(CNC(c2cnc3ccccn23)=O)C1 N1(C(=O)CN2CC3CC3C2)CCC2(CC1)CN(C(C1OCC3CCCC13)=O)C2 c1(C(=O)NCC(CC)NC(=O)CCOC)n[nH]cc1C1CC1.C(C)(=O)N N1(C(C2C(C(C)C)C2)=O)CC(O)CC1C(=O)NCCC(C)N(C)C C1(NC(C=C(CC)CC)=O)CC2COCC(C1)N2C(=O)C#CC(=O)N(C)C N1(C(CCSC)=O)CC(C(=O)NCc2ncc(C)cc2C)CC(C)(C)C1 C1(C(N2CCC(CC=C)(NC(=O)C#CC(C)C)C2)=O)OC(C)(C)OC1(C)C c1(SC)cc(C(=O)NC2COCC2C)ccc1.C1(C=O)(C(C)C)COC1.N c1(C(N2C3CCC(CC3)C2)=O)cc2c(s1)CCC(C)(C)C2.C(C(C)C(=O)N)SC c1(NC(CC)C(C)C)nc2ccccc2nc1N1CCC(N(CC)CC)C1 c1(C(=O)NCC2(C)CCC(NC(=O)CCC3CCCC3)C2)cc2ncccc2[nH]1 Cc1ccc(C(N2CC(C)(C)CC2C)=O)cc1[N+](=O)[O-].c1(C(=O)N)csc(Cl)n1 C1(C=O)CC2(CC2)CO1.C(=O)(CCn1cncn1)NC1(CC(C)(C)C)CC1 N1(C(c2n(C)cc(CO)c2)=O)CCC(NC(C2(C)CC3(CCC3)C2)=O)C(C)C1 C(CC(=O)N(C(CO)C(C)C)C)(CC(C)C)NC(CCCOC)=O C(C)(C)(CC(=O)NC1(CCNC(C2COCCN2C)=O)CC1)SC C(CCN=c1cc(Cl)nc(C2CC2)[nH]1)NC(c1ccc(C(F)F)nc1O)=O C1(C(=O)NCc2ccc(-c3ccc(F)cc3)o2)CCc2nc(O)ccc2C1 Cc1c(C(N2CC(N(C(=O)CCCC3CC3)C)C(F)C2)=O)cnn1C1CCC1 CCCCCC(O)C(=O)NCC1N(C(=O)CNS(=O)(=O)CC)CCCC1(C)C C(=O)(C1CCCc2sccc21)N(CCNC(c1cc(F)c(OC)c(Cl)c1)=O)CC C=CC(CC)CC(=O)NCC(c1ccccc1)NC(=O)CN(C)C(N)=O c1(CC(N2CC(OC)C(CNC(=O)C(C)(C)C)C2)=O)cccc(F)c1O.O CCC(CC)CC(F)C(=O)NC1COCCN(C(c2ncccc2F)=O)C1 C1(NC(C=CC2N(C)CCC2)=O)CC2CC1CN2C(=O)COCC1CC1 CC1CC(NC(C2CCCCC(=O)N2)=O)CN(C(=O)C(=O)N(C)C)C1 c1(C(=O)NC2CCCC(C(N3C4CN(C)C(C4)C3)=O)C2)ccc2c(c1)OCO2 C1(C(C)NC(C2(CCOC)CCC2)=O)CCCCN1C(=O)C(C)=C1CCC1 n1(C(C)(C)C)ncc(C(=O)NC2CCC(NC(C3(O)COC3)=O)C2)c1Br c1(CN2C(C)(C(=O)Nc3ncc(-c4ccccc4)s3)CC2)cncc(Cl)c1 O(NC(=O)C(CC)CCCCC)CC(=O)NC1(C#C)CCCOC1 N1(C(C(c2n(C)ccc2)=O)=O)CCCCC(NC(=O)CSC2CC2)C1 C1(N(C)C)(CNC(C2N(C(CC3CCC(C)O3)=O)CCC2)=O)CCCCC1 C1(C(=O)NCCN(CCC)C(c2cc(Cl)c(Br)[nH]2)=O)CCCCN1N=O N1(C(c2c(C)cc(CNC(C3CC(C)(O)C3)=O)o2)=O)CC(C)(C2CCC2)C1 C1(CCC)CN(C(=O)CC(C)C)CCN1C(=O)Cc1csc(C)c1.[SH](C)(=O)=O C1(CNC(=O)CCc2ccc[nH]2)CCCN1C(C1CC1F)=O c1(OCC)cc(C)c(O)c(C)c1.N1(C(CC2CC2)=O)CC(C=O)CC1(C)C.N c1(CC)cc(OC)ccc1F.c12cn(nn1)CCCC(=O)N1CC(C1)C2 C1(CCC(=O)NC(COC)(C)C)CCCCN(C(=O)C(C)n2cncn2)C1 CC(CC(=O)c1cccs1)NC(=O)NC(Cc1cccs1)CO Cc1c(CC(=O)N)ncn1C.C1CCN(C(=O)CC2CN(C(C)C)C2)C1C(C)C C#CCC(C)(C(=O)N1CCCOC(CC)C1)NC(c1cccc(F)c1C)=O C(=O)(C1=CCCN(C(C2CCN(C)C2=O)=O)C1)NCCOCC(=C)C c1(C2C(C(=O)NCC(CC)NC(c3ncccn3)=O)C2)cccc(F)c1F C1(NC(c2c(C)n(CC(F)F)nc2)=O)CCC(C)N(C(c2nc(Cl)cs2)=O)C1 C(=O)(CS(=O)(=O)CCO)NCCOCCNC(c1c(CC)scn1)=O c1(C=O)cc2c(nn1)CCCC2.C1(NC(c2cc(O)cs2)=O)CC(F)(C)C1.N Cc1ncc(C(=O)NCC2CN(C(c3cnn(C)c3Cl)=O)CC23CC3)cc1C#N c1(C=O)cn(C)nc1C(F)F.C(CNC(=O)CC1CC=CC1)(C)OC.N CC1(NC(=O)CC(C(F)F)n2cccn2)CCCN(C(=O)COC(F)F)C1 CC1CSCC1NC(C1CCC1NC(c1ccoc1C1CC1)=O)=O N1(C(C2C(C(=O)NCC#C)CC2)=O)CCC(C)CC1.C(=O)CC(C)C=C.N N1(C(C(c2scc(C)n2)C)=O)CCC(NC(=O)C=CC=C(Cl)Cl)C(F)(F)CC1 c1(-n2cc(CCC3(O)CN(C(CCSCC)=O)C3)nn2)cccc(F)c1C N1(C(C2C(C#N)C2)=O)CCN(C(c2ccc(F)cc2)=O)CC1CF c1(C(=O)NCCC2CN(C(C3C(CC)OCC3)=O)C2)snc(C)c1N C(CC(C(C)(C)C)NC(=O)C(C)c1ccco1)N(C(Cn1c(C)ccn1)=O)C C1(F)(C(=O)NC(C(C)SC)C)CCCN(C(c2n[nH]c(C)c2O)=O)C1 C(N=c1[nH]c2c(c(=NCCCCC(N)=O)[nH]1)COC2)c1cnc(SC)s1 CC(CCC(C)(C)C)C(=O)NC1(CCCNC(c2ccc(C3CC3)s2)=O)CC1 C1(C(=O)NCCC(C=C)(C)C)CCCCC1(C)NC(c1cccc(O)c1C)=O C(=O)(C(F)(F)C(F)(F)F)N(C)CCOCC.C1(C=O)CC(O)C(F)C1.N CC(C)CCCCCC(=O)NC1CCCCC1CNC(c1cc(C(N)=O)c[nH]1)=O Cc1nn(C)c(C)c1OCC(N1CC(NC(=O)CC2CC2)CC(C)C1)=O CCC(CC)CC(F)C(=O)NCc1n[nH]cc1C(=O)NC1CCOC(C(C)C)C1 CC(O)(C(=O)NCCN(C1CCCCC1)C(C1CC=CCC1)=O)C(F)(F)F c1(C(C(=O)NCC(C(C)C)C)=O)ccc(Cl)cc1O.C(=O)(C(C)n1cncn1)N C1(CC(=O)N(CC(C)O)CCNC(C2CC2C)=O)CCC2(CC1)OCCO2 CC1COCCC1C(N1CC(O)(CNC(=O)COCC2(F)CC2)C1)=O C1(C(N2C3CC(NC(C(C4CC4)OC)=O)(C3)C2)=O)CC2(C)CCC1(C)O2 c1(C(=O)NC(CC)CN(C)C(C2CC3C=CC2C3)=O)ccc(Br)cc1C#N CC1(C(=O)NCc2ccns2)CN(C(c2ccnn2CCF)=O)C1 N1(CC)CCOC(C(=O)NCCNC(C2CC=CCC2C)=O)C1 c1(C(=O)NCC2CCCN(C(C(C(C)C)C)=O)C2)ccc2oc(=N)[nH]c2c1 CC12CCC(C(=O)NCC(CNC(C3CC3F)=O)CO)(CC1)OC2 N1(CC(=O)NC2CCCC2NC(C2(CF)CC(F)(F)C2)=O)CC2CCC1C2 c1(C(=O)NCCN(C(C(C)(C)OC(C)=O)=O)C)c(F)c(F)cc(F)c1F N#Cc1ccc(-c2cn(C3CCC(C(=O)NC4CCCC4CO)CC3)nn2)cc1 C1(C(=O)NCCCC(C)NC(C(c2ccc(C)cc2)O)=O)CC(=O)NC1(C)C n1(CCCC)nc(C(=O)NCCCCCCNC(C2(CCO)CC2)=O)ccc1=O c1(N2CCC(CCOC)(NC(=O)CC)CC2)cc(O)nc(=O)n1C.C(=O)CO.N C(=O)(C(CC)CCOC)N(CC(=O)NC1CN(C(C)C)CC1OC)CC#C CC(C)C(C(=O)N1CCC(O)C1)C(C)C.C(=O)(CN(S(C)(=O)=O)C)NC.C CC1CN(C(=O)CN2OC(C)(C)CC2=O)CCN1C(c1cccnc1N)=O C=CCCCCC(=O)NC1CCN(Cc2cccc(NC(C)=O)c2)C(C)C1 c1(C(=O)N)ccc2sccc2c1.c1(C(N(CCOC)CC)=O)cc(C)c(C)[nH]1 C(=O)C1=CCS(=O)(=O)C1.C(C(C)(C)CC)NC(CCC)=O.C1(C=O)CCCC1 Cc1cc(C(=O)NCc2cc(C(=O)NCC3CCC4CC34)cs2)n(C)n1 c1(N(C)C)ccncc1C(=O)N(C1CCN(C(c2ccc(C(F)(F)F)o2)=O)C1)C O=C1OCc2ccc(C(N3CCOC(C(=O)Nc4ncc(O)cc4Cl)C3)=O)cc21 C1(CNC(C2(F)C(C)OCC2)=O)CC2(CC2)CN1c1ncc(O)cn1 Cc1cccc(NNC(=O)C2CCNC23CCCCC3)n1 C(=O)(C1=NOCC1)NCC1(C(C)(C)O)CN(C(=O)CC(F)F)C1 c1(C(=O)NC)cc(F)c(C(=O)NCC2(C(=O)O)CC2)c(F)c1 N1(C(C2CCCN(C(C)C)C2)=O)CC2CC1CN2CCCCCF c1(OCCC(N2C(CNC(c3c[nH]c(=O)cn3)=O)CC2)=O)ccc(Cl)cc1 C1(NC(C2(CCNC(c3nn(CC)c(C)c3)=O)CCCC2)=O)CCC=CCCC1 CC(C)(C)CC(O)C(=O)N1CC2(C1)SCCC2NC(=O)CO.c1cccc(F)n1 c1(C(=O)N)ccc(N)cc1F.c1(CC(=O)N(C2CCCC2)C)ccn(C(F)F)n1 C(=O)C(F)(F)C(F)F.c1(OC)ccccc1OCCC(=O)N(C(C)C1CC1)C C12(CC)CN(C(=O)CCc3cccnc3Cl)C(C)(C1)C2.C(=O)(CC(C)(C)O)N C(=O)(C1=CCCCCC1)NC1CC(CNC(C=CS(C)(=O)=O)=O)C1 C1(C(N2CCC(CNC(Cc3cccc(C)c3)=O)CC2)=O)CCn2cnnc2C1 CC(CNC(=O)CCC1(O)CCC1)CNC(=O)C.C1(C=O)CCCC1.N c1(CNC(c2ccc(-c3cc(C)c(C#N)nc3)cc2)C)ccc2nc(O)[nH]c2c1 c1(OC)cc(C(=O)NCC(C)N(C(=O)Cn2ccccc2=O)C)c(F)cn1 Cc1cc(C(=O)NCC2CCN2C(=O)CC2COCCO2)nnc1C C1(CC(=O)N(C2CN(C(c3c(C)nco3)=O)CC2O)C)CC2C=CC1CC2.CC c1(C(=O)NCCC(=O)NC2CON(CC)C2=O)cc(C)c(C)cn1 CCC(C)C(CC(=O)N1CCC(CCCO)CC1)NC(=O)C(O)C(C)(C)C N1(C(CCCCCNC(c2cnn(C)c2Cl)=O)=O)CC2(C)CC1CCO2 C#Cc1cc(C(=O)NC2CC3(C2)CC(NC(=O)C(C)C)C3)cc(F)c1.CCC C1(CC(=O)N(C(C)C(C)(C)O)C)CN(C(c2ccc(=N)[nH]c2)=O)CC1C c1(OC)cc(NCCC2CCN(C(=O)CC3CCOCC3OC)C2)nc(OC)n1 c1(OC)cc(Br)cnc1C(=O)NC1(C)CCN(C(C2CCC(C)O2)=O)C1 c1(C(C)=O)cc(C(=O)NCCC(C)(C)C)ccc1C.n1(CC(=O)N)ccsc1=N c1(OC)ccc(C(C)=CC(=O)N(C)CCNC(=O)C(C)n2ccnn2)cc1 Cc1ccc(Cl)cc1-n1nc(-c2nccs2)nc1C1CC1F CC1CC(NC(c2ccnc(-c3cccnc3)n2)=O)CN(C(c2cnsn2)=O)C1 c1(C(=O)NCC2OCCN(C(c3ncc(C)cn3)=O)C2)ccc2nncn2c1 c1(OCC)cc(C(=O)NC2CC(C)C2)oc(=O)c1.C1(C=O)CC1(C)Br.N C1(CCNC(C2CC(C)(CC)C2)=O)CSCCN1C(C1CC(O)(C#N)C1)=O C1(NC(c2cncc(NC)n2)=O)CCCCCC1NC(c1coc(C(C)C)n1)=O C1(O)(CC(=O)N)CCCCCC1.n1(CCCC)ccc(C(=O)NCC(C)(C)C)n1 c1(C(OCC)OCCC(O)C2CC2)cn(CC(=O)NCC)nn1 Cc1ccc(NC(=O)C(C(C)C)NC(C2(C3CCCO3)CC2)=O)c(O)c1 C(=O)(CCC(=O)NC1CC1NC(c1ccc(C(=O)N(C)C)cc1)=O)NC C1(N(C(C2C3COCC23)=O)CC)CCN(C(c2cnc(C)nc2)=O)CC1 C(C1=NOC2(CCC2)C1)NC(c1occc1CNC(c1cncnc1)=O)=O Nc1c(C(N2CCC(NC(=O)Cc3csc(S)n3)C2)=O)cccc1F c1(C(=O)NCC(CN(C(=O)CN2CCCCC2=O)C)O)ccc2cnsc2c1 C1(NC(c2cc(C)on2)=O)CCC2CN(C(c3sc(CO)nc3C)=O)CCC2C1 N1(C(C(CC)n2cncn2)=O)CC(C)CN(C(C2CC(=O)N2)=O)C(C)C1 C1(CNC(C(c2cnccn2)C)=O)CN(C)CCN1C(=O)CN1CCC1 CCC(F)(C=O)C(=O)NCC1CC(F)CN1C(C1CC2(CCC2OC)C1)=O C1(NC(C(CSC)O)=O)CC(NC(=O)C(c2ccc(F)cc2)O)CC1O C#CC1(NC(C2C=CCN2C(=O)CC2CC(C)=NO2)=O)CC(F)(F)C1 C=CCC(CC)C(=O)N.C1(C(N(CCC)CCO)=O)CC(=O)N(CC(F)(F)F)C1 c1(C(=O)OC)cnn2c1CN(C(=O)C(=O)NCC(=C1CCCCC1)F)CC2 C1(C(N(C(C)C2CC2)C)=O)Cc2cc(Cl)ccc2O1.c1(C(=O)N)cnc(N)cn1 c1(CNC(CC)CC(C)CO)sc2ccc(Cl)cc2c1C C(=O)(CCC(=O)OC(C)(C)C)NCCCCN(C)C(c1cncc(CO)c1)=O C(c1cc(F)cc(F)c1)=CC(=O)NCC(CO)NC(C(CCC)C#N)=O C(CCC(=O)N=c1cc2ccccn2[nH]1)C1(CNC(C(CC=C)(C)C)=O)CCC1 c1(C(N(CCC)C)=O)cccc(S(=O)(=O)N(C)C)c1.C1(F)(C=O)CC=CCC1 c1(CC(N2CC(n3cc(CC(C=C)O)nn3)C2)=O)sc(C)nc1C C1(C(=O)NCC(C)NC(C2CCC=CCC2)=O)CN(C)CC(C)O1 c1(C(N2CC3CN(C(c4n(C)ncc4Br)=O)CC32)=O)ccc([N+](=O)[O-])c(Br)c1 N1(C(C2N(C(C)=O)CCOC2)=O)CC(C2(NC(C3CCC(O)C3)=O)CC2)C1 N1(C(COC2CC(NC(c3cc(CCC)[nH]n3)=O)C2)=O)CC2CC2C2CC12 c1(NC(C(=O)NCCC2COCCN2)=O)ccc(Cn2cncn2)cc1 c1(NCCCN(C(=O)NC(C(=O)N(C)CC)C)C)cccn2ncc(Br)c12 C(C#CC(=O)NC(C)CCCNC(C1(CCO)CC1)=O)(OCC)OCC C=Cc1cncc(C(=O)NC(CC(=O)NCCSCCOC)C(F)F)c1 N1(C(=O)OC(C)(C)C)CCC2(C1)CN(S(=O)(=O)CC1CC1)C2 CCCC(CCC)CCCC(=O)N1CCC(N(C(=O)C(C)CCCOC)CC)C1 CCC(C)(C(=O)NC1CC2(C1)CN(C(c1cnoc1-c1cccs1)=O)C2)C(N)=O c1(NC(C2SCCN(C(c3cc(C)nn3C)=O)C2)=O)c([N+](=O)[O-])ccc(Cl)c1C C1(NC(CC2C(C)C2)=O)CCCCC12CCN(C(C1CCSC1)=O)CC2 Cc1ncnc(C(=O)NC(C)CN(C(=O)Cc2cncs2)C)c1C N1(C(CS(=O)(=O)NCC)=O)CCCC(C)C1CCNC(c1cscc1F)=O c1(C(=O)N)cc(N)c(Cl)c(O)c1.Cc1c(CC(=O)NC2CCCC2C)cnn1C C1(NC(Cc2nnc(C)o2)=O)CCCC(NC(=O)CC2(C)CCCO2)C1 N1(C(C2C(C(C)C)CN(C(C3(CO)COC3)=O)C2)=O)CC(C)SC(C)C1 c1(NC)c(C(N2CC(OC)CC(NC(c3ccc(Cl)cc3)=O)C2)=O)cccc1F C(=O)(C#CC1CCCC1)NCC1CC(OC)CN1C(=O)C(C)n1cncn1 CCC(CC(=O)N(CC(O)CNC(c1cc(C)cs1)=O)C)C1CCC1 CN1C(=O)c2ccc(C(N3CCCN(CC(F)F)CC3)=O)cc2S1(=O)=O c1(C(=O)NCC(CCOC)NC(C2CC2(F)F)=O)cc(NC)cc(Cl)c1.C O=C(N=c1cc[nH]c(CCO)c1)C1CN(Cc2ncc(Cl)cc2Cl)CCC1(F)F C1(O)(c2n(CCC)ccn2)CCN(C(c2c(C)cccc2F)=O)CC1 c1(OC)ncc(Cl)c(C(N2CCN(C(=O)CC3CCCS3(=O)=O)C(C)C2)=O)c1Cl N1(c2nnn(C)n2)CC2CC1CCC2NC(c1ccon1)=O c1(C(N(C)CC2CC(F)CN2C(=O)CS)=O)ccc(Cl)nc1N.c1nccn1C N1(C(C2(C(F)(F)F)CC(=C)C2)=O)CCOC(CCCNC(=O)CC=C(Cl)Cl)C1 N1(C(c2cc(CSCC)on2)=O)CCC(C)CC1.c1(C=O)cc(O)nn1C.C C=CCC(C)C(=O)NCC(N1CCN(C(=O)C=C(C)CN2CCOCC2)CC1)=O C1(N(C(c2nc(C)nn2C)=O)C)CN(C(=O)Cc2c(Cl)cnn2C)CC12CC2 Cc1nc2ccc(C(N3CCN(C(=O)CCn4cccc4)C4CC34)=O)cc2s1 C1(NC(C23CCCC2CNC3)=O)CCc2nc(C(F)(F)F)cn2C1 N1(C(CN(CC)CC)=O)CC(C(C)(C)C)CCC1.c1(C=O)cnc(C)cn1.C C(CC(F)F)(C(=O)NC1(CO)CCC1)N(C(Cc1c(C)nsc1)=O)C C1(C(N(CCCNC(c2cnn(CC)n2)=O)CC)=O)ON=C(C)C1C CCS(=O)CC(=O)N1CC(O)CC1Cn1cc(C2CCC(C(=O)NC)CC2)nn1 c1(C(N2CC=C(CNC(c3n(C)cnn3)=O)CC2)=O)ccc(O)c([N+](=O)[O-])c1 Cc1ncnc(C)c1C(N1CC(O)(CNC(c2cscc2C(N)=O)=O)C1)=O Cc1cc(N(C)C)ccc1C(=O)NC12CCC(CC1NC(c1cnco1)=O)C2 N1(C(C2(CC=C)CCC2)=O)CC2CCC1CN2CC(C)C N1(c2c(C#N)cc(C)c(O)n2)CC2CCCC(=O)NC2C1 NS(=O)(=O)c1cncc(C(N2CCOC(CNC(C3OCCO3)=O)C2)=O)c1 N1(C(c2cnn(C(C)C)c2F)C(=O)NC(C(=O)OC)C)CCOCC(O)C1 C1(NC(CCCCC#N)=O)CC2CC1CN(C(c1cn(CC3CC3)nn1)=O)C2 C(=O)CC(F)(F)C(F)F.C(CCS(=O)(=O)NCC(=O)N)OC.C1(C)CCC1 C1(C(N2CC(CNC(C(C3CC3)OC)=O)C2)=O)CCC2(CCOCC2)O1 C1(C(N(CC(CNC(c2c(C)nn[nH]2)=O)O)C)=O)CCN(C2CC2)S1(=O)=O c1(NCc2c(CC)cccc2)ncc(C)cc1S(=O)(=O)N1CCCC(CC)CC1 C1CCCN(CCc2ccc(C)cc2)C1.C1(C2CCCC2)C(=O)N1.CC(=O)NC c1(CNc2nccc(N3CCCC(c4[nH]n(C)c(=N)n4)C3)n2)c(O)ccc(F)c1Br N1(C(c2c(OC)ccc(O)c2)=O)CCC(C2(NC(=O)C(F)n3cccn3)CC2)C1 c1(C(NCC(CNC(C2N(CC)CCC2)=O)(C)C)=O)cccc2c[nH]nc12.C CCCCC(CCCC)C(=O)N1CC(C)(C)CC1C.C(C)(C(C)(C)C)=CC(=O)N c1(C(=O)NCCCCNC(CC2C(C)=NNC2=O)=O)cnn2c1CC(C)CC2 Cc1nc(O)nc(O)c1CC(N1CCC(C(C)NC(=O)CCC2CC2(C)C)C1)=O C1(NC(c2cc(C)sc2C)=O)CC2CCC(C1F)N2C(=O)C(C)CF Cc1c(C=CC(=O)NCC2CCCCC2)cnn1C.C1(C#N)(C=O)CCC1.C C1(C(=O)NCCCN(C(C(Cc2c(C)nc[nH]2)O)=O)CCO)CC12CC(O)C2 C1(C(C)C)CN(C(CC2(C)CC2)C(=O)NC2CC2)CCO1 C1(C(N(CC(F)F)C(C)C)=O)CC2CC1CN(C(C1CC13CCCC3)=O)C2 c1(CNC(CC(=O)NC)(C)C)cc(Br)cc(F)c1OC N1(CC(=O)N)CCS(=O)(=O)CC1.C1(CC)CCCN(CC(=O)N(CCCC)C)C1 C(=O)(C(CC(C)C)c1ccccc1)NC(CCCC)CNC(C1(C(C)=O)CC1)=O N1(C(Cc2nc(C)[nH]n2)=O)CCOCC(C(N2CC(N3CCC3)C2)=O)C1 N1(C(CC(=O)NC)=O)CCCCC1C1CCCN(C(C2CN(C(=O)NC)C2)=O)C1 C#CCCCCCC(=O)NCC1CN(C(c2ccc(OC(F)F)cn2)=O)CCO1 C1(C(=O)NCc2cnc(C)o2)CCC(O)CN1C(C1COCCC1C)=O CCCC(CC(C)C)C(=O)NCC1CC(O)(C)C1.C1(C=O)(C(F)F)CC1.N N1(C(c2n(CCN(C)C)cnc2)=O)CCC2C(C(=O)O)C12 C(C(C(F)(F)F)N1CCN(C(=O)C(C)OC)CC1)NC(c1c(OC)scc1)=O C#Cc1ccc(C(=O)N(C2CC(NC(c3cnccc3Cl)=O)C2)C)c(F)c1 C#CCC(C(=O)NC(C)CF)NC(c1ccc(SC)o1)=O Cc1ccc(SC(C)C(=O)N(C2CN(C(c3c(C)coc3C)=O)CC2O)C)cc1 CS(=O)CCCNC(c1nnnn1CC1CCOCC1)c1cnnn1C1CC1 CCCCC(CC(=O)NC(c1ccnc(C)n1)C)NC(=O)C(C)NC=O c1(NC(C)=O)ccc(N)c(C(N2CCC(C)C2)=O)c1.c1(C(=O)N)c[nH]ccc1=O CC1CC(NC(c2cc(CC3CC3)on2)=O)CCN1C.C1CC(=O)NC(=O)C1 c1(C(N(C2CCN(C(C(C(=C)C)(C)C)=O)CC2)C)=O)cc(F)cc(C)c1C c1(C(=O)NCCOCC2CCCC2)c(F)cc(Cl)cc1F C1(N(C(=O)CCc2ncccn2)CC)CCN(C(c2cscn2)=O)CC1 C1(NC(CCc2scc(C)n2)=O)CC2CC1N(C(=O)CCN1CCC(F)C1)C2 Cc1nc(CCC(=O)NCC2CC(CNC(c3cscn3)=O)CO2)cs1 Cc1cnc(Cl)cc1NC(C1C2CC1N(C(c1cccnn1)=O)C2)=O c1(OCC(=C)C)cc(CN(C2CCN(C)C(C)C2)C=O)ccc1OC c1(C(N2CCCC(CCNC(Cc3scc(C)n3)=O)C2)=O)cc(N)c(N)cc1F c1(CCC(N2C(C3CCN(C(CN(C)C4CC4)=O)C3)CCC2)=O)cccnc1F C=C(C)c1cn(CC(N2CCCC2c2ccc(C(=O)NCC)cc2)=O)nn1 n1(CC(=O)N)nc(C2CC2)n(C)c1=O.CC1OCCC1C(=O)NC1CCCC1 N1(C(=O)C=Cc2ccsc2)CCC(CNC(C2(O)CCSC2)=O)CC1 c1(CC)onc(C(=O)NCC(C)N(C)C(c2cc(C)n(CCO)n2)=O)c1C C1(C)(C(=O)NC2CCN(C(c3ccc(COC)[nH]3)=O)C2)CCC(C)=C(C)C1 c1(CNC(C2N(C(c3c(C)scn3)=O)CCC2)=O)cnn(C)c1C N1(C(c2n(CC)ccn2)=O)CCC(n2cccn2)C1.n1(CC(=O)N)nnc(C)n1 c1(C=O)cnc(C(F)(F)F)c(F)c1.CC(C)CC.C1(CC=O)CCC(=O)N1.N C(CN=C(NCC(C)C)NCC1(CN2CCCC2)CCCC1)c1c(C)nccc1 CS(=O)(=O)c1coc(C(N2CC=CC2CNC(c2nc(Cl)sc2Cl)=O)=O)c1 C1(F)(C(N(CC(C)(O)C2CC2)C)=O)CCN(C(=O)CC2CC(F)(F)C2)C1 N1(C(C(C(C)(C)C)=O)=O)CC(C2CCCN(C(C3(CO)CC3(F)F)=O)C2)C1 C(=O)(CCCCCCCC1CC1)N1C2C(NC(c3cc(C)on3)=O)CC(CC2)C1 c1(C(=O)OC)cnccc1C(=O)NC(C)CCOC.C1(CC=O)CC=CC1 N1(C(c2ccc(SC)s2)=O)CCN(C(=O)C=Cc2ccc(F)cc2)C2CC12 N1(C(C2(F)C(C)OCC2)=O)CC=C(C(=O)N(C)CC2CCCCCC2)C1 c1(N2C(C(=O)NCc3cccnc3Br)CCCC2)ncnc2c1CCCC2 c1(N(C2CCN(C(c3c(OC)nccc3)=O)C2)C)cccc(SC)c1[N+](=O)[O-] c1(OC)ccc(CN2CC(NC(=O)C(C)Cc3ccc(O)cc3)C2)cc1Br C#Cc1ccc(C(=O)NC(c2cccnc2)C(=O)NCCC(C)(C)OC)cc1C N1(C(CC2(OCC)CC2)=O)CCCCC1.C1(C2(C(NC)=O)CC2)CCOC1=O N1(C(c2cncc(C)c2)=O)CCN(C(=O)Cc2ccoc2C)C(c2cn[nH]c2)C1 c1(C(=O)NCCN(C(c2[nH]c3cc(C)sc3c2)=O)C)cc(S(N)(=O)=O)sc1C c1(C(=O)NC2COC3CCCCC23)cc(Br)cc2cccnc12 c1(C(=O)NCC(O)CCNC(C2(O)CCCC2)=O)ccc(C(F)F)cc1Cl Cc1ccc(S(=O)(=O)N2CCC(NC(=O)CCc3ccc(F)nc3)C(F)C2)c(C)c1 CC(C)C(C(=O)N1CCC2CC12C(N1CCCC1)=O)N(C)C.C(=O)(C1CC1)N N1(C(C2(C(C)(C)OC)CC2)=O)CCC2CC2C1.c1(CC(=O)N)ccc(Cl)s1 c1(C(=O)OC)cc(C(=O)NC)cn1C.C1(O)CN(C(=O)Cn2cnnc2)C1.C N1(C(c2c(CC)onc2)=O)CC(NC(=O)CP(C)(C)=O)CC2(CC2)C1 CC1CN(C(=O)CCN2CCC(O)CC2)CCCN1C(=O)CC1OCCCO1 c1(C(=O)NCC(CC)NC(=O)C(C)OC2CCCC2)ccc(OC)c(F)c1 c1(C(N2C(C3(NC(C4C(C)N(C)CC4)=O)CC3)CCC2)=O)ccc(F)c(F)c1N Cc1oc(S(C)(=O)=O)cc1C(=O)NCC(C)N(C(=O)CCCN1CCCCC1)C c1(C(=O)NCCCOC2CCN(C(c3cncnc3)=O)CC2)cccc(Cl)c1F c1(N(C2CCNCC2)C(C(C)OC)=O)ncnc2c(C)cccc12 CC1(C)CN(Cc2ncc3ccccn23)CCC1NC(c1cncc(F)c1)=O C1(C(=O)NCC(CC=C)(C)CO)CCC(C)(C)N(C(=O)C(C)(CSC)CC)C1 Cc1cc(C(F)(F)F)ccc1NC(c1cn(Cc2cnn[nH]2)nn1)C C1(C(=O)NC(C)CC2CC2)CN(C(=O)CN(C)C(N)=O)CCN1C N1(CCC)CCCC(C(N2CCCCC2CCN(C(=O)CC2CC=CC2)C)=O)C1 N1(C(c2scnc2C(F)(F)F)=O)CC2CN(C(C3CCC4CC3CO4)=O)CC2C1 C12(NC(=O)NC(C3(C)OCCO3)C)CCN(CC1)CC2 c1(C(N(CCN(C(c2ccc(CCN(C)C)cc2)=O)C)C)=O)cc(N)cc(O)c1 CC(C(=O)NCCCN(C(C1CCC1c1nc[nH]n1)=O)C1CC1)n1cncn1 Cc1cc(C2CCC2)ncc1C(=O)NC1CCN(C(C2CC3CC2C3)=O)CC1 C=C(C)C(C)(O)C(=O)N(C)CC1CCCN(C(=O)CCC=CC(C)C)C1 Cc1ccc(C(=O)NCC2CN(C(C3CC4CCC3C4)=O)CC2C)c([N+](=O)[O-])c1 CC(C)C(F)C(=O)NCC1CCC(CN(C(=O)CC(C)(C)O)C)CC1 N1(C(CC(C)CN(C)C)=O)CCN(C(c2cc3c(s2)CCSC3)=O)CC(O)C1 C(=O)C(C)(C#N)CC.c1(CC)c(C(=O)NCCCCO)cnn1C(C)(C)C C(CN=c1ccnc(N2CCC(c3ccc(F)cn3)C2)[nH]1)(c1ccccc1)OC c1(C(N(C(CC)CNC(=O)CS(=O)(=O)N(C)C)C)=O)cc([N+](=O)[O-])n[nH]1 N1(c2n(-c3ccc(C)cc3)nnn2)C(C)CC(Cc2sc(Cl)nc2C)CC1C c1(C(=O)NC(CC(C)NC(COc2cc(C)on2)=O)C)ccc2occ(C)c2c1 Cc1nc(CC2CCC(CCNC(C)=O)C2)cs1.C1(C=O)CC(=C2CC2)C1 C(=O)(C1CCCc2ccnn21)NC1(CN(C(=O)Cn2cncn2)C)CC1 C(=O)(CC(C)(C)CC(=O)OC)NC1CC(NC(Cc2cccc(CC)c2C)=O)C1 C(=O)(C(C)(C)C(=O)N)OC.C1(F)CCCC1.c1(C=O)ccc(C(N)=O)nc1 c1(C(=O)NCC2(C)CN(CC(=O)NCc3ccco3)C2)noc2c1CCCC2 CCC(CC(=O)NC1(C2CCCN2C(=O)COc2cccc(Br)c2)CC1)OC CC(C)CC(C(=O)N1CC2(CC2)CC1NC(N)=O)N(C(=O)C(CO)N(C)C)C C1(CCNC(c2n(CCSC)nnn2)(C)CCn2cccn2)NC(=O)NC1=O N1(C(c2ccc(C#N)s2)=O)C2COCC1CC(NC(C1CC(=O)NC(=O)N1)=O)C2 C1(C)(C(=O)NC(C)CCNC(C2(CF)CC2)=O)CCN(C)C1 CC1CN(C(C23CC(CCO2)C3)=O)CCN1C(=O)C(=Cc1c[nH]cn1)F C1(CCNC(C=C2CCC(C)CC2)=O)CCN(C2CCc3ccc(F)cc32)CC1 N1(C(=O)Nc2cnc(C)c(Br)c2)CCC2C(CCN2C)C1 C(CC(C)C(=O)NC1CN(C(=O)C(=O)NCCO)CC1O)OC.CCC(N)=O Cc1cc(C(=O)NCC(C)(C)C)cc(O)c1.C(=O)(CC)N.C1(C=O)CCCO1 c1(C(N2CCN(C(C=C(C)c3cccs3)=O)CC2)=O)ccc(CO)cc1F c1(OC)nc(Cl)ccc1CN1CCC(C(C)C(=O)Nc2ccc(C)cc2Br)CC1 C1(NC(C2(OC)CC2)=O)CS(=O)(=O)CC1.c1(C(=O)N)sc(C#N)cc1Cl c1(C(N2CC(C3(Nc4ncc(C#C)cn4)CC3)C2)=O)cccc2nncn12 CC1=C(C(=O)NCCC2CN(C(c3c[nH]nc3C3CCCO3)=O)CC2C)CCO1 N1(C(C(C(=O)OC)(C)C)=O)CC(NC(=O)CCS(C)=O)C(C2CC2)C1 c1(C(N(C(CC)C(=O)NCCC2CCOCC2)C)=O)cc(F)cc(F)c1 N1(C(c2nccc(OC)c2)=O)CC2(C1)CN(C(=O)CCOCC1CC1)CC2 C#CCC(C)C(=O)NC(c1ccc(C(F)(F)F)cc1)(C)C(=O)NC(C)CC=C N1(C(CN(C(C)=O)C)=O)CCC(C(C)C(=O)NC(c2cncs2)C)CC1 C1(CC(=O)Nc2c(OC)nsc2)CC2(C1)CN(C(C1CC(=O)C1)=O)C2 C(CCCCC(=O)NOCC1(C)CC1)N(C(C(CSC)C)=O)C N1(C(C(CC)CN(C)C)=O)CCCC(C)(C(=O)NC(c2cnc(C)s2)C)C1 c1(N2C(C#N)CN(C(C3CC3(F)F)=O)CC2)ncc2cc(F)cc(Br)c2n1 C1(O)(C(C)NC(=O)CSC(F)F)CN(C(c2cscn2)=O)C1.c1ccccn1 c1(OCC)ccc(=NC(=O)c2n[nH]c3c2CN(Cc2ccccc2OC)C3)[nH]n1 c1(C(N2CCN(C(c3c(C)c[nH]c3)=O)CC2C)=O)ccc2ccccc2c1F c1(OC(C)C)cnc(C(N2CCCCC2C2CC2)=O)cn1.C(=O)(C(C)C(F)F)N c1(C(=O)N)cc(Cl)cc(Cl)c1OC(F)F.C#CCCC(O)C(=O)N1CC(F)(C)C1 C(C)(CO)(C(=O)N1CC2CC2(NC(=O)C(c2ccc(Cl)s2)=O)C1)OC CC1(C(=O)NCCCCCCO)CC(O)CN1C(=O)C=Cc1cnccn1 CC1CCCCC1OCC(N1CC(CN(C)C(c2cc(Cl)ccn2)=O)C1)=O CC(C)C(C(=O)NCC(CO)C1CCC1)NC(C1(C)CCC1)=O C1(NC(c2snnc2C2CC2)=O)C2CN(c3ccnc(NC4CC4)n3)CC12 c1(CC(=O)N)cnn2c1OCCC2.N1(C(C(C)OCC#C)=O)CCC(CC=C)C1 C(=O)(C#CC1CCCCO1)N(CCN(C(c1cc(CC(C)C)[nH]n1)=O)C)C(C)C C(=O)(CCC(=O)NC1CCCC1)NCC(C)(CO)NC(C(C)CC1CC1)=O Cn1ncc(I)c1C(c1nnnn1C1CCCC1)NCC(=O)Nc1ccccn1 c1(OC)ccc2[nH]c(C(N3CCC(F)(C(N)=O)CC3)=O)c(CC(=O)O)c2c1 c1(NCCNC(CC(n2c(C)cc(C)n2)C)=O)nc[nH]c2ncnc1-2 N1(CC(=O)NC(c2nocc2C(=O)NC(CO)C2CC2)C)CCC(F)CC1 c1(C(=O)N)ccc2c(c1C)CCC2.c1(C(C)NC(C(F)OC)=O)ccc(F)cc1 CCCC(CCC)=CC(=O)NCC1(C)CCN(C(=O)CCN2CCCC2=O)C1 c1(C(N2C(CCOC)CN(C(=O)C3=COCC3)CC2)=O)cc(C)cn2ccnc12 C1(C(C)C(=O)NCCc2ccns2)CCCN(C(=O)C(=O)NCC2CC2)C1 C1(NC(C(c2ccc(C)o2)C)=O)CC(F)CN(C(c2ccncn2)=O)C1 C1(C2(C)CC2)(C(=O)NCC(=O)NCC(=O)NCCCCC#C)CC1 C1(C(=O)NCC(C)CN(C(=O)CC(C)N(C)C)C)Cc2n[nH]cc2C(=O)N1 Cc1c(N)ccc(C(=O)NCCCN(C)C(C2CC(O)C(F)C2)=O)c1Cl N1(c2c(C(=O)OC)nccn2)CCCC(CNC(C2(CO)COC2)=O)CC1 CC(O)CCC(=O)OCc1nnc(CCC(N)=O)n1-c1cccc(Cl)c1 Cc1c(C(N2CC(N(C)C(c3cn(C4COC4)nn3)=O)C2)=O)cnn1C(C)C CCC(C)(C)CC(=O)NCCC1CC(C(N2CCC(C)(CCO)C2)=O)C1 N1(C(c2cnn(C3CCS(=O)(=O)C3)c2)C(=O)NC(CC)C)CCC(C)=C(F)C1 c1(CC)cnc(C(=O)N(C2CCC2)C)nc1.c1(CC=O)ccc(C(C)C)cc1.N N#Cc1cncc(CN2CCC2C(=O)Nc2nc3c(s2)CCC3)c1 C=CC(CCC)CC(=O)NC1(CO)CCN(C(=O)Cc2cc(C(F)(F)F)n[nH]2)C1 C1(C(=O)NCC2CCN(C(CC)C)CC2)Cc2ccc(Cl)cc2S1 c1(C(N(C2C3CN(C(=O)CSC(C)(C)C)CC23)C)=O)cnc2n1CCCCC2 C1(C(N2CCCN(C(=O)C=Cc3cncs3)C(CO)C2)=O)CCn2cnnc2C1 C(=O)(C(F)CCC(C)(C)C)N1C(C(=O)NCc2c(OC)n(C)nc2)CCC1 C1(C)(C(C)C)CN(C(C2(N)CCCC3CC23)=O)CCO1 C1(C)(NC(CN(C)C)=O)CCCN(C(=O)CC2C=CCCC2)C1 C=Cc1ccc2c(c1)CN(C(=O)NCCOCC(F)(F)F)C2 c1(C(N2CC(C(C)NC(C3(C4CC4)CCC3)=O)C2)=O)cc2ccccn2n1 N1(C(C2C(C)C2)=O)CCCC(C2CN(C(C3CCCN(C(N)=O)C3)=O)C2)C1 CC(F)(F)C(F)C(=O)N1CC(NC(c2n[nH]cc2Cl)=O)CC1CO C(C(N=[N+]=[N-])C(=O)N)OCC.C1(O)CN(C(c2ncc(C(F)(F)F)s2)=O)C1 C12(C(=O)NCC(C(=O)NC(C#C)C)C)CC(C#N)(C1)C2 Cc1ccsc1C(N1CC(N(c2nnc(-c3ccco3)o2)C)C1)=O O=C(C1SCc2cccnc21)NC1CCC(NC(C2CCCC3(CC3)C2)=O)CC1 c1(C2(C(N(C3(C(=O)OC)CCCC3)C)=O)CC2)cc(C)cc(OC)c1O C=CC(C)(CCOC)C(=O)N1CC2CC1(CNC(c1oncc1CC)=O)C2 c1(C(=O)NC2C3CN(C(C(CC)n4ccnc4)=O)CC32)ccc2[nH]c(=N)oc2c1 N1(C(C2(C)CN(C(c3ccccc3)=O)C2)=O)CCC2(CC1)N=N2 c1(C(=O)OC)cc(C(=O)NCCCCC)ccc1F.C(=O)(C(C)CC1CCC1)N C(=O)(C1c2c[nH]nc2CCC1C)NC1c2cccc(C)c2OCC1 c1(C(=O)NC2C3CC(NC(CS(=O)(=O)NC)=O)CC32)sc2nccn2c1C c1(C(=O)NCC(=O)NCC2CC(C)OCC2)cc2c(s1)CCCC2 N1(C(c2cc(OC)co2)C(=O)NC)CCCN(C(=O)OC(C)(C)C)CC1 c1(-c2cc(C)nnc2)cnc2[nH]c(C(=O)Nc3cnn(C)c3)cc2c1 CCCC(CCC)CC(=O)NCCC1(C)CCCN(c2cc(Cl)nc(SC)n2)C1 N1(C(C(=O)NC(CC)C)C(C)C2CCOCC2)CC(O)CCC1C c1(C(N2CC3C(NC(C4C(=C)CC4)=O)(C3)C2)=O)cc2c(Cl)ccnc2s1 Cc1cc(C(N2CC3CC2CN(C(=O)CC2CCC(C)CO2)C3)=O)c(Cl)cc1F N1(C(C(C(CC)C)OC)=O)CCC2(CC1)CC2NC(=O)Cn1nnnc1C(C)C C(CN=C(NCC(C)OC(C)(C)C)NCc1ccco1)c1cnc(C)s1 N=c1cc(C(=O)NC2CCN(c3ccc(Br)cc3)C2)cc(N)[nH]1 C(=O)(CCC(CF)CF)NCCCN(C(=O)CC1CCC(C)(C)O1)CC C(=O)(CCS(C)(=O)=O)NCC1N(C(CCCCOC)=O)CCC1C N1(C(c2noc(C)c2C)=O)CC(NC(=O)Cc2cccc(Br)c2F)CC(C)C1 C1(C(=O)NCCC(C)NC(c2cc(C)[nH]n2)=O)(OC)CCCC1.c1ccccc1 c1(C(=O)N)ccc2nc(=N)[nH]n2c1.C1(OCC)C(C(=O)NC(C)CC)C1C C1(CC(=O)NC2(C)CC(C(N(CC(Cl)Cl)C)=O)C2)CC2CCC1O2 c1(C=O)cnc2c(c1)CCCC2.CC1CCN(C(=O)CC2CC(C)(C)C2)C1C.N CC1CN(C(=O)COC2CC2)CCCN1C(=O)CCC1CC1 C1(C(N(CC=C)CC2CC2)=O)CCCCCC1.C1(C=O)C=CC1C=O.N C1(CCC(=O)N(C)CC2COCCO2)CCN(C(=O)CC2(O)CCOCC2)CC1 C(=O)(C(F)(F)CC(C)C)N1CCC(NC(Cn2nnc(C)n2)=O)C(CO)C1 c1(CC)nc(C)c(C(=O)NCCN(C(=O)C(C)CC(C)CC)CC)c(C)n1 C1(C(=O)NC(C)CCN(C)C)(NC(Cc2cnc(C)s2)=O)CCCCC1 c1(C(=O)N)nccc2ccsc12.CC(CN(C)C)CCC(=O)NCC1(F)CCC1 CC1CCC(C)(C(N2CCC(CCC(=O)NC3CC4CC4C3)CC2)=O)C1 c1(C(N2CC(C=C)C(NC(C)=O)C2)=O)sc2ccccc2c1CC N=c1[nH]c2ccc(C(=O)NC34CCCN(C(c5cnn[nH]5)=O)C3C4)cc2s1 N1(C(c2cn(CC)nc2)=O)CCC(O)C(N(C(=O)CN(C2CC2)CC)C)C1 c1(C(NOCC(=C)Cl)=O)coc2c1CN(C(C1CC13CC3)=O)C2 C(C1=NOC2CCCC12)NC(C1(C#C)CCN(C(=O)CCC=C=C)C1)=O CCCC(C(=O)N1CC(C(C)NC(c2cnn(C3CCC3)c2C)=O)C1)N(C)C c1(C(N(CC(CC)NC(C2CC(C)CCO2)=O)C)=O)ccc(S(N)(=O)=O)s1 C(=O)(C(O)CC(F)(F)F)N1CCSCC1.c1(OCC(=O)N)cc(F)cc(F)c1.C N1(C(C2(NC(Cc3c(C)ncs3)=O)CCSC2)=O)CC2OCCOC2C1 CCC(C)CCC(=O)NCC(CNC(c1cc(-c2ccccc2)on1)=O)OC Cc1cc(C(=O)NC2COCCN(C(=O)C(c3cccn3C)=O)C2)ncc1CO c1(N2CCSCC(C)C2)ccncc1S(=O)(=O)N1CC(C)(C)C2COCC12 C1(NC(c2cn(CC(C)C)nc2)=O)CCCC(NC(c2sc(F)cc2Cl)=O)C1 c1(C(=O)NC(C(C)NC(c2cnn(C)c2F)=O)CO)ccc(Cl)c(C#N)c1 Cc1ccc(C2CCN(C(c3ocnc3C3CCC3)=O)C2)c(C)c1 CN1C(=O)CCCC1C(=O)NC1CCN(Cc2cn(-c3cccc(Cl)n3)nn2)C1 Cc1cc(C(=O)NC2CCN(C(c3ccn(C)c3)=O)C(C)C2)c(O)c(C)c1 C(C1=CCCN(C(=O)Cn2cnnn2)C1)NC(CC1(N(C)C)CC1)=O CC1CCN(C(=O)CCCC(=O)N(C(C)(C)C)C)CC1NC(c1nncn1C)=O C(c1cn[nH]c1)=C(C)CN1CCC1CC(N1CCC(CC2CC2)C1)=O c1(C(=O)NCCCC(=O)Nc2cccc(C(C)=O)c2)ccc(=O)n(C)c1 c1(C(=O)NCCN(C(C(CC(=C)C)C)=O)CC)ccc2sncc2c1 c1(C(=O)NC(CC)CN(C)C(c2nccn2C)=O)cn(C)nc1C1CC1 Cc1ccc2c(=NC3CCC3C)[nH]c(=NCCCCCCCCC3CC3)[nH]c2c1 C1(F)(C(=O)NC(c2n(CC)ncn2)C)CCN(C(=O)C(F)(F)C(F)F)CC1 C1C(C)CCN(C(c2cc(C(C)=O)cn2C)=O)C1C.C(C)(C(=O)N)NC(CC)=O CCCC(C)(O)C(=O)NCc1nc(C(=O)NC(C2(O)CCCCC2)C)co1 c1(OC)cncc(C(=O)NC(C2(C)CC2)C)c1.C(=O)(CC)N.C1CCOC1 c1(OC)cccc(-c2nc(C(=O)Nc3ccccc3Cl)c(C)s2)c1OC C1(Nc2cccc(CS(C(C)C)(=O)=O)c2)CCCCCC1(F)F N1(CC(=O)N(c2c(C)cno2)c2ccccc2)CCCCC1C Cc1sc(C(=O)NNc2ccccc2)cc1S(N)(=O)=O O=S(=O)(c1c[nH]ccc1=NCCCCC1CC1)NC1CCC2C(CC1)C2(F)F N1(C(c2c(COC)ccs2)=O)CC(NC(c2c[nH]nc2O)=O)C(C2CC2)C1 c1(SC)ccnc(N2CC(CN(C)C(C3CCN3C3CCCC3)=O)C2)n1 c1(C(C(=O)N(CC(CN(C(CCC#C)=O)C)O)C)C)ccccc1C(F)(F)F C(=O)(C#CC(C)(C)O)NCCN(C(C(C(C)C)c1cc(C)no1)=O)CC(C)O c1(C(N2CC(CCNC(=O)COC3CCCCC3)C2)=O)cncnc1O.C1CC1 C1(C(=O)NCC(CC)(F)CC)CCOCCN1C(=O)Cc1cc[nH]n1 n1(CC(N2CCC(C)CC2)=O)cc(S(N)(=O)=O)cn1.CCC(C(=O)NC)SC CC1CN(C(=O)C=CCN(C)C)CC1C.c1(C(=O)N)c[nH]nn1.C1CC1 N1(C(C(C)c2ccsn2)=O)CCC2(CCN(C(c3cnnc(O)c3)=O)CC2)C1 C1(CNC(c2c(C)cno2)=O)(CO)CCCN(C(=O)C(N2CCOCC2)C)C1 C(=O)(CCC(C)(C)O)N1CC(CN(C(C(c2cccc(C)c2)C)=O)C)C1 CC(CC(=O)NC1CCCC1NC(C1CCN(C2COC2)C1)=O)c1ccccc1 N1(C(C(CC)NC(c2nc(O)sc2C)=O)=O)CC2COCC2(CO)C1 C1(CN(C(c2c(OCC)nccc2)=O)C)CN(C(C2CCC2)=O)CC12CC2 c1(C(C(N2C(CN(C(C(C)C3CCC3)=O)C)CCC2)=O)O)ccc(F)cc1 C(=O)C(F)(F)C(C)O.c1(OC)ccncn1.C1(CNC(=O)C)CCCO1.C CC1CCC(NC(=O)C(F)(F)F)CN1C(=O)C(=O)NC1CC12CC(O)C2 c1(C(=O)NC2CN(C(C3Cc4ccccc4S3)=O)C2)cc2c(nn1)CCCC2 C(CCCC(=O)N1CC(OC)CC1CNC(C1CC(c2ccccc2)C1)=O)OC C(=O)(C(O)CC(N)=O)NCC1CC(NC(C(CN2CCN(C)CC2)(C)C)=O)C1 N1(C(C2(C)CCC(=O)N2)=O)CC2CCC1C2NC(=O)Cc1cccc(O)c1 c1(C(N2CC3C(NC(c4cscc4F)=O)(C3)C2)=O)ccc2nnnn2c1 C1(OCCNC(COCCOC)=O)CCN(C(=O)Cc2ccccc2O)CC1 Cc1cn2cccc(C(=O)N(C3CN(C(C4(Cl)CC4(F)F)=O)CC3O)C)c2n1 C1(NC(CNS(NC)(=O)=O)=O)C(C)(C)CC1(C)C.C12(C=O)CSCC1C2.N N1(C(C(C2CCCO2)OC)=O)CCC12CN(C(c1cc(C)cc(O)c1)=O)C2 CC1CCCC(C(N2CC(CCNC(c3csc(O)n3)=O)C2)=O)CC1 N1(C(CC(C=C)C)=O)CCN(C(c2ccc(COC(F)(F)F)cc2)=O)C2CCC12 CCCCCC=CCC(=O)N(C)CCOCCC(=O)Nc1ccsc1C CCCCC(C)C(=O)N1CCN(C(c2occc2C)=O)C(c2ccccc2Cl)C1 CS(=O)(=O)C(CNC(c1cc(CF)on1)=O)CNC(C1COCCO1)=O C(CC(CC)C(=O)N1CCCN(C(=O)CCc2cccc(Cl)c2Cl)CC1)=CC N1(C(C2C(C(C)=O)C2(C)C)=O)CCOC(CCNC(C2CCCCCC2)=O)C1 c1(C(N2CC=CC(NC(c3cn(CC)nn3)=O)C2)=O)ccc2c(c1)COC2(C)C CC(C(=O)NC(C)(CNC(C1CC(F)C1)=O)CO)S(C)(=O)=O Cc1oc(C(=O)NCC2CC(NC(c3ccncc3)=O)C2(C)C)cc1Br C#Cc1ccc(C(=O)NCC2CN(C(c3c(Br)nnn3C)=O)CCC2C)cc1 C(=O)(C#CC1CCCO1)NC1(CC)CCN(C(c2cccc(CO)c2)=O)CC1 C12(C(N(C3CN(C(c4ncncc4F)=O)C3)C)=O)CC3CC(C(=O)N1)C2C3 C1(NC(c2scc(COC)c2)=O)CCCC(C(=O)N)C1.C1(C2CCC2)CC1 C(C(C)(CC(=O)NC1CN(C(c2cc[nH]c2)=O)C1)C(F)(F)F)N(C)C N1(C(C(F)(F)C2(OC)CCC2)=O)CCCC(C2CC2)C1.C1(C(=O)N)CCC=CO1 CC1CN(C(c2scnc2Cl)=O)CCCN1C(c1ccc(OCCF)cn1)=O N1(C(C2C(C)(CC)C2)=O)CCC2(CC1)CC(NC(c1cocn1)=O)C2 c1(C(N)=O)ccc2c(c1)CN(Cc1ccnc(O)c1)C2 Cc1cc(=NCC(F)C2CC3CCC2C3)c([N+](=O)[O-])c(C)[nH]1 c1(CC(N2C3CC(NC(C4CC4F)=O)C2CC3)=O)c(F)cc(F)cc1F CN1CCCCN(C(C2(C)CC(O)CN2C(c2c[nH]c(=N)o2)=O)=O)CC1 CCC(CC)CCC(=O)NC1(COC)CCCN(C(c2ccc(C)s2)=O)C1 CCCCCS(=O)(=O)CC(=O)NC1CC1NC(=O)CC(C)n1cccn1 C(CN=c1[nH]ccnc1C#N)N(C(c1c(C)n(CCO)nc1)=O)CCO C1(C(=O)NCC2(NC(C(C)n3cccc3)=O)CCCCC2)CC2CCC(C1)O2 c1(C(=O)NCC(C2CCC2)NC(CCC(C)OC)=O)cnn2ccncc12 S(=O)(=O)(c1cc(-c2cccc(N)c2)ccc1OC)N1C(CNC)CCC1 Cc1cc(NC(C2COCCN(C(=O)C(C)Sc3nncn3C)C2)=O)ccc1Cl CC(C)S(=O)(=O)CC(=O)N1CC(NC(c2cc3ccccc3[nH]2)=O)C(C)C1 C1(CNC(c2n[nH]c(C)c2C)=O)CCN(c2ncnc(Cl)c2F)C1(C)C c1(OC)cccc2c1OCCC2N=c1[nH]c(N(CC(C)(F)F)C)nc2cc[nH]c12 C1(CNC(CC2OCCC(C)C2)=O)CCCCCN1C(=O)CN1CCCNC1=O C1(NC(CCN(C(C)=O)C)=O)C2CCC1N(C(=O)C(C(C)C)N(C)C)C2 C1(C(=O)NCCC(C)NC(=O)CC2CCSCC2)CCC12CCC2 C1(NC(Cc2c(C)n(C)cn2)=O)CCC(C)N(C(c2cnn(C(F)F)c2)=O)C1 C(=O)(C(C)C(O)CC(C)C)NC1(CC)CCN(C(c2n(CCC)ncc2)=O)CC1 C12(NC(C3C(CC)C3)=O)CCOC(C)(C1)C2.C1(C=O)CC(C)OC1=O.N C1(NC(C(CCC)OC)=O)CN(C(=O)C(=O)NC2CC2)C2(CCOCC2)C1 C(=O)(C(C(C)N(C12CC(C1)C2)C(=O)OC(C)(C)C)C(C)C)OC C(C)(CC(=O)N1CCC(O)C1)(C(F)(F)F)N(C)C.c1(CCC(=O)N)cnc(O)[nH]1 C(=O)(C(CCC)S(N)(=O)=O)N1CC(NC(CCSCCCC)=O)C2C(C1)C2 c1(C(=O)NCC2C(NC(CCCC#C)=O)CCC2)ccc2cccnc2n1 Cc1c(C(N2CCC3C(NC(=O)CC(F)(F)F)C23)=O)[nH]c2c(F)cc(F)cc12 C1(C(N(CCC(O)CO)C)=O)CN(C(c2cnn(C)c2N)=O)CCC1(C)C Cc1csc(Cl)c1C(N1CCC(n2cc(C)nn2)C1)=O.C1(C=O)CCC(=O)O1.N N(C)(C1CCc2c(F)ccc(F)c21)C(C(CC(=C)Cl)N)=O C12CCC(CN(C(=O)C=Cc3nccs3)C1)C2.c1(OC)cc(O)ncc1C=O.N N1(C(C(C2CCOC2)NC(Cn2ccc(C)c2)=O)=O)C2C=CCC1CCC2 c1(C(N2CC(CC=C)(NC(c3ccsn3)=O)C2)=O)cccc(OC)n1 c1(C(N2C(C3CCN(C(C(CC)OC)=O)C3)CCC2)=O)ccc(Cl)nc1OC S(=O)(=O)(CC(c1ccccc1)OC)N(CC=C)CCc1ccco1 C(=O)(C#CC1CCCOC1)NCC1N(C(C(=Cc2ccco2)C)=O)CCC1C C12(NC(=O)CC3CCCCCCC3)CC3CCC(C1C2)N3C(c1cc[nH]n1)=O c1(CC(C(=O)OCCC)F)ccccc1.C(=O)(C)N(CCC)C.C(=O)(CC)O Cc1n[nH]c(C)c1CCNC(c1cscc1)=O.c1(C=O)c[nH]nc1C1CC1.C C(C(=O)N1CCC(N(C(c2ccsc2)=O)C)C1)(C(C)C)NC(C)=O.C1CC1 c1(OC)ccc(C)c(NC(C2C(O)CCN2C(=O)Cc2cccs2)=O)c1 C1(CC=C)(NC(C2CCCC2OC)=O)CCN(C(C2(CC)CC2(F)F)=O)CC1 c1(-c2cc(C(=O)NCC(CNC(C(CSC)C)=O)CO)no2)ccccc1C c1(CC)sc(=N)[nH]c1C(=O)NCC1C=CCC1.c1(CC=O)csc(C)c1 C(CC(F)F)(C(=O)NCc1nocc1C)N(C(C=C(C)c1ccco1)=O)C CC1CN(C(=O)Cc2sc(O)nc2O)CC1(C)CNC(=O)C(C)(C)N(C)C c1(SC)cccc(F)c1C(N1CCC(C)C(C)C1)=O.n1(CC=O)ccsc1=N.N c1(C(=O)N)ccc2oc(O)nc2c1.C(C)(C)(CC(=O)NCC1CCCC1O)SC c1(C(N(CCCNC(=O)C(C)N(C)C)CC)=O)cc(Br)oc1C c1(C=O)cc(F)c(N)c(F)c1.C1(C(=O)NC(C)CCO)CCC2C(C1)C2(F)F.N c1(CC(=O)N(CCC)C(C)C)c(C)noc1C.c1(C=O)[nH]ccc1C=O N1(C(C23OCC(C)(C2)C3)=O)CCCN(CCNC(C2(C)CCC(O)CC2)=O)CC1 N1(C(CCC(=C)Br)=O)C2CCC1CC(CNC(c1cncnc1)=O)C2 Cc1cc(C(N2CCCC(C(=O)NCC3CC(=O)N(C)C3=O)CC2)=O)ccc1O C1(NC(=O)CC2C(NC(=O)Cn3c(O)nnc3O)CC2O)CCC=CCCC1 C(CC(C)C(=O)N1CCCCC1CCNC(=O)COCc1nc[nH]n1)=CC Cc1cc(C=CC(=O)NCCC(C)NC(=O)C(C)N2CCC2)ccc1Br C1(CC(=O)N)CCCC12NC(=O)NC2=O.n1(CC)cc(C(=O)NCCCC)cn1 C1(NC(CCCOCC=C)=O)CN(C(C2CCC2)=O)C(C)(C)C1.C(C)(C)C C1(OC)CN(C(=O)C#CC(C)C)CC1NC(C1(F)CC=CC1)=O C1(N(C)C)C2CN(C(C3CCCN(C(=O)COC4CCCOC4)C3)=O)CC12 C(=O)(C#CC1(C)CCCO1)NCC1CN(C(CCCOC(C)C)=O)CC1O C1(C(N)=O)C2CCC1CN(C(c1cn(CC3CC3)nn1)=O)C2 C12(Cc3sc(C(N(CC(CC)(C)O)C)=O)c(C)n3)CN3C(C1)(C2)C3=O.OC C12(NCC3=NOC(C)C3)CCC1CN(Cc1ccccc1)C2 Cn1ccc(CC(N2CCC(CNC(C3CC(N4CCCC4)C3)=O)C2)=O)n1 C1(C(N(CCC)CC)=O)CCC2CCC1N2C(c1ccc(O)cn1)=O C(=O)(C(O)CNC(C1CCOCC1)=O)NC(c1cnn(C)c1)CC c1(C(N(CCC(NOCC#C)=O)C)=O)nc(C)ccc1F N1(C(c2c(C)cco2)=O)CCN(C)CC1CNC(=O)C(C)(O)c1ccccn1 C1CN(C(=O)Cc2ccc(O)c(Cl)c2)CCN1C.c1(CC)nc[nH]c1C(=O)NC C1(C(N(CCCCNC(=O)CSC(F)(F)F)C)=O)CCc2ccnn2C1 N1(C(C(CC)N(C(=O)CC(C)C(F)F)C)=O)CCN(C)C(=O)C1 CC(CCCCNC(c1ccc(C(C)O)cc1)=O)NC(=O)C(C)(C)C1CCCO1 C1(CNC(c2cc(OC)no2)=O)(NC(c2cn(C)nn2)=O)CCCCC1C C#Cc1cccc(C(=O)Nc2cccc(CNC(C3(SC)CC3)=O)c2)c1 C(C(C)(C)C(=O)NCc1nc(C(=O)N)co1)N(C)C.c1(CCC)ncn(C)n1 c1(OCC)ccc(S(=O)(=O)Nc2ccc(Nc3cnccc3[N+](=O)[O-])cc2)cc1 c1(C(=O)NC23CC(c4ccccc4)(C2)C3)ccc2c(c1)C1CCC2O1 N1(C(c2c(CC)nc(C)[nH]2)=O)C2CCC1CC(NC(C1CCCC13CCC3)=O)C2 Cc1coc(C)c1C=CC(=O)N.C(CCC)N(CCC)C.O(C(F)(F)F)CC=O N1(C(c2c(CC)cco2)=O)CCOCC1C(=O)NCC(O)CC(C)C CN1CCC(C)(C(=O)NCCC2CCN(C(C3CCC(=O)NC3)=O)C2)CC1 C1(CC(=O)OCC)CCN(C(C2(C)CN(C(c3cnccc3C)=O)C2)=O)CC1 C1C(C2CC2)CCN1C(=O)CN1CCOC1=O.Cc1nc(C)n(CC(=O)NC)n1 Cc1cc([N+](=O)[O-])cnc1C(N1CC2(CCN(C(=O)CCOCC(F)F)C2)C1)=O c1(C(=O)NCc2occc2C(N2CCOC3(CC3)C2)=O)cc2ccccc2o1 C(=O)(CCCCCCCCCO)N(C1CCC(NC(CC(C=C)C)=O)CC1)C C(=O)(CCCCC(=O)NC(CC(=O)NC1(CF)CCC1)C(C)(C)C)OC C12(C(=O)NC(C3OCCN(C(Cn4c(C)ccn4)=O)C3)C)COC(CCO1)C2 N1(C(C2N(N=O)CCC2)=O)CC2CN(C(C3CCCCO3)=O)CC(C1)O2 N1(C(C2CC(SC)C2)=O)CC2(CC)CC1(C)C2.c1(C(=O)N)cnn2c1CCC2 C1(N(C(C(C)NC(C)=O)=O)C)CCN(C(C2CCCC2)=O)CC1.c1ccncc1 C1(CNC(C2CC(C)C(C)CC2)=O)CC2CCC(C1)N2C(=O)C(C)S(N)(=O)=O C(CCC(=O)NC(CC1CCCC1)C(=O)NC(c1ncnn1C)CC)OCC=C C(=O)(C1=CCN(C(C2C(C)(C)C2(F)F)=O)CC1)Nc1c(C)cc(O)nc1 c1(CCC(=O)NC(C2CCCN(C(=O)CC3CC(F)(F)C3)C2)C)cncnc1O Cc1ccc(C=O)cc1.c1(C=O)coc(C)c1.C(C)(C)C.C1(C(=O)N)CC1 c1(C(=O)NCCC)ccc2c(c1)NC(=O)C2(C)C.c1(C=O)cc([N+](=O)[O-])n[nH]1 C1(CC)CN(C(c2c[nH]c(Br)c2)=O)CCC1NC(=O)C(c1ccccc1)O C1(CC)(CC)CCCN1C(=O)CC1=CCCC1.n1(CC=O)cc(C2CC2)nn1.N C1C2CS(=O)(=O)CC12.c1(CC(C)C)cc(C=O)no1.CCNC.C1CC1 c1(C(=O)NC2CCC(NC(c3ccc(CC)cc3)=O)C2)ccc2c(c1)CCNC2 N1(C(Cc2cn(CC)nn2)=O)CCCCC1C(=O)NCc1cccnc1Cl c1(CNC2C(CN(C)C)COC2)cnc(C2CC3(CC3)C2)nc1 c1(C(N2CCN(C(c3cc(OC)ncc3)=O)C(CO)C2)=O)c(C)ccc(Cl)c1O C(c1ccc(=N)[nH]c1)=CC(=O)N(C(C)C)C.C1(C=O)CC(C(F)(F)F)C1.N C1(NC(c2cc(C3CC3)[nH]n2)=O)CCC(NC(C2CC3CCC2O3)=O)CC1 n1(C(CC)C)nnnc1C(c1csnc1C)NCc1cnc(C(F)(F)F)s1 c1(C(=O)NCC2N(C(C(C)C)=O)CCCCC2)cc(Br)c2c(c1)CCO2 c1(CC)cncc(C(=O)NC2CCC(CCNC(=O)Cc3cn[nH]c3)C2)c1 C(=O)(C(F)(F)C(O)C1CC1)NCC(C1CCC1)NC(C#CC(C)C)=O Cc1cc(C(N2CCC(C)C(C(N)=O)C2)C(=O)NCc2ccco2)c(O)c(Br)c1 C#CCCCCCC(=O)NCC1CN(C(c2ccn(C)n2)=O)CC1C(F)(F)F c1(CC(=O)NC2CCCN(Cc3c(C)cc(C)[nH]3)C2)cccc2[nH]ccc12 CC1(C)COC1C(=O)NC1CC(CNC(c2nccs2)=O)C1 CC1CC(NC(=O)C(Cc2ccoc2)NC(C2CC23CC3)=O)C(=O)O1 C1(NC(c2cnco2)=O)CCCCC1C(=O)Nc1ccccc1O C1(NC(CCSCC(=O)OC)=O)CCN(C(=O)C(C2CCOC2)OC)CC1 c1(OC)cc(C(N2CCC(C)C2CNC(=O)CC)=O)nn1C.c1ccccn1.O N1(C(C(Cc2cc[nH]n2)NC(C2NC(=O)OC2)=O)=O)CCC12CC(CO)C2 c1(Nc2nc(NC(COC)=O)c(C)cc2C)cc2c(cc1Cl)OCCCO2 C1(C(N2C(CC)C(O)CC2)=O)N(C(C2CC2(Cl)Cl)=O)CC12CCCC2 c1(CCC(=O)NC2CCCN(C(C(C)OCC)=O)CC2)cnc2ccccn12 n1(C(C(=O)OCC)C)cc(C2(NC(=O)Cn3cc(I)nn3)CCC2)nn1 c1(C(C)C)nc(NCc2ccoc2)cc(N(CCCc2c(Cl)cccc2Cl)C)n1 O=C1C(O)CN1.C(=O)(C(O)C1CNC1)NC1CC1 N1(C(c2c(CC)ccs2)=O)CC2CCOCC2(NC(c2cc(C)cc(Cl)c2)=O)C1 C#CC1(O)CCN(C(=O)C(CCC=C)NC(c2cc(Cl)cs2)=O)CC1 CC1(C#CC(=O)N2CC(NC(C3CCCN3c3ccncn3)=O)C(O)C2)COC1 C1(CNC(CSCC=C)=O)CN(C(=O)C)C2CCN1C2.c1c(C)n[nH]c1C.S C1(CC(=O)NC(C=CC(=O)NC(CSC)(C)CO)C)CC(=O)NC1=O c1(CC)ccc(CCC(N2CCSCC2CCNC(C2CC2(Cl)Cl)=O)=O)cc1 N(C(=NCCN1CCOCC1)N(C)Cc1ccc(Cl)c(Cl)c1)CC(C)F CCC(C(=O)NCCCCn1cc(CCC2CCCC2)nn1)C(C)(C)CC C(CC(=O)NC)(C1=CCCC1)OCC.c1(C(N2CC(F)C2)=O)cccc(N)c1 C(=O)(C(CC=C)C(C)C)NC1(CC=C)CN(C(c2cccc(O)c2C)=O)C1 CC(C)C(CNC(=O)C(F)C1CCCC1)NC(c1c[nH]c(=N)s1)=O C(=O)(CCC(=O)NCC1CN(C(C2(SC)CC(O)C2)=O)CC1C)OC c1(CC)ccc(C(=O)NCCC2CCCC2)nc1.C1(C=O)CC1(C)C(C)C.N C1(NC(C2C(OC)CCC2)=O)CC2CC(NC(c3cc(F)cnc3O)=O)C2C1 C1(C)(C(=O)NCCN(CC(C)O)C(=O)Cc2ccsc2)CCCNC1=O N1(C(Cc2ncc(C)s2)=O)CCC(C2CCCN(C(=O)Cc3cccs3)C2)C1 CCCC(CC)CC(=O)NCC12CCC(C1)N(C(=O)CCCC(C)C)C2 Cc1ccc2c(c1)C=C(C(=O)NC(C)CN(C(=O)CCC1CC1(F)F)C)CO2 c1(C(N(C(c2cncc(O)c2)=O)CC)C)ccc(F)cc1 N#Cc1ccc(NC(=S)NNC(=O)c2sc(Cl)cc2Br)cc1 Cc1cc(C(=O)N(C)CC2(O)CN(C(c3nscc3C)=O)C2)ncn1 c1(OC)ccc(CC)c(NC(C2CC2)=O)c1.c1(CC(=O)N)ccc(F)cn1 C1(NC(c2c(C)ncs2)=O)CN(C(=O)COC2CCCC2)Cc2nccn2C1 c1(C2C(C(=O)NCC(C3CC3)NC(CCc3cn(C)nn3)=O)C2)ccncc1F c1(C(C)C(=O)NC2CC2NC(=O)C)ccc(F)cc1.c1(C(=O)N)cccs1 C(=O)(CC(F)(F)CS(C)(=O)=O)N(C1CCN(C(=O)C(F)(F)CO)C1)CC CCCN=C(NCC(C)(C)C)NC1CC(C(C)(C)C)C1.C(CC)N(C)CC N1(C(c2c(C)cc(F)s2)=O)CCC2C(C1)NC(=O)CN2C(=O)CNC=O N(C(=NCCN1CCCC1)NCCN1CCC1)Cc1n(C)ncn1 Cc1nnc2n1CC(C(=O)NC1CCCCC1)C2.C1(CC(=O)N)(N(C)C)COC1 CN1CCN(C(=O)C=Cc2cn(C)cn2)CC1.C1(C(C)(C)C)(C=O)CCC1.C c1(OC)cncc(C(=O)NC2CC3CC(NC(=O)Cn4nnnc4C)C2C3)c1C CC(C)CCC(=O)C(=O)N1CC(F)(F)CC1CNC(c1ncoc1C(C)C)=O C(C(C)(C)CCNC(c1ccsc1Br)=O)NC(CC1CCC(C)C1)=O S(=O)(=O)(C=Cc1ccccc1)N1CC2(C(C(=O)NC(c3ccccc3)CO)C2)C1 c1(C(=O)NC(CC=C)CNC(=O)C(=O)NC2CC2)ccc2c(c1)COCC2 CCC(C)(COC)C(=O)N1CC(NC(c2nnsc2C(F)F)=O)C(F)C1 N1(C(=O)NCCCCCCCC)CC2OCC(C(N3CC4(CCOC4)C3)=O)C2C1 Cc1cnc(C(=O)NC2CC(NC(=O)CC(c3c(C)noc3C)C)C2)cn1 Cc1[nH]c(C)c(C(N2CCOC(C(C)NC(c3ccnc(Cl)c3N)=O)C2)=O)c1C c1(N2CCC(C(N(C3CCCC3)Cc3cc(C)no3)=O)CC2)cncc2nnnn12 c1(C(=O)NCCCN(C(=O)Cn2cnccc2=O)C)cc2c(cn1)COCC2 c1(OCC)ccc(CN2CCCC(C)(C(N3CCC(OC)CC3)=O)C2)c(O)c1 c1(N2CC(C(C)C)OCC2)ncnc2sc3ccccc3c12 C=CCC(CNC(c1cc[nH]n1)=O)C(=O)N(C)Cc1cnc[nH]1 CS(=O)(=NC(=O)c1cc(Cl)c2n[nH]cc2c1)C1CNC1 CCC(CNC(=O)CN1CCOCC1)(CC)NC(=O)CC(C)(O)c1ccccc1 c1(CN2CC(n3ccc(I)n3)(CC(=O)OC)C2)cn(C)nn1 N1(C2CCC(CC)C2)Cc2nccn2CC(NCc2nnc(C)s2)C1 O=C(NNC(=O)C1(c2ccc(O)nc2)CCC1)C1CCOC1c1ccccc1 c1(CC)nc(C)n(C)c1C(N1CCCC(NC(c2cc(OC)ccn2)=O)CC1)=O c1(C(=O)NC(CNC(c2cc(C(C)=O)c(C)nc2)=O)C)cnn2c1OCCCC2 c1(C(=O)NC(CN(C(CCC(CC)CC)=O)CC)C)cnn(C)c1S(C)(=O)=O C1(C(=O)NCCC(C)NC(N)=O)CCCN1C(c1cc(CF)on1)=O Cc1nc2c(o1)CCN(C(=O)C(F)C(C)CNC(c1cc(C)n(C)c1C)=O)C2 c1(C(=O)NC23CN(C(c4cnc(C(C)O)s4)=O)C(CC2)C3)onc2ccccc12 C(=O)(CC(C)C(F)F)N1C(CNC(Cc2cc(C)on2)=O)CC1 C=C=CC(C)C(=O)NC(CCN(C)C(C1CCCC1)=O)c1cccs1 c1(C(N2CCC(NC(c3cnc(SC)s3)=O)C2)=O)cnccc1C(F)F N(C)(S(N)(=O)=O)CC(N1CC(CC(C)NC(C2CC3CC3C2)=O)C1)=O N1(C(C(C(C)(F)F)(C)C)=O)CC(NC(=O)CCN2CCOCC2)C2CCCCC12 N1(C(CCNC(COC)=O)=O)CCN(C(=O)CCCn2cccn2)C(CO)C1 c1(C=O)c(C)nn(C)c1C.c1(C(=O)OC)cnc(C=O)cn1.C(CC)C(C)C.N c1(SCCC(=O)Oc2c(C)csc2C)ccc2c(c1)OCCO2 c1(C(=O)NCCCN(C(CSCCOC)=O)C)nn(C)c2ccc(F)cc12 Cc1ncncc1C(=O)NCCC(N1CCOCC1)C CN1CCOC(C(=O)NCC2CCCN2C(c2ccc(-c3cc[nH]n3)s2)=O)C1=O C1(CC(=O)N(C(c2ccc(Cl)cc2)CO)C)COc2ccccc2C1 c1(N2CCCC(n3nccc3)C2)nc(=NC2CCCCC2)[nH]c2cc[nH]c12 C(=O)(CC(F)(F)Cl)N(C(CC)CNC(=O)C(N1CCCCC1)C)C n1(C(CC)C)cc([N+](=O)[O-])c(C2=CCC3(C2)NC(=O)NC3=O)c1 C1(C(C)C(=O)NCc2ccccc2)CCCN(C(c2nc(=N)cc[nH]2)=O)C1 c1(C(N2C(C)(CC(N3C(C(=O)OC)CC3)=O)CC2)=O)cnccc1C#N c1(SC)cc(C(=O)N(CCCCN(C(=O)CN2C(C)CCC2C)C)C)ccc1F c1(-c2cn(CC3CCN(C(C)C)C3)nn2)ccc(C(C)(C)C)cc1 CCCCC(C(=O)NC1CC(=O)N(C)C1=O)NC(c1cncc(C#N)c1)=O N(C1c2ccccc2CC1F)C(c1cc[n+]([O-])cc1)=O c1nccc(C(F)(F)F)n1.C1(C(N(C2(C#N)CCNC2)C(C)C)=O)CCOCC1 N1(CCC(=O)NC2(CF)CN(C(C(CSC)OC)=O)C2)CCOCC1=O CC1CN(C(=O)CCCNC(N)=O)CCC1N(C(=O)CC1CN2CCN1CC2)C C1(C(=O)NC2C(SC)CCC2)COCCC1NC(C1(O)CC1)=O c1(C(N2CCC(CCNC(C3CC(C)C3)=O)C2)=O)ccc([N+](=O)[O-])c(N)n1 N1(CCC)C(=O)CCC(C(=O)OCCC2CCCN2)C1c1cncn1C CCC(C)(CC)C(=O)NCC(C1CC1)N(C(=O)CCCCCOC)C Cc1cc(C(=O)N)cnn1.C1(C(N)=O)CN(C(c2cc(C(F)(F)F)c[nH]2)=O)C1 c1(C(=O)NC(CCNC(Cc2nc(CC)sc2)=O)(C)C)cn(C)nc1OC O=C(CC1=CCCCC1)NC1COCCN(C(=O)COCC2CCCO2)C1 c1(C(C(N2CC(C)(NC(=O)CCc3cnco3)C2)=O)O)ccc(F)c(Cl)c1 C#CCCCC(=O)NCC1CN(C(C2CCC2c2ccc(F)cc2)=O)CC1C c1(OC)cc(C(C)=O)ccc1NCC(=O)NC1CC(NC(=O)CCF)C1 [N-]=[N+]=Nc1cccc(C(N2CC(CNC(=O)CCOC)C2)=O)c1.C1CCCO1 Cn1nc(C2CCC2)cc1C(=O)NCCOC1CCN(C(c2ccccc2)=O)C1 N1(C(CC(CCCCC)O)=O)CC2(C1)OC1(C)CC2(NC(c2ccsc2C)=O)C1 C1(C(N2CCC(C)(CCC)C2)=O)COCCN(C(c2cc[nH]c(=N)n2)=O)C1 N1(C(CC(CNC(CCCC2C(C)C2)=O)O)=O)CCCCC2(CCC2)C1 C1(NC(c2ccsc2)=O)CC1C1CCN(C(=O)C2=C(Cl)CCC2)CC1 N1(C(c2c(OC)ccc(C)c2)=O)CCN(C(C2CCCC(O)C2)=O)CC12CCC2 CCCC(O)C(=O)N1CCC1C(=O)NC1CC2(CC2)C1 C1(NC(C(c2cn(C)nc2)O)=O)COc2ccccc2N(C)C1=O C(CC(C)C)(C(=O)NC(C(=O)NC)C1CCC1)ONC(COCCOC)=O C1(COC)(C)CCCN1C(=O)CC1CC1.c1(C=O)cccc(C(F)F)n1 CC1CCC(C)(C)CN1C(C12CCC(CN(C(=O)C(C)(C)CC(F)F)C1)C2)=O C1(NC(C=C(C)C)=O)CC2CCC(C1F)N2C(=O)CCCc1ccc(O)c(F)c1 c1(C(=O)N)ccc(C)c(Cl)c1.C1(CNC(C(C2CCC2)OC)=O)CCCCO1 C12(C(N(C(CCO)C(=O)NC3CNC(=O)C3)C)=O)CCC(CC1F)C2.CCO CC(C)C(C(=O)NC1CC(C)N(C(c2cccc(O)c2)=O)C1)N1CCCCC1 c1(CN(C)C)ccsc1C(=O)NC1CCC(C)C1.c1(CC(=O)N)cnoc1 C1(NC(c2c(C)cnnc2)=O)CCCC(C(=O)NCC2C3CCCOC23)CC1 CCC(CC)C(C)C(=O)NCC1CC(F)CN1C(=O)CC1CCCNC1=O C#CCC(CC(=O)NOCCO)NC(C1CC(C)(C)CO1)=O C(=O)(C=C=C(C)C)NCC1(C(N2CCC(C(CC)CC)C2)=O)CC(=C)C1 N1(C(c2nn(C)c(Cl)c2Cl)=O)CCN(C(c2ccc(=O)n(C)n2)=O)CC12CCC2 c1(CCC=O)ccc(F)c(F)c1.Cc1nc(C)c(C(=O)NC2CC23CCC3)o1.N C1(C(=O)NC(CNC(CCC(c2cc(OC)ncc2)=O)=O)C)CCCCC1(F)F c1(OC)ccc(F)cc1C(=O)N(C)CCC1CCCCN1C(c1cnsc1)=O c1(C(C)NC(C(C(C)C)C(=O)OC(C)(C)C)=O)cccc2ccccc12 C(=O)(CCCC(=O)NC(Cn1ccnn1)C(=O)NC1CC12CCCC2)N(C)C C1CCC(C)CN1C(=O)CCc1ncc[nH]1.C12(COC)COC(C=O)(C1)C2.N c1(C(N(C2CN(C(C34CCC3C4)=O)C2)C)=O)ccc(C#Cc2ccccc2)cc1 c1(C(=O)NC2C(NC(CCCOC(C)(C)C)=O)CC2)cc2cnc(Cl)cc2s1 C1(NC(C2CCC(CNC(C3CN(C(C)C)C3)=O)O2)=O)CN(C)CC12CC2 N1(C(CC2CN(C(C=CC(CC)C)=O)CC23CC3)=O)CC(C)c2ncccc21 Cc1cc(Cl)cc(C(=O)NCC2CC2NC(=O)C(O)c2ccsc2)c1O c1(OC)cc(OC)cc(CC(N2CCOCC(NC(=O)CCC(C)(C)C)C2)=O)c1 C1(NC(Cc2cn(CC)nc2)=O)CCN(C(=O)C2=COCCO2)CC1F N1(C(CCC)=O)CCC2(CC1)CC2C(=O)NC1CC2OCCC12 N1(C(CN2C(=O)CN(C)C2=O)=O)CCC(C)(C)C(C)C1.c1(CC=O)ccno1.N C1(N(C(C=C=C(C)C)=O)C)CCCC2CN(C(c3ccc(C)c(O)n3)=O)CC12 N1(C(=O)OC)CC2CCC1C(C(N1CC(CCNC(=O)CCOC)C1)=O)C2 CC1CCc2n[nH]cc2C1C(=O)NCC1(C)CC1.C(c1ccnn1C)=CC(=O)N c1(C(=O)NCC(C)CNC(C2CCNC2=O)=O)ccc(Cl)c2ncccc12 c1(CCC(=O)NC2(C)CN(C(C3CC(C)(F)C3)=O)C2)ccccc1F Cc1ccc(C(N)=O)cc1C(N1CCN(C(c2cnccc2Cl)=O)C(CF)C1)=O Cn1cnc2c1CN(C(=O)CC1CC3(C1)CN(C(c1ccon1)=O)C3)CC2 C=CC1(C(=O)NC(C)C(C)NC(=O)Cc2ccc(CCCC)cc2)CCCCC1 C(=O)(C(C)CC=CCC)NC1C(NC(COCCC#C)=O)CC1 N1(C(C2C(C)(C)N(C(C3Cc4nccn4C3)=O)CC2)=O)CC2CC(O)CC1C2 N1(C(C(CCNC(c2ccsc2)=O)OC)=O)CC2(CNC(=O)OC2)C1 C1(NC(C(C)O)=O)CN(C(c2[nH]ccc2-c2ccccc2)=O)CC1(C)C Cc1cc(C(=O)NC2CCC(NC(=O)C(C)C(C)C)C2)c2c(c1)CCCN2 CC1CC(C(=O)NC2CC(NC(c3ccc(N)nc3)=O)C2)C(=O)O1.C1CC1 c1(C(N(CCCN(C(c2nc(C)sc2)=O)C)C)=O)ccccc1N1CCCCC1 c1ccc(F)c(O)c1.C1(C(=O)NC2(CCCC(=O)NC)CCC2)CCCC(F)C1 C1(C=O)CCC2CC2CC1.Cc1ccc(SCC(=O)NC2CC(F)(C)C2)cc1.N c1(C=O)csc(CC)n1.C(=O)(C(C)CC1CCCC1)N(CCOC)CC.N C1(CCNC(=O)C=Cc2cc[nH]n2)CN(C(c2ccn[nH]2)=O)CCO1.C1CC1.C c1(CC)cc(C(=O)N(C(C)CNC(c2cn(C)nc2)=O)CC)ccc1C.S c1(C(=O)OC)ccc(C(N2CCC(O)(c3cccc(F)c3)C2)=O)nc1 C1(CNC(C2C(CC)C2)=O)CN(C(c2nn[nH]c2C(C)C)=O)CCN1C.C N1(C(C2(CCC=C)CC2)=O)CCC(NC(c2cn(C)nc2C)=O)C(CC)C1 O=S1(=O)CCc2c(Nc3ccnn3CC3CC=CCC3)cccc21 C1(CC)CN(C(C2CC3(CSC3)C2)=O)CCN1C(=O)COc1c(C)cccc1C c1(C(N2CCCC(CCC)(NC(c3ccc[nH]3)=O)C2)=O)csc2cc(Cl)cnc12 c1(SC)ccc(C(=O)NC2C3CCN(C(c4cn(C)nn4)=O)C23)cc1Br S(=O)(=O)(c1ccc(Cl)cc1OC)N1CC(CC)C(N)C1 c1(OC)cc(NC(C2C(C)CN2C(c2ccc([N+](=O)[O-])[nH]2)=O)=O)cc(O)c1 c1(C=O)ccc2c(c1)OC(F)(F)O2.n1(CC)ncc(Cl)c1C(N1CCCC1)=O.N Cc1ccc(C(N2CCOCC(NC(=O)CC3C=CCC3)C2)=O)c(C2CC2)n1 CC(C)C(CN(C)C)C(=O)NC(C1CCCN(C(C2(F)CC2(Cl)Cl)=O)C1)C C(=O)(C(C)(C)C(C)NC(=O)C(CN(C)C)N(C)C)N(CC#CC)C C#CCC(C(=O)NCC(F)(F)C(F)F)NC(C1CCSC1)=O c1(C(=O)Nc2cccc(C)c2C(F)(F)F)cnc2ccccc2c1N C1(C2CCC2)(C(N2CC(C(C)NC(=O)Cc3cccnc3)OCC2)=O)CC1(F)F C(=O)(CCC(C)NC(C1(O)CC1)=O)N1CCC(OCC#C)C1 N1(C(c2sc(C)c(Br)c2C)C(=O)NCCOC)C2CCC1CC(N=[N+]=[N-])C2 C=CCCC(C)N(C(=O)COC1CC(NC(=O)C(C)(C)C)C1)CC N1(C(C(C)N=[N+]=[N-])=O)CCC2CCN(C(C3CCS(=O)(=O)C3)=O)CC12 c1(OC)ncc(C(=O)NC2CCCC2CNC(c2cnc(Cl)s2)=O)cc1C C#CC(C)(C)C(=O)NCC1CCCC1NC(c1cnn(CCO)c1C)=O N1(C(C(CCC)OC)=O)CCN(C(=O)CC(=O)OCC)CC(CO)C1 C(C)(CO)(C(=O)NCCN1CCCCCC1)NC(CNC(=O)OC)=O c1(CC(=O)NCC2C(NC(C(C)SCC)=O)COC2)cc(Cl)ccc1Cl CCCCCS(=O)(=O)CC(=O)NC1CCC(C)(NC(=O)CN2CCCC2C)CC1 N1(CC)CCCC(C(=O)NC2(CNC(=O)C(C)O)CCC2)C1 C(CC(C(=O)NC1CC(CNC(=O)C=O)C1)NC=O)SC.CCC(N)=O.N C1(C(=O)NCCCC)CSCCN1C(=O)C#CC1CC1 N1(C(CC2CC(CC)C2)=O)CC(C)CC1C(=O)N(CC)Cc1cccs1 c1(NC(C2(NC(c3sccc3C#N)=O)C(C)(C)C2)=O)cncc2ccccc12 N1(C(c2nc(C)oc2)=O)CCC2(CCC2NC(c2cc(CO)c(C)o2)=O)CC1 c1(NC(C2CC(=C)CN2C(c2cnc(Br)o2)=O)=O)cnc(Br)c(F)c1 Cc1sc(C)c(C(=O)NC(CO)C(C)NC(c2cc3c(s2)CCOC3)=O)c1C#N N1(C(C2CC=CCO2)=O)CCCC2C1CCCN2C(c1ccc2cccnn12)=O CCCC(C)(C)CC(=O)N1CC2CCC2(CNC(c2ccnc3ncnn23)=O)C1 N1(C(C#C)=O)CCC2(CCCC2C(=O)Nc2cccnc2F)C1 CC(C#N)C(=O)N(C(C)CNC(=O)CN(C1CCSC1)C)C C(=O)(C(C)S(C)(=O)=O)NCCn1cc(C(=O)NCC#CCC)nn1 C(=O)(C(C)C(C)CO)N1CC(C(C)NC(C(C)NC(=O)NC)=O)OCC1 c1(C(N2C(C)CCC(CNC(C#CC(C)C)=O)C2)=O)[nH]nc2cnccc12 c1(CC=C)cc([N+](=O)[O-])ccc1OC(c1c[nH]c(Br)c1)=O CCC(C)C(C(=O)NOC(C)(C)CO)NC(=O)CC1C(C)(C)C1(C)C O=C1NCCc2ccc(S(=O)(=O)NC3CNCc4ccnn4C3)cc21 CC1(C(=O)N(CCCNC(C2CCC2(F)F)=O)Cc2cccnc2)CCCCC1 N1(C(C(CCC)NC(=O)CS(=O)(=O)CC)=O)CCCN(C)CC1C N1(C(CC2(COC)CC2)=O)CC(NC(=O)C(O)CC(C)C)CC12CCC2 CC1(C(=O)NC2CN(C(C3CC(O)(C(F)F)C3)=O)C2)CC=CCC1 C(C)(C(CC(=O)O)NC(=O)Cn1cc(-c2ccc(C(F)(F)F)nc2)nn1)OC CC1OC2(C(=O)NC3CC34CCN(C(=O)C=CC(C)(C)C)CC4)CCC1CC2 c1(C(C)NC(C=C(C)CNC(c2cc[nH]n2)=O)=O)nc(=O)o[nH]1 c1(C(=O)NC2C(C)CCN(C(=O)CCOCC(F)(F)F)C2)cc(Cl)c(N)cc1F C=C1CCN(C(=O)CSCC(F)F)C(C(=O)NCC(Cl)C(C)(F)F)C1 Cc1c(NC(c2nc(NC(C3CCCCCC3)=O)cn2C)=O)cnc(Cl)c1Br Cc1ccccc1NC(C1(NC(=O)CCc2nncn2C)CSC1)=O CCC(CCC(=O)NC1(CN(C)C)CCC1)NC(C1CC1C(C)C)=O C1(NC(c2cc(C)c(Cl)cc2)=O)C(C)CN(C(=O)CC2CCCCCC2)CC1C c1(C(=O)NC2CCN(C(CC=CCCCCC)=O)CC2C)ccc2c(c1)CCO2 C1(C(=O)NCC(CC(C)C)NC(C2(CF)CCC2)=O)CC2C=CCC(C1)C2 CCCC(CC)CCC(=O)NCCOC1CN(C(c2nn(C(F)F)cc2Cl)=O)C1 C1(C=O)(C(C)C)CNC(=O)C1.C1(CC(N2C(CC)CC2)=O)CC2(CC2)C1 Cc1cc(C(N2CC(=O)NCC2C(N2CCOC(C(N)=O)C2)=O)=O)nc(C)n1 N1(C(c2cc(CC)c(C)cc2)=O)CCC2(CCN(C(C3CC(OC)C3)=O)CC2)C1 c1(C(c2nnnn2C2CCC2)NC(CC)CCCO)c(C)nn(CCCl)c1Cl c1(C(C(=O)N)N(CC(C)(C)C)CCC#N)cnn(C2CCC2)c1C.C=C(C)C C(=O)(C(CO)C(F)(F)F)NC12CCN(C(c3c(CC)n(C)nc3)=O)CC1C2 CC1CCN(C(=O)CC2CCNC2=O)CC1CNC(=O)C(c1ccccn1)O C(CCS(C)(=O)=O)(C(=O)N(CCCCCNC(=O)C(C)(C)C(C)C)C)OC Cc1nc2cccc(C(=O)NC(C)C(C(C)C)NC(c3cc(Cl)cnn3)=O)c2[nH]1 CC1CCC=C1C(=O)NC1(CCNC(=O)CCCSc2ccccc2)CC1 N1(C(Cc2cc(C)ns2)=O)CCCCC(CNC(=O)CCc2cc(C)on2)C1 Cc1cccc(CC(C)NC(C2C3CN(Cc4nc[nH]n4)CC23)=O)n1 C(=O)(CCCC(C)(C)C#N)NCCC1N(C(C(C=C)OC)=O)CCCC1C N1(C(C2(OCC)CCOC2)=O)CC=CC(C(N2CC(OCCO)C2)=O)C1 CCC(C)(C)CCCC(=O)NCCC(C)(CC)NC(=O)CC(C)(C)C c1(NC(C2CCN(C(CC3CC(C)C3)=O)C2)=O)ccc2nccnc2c1 c1(COC)cc(C(=O)NC2CCCN(C(c3cn(C)c(O)n3)=O)C2)n(C)c1 C1(NC(CC(C)n2ccnc2)=O)CN(C(c2cnn(C)c2F)=O)CC1CC1CC1 c1(CNC2(C)CC2(Cl)Cl)cccc(Cl)c1O c1(SCCC)c(OC)cccc1C(=O)N.c1(CC(N2CCC2)=O)nnc(O)s1 c1(C(N2CC(c3cn(Cc4cc(OCC)no4)nn3)C2)=O)cc(C)nn1CC Cn1cc(S(=O)(=O)CCNC(c2ccc(C3CC3(F)F)cc2)=O)cn1 C(CCCCCNC(=O)C(F)(F)CO)NC(c1ccccc1)=O.C1(O)CC1(F)F c1(CC(N2CC(C(C)NC(=O)COC3CC=CC3)C2)=O)cccc(F)c1F N1(C(C(C(C)C)SC)=O)CC(NC(c2cc(C#N)c[nH]2)=O)C2CCCCC12 c1(C(=O)NC2CC(C)N(C(=O)CC3COC(C)(C)C3)C2)cc(=O)cc(Cl)[nH]1 C(CC(CNC(=O)CCc1ccoc1)NC(c1cnco1)=O)OC C(=O)(C(C(C)CC)NC(=O)C=Cc1ccnn1C)NCCC(CC)C CC1(C)CCC(C(N2CCC=C(F)C2)=O)(NC(=O)C=C(C2CC2)C2CC2)C1 Cc1cc(=NC(=O)C(=O)NC(C2CCCN2C(=O)Cn2nnc(=O)[nH]2)C)[nH]o1 N1(C(=O)C2=CCCO2)CCCC(C2CN(C(c3coc4cc(O)ccc34)=O)C2)C1 c1(NCC2(C)CCCN(C(C=C(C)C)=O)C2)cc2nn[nH]c2cc1[N+](=O)[O-] Cc1c[nH]cc(C(=O)NCCC(C)(C)NC(C2CC2(C)C(C)C)=O)c1=O N1(C(CCC=CC)=O)CCC(C(F)(F)F)C(CNC(c2ccnc(C)c2)=O)C1 CC1(C(=O)NC2CCC2C(=O)NCc2ccc(F)cn2)CCC(=O)N1 C(=O)(C(CC)C(C)O)N(CCC1N(C(CN(CCC)C)=O)CCSC1)CC CCCCC(CC)C(=O)NCC1CC(O)CN1C(=O)CC1CCOCC1 S(=O)(=O)(c1ccc(N(C)CCn2cncn2)c(C#N)c1)N1CC(C)SC1 n1(CC=O)nc(C)c(C)c1C.C1(OC)CCN(C(=O)CC2(C)OCCO2)C1.C c1(C(N2CC(CN(C(C3C(C4C(C)C4)C3)=O)C)C2)=O)cnc2c(c1)CCOC2 c1(C(C)=O)cc(C(=O)NC(C)CC(C)NC(C23CC2C3)=O)co1 C1(CC)CCC(C(=O)NC(C)CN(C(c2sc(O)nc2C)=O)CC)CC1 CC1(C)CC(CNC(C2CCCNC2=O)=O)N(C(c2csnc2Cl)=O)C1 Cc1cc(C(N2CC(C)C(C)C2)=O)c(C)o1.c1(C(=O)N)cc(-c2ccco2)no1 C1(C(=O)NCC(C)(C)CO)(NC(Cn2ncc(C)c2)=O)CCC(C)(C)C1 C(=O)(CCCC(CC)CC)NC(C(NOCC=C)=O)(C)CO Cc1oc([N+](=O)[O-])cc1C(=O)N.C1(C(C)C)CCN(C(=O)C=O)CC1.C(C)C C1(CO)CN(CC23CCCC2C3)C2(COC2)C1.c1ccccc1 C1(C(=O)NCC2CN(C(CC3CN(C)C3)=O)C2)CCCCC1 C12(CC)CCC(C(=O)NCCNC(c3sc(OC)nc3Cl)=O)(CC1)CO2 Cc1ccc(OC(C)C(=O)NCC2CCN2C(=O)C=C(Cl)Cl)c(C)c1 N1(C(c2c(CC)[nH]nc2Cl)=O)CCC(NC(c2nonc2N)=O)C(F)(F)CC1 N1(C(C(C(C)SC)O)=O)CCC2(CCCN(C(=O)CCc3cncn3C)C2)CC1 N1(C(c2[nH]cc(C(N)=O)c2)=O)CCC2(CC(NC(=O)Cc3cc[nH]n3)CO2)C1 N1(C(C2(CNC(c3cnco3)=O)CC(=C)C2)=O)CC=C(C(C)(C)C)CC1.C N1(C(C(C(=O)OC)C)=O)CCC(C)(C(=O)N(CC(O)C(F)(F)F)C)CC1 C1(CC#C)CN(C(C2(CO)CCN(C(c3nonc3C)=O)C2)=O)CCO1 CCC(C(=O)NCCC(C)NC(c1c[nH]nc1OC(C)C)=O)C(F)(F)F N1(C(C2N(C(C(C)C)=O)CCC2)=O)CCC(C)(NC(=O)C)C1.C1CCCOC1.O c1(C(=O)NC2CCN(C(C(N(C)C)C3CC3)=O)CC2O)cc2cccc(F)c2o1 CC1CC(C)CN(C(c2ccc(CNC(N3CCCC3)=O)cc2)=O)C1.C1CC1.C C1(OC)CCCC(NC(C2C=CC(NC(C3CC3(F)Cl)=O)C2)=O)C1 c1(C(=O)NC2C(NC(C(CCOC)(C)C)=O)CCC2)cc2oc(Br)cc2[nH]1 c1(C(=O)NC2C(NC(CC3CC(=O)NCC3)=O)C2)ccccc1[N+](=O)[O-] Cc1nc2ccc(C(N3CC(N(C)C(c4ccc(P(C)(C)=O)o4)=O)C3)=O)cc2[nH]1 c1(C(N(C(CO)C2CC2)C)=O)cc(-c2ccccc2F)nc2onc(C3CC3)c12 C1(NC(C)=O)CN(C(c2ccc(C(=O)OC)nc2)=O)CC1C1CC1 c1(C(N(C(C)C(=O)NCc2cscc2C)CC)=O)n[nH]c2c1CCC2 C(C(C)(COC)C(=O)NCc1ccnc(C(=O)NCC2CC2Cl)c1)OC CC1(C)CC(NC(=O)COC2CCOCC2)CCN(C(=O)CCc2cnoc2)C1 CC1(C)CN(C(c2nsnc2O)=O)CC1CNC(=O)Cn1cc(CO)nn1 CCCCCCC(C)C(=O)NCC12CC(NC(c3sccc3C#N)=O)(C1)C2 C(=O)(C(C)CC(C)C)N(CCCN(C(c1c(C)sc(Br)n1)=O)C)C c1(OC)ccc(C(N2CCCC(CN(C(=O)CC3(C)CC3)C)C2)=O)nn1.S CC1(C)CC(CNC(c2cc(-c3ccccc3)cs2)c2nnn[nH]2)C1.C1CC1.C Cc1c(Cl)ccc(C(=O)NC2CN(C(C3(CO)CC3)=O)CC2C2CC2)c1Cl N(S(=O)(=O)N1CC(C(=O)OC)Cc2ccccc2C1)(CC)CC C(=O)(C#CC1CCOCC1)NC1CCN(C(COC2(C)CCC2)=O)CC1F C(=O)(C#CC1CCCCC1)N1C2CN(C(C3(C(=O)NC)CC3)=O)CC1CC2 C1(O)(CC)CN(C(c2ccn(CC(F)F)n2)=O)C1.C1(C2(C=O)CC2)CCCO1 C1(CNC(C=C(C)C(F)F)=O)CCCCC1.C1(C)(C=O)CC1C(F)(F)F c1(CN(C)CCOc2ccccc2[N+](=O)[O-])ccc2c(c1)OCC2(C)C C12(C(=O)N)CCCN1CC(O)C2.c1(CCC(=O)N(CCC)CC)c(C)noc1C C1(NC(c2c(C)nns2)=O)CCC2(CC1)CN(C(c1ncc[nH]c1=O)=O)CCO2 CC(CNC(C1CCCC1)=O)C(F)C(=O)N1CC2CC1CC2CF C#Cc1cccc(NC(=O)C(CCN(C)C)NC(C2CC23CCC3)=O)c1 CC1=C(C(=O)NCC2(O)CN(C(=O)C(C3CCC3)C3CCC3)C2)COCC1 Cc1nc2ccccc2cc1NCc1ccc(OCC(F)(F)F)cc1 CC1CN(C(=O)C(C2CCCO2)NC(=O)Cc2cccc(F)c2)CCS1 Cc1cc(F)cc(C(=O)NC(C)CCNC(=O)C(C)Cc2cccnc2)c1N c1(NC(c2ccccc2)CN(C)C)nc(=NC2C=CCCC2)[nH]c2ccccc12 CC1(C)CN(CC(=O)NC2(CNC(=O)CC3CCC(=O)C3)CCOC2)C1 N1(C(c2[nH]cc(C)c2)=O)CCN(CC(=O)NC(C)CCCCO)CC1 C(=O)(CCCONC=O)N.C1(C(N(C(C)C)CC)=O)CCC=CO1.C(C)(C)C c1(C(N(C2(CC(=O)N)CC2)C)=O)cn(C)c(=O)cn1.CC1CCCN1CCC CCCC(CCC)NC(C1(NC(c2c[nH]nc2C(F)F)=O)CC1(C)C)=O C(=O)(C1Cc2ccccc21)N1CCC=C(C(=O)N(C)Cc2cocn2)C1 Cc1cc2cc(OCn3cc(C4CCCNCC4)nn3)ccc2[nH]1 N1(C(C2(C)OCCN(C(C)=O)C2)=O)CCN(Cc2ccccc2)C2(CCC2)C1 C1CN(C(=O)CC23CCC(C)(C2)OC3)CC(C)(C)C1.C(C(C)(O)C=O)OC.N N1(C(c2cc(C(C)(C)C)nn2C)C(=O)NC)CC(C)CC(C)C1C C1(CNC(c2cc[nH]n2)=O)CN(C(c2ccccc2)=O)C2CC12.[nH]1cccn1.C Cc1csc(=Nc2ccccc2)n1CC1CCn2c(O)nnc2C1 C(c1csc(C)n1)=CC(=O)N(C1CCCC1)C.Cc1cn(C(C)(C)C=O)cn1.N O=C1NCCn2c(CNC(c3nnnn3CC3CCC=CO3)C3CC3)nnc21 c1(C(=O)NCC(C(N)=O)Cc2ccccc2Cl)cc(C(F)(F)F)ccc1F c1(N2C(CN(C)C)CCC2)cc(Cl)c2n[nH]cc2c1 CC1(C)CC(C)(C(=O)Nc2cnn(CC3CC3)c2)CN1C(=O)C1CC1 CC(C)(C)C#CC(=O)NC12COC(C)(C1)C2.C12(C(=O)N)CCC(C1)OC2 c1(C(=O)NC2(CNC(CC3C(C)OCC3)=O)CCC2)ccc2nnc(O)n2c1 c1(NCc2n(CC)cnn2)[nH]c(=NCCCC(C)(C)C)nc2ncn(CC)c12 c1(C(N2CCC(NS(=O)(=O)CCBr)C(F)C2)=O)cc2cccn2cn1 Cc1ccnc(O)c1C(=O)NCCC(C)CCNC(=O)CN1CCOC1=O c1(C(C(=O)NCCCC)N(c2cc(F)c(C)cc2F)C)ccc2c(c1)OCCC2 N1(C(C=CC=O)=O)CCN(C(=O)CC2(O)CCCN(C)C2)C(C(C)C)C1.C Cc1cc(C(N2CCC(C(F)CNC(=O)C(C)C(C)C)CC2)=O)nc(C)c1 N1(C(CN(C2CCCC2O)C)=O)CC2CC3CC2C1C3NC(C1CC2CC2C1)=O N1(C(C2C(OC)C2)=O)CCN(C(c2cc(C)nc(O)c2)=O)CC2(CC2)C1 c1(OC)ccc2oc(C(=O)NCC3CN(C(=O)C(OC)O)C4CC34)cc2c1 C1(NC(=O)NCC2(c3nn[nH]n3)CC2)CC(O)C(F)C1 CCS(=O)(=O)CC(=O)NCCCCCCN(C(=O)COCCc1ccccc1)C c1(OC)c(Cl)ccc(C(=O)NC2COC3C(NC(c4cn[nH]c4)=O)COC23)c1F C1(C(N2CC(CNC(c3cc(N(C)C)ncc3)=O)C2)=O)COC2COCC12 c1(C(=O)NC(C2CCCN(C(=O)CC(C)C(C)C)C2)C)cccc(N)c1C(F)F c1(C(=O)NC2(C(N3C(CN(C)C)C=CC3)=O)CSC2)ncccc1F Cc1cc(C)c(C(=O)NC23CC(C2)C3)c(O)n1.c1(C=O)cn2c(n1)COCC2 N1(C(CC(CCC)O)=O)CCCN(C(=O)C=CC(C)(C)SC)CC1C c1(C(N2CC=C(CNC(CSCCCC)=O)CC2)=O)cncc(S(N)(=O)=O)c1 C(=O)(C(C)(F)C(C)(C)F)N1CCCCC1.c1(OCC#C)ncccc1C(=O)N C(=O)(C1=CCOCC1)NCCc1cc(C(=O)NCC(=O)OCC)no1 C(=O)(C(C(C)(C)C)NC(=O)C(CC)CCOC)NCCCCCN(CCC)C C=CC(O)C(C)(C)C(=O)N1CC2CCC(C1)C2CC(=O)Nc1ncn(C)n1 CC1C(NC(=O)CC(O)C2CC2)CCCN1C(=O)Cn1ncc(O)nc1=O Cc1ccnc(Cl)c1NC(C1(O)CCN(C(=O)NC(=O)C(Cl)(Cl)Cl)C1)=O CCC(C)C(O)CC(=O)N1C(CC(=O)NCCc2ccsc2)C2CCCC12 C1(C(N2CC(CCNC(c3cc4scnc4[nH]3)=O)C2)=O)CC12CC(F)(F)C2 c1(C=O)cccc(C2(F)COC2)c1.C1(F)CCC1.C(F)(C(=O)NC)=C(C)C c1(CCC=O)cc(F)ccc1F.C1(NC(C2(CCOC)CC2)=O)CCCCC1.N C#Cc1ccc(Cl)c(C(=O)NC2CN(C(=O)C(CC)CC(C)C)CC2C=C)c1 C1(C(=O)NCCCNC(c2scc(C(N)=O)c2)=O)CCC([N+](=O)[O-])CC1 Cc1cnc(O)n1-c1cccc(C(=O)NCCCOC2CCCC2)c1 C(CC(C(=O)NCC1CCC1C(=O)OC)NC(=O)CC1CC1)=CC C=C(F)C1(CC(N2CCC(C)(CC(=O)N(CC(C)O)C)C2)=O)CCC1 c1(CC(=O)N(C2CN(C(C(CC=C)(C)C)=O)CC2F)C)c(C)nc(O)nc1O N1(c2cc(NCC3CCCCN(C)C3)nc(C)n2)CCC(O)CC(C)(C)C1 c1(N(C)C)ccc(Br)c(S(=O)(=O)NCCCN(C)C(C2CCOC2)=O)n1 Cc1cc(F)c(C(=O)NC2CCN(C(=O)C=CC=O)CC2C)c(F)c1.C1CC1 C1(C(=O)NCCCCN(C)C(c2csc(C(C)C)n2)=O)(COC)CCCC1 [N-]=[N+]=Nc1cnccc1C(N1CCC(NC(c2cccc(F)c2F)=O)C1)=O C1(O)(CNC(C(COC)(F)F)=O)CCCN(C(c2cnccc2C)=O)CC1 c1(CNCC(c2ccc(F)cc2)OC(C)C)ccc2c(c1)CNC2 C1(CC=C)(NC(=O)CCNC(c2n[nH]cc2Cl)=O)CC=CC1 c1(-c2cn(C(C(N3C(CCC#C)CCCC3)=O)C)nn2)ccccc1C=C C(CC(C)N=c1nc(N2CCC3(CCN(C)C3)C2)c2[nH]ccc2[nH]1)OC C12(CNC(CSCCCC)=O)CCC1CN(C(c1nc(O)sc1C)=O)C2 C1(CNC(=O)CCOC2CCC2)CCCN(C(=O)C2=CCCCO2)CC1 CC(C)C(F)C(=O)N(CCCNC(=O)CN)C.c1(C[SH](=O)=O)ccccc1 N1(C(CC2(C=C)CCC2)=O)CC2CC1CC2NC(c1cccc(N(C)C)c1)=O C12CCCC1CCN2C(c1cc(C2CC2)on1)=O.c1(C(=O)N)ccc(=O)oc1.C c1(N(C(CC2CCC(NC(=O)CN3CCNC3=O)C2)=O)CCO)cccc(O)c1 C1(N(C)C)CN(C(=O)Cn2cc(C3(S(=O)(=O)N(C)C)CC3)nn2)CCC1O C(=O)(C1=CCCCC1C)N(C1CCN(C(=O)CNC(N)=O)CC1)CC#C C1(NC(c2ccc(NC(C)=O)cc2)=O)CN(C(c2c(O)noc2C)=O)CC1(C)C C1(C(N2CCC(C)(CNC(c3cnc(S)nc3)=O)C2)=O)CC(=O)C12CCC2 N1(c2nc(C#N)cc(C)n2)CCCC2C1CCN2Cc1ccc(C(=O)N(C)C)[nH]1 c1(C(NOCC(=O)NC(C)(C)C)=O)cnccc1Br.C(=O)(CO)O C1(NC(CCc2onc(C)n2)=O)CCN(C(=O)COc2ccc(F)cc2)C2CC12 N1(C(C(C(C)C)SC)=O)CCC(O)(CNC(C2COC(=O)O2)=O)CC1 c1(C(=O)NCC=CCCC)c[nH]nc1CNC(=O)C(C)c1ccco1 C1(C(C)C)C(=O)NCCN1C(=O)CNC(C1COCOC1)=O N1(C(C2N(C)C(=O)CC2)=O)CCN(C(c2nc(Br)c[nH]2)=O)CC1CCO C1(C(N(C2CCC(O)CC2)C)=O)CCN(C(=O)C2=CCCCC2)CC1O CCC(C)(CO)C(=O)NC(COC)CC(=O)NCCC1(OC)CCC1 N1(C(CCC(C)OC)=O)CCCC2CN(C(c3c[nH]nc3C(F)(F)F)=O)CCC12 c1(CCC(=O)N)ccc(C(F)(F)F)cc1.CCCCN(C)C(C1(CF)CC1)=O c1(C(N2CC(CCNC(c3c(CC)ncs3)=O)C2)=O)cccc2cnccc12 C1(C)(OCC(N2CCC(C(C)NC(C3(SC)CC3)=O)C2)=O)CCOCC1 C(=O)(C(CO)C(F)(F)F)NC(C)CC(=O)NC1(C)CS(=O)(=O)C1 c1(CC(=O)N)cn2c(n1)CCCC2.N1(C(C2(CC)CCC2)=O)CCC(CO)CC1 CCCCC(C(=O)NCCC1CCN(C(c2cccc(Cl)c2)=O)C1)NC(N)=O CC(CN(C)C)CCC(=O)NCC1CC1C.C1(=CC(=O)N)CCSCC1 c1(CN2C(C)(C(=O)NCC3CCO3)CC2)ccc2n[nH]cc2c1 Cc1cc(=O)oc(C)c1C(=O)NCC1CCOCC1.C1(C=O)CC1C1CC1C.N c1(NC2C(C)CN(C(c3ccc(C(F)(F)F)[nH]3)=O)C2)c(C#N)cccc1[N+](=O)[O-] N1(C(CCC=C=C)=O)CCC2CCCN(C(=O)CCOCCN(C)C)C2C1 CC(C)C(C(=O)NCC(C)(CO)NC(C1CCSCC1)=O)N1CCCCC1 Cc1ccc2c(c1)CCC2C(=O)N(C(C)C)CC1CCCO1 CCCC(C)(C)CC(=O)NCC1(CO)CCN(C(=O)CC2CCC3CC23)CC1 Cc1cc(C(N2CC(C)(NC(C3CCCCC3(F)F)=O)C2)=O)cnc1Cl c1(CC)ccc2[nH]nc(NC(C3CC=CCC3NC=O)=O)c2c1.C(C)(C)C.O CN1CCCC(C(=O)NC(C)(CNC(=O)CCc2ccccc2)CO)C1 N1(C(c2ccc(OC)s2)=O)CC2CCC(C1)N(Cc1ncccc1Cl)C2 C(=O)(CS(=O)(=O)C1CCCC1)N1CC2C(CNC(CCC3(C)CC3)=O)(C2)C1 C1(CNC(c2nc(C(N)=O)sc2)=O)COCCN1C(=O)CC1(C)CC1.S C(=O)(C(CC(C)C)N(C(=O)C(c1cnn(C)c1)=O)C)NCc1c(C)ncs1 C(=O)(C1=CCCN(C(=O)CCC2CC2(F)F)C1)NC(CC=C)(C)C C1(CNC(C2(C)N(C)CCC2)=O)CCC2CN(C(c3cc(=O)cc(Cl)[nH]3)=O)CC12 N1(C(C(CSC)O)=O)CCc2sc(CNC(C3CCN(C)C3)=O)nc2C1 N1(C(CC(C=C)CC)=O)CCCC(C)(C)C1C(=O)Nc1cc(C)c(F)c(C)c1 CCCCCC(CC)C(=O)NC(CC1CC1)C(=O)NC12CC1CN(C)C2 N1(C(C)C)CCC(CNC(=O)C(C2CCCC2)NC(c2sccc2F)=O)C1 c1(C(C)(C)C)ccccc1COC(=O)CCc1sccc1Br c1(C(=O)NC2(CO)CN(C(Cc3nc(C)sc3)=O)C2)nc(Cl)oc1C c1(CC)cc(=NCC2(O)CCCN(C(=O)C(C(C)CC)OC)C2)[nH]c(CC)n1 c1(C(=O)NC(C(=O)NC(C#C)C(C)C)CN(C)C)cccn2cncc12 N1(C(C(C(C)O)(F)F)=O)CC(NC(c2cccc(O)c2F)=O)C2(CCOCC2)C1 Cc1cc(C(=O)NC2CCCCC2NC(c2cccn2C)=O)cc(C)c1C#N N1(C(=O)NCC(C)OCC)CCC(O)(c2cccc(CC)c2)CC1 CCS(=O)(=O)N1CC(C(=O)NCC2CC2CC(C)C)C1 Cc1ccc(C(CN(C(=O)CC23CCC2C3)Cc2occc2C)C(=O)O)cc1 Cc1cnc2n1C(C(=O)N1CCC(C)(NC(c3cnn(CCF)c3)=O)C1)CCC2 C(=O)C(C)C(=O)N1CCC(C(F)CNC(=O)CC2CNC(=O)C2)CC1.CO C1(CC)C(=O)N(C)CCN1C(C1C(O)CCN1C(=O)CC#N)=O c1(CC(=O)NCCN(CCOC)Cc2nnnn2C)ccc(F)c(Br)c1 C1(CC(C)N)CCN(C(=O)CC2CCC2c2ccccc2)CC1.C(C(=O)O)N1CC1 c1(SCC(=O)N(C2CC(C#N)C2)C)coc(C)c1.C1(CC=O)CCCCO1 C=CC1(CC(=O)NC2CC(O)C2)CN(C(C2(F)CC=CCC2)=O)C1 c1(CC)[nH]ccc1C(=O)NOCC(=O)N(C)Cc1scnc1C Cc1ncc(Cl)c(C(=O)NC(C2(O)CCN(C(c3c[nH]ccc3=N)=O)C2)C)n1 C1(C(=O)N)C2CCN(C(=O)C=C(C)c3ccco3)CC12.C1(OCC)CCC1 N1(C(CC(C(C)C)C)=O)CCC2(CCOCC2)CC1 C1(C(=O)OC)CN(C(=O)NCC2CCCN2CC(C)C)CC(F)(F)C1 C1(O)(C(C)NC(C2CC(C)(C)C2)=O)CCN(C(=O)Cn2nnc(=N)[nH]2)C1 C(=O)(CCCC(=O)NC1CCCC1)OCC.c1(C=O)cc(C)n(C(F)F)n1.C C=CCC(C(=O)NCc1cnn(C)c1OC)NC(C1CC(CF)C1)=O C(=O)(C(CC(F)(F)F)c1cccc(F)c1)NCC(CCOC)O c1(C(=O)NC(CNC(C2C(CC)OCC2)=O)C)cc2c(O)ncnc2cn1 CC1(C)C(NC(c2nc(Cl)sc2Cl)=O)C2CCCN(CC3CC3)C12 C1(C(=O)NCCCCCNC(Cc2cccc(SC)c2)=O)CCn2nncc2C1 c1(C(=O)OCC)nc[nH]c1NC(C1CC(NC(c2ccncc2)=O)C1)=O Cc1cc(C)c(C(=O)NCC2CN(C(C3(C)CCC3)=O)CCC2C)c(O)n1 C(=O)(C(C)N=c1cc[nH]cc1)N1CC(C2CN(C(CC=CCCCCC)=O)C2)C1 N1(C(CCC(=C)C)=O)CCN(C(=O)C(C)(C)c2cncs2)CC1c1cnn(C)c1 C12(C(N(C(C(=O)OC)C)C)=O)COCC1CN(Cc1nc(C)cs1)C2 Cc1oc(C(N2CC3CCCCC23)C(=O)NCC(F)F)cc1S(C)(=O)=O CCCCCC(CC)C(=O)N1CCC(C(=O)NCc2snnc2CC)O1 C(=O)(C1c2c[nH]nc2CN1C(=O)Cn1cnnc1O)N(CCCC)CCOC C1(C)(CNC(C(C=CC)O)=O)CC(F)(F)CN1C(=O)CCn1cnnn1 Cc1ncc(Cl)c(C(N2CCC(NC(c3c(Cl)c(C)nn3C)=O)C(CO)C2)=O)n1 C1CCN(C(=O)C=C(C2CC2)C2CC2)CC1.C(c1ccncn1)=CC(=O)NC C(=O)(CCC(=O)NCC1(C)CCCC1)NCCC.C1(C(=O)N)CC=CCC1 c1(C(=O)N)cccnc1.C1(C(=O)OC)CC(C(=O)NCCC2CCOC2)C1 C(=O)(CCCN(C)C)NCC(C1CCCCC1)NC(C1C(C)(CC)C1)=O Nc1ccc(C(=O)NCC2(NC(=O)CC3CC3)CCOC2)nc1 N1(C(C2N(C(c3cc(C)c(N)cn3)=O)CCC(=C)C2)=O)CCCC(C)(C)C1C c1(NC(C(N2CC(C)N(C(COC)=O)C(C)C2)=O)=O)cc2c(cc1Cl)OCO2 C1(CO)(NC(CCCCc2ccc(CCCC)cc2)=O)CCCc2ccccc21 C1(C(=O)NC2CCN(C(c3coc4c3COC4)=O)C2)CC2CCC1C21CC1 CC1(C)CCC(C)N(C(c2csc(-c3cn[nH]c3)n2)=O)C1.C(=O)(CC1CCC1)N Cc1nn(C)c(C(F)F)c1C(=O)NC(c1ccccc1)C.C1(C=O)CC1F.C C(=O)(C1=CCC(F)(F)CC1)N1C(C)C(NC(c2ccc([N+](=O)[O-])n2C)=O)CCC1 CC1(C(=O)NCC(c2ccccc2)NC(=O)CC2CCC=CCC2)CCCCC1 c1(CN2CCN(S(=O)(=O)Cc3cccc(Br)c3)C3C2C3)ccc2nonc2c1 N1(C(C2C(C)C2)=O)CC2CC1C2CNC(C1(C(F)(F)F)CC1)=O C1(C)(CC)CC(NC(=O)CSC(C)C)CN1C(=O)C=C(C)C(C)C CC1(C(N2CCC(NC(c3ccc(F)c(O)c3)=O)C2)=O)CCC12CCC2 c1(C(N2CC(N(C(C3=C(C)CCC3)=O)C)C2)=O)cnc2c(c1)COC2 c1(N2CCC(C)(N(C)C)CC2)nc2ccccc2nc1NCCC1CC1 C(C)(c1cccnc1)=CC(=O)NCC1N(C(C(CC)SC)=O)CC(F)C1 C(=O)(CN=S(C)(C)=O)NCCN(C)C(C1CCCCN1Cc1cccnc1)=O c1(-c2cc(C=O)no2)ccccc1Br.C(C1CCCC1)=CC(=O)NCC=CC.N c1(C(=O)NCCN(C(C2C(CCC)CCC2)=O)CCC)ccn2cnnc2c1 C1(NC(C2CCN(C(C)=O)C(C)C2)=O)CCc2nn[nH]c2C1 C(N=c1cc(C)c(S(=O)(=O)NC2C3CCCCC23)c[nH]1)c1c(C)csc1 N1(C(CC2CCC(C)CC2)=O)CC2(C(=O)NCCCOC(F)(F)F)CC1CO2 C#CCC(C)C(=O)NCC(C(C)C)NC(=O)CCc1csc(-c2ccco2)n1 C1(CNC(C#CC2(CC)CC2)=O)CC12CCN(C(=O)CCC1CCC1)CC2.C c1(C(N(CC(Cc2ccccc2)NC(CCC#C)=O)C)=O)cc2c(ncn2C)[nH]1 C1(NC(CC2(N(C)C)CC2)=O)CN(C(c2cn3ccnc3s2)=O)CC2(CCC2)C1 C1(NC(c2c(C)nn(C)c2C)=O)CC2CN(C(=O)CC(=O)NC3CC3)CC2C1 c1(CC)nc(C)ncc1C(=O)NCC1CCN1C(C1CCCN1CC)=O C1(OC)CCC2CN(C(=O)C(C)=CCNC(C3CCC(=O)O3)=O)CC12 CC1C(NC(c2cccc(O)c2F)=O)CCCN1C(=O)CC1CCCCCC1 c1(C(=O)OCC)sc2[nH]c(CN3CC(COC)CC3C)nc(=O)c2c1C N1(C(COCCCC)=O)CCC2CCCC12CNC(c1snc(C)c1N)=O Cc1nc2cccnn2c1C(N1CC(c2ocnc2C)C1)=O.C1(O)(C(=O)N)CC1 C1(C(=O)NCc2ccc(SC)o2)CCC2CCC1N2C(C1CC1)=O.C1CC1 C1(NC(CCCSC)=O)CC2CN(C(c3ccc(OC)nc3)=O)CCN2C1=O C1(C(N2CCC(COCC)C2)=O)CC(F)(F)CN1C(c1scc(C)c1C)=O N1(C(C(=O)NC(C)C)CC2CCCO2)CCN(C)CC(O)C1 Cc1cc(C(=O)NCC(N2CCOCC2)C2CCOC2)cc(C)n1 C(C(=O)NC(CCN(C)C)C(=O)N)(C(C)(C)C)OC.CC(O)C.C(N)=O C#CCC(C)(C)C(=O)NC1CNCC(C(F)(F)F)C1 O(NC(=O)CC1(C)CC1)CCOCCOC.C1(CC=O)COC(=O)C1.N C1CC2(CC2)CN1C(C1CC12CCSCC2)=O.c1(C(=O)NC)cn(CCO)nn1 c1(C(=O)NC2C(NC(C(C)CSc3ccccc3)=O)CCC2)ncc(F)cc1F C1(CCC)CN(C(C2CSCC(=O)N2)=O)CC1C(=O)NCC(C)(Cl)CC c1(C(N2CC(NC(c3c(C)c(N)cnc3)=O)C3(C2)CC3)=O)ccc2nn[nH]c2c1 c1(SC)ccc(Cl)c(C(=O)NC(C)(CNC(=O)CC(C)O)CC(C)C)c1 CS(C)(=O)=NCC(=O)NC1CC(CCNC(c2cccc(F)c2Cl)=O)C1 c1(C(=O)NCC2CN(C(c3cnc(SC)s3)=O)C(C)C2)cccc([N+](=O)[O-])c1Cl C1(C(N(CCNC(CC(CC)C)=O)C(C)C)=O)CCc2c[nH]nc2C1 CN=c1nc(N(C)CC2CCCN(C)C2)[nH]c(N2CCS(=O)(=O)CC2)n1 c1(C(N2CCCCC(CNC(Cc3c(C)cco3)=O)C2)=O)noc(C)c1[N+](=O)[O-] Cc1cc(C(N2CCCCC2CCC(N2CCCC(C)C2)=O)=O)oc1C C(=O)(C(F)C(C)CC(C)(C)C)N1CCC(C#N)(CC(C)C)CC1 N1(C(c2ccc(C)c(C)c2)=O)CC(NC(=O)C(C)(O)C(F)(F)F)CC2(CC2)C1 c1(C(N(CC(CN(C)C(c2cc(Cl)ccc2F)=O)O)C)=O)ccc(F)c(Cl)c1N c1(C(=O)OC)ccc(C(=O)NC(c2ccc(C(C)(C)C)cc2)C(C)C)c(N)n1 C1(CNC(=NCC)NCC(C)(C)c2cccs2)CCCC(C)(C)C1 c1(CC(=O)NC(C2CCN(C(C3(C(C)=O)CC3)=O)C2)C)cncc(C)c1 c1(C(N2CC34COCC3(C2)C4)=O)c(Cl)ccc(Cl)c1Cl c1(C(=O)NCC(CN(C)C(C2(CCF)CCC2)=O)O)cn(C2CCCC2O)nn1 C(CCCCC(=O)N1CC(F)(C(N2CCC(CO)CC2C)=O)C1)=CC c1(C(N2CC(OC)C(NC(c3coc(N(C)C)n3)=O)C2)=O)c(N)sc(C)c1C N1(C(CCC=C(C)C)=O)CCCN(C(C2CC2C(C)(F)F)=O)CC1C(C)C C#Cc1ccc(C(=O)NC2CC(O)CN(C(c3ocnc3C)=O)C2)nc1 c1(CC(=O)NCC2CN(C(=O)CCc3cnccn3)CCO2)cccnc1Cl C12CCCN(C1)C(=O)N2.C1(CN2CCC(n3ccc(C)n3)C2)(CO)CC(F)(F)C1 CCCCC(=O)C(=O)N1CC2CC1(CNC(=O)Cc1cnc(C)s1)C2 c1(NC(C)=O)ccc(Cl)c(C(N2CCC(c3cccc(C)c3)C2)=O)c1 c1(C(C(=O)NCCSC)N(CCCO)CC)csc2ccccc2c1=O C(=O)(C(C)(C)C(F)F)NCC(C)CN(C(=O)CC1CC12CC2)C CC(C)(C)C(C#N)C(=O)NC.c1(C=O)cc(C(F)(F)F)cc(F)c1.C1CC1 C1(C(=O)NCCCN(C)C(c2ccn(C(C)(C)C)c2)=O)CC1C1CCCC1 N1(C(C#CC(C)(C)C)=O)CCN(C(=O)CC(O)C2CC2)C2(CCC2)C1 c1(C(=O)NCC2(C(N3CC(c4nc(C)[nH]n4)C3)=O)CCOCC2)snc(C)c1N CC1CN(C)CC(C(=O)NCC2(C(N)=O)CN(C(c3ccns3)=O)C2)O1 c1(CC(N2CC=CC(NC(CC(C)(O)C3CC3)=O)C2)=O)csc2ccccc12 C(C)(CCCCNC(C1CC(SC)C1)=O)NC(C1C(CC)C1)=O c1(C(N2CCC(C3N(C(C4C(C)(C)CO4)=O)CCC3)C2)=O)cc(Cl)c([N+](=O)[O-])[nH]1 C1(C(=O)NCCNC(C(N2CCSCC2)C)=O)CCC(SC2CCCCC2)CC1 C#Cc1cc(NC(C2(C)C=CCN2C(=O)CCOCCC)=O)ccc1C C(=O)(C1=CCCCCC1)NCC1(OC)CCN(C(c2cncnc2C)=O)C1 N1(C(c2ccc(C(C)C)s2)=O)CC2CCC(NC(=O)Cc3cnccn3)CC2C1 Cc1nn(C)c(C)c1S(=O)(=O)N1CCN(c2ncc([N+](=O)[O-])c(=N)[nH]2)CC1 C(=O)(C=CS(C)=O)NCC1C(NC(CC=CC)=O)CC1 C(c1ccc(Cl)cc1F)=CC(N1CCCN(S(=O)(=O)Cc2ccc(F)cc2)CC1)=O C(CCCC(=O)N(CC(C)CNC(c1cn(C)nc1O)=O)C)SC c1(C(=O)NCCCCNC(Cc2c(C)n[nH]c2)=O)cc(C)c2[nH]cnc2c1 c1cc(C)ccc1F.N1(C(C=CCN(CCOC)C)=O)CCOC(CN=[N+]=[N-])C1 Cc1cccc(C(=O)NC2CN(C(c3cccc(CCO)c3)=O)CCC2C)c1Cl c1(CC)ncc(C(N2CC(OCC)C2)=O)s1.C(=O)C(C1CCCO1)C1CC1 c1(C(=O)NC(CSC)(C)C(N2CCC(C#N)CC2)=O)ccc(C#N)c(C)c1 CCC(C)C(C(=O)NC1CC(NC(c2cc(C(F)(F)F)ccn2)=O)C1)OC C1(NC(C=Cc2ccc(SC)s2)=O)COCCN(C(=O)C#CC2CC2)C1 Cc1cc(C(N2CCCC(C)(CNC(=O)C(C)(O)C(C)C)C2)=O)c2nccn2c1 c1(C(N2CC3CN(C(c4c(C)cc(Cl)nc4)=O)C3C2)=O)c[nH]c2cccc(Cl)c12 C(=O)(C(CCC(C)C)NC(=O)CC1=CCCC1)N1CC(C)(COC)C1 Cc1ncc(C(=O)NCCN(CC(C)O)C(=O)Cc2cccc(F)c2)cc1N C1(C(=O)NC2CN(C(c3c(C)c[nH]n3)=O)CC2C(F)F)CCc2ncncc2C1 Cc1cccc(C)c1CC(=O)NC1CN(C(c2ccc(Br)cc2)=O)C2CC12 C#Cc1cccc(C(=O)NC2CCC(C(=O)NC(c3ncc(C)o3)C)CC2)c1 C1(NC(c2ccc(OC)nn2)=O)C2CC3CN(C(=O)C(C)c4ccco4)C1C3C2 CCCCCC(C(=O)O)NC(c1c(C)nc2sccn12)=O c1(C(=O)NCC2CCCCN(C(C(C)C(F)F)=O)C2)ccc2c(c1)CCC2 c1(CC)oc(C(=O)NCCC2CCCN2C(=O)COC2CC=CC2)cc1C C(C(=O)Nc1ccccc1Br)(C(C)CC(C)C)N(C1CCCN(C)C1)CC c1(CC=O)c(C)nc(S)nc1C.c1(C(N(CC)CC)=O)cc(C)c(C#N)cn1 N1(C(C)=O)CCC(C(=O)NCC(C)N(C(=O)CCCc2csc(=N)[nH]2)C)C1 N1(C(C2N(C(CC3C(C)OCC3)=O)CCC2O)=O)CCN2C(=O)OCC2C1 C=C(CNC(c1c[nH]nc1C1CCCO1)=O)CCNC(=O)Cc1[nH]cnc1C C1(NC(c2c(C)nn(C)n2)=O)CCN(C(=O)C#CC2CCOC2)CC(C)(C)C1 CC1(C)CCCC(C(N2CC(n3cc(CNC(c4cn[nH]c4)=O)nn3)C2)=O)O1 C1CC2(CCN(C(=O)CC3CC(F)(F)C3(F)F)CC2)C1.C1(C(=O)N)CC=CC1 c1(C(N2CCCC2)=O)ccc(C(C)(F)F)cn1.C(C(F)(F)F)=CC(=O)N C(CCC(=O)NCc1nocc1C(=O)NCC(O)C(C)O)SC C1(NC(CNC(=O)CNC(c2ccncc2)=O)=O)C(O)CC1O N1(C(C2CCC(C)CC2)=O)CCN(C(=O)C(N2CCOCC2)C2CC2)CC(O)C1 C1(N(C(CN(C2CC2)CC)=O)C)CCCCC1N(C(=O)C(C(C)C)OC)C C1(CC=C)(NC(C2CC3C(C2)C3(C)C)=O)CCCN(C(c2cnn(C)c2)=O)C1 C=C(Cl)CC(C(=O)N1CC2(CC2)C1)NC(C1CCCO1)=O C(c1c(F)ccc(Cl)c1F)=CC(N1CC(F)CC(NC(C(C(C)C)C)=O)C1)=O CP(C)(=O)C1CCCCC1NC(N1CCCC(C2OCCO2)C1)=O c1(-c2cn(C(C(=O)NCC3C(C(=O)OC)COC3)C)nn2)cccc(C#N)c1 CC(C)(C(=O)NC1CCN(C(C2CC2C(F)F)=O)C1)C1CCC1 C1(C(=O)NCCN(C(C)=O)C)(NC2CCC2)CCCCC1 c1ccc(F)c(F)c1.C1(NC(=O)CCc2cscn2)CCC(NC(=O)CS)C1 C(=O)(C(CO)C(F)(F)F)N.c1(CC)ccc(C(=O)N(CC(C)(C)C)C)c(C)c1 C(=O)(C(C)(C)C(=O)NC(C)CC(=O)NCCc1ncn(C)n1)OC C1(CNC(c2cnc(C)[nH]2)=O)CN(C(=O)C(c2ccccc2)O)CC(C)(C)O1 c1(C2(NC(C3CCCN(C4CCC4)C3)C)CC2)ccccc1C1CCC1 CCC(C)CCC(=O)N(C)CC1(O)CCCN(C(=O)CCP(C)(C)=O)C1 CC1CN(C(=O)CCc2ccsc2)CCN1C(C1CC1c1ccn(C)n1)=O Cc1n[nH]cc1C=CC(N1CCC1CNC(C1CCOC1=O)=O)=O Nc1cccc(C(CC2CCC2)N(C(=O)CC(=O)O)C(=O)Cn2cccn2)c1 C(=O)(N=c1cc(C)nc(Cl)[nH]1)c1c(NCCCC)cc(Cl)cc1 C1(c2n(CCC)nnn2)(Nc2cnn(C[Si](C)(C)C)c2)CCOC(C(C)C)C1 c1(CNC(CC#C)C(=O)NC)ccc2c(c1)CC(C)(C)O2 c1(N2CCC(C)C(NC(=O)CC)C2)c(C#N)c(=O)n(C)c(=O)n1C.C(=O)CO.N Cc1cc(C(=O)NC2CC3(C(=O)NCC(C)(C)F)COC2C3)c[nH]c1=N Cc1oc(Br)c(C)c1C(=O)N(C)CCc1cnccn1 N1(C(C=C2CCN(C)CC2)=O)CCCC(F)(CNC(C2CCS2(=O)=O)=O)C1 C(=O)(C(C)(C)C(C)O)NCCCC(=O)NCC#C C1(C(N(CC(=O)NCC(C2CCCO2)O)C2CCC2)=O)CCS1(=O)=O O=C(N=c1cc(C(F)F)cn[nH]1)C1CCCN1Cc1ccc(-n2ccnc2)cc1 C(=O)(C1=CS(=O)(=O)c2ccccc21)NCCCN(C(=O)C)C.C1CCOC1.O c1(C=O)cccc2c1S(=O)(=O)CCC2.N1(C(C=C(C)C(C)C)=O)CCCC1C.N c1(OC)ccc(C2(CC(=O)NC)CCCCC2)cc1.C1(C)CNC(=O)N1C Nc1oc2ccccc2c(=O)c1CN1CCC(CC(=O)O)c2ccccc21 c1(C(=O)NC(CNC(C2N(C)C(=O)OC2)=O)(C)C)nn(C)c2c1CCCC2 n1(NC)cc(CC(=O)NC(=O)CN2CCC(SCC(C)C)C2)c2ccccc12 c1(C=O)sc(-c2ccsc2)nc1C.C1CCC1.C(=O)(C=CC(=O)N)OCC c1(COC(=O)CN2CCS(=O)CC2)nc2ccc([N+](=O)[O-])cc2[nH]1 N1(C(c2n(CC#C)ccc2)=O)CCOC(C(C)NC(c2cncnc2CC)=O)C1 N1(C(CCSCCC)=O)CC(NC(=O)C(C(C)C)OC)CC(O)C1 Cc1nc(N2CCN(C(=O)Cc3cn4c(C)csc4n3)CC2C)c2cc[nH]c2n1 C(=O)(C(CN(C)C)C(C)C)N1CCC(C)(NC(c2c(C)nn[nH]2)=O)C1 CCCCCCC(CC)C(=O)NCCC1CCN(C(=O)CC(C)C)C1 c1(CCNC(NC(C#C)C(C)C)=NC)cc(Cl)ccc1N(C1CCOC1)CC N1(c2nccc(C#N)n2)CCCC1C1CCCCN1C(=O)CC1(O)CCOC1 N1(C(COC2(C)CC2)=O)CC(NC(=O)CC(C)(C)c2ccccc2)C(C2CC2)C1 C(=O)(C(CCSC)NC(N)=O)NC1(CO)CN(C(CC2(C=C)CCC2)=O)C1 C(C(F)(C(=O)N1CCCC2COCC12)C(C)C)NC(Cc1cc(C)sc1)=O C#CCC(C(=O)NCc1occc1C(=O)N)C1CC1.c1noc(C(N)=O)n1 CN=S1(=O)CCN(C(=O)C(C)(C)CCCS(=O)(=O)CCC(F)(F)F)CC1 C1(C)(CNC(c2c(CC)nco2)=O)CCCC1.c1(CC=O)cnn(C)c1.N c1(NC(c2cn(CCO)nn2)=O)cccc(C(N2CC(n3ncc(Br)n3)C2)=O)c1 N1(C(C(C)(C)C)=O)CCC(NC(c2cncc(C(F)(F)F)n2)=O)C(C)(C)C1 C(CS(=O)(=O)CC(=O)N=c1cc2n([nH]1)CC(C)OC2)NC(C)=O n1(C(C(=O)NCC(C)F)C)cc(CC2(CCO)OCCO2)nn1 C(=O)(CC(F)(F)C(F)F)NC1CCC(NC(C=CC2COC(C)(C)O2)=O)CC1 N1(CCC(=O)NC23CN(C(c4c(OC)scc4)=O)C(C2)C3)C(C)CCCC1C C#CCC(O)C(=O)NC1CCC(CNC(c2nc[nH]c2C(F)(F)F)=O)C1 C(CCC(O)C(=O)NCCC12CC(CO1)C2)NC(=O)C=Cc1ccncc1 Cc1cc(C(=O)N(C2CCN(C(C3CCCC(F)(F)C3)=O)C2)C)ccc1C(F)F CC(C)(O)C(F)C(=O)NCc1cccc(CNC(=O)C(O)C2CCCC2)c1 C1(NC(C2CCCC(C)C2)=O)CCN(C(=O)C(F)CC2CC2)C12CCCC2 C1(NC(C2CCC23CCCO3)=O)CNCC2(CCC2)C1 Cc1nc(CC(=O)NC(C)C(C)NC(=O)CCc2nc(C)c(C)[nH]2)c(C)s1 C(=O)(C(C)CC(F)F)N1C(CN(C(c2n(CCCC)ncc2)=O)CC)CCCC1 c1(OC)ccccc1CCC(=O)NC(C)CN(C)C(c1cc(O)nn1C)=O c1(C(N2C3CC(NC(C4CC4(Cl)Cl)=O)C2CC3)=O)c(F)ccc(O)c1F CCCCC(C)C(=O)NC(C)(CNC(c1cn(C2CCC2)nn1)=O)CC(C)C C1(CNC(C2(OCC)CCCC2)=O)CCN(C(C2CC23CC(O)C3)=O)C1 C1(NC(=O)C(c2ccccc2)O)C2CC(NC(C3CC(=C4CC4)C3)=O)CC12 c1(NCC(C)Oc2ccc(OC)cc2)cc(C)cn(C)c1=O C(=O)(CC1C(=O)Nc2c(F)cccc21)NCC(=O)NC1CCCN(C(C)=O)C1 C1(C(=O)N)CCN(C)C1=O.C1(OC)(CN(C(=O)CCC2CC2)C)CCCC1 N1(C(c2cc(C)oc2)=O)CC2CCN(C(=O)CC3CC4(CC4)CO3)C2C1 C1(n2cc(C(C)OC)nn2)(C(=O)NC(CN2CCCC2)C(=O)O)CCOCC1 C1(C(=O)NCCC2CCN(C(Cc3cn(CC)nn3)=O)C2)CCC(=O)NC1 c1(CNc2cccc(C(=O)N=c3cc[nH]cc3F)c2)cc(=O)n2ccccc2n1 c1(OC)cccc(C=CC(N2CCCC(C(C)NC(=O)C3=CCCC3)C2)=O)c1 N1(C(c2cc(C)c(O)c(C)c2)=O)C2CCCC1CN(C(=O)C1=CCCC1C)CC2 C1(NC(c2ccc(F)cc2)=O)CC(NC(C2(F)CCOC2)=O)C(O)C1 C1(CCC(=O)NC2C(C)(C)C2)CCCN(C(=O)COCC2CCCO2)C1 c1(NC(c2n(CC)ccn2)c2nnnn2C2CCOCC2)cccc(COC)c1 C1(C(=O)NCCN2CCN(c3nnc(CCC)s3)CC2)CC1C1CCCC1 N1(C(C(C)C(C)NC(=O)CC2CCCC(=O)C2)=O)CCc2ncn(C)c2C1 O=C1CCC(C(F)C(=O)N(Cc2ccc(O)cc2)CC23CCC(CO2)C3)CC1 C(CC(=O)N(C)CC1CCCCC1)(C1CC1)NC(CN(CCC)C)=O c1(CC)onc(C)c1C(=O)NC1C2CC3C(C2)C13 C1(NC(C2CC(=C)C2)=O)CCCCCN(C(=O)CCC(N)=O)C1 c1(C(NC)=O)ccc2nc(N(C)C)sc2c1.Cc1ccc(C(=O)NC2CC2)o1.C C(=O)(CCC)NCC(=O)NCC(=O)N(CCN(CCCC)C)CC.S C1(C)(CNC(C2CC(C)C2)=O)CCN(C(c2cc(Br)sn2)=O)CC1 c1(C(N2CCC(COC)(NC(C3CCC(=O)N3C)=O)C2)=O)cccn2ccnc12 C12(NC(=O)CCCn3ccnn3)CCN(C(=O)CO)CCC1C2 C1(NC(c2c(CC)nc[nH]2)=O)CCCN(S(=O)(=O)N2CCOCC2)C1 Cc1cc(C)c(C(=O)NC2C=CCN(C(c3[nH]nc4ncccc34)=O)C2)cc1C C(=O)(CCC(C)CC)NC(CCOC)C(=O)N(C1CC2CCC1O2)C O=C1CC2(CCC2)C(C(=O)NCCNC(C2COCC3(CCC3)O2)=O)CN1 c1(NC(C2CN(C(=O)Cc3cccc(Cl)n3)CCC2O)=O)ncc(Cl)cc1F CC(C)(CCCCNC(=O)CCc1nccs1)NC(c1cc([N+](=O)[O-])c[nH]1)=O CN1CC(C(=O)NC(CNC(=O)Cc2ccc(Cl)s2)CO)NC1=O C1(CC)C(NC(c2c(C)ccn2C)=O)CCN1C(=O)CCOCCOC C1(C(N2CC(C)CC(CNC(C(C)=C3CC3)=O)C2)=O)Cc2cccnc2C1 c1(C(N2C(C)CC(NC(c3c(CC)c(C)sc3)=O)C2)=O)cccc(OC)c1OC C1(CC(=O)NCCC(C)CC)CCC(=O)NC1=O.c1(C(=O)N)cn(CCO)nn1 c1(C(=O)NCC(CC)NC(c2ccncn2)=O)cnn(C2CC2)c1Cl C1(C)(NC(c2cnn(C)c2Cl)=O)CN(C(=O)COc2cccnc2)C(C)(C)C1 C#CC(CC1CC1)NC(=O)C(C)c1cccs1 Cc1oc(C(C)C)cc1C(N1CCC(O)(CNC(=O)CS(N)(=O)=O)C1)=O CCCCC(=O)NCCCC(C)NC(=O)CN(C)C(C)=O.OC c1(C(=O)NC2(C)CCCN(C(c3c(C)cno3)=O)C2)ccc(S(=O)C(C)C)cc1 C(=O)(CCCCCN(C)C)N(C1CN(C(c2cc(C(F)(F)F)on2)=O)C1)C C1(C(N2C(C)CC(CNC(=O)C3=COCCC3)CC2)=O)CC2CCCCN2C1 C1(C(N(C(C2CCCCC2)C)C)=O)CCN(C(c2ccc(C#N)cc2)=O)CCO1 C1(CC(=O)N(C(CCNC(C(F)=CCC)=O)C)C)CC2CCC1C2 C1(CNC(C(CC=C)C)=O)CCCN(C(C2CC(C)(C)C2C(F)(F)F)=O)CC1 C(=O)(C(CC(C)C)OC)NC(CNC(CN(C)Cc1ncc(C)o1)=O)CC(C)C n1(CCCC)nc(C(=O)N(C)CCN(C)C(C2CC2C(C)(C)C)=O)ccc1=O c1(C(=O)NC(C)CCCNC(C2CS(=O)(=O)C2)=O)ccc(C2CC2)cc1F C1(CC)CN(C(c2cccc(C(F)(F)F)c2O)=O)CCN1C(=O)CCSC n1(CC(=O)NC2C(NC(C3C(=C)CC3)=O)CC2)cc(C(=O)O)nn1.C CC(C(=O)NCC1CN(C(=O)CC2(C)CCOCC2)C1)C(C)S(C)(=O)=O c1(CC(=O)NC2CCCN(c3ncncc3I)CC2)c(O)ncnc1O CC1CN(C(=O)COCC(F)F)CCC1N(C)C(c1ccc(C2CC2)cc1)=O CN=c1ccc(C(N2CCCC(C(=O)NCC(C)(C3CC3)OC)(CC)C2)=O)c[nH]1 C1(NC(CCS(C)=O)=O)CC2CC(NC(=O)Cc3cncnc3)C1C2 c1(C(CC(=O)NCC(CCC=C)O)C)c[nH]c2ccccc12 C1(C(N(C(C)C(=O)NCC2(C)CC2(F)F)C2CC2)=O)CC2(CCC2O)C1 C1(CC)COCCN(C(=O)CCC2(NC(c3cc(C)nn3C)=O)CCC2)C1 N1(CC(=O)NCC(CC(C)C)NC(=O)C(F)C2CC2)CCCCS1(=O)=O C1(C(=O)OCC)CC(O)CN1S(=O)(=O)Cc1ccsc1 N1(C(c2ccc(C)c(C)n2)=O)CCC2CN(C(=O)CCCn3cccc3)CC2C1 C1(C(=O)NCCS(C)(=N)=O)CN(C(C2CCC(=O)CC2)=O)CC1(C)C N1(C(c2ccc(=N)[nH]c2)=O)CCCC(F)(C(=O)Nc2ccc(CCF)cc2)C1 C1(CCC(=O)N(C2CCC2)C)NC(=O)NC1=O.C1(C=O)(NC(C)C)CC1.N c1(C(=O)NCC(C)NC(COCC=C)=O)cc2nccc(C(F)F)n2n1 c1(C(C)C)cc(CNC(=O)C)[nH]n1.C(C)(C)C.C(=O)CCc1cncs1.O CCCCCC(O)C(=O)NCCNC(c1c(SC2CCCC2)cccc1F)=O N1(C(CCC2C(C)C2)=O)CCCC(CNC(=O)Cn2[nH]cnc2=N)C1 N1(C(CSC)=O)CCC(C2CCCN2C(=O)CNC(c2ccccn2)=O)C1 Cc1ccc(CNC(c2nccnc2C)c2nnnn2C2CC2)c(C)c1 c1(C(N(CCC(=O)NCC(COC)(C)O)C)=O)ccc(=N)[nH]c1 C1(NC(Cc2ccc(C)o2)=O)CC2(CCCCN2C(=O)CC(O)C(C)C)C1 C1(CNC(COC)=O)CC12CCN(C(c1ccc(C(C)C)nc1CC)=O)CC2 c1(C(=O)N)ccc(F)c(F)c1.Cc1csc(C)c1C(N1CCC(OCC)CC1)=O Cc1ccc(C(N2CC3CC3(C(=O)NCC3(C)CCCC3)C2)=O)cc1 c1(CC(=O)NC2C(CNC(C(C)=CC)=O)CC2)ccc(CO)c(C)c1 C1(C(=O)NCC(C(C)C)OC)C=CCN(C(c2oc(C)cc2C)=O)C1 CC1(CNC(c2cccnc2N2CCCC2)=O)CCCN1C(c1cc[nH]c1)=O c1(CCNC(=O)OC(C)(C)C)ocnc1CNS(=O)(=O)CF C1(NC(Cc2cccc(C)c2)=O)CN(Cc2ccc(F)cc2C)CC1(F)F C(=O)(CCCCCOCC)NC1CCN(C(c2cn(CCC)nc2)=O)CC1 N1(C(C(c2ccccc2)SC)=O)CCOC(CN(C)C(c2cnc(C)s2)=O)C1 C12(NC(C3CC4CC3CN(C(C3(F)CC=CC3)=O)C4)=O)CCC(O)(CC1)CC2 CC(C)C(CCNC(=O)C=Cc1ccnn1C)NC(c1cnn(C)c1Cl)=O N1(C(CCC2C(C)C2)=O)CC(CNC(=O)CC(F)(F)Cl)N2CCC1C2 c1(SC(C(=O)OC)Cc2cnc(C)cc2C)nc(C)ccc1O N1(C(C(CCOC)OC)=O)CCC2(CC1)CC2C(=O)N(C1CCCC(C)C1C)C c1(CC)cc(C(=O)NCCC2CSCCN2C(C2CCC(CO)CC2)=O)c(C)o1 c1(C(N(CCCNC(CC=CC)=O)C(C)C)=O)cc(CCC)cnn1 C1(CNC(c2n(CC)cnn2)=O)CCC12CCC2.C(c1scnc1C)=CC=O Cc1c(CNC(=O)NC2CCN(C(C)(C)C)C2=O)cccc1Cl c1(CCN2CCC(NC(c3ccc(CO)cc3)=O)C2)ccc(F)cc1 C#Cc1ccc(C(=O)NCC2CCCC(NC(=O)Cn3nccc3C)C2)c(C)c1 C1(CNC(C(CC=C)OC)=O)N(C(C2CCC(C)O2)=O)CCCC1(C)C n1(CCC(=O)NC(C2CCCN2C(=O)C)C)ncn(C)c1=O.c1nncn1C.S C1(OCC)CN(C(=O)CC2CC2)CC1.c1(C(C=O)(C)C)c(C)noc1C.C C1(C(=O)NC(C)CNC(=O)C(O)CC2CC2)C2CCC3(COC(=O)C13)O2 c1(C(=O)NCC(CNC(C(C2CCOCC2)C)=O)O)ccncn1 CC1CN(c2ccnc(NCC(Cc3ccc(Cl)cc3)CO)n2)CC1C(F)(F)F C(C1Cc2ccccc21)NC(C(C(C)C)NC(C12CSCC1C2)=O)=O CC(C)CC(C(N)=O)N(C(=O)C(=O)NC1CC2CCC1N2)C N1(C(C2(NC(CC)=O)CCC(C)(C)C2)=O)CCN2C(=O)NCC2C1 c1(C(C(=O)NCCSCC)N(CCCSC)C)ccnn1CCF C(=O)C(F)(F)C(F)(F)C(F)F.Cn1ncc(C(N2CCC2)=O)c1C(F)(F)F.C C1(NC(c2cc[nH]n2)=O)CN(C(c2cnc3n2CCCC3)=O)C2(CCOC2)C1 C(=O)(N=c1ncn(CCc2ccncc2)[nH]1)NC(CCCC)C(C)O Cc1cccc2c(C(=O)NCC(C)(C)Cn3cc(C4(C)CC4)nn3)c[nH]c12 O=C1NC(CC(=O)N2CCSCC2CNC(=O)CC23CC(C2)C3)c2ccccc21 c1(C(=O)NCC(CCNC(C(C=C)(C)C)=O)O)cc2nc(Cl)ccc2s1 C(=O)(C(C)(C)CC(=O)N1CC(CCC)C1)OCC.C(=O)C(C)(C)N1CCCC1 N1(C(CC(C2CCCCC2)OC)=O)CCCCC1CCN(C)C N1(C(c2c(Cl)ncc(C)c2)=O)CC2CCC(C1)C2NCc1c(F)ccc(F)c1C C(=O)(CCN(OC)C(=O)C1CC1CNC(=O)CCN1CCCCC1)OC c1(C(N2CCN(C(C3(O)CCCCC3)=O)CC2CO)=O)c[nH]c2ccc(F)cc12 c1(C(=O)NC2C(NC(C(CC)NC(C)=O)=O)CC2)cccnc1O.C(C)=O c1(CC(=O)NC2C(C(C)NC(=O)C(C)(F)F)C2)c(F)ccc(F)c1F N1(C(C(CC)N(C)C)=O)CCCCC1Cn1cc(-c2ccc(C)nc2)nn1 C(=O)(N1OC2C=CC1CC2)C1(CNC(c2c(CC)con2)=O)CC(C)(C)C1 C=CCCCCC(=O)N1CCCC(O)(C(F)(F)F)C1 C=CCN=C(NCCc1nc(C2CC2)no1)N(C)Cc1cnn(CC(F)(F)F)c1 C(=O)(C1CCc2nccn21)NCC(C(=O)NCC(N1CCCCC1)C)N(C)C C1(c2c(CC)n(C)nc2)(CO)CCCN(C(=O)C(C)Nc2ccccc2)C1 c1(C(N(CC(CO)(CO)NC(C2CCOC2)=O)C)=O)ccc(S(N)(=O)=O)cn1 c1(OC)cccc(C(=O)NC(CNC(C2CC(C(F)(F)F)C2)=O)CO)c1 N1(C(C2CC(NC(=O)OC(C)(C)C)(C)C2)=O)CCC2(C1)NC(=O)NC2=O C1(NC(C2(NC(C3CCS(=O)CC3)=O)CC(F)C2)=O)CCn2ncnc2C1 C1(OCCNC(C(C)OCC)=O)CCN(C(=O)C(C2CCCCC2)C)C1 c1(C(=O)NCC=CCNC(C23CCCC(CO2)C3)=O)ccc2nc[nH]c2c1 c1(C(=O)NC2C(CNC(CC(CCC)O)=O)C2)cccc(NC)c1[N+](=O)[O-] CC1(C)CCOC1CC(=O)NCc1ccc(C(N2CC(N=[N+]=[N-])C2)=O)cc1 c1(N2CCCC(=C)C2)nc(N2CCN(c3ccccc3C)CC2)nc2ccsc12 C12(C(N(C3CN(C(=O)CC4CCC(=O)NC4)CCC3O)C)=O)CC3CC1C2C3O Cc1cc(=NCC2CCCCC2NC(=O)Cc2cnoc2)[nH]c(S(C)(=O)=O)n1 C(CC(C(=O)NCC(CC1CC1)CO)NC(c1ccc(Cl)cn1)=O)N(C)C CCCC(C(=O)NCC1(F)COCCN(C(=O)C)C1)S(N)(=O)=O.C(N)(=O)N CCCC(C)(O)CC(=O)N1CCC2CC1CN2C(c1csc(Cl)n1)=O N1(c2ccnc(C)n2)CC(C(=O)N(C2COCC2O)Cc2cccs2)CC(F)C1 c1(C(N2CCC(N(C(CCc3ccc(C)s3)=O)C)C2)=O)cc2n[nH]cc2cc1C C1(CC(=O)NC(c2nn[nH]n2)CC)CCCN(C(=O)Cn2ccc(C)c2)CC1 C(=O)(C(C)CC(C)C(C)=O)N1CCCC(CC(N2CCCC2)=O)C1.CC(=O)N.C Cc1ccc2oc(C(N3CCC(O)C(NC(=O)C(C)P(C)(C)=O)C3)=O)cc2c1 N#Cc1ccc2nc(Cn3ccnc3-c3ccc(-c4ccnc(F)c4)cc3)[nH]c2c1 n1(CC)c(C(N2CC3CCN(C(c4cnn(C)n4)=O)CC23)=O)nc2ccccc12 C1(C2CCCN(C(=O)C(F)n3ccnc3)C2)(NC(=O)CCCN2CCCC2)CC1 N1(C(C2C(C(C)C)(CC)C2)=O)CCC(C2CC2)(CN)CC1 Cc1nc(CCNC(C2CCN(C(=O)CN3CCSCC3)C2)=O)cs1 C1(CC(N2CCCC(CC)C2)=O)C2CCCC2N1C(c1cnco1)=O C1(C(=O)NC(C2C(C(=O)OC)C2)C)C=CCCN1C(C1CCOCC1)=O C(CC(C)(C)C(=O)N1CCCC(n2cc(CNc3nn(C)nc3C)nn2)C1)SC C(=O)(C(C)CC(C)C)N1CCC(CC#C)(C(=O)NC23CC(F)(C2)C3)C1 C=C1CC2(C1)CC(C(=O)N(CCCCN(C(=O)Cc1cnc(C)[nH]1)C)C)C2 CC(CC(=O)N)C(C)(C)C.c1(C(C(N2CCC2)=O)=O)cn(C)nc1C(F)F.C CCCC(C)(C)CC(=O)NC1(C(=O)NOC2CCOC2)CCSC1 C1(F)(C(c2nnnn2C)NC(c2cc(Br)cs2)C)CCCCC1 C1(C(=O)NCC=CCNC(c2cnc(O)s2)=O)CC2(C1)CC21CCC1 C(=O)(CCC(F)F)N(CC(O)CNC(c1nc(Br)c[nH]1)=O)C C1(NC(C2(SCC)CC2)=O)CCC(NC(=O)C(c2ccccc2F)O)CC1 CCC(CC)(CCNC(=O)C(O)C(C)c1ccccc1)NC(c1coc(Cl)c1)=O N1(C(c2cn(C)nn2)=O)CCC2(CCC(NC(c3ccc(CO)nc3)=O)C2)C1 C1(OC)CCn2cc(C(N3C4CCC3CN(C(=O)CC(C)C3CC3)C4)=O)nc2C1 C(=O)(N=c1cc(C2CCOC2)[nH][nH]1)C1N(Cc2ccc(OC)nc2Br)CC(C)C1 N1(C(C(CC(N)=O)NC(c2c(OC)noc2C)=O)=O)CCC2(CCCC2)C1 C12(C(=O)NC(CC)(CNC(=O)CN(C)CCO)CC)CC1COC2(C)C N1(C(C2(C#C)CC2)=O)CC(C2CCCN(C(c3ccc(CCCCC)o3)=O)C2)C1 c1(OC)ccccc1NC(=O)CCC1(C)CCCN1C(=O)CCO.C(N)(=O)N N1(C(c2ncc(C(N)=O)nc2)=O)CC2CC(NC(c3cscc3CO)=O)CC2C1 N1(c2nc(=N)nc(N3CC(C)=C(C)C3)[nH]2)Cc2nncn2C(C)C1 c1(C(=O)NCC2(NC(C3=C(C)CCC3)=O)CCOC2)cccc2nnn(C)c12 O=S(=O)(c1c[nH]ccc1=NCc1cn2ccsc2n1)NC1CCCCN1C1CC1 C(=O)(C1CCCn2ncnc21)NC(C1(O)CCN(C(=O)Cc2cnoc2)C1)C N(C(=NCC1CC1)NCc1ccccc1F)CC(c1cccs1)C O(NC(=O)C(Cc1cnc[nH]1)NC(c1ccncc1N)=O)CCC=C N1(C(CC=CCC)=O)CCN(C(c2cocn2)=O)C(c2ccccn2)C1 C1(OCC)CC(NCCc2[nH]cnc2C)C12CCOCC2 c1(NC(C2C(NC(CCOCCC)=O)CC2)=O)cccc(COC)c1C c1(C(C=O)O)ccc(O)c([N+](=O)[O-])c1.c1(OC)n[nH]cc1C(=O)NC1CCC1 C1(C(=O)NC(Cc2cc[nH]n2)C(=O)NCCO)CC2(CC2)CO1.C1CC1 c1(C(=O)N)ccc(C)cc1O.C(C(=O)NC1CC(C)C1)(C1CCC1)OCC O=C1NC2CCN(C(=O)Oc3ccccc3F)CC2O1 C12(CCS(=O)(=O)N3CC(=CC(F)(F)F)C3)CC3CC(CC(C3)C1)C2 C(F)(C(=O)NCCOCCNC(C1(CCOC)CC1)=O)=CCC N1(C(c2n(C)c3c(c2)ccs3)=O)CC2(CCOCC2)CC1CO Cc1cc(NC(C2CCCC(NCc3cccc4[nH]ccc34)C2)=O)c(F)cc1F c1(CC)ccc(F)cc1C(C)NC(C1OC(C)CC1C)=O c1(CC(=O)NCCCN(C(C(C(CC)(C)C)O)=O)C)ccc([SH](=O)=O)cc1.N N#CC(C(=O)Cc1ccn(C2CC2)n1)c1ncc(Br)cn1 CC1(C)CN(C(=O)CC2(c3ccccc3)COC2)CCC1NCc1ccc(Cl)o1 N1(C(CC2CCCC(C)C2)=O)CCC(C)(NC(C2CC2C(=O)N)=O)CC1.CCO C1(NC(c2n(CC)nc(C)c2)=O)CCCCCC1NC(C1CN(C)CCO1)=O n1(CCC#C)c(N2CCN(CC(F)(F)F)CC2)nnc1Cc1nc(C)no1 c1(C(=O)NC2CCCC(NC(CCCOCC)=O)C2)cccc2nc(C)[nH]c12 CCCC(C)(C)CC(=O)N1CCN(C(c2cnncc2O)=O)CC1CCOC c1(CC)cc(CC(N2CC(C(N3CCC4CC34)=O)(CC)C2)=O)on1 S(=O)(=O)(c1csc(C(C)Oc2ccccc2Cl)n1)Nc1c(C)noc1C C(CC(=O)Nn1cncn1)NC(Cc1c(C#C)cccc1)=O c1(C(C)C)ccc(C(N2C(CNC(=O)COC3CC3)CC3CC23)=O)cc1Cl C(=O)(C1CCCc2c[nH]nc21)N1CCC(C)(NC(C2CSCCS2)=O)CC1 C(=O)(C(C)C(O)C(C)CC)N1CC(SCCC(N2CCC(CCC#C)CC2)=O)C1 N1(C(c2ccc(C3(C)CCO3)cc2)=O)CCOC2(CCN(C(=O)C3CC3)C2)C1 C(=O)(C1=NOC(C)(C)C1)NCC1(NC(C(C)=C(CC)C)=O)CCCCC1C C(C)(CC(=O)NC(C)CN1CCCCC1)NC(C(C)=CC=C)=O c1(C(CNC(C2(C)CCCS2)=O)NC(c2ccoc2)=O)cccc(Cl)c1Cl N1(C(C(CC)=CC)=O)CCC(CN(C(c2cc(C(C)C)n[nH]2)=O)C)CC1 c1(CC(N2CC(C)C(CNC(c3c[nH]c(=N)o3)=O)C2)=O)ccc2ncccc2c1 C1(O)(CN(C)C(c2csc(=N)[nH]2)=O)CCCN(C(C2CCS2(=O)=O)=O)C1 c1(SC)ccc(NC(=O)C(=O)Nc2cscc2C2CC2)c(C)c1 CN1CCC(O)(CNC(=O)C(C2CCCO2)NC(=O)Cc2cnoc2)C1 c1(N2CC(C(C)NC(C3C(C)=C3)=O)OCC2)c([N+](=O)[O-])cnc2ccc(F)cc12 c1(OC)ccccc1S(=O)(=O)N1CCC(NC(c2ccnc(Cl)c2C)=O)C1 N1(CC(=O)OC)CCCN(C(c2sc(C)c(C)c2Br)C(=O)NC2CC2)CC1 N1(C(c2c(OC)ccnc2)=O)CCCCCC1C(=O)NCC1(O)CCN(C)C1 CCC(C(=O)NOCc1cccc(C)n1)N(C)C(C1CC2(C1)CC2(F)F)=O n1(CC(=O)NC(C(C(C)C)NC(=O)C=C2CCC2)C)ccc(O)nc1=O C1(C(=O)Nc2ccc(CC)cn2)CCCC12CCN(C(c1c(C)noc1N)=O)C2 c1(C(N(CC(C)NC(=O)CC(C)(C)CN(C)C)C)=O)ccc(F)cc1Br N1(C(C2CNC(=O)N2)=O)CCCC2(CCCN2C(c2nccc(Cl)c2O)=O)C1 N1(C(CCCCC(C)C)=O)CCC2(C1)CN(C(C1CCSC(C)C1)=O)CCO2 N1(C(c2ccc(CCC)s2)=O)CC(NC(c2ccc(CF)cc2)=O)CC1(C)CC C=Cn1nccc1CNc1cccc(CN2CCCCC2C)c1 c1(C(N2C(C)CCC(NC(=O)C(O)CN(C)C)C2)=O)ccc2oc(S)nc2c1 Cc1nn(CCC(=O)NCCCN(C)C(C2CC3CC3C2)=O)cc1Br Cc1ccc(-n2c(SCCN3CCN(CCF)CC3)nnc2-c2ccco2)cc1 N1(C(CNS(NC)(=O)=O)=O)CCC(NC(=O)C(F)C=O)CC1C.C(C)(C)C.O CC1CCC(C)(C)CN1C(C1CN(C)CCN1C(c1sccc1C#N)=O)=O C1(C(=O)NC(c2noc(C)n2)CC)CCN(C(=O)Nc2cccnc2)C1 c1(C(N2CC(NC(C34CSCC3C4)=O)C(O)C2)=O)ccc(C2CC2)nn1 C1(CC)CN(C(=O)CCc2cccc(OC)n2)CC1.C1(C(=O)N)CCC2(CC2)C1 C1(CC)CCCN(C)C1.c1(C(N(CC=O)CCOC)=O)ncoc1C1CC1.N C(CCNC(c1oc(C)cc1C)=O)(C(=O)NC(c1ncc[nH]1)C)OC N1(C(C=C(C)CNC(c2c(C)ncn2OC)=O)=O)CC(=O)NC2(CC2)C1 C(c1c(C)coc1C)=CC(=O)NC(C1CCCN(C(C2(CC)CCC2)=O)C1)C c1ccc2nsnc2c1.c1(NC(=O)NC23CC(C2)C3)nccc(C(F)(F)F)n1 C(=O)(C(F)C(C)CNC(C1CNC(=O)N1)=O)N1CC2C(CC)(C2)C1 C(=O)(CC(C)NC(N)=O)N(CC(C)NC(c1nocc1Cl)=O)CC CCCCC(C)CCC(=O)N1CCCN(CCNC(C2COCC2(C)C)=O)CC1 Cc1cc(N)c(C(=O)NCC2CCN2C(c2cc(Cl)cc(Cl)c2F)=O)nc1C c1(N2C(C(C)(C)CNC(=O)C(=O)N)CCC2)ncc(C(F)F)cn1.c1ncc[nH]1 Cc1cc[nH]c1C(=O)NCC1CCC1NC(C1OCCC1c1ccccc1)=O c1(C(N2C(Cn3cc(C(C)(C)OC)nn3)CCC2)=O)cn2c(n1)COCC2 C1(NC(=O)C=CCO)CCN(C(=O)CC(=O)Nc2ccccc2O)C12CCC2 c1(C(=O)NC(c2cn(CCCN(C)C)nn2)(C)C)cc(F)c(F)cc1Br N1(C(COCCCC(C)C)=O)CCOCCC1.N(C)(S(=O)(=O)N(C)C)CC=O.N N1(C(c2n(CC)c(O)nc2)=O)CCCC2(NC(c3cnn(CCF)c3)=O)CC2C1 Cc1nc(Cl)ccc1NC(C1CCCCC1NC(=O)CCC(C)(C)F)=O Cc1cc(O)nnc1C(=O)NC1CCN(C(C2CC2c2sccc2C)=O)C(C)C1 C1(OC)CN(C(c2cc(C)n(C)n2)=O)CC1C(N1CCCC(C(C)(C)C)C1)=O c1(N(CC(C)NC(=O)C=Cc2ncc[nH]2)C)ccnc(C(=O)N(C)C)n1 C(c1ccc(Cl)cc1F)=CC(=O)N.Cn1ccc(C(=O)NC(C)(C)CO)cc1=O C=C1CCC(C(=O)NCC2CCCN(C(c3conc3C(F)(F)F)=O)C2)CC1 N12CCCC1C(=O)N(C)CC(C)NC(=O)C2.C1(SCC)(CO)CCC1 Cc1ccccc1-n1nnnc1C1(NC(C)C(=O)Nc2ccccc2)CCOC1 C1(C(=O)Nc2ccc(C(=O)OC)c(Cl)c2)CC2OCCC2N(C(=O)C(C)CN)C1 CC1(C)CN(S(C)(=O)=O)CCC1NCC(C1CCOCC1)O c1(C(N2CCN(C(C34CCC3C4)=O)C(c3cccnc3)C2)=O)cc(=O)cc(Cl)[nH]1 c1(CNC(C)CC(O)Sc2ccccc2)c[nH]c2c(OCC(=O)O)cc(Cl)cc12 c1(C(N2CCCC(CCNC(C(C)c3ccsc3)=O)C2)=O)ccc(F)c(Cl)c1F c1(C(N(C(C)CNC(C2CCCC(CF)C2)=O)C)=O)cncn(C)c1=O c1(C(N2CC(C(=O)NCC(F)(F)F)C2)=O)c(-c2ccccn2)nc2ccccn12 c1(C(=O)NC2CN(C(CC(CC)(C)C)=O)C(C)(C)C2)cc(C)c2nc(C)nn2c1 C1(C(=O)NCCN(C(=O)C(C)C2CC2)CCOC)CCc2c(nnn2C)C1 N1(C(CC2CCCN(C)C2)=O)CCCC(C(=O)Nc2ccc(N(C)C)cc2)CC1 C1(CC(N2CCCC2)=O)CCCNC(=O)C1.C1(C=O)CS(=O)(=O)C1.CCO C12(NC(C(N3C(CC)CCC3)=O)=O)CC1CN(C(c1cccc(C)n1)=O)C2 C1(C)(CC)C=C(C(=O)N2CCC(C(C)C(=O)Nc3ccc(F)cc3C)CC2)C1 C1(NC(=O)C=CCO)CN(C(c2ccc(C3CCCO3)[nH]2)=O)CC2(CC2)C1 N1(C(c2c(CCCC)ocn2)=O)CC(NC(=O)C(C)COCC)CC(C)(C)C1 c1(N(C)Cc2cscc2Br)nc2c(c(=NC3CSc4ccccc43)[nH]1)COCC2 C1(NC(c2c(CC)con2)=O)CCCCN(C(C2CCCC(C#N)C2)=O)C1 N1(C(C2CCCN(CC)C2)=O)CCC(F)C(NC(=O)C(C(C)O)N(C)C)C1 C(=O)(C(CNC(C1CCN1C)=O)N(C)C)NC(c1cc[nH]n1)C c1(C(=O)NC2CN(C(C3CC(SC)C3)=O)CC2F)cn2ccc(F)cc2n1 CCCC(C(=O)OC)C(=O)NCC(C)CNC(=O)CC(O)CCC C1(C2CC2)(C(N(CC#C)C)=O)CN(C(=O)C(C)C=C=C)C1 C=Cn1nncc1C(=O)NC1(CCOC)CCN(C(C2(C)CCCOC2)=O)C1 C(=O)(C1=Cc2ccccc2C1)NC1(C)CCN(C(C(C)OCC)=O)CC1 N1(C(c2cc(C)no2)=O)CC2CCCCC2(CNC(c2cccc(Br)c2)=O)C1 N1(C(C(C)NC(CC)=O)=O)CCSCC1CCNC(=O)CSCC(=O)O c1(C2CCC(NC(=O)NC3CCC(=O)NC3)CC2)ccc(Cl)c(Cl)c1 C1(NC(c2c(SC)csc2)=O)CCCCC1NC(=O)CCCc1ccc(N)cc1 C1(CC=C)(C(=O)NCc2cnnn2C)CCN(C(=O)CCN(CC)CC)C1 C1(CNC(C2N(CC)CC2)=O)CC(C)CCN1C(=O)C.c1c(C)cccc1C N1(C(=O)NCCC2CC(CC)C2)CCc2c(Cl)cccc2C1 c1(NC(CCC)C)ccc(S(=O)(=O)NC(c2cccc(Br)c2)CC2CC2)c(Br)c1 O=C(C(CC(F)(F)F)c1ccc(F)cc1)NC1CC(NC(=O)C(F)=CCCF)C1 n1(C(CC)CC(C)O)cnc2c(N(c3cccc(F)c3C#N)C)ncnc12 C(=O)C1=CS(=O)CCC1.C1(C(C)(C)C)CCCN1C(=O)CC1CC(F)(F)C1.N C1(CC=C)(NC(=O)CC2COC(=O)C2)CCN(C(c2cccnc2F)=O)C1 N1(C(C(C)CC(F)F)=O)C2CCC1CC(C(=O)NC1(C)CCC(=O)N(C)C1)C2 C(=O)(N=c1[nH]nc2[nH]ccnc1-2)C1N(C(c2c(Br)ccc(C)c2)=O)CCCC1 C1(NC(C(C2CCN(C(c3c(CC)ocn3)=O)C2)(C)C)=O)C=C(C)CCC1 C1(NC(c2c(COC)nn(C)c2)=O)CCCN(C(=O)CC2CSCCS2)CC1 N1(C(CCC2(NC(=O)COCCF)CCCC2)=O)CCCC2(CCCO2)C1 Cc1sc(O)nc1C(=O)NCc1cc[nH]c1C(=O)N(C1C2CCCC12)C C12(C(=O)OC)CCCCCC1N(C(c1c[nH]c3nccc-3c1C)=O)CC2 c1(C(=O)OC)ccc(C#CC(=O)N2CCC(C(N3CCCCC3)=O)CC2)cc1 C(=O)(CC1COc2ccccc21)N(C(C)CNC(=O)COC(F)F)C c1(C(C)C)ccc(C(=O)NC)c(O)c1.C1COCCN1C(=O)C(F)CC1CCC1 C(=O)(CCCC(=O)C1CC1)NCC1CC(O)(CNC(CC2C(C)C2)=O)C1 N1(C(c2cn(C(C)(C)C)nn2)C(=O)NCC)CC(O)C(O)C1C(=O)OC Cc1cc(NC(C2CCC(C)(C)N(C(=O)C=CC(C)C)C2)=O)cc(C)c1F C(=O)(CCC(CC)CCC)N1CCC(O)(CNC(C2(C#C)CCCCC2)=O)C1 c1(CC(=O)NC2C=CCN(C(CC(C(=C)C)O)=O)C2)c(C)cc(Br)cc1C C1(C(=O)NC(C)CC(C)O)(COC)CN(C(c2ccc(Cl)o2)=O)C1 CN1CCN(C(=O)CSc2ccc(CNc3cc(OC)ncn3)cc2)CC1CF c1(C(=O)NCCC2CC(NC(C3NC(=O)OC3)=O)C2)ccc([N+](=O)[O-])cn1 C(=O)(CC(C(F)F)c1ccccc1)NCCN(CC(C)O)C(c1ccc[nH]1)=O C1(NC(Cc2cc(C)n(C)n2)=O)CCCC12CN(C(c1ccnc(CO)c1)=O)C2 n1(CCCN2CCCC(Nc3c(OC)c(Cl)ncn3)C2)nc(C)c2cccnc12 N1(C(C2C(CC)CCN2C(c2csc(C)c2C)=O)=O)CCC(N(C)C)C(C)C1 S(=O)(=O)(c1cnn2ccc(=NCCCOC3CCCCC3)[nH]c12)NC1(C)CCC1 C1(COC)CCCN1N(C)C1CCc2ccc(C)cc21 N1(C(c2n(C)ccc2)=O)CCCC(O)(CNC(c2cnc(N)s2)=O)C1.C1CC1 N#Cc1cc2cc(C(N3CC(NC(=O)C=CCO)C(O)C3)=O)[nH]c2cn1 C1(NC(=O)CCn2cnccc2=O)CC(O)CN(C(c2cc(O)cc(Cl)c2)=O)C1 CCCCCC(=O)N(CC(=O)NC1CCCC1C(=O)OC)CCC C(=O)(CC(C(F)F)C(C)(C)C)N1CC(C)C(NC(c2c(F)ccnc2F)=O)C1 C(=O)(C=O)NCCN(C(=O)C(C)c1ccon1)CCOC.CC(F)(F)F Cc1cccc(OCC(=O)N(C2CCC(NC(=O)C(C)(Cl)Cl)CC2)C)c1C N1(C(c2ncc(N(C)C)nc2)=O)CCC2C(CCN2C(C2C(Cl)(Cl)C23CC3)=O)C1 Cc1cc(C)c(C(N2CC3OCC(NC(=O)C4=CCCCCC4)C3C2)=O)cc1N C1(C(N(C2CCCN(C(=O)Cc3ccon3)C2)CC)=O)CC12CC(F)(F)C2 CCCCCCC(=O)NCC(C)NC(=O)CCCc1cc(C)sc1C C1(C(N2C3CN(Cc4c(OC(C)C)cccc4)CC32)=O)CC(=O)NC(=O)N1 Cc1cc(CN2CC(NC(=O)C(C)Cc3ccc(F)cc3)C(O)C2)cn1C c1(C(=O)OC)ccnc(C(N2CCOCC2C)=O)c1.C(=O)CN(C)C(N)=O N1(C(C2C(C(C)C)CN(C(C3(C)CCN(C)C3)=O)C2)=O)CCC2CN(C)CC2C1 c1(CC)occ(C(F)(F)F)c1C(=O)N(CCC)C.C(c1ccccc1)=CC=O C12(C=O)CCCC(CO1)C2.C(=O)C(C)CC1CC1.n1(CC)ccc(CC)n1.N C1(NC(C(CCC=C)NC(=O)C(C2CC2)OCC)=O)CC(C2CCCC2)C1 CCC(F)C(=O)N(CC(=O)Nc1ccc(S(=O)(=O)NC)cc1)OC N1(c2snc(C(=O)OC)n2)CCCC(CCNC(=O)Cc2cn(CC)nn2)CC1 c1(C(=O)NCC2CCCC(NC(c3cccc(C)c3)=O)C2)ncc(Cl)cc1F C1(CC(=O)N(C(CC)C)C)CCN(C(C2CNC(=O)C2)=O)C1(C)C C1(OCC)CC(NC(=NCCc2ccc(N(C)C)nc2)NCC(C)C)C12CCC2 C=CCCC(C1CC1)NC(=O)CSCCNC(=O)CO.C1CC=CC1 N1(C(C2(C)CC2(F)F)=O)CCC12CN(C(C1CC(F)(CF)C1)=O)C2 C(=O)(CCCNC(=O)CSC1CC1)N1C(C(N(C)C)=O)CC1 c1(CC)cccc(C)n1.CCC(C(=O)NCC1CC1CC=O)NC(N)=O.N C(c1ccc(Cl)cc1)=CC(=O)NCC(CC(C)C)NC(c1c(C)scn1)=O C#CCC(C)(C)NC(C1C(CNC(=O)CCCOCCO)C1(C)C)=O C(=O)(C(C)(CC)C(N)=O)N.N1(C(c2cc(C(CC)CC)no2)=O)CC(F)CC1C CCCC(CC)CCC(=O)NC(C(=O)N(CC(O)COC)C)c1cccs1 C(=O)(C1CCCc2c1ncn2C)N1CCC2(CN(C(C)=O)C2)CC1 N1(C(CS(N)(=O)=O)=O)CCCC2C1CCCN2C(c1cnccc1Cl)=O C(C1CCN(C(c2ccsc2Cl)=O)CC1)=CC(=O)NC(CC)(C)CO c1(SC)ccc(N)cc1C(N1CC(C(C)NC(=O)C)C1)=O.CC(C)(C)C.O CCC(C(=O)N1CCC(CC2CCN(C(=O)C(C)CCOC)CC2)CC1)C(C)C N1(C(C)=O)CC(C(=O)Nc2n[nH]c(C3CC3)c2Br)C(C2CC2)C1 C1(NCC(=O)NCC=C)CCCCC1NC(c1ccoc1)=O C(CC1CCC1)(C(=O)NC(Cc1cc[nH]n1)C(=O)NCCCCO)OC S(=O)(=O)(c1cccnc1NCCC(C)(C)CO)NC(C(OC)OC)C N1(C(C2C(CCC)C2)=O)CCN(C2CN(C(=O)C=CSC)C2)CC1 c1(C(=O)NC(c2cncn2C)C)ccc(C2(C)CCO2)cc1F c1(-n2cc(C(CCC)=O)nn2)cc(C(=O)NC2CCOCC2(C)NC)ccc1C C1(C(C)C)CN(C(=O)CC2CCN(CCc3ccc(F)cc3)C2)CCO1 Cc1nc2ccc(C(=O)NC3(CNC(C4CCC4C)=O)CC3)cc2n1C C1(NC(Cc2n(C)ccn2)=O)CCCN(C(c2cc(-c3ccn(C)n3)on2)=O)C1 S(=O)(=O)(c1cccc(=NCC2CC2C)[nH]1)NCc1cc(OC)no1 N1(CC=CC(=O)NC2CCN(C(C3CCC(=O)O3)=O)C2)CCOCC1 c1(C(N2CCC(N(C(COC(C)C)=O)C)C(C)C2)=O)cn(C)c(=O)c2cncn12 Cc1cc(C(=O)NCC2(O)CC(C)C2)cc(C)c1C.c1(C=O)cccc(N)c1 N1(C(CN2CC(C)(C)C2)=O)CCC(C2CCN(C(c3ccc(F)cc3N)=O)C2)C1 CCCCC(CNC(=O)C(C)(C)C1CC1)NC(C1(C)CCN(C(C)=O)C1)=O c1(C(N2CCC(O)(C(N3CCOC(CO)C3)=O)C2)=O)cnccc1Br Cc1cc(C(F)F)nn1CC(=O)NCC(C)N(C)C(C1CCOC(C(C)C)C1)=O C(=O)(C1CCCc2c[nH]nc21)NC(CNC(C1=CCN(C)C1)=O)CC(F)(F)F Cc1cc(O)ncc1C(=O)NC(C1CC1C(=O)N(C)CC1CCSC1)C CC(C)(CC#N)C(=O)NCC(CNC(c1ccc[nH]1)=O)S(C)(=O)=O CN1CC(C(=O)NC2C=CCN(C(=O)Cc3ccc(Cl)cc3Cl)C2)CCC1=O c1(N(C(c2ccc(C(C)(C)C)s2)C=O)C)ccc(C)cc1C.C(C)OCC.N c1(C(=O)Nc2cc(C(=O)OC)ncc2)cc2n(n1)CCCN(S(=O)(=O)CCCl)C2 C1(CNC(Cc2c(C)occ2)=O)CCC(NC(c2snc(O)c2Cl)=O)CC1 C1(NC(c2c(C(C)C)scn2)=O)CC2CN(C(=O)CCCn3cccn3)CC2C1 C(CC(=O)NCc1cnc(OC)cn1)(C(C)(C)C)NC(CCC(CC)C)=O c1(CC)cccc(C(=O)NCC2CCN(C(C3CCS(=O)CC3)=O)C2(C)C)c1N C1(C(=O)NC2CN(C(CC(=O)NC)=O)C2)(C(=O)OC)CC1S(C)(=O)=O CC(=O)C(C)CC(C)C(=O)NCc1csc(C(=O)N(C)Cc2ccoc2)c1 C1(C)(CNC(c2c(CC)noc2C)=O)CCN(C(c2cnn(C)c2Br)=O)CC1 CC1CN(C)CCN1C(c1cncc(Br)c1)C(=O)NCC1CCOCC1 CCC(CC)C(F)C(=O)N1CC(C(=O)NC2CC(n3cncn3)C2)C(C(C)C)C1 O=C(CCCCCF)NCC1CCN(C(=O)C(c2ccc(Br)cc2)O)C1 c1(CC(=O)NC2CCC2NC(c2ccn(C3CC3(F)F)n2)=O)ccc(O)cc1 N1(C(c2c(SC)cccc2)=O)CC2CC(C1)C2NC(=O)CC(O)c1ccccc1 CCCC(C(=O)N1CCCCC1CCNC(c1cc(C)nnc1O)=O)S(N)(=O)=O C1(O)(CNC(C2CC(CNC(C(C)OCOC)=O)OC2)=O)CCN(C)CC1 C1(O)(CN(C(C2C(C)C2C)=O)C)CCCN(C(c2cnnc(O)c2)=O)C1 C1(NC(=O)C#CC2CC2)CCN(C(C2CC3CC2C3)=O)C(c2ccccc2)C1 N1(C(CC(CNC(C(C)CC2CCC2)=O)(C)C)=O)CCN2C(=O)CCC2C1 Cc1cc(C(N2CCC3(NC(=O)CCOC4CC4)CC3C2)=O)cc(C)c1Cl c1(C(=O)NCCCCCNC(c2n(C)cnc2)=O)c(C(C)(C)C)nsc1N c1(CC)cc(C(=O)NC(CCOC)C(=O)NC2CCCC2(C)N(C)C)ccn1 CC1Cc2c[nH]nc2C(C(=O)NC2CC(CNC(=O)CS)C2)C1.c1cccs1 C(=O)(C(C)(C)CC(C)=O)NC1CCC(NC(C(C(CC)C)OC)=O)CC1 Cc1cc(C(=O)NC2CCCCC2CC(=O)Nc2ccc(C3CC3)cc2)n(C)n1 c1(C=O)c(F)ccc(F)c1Cl.C(CC(=O)N(CC)C1CC1)C(N)=O.CC=O.N c1(C(N2CCCC(n3cc(CCC(=O)O)nn3)C2)=O)c(Cl)nc2ccccn12 C(=O)(CCCC(C)=O)NCCCN(C(=O)C(C)CC1CCCC1)CCC C(=O)(C(F)(F)SC)NCCN(C(COCCCC)=O)CC.C(N)=O c1(C(=O)NC2CC(NC(c3c(CC)csc3)=O)C2)cc(Br)c(C)s1 Cc1cc(F)c(C(N2CC(O)CC2COc2ccc(Cl)cc2)=O)cc1Cl C(=O)(C1=CC2CCC=CCCC12)N1CC(NC(CCCOC)=O)C1 N=c1[nH]c2c(s1)CC(NC(=O)C(=O)NCc1ccc(N3CCCC3)nc1)CC2 C1(C(=O)NC2(CCCNC(=O)C=Cc3cocn3)CC2)CC1C1CCCC1 Cc1cc(C(=O)NCC2CCN(C(=O)CO)CC2C)nc(C)c1.C1(C)CCCC1 CSC1=C(C(=O)NC(C)C(C)NC(=O)C(C)(C)CC#N)CCCC1 C1(CC(=O)N(CC)C(C)C)CCNCC1.CCCCC1(C=O)CC1.C1CC1 C1(NC(COC(CC)C)=O)CCN(C(c2cc(C(N)=O)cn2C)=O)C1C Cc1ncsc1C(=O)N(CCC(C)NC(C1(CO)CCCO1)=O)C C1(NC(C(C=C)(C)O)=O)CCN(C(C2COC(=O)N2)=O)CCC1c1ccccc1 Cc1ccc(C(=O)NC(C)CNC(=O)CN(S(C)(=O)=O)C)c(O)c1C CCC(CC(=O)NCC(COC)NC(=O)C(c1cnn(C)c1)O)C(F)F C(=O)(CC1=CCN(C)CC1)NCC1CN(C(c2ccc(C)s2)=O)C2(C1)CCC2 N1(C(c2nn(C)c(=O)cc2)=O)CCN(C(=O)Cc2cccc(F)c2)C2CCC12 C1(C(=O)NCc2nnnn2CC2CCOCC2)(CC)CCCC1 c1(C(=O)NCC2N(C(c3n(CC)ncn3)=O)CCOC2)cc(F)cc2nc[nH]c12 C12(CNC(c3n(C=C)nnc3)=O)CCC(C(=O)OCC)(CC1)CO2 C1(C(N2CC(NC(C)=O)C2)=O)CN(C(=O)CCC=C(C)C)CC1F C1(CNC(c2c(Cl)cn(CC)n2)=O)CC2(CC2)CN1C(C1CCCC1C)=O CS(=O)(=O)c1csc(C(N2CC3C(NC(c4csnc4Cl)=O)C3C2)=O)c1 CC(C)C(F)(CNC(c1ccccc1O)=O)C(=O)NCC1(O)CCCC1 c1(C(=O)N)cc(F)cc(N)c1F.c1(C(=O)NCC(C)C)c[nH]nc1-c1cccs1 N1(C(CCCSC)=O)CC2(CCCC2)C1.c1(C=O)cc(S(=O)(=O)N(C)C)c[nH]1.N c1(C(=O)Nc2cncc(C(=O)NCCc3cccc(Cl)c3)c2)cc(I)cnc1Cl CN1CCOc2ccc(C(=O)NCC3C=CCN3C(=O)C=CCF)cc21 O=C(C1Cc2ccc(Cl)cc21)NCC(O)CNC(C1CC(n2ccnc2)C1)=O CCCCCC(F)C(=O)N1CCCC1C1(C(=O)N(CCC(C)CCC)CC)CC1 CC(CC#N)C(=O)NC(CCSC)C(=O)NCCc1cc(O)ncn1 N1(C(c2ccc(OC)cc2OC)=O)CC(C(=O)O)C2(C1)CN(C(=O)CO)C2 CC(C(=O)N1CC=CC1CNC(c1cccc[n+]1[O-])=O)C(C)(C)O CCCC(C)C(=O)N1CCC(CCNC(C2(C)CC(C)(C)C2)=O)C1 c1(C(C)NC(c2c(C)csc2)=O)ccc(C)cc1.c1(CC(=O)N)cn(C)nn1 C(=O)(C(CNC(=O)Cc1ccn(C)n1)CC1CC1)NC(C#C)C(C)C CC(CC(=O)N)CC(C)C.C12CC(C1)C2.C(=O)(C(C)CC1CCCO1)CCC.C N1(C(C)=O)CCC(CCCCCNC(=O)C(=CC2CCCCC2)F)CC1 N1(C(C(COC)O)=O)CCC(C2CCN(C(=O)CCc3ncccn3)C2)CC1 C1(CNCC(c2ccc(Br)cc2F)O)CCC12CC(F)(F)C2 N1(C(Cn2c(C)ncc2)=O)CCCC(NC(c2cccnc2O)=O)C1C Cc1nc(=N)[nH]cc1C(=O)N(C)C.C1CCN(C(=O)CC2SC(=N)NC2=O)CC1 C1(NC(c2c(OC)nccc2)=O)CCN(C(c2ccc(C)[nH]2)=O)C1(C)C C1(CNC(c2ncoc2-c2ccccc2)=O)C2CCCC1N(C(=O)CO)C2 c1(C(N(C2CCN(C(C(CC)(C)F)=O)CC2)CCO)=O)ccc(OC)c(Cl)n1 CCCC(C(=O)NC(c1nc(C)cs1)C)NC(c1cnnc(C)c1)=O N1(C(C(C)NC(=O)OC)=O)CC2CCCC2(F)C1.c1(C(=O)N)nc(Cl)oc1C c1(C(=O)NCCCN(C(c2cnc(O)s2)=O)CC)cn2ccccc2n1 CCCCC(CC(=O)N1CC=CC1CN(C)C)NC(=O)C(C)(C)CCF n1(CC(=O)NCC2CCCN2C(C2COC(=O)O2)=O)cc(Br)ccc1=O C1(C)(C(=O)NC(CCCNC(C(C)(C)OCC)=O)C)CC(C#N)C1 C1(CC(=O)NC(c2nnc(C)s2)C)CCCN(C(C2CC(=O)C2)=O)CC1 N1(C(CNC(C(CC)C)=O)=O)CC2CCCC2(NC(c2sc(CO)nc2C)=O)C1 C(N=c1nc(N2CC(C)N(C)C(C)C2)c2cccc(F)c2[nH]1)c1cnc(CC)[nH]1 C(=O)(CC(C)CC(C)C)NC(CC)CNC(C1CNC(=O)CC1C)=O c1(CCC(N2CCC(NC(CCCC#N)=O)(CO)C2)=O)ccc(F)cc1F N1(C(C(c2cccs2)NC(Cc2n(C)cnn2)=O)=O)CCC(O)CC(C)C1 c1(NC(C2N(C(C3(C)CC3)=O)CCOC2)=O)cc(-c2ccccc2)ccc1Cl N1(C(CC2CCC(OC)CC2)=O)CCN(CC(c2ccccc2)C)C(C)C1 c1(C(=O)OC)ccnc(N2CCN(C(C3CCC(F)(F)CC3)=O)CC2)c1[N+](=O)[O-] Cc1ncc(Cl)c(C(=O)NC(C)CN(C)C(c2ccccc2C2CCOC2)=O)n1 C#CC1CCCC1NC(C1CC(O)CN1C(C1CC1OC(C)=O)=O)=O N1(C(CCCOC)=O)CCC2CN(C(C3CCCC(C)(C)O3)=O)CC2CC1 CC1=C(C(=O)N2CCCOC(CNC(C3(C)CC(O)CN3C)=O)C2)CCC1 C(=O)(C1CCCn2cncc21)N(CCNC(c1c(C)n(CC(F)(F)F)nc1)=O)C CC1(CCCCNC(c2cccc(CN3CCCCCC3)c2)=O)NC(=O)NC1=O C(=O)(CCCCCC#N)NCC1(C(=O)NC2CC(C)N(C3CC3)C2)CC=CC1 N1(C(CC2(C)CCOC2)=O)CC(C(=O)N)C(C2CC2)C1.C1(Cl)CC1(F)F c1(N(CCc2nc(CC)sc2)C)nc(=NC(C)c2scnc2C)[nH]c2c1CCC2 C(=O)(C1CCc2nccn21)NCC1N(C(c2n[nH]c(C)c2Cl)=O)CCN(C)C1 Cc1nc(O)c(Br)cc1C(=O)NC(C)CN(C(=O)CC1NC(=O)NC1=O)C CC1CCCCC1CC(=O)NCC1(CC(=O)NCC2(CCCO)CC2)CC1 C1(CC)CN(C(c2csc(-c3cccs3)n2)=O)CCN1C(=O)C(C)CC(N)=O C1(C(=O)NC(C(C)C)CCN(C)C(C2CC(O)C2)=O)(CF)CC2(CCC2)C1 c1(CC(=O)Nc2c(C)cncn2)c[nH]c2nccc(Cl)c12 C1(C(=O)OC)C2CCC(O2)C1C(=O)N.C1CCN(C(=O)CC2CCCO2)CC1 c1(CNC(C2(CNC(=O)C(F)OC(F)(F)F)CCCC2)=O)ccccc1.C C1(F)(C(=O)NCC(CC)(C)O)CCCN(C(=O)CC2(C#N)CC2)C1 c1(C(N2CCN(CCC(C)(C)C)CC2)C(=O)NCCOC)cc(Br)c(OC)cn1 C=CC(C)(C)CC(=O)NC1(CO)CCN(C(c2cncc(COC)c2)=O)C1 N1(C(C2C(CCC)C2)=O)CCC(C)CC1.c1(C=O)ccc(OC(F)(F)F)nc1.N C(=O)(C(CCC)S(N)(=O)=O)N1CC(N(C(CCOCCC)=O)C)C(C)CC1 c1(C(N2C3CN(C(CCC=C=C)=O)C(C3)C2)=O)[nH]c(C)c(S(N)(=O)=O)c1C C(CCCCNC(=O)C=C1CCOCC1)N(C(C1C(CCC)C1)=O)C(C)C C(C)(CO)(C(=O)NCC1CC(C(=O)NCCCN2CCCC2C)CO1)OC Cc1ccc(CNC(C2COCCC2NC(C2CCCCC2)=O)=O)c(O)n1 CC(F)(F)CCCC(=O)N1CCC(NC(c2cnc(S)nc2)=O)C(C)(C)C1 N1(C(c2cc(CCC)[nH]n2)=O)CC(NC(C2(c3ccnn3C)CC2)=O)CC1C c1(C(N2CCN(CC(C(=O)OCC)(C)C)CC2)=O)cccc(Cl)c1F c1(NCc2n(CC)ccn2)ccc(S(=O)(=O)NC2CCC(C3CC3)C2)cc1Br c1(CC)c(C=O)nn[nH]1.C1(C(N(C2CCC2)C)=O)CC(O)CN1C(C)=O.N C1C2CC3C1C3C2C(N1CC(O)C(C)(C)C1)=O.CC(C)CCCOCC(=O)N c1(C(N2CCC(O)(C(C)NC(CCC)=O)CC2)=O)c(Cl)nc2ccccn12 N1(C(CC(C=C)(C)C)=O)CCOCC(F)(CNC(c2c(OC)cccc2C)=O)C1 C1(CN(C(CNC(COCCCOC)=O)=O)C)OCCC1(C)C.C1CC1.C C1(NC(C(c2ccccc2C(F)(F)F)C)=O)CCN(C(C2CCC2)=O)CC1CO CC1CC(NC(c2ncoc2CNC(c2ccn(C(F)F)n2)=O)=O)CCN1C N1(C(CC2NCCC2)=O)CCN(C(=O)CC2(N(C)C)COC2)C(C(C)C)C1.CC c1(C(N2C(C)(CCOCCO)CCC2)=O)cc(Br)ccc1O c1(C(c2nnnn2CCCF)(CC)NC2CCCC2F)cccc(OC)c1OC Cc1ccc(CNC(=O)C(C)N(C(=O)C#CC2CC2)C2CC2)c(F)c1 C1(O)(CC)CCC(NC(C2(NC(=O)CCCC3CCCC3)CC2(C)C)=O)CC1 CCCCCC(C)(C)C(=O)NCc1ccc(CNC(=O)C(F)C(C)(C)O)cc1 C(Cc1cn[nH]c1)(C(=O)N(C)CC1COC(=O)N1)NC(CSCCCC)=O c1(NC(C2(C)N(Cc3ccc(C(=O)OC)cc3)CC2)=O)cccc2cn(C)nc12 CC1CCCC(C)N(C(=O)CC2C=CC(NC(c3ccc[nH]3)=O)C2)C1 Cc1cc(CN2CCCC(C(C)NC(C3CCC(=O)N3)=O)C2)cc(C#N)c1 C1(SCC)CCCC(N=c2cc[nH]cc2S(=O)(=O)NCc2ccc(SC)nc2)C1 C1(O)(CC)CCN(C(c2cscc2C(F)F)=O)C1.CN(S(N)(=O)=O)CC=O.N c1(NC(C2C=CCN2Cc2cc3cc(Cl)ccc3s2)=O)c[nH]c2nccc(Br)c12 Cc1cc(C(N2CCN(C(=O)C(C3(O)CCCC3)F)CC2CF)=O)cc(C)c1O c1(NC(C2CC3CC3N2)=O)cncc(F)c1 C1(NC(=O)Cc2cscn2)CN(C(=O)CCn2cccnc2=O)C2CC12 c1(CC(=O)NCCN(C(C(CCC)OCC)=O)CC(C)O)cc(O)ccc1Cl C1(CNC(C(C(C)O)NC(C23CCCC2C3)=O)=O)CCC2(CC1)CC2 N1(C(c2c(C)nn(C3CC3)c2)=O)CCN(C(C2CC(OC3CC3)C2)=O)CC1.C CC1CCN(C(=O)CC2CC(=O)NC(=O)C2)CC1.C1(O)(C(=O)N)CCC(C)CC1 c1(CN(C)C)cn(C)nc1C(=O)NCCCN1CCN(Cc2ccon2)CC1 CCC(CCCC(=O)NOCCC1CC1)NC(=O)C(O)CC(C)(C)C C(C)(CC(C)C(F)F)NC(C(CC=CC)NC(C1(C=C)CCC1)=O)=O N1(C(C)=O)CCCC(C(=O)NCC2C(CC(=O)Nc3cncnc3C)C2)C1 C(=O)(C(C)(C)CF)NCC1(CN(C(=O)C2=CCCC2)C)CC1 C(=O)(C1CCCc2nn(C)cc21)NC1CC(F)(CNC(CS(CC)=O)=O)C1 CN1CCC(C(=O)N2CCN(c3cc(O)cc(O)c3)CC2)c2ccccc21 C1(CC(=O)NC(c2nccn2C)C)(NC(C2OCCO2)=O)CCCCC1 C1(NC(=O)CCC(F)F)CN(C(C2CSCCS2)=O)C2CCCCC12 C1(NC(c2c(OC)nsc2)=O)CCCC(N(C(=O)CCc2cnoc2)C)C1 CC1CC(C(=O)NC2CN(C(=O)CCN3CCN(C)CC3)C2)C1(C)C Cc1cccc(OCC(=O)NC(CNC(=O)C(=O)C(C)(C)C)CO)c1C c1(SC)nn(C)cc1C(=O)NCCCCCN(C)C(C1CCN(C)C1C)=O c1(CC(NOCC(=O)NCc2n(CC)ncn2)=O)ncn(C)c1C C(=O)(C(C)(C)C(F)(F)F)N1CC2C(C(F)(F)F)(C1)C2.CCC(=O)NCC=O C1(C(N(CC(F)(F)CO)C)=O)CCN(C(C2(C)CCCCC2)=O)CC1O C(=O)(CCc1cnoc1)N(CCOC)C1CC1.C1(=O)CCC2CC(C2)N1 C12(CNC(c3c(CC)scn3)=O)CC(CO1)N(C(c1[nH]ncc1C#N)=O)C2 c1(CNC(C2(C#C)CCCCC2)=O)ccc2ccc(O)nc2n1 C1(CNC(C(C)C2CCCO2)=O)CCCC2(CN(C(C3(O)CCOC3)=O)C2)O1 C(=O)(C1=CCCCCC1)NC1CCN(C(C(C)c2cc[nH]n2)=O)C1(C)C C1(CCC)CCN(C(c2cnc(C(N)=O)s2)=O)CC1.c1(C(=O)N)cc(C#N)cs1 C1(CNC(C2(COC)CC2)=O)CCC1(C)C.c1(C=O)cc(C)sc1C.N N1(C(CC2(N(C)C)CCC2)=O)CCN(C2CN(C(=O)CN3CCCCC3)C2)CC1 C(=O)(C=CSc1nc[nH]n1)NC(C)CN(C(=O)CC1CC1C(F)(F)F)C CC1(C)CC(C(=O)NCC23CC(CCO2)C3)CCO1.c1(C(=O)N)ccncc1F N1(C(C=NOC)=O)C2CCC(C2)C1CC(=O)NCCC(=O)N(C(C)C)C1CC1 c1(-c2cn(CC3CCCN(CCC)C3)nn2)cc(C)cc(C)c1.C(=O)C(C)C(=O)O c1(CC(=O)NC2CCC(NC(CN(CCC#C)C)=O)CC2)cn2c(C)csc2n1 N1(C(C2(C)CCOC2)=O)CCC2(CC1)CCN(C(c1cc(Cl)c(F)c(Cl)c1)=O)C2 c1(C(=O)NC2CC(CNC(CCCOCC)=O)C2)ccc2nnn(C)c2c1 C1(NC(NNC(=O)Cc2cccc(F)c2)=O)OC(=O)CC12CCC2 N1(C(C2(C)COC2)=O)CC2(CCCC2NC(c2cc(O)cc(O)n2)=O)C1 c1(C(=O)OC)cnc(N(C(C)CNC(=O)COc2cccnc2)C)nc1 N1(C(c2cnn3ccccc23)=O)CC2(C1)CN(C(C1CC=CCO1)=O)CC2CO c1(C(N2CC(CCNC(COCC#C)=O)C2)=O)cnn2c1OCC(O)C2 C1(CNC(=O)Cn2cnnc2O)CN(C(=O)CC2CCCC2(F)F)CC12CC2 Cc1c(Cl)ccc2cc(OCC(N3CC(c4ccccc4)CCC3=O)=O)cnc12 CC1(C)CCCC(C(=O)NCCCC2CCCCN2C(=O)C2=CCCCO2)C1 CC1(C)CC(C)(CNC(c2coc(Cl)n2)=O)CN1C(c1cc(CO)on1)=O C1CN(C(c2ccc(N)c(F)c2)=O)C(C)(C)C1.c1(SC)cnn(C)c1C(=O)N Cc1ccc(O)cc1C(=O)NCc1ccccc1CC(=O)NC1CNC(=O)C1 c1(CC)cccc(C)c1C(=O)N.C(=O)(CCC(N)=O)N1CC(F)C1.C(C)=O CS(=O)c1ccc(C(=O)NC2CC2NC(c2ccc(Cl)c(O)c2)=O)cc1 N1(C(C(C)=C(CC)C)=O)C2CCC1CN(C(C1CCCS1(=O)=O)=O)C2 C1(NC(C2CCO2)=O)CCC(NC(c2csc(Cc3ccccc3)n2)=O)CC1 CC1(C(N2CC(C(N3CC(c4ccncc4)C3)=O)C(F)C2)=O)CCCCO1 C(=O)(C(F)(F)CF)NC(C)CNC(=O)CC(C)n1ccnc1 n1(CC(=O)NCCNC(C(c2ccccc2O)OC)=O)nc(C)oc1=O C1(C(C)NC(CN(C(C)=O)C)=O)CCCN(Cc2nc(C)c(C)o2)C1 N1(C(c2cc(CCC)ncc2)=O)CC(F)(F)CC1CC.c1(C(=O)N)cc(C)sn1 C(=O)(C1CN(C)C(=O)c2ccccc21)NCC(C)N(C(c1c(C)coc1C)=O)C n1(CC)nc(C(=O)N(C2CCN(C(=O)Cc3cnc(C)[nH]3)CC2)C)c(C)n1 CC(C)(Cc1cnn[nH]1)C(=O)NCC(C)CO.C(=O)CC(C1CC1)C1CC1.N Cc1cc(C(=O)NC2CN(C(=O)CN3CC(=O)NC3=O)CC2C(F)F)ncc1F CC1CN(C(c2ccc(CNC(=O)C=CC3CC3)o2)=O)C(C)CO1 c1(OC)ccccc1NC(=O)COCCF.C(C1CCCN1C)=CC=O.CC N1(C(c2ncn(C)c2)=O)CC2CCCC2(NC(=O)Cc2c[nH]c3ccccc23)C1 C1(CNC(C2(CC#C)CCCCO2)=O)CC2(CCC2)CN1C(=O)CCC(C)OC C1(C(=O)NCCN(C)C(c2nnc(O)nc2O)=O)Cc2ccccc2C1(C)C C1(NC(C2(NC(CCN(C)CCO)=O)CSC2)=O)CCOCC1F N1(C(C=C(CC)C)=O)CCN(C(c2ncsc2CC)=O)CC1C1CC1 CC12CCC1(C)CN(C(C1(C3CCCN3C(=O)CC3C=CCC3)CC1)=O)C2 N1(C(C2(NC(c3cnc(C)o3)=O)CCC(C)(C)C2)=O)CCCC2(CCC2)C1 C1CN(C(=O)C(C)(C)C2CCOCC2)CC(C)(C)C1.CC1=NOC(C(=O)NC)C1 N1(C(C2N(C(c3ccc(C)o3)=O)CC=C2)=O)CCC(O)(C(F)(F)F)CC1 Cc1cnn(C)c1CC(=O)N(C)CCNC(C1CC(N(C)C(C)C)C1)=O N1(C(c2ccc(CC=C)cc2)=O)CCC(C)(C(N2CC3CC3C2)=O)CC1 c1(NC(=O)CNS(=O)(=O)Cc2ccccc2)ccccn1 Cc1cc(C#N)ccc1C(N1CCSCC1C(=O)NC)=O.C1(O)CCC(C)(C)C1 CC1=C(C)CN(C(c2cc(CNC(=O)Cc3n[nH]c(C)n3)cs2)=O)C1 C(CCCCNC(=O)CC1CCCOCC1)(OC)OC c1(NC(=O)NC(C)C(c2ccccc2)N)cc(Br)c(Cl)cn1 N1(C(C2CC(C)(CC)C2)=O)CC2CCC1C(NC(c1ccnc(Cl)c1O)=O)C2 N1(C(C(C)(C)N(C)C)=O)CC2(CCC(CNC(c3cc(O)nn3C)=O)O2)C1 CC1(C)COC(CC(N2CCCC2C(=O)NCC2C3COCC23)=O)C1 c1(C(=O)NC(CNC(CCC(=C)Br)=O)(C)C2CCC2)cc(C)nc(O)n1 CC1C(=O)CC1C(=O)NCCC1CN(C(=O)C)C1.C1(CC=O)CCCC1 Cc1cc(NC(=O)CC2CC(O)CN2C(=O)CCc2ccoc2)cc(C)c1 C1(CCNC(c2ccns2)=O)CCCN1C(C1CCCC1c1nc[nH]n1)=O C1(CCC)(C(=O)S)CC(=O)C1.n12cc(nn1)CN1CCC1C2.c1ccccn1 Cc1ccc(C)c(SCC(N2CCCC2C2(O)CN(C(c3cnc[nH]3)=O)C2)=O)c1 c1(-c2nnc(N(C3CCCCC3)C)n2CCC#N)ccc2c(c1)OCO2 N1(C(c2ncccc2F)=O)CCC(NC(C2(CO)CCC2)=O)CC1C1CC1 CC1CN(C(c2ccccc2)=O)CCC1CNC(c1cc2n(n1)CCC2)=O C1(C(=O)NCCc2ncc(C)o2)CCCC(NC(=O)CC=C(Cl)Cl)C1 c1(C(=O)NCC(CC)NC(c2cc(C)cc(N)c2)=O)c(C)ncnc1O C=C(C)C1OCCC1C(N1CC(C)(OCC(=O)NCC(O)CN(C)C)C1)=O c1(CC(=O)N(c2cccc(OC)c2)C2CCOCC2)cnc2n1CCCC2C N1(C(C2(C(=O)NC)CC2)=O)CCCC(C2CCN(CC3CCCCC3C)CC2)C1 C12(CNC(C3(C)CCOC3)=O)CCC1CN(C(=O)CN1C(=O)CNC1=O)C2 C1C(C)(C)CC1(C)C.c1(NC)cc(C(=O)N)cc(Cl)n1.c1(CC=O)cc[nH]n1 Cc1cc(P(C)(C)=O)oc1C(=O)NCC(c1ccc(C(F)(F)F)cc1)C C1(CCNC(C(N2CCOCC2)C)=O)CCCCN1C(c1c(Cl)cnn1C)=O C(C)(C(=O)NCC1CC1)(c1ccccc1)OC(C)C.CCC(C)C.C(=O)C C1(NC(C2(CC)CCNC2=O)=O)CCN(C(=O)CC2(O)CCCC2)CC1F CC1CCCC(OCC(=O)NC2CCN(C(=O)CC(F)F)C2C)C1 N1(C(CCSCCCC)=O)CC2(C1)CN(C(=O)CC1CN3CCC1CC3)CCO2 c1(C(C(=O)NC(C)C(=O)OC)N(CC)CC2CC2)cc(I)n(C)n1 Cn1cc(C(N2CCCC(C(N3CC(O)CC3(CO)CO)=O)C2)=O)ncc1=O N1(C(CCCC)=O)CCN(C(c2cnn(C)n2)=O)C(C2CC2)C1 C1(C(=O)NC2CN(C(c3n(CC)nnc3C)=O)C2)COc2ccc(OC)cc2C1 N1(C(Cn2c(C)nnn2)=O)CC2CC(NC(C3CC3(C)C(F)F)=O)C(C2)C1 N1(C(CCC(CC)C)=O)CCCCC(C2CN(C(C3CC=CC3)=O)C2)C1 C(=O)(C1=NOC2(CCC2)C1)NC(CCOCC)C(=O)NC.C1CC(C)=NO1 N1(C(C(C)(C(C)C)OC)=O)CC2CCC1C(CNC(c1cncc(O)c1)=O)C2 C1(C(=O)N(NCC)C)CN(C=O)C1.C1CCC(C)C1.C(C)(C)C.CC N1(C(C(C=CCCC)O)=O)CCC(F)(c2cn(Cc3csc(Cl)n3)nn2)CC1 C1(NC(C(C(C)C)N2CCCCC2)=O)CCN(C(=O)CN(S(C)(=O)=O)C)CC1O Cc1ccncc1CC(=O)NC(C)CCCCNC(C1CC1c1cnn(C)c1)=O C1CCN(C(c2csc(O)n2)=O)CCC1(F)F.c1(CC)cc(C(=O)NC)n(C)n1 c1(C(CNC(c2cc(Br)no2)=O)NC(C23CCC2CC3)=O)ccccc1 C1(CC=O)CC2(CCC2)CO1.CC(C)(C)CCNC(=O)CC(=O)N.C1CC1 N1(C(C2CC(=C)C2)=O)CCC(C)CC1CNC(=O)CC(c1cccc(F)c1)C Cc1nc2c(C(N3CC4CC(NC(c5ccnnc5)=O)C3C4)=O)cccc2o1 N1(C(C2(C)ON=C(C)C2)=O)CCCC(F)(C(=O)NCC#CCCO)C1 N1(C(C2(CC=C)CCOCC2)=O)CCC2(C1)CN(C(C13CCCC1C3(F)F)=O)C2 C1(CC(=O)N(CCCNC(=O)C(F)CC(C)C)CC)CC2(CCOCC2)CO1 N(C1c2ccccc2CC1(F)F)C(=O)NCC(C#C)O N1(C(c2cc(C)ncn2)=O)CC(C)CN(C(c2cc3ccccc3s2)=O)CC1C C12(C(=O)N(S(=O)(=O)Cc3ccccc3)CCO)CCC(O1)c1ccccc12 N1(C(c2c(C)nsc2)=O)CCC2(COC(CNC(=O)C3=CCCS3)C2)C1 c1(C(N2CC(NC(C(CC)(C)O)=O)C(n3cccn3)C2)=O)cc([N+](=O)[O-])c[nH]1 c1(C(N2CCC(C(=O)NCCC3N(C)CCC3)C(O)C2)=O)cn2ncccc2n1 C1(COC)(NC(=O)C(F)OC)CCN(C(c2cc(F)ccc2OC)=O)CC1 N1(C(c2cnc(-c3ccsc3)s2)=O)CCC(N(CCO)C(c2ccoc2)=O)C1 C(CC(C)CCNC(=O)CSc1nncs1)NC(c1c(N(C)C)coc1)=O Cc1c(C(=O)NC)nnn1-c1cnn(C)c1.C1CCC1.N1(CC=O)CC=CC1 c1(C(=O)NCCC23C(CN(C(CNC(N)=O)=O)C2)CC3)cc2cccc(F)c2o1 c1(CN(C=O)C)ccc(C(C)C)cc1.C1(N(C(=O)NC)C)CC2CC2C1 N1(C(c2ccc(C(=O)OC)[nH]2)=O)CCC(C)C(NC(=O)CC2(O)CCC2)C1 N1(C(Cc2ncc(C)o2)=O)CCC(C2CC2)C1CNC(C1CCOCC1)=O N1(C(C(CCNC(CC(C=C)C)=O)(C)C)=O)CCn2c(C)nnc2C1 C(c1ccc(C(N)=O)o1)=CC(N1CCC(NC(c2ccn(C)c2)=O)C1)=O C1(NC(C2CC3CC2C2CC32)=O)CC2CC(C1)N(C(=O)C1=CCCCO1)C2 C1(NC(CSCC=C)=O)CC12CCC(NC(=O)C(F)(F)c1cnccn1)CC2 C1(NC(COCC(=O)OC)=O)CCC(C)N(C(=O)CCCC2CCOCC2)C1 c1(CC(=O)NCC2N(C(c3c(CC)noc3)=O)CC2)cn[nH]c1.C1CC1 CCN=S(C)(=O)c1ccc(NC(=O)C(=O)NCC(C2CCC(C)(C)CC2)C)cc1 N1(C(c2nc(C)c(Br)s2)C(=O)NCCCF)CC(C)Oc2ccccc21 Cc1[nH]nc(C(=O)NC2CCCCC2NC(c2ccc(Cl)s2)=O)c1C(F)(F)F Cn1nnnc1CCNC(C1(n2cc(CCF)nn2)CC1)=O.C(CO)C C(CCC(CO)NC(c1cscn1)=O)NC(C1C(CC)OCC1)=O N1(C(Cc2c(C)scc2)=O)CC(C2CCCN(C(C3CCC(C)(C)OC3)=O)C2)C1 CC(C(=O)NN=c1nc(-c2cccc(Cl)c2)[nH]o1)C(F)(F)CC(=O)N(C)C Cc1noc2ncc(C(=O)NC3CN(C(=O)C(C)C(F)F)CC3C(F)F)cc12 C(CCNC(c1cc(C)ncn1)=O)(C(=O)N(CCCO)C)OC CN=c1[nH]cc(C(=O)N(CC(C)NC(C2CC2c2ccc(F)cc2)=O)C)o1 C1COC(C)(C)CN1C(=O)CCCCC1CC1.c1(SC)ccc(C(=O)NC)cc1 C(C(O)(CNC(=O)CNC(C1CCOC1)=O)CO)OC N1(C(=O)Cc2csnn2)CC(C2CCCN(C(c3ccc4nncn4c3)=O)C2)C1 c1(OC)ncccc1CC(N1CCCC(CNC(=O)COc2ccsn2)C1)=O c1(C(=O)NC2CN(C(CCCC#CC)=O)CC3C2C3)c(C)[nH]c2ncccc12 CC1CC(=O)NC(C(=O)NCCN(C)C(c2cnc(Cl)[nH]2)=O)C1 C1(C)(CC)C=C(C(=O)NCCCC(C)NC(c2ccc(C3CC3)nc2)=O)C1 CCCCC(C)CCC(=O)NC1CCN(CCNC(=O)C(C)CF)CC1 CN1CCC(CC(=O)NCC2OCCO2)(C(=O)O)CC1 CC1COc2ccc(C(N3CC(NC(c4ccccc4OC(F)F)=O)C3)=O)cc21 Cc1cc(C)cc(C=CC(N2CC3C(N(C(=O)C(C)C(C)(C)C)C)C3C2)=O)c1 c1(C(=O)NC2(C)CC(NC(C3(c4nccs4)CC3)=O)C2)cnc(Cl)cc1N c1(C(=O)N)nc(Cl)ccc1N.CCC(C(=O)NCc1ccccc1)N(CC)CC CCC(C)CCC(=O)NCCC1(C(=O)Nc2cccnc2CC)CCC1 c1(C(N2CC(CCNC(=O)Cc3cncs3)C2)=O)ccc2cc[nH]c2c1F C#Cc1ccc2c(=NC(=O)CCCF)nc[nH]n12.C(CCCOCC)O N1(C(CCC2(NC(=O)C(F)n3ccnc3)CCC2)=O)CCCC(CF)C1 c1(CNC(C2C=CCC2)=O)cn(C2CCN(C(=O)Cc3ccsn3)C2)nn1 N1(C(CC(C)(C)C)=O)CCN(C(c2cc(Cl)cc(Cl)n2)=O)C(C#N)C1 c1(C2(CNC(c3scc(C(=O)O)c3)=O)CC2)cccc(Cl)c1F C(=O)(C1=CCC(C)CC1)N1C(CC)C(C(N2CC(OC(=O)CC)C2)=O)CCC1 c1(CCCC)nc(C)c(CC(=O)NC2C3CN(C(c4ccc(=O)oc4)=O)CC23)s1 Cc1nc(C)n(CCC(N2CCCCC2CN(C)C(C2CC(C)(F)C2)=O)=O)n1 c1(C(=O)NC(C(C)NC(C(=Cc2ccc(Br)o2)C)=O)C)ccc(=O)n(C)c1 C(=O)(C(C(=O)NCC#CC(=O)NC(C)C(C)C)OC)OC N1(C(CC2CCCN(C(c3n[nH]c(=N)[nH]3)=O)C2)=O)CCC2(CCCO2)CC1 c1(OC)nc(OC)nc(N2C(C(=O)Nc3cnc(C)c(Cl)c3)CC3CC23)n1 N1(C(c2c(C(C)=O)cn(C)n2)=O)CC(C2CN(C(c3ccc(CO)nc3)=O)C2)C1 N1(C(=O)C2=C(Cl)CC2)CCN(C(=O)CN)CC(O)C1.c1cc(Cl)ccn1.C(=O)CO c1(N2CCC(COC)C2)ccc(S(=O)(=O)NCC(C)COC)c(Cl)c1 C1(C#N)(C(N2CCC(CN(C(C3C(C)C3C)=O)C)CC2)=O)CC2CC2C1 O=C(C1=CC2CCC(C1)C2)N1C2CCC1C(C(N1CCc3ccsc3C1)=O)C2 c1(C(=O)NCCCN(C(C(C=CC)O)=O)CCO)cc[nH]c1C.C(C)=O.N C1(N(C2CN(C(=O)C(c3cc(Br)cs3)N(C)C)C2)C(C)=O)CCC(F)CC1 c1(COC)ncc(NC(=O)C(=O)NCC2CC2[N+](=O)[O-])c(C)n1 C#CC1(C(N2CCC2C2CCCC2)=O)CCN(C(=O)C=Cc2nccs2)C1 CCCCS(=O)(=O)CC(=O)NCCCCCCNC(C1CN(C(N)=O)C1)=O C(=O)(CC(CCCC)NC(=O)CCc1cccs1)N(CCOCC=C)C Cc1ccc([N+](=O)[O-])cc1CNC(=O)C(=O)NC1CC1c1ccnn1C CCC1=C(C(=O)NC(C)CCC(N2CC3CC(CO)C(C3)C2)=O)CCCO1 N1(C(C(CCCCC)(C)CC)=O)CC(C)OC2(CCN(C(=O)CCC(C)O)C2)C1 CC(CN(C(=O)C(c1ccco1)NC(=O)CCC1(C)N=N1)C)CO N(C(=NCCc1cccc(C)n1)NC1CC1)CCOC(N(C)CC)=O c1(C(CO)NC(=O)NC2C(O)(C(=O)OC)CCC2)ccc2ccccc2c1 N1(C(C2(OC(C)C)CCOC2)=O)CCCCC1CNC(c1cc(Cl)cn1C)=O CCS(=O)(=NC(=O)Cc1ccc(C(=O)OC)o1)C1CCCCC1 N1(Cc2cccc(OC(C)=O)c2)CC2CCC1CN2C(c1n[nH]cc1Br)=O C(=O)(CCCC(=O)N1CCN(C(=O)C(C)(C)C(C)C)CC1C(F)F)OCC c1(C(NC2CCN(C(=O)CC3CC3)C2)=O)ccc(N(C)C)cc1.C(C)=O CCCCCCCCCC(C)CC(=O)N(CCNC(=O)CN(C)CC)C(C)C c1(C2C(C(=O)NCC)C2)ccc(OCC)cc1 N1(C(CC=C(C)C)=O)CCC(OCC)CC1.c1(C(=O)N)cc(C2(C)CC2)on1 Cc1ccc(C(=O)NCC2(C(N3CCCC(O)(CO)C3)=O)CCC2)c(O)c1 Cc1cc(C(N2CC3C(CNC(=O)CCOC4CCOC4)C3C2)=O)c(C)n1C c1(C(=O)NCCc2cccc(OC)n2)cc(S(N)(=O)=O)ccc1Cl N1(C(Cc2c(C)nc[nH]2)=O)CCC(NC(=O)CC2CCCC2C)C(F)C1 C(=O)(C(C(C)(C)C)SC)NCc1ccc(CCNC(C(C=C)(C)O)=O)cc1 N1(C(C(=O)NC(CS(C)(=O)=O)CO)CCC(N)=O)C(=O)c2ccccc2C1=O CCCCC(C(=O)NC(CCO)C(C)C)NC(c1nnc(S)n1C)=O C=CCC(CNC(c1coc(C(N)=O)c1)=O)C(=O)NC1CC(=O)N(O)C1 C1(CC(=O)N(CCCCO)CC)CCCN(C(c2ccc(F)cc2C)=O)CC1 S(=O)(=O)(c1ccc(Br)c(F)c1)N1C(C(=O)Nc2cnncc2Br)CC(O)C1 Cc1cc(C(N2CCN(C(=O)C=CC3CC3)C3CC23)=O)cc(C)c1F C(=O)(C(C)C(O)C(C)C)NCCCC1CCN(C(C2=C(C)OCC2)=O)CC1 N1(C(C(CCNC(C2C(CC(C)C)C2)=O)(C)C)=O)CC(C)OC(C)(C)C1 c1(C(=O)NCC(CNC(c2c(SC)cccc2)=O)C)ccc2c(c1C)CCC2 N1(C(c2ccc(C(C)(C)C)nc2)=O)CCC2(CCN(C(=O)Cn3cccn3)C2)C1 C1(CC(=O)NCCCN(C(=O)Cc2cnns2)CC)COCC1(C)C C(=O)C(C)S(=O)(=O)C(C)C.n1(CC(=O)NCCCCCC)nc(C)n(C)c1=O C=Cc1ccc(N2CCCC(C(=O)NC(C(=O)OC)C(C)O)C2)nc1 C12(C(=O)NCC(C)CC3CC3)CC1CN(C(=O)CN1CCCC1)C2 S(=O)(=O)(c1cccc(C(=O)NC2CCCCCN(C(=O)C(O)C3CC3)C2)c1)NC N1(C(C(CC(N)=O)NC(CC(C)SC)=O)=O)CCCN(C)CC1C c1(C(N2CCN(C(C(CC)COC)=O)CC2CC(F)F)=O)ccn2c1CSCC2 C(C(O)C(=O)N1CC(C(N2CC(C(=O)NC)C2)=O)(SC)C1)=CC C1(C(N2CCN(C(CC(CC)(F)F)=O)C(C(F)F)C2)=O)CCOC2(CCCC2)C1 CC1(C)COC(C(=O)NCC(=O)NCCCC2CCOC2=O)C1 N1(C(c2c(C(C)C)noc2)=O)CCOC(C(=O)N(CC(C)(O)C2CC2)C)C1 c1(C(=O)NC2C(CNC(CCCCCOC)=O)C2)cccc2c1COC2 c1(C(c2n(C)nnn2)NCc2nnnn2C)cc2ccccn2n1.C1(Cl)CC12CCC2 C(=O)(C1=C(C)OCCS1)N1CCCC(N(C(c2sc(CC)c(C)c2)=O)CCO)C1 C1(C(N(C2(C#C)CC2)C)=O)CC(F)(F)CN1C(=O)C1=CC(C)(C)C1 c1(NC2CC(CC(N3CCc4n[nH]cc4C3)=O)C2)ncc2ccsc2n1 N1(C(C2C(NC(c3c(CC)n(C)nc3)=O)CCC2)=O)CC2(CCCO2)C1 c1(C(N2CC(NC(C3(O)CCC3)=O)C2)=O)ccc2cccc(F)c2n1 c1(C(N(CC(C)NC(=O)CC2(C(=O)O)CC2)CC)=O)sc(C)cc1C n1(CC)ncc([N+](=O)[O-])c1C(=O)NC1CCC1.c1(C=O)cn(C)c(=O)cn1 C(CC(CC)C(=O)NC(=O)CC=CC(C)(C)C)=CC c1(CNC2CCC(C(=O)Nc3cc(C)no3)C2)cccc(-n2cncn2)c1 O=C(CCC(=O)c1ccc(F)cc1)NC1CN(C(C2CCCCC2F)=O)C1 C(=O)(C(C)CS(C)(=O)=O)NCC1N(C(c2ccc(C)c(C)c2)=O)CC(C)(C)C1 CC1(C)CC(C(=O)NCc2ccc(F)c(O)c2)CN1C(=O)CO.CC(F)F C1(C(N(C(C#C)C)CCCC)=O)CCC(NCc2csc(C)n2)CO1 c1(CC(=O)NCCCNC(c2ccc(C3CCOC3)s2)=O)ccc(F)c(F)c1 C(=O)(CCS(=O)(=O)N(C)C)N(CC(CNC(c1c(C)noc1N)=O)O)C c1(CN2CC3(C(C(=O)Nc4cn(C)nc4)C3)C2)cc(O)ncc1Br C1(CC(N2C(C(=O)Nc3c(C(=O)OC)n[nH]c3)CC2)=O)COc2ccccc2O1 C(=O)(NNc1ncc(Br)c2ccccc12)NCC1N(C)CCOC1 C1(CC=C)COCC1NC(=O)CCOC1CN(C(C2(C)CC2(F)F)=O)C1 C(=O)(C1CCc2cc(F)ccc21)NC(CNC(C(C(=O)NC)(C)C)=O)(C)C N1(CC(OC)OC)CCC(C(F)(F)F)C(CO)C1 c1(C(=O)NC(C(C)C)CC)cc([N+](=O)[O-])n[nH]1.c1(C=O)ccnc(C2CC2)n1.N c1(N2CC(NC(C(C)NC(N)=O)=O)C2)ncnc2c1ncn2CC(F)(F)CO C1(CNC(c2cnns2)=O)CCC(NC(c2scnc2C(F)F)=O)CC1 Cc1cc(C(=O)NCC2CCN(C(c3cc(C(C)C)[nH]n3)=O)C23CC3)ccc1Cl c1nc2nccnc2s1.N1(C(CNC(=O)OCC)=O)CCCC1C.C1CC1.N C1(C(=O)NC2(C)CCCN(C(=O)CCC3CCCC3)C2)Cc2cccc(F)c2O1 c1(NC(=O)CC2CCCN2Cc2c(Br)cncc2Br)cnc2ccc(F)cc2c1 C1(C2CCCN(C(C3CC4CC4C3)=O)C2)(NC(CC(CCOC)(C)C)=O)CC1 c1(C(N2CC(C(C)C)CCC2C)C(=O)NCCOC)cnc(C)cc1OC C1(C)(NC(CSc2c(NC(=O)OC(C)(C)C)cccc2)=O)CCC12CCC2 c1(N(C2CCN(C(C3CCN(C)CC3)=O)C2)C)nc(Cl)ncc1F C1(N(CC#C)C(C2CC2C)=O)CCN(C(C2(CCOC)CCC2)=O)CC1 C(=O)(CCC1=NNC(=O)CC1)NCC(CC)(C)NC(C1Cc2nnc(C)n2C1)=O C(=O)(CC(F)F)NC(CNC(C(C1CCOCC1)OCC)=O)CC CC1CCC(C)(C(=O)NC2CCN(C(c3cncc(F)c3)=O)C(C)C2)CC1 C1CN(C(=O)CN(C2CCC2)C)CC(C)(C)C1.c1(C(C)C)ncc(C(=O)N)o1 C1(NC(C(C2CC(F)(F)C2)OC)=O)CC2CCC(C1)N2C(c1ccoc1C)=O C1(NC(c2ccoc2Cl)=O)COC2(CCCN(C(=O)C=Cc3cccs3)C2)C1 C1(C(N(CC(C)OC)CC)=O)CCN(C(c2cnn(CCF)c2)=O)C1 c1(C(=O)NC2C3CC(NC(c4ccn(C(C)C)n4)=O)CC32)cc(N)ccc1Cl c1(CN2CCN(C)C(c3nc(C4CC4)no3)C2)ccc(S(=O)(=O)C2CCC2)cc1 Cc1ccc(C(CNC(=O)C(CO)N(C)C)NC(c2ccc(Cl)s2)=O)cc1 C(=O)C(C(F)(F)F)C(F)(F)F.C1(NC(COc2cc(C)on2)=O)COCCC1.N CCCC(CCC)C(=O)NC(C1CCCN1C(c1c[nH]ccc1=N)=O)C N1(C(C2CN(C(c3c(C)oc(C#N)c3)=O)CC2(F)F)=O)CCC2CCNC(=O)C12 c1(CC(=O)NCC2CC2NC(c2ncncc2F)=O)ccccc1Cl C12(CNC(C(N)=O)=O)CCCC1N(C(C1CCN1C1CCCC1)=O)CCC2 c1(COC)nc(NCCOc2ccccc2)cc(=NCCc2nnc(C)n2C)[nH]1 N1(C(c2cc(CCC)[nH]n2)=O)CCOC2CN(C(C3(F)CCCC3)=O)CC12 c1(OC)ccc(CC(=O)OCC2(C)CCSC2)c(Br)c1OC N1(C(C(C)Oc2cccnc2)=O)CCC(CO)(NC(=O)CN(C2CCC2)C)C1 CC1CCC(C)N1CC(=O)N(CCCC(=O)Nc1cccc(C2CC2)c1)C C(=O)(C(CCS(C)(=O)=O)NC(c1c(OC)c(Br)ccc1)=O)N.C(C(C)C)SC Nc1ccc(C(N2CC=CC2CNC(c2sccc2Cl)=O)=O)c2ccncc12 C1(C(=O)NC(C#C)C2CC2)CN(C(c2c(C#N)cnn2C)=O)CC1(C)C c1(C(=O)NCC2(C)CCCC2)ccccc1N(C(=O)C(F)(F)F)C1CC1 C1(CNC(CC(C=C)C)=O)CN(C(c2ccn(C3CCC3)n2)=O)CCC12CCC2 C(C(C)(C)CCO)NC(CN(C(=O)Cc1cncnc1)CC#C)=O N1(C(CC(C)SC)=O)CC2CC(NC(=O)C(F)(F)c3ccccn3)C(C2)C1 C#CC1(C(=O)N(CC(C)CNC(=O)CSC)C)CC(=O)C1 c1(C(N(C)CCNC(=O)CC(F)F)=O)ccc2c(n1)NCCO2 c1(C(=O)NC2C(C)CCN(Cc3cnc4ccnn4c3)C2)cccc([N+](=O)[O-])c1 N1(C(C(c2ccc(OC)cc2)C)=O)CCCC(C2CCN(C(C3CSC3)=O)C2)C1 C(CCN(C)C(C1CCCC1)=O)(C(C)(C)C)NC(C(C)OCC=C)=O C1(CC)CCCC1(C)C(=O)NCCC(C)OC c1(OC)ccnc(F)c1C(=O)N(C1CCN(C(=O)CCc2ccc(C)cc2)C1)C C1(NC(c2c(C)nns2)=O)CC(NC(C23CCC(C2)C3)=O)C12CCOCC2 Cc1csc(=O)n1CC(=O)NCC(C)(O)CNC(=O)CCCc1ccccn1 Cc1nnc2n1CCCN(Cc1c[nH]nc1-c1ccc3c(c1)OCCO3)C2 c1(CC)cc(C(=O)NC(C)(C)CCCNC(=O)C(C)(C)SC)ccc1O CCC(C)(CNC(=O)C(CC1CC1)NC(=O)CC1CC2C=CC1C2)CC c1(OC)nc(Cl)ccc1C(N1CCN(C(c2ccc([N+](=O)[O-])o2)=O)CC1)=O c1(NCC2(NC(C(CC)CC3CCCC3)=O)COC2)nnccc1C#N c1(C(N(CC=CC(=O)NCCC(COC)OC)C)=O)c(C)n[nH]c1C C(c1cccc(F)c1Cl)=CC(=O)NC(CC)(C)CNC(C1CC(O)C1)=O Cc1ccc(C(=O)NC2CC(N(C(=O)C=CC3CCCN3C)C)C2)c(O)n1 C1(NC(=O)CC=C(Cl)Cl)CCC2(CC1)CN(C(c1cnc(O)s1)=O)C2 C1(NC(Cc2ccc(C)cc2)=O)CC2CCC1N2C(=O)C(C)(C)c1ccccc1 N1(CC(=O)N)CC(c2nn[nH]n2)C2(CCC2)C1.c1(C(C)(C)C)ccccn1.C1CC1 c1(C(=O)NC(CC)(CNC(=O)C(C)(C)O)CC)cnc2occc2c1 c1(N2C(C(=O)NCC(C)C3CCC3)CCC2)ccc([N+](=O)[O-])cc1.C(N)(=O)N N1(C(C(CNC(c2ccc(O)c(F)c2)=O)OC)=O)CCc2ccncc2C1 c1(CC)ccc(CNC(=O)CC2CC2)nc1.C1(C=O)CC2(CCC2)C1.C C1(n2cc(CSC)nn2)CCCN(C(c2cncc(C(C)(F)F)c2)=O)C1 CC(CCN=c1[nH]c(=NCCc2cc(Br)no2)[nH]c2c1CCC2)N(C)C c1(C(=O)NCC2(OC)CN(C(c3csnc3C)=O)C2)c(C)cc(=O)oc1C CC(C)C(O)C(C)(C)C(=O)NCC1CCCCC1.C(=O)CS(=O)(=O)C(C)C.N c1(C(N2C3C(NC(CC(=C=C)C)=O)C(C3)C2)=O)ccc(Br)c(N)c1 C1(C(=O)Nc2c(C)ncc(CC)c2)CCN(C(=O)Cc2cc[nH]c2)CC1(C)C Cc1c(C(=O)NC)oc2ccc(Cl)cc12.C(=O)(C(C)C(F)(F)C(F)F)N1CCC1 C1(C=O)CC(=O)NC1(C)C.c1cnn(CCO)c1.C1(CC(=O)N(C)C)CCC1 N1(C(C(CC)N(C)C)=O)CCC(C2CC2)(CNC(C23CC2COC3(C)C)=O)C1 CCC(O)C(C)(C)C(=O)N1CCC(N(C(=O)CCc2cc(Cl)no2)CCO)C1 C=CC(C)C(C)C(=O)N1CC(CO)(NC(c2cccnc2)=O)C1 C1(OC)CC(CN(C(C=CC(=O)NC2CC(C)C2)=O)C)C1.C1CC1 N1(C(c2cc(C)c(Cl)cc2)=O)CC2CCOCC2(NC(=O)CN2CC(C)(C)C2)C1 C(=O)(C1CCc2c[nH]nc21)NC1C(C(=O)NCc2cccc(O)c2F)COCC1 C(CC(=O)NCC1CCC1)(C1=CCCC1)OCC.c1(CC(=O)N)nc[nH]n1 N1(C(C(C(C)C)O)=O)CCCC12CCN(C(c1cccn3cnnc13)=O)CC2 c1(C(=O)NC(C)CCN(C)C(C2(C#N)CCC2)=O)cc2ncccn2n1 N1(C(COCC(=O)NC)=O)CCCCC(C(=O)NCCSC)C1 C1(OC)CC(NC(c2ccc(C(F)(F)CF)cc2)=O)C1(C)C C(=O)(C(CC(F)F)C1CCC1)NC(CNC(CCC=CCC=C)=O)CO O=C1CCC2C(C(=O)NC3(C(=O)NOCCC4CC4)CC3)C12 c1(OC)ccn2cc(C(=O)NCC3CCCN3C(C3CC3F)=O)nc2c1 C1(C(=O)NCCNC(Cc2cn(CC)nn2)=O)CC(c2cccc(Cl)c2F)=NO1 C(=O)(C1CCCn2ccnc21)NCCN(C)C(c1conc1C1CC1)=O C(=O)(C(F)CC(C)(C)C)NCC(CC)NC(c1nscc1C)=O CN1CCC(C(=O)NCc2ccc(N3CCNC(=O)C3)cc2)C1c1cccnc1 C1(C(=O)NCC2CC(CNC(CC(CC)C)=O)C2)CCCCN1N=O CC1CC(C(=O)NCCCCCN(C)C(c2coc(CO)c2)=O)CCS1 Cc1cnc(CC(=O)NCCCN(CCCNC(=O)C=CI)C)[nH]1 C1(CNC(C(C=C)(C)C)=O)Cc2ccccc2CN1C(=O)Cc1cccs1 S(=O)(=O)(c1cc(C(F)(F)F)cc(Cl)c1)N1CC2N(C(c3ccco3)=O)C2C1.C C1(NC(C2(CC#C)CCCC2)=O)CCN(C(c2cc(Cl)cc(Cl)n2)=O)CC1CC c1(C(N(C)CC2CCN(C(C(CC=C)N(C)C)=O)CC2)=O)c(C)cc(O)nc1C N1(C(COCCCC)=O)CCC(NC(c2cc(OC)cc(C)c2N)=O)C12CCC2 C1(C(N(CCOCCNC(C(n2cc(Br)cn2)C)=O)C)=O)CC(C)(F)C1 Cc1ccccc1CCC(=O)NC(CCNC(C1CNC(=O)N1)=O)C(C)C C12(NC(c3cn(Cc4onc(C)n4)nc3)=O)CCN(C(=O)CNC=O)CCC1C2 CC1CN(C(c2ccc(Br)cc2F)=O)CC(C)N1C(C1(CCO)CC1)=O C=CCC(C(=O)N(C(CC)C(=O)NCCCS(N)(=O)=O)C)C(C)C C=CCC(CC(F)F)C(=O)NCC1(O)CCN(C(C2(C#N)CC23CCC3)=O)C1 c1(C(N2CCN(C(C(CC)O)=O)C3C2CCC3)=O)cc2c(C)cc(OC)cc2[nH]1 Cc1ccc(I)c(NC(c2cccc(NC(c3ncoc3C)=O)c2)=O)n1 c1(CC(=O)NCC(O)CNC(c2cnn3cccnc23)=O)ccc2nc[nH]c2c1 CCC(CC)C(F)C(=O)NC(Cn1cccn1)C(=O)NC.C12CC=CC(C1)OC2 c1(C(N2CC(O)(C3CCCN3C(c3ccccc3O)=O)C2)=O)cc2scnc2[nH]1 C(=O)(C(C)C(=O)NCC(C)NC(c1ncccc1C(F)(F)F)=O)OC S(=O)(=O)(c1ccc(Br)cc1NCCOc1cccnc1Cl)NC1(C)CCC1 N1(C(C(C)(O)C2CCC2)=O)CC2(CCCC2NC(c2ccc3occc3n2)=O)C1 C1(S(C)(=O)=O)(C(=O)OCc2nc(C)c(Br)s2)COC(=O)C1 C(C(C)(C)C(=O)N1CC2CC2(NC(=O)CSC2CCCCO2)C1)OC N#CC1CN(C(C2CC3CC3N2Cc2cnc(Br)s2)=O)CCO1 N(C1CCC(NC(=O)Cc2ccsc2)c2ccccc21)C(c1nc(C)n(C)c1)=O C=C=CC(C)C(=O)NCC1(NC(=O)CC2CC3(CCC3)C2)CCOC1 N1(C(=O)CCc2nc[nH]n2)CCC(N(C(=O)C(F)n2ccnc2)CCO)C1 c1(C(N2CCN(C(COCC)=O)CC2C)=O)cccc2c1nc(O)n2C C12(C(N(C(C)CC)C)=O)CCC(CC1)C(C)O2.C(=O)C(C)C=O.C(C)(C)C.N C1CCC(=O)N(C)C1=O.C1(C)(CC)C=C(C(=O)NC(C=O)C(C)(C)O)C1.N N1(C(c2cc(C)ns2)=O)CC2CN(C(C3(C)CC(C)OC(C)C3)=O)CC2C1 N1(C(C2CC(C)(CC)C2)=O)CCC(NC(=O)C(c2ccc(C)cc2)(F)F)C1C N1(C(C2N(C(C)=O)CCC2)=O)CCN(C(=O)CC2(c3ccccc3)CCC2)CC1 C(=O)(CC(CC)CC)NC(CC(N1C(C=C)CCC1)=O)C1CC1 c1(C(C(=O)NCCC#N)N(C)Cc2cocn2)ccc([N+](=O)[O-])cc1 N1(C(CC(C)F)=O)CC2(CC(NC(C3(COC(C)C)CC3)=O)C2)C1 c1(C(=O)NCCN(C(C2COC(=O)O2)=O)CC)nc(C)c(C)s1 c1(C(N2CC3CN(C(C(N4CSCSC4)C)=O)CC32)=O)nccc2nc[nH]c12 c1(CC)ccc(C(=O)NC(C)C(C)NC(c2ccn(C3CCOCC3)n2)=O)nc1 c1(C(=O)NCC(=O)N(CC)C)cc(CC)[nH]n1.CCOCC c1(OC)ccnc(C(=O)NCC23CC2CN(C(=O)CC24CCCC2C4)C3)c1 Cc1nn(CC(=O)NC2(CNC(=O)CCC(C)C#N)CCC2)c(C)c1[N+](=O)[O-] n1(C(CC(N2CCC(CNC(c3ccc(SC)s3)=O)C2)=O)C)nc(C)cc1C C12(CC)CN(C(c3ccccc3)=O)C(CNC(C3CC4CCC3O4)=O)(C1)C2 N1(C(c2cc(=O)c(O)c[nH]2)=O)C2CCC1CN(C(=O)C(F)(F)C1CC1)C2 CCCCC(O)C(=O)NC12CC1CN(C(c1coc(SC)c1)=O)C2 C(C)(C)(C#Cc1cn(CCC(C)C)nn1)C.CCCC(C)CCNC(=O)CC1CC1 N#Cc1cc(S(=O)(=O)N2CCn3nncc3C2)ccc1NCC1CCC(F)C1 C(=O)(C(C)C(O)C(C)CC)NC(C1CCCCC1)C(N1CCN(CC=C)CC1)=O c1(C(=O)NC(CCCCNC(C=Cc2ccc(C)o2)=O)C)cccn(O)c1=O C1(CCNC(c2n(CC#C)cnn2)=O)CCCCN1C(=O)C(CC)OCC C1(C(N2CCCC2CCCc2ccccc2)C(=O)NCC)CCC(C)(C)O1 C1(C(N2CCC(CN(C(=O)CS)C)CC2)=O)CCCCC1(C)C.c1cscn1.C C1(NC(=O)OC(C)(C)C)CC(S(C)(=O)=NC(=O)c2cc(F)c(N)cc2F)C1 c1(C(=O)NCC(C)(C)NC(=O)CC)cc(-c2ccccc2)co1.C(N)(=O)N C12(CNC(CCCC(C)=O)=O)CN(C(C3(C)CCCOC3)=O)CC1CCO2 Cc1cccnc1CCC(=O)NCC(C)CNC(=O)CCN1CCC(C)CC1 c1(C(=O)NC2CC(C)N(C(c3cncnc3)=O)CC2)cccc2ccnn12 C(C(C)(C)C(=O)NCCCCC1CCCC1)N(C(=O)CN1CCCCC1)C N1(C(C2(C)CCN(C(C=CCCC(C)C)=O)C2)=O)CCCN2CCCC2C1 C#CC1(C(N2CC(CNn3cncn3)C2)=O)CCN(C=O)CC1.C(C)(C)C.O Cc1cc(N2CCN(CC3CCC3)CC2)ncc1S(=O)(=O)N1CCC(C)CC1 C1(CNC(c2c(C)nn[nH]2)=O)CCCCCN1C(=O)CSCC(N)=O C(=O)(NNc1c(F)cccc1I)c1cccc2nn(C)nc21 C1(CNC(COCCCC(C)C)=O)C2CC1N(C(C1CC1)=O)C2.C1CCC1 c1(C(=O)NCc2cc(Oc3ccc(OC)cc3)ncc2)nn(C)c2c1CCC2 C(CCCCN(C(=O)C(F)=C(C)C1CC1)C)NC(C1(COC)CC1)=O C1(NC(C2CCn3nnnc3C2)=O)CCN(C(c2ccncc2O)=O)CC(O)C1 c1(C(N2CCC(NC(=O)CC3CC3)C2)=O)ccc(N2CCOCC2)c([N+](=O)[O-])c1 N1(C(C(C)=C2CCC2)=O)CCCC(C(C)NC(=O)CSS(C)(=O)=O)C1 CCCCC(CC)CC(=O)NCC(C1CCN(C(=O)C(C)C(C)(F)F)CC1)(C)C n1(CC(N2CC(NC(C3CC34CC4)=O)C(O)C2)=O)[nH]cc2c(=O)ncnc1-2 Cc1cc(O)cc(=O)n1CC(=O)NCCCOCCN(C)C(c1cn[nH]c1)=O [SH](=O)(=O)c1ccc(C#N)cc1.C1(N(C(CN(C)CCO)=O)C)CCC1.C(=O)CO C1(NC(CNC(C)=O)=O)CCCCC1C.c1(C(=O)N)nccnc1C(N)=O C1(NC(C2(C)COC2)=O)CN(C(c2cc(-c3cccnc3)on2)=O)CC1C1CC1 N1(C(=O)OC)CCCC(C(=O)NC(C2(O)CN(C(c3nsnc3O)=O)C2)C)C1 c1(C(N(C2CN(C(C(C3CC(F)(F)C3)OC)=O)C2)C)=O)cc(=O)cc[nH]1 C1(NC(c2nc[nH]c3ncnc2-3)=O)CCC2CCN(C(C3CCC3)=O)C1C2 C1(CC(N2CCC(CCCNC(C(C)(C)F)=O)CC2)=O)CCCC2(CCC2)O1 N1(C(C(Cc2ccco2)NC(CC(C)N(C)C)=O)=O)CCC2(CC2C(N)=O)C1 O=C1CC(CC(=O)NC2CCCC2CNC(c2ccccn2)=O)CC(=O)N1 CC(O)(CC(O)CNC(=O)Cc1ccccc1OC(F)F)C1CC1 c1(OC)cccc(C2=NOC(C(N3CC4CC4C3)=O)C2)c1.C(=O)C(=O)N(C)C.N C=CC(CCC)CC(=O)NCC1CC(NC(c2cccc3c2COC3)=O)C1 CCCCCCCCOCCCNC(=O)CC1CN(C(=O)C(F)(F)Cl)CCO1 c1(C(=O)NCC(C)NC(=O)C=CC2CCCO2)cnc2c(F)cccn12 c1(CN(C)CC2(C)CCC2)cc2cc(Cl)ccc2s1 C#CCC(C)(CC)C(=O)N1CC2=C(C1)CN(C(=O)COc1cccc(Cl)c1C)C2 c1(C(N2CCN(C(c3scc(C)n3)=O)C(C)C2)=O)c(C)cc(Br)cc1Cl C(=O)(CCCCC(N)=O)NC1C(C)(C)C1C(=O)NCC1CC2CCC1O2 Nc1c(C(N2CCCN(C(c3ccon3)=O)CCC2)=O)ccc(Br)c1F c1(-c2scc(NC(Cc3c(OC)cccc3)=O)n2)ccncc1C#N c1(C(=O)NC(C)C(C)C)cnc2n1CCOC2.c1(C2C(C(=O)N)C2)ccn(C)n1 C1(NC(C(CC)OCC)=O)CN(C(c2ccc3cnsc3c2)=O)C2(CCC2)C1 N1(C(=O)NCC(Cc2ccc(OC)c(OC)c2)(C)O)CC(O)C2(CCC2)C1 c1(C(=O)N)noc2cc(F)ccc12.N1(C(C2C(C(N)=O)C2)=O)CCC(C2CC2)C1 N1(C(=O)NC2CCCC(F)C2)CCn2nc3c(c2C1)CCCC3 c1(C(=O)NCC(CCCC)NC(=O)CCc2ccc(Cl)s2)c(C)cc(C)nc1O Cc1ccccc1Oc1ccccc1C(C)NC(=O)N(C)CC1CCCC1O Cc1ccc2c(C(=O)N(C)CC3CN(C(=O)CCCCCN(C)C)C3)c[nH]c2c1 C(=O)(CC(F)(F)Cl)N(CC(C)NC(=O)CSCc1ccncc1)C c1(OC)cc(C(N2CC(N(C)C(C3(C)CCOC(C)C3)=O)C2)=O)ccc1[N+](=O)[O-] C#Cc1ccc(C(N2CCC(C(C)(C)C)CC2CNC(=O)C2CC2)=O)nc1 CCC(CCC(=O)Nc1ccc(F)cc1C)NC(C1C2CCC(F)C12)=O C1(CC=C)CCN(Cc2cc(C(F)(F)F)c[nH]2)C1.C1(C)(CC=O)CC1(F)Cl C12(C(N(CCC(C)C)CCO)=O)COCC1CN(C(C1CCOC(=O)CC1)=O)C2 Cn1ccnc1CNC(C1(C)CCN1C(c1cc(C(C)(C)C)on1)=O)=O C1(CNC(CCCC)=O)CC(NC(c2ccc(COC)o2)=O)C1(C)C C1(CC(=O)NCCOCC#C)CN(C(c2nc(-c3ccsc3)cs2)=O)CCO1 c1(CCC(N2CC(NC(CC(C)OC)=O)C3C(C2)C3)=O)c[nH]c2cc(C)ccc12 C=C(C)CC(C(=O)N)NC(C)=O.c1(CC(N2CC(O)C2)=O)cncc(O)c1 c1(C(C)C)ccc(C(=O)NCC2(C(N3CCC3C3CCCCC3)=O)CCCO2)o1 Cc1c(C(=O)NC2CCC(C)C2)n[nH]c1C1CC1.C(=O)(CCc1ccoc1)N C1(O)(C(=O)OC)CN(C(=O)C(C)N(C(=O)CCC2CCOCC2)C2CC2)C1 Cc1cc(=O)c(C(N2CCN(CCNC(C3CCC(=O)NC3)=O)CC2)=O)cn1C Cn1ncc(-c2cn(C3CCCOC3c3ccccc3)nn2)c1N C(CS(=O)(=O)CC(=O)NC(C(=O)NC1CCC12CCCC2)C1(C)CC1)OC N1(C(C2(C)CC2F)=O)CCC(F)(CNC(c2ccnn2C2CCC2)=O)CC1 O=C1COC(CNC(C2CCCN2c2nccs2)=O)CN1 C1(C)(C(=O)NCCC(CC)(CC)NC(c2cncs2)=O)CC2CCC(C1)S2 N1(C(c2ccc(CCC)s2)=O)CCC2CC1CN(C(=O)Cc1cnn(C)c1C)C2 N1(C(C=C2CCC(C)C2)=O)CCCC(C)(NC(=O)COc2cccnc2)C1 CC(C)CCN(C(=O)N(C)CCn1cncn1)C1CC1 c1(CNC(c2c(C)nn[nH]2)=O)ccc(CNC(C2CC(C)CO2)=O)cc1 c1(C(=O)NC2CCCN(C(C(COCC)C)=O)C2CC)ccn2[nH]c(=N)nc2c1 N1(C(C=CCC(C)(C)NC(c2ccnnc2)=O)=O)CCC(F)C(O)C1 C#CC1(O)CCCN(C(c2conc2C(C)NC(c2cnn(CCC)c2)=O)=O)C1 c1(C(=O)NCC(C)NC(c2ncc(C(F)F)s2)=O)cc2cc(F)ccc2s1 c1(CC=O)ccc(F)nc1.c1(COCC(=O)N(C2CCCC2)C)ccnn1C c1(C(N2CC(C)C(CNC(=O)Cc3cccc(F)c3F)C2)=O)[nH]cc2c1CCC2 C1(C(=O)NC(C(=O)N(CC(CC)(F)F)C)C2(O)CCC2)CC12CCCCC2 C(=O)(C1CCc2ccccc21)N(CC(=O)NCc1ccc(C)cc1C)CCC CCCCC(C)CCC(=O)NC12CC1CN(C(c1cc(F)c(C)cc1N)=O)C2 c1(C(N(C2CCCN(C(c3ccnc(C)c3O)=O)C2)C)=O)cccn2cncc12 N1(C(C2(C)CCOC2)=O)CC(NC(=O)Cc2ccc(Br)cc2F)CC(F)C1 c1(NC(C2(c3ccccc3)CC2)=O)nc(Br)ccc1I C1(C(C(=O)NCC=CCNC(c2ccncn2)=O)OC)CCC(F)(F)CC1 c1(C(=O)NC2(CO)CN(C(c3cccc(C)c3N)=O)C2)cnc2cccnc2c1 C1(NC(C(C)SCC)=O)CCC2(CC1)CCN(C(C1C3CCOCC13)=O)CC2 C(C(CC(C)C)C(=O)N1CCN(C(c2ccc(C)nc2O)=O)C(C)C1)OC C(C(C)C)(C(O)C(=O)NCC1CCC(C=O)C1)OC.C(C)CCC1CC1.N N1(C(C2C(C(=O)OC)C2)=O)CCCCC1.c1(C(NC)=O)ccccc1C(F)F C(C(=O)N1CCCC(N2CCCC2=O)C1)(C(C)(C)O)NC(=O)OC(C)(C)C C1(NC(=O)C=C2CCC2)CC1C1CCCN(c2cc(O)nc(O)n2)C1 C1(O)(C(C)NC(c2c(C)nn[nH]2)=O)CCN(C(=O)Cc2cccc(Cl)c2Cl)CC1 Cn1cc(CNC(=O)CCC2CCN(C(c3ncncc3Cl)=O)C2)ccc1=O c1(C(N(C(C(=O)N(CC#C)CC=C)C)C2CC2)=O)cc(C)cc(O)c1 C(C)(CO)(C(=O)NC1CCC(NC(=O)C=Cc2ccc(SC)s2)CC1)OC c1(NC(c2n(C(CC)(C)C)nnn2)c2ccc(C3CC3C)o2)ccc(O)c(Br)c1 c1(OC)c(F)c(C(=O)NC(C)CCCC)cc(F)c1F.C(=O)(C=C1CC1)N c1(NC(C2CC(SC)C2)=O)cc(O)nn1-c1ncccn1 c1(C(CCC(=O)Nc2cnc(C)c(Br)c2)=O)cccc2ccccc12 C(=O)(C(S(C)(=O)=O)C1CC1)N1CCC(C)(C)C1.c1(C=O)ccnn1C1CC1 C1(C)(C(=O)NC(c2cccc(O)c2)C(C)C)CC=CCO1 c1(C(=O)NCC(C)C)c[nH]c2c(F)c(Cl)ccc2c1=O.C1(C=O)CNC(=O)N1.N N1(C(c2ccnc(C)n2)=O)CCC(C)C(NC(=O)CCC2CCCCCC2)C1 C1(C(=O)NC(C)CCC(=O)NC2COC(C(F)F)C2)Cc2nccn2C1 C(c1csnc1C)=CC(=O)NCC1C(NC(C2CC(SC)C2)=O)CCC1 C=CCCCC(C)N=c1[nH]c(=NCc2ccc(C)n2C)[nH]c2ccc(Cl)cc12 n1(CC(CC)O)cc(C(=O)NCC(C)CNC(=O)C=NOC)nn1 C(=O)(C(C)CCCOC)NCC1C=CC(NC(C(CC)OC)=O)C1 CCC(C)(C(=O)NC1CC(NC(=O)CCCNC(N)=O)C(O)C1)C(N)=O CC1CC(NC(c2[nH]nnc2-c2ccccc2)=O)CN(C(c2cnn(C)c2)=O)C1 C1(CC)(OC)CN(C(=O)CC2CCCCO2)C1.c1(C=O)cn(C(C)(C)C)nn1 c1(CC)cn2c(n1)CC(C(N1CCOCC1C)=O)CC2.C(=O)C(C)(C)C(C)C.N N1(C(CCOC)=O)CCC(CCOC)(NC(=O)CCCc2nnc(C)n2C)C1 c1(OCC=C)c(C(=O)N)cccc1C.C1CC2(CC2)CN1C(=O)C.C(C)=O c1(CC(C)(O)C2CC2)nc(-c2cccc(N)n2)nn1-c1ccc(F)nc1 C1(C(=O)NCCC=CCCC)COCCN(C(=O)Cn2ccc(C)n2)C1 Cc1oc(C(C)C)nc1C(N1CC(NC(=O)C(n2ccnc2C)C)C(C)C1)=O n1(CC)ncc(C(=O)NCCCC2CCCN2C(=O)C=CC(C)(C)C)c1C N1(C(=O)NC(C(C)(C)C)c2ccccc2)CC(C)(C)C12CCOCC2 Cc1csc2cc(C(=O)NC3(C)CN(C(C4CCOCC4C)=O)C3)[nH]c12 C1(C(=O)N)COCCC1C.C1(C(=O)NC(C2(C)CC2)C)(N(C)C)CCCC1 c1(C(N2C(CNC(C(COC)O)=O)CC2)=O)cnn2cccc(C)c12 Cn1nnc2cc(C(N3CCN(C(=O)CCOC4CC4)CC3CCO)=O)sc12 CC1CC(NC(c2n[nH]cc2CNC(=O)CC2CCCC(=O)N2)=O)CCO1 C(CCN=c1[nH]cc(Br)c2cc(Br)ccc12)N1C(C)CCCC1C C(=O)(C(C)(C)CC(C)(C)C)N1CCCC(C)C1.n1(CC(=O)N)cc(C2CC2)nn1 CC(CC(C)(C)C)C(F)C(=O)NCC1(C)CCCC1.C(=O)(CSC(F)F)N c1(C=O)ccc([N+](=O)[O-])cc1.c1(OC)cc(F)ccc1C(=O)NC(C)C(C)C C(=O)(CCCCNC(=O)CCOC)NCCOCCC=C c1(C(=O)NC(CC=C)CNC(=O)C(F)=CC2CC2)cnc2cccnn12 C1(CN(C)NC(CCSCC)=O)CN(C(=O)C(C)N(C)C)CC12CCC2 CCCC(CCCNC(c1scnc1C(C)C)=O)NC(C1(CF)CC1(F)F)=O C1(C)(NC(C(C)CSC(F)(F)F)=O)CCCN(C(C2(C)CCOC(C)C2)=O)C1 O=NN1CCCCC1C(=O)NC.c1(CCC(N2CC(F)C2)=O)ccc(Cl)c(Cl)c1 C12(C(=O)N)C3CC(CC13)C2(F)F.c1(CC)c(C(N2CCC(C)C2)=O)csc1C C(CCF)(C(=O)NCCCc1cnn(C)c1)NC(C(CC)C)=O N1(C(C(CC)(C)OC)=O)CC2CCN(C(c3ccc4nc(C)nn4c3)=O)CC2C1 Cc1cc2ncc(C(N3CC4C(C(=O)NCC5(C)CCCC5)C4C3)=O)cn2n1 c1(C(=O)NC(Cn2cc(C(COC)(C)O)nn2)C)ccnc2nccnc12 Cc1cccc(SCC(=O)NCC2CCC(N(C)C(c3cc(O)cs3)=O)CC2)c1 O=C(C1CCCc2c[nH]nc21)NCCNC(C12CCC(CO1)C2)=O c1(OC)cc(C(=O)NCC2CC(C)C2)ccn1.C(=O)(CC)N.C1CCOC1 C1(NC(=O)C2=C(Cl)CC2)CC2(C1)CC(NC(C1(C3CCCCO3)CC1)=O)C2 Cc1ccc(NC(C2CCC(C)CC2)=O)c(-n2cc(COCCCO)nn2)c1 c1(CC)ccc2c(Cl)c(C(N3CC(NC(=O)COCCF)C(C)C3)=O)sc2c1 c1(C(=O)NCC2OCCCN(C(C(C)(CO)OC)=O)C2)cc2ccc(C)cc2o1 CC1(C)CC(NC(=O)OC(C)(C)C)CN(C(c2n[nH]c(CCCO)n2)=O)C1 c1(-c2c(SC)scc2)nc(C(=O)Nc2cc3c[nH]nc3cc2F)n2ccccc12 C12CCCC1(F)CN(C(c1cc(S(C)(=O)=O)oc1C)=O)C2.C(C=O)=CCOC c1(C(=O)NCCCNC(C2C(C)OCC2)=O)ccccc1.c1(C=O)cccs1.N CC(C)CC(C)(C)C(=O)NCCN(C)C(C1CCN1S(C)(=O)=O)=O N1(C(=O)COCC2CCCO2)CCC(O)C(NC(C2CC(CF)C2)=O)C1 C1(CC)CN(C(c2ccc(C)[nH]2)=O)CCC1NC(C1(C(=O)OC)CC1C)=O N1(C(C2(CC)CCCCCC2)=O)CC2CCN(C(c3ccc(C)nc3)=O)C2C1 C(C(=O)NNc1nc(F)ccc1Cl)(C1CCNCC1)OC C(c1ccccc1)(C(F)(F)F)=CC(N1CC(NC(C(C)(C)C)=O)C(N=[N+]=[N-])C1)=O CC1CN(Cc2c(Cl)sc(Cl)c2Cl)CCN1c1cnccn1 CC1(C)CN(C(=O)C(O)CC(F)(F)F)CC(C)(C)C1NC(c1c[nH]nc1F)=O c1(OC)ccc(C(C)=CC(=O)NCCc2ccc(Br)s2)cc1 N1(C(c2cnn(C(CC)C)c2C)=O)CCc2c(C(=O)OC)c(OC)ccc2C1 C1(CC)CN(C(c2oc(C(F)F)cc2C)=O)CCN1C(c1c[nH]nc1OC)=O C(CC(C)(C)CNC(=O)COC1(C)CCCC1)NC(c1c(C)noc1)=O CC1(C)CC(CNC(=O)C(C)(C)CO)N(C(C2CCC(=O)C2)=O)C1 c1(C(=O)NC2CC(C#C)(C)C2)cc(C)nc(N(C)C)n1 C(CCCC)(C(=O)N1CC2(CO)CC2(CO)C1)NC(C1C(=C)C1)=O CCC(CCCC(=O)NC(CCO)c1ccco1)NC(=O)C(F)C(C)(F)F c1(NC(C2(C)CCCN(C(=O)Cn3cc(Cl)cn3)C2)=O)ccc(F)cc1[N+](=O)[O-] c1(N)cccc(Cl)c1C.C1(C(C(=O)CC)N(C(CC)CC)C)CCSCC1 Cc1cc(F)c(N)cc1C(=O)NCC1CCCCC1.C(=O)CC(C)(C)C(F)F.N Cc1c(C(=O)N(C)CCN(C)C(c2cc(C)n(C3CC3)n2)=O)cc(N)cc1O Cc1nscc1C(=O)NC(CNC(C1CCCC1C(F)(F)F)=O)C1CC1 n1(CC)ccc(C(=O)NCCOCC(N2CCC(C(=O)OC)CC2)=O)c1C C1(C)(C(N2CC3N(C(C=CSC)=O)C(CC3)CC2)=O)Cc2ccccc2NC1=O c1(C(=O)N)csc2nccn12.C1(CC)CCN(C(c2ccc(C(F)(F)F)[nH]2)=O)C1 C1(NC(CCP(C)(C)=O)=O)CC2(CCC(NC(=O)CCc3nncs3)CC2)C1 Cn1cc(C(N2CCC(CO)(NC(=O)CCOC3CCC3)C2)=O)c(Cl)n1 C1(C=O)CCCC(C)(C)CC1.C(CC(C)(C)C)N(CCC(=O)N(CC)CC)C N1(C(C(CCCC)C)=O)CC2CN(C(C3CCOC3C3CC3)=O)CC(C1)O2 C1(C(N2CCN(C(c3cc(C)nc(C(F)F)n3)=O)CC2)=O)CC2C=CC1C21CC1 c1(NCC2(F)CCCC2)nccc2sc(Br)cc12 C1(NC(C2C(C=C)C2)=O)CCOCC1NC(C1(C#N)CC1)=O Cc1nc2cccc(C(N3CCN(C(=O)Cn4nccc4C)C4CCC34)=O)c2[nH]1 CC(C)CCCCCC(=O)NC1(C)CCCC1NC(=O)CC1CCCN1C(C)C C1(NC(=O)CNS(=O)(=O)C2CC2)COCCC1.N1(CC(=O)N)CCCCC1 c1(C(=O)NCCC(C)NC(=O)C#CC2CCOC2)nsc2cc(Br)ccc12 C(=O)(C#CC1CCCCC1)N1C2CC(C(=O)NCC3CC(C)OCC3)(OCC2)C1 N1(C(CCC(=C)Cl)=O)CCCC2CCN(C(c3ccccc3N(C)CC)=O)CC12 Nc1nc(Cl)ccc1C(=O)NCCC1CCCCN1C(C1CC2CC2C1)=O C1(NC(CSCC#C)=O)CCCC12CCN(C(c1ccc(CCO)cc1)=O)C2 c1(OC)cc(Br)c(C(=O)NC2CC2CNC(=O)C(C)(F)F)cc1F C1(O)CCN(C)C1.c1[nH]c(=N)sc1C(F)(F)F.C1(CC(=O)NC)CCCOC1 C1(N(C(=O)COC(F)F)CCC)CCN(C(c2cc(C(F)(F)F)cs2)=O)CC1 C1(NC(CC2(NC(Cc3c(C)ccs3)=O)CC2)=O)CC(C)CC(C)(C)C1 c1(C(N2CCN(C(CCC(=C)C)=O)C(CCO)C2)=O)cc2cc(Cl)sc2[nH]1 C1(NC(c2c(OC)nccc2)=O)CN(C(C2CCN2CC)=O)C2(CCCC2)C1 N1(C(CCC)C)CC(C(=O)NCC2(NC(=O)C=CC)CCCCC2)CC1=O C1(NC(C)=O)CCN(C)C1.c1(C2(CNC(=O)C=CCl)CC2)ccccc1.CC c1(C(=O)NC(C2CCCC2)CC2CCCN(C(C(C)C)=O)C2)ccc(F)cc1F Cc1nc(CC(=O)N(C(C)C(=O)N2CCC2CO)C2CC2)co1 c1(C(N2CCC(CCOC)C2)=O)c(C)nn(C)c1C.c1(C=O)cc(C#N)c[nH]1.N c1(C(=O)NCCC2(OC)CN(C(=O)CO)C2)ccc(C(C)(C)C)cn1 C1(n2cc(C(CSCC)C)nn2)CN(C(c2ccc(C)s2)=O)CC1O Cc1noc(C)c1CCNC(=O)C(c1cccs1)NC(C1COCC(C)O1)=O N1(C(C(=Cc2cnc[nH]2)C)=O)CCCCC1Cc1ccc(Cl)cc1 Cc1ccc(Br)c(C(c2nnnn2C2CCOCC2)NCC2(C)CCCCO2)n1 C1(C(=O)NCCC2(NC(c3cccs3)=O)CC2)COc2cc(Cl)ccc2C1 Cc1cc2sc(C(=O)NCC(C)(C)CC3CN(C(c4cn[nH]c4)=O)C3)cc2s1 CC(CCCCNC(=O)CC1(C)CC1)NC(c1c[nH]cc1C1CC1)=O N1(C(COc2ccc(C(N)=O)cc2)=O)CC2(CCC2NC(=O)CCCF)C1 c1(C(=O)NCCNC(C(C)CC(C)(C)C)=O)cnc2c(n1)CCCC2 Cc1oc2cc(C(N3CCCC3(C)CNC(=O)C(C)n3cncn3)=O)[nH]c2c1C CCCC(C(=O)OC)C(=O)NC1(C(=O)NOCc2nncn2C)CC1C C(=O)(C(CNC(=O)Cn1ccnn1)C(C)(C)C)N1CC(C(C)C)OCCC1 c1(CC)nc2ccccn2c1C(=O)N.C1(CC=O)CC(C)=NO1.CCC1CC1 CC(C)C(C)C(C)CC(=O)NC1CCN(C(=O)C(C)Cn2ccnc2)CC1F c1(NCC(CC(C)(C)C)OC)cc(=NCc2cc(=O)n(C)c(=O)n2C)[nH]cn1 C1(CNC(=O)CC2C=CCCC2)CCCN(C(=O)CC2CC(=O)NC2=O)C1 [N-]=[N+]=Nc1cccc(NC(=O)C=CCNC(=O)COCCCN=[N+]=[N-])c1 Cc1nc2nccc(C(=O)NCC(C)(C(C)C)NC(=O)C=O)n2n1.CC(F)F.N c1(C(=O)NC2C(CC)CN(C(C3(CCF)CC3)=O)CC2)ccc(C)c(F)c1N CC#CCC(C(=O)N=c1ccn(C(C)CC)[nH]1)NC(c1cc(CO)oc1C)=O C1(CC(=O)NC(CC)CN(C(=O)Cc2nccn2C)C)CCC12CCC2 N1(C(C2=NOC(C)C2)=O)C2CCC1CC(O)(CNC(=O)CO)C2.c1ccccc1 C1(C(=O)NCC2CCN(c3c(C(C)C)c(Cl)ncn3)C2)CCC2C(C1)C2(F)F c1(C(=O)NCC(CNC(C(CC)CC)=O)OC)ccc(O)c(Cl)n1 C=CCC(C)C(=O)N1CCC(CO)(NC(c2cc(O)nn2C)=O)C1 N1(C(C(COC)NC(C)=O)=O)CC(C(=O)Nc2cncnc2C)CC2OCCC12 C1C2CCN(C(=O)CC3C=CS(=O)(=O)C3)C12.Cn1nccc1C1(C=O)CC1 c1(OC)cc(Br)ccc1C(=O)NCCC1CCN(C(=O)C(C)CF)C1 c1(NC(=O)CCCOC2CCOCC2)ccc2ccc(O)nc2n1 CCC(CC(=O)N(CC(C)NC(c1oc(C)nc1C)=O)C)c1ccc(OC)cc1 Cc1cc(C(=O)NCCCCC2CN(C(C3CCCCC3F)=O)C2)sc1C n1(C2CN(CC)C2)cc(CC)nn1.c1ccncc1.C1(CC(=O)NC)CCOC1 c1(C(N(CCC(C)NC(C2CC(O)C2)=O)C)=O)cc(C#N)ccc1Br C(=O)(CCC(C)(C)c1ccccc1)N(C)CC1(NC(=O)C2=CCC2)CC1 c1(CC=O)cc(C)[nH]c(=NCCN(C(=O)Cn2ccc(=O)n(C)c2=O)C)n1.C N1(C(c2n(CCC)ccc2)=O)C2CCC1CC(NC(=O)CC1CCCC(C)O1)C2 C(=O)(C(C)(C)C1=CCN(C(=O)C(N=[N+]=[N-])C(C)C)C1)Nc1c(C)n(C)nc1 C1(NC(C2N(C)CCN(C(=O)C(C)(C)O)C2)=O)CCC(N=[N+]=[N-])CC1 c1(NC(C2CCCC(NC(C#CC(=O)O)=O)C2)=O)cc2c(cc1[N+](=O)[O-])OCC2 CCC(Cc1nc(-c2nc(C(F)(F)F)cs2)nn1CCCO)C(C)C CS(=O)C=CC(=O)NCCCC1CCCN1C(c1cnc(C2CC2)nc1)=O Cc1cccnc1CCC(=O)NC12CC(C1)C2.C1(C=O)CCC(C(N)=O)C1.C C(=O)(C(N)CCC(C)(F)F)Nc1ccc(Cn2c(C)cc(C)n2)cc1 c1(C=O)ccc2c(c1)OC(F)(F)O2.C1(C)CC1C(=O)N(C)CC.CC.CC C(CCCCCN=c1[nH]ncs1)N(C)C(C1CCC2CC2C1)=O C1(CC(N2CCC(CCC#C)CC2)=O)CC2(CC2)CN1C(=O)CC(=O)NCC c1(CC(N2CCC(N(C)C(C3CC(C)(O)C3)=O)CC2)=O)cc(F)c(F)cc1F n1(CCC)ncc(C(=O)NC2CC(CCNC(=O)CC3CCCOCC3)C2)c1C C1(C#N)(C(=O)NCCCC(N2C(C(=O)NC)CCC2)=O)CC12CCC2 c1(N(C(C)CNC(C23CC(C)(C2)OC3C)=O)C)ccncc1[N+](=O)[O-] CS(=O)(=O)c1sccc1C(=O)NC1CC(C)C1.C(=O)C1=CS(=O)CCC1.N N1(C(C(C)(C)c2ccccc2)=O)CCC(NC(=O)CC2CC(F)C2)CC1 c1(OCCC)ccc2c(c1)CCN(C(c1cc(OC)ccc1OC)C(=O)NC)C2 C1(NCC(C)(C)CF)Cc2nc3ccccc3nc2C1 N1(C(C(CC(C)C)NC(C2CC(OC3CC3)C2)=O)=O)CCCCCCC1C CN1CCCCC1C(=O)NC1CC(CCNC(=O)C(c2cncn2C)O)C1 C(=O)(C1CCCc2sccc21)N1CCN(C(c2c(CC)ncnc2)=O)CC1C N1(C(C(C)(F)c2ccon2)=O)CC2(CCCN(C(c3cc(C4CC4)no3)=O)C2)C1 C1(C(C(=O)O)OC)CCN(C(C2CCCNC2=O)=O)CC1 C1(CC(N)=O)CN(C(=O)CC2CCN(C(=O)Cc3ccccc3)C2)CC1O c1(SC)ccc(Cl)c(C(=O)NC2CCC(NC(=O)C(C)(C)C(C)O)CC2)c1 C(CCN(C(=O)C=CC(F)(F)F)C)(C(C)C)NC(C=C(CC)CC)=O N1(C(Cc2cn(CC)nc2)=O)CC(C2CC2)(C(N2CCCC(F)(F)C2)=O)C1 Cc1cnc(CC(=O)Oc2ccc(OCc3ccccc3)cc2)cn1 C(=O)(C(C(C)(C)C)NC(C1CCCN1C(c1cc(C)nnc1O)=O)=O)NC C1(C(N2CCC(CC)C2)=O)CCCCS1(=O)=O.C(C=O)=CCN(CC#C)C.N C(=O)(C1=C(C)OCC1)NCC(CNC(c1cc(COC)oc1C)=O)CO C(CNC(=O)CCCc1nc(C(C)C)no1)(C(C)C)NC(CCOC)=O c1(NC)cccc(OC)c1C(N1CCN(C(C)C)C(=O)C1)=O.N12CCC(C1)C2=O C(CN=c1[nH]n(C)cc1[N+](=O)[O-])N(C)C(c1csc(-c2cn[nH]c2)n1)=O C1(OC)C(NC(c2ccc(Cl)cc2C(F)(F)F)C)COC12CCC2 C1(C(=O)NCC2C=CC(NC(=O)Cc3ccno3)C2)CCN(C2CC2)C1=O CC(C(C)(C)NC(c1ncn(C(C)(C)C)n1)=O)NC(C1CCC(=O)N1)=O C1(N(CCCNC(=O)C)CC)CC2CCCCC2NC1=O.C(=O)(C(F)(F)F)N C=CC(F)(F)C(=O)N1CCOC(CNC(c2sncc2Br)=O)C1 c1(C(=O)NC(CCSCC)C)cccnc1CNC(=O)CNC=O C(N=c1[nH]c(=N)[nH]c(=NCC2(CCN(C)C)CC2)[nH]1)c1cc(OCCC)ncc1 Cc1cn(CC(N2CCC3(CC(NC(=O)C(C)CN(C)C)C3)C2)=O)c(=O)nc1O C1(C(=O)NC(C)(CNC(c2ncccc2F)=O)C2CCC2)CCn2cncc2C1 N1(C(CC2(C=C)CCC2)=O)CC2CCCC2(CNC(C2CCN(C)CC2)=O)C1 Cc1nc(NC2CCSC2)ccc1NC1CCC(CN)C1 N1(C(C(C)OCC#C)=O)CCN(C(c2ccc(CCC)s2)=O)CC1 C=CCC(C)(O)C(=O)N(CC(C)C(=O)NCCNC(C1CCC1)=O)C C(=O)(CC(C)(C)C1CC1)NC(C)CC1CN(C(C2COCCO2)=O)C1 N1(C(Cc2c(C)n[nH]c2)=O)CC2=C(C1)CN(C(=O)COCC1CC1)C2 CN1CC=C(C(=O)N2CC(F)CC2CC(=O)NC2CN3CCCC2C3)C1 N1(C(c2n[nH]c(CC)c2C)=O)CC2CCC(N(C(=O)C(C)CC3CCC3)C)C2C1 C1(C(=O)NC(C(CC)(C)C)C)CC2CCC(C1)N2C(=O)CC(C)(C)C#N N1(C(C2N(C(c3cc(Cl)c[nH]3)=O)CCN(C)C2)=O)CCn2ncnc2C1 C(CC(=O)NCC1(O)CCOC1)(C(C)CC)NC(c1ccc(C#C)cc1)=O c1(NC(c2n(CCCSC)nnn2)c2ncc(SC)s2)cncc(C(F)F)c1 C1(C(N2CC3CCC2CN3C(C2CCCSS2)=O)=O)Cc2ccccc2N1 C(CC(C)CC)NC(c1cc(CSCC)on1)=O.c1ncccc1C(C)=O.N C1(CNC(C=CC(C)C)=O)CN(C(=O)CCc2ccc(F)cc2)CC1C CC1(C)CC(NC(=O)C(CCc2ccccc2)NC(=O)OC(C)(C)C)CCS1 c1(C(N2CCC(C)C2CNC(=O)CC2CN(C)C2)=O)cccc2occc12 C(=O)(CN=c1cc[nH]cc1)N1CC(OCC(=O)N(C23CCC(CC2)C3)C)C1 c1(C(N2CCC(NC(=O)Cc3cncnc3)C2)=O)cc(Br)cnc1Br C(=O)(C(O)CC(F)(F)F)NC1(C(=O)NCc2cc(C)c(C)nc2)CCOCC1 C(=O)C(O)CCS(C)=O.c1(OCC)ncc(C(=O)NCC2(CC)CC2)s1 c1(CC(N2CC(O)(C(C)NC(CC(COC)C)=O)C2)=O)cc(O)cc(Br)c1 c1(SC)cc(C(=O)N(CC(O)CNC(C2CC(n3cnnc3)C2)=O)C)oc1C CN1N=C(CC(=O)NC2(CO)CCN(C(C3CCC4(COC4)OC3)=O)C2)CC1=O N1(C(c2ccc(C)cc2Cl)=O)CC(NC(=O)C(C)(C)n2cnnn2)CC2(CC2)C1 c1(C=O)cnc(C2CC2)nc1.c1(CC(C)C)cc(C(=O)NCC(C)CO)n[nH]1.N c1(C(N2CC(OC)CC23CCC3)=O)cc2c(F)cccc2s1 c1(C(=O)N)csc(C2CCCCC2)n1.C(C(C)C)N(C(=O)C(F)=C1CCCC1)C Cc1ccc(NC(c2ccc(C(F)(F)F)c(C3CC3)c2)=O)cc1[N+](=O)[O-] N1(C(CC)CC)CC(C(=O)NC2CC(C)N(C(=O)Cc3cccnc3)C2)CC1=O N1(C(c2cc(OCC)ncc2)=O)CCC2(CCCC2C(=O)OC)C1 N1(C(C2(CCN(C)C)CC2)=O)Cc2ccccc2C(NC(c2ccc[nH]2)=O)C1 C(=O)(C1=CCCCO1)N1CC(C(=O)NCc2ccc(C(=O)OC)[nH]2)SCC1 c1(OC)cc(Br)cc(F)c1CN1CCOC(C(=O)Nc2ccc(C#N)cc2)C1 c1(OCCC)ccc(NCC2CNCC(C)(C)O2)cc1OCCC c1(-n2cc(C3(C)N(C(C(C)OCCC(C)C)=O)CCC3)nn2)ccc(Cl)c(F)c1 C1(CNC(CC(C)CNC(c2cnc(N)cn2)=O)=O)OC(=O)CC1(C)C N1(C(CC(=O)OC)C)CCN(CC2CC(c3ccccc3C(=O)O)C2)CC1 CC1=NOC(C(=O)NCc2c[nH]nc2C(=O)NC2COCC2)C1.N(C)C.C c1(SC)ccc(CCCC(=O)NC(C)CNC(c2cn(C)nc2Br)=O)cc1 CC1CN(C(c2cn(C)c(=O)cn2)=O)CC1(C)C(=O)NCCCc1nccs1 Cc1cc(Cl)ccc1-n1nc(CCO)nc1-c1cccc(SCc2nc[nH]n2)c1 CC1CCc2nc(N3CC(=O)NC(=O)C3)nc(N3CCC(C)(N(C)C)C3)c2C1 c1(-n2cc(CC(C(C)C)O)nn2)ccccc1C(N1CCCC1C1CC1)=O c1(C(N2CCCC(C)(CNC(c3c(C)ocn3)=O)C2)=O)cc([N+](=O)[O-])cnc1O c1(C(=O)NC(C(C)CO)C(=O)O)[nH]c2ccccc2c1-c1ccccc1 Cc1ncncc1C(N1CCCC1C(C)NC(=O)CC1(O)CCCCC1)=O C1(C(N2CCC(CC=C)(C(=O)N)C2)=O)CCCC2(CC2)C1.c1cncc(O)c1.C c1(OC)ccc(C(=O)NC2CN(C(=O)NC3CCCCC34CC4)C2)c2sccc12 C(=O)(CCC(=O)c1cccc(Cl)c1)N(CCCN(C(C(C)n1cncn1)=O)C)C C1(C(N(CCC)C2CC2)=O)CCCN1C(=O)CO.O=CCCC1CC1(Cl)Cl.N CCN=c1[nH]c(C)c(C(=O)NC(C)CC(C)NC(c2cc(C)ncn2)=O)s1 N1(C(=O)OC(C)(C)C)CC2CCC(NC3CS(=O)(=O)CC3C(N)=O)CC2C1 C=C(C)CCCC(=O)NCC1OCCC1C(N1CCCC1)=O N1(C(c2n(CCC)nc(C)c2)=O)Cc2ccccc2CC1CNC(C1CC1C)=O c1(C(=O)NC)cccc(S(=O)(=O)NCCCc2noc(C3CCCCC3)n2)c1 C1(NC(c2c(C)noc2)=O)(CO)CCN(C(=O)Cc2sc(C3CCC3)nc2C)C1 N1(C(C2CCC(CC)CC2)=O)CCC(F)C(NC(=O)CC23CCC(CC2)OC3)C1 C(CC(F)(F)F)N(C(=O)C(C1(O)CN(C(c2cc(C(F)F)[nH]n2)=O)C1)F)C Cc1cc(CNC(=O)C(CO)NC(=O)CCc2cnn[nH]2)sn1 n1(CC#C)cccc1C(c1nnnn1CCC)NC1(C(=O)N(C)C)CC1.S C(=O)(C#CC1CCCC1)NCCC(C(C)C)NC(C=Cc1n(CC)ccn1)=O C1(CNC(COCCC(C)C)=O)CCN(C(=O)Cc2c(F)cccc2F)CC1O C=CCC(C)(CNC(c1ccoc1CNC(C1CC(N=[N+]=[N-])C1)=O)=O)CO C1(C(=O)NCc2cnco2)CC(F)CN(Cc2ccccc2OC(F)F)C1 C(C(=O)N1CC2C(CN(C)C(C3(C)CCCO3)=O)C2C1)(C(C)C)NC(C)=O c1(C(=O)NC(CNC(c2nncc(CCC)c2)=O)CC)ncccc1S(C)(=O)=O N1(C(Cc2c(C)n(C)cn2)=O)CCCCCC(NC(=O)CNC(=O)CC(C)C)C1 C(=O)(C(F)C(=O)N1CCCC(NC(=O)CC2CC(F)(F)C2)C1)OCC.C c1(CSc2scc(C)n2)cccc(NC(=O)Nc2ccccc2)c1 N1(C(COCCOC)=O)CC(C)C(NC(c2ccc(O)c(Cl)n2)=O)C(C)C1 C1(C)(C(=O)NCCC(C)NC(c2coc(CO)c2)=O)CCN(C)CC1 C1(NC(c2c(C)n[nH]c2)=O)CN(C(=O)COC2CCCCCC2)C2CCCCC12 C(COC(C)C)(C(=O)NC1CCN(CCCc2ccccc2)C1)NC CCC(C)CC(C(=O)NCC1CCOC1C)NC(c1ncccc1Cl)=O C(c1ccccc1)=CC(=O)N.C1CC(O)CN1C(=O)CC1(C(F)(F)F)CC1 C12(CNC(N3CCOCC3c3ccccc3)=O)CCC(CC1)OC2 N(C1CCCCc2ccccc21)C(c1cc(Cl)c(F)cc1F)=O CC1CN(C(=O)C=Cc2cncc(F)c2)CC(CCNC(c2cnc(Cl)[nH]2)=O)O1 N1(C(C2(OC)CCCC2)=O)CCC(C=CC(=O)NOCC2CCCC2)CC1 n1(CC)cc(C(=O)N(CC(CO)(CO)NC(=O)C(C)SC)C)c(C2CC2)n1 c1(CNC(c2n(CC)cnc2)c2nnnn2CC)cccc(C2CC2)c1 Cc1cc(C(=O)NCC(CNC(c2cncc(F)c2)=O)C(F)(F)F)ncc1C#N c1(N2CC(O)(CC)C2)ccn2c(Br)cnc2n1.c1(C(=O)N)scnc1C(C)(C)C CCC(C(=O)NCCOC1CCN(C(=O)C(c2cccc(F)c2)C)CC1)C(C)O C(C(=O)NC1CC(C)C1)(C(C)C)n1ncc(C)c1.C(=O)C(C(C)C)N(C)C.N c1(NC(=O)NC2CCCN(C(C)C)C2)nc2cccc(Br)c2s1 c1(C(N(C2CCCC2)C)=O)cnccc1C(F)(F)F.c1(C(=O)N)ccc(Cl)cc1 c1(C(CC(=O)N(CCCCNC(c2cnn(CC)n2)=O)C)C)ccccc1C Cc1c(C(=O)NC2CC(CNC(C3SCCS3)=O)C2(C)C)cnn1C N1(C(C=CC2N(C)CCC2)=O)CC(CC(=O)NCCC(O)C(F)F)CC1(C)C N1(C(CN(CC(C)C)C(c2cccc(C)c2F)=O)=O)CCC12CCN(C)C2 Cc1cccc(C)c1C(=O)NC1CC2CC1CN2C(C1CC(F)C1)=O c1(-c2ccc(OCCC)cc2)ccc(C(=O)Nc2ncncc2Cl)c(OC)n1 C1(C(=O)NCC(=O)N(c2nccn2C)C)CCCN(C2C3CNCC2C3)CC1 c1(C(NC)=O)cc2c(s1)C(C)(C)CCC2.C1CCCN1C(C1CC12CCC2)=O.C C(CC1=CCN(C(=O)CN(c2ccncc2)C)CC1)NC(C(F)OC)=O c1(C(=O)NCCC(C)NC(C2(CCCC)CC2)=O)ccsc1S(N)(=O)=O C1(C(=O)NCc2n(C)ncn2)CC=CC(n2cc(C3CCOC3)nn2)C1 C1(S(C)(=O)=O)(C(N2CCC(NC(CCSCCCC)=O)C2)=O)CCCCC1 c1(NC(C2CCN(C(C(CCC)C#N)=O)C2C)=O)cc(C)cn(C)c1=O c1(C(N(CCC(=O)NCC2CNC(=O)CO2)C2CC2)=O)n[nH]c2c1COC2 Cc1ccn2cc(C(=O)NCC(O)CNC(=O)C(C)(C)CCCO)nc2c1 c1(C(=O)NC(C(C)NC(CCC(CC)OC)=O)C)ccn2cncc2c1 C(CC(F)(F)C(C)C)NC(C(CC=C)NC(C1OC2CCC1C2)=O)=O C1(C(=O)NCCOCC(C)(C)C)CCC(n2cc(CC(=O)O)nn2)C1 C1(CCNC(C2C(OC)CC2)=O)CCCN(C(c2cnn(CCC#N)c2C)=O)C1 c1(C(=O)OC)cccc2c(NC(=O)C(=O)NC3(O)CCNC3)cccc12 CCCCN=C(NCCc1cccc(F)c1)NC1CC1(C)C(C)C N1(C(C(=O)NCCOCC)c2cnsc2)CCN(C(c2ccncc2)C)CC1 N1(C(c2c(C)cccc2C)=O)CCC2(CCN(C(C3(CO)CCOC3)=O)C2)C1 C1(NC(C(C)SC)=O)CCCCN(C(c2cn(C(F)(F)CO)nn2)=O)C1 c1(C(=O)NCCN(c2ccc(C#N)nn2)CCC)cn2c(C)cccc2n1 C(=O)(C1=CCCOCC1)NC(C(N1CC(C)(CC)OCC1)=O)C C1(SC)CN(C(=O)C(C)(C)c2cnn(C)c2)CC1NC(=O)CCn1ccnc1C C(=O)(C(CCS(C)=O)N(C)C)N(CC)CC1CCCN1C(=O)C=CCF c1(CC(=O)NC2C(C)N(C(=O)C=CC(C)(C)C)CC2)cccc(Br)c1Cl c1(CC(=O)NCC2CCC(OC(CC)C)C2)cnc(On2cncn2)c(C)c1 c1(N(C(=O)C(O)C2CCCC2)CC)ccc(Cl)c(F)c1 CP(C)(=O)CC(=O)NCC1CCN1C(C1(C(F)(F)F)CCOCC1)=O C=CCCCCC(=O)NC1CC=C(C(=O)N(CC)Cc2cccnc2)C1 c1(C(=O)NCC(C)(C)CNC(c2cn3cnnc3cn2)=O)nnn2c1CSCC2 Cn1nnc(Br)c1CNC(c1nnnn1CC1CC1)CCC1CCCO1 C1(C(N(C(C(N)=O)CCC)C)=O)CC2(CCN1C(c1ncc(F)cc1F)=O)CC2 N1(C(c2cc(OC(C)C)ncc2)=O)CCN(C(c2cc(Cl)ncc2Cl)=O)C2CC12 C1(C)(CNC(C(CCSC)NC=O)=O)CN(C(c2ccc(C)nc2)=O)CCO1 n1(CC)cc(CNC(CN2CCOCC2)C(=O)O)cn1 C(=O)(C1=CCCCC1C)Nc1c(NCCC)cc(O)cc1 n1(CCC)cc(C(=O)NCCC2CCCC2)cn1.C1(C=O)CC1.C(C)=O.N N1(C(c2ccoc2)=O)CCN(N2CCC(C3CCCCC3)C2)CC1 C12(CNC(CC3CC(C)C3)=O)CCCC(CN1C(c1cnn(C)c1N)=O)C2 C1(NC(C(F)=CC)=O)CC(C)CN(C(c2cc(O)ccc2C)=O)C1 C1(C(=O)NC(C(C)O)C(=O)NCc2ccc(O)nn2)Cc2ccccc2C1 CC1CN(C(=O)CNC(=O)Cc2ccccc2)CCCN1C(=O)Cn1cncn1 Cc1cc(CC(N2CC(O)C(O)C2CNC(=O)CC2COCC2O)=O)cc(C)c1 N1(S(c2cccc(N3CCC(=C)C3)n2)(=O)=O)CCc2cc(OC)c(OC)cc2C1 C1(NC(C2C(C(=O)OC)CCC2)=O)CN(C(c2cncc(OC)n2)=O)CC1.O C(=O)(C(O)C(C(C)C)OC)Nc1c(CC)cc(O)cc1 C#Cc1cnc(C(=O)NCC2CCN(C(=O)CC(C)CC)C2(C)C)c(C)c1 c1(CC)nnsc1C(=O)NC1CC(C(F)C(=O)NCc2snnc2C)C1 c1(C(=O)NCCOC2CCN(C(CCSC)=O)C2)[nH]nc2ncc(Br)cc12 c1(C(=O)NC2(C3CCN(C(c4c(C)coc4)=O)C3)CC2)nc2ccccn2c1F C#Cc1cnc(O)[nH]c1=NC(=O)NC(C)Cn1cncn1 C1(CCCC)CCN(C(=O)C(CC2CCC2)NC(=O)C=CCN2CCC2)C1 C12(CNC(C3CCCOC3)=O)CCC(CC1)N2c1cc(C(F)(F)F)ncn1 C1(CNC(c2c(C(C)OC)noc2)=O)COCC(C)O1.C1CCC(=O)N1 C(Cn1cccn1)(C(=O)N=c1ccn(CCF)[nH]1)NC(CNC(CC(C)C)=O)=O C1(NC(C(C)Oc2ccc(F)cc2)=O)COC2CN(C(=O)C(C)(C)N(C)C)CC12 c1(CC(=O)NC(CC)CNC(c2nnsc2C)=O)cc(=O)n(-c2ccccn2)[nH]1 Cc1ccccc1C1(CNc2cnc(-c3ccoc3)s2)CCOCC1 C(CCC(=O)N1CCCC1C(C)NC(=O)C=Cc1ccoc1)N(C(C)=O)C N1(C(CCCCN(C)C)=O)CC2(CCCC2NC(C2CC2CC(C)(C)C)=O)C1 C1(C(N2CC(O)(CCNC(C(N3CCOC3=O)C)=O)C2)=O)CC12CCOC2 c1(C(=O)NCCC2CCCC2)nnn2c1CCCC2 CC(C1=CCN(C)CC1)NC(=O)CNC(C1CCC(C)(C)C1)=O O=C(C1COc2ccccc21)NC1CN(C(=O)Cc2ccc(Cl)s2)C2(CCC2)C1 c1(CN2CC(C)(C(=O)Nc3cnc(Br)c(Cl)c3)C2)ccc(O)c(C(=O)O)c1 CC(C)CC(C)C(=O)N1CCCC(C(C)Nc2ncncc2Br)C1 C#CCC(CC(=O)OC)NC(C1CCCCCN1C(=O)CC(C)CN(C)C)=O C1(C(=O)NC(CCC)C(=O)OC)CCN(C(C2(F)CCCC2)=O)CC1O c1(OC)cc(CNCC2CC(=O)N(C)C2)c(Cl)cc1O c1(C(N(C2CCC(NC(c3ccc(F)cc3)=O)C2)C)=O)cc2ccccc2nn1 N1(C(CNC)=O)CCC2(CC1)CC2(C)C(=O)NC(C)CCCC(C)(C)O N1(C(C(C(=O)OCC)CC)=O)CCCC(C2CCN(C(=O)C(C)(C)C(F)F)CC2)C1 C1(NC(CCSC)=O)CN(c2ccc(C(F)(F)F)nn2)CC(C)(C)C1 C1(CC)CN(C(=O)Cc2ccsn2)CCC1NC(c1nc(=N)cc[nH]1)=O c1(C(=O)NCC(c2ccccc2)NC(C(C=C)O)=O)cccc(Br)c1C C1(C(=O)NC2CC(C)N(C(c3cc(O)n(C)n3)=O)CC2)CNC(=O)CC1(C)C [nH]1cc(C2OCCC2C=O)cn1.n1(CC=CC(=O)N(CC)C)cncn1.CC C(=O)(CCC(=O)NCCNC(C1(CO)CCCC1)=O)c1ccc(C)s1 c1(C(=O)NC2CCCC(N(C(c3ccn(CC)n3)=O)C)C2)cc(O)cc(C#N)c1 N1(C(C2CC(OCC)C2)=O)CCC(CNC(c2nnn(C)c2N)=O)(O)C1 C1(C(N(C2CCCN(C(=O)CC3CCC(=O)CC3)C2)C)=O)CCCC(CF)C1 C1(C(N2CC(CC)(CO)C2)=O)CCCN(C(C2C3CC4C(C3)C24)=O)CC1 C1(N(C(c2c(CC)occ2)=O)C)CN(C(=O)C(C)n2cncn2)CCC1C C(=O)(C1CCCc2sc(C)nc21)N1C(CNC(C(CC)n2cccn2)=O)CCC1 N1(C(COCC)=O)CC(NC(c2snc(-c3ccccc3)c2N)=O)C(C(F)F)C1 C1(C(=O)NCC2C(C)CN(C(c3cnc(Cl)cc3Cl)=O)C2)C2CCCCCCC12 C1(C(=O)NC(C(C)O)CO)CN(C(=O)C(C#N)C(C)(C)C)CC12CCC2 C(=O)(C(C#N)C(C)C)NC1CCC(NC(c2ccc(C)n2C)=O)C1 CC(CC(N)=O)C(=O)N1CCN(CCN(C(=O)C(O)Cc2cnc[nH]2)C)CC1 C1(CN(C)C(c2cc(O)n(C)n2)=O)CCN(C(C2CC3CC3N2)=O)CC1 C12(C(NOCCCOCC)=O)CCCC1CN(C(C1CCCC(F)C1)=O)C2 C1(C=O)CCC(C(F)(F)F)N1N1CCC(c2scc(C)n2)C1 c1(C(N2CC3C(CCNC(CCCNC)=O)C3C2)=O)cc2ccc(Cl)cc2nn1 c1(C(N(CC)CC2CC2)=O)sccc1CNC(=O)CN1CCOC1=O Cc1ccnc(C(=O)NC2(C(N3CC4(CCOC4)C3)=O)CSC2)c1N c1(SCCOC)ccc([N+](=O)[O-])cc1C(=O)Nc1cc([N+](=O)[O-])ccc1Br Cc1ccncc1C(=O)NCc1cccc(NC(=O)Cc2ncoc2C)c1 N1(C(c2nc(C)n(C)c2)=O)CCC(C2CC2)C1C(=O)Nc1cccc(Cl)c1C C(=O)(C(C)CC(C)C)NC(C(=O)NCc1c(CC)nn[nH]1)C1CCC1.O C(=O)(CC(O)CC(C)(C)C)NCC1(CC(=O)NCCS(CC)=O)CC1 N1(C(CCC)=O)CCC(C(=O)NCC(C)CN(C)C(c2cnc(SC)s2)=O)CC1 C1(C(=O)Nc2c(C(N)=O)ccs2)CC(F)CN(Cc2ccc(O)c(I)c2)C1 C1(SC)CN(C(c2cnc(-c3ccccc3)o2)=O)CC1NC(c1cscc1F)=O Cc1nc(NC(C2CCC(NC(c3cscc3Br)=O)C2)=O)c(Cl)cc1Cl C(CC(O)CC(=O)N1CCC(NC(=O)C(c2ccccc2F)C)C1C)SC Cc1cc(C2CC2)cnc1C(=O)NCC1CCCN1C(=O)Cn1cnnc1 C(=O)(C1OCCc2c(O)cccc21)NC(C(=O)OCC)Cc1ncccn1 N1(C(CN(C)C(c2ccncc2)=O)=O)CC2CC(C1)C2NC(C1CCSC1)=O N1(C(C(C)OCCOC)=O)CC2(CCC2)CCC1C.c1(C(=O)N)ccns1 C(=O)(CCC(C)NC(=O)CN1CCCC1)NC1(CCCC)CC1 C1(CC)CCC(C(=O)NCC2(C(N)=O)CN(C(=O)CC)C2)O1.CC(F)F c1(C(N2CC(C)C(NC(c3ncccc3N)=O)C2)=O)c(OC(F)F)cccc1F c1(C(=O)NC2CN(C(CSCC#C)=O)C(C)(COC)C2)cc(F)cc(F)c1O n1(CCC(=O)NCC(C2CC2)NC(c2cscc2Cl)=O)cc(Br)cn1 C=CCCC(CC(C)C)C(=O)NCC(C)(C)CNC(C1CC=CCC1)=O c1(CNC(C2CCOCC2)CCOC)cccc(I)c1 c1(C(N2C3CN(C(C(C)NC(C)=O)=O)C(CC3)C2)=O)ccnc2ccncc12 N1(CC)CC(C(=O)N(C)C)CC1=O.C1CC1.C1(C=O)(CCN(C)C)CC1 N1(C(CCC)=O)CCCC(CNC(=O)CN(C2CCCC2)C)C1CC c1(COC)ccc(C(=O)NCC(C(C)C)NC(=O)C)[nH]1.c1csc(=N)[nH]1 CCC(C(=O)N(CC(=O)O)Cc1cn(-c2ccc(F)nc2)nn1)C(C)C Cc1ccc(Cl)cc1NC(=O)CCC1CCCN(C(C2(F)CC=CC2)=O)C1 Cc1cc2nccnc2cc1C(N1CCCC2C1CCN2C(C1CC(F)C1)=O)=O Cc1cnc(CC(=O)NCC(C)(Cn2cccn2)NC(c2cnccn2)=O)s1 C=C=CC(C)C(=O)N1CC2CC1C2NC(c1cc(-c2ccc(F)cc2)c(C)s1)=O N1(C(c2cccc(F)c2)C(=O)NCCCSC)CCC2(CC=CCO2)C1 CCCC(C#N)C(=O)NC(c1ccnn1C)C(=O)NC1C(C)(C)C1(C)C Cc1cccc(C(O)C(=O)NC(C)CCNC(=O)Cc2ccco2)c1 N1(C(C(C)NC(C)=O)=O)CCC(C)C1.c1(C=O)ccnc(OC(F)(F)F)c1.C N1(C(C(C)SCC)=O)CCC2(CCN(C(c3c(C)oc4ccccc34)=O)C2)C1 C1(NC(C2CC23CCC3)=O)COCC1NC(C1(Cc2cccnc2)CC1)=O c1(OC)cncc(C(=O)NCC(C)CN(C)C(C2(CSC)CCC2)=O)c1 c1(C(=O)N)cccc(C=O)n1.C(C)(CCNC(=O)CC1CC1(C)C)OC C1CN(C(=O)CCC2CCCO2)CC(F)(F)C1.c1(C=O)ccc(C(F)(F)F)[nH]1.N CC1(C)CCCN(C(C2(NC(=O)CCSC3CCCC3)CSC2)=O)C1 CC1CCC(NC(c2cnoc2C2CCC2)=O)CN1C(c1cc(O)no1)=O C1(N(C(C(CSC)C)=O)C)CCC(NC(=O)C(CO)N(C)C)CC1 N1(C(c2c(C)noc2C)=O)CC2CN(C(c3c[nH]c(C#N)c3)=O)CC2(C)C1 c1(OC)cc(C(=O)N(C(C)CCNC(C2CCC(C)(C)O2)=O)C)sc1Br C1(CO)CCC2(CCOCC2)CN1Cc1ccc(Cl)cc1F C#CCCCCCCCC(=O)N(CCCNC(=O)CC(C)(C)C)C C(C)(N=c1cccc(S(=O)(=O)N2CCSCC2C)[nH]1)c1scc(CC)n1 CCC(C(=O)NC1CC2CCC(C1)N2C(=O)CCCn1cncn1)C(C)(F)F c1(C(=O)NCC2C(NC(c3cnccn3)=O)C2)ccc(C(F)F)cn1 c1(C(=O)NCCC2CCN(C(C(C)C(F)F)=O)C2)c(Cl)ccc2ccoc12 c1(OC)cc(C)cc(C(N2CCC(NC(C3CCC4(C3)N=N4)=O)CC2C)=O)c1C C(=O)CC(O)C(C)(C)C.c1(OCC#C)ncccc1C(=O)Nc1ccccc1.N N1(C(C2CC(=C)C2)=O)CCC(C)C1CNC(C1(C(N)=O)CCC1)=O S(=O)(=O)(c1ccc2[nH]c(=NCC3CCCOCC3)sc2c1)N1CC(C)OCCC1 N1(C(CCSCC(N)=O)=O)CC(F)(F)CC1CCNC(=O)C=C(Cl)Cl CCC(CC)C(CN=c1[nH]c(=NCCSCCOC)[nH]c2c1SCC2)OC C1(C(N2C(C(=O)NCCOC(C)C)CC2C)=O)CC1C1(C)COC1 N1(C(C(=O)NC)CCCCCO)Cc2ccccc2N2CCCC2C1 N1(C(C(C)(C)CNC(=O)C=CC2CC2)=O)CCNC(=O)C1CCO n1(CC(N2C(C(C)(C)NC(C(C=C)O)=O)CCC2)=O)nc(C)oc1=O N1(C(CCCC(=O)NCC)=O)CCCC12CCN(C(C1(OC)CCCCC1)=O)C2 N1(C(c2ccc(OC)o2)=O)CC(CNC(=O)C2=COCCO2)CC12CCC2 CC1CN(C(C2CCOC2(C)C)=O)CC1CCNC(=O)CCc1cscn1 C=CCCC(C(=O)NCCC(C)C(F)(F)F)NC(=O)C(CC(=C)C)OC S(=O)(=O)(c1ccccn1)N1C(C(=O)NC(c2cc(C)cc(C)c2)C)CC1 c1(C(N(CCC)CCNC(C2CC(F)(F)CS2)=O)=O)cccc(C#N)c1C Cc1cc(C#N)sc1C(N1CCCC1C1(C)CC1)C(=O)NCCCOC(F)F C1(NC(=O)COCC2CC2)CC2CCCC2C1.c1(C=O)nnc2ccccn12.N c1(OC(C)C)ccc2c(c1)CN(c1ccnc(NC3CCC=CCC3)n1)C2 C1(NC(C(C)c2cccs2)=O)CC2CC(C1)CN(C(=O)CN1CC(C)(C)C1)C2 c1(CC(=O)N(CC=O)C)ccn(C)c1.C(CCN(CC)C(N)=O)N(C)C c1(COC(c2cn(C3C(OC)COC3)nn2)=O)c(C)nc2ccccn12 N1(CCNC)CCN(CCN(C(=O)CC2CCC3CC23)C)CC1.c1cc(C)nn1C c1(C(=O)NCCC2CCC(NC(=O)CO)C2)cc(Cl)c(N2CCCC2=O)c(Cl)c1 c1(CC(=O)Nc2ccc(CCOC(C)C)cc2)ccc(C2=CCCCC2)c(F)c1 c1(C(N(C2CCN(C(c3nc(C)no3)=O)C2)CC)=O)ccc(C(C)C)cn1 Cc1cc(Br)c(C(C(=O)NC(C)C)N(C)CCOCCN(C)C)cc1Cl C1(CC(=O)OC)(CC(=O)C2CC2)CCCC1.C1(C=O)CCCSC1.C1CC1.N C1(CC(N2CCC(F)C2)=O)CN2CCN1CC2.C1(COCC(=O)N)CCOC1 C(=O)(C1=CCN(C(=O)Cc2cncnc2)CC1)NCC(CCC=C)O c1(C2C(c3n(CC(C)O)nc(C4CC4)n3)C2)c(Cl)cccc1Cl Cc1cc(C=CC(=O)NCCCCCCNC(C2(Cl)CC2(C)C)=O)c[nH]c1=N N1(C(C(CCC)F)=O)CC(C2CC2C(N2CC(O)(C(=O)OC)C2)=O)C1 Cc1cnc(O)c(NC(=O)CCC2CCN(C(=O)C(O)C3CC3)CC2)c1 C1(C(N(CCCNC(c2c(C)[nH]cc2)=O)C)=O)C2CCC3C(C2)CC13.C1CC1 c1(C(=O)OCc2c(C)nc(C)c(C)n2)c(S(N)(=O)=O)ncn1C N#Cc1cccc(NC(C2C(C3CC3)CCN2C(=O)CCn2cccn2)=O)c1F c1(C(=O)NCCCCCN(C(=O)CC2CCC2)C)cnccc1C1OCCO1 Cc1nc(C(=O)NC2CCN(C(c3cccc(F)c3)=O)CC(O)C2)c(=O)[nH]c1C C(=O)(CC(C(F)F)NC(c1cccc(C)n1)=O)NCC1(OC)CCC(C)C1 c1(CC(=O)NCC2CCN2C(c2c(F)ccc(F)c2O)=O)ccc2c[nH]nc2c1 N1(C(C(=O)NCC)=O)CCCC1CCNC(=O)C(C1CCCCC1)O.C O(C1CCCc2ccccc21)CC(=O)NCC(C(C)(C)C)NC(CC=CC)=O C1(CNC(c2cn3ccsc3n2)=O)CCCN(C(=O)C=Cc2cscn2)CC1 c1(C(=O)Nc2cn(-c3ccccc3)nc2Cc2cccs2)ccc2c(c1)CCO2 Cc1ccccc1OCCC(=O)NC1CCC1NC(c1nccn1C)=O c1(C(=O)NCC23CC(CO2)C3)ccc2cc[nH]c2c1.C1(C=O)CC12CCC2.C c1(OC)cc(Br)cc([N+](=O)[O-])c1NC(C1CCCC(NC)C1)=O.c1cncnc1 Cc1cccc(CC(=O)NC2C3CC(NC(c4ccncn4)=O)CC23)c1 C1COCCN1C(=O)CC1C(C)(C)C1(C)C.C1(CC=O)CC2(CC2)CO1.CN CCC(C)C(O)C(C)C(=O)N1CC2CC1(C(=O)NOCCN(C)C)C2 CCC(CC(=O)N1CCCCC1C(=O)NCc1ccn(C)n1)C(C)C c1(C(=O)NC2C(C)(C)CN(C(c3c[nH]c(C#N)c3)=O)C2)cnc2ccsc2c1 N1(C(Cn2cccc(C)c2=O)=O)CCC(C2CCN(C(=O)C(F)F)C2)C1 CC(C)CCCC(C)C(=O)NCC(C)(F)CNC(c1n[nH]cc1[N+](=O)[O-])=O CC1CCC(CNC(c2ccc(F)cc2)=O)N(C(=O)CSC)C1.c1ncc[nH]1 Cc1cc(-c2cccc(C(C)C)c2)c[nH]c1=NCNC(=O)Cc1ccccn1 Cc1cccn(CC(=O)NC2(C)CCCN(C(C3(C)CCOC3)=O)C2)c1=O c1(C(N2C3CC(C3)C2)=O)ccc([N+](=O)[O-])c(S(N)(=O)=O)c1.CCC(C)=CC=O N1(CC(c2c(OC)cccc2)OC)CCS(=O)C(C)(C)CC1 C1(NC(c2noc(CC)c2C)=O)CN(C(=O)C(O)CCSC)CCC1F c1(CCC(=O)NCCN(C(C2CCC2OC)=O)CC)ccc(Br)c(Cl)c1 c1(Cc2nnc(N3CCC(CCCOC)C3C)n2C)ccc(OC)c(OC)c1 C1(CC=O)CC(C)(C)CN1C(=O)CN1CCC(F)CC1.Cc1nc(C)oc1C.N C1CCC2(CN(C(C3(F)CCCC3)=O)C2)O1.c1(SC)cc(C)c(C(=O)N)o1.C c1(C(=O)NCC(CNC(C2C(C)(C)CO2)=O)O)cc(Cl)c([N+](=O)[O-])[nH]1 CC1C(NC(=O)C=CBr)CCCN1C(=O)CCN(CCCCN(C)C)C C1(NC(C2N(C(CCc3ncn(C)c3)=O)CC=C2)=O)CCN2CCC1C2 c1(C(=O)NC2C(CNC(c3cnc(C)n3C)=O)CCC2)cc2cccc(C)n2n1 C1CC2CCC(C1)N2C(=O)CCN(S(C)(=O)=O)C.c1c(C=O)cnn1C.CS C1CCC(C)(C)CC1.C(=O)(CCOCC(=O)NCCC)OCC.C=O.N C=Cc1cncc(C(=O)NC(CO)CCCNC(=O)CCC(=O)NCC)c1 C1(CNC(CCC)=O)CCN(c2cc(OC)nc(OC)n2)CC1C c1(C(=O)N)cc2cc(C)cc(C)c2[nH]1.N1(C(COCC#C)=O)C(C)CC2CC12 C1(CC=O)CCCS(=O)(=O)C1.Cc1ccc(CCNC(=O)C=C(Cl)Cl)cc1.N CCCCC(CC(=O)NCCC1CCOC1(C)C)NC(=O)COCCC(C)C n1(CC)c(C(=O)N(CCCCC(=O)NCC2(C(N)=O)CC2)C)cnc1O C(c1ccc(C)cc1C)=CC(=O)NC(CNC(CC(CC)OC)=O)(CC)CC N1(C(c2ccc(CSCC(C)C)cc2)=O)CCC(C2(O)CCCC2)CC1 N1(C(C(F)=CC)=O)CCCC12CCN(C(=O)C1CCc3nccn31)C2 c1(OC)ccc(CC(=O)NCC2CN(C(c3ccc[nH]3)=O)CC2(F)F)c(C)c1 N1(C(c2c(C)snc2)=O)CCN(C(C2CCCN(C)C2)=O)C(C2CC2)C1 C#CCCC(O)C(=O)N1CCC(CO)(CNC(=O)CC(F)(F)F)CC1 Cc1ccc(C#N)c(N(C)CC2CCCN(C(C3(O)CCCC3)=O)C2)n1 N1(C(c2ccc(CNC(C(C)=C3CCCC3)=O)s2)=O)CC(C)CCC1C C1(C(=O)NC(C)CCNC(=O)C(c2ccc(C#N)cc2)C)CCc2n[nH]cc2C1 c1(C(=O)NCC(CC)(C)NC(=O)CCCC2CCC2)ccc(-c2ccsc2)nc1 N1(C(Cn2ncc(C)cc2=O)=O)CCC2C(CCN2C(=O)CSc2cccs2)C1 N#CC1(C(N2CCOC(CNC(c3nnc(O)nc3O)=O)C2)=O)CCCCC1 Cc1cc(N2CCCC(C)(NC(=O)C(C)C(C)O)C2)nc(-c2ccccn2)n1 CCCCCCC(CC)(CC)C(=O)N1CCC(NC(C2CCOC2C)=O)CC1 c1(Nc2ccc(NS(c3cnn(CC)n3)(=O)=O)cc2C)nc2c(C)cccc2s1 C1(NC(c2cnc(C)[nH]2)=O)CCC2CCN(c3cc(O)nc(=O)n3C)C1C2 c1(OCC(=O)NC2CC(NC(C(c3ccccc3)SC)=O)C2)ccccc1F N1(C2CN(C(c3ccn(SCCOC)n3)=O)C2)CCN(C(c2ccco2)=O)CC1 C1(NC(C(CCC)O)=O)CCCCCC1NC(c1scc(Cl)c1Cl)=O c1(C=O)c(N)cc(F)cc1F.N1(CC(C)C)CC(C(=O)NC2CC2)CC1=O.C c1(C(N2CCC(Cn3cc(CO)nn3)CC2)=O)ncnn2cccc12 N1(C(C(C)N(C)C)=O)CCN(C)CC1C(=O)NCC1CCN(C)C1 C1(C2(O)CCN(C(c3cc(Cl)cc4ccncc34)=O)CC2)(NC(=O)CCF)CC1 c1(C(N2CCN(C(c3ccc(C)nn3)=O)C(C)CC2)=O)ccc2[nH]c(=N)sc2c1 C(CC(C)C(=O)N1CCCC1CC(N1CC(CC)(CC)C1)=O)=CC N1(C2CN(C(CC(C)n3ccc(C4CC4)n3)=O)C2)CCN(C(=O)CC2CC2)CC1 N1(C(CC(CC=C)NC(=O)CC(C)(C)CCC)=O)CCCC12CCOCC2 C(=O)C(C1CCCO1)N(C1CCC1)C1CC1.CC(C)=CC=O.CCCCC C1(n2cc(-c3n[nH]c(C)c3C)nn2)CC2CCC(C1)N2C(=O)C(C)(C)C1CCC1 CC1(C)C2CCC1(C(=O)NC1CCN(CCN3CCCC3=O)CC1O)CC2 C(=O)(C(C#N)C(C)(C)C)N1C(C)C(NC(c2conc2C(F)(F)F)=O)CCC1 CCC(F)(F)CC(=O)N1CC(C(=O)NC2CCN(CCCO)C2)(CC)C1 C1CN(C(C2C(C(F)(F)F)C2[N+](=O)[O-])=O)CC1C.c1(CC)nnsc1C(=O)N C1(C(=O)NC2(CO)C(C)CCCC2)C2CCCC2CN1C(=O)C1=C(Cl)CC1 c1(NC(C2C(CC)CCN2C(=O)Cc2cc(C)[nH]n2)=O)cccc(F)c1O C(=O)(C(C)CC(F)F)N(CC(C)N(C(c1cnc(CC)nc1)=O)C)C C(=O)(C1=C(Cl)CCCC1)N(CCN(C(c1n[nH]c(CC)c1Cl)=O)C)C(C)C CC(C)(N=[N+]=[N-])C(=O)NCC1CCCC1C(=O)NC1(c2ncc[nH]2)CC1 C(=O)(C(C(C)CC)OC)N(CCC(=O)NC1(CC=C)CCCCC1)CCO CC1CN(C(=O)NCCCc2ccc(C(=O)N(C)C)cc2)CC(c2ccsc2)O1 C(=O)(C(F)C(F)(F)F)NC1CC(CCNC(C2CC(CC)C2)=O)C1 CS(=O)(=O)CC(=O)NC1CCOC(CNC(C2CNC(=O)C2)=O)C1 C#CC1CN(C(=O)C(CC(C)C)ONC(C2C3CC(=O)CC23)=O)CCN1C N1(C(c2n(C(C)C)cnc2)=O)CC2CCCC2(NC(=O)CCCCC2CC2)C1 C1(C(NOCCC#C)=O)CCCCN1C(c1nn(C)cc1C)=O C(CCC(N)=O)(C(=O)NCC#CCO)n1cc(C(C)N(C)C)nn1 N1(C(c2cc(C)c(C)[nH]2)=O)CC(NC(=O)C(N2CCOCC2=O)C)C2(CC2)C1 c1(C(N2CCC(C(N3C(C(=O)OC)C3)=O)CC2)=O)c[nH]c2ccccc2c1=N c1(C(=O)NCC(CCNC(C(CCC)OC)=O)(C)C)cn(CCO)c(=O)nc1O N1(C(C(CCN(C)C)(C)O)=O)CCN(C(=O)CC2CC3CC3C2)C2(CC2)C1 C1(C(C)C)CN(C(=O)CC2(C)CC2)CCN1C(=O)Cc1ccc(F)cc1 c1(OC)ccc2c(c1)CC(C(=O)NCCC(C)NC(=O)C1=CCCC1(C)C)O2 n1(CC)ncc2c1CCCC2Nc1nc(N)cc(=N)[nH]1 C1(NC(C23N(C(CC4CN(C(C)=O)C4)=O)CCC2C3)=O)COCC(C)(C)C1 Cc1cc2[nH]c(C(=O)NC3CC(C)C3)cc2s1.c1(C=O)cnc(C(N)=O)cn1.N C1(C(C)C)CN(C(C2(N(C)C)CC2)=O)CCCN1C(=O)CCc1cncn1C CCCC(CCC)CC(=O)NC(C1(O)CCN(C(=O)Cn2nnc(=N)[nH]2)CC1)C C1(CCCNC(CCCOCCC)=O)CCN(C(=O)CN2CC=CC2)CC1 Cc1cc(O)c(F)cc1NC(=O)CC(C(F)F)NC(=O)C(C)(C)CN(C)C CC1(C)C(C(=O)NCCCC(=O)N2CCC(CC(F)F)C2)C1C#N C(=O)(C(=O)C(C)CC)NC1CC(CCC(=O)N(CCCCCC)CCO)C1 N1(C(c2c(COC)cccn2)=O)CCC2CN(C(c3ccoc3C)=O)CC2C1 C(=O)CS(=O)(=O)C(C)C.C1(NC(COCC(=C)C)=O)CC(O)(C)C1.N C1(C2CC2)(NC(c2ccc(CO)nc2)=O)CCN(C(=O)C=C2CCCCC2)C1 CCCCC(O)C(C)C(=O)N(CCC(=O)NCC(C)(O)C1CC1)CCO C12(CNC(c3nccc(C)c3)=O)CC(C1)C(C)O2.C1(C=O)CC12CCCC2.N C(=O)(CS(=O)(=O)CCCC)NC12CC(CNC(CC(C=C)CC)=O)(OC1)C2 C(=O)(C(CC)CCCCC)CC(N1CC(CCCC)C1)=O.C1CC(C#N)C1 CCC(F)(C(=O)OC)C(=O)N1CC(NC(=O)CCC(=O)N(C)C(C)C)C(F)C1 C1(CS(=O)(=O)NC(=O)NC)(C(C)C)CC(C)(C)C1.C1CCC1N(C)C.C Cc1ccc(CNC(=O)C(C)CC2CC2)cc1F.C1(CC=O)CCCC(=O)N1 c1(C(=O)NCCN(C(CC2CN(C(C)=O)C2)=O)C2CC2)cnncc1O CCCCC(O)CCC(=O)NCCCC(C)NC(=O)CCCS(C)(=O)=O N(C1CCCc2cc(CNC(=O)C(C)O)ccc21)C(Cc1ccc(C)nc1)=O C1(NC(C(c2ccccc2)SC)=O)CN(C(c2ccc(N)c(F)n2)=O)C(C)(C)C1 c1(C(=O)NCCC(C)NC(c2cccc(-n3cncn3)n2)=O)ccccc1C#N Cc1nn(C)c(C)c1.n1(CC2(N(C=O)C)CC2)cc(CCO)nn1.C(C)(C)C C1(C(=O)N)CCCNS1(=O)=O.C(c1ccccc1)=CCCC(N1CC(F)C1)=O.C CC(C)(CC(F)(F)F)C(=O)NCC1CN(C(=O)CC2CC3(CC3)C2)C1 C1(CNC(C2(C3CC3)CCCO2)=O)CCC(C(N2CC=CC2CF)=O)C1 C=CC1(O)CN(C(=O)CCN(C)C(C2CCCC(C)C2)=O)C1 CC1(C)CCCC(C(=O)NCC2(NC(c3cccc[n+]3[O-])=O)CCOCC2)O1 N1(C(C(CC)(C)COC)=O)CC(CNC(=O)Cc2ccco2)OC(C)(C)C1 C1(C)CCN(C(C2(F)CCCC2)=O)C1.C(Cc1ccccc1)(C=O)NC(C)=O.N c1(C(C)NC(C2(COC)CN(C(=O)C=CC3CC3)C2)=O)ccccc1O C1(C(=O)N(C)Cc2ncn(C)n2)(NC(C(C)C2CCC2)=O)CCOCC1 CCCC(C)C(=O)NC1CCCC1(C)CNC(=O)C=C1CCOCC1 CC(C)(C)C(O)C(=O)NCC1CC(NC(C2CC2c2ccccc2)=O)CCO1 CCC(C)C(C)C(=O)NC(CN(C)C(C1CCC(C(N)=O)CC1)=O)(CO)CO c1(OCC=C)cc(Cl)ccc1C(=O)N.C1CC2CN(C(=O)C(C)CCC)CC12.C C(CC(O)CNC(=O)CC1(n2ccnc2)CC1)NC(C(C)C1CCC1)=O c1(C(=O)NCC(CNC(C(C)(C(C)C)OC)=O)F)ccc2ncsc2c1 C1(SC)CN(C(=O)C(C)C2CCC2)CC1NC(=O)C(c1ccc(C)s1)C c1(OC)nc(Cl)ccc1C(=O)N.C1CCN(C(=O)CNS(N)(=O)=O)CC1C.C C=CC(CCC)CC(=O)NC1CCCC1C(=O)NC(c1cccc(C)n1)C N1(C(C(CCC)(F)F)=O)CC2CCN(C(c3cccc(=O)n3C)=O)CCC2C1 C(C(C)CC(=O)NC1CC(O)(CO)C1)NC(C1(CCC)CCC1)=O Cc1cccc(C(=O)NC2CC(N(C(=O)CSCCC#N)C)C2)c1C N1(C(c2cc(C(C)C)on2)=O)CC2C=CC1C(C(=O)NCC1CCOC1=O)C2 C=CCCCCCC(=O)NCCC(O)CNC(c1cc(C(C)C)nc(O)c1)=O C1(C(=O)N)CCS(=O)(=O)CC1.n1(CCC=C(C)C)cc(CN2CCCC2)nn1 c1(NC(C2C(NCc3ccc(OC)c(O)c3Br)C2)=O)cnc2c(ccn2C)c1 Cc1cccc(Cl)c1OCC(N1CCC1CNC(=O)CS(N)(=O)=O)=O Cc1cccc(Br)c1C(=O)NCC1(C)CCC1.C(=O)(C(O)CC1CC1)N c1(C=O)c(C)noc1CCC.C1(O)(CC#C)CC(C(=O)NCC2CC2)C1 c1(C(=O)Nc2cncc(COC(C)C)c2)cc2c(C3CC3)cccc2[nH]1 N1(C(c2cnc(CC(F)(F)F)s2)C(=O)NC(CC)(C)C)CCC(C2CCCC2)C1 N1(C(CCC#C)=O)CCC2C(CCN2C(c2cc(F)c(F)c(F)c2F)=O)C1 C(=O)(C1=C(Cl)CCCC1)N1CC(NC(c2c(OC)c(C)ncn2)=O)C(C)C1 C(=O)(C(C)C(O)C(C)C)NCCNC(c1c(C)ccs1)=O CCCC(C)(CCCC(=O)OC)NC(C1CC(C)(F)C1)=O C(=O)(CC(C)C(C)C)NCC1C(NC(c2ccc(CCCC=C)cc2)=O)CC1 C1(C(=O)NCC(C)CNC(=O)CC(C)(C)F)Cc2ccccc2OC1C(F)F C1(O)CN(C(=O)CC(c2cccs2)n2cccc2)C1.C1(C=O)CC1C(F)F.N c1(C(=O)OC)c(NC(=O)COC(C2CCc3n[nH]cc3N2)=O)sc2c1CCC2 CC1CC(CC(=O)NCCCC2CCOCC2)CN1C(c1ccncn1)=O c1(C(=O)NCC2CCC(NC(C=CCC)=O)C2)ccnc(P(C)(C)=O)c1 c1(N2CC(OC)C(O)C2)ccc(Br)c(S(=O)(=O)NC(C)Cc2ccncc2)n1 c1(C(=O)N(c2ccccc2)CC)cc(-c2cnn(CCCO)c2)c2[nH]ccc2c1 CC1(C)CCCOC1CNc1ccc(C(=O)O)cc1 c1(CC(=O)NCC2(C)CC(NC(c3ccc(CC)s3)=O)C2)ncccc1C c1(OC)cn(C)c(C(N2CC3CC2CN(C(=O)CC2CC4(CC4)C2)C3)=O)cc1=O C12(C(=O)NCC(C(C)C)O)CC1CCN2C(c1ccoc1Cl)=O N1(C(C=C(C)C)=O)CCC(C(=O)Nc2cc(C)ccc2O)C12CCC2 C1(CNC(C=CC)=O)CCC(C)CN1C(=O)CCc1cc(Br)ccc1Cl C#CCC(CC(F)F)NC(=O)C(C1CC=CCC1)NC(=O)CCn1ccnn1 c1ccc(Cl)cc1.C1(NC(C=CC=CCC)=O)CC(NC(=O)CS)C1 C12(C(=O)NCc3c(C)ccc(O)n3)CCCC1CCN2C(C1SCCS1)=O N1(CC)CC2CC1CN2C(C1CC(C)CN(C(c2nccn2C(C)C)=O)C1)=O C1(C(N(C)Cc2c(C)nsc2)=O)CCC(C(C)C)N1C(=O)CC1(C)CC1 N(C(=NCCc1cccs1)NC1CC(OC(C)C)C1)CC1CCC(C)(CC)O1 O=C1NCc2c(C(=O)NCC3CCCC3)cccc21.C(=O)C1=CCS(=O)(=O)C1 n1(CCCC#C)c(N2CCOC(C3CC(F)(F)C3)C2)nnc1-c1ccco1 N1(C(c2c(CC)ocn2)=O)CCN(C)CC1.C1(C(N2CCC2)=O)C2CC2C2CC12 CC1=C(C=O)CCC1.C1CN(C(c2cc(C(N)=O)cs2)=O)CCC1C(F)(F)F.N c1(C(N2CC(F)C2)=O)cnnc(C2CC2)c1.c1(C(C)C)ccoc1C(=O)NC Cc1cc(C)c(C(=O)NCC(C(=O)NCCN2CC3CCC2C3)N(C)C)cn1 N1(C(=O)C=Cc2ccsc2)CCCC(C2CCN(C(=O)CC=C(Cl)Cl)C2)C1 Cc1cccc(C=CC(=O)NCC#CCNC(=O)Cc2cncc(C)c2)c1 C(c1ccc(C)o1)=CC(=O)NCC(CN(C(C1N(CC)CCC1)=O)C)C Cc1cc(C(=O)NC(C2CC(NC(C3(CO)CCOCC3)=O)C2)C)cc(C)c1F C(=O)(C(CNC(=O)C)C(C)C)Nc1cn(C(C)C)nc1.C(=O)C1CC1.N C(=O)(C(F)CCC(C)C)NC(CCOCC)C(=O)NC1Cc2cccnc2C1 C1(C(=O)NCC2CCC(NC(c3nncc(OC)c3)=O)C2)CCCCNC1=O Cc1ccncc1C=CC(=O)NC1CCOCC1NC(=O)C(O)C(F)F c1(C(N2C(CNC(C3C(OCC)C3)=O)COCC2)=O)cccc2ccsc12 CCC(C)(C)C(O)C(=O)NC1CCCCC1NC(C1CCC(=O)N1)=O c1(NC(=O)NC2(C(=O)OC)CCC2)ncnc2cc(F)ccc12 c1(C(N2CCC(C(C=O)C)CC2)=O)cc(C)cc(Cl)n1.C1(C(=O)OC)CCC1.N C(=O)(CCCc1cnn[nH]1)NC(CNC(CCSCC)=O)COC c1(CC)cc(C(N2CCCCC2C(C)NC(C2(C(F)F)CCCC2)=O)=O)ncn1 CC1C(NC(=O)Cc2nncn2C)CC2CCC1N2C(c1ccc(=O)n(C)n1)=O C(=O)(CC(C)(C)N(C)C(c1ncn(C)c1C)=O)NC(C1CCCO1)CC c1(C=O)ccnc(C2CC2)n1.c1(CCCC)nc(C(=O)NCC2CC2)cs1.N C1(NC(c2nc(CCCCC)sc2)=O)CC(F)CN(C(c2cc[nH]c2CC)=O)C1 CCC(F)(F)C(=O)NC1CC2(C1)CC2C(=O)NCC(O)COC(C)C CC(C)(O)C#CC(=O)N1CCC(CC(=O)NCc2cc(F)ccc2O)CC1 N1(C(CC(=O)OC)=O)CCCN(C(c2n[nH]c(C)c2C(F)(F)F)=O)CC1 C1(COC)CN(C(C2(c3n[nH]cc3C)CC2)=O)CCN1C(=O)Cn1ncnn1 Cc1cc(C(F)F)ccc1C(N1CC(N2CCC(O)CC2)C1)=O N1(C(CC(CCC)C)=O)CCC2CN(C(c3sccc3S(N)(=O)=O)=O)CC12 C12(C=O)CCCCC1CS(=O)(=O)C2.S(=O)(=O)(CC=O)NC.C1(CC)CC1.N N1(C(C2CC(=O)NC2)=O)CCN(C(=O)C2=CCCCO2)C(CCO)C1 C(C(C)C(C)C(=O)N1CCC(C(C)CNC(c2cnc(O)n2C)=O)CC1)OC C1(NC(C=C(COC)C)=O)CC(F)C1.C1(c2ccccc2)(CC=O)CCCO1 C(=O)(CCCC(C)(C)C)NCC1CN(C(c2cc(C)c(O)nn2)=O)C2(C1)CC2 c1(OC)ncc(C)c(C(=O)NCC(C)N(C(=O)CCc2nc[nH]n2)C)c1Cl c1(CC)nn(C)c(Cl)c1C(=O)NCCN1CCN(C)CC1.C1CC(C)(C)CO1 c1(C(N2CCC2)=O)ccc(Cl)c(S(N)(=O)=O)c1.c1(COC)nc(C=O)cs1 N1(C(c2n(CCC)ncn2)C(=O)NC(C)CC)CCn2cc(C)nc2C1C C1(CC=C)(NC(C2CC3C=CC2C3)=O)CCN(C(=O)CCC(C)OC)CC1 C1(C(=O)NC(c2cc(C)on2)C)(CC)CCN(C(C2C=CCC2)=O)C1 O=c1cc(N2CCc3c(Br)ccnc3C2)c2cnccc2[nH]1 Cc1cc(CNC(C2CNC2(C)C)=O)ccc1S(C)(=O)=O c1(C(=O)OC)cn(CC(=O)NCC(C)(C)CN(C)C(C2CCCC2)=O)nn1 c1(CN2CCC(C(=O)NCc3cccc(OC)c3)C2)c(O)ccc(Cl)c1Cl CC(C)CCC(C)N(C(=O)CC(O)CNC(=O)Cc1csnn1)C CC1(C)CC(NC(=O)COC(F)(F)F)CN(C(=O)C(c2ccccc2)F)C1 N1(C(C2(C)CCCC2)=O)C2CCC1CC(NC(=O)CSc1nncs1)C2 C1(C(=O)NCC(C)NC(c2cccc3c2COCC3)=O)CCn2c(O)nnc2C1 CC(CCCNC(c1nccn1C)=O)NC(c1cc(C2CC2)ns1)=O CC1CC(C(=O)NCC(C)N(C)C)CN(C(c2cnn[nH]2)=O)C1 C#CC1(C)CCN(C(=O)C(CCC)NC(=O)CCOC2CCC2)CC1 N1(C(c2ccc(C)s2)=O)CCC(C2(NC(=O)C=CC3CCOC3)CCC2)CC1 N1(C(C(CC)CC)=O)CCCC(CNC(=O)CNC(c2ccco2)=O)CC1 c1(C2(CC=O)CCC2)ccccc1.C1(C2(C(NC)=O)CC2)CCCO1.C1CC1 S(=O)(=O)(c1ccc(C(=O)O)o1)N1CC(C(F)(F)F)(CC)OCC1 c1(OCC(=O)NCCC(C)N(C)C(c2ccc(Br)o2)=O)nc(O)nc(O)n1 c1(C(=O)NCC(CC)NC(=O)C(F)CC2CCOC2)cnc(SC)n1C C12(COC)COC(C=O)(C1)C2.c1(C(C(N2CCCC2)=O)C)cc(C)oc1C.N c1(C(NC2CCN(C(c3ccsc3)=O)C2)=O)cc(S(C)(=O)=O)cc(C)c1C.C N1(C(Cc2c(SC)cccc2)=O)CCN(C(C2CCSCC2)=O)C(C(F)(F)F)C1 c1(NC(=O)CC2CN(C(c3ccc(F)cc3Cl)=O)C2)cc(F)cc2[nH]ccc12 c1(CC)cccc(C2CC2)c1.Cc1ccsc1.C(=O)(C=O)N(CCN(C)C)C c1(OC)nc(C)ncc1C(=O)NCC1CCC1.N1(C(C(=O)N)C)CCSCC1 Cc1ccc(S(=O)(=O)NC(C2CCCN(C(=O)Cc3ccccc3)C2)=O)cc1Cl c1(C(=O)OCC(C)C(C)(F)F)noc2c1CCc1sccc1-2 C(=O)C(C(C)(C)C)N(C)C.C1(C(N(C)CCOCC)=O)CCC12CCC2.N N1(C(C(F)OC)=O)CCOC(CCNC(=O)C)C1.c1cccc(C(F)(F)F)c1 C1CN(C(=O)C(C)N(CC(F)(F)F)C)CCN1C(=O)C=Cc1ccc(C)o1.C C(=O)(C1=CCC(C)(C)CC1)NC(CC(=O)NCC(CCC)C)COC N1(C(CCN(C(C)C)C(C2C3CC4C(C3)C24)=O)=O)CC=C(CO)CC1 C1(C(N2CCC(NC(c3cccc(C)n3)=O)C2C)=O)CCn2c(C)cnc2C1 C1(NC(CC2CC(NC(CCc3cnc(C)o3)=O)C2)=O)CC(C)(C)OC1(C)C c1(-c2nc(C(C(CC)C)C)n(-c3cnnn3C)n2)ccc2ccccc2n1 c1(CN(C(=O)C)CC)ccc(C(C)(C)C)cc1.c1nnnn1C1CCCC1.N C1(C(=O)NC2C(C)COCC2)CCC2CCC1N2C(C12CCC(CO)(CC1)C2)=O C1(C(=O)OC)CCC(OC(=O)NCc2noc(C3CCCC3)n2)C1 c1(C(=O)NCC(CNC(CC(C)OC)=O)O)cn2cccnc2n1 N1(C(CCC(C)OC)=O)CCCC(CCNC(C2CC3CC3CC2C)=O)CC1 c1(C(N(CCCCN(C(=O)CSS(C)(=O)=O)C)C)=O)cc2c(nn1)CCC2 C(C(C)(C(C)C)C(C)C)NC(C1C(CC)N(C(=O)CCC2CCOCC2)CC1)=O C1(C(=O)NC2(CC)CN(C(c3cnc(S)nc3)=O)C2)CN2CCCN1CC2 N1(C(c2c(C(C)C)ocn2)=O)CCC2CN(C(c3cc(Cl)n[nH]3)=O)C2C1 C1(C(=O)NCc2c(C(=O)NC(CC)(C)C3CC3)scc2)Cc2ccccc2C1 N1(C(c2ccc(C)c(C)n2)=O)CC2CC(O)C1C2NC(=O)C(C)(F)F C1(C)(CNC(CCc2onc(C)n2)=O)CCCN(C(C23CC(F)(C2)C3)=O)C1 C1(C)(COC)C=CCN1C(=O)CC(O)CNC(=O)CC1CCC(=O)CC1 C1(NC(C2C(NC(Cc3c(C)cnn3C)=O)CCCC2)=O)CCN2CCC1C2 N1(C(c2occ(OC)c(=O)c2)=O)CC2CC3CC2C1C3NC(c1csc(Cl)c1)=O c1(C2C(C(=O)N)C2)ccc(C#N)cc1.Cc1cc(C(=O)NC2CC(C)C2)cs1 c1(C(=O)NC2C(NC(C(C)SCC)=O)CCCC2)cnc2[nH]nc(O)c2c1 n1(CC(N2CC(C)CC2(C)C)=O)ncc2ccccc12 c1(OC)ccccc1C1CCN(C(=O)Nc2csc(Br)c2)C1 C#Cc1ccc(C(=O)NCCOC2CCN(C(C3(C)CC3C)=O)C2)c(C)c1 c1(C(=O)NC(CC(C)NC(C(C=C)O)=O)C)ccc(C2(OC)CCC2)cc1 C1(CC(N2CCN(C(c3cncnc3)=O)CC2CF)=O)CC2(CCC2)CCO1 Cc1ccc(Cl)cc1C(=O)NC1CC2CC1CN2C(c1[nH]ncc1C#N)=O C1(C)(COC)CCCN(C(C23CC(CO2)N(C(c2c[nH][nH]c2=N)=O)C3)=O)C1 C1(C(=O)OC)C(C(=O)OC)C2CCCC1N2C(=O)Nc1cnc(C2CC2)nc1 c1(NC(C(=O)NCCc2cnc(C)s2)=O)c(C)nn(C(C)(C)C)c1C C=CC(C)(O)C(=O)N1CCC(OCCNC(=O)C(C)OC2CCOCC2)CC1 C1(COC)CN(C(c2cnc(Cl)[nH]2)=O)CCN1C(=O)CCc1ccccn1 Cc1cc(Cl)ccc1OCC(=O)NC(C1CCN(C(C2(Cl)CC2)=O)CC1)C c1(CN2CCC(NC(C(N)=O)=O)C2)c[nH]c2cccc(C(=O)O)c12 C1(C(N(CCNC(C(CCC)CC)=O)CC)=O)CCC(N=[N+]=[N-])CC1 N1(C(C)=O)CCC2CCC(C1)N2C(c1cc(CO)c(C)o1)C(=O)NC1CCCC1 C1(C(=O)NC(C2(O)CCN(C(C3CCOC3)=O)C2)C)CCC(N=[N+]=[N-])CC1 Cc1cnc(C(=O)NCC2(C)CCCN2C(c2cnn(C)c2F)=O)cc1Cl N1(C(COCC=C)=O)CCOC2(CCN(C(c3noc4cc(F)ccc34)=O)C2)C1 CC(C)CS(=O)(=O)CC(=O)N1CCCC1CN(C)C(c1cc2n(c1)CCSC2)=O C1(C=O)C2CCCC2CN1C(=O)CC1C=NN(C)C1=O.CC(C)COCC.N Cc1nn(-c2ccncc2)cc1C(N1CCC(C(NS(N)(=O)=O)=O)CC1)=O C(C(=O)NCCN(CC(C)O)CC)N(CCC)C c1(NCC2CC(NC(c3cn(CCC)nc3C)=O)C2)ncnc2cccc(Br)c12 N1(C(C=CC(C)(C)NC(C2CCSCC2)=O)=O)CCC(F)(F)C1 C1(C(=O)NCC(C)CN(C(=O)C(F)(F)C(C)(C)O)C)COc2ccccc2C1 N1(C(Cc2c(C)nc(S)s2)=O)CC(NC(=O)CC(C)(C)C(F)F)CC12CCOC2 N1(C(C(CC)F)=O)CC(F)(F)CC1CCNC(c1ccco1)=O.n1(C)cccn1 N1(C(C(C=C)(C)C)=O)CC2CC(CNC(C3CCC(C)CC3)=O)C2C1 C(=O)(CCCC(C)(C)C#N)NCC(CC(=O)NCCCCC#C)C1CCC1 Cc1ccc(C(=O)NC2CN(C(=O)CC3NC(=O)NC3=O)CC2(C)C)c(O)c1 C1(C(=O)NC2C=CC(C(N(CC(C3CCC3)OC)C)=O)C2)COCCN1C c1(C(N2CCC(C(C)NC(c3n[nH]cc3I)=O)CC2)=O)ccc(C#N)cc1Cl C(=O)(C(C)(C)CCCNC(=O)Cc1coc(C)n1)Nc1c(OC)c(F)ccc1 c1(OC)ccc(CN2CCOCC(NC(=O)C(C)O)C2)c(Br)c1OC C(=O)(C(C)(C)S(C)(=O)=O)N1CC=CC(NC(C2C(C)OCC2)=O)C1 C1(NC(C(CCC)N(C)C)=O)CC2(C1)CC(NC(c1cnn(C)n1)=O)C2 C(=O)(CC(C)CC(F)(F)F)NCCC(=C)CNC(c1cc(C)c[nH]1)=O C1(CNC(=O)CNc2ncccn2)CN(C(c2occc2Cl)=O)CC12CC2 C1(C)(C(N2CCN(C(=O)NC)CC2)=O)CCCN(C(C)CN2CCCCC2C)C1 C1(CNCC2CCC(c3ccccc3)O2)CCC2(CCOC2)O1 N1(C(c2c(C)ccnc2)=O)CCOCC(C(=O)NCCSC(C)(C)C)C1 N1(CC(=O)N(C2CCCN(C(=O)C3=COCC3)C2)CC)CCCCC1=O Cc1cn(C)cc1C(=O)NCC(C1CCN(C(C2(C)CSC2)=O)CC1)O c1(C(C)C)cc(CC(=O)NCC2(NC(c3csc(S)n3)=O)CCCC2)on1 Cc1ncccc1C(=O)NC(C(N1CCCCC1CN(C)C)=O)c1cccs1 CC(C)CCCC(=O)NCC(C)CNC(C1CCCCN1CC(F)F)=O c1(C(=O)NC2CCC(F)(CNC(CCC=C)=O)C2)ccn2cncc2c1 CC(c1cccs1)=CC(=O)NC12COC(C)(C1)C2.c1(CC(=O)N)cscn1 C1(NC(N2CCCC2c2nc(C(F)F)no2)=O)CC(=O)N(C2CNC2)C1 CCCC(C(=O)NC)NC(=O)C(C1CCCO1)NC(c1cc(C)sn1)=O n1(CCC(=O)NCC(C)NC(c2c(C)noc2)=O)nc(C)c(C)c1C C1(NC(CSCCC)=O)CCC(NC(=O)CC2(CCOC)CCCC2)C1 N1(C(c2c(CC)occ2C)=O)CCCCC(NC(c2ccc(Br)cc2)=O)C1 n1(CC(=O)NC2CN(C(=O)C=CC3CCC3)C3CC23)cc(F)ccc1=O C1(C2CCC2)(NC(c2nnnn2CC2CCOCC2)(CC)C2CC2)CC1 C(=O)(C1=CC2CCCC12)NC(C1CCCC1)CNC(CCC(=C)C)=O CC1CN(C(C2CC3(CC3)CO2)=O)CC1NC(=O)CN1CCN(C)CC1 CS(=O)(=O)CC(=O)N1CC(NC(C23COCC2C3)=O)C(c2ccccc2)C1 N1(C(c2cc(OC)no2)=O)CC(C(=O)NC2CC23CCC3)CC(C)(C)C1 CC1CC(NC(c2cc(C(F)F)n(C)n2)=O)CN1C(c1ccc(CO)nc1)=O c1(C(=O)NC(C2(C(N3CCC(C)(O)C3)=O)CC2)C)cc[nH]c(=N)n1 C(=O)(C(O)C(C)(C)C)NCc1cc(C(=O)NCC#CC)n[nH]1 Cc1cc(C(=O)NC2CC2)ccc1C(C)C.c1(C=O)nn(C(F)F)cc1Cl.C C(=O)(CCCC(C)C)NCC1(O)CN(C(C=C(COC)C)=O)C1 N1(CCC)CCS(=O)(=O)CC1.CCC(C(=O)N1CCCC1C=O)c1ccccc1 CC(C)CCC(F)C(=O)NC(C(N1CC(=O)N(C)C(=O)C1)=O)C1CC1 c1(OC)cccc(C(N2CCC(O)(C(=O)Nc3nc(Br)ccc3Cl)C2)=O)c1Br C(=O)(CCCCC(=O)NCC1C(C)CCCN1C(c1cc(Br)n[nH]1)=O)NC C1(CNC(C(C)c2cncs2)=O)CCCN1C(=O)CCC1CC1 C1(C(=O)NC(CCN(C(C(COCC)C)=O)C)(C)C)CCOC1(C)C Cc1ccc(C(=O)NC2CN(C(c3c[nH]nc3C)=O)CC2C)cc1C1CC1 C1(CNC(CC(CC)C)=O)CCCC2(CN(C(c3cc(F)cnc3Cl)=O)C2)O1 C(=O)(C1=Cc2ccccc2OC1)NCCNC(=O)Cc1cc(Cl)cc2c1OCC2 C(=O)(C(N=[N+]=[N-])C(C)C)NCC1CCC(C(N(CC(CC)O)C)=O)CC1 c1(SC)c(C(=O)NCCC2(O)CN(C(=O)C(C)C3CCC3)C2)cccc1F Nc1cc(Cl)nc(C(N2CC(NC(=O)CC3CCOC3)CC(F)C2)=O)c1Cl CC(C)C(CC1CCCCC1)NC(=O)COC1CCC1.c1(C=O)cc(Cl)no1 C(=O)(C(C)C(O)C(C)C)NCC(CCCC)NC(=O)CCNC(=O)COC c1(OC)ccc(-c2cncc(C(=O)N(C3CC3)Cc3csnc3OC)c2)cc1 N1(C(C(C(C)C)OCC)=O)CC(C)N(C(=O)C(C2CC(F)(F)C2)O)C(C)C1 c1(C(N2CCCCCCC2C)C(=O)NCCOCC)ccc2c(c1)ncn2C c1(OC)ccc(CN(C=O)CCNC2CCSC2)c(C)c1OC c1(C(=O)NCCCNC(c2cncc(COC)c2)=O)cc(Cl)c(Cl)n1C C1(n2cc(CNc3c(C#N)c(Cl)ns3)nn2)CC2CCCC(C1)N2C1CC1 CCC(CC(=O)NCC(C)N=[N+]=[N-])NC(c1ccnc(C)c1)=O c1(CC2N(C(C3C(C)C3)=O)CCC2)nc2ccccc2[nH]1 C1(C(=O)NCC(C(=O)Nc2cccc(OC)c2)C)CCCC12CCC2 c1(C(=O)NCC2C(C)(C)CN(C(=O)Cn3ncnn3)C2)cnc2[nH]ccnc1-2 C1(C(=O)NCCOCC(C)C)CCN(C(=O)CCc2ccsc2)CC1 C#CCC(CC(=O)NC1CN(C)CC12CC2)NC(c1cnc(Cl)s1)=O C(CC(=O)NCCC1CN(C(c2cc(O)n(C)n2)=O)C1)(C(F)(F)F)OC.O CCCCC(F)C(=O)NCCCCC(=O)Nc1cc(Cl)ccc1O C=CC(CCC)CC(=O)NCC1(NC(c2cc(F)ccc2CC)=O)CCC1 c1(CC(=O)N(C(CNC(COCCC)=O)C)C)ccccc1S(C)=O Cc1cc(F)cc2[nH]c(C(=O)N(C(C)CCNC(=O)CCn3cccn3)C)cc12 CCC1=NOC(C(=O)NCCC2(O)CCN(C(=O)CS(C)(=O)=O)C2)C1 Cc1ccc(C(C)C)cc1C(N1CC(NC(c2csnn2)=O)CCC1C)=O c1(OC)cc(CCC(N2CCCCC(NC(c3ccon3)=O)C2)=O)ccc1Cl C1(C(=O)NC(C(N2CC(CS(C)=O)C2)=O)c2cccs2)CCC2(CC1)CC2 Cc1cc(C(N2CCCC(NC(=O)CC(C)C(F)F)CC2)=O)c(C)cn1 N1(C(C(CC)(F)F)=O)CC(CNC(C2(C(=O)OC)CC2C)=O)C2(CCC2)C1 N1(C(CCNC(CC(C)C)=O)=O)CCN(C(C2COCCOC2)=O)C2COCC12 C1(CN(C)C(c2cc(CCO)on2)=O)COCCN1C(c1cocn1)=O c1(CNCC2CCCN(C(C(CC)(C)O)=O)C2)cc(Br)cc(I)c1 CC(CC(=O)N1CCC(N(C(=O)Cn2cc(CO)nn2)C)C1)SC C(=O)(CC(C)(C)C(F)F)NCC(CC(F)(F)F)NC(c1cc(C)oc1)=O C(C)(C(C)(C)C(=O)NOCC(C)(C)C)NC(C1CCN(CC)C1)=O c1(C(C)NC(=O)CC2CCCN2Cc2csc(Br)n2)ccc(I)cc1 c1(C(N(CC(O)CN(C)C(c2c[nH]c(=O)cn2)=O)C)=O)cc2c(cn1)OCCC2 N1(CC(=O)NCC2CCCN2c2ccnc(-c3nccs3)n2)CCCS1(=O)=O c1(C(N2CCCC(N(C(C(CC)COC)=O)C)C2)=O)cc(N)ccc1Br N1(C(=O)NC(CCC)CC)CCC2(C=Cc3ccccc3O2)C1 CC(C)CCC(O)C(=O)NCCC(C)(C)C(=O)N1CCC1C(N)=O C1(C)(C(=O)NCCC(C)N(C(=O)CCCn2cnc(C#N)n2)C)C=CCCC1 C1(C(=O)NC2(c3ccncc3O)CC2)C2CC(CC2F)N1C(c1ccccc1)=O Cc1cc(F)c(C(N2CC3(C2)CN(C(C2C4CCC(=O)C24)=O)C3)=O)c(F)c1 c1(COC)onc(C)c1C(F)(F)F.C1(Cc2ccccc2)C(=O)N1.C1CC1 C(C1CCN(C(=O)Cc2nocc2C)CC1)=CC(N1C(CC)(CC)CC1)=O C1(NC(CC(C)(C)OC)=O)CC2(CCCN(c3ncc4ccsc4n3)C2)C1 C1(CNC(CCC2(NC(C(CSC)OC)=O)CCC2)=O)CN2CCC1C2 S(=O)(=O)(c1ccc(N2CCCC(C)CC2)c(Cl)c1)NC(C)CCn1cncn1 CCC(CCOC)C(=O)NCCOC1CCN(C(c2cccnc2O)=O)C1 S(=O)(=O)(c1ccc(NCCC(C)(C)C2CC2)cc1Br)NC1CC(CCC)OCC1 c1(CC)ocnc1C(=O)NCc1csc(C(=O)NCC=CCSC)c1 CC(O)(CNC(=O)C(c1cccs1)NC(C1CC(=O)C1)=O)C1CCC1 N(C1CN(C(=O)Cc2cccnc2C)CCc2ccccc21)C(C)=O c1(CNC(CSCCCC)=O)n[nH]cc1C(=O)NC1CCC1N(C)C C1(O)(C(N2CC(C)(NC(c3n(C)c4c(c3)ccs4)=O)C2)=O)Cc2ccccc2C1 N1(C(C2(CCC)CCC2)=O)CCC2(CC1)CC2C(=O)NC1CCN(CC)C1 N1(C(C2CC(C3CC3)C2)=O)CCCC(F)(CNC(=O)C(F)(F)CO)CC1 c1(OC)c(C)cc(C(=O)NC2(C)CCCN(C(=O)C#CC3CC3)C2)cc1C c1(C=O)cc2c(s1)CCCCC2.C1(COC)(C)CCCN1C(C1CCCO1)=O.N CCCCC(C(=O)N(C)CC1CCCN1C(=O)C(CCCC)NC(N)=O)C(C)C c1(C2CCCC2)ccc(C(C)(C)C)cc1.C1(CCN(C)C)CCCN1C(=O)NC C(=O)(C1=CCCSC1)NCC(CCNC(c1coc(C(F)F)n1)=O)OC CC1(C)CCCCC1CC(=O)NCC1CC1CNC(=O)CCCN=[N+]=[N-] C1(NC(CC2CN(C(C)=O)C2)=O)CCCN(C(=O)CCC(C)C#N)CC1 Cc1nc(Cc2ccc(F)cc2)sc1C(=O)NC.C(=O)C1=CCSC1.C1CC1 c1(OC)ccc2[nH]c(=NC3CC4CCCCCCC34)[nH]c(=NCCOCCO)c2c1 c1(CN2C(C(=O)NCC3COCCO3)CCCC2)cc2ccccc2s1 C1(C(=O)N(C2CCCCC2)CCO)CC(F)CN(C(c2cc(I)ccc2Br)=O)C1 N1(C(C2(C)CC(C)(C)C2)=O)CC2CC(C(=O)NC)(C2)C1.c1cc(F)ccc1O Cc1nn(C)nc1C(=O)NCCCCC1(NC(c2ccnnc2O)=O)CC1 C1(CNC(c2c[nH]nc2-c2cccs2)=O)CCCN(C(C2CCCCCC2)=O)C1 N1(C(c2cncc(C#C)c2)=O)CC2(CCCCN(C(C3CCC(CC)CC3)=O)C2)C1 C(=O)(CCCCCC#N)NCCC(C(=O)NCc1cc(C)ncn1)OC Nc1nccnc1C(N1CC=CC1C(N1CCC(OC2CC2)C1)=O)=O N1(C(COC(CC)(C)C)=O)CCC2CC1CN2C(c1ccccc1F)=O c1(CC=C(C)C)cc(C(N2CC3CCC2C3C(=O)O)=O)ccc1F.C(=O)CCCC N1(C(CCN(CCC)C)=O)CC2CCC1C2NC(c1cc(C2(O)COC2)on1)=O c1(C(N2CCCC(CNC(C(CC)C)=O)C2)=O)cc(Cl)ccc1C C1(C(=O)NCCOCCNC(C#CC(C)C)=O)CNC(=O)CC12CCOC2 CCCC(C(=O)N(CC(C)(C)NC(C1NC(=O)OC1C)=O)C)S(N)(=O)=O N(C1CN(C(C2CCCO2)=O)CCc2ccccc21)C(c1n(CC)ccn1)=O c1(C(=O)OC)c(C)cc(NC(c2cc(-c3csc(C)n3)cn2C)=O)cc1C C1(CC)CN(C(=NC)NCCSCc2cccnc2)CCC1O c1(C(=O)NCC2(NC(=O)Cn3ccnn3)CCOC2)ccc2c(O)ncnc2c1 C1(CNC(c2n(C)ncc2)=O)COCCN(C(C2CC(C)(C)O2)=O)C1 N1(C(c2c(COC)cccc2)=O)CC2(CCCC(C)O2)C1.C(=O)(CC(C)C)N c1(C(N2CC3(C(NC(C(C)CC4CC4)=O)CC3)C2)=O)ccc(Br)c(F)c1F N1(C(C2CCC(C)O2)=O)CCC2(CCN(C(C3C4CC5C(C4)C35)=O)CC2)C1 CCC(CC)C(F)C(=O)NC1(C(=O)NCC2C(C)C2C)CSC1 CC(C)CS(=O)(=O)CCC(=O)NC1CCC1NC(c1ccc2c(c1)COC2=O)=O N1(C(=O)OC(C)(C)C)CCC(C#N)(C(N2CCC(O)(C(C)(C)C)CC2)=O)C1 C1(C(=O)NC2(c3nc(C)on3)CC2)COCCN1C(C1C(C)=NOC1C)=O c1(C=O)ccc2c(cnn2C(F)F)c1.CS(=O)CCC(=O)NCCC1CC1.C C1(C)(C(N2CC(O)(C(C(N3CC(O)(C=O)C3)=O)F)C2)=O)CC(C)=NO1.C C1(C(N2CC(OCCOC)C2)=O)CCCC(NC(C2CCCSC2)=O)C1 C=C=C(C)CC(=O)NCC1CN(C(c2cccc(CNC(C)=O)c2)=O)C1 C12(NC(=O)CCCc3cnccn3)CCCC1(F)CN(C(C1CCCS1)=O)C2 O(NC(=O)CC(C)C(C)(C)NC(=O)CC(O)C(C)C)CCC Cc1cc(Cl)ccc1C(N1CCC(OCC2=NOC3CC23)C1)=O C(=O)(CCN=C(NCC1CN(CC(C)C)C1)NCC1CCN(C)CC1)NC c1(OCc2snc(C(C)C)n2)cccc(NC(c2ccc(F)cc2)=O)c1 CCC(O)C(C)(C)C(=O)N(CC(C)C(=O)NC1CCCC1CN(C)C)C CC1(C)CCCC(CCN(C2CC3CCC2C3)C(c2cc(F)cnc2O)=O)C1 c1(C(=O)NCC2(CN(C(C(C(CC)C)O)=O)C)CC2)ccc(Cl)c(C)c1O CC1(C)CC(C)(CNC(=O)CCCN=[N+]=[N-])CN1C(c1ncc[nH]c1=O)=O c1(-n2nnc(C(=O)NCCC(CN)OC)c2C)ccc(F)c(C)c1 c1(C(=O)OC)nccc2cc(NC(=O)CC3(O)CCNCC3)ccc12 C(=O)(C(C)(F)C(=O)NCC1(NC(=O)CC(C)(C)C2CC2)CCC1)OC CC(C(=O)N(C(CNC(=O)Cn1ncc(Br)n1)C1CC1)C)C(F)(F)F N1(CC(=O)NC2(CCCC(=O)NCC3C(C)CCC3)CCC2)CCC(F)CC1 C(C)(CCC(=O)NC(CNC(=O)Cc1cccc(OC)c1)C(C)C)OCC c1(-c2nc(OC)c(C(=O)NCCS)cc2)ccc(O)c(C=O)c1.c1cccs1.C c1(C(=O)NCC(C)NC(c2cnn3c(=O)cc[nH]c23)=O)cnn2c(N)ccnc12 N1(C(C2CC(C#C)(O)C2)=O)CC2CCC1C(NC(=O)CCC1CC1(F)F)C2 C1(NC(N2C(C)CC2)=O)CCCC1Oc1ccccc1 N1(C(C(C=C)O)=O)CC2CCCC(NC(=O)C)(C2)C1.c1(C=O)cc(C)oc1C.N C(=O)(CC(C)CC(C)C)NC(CCCC)C(=O)Nc1cc(C)ccc1OC CCCC(C)CC(=O)NCC1CC(OC)CN1C(=O)Cn1nc(C)n(C)c1=O C1(CC(=O)NC2C3COCC23)CC(F)CN1C(=O)C(F)C1CCC1 N1(C(C2(C)CCOC2)=O)C(C(=O)NCc2cccs2)C2CC(O)C1C2 C(=O)(C1=CCN(C(c2ccc(C(F)F)o2)=O)C1)N1CCN(CCC#C)CC1 c1(C=O)cccn2c(C)nnc12.C(C(COC)CC(=O)NCCC1CC1)OC.N N1(C(Cc2c(C)nc[nH]2)=O)CCN(C(C2(C#N)CC=CC2)=O)CC(C)(F)C1 c1(CC(=O)NC(C2N(C(C(C)SC(C)C)=O)CCC2)(C)C)ccc(Cl)nc1 CC1CN(C)CCC1N=c1[nH]c2c(c(=NCCc3cn[nH]c3)[nH]1)CCCCCC2 Cc1[nH]c2ccccc2c1CC(F)(F)C(=O)N1CC(NC(=O)C(=O)N)C1.C(C)C c1(CC(=O)NC)nc(C(CN)OC)no1 C1(CC)CCCCC1OCC(=O)NCCN(c1ccccc1)C(C1CC1C)=O c1(OC)cc(O)ncc1C(N1CCC2C(NC(c3nc(C)c(C)s3)=O)C12)=O C(C(O)CC(=O)NCC1CCCCC1O)NC(=O)Cc1ccccn1 C1(N(C(c2c(CC)cco2)=O)C)CCCN(C(c2cc(C)n(CCO)n2)=O)C1 c1(OC)nc(C(=O)NCC2CN(C(=O)CSSC)CCC2C)cc(O)n1 C(=O)(N=c1ccn(Cc2cccc(C#N)c2)[nH]1)NCCCNS(CC)(=O)=O CC1SCCN(C(=O)CC2CCN(C(C3(C)CC3C)=O)CC2)C1C c1(C(N2CCC3(NC(C=NOC)=O)C(CC2)C3)=O)coc2cccc(Br)c12 n1(CCNC(C(N2CCSCC2)C)=O)cnc(C(=O)NCc2ncsn2)c1 CCCCC(O)C(=O)NC1(O)CN(C(=O)C(CC#N)NC=O)C1.C(C)(C)C.O C1(CC)(CC)CC(NC(=O)COCCCF)CN1C(=O)Cn1ccc(C)n1 CCC(CC(=O)N1CCOC(CN(C(=O)CC2CC(C(F)F)C2)C)C1)C(C)(C)C c1c(F)cccc1Cl.C(C(C(C)(C)C)NC(=O)CC)NC(C1N(CC)CC1)=O C(CCOCC)(C(=O)NCC1CNC(=O)CO1)NC(C1(C#C)CC1)=O c1(C(=O)NCC(C)NC(c2cc(C#N)no2)=O)cn(C)nc1C1CCCCC1 c1(C(C)NC2CCC(N)C2)ccc(Cl)c(F)c1 C(C(C(C)C(C)C)NC(c1nnc(O)cc1O)=O)NC(c1cc(CCC)[nH]n1)=O c1(C(=O)OC)ccnc(C(=O)NCC(C)NC(C2CCCCN2C)=O)c1 c1(OC)nc(C(=O)NCC2CC(O)CN2C(=O)C(C)OCC(C)C)sc1C C(=O)C1=C2CCCN=C2NN1.c1(OC)ccccc1OCC(N1CCC(C)C1)=O.N N1(C(c2cccc(CCC)n2)=O)CCN(C(=O)C(CN(C)C)CC)C(CC)C1 C1(C)(CNC(CCOCCCOC)=O)CCCC1NC(=O)CC.CC.O c1(NC(C2N(CC)C(=O)CC2)=O)ccc(NC(=O)CCC(C)(F)F)cc1C c1(C=O)ncc(C(N)=O)cc1Cl.c1(CC)cc(C(N2CC(C)C2)=O)n(C)n1.N C(CNC(C1CCN(C(=O)NC)C1)=O)(CCCC)NC(CCC=C)=O c1(CCC=O)ccc(Cl)c(F)c1.C(C(O)CC)NC(C(C)NC(=O)NC)=O c1(C(=O)NC2C(NC(C3(C)CC(F)C3)=O)CCC2)cc(C(F)(F)F)ncc1N C(CC(=O)N(CC(=O)NCC(=O)NCCCN(C)C)C)SC N1(C(c2ncc(OC)nc2)=O)CCC(C)(C)C(CNC(c2ccnnc2O)=O)C1 CC(CC(F)F)C(=O)N(CC(N1CCN(C(C2CCN(C)C(C)C2)=O)CC1)=O)C c1(C(N2CC(C(C(=O)N(C(CC)CO)C)O)C2)=O)cc(Cl)n(C)n1 Cc1c(C(N2CC(C)(C(=O)NCc3ccc(C#N)o3)C2)=O)ccn1C N1(C(CCOCC)=O)Cc2ccccc2C1CNC(C1CSCC(=O)N1)=O Cc1cc(C(N2CCOC(CC(=O)N(C3CCN(C4CC4)C3)C)C2)=O)cn1C c1(C(=O)NC2CCC(N(C(CCC=C=C)=O)C)C2)ccn2cc(C3CC3)nc2c1 C1(NC(CSCC(C)C)=O)CCCCC1.C1(C=O)CC(O)CN1C(N)=O.C C1(C(N(C2CCCN(C(=O)Cc3ccon3)C2)C)=O)C2CCCCCC12 c1(CC(N2CCN(C(C(C)SC)=O)CC23CCC3)=O)c(C)[nH]c2ccc(F)cc12 Cc1cc(Br)cc2c1CCN(C(=O)Cc1ccc(-c3nn[nH]n3)cc1F)C2 c1(C(=O)NCC2CC(NC(C3CCC(SC)C3)=O)C2)cccc(F)c1C#N Cc1cnsc1C(N1CCC(C(=O)NCC(C)C(C)O)C1)=O C#CCC(CC#C)C(=O)NCC1CCC(NC(c2cccc3c[nH]nc23)=O)CC1 C=CCC(C)(CNC(C1CCCCC1NC(=O)CC(C)(C)C#N)=O)CO C1(C(=O)NCC(C)CN(C)C(C2CCCO2)=O)CCc2cnn(C)c2C1 C1(N(C(=O)CO)C)CCCCN(C=O)C1.N1(C(C2CC2)=O)CC=CC1.CCF c1(C(N(C2CCCN(C(C3CCCS3)=O)CC2)CC)=O)nnn2c1CCC2 C=CCC(C(=O)N1CC(O)CC1CNC(C1(N(C)C)CCC1)=O)OC C(=O)(CC1CCCc2ccccc21)NC1C(SC)CN(C(=O)CO)C1 c1(C(=O)NC2(CNC(c3c(OC)scc3)=O)CCC2)ccc(Cl)c(N)c1Cl O=C(C1=CC2CCCCCC12)OCCC12CC3CC(CC(C3)C1)C2 c1(CNCC2CCC(C(=O)NCC3CCCO3)CC2)cccc2c1OCC2 c1(C(N2CCCC(CNC(CSCC)=O)C2)=O)cc(=O)c(OC)c[nH]1 CC1CC(NC(c2cccc(Cl)c2Br)=O)CN(C(C23CC(F)C2C3)=O)C1 N1(C(CCNC(COC)=O)=O)CC=CC(NC(=O)CN2CCOCC2)C1 C1(CCCCNC(C2(C)CSC2)=O)CCCN(C(=O)C(C)(O)C2CCC2)C1 N1(C(C(C)SCCCC)=O)CCCCCCC1C(=O)NCc1cnn(CCF)c1 c1(CNC(=O)CCCNC(=O)C2=CCCC2)ccc(F)cn1 C(=O)(C1=Cc2ccccc2C1)NCC(C)=CC(=O)N(C1CC1(C)C)C Cc1n[nH]c(C)c1S(=O)(=O)N1CCC(NC(c2cnc(O)[nH]2)=O)C(OC)C1 c1(CC(C)C)ccc(C(=O)NC)cc1.C1(C=O)CC(C)N(C)C1.C1C=CCC1 CN=c1[nH]c(C(=O)N(C)CCNC(C2CCCCN2C(=O)C(C)C)=O)cs1 CCC(C)(CO)C(=O)N1CC(N2CC(NC(C3(O)CC3)=O)CC2=O)C1 N1(C(CC(C)F)=O)CC2CC2(C(N2CCCCC2CC(N)=O)=O)C1 N1(CCCCN2C(=O)CCC2)C(=O)CN(Cc2cc(F)cnc2Cl)C1=O C1(C(=O)NC2CCCC2(F)F)CC2CCC1N(C(C1Cc3ccccc3O1)=O)C2 Cc1nnn(CC(=O)NCCC2(CNC(C3CC34CC4)=O)CC2)n1 C1(CC)CN(C(c2cc(OC)ccc2I)=O)CCN1Cc1ncc(C)s1 N1(C(CN(C(C)(C)C)CC)=O)CCCC(CNC(=O)CC(C)(C)O)C1 C1(C(N(C2CCCC(NC(c3cnn(CCF)c3)=O)C2)C)=O)C2CC3C(C2)C13 C1(C(=O)NC(C(C)NC(=O)CN2CCCCS2(=O)=O)(C)C)CCC12CCOCC2 C=CC(C)(O)CC(=O)NCC1(F)CC(C)C1.c1(C=O)ccccc1.CCF.N Cc1cc(Br)cc(C(=O)NC2CC(C)N(C(c3cccn3C)=O)C2)c1F c1(CN2CCCC(C)(C(=O)Nc3cncs3)C2)ccc(Br)c2nsnc12 Cc1nn(C)c(Cl)c1C(=O)NCC1CN(C(=O)C2CC2)CC12CC2 C=CC1(C(=O)Nc2cc(Cl)ccc2O)CCN(C(=O)CC2CC3CC3C2)C1 C=CCC(CC=C)C(=O)NC1(C2CCCN2C(C2C3CC4C(C3)C24)=O)CC1 CCC(F)(F)C(=O)NCc1csc(CNC(C2COC(CCC=O)C2)=O)n1 c1(C(=O)NCC(C(C(C)C)C)NC(c2ccc(Cl)s2)=O)cnn2c1OCCC2 C1(NC(c2cc(CC)[nH]n2)=O)CCC(N2CCN(C=O)CC2)CC1.C(C)(C)C.O N1(C(C(CC)(C)F)=O)CC2CCC(C1)C(NC(c1cc3c(F)cccc3s1)=O)C2 N1(C(CCC(=C)C)=O)CCN(C(=O)Cc2ccnn2C)CC1CC c1(C(N2C(CNC(C(C)OCC=C)=O)CCC2)=O)cn(C)nc1C(F)F Cc1cc(Br)cc(C)c1NNC(=O)N1CCCc2ccc(Br)c(Cl)c21 c1(C(N2C3C(NC(C4CC=C(C)CC4)=O)C(C3)C2)=O)cnn2c(C)ccnc12 c1(C(N(CCC)C2CC2)=O)ccc2c(c1)CCC(O)C2.O=CCOCCCF.N C(=O)(CC(C)C(=O)N1CCC(C(=O)NC2COCCOC2)C1C(C)C)OC C1(CNC(c2c(C)nc(CC3CC3)s2)=O)CN(C(=O)C(C)C(C)C)CCN1C C1(C(=O)OC)CC12CCN(C(C1(C)CCCN(Cc3cc(C)c(C)[nH]3)C1)=O)CC2 C1(N(C(c2ccc(SC(F)(F)F)cc2)C(=O)NCCCF)C)CCCC(O)C1 n1(CC)ncnc1C(=O)NCCCC(C)NC(=O)CCCNS(C)(=O)=O C(CCCCCCNC(c1ccc(C#N)cc1)=O)n1cc(CS(C)(=O)=O)nn1 C(=O)(CCCCC(=O)OC)N(C1CCN(C(C(C2CC(F)(F)C2)OC)=O)CC1)C c1(C(N2CCC(C)(C)C2)=O)ccnc2[nH]c(C)nc12.C=C1CC(C)(C(=O)NC)C1 c1(-c2n(CCCOC)nc(CN3CCSC(C)(C)C3)n2)ccc(=O)n(C)n1 c1(C(N(CC(CN(C(C(C(C)C)F)=O)C)O)C)=O)c[nH]c2cccnc12 c1(C=O)ccc(C2CC2)nc1.c1(OC)ccc(C(=O)N(CCC)C(C)C)s1.N C1(=O)C2=NOC(C2)CN1.C12(C(N(C(CC)CC)C)=O)C=CC(CC1)C2 Cn1nc(C(N2CCCC2CNC(=O)Cc2cncc(C#N)c2)=O)ccc1=O Cc1c(C(=O)NC2CC(F)CN(C(=O)COC(C)C)C2)ccc2ccccc12 C(C)(C(O)C(F)F)NC(C1N(C(Cc2ccc(C)s2)=O)CC=C1)=O c1(NC(N2CCOC(C(F)F)C2)=O)ccc(COCc2ccccc2)cc1F c1(C(N(C(C)C(=O)NCc2ccncn2)CCC)=O)csc(C)c1 C1(C(=O)N)CCC2CCC1N2C(C1(N(C)C)CC1)=O.CC(C)CN(CCC)C C#CC(CC(C)C)NC(C1(N(C)C(C2CCCN2C=O)=O)CC1)=O N1(C(c2ccc(COC)cc2)=O)CCN(C(=O)CO)CC1C.c1nnc(C)s1.C c1(C(N2CCC(C)C(NC(C3CC(=C)C3)=O)C2C)=O)c(C)cccc1[N+](=O)[O-] c1(C(N2C(CCC)CN(C(C3(CF)CC3(F)F)=O)CC2)=O)c(F)ccc(F)c1F c1(C(N2C(CNC(C3CCN(CCC)CC3)=O)C=CC2)=O)cnc2[nH]nnc2c1 CC(CS(C)(=O)=O)C(=O)NCC1CC2CCC1N2C(=O)Cc1ccc(N)cc1 c1(OC)ncc(Cl)cc1C(=O)NC1CCC1NC(c1ccc(NC=O)cc1)=O C=C1CC2CCCC(C1)N2C(C1CN(C(=O)C(C)(CC)CCC)CC1F)=O C(=O)(CCC(C)(C)NC(C1CCCC(C)(C)C1)=O)N(C1CC(=C)C1)C c1(CCC)cccc(C(=O)NC2CC(NC(c3cnn(C)c3OC)=O)C2)c1 Cc1cc(F)sc1C(=O)NC1(C(N2CC(C(F)(F)F)C2)=O)CC(O)C1 CCC(C)(C)C(O)C(=O)N(C)CCN(C(=O)C(C)C1(O)CCC1)C c1(OC)nc2ccccc2cc1C(=O)NC1CC(F)CN(C(C2CCCS2)=O)C1 C1(C2CCCN(C(c3cccc(C(F)F)n3)=O)C2)(NC(C2C3COCC23)=O)CC1 c1(NC(=O)CC2CCCN(C(C3CC3F)=O)C2)cccc2c1CCCC2 C1(NC(CC2N(C(c3c(C)cc(C)s3)=O)CC2)=O)CC2CCC1(CO)C2 CN1CCN(C(C2C3CC4C(C3)C24)=O)C(C(=O)N(C)Cc2ccc(F)cc2)C1 N1(C(CCN(C(=O)C(C)S(N)(=O)=O)CC=C)=O)CCC2(C=CCO2)CC1 C1(C(=O)NCc2ncn[nH]2)(CNC(=O)COc2ccsn2)CCCC1.C CC1CC(C)(C(=O)NCc2ccc(C(=O)NCC3CCC=CCC3)o2)CCO1 Cc1ccc(OC(C)C(=O)N(C(C)CC)C)c(C)c1.C1(C=O)CCC(=O)NC1.N C1(C(=O)NC(c2nn(C)cc2O)C)(NC(C(CC)=CCCC)=O)CCCCC1 c1(C(N(CCCN(C(=O)C(O)Cc2cnc[nH]2)C)C)=O)csc(-c2cn[nH]c2)n1 C1(C(=O)NCC2(CC(C)C)CCC2)CCCC(NC(c2cncs2)=O)CC1 N1(C(=O)NC)CCCC1C(=O)NCCC(O)CNC(=O)CCN(C)CCO C1(NC(c2cc3nc(C)sc3[nH]2)=O)CN(C(C2CCCS2)=O)CC2CCCC12 C(=O)(C(CO)C(C)(C)C)NC(CC(=O)NC1CCN(CC)CC1)C C1(NC(c2cccc(OC)n2)=O)CC2CCC(C1C)N2C(c1ccc[n+]([O-])c1)=O C1(CNC(CC(CCC)(C)C)=O)CCC2(CC1)CC(NC(=O)C1=COCCO1)C2 Cc1ccc(=N)[nH]c1C(=O)Nc1cc(C(F)(F)F)cnc1N1CCOCC1 N1(C(CC(=O)OC)=O)CC(NC(=O)Cc2sccc2Cl)C(F)C1 C1(C(=O)NCC(=O)N(CC)CC)CC(C)CN1C(=O)CNC=O CC1(C)CCN(C(=O)C(=O)Nc2ncc[nH]2)CC1C.n1(CC(=O)N)nccn1 O=C1CC(CC(=O)NC2CN(C(=O)CC3(O)CCC3)CC2n2cccn2)=NN1 S(=O)(=O)(c1cccc(N2CCN(CC(F)(F)F)CC2)n1)N1C(CCC)COCC1 c1(OC)ccc(F)c(C(=O)NCC(C)(CNC(C2C=C(C)CS2)=O)O)c1 C1(NC(c2cc(C)sc2C)=O)CCN(C(c2ccc([N+](=O)[O-])o2)=O)C(C)C1 N1(C(c2n(CCC)nc(C)c2)=O)CCC(C)(C)CC1.c1(C(=O)N)ccc[n+]([O-])c1 C=CC(CCC)CC(=O)NC(C1CC1C(=O)Nc1ccc2c(c1)COC2)C C(CCCC(C)(C)C)NC(CC1(C=C)CN(C(c2cc[nH]n2)=O)C1)=O C1(C(N(C)CC2(CO)CC2)=O)CCC(O)CN1C(=O)CCC1CCC1 n1(CC2CC3(CC(C)(C)C3)C2)c(CC2CC2)csc1=Nc1ccc(F)c(F)c1 c1(-c2n(C(C=C)C)nc(C3CCCCC3)n2)c[nH]c2nccc-2c1 N1(C(c2cc(C)sn2)=O)CCC(S(C)(=O)=O)C1.C1(C=O)CCCN(C(C)C)C1.N C(=O)(C(C)=Cn1ccnn1)N1CC2C(CNC(C(CC)(C)OC)=O)(CC2)C1 c1(C(N(CCNC(C(C(CC)O)(F)F)=O)C)=O)cc(N)c2ccccc2n1 c1(C(N(CC(C)NC(C2COC(=O)C2)=O)C)=O)cnc2ccc(F)cc2c1 CN=c1[nH]ccc(C(=O)NC(CNC(=O)Cc2cc[nH]n2)C(C)C)c1N N1(C(COCCC)=O)CCC(C(F)(F)F)C(NC(C2(C)CCOC(C)C2)=O)C1 N1(C(C2C(C)(C(=O)O)C2)=O)CC2(C1)CN(C(c1ccccc1F)=O)C2.CC Cc1cc(C#N)cnc1N1CCCC(CNC(c2cccnc2O)=O)C1 c1(CNC(C(c2n(CCCCCC)ccn2)NC)=O)ccc(OCC)nc1 C1(CC(N2CCCC2)=O)CN2CCN1CC2.c1(CC)occ(C)c1C(=O)N(C)C CC1=C(C(=O)N2CCN(C(c3ccnn3C)=O)C(CC3CC3)C2)C(C)(C)CCC1 N1(C(C)=O)CC(C)CN(C(=O)NCc2cc(C3(C)CC3)n[nH]2)C(C)C1 c1(C(=O)NCCN(C(c2c(NCC)cncc2)=O)C)cc(CC)ccc1F c1(C(=O)NCCCN(C)C(C2COCC2c2ccccc2)=O)ncc(F)cn1 N1(C(CC(C(C)C)O)=O)CC2(C)CN(c3nnc(C(F)F)s3)CC2(C)C1 N1(C(C(=O)NCCOC)CCC2(C#N)CC2)CCCCCC1C1CCCO1 CCCC(C)C(=O)NCC(CC1CC1)C(=O)N1CC(OCC(=O)NC)C1 c1(C(=O)NC2C(C)(C)C(OCc3ccccc3)C2)cccn(C2CCOC2)c1=O CP(C)(=O)c1ccc(C(=O)NCC2CCCCC2NC(c2ccncn2)=O)cn1 CCCCCCC(=O)NC1(C)CC(NC(C2CCCCN2CC2CCCC2)=O)C1 N1(C(CCC#N)=O)CC2CCC1CN2C(=O)COC1CCCCCC1 C1(CNC(C2C(=C)C2)=O)CN(C(c2c[nH]nc2C2CC2)=O)CC(C)(C)C1 CCCC(C(=O)N1CCC(NC(c2ccc(C(C)C)cn2)=O)C1)C(C)C CCCCCCCCCn1cc(C2(C)CCCN2C(=O)C(C)NC(=O)CC)nn1 N(C(=NCCSCc1ccccc1)NCC1CC1C(C)C)C(C=C)C C(CC(C(=O)NCCCn1cccn1)NC(C1COC(=O)N1)=O)=CC c1(NC(CC2(OC)CN(C(=O)CCC(F)(F)F)C2)=O)cc(C)c(F)c(C)c1 C(=O)(CCCCC(C)C)NC12CN(C(c3c(C)nn(C4CC4)c3)=O)C(C1)C2 N1(C(C2(CC#C)CCC2)=O)CCC(C(C)(C)NC(=O)CCc2ccnn2C)CC1 C1(NC(c2ccn(CCCC)n2)=O)CCCCC1NC(=O)C(C)=CCO c1(C(=O)Nc2c(C(=O)OC)cccn2)c(C)cc(C#N)cc1C C1(CNC(C2N(C(COC3(C#C)COC3)=O)CC2C)=O)COCCN1C C1(C(N(CC(=O)NC(CC)CN2CCCC2)CC)=O)C2COCC12 c1(C(N(CC(C)NC(c2cnc(Cl)[nH]2)=O)C)=O)cnc2ccoc2c1 c1(NC(C2C3CN(C(=O)CCc4ccccc4)CC23)=O)ccc2ccccc2c1 CC(CC(=O)OC(C)(C)C)NC(=O)NCCN1CCOCC1 N1(C(Cc2cn(C)nc2)=O)CC2CCC2(CCNC(C2CCOCC2)=O)C1 C1(NC(C(COCC)NC(c2csc(F)c2)=O)=O)CC2CC1CC2(C)O c1(C(=O)NCCCN(C(=O)C(C2CCCCC2)F)CCO)cnc2cccnn12 c1(C(=O)NCCC(CNC(=O)COCC(F)F)O)cccn(C2CCC2)c1=O C#CCCCCCC(=O)NC12CCC(CNC(=O)CC(C=C)CC)(C1)OC2 C(=O)(C(C1=CCC(C(C)C)CC1)N(CC1Cc2ccccc21)C)N(c1ccccc1)C C1(C(=O)NCC2N(C(Cn3c(C)ncc3)=O)CC(F)(F)C2)C2CCCCCCC12 Cc1oc(Cl)nc1C(=O)NC1CCC(NC(C2(NC(N)=O)CC2)=O)C1 c1(OC)cc(C(=O)N(C2CCN(C(C3(OC)CCSC3)=O)C2)C)ccc1[N+](=O)[O-] c1(C(N(CCCNC(COCC(=C)C)=O)C2CC2)=O)ccc(OC)cc1 Cc1cc(C)c(CC(=O)NCC2(CC)CC2)c(C)c1.C(=O)(C)N.C1CC1 Cc1cc(C(=O)NCC(C)CNC(c2nsnc2O)=O)c(C)nc1C C1(C=O)CC(F)(F)CS1.c1(C(=O)NCC2C(C)C2(F)F)cnc(S)nc1 C1(F)(C=O)CCN(C)CC1.N1(C(C(C)OCC2CC2)=O)CCC(C)(C)C1.N N1(C(C(C(C)C)NC=O)=O)CCCC(C2CCN(c3nc(Cl)ncc3Cl)CC2)C1 C(=O)(C1CC(C(F)(F)F)Cn2ccnc21)N(c1c(C)nc(Br)cn1)C c1(C(N2CCC(F)(C(=O)OC)C2)=O)cc(S(=O)(=O)Nc2cccs2)ccc1O C1(CC(=O)NCC2(F)CN(C(CC3C(C)OCC3)=O)C2)CCC(F)(F)CC1 N1(C(CC2C(C)CCC2)=O)CCCC2(CCC2NC(=O)CCc2ccoc2)C1 CCC(O)C(=O)NCC1(O)CC(C(=O)N)C1.CCN(C(C)C)C(C)C c1(C(=O)NC(C)CNC(C2CCOC2=O)=O)cc(Br)c2c(c1)nnn2C C12(C(=O)NCC3(NC(C)=O)CC3)CCC(CC1Br)C2 N1(C(C(=O)NC(C)C)=O)CCOC2CCN(C(c3ccn(C)c3)=O)CC12 Cc1sc(Cl)nc1C(=O)NC1CCC(N(C(=O)CC2CCCOC2)C)CC1 c1(C(=O)NC(C2CC=CCC2)C(=O)NCC(C)OCCO)cc(O)ncc1F C1(CC(N2CCC(CN(C)Cc3nc(C(C)C)on3)C2)=O)CC(C)NC(=S)N1 c1(C(=O)N)cn2c(n1)CCC2.C1(CC)(CC)CCN(C(=O)CCn2cncn2)C1 CCCC(C(=O)NCCOC1CCN(C(c2nscc2C)=O)C1)NC(C)=O c1(OCC)ccc(Cl)cc1CNC1CC(C)CN(C(c2ccc(C)cc2)=O)C1 Cc1ccc(Cl)c(C(=O)NCC2CN(C(C3CC3CF)=O)CCCO2)c1O C1(CC(N2CC3CC3C2)=O)CC(=O)NC(=O)C1.n1(CCC)ncc(C=O)c1C.N N1(C(c2nn(CC)c(C)c2)=O)CCC2CN(C(=O)CCCn3cccc3)CC2C1 C1(C)(C(N2CCC(CC(=O)OC)C2)=O)CCCN(C(C2(C)CCCCO2)=O)C1 c1(OC)ccc(NNC(=O)C(=O)N(C)Cc2nc3c(s2)CCCC3)cc1Cl C1(NC(CC=C=C)=O)CCCC12CCN(C(c1cscc1S(C)(=O)=O)=O)C2 N1(C(C(C)C(=O)OC(C)(C)C)=O)CCC2(CC1)CCC2.C1(C(=O)N)CCCOC1 O=S(=O)(c1ccc(Cl)s1)NC1CN(Cc2cncc(Br)c2)CC1O S(=O)(=O)(C1CCN(CC)C1)NCC.C1(CC)CC(C)(C)C1 CC1C(NC(C2CC(C)(C)CN2C)=O)CC2CCC1N2c1cnc(F)cn1 C(=O)(C(CNC(c1scnc1CC)=O)C(C)C)NC(CC=C)C C1(C(=O)NCCCCCSC)CC(NC(=O)CCc2nc(C)no2)C1(C)C c1(C(CC)(C)O)cn(C2(C(=O)OC)CN(C(=O)C(N3CCOC3=O)C)C2)nn1 n1(CCOC)c(C)cc(CN2CCN(C3CCOCC3)CC2C)c1C c1(C=O)cccc2oc(O)nc12.C(C)C(C)(C)C.C(C)(C(=O)N)OCC(C)C N1(CCC)CCC(C(=O)NC(C)CC)CC1.c1(C=O)ccc(SC(F)(F)F)o1.N N1(CC(=O)N(C(=O)CN2CCOCC2)C)CCC(N=[N+]=[N-])C1 O=C(C(O)CC1CCCCC1)NCC1(O)CN(C(C2CSC2)=O)C1 Cc1[nH]c2ccc(C(=O)NC(C)CCCCNC(=O)C(O)CC(C)C)cc2c1C O=C(C(F)(F)C(O)C1CC1)N1CC(CNC(C2(C3CCC3)CC2)=O)C(O)C1 n1(CC)ncc(C(=O)NCCN(C(=O)C=CCF)CCO)c1Br.CCO C1(C(=O)NCc2cccc(F)n2)C(C2CC2)CCN1C(=O)Cc1cnsc1 c1(C2(C(=O)NCCCCNC(=O)CCc3cnoc3)CC2)ccnc(Cl)c1 C1(NC(C2CSCCS2)=O)CCOC12CCN(C(c1coc(C(F)F)n1)=O)CC2 C1(C(=O)NC2C(NC(CC3CC(OC)C3)=O)CC2)CC2CCC(C1)C2 c1(C(=O)NC2C3CN(C(C(CCCCC)O)=O)CC32)c(S(N)(=O)=O)ncn1C n1(CC)nc(C(=O)N(CCC(C(C)C)NC(C2CCC(F)(F)C2)=O)C)ccc1=O c1(NC(C2CC2NCc2ccc(Cl)cc2)=O)c(OC(F)(F)F)cccc1O c1(CCNC(CN(C(c2conc2C)=O)CC)=O)cnnn1C C1(OC)CN(C(=O)Cc2cnoc2)C(C)(C)C1.C(=O)(CCCC=O)N.C(C)C N1(C(c2cn(CC)nc2C)=O)CCCCC(CCC(=O)N(CC(O)CF)CC)C1 Cn1cc([N+](=O)[O-])c(OCC(N2CCN(C(=O)C#CC3CC3)C3(CC3)C2)=O)n1 c1(C(=O)NCC2N(C(c3c(C)ccnn3)=O)CC2)cnc(O)c2ncccc12 C(=O)(NNC(=O)c1cn(-c2ncccn2)cn1)C1C(N)C1 CSC1=C(C(=O)NC2CC2CNC(c2ccc3nc(S)oc3c2)=O)CCCC1 CCCC(O)C(=O)NCC1(C)CCN(C(c2cc(C(N)=O)[nH]n2)=O)C1 CC1(C)C2CCCN(C(c3cc(C(F)(F)F)ccc3O)=O)C1C2 O=C1CCC(CC(N2CCN(CCNC(c3cnc(O)s3)=O)CC2)=O)C(=O)N1 N1(C(COCCCC)=O)CC(COC)CC1C.C1(C=O)(C(F)F)CCCOC1 c1(C(N2CC(OC)CC2)=O)cc2c(s1)CCCNC2=O.O(C(F)(F)F)CC(=O)N Cc1conc1C(=O)NC1CN(C(=O)CC(C)C2CCCO2)C1 N1(C(C(CSCC)NC(=O)C(CN(C)C)CC)=O)CCNC(=O)CC1 c1(OC)ccc(C(O)Cn2cc(C(=O)NCC(C)C)nn2)cc1NC(C)=O Cc1cc(C(c2ccsc2)NCCCc2cc(-c3cccc(F)c3)n[nH]2)nn1C c1(C(N2CC(C)C(CNC(=O)CO)C2)=O)cc(F)cc(Cl)c1N.C1CC=CC1 N1(C2(C(=O)OC)CC2)CCN(C2(C(=O)O)CC2)CC1 C1(NC(=O)CONC(=O)C2CCOC2)CC2(C1)CC2(F)F c1(C(N2CCC2)=O)ccc(N)c(N)n1.c1(OC)ncccc1CC(=O)NCC.O C1(C(N(C(C#C)C)C)=O)CN(C(c2c(C)noc2C)=O)CC1C N1(C(C2(CCCC)CC2)=O)CCC2(CCN(C(=O)C=Cc3ccco3)CC2)C1 Cc1cc(C(=O)NCC(C)(C2CC2)NC(C2CCOCC2)=O)cc(C)c1 c1(C(=O)NCC2C(C(=O)NCCOC(CC)CC)C2)cc2ncccc2[nH]1 CCCCC(O)C(C)C(=O)NCC1CCC2(CCC2)CN1C(=O)C(F)C(F)(F)F Cc1cn2c(n1)CC(C(=O)NCCCC(C)NC(=O)C(C)(C)CC1CCOC1)C2 C(=O)(CC(C)C(C)(C)N)NC(CC)C(=O)O c1(OC)cc(C(N2CC(NC(C3(O)CC3)=O)C3CC3C2)=O)ccc1.CC(C)C c1(C=O)ncc(C)cc1C.C1(NC(C)=O)CCC(C(=O)NC2CC(F)C2)C1.C N1(C(C(c2ccc(F)cc2F)C)=O)CC(NC(c2csc(Cl)c2Cl)=O)C(C)(C)C1 c12cccc(c1)OCC(=O)N(CC)C(=S)NC2.C1(CN)CCC1 C12(C(N3CC(CNC(c4cnc(C(F)F)cn4)=O)C3)=O)CCCC1CCC2 CC(C)CC(C)(C)C(=O)NC1CC=C(C(N2CCC(F)(F)C(C)C2)=O)C1 CC(C)C(CC(=O)NCCOCCCF)NC(=O)CC1CCCN(C)C1 N1(Cc2ccc(OCC)cc2Br)CCc2cc(OC)c(C)cc2C1 C(=O)(CCS(C)(=O)=O)NC(CNC(c1cc(OC)n[nH]1)=O)C(C)C C(CC(CO)NC(=O)CCSCc1ccsc1Cl)OC CC(C)(CC(F)C(=O)NOCCC(F)(F)F)NC(C1COCOC1)=O N1(C(CC(=O)NCC)=O)CCCCC(NC(c2ncc(C(F)(F)F)cc2N)=O)C1 N#Cc1cc[nH]c(=NCC2CCCN2C(c2n[nH]c3c2CCCC3)=O)c1F CCC(C)(CNC(C1CC(CC2CC2)C1)=O)C(=O)NC(C)(C)CCCO c1cccc(Cl)c1.CC(C(C)C)NC(=O)CS.C(=O)CC1(C(F)F)CC1 N1(C(C(OC)OC)=O)CCC(C)C1c1cn(CC2CCOC2)nn1 c1(N(C2CC(=C)C2)CC)nnc(CN2CCCC2=O)n1CCC#N.C1CCCO1 C(=O)(CCCCCCNC(C12CCCCC1C2)=O)NC(C(CC)(F)F)(C)C C1(C)CC(F)(F)CN1C(c1nc(C(C)C)oc1C)=O.C(CCCC(=O)NC)OC N1(C(C2(CCCC)CC2)=O)CC(C2CCN(C(C3CC4(C3)CC(F)C4)=O)CC2)C1 c1(OCC)cnc(C(=O)NC2CN(C(=O)C(C)C(C)C)CC23CC3)c(Cl)c1 Cc1cc2nc(Cl)cc(N3CCN(C(c4ccc(F)cc4)CO)CC3)n2n1 CCC(C)C(C(=O)NCCCCC(C)(F)F)N(C)C(c1cc(Cl)n[nH]1)=O C(C(C(F)(F)F)c1ccccc1OC)NC(CCCOCCOC)=O CC1CCN(C(C2CC3(C2)CC(F)C3)=O)CC1C.C(C1CCOCC1)=CC=O.N c1(C(=O)NCC(C)NC(C2(OC)CCOCC2)=O)ccnn2ccnc12 C#Cc1ccc(C(=O)NCCCCN(C(=O)CC(F)(F)c2ccccc2)C)nc1 c1(-c2c(C)cc(CO)cc2)ccc2[nH]cc(C(=O)Nc3cc(Cl)cnc3Cl)c2c1 c1(OC)cc(C)ccc1-c1cn(CC2CCCN(C(=O)Cc3cc[nH]n3)C2)nn1 c1(C(=O)NC2CCOCC2NC(C2COCCO2)=O)n[nH]c2c1CS(=O)(=O)CC2 C#Cc1ccc(Cl)c(C(N2CC3CCC3(NC(c3cc(C)oc3C)=O)C2)=O)c1 C1(CCC(NOCC(=O)N(C)C)=O)CCCCN(C(C2CC(=C3CC3)C2)=O)C1 C(=O)(CC1OCc2ccccc21)NC1CCN(Cc2ncc(C)nc2)C(C)C1 CC1CN(C(=O)CC2OCCCO2)CC(C(=O)NCC2(C)CSC2)O1 n1(CCC)ncc(C(N2CCN(C(=O)CCCc3ccccn3)CC2)=O)c1Cl C12(NC(Cc3c(C)con3)=O)CCOCC1CN(C(c1cc(O)cc(F)c1)=O)C2 C(CC(=O)NC1CC(CC(=O)NCC(O)CF)C1)OCC c1(COCCC(=O)OC)cccc(NC(C2CCCOCC2)c2nnnn2C)c1 Cc1cccc2c1OC(C(=O)NC(CNC(c1cc(Cl)c(N)c(Cl)c1)=O)CO)C2 N1(Cc2cccc(OCC)c2)CC2(CC2)CC1C(N1CCC(SC)CC1)=O c1(C(N(C2CCCN(C(C3C(C=C)OCC3)=O)C2)CCO)=O)cnn2ccsc12 c1(C(=O)NCCOCCCOC(=O)CC(F)F)cccnc1OC(F)F Cc1c(C(=O)NC2(CNC(=O)CC3CNC(=O)O3)CCOC2)cccc1O C1(C(C)C)CCC(C(N2CCC(NC(=O)CN(C)C)C2)=O)C(=O)N1.C1CC1 C1(C(N2CC(O)(CNC(c3n(C(C)C)ccc3)=O)C2)=O)CCC(C)(O)CC1 c1(SC)cc(C(=O)NC(C2(C(N3CC(C4CCCO4)C3)=O)CC2)C)co1 CCC(F)(F)C(C)(C)C(=O)NC1CC2CN(C(c3cc(C)c(C)s3)=O)CC12 N1(C(Cc2cc(C)ns2)=O)CCN(CCNC(=O)C=Cc2cccnc2)CC1 N1(C(C)=O)CCCC1CC(=O)N(CC(=O)Nc1ccccc1)C C(=O)(C1=C2CCN=C2NC=C1)N1CCC(CN(C(c2oc(CC)c(C)c2)=O)C)C1 Cc1cc(Cl)cc(C(=O)NCC2CC2)c1C.c1(CC(=O)N)cnn2c1OCCC2 N1(C(c2c(C)nc(C)s2)=O)C(C)CC2CN(C(=O)CCC3CCCOC3)CC12 c1(C(=O)NC2CC(C)N(C(c3coc(CO)c3)=O)C2)nc(O)nc(O)c1N CCC(C)(C)C(=O)C(=O)NC1(C)CC(C(=O)Nc2cnn(C(F)F)c2)C1 c1(C(=O)NC2CN(C(=O)Cc3sccc3Cl)C3CC23)cccc2cncn12 Cc1cc(C)c(C(=O)NCC(C)(C2CCC2)NC(=O)CCS(C)=O)cc1C c1(C(=O)NC(CN(C(=O)C(n2nccc2C)C)CC)C)cnoc1-c1ccoc1 c1(NC(C2CC(F)CN(C(c3c(F)cccc3Br)=O)C2)=O)cc(Cl)ncc1Cl C12(C(=O)NCCCCC)CCCCC1NC(=O)C2.C1(C(F)(F)F)(C=O)CCC1.N C(CCC(O)C(=O)N(C)Cc1ccon1)NC(c1cc(C)[nH]n1)=O C1(CC(=O)N(CCC(N2CCC(OCC#C)C2)=O)CCO)CCCNC1=O c1(NC(C(CC)CC)=O)nc(NCC2CCC3CCCC3O2)nc2c1cnn2C N1(Cc2cccc(OC(C)=O)c2)CCN(CCNC(C)=O)C(=O)C1 C1(C(=O)NC(C)CC)C2C3CCC(C3)C12.N1(CCCC(=O)N)C(=O)CCC1=O C(=O)(C1=CCC(C)(C)CC1)NC(C1C(C(=O)NCCC(C)OC)C1)C n1(CC)nc(C(=O)NC2CCC(CC(=O)N(CCCC(=O)NC)C)C2)cc1C N1(C(c2c[nH]nn2)=O)CCC2CN(C(=O)Cc3ccc(S(N)(=O)=O)s3)CC12.CC c1(NC(=O)CN(C2CCC2)C(=O)Cc2cncs2)cnn2c1CCCC2 CCC(C(=O)NC1(NC(=O)C(=Cc2c[nH]cn2)F)CC1)N(C1CC1)CC CC(CN=c1ccnc(-c2ccccc2)[nH]1)NC(C12CCOC1CCOC2)=O c1(CC(=O)N(CCNC(CC(=C)Br)=O)CCO)ccc(C)c(C)c1.CCO C1CC2CCC2C1.C(C)(C(=O)N(CCC(=O)NC)C(C)C)NC(=O)NC [nH]1ccc([N+](=O)[O-])n1.C12CC(C(=O)CC3CC(C)(F)C3)(C1)C2.CCCC.C C1(NC(c2c(C)coc2C)=O)CCC(O)CN(C(C2CCCC(=O)O2)=O)C1 C1(C(N2CC(NC(=O)CN3CSCC3=O)C3(CC3)C2)=O)(OC)CCCCCCC1 c1(C(C)OCC)nc(-c2c[nH]nc2C)n(CCSc2ccccc2)n1 N1(C(CCOCC#C)=O)CCC(C(=O)NC(CC#C)C(N)=O)C(C)C1 C1(CCC)CCCC1C(=O)NC(C)(C)CNC(=O)CCCc1ccsc1 CC1C2CC(C2NC(c2cccc(=O)o2)=O)N1C(c1cnc(C2CC2)nc1)=O Cc1occc(=O)c1OCC(=O)N.C1CC(F)CN1C(C1CNC(=O)N1)=O.C c1(Nc2scc(SCC(=O)NC(C(C)c3ccccc3)CO)n2)ccccc1F c1(C(=O)NC2C(CNC(c3csc(CO)n3)=O)CCC2)ncc(Cl)nc1Cl c12ccc(cc1)N(C)C(=O)C(C)S2.c1(CCC)cccc(OC)c1 CC1CC(C(=O)NC2CCCC2C(=O)NCCOC2CCC2)CN1C c1(C(=O)NCC(CCCC)NC(C2CC3(C2)CC3F)=O)cccc2ccnn12 c1(CC)cc(C)ccc1C(=O)NC1COCC1NC(=O)C=CCO Cc1ccn(CC(=O)NC(C2CCCN(C(C3CC(F)(CO)C3)=O)C2)C)c(=O)c1 C1(CNC(C(CC)N(C)Cc2ccccc2)=O)OCCCC1(C)C C1(NC(C2C(C(=O)OCC)CC2)=O)(C)CCOCC1.C(=O)(C(N)=O)N c1(C(C(=O)N(CC(C)CNC(=O)CC2CCC(O)C2)C)(F)F)ccccc1F c1(NC(C)Cc2cccs2)nc2ccccc2nc1N(CC(C)(C)C)C N1(C(c2nc(CC)oc2)=O)CCN(C(=O)CCOC2CCCOC2)C(COC)C1 C(CCC(O)C(=O)NC(c1ccncc1)C)NC(CCSCC)=O C=CC(C)(C)CCCNC(C1CC12CCN(C(=O)CCn1cnnn1)C2)=O Cc1ccnc(O)c1C(N1CCC(CC(=O)NC2(C)CC(O)C2)C1)=O C(=O)(CCCC(=O)N(C)C)NCC1CCN(C(C(C)(CO)OC)=O)C1 c1(N2CC(C(C)NC(c3ncc(C)c(C)c3)=O)C2)cc(=O)n2ccccc2n1 C1CN(C(=O)C(F)(F)c2cnccn2)CCC1C(F)(F)F.C(C=O)NC(C)=O.N C(C(CC=C)C(=O)NC)NC(C(CC=C)NC(C)=O)=O.C1CCC(C)(C)CO1 c1(C(=O)NCC2N(C(Cc3cn(C)nc3)=O)CC(O)C2O)ccc2nonc2c1 c1(OCCC)ccccc1-c1cn(C2CC(NC(=O)Cc3occc3C)C2)nn1 Cc1ncnc(C)c1C(N1CCC(NC(=O)C(O)P(C)(C)=O)C1)=O c1(C(=O)NC2CCC(NC(C3(C(C)C)CCC3)=O)C2)cccc(N)c1 N1(CC(CC)(C)C)C(=O)CN(CC2(C3CC3)CCCO2)C1=O c1(C(CC)C)ccc(C(=O)OC(c2ccc(F)cn2)C)cc1 C1(C(=O)OCC)CC12CC(C(=O)NC(C)(C)C)C2.C(=O)C(C)(O)CC N1(C(C=CC(C)NC(C2=C(C)CC2)=O)=O)CC(C)OCC1C O=C(C1=CC2C=CC(C1)C2)NC1COCCN(C(=O)C=Cc2cocn2)C1 N1(C(c2ncn(C(C)C)c2)=O)CCC2CC2(C(N2CCC(F)(CF)C2)=O)CC1 c1(C(=O)NCC(CC)NC(c2[nH]c(C)c(C(=O)O)c2C)=O)coc2c1CSC2 N1(CC(=O)NC2CCN(C(C3CCCCS3)=O)CC2CO)Cc2ccccc2C1 Cc1ccn2cc(C(=O)NC(C3CCCC3)CNC(c3cc(F)c[nH]3)=O)nc2c1 N#Cc1ccc(S(=O)(=O)NC2CCN(C(C3CCC4CCC(=O)N4C3)=O)C2)cc1 C1(NC(c2nccc(C)c2)=O)C2CC1N(C(c1ccsn1)=O)C2C N1(C(CC(C=C)(C)O)=O)CC(NC(=O)C(Cc2ccccc2)OC)CC2(CC2)C1 c1(C(=O)NCC2(C)OCCN(C(C(C)OCC=C)=O)C2)ccc2ncccc2n1 C#Cc1cc(F)c(C(=O)NCCCNC(C2COC(=O)N2)=O)c(F)c1 c1(C(=O)NCc2cncc(Cl)n2)cnn2ccc(-c3cc(F)c(O)c(F)c3)cc12 c1(C(=O)NCCCCCC)ccc(F)c(C(=O)OC)c1.c1(C(=O)N)cnc(Cl)s1 Cc1ccc2[nH]c(C(=O)N(C3CCN(CCC4CCCCO4)C3)CC)c(C)c2c1 Cc1ccc(N)c(C(N2CC3CC3C2)=O)c1.c1(C(N(C)C)=O)ccc(=O)n(C)c1 CC1(C(=O)NC2CCC(F)(C)C2)CCCC1(F)F.c1(C(=O)N)c[nH]c(C#N)c1 N1(C(c2cc(OCC)ncc2)=O)CC(C)OCC1=O.c1(C(=O)O)ccc(C)cc1 C(=O)(C1CCCc2ncnn21)N1CC(Nc2cc(OCC)ncn2)C(C)C1 c1(CC(=O)NC(C2CCCN2C(c2cc(Cl)ns2)=O)C)cccc(C(F)F)c1 C1(NC(c2c(CC)csc2)=O)CCC2CC1CN2C(c1cc(C)n(C)c1C)=O C1(C(=O)NC(CC)C2CCC2)CC2CCC(C1)N2C(C1COCC1(C)C)=O C(=O)(C#CC1CC(F)(F)C1)NCCC1N(C(C2=C(C)OCCS2)=O)CCCC1 C1(N(C(CCC2(C)CN(C(CC3ON=C(C)C3)=O)C2)=O)C)CC(C)OC(C)C1 C(=O)(NN1CCCC1C(=O)N(CC(N1CCCC1)=O)C(C)C)C1C(=C)C1 Cc1ccc(F)cc1C(N1CCOCC(CNC(C2CC3CCC2C3)=O)C1)=O N1(C(c2c(CC)noc2C)=O)CC2CCC(C)C2C1.C1(C(=O)N)OCCC1(C)C c1(CC2(C(=O)NCC3CCCO3)CN(Cc3nnn(C)n3)C2)ccccc1Br CCC(CC)(CCNC(=O)C(C)CC1CCCO1)NC(=O)COC(F)F C(=O)(C(O)CC(C)(C)C)NCCCC(C)NC(C1CC(=O)CCO1)=O Cc1ncc(C(N2CC(NC(C3CN(C)CC3C)=O)C2)=O)c(C2CC2)n1 C12(OCC)CCC(C(N3CCC3)=O)(CC1)C2.c1(C=O)ccc(N)c(Cl)n1.C C(Cc1cccc(C(F)(F)F)c1)CC(=O)N(CC(C)O)C(C)C.C(C=O)=C.CC Cc1cc(C(=O)NC(C)CNC(=O)CC(c2cccc(F)c2)C)cc(F)c1C C1(C(N(CC(CN(C(=O)C=O)C)O)C)=O)CC(=O)NC1(C)C.c1ncc[nH]1.N C#Cc1ccc(C(N2CCCC(C)(C)C2C(=O)NCC(C)(O)CO)=O)c(C)c1 c1(C=O)cc2c(s1)CC(C)(C)C2.C(C)C(C)C.C(C(=O)N)N(CCOC)C C1(CNC(C(C)SC)=O)CCC(F)(CNC(c2cc(O)n(C)n2)=O)C1 C1(OC)CCCS(=O)(=O)C1.N1(C)C(=O)CN(CCn2ccc(C(C)C)n2)C1=O N1(C(C(=O)NC2(c3c(F)cccc3Br)CC2)=O)CC2C3CCC(CC3)C2C1 CCC(CC)N=c1[nH]c(=NC)[nH]c(=NCCC2CCCC2(C)C)[nH]1 c1(C(N(CCN(C(C(CSC)C)=O)C)C(C)C)=O)ccc2c(ccn2C)c1 N1(C(C2CCC(C)N(C(C3CCCCC(=O)C3)=O)C2)=O)CCc2ccccc2C1 N1(C(C)C)CCc2onc(C(=O)NC3(C)CCN(C(=O)CCC(C)(C)F)C3)c2C1 CC(=O)C(C)(C)CC(=O)NC(CNC(c1csc(O)n1)=O)C1CCC1 N1(C(N2CCC(=C)C2)=O)CCC(C(=O)NCCO)CC1 C(CCCCC(=O)N1CC(NC(c2ccc(N(C)C)cn2)=O)C(C)(C)C1)N(C)C N1(C(=O)C(F)F)CCC2(CCN(C(C3CCN(Cc4ccccc4)C3)=O)C2)C1 CC1CN(C(c2ccnnc2)=O)C1C(=O)NC1CC(O)(CO)C1 C(=O)(C1=CCC2CCC1N2C(C1CC12CC2)=O)NC1C(C#C)CCC1 c1(OC)ccc(C(C)C(=O)NCC(c2ccc(C)cc2)C)cc1OC C1(OC)CCC2(CCN(C(C3(CCNC(=O)CC4CC4)CCCC3)=O)C2)C1 CP(C)(=O)CCC(=O)NC1CCC(NC(C2CN(C3CCCCC3)C2)=O)CC1 c1(C(=O)NC(C2CC3(CCC3)C2)C(=O)OC)ccccc1CC#N Cc1ccc2c(c1)CC(C(N1CC3CCN(C(=O)CSC4CC4)C(C3)C1)=O)S2 c1(N2CCC(NC(COC3(C)COC3)=O)CC2)ccc([N+](=O)[O-])cc1 C(C)(C)(CC(C)(C)C)NC(CC1CCC(NC(Cc2cc(C)nn2C)=O)C1)=O Cc1ccc(C)n1CC(=O)NCC1(NC(=O)CC2OCCC2(C)C)CCC1 C(C)(C)(CC(F)C(=O)NCc1cc(C)c(C)o1)NC(C(C=CC)O)=O c1(CNC(CN(C(=O)C)CCC)=O)cccs1.C(=O)C(C)CC.CCO.C C1(N(CCC)C(C2CC2(C)CC)=O)CCN(C(=O)C(c2cccc(C)c2)=O)CC1 C(=O)(C1CCc2snnc21)N1C(CCNC(=O)C(F)=CC2CC2)CCC1 Cc1cc(F)ccc1C(O)C(N1CCC(CCNC(c2sccc2C)=O)CC1)=O C#Cc1cc(C(=O)NCC2(NC(=O)CCF)CCCCC2C)cc(F)c1 N1(C(C2(C)C(C)C2)=O)CCCC(C(N2CC3CC(N4CCN(C)CC4)C2C3)=O)CC1 N1(C(CCn2c(=O)cc(C)nc2)=O)CCC2(C1)CN(C(c1ccsc1)=O)CCO2 c1(N2CCCC3(NC(c4nc(C)oc4)=O)C(C2)C3)nccc2c1C(=O)OC2(C)C N=c1[nH]c(Cl)c([N+](=O)[O-])c(=NCCOCCNC(c2ccc3ccncc3c2)=O)[nH]1 N1(C(C2C(C(=O)OC)C=C2)=O)CCC(C)(C)C(C(N2Cc3ccncc3C2)=O)C1 c1(C(N(C)Cc2ccccc2N2CCOCC2)=O)cccn(CC(=O)OC)c1=O c1(C(=O)NCC(C)N(C(=O)CCC(C)OC)CC)n[nH]cc1[N+](=O)[O-] C1(O)(CCNC(=O)C(C2CCCCC2)O)CN(C(c2ccoc2C2CC2)=O)C1 CCCC(CNC(=O)CCC(C)(C)N(C)C)C(=O)N(C)Cc1ncc(C)o1 C(=O)(CCCC1OCCO1)NCC(C)CNC(c1cnc(C2CC2)[nH]1)=O Cc1onc(C(=O)NC2CCC2CNC(=O)C2=COCC2)c1Br c1(C(=O)NC2CC(NC(COC3(C)CCCC3)=O)C(O)C2)cccc2cnsc12 CCCC(C(=O)NC(C)(C)C(=O)NC)NC(=O)CN1CCC(C)CC1 C1(c2n(CC=C)nnn2)(Nc2cccc(N3CCCCC3)c2)CSCC1C C1(NC(CCOCCOC)=O)CCC(O)CN(C(=O)CC2(OC)CCC2)C1 c1(C(C(=O)N(C2CCN(C(c3ccc(Cl)s3)=O)C2)CCC)O)cccc(F)c1 CC(CCCCNC(=O)Cc1n[nH]c(=N)s1)NC(c1ccc(C2CCC2)nc1)=O N1(C(c2cncc(SCC)n2)=O)CCC2(CC2)C1.c1(C=O)ccnn1CCF.N C1(NC(CN2CCCC(CC)C2)=O)CN(C(c2nnn(C)n2)=O)CC12CC2 C12(C=O)CCC(C)(C1)OC2.Cc1ccc(C(=O)NCC23CC(CO2)C3)cn1 C1(N(C(CCCN(C)C)=O)C)CCN(C(C2CCC(C)(C)OC2)=O)CC12CC2 CON=CC(=O)NC(Cn1cccn1)C(=O)N1CCC1C(N)=O c1(C(=O)NC2CCN(C(c3cc(CCC)[nH]n3)=O)C2)oc(C)nc1CC C(CCC)(C(=O)NCC1CCN1C(=O)CCSCc1ccccc1)=CCC C1(C)(CNC(CN2C(C)CC2)=O)CCN(C(c2c(C(F)F)cnn2C)=O)C1 C(C(C)(C)C(=O)NCc1ccncc1)N(C)C(c1cn(C2CC2)cn1)=O C(=O)(C(F)(F)C(C)O)N1CCC(N(C(CC(=O)N)=O)C)C1.CC(=O)NCC c1(C(=O)OCC)sccc1-n1cc(C(C)NC(=O)CC2(C)CCOC2)nn1 c1(CC)c(C(=O)NCC(C)NC(c2ccn3nccc3n2)=O)cnc2ncnn12 C=CC1(CC(N2CC(CC(C)NC(c3cnco3)=O)C2)=O)CCCCC1 Cc1c(NC(N2CCC3OC(=O)NC3C2)=O)ccc(C#N)c1C#N CC1(C)CC(=O)c2ccc(NC3CC4CCC3N(C(C3(CO)CC3)=O)C4)nc2C1 C(=O)(CC(C)(C)CC(F)F)NC(C)CC1CN(C(c2cc(Br)no2)=O)C1 C1CC2CCC1N(C(=O)Cn1nnc(=O)[nH]1)C2.C1(C)(CC)CC1C(=O)N.C c1(OC)ccc2c(c1)C(n1cc(C(C)N(C(=O)CCC=C(C)C)C)nn1)CCO2 Cc1cccc(C(=O)NC2CC3(C2)CC3C(=O)N(CC(O)CO)CCO)c1O c1(C(N2CCC(F)(CNC(CCOC)=O)C2)=O)cccc2cc(O)ccc12 N1(C(C2(C(C)C)CC2)=O)CC2CC(NC(=O)CC3(O)CCCN(C)C3)CC2C1 C1(CCC(=O)N(CCC)CCC)CCCCN(C(C2CSC2)=O)C1 c1(NCC2N(N(C(C3(CO)CCN(C)C3)=O)CC)CCC2)nccc(C)c1N c1(CCC=O)cnc2n1CCOC2.C1(F)CCC1.C1(CC=C)(C(=O)NC)CC1 c1(N2CC3(CCOC3)C2)cc(C)c([N+](=O)[O-])cc1C#N.C(C)(C)(C(=O)N)OC.C C=CC1CN(C(C2CC(O)CN2C)=O)CC1NC(=O)Cc1c(C)cccc1C c1(C(N2CCN(CCCCCNC(CCCC#C)=O)CC2)=O)c(Cl)c(C)nn1C C1(C(=O)NC(C(=O)NCC(CC)C#N)c2cccs2)CN(C)CC(C)O1 Cc1sc(C)c2sc(C(N3CC(NC(=O)CC4(N5CCCC5)COC4)C3)=O)cc12 C1(CNC(CCCc2ccc(C)s2)=O)CC(NC(=O)C2=NNC(=O)C2)C12CCC2 C1(NC(c2n[nH]cc2[N+](=O)[O-])=O)CCOC12CCN(C(=O)C1=CCOC1)CC2 c1(OC)ccc(Cl)c(Cl)c1C(=O)NCCCNC(=O)CC(C)(C)F C(=O)(C1=NOC(C)(C)C1)N1CC(C)C(NC(c2ccc3ncccn23)=O)C1 N1(C(CCN(CCCCC)C)=O)CCC2(CC1)CN(C(=O)C(C)OC)C2C(C)C C1(C(N2CCC(C)C2CNC(c2ccncc2F)=O)=O)CCOC(=O)CC1 c1(C(=O)NCC(CC=C)NC(c2ccc(CO)s2)=O)cc(Cl)sc1Cl c1cccc(C)n1.C12(CCOC1)C(=O)N2.c1(COC)ccoc1C(=O)NC.C C1(C(=O)NCCCC2(NC(C=C(C)C)=O)CC2)CC2(C1)CC(C#N)C2 Cc1cc(N)c(C(=O)NCCC2CCCC2)c(F)c1.C1(C(=O)N)CN(C)CCO1 c1(N2CC(C(C)NC(=O)CCc3ccncn3)OCC2)ccnc(C#N)n1 c1(C(=O)NC(CC(C)NC(c2cn(-c3cnn(C)c3)cn2)=O)C)cc(C#N)c[nH]1 C(=O)(C(C)(F)C(=O)OCC)NC12C(CN(C(C(C)SCCCC)=O)C1)C2 CC(C)CC(O)C(=O)NC1C2CN(C(C3CC3C3CC3)=O)CC12 N1(C(C2N(C(=O)OC(C)(C)C)CC(F)C2)=O)CCCCC1.C(=O)C1CC1.C C(CCC(C)C)(C(=O)N)NC(c1n(CC#C)cnn1)=O.C1(C(C)(F)F)CC1 c1(C(N(C2CCN(C(c3coc(Cl)n3)=O)C2)CCO)=O)cnc2n1CCCC2 N1(C(C(C=C)(C)C)=O)CCC(O)C(NC(=O)C=Cc2cocn2)C1 Cc1cc(CC(=O)N(CCCNC(C2C3COCC23)=O)C(C)C)n[nH]1 Cc1ccncc1CC(=O)NC1CCCC1.c1(C(=O)N)c(C)coc1C(C)(C)C c1(C(=O)NCCCN2CCN(c3c(N)cccc3)CC2)cccc2nc[nH]c12 Cc1cc(C(=O)NCC(C)(C)CNC(=O)Cn2cccn2)cn1C c1(CC)ccc(C=CC(=O)NCC2CC(NC(c3oncc3Br)=O)C2)o1 Cc1ccc(C(=O)Nc2cccc(NC(=O)COC(F)F)c2)c(F)c1F C1(C(=O)N(CCO)C2CC2)CC(F)CN1C(C1CC(O)C1)=O C1(C(N2CCN(C3CN(C(CC(C=C)CC)=O)C3)CC2)=O)CCc2nc[nH]c2C1 N(C1CC(C(=O)O)c2ccccc21)C(c1c(-n2c(C)nnn2)cc(N)cc1)=O c1(-c2ccc(C(=O)NC)cc2)ccc(Br)nc1C C1(CCNC(C2CN(C(C)C)C2)=O)CN(C(=O)CN(C)C2CC2)CCO1 C1(CCN(C)C(C2CCCN2C(c2coc(CO)c2)=O)=O)CCCN1C C1(COC)CN(C(=O)C=Cc2cccc(OC)c2)CCC1.C(=O)C#CC(C)C.N O=[N+]([O-])c1cc(Br)cc(F)c1SCCS(=O)(=O)CC1CC1 N1(C(c2ccn(C)c2)=O)CCCC1(C)CNC(C1CC(=C2CC2)C1)=O Cc1ccnc2c(C(=O)NC3CN(C(C4CCCN4C=O)=O)CCC3F)cnn12 C1(NC(CCC=C)=O)CN(C(c2ccnc(OC)n2)=O)C2CC12 c1(CC)ccc(F)c(C(=O)NCCC(O)C)c1F.c1(C=O)ccc([N+](=O)[O-])[nH]1.N C1(NC(c2ccc(C(F)(F)F)cc2Cl)=O)CC2CSCC2C1 C1(C(=O)NCC(Cc2ccccc2)NC(CCC(=C)Cl)=O)CNC(=O)CC1(C)C CCCCCCCC(=O)N1C2CCC1C(CNC(c1ncsc1CC)=O)C2 CC1(C(=O)Nc2cccc(CO)c2F)CCCN(C(=O)CCc2ccoc2)C1 c1(C(=O)NCC2(O)CN(Cc3nccc(OC)c3)C2)cc(C)cc(C)n1 c1(C(=O)NC(C2CCN(C(C3(CC)CC3)=O)CC2)C)[nH]c(=N)ccc1C C1(CC(=O)N)CCCCC12CC2.c1(C(=O)OC)nc(C(=O)NC2CC2)cs1 C1(NC(C(C=C)CC)=O)CC2(CCN(C(c3c[nH]cc3C(C)C)=O)CC2)C1 c1(CC(N2CC(F)(C(=O)NC3CC(=O)OC3)C2)=O)ccc(Br)cc1 N1(C(C(C)SC)=O)CC2(C1)CN(C(=O)CC1CCCCC1(F)F)CCO2 CN1C(=O)COC(CNC(C2(CN)CC(O)C2)=O)C1c1ccccc1 C1(CNC(C2(CNC(Cc3cn(C)nc3)=O)CCC2)=O)CCCOC1(C)C C1(C(=O)NCC2(C)CN(C(C3(O)CC(F)(F)C3)=O)CCO2)CCc2nn[nH]c2C1 C1(OC)CN(C(c2ccc(F)cn2)=O)CC1NC(C1CN(C)C1)=O N1(C(c2nccc(OC)c2)=O)CCC2(CC1)CCN2C(=O)C(S)C(C)C N1(C(C(CC=C)CC)=O)CCC(=O)NC2CN(C(=O)Cc3coc(C)n3)CCC12 C(C(=O)N1CC(OC)C1)(C1CN(C(=O)C(C)OCOC)C1)OC c1(C(=O)OC)cnc(N2CCC(CC)CC2)c(Cl)c1.C(C=C(Cl)Cl)=CC(=O)N c1ncccc1C(=O)N(C1CN(C(=O)C(n2ccc(C(F)(F)F)n2)C)C1)C.CO c1(C(=O)N)cnc(N)c(Cl)c1.Cc1n[nH]cc1CC(=O)NC12CC(C)(C1)C2 CC(C(=O)N(CC(O)CNC(C1(OC)CS(=O)(=O)C1)=O)C)S(N)(=O)=O C1(CNC(=O)C=Cc2ccc(F)nc2)CN(C(=O)COC(F)F)CCC1(F)F C#CCCCC(=O)NCc1nc(C(=O)N(CC)CC2CCC2)c(C)o1 C12COC(CS)(C1)C2.C(CCC(=O)NCC(=O)NC1CCCC1)OCC C1(CN(C(CCN(CC=C)C(c2csc(F)c2)=O)=O)C)CCOC1C N1(C(c2cn(C3CCN(C)C3)nn2)=O)CCN(C(=O)CCOC2CC2)C(CF)C1 CC1(C)CCC(n2cc(CS(C)(=O)=O)nn2)CN1C(c1cccc(Br)c1F)=O Cc1oc(C)c(C(N2CC(NC(=O)C=Cc3ccc(F)cc3)C2)=O)c1C c1(C(N2CC(CNC(c3cc(OC(F)F)n[nH]3)=O)C2)=O)nc(Cl)sc1Cl CC(C)C(O)C(C)(C)C(=O)N(C)CC1(NC(=O)CN(C)C)CC1 C(=O)(C(CC)CC(F)(F)F)N1CC(CNC(CCSCCC)=O)C(C)(C)C1 C(c1ccc(OCCn2ncnn2)o1)=CCNC(CC1(N(C)C)CCC1)=O C12(CNC(C3C(C)C3C)=O)CCC(NC(c3ccnc(CO)c3)=O)(CO1)C2 Cc1c[nH]cc([N+](=O)[O-])c1=NCCCCNC(=O)COc1ccccc1Cl Cc1[nH]c2ncccc2c1C(N1CCCC1CNC(C1CC1C(F)F)=O)=O c1(C(=O)NCCNC(C2C(OC)(OC)CC2)=O)cc(N2CCCCC2)ccn1 C(=O)(NNC(=S)NCCOCC)c1cc(CCC)c(C)s1 N1(C(C(C)OCC)=O)CCC2(CCC2C)CC1.c1(C=O)cn(C)c(C)cc1=O C1CCC12CC(C(N1CC(n3ccnn3)C(C)C1)=O)C2.C(C)=O.CC=CC.N c1(CC(=O)NCC2CCN(C(C(C)OC)=O)C2)ccc(Br)c(O)c1 C1(NC(C(CC)OC)=O)CC2CCCC(C1)N2C(c1cnc(CC(C)(C)C)s1)=O N1(C(C2N(S(C)(=O)=O)CCC2)=O)CCCCC(NC(=O)CC2COC3CC2C3)C1 N1(C(=O)OCC)CC(C2CN(C(=O)NCCC)C2)C1 c1(NCCCCCCC)ccc(COC)c(C#N)c1 N1(C(C(C(C)C)F)=O)CC(C)(C)CC1CC(=O)NOCCOCCF c1(C(=O)NC2C(NC(=O)Cc3ccoc3)CCC2)ccncc1Br CC(C)C(CC(=O)NC1CC1NC(=O)CCCc1cccnc1)c1ccccc1 C1(CCC#N)NC(=O)N(Cc2ccc(CN3CCCC3=O)cc2)C1=O C1(C(=O)NC(c2ncccn2)CC)COCCN(C(C2CC(CF)C2)=O)C1 C1(C(N2C(C)CCCC2)=O)N(C(C2CC(C)N(C)C2)=O)CCCC1(C)C Cc1nc2cc(C(=O)OC(C)C(=O)NC(C)(C)C)ccc2o1 C1(CNC(c2c(C)onc2)=O)CCCCCN1C(C1OCC2CCCC12)=O C12(C(=O)NC(c3c(C(N(C(C)C(F)F)C)=O)con3)C)CCC(CC1)C2 CC1(C)C(NC(c2cnc(-c3ccoc3)s2)=O)CCN1C(=O)CO.C1CCOC1 C(CC1=CCN(C(c2ccc3ncnn3c2)=O)CC1)NC(=O)CC(F)(F)F C(CNC(C1CCSCC1)=O)(C(C)C(C)C)NC(C(c1nccc(C)c1)(C)C)=O C(=O)(C(C)(CSC)NC(=O)Cc1cccnc1O)N(CC#C)CCF C1(C=O)C2CC3C(C2=O)C13.C(=O)(CC(F)(F)F)N(CCCc1cccs1)C.N Cc1cc(C2CC2)ccc1C(N1CC(CNC(c2nccc(F)c2Cl)=O)C1)=O Cc1cccc(C(C)C)c1C(=O)NCCNC(=O)C(F)Cc1ccccc1 N1(C(COCCCOC)=O)CCC(NC(C2CCC(=O)N2C)=O)C12CC2 c1(NC(C)(C)C)ccccc1C=O.C1(C=O)CCC(=O)N1.C1CC(CC)C1.N c1(C(N2CC3(C(NC(CS(C)(=O)=O)=O)CC3)C2)=O)cc(C#N)c(N)cc1O c1(C=O)cccc(C(F)(F)F)n1.CC1CCC(=CC(=O)N)C1.C1(F)CCC1.C C(=O)(N1CCC(C(=O)NCCC2CCC(=O)N2)O1)C1C(C)C1C N1(C(c2ccc(C)n2C)=O)CC(C)C(C)(C)C1.C1(C(F)(F)F)(C(=O)N)CC1 c1(NC(=O)Cc2cn(-c3ccccc3)cn2)ccc(N2CCCS2(=O)=O)c(F)c1 C(=O)(C(CC=O)C(C)=O)OCC.C1(C=O)CC(O)CN1C(C)=O.C1CC1 c1(C(C(=O)NCCN(C(c2cnc(CCC)s2)=O)CCC)C)nc(F)ccc1Cl N1(C(CC2(NC(C)=O)CC2)=O)CC2CC1CN2C(=O)C(C)N.c1nc(C)cs1 C1(C(=O)OCC(c2cnc3ncccn23)=O)CCc2ccc(F)cc2O1 C(=O)(C1Cc2ccccc21)NC(C1CCN(C(c2c(OC)noc2C)=O)C1)(C)C C(C)(C(C)(C)C)NC(CC(n1ccc(C)n1)C)=O.c1(C(=O)N)cnn(CCF)c1 N1(CC(=O)N(C2CC2)Cc2nc(C)sc2)CC(O)CC1C(C)C C1(C(=O)NC(C23CCC(CO2)C3)C)CC2CC2N1C(C1CC(O)C(F)C1)=O C(=O)(CC(O)CCSC)NC(c1ccc(C)cc1)CNC(C=C(CC)C)=O CN1C(=O)CCC1C(=O)N(C1CC(NC(C2(C(F)(F)F)CCC2)=O)C1)C C(=O)(C1=CC2CCC1C2)N1CCC(N(C(Cc2cnc(C)s2)=O)CCO)CC1 c1(C(N(CC(N2CCOC3CC23)=O)CCOC)=O)cc(O)ncc1F c1(C(N2CCN(C(C3CC4CC4C3)=O)CC2C2CC2)=O)cc2cccc(Cl)c2o1 C(CN=C(NCc1ccc(F)cc1OC)N1CC=C(F)C1)OC C1(CC)(CC)CCCN1C(C1CCS(=O)(=O)C1)=O.C1(C=O)CC(F)(F)CS1 Cc1cccc(CN2CCC(O)(C(N3CCN(C(=O)N(C)C)CC3)=O)C2)c1 N1(C(c2cn(C)nc2)=O)CCC2CCN(C(C3(C#N)CCCO3)=O)CC12 CC(=O)CC(C)(C)C(=O)NCCC(O)C(=O)N(CC(C)C(C)C)C N1(C(C2N(CC)CC2)=O)CCC2(CCC2C)CC1.c1(C=O)occc1C(C)C n1(C(C(=O)N(CC)CC)(C)C)cc([N+](=O)[O-])cn1.C1(C=O)CCN(C)C1C N1(C(C(=Cc2ccccc2)CC)=O)CC2CCN(C(=O)C(C)SC(C)C)CC2C1 CC1CCCCC1C.c1(C=O)ccc(F)c(C(C)(C)F)c1.C(=O)(CNC=O)N N1(C(CSc2ccc(C)cc2)=O)CCCN(C(=O)CC2(C)CC2)CC1C C(=O)(C(F)CC(C)(C)NC(=O)C(C)CC1CC1)NC1C(OC)COC1 Cc1cc(C(=O)NC2CC3(C2)CC3NC(C2CCOC2)=O)nnc1C.C(C)C c1(C(C(=O)NCCOC)N(CCC2=CCCCC2)CC)ccc2nonc2c1 C(=O)C1CCCc2ncnn21.C1(CCC2N(CC=C(C)C)CCC2)CC(F)(F)C1 C(=O)(C(C)(C)C(N)=O)NC(CC(C)C)CNC(C1CCCOC1C)=O C1(O)(C(C)NC(C(C)N2CCC2)=O)CCN(C(c2cc(Cl)n[nH]2)=O)CC1 C1(CCNC(CCN(C(C)=O)C)=O)CCCN(C(c2coc(C)n2)=O)CC1 CC(C#N)C(=O)NC(C)CNC(=O)COC1CCC1 N1(C(c2c(C)n[nH]c2)=O)CCC=C(CNC(=O)CC=C(Cl)Cl)C1 C(C)(CC(=O)N1CC(C(O)C(=O)NCc2nncn2C)C1)OC N1(C(C(CC)NC(C)=O)=O)CC(NC(=O)Cc2cnc[nH]2)CC2(CCC2)C1 C(=O)(CC(C)CC(F)(F)F)N1CCCC(C)(CNC(Cc2nc(C)c(C)[nH]2)=O)C1 O=C(CCC(Br)Br)NCC1CNC2CC2C1 CC1(C)CN(C(=O)C(F)F)CC1NC(c1cc(Cl)c(Br)cn1)=O c1(N(CCN(C(c2c(C(C)C)n(C)nc2)=O)C(C)C)C)ncnn2cccc12 C1(CNC(C(C)=C2CC2)=O)CCC2CN(C(=O)C(N3CCOCC3)C)CC12 c1(C(=O)N)ccc2nnc(O)n2c1.c1(C(N(CC(C)C)C)=O)ncoc1C1CC1 N1(C(c2cnn(CC)n2)=O)CCCC(C2(NC(=O)CCC3(C)CC3)CC2)C1 c1(C(=O)NC(CCNC(Cc2c(F)ccc(C)c2)=O)C)cc2nccn2c(O)n1 c1(-c2c(OC)nccc2C)cnc2ncc(C(=O)NCc3ncccc3C)n2c1 N1(C(C2CCCC(CC)C2)C(=O)NC2CC2)CCc2sccc2C1CC C1(NC(C2CCC=CCC2)=O)CCOC12CCN(C(=O)CN1CCCCC1)CC2 c1(C(C)C)ncc(Cl)c(C(=O)NCC(O)CNC(=O)C(C)S(N)(=O)=O)n1 Cc1ccn(CC(=O)NC2(CN(C)C(C3CC4CC4C3)=O)CC2)c(=O)c1 CC1CCC(C(N2CC(F)(CF)C2)=O)N(C(=O)C=CC2CC2)C1 N#Cc1ccc(N2CC(C(N3CCC(N4CCCS4(=O)=O)C3)=O)CC2=O)cc1 C(C(N=c1cnc(C(=O)OC)c[nH]1)C(C)C)NC(c1c(CCC)n(C)nc1)=O C1(n2cccn2)(CC(=O)NC(CC)C)CCN(C(=O)CC2C(=O)NN=C2C)CC1 C1(O)(C(=O)NCc2cn(CC(=O)NC(CC)C(C)(F)F)nn2)CCCCCC1 C1(NC(N2CCN(CCN)CC2)=O)CCCC(C(F)F)CC1 C1(N(C(=O)C=Cc2ncco2)CCO)CCCN(C(=O)COCC(F)F)C1 C1(NC(CC(C)C)=O)CC(F)CN(C(=O)CN2CCCC2CO)C1 C1(C(N(C)CCn2cccn2)=O)CC2C=CC1N(C(c1[nH]nnc1C1CC1)=O)C2 N1(C(C2(COC)CCOC2)=O)CCC2(CCCN2C(c2ccc(C)s2)=O)C1 C12(C=O)CCN(C1)S(=O)(=O)C2.c1(CC(=O)NC2CCCC2)cccc(F)c1F c1(C(=O)NC2CC3C(NC(CC(COC)C)=O)C3C2)cnc2cc[nH]c2c1 c1(N(C(C2CCC(N)CC2)=O)Cc2cccc(OC(C)C)c2)ncc(Cl)cc1F C1(C(=O)NCCC(=O)NCC)CC2CC1CN(C(c1cccs1)=O)C2 C1(CNC(CC(C)(C)C2CC2)=O)CC2CCC1N2C(=O)CCc1ccncc1 c1(OC)nc(C)ncc1C(N1CCC(c2ccc(OC)cc2)CC1)=O CC(C)C(C)CC(=O)NCCCOCCNC(=O)C(C)CN(C)C N1(c2nc(CCOC)on2)CCCC1=O.c1(C(=O)N)cncc(C(=O)C2CC2)c1 c1(C(=O)NC2CCCN(C(=O)CCc3ccon3)C2)cnc2ncnc(O)c2c1 c1(C(=O)NCC(C)Cc2cn[nH]c2)ccc(C)s1.C(=O)(CCn1cccn1)N C1(O)(CC)CN(C(c2ccc(C3CC3)o2)=O)C1.C1(C=O)CC(N(C)C)C1.N C1(C(N2CC(CNC(=O)CC3CCCCO3)C2)=O)CCCCN1CC(F)F c1(SC)cccc(C(=O)NCCC)c1.c1(C(=O)N)cc(C)n(CC(F)(F)F)n1 N1(C(C(CC)CC(F)F)=O)CCCC2(C1)CN(C(c1cnsc1C)=O)C2 c1(C(N2CC(COC)(NC(=O)CC(O)CC)C2)=O)ccc(F)c(F)c1F c1(N(CC(C(C)C)C)C)nc(N2CCC(P(C)(C)=O)C2)nc2ccsc12 C(=O)C(O)(C(C)C)C(F)(F)F.C(C)(C)C(C)C.C(CC(=O)N)SCC(C)C Cc1cc(=N)[nH]cc1C(N1CC(NC(=O)CCCC(=O)N(C)C)CC(F)C1)=O c1(C(=O)NCC(CNC(C(C)OCCCC)=O)C)cc(N)cc(N)c1 C1(C(=O)NCCCCN(C(CC(C)NC(N)=O)=O)C)OCCC1(C)C C1(CC(=O)NCCc2cn(CC)nn2)COCCN1C(=O)Cc1cc[nH]c1 CCCC(CNC(c1cn(C2CC2)nn1)=O)C(=O)N(CC(O)C1CC1)C CCCC(C#N)C(=O)N1CCCC(CC(N2CCCCC2C(=O)OC)=O)CC1 c1(C(N2C(CNC(=O)Cc3cnc(C)[nH]3)CC(OC)C2)=O)ccc(F)cc1Cl c1(NC(c2n(C)nnn2)c2cnc(-c3ccccc3)s2)ccc2c(c1)COC2 c1(CN2CCC(O)(C(N3CCC(n4cc(I)cn4)CC3)=O)C2)cccc(O)c1Br N#Cc1ccc(CN2CCC(CNC(c3c(O)cc(Br)cc3F)=O)C2)cc1F N1(C(C=CCCC)=O)CCC2(CCCN(C(=O)C(C)CC(F)F)C2)CC1 N1(C(CCCCC(C)C)=O)CC(C)OC2(CCN(C(C)C(=O)N(C)C(C)C)C2)C1 C(=O)CCS(=O)(=O)N(C)C.CC1CC(=O)NC1C(=O)NCC1CC(F)C1 c1(C(=O)NCCN(C(C#CC(C)(C)C)=O)C2CCCC2)nc2ncccn2n1 CC(C)C(C#N)C(=O)NCC1(C(=O)NCC(C)(F)F)CC1 c1(-c2cc(C=O)on2)ccccc1F.CCC(CNC(C1CC1)=O)OC(C)=O c1(C(N2CC(C)(NC(CCSCCC)=O)C2)=O)cc2cnn(C(C)C)c2nc1C c1(CNC(=NC)N(C)Cc2ccc(Cl)s2)nnc2cccnn12 c1(C=O)ccc(C)c(C)c1O.C1(C(F)(F)F)(C(NCCC)=O)CCCCO1.CC c1(OC(C)C(=O)OCC(C2CCOCC2)F)cnc2ccccc2c1 C=C(Br)CC(C)(C)C(=O)NCCC(C)NC(=O)CC=C(C)C CCC(C)C(O)C(=O)N(CCNC(=O)CC(C)F)C1CC1 C(C(C(=O)NCc1cnn(CC(F)(F)F)n1)NC(c1ccccc1)=O)OC c1(NC(CCC)CCC)ccc(S(=O)(=O)NC2CC(CC)C2)c(Cl)c1 c1(C(=O)OCC)ncc(Cl)c(=NCC(C)(C)NC(=O)COC)[nH]1.CC c1(CC(=O)N)ccc(C)c([N+](=O)[O-])c1.C1(C(=O)NCCCC)CN2CCC1CC2 CC(CCC(=O)NCC1CN(C(c2ccnc(C(F)(F)F)c2)=O)CCO1)N(C)C CC1CN(C(C2(C(F)F)CCC2)=O)CC2(CCN(C(=O)CC(F)(F)F)C2)O1 c1(C(=O)NC(C(=O)NCc2cn(CC)nc2)C2CCOC2)snc(C)c1N C1(NC(C(C2CCCCC2)N(C)C)=O)CN(C(=O)CN2CC3CC3C2)CCC1F N1(C(C(c2ccccc2)OC)=O)CCN(CCCNC(C2CC(C)(C)O2)=O)CC1 C=CC(CCC)CC(=O)N1CC2C(NC(c3ncc(C)nc3OC)=O)C2C1 C1(C(=O)NCC2CC(NC(c3c(CC)cncc3)=O)C2)CCCCCC1(F)F c1(OC)ccc2cc(C(=O)NCC3CC3NC(C3CCCC3)=O)n(C)c2c1 CCC(O)C(C)C(=O)N1CCC(CCNC(C2(c3cc[nH]n3)CCC2)=O)C1 c1(C(N2CCC(c3nc[nH]n3)CC2)=O)ccc(Cl)c(F)c1.CC1(C(=O)NC)CC1 n1(CC(=O)NC(CNC(c2c(C)scn2)=O)C(C)(C)C)ncn2nccc2c1=O Cc1c(Cl)ccc2[nH]c(C(=O)NNC(c3ccc(F)c(Br)c3)=O)cc12 C1(CNC(=O)CCN2CCOC2=O)CCC2(CCC2)C1NC(=O)CC=C(Cl)Cl Cc1ccc(C(C2CC2)NCC2CCCC(C(F)(F)F)O2)cc1C CCCC(C)(C)CC(=O)N(C(C)(C(=O)NC1CC2CC1C(O)C2O)C1CC1)C C1(CCC)CN(C(c2ccc(Cl)cn2)=O)CC1C(=O)N(CC)Cc1cccs1 c1(C(C(=O)NC2CC2)N(CCC)CC)cnn(C)c1.C(C)(C)C.C=O.N c1(OC)cncnc1N1CCCCC1CCNC(=O)C(C)Sc1ccccc1 c1(OC)ccc2c(c1OC(=O)C(C)Sc1cc(Cl)ccc1Cl)CCC2 N1(C(C(CC(C)(C)NC(=O)C=C2CCCCC2)F)=O)CCCC2(CCCO2)C1 N1(C(C=CC)=O)C2CCC1C(NC(=O)CC1CCC(=O)N1)C2 C12(CNC(C=CS(C)=O)=O)CCC(CNC(=O)C3=CCCC3)(CC1)CO2 c1(C(N2CCC(C)(CNC(c3csc(O)n3)=O)CC2)=O)c(F)cccc1[N+](=O)[O-] c1(C(=O)N)cccc(Cl)c1.C=CC(C)CC(=O)NCC1CC1C.C(C)C c1(OCCOC(C=Cc2ccc(C3C(C)C3)o2)=O)ccc(Cl)c(C)c1Cl C(N=c1cc(C)n(CCO)[nH]1)(c1n(CCC)nnn1)c1cncn1C(C)C C=C(C)CCC(C)N=c1[nH]c(N2CCC(SC(F)F)CC2)nc2c1CC(C)CC2 c1(NCC)cncc(C=O)c1.C1(C)CCN(C(C2CCCN2C(N)=O)=O)C1.N Cc1cc(O)ncc1C(=O)NC(C)(C)C(C)C.C1(C)(CC=O)CC1(Cl)Cl.N Cc1nc(C)c(C(=O)NC2CC(C)C23CCC3)nc1C.C(=O)C(F)(F)C(F)F.N N1(C(C(C#N)C2CC2)=O)CCN(C(=O)CSC2CCOCC2)CC1c1cn[nH]c1 C(=O)(C1=CC2CC=CCC12)NC1CC(N(C)C(c2coc3c2C(=O)CCC3)=O)C1 N#Cc1ccc2c(c1)CN(C(=O)CCC1CCCN(C(C3CCNC3=O)=O)C1)C2 C1(CN(C)C(C2CC2Sc2ccccc2)=O)CCN(C(C2COCCO2)=O)CC1 C1(N(C)C(c2cscn2)=O)CN(C(=O)C#CC2CCC2)CC1(C)C C1(n2cc(CNS(N)(=O)=O)nn2)CC2CCC1(NC(C1CCC(=O)O1)=O)C2 N1(C(C(N2CCCCC2=O)C)=O)C(C)CC2CN(C(C3CCC3)=O)CC12 C(=O)(CC1CCc2ccccc21)N1CC(OCCC(=O)O)C1 Cc1c(NCCc2c(F)cccc2F)nc[nH]c1=NCC1CC2(CCC2O)C1 c1(CCC(=O)N(C)CC2N(C(C3CCC(CC)O3)=O)CCC2)cccc(F)c1F c1(C(N2CCC(NC(c3ccc(Cl)c(O)c3)=O)C2)=O)ccc2nc(Cl)nn2c1 c1(OCC)ccnc(N2CCCCC2CCNC(C2CCC2(C)C)=O)n1 c1(CC(=O)N(CC#C)CC)cccc(C(F)(F)F)c1.C(=O)CCC1CCC1 N1(C(c2cnc(CC)s2)=O)CCC2(NC(c3ccc(O)nc3)=O)CC2C1 c1(CC(=O)NCC(=O)N(CC)Cc2cn[nH]c2)csc(C)c1 c1(C(=O)NCC23CN(C(CSCCC(C)C)=O)C(CC2)C3)cccc2cc[nH]c12 N1(C(C2C(=C)CC2)=O)CCN(C(c2c[nH]cc2-c2csc(C)n2)=O)CC2(CC2)C1 c1(CC(=O)NCC2C3CN(C(C(CC)OCC)=O)CC32)ccc2n[nH]cc2c1 N1(C(c2c(C)c(C3CC3)on2)=O)CC2CCC1CN2C(=O)C(C)C1CCCO1 C1(OC)CC2CCC(C1)N2C(=O)CC(C)(C)NC(c1cccnn1)=O N1(C(C2C(CC)CCCN2C(=O)CCC2CC2(C)C)=O)CC2(C)CC1CCO2 N1(C(C(C2CCOC2)OC)=O)CC2=C(C1)CN(C(=O)C=CC1CCCCCC1)C2 C(=O)(C1=CC(O)C(NC(C23CCCN2CCC3)=O)C1)NC(C#C)(C)C Cc1cc(N(C)Cc2ccc(F)c(C)c2)nc(N(CC(C)(C)CN(C)C)C)n1 C(CCCCN(C(=O)CC12CCCC1C2)C)NC(C1(CC)CCC1)=O N1(C(COc2ccn(C)n2)=O)CC2CN(C(c3cc(O)nc(Cl)c3)=O)CCC12 N1(C(C(CC=C)NC(C)=O)=O)CCCC(CC)(NC(c2cnc(SC)s2)=O)C1 C=C(C)CCCC(=O)NCCOCCCN(C)C(c1cnc(O)cc1OC)=O C1(C)(NC(C(C=CCCC)O)=O)CCN(C(=O)CCOc2ccccc2F)CC1 c1(C(N2CCC(C(=O)Nc3c(C)cccc3O)C2)=O)c[nH]c2cnccc12 N1(C(CCCOCC)=O)CC2CC(NC(=O)CCc3ncc[nH]3)C2C1 N1(C(c2ccc(SC)o2)=O)CC(NC(C2CC2c2ccc(C)o2)=O)CC(F)C1 c1(C(=O)NCC(CC)(C)NC(=O)CC(C)COC)cc(OC)nc(OC)c1 Cc1ccc(CCNC(c2cnn(C)c2Cl)=O)cc1.C1(CC(=O)N)CCC(C)C1 N1(C(C(C)NC(c2ccco2)=O)=O)CCN(C(C2(C)CC(O)CN2C)=O)C(C)C1 N1(C(=O)NC2C3CC(OCC)CC32)CCCc2ccc(C(=O)OC)cc21 c1(OC)c(C(=O)N)csc1C.C1CC(F)CN1C(C1CSCN1C(C)=O)=O.C O=C(CC1OCc2cc(Cl)ccc21)NC(CC1CC1)C(=O)O C1(CC)CN(C(C2(C(C)NC(C(=O)Cc3c[nH]nc3C)C)CC2)=O)CC1O c1(C(C)NC(C(C)c2nn[nH]n2)=O)ccc(Br)s1 c1(C=O)ccc([N+](=O)[O-])s1.N1(CC(=O)NCC2CC(F)C2)CCS(=O)CC1 c1(NC(C2CN(Cc3cc(Br)ccc3OC(F)(F)F)C2)=O)nc2cccnc2s1 C#CCCCCC(=O)N1CCN(C(=O)Cc2ccc(Cl)c(C)c2)C(CC)C1 C=C(Cl)CC(C(=O)N(CCCN(C)C)C)NC(=O)CCc1cn[nH]c1 N1(CCC(N2CC(NC(c3c(Br)cnc(C)n3)=O)C2)=O)Cc2ccccc2C1=O CCCCCC(C)CC(=O)NC12CCC(CC1NC(c1coc(O)n1)=O)C2 N1(c2ccc(C)cc2)N=C(C(=O)NCCN2CCC(C(=O)O)CC2)CCC1=O N1(C(=O)C=Cc2ccco2)CC2CC(C(=O)NC3C=CCCC3CO)(C2)C1 c1(NC(C2N(C(C(C(CC)O)C)=O)CC(C)C2)=O)cncc([N+](=O)[O-])c1 C(=O)(C(CCC(C)C)N(C)C)NCC(CC=C)NC(=O)CSCC(N)=O c1(N(CCCC)C)ccnc(C(N2CC(NC(c3cccc(CC)c3)=O)C2)=O)c1 NC1CCOc2ccc(NC(N3CCC4(CC3)CC(O)(C(F)(F)F)C4)=O)cc21 c1(C(=O)NCC(CNC(=O)C=Cc2cc[nH]n2)O)cc2c(nc1O)CCCC2=O n1(CCC)ccc(C(=O)NCC(CC)NC(C2CN(S(C)(=O)=O)C2)=O)n1 c1(C(=O)NCCCCCC)nccc(C#N)c1F.C1(CC(=O)N)CCS(=O)(=O)C1 C1(C(=O)NC2(C(=O)NC3(CO)CC(C)C3)CCCC2)CCC=CCC1 C(=O)(C1Cc2c(Cl)cccc21)N1CC(NC(c2cc(OC)cc(CC)c2)=O)C1 N1(C(C(C2CC2)OCC)=O)CCC2(C)CN(C(=O)CCC3CCCCCC3)CC12 C=CC(CC)CC(=O)N1CCOC(C(=O)NCCC(O)CO)C1 C1(c2ccc(Br)cc2)(NC(=O)NC2CCC(OCC)C2)CCOCC1 C#CCCCCC(=O)NC1CC(CCNC(=O)C(C)OC)C1.c1ccc(C)cc1 N1(C(=O)Cc2c(F)cc(Br)cc2Br)CCCc2cc([N+](=O)[O-])ccc21 c1(C(N2CC3C(NC(C4CCC(C)(O)CC4)=O)(C3)C2)=O)cc2ccc(F)cc2s1 N1(C(=O)NC(C#C)CC(C)C)CC(C)Cc2cccc(O)c21 CC(C)C(C(C)NC(=O)CCn1cncn1)NC(c1cncc(N)n1)=O c1(CC(C)NC(N2CCN(C(C#N)C(C)C)CC2)=O)cccc2sccc12 c1(CC)conc1C=O.C1(C(N(CC)C(C)C)=O)CC1(C)C(F)(F)F.N Cc1cccn2cc(CNC(C34CCCC3N(C(=O)C(N)CN)CC4)=O)nc12 c1(N2CC(C)CS(=O)CC2)nc(N2CCn3cncc3C2)c2sccc2n1 Cc1nn(CC(=O)NCC(C)CN(C)C(C2CCS2(=O)=O)=O)c2ncccc12 N1(C(c2ncc(F)cn2)=O)CC(n2cc(CN3CCCCC3=O)nn2)C(O)C1 Cc1cc(Cl)c(C(=O)NCC(F)CNC(=O)CC2CC2(C)C)cn1 N1(C(C(C)NC(=O)NC)=O)CCC(NC(=O)C(C)O)C1 C12(CC)CN(C(=O)C(C)C(F)F)C(CNC(=O)CCCn3ccnn3)(C1)C2 c1(C(N2C(CNC(CCOCCOC)=O)CCCC2)=O)n[nH]c2cccnc12 CC1(C)COC(CCNC(=O)CCN(CCCO)C(c2n[nH]cc2Cl)=O)C1 c1(C(N2CC(NC(C3CC(C)OCC3)=O)C(C)(C)C2)=O)ccn2nncc2c1 Cc1cc(C(=O)N(CC(C)(C)CNC(=O)C2=NOC(C)C2)C)c(F)cc1F c1(CC)ccc(O)c(C(N2CCC(C(C)NC(c3c(C)ncnc3C)=O)C2)=O)c1 CC1CCC(NC(=O)C2=CSCCO2)CN1C(c1cn(C(F)(F)CO)nn1)=O CCC(C(=O)NC(C)CCNC(=O)C=CC1CCCCCC1)C(F)(F)F CCC(CC1CCCC1)C(=O)N1CC(c2ccccc2)C1.C(=O)CCCC1CCCCC1.C N1(C(c2cccc(C(C)C)n2)=O)CC(NC(C2CCCC2)=O)CC12CCOCC2 C(=O)(C1=C(F)CN(C(C23CCCCC2C3)=O)CC1)NC(c1c(C)nc(C)[nH]1)C C1(COC)(NC(c2nc(C)oc2O)=O)CCN(C(c2nnn(C)c2C)=O)C1 C=CCCCN(C(C1CCN(C(=O)CC)C1)=O)CC.C(=O)CCC.C(C)=O.N C1(COC)CN(C(C2CN3CCCC2C3)=O)CCN1C(=O)CCC1CC(C)C1 c1(C(=O)NC2CCN(C(C3CC3F)=O)CC2)ncc(C2CC2)cc1F C#CCC(CC(=O)NCC1CC(CC)=NO1)NC(c1ccc(O)c(C)c1)=O CC1CN(C(c2ccccc2SCC(=O)NC2(C#N)CC2)=O)CC1.C1CC1.N Cc1cc(Cl)ccc1OCC=O.c1(C(N2CC(C)C2)=O)cc(C2CC2)n(C)c1C c1(C=O)cc(N)nc(Cl)c1.c1(SCC)ccccc1C(=O)N(CC)C(C)C C1(CC)OCCCC1C(=O)NC1(CC)CN(C(=O)CSC(C)C)C1 c1(OC)cccc2sc(C(=O)NC)cc12.C12CCC(C1)N(C(c1ccon1)=O)C2 c1(-c2cn(C(C)C(=O)NC3CCCN(Cc4ccccc4)C3)nn2)nccn(C)c1=O c1(-c2n(CC)nc(-c3nccs3)n2)cnn2cccc(Br)c12 N1(C(C2(C)CCCN(C(CCSC)C)C2)=O)CCC2(C1)CN(C)C(=O)CO2 N1(C(=O)CC2CS(=O)(=O)C2)CCN(C(C2OC3CCC2C3)=O)C(CC(F)F)C1 c1(C(=O)Nc2ccccc2Cn2ccnc2)nc2cc(F)c(Br)cc2[nH]1 C1(NC(C(CC#C)O)=O)CCN(C(c2cncc(N)c2C)=O)C(C)C1 c1(CCC(=O)N)csc2nc(C)cn12.C=C(C)CCNC(=O)C(C)c1ccco1 C1(N(C(C(F)=CCC)=O)CC)CCN(C(C2CC2c2ccc(C)o2)=O)CC1 C1(O)(c2cn(CC(C)NC(CC(C)(C)SC)=O)nn2)CCC2COC1O2 N1(C(C(C=C)c2ccccc2)=O)CCC2CC1CN(C(=O)CCCC1CC1)C2 N1(C(CC=CCNC(c2cc(C)sc2)=O)=O)CCC(O)CC1C1CC1 O=C(C1=CCCCCC1)NC1CC2CCC1CC2NC(c1n[nH]cc1Br)=O n1(CC(N2CCC(NC(CCCCC)=O)CC2C)=O)ncn2cccc2c1=O N1(C(c2occ(C)c2)=O)CCCCCC1C(=O)NCCCCC(C)(F)F CC(CSC(F)(F)F)C(=O)N(CCCCN(C)C(C1CCOC1C1CC1)=O)C CCC(CC(=O)N1CCN(C(=O)CC2CCCC2(F)F)CC1CCO)CC(C)C C12(C(=O)NC3C(C)(C)CN(C(=O)CCc4nc[nH]n4)C3)CCCCC1C2(F)F c1(C(N(CC(CC)NC(c2csnc2Cl)=O)CC)=O)nn(C)c2c1CCCC2 Cc1cc(C(=O)NC2CC2C(N2CC3CC3C2C#N)=O)c(Br)cc1F Cc1ccc(S(=O)(=O)C2CCCCC2NC(=O)C(C2CCCNCC2)F)cc1 N(C(=NCCCc1ncn(C)n1)NCc1nnc2cccnn12)C(CC)C c1(-c2c(C3(C(=O)NCc4cn[nH]c4)CC3)cccc2)ccc2c(c1)CCC2 C1(C(=O)NCCCCCNC(C2C(CCOC)C2)=O)CCCN1N=O C(=O)(C1CCCc2nccn21)NCC(CNC(c1cc(F)c(F)cc1O)=O)OC c1(C(=O)NC2CCN(C(C=NOC)=O)C2)cc(Cl)ccc1F Cc1nc(C(=O)NC(C)CCCNC(=O)C(C)O)c(C)n1C.c1ccc(Cl)cc1 c1(C(=O)NC(C)CCO)ccc(S(=O)(=O)N(C)C)o1.C(=O)(C(C)(C)C#N)N c1(C=O)ncc2[nH]ncc2n1.C(C(C)C(C)C)NC(C1(COC)CC1(F)F)=O N1(C(CC2CN(C(C3C4(CC4)C34CC4)=O)C2)=O)CCCC(C(C)(C)O)C1.CO CC(O)C(F)(F)C(=O)NCCCCN1CCCN(C(c2ccccc2Cl)=O)CC1 N1(C(C=C(C)C(=O)O)=O)CC(C(N2CC3CC(C2)O3)=O)CC(F)(F)C1 c1(C(=O)NCC2OCC(CNC(CCCCSC)=O)C2)cc(=O)cc(Cl)[nH]1 Cc1cn2cc(NCCc3ccccc3)ccc2n1 N1(C(CCC=C)=O)CC(NC(c2nnn(C(C)C)c2C(F)(F)F)=O)CC(C)C1 c12ccnc(n1)-c1cccc(c1)NCCCN2C.C=CCOCCOCCC C(=O)(C1=CCOCC1)NCC(CNC(=O)CC1CC=CC1)O C1(c2occ(C)n2)CCCCN1C(=O)NCC1CCCC(=O)N1 O=C(CCCCn1ccnn1)NC1C=CC(C(=O)NC2CCCCC2)C1 C#Cc1cccc(C(=O)NCC(C)NC(C2CCN(CC)C2)=O)c1 C(=O)(CCC1=CCCCC1)N1CC2C(C(N3CC4C(C(N)=O)(CCC4)C3)=O)(C2)C1 C(=O)(CC(Cc1cccs1)NC(C1CCCCN1C)=O)NC(C)CO C1(CC)(NC(=O)CC2CCCC(C)(C)C2)CCCN(C(c2nnccc2C)=O)C1 C1(C(=O)Nc2cnn(CC)c2C)CCN(C(=O)CCCC2CC2C)C12CC2 C1(NC(c2n(CC)ncn2)=O)CN(C(=O)COC(C)(C)CC)CC1C1CC1 Cc1ncc(C(N2CC3CCC3(CCNC(=O)CCc3nncs3)C2)=O)c(C)n1 C(=O)(CCC(=O)N1CC(O)C1)OC.c1(C=O)cnc(C2CC2)s1.C(C)(=O)N N#Cc1cc(NC(=O)CC2COCCN2C(c2ccnc(Br)c2)=O)ccc1F [SH](=O)(=O)c1ccncc1C.Cc1cc(C)n(Cc2ccccc2OCC2CC2)n1 C(C(C)(C)C(=O)N1CCC(C(F)CNC(=O)C(C)OCC)CC1)OCC c1(C=O)c(C)c[nH]c1CC(N)=O.C(CC(=O)NCC1CC1)N(C)CC.C C1(CNC(c2ccc(OC)s2)=O)(NC(=O)CN2CSCC2=O)CCOCC1 N1(C(C(CC)C(=O)OC)=O)CCN(C(c2ncnc3sccc23)=O)C2CCCC12 C1(O)CC2CCC1C2.C1(N(C)C(C2(NC(=O)CO)CC2)=O)CCOCC1.C C1(CC(=O)N(C(C)CC)C)CCS(=O)(=O)CC1.C(=O)(C(C)Cc1ccco1)N C#CC(CNC(C1(NC(=O)C(C)C(C)C)CCN(C)C1)=O)CC(C)(C)C C1(NC(=O)CCCc2ccccc2)COC2(C1)CN(C(c1ncc[nH]1)=O)C2 c1(C(N(CC(C)N(C)C(c2cc(=O)n(C)cn2)=O)C)=O)cc2ccc(F)cc2[nH]1 C(=O)(C1=COCCO1)NC(CNC(C1(COC)C=CCC1)=O)C1CC1 c1(C=O)ccc(=O)n2c1COCC2.C1(NC(CN(CCC)C)=O)CC2(C1)CC2.N c1(N2CCC(CNCc3nn(CC)c(C)c3)CC2)ncnc2sc(C)nc12 c1(C(=O)NCC2CC(F)CN2c2cc(O)ncn2)nc2ccccn2n1 c1(C(=O)NCC(CNC(C2C(C)C2C)=O)CO)c(N)cc(F)cc1F N1(C(CC=C(C)C)=O)CCCC(C)(C)C1CNC(c1ncn(C(C)C)n1)=O C(CC(C)(C)C)(C(=O)NCC(F)Br)NC(CC1CCN(C)C1=O)=O c1(CC)nc(C)ncc1C(N1CCCOC(CCNC(=O)CCCC(N)=O)C1)=O C1(CCC)CN(C(=O)CCn2nc(C)cc2C)CCN1C(=O)C(CCSC)OC c1(C(C)=O)c(C)[nH]c(C(=O)NCC(CC(C)C)NC(=O)C2=NOC(C)C2)c1C C(=O)(C(O)CC(F)(F)F)NC(C(C)OC)C(=O)NCCc1cc(C)on1 c1(C=O)cc(C(N2CCC(C)C2)=O)[nH]c1C.C1(C=O)C2CNC(=O)C12.CC.O c1(C(C2(C=O)CCC2)=O)ccccc1.C(CN1CCC1)C.C(=O)C=CCF Cn1nc(C2CC2)nc1CC(=O)NCCC1CN(C(C2CC(C)(F)C2)=O)C1 c1(CC(=O)Nc2c(COC)cccc2)c[nH]c2ccc(Cl)cc12 C1(CNC(=O)Cc2cn[nH]c2)CCN(C(=O)CCSc2ccccc2F)CC1 c1(C(N2C(C)(C(=O)Nc3ccno3)CCC2)=O)ccc(C#N)cc1Cl c1(N2CCC(CC=C)(NC(c3ccc4[nH]ccc4n3)=O)C2)ccncc1[N+](=O)[O-] C1(C(=O)NCC(c2cnc[nH]2)C)CC1C1CN(C(=O)Cc2nncn2C)C1 C#CCC(C)(CC)C(=O)NCC1C=CC(NC(=O)CC2(O)CCC2)C1 c1(CC(N2C(CN)C(O)C(O)C2)=O)ccc([N+](=O)[O-])c(N)c1 C(C(=O)NC)(C(C)(C)C)NC(c1c(C)cc(F)s1)=O.c1c[nH]nc1C(C)C N1(C(CC2C(=O)NC(=N)S2)=O)CC2(CCCC2NC(c2cnoc2)=O)C1 C1(C(N2CC(OC)C(NC(c3coc(C)n3)=O)C2)=O)Cc2cc(Br)ccc2O1 C1(CC(C)NC(=O)C(F)C2CCC2)CCN(C(=O)CC2COCC2O)CC1 c1(OC(CC)C)ccc(CNCC2CC2c2cnn(C)c2)cc1 CCCCCCCCOCC(=O)NC1CC1NC(c1cncc(C(=O)OC)c1)=O C(=O)(CCCC(C)=O)N.n1(CC)nc(C)cc1C(=O)NCC1COC(C)C1 N1(C(C)C)CC(NC(=O)C(N)C2(C(F)F)CC2)CCC1=O N1(C(C=C2CCC(C)C2)=O)CCOC2CCN(C(c3cc[nH]c3C3CC3)=O)CC12 S(=O)(=O)(c1ccc(N2CCS(=O)CC2)cc1Cl)N1CCC(C(CC)CC)CC1 Cc1cc(CNC(=O)NCCNc2ccccc2F)nc(-c2ccccc2)n1 C(=O)(C1CC(=O)Nc2ncccc21)N.CC(CNC(=O)COCCF)C1CC1 O=C1NCCC2=C1C(c1ccc(CO)cc1)NC(=O)N2CCc1ccccc1 C1(NC(C#CCNC(=O)OC(C)(C)C)=O)CCc2ccccc2C1 N1(C(CC=CC)=O)CCC2(CC1)CC2NC(C1CCN(CC(F)F)CC1)=O C1(NC(c2n(C)cnc2)=O)C2CC3C1C3C2C(=O)NCC1CCC(=O)O1 c1(CC(=O)NC2(C)CCCN(C(C3CCS(=O)(=O)N3)=O)C2)nnc2n1CCCC2 [nH]1ccc(C(N2CCC(C(C)C)C2)=O)n1.C12(CC=O)CCCC1C2.C(C)OC c1(C(N(CCNC(C(C)C#N)=O)C2CC2)=O)cnc2ccoc2c1 C1(C=O)CC2CCC1CC2.C1(NC(=O)CSCc2ccncc2)CC12CCC2.N c1(NC(C2CC3C2CCN3C(=O)C)=O)ncnc2ccsc12.C1CC(F)(F)C1.O N1(c2cc(OC)ncn2)CC23CCCC2(CN(C(=O)CC2(C)CC2(F)Cl)C3)C1 CC1CCCC1N=c1[nH]c(=NCCc2cccc(C#N)n2)[nH]c2ccsc12 c1(C(=O)NCC=C2CCN(C(C(C=C)(C)O)=O)CC2)cnc2n1CCCC2 c1(C(N2C(C(=O)NCCNC(C)=O)CC3CC32)=O)cnc(O)c(Br)c1 CC#CC1CCN(C(C2CC2C=O)=O)CC1.c1(C(=O)OCC)ccnc(Cl)n1.N c1(CC(=O)NCC(CNC(C(CCC)O)=O)C(F)(F)F)cncc2ccccc12 Cc1cc2cccnc2nc1C(=O)NCC(C)CN(C)C(C1CCCC(=O)O1)=O C12(CNC(C3CCN(C(COCC(C)(C)C)=O)C3)=O)CC(C)(CO1)C2 C1(C(=O)NCc2ccn(C)n2)(CC)CCN(C(c2cc(C)on2)=O)CC1.O Cc1cc(C)c(CC(=O)NCCC2C(C)CCCN2C(c2ccsc2)=O)c(O)n1 c1(C(N2CC(NC(CN(CC)CC)=O)C(C)(C)CC2)=O)cccc2c(C)[nH]nc12 N1(C(CC(C)C2CC2)=O)CC2CCC2(CC(=O)NC2CCC2)C1 C(=O)(CCC(=O)C(C)(C)C)N1CCC(C(=O)NCC(C)CN(C)C)C12CCC2 c1(C(C)OC)nc(C(=O)N)co1.C1(O)CN(C(C2CC2(F)C=O)=O)C1.C C1(OCC)(CN(Cc2ccc(C)cc2)CC2(C)CCCO2)CCCCC1 c1(C(=O)NC2(CO)CN(C(C(CC)=CC)=O)C2)ccc(C(F)(F)F)cn1 C(=O)(CCC(C)(C)C)N1CCC(C(C(C)C)NC(c2c(CC)noc2)=O)CC1 c1(C(=O)NCC2C=CC(NC(CC(C)OC)=O)C2)ccc2n[nH]cc2c1Cl c1(C(C)NC(C(=O)N(C2CCCC2)CCCOC)=O)ccc2c(c1)CC(C)O2 C1(C(=O)NC(C(N2CC(S(C)=O)C2)=O)C2(C)CC2)C2CC3C(C2=O)C13 c1(C(N2CCCC(C(=O)NCCCSC)CC2)=O)cn2c(n1)CCNCC2 C=CC1CCCN(C(C2CCCN(c3ncc(CC)cn3)CC2)=O)C1 C1(C(N2CC(NC(C3C(C)(C)CC3)=O)C2)=O)CCC2(CC1)CC2 Cc1cc(C(=O)NCC2CN(C(=O)C(F)(F)CF)C2)n(-c2ccccc2)n1 c1(C(=O)OC)ccc(N2CCCC(C3CCCN3)C2)c(C(F)(F)F)c1 N1(C(c2c(C)nc(CC)s2)=O)CC(NC(c2cnn(C)c2N)=O)CC1(C)CC c1(NC)ccc(C(=O)N)cc1[N+](=O)[O-].C1(C)CCN(C(=O)Cn2ncnn2)C1.C c1(C(=O)NCCC(C)(C)NC(=O)COCC)cn2c(n1)COCC2.CCO Cc1c(C(=O)NCC(O)CN(C)C(c2nocc2Br)=O)ccn1C CC1CC(C(=O)NCCCCCNC(=O)C=Cc2ncco2)CCS1(=O)=O C1(CNC(CCNC(=O)OC)=O)CC2CCC1N2C(=O)C(CO)N(C)C N1(C(C(CC)N(C)C)=O)CC=C(CCNC(c2cc3scnc3[nH]2)=O)CC1 CCCCCCC(F)C(=O)N1CCC(N(C(=O)Cc2ncccc2F)CCO)C1 C1CC(C)(C)CN1C(c1cccc(Cl)c1)=O.c1(C(C)O)ccc(C(=O)NC)cc1 c1(Nc2ncnc(NCC(CN(C)C)OCC)c2C)[nH]c2cc(C)ccc2c1C c1(C(=O)NC2C(CNC(C(CC)(C)O)=O)COC2)cc(F)c(Br)cc1C C1(CC)C(NC(=O)Cc2cnc(C)[nH]2)CCCN1C(c1cc(C)nc(C)n1)=O C(=O)(CC(C)C(=O)N1CCC(C(=O)NCC(n2ccnn2)C)(C(C)C)C1)OC c1(C(=O)NC(C2CN(C(=O)CN3CC4CC4C3)C2)C)ccoc1C1CC1 c1(C(=O)NCCC2(C)CCN(C(C(CC)=CC)=O)C2)c(C)cc(C)nc1O C12(C(=O)NCC3(O)CCN(C(=O)CN4CCCC4=O)C3)CC=CCN1CCC2 C1(CNC(C=CC(C)(C)SC)=O)CN(C(C2(CCO)CC2)=O)CCO1 Cc1cc2ccc(C(N3CCCCC(c4ccccc4)C3)=O)cc2s1 NS(=O)(=O)CC(=O)NCC1CCN(C(=O)CC2CSC2)C1c1ccccc1 C1(NC(=O)CCC2CCOC2)CCC2CCN(C(c3cc(C(F)(F)F)no3)=O)C12 N1(C(CCC(=O)NC)=O)CCCC(NC(=O)C(=O)Nc2ccccc2)C1C c1(C(N2CC(CC=C)(NC(C3COC(C)C3)=O)C2)=O)cn(C)c(C)n1 C(=O)(C(F)C(=O)NCC1CCCN1C(c1ccc(NC=O)cc1)=O)OCC C1(NC(C(c2cccc(Br)c2)CC)=O)CCN(C(=O)C(C)(C)O)CC1 c1(OC)ncnc(NC2CCN(c3ncccn3)CC2)c1OC C(=O)(C1CC(=O)c2ccccc21)N1CC(NC(CC(C(C)C)(F)F)=O)C(F)CC1 Cc1cc(CC2CCCC2NCC2CCOC2C)n(C)n1 Cc1nc2ccc(C(N3CCOCC3CNC(=O)C3=NOC(C)C3)=O)cc2[nH]1 c1(CN(C(C(N2C3CC(N)C2CC3)=O)=O)C2CCCC2)ccc2c(c1)OCCO2 Cc1ccc(O)c(C(N2CCOC(CC(=O)NCCN(C)C3CC3)C2)=O)c1 Cc1cc(NC(C23CC2CCN3C(C2CCC3(CC3)C2)=O)=O)cc(O)c1 c12cc(cc(F)c1)CC(=O)O2.c1(CC)ccc(C(C)OC)o1 N1(C(=O)Nc2c(C(C)C)ncnc2)CCC(F)(F)C2(CCOC2)C1 C1(F)(CNC(C(CC)(C)OC)=O)CC2CCC(C1)N2C(c1ccc(C)s1)=O CCCCC(C)CCC(=O)NCC1CN(C(c2cc(C(N)=O)[nH]n2)=O)CC1(F)F C=C(C)CC(C(=O)NC(CC1CC1)CO)NC(C1C=CC=CC=C1)=O C1(C(CNC(=O)Nc2cncnc2)F)CCOCC1 c1(C(CC)NC(=O)C(=O)NC2CCC(C)(CN)CC2)cn(C)c2ccccc12 c1(C(=O)NC2CCC(NC(C(C)n3cnnn3)=O)C2)cccc(=S)n1O C1(C(=O)NC(CC(=O)NC)C)CCOCCN1C(c1ncn(C)c1C)=O C1(CCNC(=O)C(Cl)=CCl)CCN(C(=O)CC2(O)CCCOC2)CC1 Cc1cn2ccc(C(=O)NC3CC(O)CN(C(C4(CCO)CC4)=O)C3)cc2n1 c1(OC)ccc(F)cc1C(=O)C(=O)NCC(C)(CC(C)C)NC(=O)CCC.O Cc1cc2c(cc1C)C(C(=O)N(C)C(c1c(F)cccc1F)C)CO2 C=CCCCC(=O)NC(C)C(=O)NCCc1ccnc(O)c1 CC1=C(C(=O)NC2(CCNC(c3nn(C)cc3N)=O)CCCC2)SCCO1 c1(NC)ccc(C(=O)N(C(C)C(N2CCC(CO)CC2)=O)C2CC2)nc1 c1(OC)ncc(C(=O)NCCC(C)(C)C)cc1C.C(=O)(C(C)CC1CCCO1)N C1(C)(n2cc(-c3cnc(CC)o3)nn2)CCN(C(c2csnc2C)=O)C1 N1(C(C(CC)OC)=O)CC(NC(=O)CC2(c3ccccc3)CC2)C(C)(C)C1 c1cnc(F)c(C)c1.n1(CC(=O)NCCN(C(=O)C)CC)ccnn1.C c1(NC(CNC(C(C(C)(C)O)(F)F)=O)C2CC2)nc2cc(Br)cnc2s1 C1(C)(C(=O)NCC2CC(OC)C2)CCCN(C(=O)Cc2cccn2C)C1 c1(Cn2cc(C3N(CC(c4c(F)cccc4F)O)CCC3)nn2)cc(F)cnc1Br C1(C(=O)NC(c2nccn2C)CC)COCCN(C(c2ccnc(C)n2)=O)C1 c1(C(N2CC(CCOC)N(C(C3CCCO3)=O)CC2)=O)ccc2ncsc2c1 C(N=c1nc2sccc2c(N2CCCC(CSC)C2)[nH]1)c1c(OC)nn(C)c1 Cn1ncc(C#N)c1C(=O)NCC1CCCN1C(C1(S(C)(=O)=O)CC1)=O C1(NC(C(C)NC(=O)C2CC2)=O)C2CC(NC(C3CCC=CCC3)=O)CC12 c1(CNC(C(C(C)C)SC)=O)ccc2c(c1)CN(C(c1cc(O)ncn1)=O)C2 C12(NC(C3CCCCO3)=O)CCC(C1)N(C(=O)C(=O)Nc1ccccc1)C2 Cc1ccc(F)c(O)c1C(=O)NC1CCCC1C.c1(C=O)cc(C(C)C)on1 c1(NC(=O)CC2CN(Cc3ccn(-c4ccccc4)n3)C2)ncc(F)cc1Br c1(OC)cc(C(N2CCC(C)(C(=O)NC)C2)=O)cc(C#N)c1.c1csc(C)n1 c1(CN2CC3CN(C(c4cnc(Br)s4)=O)CC32)ccc([N+](=O)[O-])cc1O N1(C(C=C(C)C)=O)CC(NC(c2ccco2)=O)C2(CCS(=O)(=O)CC2)C1 C12(CNC(CCC(=C)C)=O)CC(NC(c3cccn3CCC)=O)(C1)C(C)O2 CCC(CCC(=O)N1CCC(CSC)C1)NC(=O)C=CC(C)C c1(CC)nc(O)c(C(=O)N(C)CC2(O)CCCN(C(C3CCC3)=O)C2)cc1C c1(NC)cncc(C(N2CCC(C(C)NC(=O)CC3SC(=N)NC3=O)C2)=O)c1 n1(C(CC)C(=O)NC2CCCC2O)cc(I)c(C)n1 Cc1nccc(C(=O)NCC2(CC)CC2)c1N.c1(CC=O)c(C)cccc1C.N c1(C(N2CC(NC(C34CCC(F)(CC3)C4)=O)C3CC23)=O)ccc2nnnn2c1 C(=O)(C(F)CC(C)(C)NC(c1cccc(C)c1N)=O)NCC=CCSC C(CCCC(CO)OC(c1ccc(CO)cc1)=O)NC(CC(CC)C1CCC1)=O C1(NC(C(CC)N2CCCC2=O)=O)CC1C1CCCN(C(c2[nH]cnc2C)=O)C1 CC1CCCC1(C(=O)NCCc1cccc(F)c1)NC(c1cc[nH]c1)=O O=C(C(C1=CCCSC1)N1CC(CO)CC12CCC2)NCCC1CC1 c1(CCC(N2CCC(CNC(CC(=C)C)=O)CC2)=O)cc(Br)ccc1C N1(C(Cn2nnc(C)n2)=O)CCC2(NC(C3CCOC(C(C)C)C3)=O)CCCC12 CCC(C(=O)NC1(CNC(c2ccn(C)c2)=O)CCC1)c1cccnc1 Cc1cc(=NC(=O)NC(c2ccc(CN3CCOCC3)o2)=O)[nH]n1C(C)C1CC1 N1(C(c2ccc(CC)o2)=O)CC=CCC1C(=O)NC1COCC1O c1(C(=O)NCCCNC(c2ccc(C)s2)=O)cc(Cl)ccc1Cl C(=O)(C(CN(C)C)C(C)C)N(CC(=O)N(CC)Cc1cccs1)CC C1(C=O)CC2(CSC2)C1.c1(C(=O)NCC2CCC2)nocc1-c1ccccc1 CC(C)CC(CNC(=O)CC1CNC(=O)O1)NC(=O)C(C)(C)F N1(C(c2sc(CCC)c(CC)c2)=O)CCC2CN(C(=O)C3=CCCSC3)CC12 C(=O)(CC1CC(=O)Nc2ccccc21)NC(CNC(C1=C(C)CCC1)=O)C n1(CC(=O)N)nc2ccccn2c1=O.C(C)(CC)(CC)NC(COCCC#C)=O C(=O)(CCN(OC)C(=O)C1CC(=O)NC(=O)C1)N(CC(=O)O)C1CC1.CC [N-]=[N+]=Nc1ccc(COC(C2CCC(O)CN2C(=O)Oc2ccccc2)=O)nc1 CCC(CC(C)C)C(=O)NC(CC(=O)N(CCCC(C)(F)F)C)C(C)C C(=O)(CC(C)P(C)(C)=O)N(CCNC(C(CCCC)C)=O)C C(=O)(C1=COCCC1)N1CCC(C(=O)NC2CCN(C(C)C)CC2)C1C C(=O)(Nn1cnnc1)C1(CO)CCN(C(C(=Cc2cn[nH]c2)C)=O)C1 c1cc(Cl)c2c(c1)OCO2.CC=O.C(C)(C)C.C(COCCOCC)OC N1(C(C(CC)=CC)=O)CCC(OCCCNC(c2ccnnc2OC)=O)CC1 C1(NC(CN(C(C(C)C)=O)C)=O)CC2CCC(C1)N2C(c1cn(C)nc1O)=O c1(C(=O)NC(C(C)NC(C(C)=C2CCC2)=O)C)cccn2cc(C)nc12 c1(C(=O)NC2CC(NC(C3(OC)CCC(C)(C)C3)=O)C2)cncc2c[nH]nc12 C(=O)(C1COc2ccc(Cl)cc21)NCCCCCNC(c1cnc2n1CCS2)=O N1(C(c2ccc(C)c(C)c2)=O)CC(O)(C2(CNC(=O)Cc3csnc3C)CC2)C1 c1(OC)ccccc1OC(C)C(N1CC=CCC1)=O.C(c1cnc[nH]1)=CC=O.N c1(C(=O)NC(C)CCCNC(C2CCCC3CC23)=O)cnc2c(cnn2C)c1 c1(C(=O)NCC(C2CC2)NC(CCCNC(C)=O)=O)ccc(Br)cc1F C(=O)(C(C)(C)CC(=O)N(C1CN(C(c2csc(S)n2)=O)CC1(C)C)C)OCC c1(C(C)C)nc(C(=O)N(C2(CC(=O)N(C)Cc3cscn3)CC2)C)co1 CCCC(C(=O)OC)C(=O)N1CCN(C(=O)CNC(N2CCCC2)=O)CCC1C C(=O)(C1=NNC(=O)C1)NC(C)CC(C)NC(=O)Cc1ccc(OC(F)F)cc1 c1(C(=O)NCCCNC(CCC(=O)NC)=O)cnc2cc(OC)ccn12 Cc1cc(Br)ccc1S(=O)(=O)NC1CCC(NCc2ccc(C#N)cn2)C1 C1(C(=O)Nc2c(SC)cccn2)CN(C(C2CCCC2C)=O)CCC1(F)F C#Cc1ccc(C2(C(=O)OC(C#C)CCC)CC2)cc1 CC1=C(C(=O)NC2(C)CCCN(C(=O)C(C)n3ccnc3)C2)CCO1 C#Cc1ccc(C(N2CC(CC(C)NC(=O)C=Cc3nc(C)cs3)C2)=O)nc1 C(=O)(CS(=O)CCC(F)(F)F)N1CC(CCNC(C(c2ccccc2)OC)=O)C1 S(=O)(=O)(c1cc(Br)c(F)cc1F)NC1C2CN(C(c3ncc(C)s3)=O)C(C2)C1 C(=O)(CCCC(F)(F)F)N1C(CNC(c2nncs2)=O)CC(COC)C1 Cc1[nH]nc2ccc(C(=O)NCC3CCN(C(=O)CC=C(Cl)Cl)C3)c(Cl)c12 c1ccc(C#N)cc1.Cc1nccn1C(C)C(=O)NCC(O)CNC(=O)CC.S C(=O)(C(C)C(O)C(C)CC)NCC(C(=O)NC(CC#C)C)C(C)(C)C C(=O)(C1CCCn2cnnc21)N1C(C)CN(C(C2(CC3CC3)CC2)=O)CCC1 C1(NC(C2C(=C)CC2)=O)CCN(C(c2cc(F)n[nH]2)=O)CC1(C)C C12(C(=O)NCC(CC)C(C)(F)F)CCC(CC1)N(C(=O)CN1CSCC1=O)C2 C1(NC(CC(=O)NC)=O)CCC2CC1CN2C(=O)CC(c1cccc(OC)c1)C Cc1cncc(C)c1C(N1CC(C(F)(F)F)C(C)C1)=O.c1(C(=O)N)cscc1F N1(C(c2ccn(C)c2)C(=O)NC(C)C)CCC(C)C(C)C1 N1(C(C2(CCNC(C3(CCC=C)CC3)=O)CC2)=O)CC(C)C(C)(C)C1 Cc1ccc(C(N2CCOCC2C(N2CCN(C(=O)C3CC3)CC2)=O)=O)nc1 Cc1c(C(=O)NCC2(NC(=O)C=CS(C)=O)CC2)sc2cncn12 c1(C(N2CC(NC(c3c(CC)csc3)=O)C2)=O)sc2ncccc2c1N Cc1c(F)ccc(C(=O)N)c1N.C12(CC(N3CCCC3)=O)CCC(C)(C1)OC2.C C(=O)(C(CCC(C)(C)C)N1CCC(C)(CN(C)C)C1)NCCCOCC C1(C)(C(N2CCCC2)=O)CC(C(C)(C)C)=NO1.C1(C)(C(C)C)CC(C=O)C1.N CCC(C)C(C(=O)NCC(F)CN)c1ccccc1 c1(C(=O)NCC(CN(C(c2c(C)snc2)=O)C)C)cncc2nc[nH]c12 C(=O)CN=S(C)(C)=O.N1(C(C2CCN(C(=O)O)C2)=O)CC=CCC1.CC(C)C CCCCCC(CC)C(=O)N(C)CCN(C(C1CCOC2(CCC2)C1)=O)C(C)C C(=O)(C1CCc2c(Cl)cccc21)NCC1(O)CN(C(C2CC(C#C)(O)C2)=O)C1 c1(CNC(=O)Nc2ccc(OCF)cc2OC(F)F)c(Cl)ccnc1Cl CCCCC(CNC(=O)C(=CC1CCCCC1)F)NC(=O)CCc1cnoc1 CC(C)C(F)C(=O)N1CC(CCCCNC(C2CCCC2(C)C)=O)C1 C1(NC(c2cc(CC)n(C)n2)=O)CN(Cc2ccc(O)c(C)c2)CC(F)(F)C1 C(=O)(C(CC(C)C)C(C)C)NC(CC(C)NC(CN(CCC#C)C)=O)C c1(CCC(=O)NC2(C)CN(C(C3(O)CC3)=O)C2)ccc(F)nc1 c1(C(N2CC(COC)N(C(c3cn(C)nc3Cl)=O)CC2)=O)cc(C)c(F)cc1N CCS(=O)CC(=O)N1CCCC(N(C)C(c2cccc(F)c2)=O)C1 Cc1ccc2c(C=CC(=O)NC3CN(C(c4csc(Cl)n4)=O)CC3F)c[nH]c2c1 C1(NC(c2c(OC)noc2C)=O)CC(C(=O)N2CCC(C(F)(F)F)C2)=CC1O c1(SCC)ccc(CC(N2CC3C(NC(C4CCCC(=O)O4)=O)C3C2)=O)cc1 c1(C(=O)NCCCCNC(=O)C=CC2CCOC2)ccnc(OC2CCC2)c1 CCN(CCc1cccc(F)c1)N1CCC(N(CC(C)O)C)CC1 c1(CCC)ccc(CC(N2CC3C(NC(C4CCC5(C4)N=N5)=O)C3C2)=O)cc1 Cc1cc(C(=O)NC2CC(NC(C3CC3(Cl)Cl)=O)C2)c(C)cc1Cl N1(C(CC(CC)(C)C)=O)CCCC(C2CC2NC(=O)C(O)COC)C1 c1(-c2cn(C(C)CNC(C(C(F)(F)F)C3CC3)=O)nn2)cccc2cnccc12 Cc1cc(C(=O)N(CC(C)N(C)C(c2n[nH]c3c2CCC3)=O)C)cc(Cl)c1 c1(CC)cc(C(=O)N(C2CCCC(NC(=O)CC3CC(=O)C3)C2)C)n(C)n1 CC(CNC(C1CCCS1)=O)(C1CC1)NC(=O)CCNS(C)(=O)=O c1(NC(=O)NCC(c2ccc(F)cn2)(C)C)nccnc1-c1ccccc1 Cc1c(-c2cn(Cc3ccccc3NC(=O)CN)nn2)cnn1C.[SH](C)(=O)=O CC1CN2CCN1CC2C(=O)NCC1CN(C(=O)CCc2nncs2)CCCO1 CC(C)CC(O)C(C)C(=O)NC1CCN(C(=O)C(C)NC(C2CCC2)=O)CC1 c1(C(N2CCN(CC(C)NC(C(CCOC)C)=O)CC2)=O)cc2ccccc2s1 C1(N(C(CC)=O)C(C)C)CCCN(C(=O)CC)CC1.CC(C)(C)C.CC(=O)O C1(C(=O)NCCCCCNC(c2c(CC)noc2C)=O)CC2(CCC2)CCO1 n1(CCC)ccc(C(=O)NC2(CCC)CC2)n1.C1(C(C=O)C)CCC(=O)N1.N c1(C(N2CCCC(C)(CC)C2)=O)ccc2nc(O)n(C)c2c1.C(=O)(C=O)N.N C1(NC(C(=Cc2ccncc2)C)=O)CCCC12CN(C(c1snnc1C)=O)C2 c1(CC)ncc(C(=O)N(C)CC=CC(=O)NCc2cncn2CC)s1 N1(S(=O)(=O)CCOC2CCCCC2)CCCN(C2CC2)CC1 c1(C(=O)NCC2CCCCC2NC(c2scnc2Cl)=O)ccc(Cl)cc1O Cc1cc2sc(C(=O)NCC(O)CC)cc2s1.c1(C(=O)N)c(C)noc1C1CC1 CCCC(C)(CC)C(=O)N1CCC(OCCNC(c2nscc2C)=O)C1 c1(C(N(C)CC2CCN(C(CCC=C(C)C)=O)C2)=O)cccc2ccc(C)nc12 C1(C(=O)NCC2CCN(C(C=C(CC)C)=O)C2)(CF)CCC(F)(F)CC1 C#CC1(C(N2CCOC(CCOC)C2)=O)CCN(C(=O)C(CC=C)OC)C1 C12CCC(CC1n1ccnc1)C2.C(C)(C(=O)N(C1CCCC1)C(C)C)OC CCCCC(CNC(=O)CCCC#N)NC(C1(C(F)(F)F)CC1)=O c1(C(N2CCC(CNC(C34CC(C#N)(C3)C4)=O)CC2)=O)cc(F)c(F)cc1Cl C1(N(C(=O)C(Cc2ccccn2)NC=O)C(C)C)CC2CC1CN2.C(C)(C)C c1(OC)ccc(C#N)cc1CNC1CC1C(=O)N.c1cc(F)c(I)c(F)c1 N1(C(CC(CC)C)=O)CC(CNC(c2ncc(OC)cc2F)=O)C2(CCC2)C1 c1(C(=O)NCCC)cnc2c(c1)OCC(=O)N2.C(=O)C(C1CCC1)C1CCC1 c1(CC(N2CCC(CCOC)(NC(=O)C(F)O)C2)=O)c(C)nc2ccccn12 Cc1nc(C(C)NC(c2ccnc(-n3ccnc3)c2)=O)c(C)o1 N1(C(CCn2c(C)nc(C)n2)=O)CCC2(CCCN2C(C2COC(=O)N2)=O)CC1 C1(N(C(CC2CCC(=O)O2)=O)CC)CCCN(C(=O)COc2ccc(F)cn2)C1 N1(C(C2CCN(C)CC2)=O)CC2CCCC1(CNC(c1cc(=O)n(C)o1)=O)C2 c1(C(C)NC(C2CCC(NC(c3c(C)n[nH]c3)=O)C2)=O)cnc2c(C)cccn12 C(C1=CN(C(=O)OC)CCC1)(c1n(CCCOC)nnn1)NCC(C)SC Cc1ccc(C(C)NC(c2ccc(CNC(c3cnsn3)=O)cc2)=O)cn1 n1(-c2nc(C)cc(C)n2)ccc(=NC(=O)CC(C)(C)C(=O)OC(C)(C)C)[nH]1 c1(CC(=O)N(C2CCCN(C(=O)C(F)C(C)(F)F)C2)C)cccc2occc12 C1CN(C(c2cc[nH]c(=N)c2Cl)=O)C(C)(C)C1.C1(CC)CCC(C(=O)NC)O1 N1(C(C(C)Cc2cccnc2)=O)CCN(C(=O)CC2CCOC2(C)C)CCC1C c1(CN(C(CN(C(c2ccccc2)COC)C)=O)C2CCC2)nc(SC)nn1C C1(CN(C(COCCC#C)=O)C)CCC(NC(c2[nH]c(O)nc2C)=O)CC1 C1(NC(=O)NC(C)C(=O)N)CCc2nnn(C)c2C1.c1cc(C(F)F)cc(F)c1 N1(C(CC(=C=C)C)=O)CC(O)CCC1C(=O)NCC(C)(C)O Cc1noc2ncc(C(=O)NC3CCC(N(C)C(c4csc(Cl)n4)=O)C3)cc12 c1(NC(=O)CC2CCC3CC23)ccc(Nc2ccc(C(=O)N(C)C)cc2)cc1 C(=O)(C(CC(F)F)C1CCC1)NCC(CC)NC(C1CCN(OC)CC1)=O C(c1ccc(C2CC2C)o1)=CC(N1CCC1)=O.C(CCC(=O)N)OCC=C.C c1(CC)ccc([N+](=O)[O-])cc1C(=O)NCC.c1(C(=O)N)cc(C)c(F)cc1Cl C1(CNC(CSCCC)=O)CN(C(C2CC2C2CCOCC2)=O)CCC1(C)C S(=O)(=O)(c1ccc(N2CCn3cccc3C2)nc1)NC1CC(C)S(=O)(=O)CC1 C1(NC(C(C)C23CC(C2)C3)=O)COCCC1(F)F c1(C(N2C(CC(=O)NC(c3cccnc3)CC)C=CC2)=O)ccn(CC)c1C c1(NC(C2CCCCN2C(=O)C(C2(O)CCCC2)F)=O)cccc([N+](=O)[O-])c1 c1(C(C(=O)NC2C(CNC(Cc3cnc(C)[nH]3)=O)CC2)O)ccc(Cl)cc1 CCC(CC)(CO)C(=O)N1CCC(C)(NC(C2OCCN(C)C2=O)=O)C1 C(=O)(CC(F)(F)CC)NCC(C1N(C(C(C=C)OC)=O)CCC1)(C)C N1(C(CC2(OC)CCC2)=O)CCC(NC(=O)C=Cc2cccs2)C(CO)C1 N1(C(CC2CCN(C)C2)=O)CCC2(C(=O)Nc3cc(F)cc(F)c3)CC2C1 C#CCC(C(=O)N(C)C(C1CCCC1)C)NC(=O)C(COC)OC CCCCCC(O)CC(=O)NC1CC2C(NC(=O)C(c3c(C)n[nH]c3C)C)C2C1 C1(NC(CCCC)=O)CN(C(c2sc(F)cc2Cl)=O)C2(CCC2)C1 N1(C(C(CC(=O)OC)(C)C)=O)CC2(CCCN(C(C3CCC3)=O)C2)C1.C(C)=O c1(C(N2CCC(n3cc(CCO)nn3)C(O)C2)=O)cc(=O)nc2sccn12 CCCC(C)(O)CC(=O)N1CCC(CCNC(C2(F)CCCOC2)=O)CC1 Cc1cc(C(N2CCC(O)(CNC(=O)Cc3sc(C)cc3C)C2)=O)cc(C)c1 C1(C(=O)NCc2c(C)n(C)nc2)CCC2CCC1N2C(=O)Cc1cncnc1O C(=O)(CC(F)(F)C(C)C)NC(CC)(CNC(C12CCCCC1C2)=O)CC C1(OC(N(C)C)=O)CCN(C(=NCCCCl)NCC2CCC(F)(F)CO2)C1 C(=O)(CC(C(C)OC)NC(C1(CCOC)CC1)=O)NC(CC=C)C c1(C(=O)NC2CCCN(C(c3c(Cl)cn(CC)n3)=O)C2)cnn2c(=O)cc[nH]c12 N1(C(c2ccc(C)cc2)=O)CC2CC(NC(=O)CN3CC(=O)N(C)C3=O)CC2C1 C1(NC(c2ccc(C)cn2)=O)CN(C(C2CC2CC(C)C)=O)CC2(CCC2)C1 Cc1ccc2c(c1)CCN(C(C1CCNC1=O)=O)C2CN N(C(=NCC1CCC2(COC2)O1)N1CCN(S(C)(=O)=O)CC1)C(COC)C c1(C(N2CC(O)(C(C)NC(C(CCC#C)O)=O)C2)=O)cnc(O)c2cnccc12 c1(CCC)ccc(C(=O)NC2CCCC2NC(c2nnccc2C)=O)cc1N c1(N(CCOCCNC(C(C)Sc2ccc(F)cc2)=O)C)n[nH]c2c1CCSC2 n1(CC)ccnc1C(=O)N(C)CCN(C(=O)CO)C(C)C.C1CCOCC1 c1(-n2cc(CC)nn2)cc(F)cc(Br)c1.C1(C(=O)OCC)CCCC(C=O)C1.N C(=O)(C(C)(C)C(=O)N1CC(NC(=O)Cc2coc(C)n2)C(SC)C1)OC Cc1nncn1NC(=O)C(C1CCC1)NC(C1CC2CCC1O2)=O c1(N(Cc2cnn(-c3ccc(F)cc3)n2)CC)c(C)ccc(Br)c1C.N1CCn2ccnc2C1 CCC(CC(=O)N(C(C)CO)C)NC(=O)CC=CC(C)(C)C Cc1ccc(C(=O)NC(C)CNC(=O)CC2CNC(=O)O2)c(N)c1F C1(C(=O)NC(CC(C)C)CCO)CN(C(=O)CCc2cncs2)C2(CCC2)C1 Cc1ccc(C)c(C(=O)O)n1.C12CCCC(O1)C2=O.c1(NC(=O)O)ccccc1 C1(NC(CC(CN(C)C)O)=O)CCN(C(c2cc3c([nH]2)CCC3)=O)CC1F C1(NC(C2=C(C)OCC2)=O)CCCC12CCN(C(c1csc(CC(C)C)n1)=O)C2 C1(C(N2CCC(CC)(CO)CC2)=O)CCN(C(=O)C(C)(O)CC(C)C)CC1(C)C CC(CN=c1[nH]c(Cl)ncc1Cl)N(C(=O)CC1CSC1)C N1(C(CCC)C(N)=O)CCCC(COC(=O)C(F)(F)F)CC1 c1(C(N2CCN(C(c3c(C)noc3)=O)C(C3CC3)C2)=O)cn2ccccc2n1 N1(C(CC2CC(CC)C2)=O)CCC(NC(=O)C#CC2(C)CC2)C2(CCC2)C1 c1(C(C#N)OCC(C)OC(c2ccc(CC)o2)=O)ccc(Br)cc1 C(C)(c1ccccc1)=CC=O.c1(COC)nc(CC(=O)NC2CCCC2)cs1 N1(CC)CC(C(=O)N(C(C)(C(=O)NC(CC)C(N)=O)C2CC2)C)CC1=O N1(C(C)C(=O)NC2CC(F)(CNC(c3scnc3Cl)=O)C2)CCCCC1=O c1(-c2ccc(OCCCC)c(CC)c2)ccc(OC)c(S(N)(=O)=O)c1 C(N=C(NCC1CCCCC1)N1CCC(c2ccccc2)C1)C1CCN(C)C1=O N1(C(c2cc(O)no2)=O)CCN(C(=O)CC2CCC3CC3C2)C2(CCC2)C1 C(Cc1cn(Cc2nnc(C3CC3)o2)nn1)(C(=O)O)NC(c1scnc1Br)=O C1CN(C(=O)CC(C)(C)N(C)C)CC1C(F)(F)F.C(C(=O)N)N(C)CC.C c1(N(C2(C(=O)NCC(Cc3ccsc3)CO)CC2)CCO)ccc(Cl)cc1 c1(CNC(CC)Cc2ccc(I)cc2)c(C(=O)O)ccnc1O N1(C(C2(F)CCN(C(C3CCC(CC)O3)=O)C2)=O)CCC2CCCC2C1 C12(CNC(c3c(Cl)ccc(CC)c3)=O)CCCC1CN(C(c1cnco1)=O)C2 c1(CC=O)ccc(F)c(Cl)c1.C1(C)CCCC1.C1(OC)CC(CC(=O)N)C1.C N1(C(C(CC=C)C)=O)CCC2(COC(CNC(=O)CO)C2)C1.c1cc(C)on1 C#Cc1ccc(C(N2CC(C(N)=O)(C)C2)=O)o1.c1(C=O)ccnn1CC(C)C c1(C(C)=O)cnc(F)c(NC2C3CCN(C(=O)OC(C)(C)C)CC23)c1 C(C)C1=CCN(C)CC1.c1(C(C)=O)ccc(C(=O)NCC2(C=O)CC2)o1.N n1(CC)cc(C(=O)NC2(CF)CCN(C(c3ccccc3O)=O)C2)c(C(C)C)n1 Cc1cc(F)ccc1C(=O)NCC1C=CCN1C(C1(C)CCN(C)C1=O)=O CC1CC(C(=O)NCC2CN(C(=O)CN3CCC(=O)NC3=O)CC2(F)F)=NO1 c1(C(N2CCC(COC)CC2)C(=O)NC2CC2)ccc(OC)c(OC)c1 Cc1cccc2c1CCOC2C(=O)NC1CCCCC1NC(=O)CN1CC=CC1 C1(C(=O)NCC(CC)NC(C2(C)CCNC2=O)=O)CC=C(C)CC1 C1(C2CC2)(CNC(c2c(C)nc(C)s2)=O)CCN(C(c2cnco2)=O)C1 c1(C(=O)NCC(CCCC)NC(c2ccc(NC)cn2)=O)coc2ccccc12 N1(C(C(C(C)C)O)=O)CCC(C)(C)C(C(=O)N(C)C(C)C)C1 CC1(C)CC(NC(C2CCCN(C(c3ccc4c(c3)CC4)=O)C2)=O)C(C)(C)O1 C1(CC(C)NC(CN(C)CC)=O)CCN(C(=O)CCC2CCN(C)C2)CC1 c1(N(C)CC)cc(C(=O)NCC2(C(=O)N)CC2)ccn1.c1ccncc1.C N1(C(C(CC)C(C)C)=O)CC2CN(C(c3nccc(Cl)c3O)=O)CC2C1 CCC(C=O)C(=O)NCc1cn(CC(C)NC(=O)CSCCOC)nn1 CC(C)(Cc1cnn[nH]1)C(=O)N.C(C)C(C)(C)C.c1(C2(C=O)CC2)ncco1 CCCC(C(C)(C)C)NC(=O)CSCCNC(=O)C(C)n1ccnn1 C1(F)(CNC(=O)CCN2CCC(F)C2)CCCC1.c1(C=O)cn(CCO)nn1.N C(CC(C(=O)Nc1cncc(C)c1)NC(c1cncn1C)=O)OCC c1(C(N2CCC(N(C(CCCC=C)=O)CC)C2)=O)c(C#N)cnn1C C1(C(=O)NCC(C(C)C)(C)NC(=O)CCCn2ccnn2)CCC=CCCC1 CCN=c1[nH]c(C)c(C(N2CC3CC(NC(C4(C)CCCCO4)=O)C2C3)=O)s1 N1(C(CCCCC)=O)CC2COCCC2(NC(=O)Cc2c(C)nn(C)c2Cl)C1 C(=O)(C1=CC2(CCOC2)C1)N1CCC(C)(CC(N2CC3(CCC(=O)N3)C2)=O)C1 c1(CC)cccc2c[nH]nc12.Cc1cc(C(C2CC2)NC(=O)C(=O)N)cc(F)c1 c1(C(=O)NC2CN(C(c3cn(CCC)nn3)=O)C(C)C2)ccc(OC)nc1C c1(C(=O)OC(C)(C)C)cnc(N2CC3(CCC3)C2C2CCOCC2)c(Cl)c1 C1(NC(c2cn(C)nn2)=O)CCN(C(=O)C(C)(F)c2ccon2)CC1CO c1(C(=O)NC(CNC(C(C=C)OC)=O)(C)C(C)C)ccc(C)c(C)n1 N1(C(C(=O)NCC)=O)CCCC(C)C1CNC(c1cc(C)cc(Br)c1)=O C1(C(N2CC(c3cn(Cc4ncccn4)nn3)C(O)C2)=O)CC(O)C12CCC2 CCCC(C(=O)OC)C(=O)N1CCC(N(C)C(c2cc(Br)ccc2F)=O)C1 C1(NC(C(Cn2ccc(C)n2)C)=O)(CNC(=O)Cc2csnn2)CCCCC1C CC(C)C(CC(=O)NCC1CCN(C(=O)Cc2ccco2)CC1C)C(C)C CC1(CNC2CCN(CCC(F)(F)F)CC2)CNC(=O)O1 N1(C(c2cnc(O)n(C)c2=O)=O)CC2CC(NC(=O)CCC3CC3)CC(C2)C1 C(C)(CC(=O)NCCNC(=O)C(O)(c1ncnn1C)c1ncnn1C)SC N1(C(C(C2CC(NC(c3c(C)csc3)=O)C2)F)=O)CC([N+](=O)[O-])C1 N1(c2cccc(CN3CCC(F)(C(=O)NC)C3)c2)CCC(=O)NC1=O c1(OC)ccc(C=CC(=O)NC(C)CCC)nc1.C1(C(=O)N)CCNC(=O)C1 C(=O)(C(C)(C)S(C)(=O)=O)N1CC=CC(NC(CCC2N(C)CCCC2)=O)C1 c1(OC2C(CC)N(C(=O)OC(C)(C)C)CC2)cnc(F)c(C)c1 N1(C(COCCC)=O)CCCN(CCCCNC(=O)CC2CCC(F)(F)C2)CC1 CN1CCN(C(=O)C(N2CCC(F)(c3ccc(F)cc3)C2)=O)CCC1=O C1(C#CC(=O)N2CCCCC(NC(c3cnc(OC)nc3)=O)C2)(CC)CC1 Cc1cc(O)cc(C)c1CC(N1CC2(CCCC2NC(=O)CP(C)(C)=O)C1)=O NC(CC(F)F)C(=O)NCc1ccccc1CC(F)(F)F C(=O)(CC(C)(C)CCOC)NCC(=O)NCC(=O)N(C(CC)CC)C N1(C(C2CCC(C)=CC2C)C(=O)NCCCSC)CC=CCC12CCC2 C(C(=O)NCC1CC(F)(C)C1)(C(C)C)OCC.c1(C=O)cscc1.N C(=O)(CCC(CC)OC)N(CC(N1CC(=CC)C1)=O)C(C)C C(C(=O)NC(c1cnn(C)c1)CO)(C(C)CC)NC(c1c(CC)ccs1)=O N1(C(C(C)OCCCC)=O)CCC(CO)(NC(=O)CN(c2ccccc2)C)C1 N1(CCC(=O)NCc2cncc3c2CCC3)C(=O)C2CCCCC2C1=O C1(C(=O)NC(CC)(CNC(C2CCC(C)CC2)=O)CC)CCOCC12CCCC2 C1(NC(c2cccc[n+]2[O-])=O)CN(C(=O)Cc2ccc(Cl)nc2)C2CC12 N1(C(c2n(CC)ccn2)=O)CCC2(C1)CN(C(C13CCCN1CC(O)C3)=O)C2 Cc1nc(C(C)C(=O)C2CC2)no1.C(=O)(C(CO)NC(=O)CC)NC=O.N N1(C(C2CCn3c(C)ncc3C2)=O)CCN2CCN(C(=O)C#CC3CC3)CC2C1 c1(CN2CC(NC(C(CCC)C)=O)C(F)C2)cc(Br)c(OC)c(Br)c1 CC1CC(C(=O)NC2CC(C)C2)CCS1.C(=O)(CCCCN1C(=O)CCC1=O)N c1(C(N2CCC(CN(C(c3cc(C)ncc3)=O)C)C2)=O)ccc2c(c1)CC2 c1(C(=O)NC2(CCC(N3C(C(N(C)C)=O)CC3)=O)CCC2)n[nH]cc1Cl c1(C(N2Cc3c(ccc(C(=O)OC)n3)C2)=O)c2cc(Br)ccc2nn1C c1(C(=O)NC2CCN(C(C(CC)(F)F)=O)C2)c[nH]c(C)c(Br)c1=O Cc1cccc2c(C(N3CCC4CN(C(C5OCCC5C)=O)C4C3)=O)c[nH]c12 Cc1o[nH]c(=NC(=O)C2CCC(NC(=O)Cc3cc(C)n(C)n3)C2)c1Br c1(NC(C)C)cccc(C(=O)Nc2ccc(C(F)(F)C(F)(F)F)cc2)c1 C(=O)(C(C)(C)CN(C(=O)CC1CC2(CCC2)C1)C)NC1CCC(SC)C1 Cn1ccc2cc(C(N3CC4CN(C(c5ccnnc5)=O)CC4C3)=O)ccc12 c1(C(=O)NCc2cccc3c2CCN3)cccc2c(Br)ccnc12 c1(C(=O)NC(CC=C)CNC(c2cc3ccsc3s2)=O)c([N+](=O)[O-])c(C)nn1C Cc1cc(=O)n(C)cc1NC(C1CCCN(C(c2nc(O)sc2C)=O)C1C)=O CCC(C(=O)N(CCCCNC(=O)C=C1CCN(C)CC1)C)C(F)(F)F c1(NC(CCC=C)c2ccccc2)nc(=N)[nH]c(N)c1C c1(C(NOC(C(C)C)C(=O)O)=O)ncn2c(=O)n(C)nnc12 C1(C(N2CCC(CNC(c3ccc(O)nc3)=O)C2)=O)CCCC(C(F)(F)F)C1 C(=O)(C(CC(C)C)n1ccnc1)NCC1OCCN(C(c2c(C)sc(Cl)n2)=O)C1 Cc1cc(C(N2CCC3(CC3NC(C3CCOC3C)=O)C2)=O)cc(C)c1C#N c1(NCc2c(CC)nccn2)nc(N2CCCC(C)(CC)C2)nc2ncn(C)c12 c1(CCOC(C(CC)(C)CN)=O)ccc2sccc2c1 N1(C(c2ccc(CSC)o2)=O)CC2CC(NC(C3COC(C)(C)C3)=O)CC1C2 C1(c2nnnn2CCSC)(NC(COCC)C(C)C)CCC2(CC1)CNC(=O)C2 c1(CNC(C(C2CCC2)NC(COCCC#C)=O)=O)cc(=O)cc(C)[nH]1 Cc1nn(C)cc1C(C)C(=O)NCC(C1CC1)N(C)C(c1ccccc1Cl)=O C(=O)(C1=C(C)C(C)(C)OC1=O)NC1CC(NC(CCC=C(C)C)=O)C(O)C1 N1(C(C(=C(C)C2CC2)F)=O)CCOC(CN(C(=O)CCN2CCC(O)CC2)C)C1 N1(C(COCC#C)=O)CCC(O)CC1C(=O)NCCCCCCCO c1(OC2CCN(C(=O)CCCn3ccnc3)C2)cc(CO)ccc1F.CN(C)CC C1(F)(C(=O)Nc2cc(OC)n[nH]2)CCN(C(c2cccc(O)c2)=O)C1 CCCCCCCC(=O)N1CCC(NC(=O)Cc2ncsc2Cl)C(CC)C1 O=C(C1CCCc2cncn21)NC1CCN(C(=O)COc2cccnc2)CC1O n1(CC(N2CCCC(N(C(C(C=C)C)=O)CC)C2)=O)ccc(=O)cc1C C1(C(N2CCOC(CCNC(C3COCCO3)=O)C2)=O)(OC)CCC(F)(F)CC1 N1(C(c2cc(C3CC3)no2)C(=O)NCC)Cc2ccccc2OCC1C CC1C(NC(=O)CC2(O)CCOCC2)CCN1C(C1CCC(OC(F)F)CC1)=O C(=O)(CCCCC(F)(F)F)NC(CC(C)NC(Cc1c(F)cc(C)c(F)c1)=O)C C(=O)(C1CCc2nccn21)NCCCCN(C)C(c1cc(N)ccc1F)=O C(=O)(C(CCCCOC)N(C1CCSC1)C)NCCC N1(C(CNC(CC)=O)=O)CCCCC1Cn1cc(-c2cncc(F)c2)nn1 c1(SC)cc(C(N2CC(NC(=O)C(C)C3CCCC3)C(O)C2)=O)c(C)o1 Cc1cnc(Nc2cn(C)c(C(=O)Nc3ccc(C(N)=O)cn3)n2)nc1 N1(C(C=Cc2ncc(C)[nH]2)=O)CCCN(C(c2ncsc2Br)=O)C(C)C1 CN1CCC(CO)(CNC(C2CSC2)=O)C1.c1(CCC(=O)N)cnn(C)c1O C1(N(C(c2nc(CCC)sc2)=O)C)CCCN(C(C23CCCC2OCC3)=O)CC1 N1(C(c2ncc(OC)nc2)=O)CC(C2CC2C(=O)N(C2CCCCC2(C)O)C)C1 Cc1cnc(C=CC(=O)NC(C)C(C(C)C)NC(=O)Cc2cncs2)[nH]1 Cc1cc(C(=O)NCC2(C(N3CC(O)(C(F)F)C3)=O)CCC2)on1 C(CN=c1nc2c(cnn2C(C)C)c(N(C)CC)[nH]1)=CCCOC.[SH](C)(=O)=O c1(C(N2CC(OC)C(NC(=O)CC3CCC4CC34)C2)=O)cn(C)ccc1=O C1(C(=O)NC2(COCC)CC2)CCCCCN1C(=O)C1=CCCOC1 N1(C(c2ccc(C#C)o2)=O)CC2(CNC(c3cn(CCC)nn3)=O)CC1CO2 c1(NCc2occ(NC(=O)OCC(C)C)n2)ccc(SC2CC2)cc1 CC1(C(=O)NCCCC(O)CO)CCN(C(c2c[nH]nc2Cl)=O)C1 N1(C(C2CCN(C)C2)=O)CC2OCCN(C(c3ccc4scnc4c3)=O)C2C1 C1(C(=O)NCC(CC)CO)CC=CC(NC(c2ccoc2C)=O)C1 C(CC(F)F)(C(=O)N1CCC1CC(C)(C)C)N(C(=O)CC1CCOCC1)C C(=O)C(C)C(C)S(C)(=O)=O.N1(C(CC)=O)CCC(O)(CC)CC1.C(=O)NC N1(C(COC(CC)C)=O)CCCC12CCN(C(C1OC(C)CC1C)=O)CC2 C1(NC(C2CCN(C(COCCCC)=O)C2)=O)CC2(CCCCO2)C1 C1(CCNC(C(Cc2ccccc2)N(C)C)=O)CSCCN1C(=O)C(Cl)=CCl CC(C)(CNC(C1CCCC1NC(c1ccc2cc[nH]c2c1)=O)=O)C1=CCCC1 c1(C(=O)N)cc(C)c2c(O)n[nH]c2n1.C(CC(=O)N(C(C)C1CC1)C)OCC c1(CN2CC(CNC(=O)CCNc3ccccc3Br)OCC2)ccc(O)cc1Cl CC(C)C(O)CC(=O)N1CCN(C(=O)CCOC2CC2)C(C(F)F)C1 CC1(C)CN(C(=O)C=C(Cl)Cl)CC1CNC.C(=O)C1=CSCS1.c1ccccc1.C C(c1ccc([N+](=O)[O-])s1)=CC=O.c1(C(N(CCOC)CC)=O)scnc1C c1(C(=O)NCC23CCCC2CCN3C(=O)C2CC2)cc2ccncc2c(O)n1 C1(N(C(c2c(SC)cccn2)=O)C)CN(C(=O)CC(=O)N(C)C)CC1(C)C c1(C(=O)NCC2(C(=O)NCC(C)(C)O)CCCO2)cccc[n+]1[O-] CC1COC2(CCC2)CN1C(C1(CF)CCN(C(=O)CC2(N(C)C)CC2)C1)=O N1(C(C(CNC(C2C(C)C3CCC2C3)=O)C(C)(C)C)=O)CCc2nnnn2CC1 C#CC(C)(C)C(=O)N1CCC(C(C)NC(C2(c3ccc(F)cc3)CCCC2)=O)C1 c1ncc(C(=O)NC(C)C)cn1.C(C(=O)NC)(C1CC1)OC.C1CCCO1 C#Cc1ccc(OCC(=O)NCC2CC3CN(C(=O)Cn4ccnn4)CC23)cc1 N1(C(C=C(C)C)=O)CCCC(CNC(=O)C=CC2CCCO2)CC1 C(=O)(C(C(C)C)NC(=O)CN1CCCCC1C)NCc1scc(CC)n1 C1(CNC(CC2(C)N(C(c3c(CC)n(C)nc3)=O)CC2)=O)(OC)CC2CCC1C2 c1(C(N(C2CN(C(c3cnc(CC)[nH]3)=O)CC2(C)C)C)=O)n[nH]c2c1CCCC2 Cc1nc(C(N2CCN(C3CCN(C(C4CC4(Cl)Cl)=O)C3)CC2)=O)ccc1C#N N#Cc1ccc(C(N2CCCC2CCNC(=O)CS(N)(=O)=O)=O)o1 C1(CC)CCC(C(=O)NC(C)C(CO)NC(c2cnc(C(C)C)n2C)=O)CC1 C(=O)(C(F)(CNC(=O)C(C)CO)C(C)C)N1CCCC(C(=O)OC)C1 c1(NC(C2C3(CCN(C(C(C)CC(N)=O)=O)C3)C2)=O)ccc(Br)c2ccncc12 c1(NC2CN(C(C(C)C(C)(C)C)=O)C2)ncnc2cccc(F)c12 c1(C(=O)NC(C(CC)C)C(=O)NCCN2CCOCC2)nn2cccnc2c1Cl N1(C(C2C(C)OC(C)C2)=O)CC2CCN(C(=O)C(C)CSC(F)(F)F)CCC2C1 N1(C(CC(CCSC)O)=O)CCN(C(c2cccnc2S)=O)C2(CC2)C1 C1(NC(CCc2c(OC)cccc2)=O)CC(O)CN(C(c2ccc(O)nc2)=O)C1 S(=O)(=O)(c1ccc(OCCOCC)cc1)NC(C(CCC)O)CO c1(C(N2CC(C3OCCN(C(C(C)(C)F)=O)C3)C2)=O)cncc2c1CCCC2 c1(CNC(=O)C)cn(C)nn1.c1ncoc1.CC1(C(=O)O)CCC1.CCCO O=C(O)C(CC(F)F)NC(C1(c2c(Cl)cccc2Cl)CCC1)=O N1(C(CCNC(COC)=O)=O)CC(NC(c2cscc2OC)=O)C2(CC2)C1 c1(C(=O)N)ccc(F)c(C(F)F)n1.C1(CNC(c2ccon2)=O)CCCCC1 C1(NC(CCC#C)=O)CN(C(=O)CNC(=O)CC(C)(C)C)C2(CCCC2)C1 C(CCC(O)CO)N(C(=O)C(CC1CC1)NC(=O)COCC(F)F)C Cc1cnn(CCC(=O)NC(C(=O)NCCC(C)(O)C2CC2)C2(C)CC2)c1 Nc1ccc(C(N2CC3CC(NC(C4CCC5CC5CC4)=O)C3C2)=O)c(F)c1 C1(C(=O)NCc2nc(C(=O)OCC)sc2)CNCC1C1CCOC1 CCCC(C(=O)N(CC(=O)NCC1C=CCC1)C1CCC1)N(C)C C1(NC(c2c(F)cc(Br)cc2Br)=O)C2CCC1CN(C(=O)CCc1cnc[nH]1)C2 C(=O)(CC1COc2ccccc21)N1CC2CCC(N(C(C(C)OCC)=O)C)C2C1 CON(C(=O)C(O)CNC(=O)COc1cccnc1)C1CCC1 N1(C(c2ccc(NC)cc2)=O)CCC2(CC1)CC2C(N1CC=CC1)=O C=CC1(C(=O)NCCSC(C)C)CCN(C(C2C3CC4C(C3)C24)=O)C1 C1(C(=O)NCc2cccc(-c3ccccc3)n2)CN2CCN1CC2 c1(C(=O)NC2C(NC(C3C(c4n(C)cnn4)CC3)=O)CCC2)cc[n+]([O-])cc1 CC(CC(=O)NC1CN(CC(=O)NC(=O)NC)CCCO1)C(F)F.c1cccs1 Cc1c(Cl)cnn1CC(=O)NCCCN(C(=O)C(C)C1CCCO1)C1CC1 C(c1ccc(C2CC2)cc1)=CC(=O)NC1C(NC(C(CC)C#N)=O)CCOC1 N1(C(C(c2cc(C)sc2)(C)C)=O)CCC(C2CCOC2)C1 C1(C(=O)NC2CCN(c3cccc(SCC)n3)CC2)CCc2ccccc2C1N N#Cc1cc(CNC(C2CC(F)(COc3ccccc3)C2)=O)ccc1Br C1(CC)CN(C(C2CCCSS2)=O)CCC1NC(C1CC(C)(C)C1)=O N1(C(Cc2ccc(C(=O)OC)cc2)=O)CC(C2(NC(c3ncoc3C)=O)CC2)C1 N1(C(C2C(C)(C)C(F)(F)C2)=O)CC2CCC(C1)N2C(=O)CCN1CCCCCC1 C(=O)(C(O)C(F)(F)F)N1CCC(C)(CNC(c2ccc(C(C)C)nc2)=O)C1 C12(C(=O)NC3CCN(CCNC(c4ccn(C)n4)=O)CC3)COCC(C1)OC2 N1(C(CN(C(=O)CNC(=O)CCCCO)C)=O)CCC2(CNC(=O)N2)C1 C=CCN=S(C)(=O)NC(C1CCC(c2ccc(C)cc2)C1)=O C(=O)(C1CCc2c[nH]nc21)N1C(CCC(=O)NC2(CC)CCCC2)CCC1 c1(SC)nc(O)c(C(=O)NCCC(C)NC(=O)C(C)(C)N2CCCC2)cc1C#N C(C)(C(C)(C)S(=O)(=O)N(C)C)NC(C1CCSC1)C CCCCC(C)CCC(=O)N1CC2(CC(NC(=O)C(C)CC(F)(F)F)C2)C1 Cc1cn2c(n1)C(C(=O)N(C)CC1CCN(C(=O)Cc3cnc(C)[nH]3)C1)CCC2 Cc1nc(NC(=O)NC(c2ccc(Br)cc2)C(N)=O)c(I)cc1Br Cc1nc(O)sc1C(=O)NC(C)CCN(C)C(C1(CO)CCCCO1)=O Cc1cc(C(=O)N(C2CN(C(=O)CCc3cnco3)CC2O)C)c2c(c1)CCO2 CC1CS(=O)(=O)CCN1C(=O)C(n1cc(COC(=N)O)nn1)C Cc1c[nH]cc(C(N2CC(NC(c3coc(C4CCC4)n3)=O)C(C)(C)C2)=O)c1=O c1(C(N2C3CC(CNC(CCS(C)=O)=O)C2CC3)=O)cc2c(nc1N)CCCC2 c1(C(=O)N)ccc2c(n1)CCCC2.C12(CC(=O)NCCCC)COC(C)(C1)C2 S(=O)(=O)(c1ccc(N2CCC(C3CCOC3)CC2)c(Br)c1)NCc1c(C)occ1 C1(C(N2CCC(CNC(c3n(CC)nc(C)c3)=O)C2)=O)CC2OC1C1CC21 Cc1noc(C2CC2)c1C(=O)NCCC1(O)CN(C(C2CC2(F)F)=O)C1 c1(CCC)n[nH]c(=NCC(CC(C)C)NC(c2sc(CC3CC3)nc2C)=O)s1 CC(=O)CCCC(C)C(=O)N1CCC(CNC(=O)CCP(C)(C)=O)CC1C N1(C(CSCCC)=O)CCC2(NC(c3cnc(COC)s3)=O)CCCCCC12 c1(C(=O)NC(CNC(C(F)OC)=O)C)cc(Oc2ccccc2Br)n(C)n1 C1(NC(C(CCCNC(c2c(CC)n[nH]c2)=O)O)=O)CC=C(C(C)C)CC1 C(=O)(C1=C2CCN=C2NC=C1)N1CC(C=O)C1.c1(C(=O)OC)nnn(C)c1.C CN1CCC(OCCC(=O)NCC(C)(O)CNC(C2CSC2)=O)CC1 C(=O)(C1CCCn2nccc21)NCC(C1CCN(C(C(CC=C)C)=O)CC1)O N1(C(CCC)=O)CCCCC1C(=O)NC(C)CC.C(=O)(C(CC1CCCC1)CC)N C1(C(C)C)CC(C(=O)NC(C)(C)CNC(=O)CC(C)(C)C)CCO1 c1(CC)nnsc1C(=O)NC(CC1CCC1)C(=O)NCC1CCCCC1 C(c1c(Cl)nc2sccn12)=CC=O.N1(CC)CCCC1C(N1CC2CC1C2)=O.N Cc1ccc(Br)cc1CNC(=O)C(=O)NC(Cn1cccn1)C(C)C c1(CC)cc(C(N2CCCCC2CNC(c2csc(COC)c2)=O)=O)ncn1 c1(C2(CN(C)CC)CC2)ccc(OC(F)F)cc1 N1(C(c2c(CC)n(CC(C)C)nc2)=O)CC(N(C(=O)CC(C)C)C)C2(CC2)C1 CCC(F)(C(=O)O)C(=O)NC(C)CC1CCN(C(c2nc(C)n(C)n2)=O)CC1 CC1CN(C(C2COC(=O)N2)=O)CC1NC(c1ccc(F)s1)=O C(=O)(C1=NOC2(CCC2)C1)NCCCCCNC(C(C(C)O)C)=O c1(-c2cccc(S(C)=O)c2)ccc2c(c1NC(=O)CN1C(=O)C=CC1=O)OCO2 c1(NC(C(CCC#C)NC(c2cc[nH]c2CC)=O)=O)ccc(F)c(C)c1F Cc1cc(C(=O)NCC2CN(C(c3nc(=O)n(C)[nH]3)=O)CCC2C)ccc1O C(=O)(C(O)C(C)(C)CC)N1CCC(C(C)NC(C(CC=C)(C)C)=O)CC1 C(=O)(C(C)S(=O)(=O)CCC)NCC(CNC(CCCC#C)=O)O C#Cc1cnc(C(=O)N(C)CCOCCC)c(C)c1.C(=O)(C(F)n1cccn1)N N1(CCC)CCCCC1CNC(=O)C(C(C)C)N1CCCC1=O Cc1ccc(CN(C2CC3CC2CN3)S(=O)(=O)Nc2cc(Br)c(C)cn2)c(C)c1 C1(C(=O)NCCN(C(CCC(C)OC)=O)CC(C)O)CC2CCC(C1)C2 N1(C(C=NOC)=O)CC(NC(c2ccc(C(F)(F)F)[nH]2)=O)C(c2nccn2C)C1 N1(C(=O)NC2CC(n3cc(CCC(C)(C)O)nn3)C2)CCC(C)(CC(=O)O)C1 c1(C(N2CC(C)(NC(COc3cc(C)on3)=O)C2)=O)cccc(C(C)(F)F)c1 C(c1cocn1)=CC(=O)NC(C(C)NC(C(C)=C1CC1)=O)C C(CC(C(=O)N1CC(CF)C1)NC(=O)CCC1(C)N=N1)=CC CC1(C)C(NC(c2cccc(CC#N)c2)=O)C2CCCN(C(C3CC(O)C3)=O)C12 c1(C(=O)NC(C(C)NC(=O)C(C)N(C)C)CO)cc(Cl)c(Cl)c(Cl)c1 c1(N2CC3C(NC(=O)C(C4CCCCCCC4)O)C3C2)nc(Cl)nc2c1SCC2 N1(C(COCCCOC)=O)CCn2c(CNC(C3(SC)CC3)=O)nnc2C1 c1(N2CCC(CC=C)C2)ccc(S(=O)(=O)N(CCC(C)O)C)cc1Br c1(C(=O)OC)cc(C(=O)N(CC(C)N(C)C(C2COCCO2)=O)C)ccc1C N1(C(C(CCC)C)=O)CCC2(CC1)CC(NC(=O)C(=Cc1ccccc1)C)CO2 C#CC(CC(C)(C)C)NC(=O)C(CNC(=O)CCC1(C)CC1)N(C)C c1(C(=O)NCC2(C)CC(NC(C(c3ccccc3)C)=O)C2)nc(=O)n(C)[nH]1 C(=O)C1=C(Cl)CCC1.c1(CNC(c2[nH]cc(CC(C)C)c2)=O)cccnc1.C CS(=O)(=O)C1CN(C(c2cc(C#N)c[nH]2)=O)CC1NC(C1CCSC1)=O c1(C(=O)NCC(CC2CN(C(c3c(C)cco3)=O)C2)(C)C)ccc(N)cc1Cl C1(CNC(C2ON=C(C)C2)=O)CN(C(c2sncc2Br)=O)CC1O C1(CC)(NC(C2CCCS2(=O)=O)=O)CCCN(C(c2ccnc(C)c2)=O)C1 C1(CC(=O)NCC2CCCN(C(=O)CCC=CBr)C2)CCCC(F)(F)C1 c1(C(=O)N)ccn2nncc2c1.N1(C(c2c(CC)cno2)=O)CC(F)(F)CC1C Nc1nc(C(N2CCC2CNC(=O)C(O)CC(F)(F)F)=O)ccc1[N+](=O)[O-] c1(C(=O)NC(CC2CN(C(c3nc(C)sc3)=O)C2)C)cncc(Br)c1C CCCCC(CC)C(=O)NCCC1(C(=O)NCc2c(C)noc2C)CC1 N1(C(Cn2cnc(=N)[nH]2)=O)CCC(C)C(F)(F)C1.C(=O)C1=CCS(=O)(=O)C1.N N1(CC(c2cncc(C(=O)OC)c2)=O)Cc2c[nH]nc2C1 Cc1cn2c(n1)C(C(=O)NC1(C)CCN(C(=O)Cn3cccnc3=O)C1)CCC2 c1(C(=O)OCC)cccc(C(C)NC(C)C(=O)Nc2ccc(C)o2)c1 Cc1ccc2sc(=NCC=CCNC(C3CCCN(C)C3)=O)[nH]c2c1 C=C=CC(C)C(=O)NCCCN(C(C1CC(C)=NO1)=O)Cc1cccnc1 C(=O)(C(CCOC)OC)N1CC(C)(CCC(N2C(CC)CC2)=O)C1 c1(C(N2C(C(=O)NC(C)CCO)CSCC2)=O)cccc(OC(C)C)c1F CC(C)C(C)CC(=O)NCC1CC2CCC1N2C(c1csc2nccn12)=O CCC(CC(=O)N1CC(CNC(c2ccccc2OC)=O)C(F)(F)C1)C(C)(C)C c1(N)ccc(Cl)cc1.C1(C(=O)NCCC(=O)NCCC)CCCN1C(C)=O C1(CNC(c2cccs2)=O)CC2COCC2N1c1ncc2ncnc-2[nH]1 C1(NC(CNC(=O)CC2CCCC2)=O)CCN(CC2CCCO2)CC1 CC1(C(=O)NC2COCC2CNC(=O)Cc2ccc(Cl)cn2)CCCC1(F)F c1(COCC)ccc(NC(c2ccnc(SCCCN3CCOCC3)n2)=O)cc1 S(=O)(=O)(c1cccc(Cl)c1)NCC(=O)NC1C=CCN(C(c2cnsn2)=O)C1 c1(C(C(F)F)NCCOCC(C)O)ccnn1C C(N=c1nc(N2CCCC(C3CCC3)CC2)c2ncccc2[nH]1)C1CCC(=O)N1 c1(C(N2CCC(C)C2CNC(=O)C(C)(F)F)=O)ncc(Br)cc1C(F)F C1(NC(c2cc(C)nn2C)=O)CCN(C(=O)CC(C)Oc2ccccc2)CC1F c1(C(=O)NC2CC(C)(NC(Cc3ccc(C)cc3C)=O)C2)ccc2c[nH]nc2c1 C1(NC(c2c(C)[nH]nc2C(F)F)=O)CCN(C(=O)CS)CC1C.c1n[nH]c(O)n1 C1(C(=O)NC2C(C(=O)NCCc3nc(C)[nH]n3)CC2)C2CCC(C2)C1C C1(CC(=O)NCC(=O)OC(C)C)CCN(C(=O)C=CC2CC2)C1 C1(NC(C2C(NC(C=CC=CCC)=O)CC2)=O)CCCN(C(C)=O)C1 c1(C(N2C(C)(CNC(C3(CC#C)CCCO3)=O)CCC2)=O)nc2cnccc2s1 C1(CC(N2CC(OCC)C2)=O)CCCCN1C(C1CC=CC1)=O Cc1cccc(CC(N2CCC(n3cc(CCC(=O)C(C)C(F)F)nn3)C2)=O)c1C C1(CCNC(C2C(C)C2C)=O)CCN(C(c2ocnc2C2CCC2)=O)C1 N1(C(=O)CS(=O)(=O)NC2CC2)CC2CC1CN2C(=O)CC1CCC(F)(F)C1 c1(C(N2CCC(CCNC(C3(CC)CC3)=O)C2)=O)c2ccccc2nn1C c1(CC)conc1CC(=O)NC1CCC(N(C(=O)CCC2(C)CC2)C)C1 CCC(C)(C)C(C)CC(=O)NCC(F)CNC(=O)C.c1(C=O)ccccc1O.N c1(C(N2CC(CCC)C2)=O)cc(S(C)(=O)=O)cs1.C(=O)C(C)(C)C1CC1.N C12(C(=O)OC)CCCC1(C(=O)NC1CCN(C(=O)C)C1)C2.c1ccncc1.O c1(C(=O)NCCC2CC(NC(CCOCC#C)=O)C2)sc(Cl)c(Cl)c1.O C(C)(C)(CC(F)C(=O)NC)NC(CNC(=O)NC)=O.C1CNC(=O)CO1 N1(C(Cc2c(C)ccs2)=O)CCN(C(C2C3CCC(C3)C2(C)C)=O)CC(C)(C)C1 C1(OC)(OC)CC2(COC(CNC(=O)CC(C)c3ccccc3)C2)C1 Cc1cc(C(=O)OCc2ncc(C3CC3)o2)c2c(Br)cccc2n1 c1(CC)cccc(F)c1.c1(CC)ccoc1Cc1nnnn1CCC1(C)CC1.N C1(CC(=O)N(C2CCC2)C)CC(C)(C)CO1.N(S(=O)(=O)N(C)C)CC=O c1(N2CCC(N(C)CC3CCN(C(C=CC)=O)C3)C2=O)c(C)cc(C)cc1C c1(C(=O)N)cnn2c1N(C)CC2.C1(C(=O)OC)CCC(C(=O)NCC#CC)C1 C(c1ccn(C)c1)=CC(=O)N.C1(C)(C(C)C)CCN1C(=O)Cc1ccccc1 N1(C(C2(OC)CCN(c3ccc(Cl)cn3)CC2)=O)CCCC2OCCC2C1 CCCCCC(CC)C(=O)N(C1CCCN(C(c2ccc3nonc3c2)=O)C1)C N1(C(C=C(C)C2CC2)=O)CC(NC(c2cc(C)nc(C)n2)=O)CC(O)C1 c1(OC)ccc2[nH]c(C=O)c(C)c2c1.C1C2CC1CN(C(=O)CC1(C)CC1)C2.N Cc1ccc(C(=O)NC(C(=O)NC(C)CO)C2CC2)nc1O c1(C(C2CCCCC2)NC(CSC)=O)cc(F)cc(F)c1 O=C1CC2CC(C(=O)NCCN3CC4CC4C3)C1O2 c1(C(=O)NCCOC2CCN(C(C3(C)COC3)=O)CC2)cc(Cl)cc2c1OCC2 N1(C(c2c(C)ccs2)=O)CC2(CCCC2NC(c2ccc3ccsc3c2)=O)C1 C#CC1(C(=O)N)CCN(C(=O)C(C)C2(O)CCC2)CC1.C(CN(C)C)CC(C)C c1(C(N2C(C(=O)OC)CCCC2)=O)cnn2ccc(C#N)cc12 c1(NC)ccc(C(N2CC3(CCN3C(=O)C=C3CCOCC3)C2)=O)cc1F c1(C(C)C)cc(=NC(=O)NC2CS(=O)(=O)CC2O)[nH]n1C(C)(C)C c1(C(=O)OC(c2cccc(Cl)c2)C(=O)OCC)nc2ncccn2n1 NC1CCOC(C2CCCN(Cc3ccn(-c4ccccc4)c3)C2)C1 C(N=c1[nH]cncc1Br)C1(F)CCN(C(C(C)CSC(F)(F)F)=O)CC1 C(=O)(CC1=CCN(C(=O)C(C)(C)C(F)(F)F)CC1)N.CC1(C)OC(=O)NC1C c1(C(C)OC)nc(C)c(C(=O)NC2CCCC(NC(=O)CSC)C2)s1 N1(C(C2CC(C)(NC(c3c[nH]c(=NC)s3)=O)C2)=O)CC2(COCC(=O)N2)C1 C1(NC(C2CCC(C(=O)OC)CC2)=O)CN(C(C2CC(C)CO2)=O)CC1(C)C N1(C(C#C)=O)CC2(CC(C(=O)Nc3cn4ccccc4n3)CO2)C1 c1(NC(C2C(C(=O)NC3CC3)C2)=O)nc(Cl)c(Br)cc1I c1(CC(=O)N(CC(=O)O)Cc2ccccc2)ncc(Br)cc1Br C(CC(CC)C(=O)N1CCC(C)(C(=O)NCC2CCCC(OC)C2)C1)=CC N1(C(C2(C3CC3)CC2)=O)CC=C(CC(=O)N2CCN(C3CC3)CC2)CC1 CC1CCCN(C(=O)Cc2ccoc2)C1CO.C12(CCCCC1)CC(=O)N(C)C2 c1(N2CC(CN(C(CCc3ccc(C)cc3)=O)C)C2)ncnc2cccnc12 c1(C(=O)NC(C(C)O)C(=O)NC2CCCSCC2)c[nH]c2ccccc12 Cc1cc(Br)c(C(=O)NC2C=CCN(C(=O)C(C3CCCCC3)O)C2)s1 C(=O)(C=CS(C)=O)NC(CCOC)CNC(=O)Cc1[nH]cnc1C N1(C(c2c(OC)cnnc2)=O)CCc2ccc(C(N3CC4(CSC4)C3)=O)nc2C1 CC(CC(C)(C)C)C(=O)N1CCCC1CN(C(=O)CSc1nnnn1C)C C(=O)(CC(=O)OC(C)(C)C)NCC1CC(C(N(C2CCSC2)C)=O)C1 c1(CC(=O)N(CC(CC)NC(=O)CCC2(C)CC2)C)cc(O)nc(O)n1 C1(C(=O)NC2(C)CCN(C(c3cc4n(n3)CCCC4)=O)C2)OCC2CCCC1C2 N1(C(c2ccc(C#C)cc2C)=O)CCC2CN(C(C3CC=CCC3C)=O)CCC12 c1(C(=O)NC2CC(OC)CN(C(=O)Cc3sccc3C)C2)cc(C)c(Cl)cc1C N1(C(CCC=C)=O)CCc2sccc2C1CNC(=O)C#CC(C)(C)C C(=O)(CC1=CCN(C)CC1)NCCCOCCNC(Cc1c(C)cc(F)cc1)=O c1(COC)cc(C(=O)NC2COCC2C)cs1.C1(C(=O)N)CCC(=O)C1 C1(C=O)COC2(CCC2)CO1.N1(C(COCCN(C)C)=O)CC(C)C(C)(C)C1 Cn1ncc2ncnc(Nc3nc(-c4cccc(S(N)(=O)=O)c4)cs3)c12 C(C(N=c1cc(C)nc(C)[nH]1)C(C)C(C)C)NC(c1c(NC(C)=O)cccc1)=O Cc1ccc(C)c(C(=O)NCCC2CCC2)c1.C1(C=O)CCCN(C(C)C)C1.N N1(C(c2nc(C#C)sc2)=O)CCCN(C(c2cc(OC)ns2)=O)C(C)C1 C1(C(=O)NCCNC(c2cn(C3CC3)cn2)=O)CCN(C2COC2)C1 c1(OC)ccc(C(=O)NC)cc1.C1CCC1(C)C.c1(C=O)ccc(C(F)F)o1 N1(C(C(CC#C)O)=O)CC(C(=O)NCCC(O)C2CC2)CC12CCC2 C1(C)(CNC(C(CCCOC)C)=O)CC(F)(F)CN1C(=O)C(c1ccccc1)C C(=O)(C(F)(F)C(C)(C)O)N1CC(O)(C(C)NC(C(COCC)C)=O)C1 c1(C(N2CC(NC(CCOCCOCC)=O)C2)=O)cscc1SC C1(C(=O)NCC(C)OC)CCCC(NC(C2CN(C)CCO2)=O)C1 N1(Cc2cc(C)cc(F)c2)CC(C2CCN(C(c3ccnc(O)c3)=O)CC2)C1 c1(CNC(c2cn(CCO)nn2)=O)cn(CC)nn1.C1(C(=O)N)CC=CCC1 c1(C(=O)NC2CCCCN(C(C(CC)N(C)C)=O)C2)ccc(S(C)=O)cc1 CCCCC(C(=O)NC1COC(CN=c2nc(C(C)C)[nH]s2)C1)NC(N)=O N1(C(CN(CC(C)(C)C)C)=O)CCCC(C)(C)C1C.C1(C(=O)N)CC(O)C1 c1(C(=O)OC)ccc(C)nc1.C1(C=O)CC2CC2N1C(c1sc(Cl)nc1Cl)=O.N CCC(CC(=O)NCC1CC1C)c1ccc(C)cc1.n1(CC(=O)N)cccn1 N1(C(C2CCC(CC)O2)=O)CCC(NC(c2cccc(F)c2C)=O)C12CCC2 c1(C(=O)NC2(C(=O)Nc3cn(CC)nc3C)CC2)cc(C#N)[nH]c1C C1(NC(c2ccc(OC)s2)=O)CCN(C(=O)Cc2cnc(C)[nH]2)CC1O c1(OC)coc(CN2CC3CC3(C(=O)O)C2)cc1=O C1(C(=O)NC2C(NC(c3cc(CC)no3)=O)CCCC2)OC(C)(C)OC1(C)C C(c1cccc(CO)c1)=CC(=O)NCC1CCN(C(=O)CC2CCCCC2O)C1 C1(C(=O)NCC2(CO)C(C=C)C2)CCCCCCN1C(c1cnc2n1CCC2)=O n1(CC(=C)C)nc(CCCCC)nc1-c1cnn(CC)c1 CC(C)C(F)C(=O)NCc1csc(C)n1.c1(C=O)c[nH]nc1-c1ccncc1.N C(=O)(C1CCCc2n[nH]cc21)NC1CCCCCN(C(C2(C#C)CCCC2)=O)C1 c1(OC)ccccc1C(O)C(=O)NC1CCCC(NC(c2cc(C)[nH]c2C)=O)C1 c1(CC)cc([N+](=O)[O-])ccc1NC1CCCN(C(c2cc(OC)n(C)n2)=O)C1 c1(CN(C(CCSC)C(=O)Nc2ccccc2)C)ccc2cncn2c1 N1(C(C(CC(F)F)NC(C2CCC(C)(C)C2)=O)=O)CCOCC2(CCC2)C1 c1(C(N(CC(C)O)CC)=O)cnc(O)n(CCC)c1=O.C1(C=O)CC12CCC2 CC1CN(C(c2cnn(C)c2C(F)F)=O)CC1C.C1(O)(CC=O)CCCC1.N c1(CNc2cc(C(=O)NC(c3ccsc3)C)n(C)c2)cc(O)ccc1F c1(NC(CN(C(c2cc(C)oc2)=O)C)(C)C)nc2cc(F)cc(F)c2o1 Nc1cc([N+](=O)[O-])ccc1C(N1CCC1CNC(C1(CF)CCC1)=O)=O C1(C(=O)OC)CN(C)C(=O)CN1C(CCC1CC1C)C(=O)Nc1ccccc1 c1(C=O)cn2cccc(Cl)c2n1.N1(C(CCSCC)=O)CC(C(C)(C)O)(C)C1 C=CCC(F)(F)C(=O)N1CC(NC(c2cnc(C3CC3)o2)=O)C(SC)C1 c1(C(=O)NC2C(N3CCN(C(C(F)=CC)=O)CC3)COC2)c(C)cc(F)cc1C C(=O)(CC(C)(C)CC(=O)NC(C)CN(C)C(c1oc(C)nc1)=O)OCC c1ccc2c(c1)CC(C)O2.n1(CC=C)nnnc1C(c1cnc(C(C)(F)F)s1)N c1(N2C3CS(=O)C(C3)C2)nc2c(c(=NCc3c(Cl)cccc3Cl)[nH]1)CCCC2 C(=O)(C(S(C)(=O)=O)C1CC1)NCC(C)N(C)C(C1C=CC=CC=C1)=O c1(NC(C2CCN(CC(=C)C)CC2)=O)ccc(OCC)c(OC)c1 Cc1ccn(CC(C)(O)C(=O)N(C)C(c2ccc(-c3nn[nH]n3)cc2)C)c(=O)c1 N1(C(C=CC(=O)N)=O)CCOCC1.C1(CCC)(C(=O)NCC(C)C)CCC1 C12(CCC(=O)Nc3nc(-c4ccccc4Br)cs3)CCC(CC1)NC2 c1(C(C)=O)cccnc1N1CCC(CC(=O)NC(c2nnc(C)o2)C)C1 N1(C(C(CC#C)O)=O)CCC2(CC2C(=O)N(C(C)C(=O)OCC)C)C1 Cc1cc(CNC(=O)CCC(=O)C2CC2)oc1C=O.C1(C(F)(F)F)CCC1 N1(C(C2(C=C)CC2)=O)CCCSCC1C(F)(F)F O=C1CCCC2C(C(N3CCC3CC(=O)NCC34CCCN(CC3)C4)=O)C12 C1(NC(=O)CC2CS(=O)C2)(CO)CCN(C(=O)C(O)Cc2cnc[nH]2)C1 c1(SC)cnoc1C(=O)NC(C)C(c1ccccc1)NC(=O)CCF Cc1nc(C(C)C)nc(O)c1C(N1CCCC1)=O.C(=O)CC1(O)CC1.CC.O C1(C(=O)NCC2(NC(CC(CC)C3CC3)=O)CC2)CCCCC12CC2 C1(NC(CC(=C)C)=O)CC(CNC(c2ccccc2)=O)C12CCC2.C(=O)N C1(CNC(c2c(C)ncs2)=O)CN(C(C23CCCC(C2)OC3)=O)CCC12CCC2 Cc1c(C(=O)NCC(C)CNC(C2CC3CC2CO3)=O)[nH]c2c1CCCC2 c1(C2C(C=O)C2)cc(Cl)cc(Cl)c1.C(=O)(C(F)=C(C)C)NC(C)C.C CCCC(C)(O)CC(=O)NC1CC(C)N(C(=O)COc2ccc(Cl)c(Cl)c2)C1 N1(C(C(Br)=C(C)C)=O)CCCC(O)(CNC(=O)CC2=CCCCC2)CC1 C(=O)(C(F)(CNC(C1C2CCC(C2)C1C)=O)C(C)C)NC(CCC)C CS(=O)(=O)c1nccc(N(C2CC(N)C2)C(c2ccc(O)c(Cl)c2)=O)n1 N1(C(CCN(C(=O)COC(C)CC)CC=C)=O)C(CO)CCC12CCC2 c1(C(N2C(CNC(CS(C)(=O)=O)=O)CC(F)C2)=O)cc2c(nc1O)CCCC2 c1(OC(C)C)cc(-c2nc(C3(O)CCCCCC3)no2)cnc1F N1(CC)CC(C(=O)NCC2CC2)CC1=O.c1ccc(Cl)cc1.C(=O)(CC)N C1(C(N(C)Cc2cn(CC)nc2)=O)CC2CCC1N2C(C1CC2CC2C1)=O c1(CN(C(=O)C(N)CCc2ccncc2)CC)ccc(Cl)c(Cl)c1 C(C)(C)(C(=O)N(C)CCN(C)C(c1ccc(-c2ccco2)s1)=O)SC C1(NC(C(COC(C)C)NC(=O)C(F)F)=O)CCCC(O)CC1 Cc1cc([N+](=O)[O-])cnc1NC1CC2CN(C(=O)C(C)C(C)O)CC12 c1(C(=O)NCCCCCCN(C(C(CC)C)=O)C)nc2ncccn2n1 c1(C(N2CC(OC)CC2)=O)c(C)nn(C)c1-n1cccn1.c1(C(=O)N)ccc[nH]1 C#Cc1ccc(C(=O)NC2(CNC(c3cc(C)[nH]n3)=O)CCC2)nc1 C1(NC(c2cc(CC)on2)=O)CCCCC1NC(=O)Cc1csc(C=O)c1 C(C(C(=O)NCC(=O)N(C)C1CC1)N(C)C)NC(CN(C(C)=O)C)=O c1(C(=O)NCC(C)NC(C2CCC3CC(C)CN3C2)=O)ccc2c(c1)CCC2=O N1(CCC)CCN(C(=O)C(C)(CO)NC(=O)CCCC2CCCO2)CC1 c1(C(=O)NCCC(C)N(C(=O)COCC2CC2)C)ccc(CO)cn1 c1(N2CCC(CC(=O)NC)C2)ccncc1S(=O)(=O)N1CCOC(C(F)(F)F)C1 CCCCC(O)CC(=O)NC1CC(CO)N(C(=O)Cc2cccc(Cl)c2F)C1 C#CC(C(C)OC)NC(=O)OC.C12CC(CO1)N(CC)S(=O)(=O)C2 C(C)(C(C(=O)NC)N(C)C)OC.c1(CC)ccc(O)cc1.c1ccsc1C=O c1(C(=O)NC(C(=O)N(C2C(C)COCC2)C)CCN(C)C)ccc2n[nH]cc2c1 Cc1cc(C(N2CCC(C(=O)NCC(O)CC3CCC3)C2)=O)cc(O)c1 C1(CNC(CCC#C)=O)CN(C(C2CC=CC2)=O)C2CCN1C2 C1(CNC(c2ccc(CC)nc2)=O)CCN(C(C2SCCCS2)=O)CC1O C1(CNC(c2ccsc2Cl)=O)CCCN(C(=O)CCn2cnccc2=O)C1 C1(C(=O)N)CCn2ncnc2C1.C1(C(=O)OC)CCCC(C(N2CC(C)C2)=O)C1 c1(C(=O)NC2CC(OC)CN(C(C(C)SC)=O)C2)[nH]c2cc(C)cc(C)c2c1C c1(C(=O)N)ccc2c(c1)c(C)c(C)n2C.C(=O)(C(C)(O)CC)N(CCC)CC CCC(C)C(CC(=O)Nc1ccc(C)c(Cl)c1)NC(c1csc(Cl)c1)=O CCC(CCC(=O)NC1C2CCN(C(=O)CCc3cccc(Br)c3)C12)OC CC1CN(C(C2C3CC4C(C3)C24)=O)C(C)CN1C(C1CC2(CCCO2)C1)=O Cc1nn(C)c(Cl)c1CNC(=O)NCC(C)C(N1CCCCC1)=O Cc1nc(O)nc(C)c1C(N1CC(NC(c2cnc(O)c(F)c2)=O)CC(O)C1)=O NS(=O)(=O)c1sccc1C(c1nnnn1CCCF)NCCOCC(F)(F)F C(=O)(CCCC(C)=O)NC1CC(CNC(c2cc(OCC)no2)=O)C1 C(=O)(CC(C)(C)F)N(CCNC(Cn1cc(C(=O)OC)nn1)=O)C(C)C C(=O)(C1=CCC(C)CC1)N.c1(COC)nc(OC)cc(N2CCCC2C2CC2)n1 C12(NC(c3cccnc3Cl)=O)CCCN(C(c3nncs3)=O)CC1C2 N1(C(C(C)OC)=O)CCCCC12CN(C(c1nc(SC)ns1)=O)C2 C1(NC(c2ccc(F)cn2)=O)CC2CC1N(C(C1CCCC1)=O)C2 N1(C(C(COCC)NC(=O)C=Cc2ccncc2)=O)CCC2(CCC2)C(O)C1 c1(NC(CC2OCCN(C(C3CCC(CC)CC3)=O)C2)=O)nc(C)c(Cl)cc1Cl N1(CC(=O)Nc2cccc(F)c2Br)CCN(C(c2ccc(O)c(I)c2)=O)CC1=O c1(CC(C)C)cc(C=O)n[nH]1.c1(CCC=O)cnn(C)n1.C(C)(C)C1CC1.N O=C1CCC(C(N2CCC(C(O)C(F)F)CC2)=O)CCN1 CC1CN(C(c2c[nH]cc2C2CC2)=O)CC1NC(c1ccc(Br)cn1)=O C=CC1CCCCN1C(C1(NC(=O)CCc2cc(C)no2)CC(F)C1)=O c1(CC)cc(F)ccc1C(=O)NC1CN(C(=O)CCO)CCC1F.CC(F)(F)F Cc1nc(O)nc(O)c1NC(C1(F)CCN(C)C1)=O.c1cc(C(F)F)cc(F)c1 c1(C=O)ccnc2c(F)cccc12.CC(C)CCNC(=O)COCCN(C)C C1(c2cn(NC(=O)NCCC)nn2)CCN(C(=O)OCc2ccccc2)CC1 Cc1cc(F)c(CC(=O)NCC2=CCN(C(=O)C(C)n3cccn3)CC2)cc1F N1(C(CSCC=C)=O)CC2CCN(C(=O)C(N3CCCCCC3)C)C2C1 c1(C(C)=O)cncc(C=O)c1.C1(CC)CCN(C(c2c[nH]c(C(N)=O)c2)=O)C1.N c1(C(=O)NCC2N(C(C3C(CCC)C3)=O)CC(O)C2)cc2ccncc2cc1F Cc1ccc([N+](=O)[O-])c(N(C)CCN(C(=O)Cc2csc(Cl)c2)C(C)C)c1 C1(C(N2CCN(C(c3c(C)onc3)=O)CC(O)C2)=O)CCc2ncc(C)n2C1 c1(OC)ccc(C(=O)NC(C)CC(C)NC(c2ccc(CC#N)cc2)=O)nn1 c1(-c2cccc(NCc3ccc(CC)nc3)n2)ccc(C#N)c(F)c1 C(=O)(C1=CCCCO1)NC(C(N1CCCC(NC(C)=O)C1)=O)CC1CC1 N1(C(CCCCCN(C)C)=O)CC(C2CN(C(=O)CC3CC4CC4C3)C2)C1 CCCC(C(=O)NCC=C1CCN(C(c2cc(C#N)c(C)cn2)=O)CC1)C(C)C C1(NC(Cc2n(C)ccn2)=O)CC(C2CCN(C(=O)CCCCC(F)F)C2)C1 C1(C(=O)NC(CC#C)C)CCN(C(=O)CC2CCC2)C12CCC2 C1(OCC)CC(CC(=O)NCC2CN(c3nnco3)CCO2)C1(C)C N1(C(C=CC(C)C)=O)CCC(C)(C)C(C(=O)N(C2CC3CCC2O3)C)C1 c1(CC(N2CC(CC)OC(C)C2)=O)cc(F)c(F)cc1F.C(C=O)NC(C)=O.N C1(CNC(C(C)N(C)C)=O)CCCCN(C(c2cncc(-c3cc[nH]n3)c2)=O)C1 C(=O)(C#CC1CCCC1)NCC(C)(CO)NC(c1cc(-c2cn(C)nc2)no1)=O N(C1CCCc2c[nH]nc21)C(CONC(c1ccc(O)cc1F)=O)=O C(C)(CCC(F)(F)F)NC(C(c1ccc(C)cc1)F)=O N1(C(c2cc(CC)oc2C)=O)C2COCC1CC(NC(C1CC1(F)Cl)=O)C2 N1(C(C(CN2CCN(C)CC2)(C)C)=O)CCC2CN(C(c3cccs3)=O)CC2C1 C1(NC(c2nc(OC)oc2)=O)CCCCN(C(C2CC(O)CN2C(N)=O)=O)C1 O=C(C1SCc2cccnc21)NCCC1COCCN1C(=O)CC(F)(F)C(F)F C(=O)(C(O)C(F)(F)F)NCc1nc(CNC(=O)Cc2cnccc2Cl)sc1 c1(N2CCN(C(C3CCc4ncnn4C3)=O)CC2)nc2cc(Cl)cc(Cl)c2o1 Cn1nc(C2CN(CCC=Cc3ccccc3)CCO2)c2ccccc12 C(=O)(C(C(C)CC)NC(C12CC(C#N)(C1)C2)=O)Nc1c(CC)cccc1 c1(CCC(=O)NCCC)ccc([N+](=O)[O-])cc1.n1(CC=O)cc(F)ccc1=O.N CN1CCC(C(=O)NCC2CCCCN2c2ncccn2)C1=O Cc1cc([N+](=O)[O-])ncc1C(=O)N(C(C)CC)C.c1(C=O)cc([N+](=O)[O-])n[nH]1.N C1(NC(C(c2cccc(Cl)c2)(C)C)=O)CCCC(NC(C2CCCCS2)=O)C1 N1(C(=O)CC2CC=CCC2)CCCC(C2(O)CCC2)C1 C12(NC(c3c(C)nco3)=O)CCCN(C(c3cn(C4COC4)nn3)=O)CC1C2 C1(C)(C(=O)NC(C(=O)OCC)C)CCCC1.C(C1CCC1)=CC(=O)N CCC(C)CCC(=O)N(CC(N1CCC(F)(CO)C1)=O)C CCC(CC(=O)NCC(C(C)C)NC(=O)C(c1csc(=N)[nH]1)=O)C(C)(C)C Cc1nc2cc(C(N3CC(NC(=O)CCN(C)C)C3)=O)ccc2o1 C1CN(C(C2CC(=O)NC(=O)C2)=O)C(C)C1.C(C=O)=CCN(CC)C CC(C)(F)C(C)(F)Cn1cc(CNC(c2sccc2C(F)F)=O)nn1 CC(=NO)C1CC(C(=O)NCC2=CCN(C(c3nc(O)c(C)s3)=O)CC2)C1(C)C C1(NC(CCN(C)CC)=O)CC(NC(c2c(C)cc[nH]c2=N)=O)C12CCC2 c1(C(=O)NCC(CC(C)C)(C)NC(=O)CC2CCCO2)c(F)ccc(F)c1O c1(C(=O)NC2CC3CN(C(C(=O)NCC#C)C)C(C2)C3)ccnc2c1nnn2C CN1CC(C)(NC(=O)C(C2CCC2)NC(=O)CC)CCC1=O.C(=O)(CO)N CCC(CC(F)F)C(=O)NC(C)CCN(C(=O)Cn1cc(Br)c(C)n1)C n1(CCC)nc(C)c(C(=O)NCCC2(O)CCCN(C(=O)CC(C)CF)C2)c1C C1CC2CCCC2N1C(=O)CC1CCC1.C1(C(=O)NC)(COC)CCCC1 N1(C(c2c(C(=O)OC)nn(C)c2)=O)CCOCCC1.c1(C=O)cc(Cl)n(C)n1.N c1(CC=O)nocc1.c1(C2(C(C)NC(C3(CC)CC3)=O)CC2)ccno1 C1(C(=O)NC2C(C)(C)CN(C(=O)CC#N)CC2)CSC(c2ccccc2)=N1 C(=O)(CCCCCN(C)C)NCC(C(=O)NCC1CCN(CC)C1)C Cc1c(C(N2CCC(N(C(=O)CC#N)CCO)C2)=O)sc2cccc(F)c12 C1(NC(CCC2C(C)(C)C2)=O)CC2CCCC(C1)N2C(c1ccc(F)cc1F)=O C(=O)(C1CC(C)Cc2c[nH]nc21)N1CCN(C(c2c(CC)cco2)=O)CC12CC2 C(CC(O)C(=O)NCC1(C)CC12CCC2)SC.C(c1ccsc1)=CC=O.N C1(CNC(CCC=CCC=C)=O)CCCCCN1C(=O)CN(C)C1CC1 CC1(C)CCCN(C(=O)Cn2nnc(=N)[nH]2)C1C.c1(C(=O)N)cncc(F)c1Cl c1(CC)cc(C(=O)NC2(CNC(=O)C=CSC)CCOCC2)ncn1 N1(C(C(CC)n2cccn2)=O)CCN(C(=O)C(C)(CC)CC)CCC1C c1(C(=O)NCCN(C(=O)CC2CCCN2)CCC)c(F)ccc2nc[nH]c12.C C1(=CC(=O)NCCCOCCNC(C2CC(O)C2)=O)CCCCC1 c1(C(N(C)CCC2CCCCN2C(c2cnco2)=O)=O)ccc2ccn(C)c2c1 N1(C(c2c(F)ccnc2F)=O)CCC(NC(C2C3CCCC23)=O)C12CCCC2 N1(C(CCC(=C)Cl)=O)CC(C)OC2(CCC2)C1.c1(C(=O)N)cc(C)n(C2CC2)n1 N1(C(C(N2CC(C)C2)C)=O)CC(=O)NCC1C(=O)NCC1COC(=O)N1 c1(NC(C(=O)NC(c2ccc(Cl)s2)C)=O)ccc(C(C)(C)C#N)cc1 C(C1=CCN(C(=O)C(c2ccccc2)NC(=O)C(C)(F)F)CC1)OC c1(C(C)=O)ccc(SCC(N2CCC3C(NC(c4ccc(C)nn4)=O)C23)=O)cc1 CCC(CC)C(C(=O)N(C(C)C(=O)NC(C(C)C)C(F)(F)F)C1CC1)OC N1(CCCCCNC(Cc2scc(C)c2)=O)CCN(c2ncncc2Br)CC1 Cn1oc(C(=O)NC2CC(C)(NC(c3ccc(C4CCCCC4)o3)=O)C2)cc1=O C1(C(=O)NCC=C(C(=O)NCCC(COC)O)C)Cc2ccccc2C1 C(=O)(C(C)CC(N)=O)NC(C1(C(N2CCC(F)(F)C2)=O)CC1)C n1(CC)nccc1C(=O)N(C(C)CNC(=O)C(=O)N(C)C)CC.CC C(=O)(CC1=CCCCC1)NC1CCN(C(c2nc(N(C)C)oc2)=O)CC1O C1(CCNC(c2n(CC#C)ccc2)c2nnnn2CC=C)CCCC(C)C1 C1(CNC(COC)=O)CC2CC(C1)N(C(c1cc(C)co1)=O)C2 c1(CNc2c(C(C)NC)cccc2)c(Cl)cccc1Cl.C1(N)CC1 c1(CC(=O)NC2CCN(C(c3cc(C)sc3C)=O)C2C)c[nH]c2c(C)cccc12 C(C)(C(=O)N)(C(C)C)NC(C)=O.C1CN(C(C2(CCO)CC2)=O)CC12CC2 c1(CC)ccc(C(N2CCCC2CCNC(=O)Cc2ccoc2)=O)cc1CC c1(C(C(=O)OCC(=O)Nc2scc(C)n2)O)ccccc1F c1(C(=O)NC2CC(CNC(C3CCCS3)=O)C(O)C2)cc(F)c(F)cc1F c1(OC)ccc2c(CC(=O)NCC(O)CN(C)C(C3(C)CC=CC3)=O)c[nH]c2c1 C(=O)(C1=CS(=O)CCC1)N1CCCC(CCNC(C(=O)NC)=O)C1 C(=O)(C(O)C(F)(F)F)NCCOCCNC(C=C(C)C(F)F)=O c1(C(N(CCCN(C)C(C2(C)COC2)=O)C)=O)cc(Br)c(F)cc1F CC(C)(C)C(O)C(=O)N1CCCC(CC(=O)NC2CC2O)C1 C(=O)(C1SCc2cccnc21)N1C2CN(C(c3cnc(C4CC4)s3)=O)C(C2)C1 c1(OC)ccc(CC(=O)NCCN(C(C23CC(O)C2C3)=O)C2CC2)nc1 Cc1c(C(=O)NC(CNC(=O)CO)C(C)C)[nH]ccc1=O.c1ccnn1C.C C1(C(N2CCC3CCC23)=O)CCc2nnc(-c3ccccc3)n2C1 C(=O)(CC1CCc2ccccc21)N.C(C)(C(=O)NCC1(C)CCC1)SC(C)C c1ccc(F)cc1.C1(NC(C2(NC(C)=O)CCC2)=O)CCCC1.C(=O)CC.N c1(CC)csc2sc(C)cc12.C1(C(=O)OCC)CCOC1C(=O)NC=O.N C1(NC(COc2cccc(C)c2)=O)CN(C)CC(F)(F)C1.c1ccc(O)c(C#N)c1 N1(C(c2nnc(C)s2)=O)C(CNC(=O)CCc2ccncn2)CC2COCC12 c1(C(N(CC(O)CNC(=O)CCN)CC)=O)ccc(Cl)cc1.CC.O C(CC(=O)NC(C1(CO)CC1)C)(C(C)C)NC(C1C(C(C)C)CCO1)=O Cc1nc2ccc(C(N3CC(CCNC(c4cc(C(F)F)cs4)=O)C3)=O)cn2n1 c1(CCC(=O)N(CCCN(C(C(C)N(C)C)=O)C)C)cc(Br)ccc1F N1(C(C2(CC)CCOC2)=O)CCN(C(=O)C=CC=O)CC1.C1CC1.C1CC1 CCCCCC(O)CC(=O)N1CC2(C1)CN(C(c1cccc3ccnn13)=O)C2 N1(C(c2cc(CCC)on2)=O)CC(CNC(=O)Cc2ccco2)C(O)C1 c1(C(=O)Nc2ccc(-c3cnc(OC(C)C)nc3)s2)cc(Br)c(O)c(Br)c1 C(=O)(CCCCCC(C)O)NCCCC(CCC)NC(c1[nH]nnc1C1CC1)=O Cc1nn(C)c(C)c1SCCNC(N1CCC(CC(F)F)CC1)=O CCCC(C)CC(=O)NCc1ccsc1C(=O)NC(CO)C(=O)N(C)C C1(C(=O)NCC2CC(NC)C2)(CC)CCN(C(c2cc(C)ncn2)=O)C1 N1(C(CCn2ccc(C)n2)=O)CCC(c2cn(Cc3cnns3)nn2)CC1C c1(C=O)ccc([N+](=O)[O-])nc1.C12(C(N(CCCOCC)C)=O)CSCC1C2.N C1(Cl)(C(N2CCCC(NC(c3coc(Cl)n3)=O)C2)=O)CC12CCOCC2 N1(CCC(=O)NC(C)(C)CNC(=O)C2=CS(=O)CCC2)Cc2ccccc2C1=O c1(C(=O)NCCCCNC(c2ccc(SC)o2)=O)cccc(N=S(C)(C)=O)c1 c1(C(N2C(CNC(C3(C)C=CCC3)=O)C=CC2)=O)cnc2c(c1)CCC(=O)N2 N1(C(c2cncc(NC)c2)=O)CCC(NC(c2cncc(C(F)F)c2)=O)CC1C N1(C(C(C(C)C)O)=O)CCC2(CC1)CN(C(C1(F)CC=CC1)=O)CC(C)O2 C(C(=O)N(C)CC1CN(C(c2nc(O)sc2C)=O)CCO1)(C(C)(C)C)OC CC1CC(NC(=O)CN2CCN(C)CC2)CCN1C(=O)CCSCC(N)=O N1(C(Cc2cccc(OC)c2)=O)CC(NC(C2CSCC(=O)N2)=O)CC(C)C1 c1(CN(C(NNC(c2ccc(C)c(O)c2)=O)=O)C)oc2c(C)cccc2c1C c1(CC)ccc(NC(=O)CCN(C(C2CC(F)CN2C)=O)CC)c(C)c1 Cc1ccc(C)c(C(N2CCC3CC23C(=O)NCc2ccn(C)n2)=O)n1 C1(CNC(c2c(CC)nn[nH]2)=O)CC2CC2N1C(C1CCCN1C)=O N1(C(c2onc(NC)c2C)=O)CCN(C)C(C(=O)OC)C1 CCCC(C)(C)CC(=O)N1CCC(N(C)C(C2(C#N)CC3C=CC2C3)=O)CC1 c1(CCC(N2CCC(CCNC(c3n(CC=C)ccc3)=O)C2)=O)cccc(F)c1 C(=O)(N=c1[nH][nH]c2c1CN(C(c1cccc(Cl)c1F)=O)C2)C1CCN(C)C1 CCCC(C(=O)NC(CO)C(C)NC(=O)C)OC.c1cccc(C(C)(C)C)c1.O c1(NC(C)CC(C)(C)CO)ccc(S(=O)(=O)NCCc2cncc(Br)c2)cc1Br N1(C(C(=O)N(C)C)=O)CCC2CCN(C(=O)CSc3ncnc4[nH]cnc34)CC12 C(CC(F)CN=[N+]=[N-])NC(CC1(C)N(C(C(C(C)C)C2CCC2)=O)CC1)=O c1(C(=O)NC2C(C)CN(C(=O)CCc3ccoc3)CC2)ccc(Cl)c(F)c1F c1(C(N(C2CCN(C(=O)CCCC(F)(F)F)C2)CC)=O)ccc(N)c([N+](=O)[O-])c1 C1(CCNC(C2C(CNC(CCCSC)=O)C2)=O)CC(=O)N(C)C1 C1(N(C(C)C)C=O)CCCCN(C(C2CC2c2cnn(C)c2)=O)C1.C(C)(C)C N1(C(c2ccc(C(=O)OCC)nc2O)=O)CCC2(CCCO2)CC1 c1(C(N(CCC(=O)NC(C)CN2CCCC2=O)C)=O)cc2cc[nH]c2cn1 N12CCCC(CC1)C2=O.CCC(CN(CC)CC)CC CC1CC2(CC(C(=O)Nc3ccccc3)C2)C1.c1(CC=O)ccc2c(c1)CC2.N N1(C(C)=O)CCN(C(c2cc(C(C)(C)C)oc2C)=O)C2CCCCC2C1 C(=O)(CC(=O)OC)N(C(C(=O)NC(c1cnn(C)c1)CC)C1CC1)C CCC(C)CCCC(=O)N1CCCC(F)(C(=O)NC(CO)CCCO)C1 C1(NC(c2[nH]cc(C(N)=O)c2)=O)CN(C(=O)C2=CCC2)CCC1CO CC1CCN(C(=O)CC2(C)CC2)CC1C.C1(C=O)(C=O)CC1.C1CC1.N C1(C(C)(O)CNC(=O)CNC(N)=O)CCN(C(C2CCCCCC2)=O)CC1 c1(C(N2CC(NC(c3cnn(C)c3)=O)CC(C)C2)=O)cccc2c1NC(=O)C2=O N1(C(CCCNC(COC(CC)C)=O)=O)CCOC(C(=O)NC)C1 c1(C(N(C2CCN(c3nncs3)C2)C)=O)cc2ncccc2[nH]1 CC(=NOCC#N)C(=O)NCC(C)(C)C(=O)NCC1(C)CCOC1 C12(C(=O)NC(CC(=O)NC3CC(CC)OCC3)(C)C)CCCC1OCC2 Cc1cccc2c(C(=O)N(CCCN(C)C(c3nn[nH]c3Cl)=O)C)cnn12 CC1CC(C(=O)Nc2nc(Br)cn2C)N(Cc2cn[nH]c2)C1 C#CC1(NC2CSCCC2=O)CCOCC1 c1(OC)cc(CNc2cncc(C(=O)Nc3ccc(Cl)nc3Br)c2)c(Br)cn1 C1(O)(C(=O)NCC2OCCN(CC)C2)CCN(Cc2ccncc2Cl)CC1 Cc1ccc(S(=O)(=O)Nc2cnc(Cl)cc2C(=O)N=c2nc(C)[nH]s2)c(F)c1 C(CN=C(NCCc1ncc(Br)s1)NC1CC1)C1(CO)CCC1 Cc1ccc(O)c(C(N2CCCN(C(=O)CCc3cncs3)CC2)=O)c1 c1(C(N(C2CN(C(C3CC(N(C)C)C3)=O)C2)C)=O)ccnc2c(Br)cccc12 C1(C(=O)NC23CC(NC(c4cn(C)c(=O)cn4)=O)(C2)C3)CC2CCCCC2O1 S(=O)(=O)(c1cnc(N2CCOC(CF)C2)c(Cl)c1)N(CC=C)C1CC1 N1(C(C2C3(CC(NC(CCC#CC)=O)C3)C2)=O)CCC(C#CC)C1 N1(C(c2cc(C)ncc2)=O)CCCC12CCN(C(C1CC(S(N)(=O)=O)C1)=O)C2 CCC(C(=O)N1CCC(=CCNC(c2cnnc(C)c2)=O)CC1)C(F)(F)F Cc1ccn2c(C(=O)NCCC(C)N(C)C(c3ccc(N)c(N)n3)=O)cnc2c1 c1(CC(=O)NCC(C)C)cc(Cl)ccc1Cl.c1(C(=O)N)nc(C(C)C)ncc1Cl C(C(=O)N1CCC(C(N2CC=CC2C(=O)N(C)C)=O)O1)c1c(C)ocn1 N1(C(C2(OC)CCOCC2)=O)CC2CCC(C1)N2C(c1cc(C)oc1C)=O [nH]1ccc([N+](=O)[O-])n1.C1CCCCC1C(=O)N.S(=O)(=O)(C1CC1)NCC=O N1(C(CCC=CCC=C)=O)CCC(CN(C(C2CC(F)C2)=O)CC)CC1 c1(OC(C)C)ccccc1CC(=O)NC1CN(C(=O)CN2CCC(C)C2)CC1C Cc1c(C(=O)NCC(=O)NCCCOCCC)cccc1Cl.c1(C=O)csnn1 c1(NC(C(C=C)(C)C)=O)cc(OC)c(C(N)=O)cn1 c1(C(N(CC(O)CO)C(C)C)=O)cc(O)cc(Cl)c1Cl C(=O)(CC(C)C(C)C)N1C(Cn2cc(C3(COC)CCC3)nn2)CCC1 C12(NC(CCCCC#C)=O)CCCN(C(c3cccc(=O)o3)=O)CC1C2 C1(C2CCN(C(c3cc(Br)n[nH]3)=O)C2)(NC(c2nc(C(C)C)oc2)=O)CC1 CC1CN(C(C2CCC3(CC3)C2)=O)CCC1C(=O)NCC1CC2(CC2)C1 C(=O)(CCCS(C)(=O)=O)N1CCC(N(C(=O)COc2ccsn2)C)C1 C#CCCCCC(=O)NC12CCC1CN(C(=O)C(C)n1ccnc1)C2 C1(CNC(C(C)(F)F)=O)CN(C(=O)C(=O)Nc2c(F)cccc2F)CC1(C)C C1(NC(c2c(C)nc(CC(C)C)o2)=O)CCCCCC1.C1(C(=O)N)CC2(CC2)C1 c1(C(N2C(CCNC(C(C3CCC3)OC)=O)COCC2)=O)cc2c(ncn2C)[nH]1 N1(C(c2[nH]cc(C(C)=O)c2)=O)CCC(C(=O)NCC(C)(O)C(F)F)(CO)C1 C(=O)(CCCC(=O)N(C)C)NC(CC)CC(=O)Nc1cccnc1 Cc1nc2ccc(C(N3CCCC(C)C3CNC(c3ccncn3)=O)=O)cn2n1 N1(C(C2C(C)CC3CC3C2)=O)CCCC(CO)CC1.C(=O)(C(C)(C)S(C)(=O)=O)N c1(C(C)NC(C2CCCN(C(c3ccc(F)c(F)c3)=O)C2)=O)ccc(O)c(O)c1 C(C1=CCN(C(C2(C)C=CCCC2)=O)CC1)NC(CC1C(C)(C)C1)=O C(CCC)(CCCNC(=O)CCn1cccnc1=O)NC(C1C(=C)CC1)=O c1(OC)cc(C(N2CCC(CCNC(=O)CC3CCC(C)O3)CC2)=O)ncn1 c1c[nH]c2c(F)cccc12.C(=O)(CC1CCCC1)NCC=O.C(=O)OCC C1(NC(CC2CCN(c3ncc(C)cn3)C2)=O)CCc2cc(Br)ccc2O1 C1(C(N(c2ccccc2)CC)=O)CC(C)CN(C(c2coc(COC)n2)=O)C1 C1(NC(c2cnc(C(C)=O)s2)=O)CC2CCC1N(C(c1ccc(=O)n(C)c1)=O)C2 c1(N(CCC)CCNC(=O)C(C2CC2)O)cc(C)nc(C(C)(C)C)n1 C=CCC(CNC(c1cccc(CNC(=O)C(F)C(=O)O)n1)=O)CC(C)C CC1CC2(CCN(CC3CCC(C)(C)CC3)CC2)CN1C(C1CC12CC2)=O C1(C(N(CC(=O)N(CCCC)CCCC)CCC)=O)CCC(OC)C1 Cc1nn[nH]c1C(=O)N(CCC(=O)N1CCC1CC1CC1)C1CC1 CCC(C)(C(=O)N1CC(CCCCNC(c2ccn3ncnc3c2)=O)C1)C(N)=O c1(C(=O)NCCOCCN(C(c2ccc(C#C)o2)=O)C)nccc(F)c1Cl CCCCC(CNC(c1cc(C2CC2)[nH]n1)=O)NC(=O)C=C(C)c1ccco1 c1(OC)cc(C)c(CNC2CC(NC(C3(Br)CC3)=O)C2)cc1C(C)C N1(C(c2nc(OC)oc2)=O)CCC(CNC(=O)CC2COCCN2C)C12CC2 C1(C(=O)NCCN=c2nn[nH]n2-c2ccccc2)CC2C=CCC(C1)C2 C1(CC(=O)NCC=C=C)CC(C)N(C(=O)COc2ccsn2)C1 CCCCCC(C(=O)NC1CCC1NC(c1cccc(C(N)=O)n1)=O)C(C)C C(C(CCC)CCCC)NC(C1(C#C)CN(C(=O)COCC2CC2)C1)=O c1(CC)cccc(CC(=O)NC(C)CN(C(=O)CC2CCCC2)C)c1 CCCC(O)CC(=O)N(C1CCCN(C(c2c(N)cncc2Br)=O)C1)C C#CC1(NC(C2CC(NC(c3[nH]ccc3CC)=O)C2)=O)CC(F)(F)C1 N1(C(CC(C(CC)C)NC(=O)C(=CC2CCCC2)C)=O)CCn2ncc(O)c2C1 c1(C(=O)NCc2oc(C(NOCCOC)=O)c(C)n2)cc(F)ccc1O C(C)(CO)(C(C)(C)O)NC(C1C(NC(C(C(C)C)O)=O)COC1)=O C1N(C(=O)CC2CCCC2C)CCCC1(C)C.c1(OCC)cc(C(=O)N)[nH]n1.C N1(C(CC(C=C)CC)=O)CC2(CCN(C(C3(C)CC(CC(C)C)C(=O)O3)=O)CC2)C1 c1(C(N2CCC(CNC(CC=C)=O)(OC)C2)=O)noc2c1CCCCC2 N1(C(c2cc(C)on2)=O)CC(O)CCC1C(=O)N(C)C1CC1 C=CCCCCCCC(=O)N1CCC(NC(c2cc(Br)ccc2C)=O)C(F)C1 C1CCC(C)(C)CN1C(C12CC(F)(C1)C2)=O.CCC(C(=O)N)OC1CCCC1 Cc1ccc(O)c(CNC(C23CC2CCN3C(=O)CC2CCOC2C)=O)n1 n1(CC(=O)NCc2sc(C(=O)OCC)c(C)n2)nc(O)c2ccccc2c1=O c1(OCC(=O)NC)ccc(CNC(C2CC2(C)CC)=O)cc1 CCC(C#N)C(=O)NCC1CC1C(=O)NC(CCOC)C(N)=O C1(CCNC(C(C)(F)F)=O)CCCCN1C(c1ccnc(OC(F)F)c1)=O C1(C(N(CC(COC)O)C)=O)CCCN(C(=O)C(C)OCC2CC2)CC1 c1(NC(CC2CCN(C(c3scc(C)c3)=O)C2)=O)cc(C)c(F)cc1I c1(C(=O)NC(CCCC)CNC(c2ccon2)=O)ccc(C)c(Br)c1C C1CCOCC1.c1(C(C)N(C)C(C2CC2)=O)ccccc1.C(=O)(C)N.C1CC1 C1(NC(C2(CC#C)CC2)=O)CCOC(C2CCN(C(=O)C(C)(C)C)CC2)C1 C1(NC(CCCC)=O)CC2CN(C(c3cc(CN(C)C)c[nH]3)=O)CC2C1 C1(N(C(c2cc(COC)[nH]n2)=O)C)CCC(NC(c2ccncn2)=O)CC1 N1(C(CC(C)n2ccnc2)=O)CC2CCC1C(NC(c1cc3c(s1)CCC3)=O)C2 N1(C(CCSCCCC)=O)CCC(C2(O)CCN(C(C3CC=CCO3)=O)C2)CC1 c1(C(N2CC(CC=C)(NC(=O)CSCC(C)=O)C2)=O)cccc2cnnn12 C1(NC(c2cn(CC)nc2C)=O)CC(NC(c2ccno2)=O)C12CCC2.C C1(C(N2CC(C)(C)C(NC(c3cnsn3)=O)C2)=O)CC1C1(C)CCOCC1 C1(C(N(CC(COC)(F)F)C)=O)CCC12CCC2.C(=O)CCC1CC(C)C1.N c1(CC)cccc(C(=O)NC2CCC(CCNC(=O)C(Br)=C(C)C)C2)c1N c1(C(=O)NC(CNC(C2(CC)CCOCC2)=O)(C)C)cc(Cl)cc(Cl)c1 C1(OC)(OC)CCC1C(=O)N(C1CCN(C(C2CC(Cl)(Cl)C2)=O)C1)CCO C1(CC(N2CC(COC)(C)C2)=O)CCCC2(CCC2)O1.C(=O)(C(C)CO)N C1(NC(C(C)N(CCC)C(C2CCCC(=O)C2)=O)=O)CCNC(=O)CC1 c1cc(C(F)(F)F)ccc1Br.C(CCN)(C1CC1)NC(=O)OC(C)(C)C.C N1(C(C)=O)CCC(c2nc(-c3cccc(N(C)C)c3)n(C(C)C)n2)CC1 C=CC1(NC(c2cc(C(C)(C)C)n[nH]2)c2nnnn2C2CCC2)COC1 c1(NC(C2(CC=C)CC2)=O)ccc(NC(=O)CCCCC)cc1C.C(N)(=O)N C1(SC)CN(C(=O)C(C)N(CC(F)(F)F)C)CC1.c1(CCC(=O)N)ccncn1 C1(C=O)OC2CCC1CC2.C(CCC(=O)NC1(C)CCOC1)N(C(=O)OC)C.N c1(CNC(=NCc2nn(CC)nc2C)NC(C)C)c(OC)cccc1F c1(-n2c(-c3cscc3F)nc(CC(C)OC)n2)ccc(C)c(Cl)c1 C1(NC(C2CC=C(C)CC2)=O)CCC2(CC1)CN(C(c1nn(C)cc1C)=O)C2 CC1(C(=O)NCC2COCC2NC(=O)CCCNC(N)=O)CCCNC1=O n1(CCC(=O)NCCC(C)NC(C(C)N(C)C)=O)cnc2sccc2c1=O C(C(C)C(F)C(=O)NCCc1ccncc1C)NC(CCCOCC)=O C(=O)(C(C(C)C)N1CCCC1=O)NCC(CC)NC(C1(C)CCNC1=O)=O C1(C(=O)OC)C2CC1N(Cc1cccs1)C2C(=O)O c1(C(N2CCC(OCC(=O)N(CC3=CCSC3)C)C2)=O)cc(O)nc(O)n1 C(=O)(C(C)CS(C)(=O)=O)N(CCC(C(C)C)NC(c1cc2nccnc2[nH]1)=O)C C1(CNC(C2C(CC)C2)=O)CC2CC1CN2C(c1cc(C)nc(C)n1)=O C1(C(N(CCC(=O)N(CC#C)CCF)CC)=O)CC(=O)NC(=O)C1 Cc1cc(Cl)ccc1NC(C1CC1(C)C)=O.C12(C=O)C(=O)C3CC1C2C3.C c1(C(N2CC(NC(Cc3c(C)ncnc3C)=O)C(C)C2)=O)ccn2c1CCCC2 C1(NC(=O)Cn2cnnn2)CCN(C(c2cc(C3CCCCC3)[nH]n2)=O)CC1O n1(C(C)C)cc(C(=O)NC(C)CCCNC(=O)Cc2csc(Br)n2)nn1 N1(CC(=O)NC2C(CC(=O)NCC3CC3C=O)CCC2)CCSCC1.O Cc1nc(Cl)ccc1C(=O)NCC1(C)CCCN1C(=O)C(=O)C(C)(C)C C1(C(N(CCN(C(=O)CCc2ncno2)CC)CC)=O)CCc2n[nH]cc2C1 N1(C(Cc2c(C)noc2)=O)CCC(NC(C2CCC2)=O)C12CC2 c1(C(c2ccsc2)NC(=O)N(c2ccncn2)CCC2CC2)ccccn1 Cc1[nH]nc2ccc(NC(C3(C)CN(C(c4ccncc4Br)=O)C3)=O)cc12 C12(CNC(CCCC(=C)C)=O)CN(C(C3(OCC)CCSCC3)=O)CC1CCO2 C(=O)(C1CCCc2nncn21)NC1CC(CNC(c2n(CC)nc(C)c2)=O)C1 c1(OC(CCNC(C(C)O)=O)=O)cccc(C)c1.c1(OCC)cc(O)ncn1 Cc1cc(=O)c(C(=O)N(C(C)C2CC2)C)cn1C.C1(C(=O)N)CCOC(=O)CC1 c1(CC)cc(C(N2CCC(C)CC2CNC(=O)CC(C)SC)=O)ccc1Cl C1(OC)(CNC(c2nonc2CC)=O)CCN(C(C2CCS2(=O)=O)=O)C1 N1(C(Cc2cccc(C)c2Br)=O)CC2CN(C(C3CCOC3C)=O)CC2(C)C1 C(=O)(C(C(C)(C)C)NC(c1c[nH]c(C(N)=O)c1)=O)N1CC(c2n(C)cnn2)C1 Cn1cc(C(N)=O)cc1C(=O)N.C1CCN(C(=O)C)C1C1CC1.c1ccsn1 c1(NCC2C(C)(C)NC2)ccc2cnc(Cl)cc2c1 N1(C(Cc2c(C)non2)=O)CCCC(C)(CNC(C23CC2CCC3(F)F)=O)C1 C1CN(C(=O)C=Cc2sc(Cl)nc2Cl)CCC1.C(=O)CC1(CC=O)CC1.CC c1(C(C(=O)N)(F)F)ccc2c(c1)OCO2.C(=O)(C(C)OC)N(C(C)C)CC c1(C(C(=O)NC(C)C2CC2)NC(C(c2cnn(C)c2)C)=O)cccnc1 c1(C(N2CC(F)C2)=O)cc(C)c(N)cc1Cl.c1(CC)ccc(CC(=O)NC)cc1 CC1CN(C(C2C=CC(N)C2)=O)CCCN1C(=O)Cc1ccccc1 N1(C(C(C)=C2CC2)=O)CC2CCN(C(C3C4CCCCCC34)=O)CC2C1 c1(C(N2CCOC2=O)C)cn(CC2CCN2C(c2cc(C3CC3)on2)=O)nn1 C1(N(C(CC(CC)SC)=O)C)CCN(C(c2cc[nH]n2)=O)CC12CC2 N1(C(CN(C(=O)C(COC)CC)CCC)=O)CCCC(CC)(CC)C1 n1(CC)ncc2cc(C(=O)N)cnc12.C1CCN1C(C1CCC1C(F)(F)F)=O C(C(O)C(=O)NC(CNC(C1(O)CCC1)=O)C1CC1)OC c1(CNC2CCN(C(C34CC(C3)C4)=O)CC2F)cc([N+](=O)[O-])cc(O)c1O O=C1Cc2cc(NC(=O)Cc3cc(-c4ccc5nccn5c4)ccn3)cnc2N1 c1(C(N2CC(CN(C(=O)C3=CCCCO3)C)OCC2)=O)ccc(Cl)c(F)c1F c1(C(=O)NCCCNC(C2CC(CF)C2)=O)ccncc1C1CC1 CCC(C)C(C(=O)NCC1(C)CCOCC1)N(C(c1cn(C(C)C)cn1)=O)C Cc1ccc(OCCC(=O)NCC(CO)NC(C2(C)CCSCC2)=O)cc1 CC1(C#CC(=O)N2CCC3CN(C(=O)C=Cc4cncs4)CCC23)CCCO1 C1(CC(=O)N)COC(=O)N1.C(=O)(CCCc1ccsc1)N(C)CCOCC C(CC(=O)NCc1cncs1)(C(F)(F)F)NC(Cc1c(C)ccs1)=O C#Cc1ccc(C(=O)NC(CNC(c2nc(Cl)oc2C)=O)CC(F)(F)F)cc1 C(=O)(C(C)C(O)C(C)C)N1CC=CC(C(=O)NC(CCSCC)C)C1 C1(CNC(CC(CCC)C)=O)(CO)CC12CCN(C(C1(C(=O)N)CC1)=O)CC2 CC(C(=O)N1CCC(NC(=O)CN2CC=CC2)C1C(C)(C)C)C1=CCCC1 C1(C(N2CC(N(C)C(c3nnn4c3CCC4)=O)C2)=O)CCc2cnn(C)c2C1 c1(C(N2CCCC(F)(CNC(=O)CC3(O)CCC3)C2)=O)cc(F)cc(Cl)c1O C1(NC(=O)OCC)CCCN(C(=O)C(Cc2ccccc2)NC(C)=O)C1 c1(CC=O)ccccc1.c1(OCC)n[nH]cc1C(=O)NCCCC1CC1.N C1(CNC(C2CC(CC)C2)=O)CCC(C=O)CC1.C1CCCC1C(C)(C)C C1(C)(C(=O)NC(CC=C)C2CC2)CCCN1C(=O)Cc1ccc(O)nc1 c1(C(=O)NC2CCN(C(C#CC(=O)N(C)C)=O)C2)cc2ccncc2o1 c1(CC)nc(C(=O)NC(C)(C)CCC)c(C)o1.C1(C(C=O)O)CC(F)(F)C1 N1(C(c2cnc(C)[nH]c2=N)=O)CCC2CCCC12C(=O)NCCC(C)O Cc1oc(S(N)(=O)=O)cc1C(N1CCC(C)C1)=O.c1(C=O)cc(C(C)C)on1 CCCC(C)(C)C(=O)NC1CN(C(=O)Cc2cn(CC)nn2)CCC1C C(=O)(CCCCN=[N+]=[N-])NC1CC(C(=O)NC(CC(=O)NC)C2CC2)OCC1 CC1(C(=O)NCCC(=O)NCCC2CC=CCC2)CCCOC1 N1(C(C(CSC)O)=O)CCN(C(=O)C(C)(C)c2cnsc2)CC1CS(C)(=O)=O c1(C(N2CCC(NC(CN3CCC(=O)NC3=O)=O)CC2)=O)cccn2nnnc12 CCC(CC)(CCNC(C1(Cl)CC1)=O)NC(=O)Cc1ccsc1Cl C(=O)(C1=C(c2ccccc2)CCC1)NC1(CNC(Cc2cnc(C)o2)=O)CCC1 C(CCC(C(=O)N1CC(F)(F)C1C1CC1)NC(=O)COC)OC.C1CC1 C12(N(C(C)=O)Cc3ccccc3)CCCC1N(C(=O)CN1CCC(O)CC1)CC2 CC(C)(CCCC(=O)NCCN1CCC1)NC(=O)CCC(F)(F)F C(=O)(C(C)SC)NCC1(C(=O)NCCNC(=O)OCC)CC1 c1(CNC(C(CC2CN(C(C3(C)CC3)=O)C2)F)=O)cc(Cl)ccn1 c1(C(=O)NC2C(NC(C3(C)CC3)=O)C2)cccc([N+](=O)[O-])c1Cl C1(C(=O)NC)CCC(=O)C1.c1(CCC)nnnn1-c1ccccc1.CC(F)(F)F C#Cc1cccc(C(N2CCC3(C(=O)N=c4cc[nH][nH]4)CC3C2)=O)c1 c1(OC)cc(=NC(=O)C23CCCC2C(=O)C3)[nH]n1C C1(NC(C=CCOC)=O)CCCC(N(C)C(c2cc(CO)on2)=O)C1 CC(N=c1nc2c(ncn2C)c(NCC(C)F)[nH]1)c1nc2ccccc2[nH]1 CCC(C)C(C(=O)NC1CC(C2CCC2)C1)NC(=O)CCc1cnco1 Cc1conc1CC(=O)NC(C(=O)NC1C(O)CC1O)c1ccco1 C(CN=c1[nH]c(=N)[nH]c(=NC2CCC(C)(C)C(C)C2)[nH]1)c1nccc(COC)n1 c1(C(=O)NCC2(CNC(CNC=O)=O)CCCCC2)cnc2scnc2c1 C(C(CC(C)C)C(=O)N1CCC(COC)(NC(c2cccc(=O)n2C)=O)C1)OC N(C(=NCCC1(O)CCOC1)NC1CCOCC1)Cc1c(OCC#C)cccc1 C1(C(=O)O)CCCC(NCc2ccc(I)nc2)CC1 C=CCC(C)C(=O)N(CCN(C(=O)C(COC)OCC)CC)CC N1(C(C2(OC)CCSC2)=O)CC2CC2(C(=O)NCC2(O)CC(O)C2)C1 c1(CC(N2C(CN(C(C(C=CCCC)O)=O)C)CCC2)=O)n[nH]c2c1CCCC2 N1(C(c2nc(CC)oc2C)=O)CC(O)CCC1C(=O)N.c1(CC)cncc(C)n1 N1(C(C2CCC(C)C2)=O)CC(C)(C)CC1CNC(=O)C(C)c1cccs1 N1(C(CCC#CC)=O)C(C)CC2CN(C(=O)Cc3ccsn3)CC12 Cc1ccc(OCCC(=O)NC(C)(C)C)c(Cl)c1.c1(C=O)ccnn1CCF.N C12(NC(CN(C(c3ccc(C)o3)=O)C)=O)CCCCC1OCC2 C1(CC(=O)NCc2ccn(C(C)C)c2)C2CN(CCC3CC3)CC12 c1(C=O)c(F)cc(C(F)(F)F)cc1F.N1(C(CN(C)C(N)=O)=O)CC2CC2C1 CC1(C(=O)NC2CC3(CC3)C2)CCCN(C(=O)C(C2CCOCC2)F)C1 c1(C(=O)NCC2CCCC2)cc2n(n1)CC(F)C2.C1(C=O)CCCC12CC2.N N1(C(c2c(C)nc(Br)s2)=O)CCCN(CCN(C(=O)C(C)C#N)C(C)=O)CC1 c1(C(=O)NC(CC)CNC(c2csnn2)=O)ccnc(N2CCCCC2)n1 C(N=c1nc2ncn(C)c2c(NCC2CCCOC2C(C)(C)C)[nH]1)c1n(C)ccc1 n1(CCCCOCC)cc(C(=O)NC2CCCC2CO)cn1 C1(NC(C2CN(C(=O)C(O)C(F)(F)F)CCO2)=O)CCCC2(CCC2)C1 CC1CCN(Cc2ccc(CC#N)cc2)CC(C)O1 C1(CNC(C(COC)C)=O)CCN(C(=O)CCS(=O)(=O)N(C)C)CCC1(F)F c1(C(N2CC(NC(C(=C)F)=O)C(F)(F)C2)=O)cc(OC)c(O)c(O)c1 c1(C(N(C2CCN(C(Cn3c(CCC)ncc3)=O)C2)C)=O)cccc(OC)c1 Cn1cc2c(C(=O)C(C)(C)C)cccc2n1.C(=O)(CC(F)(F)F)N1CCCC1CC=O Cc1nnc2c(C(=O)NC3CCc4ccccc4C3)cccn12 CCCC(C)N(c1ccccc1)CC(=O)OC.c1(CC(=O)C(C)=O)nnc(C)s1 C(CC(C)C)(C(=O)NCC(C(C)C)NC(=O)CCN1CCOC1=O)OC C1(NC(c2sccc2C2CC2)=O)CCCCC1CNC(C1CCCO1)=O C(C(C)(C)C(=O)NC1CCCC(C(=O)NCC(F)(F)C(F)F)C1)OC C(C(=O)N1CCC(C)(NC(=O)Cc2[nH]cnc2C)C1)(C(C)C)OCC c1(C=O)cc(C(N)=O)cc(F)c1.C1(NC(C(C)OCC(C)C)=O)CCCC1 N1(C(C(C)(N(C)C(c2ccc(CO)cn2)=O)C2CC2)=O)CCOC2CCC12 C1(C)(CNC(CC2(OC)CC2)=O)CCN(C(=O)CCNc2ncccn2)C1 N1(C(C2(OC)CCOC2)=O)CCC(CN(C(=O)CSc2nccn2C)C)CC1 C(=O)(CC(C)(C)Cc1ccccc1)N1CCC(NC(Cc2cnc(C)s2)=O)C1 N1(C(CCCOCC#C)=O)CCC(C=O)(NC(=O)CN2CC3CC3C2)CC1.O c1(-n2c(C)nc(C(N3CCC4CC4C3)=O)n2)ccc(Cl)cc1Cl C1(NC(=O)CCF)C=CCN(C(C2CCN2C2CCCC2)=O)C1 c1(CC(C)C(N2CCCC2CN(c2ncncc2Cl)C)=O)ccccc1F c1(CCC(=O)OC)c[nH]c(C)c1NC(=O)CCNS(=O)(=O)C(F)(F)F C1(C(=O)NC2CC(C)N(C(=O)Cn3cnc(C#N)n3)CC2)CCc2nnnn2C1 CC1CCCCC1(CNC(=O)CC1(N(C)C)CCC1)NC(C1CCC1)=O c1(C(=O)CCCOC(=O)CC2CCC(=O)N2)ccccc1Cl C1(C(C(=O)NC2C(CNC(c3cc[nH]n3)=O)C2)O)CCCCCC1 Cc1nc(N2CCOCC2)sc1COC(=O)Cc1cncn1Cc1ccccc1 N(C1CCCCn2c(O)nnc21)C(=O)NC(CS(C)=O)C(C)(C)C c1(C=O)cccc2c1CC(=O)N2.c1(CC)ccc(C(N2CC(C)C2)=O)c(Cl)c1.N c1ccc(O)c(O)c1.c1(C(=O)NC2CCC(C(=O)N)C2)ccc(CCO)cc1.C C1(NC(c2c(CCC)nco2)=O)CCCC(NC(=O)C(C)C2(O)CCC2)C1 CN(S(=O)(=O)N1CCC(O)C12CCCC2)CC#N Cc1ccc(O)c(CC(=O)NCCCC(C)NC(c2occc2C)=O)c1 c1(SC)cc(C)ccc1C(N1CCCC1CNC(=O)Cc1ccncc1Cl)=O C(=O)(C1=C(C)OCCC1)N1C(CN(C(C=C(CCC)CCC)=O)CC)CCCC1 N1(C(C2C(C)CCC2)=O)CCCCC1CCNC(=O)COCc1ccncc1 N1(C(Cc2cn(CC)nn2)=O)CCN(C(c2ccc(OC)cc2C)=O)C(CF)C1 c1(C(N2CC(O)C2)=O)cnn(C)c1CF.c1(CCC(=O)NC)cnc(O)[nH]1 Cc1ccc(C)n1CC(=O)NCC(N1CCN(C(=O)NC2CC2F)CC1)=O c1(C=O)ncnc(C)c1C.C1(CC(=O)N(CC)CC2CCOC2)C=CCC1.N CC(C)CCN=C(NCCC1CC1C(F)F)NCC1CCCCO1.CF N1(C(c2scc(C)c2)=O)CCC(F)(C(N2CCCSCC2C)=O)CC1 C(=O)(CC(C(F)(F)F)NC(=O)C(C)C(F)F)NC(c1cc(C)no1)(C)C c1(C(N2C(CNC(CC(CC=C)(C)C)=O)CC2)=O)c(C)c2ccccc2oc1=O c1(C(=O)NCC(CN(C(Cc2c(C)ocn2)=O)C)O)c(F)cccc1Cl N1(C(CNC(=O)OCC)=O)CCOC(C)(C)C1.C1(Cl)(C=O)CC1(F)F.C c1(NC(C2NCCN(C(C3C=CC(=O)N=N3)=O)C2)=O)cc2ccccc2cn1 C1(C)(C(=O)NC2(C(=O)NCc3ncccc3Cl)C(C)(C)C2)CCCOC1 c1(C(=O)NCC(=C)CCNC(c2ncn(C(C)C)n2)=O)cc2nn[nH]c2cc1F C1(NC(c2cn(CCOC)nn2)=O)CCC2CN(C(c3cc[nH]c3)=O)CCC2C1 C(CC(C)C(=O)N1CCC(N(C(c2coc(Cl)n2)=O)CC2CC2)CC1)OC C=CC(CCC)CC(=O)NC(CO)C(=O)N(C)CC1C(C)(C)C1(C)C C1(C(=O)NC2CCC(NC(c3cc(C)[nH]c3)=O)CC2)CCc2nccn2C1 C1(NC(CNC(=O)C2CC2)=O)CC1C1CCN(C(c2cccc[n+]2[O-])=O)CC1 CCC(CC)C(C)C(=O)NC1CCC(NC(=O)CN2CCCC2=O)C1 CC1CCN(C(c2cc([N+](=O)[O-])sn2)=O)CCN1C(=O)C(O)CCN(C)C c1(C(=O)OCC)cnc(C)nc1N(CCCCNC(c1cncc(C)c1)=O)C C=CC1CN(C(=O)CC(C)C(F)F)CC1NC(c1c(C)cncc1C)=O N1(CC(=O)NCC2(F)CC(NC(CCCc3n(C)cnn3)=O)C2)CCOCC1=O N1(C(c2cncc(O)c2)=O)CC2(C1)CN(C(c1ccccc1C(F)F)=O)CCO2 c1(C(N(CC(CC)NC(C2CCCN2CCC(C)C)=O)CC)=O)cnnc(O)c1 N1(C(CCC2(C)CC2(F)F)=O)CCC2(CC1)CN(C(=O)Cc1ccns1)C2 C(=O)CC(C)(C)C(F)F.c1(OC)ccc(C(N2CCC(O)(CC)C2)=O)c(F)n1.N Cc1nc2cc(C(=O)N(CC(C)NC(=O)CC3NC(=O)NC3=O)C)cc(O)c2[nH]1 S(=O)(=O)(c1cc(Br)ccc1F)NC1CN(C)CC12CC2 c1(C2(C=O)CC2)ccccc1.C(C(=O)N)OCCOC.C1(CC)CC1.C Cc1nc2ccc(CN3CCc4c(ncn4C4CCC4)C3)cc2[nH]1 c1(C(=O)NC2(C(=O)NC)CC2)ccc2c(n1)CN(C(=O)C(C)N(C)C)CC2 C(CN=C(NCC1(C)CCCOC1)N1CCN(C2CCNC(=O)CC2)CC1)OC N1(C(C(CCC)NC(C2C(C)(C)C2(F)F)=O)=O)CC(F)CC(F)C1 CCCC(C(=O)NCC(C)(C)CN(C)C(c1ncccc1Cl)=O)N(C)C CCCCCC(O)C(=O)NCCCCC1CCN(C(=O)CN(C)C(C)=O)CC1 C(=O)C1=CC(C)(C)C1.c1(CC(=O)NCCCCN(CCC)C)ccc(O)cc1 C1(NC(c2c(OCC)scc2)=O)CCCC(N(C)C(c2cc(C)[nH]c2C)=O)C1 C1(C(=O)OC)CC2CC1CC2C(N1CCOCC1c1ccc(C(=O)O)o1)=O c1(NC(C2CCCC(n3ccnc3)C2)=O)cc(OC(F)F)cc(Br)c1 c1(CNC(CC)=O)cn(C2(NC(=O)C(C)(C)n3cnnn3)CSC2)nn1 C(=O)(CCN(OC)C(=O)C1CC(C)CN(C(=O)Cn2ccnn2)C1)OC N1(C(c2cnc(C3CCC3)[nH]2)C(=O)NCCCSC)CCCC(C(O)C(F)F)C1 Cc1ccc(C(=O)NCCC2CCCN(C(c3cnn(C)c3N)=O)C2)c(C)c1 C1(C(=O)NCc2n(C)ccn2)CCCCC1NC(c1cc[n+]([O-])cc1)=O c1(CC(=O)N(CCNC(C2(CC)CCCC2)=O)CCOC)ccncc1Cl CC(C)S(=O)(=O)C(C)C(=O)NC1(C)CCN(C(=O)CCc2ccnc(Cl)c2)CC1 c1(C(=O)NC2CCN(C(c3c(C)cnn3C)=O)C2)cc2nccn2c(O)n1 CCC(CC(=O)NC1CC2CN(C(c3cc4ccsc4s3)=O)CC2C1)C(C)(C)C C1(O)(C(N2C(C(=O)NCc3n(CC)c(O)nn3)CSC2)=O)CCOC1(C)C C1(C(=O)NC(C=C)(C)CC)CN(C(C2(CCC)CC(=O)C2)=O)CCN1C c1(NC(=O)C(=O)NC2CC2c2ccc(Cl)c(F)c2F)cnc(O)c2ccccc12 C12(CNC(C(CCC3CCC3)NC(C(CO)N(C)C)=O)=O)CCCC1CCC2 C1(C(N2CCCC(CNC(C(C)Cc3cccnc3)=O)C2)=O)CC(=O)NC(=O)N1 C(c1ccccc1)=C(C(N1CC(C(=O)OC)(NC)C1)=O)C C1(Nc2c(C)cncn2)CCCC12CCN(C(C1CC3CCC1O3)=O)CC2 C1(CNC(Cc2nc(C)[nH]n2)=O)CCC(C)CN1C(c1cccc(F)c1Cl)=O C1(NC(CCSc2n(C)nnn2)=O)CCCC(NC(C2CC(F)(CO)C2)=O)C1 S(=O)(=O)(c1cnc(N2CCC(SC)C2)c(Cl)c1)N(C)Cc1cccc(SC)c1 C(CC(C)(O)CNC(C1C(C)C1(C)C)=O)OC.C1(CC=O)COCCO1.N C(=O)(N=c1cc2ccccn2[nH]1)C1CCN(C(c2c(C)n[nH]c2)=O)C1C(C)C c1(OC)ccccc1SCC(=O)NC1CC(C)C1.c1(CC=O)ncn(C)c1C c1(C2(C(=O)N)CCC2)ccnc(Cl)c1.C1(OCC(=O)NC2CC2)CCCCC1 c1(C(=O)N)cccn2nnnc12.C(C)(C(C)C(C)C)NC(c1c(OC)n[nH]c1)=O N1(C(CN(C)CCO)=O)CCN(C(c2cnn(C)c2C#N)=O)CC1CCO C(c1ncccc1C)=CC=O.N1(C(C)=O)CSCC1C(=O)NC(C)C1CC1.N N1(CC=O)CCP(C)(=O)CC1.C1CCCC1O.C(=O)(C(=O)N)N(C)C1CC1 Nc1ncccc1C(=O)NC1CC1NC(=O)CSC(F)F N1(C(c2csnn2)=O)CCC2C(CCCN2C2CC2)C1 CN1CCN(C(=O)Cc2ncc(Br)s2)CC1c1cn(CC2CC2)nn1 C(=O)(C1=CCC2CCC1N2C(=O)CC1(O)CCOC1)N1C(COC)C(C)(C)C1 CC(F)(F)CC(=O)NCCC1CC(NC(c2[nH]ccc2-c2ccccc2)=O)C1 C1(CCNC(=O)CN2CCCCC2)CN(C(C2COC(=O)O2)=O)CCO1 Cc1cc(C(=O)NCC(C)N(C)C(C2(CC3CCC3)CC2)=O)ncc1N N1(C(C(C)OCCN(C)C)=O)CCC(C(C)NC(c2ccn(CCF)n2)=O)C1 c1(CCCOC)nc(C(C)CO)n(-c2ccncc2C)n1 C1COC(C)(C)CN1C(c1cnc(O)o1)=O.c1(SC)ccc(C=CC(=O)N)s1 c1(C(=O)NC2C(C)C2)cccc(S(=O)(=O)N2CCC(CN3CCCCC3)CC2)n1 C(CCC(C)C(=O)NC1CCCC1NC(=O)CCCSC)OC N1(C(C(F)OC)=O)CCC2C(C1)CN2C(=O)CNC(c1ccco1)=O C(c1ccc(Cl)cc1)=CC(=O)NC1CC(C)N(C(=O)CS)C1.CCC(F)(F)F N1(C(=O)Cn2ncnn2)CCC2(CCN(C(=O)C(O)CC3CCOCC3)C2)C1 c1(NC(CNC)=O)cc(C2(C)CC2)ccc1F.C1CCCN(C(=O)C2CC2)C1.C N1(C(c2c(-c3ccc(C)o3)onc2)=O)CCN(C(=O)CCS(C)=O)C(C(F)F)C1 N1(C(c2c(CC)n(C)cc2)=O)CC(NC(=O)C(C)c2ccsc2)CC2(CC2)C1 N1(C(Cc2c(C)ncs2)=O)CC2CCCCC2(CNC(=O)CCC2CC2)C1 Cc1ccc(C(=O)NC(C)(C)C(C)NC(C23COCC2C3(F)F)=O)nc1C c1(C(=O)NCCC(C)NC(c2c(CC)nc[nH]2)=O)cn2cnnc2cn1 Cc1ccc(NC(=O)C(C)C(C)NC(=O)CCCc2ncco2)cc1F C(=O)(CC(C(F)F)NC(=O)C=CC1CCCC1)N1CCN(C2(C)CC2)CC1 C1(C)(C(=O)NCCC2N(C(c3nnn(C)c3N)=O)CCCC2)CCCNS1(=O)=O C1(N(C(c2c(C)onc2)=O)CC2CN(C(=O)C(C)C)C2)CCC2CCC(=O)N12 N1(C(C(C(CC)O)C)=O)CC(C)N(C(=O)Cc2csnc2C)CC1C c1(C(N2CCCN(C(c3c(OCC)scc3)=O)CC2)=O)c(F)ccc(F)c1O C1(C=O)C2CCC3(COC(=O)C13)O2.CC(C)CC(C)CC(=O)NCCOCC C(=O)(C(=O)CC(C)C)N1CCC(C(C)NC(C2(CC)CCOCC2)=O)C1 C12(C(N3C(C)COCCC3)=O)CCCC1CCN2C(c1ccc(O)nn1)=O C1(CCNC(c2nc(C)sc2)c2nnnn2CC2CC2)COCC2(CCC2)O1 C(=O)(CCCCC(F)(F)F)N1CCC(CNC(c2c(N)c(Cl)cc(F)c2)=O)C1 C12(NC(c3cnc(Cl)s3)=O)CCC(C(=O)Nc3ccnc(Cl)c3)(CC1)CC2 C(=O)(CCC(CF)CF)N1C(CC(=O)NC2C(CC=C)CCC2)CCC1 O=C(C(F)C(F)(F)F)NCC1(O)CCN(C(c2scnc2Cl)=O)CC1 N1(c2ccc(ON3CC4CCCC(F)(F)C4C3)cc2)CCc2ccccc2CC1 C1(C(C)C)N(C(c2ccsc2Br)C(=O)NCc2ccco2)CC1(C)C O=S(=O)(c1nc(Br)cs1)Nc1ccc(-c2ccc(O)cc2)cc1 c1(OC)ccc(C(N2CC(C)C2)=O)c(Cl)c1.c1(C=O)cccnc1SC(F)F.N N1(C(C2(C=O)CC2)=O)CC(C=O)C(C)(C)C1.C1(C(C)O)CC(C)(C)C1.C C1(N(C(c2cc(C)no2)=O)CC)CCCN(C(c2cccnc2C(F)F)=O)CC1 c12ccc(cc1)c(=O)[nH]2.N1(C(=O)OC)CCC1CNC(C1CC1)=O.C c1(C(=O)NCC(C)NC(C2CC2c2cncn2C)=O)cnn(-c2ccccn2)c1 C(=O)C1=CC2(CCOC2)C1.Cc1cc(F)ccc1CC(=O)NCCC1(C)CC1 c1(CC)cc(C(=O)NCCCN(C(C2CCC(C)C2)=O)CC)ccc1F c1(C(=O)NC2(C3CCCN3C(=O)Cc3ncc[nH]3)CC2)ccc2cc[nH]c2c1 C=CCC(CC=C)C(=O)NCCOC1CCN(C(c2cc(C3CC3)sn2)=O)C1 NS(=O)(=O)CCC(=O)N1CCC(NCC2CCCOC2c2ncc[nH]2)C1 Cc1nc(-c2cccc(Cl)c2)sc1C(=O)Nc1ccc(OCCC(N)=O)cc1 N1(C(c2c(CC)cns2)=O)CCC2C(CCCN2C(c2ccncn2)=O)C1 N1(C(C=CC)=O)CCC2(CCC(NC(=O)CCc3cnc4ncccn34)C2)CC1 C1(CC)CN(C(C2CCCC(=O)N2C)=O)CCN1C(=O)CCC1CCN(C)CC1 N1(C(CC2(C)CC2)=O)CCN(C(C23CC2CCC3(F)F)=O)CC1c1cn[nH]c1 c1(-n2c(C(C)CO)nc(C(COC)OC)n2)nc2cc(F)c(F)cc2[nH]1 C1(CNC(C2CCS2(=O)=O)=O)CCCCN(C(c2ccc(Cl)c(Cl)c2)=O)C1 C1(NC(C)=O)CCC(C(=O)N)CC1.C1(O)(CC)CCN(C(c2ccccn2)=O)C1 C1(C(N)=O)CCCC(NC(=O)Nc2ncccc2C(F)F)C1 CC(C)CS(=O)(=O)CCC(=O)N1CC2CCC(C1)N2C(C1(C#N)CCOC1)=O C(=O)(C(CCCc1ccccc1)N(C)Cc1cc(Br)ccc1F)NCC C1(NC(C2(C)CCN(C(c3c(C)con3)=O)C2)=O)CC=C(C(C)C)CC1 C=C=CCCC(=O)NCC1CCCN1C(=O)Cc1nncs1 c1(-c2cn(CC=C)nc2)cnc2n[nH]c(C(N3CCC(C)(O)CC3)=O)c2c1 c1(C(C(=O)OC)NC(c2nccn2C)C)cccc(F)c1 N1(C(C(COC)(C)OC)=O)CCOCC(C)(CNC(=O)CCn2ccnc2)C1 C1(N(C(c2cc(C)ns2)=O)C)CCN(C(c2ccnn2CCN(C)C)=O)CC1C n1(CCC(=O)NCC(CCSC)(C)C)c(C)cc(O)cc1=O C12CC3CC(CC(C3)C1)C2.CC(CC(N)=O)C(=O)N.N(S(N)(=O)=O)CC=O N1(C(CC2C(C)=NNC2=O)=O)CCC(CC(=O)Nc2cc(C)ccc2O)C1(C)C c1(C(=O)NCC2(CNC(C3CCN(C)CC3)=O)CC2)ccnc2ccnn12 CN1CCC(N2CCN(C(C3(NC(c4cc[nH]n4)=O)CC3)=O)CC2)CC1 C1(NC(C(C)OCC2CCCO2)=O)CN(C(=O)C=CC2CCC2)CC1F C=C(Cl)CC(C(=O)Nc1cc(OC)cc(F)c1)NC(=O)C(CC1CC1)OC C1(NC(C2C(C=C)C2)=O)COC2(C1)CN(C(=O)C=CC(C)C)C2 O=C(C1=CCCC1)NC1CCC1NC(C1CCC(F)(F)C1)=O C1(CNC(C2CC(C)=C(C)CC2)=O)CCN(C(=O)CC2(C)CC2)C12CCC2 N1(C(Cc2c(C)nsc2)=O)CCOC2(CCCN(C(=O)C#CC3CCOC3)C2)C1 CCCCCCOCC(=O)NC(C)CC(C)NC(c1cccn1C1CCC1)=O C1(O)CCCN(C(=O)Cc2nc(C)no2)CC1.c1(COC)cc[nH]c1C(=O)N C1(C(=O)Nc2snc(C(=O)OCC)n2)OCCOC1(C)C N1(C(c2c(CC)con2)=O)CC2CC(C)N(C(C3CC(O)C(F)C3)=O)C2C1 N1(C(Cc2cc(C)sc2C)=O)CC(N(C(=O)Cc2c(Cl)cnn2C)C)C2(CC2)C1 Cc1nc(C2CC2)[nH]c1C(=O)NC1(C)CCC1.C(c1cnn(C)c1)=CC=O C(S(=O)C(C)C(=O)NCCO)c1c(C)nc(-c2ccccc2F)s1 c1(OC)cc(C(N2CC3OCC(NC(c4ccc(C)s4)=O)C3C2)=O)cc(Cl)c1O C(CC(=O)N=c1cc2ccccn2[nH]1)N(C)C(c1csnn1)=O N1(C(CC(N2CCCCC2=O)C)=O)CCCCC12CC(NC(=O)C(C)(C)C#N)C2 N1(C(c2cncc(C)n2)=O)CC(CNC(C23CCCC2C3)=O)CC(C)(C)C1 c1(C(N2CC=CC(NC(=O)C3CC3)C2)=O)cc(O)nc2ncccc12 C(c1cc(Br)cs1)=CC(N1CC(c2cn(CC(COC)O)nn2)(O)C1)=O c1(C(=O)NC2C(NC(=O)CCNC(c3cccs3)=O)CC2)ccnnc1 c1(C(NC(=NCC2CCOCC2)NCC(C)(F)F)C)ccc(F)cc1 c1cccc(Cl)c1Cl.c1(C2CC2)nccn1C.C(CNCCNC(=O)N)OC c1(C(C(=O)NCC)N(c2ccccc2)CC(C)(F)F)csc2ccc(C)cc12 c1(C(N2CC(O)(CCNC(=O)CCCF)C2)=O)cc2c(nc1O)CCSC2 CC(N=c1nc(N2CCC3(CCC3)C2)c2cc(F)cc(F)c2[nH]1)c1nc(O)n[nH]1 C(C(=O)N1OC2C=CC1CC2)C1C(NC(CC(C)C(C)(C)C)=O)CCCC1 CC1CC(NC(c2ccccc2-n2cnnn2)=O)CCN1C(=O)C1=CCCSC1 C1(NC(c2ccc3cc[nH]c3n2)=O)CCN(C(=O)CCOC2COC2)C12CCC2 O=C(C#CC1CCCOC1)NC1CCN(C(C2(CCF)CCOCC2)=O)C1 C1(NC(C2OCCN(C)C2)=O)CCC2(CCN(C(=O)COC(C)(C)C)C2)C1 N1(C(c2cccc(C)c2N)=O)CC2(CNC(=O)CCC3CCCO3)CC1CCO2 CC1CN(C(=O)CC2CCCOC2)CC1NC(c1ccnc(C2CC2)c1)=O C1(NC(C(C)OCC2CC2)=O)CCC2(CC1)CC2N=c1[nH]nc(C2CC2)s1 Cc1oc(Cl)nc1C(=O)NCC(CNC(=O)C(c1cncn1C)O)CO CCCCCCCCCC(C)CC(=O)NCCCNC(c1nncn1CC)=O C(=O)(CC1=CCN(C(=O)C(CN(C)C)N(C)C)CC1)N(CCC#C)C C1(NC(c2cc(C3CCOCC3)on2)=O)CC2CC1N(C(c1cscn1)=O)C2 c1(C(=O)NCC(C)NC(C2CCC2c2nc(S)n[nH]2)=O)cncc(N)n1 C1(CNC(C(C)C2CCCO2)=O)C(C)CCN1C(=O)C(c1cccc(F)c1)C Cc1ncc(C(=O)NC(CCN(C)C)C(=O)N2CCN(C)CC2)cc1C#N C1(C)(OC(=O)C2CC2)CC(F)(F)C1.c12cnc(s1)NC(=O)N2 N1(C(CC2OCCN(c3ccnc(SC)n3)C2)=O)CC2CCCC2C1 CC1(CCO)CCN(C(C23CC(CN2C(c2ocnc2C2CC2)=O)C3)=O)C1 C12CC(CO1)C2.C(CNC(c1cccn1C1CC1)=O)(C(=O)N)N(C)C.C c1(C=O)cnc2sc(C)cn12.N1(C(C23CC(OCC)C2C3)=O)CCCCC1C c1(C(N2CC3CC3C2)C(=O)NCc2cccc(OC)c2)cc2cc(C)ccc2s1 N1(C(C2CN(C(C)=O)C2)=O)CC(C)OC2(CCN(C(=O)Cc3csc(C)c3)C2)C1 C#CCCCC(C)C(=O)NCC1=CCN(C(C2CCOC2(C)C)=O)CC1 CCC1=NOC(C(=O)NC(C)CCCNC(c2ncc(CC)cn2)=O)C1 C12(C(=O)NCC(c3ncn(C)c3)O)CC3CC1C2C3.C12(C=O)CC1CNC2=O c1(C(=O)OC)c[nH]nc1NC(C1CC1C(=O)N)=O.c1ccnn1C(C)C N1(C(c2n[nH]c(C)c2F)=O)CC2CCC(C1)C(NC(=O)C(F)(F)C(C)O)C2 C(C(COC)C(=O)N1CC2CC2(CNC(C2(C(=O)O)CC2)=O)C1)OC C(=O)(C(O)C(C)(C)C)NC(C1CCCC1)CNC(C1(CC)CCCC1)=O c1(NC(C)=O)cccc(OCC(=O)NC(C)CN(C(=O)CC(C)F)C)c1 c1(C(=O)NC(C)CN(C)C(c2cn(CCCF)nn2)=O)cnn(CCO)c1N Cc1csc(=NCC(=O)N2CCC(O)(CCNC(=O)CN3CC4CCC3C4)C2)[nH]1 N1(C(C(C)OCC=C)=O)CCC2(CCCN2C(=O)CCCc2nc(C)cs2)CC1 c1(C=O)cc(C#N)c(C)cn1.C(=O)(CCC(=O)NC(C)C)N(CCC)CCC C1(NC(Cc2cc(C)nn2C)=O)CN(c2ncc(C)c(SC(C)C)n2)CCC1C O=C1CCN(CC2CC3CCC3C2)C(=O)N1CC1CCC12CCC2 C1(C(=O)NC2CN(C(c3c(C)nc(C)o3)=O)C(C)(C)C2)CCCCN(C)C1=O C1(NC(c2c(C)nc(O)cc2)=O)CC2CC1CN(C(=O)C(C1CC(F)(F)C1)O)C2 N1(C(C(c2ccnn2C)C)=O)CCC2(CCCN(C(=O)C=Cc3cncs3)C2)C1 C1(C(=O)OC)CC(C(N2CC(C)CC3(CC3)C2)=O)C12CCCC2 c1(-c2cn(CC(=O)NC3C(OCC)CCCC3)nn2)nc(C)ccc1F C(=O)(C(C)CC(C)C)NCC(CSC)(C)O.c1(C(=O)N)ccnn1C1CC1 C1(O)(CNC(C(C)NC(C)=O)=O)CCCN(C(c2cc(Cl)nnc2O)=O)C1 C(CCC(=O)NCC(C)(C)CN(C)C(C1CC1C)=O)OCCOC N1(C(C2ON=C(CC)C2)=O)CCC(C)C(C)C1.C(=O)C[SH](=O)=O.C(C)(C)C.N c1cc(F)ccc1F.O=C(COCCNC(=O)COCCCF)N.C1CC1 c1(SCC)ccc(Cl)cc1C(N1CC(CNC(C2COC(C)C2)=O)C1)=O C(=O)(C(C)(C)CN(C(=O)CC1CCOC1C)C)N1CC(F)(CC)C1 c1(C2C(C(N(CCC)C)=O)C2)cccc(C#N)c1.c1cc[nH]c1C=O.CO.C n1(CC(=C)C)nnnc1C(COC)(CC)NCCNC(N1CCOCC1)=O C(C(N)CC(F)(F)F)NC(CS(=O)(=O)NC)C C1(NC(c2cnn3ccccc23)=O)CCCCC12CCN(C(=O)C=C1CC1)C2 C1(C(N(C(CC#C)C)C)=O)(CNC(c2cccs2)=O)CC(C)(C)C1 C1(CCNC(COCCCCC)=O)C(C)CCCN1C(c1csc([N+](=O)[O-])c1)=O C1(NC(C(COC)C)=O)C(C)CCN(C(c2ccc(Cl)c(F)c2F)=O)C1C CC1=C(C(=O)NCC(N2CCN(C(=O)C(CO)N(C)C)CC2)C)SCCO1 N1(C(c2csc(C)c2N)=O)CCC(NC(=O)COCc2ccncc2)C12CCC2 C(=O)(C(C)(C)CC(F)(F)F)N1CC(C)CC(NC(c2c(C)ncnc2O)=O)C1 c1(C=O)ccc(C(C)=O)c(C)c1.c1(OCC)ccsc1C=O.C1CC(C)C1 c1(C(=O)NC(CN(C(CC2CC(OC)C2)=O)C)(C)C)csnc1Cl O=C(CCCCCCCBr)N1CCC(C(=O)N=c2nc[nH]s2)C1 C(CC(C)C(C)C)NC(CN(C1CC1)CC)=O.c1(CCC=O)c(C)noc1C c1(CC(=O)N(CCC)CCNC(=O)C(O)CN2CCCC2)ccccc1F.O Cc1nn(CC(=O)N)c(=O)o1.C1(CC)CCN(C(=O)Cc2cc(C)n(C)n2)CC1 C(N=c1nc(-c2ccccc2)nc(N2CCC(OC)CC2)[nH]1)c1n(CC)ccc1 C(=O)(C1CCN(C(c2cccc(CCO)c2)=O)c2ccc(Br)cc21)OC c1(OCCC)ccc(Br)cc1C(c1nnnn1CC)Nc1cnc(Cl)cc1C N1(C(CC(CC)C)=O)CCC(CO)C(NC(=O)CC(C)(C)CC)C1 c1(C(N2CC(c3cn(Cc4c(C)c[nH]n4)nn3)(O)C2)=O)cc(F)c(F)cc1F C1(F)(C=O)CC12CCCCC2.C(=O)(C(C)(C)C)N.C1(N(C(=O)C)C)CCC1 C1(C(N(C(C)CNC(=O)C(F)=C2CCC2)C)=O)C(F)(F)C12CC2 C(=O)(C(C)CC(F)(F)F)N1CCC(CNC(c2cc(C(C)=O)sc2)=O)CC1C c1(C(=O)NC(C#C)C)cc(CNC(c2cc(C3CC3)[nH]n2)=O)no1 C#Cc1ccc(C(=O)NC(C)(CNC(=O)CC23CCCC2C3)CO)c(O)c1 C1(C(CNC(c2c(COC)ccs2)=O)(C)O)CCN(C(c2nccn2C)=O)CC1 Cc1cc(C(=O)NCC2CCOC2)c(O)nc1C.n1(CC=O)ncn(C)c1=O.N C#CCCC(O)C(=O)N(C1CN(C(=O)CC(C2CC2)C2CC2)CCC1C)C c1(OC)ccn2ccnc2c1C(=O)NC1CCC1.C1(C=O)(C(N)=O)CCC1.N CC1COc2c(C(N3CC(NC(C4CCOCC4)=O)CC(F)C3)=O)cccc21 C1(CC(=O)NCCn2cnnc2C2CC2)CCC2COCCC2C1 Cc1oc(C(C)C)cc1C(=O)NC1CCC(C)C1.c1(C(=O)N)cnn(C)c1N CC(C)C(C)C(=O)N1CCC(CN(C)C(c2cccc(CO)c2)=O)C1 CCCCC(C)CCC(=O)NC(CNC(=O)Cc1cnc(C)s1)CCOC C1(O)(CNC(C=CC=CCC)=O)CN(C(c2cnc[nH]2)=O)C1 N1(C(c2c(C)noc2C(C)C)=O)CC2(CNC(C3CCCO3)=O)CC1CO2.C CC(C)CC(C(=O)N1CCCC1)ONC(=O)CCn1ccnn1 C1(CC)CN(C(=O)C(COC(C)C)NC(C2CC(C)C2)=O)CC(=O)N1 c1(C(=O)NCC2(O)CCCN(C(C(CSC)O)=O)C2)cc(F)cc(F)c1O c1(C(=O)NCC(CNC(CC(C)C)=O)F)cnc2c[nH]nc2c1 c1(NC(=O)NC2CCN(CC)C2=O)cc(C)c(NC(C)=O)cc1C C(=O)(C(=O)C(C)CC)N1C(C)(CC(N2CCN(C(CC)=O)CC2)=O)CC1 c1(OC)cc(CNC(=O)CCCn2cc(C)cn2)c(F)cc1Br CCC(CCC(=O)NCC1(OC)CCOC1)NC(c1cccc(=O)n1C)=O c1(-c2sc(C)c(C(=O)Nc3c(Br)ccnc3Cl)n2)cc(F)cc(F)c1 Cc1nc2c([nH]1)C(C(=O)N1CCCC1Cn1cncn1)CCC2 N1(C(c2[nH]cc(C)c2)=O)CCC2(CC1)COCCO2 c1(OC)ccc(F)cc1CNC=O.c12nc(n[nH]1)C2.c1ncc(C(N)=O)s1 C=CCC(CNC(C1CC(N(C)C)C1)=O)C(=O)N1CC2COCC2O1 c1(C=O)cc(C(C)=O)cn1C.C1(C(C(=O)NC2CCC2)OCC)CCOCC1 c1(C(=O)NC(C(C)NC(C(C)SC)=O)(C)C)cc2c(O)cccc2[nH]1 CCC(C(=O)NC(C)CCCNC(c1ccc(Cn2ccnn2)o1)=O)C(C)O CCCCC(F)C(=O)NCC(O)CC(N1CCN(CC)C(=O)C1)=O c1(C(=O)NC2(CO)CN(C(c3n(C)ncc3Cl)=O)C2)cccc2c1OCCCO2 c1(OC)cc(C)ccc1C(=O)NC1CN(C(C2CCCCN2C)=O)C1 N1(C(c2cnn(C)c2F)=O)CC(NC(c2cnn(C)c2)=O)C(C)(C)C1 Cc1nc(N2CCC(OCCNC(=O)C(C)C(C)O)C2)[nH]c(=N)n1 N1(C(Cc2cc(C)[nH]n2)=O)CCCC(C)(NC(=O)C(C)OCCC(C)C)C1 C1(C(N2C(C)CCC(NC(c3c(Cl)ccnc3F)=O)C2)=O)CCC(N=[N+]=[N-])CC1 CCCCC(=O)N1CCCCC1C1CC1.C1(CC=O)CS(=O)(=O)C1.C(C)=O.N N1(C(c2c(=N)[nH][nH]c2)=O)CCC2CCC(C1)N2C(=O)CCOc1cccnc1 N1(C(c2ccc(C)c(N)c2)=O)CC(C)CN(C(C2(C)CCOCC2)=O)CC1C C1(C(=O)NCC2C(C(=O)N3CC(O)CO3)CCO2)CCC(C2CC2)CC1 c1(C(=O)O)ccc([SH](=O)=O)c([N+](=O)[O-])c1.c1(C(c2nc(O)n[nH]2)N)ccccc1 C(=O)(C1CCCc2ccccc21)NC(CNC(=O)C=Cc1cccnc1)CO CCCC(C(=O)N1CC(NC(c2coc(C)n2)=O)C(CC2CC2)C1)OCC Cc1nnc(CCCC(=O)NC2(CO)CCN(C(=O)CCc3ccoc3)C2)n1C c1(C(=O)N)cc2n(n1)CC(F)C2.c1(CC=O)ccc(O)nc1.C(C)(CC)OC c1(C(=O)OCC)cc(=NC2CC3CC2CC3OC)[nH]c(CC)n1 CC1CCC(CCC(=O)NCCC(=O)NCc2cn(CC(=O)O)nn2)O1 c1(C(N2CCC(C(N3C(CN=[N+]=[N-])CC3)=O)(CF)C2)=O)ccn2ccnc2c1 N1(C(c2cccc(CC)n2)=O)CCC(C)(C)C(NC(=O)C(C)CN2CCCC2)C1 C1(OC)CC2CC(C(=O)NCC)CC12.c1(C(N(CCC)C)=O)csc(C)c1.O c1(CCNC(C(C)(C)C)c2nnnn2CCCF)ccc(Br)cc1 C(=O)(CC(O)C(C)C)N1CCC(N(C(CCC(=O)NCC)=O)CCOC)CC1 C(=O)(CCCCN(C)C)NCCC1N(C(c2nc(C(C)C)oc2)=O)CCC1 CCCCCCCCC(F)C(=O)NCCCCC1CN(C(C2CCOC2)=O)C1 c1(CC(=O)N(C2(C(N3C(C)CC3C)=O)CCC2)C2CC2)ccc(C#N)cc1 c1(CC)cccc(C(N2CCC(O)(CNC(c3ccnnc3O)=O)CC2)=O)c1O C1(CNC(=O)C(C2CC2)C2CC2)COCC2(CCNC2)O1 O=C(C1CCOc2c(F)cccc21)N(Cc1cccs1)CC1CCCO1 C(C)(CC(F)(F)F)NC(c1ncn(C(C)(C)C)n1)=O.C1(C)(C=O)CCOC1.N c1(CC(=O)NC2CCC(CNC(c3cncc(F)n3)=O)C2)csc2ccccc12 C1(C(=O)NC(c2scc(C)n2)C)C2CC3C(C2NC(=O)CC2=CCCC2)C13 N1(C(c2c(CNC(C(C)n3cnnn3)=O)cc[nH]2)=O)CCc2ccccc2C1 Cc1cc(N2CCCCC2c2cccnc2O)c2cccc([N+](=O)[O-])c2n1 C(C(C(=O)NC1CC1(F)F)NC(C1CCN(CC)C1)=O)SCC C1(C)(NC(c2ccc(CNC(Cc3c(C)ocn3)=O)o2)=O)CCOC1C C1(C(=O)OC(C)(C)C)CN(C=O)CC1C(F)(F)F.C1(C)(CC)CCCO1.N C#CCC(CC(=O)N(CCC)CCNC(C1CC1C(C)C)=O)c1ccccc1 CCC(C)C(C(=O)Nc1ccc(-c2ccc(C(C)=O)cc2)cc1F)OC CN=c1[nH]cc(C(=O)NCC2CN(C(C3CCCCN3C(C)=O)=O)CC2O)o1 N1(C(c2cc(COC)sc2)=O)CC(F)(F)CC1C.C1(F)(C=O)CCCC1.N Cc1ncnc(C)c1NC(=O)NCC1(F)CCOC1 c1(C=O)c(C)nn(C)c1C(F)(F)F.C1CCCCC1.C(CC(=O)N)=C(C)C.C CC(C)CC(CC(C)C)C(=O)N1CCOCC1CCNC(=O)C(O)P(C)(C)=O C(=O)(C(C)(C)C(C)C)NC(CCCC)CNC(c1cnc(CC(C)C)[nH]1)=O Cc1cccc(C)c1CC(N1CCCC(C)(NC(=O)Cc2c(C)cnn2C)C1)=O N1(C(C2(C)CN(C(c3c(C)snn3)=O)C(C)(C)C2)=O)CC(C)OC(C)(C)C1C C1(NC(c2c(C)oc(Br)c2)=O)COC2(C1)CN(C(=O)CC(C)(C)C)C2 CC1CCCN(C(=O)CC(O)C2CCCC2)C1CNC(c1c[nH]ccc1=N)=O C1(C(=O)Nc2c(CC)nsc2)CC12CCN(C(c1ccc(C#N)o1)=O)CC2 c1(CC2(C(=O)OC)CCN(c3nnc(CC4CCC4)n3C)C2)ccc(Cl)c(Cl)c1 CCC(C)(CO)C(=O)NCC(O)C.c1(C(=O)N)cc(=O)n(-c2ccc(Cl)cc2)[nH]1 C(C)(C)(C(C)CC(=O)N1CC(CS(C)=O)C1)NC(c1cnc(C)n1C)=O CC(CC(=O)N(Cc1ccccc1)Cc1ccco1)P(C)(C)=O N1(C(C(CC)N(C)C)=O)CC2CC(O)C1C2NC(C1(COC)CC1)=O S(=O)(=O)(c1ccc(N2CCCC(CO)CC2)c(Br)c1)N(CCC#N)CCC C1(CC(=O)N)CCN(CCF)CC1.C(C(O)C(=O)N1CC(O)(CC)C1)=CCCC C1(F)(CNC(c2ccc(CCC)[nH]2)=O)CCN(C(C2(CF)CCC2)=O)CC1 C1(NC(=O)CC(C(F)(F)F)c2ccon2)CN(C(=O)CC2CC2)CCC12CCC2 c1(C(N(CCC(N2CC(OC(=O)NC)C2)=O)CCO)=O)nc(C)sc1C c1(-c2nc(C)sc2)cccc(NC(=O)Nc2ccc(Oc3ccccc3)cn2)c1 C(N=c1nc2scnc2c(N(C)CCc2ccc(Cl)cc2)[nH]1)c1c(CC)n[nH]c1 c1(C(=O)NCCCCOC)cccnc1OCC(C)C.c1(C(=O)N)ccnn1C C1(NC(C(n2ccc(C)n2)C)=O)CCOCC1C(N1CC(O)C(O)C1)=O c1(C(c2n(CCOCC)nnn2)NC)cc(F)cc(C#N)c1.C1CC1(Cl)Cl CC(CCO)N=c1[nH]c(N(C)Cc2ccncn2)nc2ccc(Cl)cc12 C1(C2CN(C(C(C)CO)=O)C2)CN(C(=O)Cc2ccon2)CCO1 N1(C(C(CCSC)O)=O)CCCC2(NC(C3CC(O)CN3C(N)=O)=O)CC2C1 C1(C(=O)N)CCCC(=O)CC1.C1(OC)CC(C)N(C(C2CC2)=O)C1.N(C)C C(=O)(C(O)CC(F)F)Nc1cccc(CNC(c2c(C)cc(C)s2)=O)c1 CC1CN(C(c2ncccc2Cl)=O)CC(CCNC(c2ccc(F)cc2F)=O)O1 CC(CCCCNC(C1CC1c1cccnc1)=O)NC(=O)Cc1ccccc1F C1(C=O)CC(C)CC(=O)N1.C(=O)(CCC(=O)NCCOCC)OCC.N c1(C(N(CCCOCC)CC)=O)cc(F)c(F)c(F)c1F c1(C(=O)NC2(CC=C)CCCN(C(C3CC3CC)=O)C2)cc2ccccn2n1 c1(CO)n[nH]c2c1CCC2.N12CCC(CC1)C(=O)c1ccc(s1)C2=O Cc1cc(C(=O)N(CCC(=O)NC2CCCC(N3CCCC3)C2)C)n(C)n1 N1(C(c2cccc(CC)c2O)=O)CCC2(CCC2NC(=O)Cc2ccns2)CC1 c1(C(C(=O)NC2C(CNC(C(C)=CC)=O)C2)(C)C)cccc(C#N)c1 N1(C(C2C(C(=O)OCC)C2)=O)C(C(=O)NC2CC2(C)C)CC2CC12 Cc1cnsc1C(N1CC(O)(C(C)(C)CNC(=O)CCc2ccon2)C1)=O C(=O)(CC(O)C(C)CC)NC(CCC#C)C(=O)N1CCCC1CNC(N)=O C(CCC(C(=O)NC(C)CC(C)C)NC(=O)CCC(C)(C)OC)OC Cc1cc(Oc2ccccc2)ccc1NS(=O)(=O)Cc1ccc(C(=O)O)cc1F CC1ON=C(C(=O)N2CC3CC3(CNC(c3cn[nH]c3)=O)C2)C1C.C1CCC1.C N1(C(C2ON=C(CC)C2)=O)CCC(C)(C)C(C(N2CCC(CCN(C)C)C2)=O)C1 C1(CNC(CN(CCC)C)=O)CCC(C)CN1C(=O)Cc1cn(C)cn1 c1(C(=O)NCC(C)(C)CNC(=O)CCc2cccs2)ccccc1Cl C(N=c1[nH]c(=NCCc2ccsc2)[nH]c2c1CCCC2)c1c(C)ccs1 n1(CC)cc(C(=O)NC23CC2CN(C(=O)C=CC2CCCO2)C3)c(C)n1 N1(C(C2CC(=C)C2)=O)CCC(NC(C2CCN(CC(C)C)CC2)=O)C1C N1(C(C(C)SC(F)(F)F)=O)CC2CC(NC(=O)CSc3nncs3)C1C2 N1(C(C2CC(N(C(=O)C3=CCSC3)C)C2)=O)CC(O)C(C2CC2)C1 Cc1ccccc1C=CC(=O)NC(Cc1ccoc1)C(=O)NC1CC(C)(C)C1 N(C1COc2c(Cl)cccc21)C(C1CCC(n2cc(C3(C(=O)O)CC3)nn2)C1)=O C1(C(=O)NC(C)CN(C)C(c2cnns2)=O)(C(F)F)CCCO1 C=C=CC(C)C(=O)N(CC(C)NC(c1ccnn1CC#N)=O)C c1(C(=O)OC)c(C)ccnc1N1CC(NC(=O)OC(C)(C)C)CC(C)C1 N#Cc1ccc(C(=O)NCC2CCN2C(C2CCSC2)=O)nc1 N#Cc1cc(F)c(C(=O)NCC2CCCN(C(c3cccc(O)c3)=O)C2)c(Cl)c1 C1(=O)CCCCC(OC)ONC(=O)C2C(CC)CCN12.C#CCC(C(=O)NC)OC c1(NC(C2C(C)CCC2)=O)ccc2c(c1)CCN(Cc1ccc(C#N)nc1)C2 C(=O)(CCC(C)(C)[N+](=O)[O-])NC(CC(C)C)CC(=O)NC(C)CCC(C)(C)C C12(CNC(CCC(C)SC)=O)CCCC1N(C(=O)C#CC1CC1)CC2 Cc1oc(C)c(C(=O)NCC(C)CNC(C2COC(C)(C)C2)=O)c1C CC1(C)C(C(=O)NCCN2CCN(C(c3[nH]nnc3C3CC3)=O)CC2)C1(F)F Cc1nc(CCC(=O)NC2(CF)CCN(C(C3CCCN3N=O)=O)C2)oc1C C1(CNC(CC(CC)C2CCC2)=O)CC2CCC(C1)N2C(=O)C(F)=C(C)C C1(C(N2C(C)(COC)CC2)=O)CC2CCC1N2C(C1CC(=O)C12CCC2)=O C=CCC(CC)C(=O)N1CCOC(C(=O)NC(c2ncccc2C)C)CC1 C(=O)(C1=CCN(C(C2OCC3CCCC23)=O)CC1)N1C(C(=O)OC)CC1 C(=O)(C(C)(C)CC(C)(C)C)NCC1CCN(C(C2(C#C)CC2)=O)C1 C1(NC(C2N(CCC)CCCC2)=O)CC(OC)CN(C(c2nn(C)cc2C)=O)C1 C1(C(C)(C)C)COCCN1C(=O)CCCCNC(=O)Cc1nc[nH]n1 C1(CCNC(c2cc(CC)n(C)n2)=O)CN(C(=O)C)CCS1(=O)=O.C(C)CC N1(C(CC2(CC(=O)OC)CC2)=O)CCCCC1c1cccc(Cl)c1 C1(NC(Cn2c(C)ncc2)=O)CC(O)(C2CCN(C(=O)C=CC(C)C)CC2)C1 C1(OC)CCC(C(=O)NCC2CC2NC(=O)C(C)(C)n2ccnn2)CC1 C1(NC(C(CC)n2cccn2)=O)CC2CCC1N(C(=O)CC(C)COC)C2 c1(CNc2cncc(C(=O)NCc3ncccc3F)c2)c(O)cc(Cl)cc1Cl C#CC1CCC(CNC(=O)C(Cc2ccoc2)NC(=O)C(C)C#N)CC1 c1(C(=O)NCC(CNC(c2cnccc2C)=O)OC)cc2c([nH]1)CCC2 CC(C)CCC(O)C(=O)N1CC(NC(c2ccc(Cl)cc2Cl)=O)C1 N1(C(C(CC)SC)=O)CC2CC2(NC(c2cccc(N3CCCC3=O)c2)=O)C1 CC1CC2(C(=O)NCC3CCN3C(c3scnc3C(C)(C)C)=O)CC12 C1(C(=O)Nc2nc[nH]n2)CC2OCCC2N(C(c2cn3ccc(Cl)cc3n2)=O)C1 C(C1(C)CCC(C)C1(C)C)=CC(N1CCN(C(C(CC)OC)=O)C(C(C)C)C1)=O c1(C(N2CC(C)(CNC(=O)C(O)CC(N)=O)OCC2)=O)nc2cccnc2s1 C(=O)(CCCCCCCBr)N1CCCC(C(=O)Nc2nnc(C)n2C)CC1 C(CCCCNC(C1CN(C(N)=O)C1)=O)N(C)C(C1COCCO1)=O CC1(C)CCC=C1C(=O)NC1CCCC(NC(c2ccc(F)cc2O)=O)C1 c1(C(=O)NC(CC(=O)OC)C)cc(-c2ccc(CO)c(F)c2)cn2ccnc12 CCC(CC)C(C)C(=O)N1CC=CC(C(=O)NCc2ccccc2CO)C1 Cc1nc(N2CC(C)CN(C(C3CC(C)(F)C3)=O)CC2C)cc2nncn12 c1(C=O)c(C)coc1C(C)(C)C.N1(C(C2C(CC=C)C2)=O)CC(CCC)C1 C1(CCOC)COCCN1C(c1nc(Br)sc1C)C(=O)NCCC#N C1(NC(C(C)OCC=C)=O)CN(C(c2cncn2C)=O)CCC12CCC2 CC1CN(C(=O)CSCc2ccccc2)CC1.c1(C=O)cc(C(N)=O)no1.N C(=O)(C(C)(C)CCS(C)(=O)=O)N1CC(CNC(CCOC(C)=O)=O)OCC1 CC1(C)C(NC(=O)C(F)C2CCOC2)CCN1C(c1ccc(CCF)cc1)=O CC(C)C(F)(CNC(c1nccs1)=O)C(=O)NC(C1CCOC1)(C)C Cc1cc(NC2CC(F)(C)C2)n2nc(C)nc2n1.c1(C=O)ccc(=O)n(O)c1.N NC1CCOC(C2CCCN(Cc3c[nH]nc3C(F)(F)F)C2)C1 NC12CCC(C(=O)NCCCc3csnn3)(CC1)CC2 c12cnc(C)nc1NC2.C(C)(CCC1CC1(Cl)Cl)(c1nnnn1C1CC1)OC CC1CCN(C(=O)C=C2CCCC2)C1CNC(=O)CCCCF Cc1[nH]nc2c1CC(C(=O)NCC(CO)NC(=O)CS(=O)(=O)CC(C)C)CC2 c1(OC)cc(C=CC(=O)NC2COCC2n2ccnc2)cc(OC)c1OC Cc1ccccc1C(=O)NCC(N1CCC(CCNC(c2scnc2C)=O)C1)=O C1(NC(CCN(C(=O)CCc2cscn2)C)=O)COCC1C1CC1 N1(C(C(CC)O)=O)CCOC2(CCCN(C(=O)CSc3ncccn3)C2)C1 C1(C(N2CC(O)(CNC(Cc3cc(C)nn3C)=O)C2)=O)CC12CCOCC2 Cc1cc(CC(=O)NCC=C2CN(C(c3[nH]nnc3-c3ccccc3)=O)C2)on1 Cc1cc(=NCCOc2ccccc2Cl)[nH]c(N2CCC(CS(N)(=O)=O)C2)n1 O=[N+]([O-])c1cc(F)cc(S(=O)(=O)N2CCC3(CC2)OCCCO3)c1 S(=O)(=O)(c1cccc(=NCc2cn3c(n2)SCC3)[nH]1)NC(c1cc(Br)cs1)C c1(C(N2CCCC(NC(c3c(OC)ccs3)=O)C2)=O)cc(OC)c(OC)cc1.O c1(C=O)cc(F)cc(F)c1.c1(OC(C)C)cccc(C(=O)NC2CCCC2)n1.N Cc1noc2ncc(C(=O)NC(C)CNC(c3cnc(C(C)O)s3)=O)cc12 CC1OC2(C)CC1(C(=O)NCC(O)CN(C)C(C1CC1(F)F)=O)C2 n1(CC(=C)C)c(N2CCC(C(=O)NC)CC2)nnc1CSc1csc(C)n1 CC(C)(CC(=O)N1CC2CC1CN(C(c1cc(F)ccc1F)=O)C2)CC(F)F c1(C(N(CC)CC2CCCN(C(=O)Cn3cccn3)C2)=O)cccc2c1OCC2 N1(C(=O)CN2CCN(CCO)CC2)CCN(C(=O)C2=CCCSC2)C2(CCC2)C1 c1(N(C(=O)C(N2CCC(Cc3ccccc3)C2)=O)CC)c(C)cccc1C c1(CC(=O)NC2CN(C(=O)CN3CSCC3=O)CC2F)cccc(C(F)(F)F)n1 C1(C(=O)NCC(CNC(c2cc(C)c(O)nc2)=O)F)Cc2ccccc2O1 CCC(C(=O)N1CC(O)(C)C1)NC(C)=O.c1(C=O)cn(CC(O)CC)nn1.N c1(C(=O)NC2(C)CN(C(c3c[nH]c(=NC)s3)=O)C2)cnc2ccc(C)cn12 C1(C(N(C2CCC2)CC)=O)CCC2(CN(Cc3cc(Br)ccn3)C2)O1 C12(C=O)CC(CN1C(C1COCC1C(N)=O)=O)C2.CC1(C)CC(O)C1.C c1(-n2cc(CC3N(C(C4OCCN(CC)C4)=O)CCC3)nn2)ccc(F)c(C)c1 [N-]=[N+]=NCCC(=O)NCC1(C(=O)NCC2CCC(F)C2)CC1 CC1(C)CC(C(=O)NCC2CC(O)C2)O1.c1(C=O)scnc1C(F)F.C C(=O)(CC1C(=O)Nc2ccc(Cl)cc21)NCCSCCC=C CCCCCC(=O)NCC1CC(O)CN1C(c1cncc(C(F)F)c1)=O CCCC(CC(=O)NCC(C)(O)C1(C)CC1)NC(C1CC(=O)N(C)C1)=O C1(NC(C(C)NC(N)=O)=O)CCCCC1CNC(=O)CCc1ccccc1 C1(OC(CCS(=O)(=O)C(C)C)=O)CCC2(CC1)CN(C(=O)C1CC1)C2 N1(Cc2[nH]c(C(C)C)c(C(=O)N(C)C)c2)CCOC2CCCCC12 C1(C(=O)N)CC12CC(F)(F)C2.C1(NC(CC2(C#N)CCC2)=O)(C)CCCCC1 C(CCCC(=O)NC(CNC(=O)C(c1ccc(C2CC2)cc1)O)CO)OC N1(C(c2c(C)c(F)cnc2)=O)CC(C)C(NC(c2cscn2)=O)C(C)C1 N1(C(C(C(C)C)CNC(=O)C(F)CC(C)(C)C)=O)CCC2C(O)C(C)(C)C12 c1(CC(=O)NCCC(C)NC(C(c2cccnc2)OC)=O)ccc2nc[nH]c2c1 C(c1ccc(F)c(Cl)c1)=CC(=O)Nc1c(C)cc(Cl)cc1 CC(=O)CCN=C(NCc1cnc(C)o1)N1CCC(CF)C1 c1(OCC)ccc(OC)cc1.C1(N)CCN(C)CC1.O1NC(=N)CCNC(=O)C1 C1(CC(=O)NC2C(C)(C)CN(C(=O)C3=COCC3)C2)CCCCCC1(F)F C#CCCC(O)C(=O)NCC(CC=C)NC(=O)CCn1cc(Cl)cn1 N1(C(c2cc(O)cc(Cl)c2)=O)CCCC2(C1)CN(C(C1CCC13CCCO3)=O)C2 CC1CN(C(C2CN(C3CCC3)C2)=O)CC(C)N1C(C1CC2CCC(C1)S2)=O C(=O)(C(CO)C(C)(C)C)NC1CC(F)(CNC(c2cn(C)c(Br)c2)=O)C1 c1(C=O)ccc(C(F)F)c(F)c1.c1(CC)nc(C=O)c(C)o1.C1CC(C)C1.N N1(C(c2c(C)sc(O)n2)=O)CCN(C(=O)C(F)(F)C=Cc2ccccc2)CC(O)C1 N1(C(C2(CC)CN(C(=O)CCCCN=[N+]=[N-])C2)=O)CCn2nncc2C1 Cc1cc(C(N2CCCC(N(C)C(C3CC(N(C)C)C3)=O)CC2)=O)cc(C)c1O c1(C(=O)NC2C3CN(C(c4n(CC)cnn4)=O)C2C3)ccc2cc(C)ccc2n1 C1(C(=O)NC2C(CC=C)CCC2)CN(C(c2ncncc2C)=O)CC1(C)C c1(C(=O)NC(CCCCNC(C(C)C(F)F)=O)C)nnc(O)cc1O c1cccnc1.c1(C(N2CC(C(=O)OC)C2)=O)cn(C2(C(=O)O)CC2)nn1.O C=CC(C)(C)CC(=O)N1CCN(C(c2cnn(C)c2C)=O)CC1C(F)F c1(C(C(=O)NC(CC)C)N(C)CC)ccc(Oc2ccccn2)cc1.CCC(C)C C1(C)COCCN(C(=O)Cc2ccc(C(N)=O)cc2)C1.CC(C)C(F)C(=O)NC CS(=O)c1ccccc1C(N1CCC(n2cc(-c3cc(F)cc(Cl)c3)nn2)C1)=O N1(C(C2(CC)CCNC2=O)=O)CCC2(CC1)CN(C(=O)CC1CCC(F)(F)C1)C2 N(C(=NCCCCC(F)(F)F)N1CCC(CC(F)(F)F)C1)CCc1ccn(C)n1 c1(C(=O)NCC2=CCN(C(C3C(OC)C3)=O)CC2)ccc2cccnc2c1 C1(O)(CC(=O)NC(C(=O)N2CCCC2)C2CC2)CCOCC1 c1(C(N2CCC(CN(C(C(C)NS(C)(=O)=O)=O)C)C2)=O)occ2c1CCOC2 c1(C(=O)NC2CC(CNC(c3cc(CC)c(C)s3)=O)C2)ccc2scnc2c1 CC1(C)CCN(C(=O)C)C1.C(=O)(CC(F)(F)F)N.C(=O)CC.[SH](C)(=O)=O CCCCC(CN(C)C(C1(CC)CCCN1C(c1cccc(NC)n1)=O)=O)CC N1(CC(=O)N(C2CCN(C(=O)CC3CC3(Cl)Cl)C2)C)CSCC1=O CC1(C)CN(C(C2CCC3(CC2)CC3)=O)CC1NC(c1ccnc(CO)c1)=O CC1CN(C(=O)C(C)N(C(=O)CC2COCC(C)O2)C)CC1O C1(C)(NC(C(C(C)OC)NC(C2CC(=C)C2)=O)=O)CCC(=O)N(C)C1 C1(NC(Cc2cn(CC)nc2C)=O)CCC12CCN(C(c1ccnn1C)=O)CC2 N1(C(c2c(OC)ccs2)=O)CCN(C(=O)C2=CCC2)CC1c1cccc(OC)c1 Cc1ccc(C(C(=O)NC2COC2)N(C)Cc2occc2Br)cc1 N1(C(C(C)Cc2ccco2)=O)CCN(C(=O)CC(C)(F)F)C(C2CC2)C1 CC1C(NC(C2(C#N)CCC2)=O)CC2CCC1N2C(C1CC(N(C)C)C1)=O N1(Cc2ccc(C)o2)CCNCC1C(=O)N(CC(c1ccccc1)O)C Cc1cc(C(=O)NCC2(O)CCCN(C(c3cc(Cl)cn3C)=O)C2)ccc1C#N C1(CC(=O)NC2CCN(C(C34CC3COC4(C)C)=O)C2)CC(=O)NC(=O)C1 c1(C(=O)NC2CCN(C(C#CC(C)C)=O)C2)c(F)cc(C(F)(F)F)cc1F c1(OCCNC(=O)NCc2cnn(-c3ccccn3)c2)cccc2ccccc12 C(C(C(=O)NCc1ccnc(O)c1)C(C)C)NC(C1(CC)COC1)=O C(CC(C)(C)C(=O)NCCN(C(c1cc([N+](=O)[O-])n[nH]1)=O)C1CC1)OC N1(C(COC(c2c(Cl)cn(C)n2)=O)=O)CCC2CCCCC2C1 C(=O)(C(C)CC(C)(C)C)NCC(C)NC(=O)C(F)(F)c1ccncc1 c1(C(=O)NCC(C)NC(c2c(SC(C)C)nccc2)=O)ccc2nccn2c1 c1(C2(C)CC2)cn(CCCCNC(=O)N(C2CCOCC2)C2CCC2)nn1 C(CC)(C(=O)NC(C)(C(=O)NCCC(O)C1CC1)C1CCC1)=CCCC c1(C(N(CC(C)NC(C2(C(C)C)CC2)=O)C)=O)nn(C)c2c1C(O)CCC2 N1(Cc2c(OC)cc(F)cc2)CC2CCC(C1)C2NC(=O)CCc1ncc[nH]1 CC1CC(C(=O)NC2CC(NC(c3cccc(-n4nnnc4O)c3)=O)C2)CCS1 C1(NC(=O)N(CCO)Cc2ccccc2F)CC2CC1C(O)C2O N1(C(c2cccc(C)c2N)=O)CCN(C(C2(C(F)F)CCOCC2)=O)CC(O)C1 c1(C(N2CCC(C(C)(C)NC(C(CC(=C)C)OC)=O)C2)=O)cc2n(n1)CCCO2 C(=O)(C1OCCc2ccccc21)NCC(CC=C)NC(c1cnc(O)n1CC)=O c1(C(=O)NCC2CCN(C(C(C)C3CC3)=O)C23CC3)oc2ccccc2c1CO C=Cc1cnn(C)c1C(=O)NC(CN(C)C(c1c(C)ncnc1C)=O)CC Cc1cc(C#N)cc(C)c1C(N1C2CCC1CC2)=O.C1(C=O)CCS(=O)(=O)N1.N CC1CCN(C(c2ocnc2C(F)(F)F)=O)CCN1C(C1CSCCS1)=O c1(C(CC)C)nc(C)cc(=NC2CCCC(NC(c3cccc(=S)n3O)=O)C2)[nH]1 CCC(C)(C)CCCC(=O)NCC(C)N(C)C(c1ccccc1CC#N)=O C(CCN=C(NCCc1cn2c(n1)CCCC2)NCC(Cl)C(F)(F)F)OC(C)C C#CCC(C)(C(=O)N(C)Cc1cnn[nH]1)NC(=O)CCCOCC=C N1(C(CC=C(C)C)=O)CCC(NC(=O)Cc2cc(C)ccc2C)C1(C)C C1(CNC(CC(CC)OC)=O)CCN(C(=O)C=Cc2ccc(C)s2)C1(C)C N1(C(C(=O)NCC(=C)C)C2CC2(C)Br)Cc2ccc(Br)cc2CC1C C1CN(C(=O)CC2CC3CC3C2)CC(F)(F)C1.c1(OCC)ncc(C=O)s1.N C(C(F)(C(=O)NC1(CN(C)C)CCC1)C(C)C)NC(CC(C(C)C)C)=O C=CCCN=C(NCc1snnc1C)NCC(C)(C)C N1(C(C(COCC)C)=O)CC(C(=O)N(C)CC2CCOC2)C(F)(F)C1 C1(c2nnc(C)s2)CCN(C(=O)C(=O)NC(C(F)(F)F)C2CC2)CC1 C1(NC(C(CC)(C)COC)=O)CN(C(c2coc(Cl)n2)=O)C2(CCCCCC2)C1 C1(CNC(CCOCCCNC(CCCC)=O)=O)CCCCC1(C)C N1(C(COc2cc(C)on2)=O)CC2=C(C1)CN(C(c1ccc(C#N)[nH]1)=O)C2 c1cc(Cl)ccc1C.Cc1cc(C(=O)NC2CC2C(=O)NC)n(C2CCC2)n1 CC#CCCCC(=O)NC1(C)CC(NC(C2CC(=O)N(OC)C2)=O)C1 C(CCCCCCCO)NC(CC1CN(Cc2c(OC)ccc(Cl)c2)C1)=O c1(C(=O)NC(C2CN(C(C3(O)CCC3)=O)CCO2)C)cncc(C(N)=O)c1 C=C(C)CC(C(=O)NC)NC(=O)NOc1ccccc1 N1(C(CC2(C)CC2)=O)CC(NC(=O)C(F)CC2CCCCC2)C(S(C)(=O)=O)C1 Cc1ccc(CNC(=O)NC(c2cc(Br)cs2)C)o1 c1(C(c2n(C(CC)(C)C)nnn2)NCc2sccc2Br)cc(C(=O)O)c(C)o1 [N-]=[N+]=Nc1ccsc1C(=O)Nc1ccc(OCc2ccccc2)cc1O CCCCC(O)CCC(=O)N1CC(C(C)NC(=O)CC2CCC3CC3C2)C1 C1(C(=O)NCCCC2C(C)C2)(CCNC(=O)Cn2ccnn2)CCC1 C(=O)(C1CCCc2sc(=N)[nH]c21)N(CCNC(c1c(COC)scc1)=O)C C1(NC(C(SC)SC)=O)CC2CCCC(C1)N2C(=O)C(C)C(C)(C)C c1(OC)ccc(CCCC(=O)NC(CNC(=O)CNC=O)C(C)C)cc1OC C(CO)(CCCCNC(C1CN(C(C)C)CCO1)=O)NC(Cc1cnc(C)[nH]1)=O Cc1ccccc1C(=O)NC1(CCNC(c2sncc2C)=O)CCC1 Cc1nc(S(=O)(=O)NCCC=O)cn1C.C1(C)(C(N(CCC)C)=O)CC=CC1 Cc1ccn(CC(=O)N(C)CCOCCC(=O)N(C(C)(C)C)CCO)n1 C1(N(C(c2cc(OC)n[nH]2)=O)CC)CCCN(C(C2CC(C)=NO2)=O)C1 c1(C(=O)OC)cccnc1N(C)CCN(C)C(C)=O.C1CCC(C)O1 C=C1CCN(C(c2cc(C)cc(F)c2)=O)C(C(=O)NC2CCCC2CF)C1 C1(C(=O)NCC(CC)NC(C2(c3cncnc3)CCCC2)=O)CNC(=O)C1 N1(C(c2cc(CCC)[nH]n2)=O)CC(C)OC2(CCN(C(=O)CCOC(C)C)C2)C1 Cc1ccc([N+](=O)[O-])c(NC(=O)CC2CCCN2Cc2cc(F)c(F)cc2Br)n1 CCC(C)CCCCC(=O)N(C(C)CNC(=O)C#CC1CCCC1)C N1(C(C2(COC)CCCO2)=O)CCCC(C(=O)NCc2cc(Cl)no2)C1 C1(CN(C(Cc2ncc(C)[nH]2)=O)C)CCCN(C(=O)Cc2cccnc2O)C1 C(=O)(C(CC(F)F)C1CCC1)NCC(CNC(c1ccsc1C)=O)OC CCC(CCC(=O)N1CCOC(CN=[N+]=[N-])C1)NC(C1(C)CC=CC1)=O C1(NC(C(C2CCCCC2)C)=O)CCC(CC(=O)NCCC(C)(C)O)CC1 C(=O)(C(CC(F)F)C1CCC1)N1CCC(F)(CNC(=O)CCC2CCC2)C1 c1(C(C(=O)NCC2(O)CC(NC(COCC)=O)C2)CO)ccc(Cl)cc1 Cc1c(Br)c(C(=O)NC(CNC(c2coc(CO)c2)=O)C2CC2)nn1C N1(C(C23CCC(OC)C2C3)=O)CCCC(NC(c2cn3c(n2)CCC3)=O)C1C CC1CN(C(c2cnn[nH]2)=O)CCC1CNC(c1cc(F)ccc1F)=O Cc1cnc(NC(C2(C)CCCN2C(=O)Cc2cc(C)n(C)n2)=O)c(C)c1 Cc1cc(C(=O)NC(C)C(C)NC(c2cc(C(C)C)oc2C)=O)sc1Cl CC1CN(C(C2CC23CCC3)=O)CCN(C(=O)C(C)(C)O)C1 c1(C(c2ccc(Br)cc2)=O)cc(F)ccc1S(=O)(=O)N1C2CCCC1CC(F)(F)C2 C1(CNC(CCC#C)=O)CN(C(C2(C)CCCOC2)=O)CC1(C)C C=CCC(C)(C(=O)N1CC(CCn2cc(C(C)(C)O)nn2)C1)N(C)C c1(NCC(C)S(N)(=O)=O)nccc(=NCc2ncc(Br)cc2F)[nH]1 N1(C(C2(C)CC=CC2)=O)CC2CCC(CNC(=O)C(c3ccccc3)F)C2C1 c1(OC)ccc(C(N2CCCC(C(=O)NCCc3ccnnc3)C2)=O)cc1 Cc1cc(NC2(C)CC(C(=O)NC(C(C)C)C3CCC3)C2)ncn1 c1(OC)ccc(CC(=O)NC2CC(CNC(c3cnncc3O)=O)C(O)C2)cn1 CC1CCN(CC(N2CC(F)(C(N3CCOCC3C3(C)CC3)=O)C2)=O)CC1 CC1CN2CCN1C(C(N1CCC(N(C)C(c3cccn(C)c3=O)=O)C1)=O)C2 C1CCN(C(C2CCN(C(C)C)CC2)=O)CC1.C(C)(C(=O)NCC)=C(CC)C.C C1(C(C)(C)C)CCCN1C(c1cc[nH]n1)=O.c1(C(=O)N)csc(CC(F)(F)F)n1 CCC(C)(F)C(=O)NC1CC(CNC(=O)CCc2ccc(O)cc2)C1 C1(C(=O)NC(COC(C)=O)CO)OCCC1CNC(=O)Cn1ncnn1 c1(-c2nc(CN3CCC(CC(=O)OC)C3)on2)ccc2cnccc2c1 C=CCN=C(NCc1cccc(Cl)c1C)N1CC(C)N(C)C(C)C1 CC1C(NC(c2ccoc2Cl)=O)CCCN1C(c1cn(Cc2cccs2)nn1)=O n1(C(C)(C)C)cnc(=NC(=O)NCc2ncoc2C2CC2)[nH]1 CN=c1nc(N(CCS(N)(=O)=O)C)[nH]c(=NC(C)c2ccc(OC)cc2C)[nH]1 c1(C(=O)NCC(CNC(c2c(OC)nsc2)=O)(C)C)cccc(=S)n1O N1(C(C(C)=C(C)C)=O)CC(C2CCN(C(=O)CCOC(C)CC(C)C)CC2)C1 CC1CN(C(c2cnn3c2CCC3)=O)CCC1NC(c1ncc(C(F)F)s1)=O C1(NC(C2CC(CNC(C3CCC(=O)CC3)=O)OC2)=O)CCCCCC1CO c1(C=O)cc(C(F)(F)F)nn1C1CC1.CC(C)CNC(C1CCCS1)=O.N C1(C(=O)NCC(C(=O)NC2(C)CC(O)C2)(C)C)CCOCC1(C)C C1(NC(C2C(C(=O)OC)C2)=O)CCCCC1.C(=O)C(C)Cc1cnn(C)c1 C(=O)(CC(F)(F)F)NC1(C(N2CCC(Cc3cn(C)nc3)C2)=O)CCC1 C1(C(=O)NCC2CCCN(C(Cn3c(C)ncc3)=O)C2)CCS(=O)(=O)N1C N1(C(C(c2ccn(C)n2)C)=O)CCC2CCN(C(C3CCS(=O)(=O)N3)=O)CC12 N1(Cc2n(C)cnc2)Cc2ccccc2C1C(=O)Nc1cc(F)c2cc[nH]c2c1 C(=O)(CCCCCC#N)NC1CN(C(C2CC(C)OC(C)C2)=O)CC12CC2 CC1(C)CN(C(c2cccn(C(F)F)c2=O)=O)CCC1NC(=O)CC1C=CCC1 c1(N2CCC(COC)C2)nc(N2CCCC(F)C2)nc2ccsc12 C1(NC(CC(CC=C)NC(=O)CC2CCC(=O)C2)=O)CCn2cnnc2C1 C1(CNC(COCCCC)=O)CC(C)N(C(=O)C(c2ccc(F)cc2)=O)C1 C1(O)(CC(=O)N(C2CCCCC2)C)CCCCC1.C1(O)(C(=O)N)CC(C)(C)C1 c1(NC(CC#CC)C)ncc(S(=O)(=O)NCC2CCCCC(O)C2)cc1Cl CS(=O)C=CC(=O)NC1CN(C(c2cccc(-c3nc(O)n[nH]3)c2)=O)CC1O C(C)(CCC)NC(C(c1cnn(C)c1)OC)=O.c1(C=O)ccn(C2CCC2)n1.N C1(n2cc(C(C)(C)C)nn2)(C(=O)OC)CCN(C(C2(C)CCCCC2C)=O)CC1 Cc1cc(C=O)c(C)o1.C1(CC=O)CCCN1C=O.C1CC1.C(C)(C)C.N N1(C(C(Cc2ccccc2)N(C)C)=O)CC2CC1CC2(C)O CCCCCC(O)CNC(=O)CC(C(F)F)NC(=O)C(C1CCCCC1)O c1(C(C(=O)N(C)CCNC(=O)CCC2CCCOC2)CO)ccc(Cl)cc1 c1(C(=O)N)cncc(C2CC2)c1.C(=O)(C(F)(F)c1ccccn1)N(CC(O)C)C C(=O)(C1=CCN(C(c2cscc2OC)=O)C1)NC1(CCOC)CCCC1 c1(C(=O)NC2C(NC(=O)Cn3nccn3)CC2)ccc(-c2nc[nH]n2)nc1 N1(C(CCC(C)OC)=O)CCC(O)(CN(C)C(c2ccn(C3CC3)n2)=O)CC1 c1(C(=O)NCCCC(=O)N(CC(COC)O)C)ccc(O)nc1C C1(NC(c2cc(C(C)C)cc(F)c2)=O)CCCC12CCN(C(c1cccs1)=O)C2 Cc1nc(C2CCOC2)sc1C(=O)NCC(C)(C)NC(=O)C(O)CN(C)C C1(CC#C)(C(N2CC(CNC(c3ccc(Br)s3)=O)C2)=O)CC=CCC1 C(C)(C)(CCCCC(=O)NC(C1CCCN(C(c2ccncc2)=O)C1)C)OC CC1CCCN(C(=O)CNC(C2CCC2)=O)C1.c1(C2(C=O)CC2)nc[nH]n1.N C1(C(N2CCC(CC(C)NC(c3ccsc3)=O)CC2)=O)Cc2ccccc2O1 C1(c2cccnc2)(C=O)CC(F)(F)C1.c1(CC)scnc1C(=O)NC1CCC1 C(=O)C1=C(C2CC2)N(CCC2CC2)C(=O)NC1c1cc(C)c(I)cc1C.CC.O c1(C=O)cnc(C(C)(F)F)s1.c1(C2(C(N(CC)CC)=O)CC2)ccncc1 C(=O)(C(C(C)C)C(C)C)N(C(CCNC(c1cc(C)c(C)nn1)=O)C)C C1CCCCN1C(=O)C(Cc1ccsc1)NC=O.C(C(=O)NC)OCCOC C1CCN(C(=O)C=O)CC1.C1(CCOC)(C(=O)N)CC1.CC(F)F.C(C)C C1(C(=O)NC(C=C)(C)C)CC(O)CN1C(=O)CC1C=CCC1 N1(C(c2nnc(C)s2)C)CCCOC(CNC(c2cn(C3CCC3)nn2)=O)C1 CC1(C)CC(C(=O)NCCC(O)CNC(c2csc(-c3ccco3)n2)=O)=NO1 CC(=O)C(C)(C)CC(=O)N1CCCCC1CC(N1CCc2n[nH]cc2C1)=O CCCC(CNC(c1ccnc(O)c1F)=O)C(=O)NCC1(C)CCCOC1 c1(C(C)C)ccc2cc(C(=O)NC(CO)C(C)NC(=O)CO)[nH]c2c1.C1CC1 C1(O)(CC(C)C)CCN(C(=O)C(Cn2cccn2)NC(=O)Cc2cncn2C)C1 C1(CCCNC(C2(C)CC2)=O)CCCN1C(C1OCC1(C)C)=O c1(SC)cccnc1C(=O)NCCC1CC1.c1(C=O)coc(N(C)C)n1.C CC1CN(C(C2COC(=O)N2C)=O)CCCN1C(=O)C=Cc1cncnc1O c1(CC)ccc(N)c(C(N2CCCC(F)C2)=O)c1.C1(C=O)CC1C(F)(F)F.N n1(CC(=O)OCC)nccc1C(=O)NC1CCC1.c1(C=O)n[nH]cc1C.C C(=O)(CS(=O)(=O)CCO)NCCCCC1CCCN(C(c2ncc(N)nc2)=O)C1 C(=O)(C(F)C(=O)NC1CN(C(=O)CC2(N(C)C)CCCC2)CC1)OCC N1(CC(=O)NC(CCCC)CCC)CCC2(CCNCC2)C1 n1(CC(C)C)nc(CCOC(C)C)nc1-c1ccc(CO)cc1 C1(NC(c2ncc(C)cc2F)=O)CCC(O)CN(C(=O)C(=O)N)C1.CC(F)(F)F Cc1[nH]cc(C(=O)NCC2(C)CCCN2C(=O)C(C#N)C(C)(C)C)c(=O)c1Cl N1(C(C(C(=O)OCC)O)=O)CC(C)N(C(c2ccc([N+](=O)[O-])o2)=O)C(C)C1 S(=O)(=O)(c1ccccc1Cl)NC(C1CC(Nc2cc(N(C)C)ncn2)C1)=O C(=O)(C(C)(CNC(=O)CCCCCNC(N)=O)CC)NCCC N1(C(C(CC)CCOC)=O)Cc2nncn2C(C)C1 C=CC(C)(O)CC(=O)NCc1cn(C2(C)CCN(c3ccc(Cl)cc3)CC2)nn1 CCC(CC(=O)NC(CC(=O)NCC(C)CCCO)C(F)F)C(F)F N1(C(c2cccc(NC)n2)=O)CCC(C)CC1C.C1(C(=O)N)CC1C(C)(C)O C1(C(=O)Nc2c(OC)nc(C)cn2)CCCC12CCN(Cc1cnn(C)c1)C2 Cc1n[nH]c(C)c1CC(=O)NC(C1CCN(Cc2ccc(N(C)C)cc2)CC1)C N1(C(C(n2cc(-c3cnc(C4CC4)o3)nn2)C)=O)CCCCC(CO)C1 O=C(C1=CC2(CCOC2)C1)NC1CCCN(C(=O)CC2(O)CCCCCC2)C1 CC(CC(=O)N1CC=CC(NC(c2cnn3c2CCCC3)=O)C1)C(F)(F)F C1(NC(CSCC)=O)CCCC2CN(C(c3c(F)cccc3F)=O)CC12 CCCC(C(=O)NC(C)(CC)CCO)NC(C1CC(N(C)C)C1)=O N1(C(C2(N(C)C)CCCCC2)=O)CCCCC(NC(C2CC(C)(C)C2)=O)C1 C(C1=CCN(C(c2ccc(=O)oc2)=O)CC1)NC(C1C(CC(C)C)C1)=O N1(C(=O)Nc2cn(CCN(C)C)nc2)CC2CC(C(F)(F)F)C2C1 c1(C=O)cc(C)c(F)cn1.N1(C(CCOCCOC)=O)CCC(CO)(C)C1.N CCC(CC(C)C)C(=O)NC(C(=O)NC(C(=O)OC)C1(C)CC1)C(C)C C1(NC(C2C(C)CC(=O)NC2)=O)CCCC2CN(C(C3CCC3)=O)CC12 Cc1cc(C#N)c(O)nc1C(=O)NCC1CCCCN1C(C1CNC(=O)N1C)=O c1(CNC(=O)C=Cc2cc[nH]c2)cccc(C(=O)NCC2CCSC2)n1 CCCCC(CNC(=O)C(n1nccc1C)C)NC(=O)CCCN(C)C(C)C c1(C(=O)OC)cncc(C(=O)NC(CC)(CO)CO)n1 C1(C(N(CCC)C(C)C)=O)CN(C(=O)CCC2CCOC2)CC1(C)C C1(C)(CC(=O)NCC(C)CNC(c2cc(C3CCC3)[nH]n2)=O)CC1(F)F c1(SCNC(C(C2CC=CCC2)N(CCN(C)C)CC)=O)ccccc1F.C1CC1 Cn1ccnc1C(C1CC1)OCC(=O)N.c1ncoc1C1CN(c2nncs2)C1 c1(C(N(CC(C)NC(c2cccnc2O)=O)C)=O)ccc(CN=[N+]=[N-])cc1 c1(C(N2CCC(NC(C3OCCN(C)C3=O)=O)C(O)C2)=O)ccc2cnnn2c1 c1(C=O)c[nH]c(=O)c2ccnn12.c1(C(=O)OC)cc(C(=O)NCC(O)C)no1 c1(C(C(N2CC(CC(C)NC(c3cnsc3)=O)C2)=O)C)ccc(F)c(Cl)c1 C(C(CO)N=c1[nH]nc(C2CCCC2)s1)NC(C1(NC(=O)NC)CCCC1)=O C1(C(N(C2CCCCC2)CC#C)=O)C(O)CCN1C(=O)CCSCCCC C(=O)(CN1C(=O)COc2ccccc21)NC1(C)CCN(C(c2c(C)cc[nH]2)=O)C1 CC1CN(C(c2c[nH]nc2-c2ccnn2C)=O)CC1NC(=O)CC1CC1(C)C c1(NC(=O)CNCCOc2nsnc2N2CCOCC2)nc2c(s1)CCC2 N1(C(=O)Cc2ccc(Cl)cn2)CCN(C(=O)CCN(CCCl)CCF)C(CO)C1 C(=O)(C(CC(C)(C)C)NC(=O)C(O)C(F)(F)F)N1CC(N(C)C)C(F)C1 C(C(CC(=O)NCc1cnn[nH]1)C1CCC1)NC(C1(C#C)CC1)=O C(=O)(C#CC1CCCC1)N1CCN(CC(C)NC(=O)CCCSC(C)(C)C)CC1 CC1CCN(C(C2CCCC3(CCC3)C2)=O)CCN1C(C1CCCC1)=O c1(C(N2CC(OC)C(NC(=O)CC(O)C3CCCC3)C2)=O)cc(C)cc(Cl)c1N c1(C(N2CC(c3cnnn3C)(OC)C2)=O)cc(C)nn1Cc1ccccc1 n1(CC)cnc2nc(=NCCC3(CSC)CC3)[nH]c(NCC3CNC(=O)C3)c12 N1(C(CN(CC)CC)=O)CC2(CCC2)CC1C(=O)NC1(C)CCCCCC1 Cc1ccc(C(=O)NC(CNC(=O)Cc2ccccc2)CO)n1C.C(C)(C)O CC1OCCC1C(=O)NC1(CNC(=O)C(C)(C)c2cncs2)CC1 c1(C=O)c[nH]c2nccc(Cl)c12.N1(C(CC(=O)OCC)=O)CCN(C)C(C)C1.N C1(C(N(C)CP(C)(C)=O)C(=O)NC(C(=O)OC)C)CCCCC1C C[n+]1ccn(CC(=O)NCC2CN(C(=O)C)C2)c1.n1(CC(=O)N)cncn1 c1(C(=O)NCCCCCNC(C(COC)OC)=O)cnn(C2CC2)c1Cl CC(C)CCC(C(=O)N1CCC2(C=CCO2)C1)NC(C1CCC2(CC2)C1)=O C(CC)(C(=O)N1CCC(CC)C1)=CC.c1(CC(=O)N)cc(-c2ccccc2)on1 c1(NC(C)(C)CCNC(=O)C2=CCCC2)nc2ccc(Cl)cc2s1 C1(NC(C(CC)(C)C)=O)CCCN(C(=O)C(C)CC2CC2)C1C C(C1CCCN1C(=O)C(=O)NCC(F)F)=CC(=O)NCC(C)(C)CO c1(NCC2CCCN(C(C3(OC)CCC3)=O)C2)ncc(C)c(SC(C)C)n1 c1(N(C)C)cccc(NC(=O)CN(C(=O)CC2CC=CCN2C)C2CC2)c1 C(=O)(C(C)(C)C=O)NC.C(=O)CC(c1ccccc1)N(C)C.CC=CC.N C1(CC)(NC(c2cnsn2)=O)CCN(C(C)=O)C1 CC1CCC(NC(=O)Cc2ccsc2)CN1C(=O)CCc1ccc(N)cn1 Cc1ccccc1CC(C)C(=O)NC1CC(CCNC(c2csnc2Cl)=O)C1 S(=O)(=O)(C1CCC(C)(C)C1)NC(c1cccs1)CC C(=O)(CC(C)(C)NC(=O)C(F)C1CC(NC(c2cnsn2)=O)C1)NC c1(C(N2CCC(NC(=O)COCC3CCCO3)CC2)=O)cccc2cc[nH]c12 N1(C(C(C)Cc2ccccc2)=O)CCOC2(C1)CN(C(c1cnn(C)c1)=O)C2 CC#CCCC(=O)N1CC(NC(=O)C(C)NC(C)(C)CC)C(C)C1 c1(C=O)cc(F)c(F)cc1C(F)(F)F.CC1(C(=O)NC2CCC2)CCCO1.N c1cc(F)cc(Cl)c1.c1(CC)conc1C(=O)NCCCNC(=O)CCS CCCCC(CC)CC(=O)NC1C=CCN(C(c2cc(COC)no2)=O)C1 c1(C(N2CCN(C(CC=C)=O)C(C3CCCC3)C2)=O)ccc([N+](=O)[O-])cc1C C1(CC(=O)NCC2(C=C)CCCC2)CN(C(=O)Cn2cnnn2)CC12CC2 Cc1cc(C(N2CC(C(=O)NCC3CC(O)C(O)C3)CC2(C)C)=O)ccc1C#N Cc1cccc(C(N2CCCC(CCCCNC(=O)C3=CCOC3)C2)=O)c1 n1(CC(=O)O)ccc2c(C(=O)NCCCn3cc(CO)nn3)ncnc12 C1(CCC(=O)N)CCC(=O)NC1.C1(F)(CNC(C=CC)=O)CC(C)C1 S(=O)(=O)(C1CCCN(C(=O)OC(C)(C)C)C1)Nc1c(C)cc(F)cc1 C1(CNC(C(C(C)O)N(C)C)=O)C(O)C(O)CN1C(=O)Cn1cnc(Br)c1 C1(NC(c2cc(C(N)=O)[nH]n2)=O)CN(c2ncc(Cl)cn2)Cc2nccn2C1 C1(NC(C=C(C)c2ccsc2)=O)CC2CC1N(C(C1CC3(CC3)C1)=O)C2 CCCC(CC)C(=O)NCC1CC(F)(C)C1.c1(C(=O)N)csc(C(N)=O)n1 C12(C(N(C3CCN(C(C(C)SC)=O)CC3)C)=O)CCC(C)(CC1)OC2(C)C n1(CC(N2CCC(N(C(C=Cc3occ(C)n3)=O)C)C2)=O)nnc2ccccc12 c1(C(N2CCC(n3cc(Cl)cn3)CC2)=O)c(Cl)cc([N+](=O)[O-])cc1Cl Cc1cccn2c(COC(=O)C(c3cccc(Br)c3Cl)(F)F)cnc12 CC(C)CC(C(=O)NC1CCC2(CC2)C1)N(C(=O)CC1CCC2CC12)C O=C1CC(CC(N2CCC(OCCNC(c3cccc(F)n3)=O)C2)=O)C(=O)N1 c1(C(=O)NCC2(C)CCCC2)cccc2cc[nH]c12.N(S(N)(=O)=O)CC=O.N C12(NC(CS(CCC)(=O)=O)=O)CCCCC1N(C(=O)Cc1cnc[nH]1)CC2 C(CCCS(C)=O)NC(CONC(CC1C(C)OCC1)=O)=O N1(C(C2(COC)CC2)=O)CC2CCC2(CCNC(c2ccnn2C)=O)C1.S c1(OCCOC)cccc(C=CC=O)c1.C1(CCC)CN(C(=O)C)C1.N c1(C(N2CC3CCN(C(C(C(C)C)O)=O)C3C2)=O)ccc2nc(Cl)sc2c1 CC1(C)CN(C(C2CCN(CCF)CC2)=O)CCC1NC(=O)CCSC(F)(F)F n1(C(C)C)cc2c(n1)C(C(=O)NCCC(C)(C)C)CCC2 C1(C(=O)NC(c2ccc(C)cn2)C)CCCCCCN1C(C1CC(F)(F)C1)=O C(=O)(C1Cc2ccc(F)cc21)NC1C(C)CCN(c2ncc3c(n2)CCOC3)C1 c1(C=O)nn(C(C)(C)C)cc1Br.C(=O)(C(OC)OC)N(C(C)C)CC.N C(=O)(C1=COCCC1)N1CCC(NC(c2ncn(C(C)C)n2)=O)(CF)C1 c1(C2OCCN(CC)C2)ccc(F)c(F)c1.c12cccc(c1)Cn1ccnc1-2 CCCCC(F)C(=O)NC1CCOC1C(N1CCC(C(C)(C)C)C1)=O C1(CC(=O)NCC2CC2CNC(c2nccs2)=O)CCC2(CCC2)CO1 C=CCC(CCCCC)C(=O)NCC(C)N(C(=O)C(C)=Cn1ccnn1)C Cc1cc(NC(C2CC=CCC2NC(C2CCCC2)=O)=O)cc(Cl)c1 N1(C(Cc2c(C)cccc2)=O)CCCC2(CCCCN2C(c2[nH]cnc2C)=O)C1 N1(C(C(C(C)(C)C)O)=O)CCCC(C2CCN(C(=O)C=Cc3cncs3)C2)C1 C1(C(=O)NC(C)Cn2ccnc2)CCCCCCN1C(=O)CN1CCCCC1 n1(CC(=O)NCCNC(c2coc(Cn3cccn3)c2)=O)cnc2c1CCCC2 CC#CCC(C(=O)N1CC2CC1CS2=O)NC(=O)Cc1cnsc1 c1(OC)ccccc1CC(C)CC(=O)NCCCN(C)C(C1CC12CC2)=O C1(CC)CC(F)(F)CN1C(c1nnc(Cl)cc1N)=O.C(C)(C=O)OCCC=C.N c1(NC(C2(C)CN(C(=O)COc3c(F)cccc3F)C2)=O)cc(F)cc(Cl)c1 Cc1noc(C(F)F)c1C(=O)NCc1cn(CC)nn1.C(=O)COC(F)F CN1CCOC(C(N2CCN(C(c3nn(C)cc3N)=O)CC2CF)=O)C1=O Cc1ccc2nc(C)c(C(=O)NC3CCN(C(=O)CCSCC(N)=O)C3)cc2c1 C1(NC(CC2(C=C)CC2)=O)Cc2ccccc2C1NC(=O)Cc1ccncc1Cl C1(C2(NC(CN(CC#C)C(C3C(C)C3C)=O)=O)CC2)CCCO1 C(=O)(C1=COCCC1)N1CCC(C)C1C(=O)NCCOCC1CCCC1 c1(C(C)NC(c2ccc(OC)cc2)C2CCCCC2)cc(Br)ccc1Cl N1(C(C2CC(OC)C2)=O)CCC(O)(c2cn(-c3ccncc3Br)nn2)CC1 C1(CNC(CC(C)OC)=O)CC2CCC1N(C(c1ccc(C)o1)=O)C2 c1(N(CC)CC)ccc(CNC(=O)NC2CCCO2)cc1.N1CCCCC1.C C(CN=C(NCC(C)(C)C1CCCO1)NC1CCCC1)N(CC(F)F)C C12(NC(C(C(C)C)C)=O)COC(C1)CC2.c1(C(=O)N)ccc(CCC(N)=O)cc1 C1(c2nc(Cc3cc(C(=O)OC)nc(CO)c3)on2)CCc2nc(=N)[nH]cc2C1 c1(C(=O)NC(C2CN(C(Cc3c(C)nc(C)s3)=O)C2)C)cnn2c(Cl)cccc12 CC1=C(C(=O)NCCNC(=O)C2=CSCS2)C(C)n2ncnc2N1C Cn1c(O)ncc(C(N2CC(OCC)C2)=O)c1=O.c1(C(=O)N)c[nH]cc(Cl)c1=O C1(NC(C2C(OCC)C2C)=O)CCCCN1CC1CCC1 c1(NC(CSCCNC(C2N(C(C)=O)CCC2)=O)=O)ccc(O)cc1C c1(N(C)C)cccc(C(=O)NC2CCOCC2NC(C2(C)CCOC2)=O)n1 CCC(C)C(C)C(=O)NCC1CCCN(C(=O)CCc2cnc[nH]2)C1.C(C)=O.N C1(C(=O)NC(COC)C(C)C)(CO)CCN(C(c2cc(C)c[nH]2)=O)C1 N1(C(Cn2cnc(N(C)C)n2)=O)CCC(S(C)(=O)=O)C1.C(=O)(CC1CC1)N O=C(C1=CC2C=CC(C1)C2)NC1C2CC3CN(C(c4scnc4Cl)=O)C1C3C2 CCC(C)CN=c1nc2c(cnn2C(C)C)c(NCCN(C)C)[nH]1 C(=O)(CC1CN(C)c2ccccc21)SCC(C(=O)OC)CCc1ccccc1 CCCCCC(O)C(=O)N1CC2CCC(C1)N2C(c1cc2ccccn2n1)=O c1(C(C(C)C)NC(c2nccnc2N(C)C)=O)ccc2c(c1)OCCCO2 C1(CCC)CCC(C(=O)NC2C3CC(NC(c4cc(C)ns4)=O)CC23)CC1 C1(C(=O)N)CC(=O)C12CCC2.C1(CC(=O)N(CC(C)O)CCF)CCCCC1 N1(C(CC(n2c(CC)ncc2)C)=O)CCCCC(NC(C2CCC=CCC2)=O)C1 N1(C(C2C(C)C2)=O)CCC(C)(NC(C2CCC23CCC3)=O)CC1 c1(C(N2CCC(NC(c3cc(C)n(C)n3)=O)C2)=O)cc(N)c(F)c(F)c1F.C C1(C(N2C(C(N(C)CC3CCOCC3)=O)C=CC2)=O)CCCC(=O)C1 c1(C(C(=O)NCCCC2CC2)N(CCCOC)C(C)(C)C)csc(C)n1 c1cccc([N+](=O)[O-])c1.c1(C(=O)Nc2scc(CC)n2)[nH]c(C)c(C(C)=O)c1C CC1CCC(CN2CCN(c3nccc(C(C)C)n3)CC2)CC1 N1(C(CCC=CC)=O)CCCCC(C(=O)N(C2CCOCC2)C)C1 CCCC(C(O)C(=O)N1CCC(C)(C#N)CC1)NC(C1(Cl)CC1(F)F)=O c1(C(N2C(C)CCC(NC(C3CC34CC(O)C4)=O)C2)=O)occ2c1CCOC2 CCC(C)(CO)C(=O)N(CCNC(c1ccnn1C(C)(C)C)=O)C1CC1 c1(C(N(CCC(=O)NCC2CC23CCOC3)CC#C)=O)cccc2occc12 N1(C(CSCC(C)=O)=O)CC2C(CNC(c3cn(CCO)nn3)=O)C2C1 c1(CCN(CC(=O)N(C2CCCCC2)C)C)ccc(OC2CCCC2)cc1 C(=O)(C(CC(F)F)N(C(=O)CC1CSC1)C)NCCCCN(C)C c1(C=O)ccc(C2CC2)cc1.C1(CC(N2C(CC)CCC2)=O)CCN(C)C1=O.N Cc1coc2c(NC(=O)C(c3ccccc3)N)cccc12 c1(SCC)cc(C=O)ccn1.C1(CC(=O)NCC)CCCC1(F)F.C1CC1 N1(C(C2C(NC(CC3CC(N(C)C)C3)=O)CCO2)=O)CC(CO)CC(C)(C)C1 C1(NCC2(C)CCC2)CCC(C(=O)NCC2CCCS2)OC1 C1(C(N(C(C)CCO)C)=O)(NC(C2CCCSC2C)=O)CCCC1C CC(CC(F)(F)C(F)(F)Br)(c1nnnn1C1CCC1)NCC1Cc2ccccc21 C#Cc1ccc(C(=O)NC2CN(C(=O)C(=O)NCC3CC3)CCC2C)cc1.O CON(C)C(=O)CNC(=O)C(C)N(C)C(C1CCCC1)=O C1(C(=O)NCC(=O)NC(C(=O)OCC)C)CCc2cnn(C)c2C1 c1(C=O)cc(C(F)F)n(C)n1.C(C(=O)N)N(S(C)(=O)=O)C.CCC.CC C1(C(=O)NC2CCN(C(=O)Cn3ccnn3)C2)C2C3CC4C1C1C2CC3C41.C c1(C(=O)NCC2N(C(Cc3c(C)nc[nH]3)=O)CCN(C)C2)cc2nccnc2[nH]1 C1(CNC(c2c(C)ncnc2)=O)CCN(C(c2nc(C3CC3)cs2)=O)CC1C Cc1c(C(=O)NC2CN(C(c3cc(CO)[nH]n3)=O)C(C)(C)C2)cnc2ccnn12 N1(C(C2OCCN(C)C2)=O)CCC(NC(=O)C=C(Cl)Cl)CC(O)C1 c1(C(=O)NC2C(NC(C(CC#C)C)=O)CCC2)cc(Cl)cc(F)c1F CC1(C)CCCC1(C)NC(=O)C(C1CC1)NC(C1CC(=O)CC(=O)N1)=O c1(COC)cc(C)c(C(=O)NCC(C)(O)C=O)o1.N12CCC(C1C)C2=O.O c1(C(N2CCCC(n3ccnn3)C2)C(=O)NC2CC(F)(F)C2)cccc(Br)n1 Cn1cc(C(N2CCC(F)C2)=O)c(C2CCC2)n1.c1(C(=O)N)[nH]ccc1C1CC1 c1(C(=O)NCC2CC(F)CN2C(=O)CC2CC2)coc2c(Cl)cccc12 C1(NC(C2CCC(F)C2)=O)CCCC2CN(C(=O)C(F)C(F)(F)F)CC12 C(=O)(CC(C)(C)C(F)F)N(C)C.C1(CC(N2CCCCC2)=O)CCC(=O)NC1=O c1(OC)ccc(NC(=O)C(c2ccc(C)cc2)N(C2CSC2)C)c(C)c1 CC(C)CC(C)(C)C(=O)NC1CCC(NC(c2ccc(Cl)s2)=O)C1 c1(OC)ccc(C)c(C(=O)N(C2CCCN(C(C)=O)CC2)C)n1 C(=O)(CC(C)(C)CC)N(CCNC(c1cccc(COC)c1)=O)CC N1(C(c2cc(CC)oc2C)=O)CC(NC(=O)C)C2(CCC2)C1.c1ccsc1.O C(=O)(C1=CCc2ccccc21)NCC1C(F)(F)CCN(C(CCS(C)=O)=O)C1 Cc1nccc(CCC(=O)NC2CCN(C(=O)COCP(C)(C)=O)C2C)n1 C1(C(=O)NC2(C)CN(C(c3c[nH]nc3-c3ccncc3)=O)C2)CCCC(C)(C)O1 C1(OCCC)CCN(C(C2COCCC2NC(=O)CC23CCCC2C3)=O)CC1 N1(C(C2(CNC(c3nc(=N)cc[nH]3)=O)CC(=C)C2)=O)CCC(O)(C)C1.O C1(C(=O)NCCC(C)CCNC(c2ccncn2)=O)CCC(C)(C)CC1 c1(C(=O)NC(CN(C(C2CN(CC)C(=O)N2)=O)C)C)ccc2[nH]ccc2c1F N1(C(C(ON=C(C)C)C)=O)CCC2(CC1)CC(C(=O)N1CCCC1)=NO2 c1(OC)cccc(CC(=O)NC2CN(C(c3csc(Cl)c3)=O)C3CC23)c1 C(C(=O)NC(C1(C(=O)NC)CC1)C)(C(C)C)NC(C)=O.C1COCCO1 N1(C(COCCC=C)=O)CC(C)C(Nc2ncnc(OC)c2C)C(C)C1 c1(CCC)ncc(C(=O)NC(C)CC(C)NC(=O)CN(C)C2CC2)s1 N1(C(COC)=O)c2ccc(S(=O)(=O)NNC(=O)OC)cc2CC1C C1(C(=O)NC(CN(C(=O)CCn2cccn2)CC)C)CC2CCC(C1)C2F c1(C(=O)NC(CC(N)=O)C(=O)O)ccc2c(c1)CCC(N)C(=O)N2 c1(N2CCCC(NC(c3c(C)ocn3)=O)C2)c(C#N)cnc2c(C)cccc12 C=CC1(CC(N2CCC(NC(=O)Cc3csnn3)CC2)=O)CCCCC1 c1(CNC(C)COC2CCOCC2)cc(C(F)F)no1 C(=O)(CCC(=O)NC1CCC(C)(CNC(c2cc(Cl)cnn2)=O)C1)N(C)C CCCCC(CC)CC(=O)NCC(O)CC(=O)Nc1cnn(C(F)F)c1 CC(C)CCCC(=O)N1CCC(CO)(NC(=O)CC2CCN(C)C2=O)C1 C1(N(C(=O)CCOC2CC2)CC#C)CCN(C(C23CCCCC2C3)=O)CC1 c1(C(N2CC=C(CCNC(C#CC(C)C)=O)CC2)=O)ccc(C#CC2CC2)cc1 N1(C(C(C)C(F)F)=O)CC2CC(C1)N(C(=O)CC1CC(C3CC3)C1)C2 c1(CC)nc(CC(=O)NC(c2nnnn2CSc2ccccc2)(C)C2CC2)cs1 Cc1cc(=NCC2CN(C(=O)Cc3c(C)n[nH]c3C)CC2(C)C)[nH]c(C(C)C)n1 c1(C(N2CCCC(CC)(NC(C3CCC(C)O3)=O)C2)=O)noc(C)c1[N+](=O)[O-] N1(C(c2nnc(C)s2)=O)CCCOC(CNC(=O)CC(c2cccc(F)c2)O)C1 n1(C(C)C)cc(C(=O)NCCC(=O)NCc2csc(O)n2)nn1 N1(C(C(NOC)=O)=O)CCC2(CC2C(=O)NCC(C(C)C)C(C)C)C1 C1(C(N(C2CCOCC2)CC)=O)CC12CCN(C(=O)Cc1cccnc1O)CC2 C(C(C)NC(c1cc(CO)n(C)n1)=O)(C(C)C)NC(CSCCOC)=O N1(C(CCOC)=O)C2CCC1CC(CCNC(C1(OC)CCC13CCC3)=O)C2 CC#CCCC(=O)NCCC1CC(NC(C2CCCCC2F)=O)C1 C1(C(N(CCCCNC(C2(CC)CC2(F)F)=O)C)=O)Cc2nccnc2C1 n1(CC)cc(NC(=O)C2=CCN(C(=O)C=C(C)C(C)C)C2)ccc1=O c1(C(=O)NCCN(C(=O)Cn2cn[nH]c2=N)CCOC)ccc2cncn2c1 Cc1ccccc1C(N1C2CN(C(=O)CN3C(=O)C=CC3=O)CC12)=O C1(C(C)C(c2ccccc2)=CC=CC=O)CCN(C(c2c[nH]nc2C)=O)C1.CC c1(-c2ncc(CSC)s2)cccc(NC(C2(CSC)CC2)=O)c1 C1(O)(CNC(C(C2CCCN(C)C2)(C)C)=O)CCCN(C(c2coc(O)n2)=O)C1 N1(C(=O)C2=CCCOC2)CC2(CCCC(CNC(C3(O)CCSCC3)=O)O2)C1 N1(C(C2CC(C)(C)C2)=O)CCC2CCN(C(c3ccc(F)c4[nH]ccc34)=O)C2C1 c1(C(=O)N)cc(O)cc(N)c1Cl.C1(NC(CNS(N)(=O)=O)=O)CC2CCC2C1 C1(C)(C(N(CC)C2CC2)=O)CCC2(CC1)CC2.C(C=O)C(C)C.CC=O.N Cn1cnc2c3c(ccc12)N(C(c1ccc(Br)c(OC(F)F)c1)=O)CCC3 C1(C(=O)N)CCCC(C#N)C1.c1(OCC)ccccc1C(=O)NC1CCCCC1 C1(CCNC(C=CC)=O)CCN(C(c2ccccc2)=O)C(C)C1.CC(F)(F)F CCC(C#N)C(=O)NC(C(=O)NCc1ccc(C)nc1)C(C)OC c1(C(N2CCOC3(CCCC3)C2)C(=O)NC2CC2)n[nH]c2c(Cl)cccc12 C(=O)(C1CCCc2nn(C)cc21)N(C(CNC(c1nn(CC)nc1C)=O)C)C CS(=O)(=O)c1cccc(Cl)c1C(=O)NC1C2CCC1C(F)(F)C2 C1(C(C)NC(=O)C(C)(C)F)CN(C(=O)C(C)N(C)C)CCO1 CCCC(CNC(C1(OCC)CCCC1)=O)C(=O)NCC(O)CN(C)C Cc1ccc(NC(N2CCC2C(=O)N(CCO)C2CC2)=O)cc1Cl c1(-c2cn(CCCC(N3CCCC(C(=O)NC)C3)=O)nn2)c[nH]c2nccc-2c1 C1(CNC(C=CCCC)=O)CC2CCC1CC2.N1(CC=O)C(=O)CNC1=O.N N1(C(CCCCOC)=O)CCC(F)(CNC(c2cnoc2-c2cccs2)=O)CC1 N1(C)CCC(F)(F)CC1.c1(N(C)C(C23CC(C=O)(C2)C3)=O)c(N)cccc1Br c1(CC)cc(CC)[nH]c(=NCCCCCCN(C(=O)Cc2[nH]cnc2C)C)n1 CCC(Cc1ccccc1C)C(=O)N1CCC(N(C(=O)Cc2n[nH]c(C)n2)C)C1 N1(C(CC(C)(C)C(F)F)=O)CCCC1C1CCCN1C(c1cc(Cl)n[nH]1)=O C1(C(=O)NCC2CCCN2C(C2(CC3CC3)CCC2)=O)CCCCC1(F)F CCCC(CCC)CC(=O)NC1(C)CN(C(=O)C(C)C(C)n2cccn2)C1 c1(C(N2C(CNC(C(C)CF)=O)CCC2)=O)ccc(C(F)(F)F)nc1N C(CC(=O)N(C)CC1CN(C(=O)Cc2cnn(C)c2)C1)(C(F)(F)F)OC.O C(=O)(C1Cc2ccc(Cl)cc21)N(CCCNC(C1N(CC)CCOC1)=O)C CC1CCCC1(C(=O)NCC1CC12CCC2)NC(=O)CCNC(N)=O C1(C)(CNC(CC(CC)OC)=O)CCCN(C(c2ccncc2C2CC2)=O)C1 C1(CNC(=O)NCCN(C)C)(NC=O)CC(O)C1(C)C.C(C)(C)C Cc1cc(C(=O)NC23CCN(C(c4cnc(C(N)=O)cn4)=O)CC2C3)cc(N)c1 CC(C)CC(C)(CNC(=O)Cn1cccc(N)c1=O)NC(C12CCC1CC2)=O N1(C(c2n(CC#C)cnn2)=O)CC2CCCC2C1C(=O)NCc1ccncc1F C1(C(=O)NCCC2(C)CCCC2)CCCCN1C(c1cc(C#N)cs1)=O CC(C)CC(CNC(=O)C(=O)NCCn1cc(C#N)cn1)CCO c1(OC)cnc(C(N2CCC(C)C2CNC(=O)CN(C)C)=O)c(OC)n1 C(=O)(C1=NNC(=O)CC1)NC1CCC(F)(CNC(=O)CCN2CCC2)C1 N1(C(COC2(C#C)COC2)=O)CCCC(CO)(NC(=O)C(CC)n2ccnc2)C1 N1(C(c2c(O)ccc3ccccc23)=O)CCOc2ccc(Br)c(F)c21 c1(C(C(=O)Nc2ccc(OCCN3CCNCC3)cc2)O)ccc(O)c([N+](=O)[O-])c1 C1(C(N2C(CNC(C=CCC)=O)CC2)=O)CCOC1CC n1(CC(=O)N(CC(CC)NC(C2CC(C)=NO2)=O)C)cc([N+](=O)[O-])ccc1=O C1(C)(C(N(CCCC)C)=O)CC2(C1)CC(F)(F)C2.Cc1[nH]nc(C(=O)N)c1C c1(OC)ccc(OC)c(S(=O)(=O)N2CCC(O)(C=O)C2)c1.c1(CC)nn[nH]n1.N C1(NC(C2C(COC)C2)=O)CCCC1O.c1(C=O)cccnc1.C(C)C.C C1(NC(CCC2(C#N)CCC2)=O)CC2CCC1CC2NC(=O)C(Cl)=CCl c1(OC)cccc2c(C(N3CC(NC(c4cnsc4C)=O)C(C)C3)=O)c(C)[nH]c12 N1(C(c2ccnc(Cl)c2Cl)C(=O)NCC)CCSC2(CCCCC2)C1 C1(C(N2C3CN(C(c4cc(CSC)c(C)s4)=O)C(C3)C2)=O)CCn2cnnc2C1 N1(C(C2N(C)CCCCC2)=O)CC2(CCN(C(=O)Cn3cc(Cl)cn3)C2)C1 C=CCCC(C(=O)NCC1COCCN1C)NC(=O)CC(=O)NCC C=CCCC(C(=O)OCC)NC(C12CC1CN(C(C1CC1C1CC1)=O)C2)=O C1(C)(CC)C=C(C(=O)NC2CCCN(C(c3coc(C4CCCC4)n3)=O)CC2)C1 N1(C(c2c(C)nc(C3CC3)[nH]2)=O)CC2(CC(C)C2)C1.c1(C=O)cnc(O)s1.N Nc1ccnc(C(=O)NCC2(NC(=O)CC3CCC(O)C3)CCOCC2)c1 C(CC(C(C)C)NC(c1cncc(OC(F)F)c1)=O)N(C(COCC)=O)C C#CC1CC2CCC1N(C(=O)C(C)NC(c1cc(F)cc(F)c1)=O)C2 N1(C(CSCCOC)=O)CCC(CO)C(NC(=O)C(c2ccc(F)cc2)CO)C1 N(C1CC(C)Cc2cc(OC)c(OC)cc21)CC(=O)NCCC=CC c1(C(N(C)CC2OCCN(C(CSC)=O)C2)=O)cccc([N+](=O)[O-])c1Cl C(=O)(CCCCCCCCCO)NC1(CC=C)CCCN(C(=O)C(C)OCC)C1 CON(C(=O)c1ccc(-c2nn[nH]n2)cn1)C1CCNC1 Cc1cc(C(=O)NC(C)C)cc([N+](=O)[O-])c1Cl.c1(C=O)cc(C(F)(F)F)n[nH]1 CN1CCCCC1CC(N1CCC(CC(N2CCCC2C2(C)CC2)=O)C1)=O C=CCCCCCC(=O)N1CC(O)(C(=O)NCC(C)(C)C2(O)CCC2)C1 C(=O)(C(C(C)C)Oc1ccccc1C)NC(CC=C)CNC(c1ccc(C)s1)=O c1(Nc2ccc(NS(C)(=O)=O)cc2)cc(Cl)[nH]c(=N)n1 N1(C(C)=O)CSCC1C(=O)NC(C)CC(C)NC(c1ncoc1C1CC1)=O C(=O)(C(C)(C)CC#N)NCC1OCC(C(N(CC(C)(O)C2CC2)C)=O)C1 c1(C(N2CCC(NC(CC(C=C)(C)O)=O)C(CO)C2)=O)cc(S(N)(=O)=O)co1 c1(OC)cc(NC(C2CC2C(=O)Nc2ncc(Br)nc2C#N)=O)cc2n[nH]cc12 Cc1nn(CC(N2C3CCC(C3)C2CNC(=O)CC2CCSCC2)=O)c(C)c1Cl CC1CCN(C(=O)C=Cc2ccnn2C)CCN1C(C1CC1Cl)=O c1(C(N(CC(C)C)C)=O)ccccc1N(S(C)(=O)=O)C.C1(C=O)CSCCS1 C(=O)(C1CCc2c[nH]nc21)NCC1CN(C(C2CC(C)(C)C2)=O)CC1O c1(C(=O)OC)cc(C(N2CCC(C)C2)=O)cc(C)c1.c1(CC=O)ccccc1.N C1(C(=O)NC23COC(C2)C(NC(C2CCC2)=O)C3)CCc2cnnn2C1 C1(NC(=O)CCC2CC2)CN(C(=O)C2=CC3C=CC2C3)C2(CCCC2)C1 C(CCC(C)C)OCC(=O)N(C(C(=O)N(CCCCO)CC)C1CC1)C N1(C(c2ccc(CC)o2)C(=O)Nc2ccccc2C)CCCC(N2CCCC2)C1 C=C(C)C1CC=C(CN2CC(=O)N(CC3(C)CCCS3)C2=O)CC1 c1(NC(c2n(CCC#C)ccc2)=O)ncc(CC(=O)OCC)cc1F C(CCCC(=O)N(C)OC)N(C(c1c(CC=C)cccc1)=O)C C=C(C)CCCC(=O)NCC1C(C)CCN1C(=O)CCNC(=O)C=CCl C=CC(C)(CC)C(=O)N1CCC(CCNC(c2ccc(F)c(CSC)c2)=O)C1 c1(C(N2CC3C(CN)C3C2)=O)nnn2ccccc12 N1(C(C2CC23CCCC3)=O)CCC(F)(CNC(C2(CO)CCCC2)=O)CC1 c1(OC)ccc(I)c(C(=O)NC2CN(Cc3cc(Br)ncc3OC)C2)c1 C1(C(=O)NC(C)(C)C=C2CC(=O)NC2=O)CC(OC(C)(C)C)C12CCC2 c1(OC)ccc(S(=O)(=O)N2CCC3C(CCN3C(=O)C3CC3)C2)cn1 c1(CC(=O)NC2CC3CN(C(c4cncc(Cl)n4)=O)CC23)cc2ccccc2s1 c1ccc(C=O)nc1.c1(C(=O)NC(c2cc[nH]n2)C)ccccc1C(F)(F)F.N CC1(C)CC(CNC(=O)C(F)(F)Sc2ccccc2)CN1C(=O)C=C(Cl)Cl c1(-c2cc(C(=O)NCCCC)c(F)cc2C)cc(C)c2n[nH]cc2c1 N1(C(CC(C=C)(C)C)=O)CCC2CCN(C(=O)C(=O)N(C)C)CC12 n1(CC)ccc(C(=O)NCC2CCC2)c1C.c1(C=O)conc1C1CCC1.N CC1CCCN(C(=O)CC(F)(F)F)C1CNC(=O)Cc1ccc(O)cn1 N1(C(Cc2cc(C(C)C)no2)=O)CCC2(CC2NC(C2CC2F)=O)C1 C(CCCCCN(C(=O)CC1CCC1(F)F)C)NC(c1ccn(COC)n1)=O c1(C(c2nnnn2C2CCOCC2)NCCCC=C)ccc(C2CC2C)o1 c1(CC(N2CCCC(NC(C3C(C(C)=O)C3)=O)C2)=O)cc(C)cc(F)c1 N1(C(Cc2nc(C)oc2)=O)CCC2C(NC(=O)CCC3CCCCO3)C2C1 C12(NC(C3C(C(C)(C)C)C3)=O)CC1CN(C(C1(C)CC=CCC1)=O)C2 c1(OCCCCC)ccc2cc(NC(N3C(C)CCC3(C)C)=O)[nH]c2c1 n1(CC(N2C(CNC(=O)CCc3cnoc3)COCC2)=O)cc(Cl)c(O)nc1=O c1(C(N2CC(Cn3cc(CC(C)(C)C)nn3)C2)=O)cc(Cc2cnn[nH]2)ncn1 C1(NC(c2ccn(CCC)n2)=O)CCCCC1NC(=O)C(C)(O)C1CC1 C1(C(=O)NC2CCC(CNC(c3[nH]n(C)c(=O)n3)=O)CC2)CCN2CCOCC12 C1CN(C(c2cc(C)c(C)[nH]2)=O)CC2(CC2)C1.c1(OC)cc(F)ccc1C=O.N C1(NC(C2(OCC)CCOC2)=O)CCC(NC(C2(C)CCC2C)=O)CC1 c1(NC(C2NCCN(C(CCC#C)=O)C2)=O)ccc(C(C)=O)cc1F c1(CN2CCN(C(c3c(OCC)ccs3)=O)C3C2C3)sc2ccccc2c1C c1(N2CC3(C(C(=O)Nc4ncc(C)c(I)c4)C3)C2)ncnc2[nH]ccc12 c1(CCC(=O)NC2C=CC(CC(=O)NCC3=NOCC3)C2)cncnc1 N1(C(C2(C)ON=C(C)C2)=O)CCCC(O)(CNC(=O)CP(C)(C)=O)CC1 Cc1ccc(C=CCNC(=O)NCC2(CCN(C)C)CC2)c(C)c1 n1(CC)nc(C)cc1C(=O)NC.C1CN(C(c2ccco2)=O)CCO1.N(C)C n1(C(C)C)ccc(=O)n(C(=O)C(C(C)C)N2CCCCC2)c1=O C(c1cc(OC)ccc1)=C1CC(C(=O)NC2CCN(C(=O)OC)CC2F)C1.O CC(C(C)(C)C(=O)NCC1CC12CCC2)NC(=O)CCCn1cncn1 S(=O)(=O)(c1cnc(NC(C)CC)cc1C)NCc1c(CC)nn(C)c1CC c1(NCc2cnn(C)c2-c2ccccc2)ccnc2cc(Cl)ccc12 C1(C(=O)Nc2cc(OC)ncn2)CCCC12CCN(Cc1cc(O)cc(Br)c1)C2 N1(C(CCCCCN(C)C)=O)CCN(C(=O)C2=CCCCO2)C2CCC12 CC1(C(N2CC=CCC2)=O)CCN(C(C2CC2(F)Cl)=O)C1 C1(NC(C2(CCCC)CC2)=O)CC2CC1CC2C(=O)NC1COCC(C)(C)C1 N1(C(c2c(C)cc(SC)o2)=O)CC2CC(NC(=O)C(C)(C)CO)CC2C1 Cc1c(C)nnn1C.c1(CC=O)cnn(C)c1.C(C(C)(C)C)N(CC=O)C.N C(CCC(C)(C)NC(C1CC(F)(C)C1)=O)NC(C1C(c2n(C)cnc2)C1)=O n1(C(C)C)cnc2c(NCCC=CBr)[nH]c(=NCC3(C)NC(=O)NC3=O)nc12 C1(N(C(C2N(C)C(=O)C(F)C2)=O)C)CC2CCC(C1)N2C(=O)Cn1cnnc1O CC1(C)CN(C(=O)C(C)(C)c2cscc2Cl)CC2(CN(C(C3(F)CC3)=O)C2)O1 c1(C(N(CC(C)N(C(=O)C(N2CCNC2=O)C)C)C)=O)cnn2ccccc12 CCC(C)(CNC(C1CC(C(=O)OC)C1)=O)C(=O)N1CC2CCC2C1 c1(C(=O)NC(CNC(C(C)(C)OCC)=O)C)ccc(C)c(F)n1 c1(OC)ncc(Cl)c(C(N2CC(CNC(C3(O)CCOCC3)=O)C2)=O)c1Cl Cc1ccc(C)c(C2=NOC(C(=O)NCC(O)C)C2)c1.C(=O)C(C)(C)C(F)F.N c1(C(=O)NC2CCC(CNC(COCCC)=O)C2)sc2ncccc2c1Cl N1(C2C(NC(c3c(C)ccs3)=O)COC2)CCN(C(=O)C=C2CCC(C)C2)CC1 N1(CC)CCN(C(=O)C(C)CCc2ccc(-c3cccc(SC)c3)o2)C(CO)C1 C1(OC)CC2CC(OC(=O)CCc3c[nH]c4ccc(F)cc34)(OC)CC2C1 c1(OCC=C)c(C(=O)NC)cccc1C.C(=O)(C1=CCCCO1)N1CCC(O)C1 C1(CNC(CCSCC(C)C)=O)CCCCCN1C(c1cccc(N(C)C)c1)=O C1(C(=O)NCCCC(CO)NC(C(C)C2CCC2)=O)CC12CC(C)(C)C2 C1(COC)(C)CCN(C(C2C=CCC2)=O)CC1.c1(CC=O)ccc(Cl)nc1.N c1(C(=O)NC2C(C)(CN)C2)cc2cc(Br)ccc2o1 n1(CC(=O)NCCC2CC(NC(C(C(C)SC)O)=O)C2)cnc2ccccc12 c1(C(=O)NCC2(F)CCN(C(CCCCC=C)=O)CC2)nc(Cl)cc(N)c1Cl n1(CC(=O)N(CC(N2CC(=C)C2)=O)C2CC2)cc(C)cn1 C(=O)(CN=c1[nH]c(=NC2CCSCC2)[nH]c2ccccc12)NCC=C C(=O)(CCC(=O)N1CCCC1CN(C(C1CC1C1CC1)=O)C1CC1)N(C)C N1(C(=O)CCc2nnc(C(F)F)o2)CCC2(CCCN2C(c2ncc[nH]2)=O)C1 C(C(C)C(C)C(=O)N1CC2CC(C1)C2NC(=O)CC(C)n1cccc1)OC C1(C(=O)NCc2ccc(C)cc2)(CN)CCCN(C(C2CCOCC2)=O)C1 CCC(CC)(CCNC(=O)COCCC(C)C)NC(=O)C=C(C)C(C)C c1(C(=O)NC(CCCCNC(c2cc(C)sn2)=O)C)ccnc2ncccc12 CCC(C(C)(C)C)NC(=O)CC(C)NC(C1CC(C)(C)C1)=O CC(C)C(CC(=O)NCC1CSCCO1)NC(C1COCOC1)=O Cc1c(Br)ccc2c1N(C(C1CCC(=O)N(CC(F)(F)F)C1)=O)CC2 C1(C(N(CCCCO)CC)=O)CCCCN(C(C2CCC(C)(C)OC2)=O)C1 c1(SC)ccsc1C(=O)NCC(C)(C)CN(C(=O)CCO)C.C1CCCOC1 CC1(NC(C2CC(=O)N2)=O)CCCN(C(=O)Cc2ccc(CO)cc2)C1 C(CCC(=O)N1CC(O)(CNC(=O)COC)C1)OCCC.c1ncnn1C c1(CC(=O)N(C(CNC(=O)COCCF)C2CC2)C)cscn1 S(=O)(=O)(c1c(Cl)cc(Br)cc1Cl)N1CC(NC(c2cc(Cl)cc(F)c2Cl)=O)C1 c1(C(=O)NCC2CCCN2C(C2CC2(F)F)=O)coc2c1COC2 N1(C(C(C)OCC#C)=O)CC(F)(F)CC1CCNC(c1ccoc1C)=O.C N1(CCCNC(CC)=O)CCN(C(=O)C(C)CS)CC1 C(C1=NOC2CCCC12)NC(C(CCC)NC(C1(C)CCN(C)CC1)=O)=O N1(C(C2(CC=C)CN(C(C3CC(CF)C3)=O)C2)=O)CC2CC(CO)C(C2)C1 CC(C)C(O)CC(=O)N1CCN(C(=O)CCC=CBr)C(C2CC2)C1 C(CCC)(C(O)C(=O)NCc1cncn1CC)NC(C(C=C)O)=O N1(C(c2cn(CC)nn2)=O)CC2C(CNC(=O)Cc3ccc(Cl)s3)C2C1 c1(C(=O)NCC2C(NC(C3(OC)CC3)=O)C2)cc2cccc(C)c2[nH]1 c1(CC(N2CC3C(NC(c4ccc(CC)[nH]4)=O)(C3)C2)=O)sc2ccccc2c1C C(CC(C)C)(C(=O)NCCC1CCCO1)NC(c1ccc(C)n1C)=O c1(OC)cc(C)cc(C(=O)NCC(C)(C)NC(C2CCc3c[nH]nc3C2)=O)c1N c1(C(=O)NC2C3CN(C(C(C#C)(C)C)=O)CC32)cnn2cccnc12 c1(C(=O)NC2CN(C(C(CC#C)O)=O)CC2C)cnc2cc(OC)ccc2c1 N1(C(C2C(C)(C(F)F)C2)=O)CCCC2(C)CCCC12.C(=O)(CCc1ccsc1)N c1(C(=O)N)cc2c(=O)[nH]ccn2n1.C1(F)(CNC(c2cc[nH]n2)=O)CCC1 c1(C(N2CCC(CCCNC(C(COC)(F)F)=O)CC2)=O)ncn2c1CCCC2 C(c1ccccc1C)=CC=O.C1(C(N(C2CCCOC2)CC)=O)OCCC1C.N Cc1ncc(Br)c(C(N2CC3CCC2C3NC(=O)CCOC2COC2)=O)n1 O=C(C1=CC2C=CC(C1)C2)NCCC1CCN(C(C23CCC2C3)=O)CC1 Cc1ccc(CS(N2CCCCC(C)C2)(=O)=O)cc1C c1(CC(=O)NC(CNC(CC(C(C)C)O)=O)C2CC2)c[nH]c2ccccc2c1=O N1(C(CCCSC(C)(C)C)=O)CC2CCN(C(=O)C3=CCS(=O)(=O)C3)C2C1 c1(NCC2(F)CC(NC(C34CCCC3C4(F)F)=O)C2)cnc2ccccc2n1 C1(NC(CSCCOC)=O)CCCC(C(=O)NCc2coc(C)n2)CC1 c1(C(=O)NC(C2CN(C(C3CCCC(C)C3)=O)C2)C)cc2c(o1)CCCC2 c1(-c2c(F)ccc(C(C)=O)c2)ccc2cc(C(=O)NC3CCS(=O)(=O)C3)nn2c1 CCCCCC(CCCCC)CC(=O)NC1CCCCN(C(c2cscn2)=O)C1 N#CC1CCCC(c2nnnn2C)(NCc2cc3n(n2)CCCC3)C1 Cc1ccc(C(=O)NC2(C)CN(C(=O)CS(=O)(=O)NC3CC3)C2)c(N)c1C c1(C(=O)NC(CCCNC(C2(OCC=C)CCC2)=O)C)ccc(F)c(C)c1 C(=O)(C(CC)NC(=O)NCC(C)(CO)c1ccccc1)NC c1(-c2cc(C(=O)Nc3c(Cl)ncc(C)c3)n[nH]2)cc(F)cc(F)c1F CCC(C)CNC(C1(c2cc[nH]n2)CC1)=O.C1(=O)CC2(CC2)CN1.O c1(CN2C(=O)CCN(Cc3ccsc3)C2=O)ccc2c(c1)OC(F)(F)O2 N1(C(c2c(C)nn(C)c2)=O)CCC(C2(NC(C3CCC4(CCC4)O3)=O)CC2)CC1 S(=O)(=O)(c1ccc(N(C)C)cc1)NC(C)CC1=CCCCC1 C(=O)(CCC1CCc2ccccc21)NCC(C1CC1)NC(CCCC=C)=O N1(C(C(C=C)O)=O)CCCCC1CNC(c1cnn(CCCC)c1C)=O n1(CC2CC(CNC(=O)CN3CCCC3)C2)cc(C2(O)CCCC2)nn1 N1(C(CC(C)C(F)F)=O)CCCC(C2CC2NC(c2cccn3ncnc23)=O)C1 N1(C(CC(=O)OC)=O)CC(NC(c2cncc(OC)n2)=O)C(C)C1 c1(C(C)C)conc1CC(=O)NCCOCCCNC(c1ccc(Cl)s1)=O c1(N(CC(C)CO)C)nc(=NCC(C)c2ccc(Br)cc2)[nH]c2c1CCCC2 C(CC(N)=O)(C(=O)NCCn1cccnc1=O)NC(C1(CN(C)C)CC1)=O c1(C=O)ccc(S(=O)(=O)N(C)C)cc1.C(CC(=O)NCC(F)C)=CC=C.N Cc1cc(F)sc1C(=O)NC(C1(C(N2CCC(c3cc[nH]n3)C2)=O)CC1)C N1(C(C2(C=C)CC2)=O)CC(NC(c2nc(C)oc2C)=O)CC(C)(C)C1 N1(CC(=O)NCC2CCN2C(c2ccc(Cl)cc2)=O)CCc2ccccc2C1 Cc1c(-n2cc(C3(NC(c4cc(C(=O)O)[nH]c4C)=O)CCC3)nn2)cccc1F N1(C(CN(S(CC)(=O)=O)C)=O)CCN(C(=O)C=C2CC2)CC(C)(F)C1 C12(NC(=O)NCC(C)C)CCCC(NC(C3CC34CC4)=O)(C1)C2 C(c1cc(Br)cs1)=CC(=O)N(C1CC(NC(C2CC(N(C)C)C2)=O)C1)C c1(C(=O)NCCC2(O)CCN(C(CC)=O)CC2)cnc2onc(C(C)(C)C)c2c1 CCC(CCC(=O)N1CCCC(N(C(c2cc(C3CC3)no2)=O)CC)C1)OC C(CC(=O)N(C(C)CC(F)(F)F)C)(C(C)OC)NC(C(F)=CCC)=O C#Cc1cccc(C(N2CCCCC2C(=O)NC2CC3CC4C(C3)C24)=O)c1C c1(C(=O)NCc2cc(C(=O)NCC3C(C)C3)on2)ccc(=N)[nH]c1 c1(C(N2CCC(c3cn(CC4CCC4)nn3)C2)=O)cc(=O)n(-c2ccccc2)[nH]1 CCC(C)C(C(=O)N1CC([N+](=O)[O-])C1)N(C)C(C1CS(=O)(=O)C1)=O C(=O)(N=c1ncnc2[nH][nH]c(Br)c1-2)C1N(C(c2c(C)c[nH]c2)=O)CCC1 Cc1cc2ncc(-c3ccccc3)c(CCCNC(=O)N=c3cc[nH]cc3)n2n1 Cc1cc(C(F)(F)F)nc(NC2CC23CC(NC(=O)CC2CC4CC4C2)C3)n1 c1(C(N(C2CCC(NC(c3cc[nH]c3)=O)C2)C)=O)cccc2c3c([nH]c12)CCC3 Cc1ccc(C)c(OCCNC(c2nn(C(C)C)cc2Br)=O)c1 CC(CS(C)(=O)=O)C(=O)NCCC1CSCCN1C(c1cc2cnn(C)c2s1)=O CC1(C(=O)NC2CCN(C(c3cn(C4CCC4O)nn3)=O)CC2)CNC(=O)C1 N1(C(C2C(CC)CCO2)=O)CC2C(C(=O)NC3(COC)CC=CCC3)C2C1 n1(CC)ncc(C(=O)NCC(F)CNC(C2(CC(C)C)CCCC2)=O)c1Cl N1(C(CCNC(C)=O)=O)CC2CN(C(C3CC34CCC4)=O)CC2(C)C1 CC(C)C(C)(O)C(=O)N1CCC(C)(NC(=O)Cc2csc(Br)c2)CC1 CN1CCCC1(C)C(N1CCCC(N(C(=O)CN(C2CCCC2)C)C)C1)=O c1(CNc2ccc(C#N)cc2F)c(N)oc2ccc(F)cc2c1=O C1(C(N2CC(CC#C)OCC2)=O)(NC(=O)Cn2ccnc2C)CCC(C)(C)C1 Cc1cc(C(F)(F)F)ccc1Cc1cccc(SC2CNC(=O)C2)c1 c1(NC(=O)C(c2cccc(Cl)n2)(F)F)ccc(S(=O)(=O)F)c(F)c1 CCS(=O)(=O)CC(=O)NC(CN(C)C)C(=O)NCc1ccc(CO)cc1 N(C(=NCCCC1CC1(Cl)Cl)NCC(=O)NC1CCCC1)C1C(C)C1 CCC(C)CCCC(=O)N1CC2C(CNC(c3cc(C)nc(C)n3)=O)C2C1 c1(C2CCN(C(=O)NC(c3ccoc3)C)CC2)nc2cc(Cl)ccc2o1 C1(C(N2C3CN(C(=O)CCOCC(F)F)C(CC3)C2)=O)CCCCC12OCCO2 C1(C)(CNC(COCCSC)=O)CN(C(c2cnc(C)nc2C)=O)CC1C c1(C(N2C(C)CC(NC(c3c[nH]ccc3=N)=O)C2)=O)cc(C(N)=O)cc(F)c1 C1(C(N)=O)CCC(C(N2CC3C(CNC(c4nocc4Cl)=O)C3C2)=O)CC1 C(=O)(C(C)(C)CCS(C)(=O)=O)NC(CNC(C(C1CCC1)OC)=O)C CC1CC2(CC2)CN1C(C1COCCN(C(=O)C(C)CO)C1)=O Cc1nc(C2CC2)ccc1C(=O)NC(C)CCN(C(=O)Cn1cccc1)C c1(C(N2CCCC2)=O)cc2c([nH]1)CCOC2.C1(C(=O)N)CCS(=O)(=O)C1.CC c1(C2(C(N3C(CN=c4nc(C)[nH]s4)C(C)CCC3)=O)CC2)nc2cccnc2[nH]1 Cc1c(C2OCCC2NC(=O)NC(CC(F)F)c2ccccc2)cnn1C C1(C(N2CC(CC=C)(C(=O)NCC3COCC(C)O3)C2)=O)CCCCC(=O)N1 C1(CCCC)CN(C(C2(C(C)(C)O)CCC2)=O)CCN1C(=O)C(F)n1cccn1 C1(NC(C(CO)OC)=O)(CO)CCCN(C(=O)C(C(C)C)c2ccncc2)C1 C(=O)(CCCC(=O)NC(C(=O)NCCc1nccs1)C1CCCC1)OC c1(C(C(=O)N(CC(CC)NC(c2ccc(C(=O)OC)o2)=O)C)C)ccccc1F c1(CC(=O)NCC(C)C)nc2c([nH]1)CCCC2.c1(C=O)cccc(CC#N)c1.N N1(C(c2c(OC)oc(C)n2)=O)CCCN(C(=O)CCc2cc(C)no2)C(CO)C1 C1(CNC(CCc2c(C)ncs2)=O)CC2CN(C(c3cccc(F)c3O)=O)CC12 CCCCCCCCC(=O)NC1CC=CCC1C(=O)Nc1ccsc1C c1(CCCC)cn(CC(=O)NCCOCC2CCC2)nn1 c1(OC)ccccc1CN(C(=O)Cc1cncs1)CCO.C(C)(C)C.C=O CCC(CC(=O)NCCCNC(c1sccc1NC(c1ncoc1C)=O)=O)SC CCCC(C)CC(=O)N1CCCOC(CNC(c2cc(OCC)ncc2Cl)=O)C1 C(=O)(C1=CCCC1(C)C)N(C)CC1CCCC1NC(C1(C)CC1)=O C1(C(N(C(CC)C2CC2)C)=O)CC2(CCN1C(=O)CC(C)(O)COC)CC2 c1(OC)cc(-c2cc(C)c(C)c(C)c2)cc2ccccc12 Cc1c(C(N2CCC3CN(C(c4cccc(CO)c4)=O)CC23)=O)sc2nccn12 Cc1oc(C#N)cc1C(N1CC2CCC2(NC(=O)CS)C1)=O.c1ccc(F)cc1 N1(C(c2cnc(-c3ccccc3)[nH]2)C(=O)NC)CCN(C)CC1CCSC c1(C(=O)NCCC(C)(C)NC(CCC(CC)C)=O)cncc2cnccc12 c1(OC)ccc(Cc2nc(-c3ccc(Br)cc3)nn2C(C2CCCCC2)C)cc1 Cc1cc(S(=O)(=O)N2CCCCC(C)(F)C2)ccc1-c1c[nH]nc1C CC(CCC(=O)N1CCC(OC2CCC2)C1)NC(=O)Cc1ccco1 c1(NC(CC)CC#N)nc(N2CC=C(C)CC2)nc2c1cnn2C C=CC(C)C(=O)N1C(C(=O)NC2CCOC2=O)CC1C N1(C(C(CNC(C)=O)(C)C)=O)CC2CCCCC2C1.C1(C=O)C=CS(=O)(=O)C1 c1(NC2CCN(c3ccc(C(=O)OC)nc3C#N)CC2O)ccc([N+](=O)[O-])cn1 c1(C(=O)NC(CNC(C(C=C)O)=O)C2CC2)ccc(C(F)(F)F)cc1C#N C1(C(F)F)(OC)CC(C(=O)NCCC(C)(C)NC(=O)C)C1.c1ccccc1 C1(C(=O)NCC2COCCN2C(c2ncccc2F)=O)CCC(C2CC2)CC1 c1(CC(=O)OCCn2c(C)csc2=O)ccccc1S(C)=O C1(C(N2CCCC(C)C2)=O)(CC)CCC(F)(F)CC1.c1cc(=O)n(C)c(O)n1.N C1(C(N2C(C3CCN(C(C(C)O)=O)C3)CCCC2)=O)CNc2ccccc2O1 c1(C(=O)NC2CCCN(C(c3cc(OC)ncn3)=O)C2C)ccc(Cl)c(F)c1N N1(C(c2cc(C)c(C)[nH]2)=O)C2CCC1CC(NC(C1(F)CCCC1)=O)C2 C1(O)(C(N2CC(CNC(CCC)=O)OCC2)=O)CC2CCC1C2 CCCCC(CCCC)NC(c1cncc(CNC(=O)C(F)C(F)(F)F)c1)=O N1(C(C#CC(C)C)=O)CCN(C(c2cc(CF)on2)=O)C(C(C)C)C1 C(c1cc2ccccc2o1)=CC(N1CCC(N(C(C(C)OCC#C)=O)C)C1)=O CC1(C)CN(C(=O)C(F)OC(F)(F)F)CC1CNC(c1cnns1)=O C1(NC(COCc2nnc(C)s2)=O)CCCCC1.C(=O)C(C)(O)C1CCC1.C c1(NC(C=C)COC)cc(S(=O)(=O)N2CCSCC2CO)ccc1C#N C1(CC(=O)OC)CCCCN1C(C1CCN(C(=O)C(C)C2(O)CCC2)C1C)=O c1(CC(=O)NC2C(NC(C3CCC(C)(C)C3)=O)CCC2)ncn2c1CCC2 C1(NC(C(C(C)C)F)=O)CCCCC12CCN(C(C1(C)COC1)=O)C2 S(=O)(=O)(C1CCC2CCC1OC2)NC1(c2c([N+](=O)[O-])cccc2)CC1 c1(C(=O)NCCN(C(c2ccc(SC(F)(F)F)s2)=O)CC)ncn(C)n1 n1(CCC)cc(-c2nnc(SCCc3ccccc3)n2-c2cccnc2)c(C)n1 N1(C(C2OCCN(CC)C2)=O)CC(N(C)C(c2cnn(C)c2C#N)=O)C2(CC2)C1 CC1CN(C(C2CC3C=CC2CC3)=O)CC1(C)CNC(c1n[nH]cc1F)=O N1(C(c2ccc(F)o2)=O)CCC(N(C(=O)Cc2ccn(CF)n2)CCO)CC1 N1(C(C(CC=CC)NC(c2ccc3[nH]nc(Cl)c3c2)=O)=O)CC(C)OCC(C)(C)C1 c1(C(=O)NCCN(C(=O)Cc2cccs2)C(C)C)nnc(O)c(Br)c1O C(C#Cc1ccc(C(=O)O)cc1)N(C)C(C1CCN1C1CCCC1)=O C1(CC(=O)NC2(CCNC(c3nn(C)c(Cl)c3)=O)CCC2)CCC2(CCC2)O1 C1(C(=O)NCCC2(CNC(C(CC)(C)CC)=O)CC2)CCc2nncn2C1 CC(C(=O)NC1CC1NC(=O)COc1ccc(F)cn1)S(N)(=O)=O C(C(C)(C(=O)NCC=C1CCN(C(C2(C(N)=O)CC2)=O)CC1)OC)OC C=CCCCC(=O)N1CCC(OCCNC(=O)C(C(C)C)NS(N)(=O)=O)CC1 Cc1cc(OCCNC(N2CC(CO)OC(C)C2)=O)ccc1Cl c1(OC)ccc2c(N3CCOC4(CC4)C3)nc(N3CC4CC4(CO)C3)nc2c1 CC(C)C(C)(O)C(=O)NC1CC2(C1)CC2C(=O)NC1C(C)CCC1C c1(C(N(CCC)CCNC(=O)Cc2n[nH]c(C)n2)=O)c(Cl)nn(C)c1Cl O=C(CN1CCCc2ccccc21)N1N=C(c2ccc(Cl)cc2)CC1C(F)F c1(OC)cc(F)c(Cl)cc1C(=O)N(CC)C1CC1.n1(CC=O)nccn1.N C(=O)(C(C)(C)Cc1cnn[nH]1)N.c1(C(=O)OC)cscc1C(=O)NCCC N1(C(COC2(C)CCCC2)=O)CC=CC(C(N2CCC(OCC3CC3)C2)=O)C1 C(=O)(C1=CCCCCC1)N1CCN(C(C)CNC(C2CC(F)(F)C2)=O)CC1 C1(C(=O)OCC)CCN(C(=O)Cc2sc(C)nc2-c2ccc(C)cc2)CC1=O c1(CC)ccnc(Oc2nc(C(N3CCCC3CNC(=O)C)=O)co2)c1.O O=C(C1=CCCSC1)N1CCN(C2CCN(C(c3cc(Cl)c[nH]3)=O)C2)CC1 N1(C(C(C2CCCC2)OC)=O)CCOC2(CCN(Cc3cscn3)CC2)C1 C1(NC(Cc2c(C)ocn2)=O)CCCC12CN(C(=O)CSC1CCOC1=O)C2 c1(CC(N2CCCC(CN(C)C(C3CCO3)=O)C2)=O)cc(F)cc([N+](=O)[O-])c1 c1(CCC(=O)N(CCC)CC)ccc(N(C)C)cc1.C(=O)CCC1CCCO1.N C(=O)(C(CO)C(F)(F)F)NC12CCN(C(c3ccc(CC#N)cc3)=O)CC1C2 C(C)(C(C(=O)NCC1CC1C1CCC1)C(C)C)NC(C1CC(=C)C1)=O C1(C(N(C2CCN(C(=O)CCC3CCCCC3)C2)CC)=O)COCOC1 N1(C(C2CN(C(C)C)C2)=O)C2CCC1CC(C(=O)NC1CC(C)OC1=O)C2 c1(C(=O)NC(CNC(CC=CCC)=O)(C)C)c[nH]cc(Cl)c1=O c1(C(=O)NCCCCC(C)NC(Cc2scc(C)n2)=O)cnn2c(C)cccc12 Cc1onc(-c2cccc(Cl)c2)c1C(=O)N(C)CCNC(=O)CCC1CC1 N1(C(CCC(C)C)=O)CC2CCC1(CNC(=O)CS(=O)(=O)C1CC1)CC2 C1CC2CC1CN(C(=O)C(c1c(C)noc1C)(C)C)C2.S(=O)(=O)(CC(=O)N)NC CC(C)C(C)(C(N)=O)NC(C1CC12CC(NC(=O)CCCC1CC1)C2)=O CCC(C)C=CC(=O)NCCOCCN(C(=O)COCCC(C)C)C N1(C(C#C)=O)CCC(C2CN(C(c3c(Br)ccc4c3OCO4)=O)C2)CC1 N1(C(C(C(C)O)(F)F)=O)CC2CCCC2(NC(=O)Cn2ncc(C#N)c2N)C1 C12(C(N3C(C4CCN(C(=O)C=CCO)CC4)CCCC3)=O)CCC(F)(CC1)CC2 CC1(C)CCC=C(C(=O)NCC2(C3(O)CN(C(=O)C=CCO)C3)CC2)C1 c1(C(=O)NCC(C2CC2)NC(c2ccnnc2)=O)ccnc(N2CCCC2)c1 C1(NC(C(CC#C)O)=O)(COC)CCCN(C(C2CN3CCN2CC3)=O)C1 c1(C=O)c[nH]nc1[N+](=O)[O-].Cc1ncccc1C(=O)NCC12COC(C1)C2.C C#CC1(NC(=O)CC2(C)CCN2C(C2(CSC)CCC2)=O)CCCOC1 c1(CC(=O)NC2CN(C(C(CC=C)C)=O)CC2F)cccc(C)c1Cl C1(NC(C(C2CC2)OCC)=O)C=CCN(C(c2nc(C)oc2OC)=O)C1 Cc1nnc2c(C(N3CC(CCCCNC(=O)C(C)(C)C)C3)=O)nccn12 c1(CCN(C(CN(CC(C)N)CC)=O)C)cccs1 n1(CC(=O)N(C)C)c(N2CC(C(N)=O)C(SC(F)F)C2)nnc1C1(C)CC1 c1(C(=O)NC2C3CC2N(C(C2CC2(Cl)Cl)=O)C3)cnc2n1CCOC2 CC(C)CCC(C(=O)NCC(O)CCO)NC(=O)Cc1csnn1 N1(C(C2(C)CC2c2ccccc2)=O)CC2CCC1CN2C(C1CCC(F)(F)C1)=O c1(C(=O)NC2C(NC(c3cnn(C(C)C)c3F)=O)C2)cc(F)cc2nc[nH]c12 C(=O)(CC(C)C(F)(F)F)NC1CCC(CNC(C2=C(C)CCC2)=O)CC1 c1(C(=O)OC)cc(S(=O)(=O)N2CCc3[nH]nc(C(F)(F)F)c3C2)c(F)cc1Cl C1(C2CCN(C(c3cnn(C4CC4)c3)=O)CC2)CC1.c1(CNC=O)ccsc1 C1(C(=O)NC(c2cnnn2C)CC)CCCCN1C(=O)C.c1ncc[nH]1 C(=O)(CC(C)(C)CCOC)N1CCC(NC(c2nc(CCC)oc2)=O)C1C C1(NC(CC(CC)C)=O)COC2(CCN(C(c3ccc4sncc4c3)=O)CC2)C1 CS(=O)(=O)C1CCN(C(C2(CNC(c3cccc(O)c3)=O)CC2)=O)CC1 C(=O)(C(C)CC(F)(F)F)N(C)CC1N(C(c2c(OC)ncc(C)c2)=O)CCCC1 C(=O)(CCC(F)(F)F)N(CCOCCNC(C(C(C)C)N(C)C)=O)C N1(C(c2c(C)csc2)=O)CCC(O)CC1C(=O)NCc1nc(N(C)C)no1 c1(NC(C(C)C2CCC2)=O)ncc(-c2cnc(N3CCN(C)CC3)nc2)cc1O C1(CNC(=NCCOC)NC2COCC2F)(CF)CC12CCOCC2 c1(CNC(=O)C(O)C2CC2)ccc(C(N2CCC(NC3CC3)C2)=O)cc1 c1(C(=O)NC(C(C)NC(c2cn(C3CC3)nn2)=O)C)cc2c(cc1F)NCCC2 c1(N(CCC)C)ccc(C(=O)NCCCn2cc(CN=c3[nH]ncs3)nn2)cc1 c1(CC(=O)NCC2(CO)N(C(C(C=C=C)C)=O)CCC2)ccc2nn[nH]c2c1 N1(C(CC2CN(C(c3ncc(NC)nc3)=O)C(C)C2)=O)CCC12CCCCC2 O(NC(=O)C(O)CCCNC(=O)CC1CCCO1)CC=C(C)C N#Cc1ccnc(N2CCC(OCCNC(c3csnc3Cl)=O)C2)n1 N1(C(C(CC)c2ccccc2)=O)CCC(CC)(NC(c2cnn(C)n2)=O)CC1 c1(CCC)ccc(OCC(=O)N(CC)C(C)C)cc1.C(=O)CC.CC(C)C.N c1(CCC)nc(=NCC2CCC(NC(c3ccn(CCOC)n3)=O)C2)s[nH]1 Cc1ccc2nc(-c3cn(C(c4ncc(Cl)cc4Cl)C)nn3)ccc2c1 N#Cc1c[nH]c2cccc(C(=O)NCC3CC(O)CN3C(=O)COCCF)c12 N1(C(CN(C)CCO)=O)CC2CCCC(CNC(=O)CS(=O)(=O)C3CC3)C2C1 c1(C(=O)NCCN2CCN(C(c3n(C)cc(Cl)c3)=O)CC2)cn(C)c(=O)nc1O C=C(C)CCCC(=O)N1CC=CC(NC(c2ccnc(C(C)(C)C)c2)=O)C1 N1(C(CC(COC)(C)O)=O)CCC(C2CCCN(C(c3cnn(C)c3C)=O)C2)C1 Cc1ncc(Br)c(N(CCC2CCCNC2)Cc2ccc(F)nc2C)n1 c1(CNC(C2N(C(C3(CC)CCC3)=O)CCCC2)=O)ccc(O)c(Cl)c1 c1(C(N(CC(=O)N(CC(O)C2CCC2)C)C2CC2)=O)occ2c1CCC2 N1(C(C(C)=C2CC2)=O)CCCC(C)(C)C1C(=O)NC(C)Cc1ccccn1 C1(C(C(N2CC(C)(COC)C2)=O)C)CCCN(C(=O)CC2(O)CCC2)C1 C(CC#C)(CC(=O)NC(C)(COC)C1CC1)NC(COCC#C)=O C(=O)(C(C)CCOC)NCC1(C)CC(NC(c2nc(CC)sc2)=O)C1 Cc1sc(-c2ccccc2N2CCCCC2)nc1C(=O)N(CCO)CCO C#CC1(O)CC(C(=O)NCC(C2CCCCC2)NC(c2[nH]nnc2CC)=O)C1 Cc1ccc2c(c1)CN(C(c1sc(=O)n(C)c1Cl)C(=O)NC1CCOC1)C2 C(CC(C)CCNC(=O)Cc1ccsn1)NC(CCSCC(C)C)=O Cc1cncc(CCC(=O)NCC(C)(O)CNC(C2CC2C(C)(F)F)=O)c1 C1(NC(COCC)=O)CCCN(C(c2ccc(C)cc2)=O)CC1.[SH](=O)(=O)CC CC(C)S(=O)(=O)C(C)C(=O)NCC1COCCN(C(c2cncn(C)c2=O)=O)C1 C#CCC(C)(C(=O)NCC1CCCC(C)C1)NC(c1cc(=O)n(C)cn1)=O c1(CC(=O)NCCC2CC(NC(=O)C(=O)NC)C2)cncnc1.C1CC1 c1(C(=O)NCC2(NC(c3ccnc(C)c3N)=O)CC2)cnc(O)c2cccnc12 S(=O)(=O)(c1c[nH]ccc1=NCc1ccccc1C1CCC1)N1C(C)CCCCC1 C1(C)(C(=O)NCC(CCC)OC)CN(C(c2ccc(C(N)=O)[nH]2)=O)CC1C N1(C(C2CCCC(OC)C2)=O)CC2CCCC(C1)N2c1ncccn1 C1(C(N2CCCCC2)=O)(OC)CCS(=O)(=O)C1.c1(C(=O)N)ccc(C)c(O)n1 C(=O)(CC(C)CC(=O)N1CCC(C)(CNC(C2(O)CCOC2)=O)CC1)OC Cc1ccc([N+](=O)[O-])cc1C(=O)N(C1CCN(C(=O)C(C)(C)CO)C1)CCO C1(NC(c2c(C)nn(C3CC3)c2)=O)CC(NC(C2(F)CCCC2)=O)C12CCC2 c1(OC(CNC(C=C)COC)=O)ccc(C)cc1[N+](=O)[O-] c1(OC)ccc(C(N2CCC(CO)(NC(=O)C(F)=CC3CC3)C2)=O)nn1 C1(C(=O)NCc2onc(CC)n2)CCCCCCN1C(=O)C(N)=O C1(O)(CC=O)CCCN(C(c2cc(Cl)c[nH]2)=O)C1.CCCCC1(C=O)CC1.N C(=O)(C1=CCCCCC1)NC1CCC(C)(CNC(C23CC(F)(C2)C3)=O)C1 c1(CCCC(=O)NC(CNC(C(=O)NCC)=O)C)ccc2c(c1)OCCCO2 N1(C(CC)C)CCN(C(=O)C(C2CN(C(=O)CCn3cc(C)cn3)C2)OC)CC1 c1(C(N(C(C(=O)NC(CCC=C)C)(C)C2CC2)C)=O)ccc(CF)cc1 C1CC(C)CN(C(c2c(C)nn(C)c2C(F)(F)F)=O)C1.Cc1cc(C=O)ns1.N CCC(C(F)(F)F)NC(C1COCCN1C(c1ccn(COC)n1)=O)=O c1(C(C)C)nc(C(=O)OCc2cc(C3CC3)on2)co1 CC(C)C(O)C(C)C(=O)N1CCC(C)(NC(=O)CCC(=O)N(C)C)CC1 Cc1cnc2nccc(C(=O)NCC3(NC(=O)CS(=O)(=O)CCO)CC3)c2c1 C1(NC(c2ccc(CC)s2)=O)C2CN(C(c3ncncc3C)=O)CC12 C1(CC)CCOCC1(c1nnnn1C(C)(C)C)NCc1cccs1 C1(NC(C2COCCN2C(=O)C=C(C2CC2)C2CC2)=O)CCC=CCCC1 c1(C(=O)NC2CCC(CC(=O)OC)C2)cc(N(C)C)cc(C#N)c1 CC(C)CC(F)(F)C(=O)N1CCCN(C(C2CCCN(C)C2)=O)C(C)C1 CC(C)(C)C(C(F)F)NC(=O)CC1CC(F)CN1C(C1CC1)=O.C(C)=O N1(C(C=CC(=O)N(C)C)=O)CC2C=CC1C(C(N1CC(CO)(CO)C1)=O)C2 C1(NC(c2ncc(OC)cn2)=O)CCOC12CCN(C(=O)C(C)C(C)(C)C)CC2 CC(C(=O)N1CC(S(N)(=O)=O)C1)C(C)(C)C.C1(C)(OC)CN(CC(=O)N)C1 c1(CC(N2CC(O)C2)=O)ccccc1C(F)(F)F.c1(C(=O)N)csc(O)n1 c1(NC2CCCC(NC(c3c(SC)nccn3)=O)C2)ncnc2ccc(Cl)cc12 C(C)(C(C)C(C)(C)C)Sc1n(CCOC)c(-c2cccc(C)c2)nn1 C1(NC(CNS(N(C)C)(=O)=O)=O)CC(N=c2[nH]c(Cl)nc3c2CCC3)C1 c1(C(N2C(C=O)COCC2)=O)ccc(I)c(F)c1F.C(=O)(CC)NC(C)(C)C.N C1(C(=O)NC(C(=O)NCCCC)C)CC(O)(C=O)C1.C1CCC1.C1CC1 N1(C(C)=O)CCC(C(N2CC(C)CC2c2cccc(F)c2)=O)C(O)C1.N(C)C C#Cc1ccc(C(N2CC3CC2C3C(=O)NC(c2n[nH]c(C)n2)C)=O)cn1 N1(C(C(CCC)CC2CCCC2)=O)C2CCC1CC(CNC(=O)CC1CC1C)C2 C(=O)(C1=CNC2=NCCCN12)NC1CCC(NC(C(C)(C)c2cccs2)=O)CC1 C(=O)(CCCS(=O)(=O)N1CCCC1)N(CCC(C(C)C)NC(=O)CNC=O)C c1(NC(CC2(C=C)CN(C(C3CC=C(C)CC3)=O)C2)=O)cc(C)cc(C)c1O C1(NC(C2(O)CC(C)(C)C2)=O)CCC2(CC1)CC2.C1(CCC=O)CCCCC1.N C1(NC(CCNC(C)=O)=O)CN(C(=O)Cc2c[nH]nc2O)CC2(CCC2)C1 c1(C(=O)OC)ccccc1C(=O)NCC.C1(O)(C(C=O)(F)F)CCCCC1.N N1(C(=O)CCC2(NC(C3C=CCS3)=O)CCC2)CCC2(CCCC2)C1 C(=O)(CCCCCC#N)N1C(C(=O)NCC(=O)N(C)CC)CC=CC1 C1(NC(=O)C=Cc2ncc[nH]2)CCC(NC(=O)C(N2CCCC2)C2CC2)CC1 CC1CC(C(=O)NC2CC(C)(C(N)=O)C2)N1C(=O)CCCC1CCC1 c1(CN(CC(C)C)Cc2ccn(CC)n2)ccc(F)cc1Br CN(Cc1ncn(C)n1)N1CCN(C(=O)Cc2cccnc2)CC1 N1(C(C(CSC)C)=O)CCC(O)(CN(C)C(c2nc(Cl)cs2)=O)CC1 c1(C(=O)OC)n[nH]c(=NCCC2CCC(NC(c3cscc3C(F)F)=O)C2)s1 C(=O)C(CO)C(C)(C)C.c1(OCC#C)cccc(C(=O)NCC2CCC2)c1 c1(NC(=O)NC2CC(C3CCN(C(C)=O)CC3)OC2)cccc2ccncc12 Cc1nc(N2CCCC2C(C)(C)CNC(c2cc(Cl)sc2Cl)=O)cc2nncn12 Cn1cc(Cl)c(CC(=O)NCC2CCN(C(=O)CC3(O)CCCOC3)C2)n1 c1(C(=O)OC)cccc(COC(C2CN(C(C)=O)CCO2)=O)c1Br C1(C(=O)NC(C(=O)O)Cc2csc(Br)c2)CCc2cc(Br)ccc2O1 N1(C(CC(CC)C(F)F)=O)CCC2(CCN(C(c3cncnc3)=O)C2)C1 C(=O)(C1=NOC(CNC(=O)Cn2cnnc2)C1)N(CCC(C)O)C CCC(CN(C(=O)CSCC(C)C)C)NC(=O)CSC(C)(C)C c1(NC(CN2CC(C(C)NC(CCCC#C)=O)C2)=O)ccc2ccccc2c1 N(C(=NCCF)NCC1CCC(C)O1)C(c1ccnc(C)n1)C c1(NC(C2(C)N(C(c3ncn(CC)n3)=O)CCC2)=O)cc(C)c(C)cc1C N1(C(C(C)c2ccco2)=O)CCN(C(c2nncn2C2CC2)=O)CC1CO c1(CCC)cc(C(=O)N(C)CC2(O)CCN(C(=O)C(C)n3cccn3)C2)sc1C c1(C(=O)NCCC2(O)CN(C(C3C=CCC3)=O)C2)c[nH]c2ccc(O)cc12 c1(NCCCC=CC)cc(=NCc2ncc(C)cc2Br)[nH]c(C(C)C)n1 CC(C(=O)NCCCC1CCCCN1C(=O)CCCC1CCCCC1)P(C)(C)=O N#Cc1c(NC(C2CC(F)CN2C(c2cc([N+](=O)[O-])cs2)=O)=O)cc(F)cc1F CCN=c1ccc(C(=O)N(CCNC(=O)C(O)CC(C)(C)C)CC)c[nH]1 c1(C(N2CCC(CNC(C(C)(O)C3CC3)=O)C2)=O)coc2c1COC2 C1(OC)CC(CNC(=O)CC2(O)CCC2)C1.C1CC12CC2.C(=O)C.N CC(C)CC(CNC(C1CCC(C)(C)OC1)=O)C(=O)NCCc1cc[nH]n1 CC(CNC(C1CC(F)(CF)C1)=O)C(=O)N1CCCC1CC1CC1 Cc1cc(CNC(=O)C(Cc2ccoc2)NC(C2CCOC2(C)C)=O)ncn1 Cc1noc(C(=O)N(C(C)CNC(c2c[nH]nc2C(C)C)=O)C)c1C O(N(CC)C(=O)C(C1(C)CC1)NC(=O)CN(C)C(=O)C1CC1)CC Cc1nnc2n1CCN(C(=O)CCC(C)NC(c1cc(F)ccc1O)=O)C2 N1(C(C(C)Cc2ccccc2)=O)CCC(F)(F)C(NC(c2ccccn2)=O)C1 C1(C(=O)OC)CCCC(C(=O)NCCO)CC1.c1(C=O)sc(F)cc1Cl.CC C(C)(C(C(C)C)NC(c1ncc(F)cn1)=O)NC(CCc1onc(C(C)C)n1)=O c1(N2CC(NC(c3cccc(Cl)c3Cl)=O)CC3(C2)CC3)ncnn2c(Br)ccc12 C=CC(C)(C)CC(=O)NC1CCCN(Cc2cn(C(C)CO)nn2)C1 CCC(CC)CC(=O)NC1CCC(CNC(c2cc(-n3cccn3)ccn2)=O)C1 O=S(=O)(c1ccc2[nH]c(=NCC(O)CF)sc2c1)N1CCC2(CCCO2)C1 N1(CC2=CCC(CC)CC2)Cc2nccc(C(=O)OC)c2C1 c1(CCC)ccc(C(=O)NCC2(O)CCN(C(C3CC=CCC3)=O)CC2)cc1N Cc1ccc(C=CC(N2CCCCC2C(=O)NCC(c2ccncc2)O)=O)o1 Cc1cc(C(=O)NCC#CC(=O)N2CCCC2CCCO)cc(O)c1 C1(C(N2CCCC(Br)C2)=O)Cc2ccccc2CN1C(c1ccc(O)c(O)c1)=O C1(C(=O)NCc2c(C(N3CCN(CC)CC3)=O)nco2)CC12CCCCC2 CCC(C)(C)C(O)C(=O)NC1CCCCN(C(=O)C#CC(C)C)C1 c1(C(=O)OCC)cc(S(=O)(=O)N2CCN(CC(F)(F)F)C3(CCC3)C2)ccn1 CC1=C(C(=O)N2CCC(C)C(CC(=O)NCc3ncc(C)o3)C2)SCCO1 Cc1cc(C(=O)NCC2CCCCN2C(c2coc(C#N)c2)=O)ccc1F C1(C#N)(C(=O)NCCc2c(C(N(CCCC#C)C)=O)c[nH]n2)CCCOC1 c1(-c2n(C)c3c(c2)cc(F)cc3)csc(=NC2CCSc3ccccc32)[nH]1 Cn1nnc2cccc(CNC(C3(N)CCC4CC34)=O)c12 C1(C(=O)NCC2(NC(C(CO)N(C)C)=O)CC2)CCc2ccc(F)cc2O1 N1(C(CC(C(C)C)C)=O)CC23CCCC2(C1)CN(c1cc(O)nc(=O)n1C)C3 c1(C(=O)NCc2cn(-c3cccc(OC)c3)nn2)cc2ccnc(Cl)c2[nH]1 C1(OC)CCC2(C(=O)NC(C)(C)CCCNC(=O)C3=C(C)OCC3)CCC12 C1(NC(=O)Nc2c(F)ccc(C)c2)CCC2(C1)CN(C(=O)Cc1ncccn1)C2 CC1(C)CCN(C(c2cn[nH]c2)=O)C1C(=O)NCc1ccon1 CN1CCN(C(=O)NCC(=C2CCOCC2)Br)c2ccccc2C1 C(=O)(CC(F)(F)C(C)(F)F)N(C1CN(C(C2=C(C)CCCC2)=O)C1)C C1(C(=O)NC(C(=O)NC(C#C)C)C)CC2CC(=O)C1O2 N(C(=NCC1CCOC1)NC(C)C1CC1)CC12CC(C)(C1)C2 N1(C(c2cnc(C)nc2O)=O)CCN(C(=O)CCC2CC2(C)C)CCC1C CC1CCN(C(=O)CCc2ccccn2)CC1CNC(c1nc(=O)n(C)[nH]1)=O Cn1cc(C(N2CCC(C)(C)C2)=O)c(O)nc1=O.C(c1ccncc1)=CC(=O)N CN1CCN(C(=O)CCc2ccc(Cl)nc2)CC1CNC(C1(C)CC1(C)C)=O c1(OC)ccc2c(c1)CCCN2C(=O)NCCNC1CCN(C2CCOCC2)C1=O C1(C(=O)NC(CC#C)C(=O)NCC2CC=CC2)CC(C)CC(=O)N1 c1(OC)cccc(C(N2CC(NC(=O)C(=O)CC(C)C)CC2C)=O)c1C C=CC(C)(CC)C(=O)NC1CC2CN(C(C3(CCc4ccccc4)CC3)=O)CC12 c1(C(=O)NCCN(C)C(c2cn3c(n2)SCC3)=O)cn(C)c2ccc(Cl)cc12 CC1CC2(CC(C(=O)NCC3CCN(C(=O)C(C4CCOCC4)O)CC3O)C2)C1 C1(C=O)CCCN(S(N)(=O)=O)C1.Cc1cc(CC(=O)N(CC(C)(C)C)C)no1.N N1(C(C2OCCC(NC(C=C(C)C(F)F)=O)C2)=O)CCCC2C(O)CC12 c1(C(N2CCC(F)(c3cn(-c4c(SC)n(C)nc4)nn3)C2)=O)c(C#N)cnn1C C1(NC(C2(C)CCOCC2)=O)CC2CC(C1)N(C(c1cc(N)ccn1)=O)C2 c1(C(=O)NCC=C=C)cc2c(s1)CCOC21CCN(CC(N2CCOCC2)=O)CC1 N1(C(C(C)OC2CCOC2)=O)CCN(C(=O)C=Cc2ccccc2)CC2(CC2)C1 c1(C(C)SCCC2CCCCC2C)ccccc1OC C#Cc1c[nH]nc1C(=O)NCC1(NC(C2CCC2C)=O)CC1 CCCC(CNc1cc(C)ncn1)C(=O)N1CCC(OCCc2ccccc2)C1 C(=O)(CN=S(C)(C)=O)N1CC(F)(CNC(C(C2CC2)SC)=O)C1 c1(NC(C2CCC(NC(C3CC3F)=O)C2)=O)ncc(Br)cc1Br N1(C(CCCc2cc(C(=O)OC)c(C)o2)=O)CCC2(CCC2)C1 N1(C(CNC(N)=O)=O)CC2C(NC(c3cnc(C4CC4)nc3)=O)C2C1 c1(C(N2CCN(C(CC(C)SC)=O)CC2C)=O)cc2c(=O)[nH]ccn2n1 c1(C(=O)NCCC2CCCN(C(=O)C(O)C(F)(F)F)C2)cc2c(cc1Cl)OCO2 c1(C(C(=O)N2CC(CNC(C3(C)ON=C(C)C3)=O)C2)(F)F)cccc(F)c1Cl c1(C(=O)NCC(CNC(C2CC2F)=O)OC)ccnc2ccsc12 Cc1cc(Cl)cc(C(N2CCC(O)(CNC(=O)C(O)CC(N)=O)CC2)=O)c1C N1(C(c2c(CNC(C(C)C3CCC3)=O)noc2)=O)CC(C)CC(C)(C)C1 CC1(C)COCC(CNC(C2CCC(n3cc(-c4ccncc4)nn3)CC2)=O)O1 N1(C(C(C(CC)C)OC)=O)CC2CN(C(c3ccc(CC)cc3C)=O)CC(C1)O2 C1(CNC(COC(CC)(C)C)=O)CN(C(c2cnn(C)c2C)=O)C(C)(C)C1 C1(F)CCN(C(=O)C=CC2(C)COC2)CC1.c1(CC)nocc1C(=O)NC C1(O)(CN(C(=O)C(C)(C)F)C)CCN(C(c2ccoc2C2CC2)=O)CC1 Cc1c(C=CC(=O)NC2(C)CCN(C(=O)C(C)(C)C3CC3)C2)cnn1C NC1CCN(CC(=O)Nc2cccc(F)c2)CC1 C(C(C)CC(=O)NC1(C(N)=O)CCC1)NC(C=C(C)C)=O c1(C(=O)NCC2(O)CN(C(=O)C(O)CN3CCCC3)C2)cn2c(n1)SCC2 N1(C(C(C)N2CCC2)=O)CC2(CCCC2NC(C2Cc3ccccc3N2)=O)C1 CCC(CC(C)C)C(=O)N1CCC(C)C(NC(=O)C(c2ccc(F)cc2)C)C1C C1(C(N(CC(=O)OC)C)=O)CC2C=CC1N(C(C1(OC)CCC1)=O)C2 c1(C(=O)OCC(CN(C)C)N(C)C)ccc(C)cc1-n1cccc1 C(=O)(CC(C)(C)COC(C)=O)NC1CCN(C(CCCC=C)=O)CC1 C#CCC(C(=O)N(C)CCc1ncccn1)NC(=O)CCc1cnn(C)c1 C(=O)(CC(C)CC(C)(C)C)N1CC(C(=O)NC2CCC(C(C)O)CC2)N(C)CC1 c1(CC)ccc(C(=O)NC2CCCC(NC(=O)Cc3c[nH]ccc3=O)C2)c(O)c1 N1(C(CC=CC)=O)CC2CCC1C(CNC(=O)C(C)Cc1ccccc1)C2 Cc1ccc(-c2ccc(CNC(=O)NCC3COCC(=O)N3C)o2)cc1C C12(C(=O)NC(C)CC3(O)CCC3)CCC(CC1)C2.C(=O)(CC(C)(C)C#N)N Cc1csc2c(C(=O)NC3CCN(C(=O)C(F)C4CCOC4)CC3)ncnc12 Cc1nc(Br)oc1C(=O)NC(C1CCN(C(=O)Cc2ccon2)C1)(C)C C(CCCC(=O)NC1CC(C)N(C(=O)CCC(=O)N2CCOCC2)C1)NC(C)=O N1(C(c2c(C)n(C)nn2)=O)CCC2(CCCN(C(C3(S(C)(=O)=O)CC3)=O)C2)C1 C12(C(N3CC(C#C)OCC3)=O)CCC(CC1)N(C(=O)CCC(C)(C)OC)C2 C(C1c2ccsc2CCN1C(C1COC(=O)O1)=O)NC(COCCN(C)C)=O N#Cc1c[nH]cnc1=NCC1(O)CN(C(=O)C(O)Cc2cccc(Cl)c2)C1 C(c1cc(Cl)ccc1Cl)=CC(N1CC2(C1)CN(C(=O)C(F)(F)c1ncc[nH]1)C2)=O CCC1=C(C(=O)NCCC2(C(=O)NC3CCN4CCCC4C3)CCC2)CCCO1 Cn1cnc2c1CCCC2C(=O)NC1COC2(C1)CN(C(c1c[nH]cc1Br)=O)C2 C(=O)(CCC(=O)NCC1COCC1)OCC.C1(C(=O)N)CC(=O)N(O)C1 C1(NC(C2(N=[N+]=[N-])CC2)=O)CCCN(C(C2CC23CCOC3)=O)CC1 N1(C(C2CCN(C(C)=O)CC2)=O)CCC2(CCN(C(c3ccc(=N)[nH]n3)=O)C2)C1 C(C1CCCC1)=CC(=O)NCC(CNC(c1ccc(C)s1)=O)OC C1(C(N2CCC(N(c3ncnc(C)c3F)C)C2)=O)CC(c2ccccn2)=NO1 N1(C(C2(C=C)CCCC2)=O)CCC2CCCC(C1)N2C(=O)CC(C)C(C)C C1(NC(C(C)=C2CC2)=O)CCC2CN(C(C3CCc4ncncc4C3)=O)CC2C1 C12CCC(CC1n1ccnc1)C2.C1C=CC1C=O.CC(C)C.C=O.C1CC1.N c1(C(N2CCC(O)(CCNC(CC(CC)C)=O)C2)=O)cc(OC)cc2c1OCC2 CCC(C)(C)C(=O)C(=O)NC1(CNC(c2ncsc2C2CC2)=O)CCCC1 C(=O)(C1CCc2cccc(O)c21)N1CCCCCC(N)C1 c1(C(N2CCOC3COCC23)C(=O)NCCOC)ccc2nc(C)sc2c1 c1(C(N2CC3(C2)CN(S(=O)(=O)CCCl)C3)=O)cccc2nscc12 c1(C(N2C(C)CN(C(C3CCOC4CC34)=O)CC2)=O)cc2ccccn2n1 c1(C(C2CN(C(=O)OCC)CCC2C(F)(F)F)=O)cnc2scnc2c1 c1(C(N2CCC(C(C)NC(c3ccc(CCC)[nH]3)=O)C2)=O)cnn2ccn(C)c12 C1(NCC(=O)N(C(=O)Cc2ccc(Cl)cc2)CCOC)CCCCC1C c1(C(C)C)ncc[nH]c1=NNC(=O)c1cccc(NC(N2CCCCC2)=O)c1 Cc1ccc(C)c(C(=O)NC2CC(O)C2CC(N2CCC2CC2CC2)=O)n1 C1(C)(CC)CCN1.N1(c2c(C(=O)OCC)ccs2)CCC(C(=O)ON)C1=O C1(C2CCN(C(=O)CC(C)n3cccn3)CC2)(NC(CC(CC)SC)=O)CC1 Cc1nn(C)c(C)c1C(=O)C(=O)NC1CCN(C(c2ccccc2F)=O)C1 C1(C(N2CCC(CNC(c3cc(C(C)(C)C)no3)=O)C2)=O)CC2CCC(C1)O2 C(=O)(CCCC(=O)NCCC1CCCN(C(c2n[nH]cc2Br)=O)C1)OCC C(C)(CC(=O)NCC(C1CC1)NC(c1coc(C)c1)=O)SC N1(C(C=CC)=O)CCC2CN(C(=O)CC3CCCC3O)CC2C1 CCS(=O)(=O)CC(=O)NCC1(C(=O)NC2CC2)CC=CC1 N1(C(CCCc2ccc(C)s2)=O)CCC(CF)(NC(=O)C(C)C(F)F)C1 N1(C(CC2(CC=C)CCCC2)=O)CC(NC(=O)C(O)C(F)(F)F)C2(CC2)C1 C(CCNC(=O)C(C)CO)(C(C)C)NC(c1cn(CCCC)nn1)=O Cc1cc([N+](=O)[O-])ncc1C(=O)N(C(C)CNC(C1CCCC(C)(C)O1)=O)C C(CC(=O)NOCCOC)C1CCC(NC(c2ccc(CC)o2)=O)C1 c1(OC)ccc(O)c(CNC2CC2C(N2CCCC2c2ccncc2)=O)c1 c1(C(N(CCNC(COCCC#C)=O)C)=O)cccc2cccc(Cl)c12 N1(C(C2C(CC)C2)=O)CCN(C(c2cn(C(C)C)nc2C)=O)CC1C1CCC1 c1(C(=O)NC(C(C)NC(c2c(C)sc(O)n2)=O)C)cccc2c3c([nH]c12)CCC3 C1(C(=O)NCC2CCCN2C(=O)C)CCC2(CCC2)C1.c1(CC)ccccc1 N1(C(C(C2CCOCC2)OC)=O)CCCCC1CNC(c1c[nH]c(=N)s1)=O N1(C(C(C)Cc2cnc[nH]2)=O)CC2CC(NC(c3cc(C4CCC4)no3)=O)C1C2 c1(C(=O)NCCNC(CN2CCN(S(C)(=O)=O)CC2)=O)cc2ccccc2cn1 Cc1cnc2c(C(=O)NCC(C)(C)CNC(c3cn[nH]c3)=O)cccc2n1 C1(C=O)CCCNS1(=O)=O.c1(CC)cnc(C(=O)NCC2(CC)CC2)cn1 N1(C(c2cc(C)cc(O)c2)=O)CCN(C(=O)C(C)CF)C2CCC12 CC1(C)CC(NC(c2ccc(C#N)[nH]2)=O)CN(C(=O)CC2CCCO2)C1 c1(OC)cccnc1C(=O)NCC1CN(C(=O)C)CC1C.c1ccc(O)cc1.O c1(CC)cccc(NC(=O)C(C2(O)CN(C(=O)C=Cc3ccoc3)C2)F)c1F c1(Oc2cccc(C(=O)OC)n2)ccc(OCF)c(C(c2ccccc2)=O)c1 c1(C(N(CCNC(C(C(C)C)Cc2ccccc2)=O)C)=O)ccn2ccccc12 CC1CCN(C(=O)C=CC(=O)NC2CC2)C1C(=O)NC.c1ccccc1 C1(CNC(c2occ(C)c2)=O)CCN(c2nnc(C(N)=O)s2)CC1C C(CC(C)(C)C)NC(C1(CCC)CC1)=O.n1(CC=O)nc(C)cc1C=O C1(CC(=O)N(C2CCN(C(C3CC(C)(C)CO3)=O)CC2)CC)CCCC1(F)F CCC(CF)NC(=O)NCC(C)N(C)C c1(C(=O)NC(C(C)NC(c2c(Cl)cnc(CC)n2)=O)CO)ccc2ccnn2c1 NS(=O)(=O)c1sccc1C(=O)NC1CC(CNC(C2CCC(F)C2)=O)C1 n1(CC)ncc2c(C(N3CC=CC(NC(=O)CNC=O)C3)=O)cc(C)nc12 C(N=c1ccc(C(F)(F)F)c[nH]1)C1N(C(C(C)OCC)=O)C2CCC1C2 c1(N2CC(C)C(NC(C3CCCN(C(N)=O)C3)=O)C2)ncccc1[N+](=O)[O-] C1(C(=O)NCCOCC(=O)NC(COCC)C)CC(C(C)C)C1 N1(C(C(CC)SC)=O)CCCN(CCCCNC(c2cnc3n2CCC3)=O)CC1 N1(C(CCS(C)=O)=O)CCN2CCN(C(=O)Cc3ccc(CO)cc3)CC2C1 C#CC1(O)CCN(C(C2COCC2NC(=O)CC(C)(C)C(C)=O)=O)CC1 c1(C=O)cc2c(s1)CCOC2.C(C)(C(=O)N)NC(=O)OC.C1CC(CC)C1 Cc1oc2ccccc2c1C(=O)NCC(CNC(C1(C)CCN(C)C1=O)=O)CO C12(NC(C(C)=C3CCCC3)=O)CCN(C(=O)Cc3cnc[nH]3)CC1C2 N1(C(CCC(C)C)=O)CC(C)C(NC(=O)COC2CCCCC2)C(C)C1 C1(C)(C(N(C)CC2CCCN(C(=O)CCC(F)(F)F)C2)=O)CCC(F)(F)CO1 C1(NC(C(C)Cc2cccnc2)=O)CCCN(C(=O)Cc2nc[nH]n2)C1 c1(N(CCCCF)CC(=O)O)ccc(Oc2cccc(Br)c2)cc1 c1(CC)onc(C(=O)NC2CCC(CC(N3CCCC3COC)=O)CC2)c1C N1(C(Cn2ccc(C)cc2=O)=O)CC2CCC(CNC(=O)C(C)C3CC3)C2C1 C1(C(=O)NCC(C2CCCCC2)C)CC2C=CC1N(C(C1(CCCF)CC1)=O)C2 CC(N=c1[nH]c(Cl)nc2[nH]ccc12)C1CN(C(C2CC(F)(F)CCC2(C)C)=O)C1 Cc1ccc(N)cc1C(=O)NC12CCC(CC1)C2.C1(C(=O)N)CC2(CSC2)C1 C1(CNC(C2(C)CC2(F)F)=O)C2CN(c3cc(-c4ccccc4)ncn3)CC12 c1(C(=O)NC23CC(NC(=O)CCCC4CCC4)(C2)C3)cnc(O)c2cnccc12 c1(C(=O)NC(C)(CNC(c2ncc(Br)cn2)=O)C2CC2)c[nH]c2ccccc12 C1(NC(C2CCCSC2)=O)CC2CCC1N2C(c1ccn(C(F)F)n1)=O N1(C(CCCOCC)=O)CCCN(C(=O)CC(C)C)C(C)C1 C1(C(=O)NC(CCOC)C)CN(C(C2(Cl)CC2)=O)CC(C)(C)C1 C1(NC(C(CCC)CCC)=O)COC2(CCN(C(=O)C=CC3CCCC3)CC2)C1 c1(C(C)C)ccccc1CC(N1CCCCC1C(C)NC(=O)CC(F)F)=O C1(CNC(COCCC)=O)C(C)CCCN1C(=O)C.c1(C=O)cccs1.N c1(C(N(CCC)CC)=O)ccc(C(N)=O)cn1.n1(CCC=O)cc(Cl)cn1.N c1(N2CC(C(C)NC(c3nc(C)nc(O)c3)=O)OCC2)nc2ccc(Cl)cc2s1 C=C(C)C(CC(=O)N1CC(C)(NC(=O)CNC(=O)OC)C1)OCC.O C(=O)(C(CC(=O)OC)OC(C)=O)N(CCC)CCNC(=O)C=CBr Cc1cc(Cl)ccc1CC(N1CCC(CCNC(=O)C(C)CC(F)F)C1)=O C=Cc1cc(C(N2CC(OC)C(NC(=O)C(CN(C)C)CC)C2)=O)cc(F)c1 CC1(C(N2CCN(C(c3cccc(C(N)=O)c3N)=O)CC2)=O)CCS(=O)(=O)CC1 c1ccccc1.n1(CC)cc(CN)nn1.C1CCN(C(=O)CNS(C)(=N)=O)C1 N1(C(CCNC(C)=O)=O)CCN(C2CCN(C(=O)CN(C)C(C)C)C2)CC1 c1(C(=O)O)ccc(N2CCC(O)C2)cc1.CC(C)COCCN(C)CC.CCO N1(C(CCC(C)OCC)=O)CCN(C(=O)CCc2nncn2C)CC1C(C)(C)C CCC(C(=O)NCC1(C(N)=O)CCCC1)N(C(=O)CC1CC(C)C1)C CCC(C)(C#N)C(=O)N1CCC(C(C)C(=O)N(C2CC(C)C2)C)CC1 N1(C(c2n(CC=C)ccn2)=O)CC=C(CCNC(c2cnco2)=O)CC1 C=CCC(CC)C(=O)N1CCCC1C1(C(=O)N(C)Cc2cccc(O)c2)CC1 CC1=C(C(=O)N)S(=O)(=O)CCO1.C1(CC)CCCN1C(=O)Cc1cc(C)no1 C1(C(=O)NCCC2CCCN(C(c3cc(C)c(C)[nH]3)=O)C2)Cc2ccccc2C1 Cc1c(Br)cnn1CC(N1CC(C)(CC(=O)NC(CO)C(C)C)C1)=O c1(C(N2C(COC)CN(C(=O)C(F)(F)CO)CC2)=O)cc2cccnn2n1 c1(C(=O)NC(CC)CNC(C2(Cl)CC2(F)F)=O)cc(Br)n(C)n1 C1(NC(C(C)(C)O)=O)CCCCCC1NC(=O)C=Cc1ccncn1 c1(C(c2n(CCC)nnn2)NCC2(CCOC)CC2)c(Br)nc(C)n1C CC(C)C(CCN(C(=O)CC1CCNC1=O)CCC#N)NCC(F)(F)F c1(C(N2C(C)CCC(NC(c3c(CC)ncnc3)=O)C2)=O)cc(Cl)c(F)c(Cl)c1 C(=O)(C1CC(=O)c2ccccc21)NCCNC(=O)CC1C=CCC1 c1(C(N2CCC(Cc3cn(CC(CC)C)nn3)C2)=O)cc2c(F)c(Br)ccc2[nH]1 C1(CC)CC2(CCC2)CN1C(=O)C.C1(C(=O)N)CCC1.C(=O)CN(C)C C1(C(N(CC(=O)NC2C(CCC)C2)C)=O)CC(=O)CC(=O)N1 N1(C(C(C)(OC)NC(C)=O)=O)CCCC(SC)CC1 c1(C(=O)NCc2occ(C(=O)NCC(C(C)C)C)c2)ccc(C#N)n1C N1(C(c2c(C)cn(C)c2)=O)CCC(NC(C2(O)CC2)=O)C(c2ccccc2)CC1 c1(C=O)ccc(Cl)c([N+](=O)[O-])c1.c1(C(C)=O)cc(C(=O)NCC(F)C)co1.N c1(OC)ncccc1C(=O)NC(CC(=O)NCC1CCCN(C)C1)C1CC1 CCC(O)C(C)C(=O)N1CCN(C(=O)Cc2cncnc2O)C(C(C)(C)C)C1 c1(CN2CCC(NC(c3nn(C(CC)C)c(C)c3)=O)C2)cc(OC)c(Br)cc1OC c1(C(=O)NC2CCN(C(C(Cc3cn(C)nc3)O)=O)C2)cncc(N)c1 C1(CCNC(c2cc(C)ns2)=O)CN(C(c2cscc2C)=O)CCS1(=O)=O Cc1cccc(CNC(C2C3CN(C(c4cc(Cl)c(Cl)s4)=O)CC23)=O)n1 C=CCC(C)(C)CC(=O)NC1CCCCN(C(c2ccnc(C3CC3)c2)=O)C1 C1(NC(C(=O)NC2CN(C(=O)OC)C2)C)CC2CC(C1)CN(C(C)=O)C2 c1(C(N(C2CN(C(C(C3CCC3)OCC)=O)C2)C)=O)cc(Cl)cc(F)c1N C1(CC(=O)OC)C=CCN1C(=O)NC(c1cnn(C)c1)C c1(OC(C)C)n[nH]c(C(=O)N(C(C)C(C)(C)C)C)c1Cl c1(C(NC2CC2)=O)csc(S(C)(=O)=O)c1.CCC(C(=O)N1CCCC1)NC C1(C(=O)NC2CC(NC(CCCC#C)=O)CC2O)(OC)Cc2ccccc2C1 c1(C(N2CCC(C(F)(F)F)CC2)C(=O)NCCCC)cc2ccncc2s1 C1(NC(Cc2ccn(C)n2)=O)CCCCC1CNC(=O)C(c1ccccc1)O C(CN=c1c(C#N)c[nH]c2cc(F)cc(F)c12)C1N(C(CC2C(C)C2)=O)CC1 C(=O)(C(CCC)C(C)C)NC1(CC=C)CCN(C(=O)C(C)(C)C2CCCCC2)C1 c1(NC(=O)Nc2nc(SC)sc2)cc(C)ncc1C N1(C(c2ccc(OC(CC)(C)C)o2)=O)CCCC(C)(NC(=O)C)C1.CCO C(=O)(C1=NOC2(CCOC2)C1)NCC1(F)CCC(CNC(=O)C=CBr)C1 N1(c2c(F)cncn2)CCC2CN(Cc3c[nH]c4ncc(Br)nc34)CCC12 C1(C(C)NC(=O)Cc2ccoc2)CCCN1C(c1cc(-c2cccnc2)on1)=O CCC(CC)CC(F)C(=O)NCCCCNC(c1cnnc(C)c1C)=O C1(CNC(c2c(Cl)cn(C)n2)=O)CCCCCN1C(=O)C=Cc1nccs1 c1(CC(=O)NCC2(NC(C3CCCC4CC34)=O)CCCC2)ccc2nc[nH]c2c1 N1(C(c2n(CC)ccc2)=O)CCCC2CN(Cc3csnc3OC)CC12 C12(CNC(C3C(C)(C)COC3)=O)CCC1CN(C(=O)CC=C(Cl)Cl)C2 C1(C#N)(C(=O)NCC2(CCNC(C(C)c3ccsc3)=O)CC2)CCCOC1 C(=O)(CC1=CCN(C)CC1)N(C1CCCN(C(C(C)CC2CCC2)=O)C1)CCF c1(C(C)C)ncc(Cl)c(C(N2CCCC2CNC(C2CCCC(F)C2)=O)=O)n1 c1(C(N2C(C)CCC(NC(c3cc(C)n(C)n3)=O)C2)=O)n[nH]c2ccc(F)cc12 N1(C(C(CCC)C)=O)CCCC(C2CCN(C(C3CCS(=O)(=O)CC3)=O)C2)C1 O=C(C1=CCSC1)NC1CC(O)(CNC(c2cnn(-c3ccccc3)n2)=O)C1 Cc1nn(C)c(C)c1CNC(=O)C(=O)NC1CNC1(C)C n1(CC(N2CC(NC(C(CC=CC)C)=O)C2)=O)cc([N+](=O)[O-])ccc1=O C1(C(=O)Nc2ccc(O)c(F)c2)C2CCCC2CN1C(c1cn2c(n1)CCC2)=O C(=O)(C1=CC2(CCN(C(C3CCCO3)=O)C2)C1)N1CCC(C#CC)CC1 C1(CNC(CCCCCOC)=O)CCN(C(C2CC(OC)C2)=O)CC1(F)F C=CC(CCC)CC(=O)N(C1CCN(C(c2cc(CO)[nH]n2)=O)C1)CC CC(C)CC(C(=O)N1CCCC1CNC(c1ccc2c(c1)COCC2)=O)C(N)=O C1(CC)CCCN(C(C2CN(C(=O)Cc3ccoc3C)CC2OC)=O)C1 N1(C(C(C)(C)SC)=O)CCC(C2CCN(C(=O)CCc3cc(C)sc3C)C2)C1 Cc1cc(=NCCCOC(=N)O)[nH]c(N2CCN(c3ccncn3)CC2)n1 c1(C=O)cnc(O)c([N+](=O)[O-])c1.c1(OC)cnc(C(=O)NCC(C)CO)nc1.N c1(C(=O)NC(CNC(C(CCC)CC)=O)CO)ccc2c(c1)N(C)CC2 c1(NC(CC)CNC(C2(c3ccccc3)CC2(C)C)=O)snc(Cl)c1C#N O=C1COCC2(CN(C(=O)C(O)C3CN(C(=O)C(C4CC4)C4CC4)C3)C2)N1 c1(CC(=O)NC(C)CN(C(=O)Cc2cocn2)C)cccc(F)c1O N1(C(c2n(C)c(S)nc2)=O)CCN(C(=O)CCc2nc(=N)[nH][nH]2)CC1CCO C1(C(N2C(C)C(N(C)C)CC2)=O)CCC2(CCC2)C1 Cc1oc(C2CC2)nc1C(=O)NCCOCCC.C1(CC=O)CC2CC2C1 C1(C(=O)NCC2(OCC)CCC2)CC(C)CN1C(=O)C(C1CCCCC1)F N1(C(c2c(C)c(F)cnc2)=O)CCC2(CC1)CC2C(=O)NC12CCC(C1)OC2C Cc1[nH]c2ccc(C(=O)OC(C)C(C)(C)C#N)cc2c1C c1(C(=O)NCCc2cc(C(N3CC4C(C)(C)C4C3)=O)no2)ccc2occc2c1 C1(NC(c2nsnc2O)=O)CN(C(=O)CCC2CCOC2)C2(CCC2)C1 N1(C(c2c(C)nc(O)s2)=O)CC2CC(C)N(C(C3OCCCC3(C)C)=O)C2C1 c1(CC(N2CCCN(C(C(C(C)C)(F)F)=O)CC2)=O)ccc2nc(O)[nH]c2c1 C(=O)(C1=CCC(NC(=O)C(C)=C(C)C)C1)N1C(C(C)(C)OC)CCC1 CC(C)C1=CCC(NC(C2CCCC2C)=O)CC1.C(=O)(C(F)OC(F)(F)F)N N1(C(c2cc(CC)ncc2)=O)CC2CCC(C1)N2C(c1c(C2CC2)noc1C)=O C1(CC(=O)N(CCCO)CCC)CC(C)N(C(c2cc(OC)n[nH]2)=O)C1 N1(C(C(C2CCCC2)OCC)=O)CCN(C(c2cc(F)ccc2F)=O)CC1CC C(=O)(C1=CCC(NC(c2csc(Cl)n2)=O)C1)NC(CCC)C1CCC1 C(CC(F)CN=[N+]=[N-])NC(CCOCCCNC(C1(OC)CCCOC1)=O)=O c1(C(=O)NCC2CC(NC(C(C)c3ncco3)=O)C2)ccc(C(F)(F)F)[nH]1 N1(C(c2cnc(CC)nc2)=O)CCN(C(=O)CCP(C)(C)=O)CC(C)C1 C1(C(=O)NCC2(OCC)CCNCC2)Cc2cc(C)ccc2O1 Cc1cc(C)c(C(N2CCCCC2CN(C(=O)C(O)CN(C)C)C)=O)c(=O)o1 CCCCCCC(C)C(=O)N1CCN(C(c2cnnn2CC)=O)CC12CC2 c1(C(C)C)c(CNC(c2nnnn2C)(C)CC2CCCC(=O)N2)cccc1F N1(CC(=O)NCCCC)CCC(C)(NC(=O)CC(C)CC)C1 N(C1CCc2cccnc21)C(C(C1CCC1)NC(C1CC(OC)(OC)C1)=O)=O C(=O)(C(CCC(C)(C)C)N1CC(COC)CC1CN(C)C)NC(CC)(C)C c1(C(N2CC(CNC(c3c(C)csc3)=O)C(F)(CO)C2)=O)nc(C)c(C)[nH]c1=O c1(COC)ccccc1C(=O)NC(C)CCC.C(=O)C(C)Cc1ccncc1.N c1(-n2cc(C(=O)NC(CCSC)C(N)=O)nn2)ccc(S(=O)(=O)C(F)F)cc1 Cc1cc(F)ccc1CCNC1(c2ccc(Cl)cc2)CC1C C1(CNC(=O)NCc2ccc(N(C)CC)cc2)CCc2ccccc2O1 C(C(C)S(C)(=O)=O)NC(Cc1cc(C)no1)=O.C(=O)C(C)(C)CC1CC1.N N1(C(CSC)=O)CCC(CC(=O)NCC=Cc2ccccc2)CC1 C1(C(N(C)CC2(O)CCN(C(CCc3nc(C)sc3)=O)C2)=O)CC(=O)NC1(C)C CCC(C)CC(C)C(=O)NC1(C(=O)NCCc2c(C)n[nH]c2C)CCN(C)C1 C(=O)(C1CCCc2nccn21)NC1CCCCN(C(c2cc(C(C)=O)sc2)=O)C1 C=CCCCC(C(=O)NCC1CCCC1)NC(=O)C(O)C1CC1 C(=O)C(C)(C)CS(C)(=O)=O.N1(C(CCCNC(=O)OCC)=O)CCCCCC1 N1(C(c2c(C)nc(CN)o2)=O)CCC(O)CC1C(=O)NOCC(F)(F)F c1(OC)cc(F)ccc1C(=O)NC1CC(C)CN(C(c2cc(Cl)c(C)cn2)=O)C1 C#CCC(C(=O)N1CC(O)CC1CNC(=O)CC)C1CC1.c1ccc(F)nc1.O C1(C(=O)NCC(C)CN(C)C(c2cccnc2O)=O)(OC)CS(=O)(=O)C1 Cc1nc2n(n1)CCN(C(C1CCCN(C(=O)CCc3cscn3)C1)=O)C2 C1(NC(=O)Cc2cncnc2O)CC2CC1N(C(C1CC(F)(CF)C1)=O)C2 C1(C(N2C(C)(CNC(c3cc(C)[nH]c3C)=O)CCC2)=O)CC(=O)NC(=O)C1 C1(O)(CC(=O)NC2CC2)CCCCCC1.C1(C(N2CCCC2)=O)CCCC1.CO c1(C(N2CCC(OC3CCN(C(C4CC4F)=O)CC3)C2)=O)cc2cccnn2n1 N1(CCCC)CCCCC1C(=O)NCCC(C)N(C(=O)CNC(=O)CC)C C#Cc1cncc(C(N2CCOCC2CCNC(C2C(Cl)(Cl)C23CC3)=O)=O)c1 C1(N(CC#C)C(C)=O)CCN(C(=O)C(n2ccc(C(F)(F)F)n2)C)CC1 c1(C(C(C)NC(N(CC)CC)=O)OC)c(F)cccc1F c1(C(N2CCC(F)C2)=O)ccc(C#N)c(O)c1.C1(C(=O)NC)(C=O)CCC1.N c1(C=O)cscc1C1CC1.C(=O)(C(Cc1ccccc1)N(C)C)N(C(C)C)C.N C(=O)C(=O)N=S(C)(C)=O.C1(COC)CN(C(c2ccnn2C2CC2)=O)C1 C1(CC=C)(NC(c2ccns2)=O)CCCN(C(c2cc(Cl)cs2)=O)C1 Cc1cc(=O)n(C)nc1C(=O)N(C1CCN(Cc2cnc(S(C)(=O)=O)s2)C1)C Nc1cccc(C(=O)NCCCCCCNC(C2(CO)CC2(F)F)=O)c1 C12CC(C1)C2.c1(C2C(C=O)C2)ccccc1.N1(C(C)(C)C)CCC1C(=O)N Cc1ccc(N(C(c2nc(C(N3CCOC(O)C3)=O)cs2)=O)C(C)C)c(F)n1 CC(Cc1c(Cl)cccc1Cl)N=c1ccnc(NCc2cn(C)nn2)[nH]1 CC(C)(F)CCC(=O)N1CCC(C(F)CNC(C2CCCNC2=O)=O)CC1 CCC(CC)CC(=O)N1CCN(C(C2SC3C=CC2CC3)=O)C(C2CC2)C1 Cc1[nH]nc(C(=O)NCC2(CNC(C3CC3C)=O)CC2(F)F)c1Cl N1(C(C(CCOC)OC)=O)CCC2(CCC(NC(=O)Cc3c[nH]nc3C)C2)C1 Cc1cc(C(=O)NC(CNC(c2ccc(=O)oc2)=O)C(C)C)cc(Br)c1C Cc1cnc2n1CCC(C(=O)NCC(C)N(C)C(c1ccc(Cl)cn1)=O)C2 C1(NC(CCCC=C)=O)CC2CC1CN2C(c1c(C2CCC2)cnn1C)=O C1(C(=O)NCc2c(C)c(F)ccc2)CNCC(P(C)(C)=O)C1 S(=O)(=O)(c1ccc(C#N)c(N2CC=CCC2)c1)N1CCCC(C)C1CCO C1(CC(=O)OCC)CN(S(=O)(=O)CC#N)C(C)(C)C1 C1(C(N2CC(C)=C(C)C2)=O)CC2(CCC2)CN1C(=O)C(C)CN(C)C C(N=c1[nH]ccc(Br)c1I)c1cc(C(=O)OC)c(OCC(=O)NC2CC2)c(N)c1 c1(NC(c2ccc(C(F)(F)F)s2)C)ncc2c(n1)SCC(=O)N2 C(=O)(C1=CCCCCC1)N1CC=CC(NC(C2CC(C(F)F)(OC)C2)=O)C1 c1(C(N2CC(F)(CNC(C(C(COC)C)C)=O)C2)=O)csc2cc(O)ccc12 C1(c2nnnn2CC2CCOC2)(NCCNC(C)=O)CCC2COC1O2 C(=O)(C1=NOC2COCC12)N(CC(C)(C)NC(Cn1nc(C)c(Cl)c1)=O)C n1(CC)cccc(C=O)c1=O.C(=O)C(F)CC1CC1.CCC1CC1.CCS c1(CC)nc(N2CCOCC(CNC(C3CCNC3=O)=O)C2)c(F)c(Cl)n1 C1(NC(C(C)N(C)C)=O)CN(C(C2(Sc3ccc(O)cc3)CCCC2)=O)CC1F N1(C(c2nc(Cl)cs2)C(=O)NCCCN(C)C2CC2)CCc2ccccc2C1 c1(C(=O)NC2CCN(C(c3c(F)cncc3F)=O)C2)ccc(C(F)(F)F)c(I)c1 C1(CNC(CSC)=O)CC(F)(F)CN1C(c1ccnc(Cl)c1F)=O C(=O)(C(C)C(O)C(C)C)NCc1cc(C(=O)NC(CCCC)C)no1 CN1CCN(CCC(=O)NCCC2CCN(C(=O)CCc3cccnc3)C2)CC1 CC1=C(C(=O)N2C(C(=O)NCC3(C(O)C(C)C)CC3)CC3CC23)CCO1 c1(C(=O)NC2C(CNC(C(=Cc3cccs3)C)=O)C2)cccc2ccsc12 Cc1c(C(=O)NCC(CC(C)C)NC(=O)COC(=O)CO)nnn1C c1(C(N2CCC(F)(CNC(c3ccoc3)=O)C2)=O)cc2c(cc1Cl)NCC2 C1(C(=O)NC(C(C)(C)NC(C=C(C)C)=O)C)CCCCC1.c1ccccc1.O O=S(=O)(c1cccc(N2CCC3CCCC3C2)n1)NCC=Cc1cccnc1 N1(C(COCCOC)=O)CC(CN(C)C(C2(F)CCCOC2)=O)C2(CC2)C1 C1(CC#C)(C(N2CCN(C(=O)C(C)Cc3cnc[nH]3)CC2)=O)CC=CCC1 N1(C(c2cccc([N+](=O)[O-])c2)=O)CC2CCN(C(=O)CN3CC4CC4C3)C2C1 C1(C(=O)N(C2CCCC2)CC2CCC2)CCCOCC1 Cc1cc2c(N3CC4(C3)CN(c3nccc(C)c3C(=O)N(C)C)C4)ncnc2[nH]1 C1(C(=O)O)CN(Cc2cc(F)ccc2F)Cc2ccnn2C1 c1(CC)ncccc1C(N1CCC(CCNC(=O)CCc2nccn2C)C1)=O CC1CN(C(c2ccnn2CC(F)F)=O)CCN1C(c1ccccc1F)=O Cc1cc(C(=O)N(CCNC2CNC2)C(C)C)c(C)n1-c1cccnc1 C12CCCC1OC2=O.C(=O)(C(C)N(C)C)NC(=O)NC C1(NC(C(c2c(C)cccc2)N(C)C)C)CCC(N)C(C)C1 c1(CC)nc(C)[nH]c1C(N1CCOCC1Cc1cn(Cc2ccncn2)nn1)=O c1(C(N(CCC(=O)NCCN(CC)CC)CC=C)=O)cnc(CC)[nH]1 C1(C2(O)CCC2)(C=O)CC1.C1(C(=O)N)CCN(CC(F)(F)F)CC1.CC(C)C c1(CNCCCCNC(=O)N)noc(Cc2ccccc2)n1.C1CCCO1.C N1(C(c2c(C)c(F)ccc2)=O)CC2(CC(C(=O)NC(C3CCCO3)(C)C)CO2)C1 N1(C(Cc2n(C)ncc2Cl)=O)CCC(C)(NC(C2CSC2)=O)CC1 c1(SCC)nccnc1C(=O)NCC1CCN1C(=O)CC1CCCOC1 c1(C(N2CCC3(NC(Cn4c(C)nnn4)=O)C(C2)C3)=O)[nH]nc2cnccc12 c1(OC)ccc2[nH]nc(CNCC3COCCN3C(=O)C(C)(C)O)c2c1 C1(N(C(=O)CCO)CCC)CCN(C(=O)C(F)(F)c2ccncc2)C1.CC(F)F C1(C2CCOCC2)(C(N2CC(C)C(NC(c3cc(N)ccn3)=O)C2)=O)CC1(F)F N1(C(c2ccncc2O)=O)CCC2(CC1)CCN(C(C1(Br)CC1)=O)CC2 c1(CC(=O)NC)ccc2c(c1)OCO2.C12CCN(C1)C(=O)C1CN(C1)C2 c1(C(N2CCC(C(N)=O)(NC(=O)NC3CCCC3)CC2)C)cn2ccccc2n1 N1(C(C2(COC)CCCC2)=O)CC(NC(=O)CC(O)C2CCCC2)C(C)C1 Cn1nc(Br)c2ncnc(NC3CN(C(=O)C4=CS(=O)CCC4)CC34CCC4)c12 C1(C(N(CCC)C2CC2)=O)CCN(C2CC2)CC1.O=CC(O)Cc1cnc[nH]1.N N1(C(C2=CCN(C(CCCNC(=O)OC)=O)C2)=O)CCc2ccsc2C1 Cc1cc(=NC2CCN(C(c3cnc4ncccn34)=O)C(C)C2)[nH]c(C)c1C#N CC(C)(C)C(CNC(=O)C=CC1CCCO1)NC(C1CCC(=O)N1)=O C1(NC(Cc2cn(CC)nn2)=O)COC2(C1)CN(C(=O)C(C)CC(C)C)C2 N1(C(c2cnn(CC)c2Cl)=O)CCCC(CC)(NC(c2ccc(C#N)cn2)=O)C1 C(CCCC(=O)NC(CO)C(C)NC(=O)C(c1ccnn1C)O)(OC)OC C1(C=O)CS(=O)(=O)CC(=O)N1.n1(CC)cc(C=O)c(C)n1.CC(O)C.CO C1(C)(C(=O)NC(CC)CN(C(=O)COCCCF)C)Cc2ccccc2C(=O)O1 c1(C(=O)NCC2OCC(CNC(=O)Cc3cc[nH]c3)C2)cnc2n1CCS2 c1(C(N2CCCC(CCNC(Cc3ccc(C)s3)=O)C2)=O)nccc(C)c1N n1(CC=O)cc([N+](=O)[O-])cn1.C(C)(CC)OC.C(=O)CC.[SH](C)(=O)=O.N c1(C(N(CCCNC(C2C3CC3C3CC23)=O)CC)=O)ncc(Cl)cc1O C1(NC(c2c(C)coc2C(C)C)=O)CCCN(C(C2CC(C)OC2C)=O)CC1 N1(CC(N2CC(CN(C(=O)CCc3ccsc3)C)C2)=O)CCCCCC1 c1(C(N(C)CCNC(=O)CC2CCC23CCC3)=O)c(Cl)nc2ccccn12 c1(C(=O)NCC(CC)NC(=O)C(F)=C2CCCC2)ccc(F)cc1[N+](=O)[O-] N1(C(c2c(N)cncc2Br)=O)CCC(C2(NC(C3CCC3)=O)CC2)C1 CC(C)C(CC(=O)N1CC=CC(NC(c2cn(C)nn2)=O)C1)c1ccccc1 Cc1cccc(C)c1N(C1CCC(C)CC1)C(=O)C(C)NCC(F)F C1(CNC(C2C(C)(C)C2)=O)(CO)CCN(C(C2CCSC2)=O)C1 C1(CC)CC(CC(N2CCCC(C)C2)=O)CCO1.C1(C(=O)N)CC1.C(C)(C)C N1(C(C2CCCN(C)C2)=O)CC=C(CNC(=O)CC2CCC(C3CC3)O2)CC1 C(C(CC(C)C)C(=O)N1CCCOCC1C)NC(C=CCN(C)CC)=O N1(C(C2ON=C(C)C2)=O)CCC2CC12C(=O)NCCc1ncccc1F Cc1cc(C2CC2NC(=O)NC(CO)CCc2ccccc2)ccc1F N1(C(C(CC=C)CNC(=O)CCCC2CC2)=O)CCn2ncnc2C1 C1(C(N(C(C)C(=O)N(C)C)C)=O)CC(C)(C)CCN1C(=O)CCCC(F)(F)F c1(SC)cc(C(=O)NCC2CCN2C(=O)Cc2ccnc(C)c2)n(C)n1 c1(CNc2ccc(C(=O)Nc3ccc(OC)nc3)nc2)ccc2sccc2c1 C=CC1(C(N2CCCC(Cn3ccnc3)C2)=O)CCN(C(=O)CC)CC1 c1(C(N(C)C)=O)cc(=NC2CC(c3cccc4ccccc34)C2)cc[nH]1 c1(C(=O)NC(C2CCN(C(c3c[nH]ccc3=O)=O)C2)C)cc2n(c1)CCCC2 N1(CCCn2c(C)nc(C)c2C)CCC2C(=O)OCC2C1 C1(C(N(C2(CO)CCC2)C)=O)CCCCC1C(=O)NOCC1(C)CCC1 N(C(=NCCSC1(c2nccs2)CC1)NCc1ccc(F)cc1)C1CC(OC)C1 C1(CC)(NC(C2C=C2C)=O)CCN(C(c2cncc(C)c2)=O)CC1.C1CC1.O CC1CN(C(C2CCCC(F)C2)=O)CC1NC(=O)CCN(C)CCO COn1cnc(C)c1C(=O)NCC1CCN(C(c2cccc(F)c2Cl)=O)CC1C C1(C(=O)NC(CN(C(C2CCN(C)C2=O)=O)C)(CO)CO)Cc2ccccc2S1 CCCC(CNC(c1ccc(C#N)cc1)=O)C(=O)Nc1c(C)noc1CC C(=O)(CCCS(C)(=O)=O)NC(CNC(C(C)C=Cc1ccccc1)=O)C n1(CCOC)nc(C(N2CCCC2CN(C(C)C(=O)N(C)C)C)=O)ccc1=O C(=O)(C(C)C(O)CC(C)C)NCc1c(C(=O)NCCC=CC)con1 c1(C(N2CC(C(=O)Nc3c(C(N)=O)n[nH]c3)C3(C2)CC3)=O)ccc2occc2c1 CC(C)(C)CC1CC1C(=O)NC1CC1C(N1CC(OC(N)=O)C1)=O c1(CCS(=O)(=O)NCCS(N2CC(C)OC(C)C2)(=O)=O)cccc([N+](=O)[O-])c1 C(=O)(C1=CCCOCC1)N(C)CC1CCC(NC(C2(C)ON=C(C)C2)=O)CC1 c1(C(N2C(CC)CN(C)CC2)C(=O)NCCCF)cc([N+](=O)[O-])c(C)cc1C C1(C(F)(F)F)(OC)CC(S(=O)(=O)NCC(=O)NC(C)(C)C)C1 c1(C(N2CCC(CNC(C(C)SC(F)(F)F)=O)C2)=O)ccn(C)c(=O)c1 N1(C(c2c(C)n(C)nc2)=O)CCC2CC2(C(=O)N(C)CCc2ccccc2)CC1 CCC(C)(CC)C(=O)NC1COCCC1NC(=O)Cc1ccnnc1O N1(C(C(C)C(F)F)=O)CCN(C(=O)CC(F)(F)C(F)(F)F)CC(C)(C)C1 N1(C(c2cccc(C(C)=O)n2)=O)CCCCC1C1CC1.C1(C(=O)N)(CCO)CC1 Cc1cc(CNC(=O)COC2CN(C(C3CCN(C)C3)=O)C2)c(C)s1 N1(C(C2CCCC(C(=O)OC)C2)=O)CC(C2CN(C(c3cnc[nH]3)=O)C2)C1 Cn1ccc2ccc(CNC3CC3C(=O)NC3CNC(=O)C3(C)C)cc12 c1(CCC(N2CC(CNC(CC3CC(=O)NC3)=O)C2)=O)ccc(F)cc1Cl CC1CN(C(=O)CC2(CS(C)(=O)=O)CC2)CC(C)C1NC(C1OCCO1)=O c1(C(=O)NC2(CO)CCCN(C(c3c(C)c[nH]n3)=O)C2)ccc2c(C)noc2n1 C1(CC(N2CC(C)(NC(CCc3ccc(SC)cc3)=O)C2)=O)COC(C)(C)CO1 C1(NC(C(C)C(C)O)=O)CCN(C(c2cc(C(C)(C)C)nn2C)=O)CC1O CC1(C)CN(C(=O)CCc2cnc[nH]2)CCN(C(=O)CC2CC3(CCC3)C2)C1 C#Cc1cccc(NC(C2CCN(C(=O)Cc3nc(C)sc3C)CC2)=O)c1 CCCCC(CC)CCC(=O)N1CCC(NC(=O)C(C)CO)CC(O)C1 C1(OCC(F)F)C(Nc2ccc(COC3CC3)cc2)CC12CCC2 C1(C2CCN(C(c3c(Cl)cnn3C)=O)CC2)(NC(CC(C(C)C)C)=O)CCC1 Cc1ccc2cc(C(=O)NCC34CCC(CO3)C4)ccc2c1.C1(C(=O)N)CC1F c1(C=O)ccnn1CC(F)(F)F.c1(N(CCC)CC)cc(C2(C)CC2)n[nH]1.N C1(CCNC(C(C)=C2CCCC2)=O)CN(C(c2ncn(C)n2)=O)CC(C)O1 Cc1ncc2n1CC(C(N1CC3(CC(NC(=O)C(F)n4ccnc4)C3)C1)=O)CC2 CC(C)C(O)C(F)(F)C(=O)N1C2CCC1CC(CNC(=O)Cn1cnnn1)C2 C(=O)(N1C(C)CCCN1C)c1cccc(NC(CCC)c2cccs2)c1 C1(C(=O)NC2CCC3(C(NC(CCCCC)=O)C3)CC2)Cc2ccc(F)cc2O1 N1(C(COCc2onc(C)n2)=O)C2CCC1C(F)CC2.C(=O)(C(O)CC(N)=O)N C1(NC(C=C(CCC)C)=O)CC2CCC1N(C(=O)CCOCC)C2 C(C(=O)N1CCCC1CCCNC(C1CC(SC)C1)=O)(C(C)C)SCC C1(NC(C2(OC)CCC2)=O)CCCC(NC(C2CCC(CSC)CC2)=O)C1 N1(C(CCCN(C(C)=O)C)=O)CCC(NC(=O)CCc2ccnn2C)C1C(C)C N1(C(N)=O)CC(CNC(=O)CCN(C(=O)C(O)C2CC2)CCO)C1 C(=O)(C(C)(C)C1=CCN(C(c2sccc2CO)=O)C1)NCCn1ncc(C)c1 c1(CNC(c2nccc(CNC(C(CC)C#N)=O)c2)=O)ccc2c(c1)CC2 O(C1CCc2cccc(F)c21)C(CCOc1c(C(N)=O)cccc1)=O C(=O)(C(C)CC(N)=O)NC(c1cccc(C)c1)CNC(C1(CF)CCC1)=O C(=O)(N1CC(O)CO1)C1C(CC)N(C(=O)CC2CCOC2C)CC1 c1(C(N(CCNC(COCCC=C)=O)CCOC)=O)sc2cncn2c1C n1(C(C)(C)C)ncc(C(=O)N)c1Br.c1(C=O)cc[nH]c1C1CCC1.CC=CC N1(C(c2c(OC)ccc(Cl)c2)=O)CCCCCC(NC(C2CC3(CC3)CO2)=O)C1 CCCC(C)(O)C(=O)N1CC(C(=O)NC2(C)CCSCC2)C(C)(C)C1 S(=O)(=O)(c1cccnc1)Nc1c(C(=O)NC)cc(Br)cc1 C1(COC)CN(C(c2cn(C)cc2C)=O)CCN1C(=O)Cc1c(F)cccc1F c1(C(N2C(CNC(C3CCCC4(CC4)C3)=O)CCC2)=O)cnn2c1NCCC2 c1(C(=O)NCC(CC)NC(C(CCC)CC)=O)cc2cccc(Cl)c2[nH]1 c1(CN2CCC(C(=O)Nc3cn(CC)nn3)C2)cc([N+](=O)[O-])c(Cl)cc1F CCC(O)CC(=O)NC12CC(C(N3CCOC(C(N)=O)C3)=O)(C1)C2 C1(NC(CC)=O)C2CC3CC(C2)CC1(CNC(c1cc2cncc(C)c2s1)=O)C3 c1(OC)cc(Br)c(NC(=O)Cn2c(-c3ccccc3)nc(O)cc2=O)c(Br)c1 CCC(CC(F)F)C(=O)NC(C1CCCN1C(=O)CC(C)NC(N)=O)(C)C CCCCC(O)CNC(=O)CC1CC(NC(C2CC3CC3C2)=O)C1 N1(C(c2c(OC)ccs2)=O)CC2(NC(C3COCCC3(F)F)=O)CCCC2(F)C1 c1(CC(=O)NCC23N(C(CC(C)C)=O)CCC2CC3)ccc2[nH]ccc2c1 CC1(NC(c2cc(CNC(C3CCC3(F)F)=O)no2)=O)CCC2(CC1)CC2 c1(C(CNC(CCOCCNC(CCNC(C)=O)=O)=O)O)cnn(C)c1 C(CCO)(C(=O)NC1(C)CCN(C(=O)C(F)n2ccnc2)C1)N(C)C c1(COC)ccoc1C(=O)NC(CNC(=O)CN1CCCC1=O)CO c1(CC(=O)NCC(c2ccco2)O)ccc(Cl)cc1Cl C12(C=O)CC(CN1C1CC1)C2.c1(CC(=O)NCC2CCC2)cn[nH]c1.C c1(NC(CN2C(C)COCC2C)=O)ccc(-c2ccncc2)nc1O CC1(C)CCCC1CCNC(C1(NC(=O)CC(F)(F)F)CC(F)(F)C1)=O N1(C(c2cc(C)n(C(C)C)n2)=O)C2CCC1C(C)C2.C1(C=O)CCS1(=O)=O.N Cc1ccc2cc(C(=O)N(C)CC3CCCCN3C(C3CCO3)=O)cn2c1 C1(OC)CC2CC(C1)N(C(=O)CN(C(c1snnc1C)=O)CC1CC1)C2 CCCC(C(=O)N(C)CC1CCC(CNC(=O)CS)CC1)N(C)C.C1CC1 C1(NC(CC=C=C)=O)CN(C(c2cc(C(F)(F)F)ccc2F)=O)CCC1C N1(C(C(c2cn(C)nn2)NC(C2CCC3(CC2)CC3)=O)=O)CCC2(CCOC2)C1 CCCC(CC)C(=O)N1CCN(C(c2cccc(NCC)c2)=O)C(C2CCC2)C1 C1(C#N)(C(=O)NC(C)CC(C)NC(=O)Cn2cccnc2=O)CCCCC1 Cc1cc(C(=O)NCC2(CNC(C3OCCC3(C)C)=O)CCC2)c(C)[nH]1 C1(C=O)CCCC(C)(C)C1.c1(C(=O)OC)c(C(=O)NCC(O)C)n[nH]c1C.N S(=O)(=O)(c1cccc(=NCC(Cc2ccoc2)CO)[nH]1)N1C(C(C)C)CCC1 N1(C(CNC(=O)OC)=O)C(C(=O)N(C2CC2)C2CC2)CCC12CC2 C1(NC(c2c[nH]nc2F)=O)CC2(CCN(C(C3CCCCC3C3CC3)=O)CC2)C1 C(=O)(C(CC(F)F)N(C(=O)C(C)OC(C)=O)C)N(CCCC(=O)NC)C c1(C(=O)N)cc(Br)cn2ccnc12.C(CC(C)(C)C)NC(C1(CC=C)CC1)=O Cc1cc(C(N2CCCCC2CN(C(=O)CC2OCCO2)C)=O)n2ncnc2n1 CC1CCN(C(=O)Cn2cnc(-c3ccccc3)n2)CC1NC(=O)C(O)C1CC1 C1(CNC(CC2CC(OC)C2)=O)CCCC(NC(=O)Cc2occc2C)C1 n1(CCCSC)c(N2CCCC(C(F)F)C2)nnc1COc1ccccc1OC N1(C(CCNC(C)=O)=O)CCN(C(c2ccc(Cl)c(C(F)(F)F)c2)=O)CC1C#N C1(c2nnnn2CCSC)(NCC(=C)Cl)CCN(CC(=O)O)CC1.C1CC1.C c1(COC)cc(C#N)ccc1NCC1CCC(N)C1 C1(C(N(C(C)CC(=O)NC(C)(C)COC(C)C)C)=O)CC12CCCC2 CC1CCCCC1(N=c1ccn(CCCC(=O)N(C)C)[nH]1)c1nnnn1C1COC1 CCCC(CC)CC(=O)N1CC(C)(C)CC1CNC(C1CCC(N=[N+]=[N-])CC1)=O c1(C(=O)NCCNC(c2ccc(N(CCCC)C)cc2)=O)nccc(Cl)c1C c1(C(=O)NC(C(C)NC(=O)CSc2nnnn2C)C)ccc2nc(S)oc2c1 C(=O)(C1=C(Cl)CCC1)NCCC1C(C)CN(C(=O)CCOC2CC2)C1 CC(C)(C)C=O.C(c1ccc(Cl)s1)=CC(N1CC(CCC)C1)=O.CC(=O)N N1(C(C2(OC)CCC2)=O)CCN(C(C2CC3CC3C2)=O)C(CS(C)(=O)=O)C1 C1(Nc2nccc(SC)n2)CCN(C(=O)COc2ccn(C)n2)C(C)C1 CC(C)(CS(C)(=O)=O)C(=O)NC1COC2(CCN(C(=O)Cc3ccns3)C2)C1 c1(C(N2CC3(C(NC(C(C)=C(CC)C)=O)CC3)C2)=O)cn2cc(Cl)cnc2n1 N1(C(C2CC=CC(NC(C3CCCCC3O)=O)C2)=O)CCCC12CCC2 N#CC1(C(N2CC(NC(C3CSCC(=O)N3)=O)CC(F)C2)=O)CC2CCC1CC2 C(CN=c1[nH]cnc(NCC=C(Cl)Cl)c1C)NS(NC)(=O)=O c1(NC(=O)OC)cncc(C(=O)N(CCC(C)NC(=O)C(C)(C)C)C)c1 Cc1cccc2c1OC(C(N1CC3CCCC(C1)N3C(C1CCCC1O)=O)=O)C2 CCC(C)CC(C)C(=O)NC12CC(C1)N(C(c1ccc(NC=O)cc1)=O)C2.N C1(NC(c2ccoc2C2CC2)=O)CC2(C1)CN(C(C1CCCS1)=O)C2 c1(NC(C23C(CN(C(Cc4c(C)noc4C)=O)C2)C3)=O)cnc2cnccc2c1 C=C(C)CC(C(=O)NCC1CCCN(C(c2c[nH]cc2C)=O)C1)OC C(=O)(CCC(C)(C)C#N)NCC1(C)CCCN(C(C2CCCN(CC)C2)=O)C1 N1(C(CN(C)CC)=O)CCC(C2(NC(c3coc4ccccc34)=O)CCC2)CC1 c1(NC(C2CCCN(C(=O)C=Cc3cc[nH]c3)CC2)=O)ccc(O)c(CO)c1 C(=O)(C1=CC2C=CC1C2)N1CC(C(C(=O)NC2CCn3ccnc3C2)OC)C1 Cc1cc(C(=O)NC2CCC(CNC(c3nocc3Br)=O)C2)cc(C)c1C c1(C(N2CC3C(NC(c4coc(O)n4)=O)C3C2)=O)cc(Cl)ccc1[N+](=O)[O-] C1(C=O)CCCC1S(C)(=O)=O.Cc1nn(CC(=O)NC2(C)CCCC2)c(=O)o1 O=c1c2ccsc2c(-c2ccccc2)nn1CN(C)CCOCF C=CC(CC)CC(=O)N(CC(=O)NC(C)(CC)C1CC1)C c1(C(N2CCC(N(C(C(C=C)C)=O)CC3CC3)CC2)=O)cccc(C)c1F CC1CN(C(=O)C(C)C(C)(F)F)CC(C)N(C(c2ccc(C(=O)CF)cc2)=O)C1 c1(C(C)C(=O)NC2CN(C(=O)C(C)(C)F)CC23CC3)c[nH]c2ccccc12 C1(C#N)(C=O)CC2CCC1C2.C(C)(C(=O)N1CCC1C)SCC(=O)OC C1(C(N2C(CNC(c3c(C)nc(C)[nH]3)=O)C=CC2)=O)CCC(F)(F)CC1(C)C C(=O)(C1=CC2CCC(C1)C2)N(C1CCN(C(=O)Cn2nccc2C)CC1)CC c1(C(C(=O)NCCN(C(C2C(C)C2C)=O)C2CC2)(C)O)ccc(F)cc1 c1(C(=O)NCCC)cc2c(cc1N)OCCO2.c1(C(=O)N)ncoc1C(C)(C)C c1(NC2(CO)CCCN(C(CNC(=O)C3CC3)=O)C2)ncc2ncnc-2[nH]1 C=CCCC(N=c1[nH]c(N2CC3C(CO)C3C2)nc2c1CSC2)c1ccccc1 c1(C(c2noc(C(C)C)n2)NCCC)ccc(Br)c(C(F)(F)F)c1 CCCC(C(=O)NC1COCCC1NC(=O)CCn1cnccc1=O)NC(C)=O Cc1[nH]c(=N)sc1C(=O)N(C(C)CCNC(C1CC1c1ccccc1F)=O)C C12(C(N3CCC(C(C)O)CC3)=O)CCC1CCN2C=O.C(C)(C)(C)CC=CC C1(OC)COCCC1CC(=O)N(C1CN(C(c2sccc2-n2ccnn2)=O)C1)C c1(SC)ccc(C(N2CCCC2CCCNC(=O)CCn2cccn2)=O)o1 N1(C(c2cc(C)[nH]n2)=O)CCC2(CCC2NC(C2CN3CCN2C(C)C3)=O)CC1 CCN=C(NCCc1ccco1)NC1CCN(C(=O)CC)C1 C1(NC(CCCOCCC)=O)CN(C(=O)C(C2CCC2)OC)CC1SC c1(NCCN(C(CN2CCC(COC)(COC)CC2)=O)C)ccc2cc[nH]c2n1 C#Cc1cccc(CC(=O)N(C(C)CNC(=O)C(c2ccccc2F)(C)C)C)c1 N=c1[nH]c2cc(C(N3CC4=C(C3)CN(C(C3CC3CF)=O)C4)=O)ccc2o1 CCC(C)C(C)OC(c1n[nH]c(C)n1)=O N1(C(C(C)Oc2ccccn2)=O)CCCCC1C1CCN(C(C2(CF)CC2)=O)C1 c1(N2CCCC(CNC(C(C)(O)C3CC3)=O)CC2)ncnc2cnccc12 C(=O)(C(CO)C(C)(C)C)N1CC(C)C(CC(=O)NCC2CSCCO2)C1 C(=O)(CC(C)(C)NC(=O)CN1C(=O)CNC1=O)NCC(C)(CO)OC O=C1CCC(C2CCCCN2S(=O)(=O)CCc2cccs2)C(=O)N1 C(C)CCC(C)C.c1(OC)csc(C(c2nnnn2C)NCCOC)c1 c1(-c2c(OC)c(F)ncc2)ccc2c(c1)CN(C(=O)C(=O)C1CC1)C2 C12(NC(CN3C(C)CCC3C)=O)CCCC1N(C(=O)Cn1cnnc1O)CCC2 c1(OC)ccc(CC(N2CC3CC2CN3C(=O)C(C)(O)C2CCCC2)=O)c(C)c1 C1(C2CC2)(CNC(c2c(C)cncc2)=O)CCN(C(c2ccc(F)cn2)=O)C1 C1(NC(CSCC=C)=O)C2CC1N(C(c1ccc(CNCC)cc1)=O)C2 C(C(C)(C)CC(=O)NC1C2CC(NC(=O)C(C3CCCCC3)C)CC12)OC c1(C(C(=O)NCCCN(C(C2CN(C)C(=O)N2)=O)C)(F)F)ccc(Cl)c(Cl)c1 C(CN=c1[nH]nc(C2CC2)o1)N(C(c1cn(C)nc1COC)=O)CC N1(C(C(C)(C(C)C)OC)=O)CC(O)(C2(C)CC2)C1.c1(C(=O)N)cccnc1S C1(C(=O)NC(C)CCF)CCC(O)CN1C(=O)CNC(=O)CN(C)C Cc1ccn2c(C(=O)N)cnc2c1.C1CC2(CC2)CN1C(=O)CN1CC(C)C1.C CC1CC(C(=O)NC2COCCOC2)CN(C(c2cc(C(N)=O)co2)=O)C1 C#CC1CN(C(=O)CC2CC(O)CN2C(c2cscn2)=O)CC1O CN1CCC(C)(C(=O)NCC2COCCN(C(c3cccc(=O)n3O)=O)C2)C1=O C1CS(=O)(=O)C2CN(C(=O)C(CO)N(C)C)CC12.Cc1ccc(C(=O)N)c(O)c1 CC(C)C(C#N)C(=O)NC(C)(CNC(=O)CCn1cc([N+](=O)[O-])cn1)CO C(C(CCCC)NC(=O)Cc1cc(C)no1)NC(COCC=C)=O c1(C(=O)NCC2CCCC2)ccccc1.C1(C=O)CC(C(F)F)C1.C1CC1 N1(C(CC=CCC)=O)CCC2(CC1)CCN(C(=O)CCS(C)(=O)=O)CC2 N1(C(c2c(CC)nn(C)c2Cl)=O)CCC2(CCC2)CC1.C(=O)(C(C)CC(C)C)N c1(CC(=O)NCC(F)CNC(C2CSC2)=O)ccc(S(=O)(=O)CCO)cc1 CN1CC(C(=O)N(C2CCCC2)CCNC(C2CC2)=O)OCCC1=O.C1CC1 N1(C(c2n(C)ccn2)=O)CCC2(CC1)CC(NC(C1CC3CC3C1)=O)CCO2 N1(C(c2n(C)ccn2)=O)CCC(NC(=O)C2=CCC2)C(F)(F)CC1 N1(C(c2c(CC)non2)=O)CCC2CN(C(C3CCc4cncn4C3)=O)CC2C1 C1(NC(C(C2CCCN(C(CC3(C)CC3)=O)C2)(C)C)=O)CCOC12CCCC2 CC(C)C(C#N)C(=O)N(C)CC1CCCN(C(c2ncsc2C2CC2)=O)C1 C12(C(N(CC(C)C)C)=O)CC(C)(CN1C(C1COC(=O)N1C)=O)C2 C1(C(N2CCC2)=O)(COC)CCCN(C(C2CCCCC(=O)N2)=O)C1.C(N)=O c1(OC)cc(C)cc(C(N2CC3CCC3(CCNC(c3ccsn3)=O)C2)=O)c1O CCS(=O)(=O)CC(=O)NCC1(O)CN(C(=O)CCC2CCOC2)C1 CC1=C(C(=O)NCC2CC(C)CN(C(C3CCN(C4CC4)CC3)=O)C2)SCCO1 C=CCC(C)(C)C(=O)NCC1(C(=O)N(C)CC2CCCN(C)C2)CC=CC1 c1(C(=O)NCC(CC)NC(CC(C(=C)C)O)=O)cc(F)cc(F)c1N c1(C(=O)NC(CN(C(c2cscc2O)=O)CC)C)cc(C(=O)OC)cs1 C1(CNC(CC(C)O)=O)CC2(CO1)CN(C(c1cncc3c1CCC3)=O)C2 CCC(C)CC(C)C(=O)N1CC(O)(CCNC(=O)C=CCN2CCOCC2)C1 n1(C(C)C)cncc1C(=O)N(CCCCCNC(=O)COCC(C)(C)C)C C#Cc1ccc(OCC(N2CCC(C)C2)=O)cc1.C1(C=O)CCN1S(C)(=O)=O N1(C(C2CC(OC)C2)=O)CCN(C(c2ccn(C3CC3)c2C)=O)C(CCO)C1 C=CCC(C)(C)CC(C(=O)Nc1ccc(F)cc1C)N(C(C)C(=O)OCC)C C1(NC(C2CC(OC)C2)=O)CN(C(c2[nH]c(C)nc2C)=O)CCC1CO C(=O)(C1Cc2ccc(F)cc21)N.C(c1ccc2c(c1)CCO2)=CC(=O)NCCC c1(C(N2C(CNC(C(CCCC)N(C)C)=O)C=CC2)=O)ccnc2ncccc12 c1(C(N2CCC(NC(c3n(C)ncc3C3CC3)=O)CC2)=O)cncc(C#N)c1 C1(NC(C2CCCC(O)C2)=O)(CO)CCN(C(c2cccc(O)c2Cl)=O)CC1 c1(C(=O)NCC(CNC(C(CC)N(CC)CC)=O)F)ccc(C)nc1C CC1(C(=O)NCC2(O)CN(C(=O)C(C)(O)C3CC3)C2)CC2CCC(C1)S2 C1(C(C)C)(C(=O)NCCCC(F)(F)F)CCN(C(=O)C=Cc2nccs2)C1 N1(C(c2ccnc(C)n2)=O)CCCC(NC(c2sncc2C)=O)C1C Cc1cc(F)c(C(=O)NC2CCC2)c(F)c1.C1(CC(=O)N)CCCC2(CC2)C1 Cc1conc1C(=O)NC1(CNC(=O)C(C)Cn2cccn2)CCOC1 c1(CCOC)noc(C(C2CCCC2)NCCN)n1 C1(C(=O)NCC(C(=O)N(C(CCC(C)C)C)C)O)CC2CCC1CC2 C1(C(C)O)CCN(C(C2(c3cc[nH]n3)CC2)=O)CC1.C12CCCN1C2 c1(C(N(C(CC)C)CC(=O)O)=O)[nH]c(C)c(C=O)c1C C1(OC(F)F)(CN)CCOCC1.N12CCC(C1)n1cc(nn1)C2 C1(CC#C)CCCN(CN(c2nnc(-c3cc(C)cc(Cl)c3)n2CC(C)C)C)CC1 CC1c2ccc(Cl)c(Cl)c2CCN1C(c1cccc2c(Br)cccc12)=O C(=O)(C(COC(C1(C)CC(=O)C1)=O)Cc1ccccc1)OC C1(CC(=O)NC2CC(N(C(=O)CSCC(F)(F)F)C)C2)COCCO1 C1(NC(c2n(C(C)C)ccc2)=O)CC2(CCN(C(C3CC3C)=O)C2)C1 C1(CC)CCC(c2nnnn2Cc2ccccc2)(NC2CCC(C)(C)C2)CC1 C1(F)(CNC(c2cnc(C)nc2)=O)CCCN(C(C2(C)CCCNC2=O)=O)C1 c1(NC(CC)=O)cccc(NC(C2CN(C(C3CC=C(C)CC3)=O)CCS2)=O)c1 c1(C(=O)NC2CCN(C(C(C3CC(F)(F)C3)OCC)=O)C2)c(C)cnn1C N1(CC(=O)NC(C(C(C)C)C)CNC(c2ccns2)=O)Cc2ccccc2C1 C1(C)(C=O)CCC(=O)N(C)C1.c1(SC)ccc(C=CC(=O)N)cc1.C1CC1 c1(C(N2CCC(C(=O)NCCSC)C2)=O)cc(F)c(C)c(F)c1 c1(C=O)nocc1C(C)(C)C.C1CC(CC)C1.C1(C(=O)NC)(C=O)CC1 c1(C=O)cnnc(C)c1.C1(C(=O)NC(C)CC)(NC(=O)OC)CCCC1.N C(=O)(C1COc2ccccc21)N1CCC(C)(CNC(c2nocc2Br)=O)C1 C(CCOCC)(C(=O)N(CC(C)(C)O)C)NC(C=CCC)=O c1(C(C(=O)NCCCSCC)NCC(C)C#N)cc(C)cc([N+](=O)[O-])c1 C(=O)(CCCCC(C)=O)NC1CCCC(N(C(C(CC(=C)C)OC)=O)C)C1 N1(C(C(CSC)C)=O)CCCC2C1CCCN2C(C12C3CC(CC13)C2(F)F)=O C(=O)(CC(C)C(C)(C)NC(=O)CCOC(C)=O)NC(CCCCC)C c1(C(N(C(C)C)CCNC(=O)Cc2n[nH]c(=N)s2)=O)snc(O)c1Cl c1(CCCCC)nc(C2CCCCC2)nn1Cc1cccs1 N1(C(CCC2C(=O)NC(=O)N2)=O)CCN(C(=O)CO)C(C2CC2)C1 Cc1ccc2sc(CNC(C3CCCC3C#N)=O)nc2c1 c1(C(=O)NC2C(NC(C(c3cnn(C)c3)C)=O)C2)ccc(=O)n(C)c1 c1(C(=O)NC(CCC)CCCNC(=O)CCCF)ccc2n[nH]cc2n1 Cc1ccc(C(=O)NCCC2CCCN2C(=O)Cc2ccns2)cc1 c1(CC)ccc(C)cc1C(N1CCCC1CN(C(c1cnns1)=O)CC)=O c1(-c2ccc(SC)c(C)c2)cnc2[nH]c(C(=O)N=c3nc[nH]n3C)cc2c1 c1(C(=O)NC2C(NC(CC)=O)C2)c(C)nc(C)nc1C c1(C(=O)NC2CC(C)(NC(C(CC=C)OC)=O)C2)cc(C)cc(C)c1 CCC(CNC(=O)CCC(C)CN(C)C)(CC)C(=O)N1CCC(C(F)(F)F)C1 C1(NC(Cn2nc(C)oc2=O)=O)CCCC12CCN(C(=O)CC=C(Cl)Cl)CC2 C(=O)(C(C)C(O)C(C)CC)NC(C(N1C(C#C)CC1)=O)c1cccs1 C12(NC(C(C)C)=O)CCC(CC1)C2.C1(C(=O)N)CC(=O)NC(c2ccccc2)C1 N1(C(C(CC=C)(F)F)=O)CCC2CN(C(c3ccn(CC)c(=O)c3)=O)CC2C1 c1(OC)ccc2cnc(C(=O)NCCCNC(C3(C)CCCC3C)=O)cc2c1 C(C)(C)(CC(=O)NC1CCC(C(N2CC(F)(CF)C2)=O)CC1)OC N1(C(c2c(C)noc2C(F)F)=O)CC=C(CNC(c2ccon2)=O)CC1 C1(CNC(C(C=C)(C)CC)=O)CN(C(c2cnsc2)=O)C2CCCC2O1 CC(C(=O)NC1(CCF)CCC1)(C1CCC1)NC(C1CC2CC2C1)=O c1(CCNC(C(C2CCC2)OCC)=O)ccc(Cl)cc1 N1(CCCNC(C(C)OC)=O)CCN(C(C)C(=O)NC2CCCC2)CC1 CCCC(CC(=O)Nc1cnn(CC(N)=O)c1)NC(=O)CC1CC=CCC1 C(=O)(CCC(C)(C)F)NC1(CF)CN(C(C(C)OCCC=C)=O)C1 C=CC(C)CC(=O)NC1CCC(CNC(=O)C(CN(C)C)CC)C1 N1(C(CCC(C)(C)NC(C(CCC)C(C)C)=O)=O)CC2CCCCC2C1C C(N=c1nc(Cl)c2c([nH]1)COC2)C1CC(=C)CN1c1cc(C(F)(F)F)c(Br)cn1 CC1(C)C(NC(c2cccc(O)n2)=O)CC1CC(=O)NOCCF N1(C(C2C(=C)C2)=O)CCC2(CCC2NC(=O)Cc2[nH]cnc2C)CC1 C1(C(N(C(C2CCOCC2)C)C)=O)CC12CC(NC(=O)CCC1CCCC1)C2 c1(N(C)Cc2nc(O)n[nH]2)nc(N2CCC3OCCCC3C2)nc2c1CCC2 N1(C(c2cc(OCC)no2)=O)CCN(C(c2csc(C3CCCO3)n2)=O)C(C)C1 CC(C)(C)C(CO)C(=O)N1CCC(CCNC(c2ccc(C(N)=O)[nH]2)=O)C1 c1(C(N(C2CCN(C(c3c(C)ccn3C)=O)CC2C)C)=O)cccc2ccnn12 C1(C(N(C2CCC2O)C)=O)C(C2CC2)CCN1C(c1cccc(Cl)c1)=O Cc1cc(C(N2CCC(C(=O)NC3C4CCCC34)C23CC3)=O)ccc1O O=C(CCC(F)(F)F)NC(C12CCC(CC1)C2)C.C1(C=O)CCC(F)(F)CC1.N n1(CC(C(=O)NCCC(C(CC)C)C)(C)O)ccc2sccc2c1=O c1(C(N(C(C(=O)OCC(C)C)C)C)=O)ccc(NC(=O)C2CC2)cc1 C(=O)(CC(C)CC(=O)OC)NC(CCC)CCCNC(=O)Cc1ccc(C)cc1 C(C(=O)N1CCC1CNC(=O)C(C)C(C)(C)C)(C(C)(C)C)OC C1(NC(Cc2ncc(CC)[nH]2)=O)CN(C(c2c(CC)cccc2F)=O)CC1(C)C CC(C)CCCCC(=O)NC1CN(C(=O)CN2CCN(C)CC2)CCC1F C(=O)(C(O)CCCNC(=O)C(C)OC)NCc1c(CC)cncc1 c1(CC)ccc(CCC(N2CCCC2C2(NC(=O)C=C(C)Cl)CC2)=O)cc1 c1(C(=O)NCCCCCCn2cc(C3(C)CC3)nn2)cc(F)cc2ccoc12 c1(CC(=O)NC2CCCN(C(c3ccoc3)=O)C2)cc2c(cc1Br)OCO2 CC1(C)CN(C(=O)C(O)CC2CC2)CC1.c1(C(=O)N)ncccc1C(F)(F)F Cc1ccc(F)c(C(=O)NCC2CC(C)CN(C(=O)CCc3cncnc3)C2)n1 Oc1ccc(Br)c(NCc2nc(-c3ccc(Br)cc3)cs2)n1 c1(CC)nc(C(=O)N(C(C)C(=O)Nc2cccc(SC)c2)C2CC2)c(C)o1 N1(c2ncc(C)cn2)CCc2nc(C(=O)NCCC3=CCCCC3)cn2CC1 CC1CCN(CCNC(=O)C(Cn2ccnn2)NC(=O)Cc2cc[nH]n2)C1 C1(C(N2CCC2)=O)CCC2C(CC1)C2(F)F.C1(C(=O)N)CC2(CCCC2)CO1.C CCC(CC)C(C(=O)N1CC2(CC(NC(c3n[nH]c(C)c3Cl)=O)CO2)C1)OC N1(C(C(C(C)(C)O)F)=O)CC(NC(c2ccc(F)c(Cl)c2)=O)C(N=[N+]=[N-])C1 c1(C(=O)NC(C(C)(C)NC(c2c(C)ccc(N)c2)=O)C)cnc2occc2c1 C1(OC)CN(C(=O)C(C2CCOCC2)F)CC1C(=O)NCC(C)CC(C)C C1(C(=O)NCC(CNC(C2(CC(C)C)CCCC2)=O)(C)O)CC12CCSCC2 C1(NC(c2c(C)scc2)=O)CN(C(=O)CCN(C2CCCCC2)C)CC(C)(C)C1 CC1OC(=O)NC1C(=O)NCC12CC(CN1C(=O)COC(F)F)C2 C1(S(N)(=O)=O)(C=O)CCCC1.c1(C(=O)O)cc(C=O)[nH]n1.C1CC1.CC C1(NC(c2c(CC)scc2)=O)CCCCN(C(c2ccc(OC)c(OC)c2)=O)C1 C1(C(=O)NC(Cc2ccco2)CO)CC2CC2N1C(c1cc[nH]n1)=O c1(NC(C)C)cccc(CNC(=O)NCCc2cn(C)nc2Br)c1 C1(COC)CN(C(=O)Cc2cnccn2)CCN1C(C1CCCN(C)C1)=O C(=O)(C1=NNC(=O)CC1)N1C(C)C(NC(c2sccc2SC(F)F)=O)CC1 C1(NC(COC2CCN(C(CCC(CC)OC)=O)C2)=O)CN(C)CCN(C)C1 CC(C(=O)NCC1(F)CCC1)C(F)F.C(=O)C(Cc1ccccc1)C1CC1.C Cc1csc(C=CC(=O)NC2CC2CNC(c2cn(C)cn2)=O)n1 CC1(C)C2CN(C(c3ccc(CCC(N4CC5C(C4)C5(F)F)=O)[nH]3)=O)CC12 C1(CN(C(Cc2ccn(C(C)C)n2)=O)C)CCCCN1C(=O)CC(C)CN(C)C C(c1ccc(Br)cc1)=CC(=O)NC1CC(NC(C2(C(N)=O)CC2)=O)C1 C1(CC=C)(NC(c2ccncc2)=O)CN(C(C2CCCN2C(C)=O)=O)C1 C(C1=NOC2C3CCC(C3)C12)N1C(=O)CC(c2ccc(Cl)c(Cl)c2)C1=O Cc1ccc(Cl)cc1C(=O)NC1CN(C(=O)CC(C)(F)F)C2CC12 c1(C(N2CCC(CC(=O)Nc3ccsc3CO)C2)=O)cc(F)cc(Cl)c1 Cc1ncccc1C=CC(=O)NCCC1(NC(=O)OC(C)(C)C)CCC1 C1(C2CC2)(C(=O)NCC2CC(CNC(c3cscn3)=O)OC2)CCOCC1 n1(CCC)nnnc1C(c1cc(OC)ns1)NCC(c1nc(C)no1)(C)C c1(C2N(CC=O)CCC2)cncc(C)c1.n1(CCC)ccnc1C.CCC(C)C c1(C(C)C)c[nH]nc1C(=O)NCC1CCCC1.C(=O)C(C)(C)n1cc(Cl)cn1 c1(SC)c(C(N2CC=CC2C)=O)cccc1F.C1(CCC(=O)N)CC(F)(F)C1 CC1CN(C(c2csc(C(C)(C)C)n2)=O)CC(C)CN1C(C1CCOC1)=O c1(SCC(=O)NCCC(C)N(C(=O)C)C)ccc(C#N)cc1.C1CCCC1.O N1(C(c2n(C)nnc2CNC(=O)Cc2cc[nH]n2)=O)CC2(C1)CC(C)(O)C2 CC(C)(CCCNC(=O)CC1(C)CC1F)NC(=O)C=C1CCC1 C=CCCCCCCCC(=O)N1CC(CO)(NC(=O)C=Cc2sccc2C)C1 C1(OC)CN2CCCC2(C(=O)NC2CCC(NC(c3ccn(C)n3)=O)C2)C1 C(N=c1[nH]c(=NCCc2ncc(C)o2)[nH]c2cccnc12)C1(COC)CCC1 C1(NC(C2C3(c4c(OC)cccc4)COC2C3)=O)CCC2(CCC2)C1 CS(=O)(=O)c1cccnc1C(=O)NCC(CO)NC(C1CCOC1)=O C(=O)(C1CCCc2ccnn21)NCC12N(c3snc(COC)n3)C(CC1)CC2 C1(NC(CCC2CCN(C(c3nc(C)sc3)=O)C2)=O)CCOCC1F Cc1ccccc1OCCC(=O)NC(C)CNC(c1cc(C(N)=O)cn1C)=O C(=O)(C1=C(Cl)CCCC1)NC(C(C)NC(c1c(C)n(CCO)cc1)=O)(C)C c1(C(N(C(C)C)CC)=O)cc(=O)cc(Cl)[nH]1.c1(C=O)ccccc1.N(C)C N1(C(C2CCCC(OC)C2)=O)CC2CCC(C(=O)N)(C2)C1.C1CCC(=O)NC1.C Cn1cnc(CC(=O)NCCC(N2CCC(C3CCCO3)C2)=O)c1 C1(CC(=O)Nc2sc(C(C)=O)c(C)n2)CC2(C1)CN(Cc1nccs1)C2 CCC(O)(CC(=O)NCCCOCCNC(=O)C1=C(Cl)CC1)c1ccccc1 c1(C(=O)NCC2CCN(C(c3ccc(N)cc3O)=O)C2)ccc(F)c2c1OCC2 N(C1c2ccccc2C2CC1C2)C(N1CCCC(c2n(C)ccn2)C1)=O C(=O)(C1CCc2ccccc21)NCC(CCC)NC(c1cc(C)c(CC)s1)=O Cc1ccc2cc(C(=O)NCCNC(=O)Cc3cnc(C)[nH]3)[nH]c2c1 c1(C(=O)NC2CCC(N(C(c3c(CC)scn3)=O)C)C2)cccc2c1CCCC2 c1(C(=O)OC)ccc(CC(=O)N(C)CCN(C(C2CC2C)=O)C(C)C)cn1 CCC(C)C(=O)N1CC(C)C1C(=O)N(C)Cc1nc(C)cs1 c1(N(C)C)nc2ccc(C(=O)NC3CC4(C3)CN(C(=O)C=CCO)C4)cc2[nH]1 C1(NC(c2c(SC)cn(C)n2)=O)CC2CCC1C2.c1(C(=O)N)cc(N)cnc1C S(=O)(=O)(c1[nH]c(=NCc2nnnn2C(C)C)ccc1Br)N1CCC(OC)C1C c1(OCc2scc(C(=O)OC)n2)ccc2c(c1)nc(C)n2CCC#N C1(NC(CCCCCN(C)C)=O)CC2CCC1CN2C(c1cnc(S)[nH]1)=O C1(C#N)(C(N2CC(C)N(C(c3ccc(CCO)cc3)=O)CC2)=O)CC2CCC1C2 c1(CC)c(C(N2CCN(C(=O)CCC(C)(C)F)CC2COC)=O)cccc1F C(C1CCCc2n[nH]cc21)NC(C(=O)NCCS(N1CC(C)OC(C)C1)(=O)=O)=O C12(CNC(C3N(C)CC(C)(C)C3)=O)CCC(CC1)CO2.C(=O)(C=C(Cl)Cl)N C(=O)(CCC(C)(C)[N+](=O)[O-])N1CC(CNC(C2(CC)CCC2)=O)C(F)(C)C1 O=C1CCc2cc(C(=O)NNC(=O)NCc3cc(Cl)cc(Cl)c3)c(F)cc2N1 c1(C(=O)NC(C(C)C)CNC(=O)COC(F)F)c(Cl)cnn1C1CCCC1 c1(OCC)ncc(C(=O)NCCCC)cn1.c1(C(=O)N)ccnc(C2CCC2)c1 N1(C(c2c(C)cc[nH]2)=O)CCCC(CCNC(=O)C)CC1.N1(C(=O)N)CCCC1 N1(C(C)=O)CCCC(O)(CC(N2CCC(CNC(c3ccon3)=O)C2(C)C)=O)C1 NC(=O)CCC(=O)N1CCC(N(C(c2cccc(N)n2)=O)CC2CC2)CC1 CC1CCN(C(=O)CCc2ccco2)CC1CC(=O)NC1CC(C)(CO)C1 C1(CCNC(CNC(C2(C(=O)OCC)CC2)=O)=O)CCOC1(C)C Cc1cccc(C(C(F)(F)F)NC(C2CC(=O)N(CC(F)(F)F)C2)=O)c1 CCCCCCC(F)C(=O)NC(C)(CNC(=O)Cn1cnc(C#N)n1)C(C)C CC1(C)CCN(C(=O)C(F)CC2CCOC2)C1C(NC[Si](C)(C)C)=O C#Cc1ccc(C(=O)NCc2cccc(C(=O)NCCC(=O)OCC)n2)cc1 S(=O)(=O)(c1cccnc1NCc1cc(Cl)n(C)n1)N1CCCC(N(C)C)C1 Cc1ccc(NCC(N2CC3CCCC23)=O)cc1-c1nn[nH]n1 C1(OC)CCCC1C(=O)NC1CC(F)(CNC(C2(C)CC2(F)F)=O)C1 Cc1cccc(C(=O)NC2(c3ccc(Br)cc3)CN(C(C3CCC3)=O)C2)c1 c1(C(=O)OC)cc(C)c(C(=O)NCC2CC(O)C2)o1.c1(C=O)ccoc1 C12(C(=O)NCCN(CC(C)O)C(=O)Cc3cscn3)CC(C)(CO1)C2 CC1CC(NC(C2COC3COCC23)=O)CCN1C(=O)C(N1CCSCC1)C C=CC(CC)CC(=O)N(CC(C)(C)C(=O)N(c1ccn(C(C)C)n1)C)C C1(NC(C23CC(CO)(C2)C3)=O)C=CCN(C(=O)CC2(O)CCCCC2)C1 N1(C(C=C(CCC)CCC)=O)Cc2[nH]nc(C(=O)NCC=C3CCCCC3)c2C1 c1(SCC(=O)NC2C(CO)CCN(C(CC=CCC)=O)C2)ccccc1[N+](=O)[O-] c1(C(N(C2CCCN(C(CS(=O)(=O)NC)=O)C2)C)=O)cc2n(c1)CCC2 c1(CC)cccc(C(=O)NCC=CCC(=O)NCC2(C)CCCO2)c1 N1(C(C2N(C(c3n(CCC)ccc3)=O)CCC2C)=O)CCc2c[nH]nc2C1 c1(C(=O)NC2C(NC(CCCSC(C)(C)C)=O)CCC2)cnc2ccccn12 N1(CC(C)C)CCN(C(=O)CC2CCC2)CC1.c1(C=O)cccc(C(N)=O)c1.N c1(C(=O)NCc2cn(CCNC(CC3C(C)CCO3)=O)nn2)c(F)cccc1Cl CC(C)CC(C)(C)C(=O)NCC1CC(C)C1.c1(CCC=O)ccc(O)cc1.N C1(NC(C(C(C)O)C)=O)C2CCC1CN(C(C1(c3ccno3)CC1)=O)C2 Cc1cc(C(N2CC3C(CNC(=O)C(O)C(C)C)C3C2)=O)c(F)c(Br)c1 C1(C2CC2)(NC(C(COCC)n2cc(CC3CCCCN3C)nn2)=O)CCC1 c1(CC)ccc(C(C)=CC(N2CC(OC)CC2CCNC(=O)CS)=O)cc1 N1(C(c2c(C)cc[nH]c2=N)=O)CC2COCCC2(NC(=O)C=Cc2cocn2)C1 N1(C(c2ncn(C(C)C)c2)=O)CC2COCC(C1)C2NC(c1cc(C#N)c[nH]1)=O CN1CC2CN(C(C3(C)CCCN3C(=O)CCc3cccnc3)=O)CC2(C)C1 c1(CN(C(C)C)C(=O)Nc2ccnn2CC(F)(F)F)ccc(Br)cc1 C1(NC(c2scc(CNC(C3(C)CCNC3=O)=O)c2)=O)COCCC1(F)F C1(CC=C)(NC(c2coc(CC)n2)=O)CCCN(C(C2CCC(C)C(C)C2)=O)C1 c1(OC)cc(OC)c(NC(=O)NC(C)(C(C)C)c2nn[nH]n2)c(OC(F)F)c1 C=C1COc2c(C(=O)NC(C)(C)CCNC(C3CC34CC4)=O)cnn2C1 c1(C(N2CCN(CC(O)C(F)(F)F)CC2)c2ncc(C)s2)cn(C)c2ncccc12 C1(C(=O)NC2CCSC2)(CC)CCCN(C(=O)C(=O)NOC)C1 C1(CC(N2CC(CC)(OC)C2)=O)SC(=N)NC1=O.C1CCOC1.C(=O)(C)N CS(=O)c1ccc(C(N2CC3CCC2CN3C(C23COCC(C2)OC3)=O)=O)cc1 N1(C(C(c2cccc(OC)c2)(F)F)=O)CCC2CC2CC1.C(=O)(C=C(C)Cl)N N1(C(c2ccc(F)cc2I)=O)CC2CCN(C(=O)C3=CCCCO3)C2C1 N1(C(CSC)=O)CCOC(C(=O)NOC(CO)C(C)C)CC1 N1(C(C2(C(C)NC(=O)CCCC3CC3)CC2)=O)CC2C3C=CC(O3)C2C1 c1(SC)cccc(C(=O)NCC2CCC(CC(N)=O)CC2)c1 N(C1COc2ccccc21)C(C1N(Cc2ccc(C)cc2O)CCSC1)=O Cn1cc(C2CC2NC(=O)CNC(=O)C(F)(F)c2ccccc2)cn1 c1(C(=O)Nc2cc(CCC)no2)csc2c1CCN(C(=O)CCCCCCBr)C2 N1(C(C2(C)CC(F)C2)=O)CCC(O)(CNC(C2CCC(CO)CC2)=O)CC1 C1(C(=O)OC)N(CCCCS(=O)(=O)N2CCCC2)CCCC1(C)C N1(C(C(CC)OC)=O)CCN(C2CN(C(c3cccc(Cl)c3)CCOC)C2)CC1 C(C(CO)C(F)(F)F)NC(C1N(C(c2c(OC)cncc2)=O)CCSC1)=O C(C)(CC(=O)N1CCC(NC(c2cc(Br)n[nH]2)=O)C1)(C1CCC1)N(C)C CC1COC(C(=O)NC(C)(C)CN(C)C(c2coc(CC3CC3)n2)=O)C1 c1(CCC(=O)NCC(F)CNC(c2ccccc2)=O)csc(-c2cnccn2)n1 Cc1cc(Br)ccc1C(=O)NC1(C)CN(C(C23CCCC(C2)OC3)=O)C1 C(=O)(CC1=CCOCC1)N1C(CC(=O)NCc2ccc(C#N)s2)CC(C)(C)C1 N1(C(c2ccc(C)o2)=O)CCN(C(C2OCCC2(C)C)=O)C(CCO)C1 CCC(C)CCCCC(=O)N1CCC(c2n[nH]c(CNC(=O)CC3CC3)n2)CC1 Cc1oc(Cl)nc1C(=O)NCCN(CC(C)O)C(=O)CO.C1CCC1.C c1(C=O)cc(Br)n(C)n1.c1(C(N(C)CC2CC2)=O)cnn(CC(F)F)c1.N C1(C)CCN(C(c2c(C(F)(F)F)coc2C)=O)CC1.C#CC1(C(=O)NC)CC1 c1(C(N2CCC(N(C(CCOCC)=O)CC)C2)=O)cc2nnn(C)c2s1 N1(C(c2c(CC)nns2)=O)CCCCC1CNC(c1csnc1OC)=O N1(C(C(=O)N(C)C)=O)CC2CCC2(CNC(c2ocnc2C2CC2)=O)C1 Cn1c(C(=O)NC2CCN(C(=O)CCOCC3CCCO3)C2)cc2ccsc12 c1(C(N2C(CNC(c3nccc4n[nH]cc34)=O)CC2)=O)cnc2ccnn2c1 c1(CC)cccc(C(=O)OC2(C)N(C(Cn3cc(C(=O)OC)nn3)=O)CCC2)n1 N1(C(CCC(CC)C)=O)CC2CCC1CN2C(c1ccc(C#N)[nH]1)=O Cc1cc(N2CCC(NC(=O)N(CC(C)(C)C)Cc3nccs3)CC2)nc(C)n1 C1(C(=O)NC(C2CN(C(CSCCC)=O)C2)C)CCCC2(C1)CC2(F)F C(=O)(C(C)(C)C(C)(F)F)N1CCC(NC(CC(C(C)C)O)=O)C(O)C1 C1(NC(C2CCCCC2)=O)CCC(n2cc(CC3(O)COC3)nn2)CC1 C12(CNC(C(C(C)C)C)=O)COCCN1CCN(C(C1CCOCC1)=O)C2 C12(NC(C3N(C(C(=Cc4ccco4)C)=O)CC=C3)=O)CCC(C1)OC2C N1(C(C(C(C)C)NC=O)=O)CC2(C1)CN(C(=O)CC1CCCCC(=O)N1)C2 c1(C(=O)NCc2nccc(OC)c2)c(-c2ccccc2O)ccc2c1OCO2 N1(C(c2c(OC)cccc2)=O)CCCN(C(=O)C(C2(O)CCCC2)F)CC1C C1(NC(c2ccn(C(CC)CC)n2)=O)C=CCN(C(=O)CN2CCNC(=O)C2)C1 C(=O)(C1=NNC(=O)CC1)NC1C(NC(c2c(CC)nn(C)c2)=O)CC1 C1(CCNC(c2nn[nH]c2Cl)=O)CCCN(C(c2cc(C(F)F)no2)=O)C1 CN1C(=S)NC(c2ccccc2C(=O)O)C2=C1CC(C(=O)O)NC2=O c1(CN2C(CC(=O)Nc3ccc(I)cc3Cl)COCC2)cc(Br)cc(F)c1F N1(C(C=CCCC)=O)CC(F)(F)CC1(C)CNC(c1ccncn1)=O c1(CC(N2CC(NC(C(CC)(C)O)=O)(CO)C2)=O)nccc2ccccc12 C#Cc1cccc(CNC(N2CCCC(CCNC)C2)=O)c1 N1(C(c2sc3ccccc3c2Br)C(=O)NC(CC)C)CCC2(CC1)C(O)CC2O c1(C(=O)NCCCOCCNC(=O)CCc2cn[nH]c2)cnn2c1CCCC2 C1(CNC(=O)CC2(O)CCC2)COCC1.c1(C=O)c[nH]nc1-c1cccs1.C Cc1cccc(C(=O)NC2(C(=O)N)CCC(C)(C)C2)c1C#N.C1CC(F)(F)C1 N(C(=NCCF)NC1CCC(=O)NC1)C(C)CCc1ccco1 CC#CCC(C(=O)N1CCC=C(C)C1)NC(=O)CC1CC2(CCC2)C1 C1(NC(=O)CSc2ccccn2)CCCCCN(C(=O)Cn2cccn2)C1 N1(C(c2c[nH]nc2C)C(=O)NCC=C)CC2(CC=CC2)C1C(C)C C1(CC(C)C)COCCN1C(=O)CN(C(=O)CC1CC1)CCC.C(N)=O C(C(CC(=O)Nc1c(OC)noc1C)C1CCC1)NC(CCC#C)=O CC(C(C)C(=O)NCC(O)CC1CCC1)NC(c1ccnn1C1CC1)=O C1(C(=O)NCCNC(C2(OCC)CCSCC2)=O)CCCCN(C)C1=O CC(C)CC(CNC(=O)CC1CCC(=O)C1)C(=O)NCCCCCCCO Cc1nc(-c2nc(-c3cccc(C(N)=O)c3)sc2C)n(CCN2CCCC2)n1 N1(C(=O)OC(C)(C)C)CC2(CC(C(=O)NCC(c3cnc(O)[nH]3)O)CO2)C1 c1(NC(c2n(CCCCCC)nnn2)CCOC)ccccc1C C(=O)(C(CO)C(F)(F)F)N1CCCC(NC(c2ncc(F)cn2)=O)CC1 C1(C(=O)NCC#CCNC(=O)CCOCC(F)F)CCOC(=O)CC1 C1(NC(Cc2cn(C)nn2)=O)CCCCCN(C(C2(C)CC(C)(C)C2)=O)C1 C1(C(N2CC(F)(C(=O)Nc3cn(CC=C)nc3)C2)=O)CCCCC1(C)C c1(C(CCC(=O)OC(C(C(=O)OCC)=O)CC)=O)csc2ccccc12 O=C1CC2CC1CC2C(=O)N(CCC(=O)N1CC(CC2CC2)C1)C.C1CC1 C(CC(F)(F)F)N(C(=O)CC)C(=O)CC1COCCO1.CC CCCC(C)(O)CC(=O)NC1(CC(=O)N(C)CC2CCOC2)CC1 n1(CCN(CC)CC)c(-c2cc(C)ccc2C)csc1=Nc1ccc(C)c(C)c1 C(CC(=O)NCC(=O)NCC(=O)NC1(C)CC1C)OCCOCC C1(C)(C(=O)NC(C2CCN(C(C3(C4CC4)CCC3)=O)C2)C)CC2CC2C1 C1(C(=O)NC(CCC)C)CCCN1NC(=O)c1ccc2[nH]ccc2n1 c1(SC)cc(NC(C2CC(c3ccccc3)OC2=O)=O)ccc1Cl NC1CN(Cc2cccc(-c3ccc(-c4cn[nH]c4)cc3)c2)CCC1F c1(OC)ccc(F)c(C(=O)NCC2CCC2)c1Cl.C12(C(=O)N)CCCC1C2 CC1(C(=O)NCc2n[nH]c3c2CCC3)CC12CCN(C(C1CCCCO1)=O)CC2 N1(C(c2c[nH]c(=N)o2)=O)CCCCC(NC(=O)CC2CCCCC2O)CC1 C12CCCCC1C(=O)N2.c1ccccc1.CC(C=O)N(C(=O)CC1(C)CCC1)C C1(C(=O)NC2(C#C)CC(F)(F)C2)CCC(C)(C)N(C(=O)C(C)(O)C=C)C1 C(CC(C(=O)N1C2COCC1C2)OC)NC(c1c(CC)ncs1)=O c1(C(N2CCC(C(C)(C)NC(CCCC(=C)C)=O)C2)=O)c(C)oc2ccccc12 N1(S(c2c(C)cnn2C)(=O)=O)CCOC2(CCS(=N)(=O)CC2)C1 Cc1ccc(C(N2CC3CC(NC(c4ccncc4)=O)C2C3)=O)cc1Cl Cc1nc(C)c(C(=O)NCc2csc(C(=O)NC3CC34CCC4)c2)o1 Cc1ccncc1C=CC(=O)NCCC(C)N(C)C(C1CCC(F)CC1)=O c1(C(=O)NC2C(CNC(C(CCC)F)=O)C2)cc(C)nnc1O c1(C(N2CCCC(CCNC(C(C)NC(C)=O)=O)C2)=O)cncc2cccnc12 C(C)(CCCC(=O)NOCCCC(F)(F)F)NC(c1ccc(C)c(F)c1)=O c1(C=O)c(C)c2cnccn2c1C.c1(CC)ccc(N)c(C(=O)NC2CC2)c1.C N1(C(C(c2ccc(C)o2)C)=O)CC2(C=C(C(=O)NC3CCC3)CO2)C1 c1(-n2c(CC3ON=C(C)C3)nc(CSc3cnn(C)c3)n2)ccc2ccsc2c1 C(CC(C)C(=O)NCCCCCN1CCN(C(c2c[nH]c(=N)o2)=O)CC1)=CCC Cc1ncc(C(N2CC(CC(F)C(=O)N3CCC(OC(C)C)C3)C2)=O)cn1 C1(NC(C(COC)COC)=O)C2CC3CN(C(C4CCC5(CCC5)O4)=O)C1C3C2 N1(C(C2CCC(F)C2)=O)CCCC2CN(c3ncc4c(n3)COC4)CCC12 c1(C(=O)NC2C(CNC(C3C(C)(C)CCCC3)=O)CCC2)ncnc2ccsc12 c1(C(=O)N)cnc2n1CCS2.c1(NC(C)=O)cccc(C(N2CCC(C)C2)=O)n1 N1(C(C=CCOCCOC)=O)CC(O)CCC1C(=O)N.CC=O.C1CC1 N1(C(C2(SC)CCC2)=O)CCC2(CCCN2C(C2CN(S(N)(=O)=O)C2)=O)C1 C1(CC(N2CCC(N(C)C(c3cc(Cl)no3)=O)C2)=O)(COC)CCOCC1 n1(CC(=O)NC2CCOCC2NC(C2(F)CC=CCC2)=O)ncc2ccccc12 C1(C(NC2CCN(C(C3CCC(=O)N3)=O)C2)=O)C(C(F)(F)F)C1[N+](=O)[O-] N1(C(C(C)NC(C)(C)C)=O)CCCCCC1CNC(C1CC1)=O.C(N)=O Cc1ccnc(C(N2CC(CNC(=O)CN3CCCCC3)C(C)C2)=O)c1 C=CCC(C(=O)OC(c1noc(-c2ccccc2)n1)C)OC C(=O)(C#CC1(CC)COC1)N(C(CC)CC(=O)NC1CC2OCCCC12)C C1(c2ccc(OC(C)C)cc2)C(C)CN1N1CCC2(CCCO2)CC1 Cc1c(C(=O)NC(C)CC(C)NC(=O)Cc2cscn2)nnn1C(C)C N1(C(c2ccc(OC(C)C)cn2)=O)CCC(CNC(c2cc[nH]n2)=O)C12CCC2 C(=O)(C1=CCN(C(=O)C(F)C2CCC2)CC1)NC1CCCN(CC)C1 N1(C(C(CC)CC(C)C)=O)CC2CCC(C1)C(NC(=O)C(C(C)C)OC)C2 C1(C(=O)NCC=C)CCCN1N1CCC(c2c(C)[nH]c3ccccc23)C1 C=CC(CCC)CC(=O)NCCCCCNC(C1(C=O)CCC1)=O.C(C)(C)C.O C1(NC(CCOC(C)C)=O)CN(C(c2n[nH]c(C(C)(C)C)n2)=O)CC1C C1(NC(c2nc(OC)c(C)s2)=O)COC2CN(C(=O)C3=COCCO3)CC12 C1(CC(N2C(CN(C(=O)CCCc3ncco3)C)CCC2)=O)CC(C)(C)CCO1 Cc1c(C(=O)NCC(C(C)C(C)C)NC(=O)C=C2CCSCC2)cccc1F C1(NC(CCNC(=O)OC)=O)CCCC1O.c1(C=O)ccc(C2CC2)cc1.C C(=O)(CC(O)C(Cl)(Cl)Cl)N1CCC(O)(c2cn(C(C)C)nn2)C1 C1(c2c(C(=O)OC)n[nH]c2)CCN(C(=O)Nc2ccc(Br)cc2)CC1 c1(C(=O)OC)cccc(C)c1S(=O)(=O)NC1CN(Cc2cc[nH]n2)CC12CC2 c1(CN(C(=O)CC(C)(C)C)CC)cc(OC)cc(Br)c1OC C(N=c1nc(N2CCOC(C(N)=O)C2)c2[nH]ccc2[nH]1)C1(C)NC(=O)NC1=O CC12CCC1CN(C(C1CCC(O)CN1C(c1cnc(=N)[nH]c1)=O)=O)C2 C1(C(=O)Nc2ccc(NC)c(C)c2)CCC2(CCCCC2)C1 c1(C(N2CC(C=C)OCC2)C(=O)NCc2ccco2)cc(F)c(Cl)cc1Cl C1(CC(=O)NC(CN(C(=O)C=Cc2ccccn2)CC)C)CCCC(=O)N1 Cn1nc(C(=O)NCC2CC2C(=O)NCc2nc(C#N)cs2)ccc1=O C1(O)(CN(C(=O)Cc2nc[nH]n2)C)CCN(C(=O)C(O)c2cnc[nH]2)C1 C1(C(=O)NC(CSCC)C(=O)NC(c2scnc2C)C)CCC(C#N)CC1 C1(C#N)(c2c(C(=O)OC)scc2)CCN(S(=O)(=O)C2COC2)CC1.C(C)=O.N N1(C(C(C)c2cccs2)=O)CC(O)(CNC(=O)C(C)(C)N2CCCCC2)C1 Cc1cc(C(=O)NCC=CCNC(=O)CCCCC#N)c2cccnc2c1C N1(C(c2c(SCC)cncc2)=O)C2CCC1CN(C(C1CCCC(OC)C1)=O)C2 N1(C(CC(CC)OC)=O)CCN(C(C2CCN(OC)CC2)=O)CC1CC1CC1 c1(C(N2CCC(N(c3nc(C)nc(O)c3)C)C2)=O)cnc2cccnc2c1 C1(CNC(C(CC=C)OC)=O)(CO)CCCN(C(=O)CCN2CCCC2)C1 C(=O)(C1=NN(CCO)C(=O)CC1)N(C(C)C)C(c1cc2c(Cl)cccc2o1)=O Cc1nc(C2CC2)oc1C(=O)N(C1CCCN(C(C2COC(=O)N2)=O)C1)CCO CCC(CC(=O)NOCCOC)N(C)C(C1CCCC12CCC2)=O c1(C(=O)NCCCC(C)NC(C2CCCCO2)=O)cc2cc(Br)cn2cn1 C1(CNCC(c2ccc(O)cc2)OC)CCCC(N(C)C)C1 c1(C(=O)NC2C(NC(CCc3onc(C(C)(C)C)n3)=O)C2)cc(F)cc(Cl)c1 N1(C(C(CC)C)=O)CCC(O)CC1C(=O)Nc1ncc(Br)nc1C CCC(C)(COC)C(=O)N1CCC(CNC(c2ccc(SC(F)(F)F)s2)=O)C1 c1(NCc2n(C(CC)C)ncc2)cn2ncnc2c(C)n1 Cc1c(-c2cc(F)ccc2F)cnc2c1N(S(=O)(=O)c1cccnc1Cl)CCO2 N1(C(C=CCN(C)CC)=O)CC2CC1CCC2NC(c1cc(SC)ccc1Cl)=O c1(C(N2CC(OCC)(CO)C2)=O)coc2c1CN(C(=O)C(F)(F)C1CC1)C2 N1(C(c2cc(OC)no2)=O)CC2(CCC2NC(c2cc(Br)cnc2O)=O)C1 c1(CNC(C(C)OC(C)=O)=O)cc(C(=O)NC)n[nH]1.C1COC(=O)N1 c1(C(N2C(CNC(c3c(C)nns3)=O)CC2)=O)nccc(Cl)c1O c1(C=O)cc2c(cc1O)OCO2.c1(C(N(C)C)=O)coc(C(N)=O)c1.C1CC1 C1(CC(=O)N(C)CCNC(=O)C2=CSCS2)Cn2ccnc2NC1=O c1(OC)ccc(CC(=O)NCC2(NC(C3CCCN(C)C3)=O)CC2)cc1O N(C(=NCC1CCCCO1)NC)C(C1CCCS1)C.C12CC(C1)C(C(F)(F)F)O2 Cc1cccc(C(C)C(N2CC(CNC(c3cccn3C)=O)C(O)C2)=O)c1 CCC(CC)CCCC(=O)NC1(CC)CCN(C(c2ccc(SC)cc2)=O)CC1 N1(C(c2c(C)cc(O)cc2C)=O)CC2CCC1C1CN(C(=O)C(C)(C)C)CC21 Cc1cc(C(N2CCC(NC(=O)C=Cc3cc[nH]n3)C23CCC3)=O)c(N)c(Cl)n1 n1(CCOC)nccc1C(=O)N.c1(C=O)ccc(-c2ccco2)s1.C1CC1.C c1ccc(C)cc1.N1(C(COCC=C)=O)CCCC1C(C)NC(=O)CS.C N(C(=NCc1ccccc1)N1CCC2(C1)CC(F)(F)C2)Cc1cc(C)no1 C=CCCC(C(=O)NCCC1CCC(C)(C)O1)NC(C1CCC(C)(O)CC1)=O c1(C(N2C(CCC)CCCC2)C(=O)NCC)cccc(C)c1Oc1ccccc1 N1(C(C2C3CCN(C(C(C(C)C)C4CCC4)=O)CC32)=O)CC2(CCC2(C)C)C1 Cc1cc(C(=O)NC2CCN(C(=O)C3=CCOC3)CC2CO)cc(C)c1Cl CCCC(CCCNC(c1cc(C)sn1)=O)NC(=O)CCNC(=O)COC c1(-c2cc(C(=O)Nc3scc(C)n3)sc2)ccc(F)c(C#N)c1 C1(C(N(CCCNC(C2(C#N)CC2)=O)C)=O)Cc2cncn2C(=O)N1 c1(NC(C2CCN2C(c2cccnc2F)=O)=O)ccc2nncn2c1 Cc1cc(C(=O)NC(C)(C)CC)c2c(c1)C(C)CCN2.C1(CC=O)CC(F)C1 c1(C(N2CC3CC(NC(C(C(C)(C)C)O)=O)C3C2)=O)ccc(O)c(F)c1F C=CCC(C)C(=O)NC(c1nocc1C(=O)NCc1nnnn1C1CC1)C c1(C(=O)NC(C(C)NC(c2c[nH]nc2C2CC2)=O)C)cccc(N)c1O C1(C(=O)NC2CC(NC(CC3(OCC)CCCC3)=O)C2)CCC(C)NC1=O CN1C(=O)NCC1C(=O)NC1CCN(C(=O)C)C1.c1ccc(C(C)(C)C)cc1 CCC(C)C(CC(=O)NC1CC=CC1)NC(=O)CC1CCC(C)(C)C1 c1(OC)ccc(C2CCNCC2NC(c2cnn(C3CCCC3)c2)=O)cc1 C1(C(N2CC(=CCC)C2)=O)C2CCN(C(c3sccc3C(C)=O)=O)CC12 C=CCC(CC=C)C(=O)NC1CC(NC(C2CC(C)(C(=O)OC)C2)=O)C1 C(=O)(C(CNC(C1CC2(CCC2)CO1)=O)C(C)C)NCc1cc(C)ns1 C1(OC)CC2(C1)CC(C(=O)N)C2.C1CCN(C(=O)C=C2CCSCC2)C1(C)C N1(C(C(CCC)NC(c2c(C)nn(C)c2C)=O)=O)CCC2(CNC(=O)O2)C1 c1(C(N2CCC(C(C)NC(c3sccc3Cl)=O)C2)=O)cnc2c(c1)NCC2 CC1CC(NC(c2cnnn2C)=O)CN1C(=O)C(c1ccccc1)F C1(NC(C2(C)C(C)(C)C2)=O)CCN(C(=O)C=Cc2ccc(Br)o2)CC1F C1(OCC(=O)N(CCC)CCC)CCN(C(C2(C)CCCS2)=O)C1 N1(C(Cc2c(C)cccc2)=O)C(C)C2CC1C2NC(=O)CCOC(C)CC(C)C c1(OC(C)C)ccc(S(=O)(=O)NC2CN(C3COC3)C2)cc1 O(N=C1CCCCCC1)CC(N1CCN(C(=O)CCCF)CC1CC(F)F)=O C(=O)(C#CC(C)(C)O)N1C2(C(=O)NCCC=CC=C)CC(C1)C2 N1(C(C(CC(CC)C)NC(c2ccc(C#N)[nH]2)=O)=O)CCc2cccnc2C1 c1(CNC(C2(C)C(C)C2)=O)ccc(C)cc1.c1(C=O)cc(C(F)F)n(C)n1 CC(CC(=O)N1CC(C(C)(C)O)(CNC(c2cocn2)=O)C1)c1ccncc1 C1(C(N2CCN(CCCNC(CCCSC)=O)CC2)=O)CN2CCCC1CC2 C(c1ccccc1F)=CC(=O)NC(C(C)(C)C)CNC(=O)CCCF CC1CCC(C(=O)N(C2(C3CC3)CC2)C)N1C(c1cc(C2CC2)no1)=O Cn1cc2c(n1)CCC(C(=O)OCC1COC(C)(C)OC1)C2 c1(C(N2CC(S(C)(=O)=O)C2)=O)cc(O)nc2c1CN(C(c1csnc1Cl)=O)CC2 c1(C(N2CC(C)C(NC(C3(O)CC3)=O)CC2)=O)c(Cl)ccc(F)c1N CC(O)C(C)C(=O)N1CC(C(N)=O)(CNC(=O)Cc2nc[nH]n2)C1 Cc1cccc2c(NC3CC3C(N3CCCC(Br)C3)=O)ncnc12 n1(COCc2onc(C)n2)c(N2CCC(C)CC2)nnc1C1CCCCO1 c1nc(C(=O)NC)cs1.C1CCCN1C(=O)C(c1cnn(C)c1)C.CCOC c1(NC(CCc2ccc(C(N(CCC)C(C)C)=O)[nH]2)=O)cnn2cccnc12 N1(C(c2cnnn2C2CC2)=O)CCC(C2CC2)CC1 C1(C(=O)NCC(CN(C(C(=CC2CCCC2)C)=O)C)(C)C)CN2CCN1CC2C N1(C(c2ccc(CC)cc2F)=O)CCC2C(C1)CN2C(=O)CCSC C1(NCc2c(C)cc(F)s2)CCCCN(C(=O)OC(C)(C)C)CC1 O=S(=O)(C1CCC2(CC1)OCCO2)N1CCN(c2ccccc2OC(F)F)CC1 N1(C(c2c(CNCCC3(CO)CC3)cccc2)=O)CCc2nocc2C1 Cc1cnc(N2CCC(C)(N(C)C)CC2)cc1Br Cc1ccnc(C)c1C(N1CCC(N(CCO)C(c2cccnc2S)=O)C1)=O CCC(C)(C(=O)N)OC.c1cnn(-c2ccc(C(F)(F)F)cn2)c1C.C(C)(C)C.C c1(CN2C(CC(=O)Nc3c(C(=O)OC)nccc3)CCC2)cccc2nonc12 C12(NC(CSc3n(C)nnn3)=O)CCC1CN(C(c1ccc(O)c(Cl)n1)=O)C2 C#CCC(C)(CC)C(=O)NC1(CC(=O)NOCC2CCCO2)CC1 C=CCC(C)(C)C(=O)NCCC(C(C)C)NC(C1(C)C=CCC1)=O c1(C(=O)NCCC(C)N(C(C(C)OCCC=C)=O)C)cc2ccc(Cl)cn2c1 Cc1cc(CCC(=O)Nc2ccc(OCC(=O)NC(N)=O)c(Cl)c2)ccc1Cl N1(C(C(C)CNC(=O)CC2CC3(CC3)CO2)=O)CCCCCCCC1 C(=O)(C(O)CC=O)N(C)CC1CC1.c1(C=O)cc(F)n(C)n1.C(C)(C)C c1(C(N2CC(CNC(c3nc(CCC)sc3)=O)C(O)C2)=O)cccc(C)c1N c1(C(C(=O)NC2CCOC2)N(C(C)COC)CC=C)ccc2nn(C)cc2c1 CCC(COC)C(=O)NCc1cncc(C(=O)NC2COCCC2OC)c1 C=C(C)CCCC(=O)NCC1CN(C(c2cnc(C(F)F)nc2)=O)CCN1C C(c1ccc2c(c1)CCO2)=CC(N1CC(NC(c2n3cc(C)sc3nc2)=O)C1)=O CC(C)(C)[Si](C)(C)OCCNC(c1cc(Br)nn1C(F)F)C1CCC1 C(=O)(CC(C)C(F)F)NCCCNC(C(C)Cc1ccncc1)=O.C1CCCC1.C c1(C(N2CC(F)CC(NC(CC(C=C)CC)=O)C2)=O)cc2c([nH]1)CCCC2 C=CCCCCC(=O)N(C(C)CNC(c1c(Br)c(CC)nn1C)=O)CC C1(CC(=O)N(C(c2ccccc2)CN(C(=O)C=CBr)C)C)CC(C)(C)CO1 C(C)(C)(CC(=O)NC(C1(O)CCN(C(=O)CNC(C)=O)C1)C)OC C(C)(C(C(=O)Nc1cc(C)cn(C)c1=O)C(C)C)NC(CNC(CCC)=O)=O C1(C=O)CCCN(CC(F)(F)F)C1.CN1CC(CC(=O)NC2CC(CC)C2)C1.N N1(C(C(CC=C)C)=O)CC2C3CCC(C2C1)N(C(=O)CN1CCC1C)C3 c1(N2CCC(=CCNC(=O)C3=CCCCCC3)CC2)c[n+]([O-])ccc1[N+](=O)[O-] CCCCC(O)CC(=O)N1CCN(C(=O)CCc2ccc[nH]2)CC1C1CCCC1 C1(CCC)CN(C(=O)CSCC(F)F)CC1NC(=O)Cc1cn[nH]c1 N1(C(c2c(C)cn(C)c2)=O)CCC2CCN(C(=O)CN3CSCC3=O)CC2C1 c1(OC)cc(C(=O)NCCC)c2c(c1)CCC2.c1(C=O)cn(C(C)(C)C)nn1 c1(C(=O)NC(C2N(C(CSCCCC)=O)CCCC2)C)c(C)cc(C)oc1=O CC1(C)CCCCC1C(N1CCC(N2CCN(C(C3(O)CCC3)=O)CC2)CC1)=O N1(C(C(C)CC2CCC2)=O)CC(NC(=O)C(C)COc2ccccc2)CC(F)C1 c1(CC)cc(C(=O)OC2CN(C(C)C)CCC2F)c2c(CC(C)(C)C)noc2n1 C1(CCNC(C(C)Cc2ccccn2)=O)CCN(C(=O)CN2CC3CC3C2)CC1 N1(CCOC)CC(C(=O)NC2CC(F)C2)CC1=O.c1(C=O)c(C)ncn1C.C N1(C(COC(CC)(C)C)=O)CC(O)(C(C)NC(c2ccncn2)=O)C1 N1(C(c2c(CNC(C3CCC(=O)O3)=O)cco2)=O)CC2CCC(CC2)C1 N1(C(C)C)N=C(C(=O)NC(CNC(c2ccc(Cl)c(O)c2)=O)CO)CCC1=O C(C(C)C(=O)N1CC(O)(CN(C(=O)CCc2cncs2)C)C1)SC C1(N(C(C(C2CC(NC(CC=C)=O)C2)F)=O)C)COCC1O C(=O)(C(C)(O)CC(F)F)NCCNC(Cc1c(C)cc(Cl)cc1)=O c1(C(N2C(C)CN(C(=O)C(O)C3CCC3)CCC2)=O)ccc2c(Br)cnn2c1 c1(C(=O)NC2C(C)N(C(C3CC4CCC3O4)=O)CC2)ccc2nccn2c1 CCCC(C)C(=O)N(C(CC)C(=O)NCc1nncn1C)C c1(CCN(C)C)nc(-c2ccc(-c3cccc(Br)c3)cc2)n(-c2ccn(C)n2)n1 c1(C(N(C)CC2(O)CCN(C(C(C=C)(F)F)=O)CC2)=O)cncc2ccsc12 C1(F)(CNC(c2c(C)[nH]c(=N)s2)=O)CCN(C(=O)CCNC(N)=O)CC1 C12(C(=O)NCCc3c(C)ncs3)COC(C1)C(NC(=O)CC1=CCCC1)C2 C(=O)(CC(CC(=O)NCC)NS(=O)(=O)CCC)OC.C(C)(C)C.C=O.N c1(C=O)ccc(S(C)(=O)=O)s1.C1(C(N2C(C)CCC2)=O)CC(C(C)(C)C)=NO1 c1(C(C(=O)NCC(C)(C)NC(c2cnc3n2CCS3)=O)=O)ccc(Cl)cc1O N1(C(C(F)OC)=O)CCC2(CCC2)C1.C(c1ccc(C(N)=O)o1)=CC(=O)N N1(c2c(C)c(NC(c3cncs3)C)ncn2)CC2C(=O)N(C)C(=O)C2C1 N1(C(C(CC)OCC)=O)CCCC(C2(NC(=O)Cn3cc(Br)cn3)CC2)C1 N1(C(CN(C(C2CCC=CCC2)=O)CC)=O)CCC2CN(C)CCC12 C1(NC(C2CN(CC(C)C)C2)=O)COCCC1NC(=O)C(=O)NC1CC1 c1(CC)nc(C(=O)NCc2ocnc2C=O)c(C)o1.C1COC(C(F)F)C1 C#Cc1ccc(OCC(=O)NCC2(NC(=O)C(C)(F)F)CCOC2)cc1.O c1(NC(C(N2CCC(=CBr)CC2)c2c(C)cc(C)s2)=O)ccc2c(c1)OCO2 CCC(C)(O)C(=O)N1CCC(NC(c2ccccc2COC)=O)C1CO C12(NC(CSCCC)=O)CCN(C(c3cc(O)nn3C)=O)CCC1C2 C1(OC)CCCC(C(=O)NCC(C2CCN(C(c3n[nH]cc3F)=O)CC2)(C)O)C1 C1(CNC(Cc2cn(C)nc2)=O)CN(C(=O)Cn2ccnn2)CCO1.N(C=O)C N1(C(=O)NCc2ccc(C)cc2Cl)CCN(C(=O)OC(C)(C)C)C(C)C1C c1(C(=O)NCC2(NC(CCC=C)=O)CCC2)c(OC)ccc(OC)c1[N+](=O)[O-] C(CCC)(CCO)NC(CC1(NC(c2nc(CCC)oc2)=O)CCC1)=O C1(C(N2CCC(C(C)O)C2)C(=O)NCc2nnn(C)n2)CCC2(CC2)C1 N1(C(C(C(C)C)N2CCCC2=O)=O)CCC(C)C(CNC(=O)Cn2cncn2)C1 O=C(CS(=O)(=O)C1CC1)N1CCCCC(CNC(C23CCCC2CCC3)=O)C1 C(=O)(C#CC1CCC2(CC1)OCCO2)N1CCCC(C(C)NC(C)=O)C1 c1(C(C)NC2CCC(OC)CC2)ccc2c(c1)CCC2 c1(C(C)NC(C(C2CCOC2)NC(COCCC#C)=O)=O)ccc(O)cc1 Cc1ccc(F)c(C(=O)NCC2CN(C(=O)C(C)(C)C3CCC3)CC2O)c1F C(=O)(CCc1cn[nH]c1)N.N1(CCC)CCCC1.C(=O)C=CCN(C)CCF C1(C(=O)NCC(CO)NC(c2cccnc2)=O)CCCN(c2cc(O)ncn2)C1 C1(OC)CC(C)N(C(c2cc(C)ncn2)=O)C1.c1(C(=O)N)ncc(C(F)F)s1 C1(C(N(CCN(C(=O)Cc2sccc2Cl)C)C)=O)CC(C(F)(F)F)CO1 CC1(C)COCC(CC(=O)NC2CC3(C2)CC3)O1.C(C1CCOCC1)=CC=O.N N1(C(c2ncc(OC)nc2)=O)CC2(CCC2)CC1C(=O)NCC(C)(C)CCCO C1(CCNC(COC)=O)CN(C(=O)CNC(c2cccs2)=O)CCO1 C1(C(N2CCC2C)=O)(CC)CCC(O)CC1.c1(C=O)ncccc1Cl.C1CC1.N C1(NC(C(CC2CCCC2)NC(C2CN(C(C)=O)C2)=O)=O)CCOCC1(C)C c1(C(=O)NC2CCCC(N(C(CCC(=C)C)=O)C)C2)cc(Cl)cc(Cl)c1[N+](=O)[O-] C(=O)(C(F)CC(C)(C)C)NCC(CCC)NC(=O)C(C(C)C)OCC Nc1ccc2nc(N3CCCC(CNC(c4nc[nH]c5nccc4-5)=O)C3)sc2c1 c1(CCOC(C)C(=O)NCCC2CCN(C(=O)C(C)N(C)C)C2)ccccc1 N=c1nc(C2CCN(C(=O)NCC3CC3(F)F)C2)[nH][nH]1 Cc1nccc(CNC(=O)CCC(C)NC(c2n[nH]c(O)n2)=O)n1 Cc1ncc2c(n1)CCC(NCc1cn(CC3CC4CC4C3)nn1)C2 N1(C(c2c(C)con2)=O)CCC(COC2CCN(C(c3cc(Cl)cs3)=O)C2)CC1 S(=O)(=O)(c1cccc(C(=O)O)c1)N1CCC(OCC)(CO)CC1 OCCC(N=c1nc(N2CCSCC2)c2cccc(F)c2[nH]1)C1CCC1 Cc1c(N)ccc(C(N2CCCCC2CNC(=O)Cc2ccsn2)=O)c1F c1(C(=O)NC(CCNC(C(Br)=C(C)C)=O)(C)C)cccc(C(C)(C)C)n1 O=C(C1=CNC2=NCCC2=C1)NCCC1CC(NC(c2ccco2)=O)C1 c1(C=O)ccc(S(C)=O)cc1.c1(C(N(C)CC)=O)cc(C(C)C)[nH]c1CC CC1(C)c2ccccc2CCN1C(=O)NCc1nc(CCc2ccccc2)no1 CCCC(C)(O)CC(=O)NC1CCN(C(c2ccc3n[nH]cc3n2)=O)CC1C c1(C(N2C3C(C(N4CCn5cncc5C4)=O)C(C3)C2)=O)c(Cl)ccc(F)c1Cl c1(C(=O)NC2(CC)CCCN(C(CC(C=C)C)=O)C2)cc([N+](=O)[O-])cnc1O N1(CCC(N2CC(c3ccccc3)C(F)C2)=O)C(=O)C2CC=CCC2C1=O C1(CNC(C(C=C=C)C)=O)CN(C(C2(C(F)(F)F)CCCC2)=O)CC12CC2 c1(CNC(c2ccns2)=O)cc(C(N2CC(N3CCC3)C2)=O)on1 c1(N(CCCCC)C2CC2)ncnc(Cl)c1C(C)(C)C(=O)OC C1(NC(Cc2c(C)non2)=O)CC2(C1)CN(C(c1cc(C(N)=O)no1)=O)C2 N1(C(C(C(CC)C)NC(=O)CC2CCOC2C)=O)CCc2oc(C)nc2C1 N1(C(c2n(CC)ncn2)=O)CCN(C(c2ccccc2)=O)C(C)C1.C(C)(C)(C)O CC1CC(NC(=O)Cc2cc(O)nnc2O)CN(C(=O)CC2(C)CC2)C1 C#CC1=CN=NC1=C(O)NCC(Cc1ccc(Br)cc1)OC C12(C(=O)NC(C3CCCO3)CC)CC(CN1C(C1C3CCC(F)C13)=O)C2 c1(C(N2CCCCC2CC(C)O)C(=O)NCC)nc(C)ccc1Br C1(NC(C2(CC)CC2)=O)CC2CCC(C1C)N2C(C1CCC=CCC1)=O C(=O)(C#CC1CCCO1)N1CC(C)(NC(=O)CCC2CCOC2)C1 C12(NC(CC3(NC(CC4C(CC)C4)=O)CCC3)=O)CC(C)(C1)C2 C1(C(C)C)CCc2[nH]nc(C(=O)Nc3ncc(C(F)(F)F)cc3Cl)c2C1 N1(C(C(CC)CC)=O)CCCC2CN(C(c3cccc4ccn(C)c34)=O)CCC12 c1(C(N2CCC(C(C)NC(=O)CC3(O)CCC3)C2)=O)snc(Cl)c1Cl c1(CCNC(c2c(CC)nn[nH]2)=O)ccc(C)cc1.C1(C=O)CCC(F)C1.N c1(N2CCCC(CC)CC2)cc(C)c(S(=O)(=O)NCC2CCCOCC2)cn1 CCC(C)(CCNC(c1csc(F)c1)=O)NC(=O)Cc1c(C)n[nH]c1C CC1(C)COC(CCNC(=O)NCc2cc(-c3ccccc3)n[nH]2)C1 c1(OC)ccc(S(N)(=O)=O)cc1C(=O)NCCC.C(=O)(CS(C)(=O)=O)N c1(C(=O)Nc2cc(OC)cc(F)c2)coc2c1CN(C(C1COC(C)C1)=O)C2 C1(F)(C(N2CCCC(C(=O)OC)C2)=O)CCN(C(=O)Cc2ccc(Cl)cc2)CC1 C1(C(=O)OC)COCCN1C(c1ncc(NC(=O)OC(C)(C)C)cn1)=O N1(C(CCSCC)=O)CCC(O)(CN(C(=O)COC(CC)CC)C)C1 C1(C(=O)NCC(C)=O)CC2CCN(c3ccncc3C)CC12 c1(C(=O)NC(C(C)C(=O)NCC2=CCCC2)C)cn2c(n1)CCC2 c1(SC)ccc(C(N2CCC(N(C)C(c3cccc(Br)n3)=O)C2)=O)cc1 C1(NC(c2cc(C)ns2)=O)CCN(C(C2(N(C)C)CC2)=O)CC1F C(=O)(CC=C(Cl)Cl)NC1(CO)CN(C(C2(C)CC(F)C2)=O)C1 Cc1cc2c(c(C)c1C)CCCN2C(c1cnc(C(F)F)s1)C(=O)NC(C)(C)C C(=O)(C#CC1CCCC1)N(CCC(N1CCCC(C)C1CO)=O)CC=C c1(C(N2CC3CCC(CNC(CCCCC)=O)(C2)C3)=O)ncnc2c1ccn2C C1(CC)CCN(C(c2cnc(C3CC3)o2)=O)C1C(N1CC=C(C)C1)=O CC1C(CONC=O)CCCN1C.C(C)(C)(C)NC(=O)NC C1(CC)COC(C)CN1C(C1(NC(c2cscn2)=O)CCN(C)C1)=O c1(CCC)nc(C(N2CCC(CN(C)C(C3CC3c3ccsc3)=O)C2)=O)co1 CC1(C)CC(NC(c2ccnc3[nH]c(O)nc23)=O)CCN(C(=O)C(Cl)=CCl)C1 C(CO)(CC(F)(F)F)NC(C1CC(O)CN1C(=O)CC1CCCC12CC2)=O N1(CCCC)CCCCC1C(=O)NCC1(C(F)F)CCN(C(=O)CC)C1.O.C c1(CC(=O)NCC(=O)NCCCCNC(c2cnsc2)=O)ccccc1 C1(NC(C=CCOC)=O)CCC1NC(=O)CCc1nc[nH]n1 N1(C(C(COC)(C)OC)=O)CCN(C(=O)C=Cc2cncn2C)C(CC(F)F)C1 c1(NC(=O)NCC(c2ccc(Cl)c(F)c2)O)cccc2c1CCCC2 N1(C(C(C)Cc2ccc(F)cc2)=O)CC(NC(=O)CCC(N)=O)C2(CC2)C1 C(=O)(C(C)C(=O)OC(C)(C)C)N1CC(CNC(c2c(C)onc2)=O)C1 C1(n2cccn2)(C(N(C(C)C)CCN(C)C(C2COC2)=O)=O)CCC1 c1(CC#N)ccc(C(=O)NC2CC(CO)N(C(=O)CCc3cccs3)C2)cc1 C1(CC(=O)NCCOCCCNC(c2ccco2)=O)(N(C)C)CCCCC1.O c1(C(C(=O)N(CC(C)NC(c2nc(Cl)oc2C)=O)CC)C)cc2ccccc2o1 CC1CC(NC(=O)C(C)CCc2ccccc2F)CN(C(=O)C)C1.[SH](C)(=O)=O.N C1(C(N(CCCNC(=O)COC2CCCOC2)C)=O)CCCCC12CCC2 N1(CBr)CCC(C2CCCCC2)C1.C1(Cc2nnnn2C(C)C)(CC)CCOCC1 N1(C(c2c(OC)cc(N(C)C)cc2)=O)CCOC2(C(OC)COCC2)C1 Fc1c(Br)cc(CN(CCc2cccc(Cl)c2)C2CC2)cc1I C1(O)(CCNC(C)=O)CCCN(C(C2(Cl)CC2(F)F)=O)C1 CC1CC(C(=O)NCC2CC[Si](C)(C)C2)CN(C(=O)CCN=[N+]=[N-])C1 c1(C(N2CC(C)(NC(CCC(C)OC)=O)C2)=O)ccc(N=[N+]=[N-])cc1 C1(CC)CN(C(=O)CN(c2cnccn2)C)CCC1NC(c1cc(C)on1)=O c1(NC(CNC(CCN(C(=O)C)CC)=O)C)ccc(C#N)nc1.CCC(C)C C1(C(N2CC(C)(CF)C2)=O)(COC)CN(C(c2ccoc2C2CC2)=O)C1 c1(N2CCC(N=S(C)(C)=O)CC2)cc[nH]c(=NCCC=CBr)n1 CN1CCN(C(C23CC(NC(C4CC5CCCC5C4)=O)(C2)C3)=O)CC(O)C1 C1(C2CCOCC2)(C(N2CC(CNC(CC(CC)C)=O)OCCC2)=O)CC1 c1(C(N2CCCC(C(C)NC(c3c(CC)csc3)=O)C2)=O)ncnc(O)c1Cl c1(N2CCC(Oc3cccc(CO)c3)C2)cc2cnccc2o1 C(=O)(C(CO)C(F)(F)F)NCCC1(OC)CN(C(CCC)=O)C1 C1(CC)C(C(=O)NCCP(C)(C)=O)CCN1C(=O)C=CCO c1(NC(C2CCN(C(c3cc(C)cc(C)n3)=O)C2)=O)ncnc2c1c(Br)cn2C Cc1nc(C)c(CNC(C2(NC(c3ccc(Cl)cc3)=O)CCCC2C)=O)o1 C1(CCC)CCC(O)(C(=O)NCC(CC)(CC)NC(C2CCC(=O)N2)=O)CC1 CC(C)(C)C#CC(=O)NC1(C)CC(C(=O)NCC2(C)CC3CCC2C3)C1 C1(COC)CN(C(C2CC2(F)F)=O)CCN1C(=O)CCn1cnnn1 N1(C(c2ccc(N)c(F)c2)=O)C2CCC1CN(C(=O)CCCc1cccs1)C2 CCC(CCCC(=O)NCCCC1(C)CC1)NC(=O)C(C#N)C(C)(C)C S(=O)(=O)(c1cccnc1NC1COCC1O)N1C(CN(C)C)COCC1 C(=O)(C1=CC2(CCOC2)C1)N.CC(C)C(C)CNC(=O)CSc1nncs1 C1(C(=O)NC(CC=C)CO)CC(F)CN1S(=O)(=O)CCCC N1(C(COCC=C)=O)CCC2(CO)CN(C(=O)C(=CC3CCCC3)C)CC2C1 C(C(C)(C)CN=[N+]=[N-])NC(c1ccn(CCNC(C(C=C=C)C)=O)c1)=O C(CCSC)(C=O)NS(CC)(=O)=O.C(C)(C)C1CC1.c1(C=O)cn[nH]c1.N CC(C)CC(CNC(=O)CNC(=O)C1CC1)C(=O)N.CCC(O)C1CCC1 N1(CC#C)CCC(CNC(c2cn(C3CC3)nn2)=O)CC1 C(=O)(C#Cc1ccc(Cl)cc1)N1CCC(O)(C(=O)NC(c2ccsc2)C)C1 C1(C(N(C2CNCCOC2)C)=O)CC12CCCNC2 c1(CC(N2CC=CC(NC(c3ccncn3)=O)C2)=O)ccc2ncsc2c1 C1(C(N(CC=C)C)=O)CN(C(=O)CCOCC(C)C)CC(C)(C)C1 C(CO)(CC(C)C)C(=O)NC1(C)CN(C(C(C2CC2)SC)=O)C1 c1(C(=O)NC(CC)CN(C(C2CC23CCCC3)=O)CC)nccn2nccc12 CON=Cc1ccc(C(=O)NC2CCOCC2NC(C2CC(O)CN2C)=O)cc1 N(C1CCc2c(F)cccc21)(CCCCCNC(c1c(C)nc(C)[nH]1)=O)CCO c1(C(=O)NC23C(CN(C(C(CC#C)(C)C)=O)C2)CCC3)nn2cccnc2c1Cl c1(C(=O)NC2CC(C(C(=O)NC(CC#C)CC)F)C2)ccc(O)cn1 N1(C(C2CCN(C(CC)=O)C2)=O)CCCC(C)(NC(c2cnc(CC)s2)=O)C1 CC(O)C(C)C(=O)NC1CC(C)(NC(c2cnncc2O)=O)C1 N1(C(c2c(C)cc(F)cc2)=O)CC2CCCC2(NC(=O)C(=O)Nc2ncc[nH]2)C1 CC(CC(F)F)C(=O)N1CCC(C)(CC(N2CC(C)(C)C2C(C)C)=O)C1 C(CC(C(C)C)NC(c1csc(C(F)F)c1)=O)N(C(CCCOCCC)=O)C C(C)(CC(=O)NC1CCN(C(c2c(N)cccc2F)=O)CC1F)(C(F)F)N(C)C CCCCC(CC)C(=O)NC1(CNC(=O)C(n2cc(Br)cn2)C)CCCC1 C(=O)(C#CC1CCCC1)N(C1CN(C(c2cocn2)=O)CC12CC2)C CCC(C)C(O)CC(=O)NC1CCCCC1CC(N1CC(C)C1(C)C)=O c1(C(N)=O)ccc(C(N2CCSCC2C(N2CCC(F)C2)=O)=O)cc1 C1(CNC(C(CC)C2CCOC2)=O)CN(C)CCN1C(=O)CCc1cncnc1 Cc1cc(C(=O)NCCCN(C(c2cn(C(C)(C)C)nn2)=O)C(C)C)ns1 c1(CC(=O)NC(C)C)ccc(C(C)=O)cc1.C1(=CC=O)CCC(C)C1 CCC(N=c1nc(N2CCCC(OCCO)C2)c2c(ncn2C)[nH]1)C1CC1 C1(C(=O)OCC)CC=CC1.c1(C(NCCC)=O)cnoc1C1CCOCC1 CC(C(=O)NCCN(C(=O)C1=CCC1)CCCN(C)C)C(C)n1cccn1 C1(CNC(c2c(C)n[nH]c2C)=O)CCC2CN(C(C3CC=CCO3)=O)CCC2C1 c1(CNC(C=C(C)C)=O)ccc(CNC(=O)Cc2cccn2C)cc1 CC12CN(C(C3(C)CCCC3)=O)C(C(=O)NC3(C)CC4CCC3C4)(C1)C2 c1(CC(=O)NC2(CCOC)CCN(C(=O)CC(C)OC)C2)cccc(Cl)c1F CCC(C)C(=O)NCC(=O)NC(C)(C)CC.c1(C2C(C(=O)N)C2)ccoc1 N1(C(C(CC#C)(C)C)=O)Cc2[nH]nc(C(=O)N(CCC(=O)NC3CC3)C)c2C1 C1(CC)CN(C(=O)C(CCOC)OC)CCN1C(c1ccn(C)n1)=O c1(NC(c2n(CC)nnn2)CCSc2ccc(Cl)cc2F)ccc(Br)c(Cl)c1C C1(C(=O)NC2(CO)CN(C(C3(OCC)CCOC3)=O)C2)CCCCN(C)C1=O C(=O)(C(C)CC(F)F)NCC(C(=O)NCCCC(N)=O)OC c1(C(N2CC(c3cccc(OC)c3)NCC2)=O)ccccc1P(C)(C)=O Cc1nn(C)cc1C(N1CC(F)(C(N2CC(O)(CC(C)C)C2)=O)C1)=O C(=O)(C(C)(O)C(C)C)N1CCCC(N2CCN(C(C(=O)NC(C)C)=O)CC2)C1 c1(C(c2nnnn2C2CCOCC2)NC2(COC)CCSC2)cccc(C)n1 C12(C(=O)NCC(CC(=O)N(CC(O)C3CCC3)C)OC)CCC(C)(C1)OC2 Cc1nscc1C(=O)N.c1noc(CS(=O)(=O)CC2(C(F)(F)F)CCCN2)n1 Cc1nccnc1C(N1CCC1)=O.C1(C=O)C(C)CCN1C=O.C(C)(C)C.C c1(CSCC)cc(C(=O)NC(C)CC)no1.C1(C(=O)N)CC2(CC2)C1 C1(NC(c2n(COC)ncc2)=O)(CO)CCCN(C(c2cccc(C)c2C)=O)C1 c1(C(N2CCC(O)(CN(C(CCC=CC)=O)C)C2)=O)ccc(OC)cc1F CC(C)CC(CNC(=O)CC1CCC=CCC1)NC(=O)C(C)NC=O c1(C(=O)NC2CCCC(N(C(=O)CC(F)F)C)C2)n[nH]c2c1CCCCC2 C1(Cc2cn(-c3c(C(=O)O)scc3)nn2)CCCN(C(C2(C)CC2(Br)Br)=O)C1 Cc1nnccc1C(=O)NC(C)CCCCNC(=O)C=Cc1ccnn1C C1(CC)CCOC1C(=O)NC1C=CC(C(N2CC(CSC)C2)=O)C1 c1(CC)noc(C(=O)N(C2CCN(C(=O)CC3CC(C)C3)C2)CC)c1C O=C(CCC1=CCCCC1)NCC1CCC1NC(=O)C(c1ccc(Cl)cc1)O C1(OC)CN(C(=O)C(C)SC(C)C)CC1NC(c1ccnnc1)=O C(C)(CCC(=O)NCC(C)CNC(c1nc(-c2nc[nH]n2)sc1C)=O)OC N1(C(C(CSC)(C)NC(c2sccc2C#N)=O)=O)CCC(C2CC2)CC1 Cc1oc(-c2ccsc2)nc1CC(=O)NCC(O)CN(C)C(C1CCN(C)C1)=O C(=O)(C1=NOC2COCC12)NC(C)CCCCNC(c1cn2ccnc2cn1)=O c1(SC(C)C(N2CCS(=O)C(C)(C)C2)=O)ccc(S(N)(=O)=O)cc1 C(=O)(CCC(C)(C)[N+](=O)[O-])NC(C(CO)NC(C12CC(OC)C1C2)=O)C c1(CC)c(C(=O)NC(C2CN(C(c3ccc(Cl)s3)=O)CCO2)C)cnn1CC C1(NC(CN(S(CC)(=O)=O)C)=O)CN(C(c2c(C)ncn2C)=O)CC2(CCC2)C1 CCCC(C(=O)OC)NC(=O)CC1CCCN(C(=O)Nc2ccc(Br)s2)C1 C1(NC(CSc2n[nH]c(=N)s2)=O)CCCN(C(=O)CC2CC3(CCC3)CO2)CC1 c1(C(N2CC3C(C(=O)Nc4cc(C(C)C)no4)(C3)C2)=O)cc(F)c(Cl)c(Br)c1 c1(OC)ccc(C2=CCN(C(c3cc(OC(F)F)ccc3C)=O)C2)cc1 CCCCC(CNC(=O)C(C)C(C)C)NC(c1cnn(CC)c1)=O Cc1cc(C(=O)NC(C2CN(C(=O)CN3CCC(C)C3)C2)C)nc2ccccc12 Cn1cnc(CN(CCO)CC2(F)CN(C(=O)OC(C)(C)C)C2)c1 c1(-n2cc(CC(CC)(C)O)nn2)cc[nH]c2nccc1-2.C1(=O)CCCCCN1 N#Cc1cccc(C(CF)NC(C2CN(C(c3ccccn3)=O)CCO2)=O)c1 C1(C2CC2)(C(N(CCCNC(C2(C)COC(=O)OC2)=O)C)=O)CC=CC1 CCCC(C)C(=O)N1CCCC1CN(C(=O)COCC1CCC1)C c1(OC)ccc(C(=O)N(C)CC2CCCN2C(=O)CC(C)(C)F)c(F)c1 N1(C(=O)OC(C)(C)C)CC2CCC(C(N3CCC4(CCOCC4)C3)=O)CC2C1 C1(C(=O)NC(C)Cc2nn[nH]n2)CC(NC(=O)COCCN(C)C)C1 CCC(CC)CCCC(=O)NCC1CCCCN1C(c1ncsc1C)=O C=C1COc2c(C(=O)NC(C)(C)CCCNC(=O)C(=O)NCC)cnn2C1 S(=O)(=O)(CC(=O)NC(C)(CNC(=O)C#CC(=O)N(C)C)C(C)C)NC Nc1ccc(C(N2CC(F)C2)=O)cc1C(F)(F)F.C1(C=O)CC1C(F)F.C c1ccc(F)cc1F.C1(C(=O)NC2CC(N3CCCC3)C2)C=CCN1C(=O)C.O N1(c2n(CCC3CC(C)C3)nnn2)CC(C)OC2(CCOC2)C1 C1(NC(CCSCCCC)=O)CN(C(C2CC(n3ccnn3)C2)=O)C2CCCC12 C#CCCCCC(=O)NC1CC(CNC(c2ccn(C3CC3(F)F)n2)=O)C1 c1(OC)cccc(C=CC(N2CCC3(CC3)C2)=O)c1.C(=O)C=CC(C)C.N c1(C(N2CCC3CCCC23CNC(=O)C(F)(F)C2CC2)=O)cnc2n1CCCC2 N1(C(c2nc(C)n(C)n2)=O)CCC(C(F)(F)F)C(NC(c2cocn2)=O)C1 CC1CC(NC(=O)CCC[N+](=O)[O-])CN(C(=O)OCc2ccccc2)C1 N1(C(C(C)OC)=O)CCC(CNC(C2(c3ccc(C)nc3)CC2)=O)C12CC2 C1C(C)CC(=O)N1C1CC1.C1(CC(=O)OC(C(C)OC)=O)CCCCC1 C1(NC(c2cc(C)nn2C)=O)CCSC12CN(C(C1Cc3cscc3C1)=O)C2 N1(C(C(OC)OC)=O)CCC(C)C1C(=O)NC1(c2ccc(F)cc2)CC1 CC1CCC(CNC(c2ccc(C#N)[nH]2)=O)CN1C(=O)CN1CCn2nccc21 N1(C(C(CC2CN(C(c3[nH]cc(C#N)c3)=O)C2)F)=O)CC2C=CC1CC2 C(CCCC(C(=O)Nc1c(C)cc(C)cc1C)N1CC(C(F)(F)F)CC1C)OC c1(CC)cccnc1C(=O)N(CC(C)NC(c1ccc(=O)oc1)=O)C C12(NC(C(C)Oc3ccccc3C#N)=O)CCCC1N(C(C1CC(O)C1)=O)CC2 c1(OC)ccc2c(C(N3CCC4CN(Cc5cncc(F)c5)CC34)=O)c[nH]c2c1 C=CCCC(C(=O)N(CCC(F)(F)F)CC)NC(=O)CCCOC N1(C(C(=O)N(CC(CC)C)C)=O)CCC(c2ccc(F)cc2)(C(=O)O)C1 C1(NC(CC=CC)=O)C2CCC(C2)C1C(N1CCC(F)(CF)C1)=O C(=O)(CC(C)C(C)C(C)C)N1CCN(C(c2c(C)nc(C3CC3)o2)=O)CC(O)C1 C(=O)(C(C)CCCOC)NCC(CC=C)NC(=O)Cc1cc(C)ccc1Br N=c1nc2ccc(C(=O)NCC3CCN(C(c4cn(CCO)nn4)=O)C3)cn2[nH]1 C1(COC)(NC(c2nc(C)c(C)s2)=O)CCN(C(C2(C)COC2)=O)CC1 CC(C)C(CCN(C)C(c1ccsc1Cl)=O)NC(C1(C(=O)C2CC2)CCC1)=O Cc1cc(OC(C)C(=O)N2CC(N(C(=O)C=CCF)C)C2)ccc1Cl c1ccc([N+](=O)[O-])cc1.C1(C=O)CC(C)N(C)C1.CCC(C)CNC(=O)C.O N1(C(C=C(CC)C)=O)CCC(NC(c2cc(C)nnc2O)=O)C2(CCC2)C1 C=Cc1ccc(C(N2CC3CC2CC3NC(C2C3CC4C(C3)C24)=O)=O)cc1 N1(c2snc(C)n2)CCN(c2cc(N(CCCO)C)ncn2)CC1 N1(C(C2C(OCC)C2)=O)CCCC(NC(C2CC(=O)N(C(C)C)C2)=O)C1 C1(NC(CC(CC)N(C)C(c2cncn2C)=O)=O)CC2(CCC2)C1O C1(C(=O)NC2CCC(NC(C(CC(C)C)=O)=O)CC2)CC2C=CCC(C1)C2 Cc1c(C(=O)NC2CCN(C(C3CC4CCC(C3)O4)=O)C2)sc2ccc(F)cc12 c1(CC(N2CCCC(N3CCN(C(C)=O)CC3=O)C2)=O)cncc2ccccc12 CCC(C(=O)NCC1(CNC(c2ccccc2O)=O)CCCC1)C(C)(F)F.S c1(C(=O)O)cc(C)c(C)nn1.c1(C(CC)C)ccc(C(C(C)C)NC(=O)C)cc1 C(=O)(CS(=O)c1ccc(Cl)cc1)N1CC(C)N(C(=O)CN(C)C2CC2)CC1 c1(OC)ccc(Br)c(CN2CC3CC2CN3C(=O)Nc2ccc(C)cc2)c1 c1(CC(C)C(=O)NC23CC2CN(C(c2ccc(O)cc2)=O)C3)cccc(Br)c1 c1(C(C)C)cc(C(N2CC3CC3(CNC(C3COC3)=O)C2)=O)nn1C c1(CCC(=O)NCCN(C(=O)C(CC(C)C)N(C)C)CC)cc(F)ccc1 c1(SCCCC)c(NC(=O)CCSCC(C)C)cncc1Br c1(C(N2CC(OCC(=O)NCCC3CCCCCC3)C2)=O)cccc2occc12 C1(NC(=O)CCc2cnc[nH]2)CC2(C1)CN(C(C1(C(F)F)CCCO1)=O)C2 C1(C(N(CCO)CC)=O)CC(C)(C)CCN1C(=O)C(C)N=[N+]=[N-] c1(OC)ccccc1C(C(=O)NC1(CO)CCN(C(C2CC=CC2)=O)C1)OC c1(C(=O)NCC2CC(F)(F)C2)cc2ncc(-c3cc(CO)ccc3F)cc2[nH]1 N1(C(c2c(C)cns2)=O)CC(C)CCC1CNC(=O)Cc1c(C)cccc1Cl N1(C(c2scc(COC)c2)=O)CC(NC(C2SCCS2)=O)C(C2CC2)C1 c1(NC(CC)CCCO)ncnc(N(C)Cc2ccc(SC)cc2)c1C C1(C(F)(F)F)(OC)CC(CNC(=O)CC(C)CF)C1.C(=O)C(C)N(C)C Cc1cc(C=CC(=O)NC2CCN(C(=O)CC3CC34CC4)C23CC3)ccc1Br c1(OC)ccc(C2CC2C(=O)NCCC(C)C)nc1.c1(C=O)csc(C)c1N.N C=CCC(C)(C)CC(=O)N1CC(CNC(=O)C(C)C)C2CC12.C=O.CCC.N c1(C(=O)NC(CN(C(=O)CS(=O)(=O)CC)CC)C)cc2nccnc2cc1C C1(NC(C(n2cc(CC(C(=O)OC)C3CC3)nn2)C)=O)CCn2ncnc2C1 N1(C(C2CC(NC(CCCC(=C)C)=O)C23CCC3)=O)CCCC(C)(C#N)C1 C(=O)C1=NOC(C(C)(C)C)C1.C1(C)(NC(C(C2CC2)OC)=O)CCCC1.N N1(C(C2(COC)CCCCC2)=O)CC2CN(C(C3CC34CCC4)=O)CC2C1 C1(C(=O)NC(c2cncc(OC)c2)C)CCC2(CCCCC2)CC1 N1(C(C2C=C(C)CS2)=O)CCN(C)C(CNC(=O)CCNC(N)=O)C1 c1(CC)ccc(C(=O)NCCCN(C(=O)CC23CCCC2C3)C2CC2)s1 Cn1cc(NC(=O)C(=O)Nc2ccccc2N)c(C(F)F)n1.c1ccccc1.C CCCC(C)(C)C(=O)N1CC2CC(NC(C3CCC(C)(C)OC3)=O)C2C1 C12(CNC(c3cc(OC)n[nH]3)=O)CC1CN(C(=O)CCC1CCC1)C2 c1(OC)cc(-c2cn(CC3CN(C(=O)CC4(OC)CC4)CCO3)nn2)cc(F)c1 CCC(CC(=O)NC1CCC1NC(c1cccnc1N1CCCCC1)=O)C1CC1 C1(CC(=O)N(CCCN(C(=O)C)C)C)CC2(CCOCC2)CO1.C1(F)CC1.O c1(C(N2CCC(C=C)C2)C(=O)NCCOC)ccc(O)c(F)c1 c1(C(N2CC3CCN(C(=O)C(O)C(F)F)CC3C2)=O)c(F)c(F)cc(F)c1F C1(C)CCOC1C1CC1.CC1(C=CC(=O)NCC2(CC=O)CC2)COC1 C=CC1(C(N2CC(CC(F)C(=O)Nc3cnn(CCOC)c3)C2)=O)CCC1 C1(c2nnc(C)o2)CCCCN1CC(=O)NC1CC1c1ccn(C)n1 c1(C(N2CCC(C)(CNC(COCCC=C)=O)C2)=O)cc2c(cc1Cl)CCCC2 C1(O)(CNC(C2C3CCC23)=O)CCCN(C(c2ccoc2)=O)CC1 c1(C(N2CCN(C(c3c(C)n(C)cc3)=O)C(C3CC3)C2)=O)cc2c(ncn2C)[nH]1 c1(OC)cc(C(=O)N(CC(C)CNC(C23COCC2C3)=O)C)cc(Cl)n1 c1(CC(=O)N(C2CCN(C(C3CC4CC4C3)=O)C2)C)c[nH]c2ccccc12 C=CCCCC(C)(C)C(=O)N1CC(NC(=O)C=Cc2ccc(F)c(F)c2)C(O)C1 CN1CCc2[nH]nc(C(N3CC(NC(=O)CSC4CC4)C4CC34)=O)c2C1 Cc1ccc(CC(N2CCC(CCC(=O)N(C)CC3CCC3)C2)=O)cn1 c1(C(=O)NCC2CCN(C(CCC=CC)=O)CC2(F)F)c(Cl)nc2ccccn12 C(CCC(C)CC(=O)NC1CN(C(c2cnc(C(F)(F)F)c(F)c2)=O)C1)=C(C)C C(=O)(C(C)(O)C(F)F)N1CCCC(n2cc(-c3ccc(C)cc3)nn2)C1 c1(C(=O)NCCC(C)NC(=O)CC)ccnn1C1CCCC1.C1(C=O)CCC1 CC1CCC(O)C(NC(C2(NC(c3cnc(N)cn3)=O)CC2)=O)C1 C1(C(N2C(CNC(CCCC=C)=O)(COC)CCC2)=O)CCc2cn(C)nc2C1 C1(CC)CC(N=c2nc3c(ncn3CC)c(NCC3(C4CC4)CCCO3)[nH]2)C1 C=C1CC2CCCC(C1)N2C(=O)CC(COC)NC(=O)CCN(C)C C1(N(C(=O)C2=CCC2)CCCC)CCN(C(c2nc(C)nn2C)=O)CC1 N1(C=O)CCC(O)(C(F)F)C1.c1ccccc1.c1(N(CC)C2CC2)ccon1.N N1(C(C2C(C=C)C2)=O)CCN(C(c2cnc3n2CCC3)=O)CC1CS(C)(=O)=O C(=O)(C1=CCC(NC(c2c(C)n[nH]c2C)=O)C1)NC(CC#C)C(=O)OC N1(C(C(C(C)S(C)(=O)=O)C)=O)CCCC(C2CCN(C(C3(F)CCC3)=O)CC2)C1 C1(C#N)(CC(=O)NCC2(C(F)F)CCN(C(C(CCC)C)=O)C2)CCCCC1 C#CC1CN(C(C2CCN2C)=O)CCN1C(c1nonc1N)=O N1(C(c2ncn(C)c2)=O)CCCCC1CCNC(C1(Cl)CC1(F)F)=O c1(CC)nccc(C(F)(F)F)c1NC(=O)NC(c1cccc(Cl)c1)CO N1(C(C=COCC)=O)CCC(C)C(CNC(=O)CCCCCOC)C1 C1(NC(CC=CC=C)=O)CCN(C(C2CCC(COC)C2)=O)C1 Cc1cc(C)c(CNC(=O)CC2CCN2C(=O)CC#N)s1 C12(CCC)CC(C(=O)N(CCCC(=O)OC(C)(C)C)CC)(C1)C2 Cc1cnc(CNC(C2COCCN2c2cc(-n3cncn3)ncn2)=O)nc1 N1(C(C(C)C2(O)CCC2)=O)CC2CC(CNC(=O)CCc3ccc(Cl)cc3)C2C1 C=C1CC2CCC(C1)N2C(=O)C(O)C(CCC)NC(=O)CC(C)C(F)(F)F N1(CC(C)NC(=O)C(c2ccccc2)C)CCN(C(C2(n3nccn3)CC2)=O)CC1 C(C1=NOC2COCC12)NC(C1(F)CCCN(C(C(C)(F)c2ccon2)=O)C1)=O N1(C(C2(OC)CCCC2)=O)CCC(C)C(NC(c2ccc(-c3cc[nH]n3)s2)=O)C1 c1(C(=O)NCC(C)(C)C(N2CC(CO)CC2(C)C)=O)cnn2ccc(Cl)c(F)c12 CC(C)C(CCNC(C1CC(F)C1)=O)NC(=O)C(C(C)C)n1cccc1 C1(C(C)(O)C)CCN(C(=O)C(O)Cc2ccccc2Cl)CC1.C(=O)C=C1CC1.N CC(CC(=O)N1CCCC1CCNC(=O)CCC(C)(C)O)C(F)F CC1CN(C(=O)CCN(C)C(c2cc(O)cs2)=O)CC1C(N)=O N1(C(C2CC(C)(C)C2)=O)CCCC(C)(C#N)C1.CC1CCC(CCC(=O)NC)O1 CC(C)(CC(F)F)C(=O)N1CCC(N(c2ccncn2)CCN2C(=O)CCC2=O)C1 C1(CC=O)CC2(CCCC2)CO1.C1CCCC1.C(C)(C(=O)N)NC(=O)NC N1(C(C(CC=CCC)C)=O)CCOC2(CCN(C(=O)C3=CC(C)(C)C3)C2)C1 N1(CCCSC)CCC(O)C(C(N2C(C)CCC2(C)C)=O)C1 C(=O)(C1CCCn2cc(C(C)(C)C)nc21)NC1C(CNC(C)=O)CCC1 c1(-c2cn(CCN(C(C(C3CCOCC3)OCC)=O)C)nn2)cccc(C)n1 C1(CC(=O)N(C2CCCN(C)C2)C)CC2(C1)CN(C(C1CNC(=O)C1)=O)C2 C1(CC=C)(C(=O)NCC(O)CCC2CC2)CCCN1C(c1cccnc1)=O O(C1CCc2c(OC(F)(F)F)cccc21)CCSCCNC(=O)OC(C)(C)C CCC(C(C)C)C(C(=O)NC1COC1)N1CCCC(c2ccccn2)C1 N1(C(c2c(CC)nccn2)=O)CCN(C(=O)C(C)Sc2ccccn2)C(C)C1 n1(CC(N2CC(CCCC)N(C(C)=O)CC2)=O)ccc2cc(Br)ccc12 CC(C)CC(O)CC(=O)N1CCC(C)(C)C1CC(N1CCOCC1)=O C(=O)(C1CCCc2nn[nH]c21)NC1C(CNC(Cn2ncc(C)c2)=O)CCCC1 CC1(C)CC(NC(C2(C)CC2(F)Cl)=O)CN(c2ncc3ncnc-3[nH]2)C1 C(=O)(NN(C)c1cnccn1)NCCC(C)Oc1ccc(I)cc1Cl C(=O)(C1=CC(c2ccccc2)=NS(=O)(=O)N1)OC(C(C)C)C(=O)N1CCCCC1 N1(C(C2CC(OC)(OC)C2)=O)CC2(CC(Nc3ccc(C=O)nc3)CO2)C1.O c1(C(=O)NCCCC(C)NC(CCSCCCC)=O)cc2ccncc2[nH]1 N1(C(C=CC(C)C)=O)CC(NC(c2cccc(F)c2Cl)=O)CCC1C N1(C(CC2N(C(CN3C(=O)CCC3)=O)CCC2)=O)Cc2cccc([N+](=O)[O-])c2C1 c1(COC)ccc(C(=O)NC2(CSC)CC2)o1.N12CCC(C1)C2=O CCC(C(=O)N(CCCNC(c1ccc(CSC)s1)=O)CC)OC Cc1cc(C)c(C(=O)NC2CCCC(C)C2)c(C)c1.C1(C=O)NC(=O)C2CC12 c1(C(=O)NCC2CC(NC(C(C)OCCC=C)=O)C2)cc(Cl)nnc1O c1(C(=O)NCCNC(CCCC)=O)cc2sc(C)nc2[nH]1 c1(C(N2CCC(Cn3cc(-c4cccc(F)n4)nn3)CC2)=O)c(Cl)cncc1Cl C(CCN=c1[nH]nc(C)o1)N(C(Cc1cccc(OC)c1)=O)C n1(CC(=O)O)nccc1C(N1CCCC1)=O.N1(CCC=O)CCC(F)C1.CC c1(SCCC(=O)NC2C(C)CN(C(=O)CP(C)(C)=O)C2)nc2ccccc2o1 C1(C)(OC)CN(CC(N2CCCC2)=O)C1.C1(C(NC)=O)CCN(CC(C)C)C1.C c1(CNC(=O)CCc2cnn[nH]2)ccc(C(N2CCC(CO)(CO)C2)=O)cn1 CC1(C)C(C(N2CCC(C(C)(C)C(=O)Nc3cccc(Cl)c3)C2)=O)C1(F)F c1(C=O)ccc(Cl)c(C(F)(F)F)c1.C(C=O)(C1CCC1)OCC.C1CC1.N C(=O)(C1=C(C)CCC1)NC(CN(C(=O)C(C)c1cccs1)CC)C c1(NC(C(c2scc(C)c2C)N(CC(=O)OC)CCC)=O)c(C)cc(C)cc1C Cc1c(Cl)c(C(=O)NC2CC(C)CN(C(c3cc4n(n3)CCC4)=O)C2)nn1C C#CCC(CC#C)C(=O)N1CCN(C(=O)CCNC(=O)CO)C(C2CCCC2)C1 N1(C(COCCCC)=O)CCCC1C(N1CCC1(C)C(=O)OCC)=O C(CCC(C(=O)Nc1cc(F)ccc1O)NC(c1csc(=N)[nH]1)=O)OC C(C(C)(C)C)NC(C)C.C(=O)C=O.C(C)CN(C)C=O.C(C)(C)C c1(OC)cc(Cl)ccc1N1CCN(C(=O)NCC2CCC3(CCC3)O2)CC1 C(C(C)C(C)C(=O)N1CCC(O)(C(C)NC(c2occc2Br)=O)CC1)OC c1(C(N2CC=CC(NC(c3c(N)nccn3)=O)C2)=O)cc2sc(Cl)cc2s1 N1(C(CONC(C2(CC)CCOC2)=O)=O)CC2(CC(CO)CO2)C1 c1(-c2nc(C(C)C)oc2)nc(C2CC2)nn1CC1CCCOC1 C1(C)(C(N(CC(C(=O)NC(CCCC)CC)C)C)=O)CC(=O)N(C)C1 Cc1cc(C(=O)NC(C)C(CO)NC(C2CCCC2)=O)n(C2CC2)n1 C1(CC)CN(C(=O)C(C2CCCC2)OC)CC1C=O.C(Cc1ccco1)CO.N c1(C(=O)NC(CN(C(c2cnc(N(C)C)cn2)=O)CC)C)ccn2nccc2c1 CCCC(COC(C)(C)C)NC1(c2nnnn2C2CCOC2)CSC1.CC c1(C(N2CC(CCNC(C=CCC)=O)OC(C)C2)=O)cc2ncccc2[nH]1 N1(C(C(CC=C)OC)=O)CCC2(CCC2NC(c2cc(C)[nH]c(=NC)n2)=O)CC1 c1(-c2c(CC)ocn2)nc(-c2ccc(N)cc2)nn1CC1(CO)CC1 N1(C(N2CCC(OCC=C)C2)=O)CC(=O)Nc2ccccc2C1C CCS(=O)(=O)c1ccccc1C(N1CC2CCN(C(=O)C(C)O)CC2C1)=O Cc1ccc2cc(C(=O)NCC3CCCN3C(=O)CSC(F)(F)F)ccc2c1 c1(CC(N2CC(NC(c3c(CC)noc3)=O)C(OC)C2)=O)c(F)cccc1Cl N1(C(C2CC(C)(C)C2C(F)(F)F)=O)CC2(CCN(C(=O)C=O)C2)C1.C1CC1 c1(C(=O)NCC2(C)CCN(C(=O)C(F)=C3CCC3)C2)cccc2c1C(=O)NC2 CCC(C)C(=O)NNS(=O)(=O)CCNC(=O)OC(C)(C)C c1(C(=O)NC2C(F)(F)C23CCC3)ncnc2[nH]cnc12 C1(CC)(NC(=O)CCNC(c2ccc(NC)cn2)=O)CCCCCC1 C(CC(C)(C)C)(C(=O)N1CC(C)CC1(C)C)OC.c1(C=O)cc(C)cc(C)c1.N N1(C(C(C2CC2)OCC)=O)CCC(C2CCCN(C(=O)CCC(C)OC)C2)CC1 N1(C(C(C)OC)=O)CCC2(CC1)CC(NC(=O)CCN1CCN(C)CC1)CCO2 C1(NC(C2(CC#C)CCC2)=O)CN(C(=O)CCn2ccccc2=O)CC1OC C1(C=O)CC(C2CCOCC2)=NO1.c1(COC)nc(NC2(C)CCC2)cc(Cl)n1 c1(N(C)C)cc(C(N2CC3C(NC(C4C(F)(F)C45CC5)=O)C3C2)=O)ccn1 C1(CC(=O)NCC2(OC)CCC2)CCCCC1NC(c1coc(C)n1)=O c1(C(=O)Nc2cc(OC)ncn2)csc2c1CCN(Cc1cn(C)cn1)C2 C1(C(N2CC(CCC)N(C(=O)C=C3CC3)CC2)=O)Cc2cccc(C)c2O1 C1(c2n(CC)nnn2)(Nc2ccc(Oc3ccc(Cl)cc3)cc2)CN(C)CC1C C1(CNC(c2ccc(C)nn2)=O)N(C(c2sccc2C(F)F)=O)CCCC1(C)C c1(OC)c(CC(N2CCC(O)(C(C)NC(C3CCCC3)=O)C2)=O)cccc1F C1(C(=O)NC2CC(OC(C)C)C2)CCCN(C(c2ccco2)=O)C1C.C(N)=O c1(OC)ccc(C(N)=O)cc1NC(c1ccc(F)cc1)CC1CCC1 CC1CC(C(=O)N2CCCC(C(=O)NCC3(CCO)CC3)C2C)=NO1 C12(NC(c3c(CC)con3)=O)CCOCC1CN(C(c1cnnn1C)=O)C2 N(C1CCCn2cnnc21)C(C1CCN(C(c2cncc(F)c2)=O)CCO1)=O C1(C(=O)NC2(C(=O)NOCC3CCCC3)CSC2)C2CCCCC12 N1(C(c2c(C)[nH]nc2C(F)F)=O)CC2CCCN(C(=O)C(C)C(O)C(C)C)C2C1 C(C(=O)NCC(N1CCCCC1)C)(C(C)O)NC(c1c(C)non1)=O CC(C)(C#N)C(=O)N1CCC(C(F)C(=O)NCCCC2CCCCC2)C1 N1(C(=O)OCC)CCC(N(C(C2(c3ccccc3)CC2(Cl)Cl)=O)CC)CC1 N1(C(C(Br)=C(C)C)=O)CC2CCCC(N=c3[nH]c4ccc(C(F)(F)F)cc4s3)C2C1 N1(C(C(C(C)O)N(C)C)=O)CCC(C(=O)NCC(=O)N(C)O)C12CC2 O1n2c(nc3ccc(Br)cc23)C1.c1(C(=O)OC)ccc(I)cn1 CC(C)(C)C(CO)C(=O)N1CC(=O)NCC1C(=O)NCCc1ccon1 Cc1ccc(N(C)C)c(C(=O)N)c1.C1(C)(C=O)C(C)(C)C1(C)C.C1COCC1 N1(C(C(C)C)=O)CCCCC1C(=O)NC1CC(F)C1.c1(C=O)csc(Cl)n1.C c1(OCC(=O)NC2(C)CCN(C3CCNC3=O)C2)cccc2ccccc12 N1(C(c2cn(C)c(=O)n2C)=O)CCN(C(=O)C(C)(O)C2CCC2)CC(C)(F)C1 Cc1csc(=O)n1CCC(=O)NC(CNC(=O)C1=CCOC1)C(C)(C)C CCCC(CC(C)C)C(=O)N1CC(F)(CNC(C2CCC2n2ccnc2)=O)C1 c1(C(=O)NC(C2CCN(C(c3c[nH]c(=N)o3)=O)C2)C)cn2ccnc2s1 C=CCC(C(=O)NC1(CC(C)C)CC1)NC(=O)C(C)OCC(C)C C1(NC(CC(C)(C)C)=O)COC2(CCN(C(=O)C=Cc3ncc[nH]3)C2)C1 C(C(CNC(C1(OC)CCSC1)=O)C(F)(F)F)NC(c1ccc(CC)o1)=O c1(OC)c(C(N2CC(NC(=O)CCC(C)(F)F)CC2(C)C)=O)nc(O)nc1O N1(C(c2nc(COC)oc2)=O)CC(CNC(c2ncccc2N)=O)CC1C N1(C(c2ccoc2)=O)CC(C2CCN(C(c3cc(C4CCC4)no3)=O)CC2)C1 Cc1c(C(N2CCC(NC(=O)CCn3c(C)ccc3C)C2)=O)nn2c1CCCC2 C1(CC(C)C)CCCN(C(=NCCC(F)(F)CO)NCC(F)F)C1 C(=O)(C(F)CC(C)(C)NC(C1CC1(F)Cl)=O)NCC1(OC)CCC(C)C1 CC(C)C(O)C(C)C(=O)NCCCCCC(=O)NCC1(O)CCCC1(C)C C(CC(C)C(=O)NC1CN(C(c2ccnc(CC)c2)=O)CC1C)=CC S(=O)(=O)(c1ccccc1F)NC1CC(C(=O)NCc2cn(CC)nc2)C1 Cc1nc(C(=O)NC(C)C)c(C)n1C1CC1.C1(S(N)(=O)=O)(C=O)CC1 c1(C(N2CCOC(C3CN(C(C4CCCOC4)=O)C3)C2)=O)cc2n(n1)CCC2 Cc1ccn(C(C)C(=O)N(C2(CC(=O)NC3CCN(C(C)(C)C)C3)CC2)C)n1 N1(C(c2c(C)cc(C)c(N)c2)=O)C2CCC1CN(C(c1nccnc1N)=O)CC2 N12CC3(CC3)CC1C2=O.N1(C(=O)NCC)CCN(S(=O)(=O)CCO)CC1 C1(NC(C2(CC=C)CC2)=O)CCCCCN(C(=O)CS)C1.c1ccsc1[N+](=O)[O-] C(c1ccc(-c2ccccc2F)s1)=CC(=O)NCC(CC1CC1)CO Cn1cnc2c[nH]c(=NCC3CN(C(c4cc(Cl)cc(Cl)n4)=O)C3)nc12 c1(C(=O)NCC(C)CNc2cccc(F)c2C#N)ccc2c(n1)OCCO2 c1(C2(N(C3CC3)C=O)CC2)ccc(Cl)cc1Cl.N1(C(=O)N)CCCC1.CCO Cc1ccc(OCCC(=O)NCC(O)CCNC(=O)CCc2ccc[nH]2)c(Cl)c1 c1(OC)cc(C(=O)NC2CCN(C(=O)C(=O)NCC3CC3)C2C)ncc1Br N1(C(c2cc(OCC)no2)=O)CCCC(F)CC1.N(C)(S(N)(=O)=O)CC=O N1(C(C(CCOC)NC(=O)C=Cc2cocn2)=O)CCCC(C)(C)C1C Nc1nc(Cl)ccc1C(=O)NCC1CCC(NC(c2csnc2Br)=O)C1 C(=O)(C(CNC(c1ccncc1N)=O)C(C)(C)C)NC(C)CCC1CC1 c1(OC)cc(CCC(N2CCN(c3ccnc(Cl)n3)CC2)=O)ccc1N C(=O)(C1=Cc2ccccc2C1C)NC(CC)(C)C(=O)O C1(CC)CN(C(=O)CN2CCN(C)C(=O)C2)CCC1.C1(C=O)CCC(=O)N1C.N c1(C(=O)NC(C(C)C)(C)CNC(=O)C(C)CF)cc(Cl)c2[nH]c(O)nc2c1 C=CC1OCCC1C(=O)OCc1ccccc1C(=O)C(F)(F)F CCC(CNC(=O)C=NOC)(CC)NC(=O)COc1cncc(Br)c1 n1(C(C)C)nc(Br)cc1C(=O)NCc1n[nH]c(Cc2cccc(F)c2)n1 N1(C(c2cnc(OC)s2)=O)CCC(C=CC(N2CCN(C)CC2)=O)CC1.C1CC1 Cc1cc(CC(N2CCCC(CNC(C3(C)CCC3)=O)C2)=O)cc(F)c1 c1(N(CCC)CCNC(=O)C(CC)SC)ncc(C(=O)OC)c2sccc12 CCC(C)(C)CCCC(=O)NCC(O)Cn1ccnc1 CC1(C)CN(C(c2cccn3cnnc23)=O)C(CNC(c2csnc2Cl)=O)CO1 CN1CCC(O)C(NC(C2CCN(C(C3CC34CCC4)=O)C2)=O)C1 N1(C(c2cc(C)on2)=O)CCN(C(C2CCC2C#N)=O)C(C)C1 Nc1cc(F)c(O)cc1C(N1CCC2CCC12CNC(c1sccc1Cl)=O)=O n1(CC(=O)NC2CN(C(=O)Cc3cnoc3)C3CC23)ccc([N+](=O)[O-])n1 C1(NC(C=CC(C)(C)C)=O)(C)CC2CCC1CC2.C1(C=O)CCCC12CC2.N N1(C(C(C)(C2CC2)OC)=O)CC(C2CCCN(C(=O)CC(=O)NC3CC3)C2)C1 c1(C(N(C(CC)C(=O)N(CC(C)(C)COC)C)C)=O)ccc(NC)cn1 c1(CC(=O)N(CCCCNC(c2c(C)noc2)=O)C)coc2cc(F)ccc12 C1(C)(NC(c2c(CC)non2)=O)CCC(Nc2ncc(Br)c(O)n2)CC1 C(N=c1[nH]c(=NC(C)c2ccnc(Cl)c2)[nH]c2cc[nH]c12)c1snc(COC)n1 C1(C2(NC(C3CC4CC4C3)=O)CC2)CCCN1C(C1(n2cccn2)CC1)=O C1(C)(C(N2CCCC(CC(N3C(C=C)CC3)=O)C2)=O)CCC(C)CC1 c1(CCNC(c2cn(CCO)nn2)=O)n[nH]cc1C(=O)NCCC1CCOC1 c1(OC)ccc(CC(=O)NC)c(C)c1.C1CC2CC2N1C(=O)C(O)C1CCCC1 N1(C(CC(C)N(C)C)=O)CCC(O)C(N(C(=O)Cc2cncs2)C)C1 C1(NC(C2CCCOCC2)=O)CC2CCC1N2C(c1cc(O)cc(F)c1)=O c1(CC(C)C(N2CCN(C(=O)C3=CCC3)CC2)=O)cccc(F)c1.C12CN(C1)C2 C1(CN(C(=O)CC2CC2)C2CC2)CCCN1C(=O)C(C1(O)CCCC1)F c1(OC)cc(Cl)c(C)cc1C(N1CCCC(C)C1)=O.C1(CC=O)CN(C)C1.C N1(C(C(CC)COC)=O)CCC(C2CC2)(CNC(c2cccn2C(C)C)=O)C1 O(NC(=O)CCN(C(=O)Cn1ncnn1)CC1CC1)CC(=O)OC c1(C(=O)NC(CN(C(CC(CC)(C)C)=O)C)C)c(C(F)F)nc2ccccn12 c1(C(N2CC(CC(C)NC(C3CC3CF)=O)C2)=O)cccc[n+]1[O-] c1(C(=O)N)cc(C(C)(C)C)nn1C.C1(CC)CCN(C(c2ccc(Cl)o2)=O)CC1 CC1OCCC1CNC(=O)CCCNC(=O)Cn1nccn1 N1(C(c2cc(C)ncc2)=O)CC(C(=O)N(C)CC2(C)CCC2)C2(CCC2)C1 c1(C(=O)NCC(CC=C)Nc2cccc(C)c2)ccc(COC2CC2)cc1 C1(CNC(C(C)CO)=O)CN(C(=O)CCC2CCC(=O)C2)C2(CCC2)C1 c1(C(=O)NCCC2CCCN2C(C2CCNC2=O)=O)cc(F)ccc1Br c1(C(N2CC(NC(c3cc(=O)cc[nH]3)=O)C(O)C2)=O)ccn2nccc2n1 C1(NC(CC(C=C)CCC)=O)CN(C(=O)CCCc2ccsc2)C2(CCCC2)C1 C(CCCCC(=O)NCC1CC(O)C(O)C1)NC(CC1CCC(C)(C)O1)=O CCC(CC(=O)NCC1(O)CN(C(=O)COCCN(C)C)C1)C1CCC1 C(=O)(CCC(=O)N)OC.C1CC(F)CN1C(C1CC(=O)N(C(C)(C)C)C1)=O c1(C(=O)NCC2(O)CC(NC(c3cc(C)[nH]n3)=O)C2)ccc([N+](=O)[O-])cc1 N1(C(c2cc(Cl)nc(=N)[nH]2)=O)CCCC2(CCCCC2NC(C2CC2(Cl)Cl)=O)C1 C1(C(=O)OC)CCCC(NC(=O)NN2CCC(CC3CCCO3)CC2)CCC1 C(C)(CC(F)(F)F)NC(COCC(C)C)=O.c1(CC(=O)N)ccc(Cl)nc1 CC1CN(C(C2OCCC2C)=O)CCCN1C(c1cnc(-c2cnn(C)c2)s1)=O N1(C(c2c(C)n[nH]c2)=O)CCCC2(CCN(C(=O)C3=CC4CC(C3)CC4O)C2)C1 c1(CN(C(C(F)OC)=O)C)cnn2c1CN(C(=O)C(F)C1CCC1)CC2 c1(OC)cc(N)c(Cl)cc1C(N1C(C)C2CC1C2)=O.C1(CC=O)CCCOC1.N Cc1nn(C(C)C)c(C)c1CC(=O)NC1CCCCC1.C(=O)(CS(C)(=O)=O)N C(C1=CCCN(C(=O)CC2CCCCC2)C1)NC(c1noc(CC)c1C)=O c1(C(N(CC)CC2CCN(C(C3OCCC3C)=O)CC2)=O)ccc2scnc2c1 C1(NC(C2C(C(C)C)(CC)C2)=O)CCN(C2CCCC2)CC1 C1(NC(C(CC)(C)C)=O)COC2C(NC(C34CC(C)(C3)OC4C)=O)COC12 Clc1cccc(C2(Cn3nc(-c4ccc(Cl)nc4)nc3C3(C4CCCO4)CC3)CC2)c1 Cn1cncc1C(=O)NCCS(=O)(=O)NC(C)(C)C N1(C(c2cc(OC)c(O)c(Cl)c2)=O)CCC2CN(C(=O)CCC(C)SC)CC2C1 c1(CN2CCC(C(n3cc(C(C4CCCCC4)=O)nn3)C)C2)nc(C#N)cs1 CCCCCCC(F)C(=O)NC(C)(CNC(c1cncc2nc[nH]c12)=O)C(C)C C1(CNc2scc(CC(=O)OCC)n2)CN(Cc2ccc(C)cc2)CCO1 O=C(C1c2c[nH]nc2CN1C(=O)CC1CCCO1)NCCCCCCO C12(CC)CN(C(c3cncn3C(C)C)=O)C(C)(C1)C2.C1(C=O)CC1(C)C Cc1cc(N)n2ncc(C(=O)N(C)CC3CCCN3C(=O)C3=NOC(C)C3)c2n1 c1(C(=O)NCCC2(COC)CCC2)sc(N2CCOCC2)nc1C C1(C(=O)NC2CN(C(c3c(C)cc(C)c(Br)c3)=O)C2)CCc2ccccc2C1O C1(NC(Cc2c(C)nc[nH]2)=O)CCCC(NC(=O)COCCF)C1 C#CC(C(C)C)NC(=O)C(c1ccco1)NC(C1CC(=O)C1)=O N(C(=NCCCC1CCOC1)NCCCCl)CC(CO)C1CCOC1 N1(C(c2ccnc3ccsc23)=O)CCCCC12CC(NC(C13CCC(C1)C3)=O)C2 N1(C(C(C2CCCC2)OC)=O)CC=CC1Cn1cc(-c2ccsc2)nn1 C1(C2CCCN(C(=O)CCC(C)C)C2)(NC(CC2(C=C)CC2)=O)CC1 C(=O)(CCC(N)=O)NCC(CCC)NC(=O)C(C1CCCC1)OC Cc1cc(C(c2nnnn2CCCSC)NC(C2(C)COC2)C)cnc1C.C c1(C(N2CC(CCC)C2)=O)cccc(C2CC2)c1.c1(C=O)nc(C2CC2)cs1.N CC(C)C(O)C(F)(F)C(=O)NC(C1CCN(C(=O)CCS(C)=O)C1)C C(C1CN(C(c2ccc(C)cn2)=O)CC1C(=O)NC(CO)CCOC)=CC Cc1cc(CC(=O)NCC(CO)NC(=O)C(F)(F)c2ccccc2)cc(F)c1 N1(C(CN2CCC(C)C2)=O)CC2COCC2(C(=O)NC2CCN(C(C)(C)C)C2)C1 Cc1cn2ccc(C(=O)NCC3COCCN3C(c3cnc(C)n3C)=O)cc2n1 N1(C(c2nc(CCC)oc2)=O)CCC(NC(c2cc(Cl)ns2)=O)C1C(C)C C1(C(=O)NCC(CNC(C23CCC(CC2)C3)=O)CO)COc2ccccc2C1 CCC(C)CCC(=O)N1CC(NC(=O)C(F)(F)c2cnn(C)c2)CC(C)C1 Cc1ccc(CN(CC(=O)N(C)CCNC(=O)C(C)(C)CC2CC2)C)cc1 c1(C(=O)NCC23CC2CN(C(c2ccsn2)=O)C3)ccc2c(c1)COCCN2 Cc1nc(=NC(=O)CN2CCN(Cc3cc(O)c(O)c(O)c3)CC2)s[nH]1 C1(c2c(OC)cncc2)NC(=S)N(c2ccc(C)cc2)C2=C1C(=O)N(C1CC1)C2 C1(C2CN(C(c3ccc(-n4ccnc4)nn3)=O)C2)(NC(=O)CC2CC2)CC1 C=CCC(C)C(=O)N1CC(C2CN(C(=O)CC3CC(OC)C3)CCO2)C1 C1(CC(=O)N(C(C)C)CC)CCCCC12CC2.c1(C(=O)N)coc(N(C)C)n1 C1(C(=O)NCc2c(CC)n[nH]c2)CN(C)CCN1C(c1cc(C)co1)=O O=C1Cc2ccc(C(=O)NC3CN(C(c4cnn(C(F)(F)F)c4)=O)C3)cc2N1 CC1(CNC(c2ccc(-c3cccs3)[nH]2)=O)CCCC1.C1(CC=O)CCCC1.N c1(C=O)c(C)nn2cc[nH]c(=O)c12.C1CCCC1.C1(CC(=O)NC)(OC)CC1 C(=O)(C(F)(F)CO)N1CCC(CN(C)C(c2cccnc2)=O)C1 N1(C(c2n(CCC)ncc2)=O)CCCCC(N(C)C(C2C3CNC(=O)C23)=O)C1 C(=O)CC1=CCOCC1.C=C=CC(C)C(=O)NCCN(CCC)C(C)=O CC(C)C(C)CC(=O)NC1CCCC1NC(=O)CCC(=O)N(C)CC.C(N)=O C(c1cnc[nH]1)=CC(=O)N(C1CCN(C(C2CC(C)CO2)=O)C1)CC N1(C(c2c(C)noc2C(C)C)=O)CCC(C2(NC(=O)C=C(Cl)Cl)CC2)C1 N1(C(C(c2cn(C)nc2)NC(=O)CN2CCCCC2)=O)CC2CC2C2CC12 Cc1cc(CNC(=O)CC2CCCCN2C(=O)CC2C=CCCC2)nnc1C c1(C(=O)NC2C(NC(c3cccc(N)c3O)=O)C2)cc(F)c(Br)c(F)c1 C1(CC(=O)OC)CC(NC(=O)Nc2cccc(-n3ccnc3S)c2)C1(C)C N1(C(C2(C(C)NC(C(CC(C)C)O)=O)CC2)=O)CCC([N+](=O)[O-])CC1 C(=O)(C(O)C(C)(C)CC)N1CCC(N(CCC)C(C2CC2CF)=O)CC1 c1(C(N2CCC(O)(CCNC(c3cnn[nH]3)=O)C2)=O)cncnc1O.C1CC1.C C(CC(C)C(C)C)NC(c1[nH]c(CC)c(Cl)n1)=O.c1(C(=O)N)ccc(N)c(F)c1 C1(CNC(C(C)OCOC)=O)CCN(C(C23CCC(C2)C3)=O)CC1(F)F C1(OC)CCCN(C(c2sccc2Br)C(=O)NC2CC2)C1C C1(c2nnnn2Cc2cccs2)(NCc2cnc(C)s2)CCCSC1 C1(C(=O)NCCN(CCOC)C(c2csc(=N)[nH]2)=O)CCC(OC)C1 C(=O)(C(C(C)(C)C)NC(N)=O)N1CCC(C)(CC(NOCCN(C)C)=O)C1 C1(NC(c2ccnnc2O)=O)CC12CCN(C(C1CCC(O)CC1)=O)C2 CCCCCC(O)C(=O)N1CC(C(=O)NCC2(CO)CC=CC2)C(CC)C1 C(C)(CCCCNC(c1cc(C)n(CCO)n1)=O)NC(COCCOC)=O C1(C)(C=O)CC(C)(C)C1.C(=O)(C(O)C)N1CC(CC(=O)OCC)C1.N CCC(C(=O)N1CCOCC1CC(=O)NC(C)C1CC1)C(C)(C)CC Cc1cc(CC(=O)NCC(C(C)(C)C)NC(=O)C2=CCCSC2)ccc1CO c1(OC)ncccc1C(c1nnnn1C)NC(c1nnc(CO)s1)C c1(CCNC(=O)C(=O)NCC2CCCCN2CC(F)F)ccc(F)cc1Cl C(N=c1cc(C2CC2)nc[nH]1)C1C(NC(CC(C)(C)c2ccccc2)=O)CCC1 C1(C(N2CC=CC2)=O)CCC(C2CC2)CC1.c1(C(=O)N)ccsc1C(F)(F)F Cc1c(C(=O)NC2CN(C(c3cncn(C)c3=O)=O)CC2C(F)F)cccc1N N1(C(C(CC)CN(C)C)=O)CC(C)CN(C(=O)CCN2CCNC(=O)C2)C(C)C1 c1(C(=O)NC(C(C)c2ccccc2)C(=O)O)ccccc1C#N Cc1scc(C(=O)NC2CCC(C(N3CCC(N4CCC4)C3)=O)CC2)c1C c1(C=O)ccccc1.O=CCCCNC(=O)C(=O)N1CCC1CO.C1CC1.C N1(CC(=O)OCC)CCC(C(N2CCOCC2)C)CC1 C1(n2cc(CNC(=O)CCN3CCC3)nn2)CCN(C(=O)COC(F)F)CC1 Cc1nn(CC(=O)NC2C=CCN(C(=O)Cc3cc[nH]c3)C2)c(=O)n1C C1(C(=O)NCC(c2ncn(C)c2)O)C=CCN(C(C2CC(C)(F)C2)=O)C1 S(=O)(=O)(c1ccc2c(c1)CCO2)N.c1(C(N)=O)ccc(NC(C2CC2)=O)cc1 CC1=NOC(C(N2CCCC2C2(NC(=O)C=CCn3cncn3)CC2)=O)C1 C12(C(=O)NC(C)CC(F)(F)F)CCC(CN(C(=O)CCc3nccs3)C1)C2 N1(C(CCOCCOCC)=O)CC(O)CC1C(=O)Nc1c[nH]ccc1=O c1(C(=O)NC2(C)CN(C(CC3C(C)OCC3)=O)C2)cn(C)[nH]c1=N c1(CC)cncc(NC(=O)NC(c2ccc(C)o2)Cc2cccc(Br)c2)c1 c1(C(N(CC)C)=O)cc2cc(Cl)sc2[nH]1.c1(CC)c(C=O)cnn1CC(C)C.N N1(C(C(CCC)NC(C)=O)=O)CCCN(C(C2CCCC2(F)F)=O)CCC1 c1(OC)cc(CN2CC3CN(c4ccnc(SC)n4)CC23)c(OC)cc1Cl c1(-c2cnc(OC)c(C(=O)Nc3cncnc3C)c2)ccc2c(c1)OCC(=O)N2 Cc1ccc(C(c2nnnn2C2CCC2)NCCc2cnccn2)cc1F C(=O)(C1CCCc2c[nH]nc21)N1CC(NC(=O)CN2CCCS2(=O)=O)C1 c1ccc(O)cc1.C(COc1ccccc1)(C(=O)NCCC)OC.C(=O)(C)N C(CCCCCC(=O)NCCC#CCO)NC(c1c(CC)noc1)=O N1(C(Cc2cccc(OC)n2)=O)CCC2CCC(NC(=O)C(O)CCSC)C1C2 CCC(C)C(CC(=O)N1CCC(C2(C)CC2)CC1)NC(=O)C1=NOCC1 CC1CCCN1C(c1ocnc1C1CC1)=O.c1(CC(=O)N)ccc(C2CC2)cc1 C#CCCCCCC(=O)NCC1CCCCC1C(=O)NC1CCC(CO)C1 N1(C(C)=O)CCC(C2CC2)C1.C1(C(=O)NCC=O)(OCC)CC1.N(C)C C1(C(=O)NCC2(n3ccnn3)CC2)CCC(O)CN1C(c1cc(Cl)c[nH]1)=O N1(C(C(C)(C2CC2)OC)=O)CCCC(CCNC(=O)CCCSC)C1 C(CCC(C)C(=O)NC1CCC(NC(c2ccc(C3CC3)s2)=O)CC1)OC C1(c2ccccc2)(C(=O)NC2C(CNC(C(C)(F)F)=O)CC2)CNC(=O)C1 Cc1cc(N(C)CC2CN(C(c3csc(C)c3C)=O)CCO2)ncc1C#N N1(C(c2cc(C#N)on2)=O)CCC(NC(c2ccccc2C(N)=O)=O)C(F)C1 N1(C(Cc2ccc(C)cc2)=O)CCC(F)C(N=c2ccnc(N3CCCC3)[nH]2)C1 C1(C(=O)NCCC(C)(O)C2CC2)C2CN(C(C3(Cl)CCCCC3)=O)CC12 C(C)(C)(CC(=O)NCC1COCC1NC(=O)C(C)C(C)O)OC C1(CNC(C(=O)NCC(c2ccccc2)CC)=O)CCCC1CC(=O)OC CCC(CCCC(=O)NCCC(C)(C)N(C)C)NC(c1cn(C)ccc1=O)=O c1(CC)ccc(C(N2CC3CC3(NC(C3CN(C)CCO3)=O)C2)=O)c(F)c1 [SH](=O)(=O)C(F)(F)F.C1(O)(C(N(C)CC)=O)CCOC1.C(=O)CC.CC.O CCC(CC)C(C)C(=O)NC1CN(C(=O)COC)C(C)(C)C1.c1nc(C)no1 C1(CC(=O)NC2(c3nc(C)[nH]n3)CC2)CCCN(C)C1.C(=O)C(C)C(F)F.N Cc1cc(C(=O)NCCN(C)C(c2coc(Cl)n2)=O)ccc1[N+](=O)[O-] c1(C=O)ccc(C2CC2)c(F)c1.C1(CNC(c2c(C)snn2)=O)CCCCC1.N n1(CC(=O)NC(CNC(C(C)N2CCC2)=O)C)ccc2ccc(F)cc12 N#CC1(C(=O)NCCc2ccc(C)cc2)CC2CC2C1.C(=O)(CC1=CCCC1)N CC1CC(C#N)(C(=O)NC2CC(CCC(=O)NCCN3CCC(O)C3)C2)C1 CC(CCN(C)C)C(=O)NCc1ncoc1CC.C1(C(C=O)F)CCOCC1.N C12(C(N(CCC)C)=O)C3C4C1C1C2C3C41C#N.C1CC1C=O.CCO.C C(C(C)(C)CNC(=O)CN(c1ccncc1)C)N(C(C(C)SC)=O)C c1(SC)ncc(CN2CC3(CC(CC=O)C3)C2)c(Cl)n1.C(C1CC1)C1CC1 C1(CC(=O)NCC(C)OCC#C)CCCCC1NC(C1CCCOC1)=O c1(SCC(N2C(Cn3cc(CCC(C)=O)nn3)CC2)=O)ccc(C)cc1C C1(CNC(c2cc(CC)no2)=O)CCN(C(=O)Cc2nnc(S)n2C)CC1C Cc1ccn(C(C)C(=O)NC(C)(C)C=CC(=O)N(C2CC(CO)C2)C)n1 c1(C(=O)NC(C)CC(C)NC(=O)CCCCc2cnn[nH]2)c(F)ccc(N)c1F c1(OCC)c(C(=O)NCC2CCC2NC(c2cnsn2)=O)cccc1F CN1CC=C(CC(=O)NCC2COCCN(C(C34CC=CC(C3)OC4)=O)C2)CC1 Cc1cc(C(=O)NC(C2CCCCN2C(c2cc(F)cs2)=O)C)cc(=O)n1C N1(C(C(=O)C2CCCC2)=O)CCCC(C2CC2NC(c2ccc(Cl)o2)=O)C1 c1(CC(C)C)ccc(C#N)c(N(CCC)C(C)C)n1.C(=O)C(F)=CC1CC1.N Cc1cccc(C)c1C(N1CC(C(N2CCC(N(C)C)C2)=O)C2(CC2)C1)=O Cc1ccc(CC(=O)NC2CC(CNC(C3CCC34CCCO4)=O)C2)c(C)c1 Cc1ccc(Br)c(C(=O)NCC(C2CC2)N(C)C(C23COCC2C3)=O)c1 Cc1cc(O)nc(CNC(=O)CONC(C2CCC(=O)O2)=O)n1 N1(C(CC(C)SC)=O)CC2(CC2)CC1CNC(=O)C(c1cccc(F)c1)C c1(Cc2n(CCOC)nnn2)ccc(Cl)cc1.c1(CC)nc(C(F)(F)F)cs1.N c1(OC)ccc(C(N2CCC2CNC(C2CCCC(=O)N2C)=O)=O)c(C)n1 C1CN(C(c2cc[nH]c2C2CC2)=O)CC2(CC2)C1.C1(CC)CCCCC1C(=O)N N1(CC(=O)NC(C(=O)OC)C(C)(C)C)CC(CC2COCCN2)c2ccccc21 CN1CCN(C(C)(C)C(=O)N2CC(F)(C)C2)CC1.C(=O)C(F)(F)c1nccs1.N c1(C(N2CC(C)(NC(c3cnn(C)c3F)=O)C2)=O)cnc(O)n(C2CC2)c1=O C1(C(C(=O)Nc2ccnc(O)c2)O)CCC(F)(F)CC1 c1(C(=O)N)ccc(=O)n(C)n1.c1(C2(C=O)CC2)cccc(Cl)c1.C=C(C)CC c1(-c2c(C(N3CCC(O)(c4cccc(Br)c4)CC3)=O)c[nH]n2)cc(Cl)cc(Cl)c1 C1(C(C)NC(c2ccc(C(N)=O)o2)=O)CN(C(C2CC(F)C2)=O)CCO1.C c1(C=O)cn2cc[nH]c(=O)c2n1.C(CCC)(C(=O)N1CC(OCC)C1)=CCC.N N1(C(CSCC#C)=O)CCCCC1C1CCN(C(=O)CCC(=O)OCC)CC1 C1(C(=O)NC2CC2)CCCC12CCN(C(C1CCCN1C(c1ccon1)=O)=O)C2 C1(NC(C(CN(C(C=C(CC)CC)=O)C)C)=O)CCCC(OC)C1 C(=O)(CC(C)(C)CC)NCC1CCN(C(C(F)=CCC)=O)CC1 c1(C(=O)NC2CCCC(NC(c3cn[nH]c3)=O)C2)ccc([N+](=O)[O-])c(O)c1 c1(C(=O)NC(CN(C(C(C)OCCCC)=O)C)C)cc(N2CCOCC2)ncn1 C1(C)(CC)CC(C(=O)NC2CN(C(=O)Cn3ncnn3)CC2C)CCO1 c1(C(=O)NCCC(C)N(C(CC2CC(SC)C2)=O)C)conc1C(F)(F)F C(=O)(C1=C(F)CN(C(=O)CC2CCC(C)CO2)CC1)Nc1c(C)ccc(C#C)c1 c1(C(=O)NC(c2onc(COC)n2)C)ccc(O)c(OC)c1 N1(C(=O)OC(C)(C)C)CC(C)(C)OCC1C(=O)NCCCc1csnn1 CON(CCC(=O)N1CCn2cc(C)nc2C1)C(=O)C1C2CC3C(C2)C13 C(CCN=C(NCc1cccnc1Cl)NC(C)CF)SC C(CN=c1[nH]c(=NC(C)c2nnc3n2CCCC3)[nH]c2c1CCC2)=C(C)C N1(C(c2cc(C)[nH]n2)=O)CC2CC2(CNC(c2nccnc2C(F)(F)F)=O)C1 C(CCCC=C)(C(=O)NCC1CC1(C)C)NC(Cn1ncc(C#C)c1)=O C1(F)(C(=O)NC2C(NC(C(c3cccc(Cl)c3)C)=O)C2)CCCCCC1 N1(C(CS(CC)=O)=O)CCN(C(c2ncccc2OC(C)C)=O)CC1CO C1(C(=O)NC(C)Cn2ccnc2)C(O)CCN1C(C1C2(CC2)C12CC2)=O C(=O)(CCC(C)(C)C)NC1(C)CC(NC(C(c2c(F)cccc2F)N(C)C)=O)C1 c1(C(=O)N)c2c(nn1C)CCOC2.CC1=C(C(=O)NCC2CCC(O)C2)CCC1 N1(C(c2ccc(OC)nn2)=O)CCN(C(=O)CC(C)F)C(CS(C)(=O)=O)C1 C=CCC(CC=C)C(=O)N1CCCN(C(C2CCCC(=O)C2)=O)CC1C Cn1cc(C(=O)N)c(-c2nccs2)n1.C1(O)(C=O)CC(C)(C)C1.C1CCC1.C CCC(CCCO)N=c1cccc(S(=O)(=O)N(C)Cc2cccc(OC)c2F)[nH]1 CC(CNC(=O)CCOC1COC1)C(=O)NC(C)CCCO c1(C(=O)OC)cnc2c(Cl)c(N3CCCC(CNC(N)=O)C3)ccc2c1Cl C(=O)(CC1CCC(C)(C)c2ccccc21)N(CC(C)(C)C)CCC#C Cc1nc2cccc(C(=O)NCC(C)(CO)NC(C34CC(C)(C3)C4)=O)c2s1 C1(NC(C(CCOC)NC(=O)CCc2nncs2)=O)CCCC(CO)CC1 C1(C(N2CCC(N(C(=O)CC3CCCCC3)C)C2)=O)CCCNC1=O N1(C(c2cnnc(C)c2C)=O)CCC(C2CC2)C1C(=O)NC1CC(CC(N)=O)C1 c1(C(=O)OC)[nH]ccc1C(N1CC(O)(CC)C1)=O.c1(CC=O)scnc1C.N C(=O)(CCC(F)(F)C(F)F)NC(C1CCOC1)CNC(CC=C)=O c1(OCOC)cc(C)c(-c2ccnc(C(=O)NCc3cccnc3Br)c2)c(C)c1 C1(C)(CNC(C=NOC)=O)CCCC1NC(c1ccn(CC(F)F)n1)=O C1(C(C)OC)CCN(C(C2CCN(C(C3CCCCS3)=O)C2)=O)CC1 N1(C(C2C(C)(C)COC2)=O)CC(NC(=O)C(=Cc2c[nH]cn2)F)C2(CCCC2)C1 C(=O)(C1=CC(O)C(NC(c2ccsn2)=O)C1)NC(C#C)(CO)CO C1(NC(C2C(C=CC)CN(C(=O)CC(=O)OCC)C2)=O)CCn2cnnc2C1 C1(NC(C23N(C(C4CN(CC)C(=O)C4)=O)CC(C2)C3)=O)CCC(O)C(O)C1 CC(C)CS(=O)(=O)CC(=O)NC1CCC2CN(C(c3cnn(C)c3)=O)CCC2C1 C(=O)(CC(C)C(F)F)NC1(C(=O)NC2CCC3(C(C)C)C2C3)CCN(C)C1 C1(OCC(=O)NC2CC(NC(c3ncncc3Cl)=O)C2)CCCC(F)C1 Cc1cc(Br)ccc1C(N1CCC(F)(CNC(=O)COC2CCC2)C1)=O C12(C(=O)NCC3(NC(c4ccc(O)cc4Cl)=O)CC3)CCCC1C2(F)F C1(CN(C)C)CC(C(=O)N(C)CC2(C)CC2)CCO1.C1(C(=O)N)CCO1 C1(C(N(CC(CN(C(CCC=C(C)C)=O)C)O)C)=O)CC2CC1C1C2C1(F)F Cc1ccc(C(N2CC3CC2CN3C)=O)c(=O)n1C C1(C(=O)N)CC12CCCCC2.C1(C(=O)NCC2(CSC)CC2)CCCCC1 C1(NC(C2CC(SC)C2)=O)CN(C(C2CCOC2(C)C)=O)C(C)(C)C1 C(CN=c1[nH]c2ccc(F)cc2s1)C1CCC(NC(C2(C)CCCC2)=O)C1 c1(C(=O)NC2(C)CCCN(C(c3cccnc3)=O)C2)cccc2nccn12 C1(C)(CCC=O)CCC(=O)N1.c1(CC)cc(C(=O)NC2(C)CC2)n[nH]1.N c1(N2CCC(=CC(=O)NC3CC(F)(F)C3)CC2)ncnn2cccc12 N1(C(C2(C)CCCN(C(CCc3ccc(C)o3)=O)C2)=O)CC(O)(C2CCC2)C1 c1(C(=O)NC2C3CC(NC(C(C)(C)OCC)=O)CC32)nc(OC)ccc1C C1(NC(C(C)OCCCC)=O)CCOC12CCN(C(c1cccc(O)n1)=O)CC2 c1(C(N2CCC(O)C2)C(=O)NCCCOC)ncc(C(C)C)s1.c1ccccc1 C(C(C)(C)CC(=O)NC1(C)CCC(C)C1)NC(CN1CCC(C)CC1)=O C1(C#N)(C(=O)N)CCSCC1.c1(OC)ccc(CC(=O)NCCC2CCC2)cc1 CC1CC(CNC(C2(CO)COC2)=O)CCN1C(C1CCSC1)=O n1(CCNC(=O)Cc2nncs2)cc(C(=O)NC2(CO)CC2)nn1 C=CCC(C(=O)NC1CN(C(c2ccnn2CCC(F)(F)F)=O)CC1O)C(C)C c1(C(=O)NCC(C)NC(CC(C)C2CCCCC2)=O)cc2c(O)cccc2n1C C12(C(NOCC(=O)N(C)CC3CCN3C(C)(C)C)=O)CCN(CC1)CC2 C(C)(C(CC(=O)NC1COCCOC1)NC(=O)C(=O)NC1CC1)OC N1(C(C=C(C)C(C)C)=O)CCCC(O)C1.C1(C)(C=O)CCC(C(C)(C)C)CC1.N Cc1ncc(C(=O)NCCSCC(=O)NC2CC2(C)C)cn1 N1(C(c2n(C)cc(Cl)c2)=O)CC2CCS(=O)(=O)C2C1.C1(C=O)CCC1.C1CC1 N1(C(CC(=C)Br)=O)CCC(n2cc(-c3ncoc3C(=O)OC)nn2)CC1 CC(C)CC(C)CNC(C1CC2CCC1O2)=O.C(=O)C(C)(C)C.C(=O)CC.N c1(CC)cncc(C(=O)N(C(C(N2CCC2CC(C)C)=O)C2CC2)C)c1 c1(OCC(=O)N(CCCNC(CC(C)c2cccnc2)=O)C)ccccc1Br C=CC(C)(C)C(=O)NC(C1CN(C(c2cncnc2)=O)CCO1)C N1(C(c2cnc3n2CCC3)=O)CCCN(C(C2CCC(C3CC3)CC2)=O)CCC1 c1(OC)ccc2c(c1)CC(C)CC2NC(N1CCC2(CCCCO2)CC1)=O c1(C(N2C(C(N3CCC(C)(N(C)C)C3)=O)C3CC3C2)=O)ccc2nccn2c1 c1(C(N(C(C)C)CCNC(=O)C=O)=O)ccc(N)c(F)n1.CCC(N)=O.N c1(OC(COC)C)ccc(NC(c2cnc(OC)cn2)=O)cc1 Cc1ccc(C(N2CC(O)(C(F)C(N3CCCC(CCF)C3)=O)C2)=O)c(O)c1 c1(C(=O)NC2CCN(C(C3=CC(C)C3)=O)CC2O)cnc2[nH]ncc2c1 N1(C(c2cncc(N)c2)=O)CC(NC(c2ncnc(O)c2F)=O)CC(O)C1 C(C(CNC(=O)CC(C)C(F)F)C(F)(F)F)NC(c1c(CC)occ1C)=O C(c1cccc2ccccc12)=CC(N1CC(N(C(=O)CC2(C)CC2)C)C(F)C1)=O c1(OC)ccc(C(=O)N(C)CCOCCNC(c2ncc[nH]c2=O)=O)nc1Br CC1(C)CN(C(c2cnc[nH]c2=N)=O)CC(C)(C)C1NC(c1cccc(=O)o1)=O CCC(C)C(C)C(=O)NCCCOC1CCNCC1 c1(C(=O)NCC(c2ccc(Cl)cc2F)F)cc2nc(Cl)ccc2s1 C1(NC(=O)OC(C)(C)C)CCC(C(=O)Nc2cncs2)C1.N1CCOCC1.C C(=O)(C(C)C(F)(F)F)N.c1(-c2nc(C)on2)cccc(C(=O)NC(C)(C)C)c1 c1(CC)cc(C(=O)NCC(O)CC(=O)N2CC(O)(CC)C2)ccn1 c1(C=O)c(F)ccc2n[nH]cc12.C12(NC(CN(CC)CC)=O)COC(C1)CC2 CC1CCC(CC(=O)NC2CC(NC(c3nc(Br)c[nH]3)=O)C2)O1 c1(CC(=O)NC2CCC(C)N(C(=O)CCS(C)=O)C2)coc2cc(F)ccc12 C1(N(C)C(C2CC2c2cccs2)=O)CCCN(C(c2cc[nH]c2)=O)C1 n1(CC)cnc2[nH]c(=NCC(C)CC(=O)NC)nc(N(CC(C)C(C)C)C)c12 N1(C(C(CCOC)C)=O)CC2CCC2(CNC(c2ccc(COC)o2)=O)C1 C(C(C)(O)CNC(C1(O)CCCC1)=O)NC(CCNC(C)=O)=O c1(C(=O)NC(c2nc(C(N3CC=CC3CF)=O)co2)C)ccnnc1O C1(C(=O)NCCN(C(=O)CC2CC23CC3)C2CC2)CC2C=CC1O2 c1(OC)ccnc(O)c1C(=O)NCC(C)(O)C.c1ccc(O)cc1.C(=O)C.N c1(CC(=O)NC(C)CNC(c2nc(Cl)sc2Cl)=O)ccc(F)cc1Cl C(C1=NOC2CN(C(C3CSC3)=O)CC12)NC(c1cn(-c2cccnc2)nn1)=O n1(CCC)nc(C)cc1C(=O)NC(C)(C)CNC(C1(C)CCNC1=O)=O c1(C(N2CCN(C(C3CCN3S(C)(=O)=O)=O)CC2)=O)cc(O)c(F)cc1N.C CCC(C)CCCC(=O)NCCn1ccc(C(=O)NCC23CCC(CC2)CC3)c1 C(C(C)N=c1[nH]c(N2CC3C(=O)NC(=O)C3C2)nc(=NC)[nH]1)N(CCCC)C CCCCC(F)C(=O)N1CCCC1C(C)(C)C(N1CCC(F)(CF)CC1)=O C1(C(=O)NCC(C(C)C)NC(CN(C(C)=O)C)=O)CC2(C1)CC2F CC1COc2ccccc2C1C(=O)NCCCC1(NC(c2c[nH]ccc2=O)=O)CC1 O=C1NCC2(CO1)COC(CF)CN2C(=O)C(c1ccc(F)cc1)C1CC1 N1(C(c2nn(CC)c(C)c2)=O)CCC2(CCCN2C(=O)Cc2cc(C)ns2)C1 C1(C(=O)NCC2(OC)CN(C(c3ccncc3C3CC3)=O)C2)COCCOC1 C(=O)C(O)(C(F)(F)F)c1cn[nH]c1.c1(C(=O)NC2CCCC2)ccc(Cl)cn1.N C(=O)(C1=C(F)CN(C(C2CC2C(F)(F)F)=O)CC1)N(CC(C)(C)C#N)C c1(C(=O)NC(CC=C)CNC(=O)C(Cl)=CCl)cccc(=S)n1O C1(NC(c2c(C)nc(C(C)C)o2)=O)C(C)CN(C(C2(O)CC2)=O)CC1C c1(C(=O)NC(CC)CN(C)C(c2cnoc2C2CCC2)=O)cn(C)nc1C C1(C(N2CCN(C(CCSC)=O)CC(C)(F)C2)=O)Oc2ccccc2OC1C c1(CC(=O)NC2(C)CN(C(C3CC4(C3)CC4F)=O)C2)cccc(Br)c1Cl Cc1ccnc(C(=O)NOCC(=O)NCC(c2ccnn2C)O)c1F Cc1ccnnc1C(=O)N(CC(C)NC(C1CC1c1nncn1C)=O)C N1(C(c2cc(C)sc2)=O)CCC2CCN(C(=O)CNC(=O)CCCCO)CC12 c1(C(=O)NC2C(NC(c3nc(C)oc3C)=O)CCC2)cc2ccccc2cc1C C(=O)(C1=COCC1)N(CCNC(C(C)Nc1ccccn1)=O)C.c1ccccc1 N1(C(CCCNS(C)(=O)=O)=O)CC2CCC1C(Nc1ncc(O)cn1)C2 c1(C(=O)NC(C)CNC(c2sc(F)cc2Cl)=O)cc2c(cc1Cl)NCC2 C1(C(=O)NCC2CC(=C)C2)CN(C(c2cccc(C)n2)=O)CC1F CCCCCCC(C)C(=O)NC1COCCC1C(N1CCC(O)CC1)=O S(=O)(=O)(c1cc(C)cnc1NC1CCCOC1)N(CCC)C(C1CCC1)C N1(C(CSCC(=O)OC)=O)CCCC1C.C(c1ccccc1)=CC(C=O)C.C O=C(CCCC1(NC(=O)COCC2CCCO2)CCC1)N.C1(CCF)CC1 N1(C(=O)OC(C)(C)C)CC2CCC1C1CN(Cc3cncc(C(=O)O)c3)CC21 C12(NC(C3N(CC)CCC3)=O)COC(C1)C2.c1(CC=O)cccc(Cl)c1.C C1(F)(C(N2CC(O)(CCNC(c3n(C)nnc3)=O)C2)=O)CCC(F)(F)CC1 CC(CC(F)(F)F)c1nc(-c2cscn2)no1 C(=O)(C1Cc2ccc(F)cc21)N1CC(N(C(=O)CCCC2CCC2)C)C(O)CC1 Cc1c(Br)cnn1CC(=O)NCCC(C)NC(=O)C=C1CCOCC1 N1(C(=O)Cc2ncccn2)CCN(C(=O)Cc2ncc(Cl)s2)C2CCCCC2C1 c1(C(C(=O)NC(CSC)C)O)cc(F)cc(F)c1 C1(NC(CCC(CC)OC)=O)Cc2ccccc2C1NC(C1CCN(C)C1=O)=O CN=c1[nH]c(=NCc2ccccc2OCCCO)[nH]c(=NCCC(C)CCO)[nH]1 N1(C(C2(C#N)C(C)C2)=O)CC2CCC(C1)N2C(c1cc(O)nc(C2CC2)n1)=O c1(C2(C)C(C(N(C)CCNC(c3cc(C(N)=O)n[nH]3)=O)=O)C2)ccccc1F C(C(C)(O)C(C)CC)NC(C1N(C(c2c(CC)nccc2)=O)CCSC1)=O C#CCCCCCCC(=O)NC(CC(=O)NC1(C)CC2(CC2)C1)C(F)F Cc1cc(Br)cc(Cl)c1C(N1CCCN(C(c2ccnc(Cl)n2)=O)CC1C)=O Cc1cnc(CCC(=O)NCCCCN(CCCNC(c2cc(Cl)ns2)=O)C)[nH]1 N1(C(C(CCC)OC)=O)CCC(NC(=O)Cc2nc[nH]n2)CC1c1ccccc1 C(CCC(C)(C)C(=O)NCc1nc(C#N)cs1)NC(c1c(F)ccc(C)n1)=O C1(=CC(=O)NCC(CNC(C(CSC)C)=O)O)CCCCC1(C)C N1(C(COCCSC)=O)CCC(N=[N+]=[N-])(C(=O)NC)C1.c1cnc2n1CCC2 NS(=O)(=O)c1coc(C(N2CCCCC2CCNC(C2CC(F)C2)=O)=O)c1 N1(CC)CCN(c2ccc(F)c(NC3CC(F)(F)C(=O)N3)c2)CC1(C)C N1(C(COCC(=C)C)=O)CCCN(C(c2cncc(N)n2)=O)CC1 c1(C(=O)NC2CC(C(=O)Nc3nnc(C4CC4)o3)C2)c(Cl)ccc(Cl)c1F c1cccc(C=O)c1[N+](=O)[O-].C1(C(F)(F)F)(C(N(CC)C2CC2)=O)CC1 C1(N(C(=O)COCC(F)F)C)CCN(C)C1.c1ncc(CCc2ccccc2)o1 c1(C(N2CCC(C(C)NC(C(CC=C)C)=O)C2)=O)ccc2c(c1)OCCCO2 N1(C(C(C)N(C(=O)C(C)n2ccnc2)CC)=O)CCC(CC2CC2)CC1 C1(C(N2CC(CC(C#C)C)C2)=O)CCCC(NC(c2ccn(C)c2)=O)CC1 N1(C(C(C)NC(CC)=O)=O)CCC2CCN(C(c3cnc(S)[nH]3)=O)CC12 C=CC1CC(N=c2[nH]c3ccc(S(=O)(=O)N4CCS(=O)C(C)(C)CC4)cc3s2)C1 N1(CC)CC(C(=O)N(C2CCCCC2N(C)C(C2CC2(F)F)=O)C)CC1=O.CO Cc1cccc(C)c1.C(=O)CC.C1CCOC1.C(C(=O)N)NC1(C=O)CC1.C C(=O)(CC1OC(=O)c2ccccc21)NC1CCN(C(C=C(CC)C)=O)CC1 Cc1cc2[nH]c(C(N3CC4(CNC(c5cc(C)c(C)o5)=O)CC3CO4)=O)cc2o1 c1(-c2n(C(C=C)C)nc(-c3ccc(C(F)F)cc3)n2)cc(F)cc2cccnc12 N1(C(C2C3CNC(=O)C32)=O)CC2CC1CN2C(=O)C1=CCCOC1 c1(NC2CCN(OCC)CC2)nc2c(c(=NC3CCC(NC)C3)[nH]1)CCCCCC2 N1(C(c2c(C)ccnn2)=O)CC(NC(=O)Cc2cnc(C(F)(F)F)s2)CC(F)C1 CC1CCC(c2cccs2)N(C(=O)OC(C)(C)C)C1.N1(C=O)CCC(OC)CC1 n1(C(C)C)cc(C(=O)NC2CC2CNC(c2ccncc2F)=O)c(Br)n1 C1(F)(CNC(c2cn(C)c(=O)cc2)=O)COCCN(C(C2(O)CCSC2)=O)C1 C(=O)(CCCCC(=O)N1CCN(C(c2cncs2)=O)C(C2CCCC2)C1)OC C(=O)(CCCCCN(C(C(COCC)C)=O)C)N.C(C)(C)C.C(=O)O C(=O)C1CCC(=O)c2cccn21.C(=O)(CSCC=O)OCC.CC.CC.N C1(C=O)(OC)CCC(C)(C)CC1.C1(C2CC2)(CC=O)CC1.CC=CC.N c1(C(N2C(C)CC(NC(c3c(C)cn(C)c3)=O)C2)=O)coc2c(F)cc(Cl)cc12 CC(C)(CCS(C)(=O)=O)C(=O)N1CCCOC(CNC(=O)CNC=O)C1 C1(CCNC(CC)=O)CCN(C(=O)C(C)Sc2nncn2C2CC2)CC1 N1(C(C(C=C=C)C)=O)CCC(C)C(N(C)C(c2cc(-c3ccncc3)no2)=O)C1 CC1CC(NC(C2(C)CC(F)C2)=O)CCN1C(C1CCCC(F)(F)C1)=O c1(C(N2C(CNC(C3CC3Br)=O)CCC2)=O)ccc2c(=O)cc[nH]c2c1 C(=O)(N1OC2CCC1CC2)C1(COC)N(C(CCC2(CCC#C)N=N2)=O)CCC1 N1(C(CCC(C)N(C)C)=O)CCN(C)CC1CNC(C1(F)CCN(C)CC1)=O C1(C2CCN(C(=O)C3=CS(=O)CCC3)C2)(NC(CC(C)(O)C2CC2)=O)CC1 c1(C(=O)NCC(CC(C)C)NC(=O)C(C2CCCCC2)O)cn2c(n1)SCC2 Cc1sc(C(N2CCN(C(c3cnc[nH]3)=O)CC2C(C)C)=O)cc1[N+](=O)[O-] c1(C(=O)NCCCN(C(C)C)C(c2occc2Cl)=O)nnn2ccccc12 C1(SC)CC(C(=O)NCCC(C)N(C(=O)CO)C)C1 CC1(CNC(c2cc(CO)[nH]n2)=O)CCN(C(=O)CC2CCCCC2O)C1 CCC(F)(F)CC(=O)NCc1nc(C(=O)NC(COC)CCOC)c(C)o1 N1(C(C=CCC)=O)CC(C(=O)N(CCCCC)C)C(C)(C)C1 c1(C(N2CCC(N(C(=O)C(O)C(F)F)CC)CC2)=O)ccc(C#N)n1C c1(OCC)cc(C(=O)N)cc(Cl)c1O.C(=O)(C(F)CC1CCCC1)N1CCC1 c1(C(N2CC(COC)(CNC(=O)CC(C)(C)C)C2)=O)ccc2cccnn12 c1(CC=O)ccc2c(c1)NC(=O)C2.C1CCN(C(C23CC2C3)=O)CC1.O=CC C(=O)(N=c1[nH][nH]c2ncccc12)C1(CNC(c2ccc(OC)cc2)=O)CC1 c1(OC)noc(C(=O)NCC(O)CNC(=O)CCn2cncn2)c1Br c1(C(N2CCC(N(CC)CC)C2)=O)ccc(C2CC2)o1.c1(C=O)cccnc1 c1(NCC(CC(C)C)(C)NC(c2cc(O)nc(O)c2)=O)cnc(C#N)c(C#N)n1 Nc1cc(C(N2CC(NC(=O)CC34CCCC3C4)C(O)C2)=O)cc(F)c1Br C(=O)(CCCC(F)(F)F)NC1CC(C)(C(N2CCC2CF)=O)C1 N1(C(C2C(OCC)C2)=O)CCCN(C(C2CC(F)C(=O)N2)=O)C(C)C1 Cc1ncoc1CN(C(C1CCCSC1)C(=O)NC1CCOC1)C N1(C(COCC#C)=O)CCN(C(=O)CC(F)F)C(CCSc2ccccc2)C1 c1(C(C(=O)NC2CCN(C(c3nc(C)on3)C)C2)C)cn(C)nc1C C1(Br)(NC(=O)NCCCN(CC(C)C)C)CCC1 CC(CC(=O)NCCC12CC3CC(CC(C3)C1)C2)CC(=O)O N1(C(CC(C)C)=O)CCN(C(=O)Cc2cccc(S(C)(=O)=O)c2)C2CCCCC12 C=CC(O)C(=O)NCCC1CC(C(=O)NCC2(C)CCCC2)C1 Cc1cc(=NCC2(F)CCCC2)[nH]c(=NCc2c[nH]nc2C)[nH]1 N1(C(CCC=CC)=O)CCCC(CCNC(c2ccc(C3CC3)cc2F)=O)CC1 C1(CNC(C(CC)COC)=O)CCN(C(=O)CCc2cccc(OC)n2)C1(C)C N1(C(C(C)CN(C)C)=O)CCOC2CCN(C(C3CC(O)C3)=O)CC12 C(=O)(CS(=O)(=O)CC)NCCCOCCNC(c1cccc(CC)n1)=O CCC(CC)C(C(=O)NCc1ccc(C(=O)NOCC2(C)CCC2)o1)OC Cc1coc(C)c1C=CC(N1CCC(F)(CNC(=O)C(C)n2ccnn2)C1)=O C12(C=O)CCCC(C)(C1)OC2.n1(CC)cc(NC(=O)C=O)cn1.C1CCCC1 C12(CNC(C3(COC)CC3)=O)CCCCC1N(C(c1c[nH]nc1C)=O)CC2 c1(C=O)ccc2c(c1)CCCC2.C1(CNC(CN2CC(CC)C2)=O)CCOC1.N C1(NC(CC2N(CC)CCC2)=O)CC2C(NC(c3coc(C)n3)=O)C2C1.O c1(CC(N2C3C(NC(CN4CC(C)(C)C4)=O)CC(C3)C2)=O)ccc2ncsc2c1 N1(C(C(C=C)(C)CCOC)=O)C2CCCC1CN(C(c1cc(C)sn1)=O)C2 S(=O)(=O)(c1cnc2ccc(Cl)cc2c1)NC(c1cccc2c1COCC2)=O N1(C(c2c(C)cc(F)c(Br)c2)=O)CCC2C(CCN2C(=O)NCCCl)C1 C1(CC)CCN(Cc2[nH]cnc2C)C1c1cccnc1.C1CN1C(C)=O C(=O)(CS(=O)(=O)C(C)C)N(CCC(C)C)C.c1(CC)cc(C=O)n(C)n1.N CC1CC(NC(c2cnn(C3CCC(=O)NC3=O)c2)=O)CCN1C C(CCCC(C)(C)C(=O)NNC(=O)c1c[nH]c(=N)s1)NC(C1C(C)CN(C)C1)=O c1(C(=O)NCC2N(C(c3n(C(CC)C)ncc3)=O)CCC2)[nH]nc([N+](=O)[O-])c1Cl C(CC(CC)C(=O)NCC1COCCN(C(=O)CCS(=O)(=O)NC)C1)=CC c1(C(=O)NCC(CC)NC(c2cnoc2C)=O)cccc2nc(C)sc12 c1(CNC(C2(C)CC2Br)=O)cn(CC2CC3CC3C2)nn1 C1(NC(COCCCC)=O)CN(C(c2ccc(OC)nc2Cl)=O)C2(CCOC2)C1 c1(C(=O)NC2CC(CC)(CC)N(C(C3CC3C)=O)C2)cnc2occc2c1 C(=O)(CCP(C)(C)=O)N1CCC(C)(CC(=O)Nc2cc(C)sc2)C1 N1(C(C=Cc2n(CC)ccn2)=O)C2CCC1(CNC(C1CCCCC1C)=O)CC2 C#CC1CCCC1NC(=O)CCN(CCCO)C(=O)C=CCN1CCCC1 c1(-c2ccc(C(N3CCC(CC)(CC)C3)=O)s2)ccc(OC)c(OC(C)C)c1 Cn1cc(Br)nc1NC(C1CCCCN1C(=O)Cc1cncnc1)=O N1(C(c2n(CCOC)ncc2)=O)CCC(C)(C)C1.C1(C=O)(C(N)=O)CCC1 CC1CN(C(c2cccc(N3CCNC3=O)c2)=O)CCN1C(c1cscc1F)=O c1(C(=O)NC2C(C(=O)NCc3c(C)ccs3)OCC2)ccc2[nH]ccc2n1 c1(C(=O)NCC(CNC(C2(C)CCC2)=O)(C)O)ccc2[nH]ccc2n1 c1(OCC)ccnc(N2CCCC(CC)C2)n1.c1(C(=O)N)cc(C2(C)CC2)on1 C1(CC(N2CC(CCC)C2)=O)COC(C)(C)C1.C(C=O)(C1CCCC1)OC.N C(=O)(CCCS(C)(=O)=O)NCC(CC)(CC)NC(=O)C=CBr C1(O)(CN(C(C(COC)(C)C)=O)C)CCCN(C(=O)C(C)=C2CCCC2)C1 Cc1conc1CC(=O)NCC(O)C(=O)NC(C)(C)C(F)F C(CCCc1ccccc1)NC(C(F)=CC)=O.C1(C=O)CCN(CC(C)C)C1.N CC1Oc2ccccc2OC1C(=O)NC1(C)CC(NC(=O)C2=C(Cl)CCCC2)C1 N1(C(C)C2CC2)CC(C(N2CC(NC(C3SCCCS3)=O)C2)=O)CC1=O CC(C)C(C(C)NC(C1CCSCC1)=O)NC(C1C2CC3C(C2)C13)=O n1(CC)nc(C(=O)N(CC(C)CNC(C2CC(SC)C2)=O)C)ccc1=O Cc1cc(F)sc1C(=O)NC1CC(CNC(c2cccc(F)c2)=O)C1 C(C)(CO)(C(=O)NCC1CCCS1)NC(c1cc(C)on1)=O N1(c2snc(SC)n2)CC2CCC(NC(=O)C3=CCCOCC3)CC2C1 CC(C)(C(=O)NCC(O)CCNC(C12C(=O)C3CC1C2C3)=O)C(F)F N1(C(C(C=C=C)C)=O)CCc2sc(CNC(c3cn(CC(N)=O)nn3)=O)nc2C1 C1(CNC(C(CC)SC)=O)CC(F)CN1C(=O)Cc1ccc(C(F)F)cc1 N1(C(c2c(CC)nn(C)c2)=O)CC2CCC1C2.C1(CC=O)CC(=O)NC(=O)C1 N1(C(C=CC=CC)=O)CCC2(CC2NC(=O)Cc2cncnc2O)C1 C(=O)(C1=CCN(C(c2cnn[nH]2)=O)CC1)N(C1CCC1(C)C)C N1(C(Cc2ccc(OC)c(O)c2)=O)CC2CCC(C1)N2C(C1CCNC(=O)C1)=O c1cc(NCC2CCCC(CO)C2)cc(NC2CC2)c1 c1(N(CCC)C(C2CC2C(=O)N)=O)cc(C)nn1C.n1(C2CC2)cncn1 C12(C(=O)NC(C)CN=[N+]=[N-])COC(C1)C(NC(=O)C(C)(C)C1CCCC1)C2 C(=O)(CC(C(F)F)NC(=O)C#CC1CCC1)N(C)Cc1c(C)cnn1C C1(C)(C(=O)NC2C(C)CN(C(=O)CC(C)n3ccnc3)C2)Cc2ccccc2C1 C=CCCCC(C(=O)NC1(C)CCC(C)(C)C1)NC(=O)CCc1nc[nH]n1 c1(C(=O)OC)nc(Cc2nnnn2C2CCC2)nn1C.C(CC1CC1)C1CC1 c1(NC(C2CC(C)OCC2)=O)ncnc2c1ccn2C N1(C(C(=C(C)C2CC2)F)=O)CCC(CO)(NC(c2cc[n+]([O-])cc2)=O)C1 C=CCCC(F)(F)C(=O)NCC1CCCN1C(C1(COC)CC=CCC1)=O C1(C(=O)NC2CCC(C(C)O)CC2)CC2(CC(NC(=O)C3CC3)C2)C1 c1(CCC=C)ccc(C(=O)NCCC2(NC(c3ccccc3)=O)CC2)cc1 c1(C(N2CC(C)(NC(C=Cc3c(C)coc3C)=O)C2)=O)cc2c(=O)[nH]ccn2n1 C=CCC(C(=O)NC12CC(C1)C2)C(C)C.c1(C=O)cn(C)nc1C(F)(F)F CC1CC(NC(=O)COCc2nc[nH]n2)CN(C(c2cc(O)ccc2F)=O)C1 C(C(C)C(=O)N(C(C)C(=O)NCCF)C)NC(CCSC)=O C(C)(C(C)C(=O)N(CCCO)C1CC1)NC(C1C(C(C)=O)C1(C)C)=O c1(C(=O)NCCC2(C(N3CCC(O)C(CO)C3)=O)CC2)coc2ccccc12 C1(CNC(C(C)N(CC(F)(F)F)C)=O)CCCCN1C(C1CCCOC1C)=O C1(C(=O)NCC(C(C)(C)C)NC(C(C(CC)O)C)=O)CN=C2N=CNN2C1 c1(C(C)C)cc(C(=O)NCCC2CCC(C)(C)O2)cc(O)n1 N1(CC(C)C)CC(C(=O)NC(C)C(C)(C)C)CC1=O.C1(C=O)CCCC12CC2 C1(CC(=O)NC(C)C)(C=O)CCCC1.c1(C=O)cnco1.CC.C(=O)CO c1(C(N2C(C3(NC(c4cnc(O)o4)=O)CC3)CCC2)=O)ccnc(C2CC2)n1 c1(C(N2C(CCC(=O)NC(CCC)C(F)(F)F)CCC2)=O)ccc2[nH]ccc2n1 C1(NC(=O)C#CC2CC2)CC12CCN(C(=O)C1=CCCSC1)CC2 Nc1cnc(Br)c(C(=O)NC2CC(CCNC(C3CCC(=O)N3)=O)C2)c1 C=C(C)CCC(=O)NCC1CCCCC1NC(=O)C(C)NC(=O)COC CC(CCCCNC(c1ccc(N)cc1)=O)NC(=O)CC1CCOC1 N1(C(CC)=O)CSCC1C(=O)N(CCCNC(=O)CSC(C)C)C CC(C)CC(F)C(=O)N(C1CCN(C(c2cnc(F)c(Cl)c2)=O)C1)C CC1CC(C(=O)NC2CC2NC(C2(C)CCCCC2)=O)CC(C)(C)C1 N1(C(C(C(C)C)OC)=O)CCC2CCC(C1)N2C(=O)COc1cncc(Cl)n1 C1(CC)CC(C(=O)NC2CON(CC)C2=O)CCN1C(=O)C(C)NC=O c1(C(=O)NCC(C2CC2)OC)cccc(-c2ccoc2)c1 C1(C(N2CCC(C(=O)NC(C(CC)(C)C)C)(CF)C2)=O)CC2CC(=O)C1O2 C(=O)(C1=C(C)N(C2CC2)C(=O)NC1c1cc(Br)cc(I)c1)OCC CCCCC(CC)C(=O)N1CC2C(NC(c3cc(Cl)c(N)cc3OC)=O)C2C1 c1(CC=O)c(C)nn(C)c1C.N1(CC(=O)NCC)CCCC(C=O)C1.CC Cc1cc(C(=O)NC(C)Cc2ccccc2)cc(O)c1.C1(CC(=O)N)CCCC1 C1(NC(c2cc(OC)no2)=O)CN(C(=O)C=Cc2cccn2C)CC1SC n1(CC)cc(NC(C2C3CC2N(C(c2n[nH]c4c2COC4)=O)C3)=O)c(C#N)n1 c1(C(C)NC(C(=O)Nc2cc(-c3ccc(C)cc3)no2)=O)c(CO)cnc(C)c1O C1(C(C)C)CN(C(=O)C2CC2)CCC1NC(c1cc(C2(C)CC2)on1)=O C12(NC(CC#N)=O)CCN(C(=O)CC3(O)CCCC3)CC1C2 N(C(=NCCCC1(O)CCC1)NCC1CCCO1)Cc1c(C)cccc1C c1(CC)nc(Cl)c(C)c(=NC2CN(C(=O)CN=c3ccc(Cl)n[nH]3)CC2C)[nH]1 CC1CS(=O)CCN1C(=O)CCC1CCCN1.c1(C2C(=O)N2)ccnn1C N1(C(C(C2CCC2)OC)=O)CC2CN(C(=O)C3=C(C)OCCS3)CC2(C)C1 N1(C(c2c(OC)n(C)nc2)=O)CCCC(CC(=O)NC2CCCOC2)CC1 c12ccnc(n1)NC(=O)C2.N1(CC(=O)N(C)CC)CCCC(CSC)C1 c1(C(=O)OC)ccc(C=O)c(F)c1.C1(C=O)CCC(C(F)F)O1.C(C)(C)C CC1CCCCC1C.N1(CCC=O)CCCS1(=O)=O.C(=O)C.[SH](C)(=O)=O.N Cc1oc(Br)cc1C(N1CC(NC(=O)CCn2ccnc2)C2CC12)=O C1(O)(CNC(c2noc(C)n2)CC)C2C3CC4C5C3CC2C5C14.C(C)=O c1(C(=O)NCC2N(C(C3C(C(C)O)C3)=O)CCCC2)cccc(N)c1O C(=O)(CC(CC)C(C)C)N(C)CC1OCCN(C(CC2(C=C)CCCCC2)=O)C1 CCC(CC)C(=O)N1CCC(CF)(NC(C2CCSC2)=O)C1 N1(C(C(N2CCC(N(C(CC(C)N)C)C)C2)=O)=O)CC2CNC(=O)C2C1.C(C)(C)C CC(CNC(C1(C)CCCCCC1)=O)C(F)C(=O)NCC1CC1 c1(N2CCC(C(CC)C)CC2)ccc(S(=O)(=O)N(C)CCOC)c(Br)c1.C1CC1 N1(C(C2(C)CC2)=O)C(C(=O)N(C2CCOC2)C2CC2)CCC12CC2 N1(C(Cc2scc(CC)n2)=O)CCN(C(c2c[nH]nc2F)=O)CC1C c1(OCC(C)C)ccc(NC(=O)C(=O)NC(c2ccc(F)cc2)CF)cc1Cl c1(NC)cccc(OC)c1C(N1CC2CC2(C(=O)N(C)C2CC2)C1)=O c1(CC)cc(C(N2C3CCC2C(NC(=O)C(C)(C)F)C3)=O)ccc1Br C1(NC(C(C)OCCC(C)C)=O)CCOCC1C(N1CC(CC(C)(C)C)C1)=O Cc1cc(CCCNC(=O)C(C2CCCC2)NC(c2ccc[nH]2)=O)on1 c1(C=O)cnc(C(F)(F)F)cn1.Cc1cc(OCC(=O)NC)no1.C1COC1 c1(C(=O)NC2C3CN(C(CS(CC)(=O)=O)=O)C2CC3)cnn2c1OCC(F)C2 C1(OC)CCC(C)(C(=O)NCCC2CN(C(=O)C(C)C)CCCO2)CC1 C1(C)(C(=O)NC(c2cnc(C)s2)C)CCN(C(=O)C=Cc2ccncc2)C1 Cc1cc(CNC(C2CC3(CCC3)C2)=O)oc1C(=O)NC1CCOC1=O c1(N(CCCC(C)O)C)[nH]c(=NCc2cccs2)nc2c1cnn2C c1(C2C(C=O)C2)cccc(C#N)c1.C1(C(N(CC(C)C)C)=O)(C)CCCO1.N CC(CCCNC(c1ccnn1C(F)F)=O)NC(=O)CC(C)C1CC1 C(C(CNC(C1(OC)CCC1)=O)C(F)(F)F)NC(c1c(CC)ncs1)=O C1(CNC(CCC(CC)C)=O)CC2CCCC2N1C(c1coc2c1COC2)=O c1(N2CCC(CNC(=O)C(F)C3CCC3)C2)c(Cl)cc([N+](=O)[O-])cc1Cl c1(C(=O)NC2(COC)CCCN(C(C3COC3)=O)C2)cc(Cl)cc2ccccc12 N1(C(=O)NC(c2cnn(C)c2)CN(C)C)CCCC(C)(Cc2cnnn2C)C1 CC1CN(C(C2(O)CC2)=O)CC(C)N(C(=O)CCn2cc(C#N)c(O)nc2=O)C1 C1(O)(CN(C)C(C2CC3(CC3)C2)=O)CCN(C(C2CCC(F)(F)C2)=O)C1 N1(C(c2c(COC)n(C)nc2)=O)CC2(C1)SCCC2NC(=O)CN(C)C c1(C(N2CC3C(NC(=O)CC4OCCCO4)(C3)C2)=O)ccnc2[nH]nnc12 C1(NC(c2nc(CCC)oc2)=O)CCN(C(=O)CC2(C)CCCC2)C12CCCC2 c1(C(C)C(=O)NCC2(NC(=O)CSS(C)(=O)=O)CC2)nc(F)ccc1Cl c1(C(N2CCC(C(C)O)CC2)C(=O)NCC)ccc([N+](=O)[O-])s1 C(C(CC)=Cc1ccccc1)(C(=O)NC(C)C)N(CCC#C)CC CC1CC2CN(C(c3cncc(N)n3)=O)CC2N1C(c1cccc(Cl)c1F)=O C1(NCc2cccc(-c3c(OC)n(C)nc3)c2)CCNC2(CCCCC2)C1 Cc1sncc1C(=O)NCC1CCN(C(=O)CCNC(C2CCCO2)=O)C1 C(=O)(CCC(C)(C)C)N(CC1C(C)CN(C(=O)CO)C1)Cc1ccncc1 C(C(CC(C)C)C(=O)NCc1nncn1C)NC(CCC(C)OC)=O n1(C(CC)C)nc(-c2cccnc2)nc1-c1ccc(OC(C)C)cc1 Cc1ccc(CC(=O)NC2(C(=O)N(C)Cc3cn(C)nn3)CCSC2)s1 C1(C(C)(C)C)CCN(C(C2(NC(=O)C(O)C3CCCC3)CC2)=O)C1 c1(C(=O)NC2CC(NC(C3CC4C=CC3C4)=O)C2)cnn2c(=O)cc[nH]c12 CCC(CC)(C(N)=O)NC(C1C2CC1N(C(=O)Cc1cc(C)[nH]n1)C2)=O N1(C(CCCCC)=O)CCOC2(CCC2)CC1.C(C(=O)N)COCCOCC#C c1(CNC(C2CCN(C)C2)=O)ccc(C)cc1F.c1(C=O)ccc(N)c(F)n1.N CC1=C(C(=O)NCC(C2CCN(C(c3csnc3C)=O)CC2)F)CCCC1 n1(CC)cnc2[nH]c(=NCCNC(=O)C(C)C)[nH]c(=NC(C)C)c12 Cn1nc(C(=O)NCC2CCCN2C(=O)CCc2cccc(O)c2)cc1F O(NC(=O)C1=CC2(CCN(C(c3ccc4[nH]ccc4c3)=O)C2)C1)CCC#C C1(CCCOC(=O)NC2CC2)CC2CCC1C2 c1(C(CC)OC(C(=O)N)OCC)ccccc1.C1(C=O)CN(C(N)=O)C1 C(=O)(C(C)CCCC(C)C)N1CC(CC(=O)NCC2CCN(CCC)C2)OCC1 C1(C(=O)NC2(CCNC(c3c(C)nc(C)s3)=O)CC2)CCN2CCOCC12 C12(C(=O)NCC(CC)(C)NC(=O)COCP(C)(C)=O)CC1COC21CCC1 C(=O)(CCCCCCCCCO)NC(C)CN(C)C(c1[nH]cnc1C#N)=O c1(OC)cc(Br)ccc1C(N1CCCC(NC(c2cnc(Cl)s2)=O)C1)=O N1(C(C(CC=C)NC(C2CCC(C)(C)C2)=O)=O)CCN(C)C2(CCC2)C1 c1(C(N2C3(CNC(c4csnn4)=O)CCC(C2)C3)=O)cn2c(n1)COCC2 C1(CC(=O)NCC(C)OCC=C)C2CCCC2N1C(C1CCCO1)=O Cc1cc(C)c(C(=O)NC2CCCC2NC(=O)Cc2cncc(O)c2)c(C)c1 c1(N2CC(OC)C(F)C2)ccc(S(=O)(=O)N(C)CC2(C)CCCO2)cc1Br C(=O)(C#CC1(C)COC1)NCC(CNC(C(C)SCC1CCCO1)=O)(C)C c1(C(N2CCC(C)C2)=O)cccc2c1NCC(C)C2.C=C(C)COCC(=O)N.C Cc1cccc(F)c1NC(=O)CC1CCN(C(=O)CC2C=CCCC2)C1 c1(-c2n(-c3ccc(C)c(Cl)c3)nc(CC3CC4CCC3C4)n2)nc2cccnc2s1 N1(C(c2n(CCC)ccc2)=O)CC(CNC(=O)C(c2ccccn2)C)C(C)C1 C1(NC(c2ccc(C#C)cc2)=O)CCC2(CC1)CC(NC(C1CCCC1O)=O)C2 c1(C(=O)NC2C3(c4n(C)ncc4)CCC2C3)c(F)ccc(Br)c1N c1(C(N2CCC(NC(C3CS(=O)(=O)CC(=O)N3)=O)C2)=O)coc2ccc(O)cc12 Cc1cc(Br)cc(C)c1CNC(=O)C(n1cc(-c2ccnc(C(F)F)c2)nn1)C C(=O)(CCCCCCSC)NC1CCN(C(c2nc(CC)oc2C)=O)C1 c1(CN2C(C(N3CCC(F)C3)=O)CC(C)C2)ccc(Cl)cc1C(=O)O C(=O)(C1=CCN(C(=O)CONC(c2cncc(F)c2C)=O)CC1)OC C1(C(=O)NC(c2c(C)nns2)C)CCC(C)(C)N(C(C2CCC3(CC3)C2)=O)C1 c1(C(N2CCC(C)(N(C)C)C2)C(=O)NCCCC)cccc(OC)n1 C1C(C)(C)CC1(C)C.C(=O)(C(CC)C(=O)N)OCC.C(=O)C=O.C1CC1 n1(CC)cccc(NC(=O)C(C)(C)CN(C)C(c2ncccn2)=O)c1=O N1(C(=O)NC(C2CCCN(C3CCC3)C2)C)CCOC2(CCS(=O)(=O)C2)C1 CS(=O)c1ccccc1CC(=O)N.c1(C(N2CCC2)=O)ccn(C(C)(C)C)n1.C C1(C(N2CC(N(CC)CC)C2)=O)CCCN1C(=O)Cc1ccoc1 N1(C(c2c(OC)oc(C)n2)=O)CCCN(C(c2cccc(C3CC3)c2)=O)C(C)C1 c1(-c2n(CC(C)NC(C3(c4ccccc4)CC3)=O)ccn2)ccc(Cl)cc1 c1(OC)cc(N(C)C)ccc1C(N1CCC1)=O.c1(C=O)sccc1C1CC1.C Cn1cc(Br)c2c(C(=O)NC3CC3C)ncnc12.C1(O)(CC(=O)N)CCC1 C(=O)(C(C)(C)CNC(c1nn(C)cc1Cl)=O)N1CCC(CC(C)C)C1 C1(C(N2CCC(N(C)C(c3cc(F)ccc3Cl)=O)C2)=O)CCc2c(nnn2C)C1 N1(C(Cc2cc(C)on2)=O)CC(NC(c2cc(C(C)C)n(C)n2)=O)C(CO)C1 C(C)(CC(F)(F)F)NC(CC(C)C1CC1)=O.c1(C=O)nnc(C(C)(C)C)s1.N C1(F)CCCC1.c1(C=O)cc(O)ncn1.C(=O)(C(F)(F)F)NCC(=O)N.C c1(C(N2CC(C3(NC(C4C(C)(C)COCC4)=O)CC3)C2)=O)ccn2ccnc2c1 C(=O)(CC(F)(F)C(F)F)N1CC(C)(NC(Cc2cc(CC)nn2C)=O)C1 N1(S(CC#N)(=O)=O)CCC2(CC1)CC2C(=O)NCc1cccnc1 N1(C(c2c(C)cc(O)cc2)=O)CCC2CCC(C1)N2C(=O)C(c1ccncc1)C C1(CCC#C)CCN(C(=O)CC2CCCCN2C(C2CC(=O)N(CC)C2)=O)CC1 N1(C(C2(CC#C)CC2)=O)CCN(C)C(C(=O)NC2CCN(C(C)=O)C2)C1 C(=O)(C1=Cc2ccccc2OC=C1)N1CC(CCNC(=O)C2=CCCS2)OCC1 c1(OC)cc(I)ccc1C(N1CCCC1(C)C(=O)NCC1(C)CCOCC1)=O N1(C(c2ccn(CCNC(CCOCC(C)C)=O)c2)=O)Cc2cccc(F)c2C1 C(=O)(CCS(=O)(=O)Cc1ccccn1)N(C)CC1N(C(CC(C)OC)=O)CCC1 C1(CN(C(=O)CCc2cnc(O)[nH]2)CC)CCCN1C(c1[nH]cnc1C)=O C1(NC(c2ccc(C)cn2)=O)CC2CCC(C1)N2C(c1n[nH]cc1Cl)=O c1(C(N2CC3CC(NC(C45CCCC4C5)=O)C2C3)=O)ccc([N+](=O)[O-])o1 Cc1nc2ccccn2c1C(=O)NCC(C)NC(c1cc(=O)n2nccc2[nH]1)=O Cc1cc(=O)ccn1CC(=O)NCCN(C1CCCCC1)C(C1CC1(C)C)=O C1(C(N2C(C)(C(C)C)CC2)=O)CC2CC1CN(C(C1CCC(C)(C)C1)=O)C2 C1(NC(c2cnoc2C2CC2)=O)CN(C(=O)CC2CCSCC2)CCC1CO N1(C(C2(CC)CCNC2=O)=O)CC2CCC(C1)C2NC(c1cnsc1)=O Cc1cc(CCC(=O)NC2CC2CNC(=O)CSCC2CCCO2)n[nH]1 CC(C)CC(C)(C)C(=O)N1CCCC(C(=O)NCC(C)Cn2cccn2)CC1 c1(C(N2CCC(OCCNC(C3CCCS3)=O)C2)=O)cc2nn[nH]c2cc1F Cc1cc(C(N2CCC3CC23C(=O)NC(C2(O)CCC2)C)=O)nc(O)c1 N1(C(c2c(C)nc(C)s2)C(=O)NCC2CCOC2)CCN(C)CC(C)C1 C(C(C)(C)CSC)NC(CCN(C(=O)CCc1cc(C)cs1)CC#C)=O N1(C(c2c(CC)nns2)=O)CCC2CCCC12CNC(c1cc(N)ccc1F)=O C1(C(=O)NCC(=O)NC2CC2)CCCN1C(=O)CNC1CCSC1 N1(C(c2c(OCC)nccc2)=O)CCC(O)(CCNC(C2SCCC2C)=O)CC1 c1(CC)nn(C)cc1C(N1CC(NC(c2cc(C#N)no2)=O)CC1C)=O c1(C(CC(=O)NCCC2CCN(C(c3c(CC)c[nH]n3)=O)C2)C)ccccc1F N1(C(C(CC)O)=O)CC(F)(F)CC1CNC(=O)C(C)(C)c1ccccc1 c1(CN(C)C(C2C3CC3CN2C(=O)CC)=O)cccc(O)n1.CC(C)(C)C.O C(C1CN(C(c2ccc(C)o2)=O)CC1C(=O)Nc1cncc(C#N)c1)=CC N1(C(c2cnc(C)c(N)c2)=O)C2CCC1CC(NC(c1c(Br)noc1C)=O)C2 CC1CCN(C(=O)C=CC2CCC2)C(C)C1.C1(C(=O)N)CCCN1C1CCCC1 N1(C(COC2(C)CN(C(=O)CSCCC#N)C2)=O)CC(O)CC12CCC2 C12(NC(=O)Cn3cnnc3)CCN(C(=O)CN3CCCNS3(=O)=O)CC1C2 c1(C(C(=O)N)O)ccc(Cl)c(F)c1.C(C(=O)NC1CC(C)C1)(C(C)C)OC c1(C(=O)NC2C(OC)CN(C(=O)Cc3c[nH]nc3C)C2)cnc2cccnc2c1 c1(OC)cc(CNC2CC(NC(=O)Cc3cc(C)on3)C2)cc(O)c1O c1(SC)ccccc1COC(=O)C(C(C)C)NC(c1cc(C)nn1C)=O C(CNC(=NCC1CCCCC1)NCC1(N(C)C)CCC1)(C(F)(F)F)OC CC(CC(=O)N1CCC(CCNC(=O)CCc2nncs2)CC1)CC(C)(C)C Fc1cc(-c2nc(C3CCOC3)nn2CC2CCOCC2)c2ncccc2c1 c12ccc(cn1)Cn1cc-2nn1.C(=O)(C(COC)N(C)C)NC(CC)CSC N1(C(c2cc(CC)on2)=O)CCC(N(C(=O)C=NOC)CCOC)CC1 C1(O)(CC)CCCN(C(C2(C#N)CC23CCC3)=O)C1.c1(CC)cnsc1C=O.N N1(C(C2(C#C)CCCC2)=O)CCC(N(C(=O)CCNC(=O)C=CCl)C)C(C)C1 C1(N(C(CC2CN(C(c3c(CC)occ3)=O)C2)=O)C2CC2)CCCC(F)C1.O c1(CC(=O)N(C(C)C)CCNC(=O)C=C(Cl)Cl)ccc2nc[nH]c2c1 C1(NC(C2CC3CCCC23)=O)CCCCC12CCN(C(C1(Br)CC1)=O)C2 C1(C(=O)NCc2nocc2CO)(CC)CCN(C(=O)CCC(C)OC)C1 C12(C=O)CC(C)(C1)OC21CCC1.CCC(CC(=O)NCC1CCC1)C1CC1.N C1(CNC(Cc2cc(C)on2)=O)CC2CCC1C2.C1(O)(CC(=O)N)CCCCC1 CC1c2cccnc2CCN1C(=O)Nc1nc(Cl)c(C(F)F)s1 C1(NC(C(C)OCC)=O)CCCC12CN(C(c1cc(N)nc(Br)c1)=O)C2 c1(CCN(C(c2n(C)nc(CC)c2Br)C(=O)NC)C)ccc2c(c1)OCO2 Cc1ccc2oc(N3CCOC(C)(CNC(=O)C(C)(C)CS(N)(=O)=O)C3)nc2c1 CC(O)C(F)(F)C(=O)N1CCC(CCCCNC(C23CCOC(C)(C2)C3)=O)CC1 C1(C(=O)NC2C=CCN(C(=O)CCC3OCCO3)C2)CCC2(CC1)CC2 C1(CC)(NC(C2CCC2(F)F)=O)CCN(C(c2sc(F)cc2C)=O)CC1 N1(C(c2c(C)sc(Cl)n2)=O)CCCC(C)(C)C1.c1(C=O)cc(C(C)C)n(C)n1.N c1(C(=O)N)cnn2c1OCCCC2.CC1(C)COC1C(=O)NC(C)(C)C1CCC1 Cc1c(NC(C)C)cccc1Cl.n12cc(nn1)C(=O)NC1CC2C1 C#Cc1ccc(C(=O)N2CCC(C(N3CC(C4CCCO4)C3)=O)O2)nc1 C(CCOCC)(C(=O)NCCCCC1CCCC1)NC(C1C(=C)C1)=O C1(CN)CC2CN(CC3(Cc4ccccc4)CCOCC3)CC2C1 C1(NC(CCCC(=O)NCCC)=O)CC2CC(C1)N(C(=O)CCC(C)SC)C2 c1(C(=O)NCC2CCCO2)ccc(CNC(C2(O)CCSC2)=O)o1 C1(N(C)C(c2coc(C(F)(F)F)c2)=O)CN(C(=O)Cc2nc[nH]n2)CC12CC2 C=CC1CN(C(c2cc(O)cc(=O)o2)=O)CC1NC(=O)CN(c1ccccc1)C N1(C(c2ccc(OC)s2)=O)CC2CC(C(=O)NC3COC(C)(C)C3)(C2)C1 C1(NC(CCNC(=O)CO)=O)CCCC(NC(c2cnoc2-c2ccoc2)=O)C1 C1(NC(Cn2c(=O)sc(C)c2C)=O)CCN(Cc2cncc(F)c2)CC1(C)C N1(C(=O)CCC2CCCN(C(=O)COCCF)C2)CCc2nc[nH]c2C1 C#CCC(C)(CC)C(=O)N1CCC(C)(CC(N2CCC(CF)CC2)=O)C1 C1(OC)CCC2(C(=O)NCCC3CN(C(=O)C=CCO)CC3C)CC12 c1(C(N2C(CCC(C)(C)NC(C=NOC)=O)CCCC2)=O)cc(Cl)ccc1C CC(C)(CC(=O)NC(Cc1cn[nH]c1)C(=O)NC1CCC2CCC12)C1CC1 C1(C(=O)NCC2CCN(C(CC(=C)Br)=O)C2)Cc2nnc(C)n2C1 N1(C(c2c(C(C)NC(c3nc(Cl)cs3)=O)noc2)=O)CC2CC1CS2 c1(C(=O)NC23C(CN(C(C(CCSC)OC)=O)C2)C3)cccc(Cl)c1N C1(NC(CS(CCOC)(=O)=O)=O)CC2(C1)CC2N=c1ccnc(C(F)(F)F)[nH]1 C1(NC(C(CCC)c2ccccc2)=O)COC2(C1)CN(C(=O)C=CSC)C2 N1(C(c2cnc(C)s2)=O)CC2CC(NC(c3cc(Cl)nc(Cl)c3)=O)CC2C1 N1(C(C=C(CNC(C2(C=C)CCCC2)=O)C)=O)CCC2(CCC(O)C2)C1 c1(C(C(=O)NC2(C)CC(NC(c3c(C)cco3)=O)C2)C)ccc(Cl)cc1 c1(C(=O)NC(CC)CN(C(=O)C(CC)OC)C)oc(C2CCC2)nc1C C1(C=O)CC2(CCCCC2)CO1.C1(O)(CC)CN(C(=O)CCC)C1.C(C)(C)C.N C1(CNC(c2ncn(C(C)C)n2)=O)CN(C(=O)C(=O)NCC(F)F)CCC1C C1(NC(c2cn(C(C)C)nn2)=O)CN(C(=O)CCC(=O)c2ccncc2)CC1O NC1(C(N2CCN(C(N3CCOCC3)=O)CC2)=O)CCCOCC1 c1(OC)ncc(C(=O)NCC(O)CNC(C2CC(=O)C2C)=O)s1 c1(CC)ccc(N)c(C(=O)NCCC(C)NC(c2c(C)nn(C)c2Cl)=O)c1 c1(C(NCC(C)NC(c2c(CC)n(C)cc2)=O)=O)cnc2c(c1)COCC2.C C1(CCC(=O)NCCC2CCCCCC2)CCCCN1C(C1COC(=O)N1)=O C1(NC(CC2(OC)CCC2)=O)CC(F)CN(C(c2coc(C)c2)=O)C1 N1(C(C(C(C)C)C)=O)CC(NC(c2cncc(Cl)c2)=O)CC(F)C1 c1(CC(N2C3CC(CC(NC(CC4(C)CC4)=O)C3)C2)=O)c[nH]c2cc(Cl)ccc12 c1(N(C(C2C(CNC(Cc3c(CC)con3)=O)CC2)=O)C)cccc(Cl)c1 c1(CC(C#C)NC(=O)C(CN)N(C)C)cccc(C)c1 C1(CNC(C(C)OC)=O)COCCN(C(=O)C(c2ccc(Br)cc2)=O)C1 C(=O)(C(C(C)C)N(C(c1cnc(Cl)s1)C(=O)NCCCSC)C)OC Cc1ccc2n1CCN(C(c1ccc(-n3cc(OCCOCCO)nn3)cc1)=O)C2C c1(C(=O)NCC(C)CNC(=O)CSCCC#N)ccc(-c2ccccn2)o1 Cc1cc(O)cc(=O)n1CC(=O)NCC1CCN1C(=O)C(C1(O)CCCC1)F C(C)(C(C)S(C)(=O)=O)OCCNCC(C)=CC(=O)O Cc1cc(C(=O)NC2(CC(=O)NCCC34CCCC3C4)CC2)sn1 C1(C(=O)NCCCCC(C)NC(=O)CC2CCSCC2)CCC(=O)CC1(C)C Cc1cc(C(=O)N(CC(O)CNC(c2ccnc(C(F)F)c2)=O)C)ncn1 N1(C(CC(c2scc(C)c2)O)=O)CCC(C)(NC(c2cc(C)c[nH]2)=O)CC1 c1(CC)cc(C(=O)NCC(O)CC(=O)NC(C)(C)C(=O)OC)ncn1 N1(C(C=CC)=O)CCC(NC(c2ccc(C(F)F)s2)=O)CC1C1CC1 Cc1cccn2ncc(C(=O)NC(C)C(CO)NC(c3nn(C)cc3N)=O)c12 C1(CNC(CSCC)=O)C=CCN1C(=O)C=CC1CCOC1 N1(C(CN(C2CCC2)C)=O)CC2CN(C(=O)C(O)CC(N)=O)CCC12 C(=O)(C(CCCOC)NC(=O)CC1CSC1)NC(CC)C1CCOC1 c1cn(C2CCN(C(c3cnn(C4CC4)c3)=O)C2)nn1.O=C(C(O)C1CC1)N.C N1(C(C=C=C(C)C)=O)CCCCC(CCC(=O)NCC(c2cnn(C)c2)C)C1 CC1(CC(=O)NCC=CCNC(c2cc(C(F)F)cs2)=O)CCOCC1 C1(C)(CS(=O)(=O)NC(C2(O)CN(C=O)C2)C)CCCO1.C(C)(C)C.O C(=O)(CS(=O)(=O)C(C)(C)C)N(CC(CC)NC(=O)Cc1csc(=N)[nH]1)C C1(C)(CC(N2C(C(C)(C)O)CC2)=O)CCN(C(c2ncc[nH]2)=O)C1 C#CCC(O)C(=O)N1CCC(C(=O)N(CC(c2nn[nH]n2)C)C)C1 C1(C(=O)NC(CCNC(CCc2c(C)noc2Cl)=O)C)Cc2c[nH]cc2S1(=O)=O C12(C(N3CCCCC3)=O)CCCC1CCC2.C1(C(=O)OC)CC(CC(=O)NC)C1 c1(C(=O)NC(CC)(CC)CCNC(=O)C(F)C2CCC2)cncc2nc[nH]c12 CC1CC(C(=O)NCCOC2CN(C(=O)CC3CCCCC3)C2)C1(C)C CC(C)C1=NOC(C)(C(=O)NC2CCC(C)N(C(c3ccncc3O)=O)C2)C1 Cc1ccc(SCCC(N2CC(CNC(c3cncnc3)=O)CC2C)=O)cc1C C(=O)(C1CCCc2ccccc21)N1CCCC(C)(CNC(=O)Cc2cc[nH]n2)C1 CCCCC(C(=O)NC1CC(N(C)C)C1)NC(C1C(C)(C)C1(C)C)=O C1(C(=O)NC(CNC(Cn2c(C)nnn2)=O)C2CCC2)CC(C)CCO1 C1(CNC(c2c(C(C)C)occ2)=O)CN(C(=O)CC(C)N(C)C)CC(C)(C)C1 c1(C(N2C3C(NC(C(CC#C)C)=O)CC(C3)C2)=O)nn(C)c2c1CS(=O)(=O)CC2 c1(OC)cc(Cl)c(Cl)cc1C(=O)NC(CO)C(C)NC(=O)Cc1c[nH]nc1O CCCC(C(=O)NC1CC1)NC(N)=O.C(=O)C(C)C.C(=O)C(F)(F)F.C Cn1cc(CC(=O)NCCCNC(c2ccc(C#N)[nH]2)=O)c(C(F)(F)F)n1 Cc1nc2c(C#N)cnn2c(NC(=O)C(O)C(O)c2ccc(O)cc2)c1Br Cc1cc(C(=O)NCC2CCN2C(=O)CCc2cncnc2)sc1Cl C(=O)(CCCCC(N)=O)N(C(CC)CNC(=O)CCOC1CCOCC1)C Cc1cc2sc(C(=O)NCC(C)(C(C)C)NC(C3CC=CC3)=O)cc2s1 N1(C(C2CC(CNC(Cc3cc(C)on3)=O)OC2)=O)CCSCC1C1CC1 Cc1cccc(Br)c1C(C(=O)Nc1ccc(Cl)cc1)NC1C=CCC1.C(C)(C)N CC1CCN(C(=O)C=CBr)CC1N(C)C(c1cc(C2(C)CC2)n[nH]1)=O C1(NC(c2cnc(OC)nc2)=O)C(C)(C)C(NC(C2CSCCS2)=O)C1(C)C CC(C)CC(C(=O)N1CC(CNC(=O)CC2(C)OCCO2)C1)N1CCCCCC1 N1(C(CSCCCC)=O)CCC2CCN(C(=O)COC(F)F)CC2C1 C1(CC(=O)NCCN2CCN(C(C3(F)C4CCCC34)=O)CC2)CC2(CC2)CO1 c1(C(N(CC(CNC(C2(CCC)CC2)=O)O)C)=O)[nH]nnc1-c1ccccc1 N1(C(C23CC(NC(CN4C(C)CCC4)=O)(C2)C3)=O)CCC2CC12C c1(OC)cc(C(=O)N)ccc1C(N)=O.C1(C)CCN(C(=O)CC2CSC2)CC1 C1(OC)CN(C(C2CC2(C)C(F)F)=O)CC1NC(c1ccc(SC)cc1)=O C12(NC(CNC(CCC)=O)=O)CC(CNC(C3CNC(=O)C3)=O)(C1)C2 N1(C(CC(CC)SC)=O)CCC2C(NC(C3CN(C4CCN(C)CC4)C3)=O)CC12 c1(C(N(C(C)CCNC(C2C3CCCCCC23)=O)C)=O)cc2c(nn1)CCC2 c1(C(=O)NC2CN(C(c3cn(C)c(=O)cc3)=O)C2)cc(F)c(N)c(F)c1F N1(C(C(CC2CN(C(c3ncn(C)c3)=O)C2)F)=O)CCCC2(C)CCCC12 Cc1cc(CNC(c2nc(C3CC3)no2)c2nnnn2C)c(C)n1C c1(C(=O)NCc2ccc(CCC)cc2)cc(F)ccc1F.C(=O)CP(C)(C)=O.N C12(CC(=O)NCC3CC(NC(C4C(C)CCCC4)=O)C3)CCCN1CCC2 N1(C(c2[nH]cc(C(N)=O)c2)=O)CCC(Cc2nc[nH]n2)CC1 c1(C(NC)=O)ccccc1Cl.N1(C(C2(SCC)CC2)=O)CCCC1.C1CC1.C C1(NC(c2cncc3nc(O)[nH]c23)=O)CCCC12CCN(C(C1COC1)=O)CC2 c1(OC)cccc(CNCc2cccc(C)c2OCC(F)F)c1C#N Cc1cc(C(N2CC3CC3(NC(=O)CC3CN4CCC3CC4)C2)=O)c(C)n1C c1(C(=O)NCC2(C)N(C(CC(C)OC)=O)CCC2)nn(C)c(Br)c1C c1(C(=O)NCCOCCCNC(=O)CCc2ccccc2)cc2c(s1)CCCC2 C1(C)CN(C(=O)C2=NNC(=O)CC2)C(C)(C)C1.C(CCC(=O)NC)OC(C)C C1(CC(=O)N(CCCC(=O)NCCc2nc(C)sc2)C)CCC(C#N)C1 C1(CNC(C(C2CCCCCC2)OC)=O)CCCN(C(=O)Cc2ccoc2)C1 C(=O)(CCC(CC)NC(C1(C#N)CCC1)=O)NC(CC#C)C(=O)OCC C1(CC)CCCCCCN1C(c1cccnc1)C(=O)NCCSC C(c1cc2ccccc2o1)=CC(=O)NC(C(C)NC(C1CCC12CCC2)=O)(C)C Cn1c(=O)c2ccc(NC(=O)C=CCCC(C)(C)C)cc2n(C)c1=O c1(CC)cccc(NCC2CCC(C(O)C(=O)O)CC2)c1 C1(NC(C2CC2(F)F)=O)CC2CN(C(=O)C(O)Cc3ccc(O)cc3)CC2C1 c1(CCC)cnnc(C(=O)NCC2(C)CCCN2C(c2cc(Cl)n(C)n2)=O)c1 CCC(O)C(C)C(=O)NCCCN(CCCNC(c1ccoc1Cl)=O)C C(=O)(C(C1CN(C(=O)C(F)=C(C)C)C1)OC)N(CC#C)CC1CC1 c1(OC)c(OC(F)F)ccc(CN2CCOC(C(C)C)C2)c1[N+](=O)[O-] CC(C)(C(=O)NCCOC1CN(C(c2cc(F)c[nH]2)=O)C1)c1ccsc1 CCCCC(O)C(C)C(=O)N1CC(NC(C2(OC(C)C)CCC2)=O)C(CO)C1 N1(C(c2csc(Cl)c2)C(=O)NC)CCOC2CC12 CCS(=O)(=O)CC(=O)N1CCC(OCCNC(C2CCOC(C)(CC)C2)=O)C1 CC1(C)CCN(C(C23CCC(C)(CC2)OC3)=O)CC1NC(c1snc(O)c1Cl)=O C#CCCN=C(NCCCNC(=O)NC)N1CCC(C)C1C N1(C(CCCCCC)=O)CC2(CC(NC(c3nc(OC)ccc3C)=O)CO2)C1 C=CCCC(C(=O)N1CC(O)CC1COC)NC(c1occc1COC)=O C1(NC(C2CCN(C(C(CC)C(C)C)=O)C(CC)C2)=O)CN2CCC1(F)CC2 C1(C(N(CCC)CCNC(=O)C(F)CC2CCCC2)=O)(C)CCCCO1.O Cc1ccc2[nH]cc(CC(N3CC4(CC4)CC3C(N3CCOC(=O)C3)=O)=O)c2c1 N1(C(C2(CC)CCCC2)=O)CCC(NC(=O)CC2CC3CCC2C3)CC1 C(=O)(C#CC1CCOC1)NC(C(C)NC(c1c(C)n(C2CCOC2)nn1)=O)CO c1(N2CCCC2)ccc(Cl)c(F)c1.N1(C(=O)OC(C)(C)C)CC(CC(=O)O)C1 N1(C(C2C(C)OC(=O)N2)=O)CCCCC(NC(C2CCCCC2)=O)C1.C(N)(=O)N N(C(=NCCCn1ccnn1)NCc1ccco1)C1CCN(CCOC)C1 c1(C(N2CCCC2CCNC(C2(F)CCOC2)=O)=O)csc(C(F)(F)F)c1 c1(C(=O)NC(C2CCN(C(CSCC(C)C)=O)C2)(C)C)ccc(F)c(O)c1F N1(C(c2c(C#C)cn(C)n2)=O)CCCC2(CCN(C(=O)C(CC)CC(C)C)C2)C1 CCC(C)(CNC(C12C(=O)C3CC1C2C3)=O)C(=O)Nc1cc(F)ccc1O n1(C(C)C)cc(C(=O)N(CC(C)C)C)ccc1=O.C(c1cn(C)nn1)=CC=O.N c1(C(=O)NC(C)C(C2CCCCC2)NC(C2CCC=CCC2)=O)ncccc1N CN1CCN(C(=O)C(F)OC(F)(F)F)CC1CNC(c1cc(O)nc(O)n1)=O C1(N(C(c2ncn(CC)n2)=O)C)CN(C(c2c[nH]c(C(N)=O)c2)=O)CCC1O c1ncncc1Cl.C1(NC(=O)CCC)C2CC(NC(C3C4COCC34)=O)CC12 CN=C1SC(CC(=O)NC2CCCN(c3cnccn3)C2)C(=O)N1C N1(C(c2ccc(C(=O)OC)cc2F)=O)CCC2(CC(NC(=O)CSC)C2)C1 C1(NC(c2cnc(C(C)=O)s2)=O)CC=CCC1NC(=O)CCc1ccccc1 C(=O)(CC(C)C(=O)NC1CC(NC(=O)CC(C)N(C)C)C1)OC C(c1ccc(C)cc1)=CC(=O)NCC(CCCC)NC(C1CC(O)C1)=O N1(C(C)=O)C(=O)CCC1C=O.C1CCCN(C(=O)C(C)(C2(C)CC2)NC)C1 c1(OC)ccc2nc(C(N3CCC4(CNCCO4)C3)=O)ccc2c1 CC(C)(N=[N+]=[N-])C(=O)NCC#CC(=O)NCCc1cccnc1 C1(C(=O)NCC(=O)NCC)C2CC1N(C(=O)CCC1CCCO1)C2 c1(NC(C2(CC)CCN(C(C(CCC)OCC)=O)CC2)=O)c(C)ccn(C)c1=O c1(NC(C2CC(CC)N(C(=O)CCc3nccs3)CC2)=O)cnc2ccnn2c1 CC(C)CCCC(C)C(=O)NC.C1C(C2CC2)CCN1C(=O)C=C1CCN(C)C1 n1(CCCNC(C2(CC(C)=O)CCC2)=O)cc(-c2cn[nH]c2)nn1 c1(NC(c2scc(C)n2)C)nc(C)cc(=NCCC(C)O)[nH]1 CCCC(C(O)C(=O)N(C1CCCC1C)C)NC(C1(C)CC=CCC1)=O CC1COCCN1Cc1cn(C2CC3(C=O)CC23)nn1.C1CC(=C2CCC2)C1.N N1(C(c2nc(Cl)ccc2Br)C(=O)NC)CCc2c(F)cccc21 C1(NC(C=CC(C)C)=O)CN(C(c2ccc(C(F)F)nc2)=O)CC1C1CC1 Cc1cc[nH]c1C(=O)NCCN(CC(C)O)C(=O)CN1CC(C)(C)C1 CCCC(C(=O)NC1CC1C(=O)OCCc1cc(N2CCCC2)ccn1)C(C)C c1(C(C)OC)ccc(O)c(C(=O)NC2CC2Cl)c1 C=CCC(C(=O)N1Cc2ccccc2CO1)NC(c1ncn(C(C)C)n1)=O C1(C(=O)Nc2n(CC)nnn2)CCN(C(=O)C(C)(C)C)CC1.c1(N)nccs1 c1(OC)ccc(C(N2CCCC2CN(C(=O)C(O)Cc2cnc[nH]2)C)=O)cc1N c1(C2(C(=O)NC(CNC(C3CCC(CC)O3)=O)C)CCC2)c(F)cccc1Cl N1(C(CCC2CCN(C(CN3C(C)CCCC3)=O)CC2)=O)CCCC(F)(F)C1 C(C1CCCN1C(=O)CC1CCCC1O)=CC(=O)N(C1CC(SC)C1)C C1(NC(C(CCOC)C)=O)C(C)(C)C(NC(=O)CO)C1(C)C.c1ccsc1 C1(NC(CC(CC)NC(=O)CCS(C)(=O)=O)=O)(CO)CCCCCC1 C(=O)(CCCCC(=O)N1CCN(CC(=O)NCc2nc(CSC)no2)CC1)OC c1(C(n2cc(CNC3(C4CCCCO4)CC3)nn2)CC)cccc(Cl)c1 N1(C(C(c2c(OC)cccc2)O)=O)CCC2CCN(C(c3csc(S)n3)=O)C2C1 c1(C(N(CC(CC)NC(=O)C(C)Oc2ccc(F)cc2)C)=O)cnc(C)cc1Cl C(=O)(C(F)C(C)(C)O)NC1(CCNC(C(CC#C)O)=O)CCC1 c1(C(N(C2CN(C(c3cnc(Cl)cc3I)=O)C2)C)=O)ccc2c(c1)C(=O)OC2 N1(C(CCCc2c(C)ccs2)=O)CC2CC(C1)N(C(=O)CNc1nccs1)C2 CC(C)C(F)C(=O)NC1(CCNC(c2ccc(CO)cn2)=O)CCC1 c1(C(=O)NCC(CC=C)NC(c2cc(OC)nn2C)=O)ccc(Br)c(N)c1 c1(C2N(C(=O)CC(C(F)F)N3CCOCC3)CCC2)nc2ccc(Cl)cc2[nH]1 C1(NC(C(C=C=C)C)=O)CCN(C(=O)CC(F)(F)F)C1(C)C c1(CC)cc(C(N2CC(O)CC2CNC(=O)C(c2ccccc2)F)=O)nn1C c1(C(=O)NCC2CC(NC(C(CC)=CC)=O)C2)ccnc(N2CCCC2)c1 N1(C(COC(C)(C)C)=O)CCOC(c2cn(-c3cccc(C(N)=O)c3)nn2)C1 C(=O)(CC(C(=O)N1CC(CCCCNC(=O)CC=C(Cl)Cl)C1)N(C)C)OC c1(C(N2CC3C(C=O)(C3)C2)=O)cn2c(n1)CN(C(=O)Cc1noc(C)n1)CC2 c1(OC)c(C(=O)NCC2CC2C)oc2ccccc12.c1(C=O)cnoc1C.N C1(NC(C=CC)=O)CCS(=O)(=O)C12CN(c1cc3nncn3cn1)C2 c1(C(N2CCC(C)C2)=O)ccc([N+](=O)[O-])c(S(N)(=O)=O)c1.C1(C=O)CC1(F)F N1(C(CCC(C)SC)=O)Cc2occ(C(=O)Nc3c(C)ccn(C)c3=O)c2C1 N1(CCC(=O)NC(CCNC(C2CN(C(=O)NC)C2)=O)C)CCOC1=O C(C)(C(=O)NCC=CC)(c1ccccc1)NC(C)C.c1(C=O)scnc1Cl.O C(=O)(C1=C(c2ccccc2)N(C)C(=O)N(C)C1c1cnc(OC)c(F)c1)OC Cc1ccc(C=CC(=O)NC2CCN(C(=O)CN3CCCNC3=O)C2C)cc1Cl Cc1cc(Cl)c(C(=O)NCC(CNC(c2ccccc2SC(F)F)=O)CO)cn1 N1(C(C2CCN(Cc3cnc(Cl)cc3Cl)C2)=O)Cc2cccc(F)c2C1 c1(C(C(=O)NCC2(Cc3ccc(F)cc3O)CC2)N(C)C)ccc(F)cc1Br C(C)(C(O)C(F)F)NC(C1N(C(CCn2ncc(C)c2)=O)C(C)C1)=O c1(C(CC)NC(=O)NCCN2CCOCC2)ccc(Br)cc1 C1(NCC(C(C)O)C)CCC(Oc2ncccn2)CC1 C1(S(C)(=O)=O)(C=O)CC1.C(c1cnc[nH]1)=C(C)C(=O)N(C1CCCC1)CC c1(C(N(C2CCCC2)CCCNC(C(C)=CC)=O)=O)cc(C)n(CC)n1 c1(C(N2CC(F)(CNC(C(C)=CC)=O)C2)=O)ccc(-n2cncn2)nc1 C(=O)(C1=CC(C)C1)NC1C(NC(Cc2c(C)occ2)=O)CCC1 C(C(C(=O)O)NC(c1cn(CCNC(=O)CCc2cnoc2)nn1)=O)OC N1(C(c2cc(C)ccc2)=O)CCC2CC(C(=O)NCC(C)C)C2C1.C(C)(C)(C)N Cc1cccc2cc(C(=O)NC3C4CCC3N(C(c3cnc(O)o3)=O)C4)nn12 C1(C(=O)NC(c2ccccc2)C(=O)NCC(CC2CC2)OC)CCCC1 C1(C(=O)NCCCCCCOC)CCOCCN1C(C1(CCOC)CCC1)=O C1(C=O)CC2(CC2)C1.C(C(C(=O)NC)N(C)C)OC.C1(O)(CC)CCC1 c1(C(=O)NC2(CNC(CC(CCSC)O)=O)CCC2)cc2ccccc2c(O)n1 C1(CC(=O)NC2(C(N3CC4CCC3C4)=O)CCCC2)CC2CCC1O2 C1(C(=O)OC)CCCC(NC(c2cc(-c3cncs3)on2)=O)CC1 CCCCCS(=O)(=O)CC(=O)N1CC2CC(NC(C3(CO)COC3)=O)CC1C2 C(=O)(CCCN=[N+]=[N-])N(C1CCC(NC(CN(CC)CC)=O)C1)C C1(CNC(CCOCC)=O)CN(C(c2cc(N3CCCCC3)ncn2)=O)CCO1 CCC(CC(C)C)C(=O)N1CCCC(F)(CNC(=O)C(C)Oc2cccnc2)C1 C1(C(N(C2CCN(C(C34CC(CO3)C4)=O)C2)CC)=O)CCCC2(CC2)C1 N1(C(c2cc(OC)c(Cl)cc2)=O)CCC(F)(F)C(C)C1.C1(O)(C(=O)N)CCOC1 CCCC(C)=CC(=O)NCC(CNC(=O)CCOC1CCC1)OC N1(C(C2CCC(C)(F)CC2)=O)CCc2sc(CNC(C3CCNC3=O)=O)nc2C1 N1(C(C2(CC)CCN(C(=O)CCCNC(N)=O)C2)=O)CC2CC1CN2C CC(CNC(C1(CO)CCC1)=O)CC(=O)NCC1CC(=O)N(C)C1 Cc1cc(Br)c(C(=O)NC2CCN(C(C3CCCC(F)C3)=O)CC2)s1 c1(CC)cccc(C(N2CCC3C(NC(c4cnc(C)cn4)=O)CC23)=O)c1F CC1CC(NC(=O)C(C)Cc2ccncc2)CN(C(=O)CCc2ccc[nH]2)C1 C1(C(N(C(C(N2CC(CCOC)C2)=O)C)C2CC2)=O)CC(=O)CC(=O)N1 C(=O)(CC(C)(F)F)NC(C(C)NC(c1cc(-c2cccs2)on1)=O)(C)C CC(C)CC(CNC(=O)CCCCCNC(c1cnc(S)nc1)=O)CO CC(C(=O)NC(C)CCN(C(=O)CC1CCCC1)C)c1ncco1 C(=O)(CC(C)P(C)(C)=O)N1C(CCNC(c2n(CC)ccc2)=O)CSCC1 n1(CCCF)nnnc1C(C1C2COCC12)NCc1cccnc1 N1(C(c2c(CC)nc(C)o2)=O)CCN(C(=O)CCCF)CC1CCO N1(C(C2(N(C)C)CCOCC2)=O)CC(NC(c2ccsc2Cl)=O)C(C)(C)C1 CC(CC(=O)NC(C1CN(C(=O)COc2cnn(C)c2)CCO1)C)CC(C)(C)C N1(C(C2C(C)C2)=O)CCC(CCNC(C2CN(c3nnnn3C)C2)=O)C1 N1(CC(=O)NCCC2CN(C(C3C(C)C3C)=O)C2)C(=O)CCC1=O CCC(CC(=O)NCC1CC(F)(C)C1)CC(F)(F)F.C1(CC=O)CCOC1.N c1(C(N2CCCC(Nc3ncc(Br)c(O)n3)C2)=O)ccnc(F)c1F CCS(=O)CC(=O)NCCC(=O)NCCCOCC(F)F CCCC(C#N)C(=O)NCC(C)NC(c1cccc(C(C)(F)F)n1)=O c1(C(=O)NC2(C)CN(C(CC(c3ccc(OC)cc3)C)=O)C2)cc(C)cnc1Cl c1(CC)cc(C)ccc1NC(=O)C#CCNC(=O)COC1CCCOC1 C1(OC)(OC)CCC1C(N1C(C(=O)NC2(C)CCSC2)CC1C)=O N1(C(C2(C#N)CCC2)=O)CC(NC(C2C3CCC2(c2cccs2)C3)=O)C(O)C1 C1(CCC(=O)NCCCN2CCOCC2)(NC(c2csnc2Cl)=O)CCCC1 CCC(CCOC)C(=O)NCC1(F)CN(C(=O)C(C)CC(F)F)C1 n1(CC(N2CC(CC(C)NC(C3CC34CC4)=O)C2)=O)cc(Br)cn1 N1(C(C2CCC(C)C2)=O)CCC(CNC(c2ccccn2)=O)C(C2CC2)C1 C1(N(CCC)C(C2CC2C2CCCO2)=O)CCN(C(C2(O)CCOCC2)=O)CC1 c1(C(=O)NC2CC(O)CN(C(=O)CCCC3CC3)C2)ccc2c(c1O)CCC2 Cc1ccc(F)c(CC(=O)N(C(C)CN(C)C(c2c(Cl)n[nH]c2CCC)=O)C)c1 c1(C=O)nn(C)c2c1CCC2.CC(C)(C)C.C1(C(=O)N)CC1C=O.C#CC C(=O)(CC(C)(C)C1CC1)N1CC(C(C(=O)NCC(C)C)OC)C1 CCCCCC(F)C(=O)NCC(CNC(=O)C(CC)CCC)OC N1(C(c2c(NCc3cccc(C)c3)c[nH]n2)=O)CC=C(c2ccccc2)CC1 c1(C(N(CC(C)CNC(=O)COC)C)=O)cccc(F)c1F.C1(F)CC1 C(=O)(C(CCCC(=O)OC)N(CCCF)C)NCC=C C(C(C(=O)NCCc1cn(CC)cn1)C(C)(C)C)NC(CCCCC)=O c1(N2CC3C(C)(C)C(C3)C2)nc(=NCCCC23CCCC2C3)[nH]c2c1SCC2 N1(CC(=O)N(CCC(C)NC(C(=O)NC(C)=O)C)C)Cc2ccccc2C1 C1(C(N(C2CCN(C(C(CC)NC(C)=O)=O)CC2)C)=O)CCC(=O)N(C)C1 C1(C(C)(C)C)(C)CCN(C(C2CCCS2(=O)=O)=O)C1.n1(CC=O)[nH]cnc1=N C1(C(=O)NCCC(C)(C)NC(C2(C(=O)NC)CC2)=O)COCCC1C C1(C(=O)NC(C2N(C(C=C(C)C(C)(C)C)=O)CCC2)C)CCOC2(CCC2)C1 C12(NC(c3c(Cl)ccc(C)c3)=O)CCCN(C(=O)C(O)C3CCC3)CC1C2 Cc1cccc2oc(N3CC(NC(=O)CCCN(C)C)CC(C)(C)C3)nc12 C1(C(=O)OCC)(C(c2nnnn2C)Nc2cnn(C)c2C)CC=CCC1 N1(C(C(C)N(C)C)=O)CCC(NC(c2ccc(-c3cccnc3)s2)=O)C(CO)C1 C1(C(N(CC(CC)O)CC)=O)CCCC1CNC(c1cc(C)[nH]n1)=O C(=O)(C(O)CC(F)(F)F)N1C(C(=O)NCCC(C)c2cn[nH]c2)CC(O)C1 c1ccccc1.C(CCC(=O)N1CCC(N(C(=O)CO)C)C1)OC.C(=O)C1CC1 N1(C(C(CCC)N(C)C)=O)CC(C)OC2(CCN(C(=O)CCCCC#N)C2)C1 C1(C(=O)OCCCCS(C)=O)CN(C(=O)OC2CC2)CCC1O C=C(C)CC(C)C(=O)N1CCCC(F)(CNC(c2ccc(F)c(F)c2)=O)C1 C1(CCC(=O)N(CCC(C)NC(=O)CCC2CC2)C)CCC(=O)C1.C1CC1 Cc1ccc(F)cc1CC1CC2CCC1C2.c12nc(Cl)c(s1)c(=O)[nH]2 c1(CC=O)noc(C)c1C#N.N1(C(C(C)NC(=O)NC)=O)CCN(CC)CC1 C1(C(=O)NC(CNC(COCC(C)C)=O)CO)CC(C)CC(=O)N1 c1(C(=O)NC(CNC(C(CC)OC2CCCC2)=O)C)ccnc(C(C)C)n1 c1(C(N2C3C(NC(=O)Cc4cc[nH]n4)CC(C3)C2)=O)cc2c(F)cc(F)cc2[nH]1 C#Cc1ccc(C(=O)NC(C)(CSC)C(=O)NC(C)Cn2cnnc2)cn1 c1(C(N(CC(C)NC(=O)C)CC)=O)[nH]c2ccc(C)cc2c1C.CCC(C)C.S c1(-c2cc(OCC)c(F)cc2)ccc2c(C(=O)OCCCC(F)(F)F)n[nH]c2c1 C12(NC(COCC)=O)CCC(C(N3CCN(C(C)=O)C(C)C3)=O)(CC1)C2 N1(C(C)C)CCCN(C(=O)COC(=O)NCCNC(C2CCCC2)=O)CC1 Nc1ccc(-c2cn(C3(C(F)F)CC3)nn2)cc1F.c1ccc(C)cc1 N1(C(C2(C(=O)NC)CCC2)=O)CCC(N(C(=O)CCS(C)=O)CCO)CC1 c1(NC(CC2CCN(C(c3ccc(COC)cc3)=O)C2)=O)ccc(Cl)nc1Cl CC(O)C(C)(C)C(=O)N1CCC(C(C)(C)CNC(c2cnsc2)=O)CC1 C1(C)(CNC(C=CCCC(C)C)=O)CCN(C(=O)C(C)CC(C)C)CC1 C(=O)(CC(F)(F)CC)NC1(C2N(C(C(CC)NC(C)=O)=O)CCCC2)CC1 C1(C(=O)NCCc2ocnc2CO)CC2CCC(C1)N2C(C1CC1Cl)=O c1(C(N2CCC(CNC(c3c(CC)onc3C)=O)C2)=O)cc2n(n1)CCO2 c1(C(=O)NCCC(C)C)c(O)ccc(Cl)c1F.C(=O)C(F)(F)CC1CCCO1.N Cc1c(C(=O)NCC(O)CN(C)C(C23CC(CCO2)C3)=O)oc2c(C)cccc12 N1(C(C(COCC)n2cc(COC(C)C)nn2)=O)CC2CCC1C(O)C2O c1(C(N(CCC(c2cccs2)NC(=O)COC)C)=O)cccnc1.C1CC1 c1(CC(C)C)ccc(C(N2CCC2(C)c2ccccc2)C(=O)NC2CC2)s1 Cc1ccc2c(C(=O)NC3CN(C(c4nc(C)sc4C)=O)CC3C)coc2c1 CC(C)(C)C1=NOC(C)(C(=O)NC2CCC2)C1.c1(C=O)cnn(CCO)c1N.N C1(CNC(c2c(N)cccn2)=O)CCN(C(=O)CC2(O)CCC2)CC1C1CC1 C(=O)(C(C)(C)C(C)NC(c1nsnc1O)=O)N1CC(CCC)OCC1 C1(NC(CCCc2onc(CC)n2)=O)CN(C(=O)CCP(C)(C)=O)CC1C1CC1 c1(C(=O)NCC(CC=C)NC(=O)CC(CN(C)C)C(F)F)nc2sccn2c1C CC1CN(C(c2cc(O)ncn2)=O)CC1C(=O)NCCCOCC1CCC1 C1(C(C)NC(CSC)=O)CCN(C(=O)CCc2cscn2)CC1 N1(C(C=CC(CC)C)=O)C(CNC(c2sccc2F)=O)CC2CCCC12 C(=O)(C(F)n1ccnc1)NCCNC(C=CC=CC)=O CC(C)CC1CCC1.C(=O)C(C1CC1)N(C)C(C1CCC1C(C)(C)C)=O n1(CCC(=O)NC(C2CCCN2C(C2CN(C)C(=O)N2)=O)C)cccnc1=O CC1CCN(C(C2(O)CCCC2)=O)CC1CNC(=O)COc1ccccn1 Cc1nc(CCC(N2CC(CNC(c3ccnn3CCF)=O)C3CC23)=O)oc1C C1(C(C)C)N(C(=O)C(C)O)CC12CCN(C(c1cccc([N+](=O)[O-])c1)=O)CC2 N1(C(c2cscc2Br)=O)CCN(C2CC(NC(=O)C(F)(F)F)C2)CC1 C(=O)(CCCCCCn1cc(CNC2CCC2)nn1)NC1C=CC(C)(C)CC1 C1(C)(NC(COCCOC)=O)CCN(c2nnc(C(C)(C)C)o2)CC1 c1(OC)ccc2c(c1C(=O)NCC#CCNC(=O)CCc1ccncc1)CCC2 CCCCC(CCCC)NC(C1(C(C)C)CCN(C(=O)C(C)N2CC(C)C2)C1)=O C(C(C)C)(C(O)C(=O)N1CC=CCC1C(=O)NCCC(C)CO)OC C(=O)(CCS(N)(=O)=O)N1CC2C(CNC(C3CN(C(C)C)C3)=O)(C2)C1 CCC(C)(C)C(O)C(=O)N1CCC(NC(=O)C=Cc2ccccn2)C1(C)C C(=O)(C(C#N)C(C)(C)C)NC1CC(OCC(=O)NC23C(CN(C)C2)C3)C1 C1(C(=O)NC(CC(C)NC(c2c(Cl)nn(C)c2Cl)=O)C)CCc2[nH]nc(O)c2C1 c1(C(=O)NCC(CC)NC(=O)CC2OCCOC2(C)C)cc2[nH]ccc2s1 c1(C=O)ncc(C(N)=O)cc1Cl.C(=O)(CCC(=O)NCC1CC1)NCCC C1(C(N(C2CCN(C(C(C)C)=O)C2)Cc2ccccc2)=O)CC(O)(C#N)C1 CC1(COC(=O)CC2CCCC2O)CS(=O)(=O)C1 c1(OC)cc(F)cc(C(N2CCN(C(C3CCN(C)CC3)=O)C(CO)C2)=O)c1N c1(CNC(COCC#C)=O)ocnc1C(=O)NOCC(=O)OC(C)=O CN1CCN(C(=O)NCCS(=O)C(C)(C)C)CC1C1CC1 S(=O)(=O)(CC(=O)N1CC(O)CC1CNC(=O)C(C)O)NC.C1CCCO1 Cc1cc(C)c(C(=O)N(C(C)CNC(=O)CCC=O)C)c(C)n1.C1CCCC1.N Cc1nc2n(n1)CCN(C(C1(F)CCCN(C(=O)C(C)CC3CC3)C1)=O)C2 C(=O)(N1CC(n2cc(C(C)(C)SC)nn2)CO1)C1C(C(=O)OCC)C1 CC1CCN(C(c2cnc(C(F)F)nc2)=O)CC1CNC(=O)CN1CCSCC1 C1(C(C)C)(C(=O)NC2CC=CCC2)CCN(C(c2ccc(F)cc2)=O)C1 C1(CC(=O)NCC(C)(CO)NC(Cc2cncc(C)c2)=O)CC2CCC(C1)N2C O=C1CCCC(CC(=O)NCC2(NC(=O)COC3CCC3)CCOCC2)C1 Cn1ccc(C(=O)NCC2CC(NC(C3CCCCO3)=O)C(O)C2)cc1=O C1(C#N)(OC)CC(C(N2CCCC(N(CCF)C(c3ncccc3Cl)=O)C2)=O)C1 c1(C(N(C2CC(NC(C3N(C)CCCC3)=O)C2)C)=O)c[nH]c2nccc-2c1 c12nc(c3ccccc3n1)N(C1CCNC1)C2=O.c1(CC)c(F)cc(Cl)cc1Cl C1(C(=O)NC(CNC(c2cc(C)c(O)nn2)=O)C(C)(C)C)CCC2(C1)CC2(F)F N1(C(c2cn(C)c(=O)nc2O)=O)CC2(CCN(C(C3COC(C)(C)O3)=O)CC2)C1 CC1COCC(CC(N2CC(CC(F)C(=O)NCCc3ccsc3)C2)=O)O1 c1(OC)cc(C(=O)NCCCC2CCCCN2C(=O)C(C)CC2CCC2)ccn1 N1(C(C(=CC2CCCC2)C)=O)CC2CCC2(CC(=O)NCc2cc[nH]n2)C1 C1(C(=O)NC(CNC(CC2CC(SC)C2)=O)C)CCCN(CC(F)(F)F)C1 N1(C(C(=O)NCCOCCCC)=O)CCSCC1CCNC(=O)C(C)CO c1(C(N2C(C)(CCC(=O)NC3C(C)(C)C3)CCC2)=O)ccc([N+](=O)[O-])o1 C(CCN(C)C(C1CCOC1C1CC1)=O)C(C)C.c1(C(C)C)cc(C=O)on1.N O(N=C1CCCCCC1)CC(=O)NC1C(NC(C2(OC)CCSC2)=O)COCC1 C1(COC(C(c2cscn2)N(C)C)=O)CCCN(C(N)=O)C1.C1CN(C=O)C1 CCC(C)C(O)C(C)C(=O)NC1CC(CNC(c2ccccc2C)=O)C12CCC2 N1(C(CCCCNC(N)=O)=O)Cc2ccc(CNC(c3cc(F)n[nH]3)=O)cc2C1 CCC(CNC(=O)N(C(C)C(=O)NC1CC1)C)(CC)N1CCOCC1 N1(C(C(C)NC(C)=O)=O)CCCC(O)(C)C1.c1(CCC=O)cc(C)nc(C)c1 C1(CC)C(C(=O)NCC(O)CCO)CCN1C(c1ccnc(C)n1)=O c1(C(N2C(CNC(C3CCC3(F)F)=O)CCC2)=O)cncc(O)c1 c1(OC)ccc(CCC(N2C(C(=O)N)CC3CC23)=O)cn1.C(C(F)(F)F)C1CC1 N1(C(C(C)SCC)=O)C(C(=O)Nc2cnccc2N(C)C)CC2CCCC12 C(=O)(C(CC)C(C)C)NCCNC(C=CC(CC)=CC)=O.C1CC1.C c1(OC)nccnc1C(=O)NC1CCC(CNC(=O)CC(C)O)CC1 C1(C(=O)OC)(COC(c2nc(CCC)oc2)=O)CCCCS1(=O)=O C(CN=c1ccnc(NCCN2CCOCC2(C)C)[nH]1)N1C(C)CCCC1 c1(C(=O)NCC2N(C(c3cccnn3)=O)CCN(C)C2)ccccc1S(C)(=O)=O N1(C(Cc2ccco2)=O)CCCCC1CC(N)=O.CC(C)(C)C(=O)NCC(=O)N c1(C(=O)NCC(C)NC(=O)C(C)CC(N)=O)ccc(N)c2cnccc12 CC1=C(C(=O)NC2CN(C(C3CC(=O)C3C(C)(C)C)=O)CC23CC3)CCO1 C12(C(N3C(C)CC(NC(=O)Cc4ccccc4)CC3)=O)C3C4C1C1C2C3C41C#N c1(CNC(c2ccc(OC)s2)=O)cccc(C(=O)NOCCCN(C)C)n1 C#Cc1ccc(C(=O)N(CCC(=O)NCCC2CCSC2)CC=C)o1 N1(C(C(CCOC)NC(=O)CC2CNC(=O)O2)=O)CCC(C2(O)CC2)CC1 C12(CNC(c3ccnc4c3CCC4)=O)CCCC1CCN2C(c1n[nH]cc1Cl)=O C(C(=O)NCC(C)(C)CC1CC1)(C(C)C)NC(C(C)OCCCC)=O N1(S(CC)(=O)=O)CCCC(C(=O)NC23CC2CN(C(=O)Cc2ccnn2C)C3)C1 c1(C(=O)NC(CC)CNC(c2cnc(C(F)F)s2)=O)cc(C(=O)O)ccn1 C1(CC(=O)NCCN(C(=O)Cc2csnn2)CC)COC1.C(C)=O.N C1(CCC(=O)NC2CC(=O)NC2)CCCCN(C(=O)C=CCN2CCCC2)C1 C1(C)(CNC(C(C)C2CCCC2)=O)CC(F)(F)CN1C(C1SCCCS1)=O C1(C2CC2)(C(=O)NCC2C(NC(CC(C)C3CCCCC3)=O)CC2)CCC1 C1(C(N2CC(N(C(c3ccc(C(C)=O)cc3)=O)C)C2)=O)C2Cc3ccccc3C12 n1(CC)cc(NC(=O)CCNC(=O)C=Cc2ccoc2)c(C)n1.C1CC1 N1(c2n(CCOCC=C)c(SC(F)F)nn2)CCC2COC(=O)NC2C1 C1(CNC(COC(C)C)=O)N(C(C2CC3(C2)CC32CC2)=O)CCCC1(C)C c1(C(=O)NC2CCC(NC(=O)C(Cl)(Cl)Cl)C2)ccc(I)c(Br)c1 n1(CC)ncc(C(=O)NC(CC2CC2)C(=O)NC(c2ncc(C)o2)C)c1C C1(C(N)=O)CN(C(=O)CC2CCCN2C(C)C)C1.C1(C)CC1C=O.CO N1(C(C(CCSC)NC=O)=O)CCCCC(N(C(=O)C(C)SC)C)C1 C1(NC(C(F)(F)C2(OC)CCC2)=O)CC12CCN(C(C1CCC(=O)C1)=O)CC2 c1(C(N2CC(OC)(C)C2)=O)ccc2nccnc2c1.n1(CC(=O)N)cc(C)cn1 C(=O)(C(F)(F)c1cnn(C)c1)N(CC(C)NC(=O)CC1C=CCC1)C Cc1ncn(C)c(=O)c1C(N1CCC(CCN(C)C(C2CCCC2)=O)CC1)=O c1(C(N(CC(CNC(c2c(CC)ccs2)=O)(C)C)C)=O)nc2cccnc2s1 N1(C(=O)C(F)(F)c2cncs2)CC2CCCC2(CNc2ncc3c(n2)COC3)C1 N1(C(C(C(CC)C)=O)=O)Cc2occ(C(=O)NCC(O)C(C)(C)O)c2C1 c1(CNC(=O)NC(CC)CO)c(C)sc2ccccc12 C1(O)(C(N2CC=CC(NC(c3ccccc3NCCO)=O)C2)=O)CC2CCC1C2 Cc1ccc(C=CC(N2CCC3CCC23CNC(c2sccc2Cl)=O)=O)cn1 C1(N(CC(c2ccccn2)C)C)CCCCN1C(=O)OC(C)(C)C c1(OC)ccc(C(N2CCC(CF)(NC(C3CCCCS3)=O)C2)=O)c(O)c1 c1(C(C)=O)n[nH]c(=NCC2CC(CNC(=O)C=CC(C)(C)C)CO2)o1 Cc1cccc(C(=O)NC2CCN(C(C3CCCN3S(C)(=O)=O)=O)C23CC3)c1C c1(C(N2CC(CNC(C3C(C(=O)OC)C3)=O)C2)=O)cc(C)c(O)nn1 c1(CCOCCCNC(C(=O)NCc2ccccc2)=O)cccc(Br)c1 C1(C2(NC(C3C=CCCC3)=O)CC2)CCCN1C(=O)C(O)CC1CCC1 N1(C(c2cc(C)c(C)o2)=O)CCC(NC(=O)C(n2ccnc2C)C)CC(C)(C)C1 c1(OC)ccccc1C=CC.C1(CC=O)CC(C(F)F)C1.C1CC1C=O.N C(=O)(C1CCc2nccn21)N1CCC(CC)(NC(c2cnc(OC)c(C)n2)=O)C1 C1(C(=O)NCC(C2CC2)NC(c2nc(CC)sc2)=O)CCC(C2CC2)CC1 C1(NC(c2n(CC)ncn2)=O)CCN(C(=O)CCN2CCCCC2)C12CC2 c1(CNC(C(c2cn(C=C)nc2)N(CC(C)CO)C)=O)cccc2ccccc12 C1(NC(c2cccc(F)c2C(F)(F)F)=O)CN(C(c2cn[nH]c2)=O)CCC1C C1(C(C)NC(C2C(C)(CC)C2)=O)CCN(C(c2coc(Cl)n2)=O)CC1 CC1(CNC(C2CC3CC(=O)C2O3)=O)CCCCC1.C1(C)(C=O)CCCCO1.N N1(C(c2[nH]n(C)c(=O)n2)=O)CC2(CC(NC(c3ccc(F)o3)=O)C2)C1 C1(O)(CCNC(C(CC)(C)O)=O)CCN(C(c2cc(Cl)cn2C)=O)CC1 N1(C(CCC(C)(F)F)=O)CCC(NC(C2CC(C(F)(F)F)C2)=O)CC(O)C1 c1(C(=O)NCCCCn2cc(CCC3CCCCO3)nn2)nc2ccccc2s1 Cc1cc(C(=O)NCC(C)(C)CNC(c2ccccc2C)=O)c(F)c(Br)c1 C#CCC(CC(=O)N1CCCC(=C)C1)NC(c1cncc(OC)n1)=O c1(C(=O)NC(CNC(c2c(CC)nccn2)=O)C(C)C)cccc(=O)n1C c1(CC)c(Cl)nc(C2CCC2)[nH]c1=NC1CCCCC1NC(=O)C(C)CN(C)C C(C(C)(O)C(=O)NCC12CC1CN(C(C1CCOCC1)=O)C2)OC c1(CC(=O)N)c(C)noc1C.n1(CC(CC)O)cc(C(N2CCC(C)C2)=O)nn1 c1(C(=O)OC)c(C)cc(C)nc1NC1CN(C(=O)C=Cc2cncs2)C1 N1(C(C(C)OC)=O)CCCC(F)(CNC(C2CC2C(F)F)=O)CC1 N1(C(C(=O)NCC)=O)CCC12CN(C(=O)C(C1CCOCC1)OCC)C2 C1(CC)CNC(=O)CN1C(=O)NCc1ccccc1CN1CCOC(C)C1 C1(NC(C(CSC)(C)NC(c2cc(C(C)C)on2)=O)=O)CC2(CCC2)C1O C(C)(C(CC(=O)NCc1ccccc1F)NC(C12CSCC1C2)=O)OC c1(C(=O)NC2C(C)CN(C(=O)CC3OCCCO3)CC2)cc(F)c(F)c(Cl)c1F C12(C(=O)NCc3scc(CC)n3)CC1CN(C(=O)COc1ccccc1)C2 CCCCCCCCCC(=O)N1CCCC(C(=O)NCC2(O)CCC2)CC1 CCCCCCCC(=O)N1CC(F)CC1C(=O)NC(C1CCC1)C c1(OCCOC)ccccc1NC(=O)NCC1(C(C)OC)CCC1 N1(C(C(C)SCCCC)=O)CC2CCC1C(NC(C13CC(F)C1C3)=O)C2 C(=O)(CC(=O)NC)N(C)C.n1(CC=O)nnnc1C1CC1.C1CC1C=O c1(C(=O)NC2C(CC)CN(C(c3nc(C)n(C)n3)=O)CC2)c(C)cc(O)nc1C N1(C(Cn2ncc(C)c2)=O)CC2CC(CNC(C3(C)CCC3)=O)CC1C2 C1(C(=O)OC)(CC)CCCCN1CC1CC12CC2(F)F N1(C(c2ccc(CC)o2)=O)CC(O)CC1CNC(C1CCO1)=O c1(C(=O)NCC(C)NC(CCc2cccc(C)c2)=O)nsc2ccc(C)cc12 C(=O)(CCCCCCNC(=O)CC1COCCO1)N1CCC(N(C)CC)C1 C(=O)(C1=C(C2CCC2)N(CC)C(=O)NC1c1c(Br)nc(C)n1C)OCC N1(C(CCN(C(=O)C(C(C)C)C2CCC2)CC)=O)CCS(=O)CC1C N1(C(c2c(C)cc(C)c(C)c2)=O)CCC2C(CCCN2C(c2ccoc2C)=O)C1 c1(C(=O)NC(CN(C(=O)CC(C)C(F)F)CC)C)cn2c(n1)CCCC2 CC1CN(C(=O)Cc2cnoc2)CCC1CNC(C1(N(C)C)CC1)=O N1(CC)CCN(C(c2cnn(CCNC(C3CCC(C)O3)=O)c2)=O)CC1 S(=O)(=O)(c1ccccc1Br)NCC(CC)(C)C(C)O.[SH](=O)(=O)C(F)F.CC.N C(CCC(=O)N1CCCC1C1(NC(=O)CN(C)C(C)C)CC1)SC N1(C(C2CCC(=O)NC2)=O)CCN(C(=O)CCc2ccc(Cl)s2)C2(CCC2)C1 C1(C(N(C(C)CO)CC2CCC2)=O)C2CCN(C(C3CS(=O)C3)=O)CC12 CCCCCCC(=O)N1CCC(CNC(c2cn(C3CC3)nn2)=O)C(O)C1 c1(C(=O)NCC2N(C(c3ccc(CCC)[nH]3)=O)CCC2)n[nH]c2c1CCOC2 C(C)(CC(C)CC)N(C(CONC(C1(OCC)CCCC1)=O)=O)C C1(NC(c2cc(CCC)[nH]n2)=O)CC2CCC(C1)N2C(c1cc(C)c(N)cn1)=O C1(CCC)(C(=O)NC)CCCN1Cc1cccc(Br)c1 C(CCC(F)(F)F)ONC(C1(F)CN(C(c2cc(C)on2)=O)C1)=O N1(C(c2ccncn2)=O)CC23CCCC2(C1)CN(C(C1SC2C=CC1C2)=O)C3 N1(Cc2ccc(C)[nH]2)CCC2CN(C(=O)C=Cc3ccc(F)cc3Cl)CCC12 c1(OCCOC)ccc(OCC2CCC2)cc1Br.C(=O)C(O)CC1CC1.N c1(NC(C(CC)(C)O)=O)ccc(OC)c(-c2ccn(C)n2)c1 c1(C(=O)NC(CC=C)CNC(=O)CCn2cncn2)ccc(Br)cc1SC N1(C(c2c(CC)cco2)=O)CCCC(N(C(c2ccn(C3CC3)c2C)=O)CC)C1 CC1(C(=O)NCC(c2ccccc2)CNC(C2CC2F)=O)CC(F)(F)C1 c1(C(N2CCC=C(CNC(C3CC=C(C)CC3)=O)C2)=O)nc[nH]c2ncnc1-2 C(CC(=O)N1CC2CC2C1)(C(F)F)NC(=O)Cc1ccon1 C1(NC(C2CC3CCC2O3)=O)CN(C(=O)CSC2CC2)CCC1O c1(C(=O)NC(CN(C(C2C(=C)C2)=O)C)C)ccc2sc(C)nc2c1 C1(C(N(C(C)C(=O)NCC2CCCCS2)C2CC2)=O)CC(=O)CCO1 CCC(CC(=O)NC1CN(C(c2ncn(C)n2)=O)CC1C(F)F)C(C)C c1(C(N2CCC(CC=C)(NC(=O)C(C)C(C)O)C2)=O)c(C)ncnc1O N1(C(C(CSC)C)=O)C2CCC1CC(C(=O)NCC1CN(C(C)C)CCO1)C2 CC#CCCCC(=O)N1CCC(CNC(c2cnn(C)c2)=O)C1 C(=O)(CCCCCN(C(=O)CCCC(=O)C1CC1)C)N1CCCC(C)C1 CCC(C)(C)CC(=O)NC(C)(C)C1CC1.n1(CC(=O)N)nnnc1C(C)C CC1CCCN(C(=O)CN(C)C)C1CNC(c1ccc(C2CC2)c(F)c1)=O c1(NC(CC2CCCN(C(C(CC=CC)C)=O)C2)=O)ccc(Cl)c(O)c1 CCCCC(C)CCC(=O)NCc1nc(C(=O)NC(C)CS(N)(=O)=O)c(C)o1 N1(C(C2OCC(C)C2)=O)CCC2(CC1)CC2NC(=O)C=CC1CCCC1 Cc1nc(N2CC3CC(C2)N3C(c2cc(F)nc(F)c2)=O)cc(C(F)(F)F)n1 C(=O)(CC1=CCCCC1)NCC(C1N(C(C)=O)CCC1)(C)C.N1(C=O)CCCC1 C1(CSCC(=O)NCCCN(C(C2C(C)=C2)=O)C)CCCCO1 O=C(O)CCCC(=O)N1CCC(n2cc(CSCCO)nn2)C(O)C1 C1(OC)CCC12CC(C(N1CCCC1(C)CNC(=O)CC(C)(C)OC)=O)C2 c1(C(=O)NCC2C(NC(C3CCC(=C)CC3)=O)C2)ccc2c(c1)CCN2C CC(C(=O)N(C)CC1CCCN1C(=O)C=CC(c1ccccc1)=O)C(C)(F)F C1(NC(c2c(C)occ2)=O)CC2CC1CN2C(=O)C1=NNC(=O)C1 CCC(C(=O)N(C(C)(C(=O)NCC1CCCN1C(C)=O)C1CC1)C)OC c1(C(CC)(CC)C(=O)NC(C)CN(C(=O)C(C)CO)C)ccc2c(c1)OCO2 Cc1cc(C(=O)NC(C)CNC(c2ccnn2CC(F)F)=O)nnc1C CC1CCCCN1CCC(=O)NCCOCCN(C(=O)C(C)CC1CCCC1)C N1(C(C2C(C(C)C)C2)=O)CC2C(CC(=O)NCC(C)C3CCC3)C2C1 N1(C(C(CC)NC(c2ccc(C)c(C)c2)=O)=O)CCc2c[nH]nc2C1 c1(NC(Cc2ccn(C)n2)=O)cccc(NC(c2csc(Cl)n2)=O)c1 C(C(C)(C)CNC(C1(C)CC1(F)F)=O)N(C)C(C1CC2CC2C1)=O c1(-c2cn(CC3C(C)(C)CN3c3nnc(C4CC4)s3)nn2)ccc2ocnc2c1 C1(NCc2c(C)n(C)nc2)(CN2CCOCC2CO)Cc2ccccc2C1 N1(c2n(CCCOC)c(C(c3ccncc3)(C)O)nn2)CCc2scc(Br)c2C1 c1(C(=O)NC(CNC(C(C(C)(C)F)(C)F)=O)CO)cn2cccc(Cl)c2n1 CCN=c1ccc(C(=O)NC2CC3(C2)CN(C(c2c(C)nc(C)n2O)=O)C3)c[nH]1 CCC(C)C(C)C.C(C=O)OCCOCC.C1(C=O)(CCN(C)C)CC1 N1(C(C(C(C)C)=O)=O)CCC(C2CC2)C1C(=O)NCCCc1ccncc1 c1(C(N2CC(C(C)NC(=O)CC3COC(C)(C)C3)C2)=O)cnc2cc[nH]c2c1 NC1CCC(NC(c2cnn(C3CNC3)c2)=O)c2ccccc21 C1(NC(C2(C(F)F)CCC2)=O)CCCC(N=c2nc(C3CC3)[nH]s2)C1 C1(NC(NCCSC)=S)CCOC(c2cccc(F)c2)C1 CC1=CCC(C(=O)NC(C)C(C)C(=O)N2CCC(O)CC2)CC1 CCC(C)(O)Cc1cn(CCC(=O)N(C(C)C(=O)NC)C)nn1 N1(C(Cc2cn(CC)nn2)=O)CCOCC(CNC(=O)CN2CCS(=O)CC2)C1 c1ccc(C(C)C)cc1.c1(CC(=O)N)cnnn1C.C(CC)N(C(=O)C)CC O=C(N=c1cc[nH]cc1Cl)NNC(=O)c1csc2ccc(Br)cc12 c1(OC)cccc(C2(C(=O)NCCCCN(c3cccc(Br)c3)C)CCCC2)c1 N1(C(CCN(CC)CC)=O)CC(C)OC2(CCC2)C1.c1(C(=O)N)cc(C)[nH]n1 N1(C(CC(CC)C2CC2)=O)CCN(C(c2ccc(C)o2)=O)CC1C(C)(C)C C1(CCNC(=O)CCc2cscn2)COCCN1C(C12CSCC1C2)=O Cc1c(C(=O)NC2CC2)oc2ccccc12.C(=O)(CCC(C)(C)[N+](=O)[O-])N(C)C C1(C)(C(=O)N)CCN(C)CC1.C1(C(=O)NCc2cc(CC)on2)CCCCC1 C(c1cccc(F)c1)=CC(=O)N(C(C)C)CC.C1(CC(=O)N)CCCOC1 C(c1ccc([N+](=O)[O-])cc1)=CC(=O)N(C)CCNC(c1cc(Br)cs1)=O C1(OCC(=O)NC)CCN(C(=O)Cc2cccs2)C1.c1(C=O)cc(F)c[nH]1 CN(C)S(=N)(=O)NC(c1cc(-c2ccc(F)cc2)no1)=O c1(C(=O)NCc2c(Cl)ccc(C)n2)cc2ccoc2cc1F c1(CNC2(c3n(C(CC)(C)C)nnn3)CCCCC2C)nc2ccccc2n1C c1(CC(=O)NCC(C)NC(CC2CC(OC)C2)=O)ccc(C)o1 C1(C)(NC(C(CC2CCCC2)NC(C2C(C)C2C)=O)=O)CCC(=O)N(C)C1 S(=O)(=O)(c1ccc2c(c1)CCN2C(C1CC(N=[N+]=[N-])C1)=O)N(C)CC N1(C(c2c(C)ocn2)=O)CCCC2(C1)CN(C(C13CC(C)(C1)C3)=O)CCO2 c1(C(N(CC)C)=O)ccc(F)c2c1OCC2.CC1CC(C)C1C(=O)NCCO C1(CC)OCCCC1C(=O)N(C)CC1CC1.C(=O)(C(F)=C(C)C1CC1)N C1(NC(C(CSC)(C)NC(C2CNC(=O)N2)=O)=O)CCN2CCC1C2 C1(NC(=O)C=C(C2CC2)C2CC2)CN(C(c2coc3c2COC3)=O)CC1C1CC1 C(CCC(C)C)(C(=O)NCC1CC12CCC2)NC(C=CC=CCC)=O.C Cc1nn(C)cc1CCC(=O)NC(CC)C(C)C.C1(=CC=O)CCC(C)CC1.N C1(NC(=O)CS(=O)(=O)NC2CC2)CCCN(C(c2ccsc2)=O)C1 N1(C(CS(CCC)(=O)=O)=O)CC(NC(=O)C(CC)SC)Cc2ccccc21 Cc1csc(=O)n1CC(=O)N.C1(C=O)C(c2nc(=N)[nH][nH]2)C1(C)C.CC(F)C c1(C(N(C(CC)C(N)=O)CCC)=O)cc(O)ccc1OC c1(C(=O)NCC(CNC(C2CC(C)(C)O2)=O)O)cc2c(cn1)OCCC2 c1(C(N2C(C)(C(=O)NC3(C=C)CCC3)C=CC2)=O)ncnc(O)c1F c1(OC)cc(C=CC(=O)NC2CCC(C)(C)C2)ccc1F.c1(C=O)ccoc1 c1(C(=O)NC2C(CC(=O)N(CC(C)OC)C)C(O)C2)cccc2ccoc12 C1(CNC(CN(CCC)C(C2CCOC2)=O)=O)CCCC2(CC2)C1 c1(C(=O)NCCN(C(C(CC)Oc2ccccc2)=O)C)ccc2c(n1)NCCO2 C1(=CC(=O)NCC2N(C(C(CC=C)C)=O)CC2)CC2CCC(C1)N2C c1(C(=O)NC23C(CN(C(C(C)C(F)(F)F)=O)C2)CC3)cc2ccc(O)cc2n1C c1(CC)cc(N)c(C(=O)NC2(C)CCOCC2)cc1F.C(=O)(C)N.C(C)=O C1(C(N2C(CC)CN(C(c3ncn(C(C)C)n3)=O)CC2)=O)CCn2nncc2C1 Cc1cc(CC(=O)NCC2CC(C(=O)NC3C=CCCC3)CO2)cs1 C1(F)(C(=O)NCC(CO)NC(=O)CC2(O)CCC2)CC12CCCCC2 Cc1ccc(C=CC(=O)NC2CCC(O)C2)cn1.C12(C=O)CCCN(CC1)C2.N N1(C(C(CC=CC)C)=O)CC(C(=O)N(CC(C)O)C)CCC1(C)C c1(C(=O)NCC(CN(C(CC(C=C)CC)=O)C)O)c(C)cc(C)c(Br)c1C C1(OC)C=CCN(C(c2c(-c3ccccc3)nnn2C)=O)C1 N1(C(=O)CC2C3CCC(C3)N2C(=O)CCCc2ncco2)CCC(C2CC2)CC1 C=C1Cn2c(C(=O)NCCCOCC)nnc2S1.C1(CC(=O)N)CCCCC1F C#CC1CCCN1C(C1COCCN1C(C1COCC(C)O1)=O)=O c1(OC)nn(C)cc1C(=O)NCCCCC(C)NC(=O)C(O)C1CCCC1 c1(CC(=O)NC2CCC(NC(c3cnsc3)=O)C2)ccn(C2CCCC2)n1 C1(CNC(C2C(C=C)C2)=O)(NC(=O)C(C)CC(C)C)CCC(C)(C)CC1 N1(C(c2cnc(CC(F)(F)F)s2)C(=O)N2CCCC2)CCN(c2ncncn2)CC1 C(=O)(C(C#N)C(C)C)NC1CCN(C2CCN(C(c3scc(C)c3)=O)C2)CC1 CC(CC(=O)NCCNC(=O)C(O)c1ccco1)c1ccncc1 C(C(C)C(F)C(=O)NC)NC(c1c(C(C)C)noc1)=O.c1cn(C2CC2)nn1 C(CNC(c1cncnc1)=O)(C(=O)N1CCCC1C1CC1)OC N1(C(C(CNC(C(C)(C)OC)=O)N(C)C)=O)CC(CO)CC1C c1(C(=O)NCCC2CCN(C(C(COC)C)=O)C2)cc(N)cc(N)c1 CC(C)C(C)C(CNC(c1ccc(Cl)cc1)=O)NC(=O)CCCC1CCCCC1 C1(CC(=O)N(CC(O)CO)C)COCCN1C(=O)Cn1[nH]cnc1=N C(=O)(C(O)CCSC)NCC(CC)NC(C1(Cc2ccccc2)CCCC1)=O CC1(F)CC(C(=O)NCC2CCN2C(=O)COC2(C)CCCC2)C1 CCC(F)(F)CC(=O)NC(CNC(c1cccc(Br)c1Cl)=O)C1CCC1 CC(C)CC(C(=O)NCCC1(O)CCN(C(=O)C2=NOC(C)(C)C2)C1)C(C)C C1(C(C)NC(=O)Cc2cccn2C)CCCN(C(C2CSCCS2)=O)C1 c1(C(=O)NCCC2CN(C(c3cn(CC)nn3)=O)C2)c(C)cc(C)cc1N CC(C)CC(=O)NC(CO)C(=O)NCCCOC(=N)O C(=O)(CCCC(C)c1ccccc1)N1CC(C(N)=O)C1.C=C1CC(C(=O)NC)C1 c1(OC)ccc(C2CCN(c3nnc(CCc4ccsc4)n3C)C2C)cc1F C1(N(C(CC(CC)C2CCC2)=O)C)CN(C(c2sc(C)c(C)c2C)=O)CC12CC2 c1(C(=O)NCC(C(=O)N2CC(F)(C(=O)OC)C2)(C)C)c[nH]c2cccnc12 Cc1cc(Cl)ccc1OCC(=O)N(C(C)C)C.C1(CC(=O)N)CC(C)(C)C1 c1(C(N(C)CCN(C)C(C2CC23CC3(F)F)=O)=O)cc2cccc(O)c2[nH]1 N1(C(=O)C(=O)N2CCC2c2cn(CCCF)nn2)CCC(O)C(CO)C1 c1(C(=O)NCC(CN(C(C2C(C)C2)=O)C)O)cccnc1S c1(C(N(CC(C)NC(C2COC(=O)N2C)=O)CC)=O)cccn2ccnc12 C(=O)(C1=C(C)OCCS1)N1CC2C(NC(c3c(CC)noc3)=O)C(C2)C1 Cc1ncc2n1CC(C(=O)NCC1CN(C(c3cocn3)=O)CC1(C)C)CC2 C1(Cn2cc(NC(CC(CC)OC)=O)nn2)CC2CCC1N2C(=O)CCC(C)(C)O C(=O)(C(F)C(F)(F)F)NC1C(C(N(OC)Cc2ccccc2)=O)COC1 N=c1nc(CCC(=O)NCC2CC(C)C2)[nH][nH]1.C1(O)(C(C=O)F)CCCC1.N c1(C(=O)NC2(CCCNC(C(C)O)=O)CC2)ccc(-n2cccn2)cc1 CC1=NS(=O)(=O)N(C)C=C1C(=O)N.C1(CCC)CCCN1C(C1CC2CC2C1)=O CCCC(C)CC(=O)N1CCN(C(=O)CCc2cnccn2)CC1C1CCC1 C1(n2cc(CC)nn2)CCN(C(=NCC(C)(C)C2(O)CCC2)NC(CC)CC)C1 C(=O)(C1=C(C)OCC1)N1CCC2C(NC(C(CCSC)O)=O)C21.c1ccccc1.C Cc1cc(C(N2CCC(C(=O)NC3CC4CCC3O4)C2)=O)cnc1F Cc1nc(C(=O)NC2CCCCC2NC(c2csc(S)n2)=O)ccc1[N+](=O)[O-] C(C(C)(O)C(F)(F)F)NC(CCC1(C)CN(C(c2ccc(F)c(F)c2)=O)C1)=O C1(C(C(=O)NCCCC)N(C2CCCC2)Cc2ccc(Br)s2)CCSCC1 C(C)(C(=O)NCCC1CC(NC(=O)CC2CSCCS2)C1)(C1CC1)OC C#CCC(CC(=O)N1CCC(OCC)C1)NC(=O)C(c1cccnc1)C1CC1 c1(C=O)cnc2ccc(C)cc2c1.C1(O)(CC#C)CC(C(=O)N(C(C)C)C)C1.N c1(C(N(C2CC(NC(c3c(-c4nc(C)sc4)c[nH]c3)=O)C2)C)=O)c[nH]c(C#N)c1 C1(CC)C(C(=O)N(C2CCN(C(C3(CF)CC3)=O)C2)C)CCN1C N1(C(C#CC(C)(C)C)=O)CCC2(CCCN(C(c3cnc(Cl)s3)=O)C2)C1 C(C(=O)NCCOCc1ccccc1)(C(C(C)C)C(C)C)N1CCC(C#C)(O)C1 C1(C(C)C(=O)N2CC=CC2)CCN(C(=O)COCC2CC2)C1 C1(C=O)C2CC(=O)CC12.C1(CC=C)(C(=O)NCC2CCCC2)CCCC1.N C=CCCCCC(=O)NCCN(C(=O)C(c1cccc(OC)c1)(F)F)C C1(CC(=O)NC(CCC)C)C2CN(C(c3c[nH]c(=S)cn3)=O)CC12 C(=O)(CC1=CCN(C(C2COC(=O)N2)=O)CC1)NCc1scc(C)n1 Cc1c[nH]c(C#N)nc1=NC(CNC(=O)C(N1CCCC(O)C1)C)C(C)C Cc1csc(C(=O)NCCCNC(c2sccc2C(F)F)=O)c1Cl C(=O)(C(C)(O)CC(F)(F)F)N1CC(C2(NC(C3CCCC(C)(C)C3)=O)CC2)C1 CN1CCOC(C(=O)NC2CC(Nc3nccc(-c4cnccn4)n3)C2)C1 N1(C(C(C)(C)C#N)=O)CC2CCC(C1)N2C(=O)C(c1cccc(Cl)c1Cl)(F)F N#Cc1c[nH]c(C(=O)NCC2CN(C3CCN(C4CCC4)C3=O)CCO2)c1 c1(C(=O)OC)ccc(F)c(OCC2CCON2C(=O)OC(C)(C)C)c1 c1(C(C(=O)NCCNC(C(Cn2ccc(C)n2)C)=O)O)ccc(F)c(F)c1 C#Cc1cc(C(N2CCCC(C)C2CCNC(=O)CCC(C)(F)F)=O)ccc1C C(=O)(C(C(C)OC)NC(c1cnn(C2CC2)c1)=O)N(CCOC)C N1(C(c2cc(OC)nn2C)=O)CCC2CCCC12C(=O)NCCO.CC(C)C C1(CNC(c2ccc(COC)cc2)=O)CN(C)CCN1C(c1cnsc1C)=O c1(SC)ccccc1C=O.C1(C(N(C(c2ccccc2)C)C)=O)CCS1(=O)=O.N C(C(=O)NC1CCC(CNC(=O)Cc2ccncc2)C1)(C(C)C)OCC N1(C(CCCCC(=O)NC)=O)CCC2CN(C(c3ccc(=N)[nH]c3)=O)CCC2C1 Cc1cc([N+](=O)[O-])ccc1C(N1CC2CCC2(NC(=O)Cn2ncnn2)C1)=O C(CCC)(C(=O)NCC(N1CCN(C(=O)CN2CCC2C)CC1)C(F)F)=CCC C1(CNC(CC2(C=C)CCC2)=O)CN(C(=O)CSC)CCC1C(F)(F)F C(=O)(C1=CCN(C(=O)C(F)=CC2CC2)CC1)NCC1(CC)CCCO1 CC1(CNC(c2ccnnc2)=O)CCCN1C(C1CC2CC2C1)=O N1(C(C(C)SCCCC)=O)CC(C(=O)NC2(CO)CCC2)C(C(C)C)C1 c1(C(N2CCC(O)(CNC(C(C)(C)F)=O)C2)=O)ncc2cc(Br)ccc2n1 c1(C(=O)NCCC(C)F)cccc(-n2cccn2)n1.C1(C[SH](=O)=O)CC1(C)C c1(NC(=O)N(CCO)CCN2CCCCC2)nc2c(F)ccc(Br)c2s1 Cn1c([N+](=O)[O-])cnc1C(=O)NC1CCN(C(c2coc(C(F)F)n2)=O)CC1F C(CC(C)N=c1[nH]c2c(c(=NCCC3CCCC34CC4)[nH]1)CSC2)SCC C(C(C)(C)C)N(C(=O)C=Cc1cc[nH]c1)C.c1(C2C(C(=O)N)C2)cn[nH]c1 C1(NC(C2CCC(O)CC2)=O)CN(C(C23CC(F)(C2)C3)=O)CC1O c1(CC)ccc(F)c(C(=O)NC(C)(C)CCNC(c2cc(OC)cs2)=O)c1 N1(C(CCCCN(C)C)=O)CCC(NC(c2cccs2)=O)C2(CCC2)C1 c1(OC)ccc(C(=O)N(CCCNC(c2cc(CC(C)C)[nH]n2)=O)C)c(O)n1 CC1(F)CCN(C(=O)C(=O)NCCC2CCCC23CC3)C1 C(=O)(CCNC(=O)CO)NCCN(C(COCCOCC)=O)C c1(C(=O)NC2CCN(C(C(CC=C)CC)=O)C2)ccc(S(N)(=O)=O)s1 c1(C(N(C)CC2(O)CCN(C(C(CC=C)(C)O)=O)CC2)=O)ccc2c(c1)COC2 n1(CCOC)c(N)c(C(=O)CN2CCC(N)CC23CC3)c(O)nc1=O C(=O)(C#CC1CCOC1)NC(CN(C(C(N1C(CC)CCC1)=O)=O)C)(C)C C(=O)(C(C)CC(C)(C)C)NC(C(=O)N(CCCOC)CCO)CCC1CC1 N1(C(CCOC2CN(C(C(C)(C)C#N)=O)C2)=O)CC2(CCCCC2)C1 C1(C(N(C)Cc2ccn(CC)n2)=O)CCCCC1.C1(C(=O)N)CC1C(F)F CC(C)CC(C)C(=O)NC12COC(C)(C1)C2.c1(C=O)cc(C2CC2)ccn1.N c1(C(CN(CC(OCC)OCc2cccnc2)C)=O)ccc(OC)cc1 C1(CC(N2CC(CN(C(COCC(C)C)=O)C)C2)=O)CC2CC2C1 Cc1ccccc1-n1ncc(C(N2CC(O)CC2CNC(=O)C=CBr)=O)c1C Cc1c(O)c(=O)ccn1CC(=O)NCCC(C)NC(=O)CC1CCC1(C)C C1(CCNC(CC(=O)OC)=O)CN(C(=O)CC(C)N(C)C)CC1C C1(NC(CC2CC(=C)C2)=O)(COC)CCCN(C(C2CC(CC)(C)C2)=O)C1 c1(OC)ccccc1OCC(=O)NCc1ccccc1OC(c1ccccc1)C C1(CNC(C2CC(OCC)C2)=O)CC(C)N(C(c2ns[nH]c2=O)=O)C1 c1(NC(c2ccc(C)cc2[N+](=O)[O-])=O)cccc2c(C(=O)O)cccc12 CCC(CCC(=O)NC1CN(C(c2cc(Br)cn2C)=O)CC1C)OC CCCC(CNC(=O)C(C)(C)C(F)F)C(=O)NCCN1C(=O)CCC1=O c1(C(=O)NC(CN(C(C(C)SC)=O)C)(C)C)ccc(SC)c(Br)c1 Cn1ncc(C(=O)NCCC2(C(=O)NCC3CNC(=O)CO3)CC2)c1C#N C1(F)(CNC(CC(C)OC)=O)CCN(C(=O)COc2cccc(F)n2)CC1 c1(C(N2C(CNC(c3cc(Cl)ncc3Cl)=O)CC(F)C2)=O)ccc2sccc2c1 C1(C)(C(=O)NCCc2nccc(C)n2)CC(O)CN1C(=O)CC1CCSC1 CN1C(=O)OCC1C(=O)NOCCN(C)C.C1(CCNC=O)(SC)CCC1 C1(C#N)(C=O)CC12CCCC2.Cn1nc(C(F)F)cc1C(=O)N.CCC1CC1 C1(CC)C(NC(=O)C(=O)C(C)(C)C)CCCN1C(c1cnn(CCO)c1)=O C1(F)(C(=O)OC)CCN(N2CC(=O)N(C)CC2C)C1 CC1CCN(Cc2ccccc2C(F)(F)F)CC1NC(c1cc2c(s1)CCC2)=O c1(C(=O)NC(CNC(C2(OC)CCC2)=O)(C)CO)cc(N)ccc1O c1(C(N(CCOC)Cc2cnn(C)c2)=O)cnn2cc(OC)ccc12 CC1COCC(C(=O)NC2CCCCC2C(=O)NC(CC2CCCC2)CO)O1 c1ccccc1.CCCCNC(=O)C=CC=O.C(=O)CC=CC(C)(C)C.N C12CCC(CC1)N(C(C1CC3(C1)CC3(F)F)=O)C2.Cc1cc(C(=O)N)nc(O)n1 C(=O)(C(C(C)CC)NS(C)(=O)=O)OCCNC(CC=C)=O N1(C(c2c(C#N)scc2)=O)CC(NC(=O)CCn2cncn2)C2CCCCC12 c1(C(c2n(CC(=C)C)nnn2)NC(C)C(N)=O)cc(F)cc2c1CCC2 N1(C(C(CC)SC)=O)CC2C(CNC(=O)C(C)Cc3ccccc3F)C2C1 C1(CNC(CCCn2c(C)ncc2)=O)CCCN(C(=O)CCOC2CCOC2)C1 N1(C(C(C2CCCOC2)OCC)=O)CC2CC(NC(=O)CCC3CC3)CC2C1 C1(NC(Cc2cc(C(=O)OC)sc2)=O)CCCCCN(C(C2CC2F)=O)C1 Cc1coc(C)c1C=CC(=O)NCC1C=CCN1C(=O)CC1CCC(=O)N1 C(=O)(CC(C)N=c1[nH]c2c(c(=NCCCN3CCCOC(C)C3)[nH]1)SCC2)NC c1(C(N2CC(CC(C)NC(C3(C4CC4)CCC3)=O)C2)=O)c(F)cncc1Br C1(C(N2CCN(C(CN(C)C(c3cnn[nH]3)=O)=O)CC2)=O)CC2(CCCC2)CO1 C1(NC(C2C(C)C2(F)F)=O)C2CN(C(C3CCCO3)=O)CC12 c1(C(=O)NC2(CO)CCN(C(CC3CC(=C)C3)=O)C2)ccc2c(c1)[nH]c(=N)n2C c1(NCC2C(C)CNCC2)ccc2c(c1)C(=O)OCC2 n1(CC=CC2CC2)cccc1C=O.c1(C=O)ncnn1C1CCOCC1.CC C(C(=O)NC1CCC(O)C1)(C(C)C)NC(C(C)=C1CCC1)=O c1ccc(CC)cc1.O(CP(C)(C)=O)CC=O.C1(C(C)C)(C(=O)N)CCC1.C c1(C(C(=O)NCCC)N(CC(=O)N)CCC)ccc(C)c(C)c1F.C(C)CC c1(C(=O)NC(C(=O)NCCCC2C(C)C2)C2(O)CCC2)cc(=O)cc[nH]1 C(c1cccc(Cl)c1)=C(C)C(N1CCC(N(C(=O)CCC(C)C)C)C1)=O CN1CCCCC1CCn1cc(CCCS(C)(=N)=O)nn1 c1(C(=O)OC)cc(Cl)c(NC(N2CC(C(OC)OC)C(F)C2)=O)c(Cl)c1 N1(C(C2C(C#N)C2)=O)CCC2CN(C(c3cn(-c4ccccc4)nn3)=O)CC12 C1(CC(=O)NCCCCNC(=O)C=CCF)CCCCC1O N1(C(c2cccc(N(C)C)n2)=O)CCC2CCCC12CNC(=O)C(C)(C)F c1(NC(C2(O)CCN(C(CC(CC)O)=O)C2)=O)cnc(Cl)c(C#N)c1 C1(C(=O)NC(CC(=O)NC23CC(C2)C3)CC2CC2)Cc2nccn2C1 Cc1nc(C(N2CCC(N3CCC(NC(C4CCOC4)=O)CC3)CC2)=O)n(C)n1 CCCC(CCC)CC(=O)N1CCN(C(c2cscc2OC)=O)CCC1C Cc1nc(C)c(CNC(=O)CC2CCCN2C(=O)C(C)Cn2cccn2)o1 C(=O)(C(C)CC(C)(C)C)N(CC(CNC(CC1(OCC)CC1)=O)C)C Cc1cc(-n2cccn2)nc(=NCC2CC(C)N(C(c3cc(Cl)c(Cl)[nH]3)=O)C2)[nH]1 C1(NC(c2cnc(CCC)s2)=O)CN(C(=O)C(C)C)CC1c1ccnn1C C1(O)(CNC(C2C(C)(C)C2)=O)CCCN(C(C2COCCN2C=O)=O)CC1 N1(C(C2C(NC(C(C)C3CCC3)=O)CC2)=O)CCOC(C2(C)CC2)C1 c1(C(=O)NCC23CC(CN2C(c2ccncc2)=O)C3)ccc2ncc(Br)n2c1 Cc1csnc1C(=O)NCCCN(C(=O)CNc1cccnc1)C(C)C c1(C(=O)NC2(C(=O)NCCSCCO)CCSC2)ccc(Cl)cc1 C1(CC)CN(C(C2CC(C)CN2C(c2cnc(Cl)n2C)=O)=O)CCS1 C1(NC(C2N(C(COc3ccn(C)n3)=O)CCC2O)=O)CCCC(O)C1O N1(C(C2(C#C)CN(C(c3ccn(CC)n3)=O)C2)=O)CCC(CO)C(O)C1 N1(C(C2N(CC)CC2)=O)CCC2(CC1)CC(F)CO2 C(=O)(C1=CSCCO1)N1CCC(CNC(CCOCCOCC)=O)C1 C#CCCCCCC(=O)N1CC2CC2(CNC(c2c(F)cncc2Cl)=O)C1 c1(C(N2CC=C(C(=O)N(CC(C)(CO)CO)C)C2)=O)c[nH]c2ccccc12 CN=c1[nH]cc(C(=O)N(C)CCC2CCN(C(c3nn(C)nc3C)=O)CC2)o1 Cc1csc2nc(CN3CCCC3CNC(C3CCC34CCCC4)=O)cc(=O)n12 Cc1cnc(C=CC(=O)N(C(C)C)C)[nH]1.c1(CC=O)ccc(C2CC2)cc1.N C(=O)(C1=CCCCC1C)N1C2C(C(=O)Nc3c(C)csc3)C(C2)C1 N1(C(=O)CC2CCCCN2C(c2ccc(F)s2)=O)CCC(C2=NOCC2)C1 N1(c2ncc(C)cn2)CC2CC1CCC2NC(c1cnn(C)n1)=O c1(NC(=O)NCC(=O)NC(C)CC)cccc(Cl)c1.c1(C=O)cscn1.N Cc1cccc2[nH]c(C(=O)N(CC(C)N(C)C(C3CC4CCCCC34)=O)C)cc12 c1(C(N2CC=CC(NC(CCC=CC(C)C)=O)C2)=O)n[nH]c2c1CS(=O)(=O)CC2 N1(C(COCC(C)C)=O)CCCC2(CCN(C(=O)C(C)C3=CCCC3)CC2)C1 C12(NC(C(c3ccccc3)NC(C)=O)=O)CC(C1)N(C(=O)C(F)(F)CO)C2 c1(C(N2CC(NC(c3c(C)nc(C)o3)=O)C2)=O)cc(S(C)(=O)=O)ccc1C C=C(C)CC(C(=O)N1CC(O)CC1CC(=O)Nc1cccc(CC)c1)OC N1(C(C(C(CC)CC)C)=O)CC2(CCOCC2)CC1CNC(c1csc(O)n1)=O c1(CC(=O)NC2CN(C(C(C)(C)CC3CC3)=O)C2)ccc([N+](=O)[O-])cc1F C1(NC(CC(C(=C)C)O)=O)CC2CCC(C1)N2C(c1[nH]c(C2CC2)nc1C)=O C1(NC(C2CC(SC)C2)=O)CCN(C(c2ccsc2Br)=O)CC1CO C1(CNC(C=NOC)=O)CC(C)CN(C(=O)C(c2ccccc2)O)C1 C(=O)(C1=CC2(CCOC2)C1)NC1(C)CC(NC(C2=C(C)CCC2)=O)C1 Cn1cncc1CN1CCCC1C(=O)NCCN=[N+]=[N-] N1(C(C(C(C)C)C)=O)CC2CN(C(=O)Cc3ccccc3[N+](=O)[O-])CC2(C)C1 C(=O)(C(C)CCC(C)(C)C)N1CC(C(N2CCOC(C)C2(C)C)=O)C1 C12(CC(=O)N)CCC(CC1)CC2.N1(C(C2C(C)(C(F)F)C2)=O)CCCC1C C(=O)(C(C)(C)CO)NC1CC(OCC(=O)NCC2OCC(C)C2)C1 N1(C(C(C(C)C)SC)=O)C2CCC1C(NC(c1cc(C)cs1)=O)C2 C#CCCCCCC(=O)NC1(CNC(=O)CN2CCCC(N(C)C)C2)CC1 c1(SC)nc(C(=O)N(C2CCN(C(C3(CF)CC3)=O)CC2C)C)c2ccccn12 c1(C(=O)OC)ccc2c(c1)CCC(C)N2C(c1ncc(C2CC2)o1)=O C1(CC)C(NC(=O)C#CC(C)(C)O)CCCN1C(C1CCCCN1CC)=O c1(C(N2CCC(C)(NC(=O)CCc3cocn3)CC2)=O)cc2ccccc2o1 N1(C(CCCOC(C)=O)=O)CCCC(C)(C(=O)NCCc2n[nH]c(C)n2)C1 C1(CNC(c2ccoc2C2CC2)=O)COCCN(C(c2ccco2)=O)C1 CCCC(C)(O)CC(=O)NCCC1CC(NC(=O)CCOC2CCOCC2)C1 C(=O)(C(C)(C)CCF)N1CCC(CCC(=O)NCC2CC(N(C)C)C2)CC1 c1(C=O)cc(Cl)ccn1.c1(C(=O)NCC(C)OC)cc(C(F)(F)F)on1.N c1(CC)cc2c(N3CCC4(NC(c5cc(CC)[nH]n5)=O)CCCC34)ncnc2s1 C1(N(C(=O)CCC2CCN(C)C2)CCOC)CCN(C(=O)C(C)O)CC1 CCCC(CNC(=O)C=CC(C)C)C(=O)NC1CC=C(C)CC1 Cc1cc(C(=O)NC(C)(CNC(=O)CCc2cnn(C)n2)C2CC2)ccn1 N1(C(CCC)=O)CCOC2CN(C(c3ccc(C(F)(F)F)c(Cl)c3)=O)CC12 C1(C(=O)NCc2onc(C)n2)CN(C(C2CCC2CN)=O)CC12CCC2 C(=O)(CC(C(F)(F)F)n1ccnc1)NCCCNC(C(C=C=C)C)=O CC1CCC(=CC(=O)N(CCCCNC(=O)C2=CCC2)C)C1 CC1CN(C(=O)CN2CCCC2)CC1NC(=O)Cc1cncc(Br)c1 C1(CNC(C=CC(CC)C)=O)CC2CC2N1C(c1ccncc1)=O.CC(F)F c1(C(N2CCC(CNC(c3n(CC)ccc3)=O)C23CC3)=O)cccc2nncn12 C#CC1CN(C(=O)C(C2CCOCC2)C)CCN1C(=O)COC1(C)CCC1 CC1CN(C(c2nncs2)=O)CCC1N(C)C(c1cc(C(F)F)cs1)=O C(c1c(F)cccc1F)=CC(=O)NCC12CC1CN(C(=O)Cc1ccoc1)C2 C(CCN(C)C)(C(=O)N(CC(N1CCCC1)=O)C)NC(c1c(C)cns1)=O C1(C(=O)NOCC(C)(C)C)(CCC=C)CN(C(=O)Cc2ccns2)C1 N1(C(=O)CCc2ccc(Cl)s2)CCC2(CCCN(c3ncnc4ccsc34)C2)C1 c1(C(N(CCN(C(C(C)=C(C)C)=O)C)C)=O)cccc2nc(C)sc12 CC1(C)CC(C(=O)NCCC2CN(C(c3ccncc3N)=O)CCO2)C(C)(C)O1 Cc1cc(=O)c(C(N2CCC(C(=O)NC3(C)CCCC3(F)F)CC2)=O)c[nH]1 CC1CCC(F)(F)CN1C(=O)C(c1ccccc1)NC(=O)C=Cc1nccs1 C1(C(N(C(C)C)CC)=O)CCC(F)(F)C1.C1(C(=O)N)CCCN1c1nccs1 N1(C(C(C)(C(C)C)OC)=O)CCC2(CC1)CN(C(C1CCC1)=O)C2C(C)C.S Cc1nc(NC2(CO)CCCN(C(=O)C(F)OC(F)(F)F)C2)c(Cl)cc1[N+](=O)[O-] c1(OCC)nc(C(N2CC=CC2)=O)co1.c1(CC=O)ccon1.C1CC1.C CC1CN(C(C2CC(O)C2)=O)CCC1N(C)C.C1(C(=O)N)COCC1C(N)=O c1(C(C)=O)ccsc1C(=O)NCC(C)N(C)C(C1CCCCO1)=O C1(C(C)C)CN(C(=O)CCC2CC2)CCCN1C(=O)CN1CCn2nccc21 CN(C)NC(=O)CCC(=O)N(C)CCN(C)C(c1cnn[nH]1)=O C1(C(=O)NC2(C)CN(C(c3ccc(C(C)=O)[nH]3)=O)C2)CN(C)CC(C)O1 C1(C(N(CCO)CC)=O)CC(O)C(O)CC1CNC(C1(C)CCC1)=O CCCCC(C)CCC(=O)N1CCC(C)(CC(=O)NCCOC2CCCCC2)C1 C1(N(C(C2C(COC)(C)C2)=O)C)CCCCC1.C(c1cnc[nH]1)=CC=O C(=O)(CC(C)CC(C)C)N1CCN(CCCNC(C(C)N(CC)CC)=O)CC1 c1(C(N(C2CCN(C(C3(CC)CCOC3)=O)C2)CCO)=O)cc2ncccc2s1 C(=O)(N=c1c(Cl)c[nH]cc1Br)C1(F)CN(C(c2c(Br)cncc2Br)=O)C1 C1(NC(CSCc2cccc(C)c2)=O)CN(C(C2CC2C#N)=O)C2(CCC2)C1 c1(C(N(CC(=O)NCC(O)C(C)C)CCC)=O)cccnc1O C#CCC(C(=O)N(CCC)C)NC(=O)COCCOC1CCCCC1.CC.O N1(C(C2SCCS2)=O)CC(F)CC1CNC(=O)C(F)(F)c1cnccn1 N1(C(C2(F)C(C)C2)=O)CCCC(NC(=O)Cn2cc(C3CC3)nn2)CC1 c1(CC)ccc2occ(C(N3CCC4C(NC(=O)CCc5cn[nH]c5)C34)=O)c2c1 N1(C(c2cc(C)no2)=O)CCC(CC(=O)NC(c2nc(C)oc2C)C)C1(C)C c1(C(=O)NCC(C)C)ccc(P(C)(C)=O)o1.C1(C)(C=O)CCN(C)C1=O.N Cc1cc(C(=O)NCCN(C(=O)CC(C)C(F)F)C(C)C)cc(=O)n1C C#Cc1ccc(C(=O)NCCCN(C(=O)CCCN2CCCC2)CC)cc1C C(=O)(C=C1SCC(=O)N1C)NC(CCCCNC(CC1(CC)CCC1)=O)C C1(C2CC2)(OC)CCC1.C(=O)(C(C)N(C)C)N.N1(C2(C=O)CC2)CCCC1 S(=O)(=O)(C1CCCC1C)NCc1cccc(NC(C(C)C)=O)c1 c1(C(=O)NCC(CNC(c2c[nH]c(Br)c2)=O)O)cc2ccsc2[nH]1 N1(C(CC)=O)CCC2CC2(NC(=O)Cc2ccc3nn[nH]c3c2)CC1 c1(C2C(C(=O)NCC34C(CN(C(c5ccon5)=O)C3)C4)C2)ccc(F)cc1F c1(C(C)C)ccccc1CC(=O)NCC1CC1.C1(C)(C=O)CCC(=O)C1.C c1(OC)c(C(N2CC(C)(C)OCC2C)=O)cc(Cl)cc1C.C(=O)CN(C)C.N CC1(C)C(C(=O)NCC(F)(F)C(N)=O)CCN1C(=O)CC1CCC(O)C1 C1(C(N2CCCC(=C)C2)=O)CN(C(=O)CC(C)N(C)C)CC(C)(C)C1 C(=O)(C(C)(C)CCC(=O)N1CCN(C(c2cnc(C)nc2OC)=O)C(C)C1)OC C1(CNC(CC(C=C)c2ccccc2)=O)CCN(C(=O)CSC(F)F)C1(C)C c1(SC)ccc(C=CC(=O)NCC(C)NC(=O)CN2CC3CC3C2)cc1 N1(C(CC(C)O)=O)CC=C(CC(=O)N(CC(O)CO)C(C)C)CC1 N1(C(C(C)CC2CCCC2)=O)CCC(N(C)C(C2(CO)CCC2)=O)CC1 Cn1cnc(C(N2CCC(F)C2)C(=O)NCC2CCOC2)c1Cl C1(C(=O)NCCn2ccnn2)(OC)CCC(C)C1.c1(CC=O)cccnc1.C Cc1cccc(C(=O)NC2COCC2CNC(C2C(C)C2C)=O)c1Cl c1(OCCC(N2CCC(O)C2)=O)cc(F)cc(F)c1.C1(Cl)(C(=O)N)CC1(F)F C(=O)(CCO)OC.C1(C)(CCC=O)CN(C(=O)CC2CC(N(C)C)C2)C1.N N1(C(C=CC=CC)=O)CC(CCNC(c2cc(=O)cc[nH]2)=O)OC(C)C1 c1(C(N2C(C(C)NC(=O)CCc3cnn(C)n3)CCC2)=O)ccccc1[N+](=O)[O-] CC1CCC(O)(C=O)CC1.C1(C(F)F)CCN(C(C2(C(F)(F)F)CC2)=O)C1.N c1(C=O)nn(C)cc1S(N)(=O)=O.N1(C(C2N(CC)CC2)=O)C2CCC1CCC2.N C1(C(=O)NCC2CC(NC(CCCC#N)=O)C2)CN2CCCN1CC2 CC1CC(NC(=O)Cn2cnnc2)CN1C(c1sccc1C(F)F)=O C(=O)(C(C(C)C)Oc1ccccc1Br)NCC=CC(CC)C N1(C(c2c(C)scc2)=O)CCC(C2(NC(c3cc(C4CCC4)nn3C)=O)CC2)C1 N1(C(CCC#CC)=O)CCC(C2CCN(C(=O)CCc3ccc(F)c(F)c3)C2)C1 C1(CCC#C)CCCN(C(C2CN(C(=O)Cc3cncs3)CC2OC)=O)C1 C1(C(=O)NCc2ccc(CNC(C(C)C)=O)cc2)Cc2cc(Br)cnc2C1 C(c1ccccc1)=CC.N1(C(C(=O)NC)C2CCC2)CCCCC1 C(=O)(C1=CCOCC1)N(C)CCn1cc(CNC(=O)C=CC(N)=O)nn1 N(C1CC2(CN(C(=O)CC3(C)CC3)C2)n2ccnc21)C(CC1CCN(C)C1)=O N1(C(CCCCCCNC(C(CC=C)NC(C)=O)=O)=O)CCN2C(=O)OCC2C1 n1(CC)nnnc1C(c1cnc(C(C)(C)C)s1)NCC(C)N(c1ccccc1)C c1(C(N(CC(C)(C)NC(c2nc(C)nc(O)c2)=O)C)=O)cnn2c1C(C)CCC2 c1(OC)ccc(I)cc1NC(C1CCCN1C(=O)CC1CC2CCC1C2)=O N1(C(C(C)OC)=O)CCC2(CC1)CC(C)N(C(c1ccnc(C(C)C)n1)=O)C2 n1(CC(C)N(C(C2CCN(C)S2(=O)=O)=O)C)ncc2ccccc12 C1(NC(C2C(CC)OCC2)=O)CN(C(c2ccc(CN3CCCC3)o2)=O)CC1 N1(C(Cc2cn(CC)nn2)=O)CC2CC(NC(=O)CS)C(C2)C1.c1nccn1C c1(NC(C2(O)CCN(C(c3cc(CC)on3)=O)C2)=O)cnc2c(O)cccc2c1 c1(N(CC(C)C(F)(F)F)C)nc(N(C)CC2(CO)CC2)c2c(n1)CCS2 c1(-c2c(Cl)nc(OC)s2)ccc2c(O)nccc2c1 C1(C(N)=O)CN(C(=O)C=Cc2ccccc2)CCC1.C1(CC(=O)N)CCC2CC12 c1(C(N2CCN(C(C(C(C)C)O)=O)C(C(C)C)C2)=O)cc2cc(F)ccc2o1 C(=O)(C1=NOC(C)(C)C1)N1CC(NC(C(CC(C)C)C)=O)C(F)CC1 N(S(=O)(=O)N1CCN(C(c2ncc(C)o2)C(=O)NC(C)C(=O)OC)CC1)CC N(C1CCc2ccc(OC(F)F)cc21)C(C(C(C)C)C)=O C(=O)(C(CNC(C1CCCN1C)=O)C(C)C)NCC1(CC=C)CCCC1 c1(CC)cc(C(=O)NCC(C)(C)CNC(=O)Cc2ccc(C)s2)n(C)n1 C(=O)(NN1C(=O)C(C)N(C)C1=O)C1(C(=O)OC)CCC2CC12 c1(CC(NOC(CC)C)=O)ccc(NC(=O)N(c2ccccc2C)CC)cc1 C12(C=O)CC(C)(C1)OC21CCC1.C(C(=O)N(C(C)C1CC1)C)N(C)CN C1(OC)CN(C(=O)NC(c2cc(Cl)cnc2F)CF)C2(CCC2)C1 CC12CC(CCO1)N(C(=O)C(O)CNC(=O)C1=C(Cl)CC1)C2 c1(C(=O)NC2(CCNC(C3=NNC(=O)CC3)=O)CC2)cccc2cc(O)ncc12 CN1CC(C)(C)CC1C=O.c1cc(C(N2CCC(C)(C(N)=O)C2)=O)n(C)n1.N CC1(C(N2CCN(C(c3ncc4n3CCCC4)=O)CC2)=O)Cc2ccccc2C1 N1(C(C2CC=C(C(C)C)CC2)=O)CC(NC(C2CC2(C)C)=O)CC12CCOCC2 c1(C(N2CC3(CC(NC(=O)COCC(F)F)C3)C2)=O)cc2ccsc2c(O)n1 N1(C(CCCCC=CCCC)=O)CC2N(C(c3sccc3Cl)=O)CCC2(C)C1 N1(C(COCC(C)C)=O)CCCCC1CC(=O)NCC1CSCCO1 CC(C)C(CC(=O)NC1CC1CNC(c1cc(Cl)cc(Cl)c1N)=O)C(C)C C(c1cncc(F)c1)=CC(=O)NC1C2CCN(C(C3CCC(C)CC3)=O)C21 C1(C)(NC(C(C)N(C(c2csnc2Cl)=O)C2CC2)=O)CCC(=O)NC1=O Cc1ncoc1C(=O)NCc1csc(CNC(C2CCSC2)=O)n1 c1(C(N2C(C(=O)NC(c3cnc(C)s3)C)CC=CC2)=O)cccc2[nH]ncc12 CCC(C)(C)C(O)C(=O)N1CC(CN(C)C(c2ccncc2F)=O)C2(CC2)C1 CC(CC(=O)NCCCCCN(C)C(c1cnc2c(c1)COC2)=O)CC(C)(C)C N1(C(CCN(C(c2ccc(F)cc2)=O)CC)=O)CC(C2CC2)(OC)C1 c1(CC(=O)N(C(C)C)C)cc(F)c(F)cc1F.c1(C=O)cccs1.C(=O)(C)N C1(O)(CCNC(CSCCCC)=O)CN(C(=O)Cc2nncn2C)C1 CC(C)C(C)CC(=O)N(C(C)CC(=O)NCCC1(C)CCCO1)C CC1(C)CC(CN=c2ccc(OCC(F)(F)F)c[nH]2)CNC1=O C1(CC)C(NC(=O)C(C)OCCN(C)C)CCCN1C(=O)C(CO)OC c1(C(=O)NC2CC(NC(CC(C=C)CC)=O)C2)c[nH]c2cccc(F)c12 C(=O)C1=Cc2ccccc2C1.CC1=C(C)CC(C(=O)NCC2CC2C)CC1.N c1(OC)oc(C)nc1C(=O)NC1CCCC1.C1(C(=O)N)CCC(C(N)=O)O1 Cn1cccc(C(=O)N(CCC)C2CC2)c1=O.c1(C(=O)N)cnc(C(F)F)nc1 CC1(C)OCCC1C(N1CCC(C(=O)NCCO)(CO)C1)=O.CCC1CC1 c1(C(=O)NC(CC)C(=O)N2CC(CC(F)F)C2)cccc2cc[nH]c12 Cc1cc(C)nc(CNC(C2(NC(C3CCC(C)O3)=O)CSC2)=O)n1 c1(NC(C2CC(C)CN2C(=O)CCC2CCC2)=O)cc(OC(F)(F)F)cc(Cl)c1 C(C(C(=O)NCC1CC[Si](C)(C)C1)C(C)(C)C)NC(c1c(C)cn(C)c1)=O CC1CCCCCCN1C(C1CCCN1C(c1ncn2c1CCC2)=O)=O N1(C(c2cn(C)nc2C(F)F)=O)CCCC(C2CC2)C1.N1(CC(=O)N)CC=CC1 C(CNC(C1(CSC)CCC1)=O)(CC(=O)N(C(C)C(C)(C)O)C)OC C1(CCNC(c2c(SC)cccc2)=O)CN(C(=O)CCc2ccon2)CCCO1 c1(C(N2CCCC(CCNC(c3cc(CF)on3)=O)C2)=O)csc2ccccc12 CCC(C)(F)C(=O)NCC(C1CC1)NC(c1cnc[nH]c1=N)=O Cc1ccc(CCC(=O)Nc2ccn(CC(=O)NC3CC3)c2)cc1Cl N1(C(CSS(C)(=O)=O)=O)CCC(CO)C(NC(=O)Cc2ccoc2)C1 c1(C(=O)NC2CC3(CN(C(C(C)C4CCCC4)=O)C3)C2)n[nH]c2c1CCOC2 c1(CC(N2CC3CC3C2)=O)cc(C)ccc1C.c1(OC)cc(C(=O)NC)nn1C c1(C(N(CCN(C(C2CCC(C)C2)=O)CC)CC)=O)onc2c1CCCC2 N1(C(C(=O)NCC2CCS(=O)(=O)C2)=O)C2CCC1C(N)C2.c1ccccc1 CCC(F)(F)C(C)(C)C(=O)NC1COCC1NC(=O)CC1NC(=O)NC1=O O=C(O)CC(O)C(=O)NC1CC(c2ccon2)C1 C1(CCNC(CCOCCC)=O)CN(C(=O)Cn2ncc(O)nc2=O)CC(C)O1 Cc1cc(C#N)ccc1COC(=O)C(C)(C)Oc1c(F)cccc1F C(=O)(C(O)CC(C)C)NCC1(OC)CN(C(c2c(OC)cc(C)s2)=O)C1 c1(NC(CC2CCCN(Cc3c(C)n[nH]c3C)C2)=O)cnc2ccccn12 C1(CC(=O)NCCC(C)SC)CCCCN1C(=O)CCC1CCCC1 N=c1nc(O)cc(C2CCN(C(c3cc(C4CNC4)no3)=O)C2)[nH]1 Cc1cc(NC(=O)C(C)(C)CCNC(=O)C2=C(Cl)CC2)c(C)c(C)c1 C1(CNC(C)=O)CN(C(C2CC(C3CC3)=NO2)=O)C2CCCC2O1 c1(C(N2CCCC(F)(CNC(C(F)=C(C)C)=O)C2)=O)cncc2ncn(C)c12 N1(C(C(C)CF)=O)CCC2(CCCN2C(=O)Cc2ccc3occc3c2)CC1 C1(C(=O)NCCCC(C)NC(c2ncc(Br)cc2O)=O)CC2(CCCO2)C1 C1(NC(COCCOCC#C)=O)CCN(C(c2n[nH]c(C)n2)=O)C12CC2 Cn1cnc2cc(C(=O)NCC34CC3CN(C(c3cc(Cl)ccn3)=O)C4)cnc12 c1(C(N(CCCCN(C)C(c2ccncn2)=O)C)=O)ccnc(F)c1F C1(CNC(c2cc(C(C)C)[nH]n2)=O)CC(C(=O)N2CCOC(C3CC3)CC2)=NO1 c1(NC)cccc(C(=O)NC(c2ccccc2F)C(=O)NCC(C)OC)n1 Cc1cc(=NCCN(C(=O)C(C)Oc2ccc(F)c(F)c2)C)[nH]c(C)n1 C1(NC(CCc2n(C)cnc2)=O)CCN(C(c2cc(C#N)c[nH]2)=O)C(C2CC2)C1 Cc1c(C(N2CCC(O)(C(C)NC(=O)COC3CCC3)C2)=O)cccc1Cl CN1CCN(C)CC(C(=O)NC2CCC(NC(=O)Cc3cc[nH]c(=N)c3)CC2)C1 C1(N(C)C(C2CC3CC3C2)=O)CCC(n2cc(C3(O)COC3)nn2)CC1 C(=O)(CCN=c1[nH]c2ccc(S(=O)(=O)NC3CC3)cc2s1)NCC.C1CCC1.C C1(c2nc(-c3ccc(CC)cc3)nn2CC)CCc2n[nH]cc2C1C c1(NC(CC2(C)N(C(c3c(OC)nccn3)=O)CC2)=O)cccc2cnccc12 C12(OCC)CCC(C(=O)NC3CCCCC3)(CC1)C2.c1(C=O)nn[nH]c1Cl.C N1(C(C2(F)CCN(C(c3ccc(C)cc3)=O)C2)=O)CC(O)C(O)C(O)C1CO c1(OC)cc(C(N2CCOC(C)(C)C2)=O)ccc1C.C(c1cnc[nH]1)=CC(=O)N C1(NC(C2(C)CC(=C)C2)=O)C2CCC1CN(C(=O)CC1CCSC1)C2 C1(C(=O)NC(CNC(CS(CC)(=O)=O)=O)(C)C2CCC2)Cc2c(F)cccc2O1 C#Cc1ccc(F)c(C(=O)NCC2CC(C)N(C(c3[nH]nnc3C)=O)C2)c1 CON1CCC(C(N2CCOC(CCNC(C3CC4(CCCC4)C3)=O)C2)=O)CC1 c1(NC(C2C3CN(C(c4cc(C)[nH]c4C)=O)C2C3)=O)c(C)ccnc1Cl C1(CCNC(c2c(CC)nco2)=O)CCCN(C(c2cc(C)cs2)=O)CC1 N1(C(CC2(C)CC2)=O)CCC2(C1)CN(C(c1c(F)ccc(Cl)c1N)=O)C2 c1(C(=O)NC(CNC(CCCCOCC)=O)(C)C(C)C)cncc2ccsc12 c1(COC)nc(Cl)cc(=NCC=CCNC(c2cnn(CCO)c2C)=O)[nH]1 Cc1ccccc1C=CC(=O)NC(C1CN(C(=O)COCC(C)C)CCO1)C c1(C(N2CCOCC(F)(CNC(C(COC)C)=O)C2)=O)cc(Cl)c2n[nH]cc2c1 C(=O)(C1=CC2C=CC(C1)C2)N(C(C)C(=O)NCCCc1cncnc1)C1CC1 C1(NC(C2C(OCC)CC2)=O)CC(C(=O)N)C12CCC2.c1cncc(F)c1 c1(NC(C(N2C(C)CC(N)C2)=O)=O)ccc2c(c1)NC(=O)C2 C(C1CCCCC1)=CC(=O)N(C(C)C(=O)N(CCCC(C)C)C)CCC C1(C(N2CC3C(CNC(COCC#C)=O)(C3)C2)=O)CC2(CCCCC2)CO1 C1(NC(c2cncc(F)c2)=O)CC(NC(c2cnc(Cl)s2)=O)C12CCC2 c1(NC(C2CCCN(CC3CC(OCC)C3)C2)=O)cn(C)c(=O)nc1O c1(CN(C(C2CC2)=O)CC)ccc([N+](=O)[O-])cc1.c1(C(=O)N)cccnc1 CC1CCOC1C(=O)NCc1cc(C(=O)NC2CCC2)co1.C(N)(=O)N CC(C)CC(C(=O)NCC(C)CCO)N(C)C(C1COCC1(C)C)=O C1(C(C)C)CCC(C(N2CC(C)(NC(=O)C3=CC(C)(C)C3)C2)=O)C(=O)N1 N1(C(CC(CC)C(C)C)=O)CCOC2(C1)CN(C(c1ncccc1Cl)=O)C2 c1(CC=O)ccc(S(C)(=O)=O)cc1.N1(C(C(COCC)C)=O)CCCCCC1.N N#Cc1csc(C(=O)NC2CCCCC2CNC(c2cc(Cl)cs2)=O)c1 C(=O)(C(O)CNC(C1(n2cnnn2)CC1)=O)NC(CCC)c1ccco1 C(=O)(CS(=O)(=O)CC(C)C)NC1CC(Nc2ncnc(C)c2F)C12CCC2 C(=O)(CCC(=O)NC1(CO)CN(C(C2(C)CCCN2C)=O)C1)N(C(C)C)C c1(N2CC(CNC(c3c(CC)noc3)=O)OCC2)nc(C(C)C)cc(C)n1 O=C(N=c1nc(-c2ncccc2Cl)[nH]s1)NCC(C1CC1)C1CC1 C1(C(=O)NCC(C)CNC(c2cncc(C#N)c2)=O)CCn2ncnc2C1 CC(C)CCCC(C)C(=O)N1CC(C(=O)NCC2CCCN(C)C2)C2(CC2)C1 Cc1cn2nc(N3CCS(=O)(=O)C(CCNC(=O)C(C)C4CCCO4)C3)sc2n1 c1(C(=O)NC(c2ccccc2)CC)cc2ccc(O)cc2n1C c1(OC)cccc(OC)c1C(=O)NC(CNC(=O)CCCSC)C1CC1 C(=O)CC(F)(F)C(C)(F)F.CC(C=O)NC(=O)C1CC1.CCCC1CC1.N C1(NC(C(C)C2CC2)=O)CC2COCC(C1)N2C(=O)C(F)OC(F)(F)F C(=O)(C(C(C)C)NC(C12CSCC1C2)=O)N(CCC(F)(F)F)CC CCC(C(=O)NC12CC(NC(=O)C(F)(F)C3CCOCC3)(C1)C2)n1cncn1 N1(C(C(C)OC)=O)CCN(C(=O)CCC2CC2)CC1CC1CC1 c1(C(C(=O)N(C)CC2N(C(CSC)=O)CCCC2)C)ccc(F)cc1F Cc1cc(N2CCCC2)ccc1OCC(=O)N(C)C.C(C)(CC(C)NC)NC C1(C(=O)N=c2cc[nH]cc2)COC2(CCN(C(=O)C3=CCCS3)CC2)C1 c1(N2CCC(NC(CC3CCN(C)C3=O)=O)C(O)C2)ccnc(S(C)(=O)=O)n1 C1(C(N2C(C)CCN(C(=O)CC3CN(C)C3)CC2)=O)CCc2nc(=N)[nH]cc2C1 c1(CNC(C2CC23CCC3)=O)cn(CC(N2CC(c3nc(=O)o[nH]3)C2)=O)nn1 C(CCCCC(=O)N1CCC(C)(NC(=O)C(C)C(C)O)CC1)NC(C)=O O=C(CC(CC1CC1)NC(=O)CC1CCC=CCC1)NCC1CCOC1=O C1(C(C)C)(C(=O)NCCC2CC(C)(C)C2)CCN(C(c2ccn(C)c2)=O)C1 c1(C(=O)NCC(CC)(CC)NC(c2cnn[nH]2)=O)cc(Cl)c(C)cc1OC C(=O)(CCCC(=O)N1CCCC(CO)(NC(=O)CCC)C1)OCC.C(N)(=O)N CN1CCN(c2cncc(Cl)n2)C(CNC(=O)CCNC(C2CCCCC2)=O)C1 C1C2COCC1CN(C(c1cc3n(n1)CCO3)=O)C2.C(=O)(COCC=O)NC.N C(C)(CCC(=O)N1CCCCC1CN(C(=O)C(n1nccc1C)C)C)OCC CCC(C)CCC(=O)NC1CC(CNC(c2cccnc2-n2cncn2)=O)C1 C1(NC(C(C2CCN(C(CCCOCC=C)=O)CC2)C)=O)C2CCCC1COC2 C(=O)(C1CCc2cc(F)ccc21)NC(C)CNC(c1cc[nH]c(=N)c1[N+](=O)[O-])=O C1(C(=O)OC)COCCN1C(C12CC1CN(C(c1cc(C(C)C)nn1C)=O)C2)=O N1(C(=O)CCC2CCOC2)CC2(CCN2C(C2CC3CC3C2)=O)C1 C(CC(Cc1ccccc1)NC(c1cnc(C2CCC2)s1)=O)NC(C(C)OC)=O c1(C(=O)NC2(C)CC(NC(c3ccc(C)nn3)=O)C2)cnc2cc(C)ccc2c1 CCC(O)CC(=O)N1CC(CC(=O)N(C)Cc2nncn2CC)C(C)C1 C#CC(C)(C)C(=O)NC(CNC(c1cnsc1)=O)CC N1(C(C(C=C)C)=O)CC2CN(C(=O)CC3CCCC(=O)N3)CC(C1)O2 Cc1ccc(OCC(=O)N)c(F)c1.C1C=CCN(C(=O)C=Cc2ncc(C)[nH]2)C1 C=CC(C)(C)CC(=O)NCc1cncc(C(N2CC(OC)C(O)C2)=O)c1 CC1(C)C(NC(C23CC2CCN3C(C2CC(C3CC3)C2)=O)=O)CC1(F)F C=CC(COC)N=c1[nH]c(N2CCC(C)(C)SC(C)(C)C2)nc(=NC)[nH]1 C1(C(=O)NCC(C(=O)NCc2c(CC)nco2)N(C)C)NC(=O)CC1C C(=O)(CCCCO)NCc1cn(CCC)nn1.C(C(C)(C)C)C1C(C=O)C1 C1(C(=O)NC2C(C(N3CC(CC)C3)=O)CCCC2)CC12C(=O)Nc1ccccc12 c1(C(N2CC(OC)CC2)=O)ccc([N+](=O)[O-])o1.c1(C=O)conc1C1CCC1.N C(C)(CC(C)N=c1[nH]c(Cl)ncc1C)NC(C1N(CC)CCOC1)=O c1(C(N(C(CNC(C(CCC)OC)=O)C2CC2)C)=O)cc2n(c1)CCOC2 N1(CC)CCN(CC(=O)N(CC)C2CC2)C(=O)C1=O.c1(C(=O)N)oncc1C C(=O)(C(CO)NC(=O)C(F)CC1CCOC1)N(C)CC1CC1 c1(SC)cc(C)c(C(=O)NC2CCC(F)(C)C2)s1.C1(C(=O)N)CC(C)C1 CCCCC(CC)CC(=O)NCCOC1CCN(C(=O)Cn2nnc(=O)[nH]2)C1 C(C)(C)(CCCC(=O)NCCCC1CCCCO1)NC(CCc1n(C)ncc1)=O Cc1cc(CC(=O)NC(c2ccnn2C)C(=O)NC(C)C(=O)NO)cs1 C1(C)(C(N(CCC)CC)=O)CCC(=O)N(C)C1.C1(C=O)(N(C)C)CC1.N Cc1[nH]nc2c(C(N3CC(O)(CNC(=O)C(C)C#N)C3)=O)cccc12 C1(NC(c2cccc(CO)c2)=O)CCCCN(C(=O)CCCCCBr)C1 C1(NC(C2CCC(OC)C2)=O)CC2CC(NC(C34CCC(CC3)C4)=O)CC12 C(C(CC(C)(C)C(=O)OC)NC(=O)NCC1(C#N)CC1)OC C1(NC(c2c(C)ccc(Cl)c2)=O)C2CCN(C(=O)CN3CC4CC4C3)CCC12 CC(CO)N(C)NC(=O)NC(C(C)(C)C)c1ncccn1 CC1CCC(NC(=O)C=CCN2CCCC2)CN1C(c1cc(CCCO)on1)=O c1(OC)ccc(CNC(=O)C(C2CS(=O)(=O)C2)N)cc1S(C)(=O)=O C(C(C(=O)N1CCC1CNC(C1CC=CCC1)=O)C(C)(C)C)OCC=C C1(C2CCCN(C(=O)CCOCC(F)F)C2)(NC(C(C)C2CCC2)=O)CC1 C(=O)C#CC1CCCC1.N1(C(C)=O)CCOCC1C(=O)NCC12CC(C1)C2.N N1(C(Cn2ncc(C#N)c2)=O)CCCC(C2CC2NC(c2csc(S)n2)=O)C1 C1(NC(c2cnc(O)c(F)c2)=O)COCCN(C(C2(CC3CC3)CCC2)=O)C1 c1(C(=O)NCC2(C)CCN(C(=O)CN=S(C)(C)=O)C2)cc2ccc(Cl)cc2[nH]1 C#Cc1cnc(NC2CCCCN(C(=O)C(C)Sc3ccc(OC)cc3)C2)nc1 c1(C(=O)NCC(C)N(C(=O)CSC2CCCCO2)C)ncc(Cl)cc1F c1(NCC(C(=O)NC)(C)C)ccc(S(=O)(=O)NC2CCCc3occc32)c(Cl)c1 C(CCCC(=O)NC(C)CC(C)NC(=O)Cc1ccsc1Cl)(OC)OC c1(CC)noc(CCCC(=O)NCC(CC)NC(c2cnn(C3CCC3)n2)=O)n1 C(=O)(CC(C(F)F)NC(c1cn2c(n1)CCC2)=O)N1C(CC#C)CCCC1 N1(C(c2cn(CC=C)nn2)=O)CCC2(CC2C(=O)N(CCN(C)C)C)C1 N1(C(c2c(C)ncc(Cl)c2)=O)CCC2C(CCCN2C(=O)CC2CC(=O)C2)C1 C1(NC(C(CCNC(c2n(C)cnc2)=O)O)=O)CN2CCCC1C2 C1(COC)CN(C(=O)CCc2cccc(OC)c2)CCN1C(=O)C1=NOCC1 N1(C(C(C)CO)=O)CCC(CO)(CNC(=O)CC2(C)CCOC2)C1 N1(C(CNC=O)=O)CCC(F)(F)C(C)C1.C(=O)(C=C(Cl)Cl)N.C1CCCC1 c1(CNC(=O)CC2CC2)cn(C2CN(C(C3CC(O)C3)=O)C2)nn1 c1(C(=O)NCC(CC=C)NC(=O)C(O)c2ccco2)cn(C)c(=O)c(C)n1 c1(N2CC(C(C)NC(C=CC)=O)C2)cc(C)nc(S(C)(=O)=O)n1 Cc1cc(Cl)ccc1NC(=O)CC1(C)CCN1C(=O)Cn1nccn1 Cc1cc(C2CCC2)ncc1C(N1CC(NC(c2nc(Cl)sc2C)=O)C(C)C1)=O c1(NC2CC(F)(CNC(CCCc3ccc(OC)cc3)=O)C2)ncc(Cl)c(O)n1 c1(C(N2C(C)CC(NC(Cc3c(C)cnn3C)=O)C2)=O)cc2c(o1)CCCC2 C12(CC)CCC1CN(C(=O)CCc1cnc(C)s1)C2.C(C(=O)N)N(CC)CC C(=O)(C(C(=O)NC1CCN(C(C2CN3CCC2CC3)=O)C1)C(C)C)OCC CC(CC(F)(F)F)C(=O)NCC1CC2(CCC2)CN1C(C1CC(CF)C1)=O c1(NC(C2CN(C(c3sc(Cl)nc3Cl)=O)CCC2(F)F)=O)c(Br)ccc(F)c1F CC1CN(C(=O)CC2CCC2)CCCN1C(=O)C(F)n1ccnc1 Cc1nc(N2CCC(O)(C3(C(=O)O)CCC3)C2)c(C#N)c(C)c1C Cc1ncc(Cl)cc1C(N1CC(CC(C)NC(C2CCN(C)CC2)=O)C1)=O Nc1ccc(C(=O)NC(C(=O)NCC(=O)NCCO)C2CC2)nc1F C1(N(C(=O)CC2CC2)CC)CCN(C(=O)CCNS(C)(=O)=O)CC1 C1(CNC(C(C)=C(C)C)=O)CCC2(CCN(C(C3CC34CCC4)=O)CC2)O1 C1(CC)CC(C(=O)NCc2coc(C)c2)CCN1C(=O)CCCC1CC1 c1(OC)ccc(C(=O)NC2CN(c3cc(C(F)(F)F)ncn3)CC2C)cc1 c1(NC(C2CN(Cc3cccs3)CCC2O)=O)c(F)ccc(Cl)c1F Cc1c(C(N2CC3CC2CN3C(=O)C(C)OC2CCCC2)=O)sc2cncn12 C1(C(N2CCC3C(NC(C(C)=C(CC)C)=O)C32)=O)C2C3CC4C1C1C2CC3C41 CCCC(C)(C)CC(=O)NC1CCC(N(C(=O)C=Cc2cncn2C)C)C1 C1(NCc2nc(C)c(C)[nH]2)CCc2cnn(C(C)C)c2C1 c1(C(N2C(CNC(c3ccc(OC)s3)=O)CCC2)=O)ccc2nonc2c1 C(C(=O)N)(C(C)C)NC(C)=O.C1CN(C(=O)C=CC)CC1C.c1ccccc1 C12(CNC(COC)=O)COC(CNC(C3(C)CCCO3)=O)(C1)C2 C1(C(=O)NCC(CNC(Cc2c(C)n[nH]c2)=O)CO)Cc2cccc(F)c2O1 C(C#Cc1ccc(I)cc1)NC(C1CCCN(c2cncs2)C1)=O C1(C(=O)OC)COCCN(C(=O)C(N2CCOC(C)(CCOC)C2)=O)C1 C1(CC)CCN(C(c2cnc(OC)s2)=O)C1C(=O)NCc1ccnc(C)c1 CN1CCN(C(=O)CC2CCCCCC2)C(CNC(=O)C(C2CC2)C2CC2)C1 c1(NC(C2C(C)C2C)=O)ccncc1C(=O)NC(C)(C)C c1(CNCC=O)cc(C)c(O)cc1C.C(=O)(C(C)COc1ccccc1)OC C1(CC(N2CCC(CNC(=O)C(=O)Nc3ncc[nH]3)C2)=O)CCC=CCC1 C1(C(N2CCC(NC(C(C)OCC=C)=O)C2)=O)CC2CCC1CC2(F)F Cc1oc(C(C)C)nc1C(=O)N(CCC)C.c1(C=O)cn(C(F)(F)CO)nn1.N c1(C(=O)NC2(CC=C)CCCN(C(=O)CO)C2)ccc2c(c1)C(=O)NCC(=O)N2 CC1ON=C(C(=O)N(C2CCCN(C(c3ccc(Cl)c(N)c3)=O)C2)CCF)C1C S(=O)(=O)(c1ccc(Br)cc1F)N(C1C(C)CCNCC1)Cc1ccc(F)c(Cl)c1 N1(C(C2CCC(NC(C)=O)CC2)=O)CC=C(C)CC1.c1(C(=O)N)cn(C)nc1C N1(C(C(C)(F)F)=O)CCC2CCN(C(c3ccoc3)=O)C2C1 c1(C(N2C(CNC(CC(=C=C)C)=O)CCCCC2)=O)cccc2oc(C)cc12 Cc1c[nH]c2ncc(C(N3CCC4CCC(C3)N4C(C3CCCN3C)=O)=O)cc12 c1(OCC)nccc(C)c1C(=O)NC1CCCCN(C(C2CCCC(F)C2)=O)C1 N1(C(c2ccc(CC)o2)=O)CC2(COC)CC1(C)C2.c1(CC=O)ccco1 Cc1ccc(C=CC(=O)NC2CC(C)N(C(=O)C(C)(O)c3ccccn3)C2)cc1 C1(C(=O)NCCCC(=O)NC)(CC)CCCN(C(=O)C(n2cnc(C#N)n2)C)C1 CC1CCCC1NC(c1cnn(CCNC(=O)CC2CC2)c1)=O C(C1CCCCCC1)=CC(N1C(CN(C(c2cncc(C)n2)=O)C)CCC1)=O C(CC1CC1)(C(=O)N1CC(CO)C1)SC.C1CC(=O)N1 C1(C(N(C(CF)CF)C)=O)CCOCCN1C(C1CCCN1C)=O C1CC2CCC(C1)N2C(=O)C=Cc1cn(C)cn1.CN1CCC(C)(C=O)C1=O.N c1(C=O)c(C)oc(C)c1S(N)(=O)=O.N1(C(CCCSC)=O)CCC(C)C(C)C1.N C=CCC(CC)C(=O)N1CCC(C(C)C(=O)N(C)C(c2ccncc2)C)CC1 C(C)(CNC(=O)Cc1csnn1)(C(C)C)NC(C1CC(CC)C1)=O Cc1c(NC(=O)CN(C)CC2CCN(C(c3ccccc3)=O)CC2)ncnc1Cl CC(C(=O)NCC1(F)CCN(C(=O)CCC2CCC(=O)C2)CC1)S(C)(=O)=O CN1CC(NC(=O)CSCCNC(=O)CCOCC(F)F)C(C)(C)C1 C=CCC(CC)C(=O)NC1(C)CC(NC(c2cc(C)nn2CC(F)(F)F)=O)C1 c1(C(N2CCC3C(NC(c4nncs4)=O)C3C2)=O)cc2ccccn2c1 C(=O)(C(F)(F)C1=CCOCC1)N.c1(CC)[nH]ccc1C(=O)N(CCC)C1CC1 c1(NC(CC(CNC(=O)C(C2CCOCC2)O)OC)=O)cc(C)cnc1O c1(NC(N2CC(C(C(=O)NC)(F)F)(O)C2)=O)nc(Cl)ccc1C(F)(F)F CS(=O)(=O)c1ccc(C=CC(=O)NC2CCC(C3CC3)CC2)o1 Cc1ccc(C=CC(=O)NCCCNC(=O)C(O)CC2CC2)o1 C1(C(=O)NC(C)CC(C)NC(=O)CSC(F)(F)F)CCC2(CC1)CC2 c1(C(N(C(C)C(=O)O)Cc2ccccc2)=O)ccc(Br)cc1[N+](=O)[O-] C(=O)(CCCCCc1ccc(O)cc1)NC1C(NC(C(COC)(F)F)=O)C1 N1(C(c2cccc(C(C)(F)F)c2)=O)CCOC(c2ccccc2)CC1 N1(C(c2cc(C)nc(O)c2)=O)CCC2C(CCCN2C(=O)Cc2ccns2)C1 c1(C(N2CCC(C(C)NC(COCC=C)=O)CC2)=O)c[nH]c2cc(Cl)ccc12 CC1CCC(C(=O)NCC2(c3cccc(Cl)c3)CCCC2)NC1 CCCC(CC(C)C)C(=O)NC1CCC1NC(c1nn(CC)cc1Cl)=O c1(N(C)C(c2n[nH]cc2NCc2ncc[nH]2)=O)ccc(F)nc1N(C)C c1(CC)cnc(OC(c2cccc(OC3CCCC(C)C3)c2)=O)c(O)c1 C1(C)(c2cn(Cc3c(C)ncn3C)nn2)CCCN(C(c2cc(Cl)c(Cl)s2)=O)C1 N1(C(C2CC(OC)C2)=O)CC2COCCC2(NC(=O)Cc2c(C)ncnc2C)C1 c1(C(N2CCCCC(NC(C(C)C(C)(C)C)=O)C2)=O)ccnc2[nH]ncc12 C#CCCC(O)C(=O)N1CC(C(=O)NCCNC(C2(C#N)CC(C)C2)=O)C1 c1(C(=O)NC(CNC(CCN(C)CCO)=O)(C)C2CC2)csc2cc(Cl)cnc12 CC1(C(=O)NCC2(F)CCC2)CCNC1=O.c1(C=O)ccnn1CC(F)F.C O(NC(=O)C(C)NC(c1cn(CC)nn1)=O)C(CC)C C1(C(=O)NC)Cc2ccccc2CN1C(=O)C=Cc1ccnn1C CCCC(C(=O)NCC1CC1(Cl)Cl)NC(=O)COC1CCCC1 CCC(CC(=O)NCCc1ncn(C)n1)NC(=O)Cc1ccc(C)o1 c1(C(N2CC3C(NC(CCCC(=O)OC)=O)(C3)C2)=O)ccc2ncsc2c1 C1(Nc2c(C)cc(C(=O)NCCO)cc2)COc2ccccc2OC1 C=CCC(CC)C(=O)NCC1CCC1NC(c1cc(N2CCOCC2)ncn1)=O c1(CC)cc(OCC(=O)NCC2(O)CN(C(=O)CNC=O)C2)ccc1Cl c1(C(=O)NC(CC)CNC(C2(C)CC2C)=O)c(C)noc1C(F)(F)Cl Cc1cnn(CC2CC2)c1.c12cn(nn1)CCCC(=O)NC21CCC1 Nc1ccc(C(=O)NCC23CCC2CN(C(c2cc[nH]n2)=O)C3)c(Cl)c1 c1(C(C(=O)NCC(=C)C)N(C2CC(C)OC(C)C2)C)ccc(C2CC2)cc1F C#CCC(CC(=O)NCC1CC(SC)C1)NC(C1(CC#C)CCCCO1)=O N(C(=NCCOC(F)(F)C(F)(F)F)NCC1(F)COCCOC1)C(C=C)C CC1(C)CC(C(=O)NC2CC(NC(=O)CC3(C#N)CC3)C2)CC(C)(C)S1 CC1CN(C(C2(CC(F)F)CC2)=O)CCN1C(c1sccc1F)=O CC1(C)C=C(C(=O)NCC2(C)CC2)C1.C1(C=O)CC2(C1)CC2(F)F.N c1(C(N2CC(NC(C3C(=C)CC3)=O)C(c3ccnn3C)C2)=O)cn(C)c(=O)cn1 C(=O)(C1c2c[nH]nc2CN1C(C1CC12CCCC2)=O)NCC(C(C)O)O c1(OC)ncc(CN2CCC(=CC(=O)Nc3cc(F)ccc3Br)CC2)cc1Cl C1(O)(CC)CCN(C(C2C(C#N)C2(C)C)=O)C1.c1(C(C)C)occc1C(=O)N c1(C(=O)NC(CCSC)C(=O)N(C(C)CCC(C)C)C)cn2c(n1)CCC2 N1(C(C(C)C2CCC2)=O)CC2=C(C1)CN(C(C1CCS(=O)(=O)C1)=O)C2 C(c1ccc([N+](=O)[O-])cc1)=CC(N1CCCC(N(C(=O)CC(C)(C)F)C)CC1)=O c1(C(N2CC3CC3C2)=O)nccc2ccsc12.C(C=CC(=O)N)(CC)=CC.C C(=O)(CCCCCSC)N1C(CN(C(c2nc(C#C)sc2)=O)C)CCC1 N1(C(C(COC)O)=O)C(C(N2CCN(C(C)(C)C)CC2)=O)CCC1C C#Cc1ccc(C(=O)NC(C2CCCN2C(=O)COCP(C)(C)=O)(C)C)cc1 N1(C(C(C(=O)OC)C)=O)CC2CN(C(c3ccc4c(c3)OCCC4)=O)CC2(C)C1 C1CCN(C(C2CC3CCC2C3)=O)C1(C)C.C(C)(C)(C=O)NC(=O)NCC C12(C(=O)NCC(C)N(C(=O)CN3CCCS3(=O)=O)C)CCCCN1CCC2 C(=O)(C(CCS(C)(=O)=O)NC(c1cc(C)[nH]c1C)=O)OC C(CC1CC1)(C(=O)NCC(C1CCCC1)O)NC(c1cc(Cl)c[nH]1)=O Cc1ccccc1C1CCN(Cc2cc(C(N3CCC(O)C3)=O)ccn2)CC1 N1(C(CC(OCC)OCC)=O)CCC(O)(CC(=O)NCc2ccco2)CC1 n1(CC)cc(C(=O)NC2CCN(C(c3cnc(C)o3)=O)CC2F)c2ccccc12 c1(OC)cc(C(=O)NCC(O)CNC(C2CC(=O)N(C)C2)=O)c(Cl)cn1 C1(NC(c2n(C)cc(Cl)c2)=O)CC2CC(C1)N(C(=O)Cc1ccccc1F)C2 c1(C2C(C(N(CC(C)O)C)=O)C2)ccc(Cl)cc1.n1(C(C)C)cccc1C=O.N Cc1noc(C)c1CC(=O)NCC1CCN(C(c2n[nH]c(C)c2F)=O)C1 C1(CNC(Cc2nnc(C)o2)=O)CN(C(c2c([N+](=O)[O-])cnn2C)=O)CC1(F)F C(CC(C)C(=O)N1CCC(NC(c2c[nH]c(C(N)=O)c2)=O)C1C)OC N1(C(c2c(C(C)C)ncs2)=O)CCOC(C(C)NC(=O)C(c2ccccn2)O)C1 C(C(CC(C)C)C(=O)N1CCC(CC(F)F)C1)NC(CNC(=O)NC)=O c1(CC)ncc(C(N2CCCC2(C)CNC(c2cc(C#N)c[nH]2)=O)=O)c(O)n1 C1(F)(CNC(C(C)(C)C)=O)CCN(C(C2CCC2CF)=O)C1 c1(NC(C2N(Cc3c(C)nc(C)[nH]3)CC(O)C2)=O)nc(Cl)c2ccnc-2[nH]1 C1(C(=O)NCc2c(OC)ccnc2)CCCCCN1C(c1ccccc1F)=O C1(C(=O)NCC2CCN(C(C(CC)(C)C)=O)CC2)CC2CCC1CC2OC C1(NC(C(C=C)(C)C)=O)CC(C)CN(C(c2cc(N)c(F)cn2)=O)C1 C(c1cn(C(C)C(N2CCC(N3CCOC3=O)CC2)=O)nn1)=CC c1(OCCC(=O)NC(CNC(CC=CC)=O)C)ccc(F)c(F)c1 c1(NC(C(C(C)C)N(C)C)=O)cccc2c1CCC2.C123CC1CN(C2)C3=O C(CCCCC(=O)N1CCC(C)(N(C)C)C1)NC(C(C)N1CCCC1)=O C1(C2CCOCC2)(C(=O)NCCCC(C)NC(c2cscn2)=O)CCOCC1 N#CC1(C(=O)NC2CC(NC(=O)Cc3c[nH]ccc3=O)C(O)C2)CCCCC1 N1(C(C23CCC(C)(C2)CO3)=O)C2CCC1CC(NC(C1CC13CCCC3)=O)C2 N1(C(CCc2cc(C)on2)=O)C2CCC1CN(C(=O)CC13COCC(C1)C3)C2 N1(C(C(CSC)C)=O)CC2(C1)CN(C(c1cc(Cl)c(C)cn1)=O)CC(C)(C)O2 C1(C=O)CC(C)(C)CC(C)(C)C1.n1(CC(=O)N)cc(C(C)O)nn1.CCCC C=C(Cl)CC(C(=O)NC(CC)C(C)(C)C)NC(c1ncc[nH]1)=O Cc1ncc(C(=O)N(C2CCCCC2CNC(=O)CC23CCCC2C3)C)cc1Cl C1(C(=O)NC(C2CCCN2C(c2ccccc2)=O)C)C=CCOC1 C1(C(=O)N(C)C)(CNC(C(C)NC(N)=O)=O)CCCC1.C1(O)CCOC1 C#CC(CNC(C1CCCCCCN1C(c1snnc1CC)=O)=O)CC(C)(C)C C(=O)(C(O)C(F)(F)F)N(CC(CC)NC(C1(C(F)(F)F)CCC1)=O)C c1(C(C)C)ccc(C(O)C(=O)NCCC(C)(C)C)cc1.C(=O)CCc1cnoc1.N C1(CC)CN(C(c2ccnc(-n3ccnc3C)c2)=O)CCC1NC(=O)CSC C=CC(C)(CC)C(=O)N1CCC(C)C(C)C1.c1(C(=O)N)cnc(C(F)(F)F)cn1 c1(C(N2CC(C(=O)Nc3ncc(Br)nc3CO)NCC2)=O)cc(Cl)nc(Cl)c1F c1(CC)cc(C(=O)N)c(C)nn1.C1(C(N2CCC2)=O)(C(F)F)CC(O)C1.C N1(C(c2c(SC)n(C)nc2)=O)CCC2(CCCN(C(=O)CC(C)C(F)(F)F)C2)C1 CC1CN(C)CCC1Nc1cc(NC(C)CC(=O)NC2CC2)ncn1 C(=O)(CCC(O)C(C)(C)C)N(C)CC1COCCN1C(C1CC2(CC2)C1)=O N1(C(C(C)(F)F)=O)CCC(CNC(c2ncccc2Br)=O)C12CC2 N1(C(c2[nH]c(C)c(C)c2C)=O)CC2CCC1CN2C(=O)C(F)=C1CCCC1 c1cc(F)cc(Cl)c1.N1(C(CC(=O)OCC)=O)CC2(CC2C(=O)NC)C1 c1(CC(=O)NC(C2CC2)C)ccccc1.C(=O)CC=CC(C)(C)C.CC O=S(=O)(c1c(Br)cc(F)cc1Br)NCC1CC2(CCCC2)CO1 c1(C(=O)NC2CC(F)CN(C(C3CC4CCC3CC4)=O)C2)cc2ccccn2n1 C1(CC)CCCN(CC(=O)N(CCCNC(=O)CCCc2cnn[nH]2)CCO)C1 C(=O)(C(C(C)C)NC=O)NCCN(C(c1ccc(CC)[nH]1)=O)C.C1CC1 Cc1ccc(-c2cccnc2)cc1NC(=O)NCc1ccc(Cl)cc1Cl Cc1cc(CCC(=O)NC2CC(C)N(C(=O)C(C)OCCN(C)C)C2)nn1C CCC(CC(F)F)C(=O)N(CCCCCNC(=O)C(Br)=C(C)C)C N1(CC)CCOCC1C(=O)NCc1ccccc1CNC(C1CC1)=O.S N1(CC2OCC(C)(C)C2)CCC2(CCCN(C(c3cc(C#N)c[nH]3)=O)C2)C1 C12(NC(C(C3CN(C(c4nn(C)c(CO)c4)=O)C3)O)=O)CCN(CC1)CC2 Cc1ccc2c(c1C(=O)NC(C)CNC(C1(F)CCOCC1)=O)CCCN2 c1(C(=O)NCC(CC(F)(F)F)NC(C=CS(C)=O)=O)cnn2c1CCCC2 c1(C(=O)NC(c2ccc(Cl)cc2)c2ccsc2)cccc2c1COC2 C1(NC(C(C=C)(C)C)=O)C2CCCC1CCC2.C(=O)(C)N.C(=O)C.C(C)=O c1(CNC(C(=O)N(C2C(C)CCC2)C)=O)ccc(C(N)=O)cc1 N1(C(C2CCC(C)CC2)=O)CC(NC(=O)CCN(C)CCO)CC2(CC2)C1 C1(NC(CC(C)F)=O)CCC(C(N2CC(O)(C(F)F)C2)=O)CC1 c1(CC)c(C(=O)NCc2conc2C)cnn1-c1cccc(Cl)c1 c1(C(c2n(CCSC)nnn2)NC)ccc(C)c2ccccc12.C1CC(C)(C)C1 C1(CC(C)C)CN1.C1(c2ccno2)(C(=O)NCC2(CC)CCC2)CCOCC1 C=CCC(CNC(c1cc(OC)n[nH]1)=O)C(=O)NCP(C)(=O)OCC CC1CC2CN(C(=O)CC3(C)CCN(C(c4coc(C(F)F)c4)=O)C3)CCN2C1 c1(C(=O)NC(c2ccnn2C)C(=O)NC(C)C(F)(F)F)cc(F)cc(F)c1 C1(NC(c2ccc(OC)nc2)=O)CC2CCC1CN(C(c1c[nH]c(=S)cn1)=O)C2 C1(CCOC)CCN(C(=O)CN(C)C(C)C)C1.c1cccnc1.C(=O)(CC)N C1CCS(=O)(=O)C12CN(C(=O)C(c1cccc(Cl)c1)O)C2.CC(C)(C)OC=O c1(C(C)(C)C)nc(=NCCCCCCNC(c2sccc2S(C)(=O)=O)=O)s[nH]1 c1(C(c2cccc(Br)c2)NC(N2CCC(C)C2)=O)cc2ccccc2o1 C12(C=O)CCC(=O)N1CCS2.N1(CC(N2CC(CCC)C2)=O)CCS(=O)CC1.N c1n[nH]c(O)n1.O=C(CCOCC1CC1)N.C(=O)(C)NCC.C1CC1 C(=O)(C1c2ccccc2C(=O)N1C)Nc1c(C)cc(Cl)c(F)c1 C12(NC(c3cc(C)nc(C)n3)=O)CCCN(C(=O)Cc3sc(C)nc3C)CC1C2 c1(C(=O)NC2(C(=O)NC)CN(C(COCCCC)=O)C2)c(C)ncn1C C1(CNC(CCCSC(C)C)=O)CN(C(C2(C)C=CCCC2)=O)CCN1C CCCCC(O)C(=O)N1CCN(C(=O)Cc2sccc2C)C(c2nccn2C)C1 CC(CCN(C)C)C(=O)NC1CCCC(CC(N2CCC3CCC23)=O)C1 C(=O)(C(C)CCNC(=O)CC1CCC1)OC.c1(C(=O)N)ccnn1CCF N1(C(C(F)=CC)=O)CC(O)(CNC(=O)CCc2cc(OCC)no2)C1 C(=O)CC(F)(F)C(F)(F)F.C(=O)(CCC(=O)Nc1nccs1)NCCCC=C.N CCCC(O)C(=O)NC1CCC(NC(c2ccc(CN(C)C)cc2)=O)CC1 N1(C(c2cc(CC)c(CC)o2)=O)CCCCC(NC(c2cncn2C(C)C)=O)C1 Cc1nccc(C(=O)NC(CNC(=O)Cc2cncn2C)C2CCC2)c1N CC(c1ccccc1)=CC(=O)NCC1(NC(=O)CC2CC=CC2)CCCC1 c1(NCc2c(C)scc2)nccc(=NCCCNS(C)(=O)=O)[nH]1 CN=c1nc(N2CCCC(CCCO)C2)[nH]c(N2CCOC(C#N)C2)n1 C1(CC(N2CC(OCC(=O)NC)C2)=O)CC(F)CN1C(c1ncccn1)=O C1C2CN(C(c3ccsc3Cl)=O)CC12.C1(C(=O)OC)C(C(=O)NC)C1(C)C N1(C(CC2CCCC(NC(C3CCCC3O)=O)C2)=O)CCCC2COCC12 CC(O)C(C)C(=O)N(CC(C)(C)NC(c1nn(C)cc1Cl)=O)C c1(NCC(=O)N(CC(=O)O)CC)ccc(N2CCCC2)c(Cl)c1 c1(C(=O)NCC2CCCN2C(=O)COCC(F)F)ccc2oc(O)nc2c1 C(=O)(C1=CCC(NC(C23CSCC2C3)=O)C1)N(C)Cc1scc(C)n1 c1(C(=O)N)c2c(nn1C)CCC2.C(C)(C(C(=O)NC1CCOCC1)N(C)C)OC C1(CN2CCC(c3cccc(C)c3)C2)CCC2(CCNCC2)CC1 c1(C(C)=O)c(C)[nH]c(C(=O)N(CC(O)CNC(=O)CC2(O)CCC2)C)c1C CC(C)(F)C(C)(F)Cn1cc(C2(NC(C3CCCCCS3(=O)=O)=O)CCC2)nn1 CC1CC(C(N2CCCC(Br)C2)=O)N(Cc2cn(C)cn2)C1 CCCCC(C)C(=O)NCC1(F)CC(NC(c2cc(I)on2)=O)C1 c1(NCc2cc(OCC)no2)nccc(=NCCc2nc(C)c(C)s2)[nH]1 C1(C(=O)NCCNC(COC)=O)CCC1.C1(C(C)(C)O)(C=O)CCC1 CCCC(C(=O)N(CC(C)C(=O)N1CCC(CC(=O)NC)C1)C)OC N1(C(CCc2c(C)ncs2)=O)CC(C)CN(C(C2CCCO2)=O)CC1C c1(CCC)ccccc1C(=O)NC(CO)C(C)NC(C1(F)CCCOC1)=O C1(CN(C(c2cocc2C)=O)CC)CCN(C(C2CCC(C)S2)=O)CC1 C=C1CCN(C(C2CCN(C)C2)=O)C(C(=O)NC(C)Cc2cccnc2)C1 C(=O)(C1CCCn2ccnc21)NC(CNC(c1ccccc1)=O)CO c1(N2C(C)(C(=O)NCC=C)CCC2)ncnc2n[nH]c(Br)c12 Cc1cc(Br)nc(NC(=O)CSc2cccc(Oc3ccccc3)c2)n1 N1(C(c2c(C)cns2)=O)CCN(C(c2csc(C3CC3)n2)=O)C2CC12 C(=O)(CC(O)CC(C)(C)C)NCCC1(O)CN(C(C(C2CCOCC2)OC)=O)C1 N1(C(C(C(CCC)NC(C2(C)CCCCO2)=O)O)=O)CCc2cnccc2C1 c1(SC)cc(C)ccc1C(=O)NC1CCCC(N(C)C(c2ccns2)=O)C1 CC12C3C4C1C1C2C3C41C(=O)NC1CCCN(C(c2ccnc(F)c2O)=O)C1 CN1CCCC(C(=O)N(CCCN(C)C(C2(C(F)(F)F)CCO2)=O)C)C1 C#CCCCCCNC(C1CN(C(C2CN(C(C)C)C2)=O)CCO1)=O C12(NC(=O)CCCF)CCCC1N(C(c1nnc(O)cc1O)=O)CCC2 c1(NC(CN2CCN(C(C(=C)F)=O)CC2)=O)cc(C)c(C)c([N+](=O)[O-])c1 N1(C(c2nnn(C)n2)=O)CCC(C(F)(F)F)C(NC(c2cnccn2)=O)C1 Cn1nnc2c(NC3CCCCC3NC(=O)C=C(Cl)Cl)ncnc12 c1(NC(C)=O)ncc(S(=O)(=O)NC2CCCN(c3nc(C)ncc3F)C2)s1 c1(CNC(=O)NC(COC)(CO)c2ccccc2)ccc2c(c1)oc(=O)n2C Oc1c(C(F)(F)F)cc(F)c(-n2cc(C(c3nccs3)SC(F)(F)F)nn2)c1F C12(NC(c3c(Cl)cc(C)nc3)=O)CCCC1N(C(=O)Cc1cncc(F)c1)CC2 N1(C(CCSCCC)=O)CC(NC(c2ccc(-c3cn[nH]c3)cn2)=O)CC(C)C1 C1(C(=O)NC2CN(C)C(=O)C2)CC2CN(C(=O)C(C3CCOCC3)=O)CC2C1 Cc1cc(C(=O)NC(C)CNC(=O)CC2CN3CCC2CC3)c(Br)cn1 C12(NC(Cc3c(C)ocn3)=O)CCOCC1CN(C(=O)CSc1nncs1)C2 N1(C(c2cc(C(C)C)no2)=O)CCN(C(=O)C(C)NC=O)CCC1C C(=O)(N=c1cc(C)n(C)[nH]1)C1CN(C(c2cc(CC)n(C)n2)=O)CC1C c1(C(N2C(CCNC(C(CC=CC)C)=O)CSCC2)=O)ccc([N+](=O)[O-])cc1N O=C1CN(N2CCCC(C3CCCCC3)C2)CCN1Cc1ccccc1 c1(OCC)ccc(NC(=O)C(C2CCN(C=O)C2(C)C)F)nc1C.C(C)(C)C C(=O)(C1=NN2CCCN=C2N1)N1CC=C(CNC(CC=CCC)=O)CC1 CC1CCN(C(c2cc(C(F)(F)F)cc(Cl)c2)=O)CCN1C(=O)CCCCCF C=CC1OCCC1C(=O)NCCC1CC(NC(C2(C)CCOC2)=O)C1 c1(C(=O)NCC2(NC(c3c(C)ncc(Cl)c3)=O)CCC2)cccc2nc[nH]c12 Cc1nnc(-c2ccc(C(=O)NCCN(C(=O)CC3CCCOC3)C)cc2)n1C CCCC(F)(F)C(=O)N1CCC(C(F)C(=O)N(C(CO)CO)C)C1 N1(C(c2c(OC)cncc2Br)=O)CC2(COC(CN)C2)C1 S(=O)(=O)(c1ccc(N2CCc3cc[nH]c(=N)c3C2)cc1Cl)NCCCC=C c1(OC)cc(F)ccc1C(=O)NC1CCN(C(=O)CCC(C)(C)OC)CC1CO N1(C(C2CN(C(c3cc(C)nc(O)c3)=O)CC(C)C2)=O)CC=CC12CCCC2 C(C(C)CC(F)(F)F)NC(CC(=O)N(C(C)C)CCOC=O)=O c1(C(C)C)ccc(C#N)c(NCC(C)CNC(c2nc(Cl)ccc2F)=O)n1 N1(C(c2n(CC)ccn2)=O)CC(OC)CC1CNC(c1ccncc1)=O CCCC(C(O)C(=O)NC1CC2CCCC(C1)C2)NC(c1cc(C)oc1CC)=O C1(NC(c2[nH]cc(C(C)=O)c2)=O)CN(C(c2nc(O)c(C)s2)=O)CC12CCC2 c1(CCC(=O)NCCC(C)NC(c2cnc(Cl)[nH]2)=O)nc(-c2cccnc2)no1 C(CCC(C(=O)N(C(C)CO)C)NC(=O)Cc1cnccc1C)OC C1(C(N2CCC(C(C)NC(CCC=C(C)C)=O)C2)=O)C2CCC1(C)C2(C)C C1(=CCNC(=O)CCc2ccoc2)CCN(C(C2CCCC(CF)C2)=O)CC1 C1(CC(=O)NCCOCC(N2CC(Cc3ccncc3)C2)=O)CCOCC1 C(=O)(C1=CCN(C(=O)C(C)(C)CC#N)C1)N(CC(O)C1CC1)C C1(C(=O)NC2CN(C(c3c(C)nc(C)o3)=O)CC2O)Cc2cc(Br)ccc2O1 C1(C(=O)Nc2n[nH]c(C3CCCN3)n2)CC2CNCC1C2 CC1(C)C2CCC1(NC(=O)CCC1CCC1)CC2.C1(CC=O)CCCC(O)C1.N C#Cc1ccc(CCCC(=O)N(C)CC2CCN(C(C3(O)CCSC3)=O)C2)cc1 Cc1cc(C(=O)NCC2CCC2)c(C)nc1C.c1(C(=O)N)ncc(Cl)c(N)c1Cl C(c1cncs1)=CC(N1CC(O)(C2CCCN2C(C2CC23CC3)=O)C1)=O c1(CC(=O)NCC(C)CN(C)C(c2coc(C3CC3)n2)=O)c(F)cncc1Cl c1(C2(C=O)CC2)ccccc1.C1(C(N(CCC)CC)=O)CN(C(C)C)C1.N N1(C(=O)CSc2ccccc2)CC23CCCCC2(C1)CN(C(c1ncc[nH]1)=O)C3 Cc1ccc(C(=O)NC)c(Cl)c1C.C1CN(C(=O)CC(C2CC2)C2CC2)CCO1 N1(C(c2ccc(C)[nH]2)=O)CCC(C(=O)NCC(N2CCCCC2)=O)C12CCC2 C1(C(N2CCC(CNC(C3CC(=C)C3)=O)(OC)C2)=O)CC2C=CC1CCC2 C=CCC(CNC(C1CNC(=O)N1)=O)C(=O)N1CC(S(C)=O)C1 C1(O)(CNC(C2CCN(C(c3c(NC)ccnc3)=O)CC2)=O)CCC(C)(C)C1 C1(C)(C(=O)NCC2CC(NC(C(CCC)N(C)C)=O)C2)CCN(C)C1=O n1(CC(=O)Nc2scc(-c3ccc(C)s3)n2)[nH]cc2c(=O)ncnc1-2 c1(CC)ccccc1CNC(c1ccc(CNC(C2CCCCO2)=O)cn1)=O N1(C(C2CCN(C(CCc3nc(=N)[nH][nH]3)=O)C2)=O)CCC(CCF)CC1 Cc1[nH]c2ccccc2c1CNC1(c2nnnn2Cc2cccs2)CSC(C)C1 C=C=CC(C)C(=O)N1CCCCC1CCCNC(c1cc[nH]c1CCC)=O c1(CN2CCCC(NC(c3cc(OC)c(F)cc3)=O)C2)cc2ccncc2[nH]1 CC1=C(C(=O)N2CCC(C(N3CCOCCC3CC)=O)C2)CCO1.C1CC1 c1(CNC(c2nnnn2CSc2ccccc2)C2(CC)CCC2)ccncc1 Cc1nn(C)c(Cl)c1C=CC(N1CCCC1(C)CNC(=O)C(F)F)=O c1(CC(=O)NCc2occ(C(=O)NCC(CC)CC)c2)cnn(C)c1C C1(C(N2CC3CN(Cc4c(F)ccc(F)c4Cl)CC3C2)=O)Cc2ccccc2O1 Cc1nccc(C(N2CCN(C(C3(Cl)CC34CCC4)=O)CC2CO)=O)c1C C(=O)(C1=C(Cl)CCCC1)NC(CCCC)CNC(C1CN2CCC1CC2)=O c1(N2CC(C)(C)C(O)CC2)nc(=NCC(C2CC2)C2CC2)[nH]c2c1SCC2 N#Cc1ccc(C(=O)NC2CCCN(c3nccc(C(F)F)n3)C2)s1 c1(C(N2CC3C(C3)C2)=O)cc(I)c(O)c(I)c1.c1(C(=O)N)cc(C(F)F)no1 Cc1cc2n[nH]cc2cc1C(N1CC(C)N(C(=O)CCc2cnco2)CC1C)=O C1(C(N2CCCC(NC(C3(C(=O)NC)CC3)=O)C2)=O)CCC(=O)CC1C C(=O)(C1CC=Cc2ccccc21)N1CC(CN(C)C(C2(C)CCCC2)=O)OCC1 Cc1cc(O)ccc1C(=O)NC1CCN(C(=O)COC(C)C)CC1C(C)C c1(C(=O)NC(CCCC)CNC(=O)C(C)n2ccnc2)cccc(C(N)=O)c1C c1(C(N2CCC(NC(=O)OC)CC2)=O)cccc2c1OC(C)C2 c1(CCC(=O)NCC(C(=O)OCC)(C)CC)nc2ccccc2[nH]1 C(C(C)(C)CC(=O)NC(c1cccc(C)n1)C)NC(C1C(CCOC)C1)=O C12(NC(c3nn(CC)c(O)c3)=O)CCN(C(c3ccc(Cl)cc3N)=O)CC1C2 c1(CN2CCN(C(CCc3ccc(C)c(F)c3)=O)C(C)C2)cc(I)c(F)cc1F C1(NC(c2cc(CSCC)on2)=O)CCCN(C(C2(F)CC2)=O)CC1F Cn1nc(C(N2CC=CC2C)=O)cc1C1CC1.C1(C)(C(=O)N)CNC(=O)C1 Cc1cnc(C(N2CCC(C)C(C)C2)=O)c(C)c1.c1(C(=O)N)cnn(C(C)C)c1 Cc1nc(CO)sc1NC(C1CC2CCC2C1)=O CCC(C(=O)NCCNC(C1(OC(C)C)CC1)=O)n1cccn1 C(=O)(CC(CNC(C1(OC)CCOCC1)=O)C(F)(F)F)OC N1(C(c2cnc(-c3c(Cl)cccc3Cl)s2)=O)CC(O)CC12CCCC2 c1(C(N2C(C)CC(CNC(c3cnc4n3CCS4)=O)C2)=O)cc(F)c(O)c(F)c1 CC(CF)CC(=O)NC1CCCCC1NC(c1cnccn1)=O N1(C(C2CCC(C(=O)OC)C2)=O)CCC2C(C1)CN2C(=O)Cc1ccno1.C N1(C(CC2(OC)CCC2)=O)CCC(CO)(NC(=O)CCc2ccccn2)CC1 N1(c2ncnc(=N)[nH]2)CC2(C1)SCCC2NC(c1ccc(C(F)(F)F)cn1)=O C1(NC(c2c(C)occ2)=O)CC(O)CN(C(c2cccc(SC(F)(F)F)c2)=O)C1 Cc1c(C(=O)NC(C)C(C)C(C)C)c(C(F)(F)F)nn1C.C(=O)CN(C)C C(=O)(CC(C(F)F)NC(C1CCC1)=O)N(C(C(=O)OCC)C)C1CC1 N1(C(C2(C)CCOCC2)=O)CCCCCC(NC(C2CCc3nnnn3C2)=O)C1 c1(NCCc2nnc(C)s2)[nH]c(=NCC2CCCC(F)(F)CC2)nc2scnc12 C1(CC(=O)NCCN(C(=O)CCCc2ncco2)CCC)C=CCCC1 C=CCC(C(=O)N1C(C(=O)OC)CC1C)NC(c1ccc[nH]1)=O c1(C(N(CCC)C(C)C)=O)ccnc2c1CC(=O)N2.C1(C(=O)N)CCC(=O)N1C N1(C(c2cc(CC)c(C)s2)=O)CCC2(CCN(C(C3CCC(C)(C)O3)=O)CC2)C1 C12(NC(C3CC(=O)N(CCC4CC4)C3)=O)CCCC1N(Cc1ccon1)CC2 C1(C(=O)OCC)CCNCC1NC(c1ccc(-c2csnn2)cc1)=O N1(C(C=CSC)=O)CCC(C)C(NC(=O)C(c2cccc(OC)c2)(F)F)C1 c1(C(=O)NCC(CC=C)NC(C2CC2C=C)=O)c[nH]c2nccc(Br)c12 N1(C(CC2(C)CCCC2)=O)CC2CC1CN(C(C13CCCCN1CCC3)=O)C2 c1(CNCC(C2CCOC2)OC)nc(N(C)C)no1 N(C1c2ccccc2CC12CCCC2)S(=O)(=O)c1ccc(NC2CCC2)c(F)c1 N1(C(CCCOC)=O)CCC(O)(CCNC(=O)C(O)Cn2cncn2)C1 C(CN(Cc1ccc(C)cc1C)N1CCC(OCC(F)(F)F)CC1)OC N1(C(CCC#C)=O)CC2CC(NC(=O)CSc3n[nH]c(=N)s3)C(C2)C1 c1(C(N2CC(NC(C3(CC#C)CCOC3)=O)C(O)C2)=O)cc2c(Cl)cccn2n1 N1(C(c2n(C)nnc2)=O)CCC2(CCCC2C(=O)Nc2nc3c(s2)CCC3)C1 c1(C(N(CCOCCOC)C)=O)ccc(C)nc1.c1(C=O)csc(Cl)c1.N c1(CC)cc(C(=O)NCCC2CC(NC(c3scc(C)c3C)=O)C2)oc1.C C(CC(O)CC(=O)NC1C=CCN(C(c2ccc(CS(C)(=O)=O)cc2)=O)C1)SC N1(C(c2ccc(SC)o2)=O)CC(NC(=O)CCC(C)SC)CC2(CC2)C1 c1(OC)ccccc1N(C(=O)C(N)CO)C(=O)C(c1ccccc1)SC C1(CNC(c2scnc2Cl)=O)C(Cn2cc(CN3CCCC3)nn2)C1(F)F c1(C(=O)NCC(C)N(C(CCCn2c(C)ncc2)=O)C)nc(C2CC2)ncc1Cl C1(Nc2cc(NCc3c(OC)nn(C)c3)ncn2)CC(C)(C)OC1(C)C N1(C(c2sc(CC)c(C)c2)=O)CCN(C(C2CN(C)CC(C)O2)=O)C2(CCC2)C1 C(C(C)C(=O)NNC(=O)CCCN1CCC(N(C)C)C1)OC Cc1csc(=NCC(=O)NC2CC(CNC(C3CCC(C)(C)CO3)=O)C2)[nH]1 Cc1cc(Cl)c(Cl)cc1C(N1CCN(C(=O)CC(C)(C)C)C2CCC12)=O C12(C(N(CCCCCCNC(C3CCC(C)O3)=O)C)=O)CCC(CC1)OC2 N1(C(CC(C)=C(C)C)=O)CCCC(C(=O)NCC(O)C2(Cl)CC2)C1 C1(OC)CC(CC(=O)NC2CC(OCC(=O)NCC=CC3CC3)C2)C1 N1(C(C2(NC(=O)OC(C)(C)C)CC23CCC3)=O)CCCC2(C=CCO2)CC1 Cc1nc(C(C)NC(C2CC(CNC(=O)COCCCF)C2)=O)no1 N1(C(c2cc(OC)ns2)=O)CCC(NC(=O)C(C)C(=O)OC(C)(C)C)C1C N1(C(C2CC(C(=O)OC)C2)=O)CCCC2(CC2)C1.C1(C(=O)N)CNC(=O)N1 N1(C(C(CC=C)(F)F)=O)CCOCC(C)(CNC(=O)C=C(C)C)C1 C12(NC(c3c(Cl)cc(C)c(N)c3)=O)CCOCC1CN(C(=O)C=CC1CCC1)C2 c1(C(=O)NCCC(C)N(C(=O)CCC2CCCO2)C)ccc([N+](=O)[O-])c(C#N)c1 Cc1ccc(C(N2CCCC2C(=O)Nc2sncc2C#N)=O)c(I)c1C c1(C(=O)NC(C)CN(C)C(C2(C#N)CC2)=O)cn(C)c(=O)nc1O c1(C(N2CCC(CNC(C3CC34CCC4)=O)C23CC3)=O)cnn2c1CCCN2 C1(NC(C(CNC(C)=O)(C)C)=O)CCC2CN(Cc3ccc(F)cc3Cl)CC2C1 C1(C)(C(N2CC(C)(NC(=O)C(F)CC3CC3)C2)=O)CCCS1(=O)=O c1(-n2cc(C3(F)CCN(C(C(NOC)=O)=O)CC3)nn2)cccc(S(N)(=O)=O)c1 CC1CC2(CCN(C(c3ccoc3Br)=O)CC2)CN1C(C1CCC(=O)N1)=O N#Cc1c(N2CCC(CNC(=O)CCC[N+](=O)[O-])C2)cccc1F CC(=Cn1ccnn1)C(=O)NCC(C)(C)CN(C(=O)C1=CCCC1(C)C)C C(C)(C(C)(C)NC(=O)CC(O)C1CCCC1)NC(COC(C)C)=O C(=O)(C1CCCc2cncn21)NC1C(OC)CN(C(C(CCCCC)(C)C)=O)C1 C(=O)(CCC(C)CN(C)C)NCC(C(=O)N(CC(C(C)C)C)C)N(C)C N1(C(c2cc(C)c(Br)o2)=O)CC(C)CN(C(c2cnc(N)c(N)c2)=O)C(C)C1 S(=O)(=O)(c1c(F)cc(F)cc1F)N1C2CN(C(c3c(F)ccc(C)c3Cl)=O)CC21 c1(NC2C(C)CN(C(C3CCCCS3)=O)CC2)ncnc2c1ncn2C1CC1 C=CC(C)(C)CC(=O)N1CCOC(CCNC(C2CCC3CC3CC2)=O)C1 C1(O)(CN(C(c2cccc(C)c2)=O)C)CCCN(C(C2(C(C)(F)F)CC2)=O)C1 c1(C2(C)C(n3cc(C(CC)O)nn3)C2)ccc(Cl)nc1 c1(C(=O)NC(CCOC)CNC(=O)C=CC(C)C)sc2cccnc2c1Cl c1(C(=O)NCc2c(C)cc(C)nc2)ccc2c(c1)C1(CC1)C(=O)N2 N1(C(C2(C)ON=C(C)C2)=O)CCCC(F)(C)C1.N1(CC=O)OC(C)(C)CC1=O N1(C(CCC=C=C)=O)CCCC2(CC(NC(C3CC(F)(F)C3(C)C)=O)C2)C1 N1(C(CCOC(C)C)=O)CCN(C(c2ccc(-c3ccco3)s2)=O)CC1CO C(=O)(CCC(C)N(C)C(C)=O)NCC(NOCC(=O)OCC)=O C1(C(=O)NCC2(CSC)CC2)COC2(C1)CN(C(=O)CC)C2.C(C)C c1(C(=O)NC2CC(C(N3CC(C)C(O)CC3)=O)C2)ccc([N+](=O)[O-])nc1 CCC(CCCC(=O)NCc1ccnn1C)NC(c1c(C)ccnc1O)=O C(C)(C)(CCC(=O)N1CCC1CF)NC(COCC(=O)NC)=O N1(C(c2nc(Cl)cs2)=O)CC2CCC1CN2Cc1ccc([N+](=O)[O-])o1 CC1(C)CCN(C(=O)CCC2CCN(C(C3(c4cc[nH]n4)CC3)=O)C2)C1 C1(NC(C(C)(C(C)C)OC)=O)CN(C(=O)Cc2c[nH]nc2C)C2(CCC2)C1 C12CCC(CN(C(=O)CC3CC3)C1)C2.Cc1nn(C(C)C)c(C)c1C(=O)N c1(C(C)C)c[nH]nc1C(=O)NC(CO)C(C)NC(=O)CS.C1CCCCO1.C N1(C(c2c(Cl)cc(C)s2)=O)CC(NC(=O)CC2CCOC2C)C2(CC2)C1 CC(C(=O)NCC1CC1NC(=O)Cc1cocn1)C1CC1 c1(-c2n(-c3ccn(C)n3)nc(-c3cnn(CCO)c3)n2)cc(F)c(F)cc1F c1(NC(C2CCCN(C(C=C(C)C)=O)C2)=O)ccc([N+](=O)[O-])c(Cl)c1Cl c1(C(CNC(N2CC(CNC(=O)OCC)C2)=O)=O)cc(Br)c[nH]1 C1(CC)CN(C(=O)CC2(C)CC2(Cl)Cl)CCN1C(=O)COC1(C)CCCC1 CC(C)(F)CCC(=O)NC1(CNC(=O)CN2CC3CC3C2)CCOCC1 Cc1[nH]nc2c1CN(C(C1CC1C(=O)NC(c1ccccn1)(C)C)=O)CC2 C1(NC(C2CCCO2)=O)CN(C(c2ncc(Br)cc2F)=O)CC1(F)F C1(COC)(NC(=O)C(O)C(C)S)CCN(C(C2CN(C(C)=O)C2)=O)CC1 CC(CCNC(=O)C(c1cccc(O)c1)C)CCNC(=O)CCc1cncs1 N1(C(c2ccccc2-c2ocnc2C(=O)O)=O)CCC(C2CC2)C1 c1(NC(C)=O)ncc(S(=O)(=O)NC2CN(CC3CCC(C)CC3)CC2C#N)s1 c1(C(=O)NCC(CC)NC(=O)C(c2ccnn2C)OC)cccnc1C1CC1 c1(CNC(=O)C(N2CCCC(Oc3cccc(F)c3)C2)=O)cc(Cl)ncc1Cl c1(C(=O)Nc2ccnn2C2CCCOC2)cccc(OCCO)n1 CC1(C)C=C(C(=O)NCCn2cc(C(=O)NCCC3COCCO3)nn2)C1 c1(CC)nc(C(=O)NC)c2ccccn12.C1(O)CN(C(=O)CN2CCSCC2)C1 C=CCCCC(C(=O)N1CCCC(CN(C)C)C1)NC(=O)CCc1cccn1C N1(C(C2N(C(C)C)CCC2)=O)CC2CC1C2C(=O)NCc1nccn1C N1(C(CC(C(C)C)NC(=O)C(C)c2ccco2)=O)CCC2CN(C)CC2C1 C1(O)(C=O)CCCC(C)(C)C1.N1(CC)CCCC1CC(=O)N(CC(C)O)CC CC(C)CCC(=O)C(=O)NC1(C(=O)NCCC(O)C2CCCC2)CC(F)(F)C1 N1(C(C(CCC#C)O)=O)CC2CC(O)C1C2NC(c1ccc(OC)c(OC)n1)=O Cc1n[nH]c(C)c1CC(=O)NCCN(C(=O)C(C(C)C)S)C.c1ccccc1.C c1(C2(C(N3CCC(CC)C3)=O)CCC2)cc(Cl)cc(Cl)c1.C1(F)(C=O)CC1.N C1(CNCC(O)COCC(F)(F)F)CC2(CCC2)CCO1 C=CCC(C)(C)CO.C1(CC(=O)N)CC2(C1)CN(C(C1(C)CC(=C)C1)=O)C2 c1(C(=O)NC(C(C)C)CNC(=O)C(O)CC(F)F)nc2ncc(CCO)cn2n1 c1(CCn2cc(CN3C(C(=O)OC)C(C)CC3)nn2)c(C)nn(CC)c1C C1(CNC(CN(CCOC)C)=O)C2CN(C(c3cnc(Cl)[nH]3)=O)CC12 c1(C(=O)NC(C)CN(C)C(C2CC2C#N)=O)cccc2c1CCO2 N1(C(c2nc(C)oc2C)=O)CCN(C(=O)CC2CCCC(C)O2)C(C2CCC2)C1 c1(NC2CC(NC(CCNS(CC)(=O)=O)=O)C2)nccnc1C#N C1(C(N2CCC(CC=C)(NC(=O)CNC)C2)=O)CC2(C)CCCN2S1(=O)=O Cc1ccc(C)c(C(=O)NC2(C)CCOCC2)c1.C1(C(=O)N)CCCNS1(=O)=O CCC(C)C(C)C(=O)N(CCCCCCNC(c1cnc(C(=O)OC)cn1)=O)C N1(C(c2cc(C)cc(C)c2N)=O)CC2COCCC2(NC(=O)C#CC2(C)CC2)C1 C(CCC(C)(C)C(=O)NC1CC1c1ccco1)NC(CCCCCC)=O C=C1CC2CCC(C1)N2C(C1CCCC1CNC(C1(F)CC1)=O)=O C1(C(N2CCCC(CCC(N)=O)C2)=O)CCCN(C2CCSCC2)CC1 C1(C(=O)N)CCn2ncnc2C1.CC(C)CCNC(=O)CC1(c2ccon2)CC1 C1(C)(C(=O)NC(C(=O)OCCC)C)CCCN(C(=O)CCOCC)C1 c1(OCC(=O)NCC2OCC(CN)C2)cccc(Cl)c1Cl.C1C(=O)N1 c1(COC)ccc(C(=O)N(C(C)CCNC(=O)C(O)CC)C)cc1F N1(C(c2cc(C3(C)CC3)on2)=O)CCOCC(C(=O)NC)C1.C12CCC(C1)OC2 c1(NC(C(=O)NC2CCC(SCC)C2)=O)ccnc(O)c1.c1cc(C)ccn1 C(=O)(C(C#N)C(C)(C)C)N1CCCC(N(C(=O)COc2cnc(Cl)cn2)C)C1 C(=O)(C(C(C)C)S)NC(C(C)NC(C=CC(C)C)=O)(C)C.c1ccccc1 C=CCC(C)(C)CC(=O)N(C(C)CN(C(=O)Cn1cccnc1=O)C)C N(C1CCc2c(C)cccc21)C(=O)Nc1ccc(OCC(=O)NC)cc1 CC(CNC(=O)CC1CCCCC1O)CC(=O)NCc1nc[nH]n1 CC(N=c1cccc(S(=O)(=O)NCC2C3COCC23)[nH]1)c1ccccc1Br N1(C(CCC(=C)C)=O)CCC(CNC(C2CC2F)=O)C12CCC2 C1(C(C)C)CCOC1C(=O)NC(C(=O)NCc1ccccc1)c1ccco1 C1(C(=O)NC2CC(c3cn(-c4cccc(CSC)c4)nn3)C2)(OC)CCCOC1 N1(C(c2c(CC)c[nH]c2)=O)CCCC(C2CC2NC(c2cc(C)nnc2O)=O)C1 CC(C)C(C(=O)NC(Cc1ccoc1)C(N1CCC(C)(F)CC1)=O)C(C)C Cc1ccc(CSCC(N2CCC(C)C2C)=O)cc1.c1(C(=O)N)cc(C)co1 N1(CC(=O)NC2CN(C(C3CSCCS3)=O)C2)CCn2nccc21 C1(O)(CNC(CC2CC(NS(C)(=O)=O)C2)=O)CCN(C(=O)C(N)=O)C1 CC1CCc2[nH]c(=NCc3cn(C)[nH]c3=N)nc(N3CC4C(C3)C4(F)F)c2C1 C(=O)(CCCC(=O)OC)N1C(CC)C(C(=O)NCCCCCCF)CC1 c1(CC)cc(C(N2CC(CNC(C3CCC4CC4CC3)=O)C2)=O)ccc1OC C1(NC(C(CC)COC)=O)CC2CCC(C1)N2C(c1csc(C(C)(F)F)n1)=O n1(CC)nc(C(F)(F)F)cc1C(=O)NC1CCN(C(=O)C)CC1.CC=O.S C=CCCCCC(=O)N(CCNC(c1ncc(Cl)cc1Cl)=O)CC1CC1 c1(C(C)NC(C(CSC)O)=O)ccc(N(C)C)cc1.c1(CC=O)ccsc1Cl.N N1(C(c2c(C)nccn2)=O)CCCN(C(c2cc3c(s2)CCC3=O)=O)C(C)C1 C1(CC)CCC(CNC(=O)C(O)CNC(=O)CC2CCSC2)CC1 CCC(COC)C(=O)N1CCOCC1CNC(c1cc(CO)oc1C)=O C(=O)(C(C(C)(C)C)C1CCC1)NCC1(O)CN(C(CC(COC)C)=O)C1 Cc1cnc2ccc(C(N3CC4(C3)CN(C(c3nnc(Cl)cc3N)=O)C4)=O)cn12 c1(C(C)C)cccc(CC(N2CCC(CO)(NC(=O)C=CBr)C2)=O)c1 N1(C(Cc2cccc(OC)n2)=O)CCCC(C)C1C.c1(CC(=O)N)cnn(C)c1 C(=O)(C(C#N)CCc1ccccc1)N(CC(CN(C(C(F)=CCC)=O)C)O)C c1(C(N2CC(NC(C3N(C)CCCC3)=O)C(O)C2)=O)ccc2c[nH]nc2c1 N1(C(c2c(CC)noc2)=O)CCCC(C)(NC(=O)C(=Cc2cnn(C)c2)C)C1 CCC(CC(F)F)C(=O)NCc1ccc(CNC(c2cnnn2C)=O)cc1 C(C)(S(=O)(=O)C1CCOCC1)c1onc(C)n1.c1(OC)ccc(C2CCC2)cc1C N1(C(CCCCN(C)C)=O)CC(F)(F)CC1C(=O)NC1CC2OC(=O)CC12 CCC(C)(CCNC(=O)C(O)Cc1cnc[nH]1)NC(c1occc1C)=O c1(NCc2c(CC)noc2CC)[nH]c(=NC2CCC(F)(F)C2)nc2scnc12 N1(C(c2ccc(C)nn2)C(=O)NC)CC2(CCC2)C1C(=O)OC C(=O)(C(O)C(CCC)NC(c1nc(=N)cc[nH]1)=O)NC(CC=C)(C)C C=CC(C)(CCOC)C(=O)N1CCCC(N(C(c2cn(C(C)C)nn2)=O)CC)C1 CCCCCC(F)C(=O)NC1(CNC(C2(C)CC2(F)F)=O)CC(OC)C1 N1(C(CN(C)C)=O)CCc2cc(-c3cncc(C4CC4(F)F)c3)ccc2C1 C1(C(N2CCC(N3CCN(C(=O)C(F)=CCCF)CC3)C2)=O)CC2(CCOC2)C1 C#CC1(O)CCCN(C(C2CN(C(=O)Cc3cnn(CC)c3)CC2(F)F)=O)C1 CCC(CC(F)(F)F)C(=O)NC1CCN(C(=O)CCP(C)(C)=O)CC1CO Cc1ncc(Br)c(C(=O)NCC2CC(C)CO2)n1.O(C(F)(F)F)CC=O.N C(N=c1[nH]c2cccc(F)c2s1)C1(O)CN(C(C2CCN(C(CC)=O)C2)=O)C1 c1(C(N2CCCC(CC)(NC(=O)C#CC3CC3)C2)=O)cc2cccc(F)c2s1 N1(C(c2c(C)n(C)cc2)=O)CC2(CCCC2NC(c2ncc(F)cc2F)=O)C1 N1(C(C(OC)OC)=O)CCN(C(=O)CCO)C(c2cccc(F)c2)C1.C1CC1.C c1(CCC(=O)NCc2cn(C3CCN(Cc4ccccc4)C3)nn2)ccncc1 c1(C=O)[nH]cnc1C#N.c1(CC(=O)NCC(C)C2CC2)cc(C2CC2)on1.N c1(C(N(CCc2cccc(OCC)c2)C)=O)ccc(OC)c(OCC)c1 CC1SCCCC1C(=O)NC(CC1CCCC1)C(=O)NCCCOCC(F)F C1(CC=C)(C(=O)NC2CC(=O)N(C(C)C)C2)CCN(C(c2ccsc2Cl)=O)C1 Cc1ccc(NC(=O)N(C(C)C)CC2(C)CC2)cc1C#N N1(C(C(C)(C)CO)=O)CC2(C1)CCCS2(=O)=O.C1(C=O)CCC2(C1)CC2(F)F.N C(=O)(C1CCCn2ccnc21)NC(C)CCN(C)C(c1ccc2nsnc2c1)=O C1(C(=O)NCCCN(C(C(CCC)CC)=O)C2CC2)CCc2nc(C)cn2C1 N1(C(c2cc(COC)on2)=O)CCC2(CCN(C(C3COC(=O)N3C)=O)CC2)C1 c1(C(N2C3CCC2CN(C(C2(F)CCOCC2)=O)C3)=O)cc2ccccc2o1 N1(C(C2C(CC(C)(C)C)C2)=O)CCOC(C(=O)NCC=CCO)C1 c1(C(=O)NC2CCN(C(C(C)C(F)F)=O)C2(C)C)cncc2cnccc12 N1(C(c2cncc(C#C)c2)=O)CC(CO)C2(CCN(C(=O)C(C)COC)CC2)C1 C(C1(C)CCC(C)C1(C)C)=CC(=O)NC1(CC)CCN(C(C(CCC)O)=O)CC1 c1(C(=O)NCC2C(C)CCCN2C(C2CCC=CO2)=O)[nH]nc2ncnc(O)c12 c1(C(=O)N)cc2ccc(Cl)cc2o1.c1(OC)ccc(F)cc1C(=O)NC(C)CO C=CCCCCCC(=O)NCC1(C)CCCN(C(=O)CC2CC3(CC3)C2)C1 C(C(CO)C(C)(C)C)NC(CC1CCN(C(COCCC)=O)C1)=O Cc1ccc2c(c1)C=C(C(=O)NC(C)CC(F)(F)F)CO2.C(=O)(CC1CC1)N c1(CC)cnc(O)c(C(N2CC(CCNC(=O)C(C)(C#N)CC)C2)=O)c1 C(=O)(CCCCCF)NCC(C1CC2CCC1CC2)(C)O CC1C(=O)NCCCN1C(=O)C=CCN(C(=O)CCS(C)(=O)=O)C C(c1cnn(-c2ccccc2)c1)=CC(=O)NCCCC(C)NC(c1cccs1)=O C1(CNC(C2CC(C#N)(OC)C2)=O)CN(C(C2CSCC(=O)N2)=O)CCC1C N1(C(c2nc(CC)oc2)=O)CCCC(NC(c2ccncc2F)=O)C(F)C1 CC1(NC(=O)Cc2cncs2)CCCN(C(=O)Cc2ccc(O)cc2Cl)C1 c1(C(=O)NCCC2CCCN(C(CC(C)(C)O)=O)C2)cc2cnc(Cl)cc2s1 C12(CC(=O)N(CCC#C)CCO)CCC1CN(C(=O)C=Cc1cn[nH]c1)C2 C1(NC(C(CC)=CC)=O)CCCN(C(c2cnn(C(C)C)c2C)=O)CC1 c1cc(S(C)(=O)=O)ncn1.C(C)(C)(CC(C)C)NC(Cc1c(C)n[nH]c1C)=O.N NC(=O)CC(N)C(=O)N1CCCCC1c1nnc(C2CCOCC2)o1 c1(C(=O)NC2(CNC(C=COCC)=O)CCOC2)ccc(OC(F)F)cc1 c1(OC)ccc(NC(C2CC2NCc2cc([N+](=O)[O-])cs2)=O)c(Cl)n1 C(Cc1ccoc1)(C(=O)NCCC1CCC1)NC(c1scnc1C(F)F)=O c1(NC(=O)NC(c2ncc(C)o2)C)cc(C(=O)OC(C)(C)C)ccc1C c1(C(=O)NC2CC(C)(CNC(C(C)n3cncn3)=O)C2)ccc2cc[nH]c2n1 C1(C)(C(=O)NCc2cn(CC#C)nc2)CCN(C(C2CC23CCC3)=O)C1 c1(C(=O)NC2C3CN(C(c4c(C)nn(C)c4C)=O)CC32)ccc2nnc(O)n2c1 C1(C(N(CC=C)CCO)=O)CCCCN1C(=O)C(C)C1(O)CCC1 c1(C(N(CC(=O)OC)C)=O)cc(CNC(=O)Cn2ccnc2)[nH]n1 c1(C(N2CCCCC(C(=O)NC(C#C)CC(C)C)C2)=O)cccc2[nH]ncc12 CCCCC(O)CC(=O)N(C)CCOCCC(=O)N(C1CCN(C)C1=O)C C(=O)(C(CC(C)C)C(N)=O)N1C(C(=O)NCCc2cccc(C)c2)CN(C)CC1 C1(CC(=O)NCCNC(c2csc(Br)c2)=O)CC(=O)c2ccccc2C1 C1(C(=O)NC2C(OC)CCC2)CCN(C(=O)CC2CC(C)C2)CC1C C(CNC(c1ncncc1Cl)=O)(CC(F)(F)F)NC(C1CCN(C)C1=O)=O c1(C=O)c(C)[nH]c(C=O)c1C.C1(C)(CC=O)CC1(F)Cl.CC=CC.CO Cc1cc(C#N)cnc1C(=O)NCC1CCN(C(=O)C2=CS(=O)CCC2)C1 Cc1cc(C)c(C(=O)N(c2ccccc2)CCC2(C(=O)O)CC2)cc1C=O N1(C(CC2(COC)CCOCC2)=O)CCC2CCCC(C1)N2C(=O)C=CC(C)C N1(C(c2c(C)occ2)=O)CCC(C)(C)C1C(=O)NCCN1CCCCC1 C(C#CC(=O)N(CC(F)F)C1CCC1)NC(C(C)c1cccs1)=O N1(C(C(CC)=CC)=O)CCC2(C(N3CCCC(N=[N+]=[N-])C3)=O)CCCC12 Cc1cc(C(N2CC(CN(C(=O)C(N)=O)C)C2)=O)cc(C)c1Br CCCC(C(=O)C(=O)OC)OC(=O)C1=CC(C)(CC)C1 c1(OC)cc(C#N)ccc1C(N1CCCC(CNC(=O)CC=C(Cl)Cl)C1)=O c1(C=O)cnc2snc(C)c2c1.c1(SCC)ccc(C(=O)N)cc1.CC=CC C(C(C)(C)CN=c1[nH]c(CO)nc2ccccc12)N(C(=O)C(O)CC[S+](C)C)C C#Cc1cnc(=NCCC2CC(NC(=O)Cc3csc(C)n3)C2)[nH]c1 C1(C(=O)NCC=CCC(=O)N(CCC)C(C)C)CCCC(O)C1 C(=O)(N=c1[nH]oc2ncc(Br)cc12)NCC(c1ccc(C)cc1)N1CCOCC1 c1(C(=O)NCC2N(C(C(C)OCC#C)=O)CCC(C)C2)cccc2c1ncn2C CC1=C(C(=O)NC2CCOC2C(=O)Nc2cccc(Cl)c2)CCC1 N1(C(C(n2cc(CCOCC(N)=O)nn2)C)=O)CCOc2nccc(Cl)c2C1 Cc1cc(C#N)cc(C)c1NC(C1CC(F)(F)CS1)=O c1(OCC(N)=O)ccc(C(=O)NCC2CC2)cc1.C(=O)C(O)C1CCC1 C(=O)(C1=CCCC1C)NCC(C(=O)NCc1c(C)nn(C)c1)N(C)C C(c1cncc(F)c1)=CC(N1C(C)CC(NC(CCOC(C)C)=O)C1)=O N1(C(c2c(CCCC)ocn2)=O)CCC2(NC(c3cc(C(N)=O)no3)=O)CC2C1 C(CCCC(=O)NCCn1ncnn1)NC(c1c(CC)nns1)=O c1(CC)nc(C(N2CCOC(C(C)NC(=O)CC(F)(F)F)C2)=O)c(C)o1 C(=O)(C1=C(C)N(C)c2nnnn2C1C)N.C1(CNC(C=CCC)=O)CCCC1O CC1(NC(C23CC(C)(CO2)C3)=O)CCN(C(=O)C=CC=O)C1.C1CC1 Cc1ccc(-n2cc(O)c(C(=O)NC3CC3)n2)cc1.c1(C(=O)N)cc(Cl)cnn1 CCCC(CCCNC(=O)C(c1c(C)noc1C)C)NC(=O)C(F)(F)CN(C)C C1(C(N(C)CC2(O)CN(C(C3C4CCC3CC4)=O)C2)=O)COCCN1C C(C(C(=O)N(C)Cc1noc(C)n1)C(C)C)NC(C(COC)N(C)C)=O C12(CC(N3CC(CN(C(=O)Cc4nncn4C)C)OCC3)=O)CCC(CC1)OC2 Cc1ccc(CC(N2CC3CC2CC3CNC(=O)Cn2cccc2)=O)cc1C C1(O)(CC)CCN(C(=O)CCC2CCCO2)CC1.C1(C=O)CC1.C(C)(C)C.N CCC1=NOC(CC(=O)NCC2(F)CC(NC(C3CC(OC)C3)=O)C2)C1 C#Cc1ccc(C(N2CC(NC(=O)C(F)CN(CC)CC)CC2CO)=O)o1 c1(CC)cccc(NC(=O)C(O)C2CN(C(=O)CCC(C)SC)C2)c1C C1(NC(C2C=CC(NC(CCC(C)OC)=O)C2)=O)CCn2ncnc2C1 N1(C(C(CC)C#N)=O)CCCC12CCCN(C(C13CC(C)(C1)C3)=O)C2 C1(OC)CCCC(C(=O)NCC2(CNC(=O)CCN3CCCC3)CC2)C1 Cc1cc(C#N)cnc1C(N1CCN(C(=O)CCCN(C)C)CC1CC(F)F)=O c1(NC23C(NC(c4cnsn4)=O)CC(CC2)C3)nc2ccc(F)cc2s1 Cc1ccc(C(=O)NCCOCCC(=O)Nc2csnc2C2CC2)c(O)c1 c1(CC(=O)NCCC2CN(C(c3cnsn3)=O)C2)csc(C2CC2)n1 C(CC(CC)C(=O)N1CC(C(C)NC(C2CC3(C2)CC3(F)F)=O)C1)=CC C1(CC(=O)NC)CCN(C(=O)CN(C(=O)C(C)C)CC(C)C)CC1 N1(C(C(CC(F)F)NC(c2ccn(C3CC3)n2)=O)=O)CC2CCC(O)C(O)C12 O=S(=O)(c1ccc(C(F)(F)F)c(F)c1)N1CCCC1CN1CCOCC1 Cc1cc(C(=O)NC(C)(C)CNC(=O)C(C)C(F)F)cc([N+](=O)[O-])c1Cl c1(COC)nn(C)cc1C(=O)NC1CN(C(=O)C=CC2CCOC2)CC1O C(C1CN(C(=O)CC(C)(C)COC)CC1C(=O)N(CCCO)C1CC1)=CC C1(C2CC2)(C(N(CCCO)CC)=O)CN(C(=O)CSC(F)(F)F)C1 c1(OC)ccc2nc(Br)nc(N3CCC(NC(c4ccc(F)cc4)=O)CC3)c2c1 CC1(C)CC(CC(=O)NC2(C)CCN(C(=O)CC(O)C3CC3)C2)CO1 Cc1nc(=N)[nH]cc1C(=O)N.C12CC(C1)C(C)O2.C(=O)CCc1nncs1.C CC(Cc1cnco1)C(=O)N(c1ccccc1)CC1CCOC1 CCC(CC(=O)NCC1CCCCC1)C(C)(C)C.c1(C=O)ccc(C(C)=O)o1.N C(c1ccc(F)c(F)c1)=CC(=O)N(C)CCNC(=O)C(C)(C)C(F)F c1(C(=O)NCC2C(C)(C)CCN2C(=O)CC2CC2)cc(Cl)c(F)cc1Br C1(NC(CSCC=C)=O)CCC(C)(C)C1.c1(C=O)ccc(C(C)=O)[nH]1.N N1(C(c2cc(CC)[nH]n2)=O)CCC(CO)(C)C1.C(=O)C(C(C)C)n1cnnn1.N C1(C(N2CC(NC(c3cnn(C4CC4)c3)=O)C3(C2)CC3)=O)CC2CCC(C1)C2O C1(CCOC)(NC(C2COCOC2)=O)CCN(C(C2CC23CCCC3)=O)C1 Cc1ccc(F)c(C(=O)N(CC(C)N(C(=O)CC2CCCC3(CC3)C2)C)C)c1Cl C(c1sccc1Br)=CC(=O)NC1CCC(CNC(C2CCOCC2)=O)C1 c1(C(=O)NCCN(C(CCOC(C)C)=O)C)cnc(C(C)O)s1 c1(-c2n(CCC)nc(-c3ccoc3)n2)ccc(S(=O)(=O)c2ccccc2)s1 c1(CC(=O)N)c(Cl)ccc(O)c1Cl.C(c1ccc([N+](=O)[O-])s1)=CC=O.C1CC1 N1(C(CC2(OC)CC2)=O)CCC(NC(c2ccc3nn[nH]c3c2)=O)C(CO)CC1 N#Cc1cc(F)c(CNc2cc(F)cc3cc[nH]c23)c(F)c1 C1(C(N2C3CN(C(C4N(N=O)CCC4)=O)C(CC3)C2)=O)CCc2nnc(O)n2C1 CCC(C)C(=O)C(=O)NC(CN(C)C)C(=O)NCc1nc(CO)cs1 N1(C(Cc2cccc(C)c2)=O)CCC(F)C(NC(c2cc3cscc3s2)=O)C1 N1(C(C(C(C)O)C)=O)CCC(NC(c2cc(O)cc(=O)o2)=O)C(C)(C)C1 c1(-n2c(C(C3CCCC3)C3CC3)nc(C(CC)O)n2)cc(F)ccc1C c1(C(=O)NCCOCCCNC(COC(CC)C)=O)cnc(S)nc1 C1(NC(C2C(C(C)C)OCC2)=O)CCC(C)(C)CC1.C1(C=O)(N(C)C)CC1 C(=O)(C(F)(F)C(O)C(C)C)N1CC2C(NC(C(CC)Cc3ccccc3)=O)C2C1 C=C1CCN(C(=O)C(N2CCOC(CF)C2)=O)C(C(=O)O)C1 N1(C(C2CC(=C)C2)=O)CC2CCCC2C1C(=O)NCC1CCCOC1(C)C CON(CCC(=O)N(C1CC(C)(C)C1)C)C(=O)CC1COCC1O c1(NC(C=Cc2ccc(C)s2)=O)ncc(-c2ccc(C3CC(=O)NN3)cc2)cc1O c1(CN(C2CC3CC2CN3)C(c2cc(C)c(C)nc2)=O)cn2cccnc2n1 N1(C(C(C)Cn2cccn2)=O)CCN(C)CC1C(=O)NC1(CO)CC(F)C1 N1(C(C2CC(OC)C(OC)C2)=O)CCCN(C(C2CC(O)C2)=O)CCC1 CC1C(O)CC2CCC1N2Cc1ccnc(NCC2CC3(CCC3)C(=O)O2)n1 CC(C)C(=O)C(=O)N1CCCC(CNC(c2cnon2)=O)C1 C(=O)(C(COC)CC(C)C)NCCC1N(C(c2c(C)cc(CC)o2)=O)CCC1 CCCCCCC(C)(F)C(=O)N1CCC(O)(Cc2cccc(F)c2)C1 C1(C(=O)NCCC2N(C(c3c(C)cco3)=O)CCCC2)CCC2(CCC2)OC1 C(C(=O)N1CC(O)(c2cc[nH]n2)C1)(C(C)C)NC(Cn1c(C)ccn1)=O N1(C(COC)=O)CCN(C(C2C(C)OC(C)C2C)=O)CC1C CN1CCn2ncc(C(N3CCCC3CNC(C3CC34CCC4)=O)=O)c2C1 CN1CC(O)CC1CNC1CCC(CNC(C2(N(C)C)CCOCC2)=O)CC1 c1(N(C(C)C)C(C2(CC3CC3)CCCO2)=O)ccc(OCC(C)(C)C)cc1 C1(CNC(Cc2ccc(C)c(Cl)c2)=O)CC2COCC2N1C(=O)CSCC(N)=O n1(CC)ccc(CC(N2CCC2CNC(=O)CNc2ncccn2)=O)n1 CC(CO)(C(=O)N1CC(C#N)C1)NC(c1ccc[n+]([O-])c1)=O N1(C(CCCSC(C)(C)C)=O)CCN(C)C(CNC(c2ccc(Cl)nc2O)=O)C1 c1(OC)ccc(OC(F)(F)F)cc1-c1nc(C)c(NC(=O)C=C(C)C)s1 C1(CC=O)CCCCC(=O)N1.c1(OCC)ccsc1C(=O)NCCC(C)C.N Cc1c(C(=O)N(CCN(C(=O)CC(C)O)C)CC)sc2cncn12.C(N)=O N1(C(C2CC(N(C)C)C2)=O)CCC(NC(=O)CCC2CC2(Cl)Cl)CC1 CC(CCCCNC(c1nccs1)=O)NC(c1cccc(F)c1)=O N1(C(c2nc(CC)oc2)=O)CCC(F)(CNC(c2sc(SC)cc2C)=O)C1 c1(CNc2cn(C(C(=O)OC)C)nc2)ccc(C2CC2)cc1C c1(N(CCOC)C)ncnc(NCc2nc(C3CC3)n[nH]2)c1C CC1=C(C(=O)NCC2(NC(c3csnc3Cl)=O)CCCCC2)CC1 c1(C(N2C(C)CCC(CNC(C3(C#N)CC3)=O)C2)=O)cnn2ccn(C)c12 c1(C(N(CC(C)CNC(=O)C=Cc2cc[nH]n2)C)=O)cnc(N)c(O)c1 CN1CSCC1C(=O)NCC1CCCN1C(c1ccc(CN=[N+]=[N-])o1)=O C(=O)(CC(C)P(C)(C)=O)NC1C(CC)N(C(c2sc([N+](=O)[O-])cc2Cl)=O)CC1 C=C(C)C(CC(=O)N1CCC2C(NC(c3cc(O)ncn3)=O)C12)OCC CC(C)(C)C(CC(=O)NC1CC2CCC(C1)N2C(=O)Cn1cnnc1)C(F)F c1(C(N(CC(CNC(C(F)=CCC)=O)C)C)=O)ccccc1.c1ccccn1.O c1(C(N2C3CN(C(CCCOCCC)=O)C(CC3)C2)=O)cccn2c(O)nnc12 Cc1cc(C(=O)NC2CC(CC)C2)on1.C1(C=O)CCCC1c1nc(S)n[nH]1.N c1(CC(=O)N)csc2cccc(Cl)c12.C1(C(=O)NCC2CC2)(CC)CC1 N1(C(C2C(OCC)C2(C)C)=O)CCC(O)C(CC(C)C)C1 CC(C(=O)N1CCC(F)(CNC(c2cnccn2)=O)C1)C(F)(F)F C1(NC(=O)NCCOc2ccccc2)CCC(Oc2nnc(CO)s2)CC1 C1(Cc2c(C(N3CCNS(=O)(=O)CC3)=O)cccc2)COc2ccccc2O1 C12(NC(CC)=O)CCN(C(c3cnc(C)n3C(F)F)=O)CCC1C2 C1(C(N2CC(C)C(C)C2)=O)CC(c2ccccn2)=NO1.C(C(=O)NC)NC(C)=O CC(F)CC(=O)NC1COCC1NC(=O)Cn1ccc(C2CC2)n1 c1(C(=O)NC(CC)CNC(C2(CF)CCOCC2)=O)nc(OC)cc(OC)n1 CCC(F)(F)C(C)(C)C(=O)NC(C)CCCNC(C12CC1Cc1c[nH]nc12)=O c1(N(C)Cc2cccc(C)n2)nc(=NCCC2CCCCO2)[nH]c2c1SCC2 C1(CC)CN(C(=O)C(C)O)CCC1NC(C1(O)CCSCC1)=O c1(C(=O)N)cc(N)c(F)cc1F.CC1(C)CCCC(C(=O)NCCC2CCC2)C1 Cc1sccc1C(=O)NCCN(C(=O)C(C)OC(C)(C)C)C c1(OC)ccc(C(=O)NCC2CC2NC(=O)CC(C)c2cccnc2)nc1 C(CC(C(=O)O)NC(=O)CCCC(=O)Nc1ccccc1)(OC)SC C1(CNC(C(C)OC)=O)CN(C(c2nccc3cc[nH]c23)=O)CCC1(C)C C(=O)C(C(F)(F)F)C(F)(F)F.c1(C(N2C(C)CC2)=O)cn2c(n1)C(C)CCC2.N CC1CN(C(C2CC(F)(F)CS2)=O)CCN(C(C2(c3cccnc3)CC2)=O)C1 C(=O)(C1=CCCCC1P(C)(C)=O)N.CN1CCCC1CCC(=O)NCCOCC C1(F)(CO)CCN(N(C)C2CCN(CCSc3ccccc3)CC2)C1 N1(C(c2ccc(C)nc2O)=O)CC2CC1CN(C(c1ccnc(C)c1O)=O)C2 CS(C)(=O)=Nc1ccc(C(=O)NC2CCCCC2NC(C2CCSC2)=O)s1 Cc1c(I)nn(C)c1C(N1CCC(CCO)CC1)C(=O)NCCCOC.C1CC1 C=C(C)CCC(=O)NCC1CCCCC1NC(c1cc(C)c(C)o1)=O N1(S(c2ccc([N+](=O)[O-])nn2)(=O)=O)CCC2(CC1)OCCc1ccccc12 C1(OC)CC2(C1)CC(C(N1CC(C)(C)CC1CNC(=O)C(C)CCO)=O)C2 c1(OC)ccccc1S(=O)(=O)N1CC2CN(C(c3cc(Cl)c(F)c(Cl)c3)=O)C2C1 Cc1cc(C(=O)NCC(O)CN(C)C(c2ncncc2Cl)=O)ccc1Br c1(C(N(C)CCC2CCCN2C)=O)ccc(-n2ccnc2)cc1 C1(CC2(c3cn(CC[Si](C)(C)C)nn3)CCC2)CCCCCN1 c1(-n2ccc(C)n2)ccccc1C(=O)NCC(O)CN(C)C(C1C=CCC1)=O CC1CC(C(=O)N)CCN1C(=O)CC1NC(=O)NC1=O.C1CCC2(CC1)CC2.C CCCC(C)(CC)C(=O)OC1CCN(CC2CCC(=O)N(C)C2)C1 Cc1scc(C(=O)NCCCCC(C)NC(=O)CN2CCC(C)C2)c1N N1(C(C(CCCC)NC(N)=O)=O)CCC(NCCO)CC(O)C1 c1(C(N2CCC(N(S(N(C)C)(=O)=O)C)CC2)=O)ccc(S(N)(=O)=O)cc1 N1(C(C2N(C(CC)=O)CSC2)=O)CCCC2(NC(C3(C)CC3(F)F)=O)CC2C1 N1(C(c2nc(OCC)oc2)=O)CCCN(C(=O)C(c2ccncc2C)C)CC1 c1(C(N2CCC(C(=O)Nc3ccno3)C2)=O)cnnc(Cl)c1 Cn1cnc2[nH]c(=NCCCC(F)(F)F)nc(N3CC4C(C3)C4(C)C)c12 C1(NC(C(C=CC)O)=O)CN(C(=O)C(CC)=CC)CCC1CO N1(Cc2ccc(OCC)cc2)CCCC2(CCN(C(c3cscn3)=O)C2)C1 c1(C(N(CCCCNC(C(C(CC)C)OC)=O)C(C)C)=O)cc2cccn2cn1 c1(C(N2CCC(C)C(NC(c3csc4nnsc34)=O)C2)=O)cccc2c[nH]nc12 CC1CN(C(=O)CCN2CCOCC2)CC1NC(c1ccc(-c2cccs2)[nH]1)=O Cc1cc(C(=O)N(C2(C(=O)NCC3(C)CC3(C)C)CC2)C)c(C)n1C C1(C(=O)N)CCC2(CCC2)CC1.C1(F)(C=O)C(F)(F)C1(F)F.CC=CC C(=O)(C(C)(F)C(=O)N1CCC(CNC(=O)C=C(C)C)C1)OC c1(OC)ncc(C=CC(=O)NC2CCN(C(=O)C(C)CSC)C2)cn1 CCC(CC)(CC)C(=O)N1CCC(CO)(NC(C2CCCOCC2)=O)CC1 C1(NC(C2CCN(CC(F)F)CC2)=O)C=CCN(C(=O)CN2CCCNC2=O)C1 Cn1cc2cc(C(=O)NCCC(N3CCCCCC3)=O)ccc2n1 C12(CC)CN(C(c3cnsc3)=O)C(CNC(=O)CN3CCCCC3)(C1)C2 C(=O)(CC(O)CCCC)NC1CC(C(N2CC3(CC(=C)C3)C2)=O)C12CCC2 C(=O)(C1=CC(C)(CC)C1)NCCCCC1CCCN(C(CCCC#C)=O)C1 C1CC2CC1CN(C(C1(F)CCC(F)(F)CC1)=O)C2.C(C=O)N(S(C)(=O)=O)C C1(C(=O)N(C)CCNC(C2CCS(=O)CC2)=O)(COC)CC=CCC1 Cc1cc(C(C)C(N2CC(F)(F)CC2C)=O)cc(F)c1.C1(C=O)CC(C)(O)C1 C1(CCNC(c2nc(C)oc2)=O)CCCCN1C(=O)CC1CCCN1C CCC(Cc1ccc(N)cc1)C(=O)N1CC2CC1C2NC(C1CS(=O)(=O)C1)=O Cc1cc(C)c(C(=O)NCCC2CC2)c(C)c1.C1(CC(=O)N)CCC(O)C1 C(c1cc(Br)cs1)=CC(=O)NC(CNC(c1cnsn1)=O)C1CC1 c1(C(=O)N(C2C(C(C=C)C)C2)C(C)CC)cccc([N+](=O)[O-])c1 c1(NC)c(C(N2CCC(c3cc(CNC(C)=O)on3)CC2)=O)cccc1N C#Cc1ccnc(C(=O)NC2CCCC2CNC(=O)C(C(=O)O)OC)c1.C N1(C(CCCc2scc(C)n2)=O)CC2(C1)SCCC2NC(=O)CC1(O)CCC1 C(C)(C)(CCCCNC(=O)C(F)=CC1CC1)NC(c1cccc(C)n1)=O c1(C(N2CCC(C)(C)C2)=O)cn2c(n1)CCCC2C.C(C(=O)NC)SCC=C N12CC3(CC(C3)C1=O)C2.Cc1cnc(CNC(c2ccc(Cl)cc2)C(C)C)cn1 c1(CN(C(=O)C(=O)Nc2cccc(C(N)=O)n2)C(C)C)ccc(Cl)c(Cl)c1 C(N(C)N1CCC(O)(SC)C1)c1ccc(OC)cc1 C1(CSCC(=O)NCC)CC2COCC2N1Cc1ccnc(C#N)c1 Cc1cc([N+](=O)[O-])cc(C(=O)N)n1.C1CN(C(C2CC2C(F)F)=O)CC1(C)C C1(CC(=O)N(CCCCC)Cc2ccccc2)Cn2ccnc2NC1=O C(CNC(c1ccccc1)=O)(C(C)(C)C)NC(C1C(OCC)C1)=O.S C1(N(C(c2cn(CC=C)nc2)=O)C)CCCC(N(C)C(c2ncn(C)n2)=O)C1 C(C)(C(O)C(=O)N(CCCCCNC(=O)CCC(=O)c1ccc(C)s1)C)OC C12(NC(CCSCC(C)C)=O)CC(C)(C1)C2.C(=O)(CC=O)N.C1CC1 c1(C(N2CC(NC(c3ccc4nccn4n3)=O)C(F)C2)=O)n[nH]c2c1CC1CC21 n1(CC)ncc2c1CC(C(N1CC3CCC1CN3C(C1CCS1(=O)=O)=O)=O)CC2 N1(C(=O)NC(CC)CC2CC2)CCC2(CCC(O)CC2)C1 CC(CN(C)C(c1cc(C(F)(F)F)n[nH]1)=O)S(C)(=O)=O c1(C(C(=O)NCCCC)N(C)CC2(C#N)CCCC2)ccc(CF)cc1 C(=O)(CCN(C)C)NCC(=O)OC(C)C.c1(C(C=O)C)ccn(C)c1.N C1(C(N2C(C)C(NC(c3c[nH]nc3[N+](=O)[O-])=O)CCC2)=O)CC12CCOC(C)C2 c1(CCCCC)ccc(C(N2CCC(N(C(=O)Cc3cc(C)on3)C)C2)=O)o1 CC(C#N)CN=c1[nH]c2c(c(=NC(C)Cc3cc(F)c(F)cc3F)[nH]1)CSC2 C1(C(=O)NC(C2(O)CCN(C(C3COC3)=O)C2)C)CCC(CCO)CC1 c1(C(N2CCC3CN(C(C4CC(O)C4)=O)CC23)=O)cc(Cl)c(Cl)cc1Cl C1(OC)CN(C(=O)C=CC(C)C)CC1NC(c1scnc1C(F)(F)F)=O c1(C(=O)NC2C3CN(C(CCCNC(C)=O)=O)CC32)cc(C2CC2)n(C)c1C C1(NC(=O)C(O)C(F)(F)F)CN(C(=O)Cn2ccc3ccccc23)CC(F)(F)C1 N1(C(C2(COC)CC(=C)C2)=O)CCC(C2CN(C(c3cscn3)=O)C2)CC1 CC1CCN(C(=O)CCOCC=CC(=O)OC)C1CO c1(C(C)C)ccc(C(=O)NC2CCC(NC(=O)CCN3CCCCC3)C2)s1 C1(NC(C2(C)CC(F)C2)=O)CCS(=O)(=O)C12CN(C(c1n[nH]cc1Cl)=O)C2 c1(OC)ccc(C(=O)NCCC(C)NC(C2(Cl)CC2)=O)cc1C n1(CC)c(=O)c(=O)[nH]c2cc(C(=O)OC(C)CCc3ccccn3)ccc12 CCC(CC(=O)N1CC(C)CC1C(N1CCc2nc[nH]c2C1)=O)C(F)F N1(C(CCC=CC)=O)CC2CN(C(C34CC(CO)(C3)OC4C)=O)CCC2(CO)C1 c1(OC)cnc(C(=O)N(C)CC2CN(C(C3COC(=O)O3)=O)CCO2)c(O)n1 Cc1ccsc1-c1cn(CC(=O)N(CCOCNCCO)CC)nn1 c1(OC)ccc(C)cc1CC(=O)NC(C1CCCCC1)C.C(=O)C(C)(C)C#N.N C1(NC(CSCCC(C)C)=O)CCC(N(C)C(c2csc(C3CC3)n2)=O)C1 c1(C(=O)OC)ccc(NC(=O)C=C2CCN(C)CC2)c(Br)n1.c1ccccc1C C=CC(CC)C(=O)NCC1CCC(NC(c2cnco2)=O)CC1 CC(C)S(=O)(=O)c1ccc(Cl)c(C(=O)NNC(=O)c2cc(I)n[nH]2)c1 C(=O)(C(C)CS(=O)(=O)N1CCCC(C)C1C(=O)OC)OC N(C(=NCC(CO)c1ccccc1Cl)NCC(=O)Nc1cccc(F)c1)C(C)C C1(NC(C(COC)(C)C)=O)CCN(C(c2cc(C)ncn2)=O)CC1O C1(NCc2ccc(C(=O)NCC)cc2)CCc2nn(C)cc2C1 c1(C(N2CCC(NC(C34CC(O)C3C4)=O)C2)=O)ccoc1I N1(C(C2N(N=O)CCC2)=O)CC2(CCCC2NC(=O)CCN2CCCS2(=O)=O)C1 c1(C(N2CC(NC(c3cccc(F)c3F)=O)C2)=O)cnn2ccncc12 c1(CN2CC(C(=O)NC(CCC)CO)SCC2)ccc(Cl)c(I)c1 CCC(C)C(C(=O)NCC12CCCCC1C2)N(C(=O)Cc1ccon1)C N1(C(C(COC)(C)C)=O)CC2COCCC2(NC(c2cccc(C)c2N)=O)C1 C1(C(=O)NC(C)CC#N)CC2CC2N1Cc1csc(Br)n1 n1(CCCOC)cc(CC2CN(C(c3nc(I)cs3)=O)C2)nn1 CCC(COCC1CC1)NC(=O)C(C)N(C)C(C1CCC1C)=O C1(C(=O)NCCCC=C)CCC(C)(O)CC1.C1(C(F)(F)F)(C=O)CC(=C)C1 Cc1ccc(C(=O)NCC(CC2CC2)C(=O)NCC(c2ccco2)O)c(O)c1 Cc1c(-n2cc(C(C)(C)NC(c3ncnc(O)c3F)=O)nn2)cccc1Cl n1(CC)ncc(C(=O)NC)c1C1CC1.C1CC(F)CN1C(=O)C.C(C)C C1(CC)CCN(C(=O)Cc2cccnc2)C1CNC(=O)CC(C)F CC1CCC(C(=O)NC2CC(NC(=O)C(C)NC(C3CCOCC3)=O)C2)CC1 C(=O)(C(C)C(=O)N1CCOC(CNC(c2ncoc2C2CCC2)=O)C1)OC O=C(CCC(=O)c1ccc(Cl)cn1)NC.C1C2CN(C(C3CC(F)(F)C3)=O)CC12 CN1CCC(CC(N2CC3CC2C3NC(C2CN(C(N)=O)C2)=O)=O)CC1 C1(C(N(CCOC)C)=O)CC(F)CN(C(c2ncc(Br)cc2Br)=O)C1 N1(C(c2[nH]cc(C)c2)=O)CC(F)(F)CC1C.n1(CC=O)nnnc1C1CC1.N Cc1cc(C(N2CC3CC(N(C)C(c4n[nH]cc4C)=O)C2C3)=O)n2nccc2n1 C1(CC(=O)NCCC(C)NC(Cc2c(C)cccn2)=O)CCC2(CCC2)O1 c1(C(N2CCC(N(C(=O)C(c3ccc(C)s3)C)CC)C2)=O)cc2c(o1)CCCC2 c1(C(N2C(C)(CNC(=O)Cc3n[nH]c(=N)s3)CCC2)=O)ncc(Br)cc1F C1(N(C)C)(C(N2CC(F)(CNC(=O)CCC3CCCO3)C2)=O)CCCSC1 c1(CC(N2CC(NC(c3cnc(Cl)c(Cl)c3)=O)C(O)C2)=O)cc(F)c(F)cc1F n1(CC)nc(C=O)c(C)n1.c1(C(N(CC)C)=O)cc(C(C)(C)C)c[nH]1.CC C(c1ccccc1)=CC(=O)NC(C)(C)CCCNC(C1(C)CC1(F)Cl)=O.C C(CC)(CCCC(=O)Nc1cnc(C)c(C#N)c1)NC(C1C(CCC)C1)=O CCCCCC(CC)C(=O)N1CC2=C(C1)CN(C(C1CCC(C#N)CC1)=O)C2 N1(C(c2[nH]nnc2C2CC2)=O)CCC2(CC1)CN(C(=O)COc1ccccc1)C2 c1(C(=O)NC(CN(C(C2CC(CCO)C2)=O)CC)C)cc(N)cnc1Cl C=CCC(C(=O)NCCC1CN(C(C2(C)CCCCC2)=O)CCO1)NC(C)=O C=CCCC(C)NC(=O)Cn1cccc1.c12cn(nn1)C2.C1CC2CC2C1 N1(C(c2cnc(C)s2)C(=O)NC2CC2)CCC2C(CCCN2C)C1 c1(OC)cc(C(=O)NC2CN(C(=O)CC(C)n3cccc3)C2)nc(C)c1 c1(COC(c2cc(S(N)(=O)=O)sc2Cl)=O)ccc2ccccc2c1O c1(CC)ccc(N)c(C(=O)NCCC2CCN(C(c3ncoc3C)=O)C2)c1 c1(CCCC(=O)NCC(CNC(=O)CC(C)CF)OC)c(F)cccc1F C1(NC(c2c(COC)cco2)=O)CN(C(=O)CP(C)(C)=O)CC12CCC2 C(=O)(C(O)CNC(=O)CC1CSC1)N1CC(CN(C)C)C1 c1(C(N(CC(N2CCCC2C(N)=O)=O)CC#C)=O)cc2ccccn2c1 N1(C(C2N(C(=O)CC3CC(F)C3)CCN(C)C2)=O)CCc2c(O)noc2C1 c1(C(=O)NCCCN(C(=O)COc2ccsn2)CC)sc2sccc2c1Cl Cc1ccnc2c(C(N3CCC4CCN(C(=O)C(C)(F)F)CC34)=O)cnn12 Cc1ccc(CC(=O)NCC(C2(O)CCN(C(c3ccco3)=O)C2)C)cc1Cl C#CC1CCCC(CNC(c2c(C)cnn2C)=O)C1.C1(C(=O)N)CN2CCC1C2 C1(NC(=O)Cc2c[nH]ccc2=O)CC2CN(C(=O)C)CC2C1.C(=O)C(F)(F)F.N c1(C(=O)NCC2C3N(C(C(CCC)OC)=O)C(CC3)C2)cc2n(n1)CCOC2 Cc1cn(C)nc1Cn1cc(CCC(=O)NC(Cc2csc(Br)c2)C(=O)O)nn1 C1(C(N2CCC(NC(c3ccc(OCCO)cc3)=O)C2)=O)CCc2cnnn2C1 C(=O)(C(F)(F)c1csc(=N)[nH]1)N(C1CN(C(C2C(C(C)O)C2)=O)C1)C CC(CCO)C(=O)NCC1CC(F)(CNC(=O)C(c2ccccc2)C)C1 CCCCCC(=O)NC1CC1NC(C1(COC)CC(F)(F)C1)=O C1(NCCOC)CN(C(=O)NC23CCCC2CCC3)CCC1=O C1(C)(C(=O)NCC(CO)NC(C(CN(C)C)O)=O)CCOCC1 c1(OC)c(F)cc(NCc2cnn(Cc3ccccc3)c2)cc1F c1(NC(CN2CCN(C)C(C)(C)C2)=O)ccc2c(c1)OC(F)(F)O2 N#Cc1ccccc1C1(C(N2CCCCCCC2C(=O)NCCF)=O)CC1 C(=O)(C1=C(Cl)CCOC1)N1CCCC(C)(NC(c2cc(C3CC3)no2)=O)C1 c1(OC)ccc(C(c2nnnn2C2CC2)NCC(C)(C)c2cccs2)c(OC)n1 CC(F)(F)C(F)(F)F.C1(NC(C(CC)OC)=O)CCC(N(C(=O)CCO)C)CC1 C(C(C)(C)C(=O)NCC1CCCCC1)OCC.c1(CC=O)ccccc1.C c1(C(N2CC3CN(C(C(CCOC)OC)=O)C3CC2)=O)ccc2nc(C)sc2c1 c1(OCC(=O)NCCC2(NC(C3CCOC3=O)=O)CC2)ccc(F)cc1 c1(NC(N2C(c3ccc(C)cc3)CCC2)=O)c(F)cc(F)cc1Br CCC(C(=O)NC1(C)CC(NC(=O)C(C)CSC)C1)Sc1nc(=N)[nH][nH]1 CC1(C)CN(C(=O)Cc2ccn3cncc3c2)CCC1NC(C1CCOC1=O)=O C1(C(=O)NC(CC)(CNC(C2CC3CCC2O3)=O)CC)CCCCC12CCC2 c1(C(C)=O)ccc(CC(=O)NC2CC(F)C2)s1.C1(C=O)CCOC1C(C)C.C c1(OC)ncccc1CN(c1nccc(N2CC(CO)C(CO)C2)n1)C N1(C(CCC(C)OC)=O)CC(C)(C(N2CC(F)(C3CC3)C2)=O)CC1(C)C N1(C(c2ccc(N)c(O)c2)=O)CCCC(NC(=O)CCC(F)F)C(F)C1 C(CCCCC(=O)NCC(C1CC1)NC(=O)C=Cc1cnc(C)s1)OCC Cc1cn(CCO)nc1NC(=O)C(O)C(C)C CC1CC(NC(=O)C(=O)Nc2ncc[nH]2)CN(C(=O)C=CC2CC2)C1 CC(C)(CCCC(=O)N1CCCC(CCO)C1)NC(C1CC2CCC1C2)=O Cc1cccn2cc(C(N3CCC(C)C(CNC(=O)C=CCF)C3)=O)nc12 C(=O)(C(C)(C)S(=O)(=O)C1CC1)N1CC2(CN(C(c3c(F)cccc3)=O)C2)C1 c1(C(=O)NC(C(C)C)CCNC(c2cnnc(Cl)c2)=O)c(F)ccc(F)c1F Cc1cc(C)n(CCNC(C2CC(O)C2)=O)n1.C(=O)CCC1CC(C)C1.C c1(C(=O)NCC(CCOC)NC(c2cc(C)sc2C)=O)c[nH]c2cccc(Cl)c12 CN1CCN(C(c2ccc(C(F)F)o2)=O)C(CNC(C2(CC)CC2)=O)C1 c1(OC)cccc2c(C(N3CCC4CC3CN4C(=O)CCCN(C)C)=O)cnn12 n1(CC(N2C(C)CCC2)=O)cccc(N)c1=O.C(C(=O)N)=CCN(C)CC n1(COC)nccc1-n1cc(CNCC2(C)CC2Br)nn1 C1(C(C)C)CN(C(C2CC(O)C2)=O)CCCN1C(=O)C(C)c1cccs1 C1(C)CCN(C(=O)Cc2ccccc2)C1.C(C(O)C(=O)N)OC.[SH](C)(=O)=O CCC(C)(C)CC(=O)NC1COCC1CNC(C1CN(S(N)(=O)=O)C1)=O C12(C(N3CC(C)CC3)=O)CCCC(C)(C1)OC2.C1(CC=O)CCC(C2CC2)O1.N C1(C(C)C)CN(C(c2ccccn2)=O)CCN1C(c1ccc([N+](=O)[O-])o1)=O N1(C(COCCOCC)=O)CCC2CC12.c1(N(CC=O)C)ccccc1.C C1(CNC(CSCC)=O)CN(C(=O)CC(O)c2ccccc2)CC12CCC2 N1(CC)CCC(N(C)C(C2CCCC2NC(C2COCC2(C)C)=O)=O)CC1 C(N=c1ccc(=O)n(CCO)[nH]1)c1occ(C(=O)O)n1 C1(C(N2CC(C(N(C)Cc3ccncc3F)=O)OCC2)=O)CC2CCC1CC2 C1(C(=O)NCC2(OC)CN(C(c3ccc(C#C)cn3)=O)C2)CN2CCN1C(C)C2 C(=O)(C1=CCCCCC1)NC(C)CCNC(=O)C=Cc1ccncc1 Cc1cc(C(=O)NCC2CCCCN2C(=O)C(N2CCCCCC2)C)cnc1C c1(NC(=O)NC2CCCN(c3ccc(C)cn3)C2)ccc2nc[nH]c2c1 c1(C(C)C(=O)N(C(C)C)C)ccc(Cl)cc1.c1(CC=CCC(=O)N)ccccc1 Cc1cccc(C(=O)NC2(C3CN(C(c4cncs4)=O)C3)CC2)c1Br C(CCC(=O)NCCC(O)CNC(c1ncoc1C(C)(C)C)=O)OC(C)C C1(CCNC(=O)C(CO)NC(=O)C=Cc2ccccc2)CN(C(=O)CO)CCO1 CCCCC(C)C(=O)NC(C)CCCNC(c1ccc(CC)nc1C)=O Cn1ncc(C(N2CC=CCC2C(N2CCC2CF)=O)=O)c1Cl Cc1ccc(C(C)C)c(C(N2CCC(NC(=O)Cc3sccc3Cl)C2)=O)c1 N1(CC)C(=O)CCC1C(=O)NCC(c1ccccc1)NC(c1nonc1)=O c1(OC(C)C)ccc(Cl)cc1C(=O)NC1CC1.c1(C(=O)N)n[nH]c2c1COC2 C1(C(NOC(C)C)=O)CC12CCN(C(c1cccn1C1CC1)=O)CC2 c1(C=O)coc2c1C(O)CCC2.c1(CC)cscc1C(=O)NCC1CC1C c1(C(=O)NCCNC(c2csc3cncn23)=O)ccc2nc[nH]c2n1.C1CC1.C CC1CCCCN1C(=O)CN1CC(C)(C)C1.c1(C=O)cc(C(C)(C)C)nn1C.N Cc1cc(=NC(=O)C(=O)NC(CC(C)C)C(F)F)[nH]o1 c1(C(N(CCOC)CC)=O)cccc(C)c1.C(=O)(CC)N.[SH](C)(=O)=O c1(CNC(c2cccc(CN3CC(C)OC(C)C3)c2)=O)cc2ccccc2[nH]1 n1(CC)cc(Cl)cc1C(=O)NCC(C)C(C)C.C1(C(=O)N)CC(C)(C)CO1 Cc1cccc(OCC(=O)N(C2CN(C(c3c[nH]c(=N)s3)=O)CC2F)C)c1 c1(NCC2OCCC2)ccc(SCC2CC2)cc1 N1(C(C(CC)C2CC2)=O)CC2CCCCC2(CNC(c2c[nH]nc2OC)=O)C1 Cc1nc(N2CCCC2CNC(=O)C(c2c(C)n[nH]c2C)C)c2c(C)csc2n1 C(C(C)(C)CCN(CCO)CC1CCN1)OC C(C1(CNC(c2cc(C(C)(C)C)ns2)=O)OCCc2ccccc21)OC CCC(O)C(C)C(=O)N1CCC(COC)(NC(c2c(Cl)c(C)nn2C)=O)C1 c1(C(N2CC(C)(NC(C3CCCC34OCCO4)=O)C2)=O)ccc2nc(O)[nH]c2n1 C(CC(=O)N(C(C)C(=O)N(CC(O)COC)C)C1CC1)=C.CCCN(C)C C(=O)(C1=NOC2COCC12)NC(CC(=O)NC1COCCC1(F)F)CC1CC1 c1(OC)cccc2[nH]nc(C(=O)NC(C)CN(C)C(C3CCC34CCC4)=O)c12 C#Cc1ccc(CC(=O)N(C)Cc2c(Br)cnn2C)cc1 C1(NC(c2c(CC)scn2)=O)CN(C(c2cc(Cl)no2)=O)CC1C1CC1 CC(O)C(F)(F)C(=O)N1CCC(C(=O)NCCC2CCCC2O)C1 c1(OC)cc([N+](=O)[O-])ccc1C(N1CCS(=O)C(C)C1C)C(=O)NCC1CC1 CCCC(C#N)C(=O)N1CCCCC(C(N2CCN(C)C(CO)C2)=O)C1 N1(C(CCC2(CCC#C)N=N2)=O)CCCC(CCNC(c2n[nH]c(=N)[nH]2)=O)C1 CC1CCCCC1CNC(=O)C=CC1CCCC1.c1(CC=O)nnc(O)s1.N C(C(C)(C)CNC(=O)CNC(=O)NC)NC(C(C)OCC=C)=O C(=O)(C(C)(O)C(C)(C)C)NCC1N(C(Cc2c(C)nc(C)s2)=O)CC(O)C1 Cc1cc(NC2C3CN(C(c4cnn(C(F)F)c4)=O)CC23)ncn1 c1(C(N2C(CCC(=O)N(CCO)CC)CCC2)=O)cc(F)n(C)n1 CCCC(C)(C)CC(=O)NC1CS(=O)(=O)CC1C(F)(F)F.C1CC1.C1CC1 C(=O)(C(CC(N)=O)NC(c1cc(C#N)c[nH]1)=O)NC1(C#C)CC1 C=C(C)CC(C(=O)NCC(C)(C)C1CCCC1)NC(C1CC=CC1)=O CC1(C)COCCC1C(=O)NCC(O)CC(=O)N1CC(OCC(F)F)C1 Cc1c(C(=O)NC2CCCC2)c2ccccc2n1C.C(=O)(C(C1CC1)N(C)C)N C1(CNC(C2CC3CCC2C3)=O)CC2(CO1)CN(C(C1CC3CCC1CC3)=O)C2 N1(C(CCCCC)=O)C2CCC1CN(C(=O)C(C)NC(=O)NC1CCCC1)C2 c1(N(CC)CC)ccc(C(c2nnnn2CCCF)NCCC(F)(F)Cl)cn1 Cc1occc1C(=O)NCC=O.C1CC(CC)C1.C(=O)CN(C)C1CC1.N c1(C(=O)NCC2C(C(=O)NC(C)C(=O)NO)C2)cnn2c1OCC2 C1(NC(Cc2n(C)ncc2)=O)CCCCC1NC(c1ccc(F)cn1)=O C(C1Cc2ccccc21)NC(C1(C(C)C)CCN(C(C(CC)CC)=O)C1)=O C1(NC(c2cnn(C3CCCC3)c2)=O)CC(F)CN(C(=O)C=C2CCC2)C1 C1(CNC(C=Cc2ccc(SC)s2)=O)CCC(C)N(C(=O)CCCF)C1 C(CCF)(C(=O)NOCc1ccccc1)NC(C(CCN(C)C)(C)O)=O c1(C(=O)NCC2OCCN(C(C3C(CC)CCC3)=O)C2)ccc(C)cc1N=[N+]=[N-] c1(OCC)ccc(C(N2CCCC2)=O)cn1.c1(N(C)C)ccnc(C(F)(F)F)n1 CCC(C(=O)NC1(C)CC(C(=O)NC)C1)N(CC)C.c1nncn1C(C)C C1(CNC(c2cccnc2)=O)CC2CC(C1)N(C(c1cccn3cncc13)=O)C2 C(=O)CS(=O)(=O)C1CCCC1.C=C=CC(C)C(=O)NCC1(F)CC(C)C1.N CC1(C)CCCN1C(C1CC(C2CC2)=NO1)=O.c1(CC(=O)N)c[nH]c(=N)nc1O CC1(CNC(=O)C(O)c2ccsc2)CCN(C(=O)C=Cc2cc[nH]n2)CC1 CC(CC(N)=O)C(=O)NCC1CC(NC(c2cc(=N)[nH]c(Cl)n2)=O)C1 N1(C(c2nc(OC)oc2)=O)CC2CCC(NC(C3CC34CC(C)(C)C4)=O)CC2C1 Cc1cc(C(=O)NC(C)(C)CNC(=O)C(C)C)cc(C)c1 Cc1cc(C(=O)NCc2ccc(-c3cccc(S(C)=O)c3)cn2)cc2[nH]ccc12 c1(C(C(=O)NC(C(C)NC(C=CCC)=O)C)O)ccccc1 C(=O)(CCC(C)(C)C)N(C1CCN(C(c2cc(C(C)=O)[nH]n2)=O)C1)CCC Cc1c(F)ccc(Cl)c1C(=O)N.C1(C)(C=O)CC(F)(F)C1.C1(CC)CCOC1 c1(C(C)NC(C2CCCO2)CN(C)C)cc(Cl)ncc1F Cn1oc(C(=O)NCCCNC(c2ccc(OC(C)(C)C)cc2)=O)cc1=O c1(C(CNC(CN(C)CC)=O)NC(=O)C(C(C)C)SC)cccc(Cl)c1Cl C1(C(=O)N(C)CCC2CCCCN2C(c2ccc[n+]([O-])c2)=O)(OC)CCCCC1 C1(OCC)CCN(Cc2ccccc2C2CCC2)CC1(C)C C(=O)(C1=C(C)OCCC1)NCC(C)CC(=O)NC.C=C1CC2(C1)C(=O)NOC2 Cc1cc(C(N2CCC(C(C)NC(c3cccn3C3CC3)=O)C2)=O)ccc1Br c1(NC2C3CN(C(c4cc(CCC)oc4C)=O)CC32)ncnc2c1CCCC2 c1(C(=O)Nc2ccc(Cl)cc2O)ccc2nc(C(F)(F)F)[nH]c2c1 C(C)(C)C(F)(F)F.C1(C(N(CCC)C)=O)CCC1C(F)(F)F.C(=O)C.N NC12COCC(CN(C(c3cn(CC4CCc5ccccc54)nn3)=O)C1)C2(F)F Cc1c(F)ccc(N)c1C(=O)NC(C)CC.c1(C(=O)N)c[nH]nc1C1CCCO1 c1(CNC(C)CSc2nncn2C)cn2cc(Cl)cc(Cl)c2n1 Cc1cc(C(=O)NCC(C)(C)C(=O)NCCCN2CCCC2C)cc(C)n1 C(=O)(C1OCCn2ccnc21)N.CC1(C#CC(=O)NCC2CC(O)(C)C2)COC1 C1(C(=O)OC(C)(C)C)CC12CCN(C(c1sccc1S(N)(=O)=O)=O)CC2 C1(C=O)CC2(CCC2O)C1.C(=O)(CCOC1CC1)NC(C1(C)CC1)C Cc1cc(C(N2CC(CCc3cn(C(C)CO)nn3)C2)=O)nn1-c1ccccn1 Cc1nsc(NCC2CCCN2C(c2cc3occc3s2)=O)c1C#N CP(C)(=O)COCCc1cn(CCSC2CCCN2S(C)(=O)=O)nn1 Cc1ccc(C2CC2C(N2CCN(C(c3ccc(Cl)s3)=O)CC2CF)=O)c(Cl)n1 N1(C(C(C)n2cncn2)=O)CC(O)CC1CNC(C1CC2(CC2)C1)=O CC1ON=C(C(=O)NC(C)C(C)(C)NC(c2cc3occc3s2)=O)C1C N1(C(C2CCC(=C)CC2)=O)CC(NC(c2nccc(C)n2)=O)CC12CCOC2 CC1(C(=O)OCC(c2ccc3c(c2)CCCC3)=O)CC(c2ccccc2F)=NO1 Cc1cc(C(N2CC(C)(NC(c3cnn(CCO)c3N)=O)C2)=O)nc(N(C)C)n1 CC(C)(CC(=O)N1CCCC(Cn2cc(CCC3CCCC3)nn2)C1)C(F)(F)F C(=O)(CCC(=O)NC(C)C)OCC.c1(C(=O)N)ccc(N2CCCCCC2)cc1 C1(C(N(CCCCC)C(C)C)=O)CC(CC)CCN1C(=O)C(C)CCCOC N1(C(=O)C2=CCSC2)CCCC1C1CCCN1C(c1cccc(CCO)c1)=O c1(C(N2CCOCC2)CNC(C)Cc2cccs2)cccc2c1S(=O)(=O)CCC2 C(c1cccc(CO)c1)=C(C)C(=O)NC(CNC(=O)Cc1cc[nH]n1)C(C)C c1(C(N(C2CCC(NC(c3cnc[nH]3)=O)CC2)C)=O)ccc(S(N)(=O)=O)cc1 N1(C(CC(c2cccc(OC)c2)C)=O)CCC2CCC(C1)N2C(=O)C1=COCC1 CCC(C)CCCCC(=O)N1CC(C)CCC1C(=O)NC1CCN(OC)CC1 CCC(C(=O)OC)C(=O)NCc1ccnc(C(=O)NC2CC23CCCC3)c1 O=C1NC(C(=O)N(CCC(=O)NC2(c3nn[nH]n3)CC2)CCO)CO1 C1(CNC(C(CCC)C)=O)CN(C(c2cc(SC)ccc2O)=O)CC1(C)C C(c1ccc(C)cc1)=CC(N1CCC(CC(N2C(C=C)CCC2)=O)C1)=O C(=O)(CC(F)(F)C(F)F)NC(C1CC1C(N1CC=CC1CF)=O)C c1(CCC(=O)N)ccccc1[N+](=O)[O-].C(C(O)C(=O)NCCC1CCC1)=CC C1(CC)CN(C(=O)CSCCC(C)C)CCN1C(=O)Cc1ccnc(OC)c1 C(=O)(C1=NN(C)C(=O)CC1)N1CCC(=C)CC1C(=O)NC1CC1c1ccccc1 CCC(O)CNC(=O)C(c1ccoc1)NC(=O)Cn1ccnc1 C1(NC(c2c(OC)cc(C)s2)=O)(CO)CCCN(C(C2CCOC(C)C2)=O)C1 C1(C)(C=O)CCCO1.C1(CN(C)C(=O)NCC(=O)NCCCO)CCCC1 C1(NC(CS(CC)=O)=O)CCC(C)(NC(c2cnc(C)c(N)c2)=O)CC1 N1(C(c2c(C)nn[nH]2)=O)CCC(NC(C2(C(C)C)COC2)=O)C(C)(C)C1 C(CC(N=c1nc2c(ncn2C)c(NCc2cnc(C(C)C)s2)[nH]1)C(C)C)OC N1(C(C(CCC)OC)=O)CCC(CNC(C2(n3nccn3)CC2)=O)C12CCC2 C1(CNC(CN(C)C(N)=O)=O)CCN(C(c2csc(C#N)c2)=O)CC1(F)F c1(C(=O)NC2C3(CN(C(C(CC)=CC)=O)C3)CC2)ccc2cc(F)ccc2n1 CC1c2cc(F)cc(F)c2CCN1N1CC(CO)(CO)C1 c1(CNC(N2CCc3ccc(Br)cc32)=O)cn2c(F)cccc2n1 CC1Nc2ccnn2C(C)C1CCC(=O)NCc1cc2c(s1)CCOC2 c1(C(N2CCC(CN(C(=O)CCn3cnnn3)C)C2)=O)cc[nH]c(=N)c1[N+](=O)[O-] c1(C(=O)NCC(CC)C)cc(C(C)C)oc1CC.C(=O)CC(C)C1CCCC1.N C1(NC(C(C)SC(F)(F)F)=O)CCN(Cc2cn(Cc3cnns3)nn2)C1 C1(NC(C(C=CC)O)=O)CN(C(c2c(C3CCC3)cnn2C)=O)CC1(C)C c1(C=O)ccc(CCF)cc1.CC(C)(C(=O)NC1CCCC1)OCC(F)(F)F.N C=CCC(C)C(=O)NC1CC1NC(c1ccc(N2CCOCC2)nc1)=O C=CCCC(F)(F)C(=O)NC1CC=C(C(=O)NC(C)C(=O)NCCC)C1 N1(c2nccc(C)n2)C2CCC1CC(CNC(C1CCCC(F)C1)=O)C2 c1(CC)ccc(C(=O)NC2CC(NC(=O)CCC3CCCO3)C2)s1 C=CCC(CC)C(=O)NC1CC2CC1N(C(c1c(C3CC3)noc1C)=O)C2 c1(C(=O)N)ccc(F)c(C)c1N.CCC(CN(C)C)CC(=O)N(C(C)C1CC1)C c1(C(N2CCCC(N3CCCOCC3)C2)=O)cc2ccc(Br)nc2s1 C1(NC(C2CC2F)=O)CS(=O)(=O)C12CCN(C(=O)Cc1ccc(Cl)s1)CC2 C1(C(=O)NCCCC(F)(F)F)CN(C(=O)CN2CCCCC2)CC1C1CC1 N1(C(C(CC=C)C)=O)CC2(CCC2NC(=O)CCn2nc(C)c(C)c2C)C1 C(CC(=O)NCC1CCC(=O)NC1)(C(C)(C)C)NC(C1C(C)(C)CCO1)=O N1(C(c2nnc(C)s2)C)CC2CN(C(c3cnc(C(C)C)s3)=O)CC2C1 C1(CNC(c2c(CC)onc2)=O)CCCCC1NC(=O)CCC(F)F c1(N(C(=O)CCCC2CC2C)CC)cc(F)cc(Cl)c1 C(C(CC(C)C)C(=O)N1CCC(C(=O)NC(C)CC2CCCCC2)C(C)C1)OC c1(OC)cc(OC)cc(NC(=O)CC2CCCN2Cc2ccncc2O)c1 C1(C(=O)NCCCNC(C2(c3ccc(C)cc3)CCC2)=O)CCC2CC2CC1 N1(C(C2CCc3nncn3C2)=O)CCCC2C1CCCCN2C(c1cc[nH]c1)=O N1(C(CC2(CN(C)C)CCC2)=O)CC2CC(C1)N(C(c1cc[nH]c(=N)c1)=O)C2 C1(CC(N2CC(NC(c3cc(C)n(C)c3)=O)CC2C)=O)(OC)CCOCC1 N(C1CCCc2cc(CNC(C3CCC(C)CC3)=O)ccc21)C(C(OC)OC)=O c12cccc(c1)NC2=O.c1(C(C(=O)N(C(C)C)CCF)C2CC2)ccccc1 C(=O)(C1=C(Cl)CCC(C)C1)NCC1OCCN(C(c2cn(C(C)C)nc2)=O)C1 C1(NC(Cc2cc(C)no2)=O)CN(C(C2CCC(=O)N2C)=O)CC1C#N C(N=c1cc(Cl)nc(S(C)(=O)=O)[nH]1)C1(NC(CC2(O)CC(C)(C)OC2)=O)COC1 N1(C(c2c(CC)sc(=N)[nH]2)=O)CCN(C(=O)CCC2CC2(Cl)Cl)CC1CO C(=O)(C(F)CC(C)C)NCCCN(C(c1cc(N)cnc1C)=O)CC C1(NC(C(=O)N(CC)CC2CCCCC2)=O)CCC(S(C)(=O)=O)CC1 C(=O)(C(C(C)C)c1ccc(Cl)cc1)N(C(CNC(Cc1cc(C)sc1)=O)C)C C(=O)(N=c1cc(C(N)=O)n(C)[nH]1)C1(CCOC)CC1.C1(C=O)(CC)CC1 c1(N2CC3N(C(c4c(OC)ccs4)=O)C(CC3)C2)ncnc2ccc(Br)cc12 C(CCN=C(NCC1CC1[N+](=O)[O-])NC1CCCCC1)c1ccc(OC)cc1 c1(C2(C(N3CCC(CC)C3)=O)CC2)ccc(F)cc1.c1(OC)cc(C=O)[nH]n1.N N1(C(C(CCC#C)O)=O)CC2CC(NC(c3ccc(S(C)(=O)=O)s3)=O)CC1C2 C(=O)(CC(C)NC(=O)CC1(NC(C2CCCCC2)=O)CCC1)OC N1(C(c2cncc(OC)c2)=O)CCN(C)C(C(=O)N)C1.C1COCC1N(C)C.C c1(NC(CC#CC)C)nc(=NCCN2C(=O)CNC2=O)[nH]c2c(C)nn(C)c12 C(=O)(CS(=O)c1cccc(OC)c1)NCC1(C(F)F)CCN(C(COC)=O)C1 c1(C(=O)NCC(CNC(C2C(C)OCCO2)=O)C)c(O)cnc2ccc(F)cc12 c1(C(=O)NCCC2CC(NC(C=C(CCC)C)=O)C2)cn(C)nc1C(F)F CCCC(CCCNC(=O)CCCN1CCCC1)NC(C1(CC(F)F)CC1)=O C1(CNC(CCOC(C)C)=O)C(C)CCN1C(=O)C=Cc1ccnn1C c1(NC(=O)NC(C(C)C)CO)cnc2[nH]cnc2c1 C1(CC=C)(NC(=O)C2=C(C)OCC2)CCN(C(=O)C=Cc2ccccc2Cl)CC1 C1(NC(c2cn(C)[nH]c2=N)=O)CCC12CCN(C(C1C(F)(F)C13CC3)=O)CC2 c1(C(C)NC(=O)Nc2cnc(I)cn2)ccc2c(c1)CCCC2 N1(C(c2cc(CC)on2)=O)CC2CCC1CN(C(c1ccnc(F)c1Cl)=O)C2 CCCC(C(O)C(=O)NC(CO)(CO)CO)NC(c1cc(C(C)C)on1)=O NS(=O)(=O)CC(=O)NCCNC(=O)CCc1ccoc1 c1(CC(CO)NC(CC)C(=O)N(C)C)ccc(F)cc1 c1(C(=O)NCC(C(C)C)NC(C2CCSC2)=O)cnc(O)c2ccsc12 c1(C(N(CCN)CCNS(=O)(=O)N(C)C)=O)ncnc2sccc12.CC N1(C(Cc2c(C)ncs2)=O)CC(F)CC1CNC(c1cccnn1)=O.C(C)C.N C1CC(C)CCN1C(c1cc(C2CC2)ns1)=O.n1(CC)ccnc1C(=O)NC n1(CC)nnnc1C(C)(CCC1CC1)NCCCOC(c1ccccc1)C C(=O)(C1CCSc2ccccc21)N(CCCNC(c1cnco1)=O)CCO C(CC(C)C)(C(=O)N1CCCC1CNCc1c(O)cccc1Cl)NC(C)=O C(c1c(F)cccc1F)=CC(=O)NC12CCC(C1)N(C(c1cccc[n+]1[O-])=O)C2 C(N=c1cc(Cl)c(O)n[nH]1)C1(CCNC(c2c(C)cccc2)=O)CC1 C1(C(=O)NC2CCC3CC23)(CC)CCN(C(=O)CCc2cc(C)no2)CC1 N1(C(C(C)OCC)=O)CCC(CCn2cc(-c3cccc(Cl)c3)nn2)CC1 C1(C(=O)NC2(C)CCCCC2)CCN(C(c2nc[nH]n2)=O)CCO1 c1(C(=O)NC2C(NC(C(CC)N(CC)CC)=O)CCC2)sc(F)cc1Br c1(CN2C(=O)CN(CC(C3CCOCC3)OCC)C2=O)cccc2ccccc12 Cc1cc2nc(Cl)[nH]c(=NC3CC(F)(CNC(=O)CCc4nc[nH]n4)C3)c2s1 c1(C(N2CCC(O)(CN(C)C(c3cn[nH]c3)=O)C2)=O)ccc(Br)c(N)n1 CC1CCC(NC(c2ccc[nH]2)=O)CN1C(=O)CN1CCCC1 C1(CNC(c2coc(Cn3cc(CCCCCO)nn3)c2)=O)CCCCC1(F)F Cc1ccc2c(C(=O)NC(C)CCNC(C3CC34CC4)=O)c(C)ccc2c1 c1(NC(C(=O)NCC2C(N)CC(CO)CC2)=O)ccc2c(c1)Cc1ccccc1-2 C(=O)(CCC(F)(F)F)N1CC=CC(NC(c2cn(C(F)(F)CO)nn2)=O)C1 c1(OCC(=O)NCCCN(C(C2C(C)CC2)=O)C)ccc(Cl)cc1F C=C(Br)CC(C)(C)C(=O)N1CCC(CCNC(=O)C(C)NC(=O)CC)C1 c1(CN(C)C(c2ccc(C)cn2)=O)cccc(O)n1.C1(C(=O)N)CCC1(F)F C=CCCCCCC(=O)N1CCCCC1CNC(C1NC(=O)CC1C)=O c1(SC)cc(F)ccc1C(=O)NCC1CCCCN1C(C1(C2CC2)CC1)=O Cc1ccc(Br)cc1C(C)NCC1CC1.C(=O)(CC)N.C(C)(C)C.C=O C1(CC=C)CCN(C(C2(NC(=O)CNC(=O)CC)CC(O)C2)=O)C1 C1(CC)CN(C(=O)CCOC(C)=O)CCO1.C1C=CCS1 Cc1nc(C2CC2)ccc1C(N1CCC1CNC(=O)CCCC(F)F)=O Cc1c(CN(C(C2CCSC2(C)C)C(=O)NCCCF)C)cccc1Br C1(N(C(c2n(CC)ccn2)=O)C)C2CN(C(=O)C(C)O)CC12.c1cccc(F)c1 C1(C(N(C2CCN(C(=O)CC(C)O)C2)CC#C)=O)CCC(=O)N(C2CC2)C1 N1(C(C2(C(C)(C)OC)CC2)=O)CC2C(C(=O)NC(c3cncs3)C)C2C1 C1(CC(=O)NCC(C)CNC(=O)CN(C2CCSC2)C)COCCOC1 N1(C(C(COC)O)=O)CCSCC1CCNC(=O)Cc1ccc(Cl)s1 c1(CNC(c2ccc(C(C)=O)o2)=O)ccc(C(N2CC(C#N)C2)=O)cc1 n1(C(C)(C)C)cc(Cl)c(C(N2CCC(C)C2)=O)n1.C1(C=O)CC2(C1)CC2F.N C1(CNC(C(C)C(F)(F)F)=O)CC2(CCN(C(=O)CC)CC2)CO1.CC(F)F.O C#CC1(C(N2CCN(C)CC(C)C2)=O)CCN(C(=O)CC=C=C)CC1 CC1(C)CCC(CCOC(=O)C(O)C2CCCC2)C1 N1(C(CCOC2CN(C(C(c3ccccc3)C)=O)C2)=O)CC2OCCN(C)C2C1 N1(C(CC2(OC)CN(C(C3CC(C=O)C3)=O)C2)=O)CCOCC1CC(N)=O.O C#Cc1cccc(NC(=O)C2=NOC(CNC(=O)C(C)(Cl)Cl)C2)c1 C1(n2cc(C3CCN(C)C3)nn2)CON(C(=O)c2ccccc2O)C1 c1(CC)ccc([N+](=O)[O-])cc1C(N1CCC(C)C1)=O.C(=O)C=CC(C)=O.N C1(NC(c2ccn(C(C)(C)C)c2)=O)CN(C(c2ncccc2N)=O)CC1(C)C c1(Sc2cccc(O)c2)cnc2cc(Br)c(Br)cc2n1 Cn1cc(C(N2CCCC2(C)C(N2CCC2C2CCC2)=O)=O)n(C)c1=O C1(NC(C2CNC(=O)N2)=O)CCCCN(C(C2(OC)CC2)=O)C1.c1ccccc1 c1(C(N(CC)C)=O)ncnc2cc[nH]c12.C1(CC(=O)N(C)CCO)(CC)CCC1 CC1C(C)CCN1C(=O)C#CCNC(C1CC1OC(C)(C)C)=O C(CS(=O)(=O)CC(F)(F)F)NC(CCC(C)(C)C)c1n(C(C(=O)OC)C)nnn1 CC1CCC(CC(=O)NCc2ccoc2C(N2CCC2(C)CCO)=O)OC1 C1CCCN1CCC1CCC1.c1cccnc1.C1(C(F)(F)F)(C(=O)N)CC1.C C12(CNC(C3N(CC)CC3)=O)CCC(CN(C(=O)CCS(=O)(=O)N)C1)C2 c1(OC)ccc2c(c1)C(CCn1cc(-c3cc(C)c(C)cc3C)nn1)=CC2 c1(C=O)cnn2c(=O)cc[nH]c12.c1(CC)ccc(C(=O)NC2CC2)c(C)n1.C C1(C(=O)NC(C2CCCC2)CC)(CNC(c2cc(CC)sn2)=O)CCCCC1 CCCCC(C)C(=O)NC(c1ccccc1F)CNC(=O)Cn1nc(C)nc1C c1(CC)ccc(F)c(C(=O)NC2CC(NC(C3CC3(C)Br)=O)C2)c1F c1(C(N2CCCC(C(N)=O)C2)=O)ccc2c(n1)CCC2.C(C)(CO)(C(=O)N)OC C1(C(=O)NC2CC(CNC(CCCC#C)=O)C2)CCn2ccnc2C1 C(CCCCC(=O)NCC1(C(=O)N(C)CCc2ncccn2)CCCCC1)OC N1(C(C(=O)Nc2cncc(CC)c2)=O)CC2(COC)CC1(CN)C2 c1(OC)ccc(C(=O)NC2CCCC(NC(c3cc(Cl)cn3C)=O)C2)cc1OC S(=O)(=O)(c1ccc(N2CCC(CC3CCCC3)C2)cc1Cl)NC(CSC)C N1(C(C(CO)N(C)C)=O)CC(F)(F)CC1C(=O)NCc1nc(=O)o[nH]1 C1(C(N(C(C)C)CC)=O)CCC2(CCC2)O1.c1(C(C=O)C)cccc(Cl)c1.N O=C1CCc2ccc(C(=O)NC3CCC(NCc4ncc(Cl)cc4Cl)C3)nc2N1 Cc1sc(C(=O)NC(CNC(C2CC2c2ccccc2)=O)C(C)C)nc1O c1(N(CC(=O)NCC)C)nc2ccccc2c(=NCc2cc(OC)ns2)[nH]1 C(=O)(CC(C)SC)NCCN(C(=O)CC1CC1(Cl)Cl)CCOC C1(NC(c2[nH]cc(-c3[nH]c(=N)sc3)c2)=O)CCCCCN(C(c2cnsc2)=O)C1 C=CCC(C(=O)NC(C(=O)N(C1CCOCC1)C)C1(C)CC1)NC(C)=O Cc1c(CCC(=O)NCC(C)(F)CNC(=O)C(C)(C)C2CCC2)cnn1C CC1(C)CCC(C(N2CCC=C(F)C2)=O)CN1C(=O)C(F)(F)C1CC1 c1(N(C(C(CNC(c2cn(CCC)nn2)=O)O)=O)CC)cccc(Cl)c1 C(=O)(CCCCCNC(C12CC(C#N)(C1)C2)=O)NCC(C#C)C(C)C C(=O)(C(CCOC)OC)NCCC(=C)C.C1CCS(=O)(=O)C1.C(=O)(C)N CC1(C)C2CCC1(CN1CCC(F)C1)C(=O)C2.c1(C=O)cnc(C2CC2)nc1.N C1(O)(C(c2cn(CCC3CC=CCC3)nn2)O)CCCCC1 c1(NC(C)(C)C)ccccc1.C12CC(C1)C(=O)COC(=O)CO2 C(=O)(C(O)C(F)(F)F)NCC=C1CCN(C(C(c2cn(C)nc2)=O)=O)CC1 c1(C(=O)NCC2CCCN2C(=O)Cc2ccc(Cl)cc2)cccc2[nH]ccc12 Cc1nn(C)cc1C(C(=O)NCC(C)C)N(CCCNS(C)(=O)=O)C C1CCC(C)CN1C(=O)C(C)C(C)(F)F.N1(C(=O)NC)CC(C(=O)N)C1.C O(C=C(C#N)C(=O)N1CCOC(CNC(c2cn(C)c(=O)n2C)=O)C1)CC c1(C(=O)NCC=C2CCN(C(=O)C3=CCOC3)CC2)cc2n(n1)CCCC2O C(=O)(C#CC1CCCOC1)N1C(Cn2cc(C=CC)nn2)CC1 N1(C(C2C(C=C)OCC2)=O)CCCN(C(c2conc2COC)=O)CC1C(C)C C1(C(=O)O)CCCCC1C.C(CCO)N(CC=O)CCC C1(C(=O)NCC(CCNC(c2cnc(O)cc2C)=O)OC)CCc2nccn2C1 C1(NC(c2n(CC)nnn2)C2(C(F)(F)F)CCC2)CCOCC1(C)C Cc1cccc2cc(C(=O)NC3(CNC(=O)CCCC(C)C)CCOC3)cnc12 CN1CCN(C(=O)Cn2ccnc2)C(C(=O)NCCCCN2CCCC2)C1 c1(C(=O)NCC2CC(NC(C(C=C)(C)O)=O)C2)cccc(CC)c1N N(C1CCc2ccc(F)c(F)c21)C(=O)C(N1CCCc2occc2C1)=O c1(OC)c(Cl)cc(C(=O)NCC(C)CNC(C2CCC(=O)N2)=O)nc1Cl Cc1csc2cc(C(N3CC4(CCCC4NC(=O)CCc4cscn4)C3)=O)[nH]c12 CCC(C)CC(=O)N1CCC(C(C)(C)CNC(=O)C=C(C)c2ccco2)CC1 C(C1=CCN(C(C2(CO)CC2)=O)CC1)NC(C1CCC2CC2C1)=O c1(SC)cccc(F)c1C(=O)NC1CCC1.C1(CC=O)CC(n2cnnc2)C1 N1(C(c2csc(O)n2)=O)CCN(C(c2ccc3ccnn3c2)=O)C2CCCCC12 c1(C(=O)NC(C(C)C)C(C)NC(=O)Cc2cscn2)c[nH]c2ccncc2c1=O c1(C(C)=O)ccc(C)cc1.C1(C(=O)N)CCCN1C(=O)CCN(C)C.CC=O N1(C(=O)COc2cccnc2)CCN(C(=O)CCc2cnoc2)CC2(CC2)C1 N1(C(C(C)(C)N(C)C)=O)CCC(C2CCN(C(c3cc(C4CC4)[nH]n3)=O)C2)CC1 C(=O)(CC(C)CC(F)(F)F)NCC(C1CCC1)NC(c1n(C=C)ncc1)=O C1(N(C(CCNS(CC)(=O)=O)=O)C)CCCCC1N(C)C(C1CCOCC1)=O CCCCC(CNC(=O)CN1CSCC1=O)NC(c1ccc(C(C)C)cn1)=O C1(CNC(C(CC(C)C)C)=O)CN(C(C2CCNC2=O)=O)CC(C)(C)O1 c1(C(=O)NCC(C)(C)NC(C(CC)OCC)=O)ccnc(COC)c1 c12ccc(cc1)S(=O)(=O)C(=O)N1CCN2CC1.C1(CC(=O)OCCC)CCOC1 CCC(C)(CO)C(=O)NC1CCCN(C(C2(Sc3ccccc3)CC2)=O)C1 c1(C(=O)NCC2N(C(C(n3ncc(C)c3)C)=O)CC2)ccc2ncn(C)c2n1 c1(C(=O)NCC(C)OC)cc(CNC(=O)C(c2cnccn2)C)ccn1 Nc1c(C(=O)NC2CN(C(=O)CC3CC3)CCC2C(F)(F)F)ccc(Cl)c1F C1(C(N(C)CC2CCN(C(C(CCC)(C)O)=O)CC2)=O)CCc2c(n[nH]c2C)C1 CC1CN2CCN1C(C(=O)NCC1CCCC1)C2.C12(C(=O)N)CCN(CC1)CC2 C(C(C(C)C)C(C)C)N(CCC(=O)Nc1ccccc1C(C)CC)CC S(=O)(=O)(c1c[nH]c(=NCCC(C)(C)C)cc1C)NCC(C1CCC1)OCC c1(C(N(CCC)CCNC(=O)CO)=O)ccccn1.c1ccc(Cl)nc1.C c1(NC(c2cocn2)=O)ccc2c(c1)CN(Cc1ccc(Br)c(CO)c1)C2 N1(C(C2C(C=O)C2)=O)CC(C=O)C2(CCC2)C1.C1(C)(CC)CCCC1.CC c1(C(N2C(CNC(C3(COC)CCOCC3)=O)CC2)=O)cc(Cl)c(Cl)n1C N1(CC)CCOCC1C(=O)NC(CNC(=O)C(C(C)C)SC)C(C)(C)C c1(CC(N2C(C)(C(=O)NC3CONC3=O)CC2)=O)ccccc1C#N c1(C(=O)NCCCC=C)ccc(=O)n(CC)c1.C(=O)(C(O)CN1CCOCC1)N C1(C(CNC(=O)COCC2CC2)F)CCN(C(=O)C)CC1.C1CCCCO1.S n1(CCNC(C2CC(=C)C2)=O)cc(C(=O)NC(CO)C2(C)CC2)cn1 c1(N(CCCCN(C(C(C#C)(C)C)=O)C)C)ncc2ccsc2n1 N1(C(c2c(CCC)n(C)nc2)=O)CC2CN(C(c3cnc(C)nc3C)=O)CC2C1 c1(C(N2CCC(C=C)C2)=O)ccc(C(N2CCOC(C)(C)C2)=O)cc1C N1(c2n(CC(C)Cc3ccccc3)nnn2)CCC(OC2CCOC2)CC1 CC(O)C(C)(C)C(=O)NC1CC2CC1N(C(=O)CSCCC#N)C2 C(=O)(CCCCC(=O)NC1CN(Cc2ccccc2OC(F)F)C1)OC C1(CC(=O)NCC(C)(F)C)COCC1(C)C.c1(C=O)ccc(C(F)(F)F)[nH]1 c1(N(C)C)ccc(C(N2CCC(CNC(=O)CCOc3cccnc3)C2)=O)nn1 C1(CC(N2CC(C)(c3cn(Cc4cccc(F)c4)nn3)C2)=O)CCCC1(F)F Cc1cc(F)ncc1C(=O)NC1COCCN(C(c2cnc(F)c(Cl)c2)=O)C1 c1(C(=O)NC2CCCN(C(CC(CCCC)O)=O)C2)ccc(N)c([N+](=O)[O-])c1 c1ccc(O)nn1.N1(C(C2C(OC(C)=O)C2)=O)CCC(C(C)(C)C(=O)N)C1 Cc1ccc(C(N2CC3(CCCC3NC(=O)CCCN(C)C)C2)=O)c(F)c1F c1(CN2C(C(N3CCCC3CO)=O)C3CCC2C3)ccc2ocnc2c1 CCC(CC(=O)NC(COC(C)C)C(=O)NC1CN(C)NC1=O)C(F)F C(=O)(CCS(C)=O)NC(CNC(COCC(=O)NC)=O)(C)CO CCCCC(O)CC(=O)NC1CN(C(C23CC(COC)(CO2)C3)=O)C(C)(C)C1 C1(NC(C(CC#C)C)=O)CN(C(=O)CC2OCCO2)C2(CCC2)C1 CC1CN2CCN1C(C(=O)N(C)CCN(C)C(c1cccnc1CO)=O)C2 C1(CNC(C2CCCOC2)=O)(NC(C2COC2)=O)CC2CCC1CC2 Cc1cnc2cccc(Oc3ncnc4c3ncn4C3CCCCO3)c2c1 C1(C(N2CC(C#C)(F)C2)=O)CCCCCCN1C(=O)C=Cc1ccccc1C C1(NC(C2=C(C)CC2)=O)CC2CC1N(C(=O)C(=O)Nc1ccccc1)C2 C=CC(C)(C)C(=O)N(CC)CC1CCCN(C(=O)C(N2CCNC2=O)C)C1 Cn1cnc2c(N3CCCCC3C(N3Cc4ccc(F)cc4C3)=O)ncnc12 c1(C(=O)N)cc(F)c(F)c(F)c1.c1(COC)c(C(=O)NCCCO)cnn1C N(C(=NCCC(C)N(C)C)NCC1CCCN(C=O)C1)CCSC.C(C)(C)C.O CC(C)(CNC(C1CCSC1)=O)CCNC(=O)CC1CCCC1 C1(O)(CO)CCCN(N2CC3CC2CN3Cc2cccs2)C1 Cc1nc(O)nc(C)c1CCC(N1CCCC(C)(CNC(=O)C(O)C2CC2)C1)=O Cc1c(Cl)cc(C(N2CC(C(=O)NCCN(CCO)CCO)C2)=O)cc1Cl CC1CC1C1CC1C(N1CCCC1CCCNC(C1CCCC(C)C1)=O)=O C1(CC(=O)NCCn2cccnc2=O)CCN(C(C2C3(CC3)C23CC3)=O)CC1 N1(C(C(c2ccccc2)OC)=O)CC(C)OC(C)(C)C1.c1(CC(=O)N)cnns1 C1(C(=O)NC2CN(C(c3ccn(C4CCC4)n3)=O)CC2CO)OC2CCC1CC2 N1(C(C(c2ccc(C)cc2)(F)F)=O)CCC(NC(c2nn(C)cc2Cl)=O)C(F)C1 c1(CC(NOCC(N2CCCC(C(C)(C)O)C2)=O)=O)c[nH]c2ncccc12 C1(NC(C2(N(C(=O)CN3CCCC3=O)C3CC3)CCC2)=O)CCOC(=O)CC1 C1(CNC(c2c(CC)ncs2)=O)COCCN1C(C1CCSC1)=O C1(NC(C(C)N(C)C)=O)CCN(C(c2cnn(C3CC3)c2)=O)C1C n1(CCCN(C)C)c(CNC(CCCC(C)(C)C)C(=O)OC)nc2ccccc12 N1(C(C2(C)CCNC(=O)C2)=O)CCC(C2CC2)(CNC(c2ccon2)=O)C1.C CC1CCCC(CC(N2CCN(C(=O)CNC(C3CC(F)(CF)C3)=O)CC2)=O)C1 c1(NC(C2CCN(C(C(C)(C)OC)=O)CC2)=O)cccc2c[nH]nc12 Cc1cc(Cl)c(Cl)cc1C(N1CC(O)(C)C1)=O.c1(C=O)ccn(C(F)F)n1.N c1(C(N(C2CN(C(c3n(CC)cc(Cl)c3)=O)CC2F)C)=O)ccc(=O)n(C)n1 CCCC(CCC)C(=O)NC1CS(=O)(=O)CC1NC(c1cc(Cl)c[nH]1)=O N1(C(CNc2n(C)ncc2)=O)CC2CCC(NC(=O)CCCN3CCCC3)(C2)C1 C1(NC(c2ccc(C)o2)=O)CN(C(c2ccc(CN=[N+]=[N-])o2)=O)CCC1C c1(C(=O)NCCC(C)NC(=O)CC2SC(=N)NC2=O)c[nH]c2cc(F)ccc12 N1(C(C2C(OCC)C2)=O)CCCC(O)(C)CC1.C1(C(=O)N)Cc2cscc2C1 C(=O)(C1COc2ccc(F)cc21)NCCCCCCNC(C(C=CC)O)=O C(=O)(CCC[SH](=O)=O)Nc1c(C(=O)OC)c(C)cs1.c1(CCCN)ccccc1 C1(C)(CNc2cc(NC3CCC(C)C3)ncn2)CCCCCC1 C1(NC(C2C(C)(C)CC2)=O)CN(C(=O)C(O)CC2CCCCC2)CC1O c1(CCC(c2n(CC=C)nnn2)NCC(COC)C(C)C)cccc(Cl)c1 C1(CN(C(C(C)OCCCCCC)=O)C)CCN(C(=O)CCc2ccon2)CC1 C(=O)(C(C)C(C)O)N1CCC(CNC(c2ccc(C)o2)=O)C1 c1(C(NC2c3ccc(C)cc3CC2)=O)c(O)cc(=O)n2c1CCCC2 C1(OC)CCCC(C(c2ccc(Cl)s2)=O)C1.N12CCN(CC1)CC2=O C1(C(N2CCCC(NC(c3sc(C)c(O)n3)=O)(CO)C2)=O)CCC(N=[N+]=[N-])CC1 c1(C(N2C(C)CC(OC)C2)=O)nnn2c1COCC2.C1(O)(CC(=O)N)CCOC1 C1(CCC(=O)N(CCC(O)CO)C)CCCCN1C(c1cc(Cl)c[nH]1)=O CC(C)C(CCNC(=O)COCCN(C)C)NC(c1cccc(Br)c1)=O C1(CC(=O)N(C)CC2CCCCO2)CCCN(C(C23CCC(CC2F)C3)=O)CC1 C1(N(C(=O)Cc2nncn2C)C)CCCCC1NC(C1CCS(=O)(=O)N1)=O c1(C(=O)N)ccc2[nH]c(=N)n(C)c2c1.S(=O)(=O)(CC(=O)N(C(C)C)C)NC c1(C(N2CCOCC2C2CCCC2O)C(=O)N)cc(S(C)(=O)=O)c(C)o1.C=CC CC(=NOCC#N)C(=O)N1CCC(C(C)C(=O)N(C2CC3CCC2O3)C)C1 CC1CN(C(c2ccno2)=O)CC(C)N(C(=O)CCSc2ccccn2)C1 N#Cc1ccc(=NCC(=O)NCC(C2CC2)NC(=O)C2Cc3ccccc32)[nH]c1 CCCC(C#N)C(=O)NCC=CCC(=O)N(C1CCN(C)C1)C C(=O)(C(C)(CSC)NC(c1ccnn1C)=O)NCC1(CO)C(C=C)C1 c1(C(=O)NCC2C(NC(c3ccc(F)s3)=O)CCCC2)c[nH]c2cccnc12 CC#CCCC(=O)NC1C2CCN(C(C3CC34CCC4)=O)C12 C1(CN(c2cc(Cl)cs2)C)CC2(CCCC2)CO1 Cn1c(NC(=O)NCC(=O)NC(c2ccc(F)c(F)c2)=O)nc2cccnc12 Cc1c(C(=O)NC2CC(C(=O)NOC(c3ccncc3)C)C2(C)C)c[nH]c1C#N c1(C(N2C(CNC(C(C=C=C)C)=O)C3CCC2C3)=O)cc2c(cn1)COCC2 C(=O)(CCCC(=O)N(C)C)N1CCC(C(=O)Nc2cncc(C)c2)CC1 CCC(C)(O)Cc1cn(-c2cnn(CCCC#N)c2)nn1 C1(C(=O)NC(CNC(C(C)n2cnnn2)=O)CO)C2C3CC4C1C1C2CC3C41 c1(CN=c2[nH]nc(CC)o2)c[nH]c2ccccc12 c1(C(=O)NC(C#C)CC2CCCO2)cc(C(N)=O)ccc1OC c1(CC(=O)NC(C2CCCCN2C(=O)CCc2cn[nH]c2)C)c(F)cncc1Cl c1cn(C2CCN(C(=O)C(F)=C3CCC3)C2)nn1.CCCCSCC(=O)NC N1(C(c2cnc(OC)s2)=O)CCOC(C(C)NC(c2cnoc2C)=O)C1 CCC(C(=O)N1CCCC1CN(C)C(C1CSCN1C(C)=O)=O)OC C1(C(N2CC(C(C)NC(CC(=O)NCC)=O)OCC2)=O)CCn2ncnc2C1 c1(N(C)CC2CCC2)nc2ccsc2c(=NCC(CCCO)c2ccccc2)[nH]1 CCCCCCCCC(=O)NCC(C)N(C(=O)CC(C)(C)CN(C)C)C CC1CN(C(c2coc(Br)c2)=O)CC(CCNC(C2(CCO)CC2)=O)O1 N1(C(CNC(=O)C(c2ccc(Cl)cc2)O)=O)CC2(C1)CN(C(=O)CO)C2 Cc1ccc(C(C)C)cc1C(=O)NCC(N1CCCC1)C.c12nc(cs1)S2 CC(C)C(C(C)NC(c1nscc1Br)=O)NC(=O)Cc1cnn(C)c1 Cc1nn(C)c(C)c1C=O.C(CCNC)C(C)(C)C.C1(S(N)(=O)=O)CC1.C C1(C(=O)NC(c2ccc(Br)cn2)C)CCN(Cc2ccc(F)nc2)CC1O c1(OCC)ccc(N)c(C(=O)NCC2CCN2C(=O)C2=CCSC2)c1 C(=O)(CCN=C(NCC(F)F)NCC1CSc2ccccc21)NC(C)(C)C CN1CC(C(=O)NC2CC(F)(CNC(c3cnc[nH]c3=N)=O)C2)CC1=O CC1=C(C(=O)NC2CCN(C(=O)C(C)(C)C(C)C)CC2)C(C)n2nnnc2N1C CCCC(CC(C)C)C(=O)NCCC(C)NC(=O)CC1CCCC1C c1(-c2cn(C)nn2)cncc(C#N)c1.c1(C2C(C)C2)cccc(Cl)c1 N1(C(C2CN3CCN2CC3)=O)CCCC2C1CCCN2C(c1c[nH]c(=O)cn1)=O C1(NC(C2=CC(C)(C)C2)=O)CC2CCC(C1)N2C(c1cccc(C(F)F)c1)=O N1(C(CC(C)C2CC2)=O)CCCN(C(c2ccnc(C3CC3)n2)=O)C(C)C1 C=CC1(CC(=O)N)CCOCC1.C1CN(C(C2CC(=C3CC3)C2)=O)C(C)(C)C1 N1(C(CCc2ccc(C)cc2C)=O)CCCC2(C1)CN(C(c1ns[nH]c1=O)=O)C2 CN1CCOC(C(=O)NC2CC(CNC(c3ccc(C4CC4)cc3)=O)C2)C1=O c1(C(=O)Nc2c(O)cc(Br)cc2Cl)ccc2nn(C(F)F)cc2c1 n1(CC(C)C)[nH]c(CC(=O)N(C2CCN(C(=O)CS(N)(=O)=O)C2)CC)cc1=O CCCCCC(C)(C)C(=O)N(CCCCNC(c1ccccc1C(C)(C)C)=O)C O=C1CSc2cc(C(=O)NC3CCCN(Cc4ccc(F)cc4Cl)C3)ccc2N1 c1(C(=O)NCC2CCCN(C(CC(C)SC)=O)CC2)cnc2[nH]c(O)nc2c1 C=CC(CC)CC(=O)N(C(C)CNC(c1n[nH]c(C2CC2)c1Cl)=O)C C(c1ccccn1)=C(C)C(=O)NCC1CCCCC1.C(C1CCCO1)=CC(=O)N C(=O)(NNc1nc2cc(Br)ccc2s1)C12OCC(S(C)(=O)=O)(C1)C2 N1(C(c2c(NC)ccc(C)c2)=O)CCC(C)N(C(=O)CCSCC(N)=O)CC1 N1(C(C2C(NC(C3(CC(C)=O)CC3)=O)CCOC2)=O)CCC(C)CC1C C12(C(=O)NCC(C3(O)CCN(C(C4CC(C)(C)CO4)=O)C3)C)CC1CNC2=O C1(NC(Cc2nnc(C)o2)=O)CCN(C(=O)CNC(c2ccncc2)=O)C(C)C1 O=C(C1CCCc2scnc21)NC1(CN=c2[nH]nco2)COC1 C(=O)(Nn1cncn1)C1C(C)(C)C(NC(c2n[nH]c(O)n2)=O)C1 C1(OC)CCCC(C(=O)N(C(C)C2CC2)C)C1.c1(C(C=O)O)cccc(Cl)c1.N C12(CNC(CCCOC(C)C)=O)COC(C)(C1)C2.C(=O)C(C)c1cccs1 C(CCCCCCCO)=CC(=O)NC(CCNC(C1=NOC(C)C1)=O)(C)C C1(NC(c2ccc(Cl)o2)=O)CCC(NC(C2CC2c2ccccc2)=O)CC1 Cc1cc(CC(=O)NCCN(C)C(c2[nH]cnc2C)=O)ccc1O N1(C(c2c(C)nc(C)s2)=O)C2CCC(C(N3CCCOCC3C)=O)C1CC2 C1(C(N(C2CC3CC3C2)C)=O)CC(=O)CN1C(C1CC1C(F)(F)F)=O CC(C)C(C(=O)NC(C1(C(N2CC(N3CC(F)C3)C2)=O)CC1)C)C(C)C c1(C(N2CCCC(C)(C(=O)NCC(CC)CC)C2)=O)cc(C)cc(C#N)c1 C(c1ccccc1Cl)=CC(=O)NC(C1CCCCC1)CNC(c1c[nH]c(=N)o1)=O C#CCC(C)(C(=O)N(CC(C)C(C)C)C)NC(c1cc(C)sc1C)=O Nc1cccc(C(N2CC3C(CNC(C4CCNC(=O)C4)=O)C3C2)=O)c1F c1(C(N(C2CCCC2)CCCNC(CC(C)SC)=O)=O)cc2nccn2c(O)n1 C12(CNC(C3CCCSC3)=O)CC(CN1C(=O)CCC1CC(F)(F)C1)C2 C1(CC(=O)NC(C)CCNC(C2CN(C3CCC3)C2)=O)CCNC1=O c1(C(N(CCCNC(C(=O)NCC)=O)C(C)C)=O)ccnc2[nH]cnc12 Cc1ccc2[nH]nc(C(=O)NC3CCN(C(C4(F)CCS(=O)(=O)C4)=O)CC3)c2c1 c1(C(C)N(C(=O)CCn2cc(C(O)C3CC3)nn2)C2CC2)ccccn1 c1(CNC(CC(N)CCc2ccccc2)=O)c[nH]c2ccc(F)cc12 N1(C(CC(CCC)(C)C)=O)CCC2CN(C(c3cc(C)n(CC)c3C)=O)C(C)C12 Cc1occc1C(N1CC(OCCNC(C2CC(n3ccnc3)C2)=O)C1)=O CC(C)(C)CCCCC(=O)NCC1CN(C(=O)CSc2nncs2)CC1(F)F C(=O)(CCCC(N)=O)N(C1CCN(C(=O)C(C)(CO)OC)C1)CC CCC(C)(C)C.c1(CC)cscc1C(=O)N.C(=O)C(C)C.C(=O)C(F)(F)F C1(CSCCNCC)CCOC2(CCCC2)C1 c1(C(N)=O)ccc2c(n1)N(C(C1CCCC3(C)CCCCC13)=O)CCC2 c1(-c2cnc(NC(C3CN(Cc4cnc(C)s4)C3)=O)s2)ccc(F)cc1 C1(NC(Cn2c(C)nnn2)=O)CCCC(CNC(=O)C=C(Cl)Cl)C1 N1(C(c2c(OC)n[nH]c2)=O)CCN(C2CCCN(C(=O)Cc3ccsc3)C2)CC1 c1(C(=O)NC(CCNC(CC(C)SC)=O)C)cnn2cc[nH]c(=O)c12 c1(C(=O)OC2CCN(C3CCCCC3)C2)ccc(NC(=O)C2CC2)cc1 n1(CC)cc(C(=O)NCC(CO)NC(C23CCCCC2C3)=O)c(C2CC2)n1 c1(OC)cc(CC(=O)NCC2CCN2C(=O)CCC(C)(C)C)cc(OC)c1O Cc1ccc(C2CNCC2N2CCCC2C=Cc2cccs2)c(Cl)c1 C(=O)(C(N)C1CCc2ccccc21)NCC(C)Oc1ccccc1 C(=O)(C(C(CC)CCCC)N1CCSC(C(F)(F)F)C1)NCC=C C(CCCCCS(=O)(=O)CCO)OC(=O)CNC1CCC12CC2 c1(C(=O)NC)ccc(F)cc1C1CC1.C1C2CN(C(C3CC(O)C3)=O)CC12 N1(C(CCN(C(CCC)C)C)=O)CCC(C)C(NC(=O)CCCNC(N)=O)C1C c1(CC)[nH]nc(C(=O)NC2CCC2)c1[N+](=O)[O-].C1(C=O)OC(C)(C)OC1(C)C N1(C(c2cc(C)nc(C)c2)=O)CCN(C(c2cnc(S)[nH]2)=O)C(C)CC1C N1(C(Cn2c(C)nnn2)=O)C2CCC1CC(NC(c1cccc3nncn13)=O)C2 N1(C(CC=C(C)C)=O)CC2(CC2)CC1CNC(=O)C[SH](=O)=O.C1CC1.N c1(CC(=O)NCCCCCC)cnc2c(=O)[nH]ccn12.C(=O)(C(C)CN(C)C)N C12(NC(CCOCC)=O)COC(C1)C(NC(C1CC(N(C)C)C1)=O)C2 c1(C(N2CCC(NC(CCNC(=O)NC)=O)C2)=O)ccc(F)cc1C N1(C(CC2C(C)OCC2)=O)CCC(OCCNC(=O)CC2CCCC2(F)F)CC1 C1(C(=O)NCC2(SCC#C)CC2)CCCN1NC(=O)C(C)=CCC N1(C(CN(CCOC)C)=O)CCCC1Cc1c[nH]nn1.c1cc(C2CC2)no1.C C1(C(=O)NC(C)CCNC(c2n[nH]c(=N)[nH]2)=O)CCCC(O)C1 c1(C(=O)NCC(CNC(C(CCCC)C)=O)C)c(F)ccc2nc[nH]c12 c1(C(=O)NCC2C(NC(=O)CC3CCCO3)C2)cnoc1-c1ccc(Cl)s1 N1(C(C(=O)NC2CC(F)(F)C2)c2csnn2)CCC2CS(=O)(=O)CC12 C1(NC(c2cc(C)[nH]n2)=O)CN(Cc2coc(C)n2)CC2(CCOCC2)C1 Cc1cc(N2CCCC(C(C)NC(C3CCC(=O)NC3)=O)C2)nc(C2CC2)n1 N1(C(CC(CCC)(C)O)=O)CCC2(CC1)CN(C(=O)C(CC(C)C)NC(C)=O)C2 C1(CNC(Cn2c(C)nnn2)=O)CCCCN1C(c1ccn(CC(C)C)n1)=O N1(C(c2c(OC)nccn2)=O)CCC2(CC1)CC2.c1(C=O)c(F)cnn1C(C)C C(=O)(C(C)(C)CC1CC1)NC1C(CNC(C(C)Cc2ccncc2)=O)C1 C1(NC(c2c(CC)ocn2)=O)CN(C(=O)CCCC(=O)C2CC2)CC2(CCC2)C1 c1(CCC(=O)NCCC)ccc(C(F)(F)F)nc1.c1(C=O)cn(C2CC2)nn1.N c1(CCCC(=O)N(CCCN(C)C(C2CC(O)C2)=O)C)ccc(Br)cc1 c1(C(=O)NC(CN(C)C)C(=O)NCC(c2ccccc2)F)ccc2cncn2c1 N1(C(c2ccc(N(C)C)cc2)=O)CC2CN(C(=O)CCc3cncs3)CC2C1 CCC(C(=O)NCCCCN(C)C(c1ccc(OC)nc1Cl)=O)C(C)C C(=O)(CC(C)CF)NC(CC1CCC1O)=O.C1(C=O)(C(C(C)C)=O)CC1.O c1(C(C=O)N(CC(=O)NC(C)(C)C)C(C)C)ccc(Br)c(F)c1.C1CCOC1 CN1CCOCC1c1nn[nH]n1.C1(c2cccc(OC(F)F)c2)CCCOC1 c1(OCC)ccc(-c2nc(-c3cn(CC4CCCO4)nn3)n(CC3CC3)n2)cc1 N1(C(C(c2ccn(C)n2)OC)=O)CCC(C(C)(C)NC(=O)C(N)=O)C1 N1(C(c2ccc(OC)c(C#N)c2)C(=O)NC(CC)C)CCc2ncnc(C)c2C1 C(=O)(C(CNC(=O)CNc1ccccn1)CC(C)C)NCC(CC)CCO N1(C(C(C)NC(c2ccc3occc3c2)=O)=O)CC23CCC2(COC3)C1 CCCC(O)(CCC)CC(=O)Nc1ccc(CCC(=O)OC)cc1 c1(C(=O)NCCCN(C(=O)C)C(C)C)ccc(=O)n(C)c1.C1CCCCO1.S Cc1cc(C(N2CC(NC(C3(C)CCOCC3)=O)C(C)C2)=O)cc(C(F)F)c1 c1(OC)c(O)ccc(CN2CCCC2CC(=O)NCCS(C)(=O)=O)c1[N+](=O)[O-] c1(C(=O)NC2CCC(C(=O)NCCn3ncc(C)c3)CC2)cnc2ccccn12 C(CC(=O)NCc1cnc[nH]1)(C(F)(F)F)NC(C(CC)(C)C)=O CC1(C)Cc2occc2C(NC2CC(O)C2(C)C)C1 CC(C)C(C(=O)NCCCNC(=O)C(O)Cc1cnc[nH]1)n1cnnc1 N1(C(CCNC(C)=O)=O)CCC2C(NC(c3c(C)ccn3C)=O)C2C1 N1(C(C=C(CC)C)=O)CCCC(CNC(=O)CCc2cn(C)nn2)CC1 N1(C(C2(C)CC2(F)F)=O)CC(NC(c2ncoc2C2CC2)=O)CC2(CCC2)C1 c1(OCCC(=O)N(CCC(F)(F)F)CC2CC2)cccc(I)c1 N1(C(c2ccn(CCCC)n2)=O)CC2CN(C(C3CC(=O)N(C)C3)=O)CC2(C)C1 c1(CC(=O)NC(CC)(C)CNC(C2CC(C)=NO2)=O)ccccc1C CC1(CNC(C2(Sc3ccccc3)CCCC2)=O)CCN(C(C2CCOC2)=O)C1 Cc1csc(C(=O)NC2CC(CC(=O)NCCCOCC(C)C)C2)c1 Cc1nc(C(N2CC(NC(=O)CC3(C)CCCO3)CC(C)C2)=O)ccc1C#N c1(CNCC23C(CN(C(c4cc(F)ccc4F)=O)C2)C3)c[nH]c2c(Br)cccc12 C12(CNC3C(c4c(Br)ccs4)C3)CCCC1OCC2 N1(C(c2nc(C)n(C)n2)C(=O)Nc2ccc(F)cc2)CCOCC(C)(F)C1 C(C(S(C)(=O)=O)c1ccccc1)NCCCN(C(C)(C)C)CCO C1(CNC(C2ON=C(C)C2)=O)CCC(N(C)C(C2CC(=O)N(O)C2)=O)CC1 C#CCCCC(=O)NCC(O)CNC(C1CC(F)(CO)C1)=O c1(OC)ccc(C(N2CC3C(C(N4CCCC(CF)C4)=O)C3C2)=O)cc1F O=C(CS(=O)(=O)C1CC1)NC(c1ccccc1)CNC(c1ccc(C)cn1)=O c1(N2C3CC(CC(NC(c4ccc(C)c(Cl)c4)=O)C3)C2)c(C)cncc1[N+](=O)[O-] S(=O)(=O)(c1ccc(Cn2nccn2)cc1Cl)NC1(CSc2ccccc2)CC1 n1(CC=C)ccnc1C(=O)NC(CNC(=O)Cc1cncnc1)C(C)C N1(C(c2cccc(OC)n2)=O)CCOc2cc(Br)ccc2C1CO C1(CC)CC(C)CN(C(c2ccc(N3CCCC3)nc2)C(=O)NCCOC)C1 c1(COCC)nc(N2CCCC(CCNC(C3CC=CC3)=O)CC2)cc(Cl)n1 C1(CNC(c2cscc2Cl)=O)CCC(C(N2CCC(N3CC=CC3)C2)=O)O1 Cc1ccc(C)c(C(=O)NC(C)CCCNC(C2CC2C(F)F)=O)c1C Cc1cccc2cc(C(N3CCC(NC(=O)CSc4nc[nH]n4)C3C)=O)[nH]c12 NC(=O)CCCCNC(C1C=CCN(C(c2cc(O)cs2)=O)C1)=O c1(CNC(CC2C(C)CC2)=O)ncccc1C(=O)NCc1cccnn1 Cc1c[nH]c(C(=O)NCc2cc[nH]c2C(=O)N(C2CCCC2C)C)c1C CCCC(C)CC(=O)N1CCOC(CNC(=O)CC2CNC(=O)O2)C1 N1(Cc2cnc(C)o2)CCCC(NC(=O)C(C)Sc2ccccn2)CC1 c1(C(N2CC(NC(COc3c(C(N)=O)cccc3)=O)C2)=O)nc(F)ccc1Cl c1(CC)sc(=N)[nH]c1C(N1CCC1CNC(c1cc(C)co1)=O)=O CCC(CCCC(=O)N1CCN(C)CC1C(C)C)NC(=O)CN(C)C(C)=O C1(C(=O)NCCCc2nc(C)[nH]n2)C=CCN(C(C2CN3CCC2C3)=O)C1 c1(CC)nc(N2CC(OCC)C2)c(CC)c(Cl)n1.c1(C(=O)N)cc(Cl)ccc1F C1(CC)CN(C(c2nc(C)nn2C)=O)CCC1NC(c1ccnc(Cl)c1Cl)=O c1(C(=O)NC(CCCCNC(C(CC)(C)F)=O)CO)csc2c1CCCC2 N1(C(C2C(OC)CN(C(C3CCCC(=O)CC3)=O)C2)=O)CC2(C1)CN(C)CCO2 c1(C(N(C)CC2N(C(C=CCCC)=O)CCOC2)=O)cccc(F)c1F N1(C(c2cc(CCC)on2)=O)CC2CC2(C(=O)NC2CC2C2CCC2)C1 c1(OCC)cncc(C=O)c1.C1(CC)CCN(C(C23CC(C)(C2)C3)=O)C1.N c1(C(=O)OCC)ccc(C)c(NC2CC2)c1.C1(C=O)CCS(=O)(=O)C1 C1(CC)(NC(C2CC=CCC2C)=O)CCN(C(=O)CC23CCCN2CCC3)CC1 C1(CC#C)(C(=O)N(C)CCOCC)CCCO1.C1(O)(CC=O)CCCC1.N C1(NC(c2c(C)nc[nH]2)=O)CC(NC(=O)C(c2c(C)noc2C)(C)C)C12CCC2 N1(C(c2c(C)nc(C)o2)=O)CCC(NC(C2CC(C)(C)C2)=O)CC(C)(C)C1.C S(=O)(=O)(c1cccc([SH](=O)=O)c1)NC1CCN(C(CC)=O)C1.CC.C(C)C.N c1(C(N(C2CCCN(c3nnc(C)s3)C2)C)=O)cc(NS(C)(=O)=O)ccc1O C(CC(C(=O)NC1CN(C)CCO1)NC(=O)C(C(C)C)SCC)OCC c1(SC)nc(N2CC3(CN(C(c4ncncc4Cl)=O)C3)C2)cc(C(F)F)n1 N1(C(c2cc(C3CC3)nnc2O)=O)CC(C2CN(C(C3(O)COC3)=O)C2)C1 C(C(CC(=O)N1CCC1(C)C(C)C)NC(C1(C)CCC1)=O)OC c1(-c2ccc(OC)c(C(=O)CF)c2)ccc2c(c1)OCO2 N1(C(C2(COC)CCOCC2)=O)CCCCC(N=c2[nH]c3cc(C)ccc3s2)C1 CC(CCO)NC(=O)C=CCNC(=O)C=CC1CCC1 c1(C=O)cccc2ccoc12.C1(CC(=O)N(C(C#C)(C)C)C2CC2)CCC1O.N C1(C(N(C(C)C(=O)NC(C)Cc2nncn2C)C)=O)CCCCC1(C)C C(C(CC1CC1)C(=O)NCc1sccc1Cl)NC(C1COCCO1)=O C1(C(=O)NCCC(C)CCNC(C2C(C)(C)C2(C)C)=O)CC(C)(C)CN1C C(=O)(CCCN=[N+]=[N-])N1CCC(n2cc(CNC(Cn3c(C)ccn3)=O)nn2)C1 N1(C(COC2CCN(C(C(n3ccc(C)n3)C)=O)C2)=O)CCSC(C)C1 c1(C(=O)NCc2cccc(NC(C(C=C)(F)F)=O)c2)cc2c(s1)CCC(C)C2 C1CC2COCC2N1C(=O)CC(C)c1ccco1.C(C(=O)NC)(C(C)C)SCC C(=O)CC(F)(F)F.c1(CC)ccsc1C(=O)NCCCOCC.CC(C)C Cc1cnnc(O)c1C(N1CCC(NC(C2(C)CCC(C)CC2)=O)C1)=O CC(CCCNC(C1CCN(S(C)(=O)=O)C1)=O)NC(c1ccsc1Cl)=O CC1CN(C(c2ccc(Cl)cn2)=O)CCN1C(c1cc(=O)n(C)o1)=O CN1CC(O)CCC1C(=O)NCC1(C(=O)NC2(C)CC(F)C2)CCCCC1 C1(NC(C2(C(C)C)CCC2)=O)CCN(C(=O)Cn2cccc(N)c2=O)CC1CO CC(N=c1nc2scnc2c(NC(c2cccs2)C)[nH]1)c1cnccn1 N1(C(C)=O)CCCC(C(=O)NC)C1.C1CCC(N(C)C(c2ccc(Cl)[nH]2)=O)CC1 c1(C(=O)NC2(COC)CCN(C(CC=CC)=O)C2)nccc2n[nH]cc12 Cc1nn2cccnc2c1C(=O)NC1CC2CCC(C1)N2C(C1CC1[N+](=O)[O-])=O Cc1cc(-c2nc(-c3cnn(C)c3C)n(Cc3cccc(Cl)c3)n2)c(C)o1 N1(C(c2cnc(OC)s2)=O)CCN(C(=O)CC2CCOC2)CC1CC(F)F c1(C(=O)NCC(CO)NC(Cn2c(C)csc2=O)=O)ccnc2ccncc12 C1(C(=O)NC(C)(C)CNC(=O)C=C(F)c2ccccc2)CCOCC12CCC2 c1(C(N2CC3(C2)CN(C(C2CC2(Cl)Cl)=O)C3)=O)n[nH]c2ccc(Cl)cc12 N1(C(CNC(=O)CNC(=O)C(=O)C2CCCC2)=O)CC2(C1)NC(=O)NC2=O N1(C(C(C)CF)=O)CCCCC1c1cn(CC)nn1.C1(NC(C)=O)CCN(CC)CC1 C1(CC)C(C(=O)NC2(C)CCSC2)CCCN1C(C1CC=CC1)=O C1(NC(C2CCCC2)=O)CCCN(C(C2CCCC2c2nc(S)n[nH]2)=O)CC1 c1(C(N2CCn3c(COC)ncc3C2)=O)c[nH]c2c(C)cc(F)cc2c1=O C=C(Br)CCC(=O)N1CCC(CC2CCN(C(C3(OC4CC4)CC3)=O)CC2)C1 c1(OC)cccc(CN2CCC(C(C)NC(=O)Cc3sc(C)nc3C)CC2)n1 Cc1c(C(=O)NC2CC(F)(C)C2)n[nH]c1C1CC1.C1(C=O)CCC(=O)NC1 CC(CC(=O)NC1CC(C)(NC(=O)CC2CCC(C)(C)CO2)C1)C(F)(F)F c1(C(=O)NCCCC(=O)NCCC2CCC(C)(C)C2)ccc(O)cc1F C(=O)(C(C)(C)C1CCC1)NCC(=O)NCC(COC)C N1(CCC)C(=O)CCC1C(=O)NCC(C)(C1CCC1)NC(c1ccns1)=O C(=O)(CC(C)C(=O)N1CC2(CCC2NC(c2ccc(Br)c(O)n2)=O)C1)OC C1(C2CC2)(OC)CN(C(=O)NC(c2ccco2)C)C1 C1(O)(Cc2cnc(CC)s2)CCCN(C(=O)C(C#N)CCc2ccccc2)CC1 C(=O)(C1=CC(O)C(NC(C2CCCCCN2C)=O)C1)NC(C)CCCCO N1(C(c2c(Cl)cc(C)nc2)=O)CCC2(C1)CN(C(=O)C=Cc1ncco1)C2 N1(C(c2ncn(C(C)C)c2)=O)CC(NC(C2(O)CCCCCC2)=O)CC(C)C1 Cc1csc(CNC(N2CCCC2C(F)(F)F)=O)n1 C#CC1(C(=O)N(C)Cc2cnn[nH]2)CCN(C(c2cnco2)=O)C1 N1(C(CCCN(C(C)=O)C)=O)CCN(C)C(CNC(C2(C)CC3CCC2O3)=O)C1 C(CC(=O)N(CCC(=O)OC)OC)N(C(CCNC(C)=O)=O)C c1(C(=O)NC2CC3(C2)CN(C(c2cc(O)nc(Cl)c2)=O)C3)ccc2c[nH]nc2c1 Cc1nc(C)c(C(N2CC(N3CCN(C(C4OC(C)CC4C)=O)CC3)C2)=O)o1 C(=O)(C1CNC(=O)c2ccnn21)NCC(C)N(C)C(c1cc(Cl)cnc1O)=O N1(C(c2[nH]c(=N)sc2)=O)CCC2(CCCCN(C(c3ccc(CO)nc3)=O)C2)C1 N1(C(c2cn(C(C)(C)C)nc2)=O)C2CCC1CN(C(C1CC1C1CCCC1)=O)C2 c1(C(=O)NCCN(C(CCN(C)CCO)=O)C)ccnc2c(Br)cccc12 C1(C(=O)NCc2[nH]nc(C(C)O)n2)CSc2ccccc2O1 C1(C2CCCN(C(C3CC4(CC4)C3)=O)C2)(NC(C2N(N=O)CCC2)=O)CC1 c1(OC)cc(OC)c(C(=O)N)cn1.C1CC(F)CN1C(=O)CC.CC(N)=O.C c1(C(C(=O)O)NC(C)CCOCc2ccccc2)cccc(Br)c1 Cc1ccnc(C#N)c1NC(C1CN(Cc2cnc(Cl)c(F)c2)CCS1)=O Cc1cc(C(=O)NC2CC(NC(c3cnsc3)=O)C(O)C2)c(C)[nH]1 Cc1cc(C(N2CCN(C(c3[nH]cnc3C)=O)CC2C)=O)c(F)cc1Cl C1(CC=O)CCCCN1C.Cc1oncc1C(=O)NC(C)C(=O)N.C1CC1.C c1(OC)cc2ccccc2cc1C(=O)NC1CC2(C1)CC2.C(=O)C(C)C(F)F.N C1(NC(CCOCC)=O)CN(C(=O)C(C(C)C)c2cccnc2)CC1OC c1(OCC(N2C(C(=O)NCCCC)CCC(C)C2)=O)ccc2c(c1)CCCN2 N1(C(C(CC2CC2)OC)=O)Cc2n[nH]cc2C1C(=O)N1CCc2oc(C)nc2C1 N1(C(C=C(C)C)=O)CCCC(C2CCN(c3cc(C)c([N+](=O)[O-])cn3)C2)C1 N1(C(CSC)=O)CCCN(C(=O)C(C)OCC(C)C)CC1 C(CC(C(=O)NCCOCCC(C)C)NC(c1ccccc1)=O)SC N1(C(c2ncn(C)n2)=O)C2CC=C(C(=O)NCC(O)C(F)F)C1CC2 C1(NC(C=CC(=O)N(C)C)=O)CC2CCC1CC2.C(=O)C(F)=CC1CC1.N C12(C(N(CCCCN(C(=O)C)C)C)=O)CCCC1(CN)C2.CC.C(N)=O.S Cc1c(C(=O)NCCC(C)Nc2cc(N3CCCC3)ccn2)cc(N)cc1O C1(C(C)C)N(C(C2CC2(C)Br)=O)CC12CCN(C(c1cc3occc3[nH]1)=O)CC2 Cc1ccncc1C(c1nnnn1C(C)C)NCC1(c2cnn(C)c2)CCCO1 Cc1cc(C(=O)O)c(F)cc1NC(c1cnn(CC2CCCO2)c1)=O N1(C(CC2C(NC(COCCCOC)=O)CCCC2)=O)CCOCCC1C C#CCCN=C(NCCCCn1ccnc1C)N1CCSC(C)(C)C1 N#Cc1ccc2c(c1)CCCC2C(=O)NC1CN(C(=O)CCCCC(F)(F)F)C1 c1(OCC)ccnc(NC(CCN(C)C(C2CC2C2CC2C)=O)C(C)C)n1 N1(C(CCCOCC=C)=O)CC2OCC(NC(c3nccnc3Cl)=O)C2C1 N1(C(c2cncc(C)c2)=O)CCC(C)C(NC(=O)CC(=O)NC2CC2)C1 C1(C=O)CC2(CCCCC2)C1.C1(C(=O)NC(C)C(C)C)(OCC)CCOCC1 CCCCC(O)C(C)C(=O)NCC1(CNC(=O)CCC(=O)NC)CCCCC1 N1(C(c2ccc(SCCC)cc2)=O)CC2CCCN(C(c3cocn3)=O)C2C1 c1(C=O)cccc2c1OCC2(C)C.C=CC(C)C(C)C(=O)N(C)CC1(C)CC1.N Cc1c(C(N2CC(C(C)NC(C3CCC(F)C3)=O)C2)=O)cccc1CO CN1CC(O)CC1C(=O)NC(c1cccc(Cl)c1)CNC(c1ccnn1C)=O CC1CN(C(c2cc(C(=O)OC(C)(C)C)co2)=O)CC1.C1(C=O)CCCC1.C c1(CS(=O)(=O)NC(c2cc(C3(F)COC3)no2)=O)ccc(Br)cc1 c1(OC)cc(OC)c(Cl)c(NC(C2(O)CCN(Cc3cnc(Br)s3)C2)=O)c1Cl C1(O)CCCN(C(C2CCCCS2(=O)=O)=O)C1.c1(COC)cc(C(=O)N)no1 C1(CC(=O)NC2CC(NC(CC(=O)NCC)=O)C2)CCCC(C#N)C1 C(=O)(CCCCCCCC1CC1)NC(CCCNC(c1ncc(CC)nc1)=O)C c1(OC)c(C(N2CCCC(C)C2)=O)csc1C.c1(C(=O)N)cc(C(N)=O)ccn1 N1(C(C(C)NC(c2cccs2)=O)=O)CCN(C(c2nnn(C)n2)=O)C(CCO)C1 CC(O)CCCC(=O)NC1CC(C)N(C(c2cc(C(N)=O)no2)=O)C1 Cc1occc1C(=O)NCC(=O)NCC(C(C)C)NC(=O)C.C1CCOCC1 O=C(C1CCc2nccn21)NCC1CC(O)CN1C(=O)COC1CC1 n1(CC)nc(C(N2CCCC2C(C)NC(=O)CC2CNC(=O)O2)=O)cc1O C(=O)(CCC(C)NC(=O)CC1CNC(=O)O1)NCC(CC)C#N c1(OC)cccc(C(C)(C)C(=O)NC2CCCN(C(C3CC4(CC4)CO3)=O)C2)c1 CCS(=O)(=O)CC(=O)N(CCC(=O)N1CCN2CCC1C2)OC C1(C#N)(OC)CC(C(=O)NC(CC2CC2)C(N2CCSC(C)C2)=O)C1 C(=O)(C1=Cc2ccccc2OC1)NCC(C1CCN(C(C2C(C)C2)=O)CC1)(C)O N1(C(CCN(C)CC)=O)CCCCC1C1(NC(=O)C(=O)NC2CC2)CC1 CC1CN(C(=O)C(C)(C)n2cnnn2)CCC1CNC(c1nccnc1N)=O C1(C(N(C2CCCN(C(c3cccc(N)c3)=O)C2)C)=O)CCN(C)S1(=O)=O C1(CC(N2C(C(N3CC(OCC#C)C3)=O)CC2C)=O)CC2CCC1C2 C1(CC(=O)NCC(CC=C)NC(c2ccc(Cl)cc2F)=O)CCC(=O)NC1=O c1(C=O)cc([N+](=O)[O-])ccc1.n1(CC)cc(C(=O)NCC2CC2)nn1.C CC12CCC(C(N3CCN(C(C4CC(C(F)(F)F)C4)=O)C4CC34)=O)(CC1)CO2 c1(OC)ccc(C(=O)NC2COCCN(C(c3c(O)cccc3Br)=O)C2)cc1O C1(C)(CC(=O)N(CCNC(C(c2ccccc2)NC(C)=O)=O)C)CCCCC1 C#CC(C(C)OC)NC(=O)CONC(C1CC(=O)CS1)=O c1(C(N2CC(NC(c3ccc(CC)[nH]3)=O)CC2(C)C)=O)cccc2c1nnn2C C1(C(=O)NCCNC(c2c(CC)n[nH]c2)=O)CCC(C#N)CC1 Cc1cc(C)c(C(=O)NC2CC(CCNC(C3CC(F)CN3C)=O)C2)cc1C c1(CN2C(COCC#C)CCC2)ccc2nccc(N)c2c1 C=Cn1nccc1C(=O)NC(c1cn(C2COCC2OCC)nn1)C Cc1nc(NCCCOCCCO)cc(=NCCc2ocnc2CO)[nH]1 c1(CN2C(CCC(=O)O)CC2)ccc(O)c(O)c1 c1(NC2CC(NC(C3C(C)(Br)C3)=O)C23CCC3)ccc([N+](=O)[O-])cc1Cl Cc1cc(C(=O)NC2CN(C(c3cc[nH]c3C(C)C)=O)CC2(C)C)c(F)cc1Cl c1(NC(C2N(C(C(C(=O)OC)C)=O)C3C(C2)C3)=O)ccc(Cl)c(C(C)=O)c1 N1(C(C(CC)(F)F)=O)CC2CC(NC(c3scnc3C(F)F)=O)C1C2 C(=O)(C1=CCCN(C(c2ncc(C)s2)C(=O)NCC(C)C)C1)OCC C(=O)(NNC(=O)NC1CCN(C(=O)NC2CCC(=O)NC2)C1)C1C(C)C1 C=C(C)CC(C(=O)N)NC(C)=O.c1(C(N2CCC2)=O)ccc(C2CC2)cc1Cl C(=O)(CCCCCC(C)O)NC1CN(C(c2c(OC)n(C)nc2)=O)CC12CC2 C(=O)C1=CCC(F)(F)CC1.c1(OC)ccc(C(F)F)cc1C(=O)NC1CCC1 c1(C(N(CCCC(C)(C)C)C)=O)cnc2ccsc2c1.C(=O)(CC=O)OCC.N N1(C(c2c(C)c(F)ccc2)=O)CCC(Nc2ncnc(=N)[nH]2)C2(CCC2)C1 Cc1c(C(=O)NCCCN(C(C2CC23CCCCC3)=O)C(C)C)sc2nccn12 N1(C(CC=C)=O)CC2COCC(C1)C2NC(=O)CC1C(=O)NN=C1C c1(CN2CC(C(N3C(CC(=O)OCC)CCCC3)=O)OCC2)cccc(C)c1C C1(C(N2C(CC)CN(C(=O)CC)CC2)=O)CCC(=O)CC1(C)C.CCN(C)C.O Cc1ccc2nc(NC(c3ccc(Oc4ccccc4)cc3)C)nc(O)c2c1 CC1OC2(CNC(=O)Cc3ccn(C)n3)CC1C2.C1(C=O)CC1C1CCC1.N Cc1ccc(F)c(C(=O)NC(C)C(C)(C)NC(=O)CC2CC(F)(F)C2)n1 C(C(C)C(C)C)NC(C1(CCOCC)CCCC1)=O.C(=O)C=CCO.N N1(C(C(CC)F)=O)CC(C2CN(C(=O)CCc3cncc(C)c3)C2)C1 c1(CNC(C2CCCS2)=O)nnc2n1CCN(C(C1CC3(CCC3)CO1)=O)C2 CC(C)=C=C1C(c2nc(-c3cccnc3C(F)(F)F)no2)C1(C)C C=C1CC2(C1)CC(C(=O)NC1CC3CC1N(C(=O)Cc1ccccc1C)C3)C2 C1(C(=O)NC2(CCCNC(C(CC)C)=O)CC2)CC(Cc2ccccc2)=NO1 c1(C(N2CCCC(CC(=O)Nc3cc(Cl)cc(Br)n3)C2)=O)cc(F)c(Cl)c(Br)c1 C1(C=O)CCCN(C(C23CC2CN(C(C2(C(F)(F)F)CCC2)=O)C3)=O)C1.CC CC(C)(CCCNC(C1CC12CC2)=O)NC(c1n[nH]c(C(C)(C)C)n1)=O N(C1CCC(C)(C)c2ccccc21)C(=O)Nc1cc(C)nc(C)n1 c1(CNC(c2c(C)oc(CO)c2)=O)nc2ccccc2[nH]1 C1(C(N2CCN(Cc3ncccn3)CC2)=O)Cc2ccccc2O1 C1(CNC(=O)CC2OCCO2)CCN(C(C2CCC3(CC2)CC3)=O)CC1O c1(C(N(C2CCCCC2)C)=O)cccn(O)c1=O.c1(COC)nocc1C(=O)N c1(C(=O)NC(CCCOC)C(N2CCCC3(CC2)CC3)=O)cnc2ccccn12 c1(NC(C=CC(=O)NC2C(NC(COCC)=O)C2)=O)cccnc1 C#CCC(C)(CNC(=O)CC1CN(C(=O)CC2OCCCO2)CCO1)CO C1(CNC(C(F)(F)C2(OC)CCC2)=O)CCCN(C(=O)C(C)C2CC2)C1 N1(C(C2CCN(CC(N)=O)CC2)=O)CC(F)(F)CC1CNC(C1CCC1)=O C(=O)(C1=CC(O)C(NC(C2CC(C)(F)C2)=O)C1)NC(C1CCCC1)C N1(CC)CCC(NC(=O)CC2(C)CC2)C1=O.c12conc1CNC2=O C(c1ccccc1F)=CCC(=O)N(CCC(C)NC(c1cc(C)nnc1)=O)C CC1=CCSC1C(=O)NCC1CN(C(C2CCC(O)C2)=O)C1 N1(C(Cn2ncc(N)c2)=O)CCCC(C2CCCN(C(C3(C(F)F)CC3)=O)C2)C1 c1(C(=O)NCC2CC(NC(C3(OC)CCCOC3)=O)C2)nc2ccccn2c1F C1(C(=O)N)CN(C(c2n[nH]c(C)c2C)=O)CCC1C.C1(CC)CC(C)CC(C)C1 CC(CCN=c1cc(CO)nc(Cl)[nH]1)NC(=O)CN1CCC(N(C)C)CC1 C1(C(=O)N(CCCN=[N+]=[N-])C)(NC(C(C)OCCC=C)=O)CCC(C)(C)C1 C1(C(N2CC(C(=O)NCC(C#C)CC)(CC)C2)=O)COCCC1C N1(c2c(Br)cnc(OC)n2)CCCC2(NC(=O)CCn3cnnn3)CC2C1 c1(OCC(=O)N(C)CCNC(=O)C(F)C2CCOC2)ccc2c(c1)CCC2 C1(COC)CCCN1C(c1[nH]nnc1C(F)F)=O.C(=O)CCc1cnoc1.C C1(C(N(CC(C)N(C(c2ccc(C)cc2)=O)C)C)=O)CC2OC(C)(C)OC2C1 C1(n2c(CC(n3c(C)ncc3)C)nc(C3CSC3)n2)CC(C)(C)OC1(C)C C(=O)(C(C(CC)CC)OC)NCC(C(=O)N1CCC(OCCC)CC1)C(C)C C12(CC(=O)Nc3c(C)n(C)nc3)CCC1CN(C(C1CC3C(C1)C3(F)F)=O)C2 CC1CN(C(c2cccs2)=O)C(C)C(C)N1CC(C1CCCCC1)=O C(=O)(CC(F)(F)C(F)(F)F)NC1CC(CNC(=O)Cc2ccsc2Cl)C1 c1(NC)ccc(NC(=O)NCC2CCCC(OC)C2)c(C(=O)OC)c1 C1(NC(c2coc(C3CCC3)n2)=O)CC(NC(C2CCCC2O)=O)C(O)C1 N1(C(CCCc2ccccc2)OC)CC(c2nc(C(C)OCC)no2)CC1=O C1CCN(C(C23CCC2C3)=O)CC1.C1(C(=O)N)CCCN(C(=O)CC2CC2)C1 C1(CC=C)CCCC1.c1(C(=O)N)conc1CC.c1(C=O)ccc(C(N)=O)o1 C1(CN(C)C(C2CC(O)(C#N)C2)=O)CCCCN1C(C1CCCOCC1)=O c1(C(=O)NC(CC)(CNC(C2CC(C)CO2)=O)CC)cnn(C)c1C#N c1(OC)cc(F)c(Br)cc1NC(C1(F)CN(C(c2ccnc(Cl)n2)=O)C1)=O c1(C(=O)N)cn(C)c2ccccc12.n1(CC)cc(CC(N2CC(O)(C)C2)=O)nn1 C=CCC(CC)C(=O)N1CCC(N(C(=O)CCc2ccc(CO)cc2)CCO)C1 C1(C(OC)OC)CN(C(C2CCCN2C(C2CC(F)C2)=O)=O)CCO1 C(=O)(C1CCN(C)c2ccccc21)N1CCC(C)(NC(c2c(CC)con2)=O)C1 C1(Oc2nnc(CN(C)CSCCO)s2)C2CN(Cc3cnc(C)[nH]3)CC12 n1(CCC)ncc(C(N2CCCC(C(C)(O)CNC(C3CC3)=O)C2)=O)c1Cl.S N1(C(c2ccc(C#N)o2)=O)CCC2(C1)CN(C(=O)CC1CCC1)CCO2 C1(C(=O)NC2CCC(C)(C)C2)CC12CCN(C(c1csnn1)=O)CC2 N1(C(CC=C)=O)CCC2(CCC(NC(C3(O)CCCC(C)CC3)=O)CC2)CC1 N1(C(c2c(CC)n[nH]c2)=O)CC2CCC(C1)C2NC(=O)C(C)O.C1CCCO1 C#CCCCC(C)C(=O)NCC1CN(C(C2(C(=O)NC)CCC2)=O)CC1(F)CO c1(C(N2CC(C)(C)C(NC(C3C=CCC3)=O)C2)=O)ccnc2[nH]cnc12 c1(C(C)(C)C)nc(C(=O)N)co1.C1C=CCC1.c1(C=O)cnc(C2CC2)s1.C Cn1cc(C#N)cc1C(=O)NCCCCC(N1CCSC2CCC12)=O c1(CN(CC(=O)O)C)cnn(Cc2ccccc2)c1 C1(NC(=O)CCOCC2CCC2)CCN(C(C2(CF)CC2(F)F)=O)CC1O C1(OC)CN(C(C2CC=CCN2C(C23CCC(CC2)C3)=O)=O)CC12CC2 C1(NC(C(C2CC2)OC)=O)CCN(C(C23COC(C=O)(C2)C3)=O)CC1.N c1(C(N2CCC(C(CNC(CCOCCOC)=O)C)CC2)=O)cccc(O)c1Cl C(c1ccc(Cl)nc1)=CC(=O)NCC1C2CN(c3cc(Cl)ncn3)CC12 C1(C)(C(N2C(C)(CC(N3CCN(CCCC)CC3)=O)CC2)=O)C(C)(C)C1(C)C Cc1cccc(C(N2CCC(CCNC(=O)CNC=O)CC2)=O)c1F CC1(C)OC2(C(=O)N3CC(C)(O)CO3)CC1(Cc1ccccc1)C2 C1(NC(=O)COCCc2cccs2)CCN(C(c2cccc(F)c2)=O)CC1F c1(C(N2CC(NC(C(C)=C(C)C)=O)C2)=O)cc(C)nc2cccc(Br)c12 C1(NC(c2c(C)[nH]c(=N)s2)=O)CN(C(c2ccc(Cl)o2)=O)CC12CCC2 N1(C(CC2(COC)CC2)=O)CCSCC1C(=O)NC(c1cncnc1)C c1(NC(C)=O)sc(Cl)cc1C(=O)NC1COCC1NC(=O)C(O)C(F)F c1(C(=O)NC2CCC(NC(C3CC(C)(O)C3)=O)CC2)nnc(O)nc1O C(CC(O)CNC(c1c[nH]cc1CC)=O)NC(CSCCC)=O C1(N(C(C2CC(OCC)C2)=O)C)CCCCN(C(C2CSCCS2)=O)C1 C(=O)(C(C)(C)C)NC(CC(=O)OC)C.n1(CC=O)nccc1.C(C)=O.N N1(C(C2(COC)CCCO2)=O)CC2(CCCN(C(c3ccc(Cl)cc3)=O)C2)C1 c1(C(N2CC3CN(Cc4cc(C)c(F)cc4)C3C2)=O)cccc2c1OCCC2 N1(C(C(C)(F)F)=O)CCCC2(CC(NC(=O)Cc3n[nH]c4ccccc34)CO2)C1 c1(C(=O)NCC(C)(O)CNC(c2nc(=N)cc[nH]2)=O)ccc2sncc2c1 N1(C(C=CC)=O)CCc2ccccc2C(N(C)C(=O)CC(C)CCC)C1 CC1CC(C#N)CN1C(c1occc1-c1ccc(F)c(F)c1)=O N1(C(Cc2c(C)cco2)=O)CCC(O)(CNC(=O)C)CC1.C(=O)N.C1CC1 CC1(NC(=O)Cc2ccc(Cl)s2)CN(C(c2cc(C3CCCC3)[nH]n2)=O)C1 CCC(C)CC(C)C(=O)N1CC2(CCC(CNC(c3csc(CO)n3)=O)O2)C1 N1(C(c2nc(CCCC)sc2)=O)CC(NC(=O)C(C)C2CCC2)CC(O)C1 c1(C(=O)NCC2(n3cccn3)CCN(C(CC)=O)CC2)c[nH]c2ncnc(O)c12 C(c1ccncn1)=CC(=O)N.n1(C(C)C)ccc(CC(=O)N(CC(C)(C)C)C)n1 CCC(C)C(O)C(C)C(=O)N1CCC2CCCC12C(=O)NOCc1nc[nH]n1 C1(C(N(CC)CC)=O)CCCCN1CC.c1(CC=O)cc(C)[nH]n1.CCO.N c1(N2C3CN(Cc4c(C)cc(O)cc4O)CC32)ccn2ncc(Br)c2n1 CC(C)(CCC(=O)NC1CC2CCCC2C1)NC(C1CCCC(C#N)C1)=O N1(C(C(CC)C)=O)CC2(C1)SCCC2NC(=O)CCc1ccsc1Br Cc1c(C(=O)NC2CCN(C(C3CC4(CCO4)C3)=O)C2)cnn1C(C)(C)C CCCCC(CC(=O)NC1CCC(N=[N+]=[N-])CC1)NC(=O)C(CN(C)C)CC c1(C=O)n[nH]c2c1COCC2.C=CCC(C(=O)NC1CC(F)(C)C1)NC(C)=O c1(C(=O)NC(C)(C)CN2CCN(C(c3nccs3)=O)CC2)cnc2n1CCC2 N(C1COCc2ccccc21)C(c1c(OC)cc(Cl)c(C)c1)=O N1(C(C2(CC)CCC2)=O)CCOC(CN(C(=O)CC)C)C1.c1ccc(F)cc1.S CC(=O)C(C)(C)CC(=O)NC1CCCCCC1C(=O)NC(C)CCC1CCCC1 C(=O)(C(CCC)CCC)N1CC(C=C)(CC(=O)N(CCCC)CCO)C1 C1(C(CNC(C2(COC)CCCO2)=O)(C)C)CCN(C(=O)C(O)C(F)F)CC1 C#CC(C)(C)C(=O)NCC12CC(CO1)C2.c1(CC(C=O)C)ccc(F)cc1 N1(C(c2ccc(=N)[nH]c2Cl)=O)CC2CCC(C)C2C1.C(c1ccoc1)=CC(=O)N c1(C(=O)NC2(C)CN(C(Cc3cnc(C)[nH]3)=O)C2)nc2c(s1)CCCC2 N1(C(c2cccc(C(N)=O)c2)C(=O)NCCCSCC)CC2CCOC2C1 N1(C(c2c(OC)ccc(Br)c2)C(=O)NC(C)(C)C)CCOCCC1(C)C CC1CCCC=C1C(=O)NC(C)(C)CCNC(c1ccc(O)c(F)c1)=O c1(C(N2C(CN(C(=O)CCC3CCCO3)CC)CCC2)=O)cncc(OC)c1 N1(C(c2c(CC)ocn2)=O)CCC(NC(c2cc(Br)c(C)o2)=O)C(F)C1 O=C(C1=CCS(=O)(=O)C1)N1CC2CC(Nc3ncc(Cl)c(O)n3)CC1C2 c1(C(=O)NCC(C)NC(C2(CC)CCCO2)=O)n[nH]c2c1CCCC2 CC1CC(O)CCN(C(C2COCCN2C(c2ccc(O)c(F)c2)=O)=O)C1 c1(-c2cn(C3(C(=O)OC)CN(C(CC(CC)C)=O)C3)nn2)cccc(Cl)c1C CC1(C)CCCC(C(=O)NC(CNC(=O)Cn2ncnn2)C2CCC2)C1 C1(C(=O)NC2(CO)CCN(C(C3(C)CC3)=O)CC2)Cc2ccccc2O1 N1(c2cc(NC3CC(C)N(C)CC3)nc(C(F)(F)F)n2)CCC([N+](=O)[O-])CC1 C(C(=O)NCC1CCOCC1)(C(C)C(C)(C)C)N(CCNC(C)=O)C c1(C(N2CC(NC(=O)C3=CCCC3)CC(C)(C)C2)=O)c(O)ccc2ccccc12 C1(CC(=O)N(CCOCCNC(C(F)OC)=O)C)OCCC1(C)C C1(OC)CCC2(C(=O)NC3(C)CCCCC3)CC12.C(=O)CCCc1cc[nH]n1.N N1(C(C(C)C2CCCC2)=O)CCC(O)(CN(C(=O)CC2CC(=O)NC2=O)C)CC1 C(=O)(C(F)(F)C(F)F)NC(C1CCN(C(c2ncccc2Cl)=O)CC1)C c1(C(N(CC(CC)NC(=O)C(C)(C)C2CCCO2)C)=O)c[nH]nc1-c1cccs1 N1(C(C(C)(C)C2CC2)=O)CC2CC2C1.C1(C(=O)N)CCCN(C(=O)C2CC2)C1 Cc1nc(C)c(C(=O)NC2CC(CNC(C3CCCC3(C)C)=O)C2)nc1C C(=O)(C(O)P(C)(C)=O)N(C(C)C)CCNC(=O)CC1CC2(CC2)C1 CCC(O)C(F)(F)C(=O)NC1CC2(C1)CC2C(=O)Nc1ccc(Cl)cc1 Cc1nn2cc(C(=O)NCC3CCN3C(=O)Cc3cnccc3C)nc2s1 C1(=CCNC(C2C(=C)CC2)=O)CCN(C(=O)C(CCC)OCC)CC1 c1(C(=O)NC2CC(NC(C3Cn4c(C)nnc4C3)=O)C2)cc2cccc(Cl)c2s1 N1(c2ncnc(N(C)CC)c2C)CCc2nnnn2CC1 c1(CN2CC(O)(CNC(c3cnc(O)[nH]3)=O)C2)c(Cl)cnc(Cl)c1Cl C1(CC)CN(C(c2nc(Cl)ccc2F)=O)CCC1NC(C1COC(C)(C)C1)=O CC(C)CC(C)(CNc1ncc(O)cn1)NC(=O)COc1ccc(Cl)cc1 S(=O)(=O)(CCCOC(=O)Cc1ccc(OC(F)(F)F)cc1)NCC(=O)O c1(C(N2C(CN(C(C(CC)SC)=O)C)CCC2)=O)ccc(C)cc1 O=C(O)CC(C(=O)NCC1CCC2(CC1)CC2)N1CCCCC1 N1(C(c2c(CC)ocn2)=O)CCC(C(F)C)CC1.c1(C=O)ccn(C(F)F)n1.N C1(C2N(C(CN(C(C)=O)C)=O)CCC2)CCN(C(=O)C=Cc2ccncn2)CC1 CC1CN(C(c2ccc(C(F)F)c(F)c2)=O)CCN1C(C1CCC1)=O C1(O)(C(N2CC(O)CC(NC(c3cc(C)n(C)c3C)=O)C2)=O)CCCC(C)(C)C1 c1(C(N2CC(CCNC(c3ccc(C(C)=O)s3)=O)C2)=O)ccc2c(c1)OCCO2 C1CN(C(=O)CN(C)S(=O)(=O)N(C)C)CCCO1.Cc1noc(C(=O)N)c1C.C c1(C(=O)NC(c2cccc(OC)c2)CC)cnc(=NCC)[nH]c1 C#CC1CN(C(C2C(C)C2C)=O)CCN1C(=O)C(C)n1cccn1 N1(C(CC(CC)O)=O)CCCC(C2CCN(C(=O)COC3CCC3)CC2)CC1 C1(NC(C2C(c3n(C)cnn3)CC2)=O)CCCN(C(=O)Cc2nc[nH]n2)C1 C1(C#N)(C(=O)NCC2C(NC(C(c3cccc(C)c3)C)=O)CCC2)CCOCC1 Cc1coc(C)c1C(=O)NC(C)C(C(C)C)NC(=O)Cc1cncnc1 C(=O)(C#CC(=O)N(C)C)NC(C(C)C)CNC(=O)CCc1cncn1C C(=O)(CC(C)(C)C(F)F)N1C(CCNC(=O)Cc2nonc2C)CC(OC)C1 Cc1cc(Cl)ncc1CNC(=O)N(C(C)C(=O)N)C(C)C.c1ccccc1F c1(C(=O)NC2CC(OC)CN(C(=O)CC3CC(SC)C3)C2)cnn2ccncc12 C(c1ccc(Br)c(Cl)c1)=CC(=O)N(C(c1cccnc1)C)CC N1(C(c2cc(C(=O)OC)on2)=O)CCC2CC(C1)CN(C(C1CC1C)=O)C2 CC1(C)C(CC(=O)NCCOC2CCC2)CCN1C(c1cc(Cl)no1)=O c1(C(N(CC(O)CNC(=O)CC2CSC2)C)=O)ccc2c(c1)COCC2 C1(NC(CCN(C(C)C)C(c2c[nH]c(C(N)=O)c2)=O)=O)CCCCCC1CO C1(CCC)CN(C(=O)COC(F)(F)F)CCN1C(C1CCCOC1)=O N1(C(C(C)SCCCC)=O)CC2(C(=O)NCC(C)(CC)C(N)=O)CCC1CC2 C(C)(C(=O)NC1C2CN(C(C3CC4(CCOC4)C3)=O)CC12)(C(C)C)OC CCCCCC(CC)C(=O)NCC.C1(C(=O)N)CN(C(C2CC2CC(C)C)=O)C1 c1(OC)cc(C)nc(NC2(CF)CCN(C(C3CC3C3CCCC3)=O)C2)n1 C(=O)(N=c1cc(-c2ccccc2Cl)[nH][nH]1)C1N(Cc2c(C)noc2C)C2C(C1)C2 C1(N(C2C3CCC2CNC3)C(=O)NCc2cccc(C)c2)CC(C)(C)OC1(C)C CC1(C#CC(=O)NC2CCCN(C(=O)CONC(=O)OC(C)(C)C)C2)CC1 N1(C(Cc2cc(C)sc2)=O)CC=C(C(=O)NC2CCC3(CCCC3)C2)CC1 C=C(C)CC(C)C(=O)NCCOC1CN(C(=O)COC2CCOC2)C1 S(=O)(=O)(c1[nH]c(=NCC2(N(C)C)CCOCC2)ccc1Br)NC1(CC)CC=CC1 c1(C(=O)NC2C(NC(COc3c(C)cccc3)=O)CC2)cc(N)cnc1C Cn1cc(C(N2CC3CC(NC(c4cnn(C5CC5)c4)=O)C2C3)=O)ncc1=O c1(C(N2CCC(CN(CC(=O)N(CC)CC)C)C2)=O)cccc(F)c1F Cc1ccc(C(C)NC(=O)NC23CCCC(CC2CO)C3)cc1[N+](=O)[O-] Cc1cc(CO)oc1C(=O)NCC1CCCCC1NC(=O)C.c1nc[nH]n1.S c1(-c2c(OC)nc(OC)c(C)c2)cc(N=c2ccn3ncc(Br)c3[nH]2)ccn1 CP(C)(=O)CCC(=O)NCC1(CNC(C2CCC3CC3CC2)=O)CCC1 C1(NC(CCN(C(CCN(C)CCO)=O)CCCO)=O)CCCC1(F)F C(c1cccc(Cl)c1)=C(C)C(=O)N1CCC1CNC(=O)CCS(C)=O N(C1CCCc2ccc(F)cc21)C(C1OC2CCC1C2)=O N1(C(CCN(C(c2ccnc(C)n2)=O)CC2CC2)=O)CCC(C)C(C)C1 C1(NC(c2nc(C)sc2)=O)CCN(C(C2CC(C#N)C2)=O)CC1O C1(C(=O)NCCCCCCNC(=O)C=CC(C)(C)C)(CC)CC(C)(C)C1 C1(CNC(=O)CC2CCCS(=O)(=O)C2)CC2CCC(C1)N2c1nnc(CO)s1 N1(C(CCCNC(N)=O)=O)CC2CC2(C)C1.c1(C(=O)N)cc(-c2ccco2)[nH]n1 C(C(C)(C)C(=O)NCCc1n[nH]cc1C(=O)NC1CC(C(C)O)C1)OC C=CCC(CC(C)C)C(=O)N(CCCNC(c1coc2c1CSC2)=O)CC Cc1cccc(C)c1NC(N1CCN(C(=O)CC(c2ccccc2)N(C)C)CC1)=O N1(C(CCCc2onc(CCC)n2)=O)CCCN(C(=O)CC2CCCC2O)CC1 CC1(O)CN(C(C2CCCCCC2NC(=O)C=Cc2ccsc2)=O)CCC1O N1(C(C(C)NC(COC)=O)=O)CCCC1CC.c1(CC(=O)N)csc(Cl)c1 N1(C(c2c(OC)ccs2)=O)CC(NS(=O)(=O)CCCl)C(C)C1 N1(C(C=C(C)CNC(C2CC=CC(O)C2)=O)=O)CCCCC(CO)C1 c1(C(=O)NC2(CNC(C(CC)N(C)C)=O)CCOC2)cc(O)n(C)n1 c1(C2(C=O)CC2)ccc(Cl)cc1.C1(CCNC(c2ccoc2Cl)=O)CCCC1.N c1(C(=O)NCC(CC)NC(c2scc3c2OCCO3)=O)c(O)nnc(C)c1C C12(CC(=O)OC)CCCCC1N(C(c1cc([N+](=O)[O-])cc(F)c1OC)=O)CCC2 C1(NC(Cc2cnc(C)o2)=O)CCN(C(=O)CC(C)C(F)F)CC1F c1(OC)ncc(CN2CCCC2C(=O)NCc2c(O)cccc2F)c(OC)n1 C1(C(C(=O)NCCCN2CCCC2)NC(C2C(C)(C(F)F)C2)=O)CCCCC1 c1(OC)cc(F)ccc1C(=O)NC1CN(C(=O)CC2CC(SC)C2)CC1(C)C O=C(CCCCCCCBr)Nc1ccccc1C1CCN(c2ncccn2)CC1 N1(C(c2c(C)scc2)=O)CCCC(O)(CNC(=O)C(C)(C)C2CCOCC2)C1 N1(C(CNC(C)=O)=O)CC(O)(CCNC(c2ocnc2C2CC2)=O)C1 C(=O)(CCCCC(F)(F)F)NC(CC)(CNC(=O)Cc1cc(C)no1)CC N1(CCCNC(C(C)Sc2ncccn2)=O)CCN(C(=O)CC(C)(C)C)CC1 CCC(C)(C#N)C(=O)NCCC1(C)CCN(C(=O)C=Cc2cn[nH]c2)C1 N1(C(C2N(C)CC(F)C2)=O)CC2CC1CN2C(C1(F)CC1)=O N1(C(CN(C(=O)COC)CCC)=O)CC(N(C)C)C(C)(C)C1.C1CCC1 C1(O)(CC)CCN(C(=O)Cn2ccc(=N)[nH]2)CC1.c1cc(C=O)sn1.CCO N1(C(C(CC)C)=O)CC2CCC1C(C(=O)NCc1cc(Cl)ccn1)C2 c1(N2CCC(NC(C3C(CC)CCC3)=O)CC2C)ncc2ccsc2n1 c1(C(=O)NCC2CC(NC(C(C)(C)C#N)=O)C2)c(F)ccc(Br)c1Cl c1(C=O)cc(S(N)(=O)=O)cn1C.C1(NC(C(=O)NCC)=O)CCCC1.C S(=O)(=O)(c1ccc(C#N)c(N2CCOCC2)c1)N1CCC(C)C(F)(F)CC1 C1(OC)CCC2(C(N3CC(CNC(=O)C(C)C#N)C3)=O)CCC12 C1(NC(COc2cn(C)nc2)=O)CN(C(c2c[nH]c(=N)o2)=O)C(C)(C)C1 C1(COC(C(c2ccccn2)C)=O)CCN(C)CC1 CC1CN(C(=O)CC2CC(NCc3cc(F)ccc3C(=O)O)C2)CCC1O C1(NC(=O)OC(C)(C)C)CS(=O)(=NC(=O)C2CNC(=O)C2)C1 C(=O)(CCC(C)c1ccc(Br)cc1)NC1C(CNC(C2CC(OC)C2)=O)C1 Cc1cc(F)ccc1C(=O)N(C(C)CN(C(=O)C(C)n1cccc1)C)C C1(NC(CCOCC#C)=O)CC2CCC1(NC(C1CC1(F)F)=O)C2 Cc1cc(O)cc(C)c1C(N1CC2CN(C(=O)C=Cc3ccc(Cl)cc3)C2C1)=O C1(C(=O)NC2CCC(N(C)C(c3cccnn3)=O)CC2)CCCC2C1C2(F)F Nc1ccc(Cl)cc1C(=O)NC1(CCO)CN(C(=O)CCc2ccccc2F)C1 c1(CNC(c2n(CCC(C)C)ncc2)=O)ccc(Br)cc1I Cn1cc(C2=NOC(C(=O)NC3CC(F)C3)C2)cn1.C1(CC=O)C=CCC1.C c1(C(N(C)CC2CC2)=O)ccc(S(N)(=O)=O)cn1.C1(C)(C=O)CCCN1C c1(NC(=O)NC)cccc(C(=O)NC2CC(NC(c3ccnnc3)=O)C2)c1 c1(C2(C(=O)NCc3csc(Cl)c3)CC2)cccc(Cl)n1.C1(C=O)CCC1.C CCC(C(=O)OC)C(=O)NCC(C)(C)CN(C(=O)CCc1cncnc1)CC CCCC(CC(C)C)C(=O)N(CC(=O)NCCC(CCC)C1CC1)CC1CC1 N1(C(C2CCC(C)N2C(c2cccc3ccnn23)=O)=O)Cc2nncn2C(C)C1 CC(C(=O)N1CCCCC1C1CCCN(C(C2(C#N)CC(=O)C2)=O)C1)C(C)(C)C CN1CCC(=O)Nc2cc(C(=O)NC3CCCC3C)ccc21.C(=O)C=CCF.N c1(CC=O)cccc(S(C)(=O)=O)c1.CC(C)C(C)C.C1(CC=O)CC12CC2 C1(NC(CCCOC(C)C)=O)CCN(C(=O)C=Cc2ccncn2)C(C)C1 c1(CN(C(=O)CCn2cnnn2)C)ccc(C)cc1.C(=O)CCc1cscn1.N c1(C(N(C(CNC(c2c(C)nns2)=O)C)C)=O)ccc2c3c(cccc13)CC2 N1(C(Cc2c(C)ccc(F)c2)=O)CC2CCN(C(c3ncc(F)cn3)=O)C2C1 c1(N(CC(C2CCC2)OC)C)nc(N2CC3C(C)C3C2)c2c(ncn2C)n1 c1(C(=O)NCCN(C(=O)C(C2CCOCC2)F)CCCN(C)C)ccccc1 C12(CNC(=O)Cc3ccc4c(c3)CC4)CCCC1CCN2C(=O)CO.CCCF N1(C(Cc2cc(C)sc2)=O)CC(NC(=O)CC2CN(C)C2)CC1(C)C C(=O)(NN1CCOC1=O)c1cc(C)cc(C)n1 Cn1ncc2cc(C(=O)N)cnc12.C12CC(CN1C(C1(C(N)=O)CCC1)=O)C2 n1(CC#C)cc(SCc2ccnc(OCCC)c2)c2ccccc12 C12(C(=O)NCC(CC)(C)O)CCCC1CCN2C(=O)Cc1c(C)noc1C C1(NC(C2(OC)CC(c3cn(C(c4ccccc4)C)nn3)C2)=O)CCCCCC1 C(=O)(C1CCCc2ncnn21)N(CC(C)NC(=O)C1=CCCCCC1)C c1(CN2CCC(N(C(C(c3ccc(OC)cc3)O)=O)C)C2)cccc2c1OCO2 C1(C(=O)NC(CC=CC)CO)(C(C)C)CCN(C(=O)CC=C(Cl)Cl)C1 C(C(F)(F)C(=O)N1CCN(C(c2cc(C(F)(F)F)ncn2)=O)CC1)OC c1(C(=O)NCC(CC)NC(C2CCOC2)=O)cnc2c(F)ccc(F)c2c1 c1(OC)cc(C(=N)NOCC2CC(=O)N(c3cccc(Cl)c3)C2)ccn1 C1(C(N2CCN(CCCC)CC2)=O)CCN(C(=O)C(C)(F)C(C)(C)F)C(C)(C)C1 Cc1ncsc1C=CC(=O)NC1CC(NC(c2ccc(N3CCCC3)nc2)=O)C1 C1(NC(C(C(=O)NC)(C)C)=O)CN(C(=O)Cc2cncnc2O)CC2(CCC2)C1 C1(C(=O)NC2CCC(C(=O)OC)C2)CCCCN(C(C2CN(C)CCO2)=O)C1 N1(C(C2(COC)CC2)=O)CC2CCC1C1CN(C(C3(C)CCN(C)CC3)=O)CC21 C(=O)(N=c1cc2n([nH]1)CCCC2)C1(CC)CCN(C(C(CCC)C#N)=O)C1 c1(C(=O)NCC(C)N(C)C(c2csc(C#N)c2)=O)cc2cc(Cl)ncc2[nH]1 C(=O)(CCCCCF)N(C(C)CCNC(c1cc(C2CC2)ncn1)=O)C CC1CCn2cc(C(=O)NCC3CCN3C(=O)CC3CCCOCC3)nc2C1 C1(CNC(c2ccc(C)c(F)c2)=O)CC2COCC2N1C(=O)Cc1ccno1 Cc1ccc(C(N2CCCC(N(S(C)(=O)=O)C)C2)C(=O)NC2(C)CC2)nn1 c1(CC)nc(C(=O)NCC(C)(O)CNC(=O)CCc2cnc[nH]2)cs1 N1(C(C(CO)N(C)C)=O)CCOC2CN(C(c3ccc(Cl)c(C(F)F)c3)=O)CC12 C1(F)CCCN(C(c2ccc(C(F)(F)F)c(F)c2)=O)C1.CC(C)(C)CC(=O)N.C c1(CC)c(OC)cc(C(=O)NC2CCC23CN(C(=O)C(C)(C)CC)C3)cc1O C=CCC(C(=O)OC)NC(C1(NC(=O)CC2CCCCCC2)CCSC1)=O c1(C(N2C(C)CN(C(c3csnn3)=O)CC2)=O)ccc([N+](=O)[O-])c(O)c1 CN=c1ccc(C(=O)NC(CO)C(C)NC(c2nn(C)c(C)c2Cl)=O)c[nH]1 c1(C(N2CC(NC(C(C)=CC)=O)C3(C2)CC3)=O)cc(N)c2ncccc2c1 C(CC(C(=O)NC1(C)CCN(C(c2cnc(C)o2)=O)C1)OC)OC C12(CNC(c3n(C)cnc3)=O)CC(CN1C(=O)CC1CCCC(=O)N1)C2 C1(C(N2CCC(N(C(CCCc3cc(C)no3)=O)C)C2)=O)CC(=C(F)F)C1 N1(C(C(C(C)(C)C)c2cc[nH]n2)=O)CCC2C(CCN2C(C2CS(=O)(=O)C2)=O)C1 c1(C(N2CCCC(NC(c3nc(C)sc3)=O)C2C)=O)cc(O)c2ccoc2c1 C(=O)(CS(=O)(=O)CC)N(CC(N1CC(O)(CC=C)C1)=O)C c1(C=O)cc(C=O)n(C)n1.c1(C(N(CCC)C)=O)cc(C(C)=O)oc1C.CO C1(OC)(CO)CCN(C(c2[nH]ccc2CNC(c2cnc(N)cn2)=O)=O)C1 N1(C(c2cccc(CC)c2)=O)CC2(CCCC2)C1C(=O)NOC(C)CC Cc1ccc(C(=O)C(C)Sc2nc(-c3ccc(Br)cc3)no2)cc1C N1(C(C2C(C)(C)C2)=O)CCCC(CNC(=O)CCn2cccn2)CC1 CC1(F)CC2(CN(C(C3(CNC(c4cc(Cl)no4)=O)CC=CC3)=O)C2)C1 CC1(C)CCCN(C(C23CCCC2C3(F)F)=O)C1CNC(=O)CCP(C)(C)=O N1(C(=O)OC(C)(C)C)CCC(CCC(=O)N2CC(CN3CCC3)C2)CC1 c1(NC(C(C)(C)N(S(C)(=O)=O)C)=O)cccc(-c2cscn2)c1 C(=O)(C(CC)C(C)(C)CC)N1C(C)CC(NC(C=C(CC)CC)=O)C1 C(=O)(CCCCCC#N)N1CC(C)CC(NC(CC(C)OC)=O)C1 c1(C(=O)NCC(C2CCOC2)NC(=O)C(=Cc2c[nH]cn2)F)ccc(F)s1 c1(C(=O)NCCC(C)NC(c2ccc(Cl)c(F)c2O)=O)cnc2n1CCCC2 N1(C(C(c2cncc(F)c2)C)=O)CCC2(NC(c3ccc(Cl)cc3)=O)CC2C1 n1(CC(=O)NCC(CNC(CC2(C#N)CCC2)=O)O)c(O)nc2ccccc12 CC1(C)CCC(C(=O)NCc2cccnc2)(NC(=O)CN2CCCNC2=O)C1 C(=O)(CCCCNC(C1CCCC(=O)N1)=O)NC(CC#C)CO c1(CN(C2CCOC(C)(C)C2)CC)ccc(I)c(Br)c1 c1(CC(=O)NC2C(NC(C3(CC)CCC3)=O)CCC2)ccc(OC)cn1 C1(C(=O)NCC(CC)C)CC(=O)N(c2nccs2)C1.c1(C=O)sc(C)cc1C.N CC1=NOC(C(N2CCC(N(C(=O)Cc3nnc(O)s3)CCO)C2)=O)C1 C(=O)(C(O)C(F)F)NC1(CNC(c2n(CC)cnn2)=O)CCC1 N1(C(C2CCCN(C(CCC)=O)C2)=O)CCCC(S(N)(=O)=O)C1 C(=O)(C1CCCc2nn[nH]c21)N1CCC(O)(CNC(c2c(O)cccc2Cl)=O)C1 N1(C(c2c(OC)n[nH]c2)=O)CCC2(C1)CN(C(c1ccoc1C(C)C)=O)C2 Cc1onc(C(F)(F)F)c1C(=O)N.C1CC(F)CN1C(=O)C(F)OC(F)(F)F C1(CC(=O)NCCCNC(C2(C=C)CC2)=O)CCCCC1C CC1CC(C(N2CCC(N(c3ccncn3)C)CC2)=O)CCS1 C1(NC(c2ncc(OCC)nc2)=O)CCC(O)CN(C(=O)C2=C(C)OCCC2)C1 C1CCN(C(C2(C(F)(F)F)CC2)=O)C1.C1(CC=O)CS(=O)(=O)C1.CO c1(CC)ncc(C(=O)NC2(CC)CN(C(c3c[nH]nc3CC)=O)C2)c(C)n1 C=CC(CC)CC(=O)N1CC(n2cc(C3CCCCC3)nn2)CC1C(=O)OC CC(CC(=O)NC1CC2C(NC(c3cc(C4CCC4)[nH]n3)=O)C2C1)P(C)(C)=O c1(SC)ccc(C(N2CCCC2C2CC2)=O)cn1.C(C(N)=O)(C=O)C1CC1.N c1(OC)nc(N2CC(CN(C(=O)CC3CCC(C)C3)C)C2)nc2[nH]cnc12 CC(C)(CCCN=c1[nH]cncc1Br)NC(C1(CS(C)(=O)=O)COC1)=O C(=O)(C1=CCC(NC(=O)CNC(=O)C(C)(C)C)C1)N1C(C(C)C)CC1 C(=O)(C(CN=[N+]=[N-])NC(c1ccncc1NC)=O)NCCCOCCCC C1(NC(Cc2ccn(CC)n2)=O)COCCN(C(=O)CCC(C)O)C1 c1(C(=O)OC)nn(C)cc1C(=O)NC1CN(C(=O)CCN(C)CCO)CC1 c1(CC(N2CCN(C(Cc3c(C)nn(C)c3)=O)CC2)=O)ccc2c(c1)ncn2C C1(C(N(C)CC)=O)OC2CCC1C2.C1(C(=O)N)CC(N2CCCC2)C1.C1CC1 C(=O)(C(C)(C)CCS)N1CCC(CC=C)(NC(C2C(OCC)C2C)=O)C1 CC(C)C(CNC(c1cnoc1-c1cccs1)=O)NC(=O)C(N1CCSCC1)C c1cc(Cl)c(Cl)cc1C(=O)NCC=O.C(=O)(C(C)n1cccn1)NCC.C C1(C(=O)NC(CC)(CNC(c2cc(C)on2)=O)CC)CC(=O)C12CCC2 C1(CC)CN(C(=O)CONC(=O)C2(C(C)=O)CC2)CCO1 C1(C(=O)NC(C#CC)(C)C)(COC)CC12CCC2.C12CCC1NC2=O.O S(=O)(=O)(c1cc(Cl)ccc1Cl)NCC1(C)CN(Cc2ccc(O)cc2)C1 c1(C(=O)NCCCN(C(C(CC)O)=O)C)cc(OC)cc(Cl)c1F CC(C)(F)CCC(=O)NCCCOC1CCN(C(c2nc(Cl)ccc2N)=O)CC1 CCS(=O)(=O)C=CC(=O)N1CC2C(CNC(c3ccc(F)c(Cl)n3)=O)C2C1 c1(OC)ccc2oc(C)c(C(=O)NCC3CC4(CCC4)C3)c2c1.C(C)(=O)N c1(CN2CCN(C(C#CC)=O)CC2C#N)cn(CC)c2ccccc12 C=C1CC2CCC(C1)N2C(=O)NC(c1nc(C)cs1)C C(c1cccc(Cl)c1)=C(C)C(=O)NCCCCCCNC(C1CC1F)=O c1(C(N2CCC(NC(c3n(CC)nnc3)=O)C2(C)C)=O)cc2sccc2cn1 N1(C(c2c(C)onc2)=O)CCC(F)(CNC(=O)CN2CCP(C)(=O)CC2)CC1 CC1CC(NCc2cccc(I)c2)CCN1Cc1ccco1 C12(NC(C)=O)CCC(C(=O)Nc3cccnc3I)(CC1)C2 c1(CNC(C=C(CNC(C2(OC)CC2)=O)C)=O)ccc(O)cc1C N1(C(CC=C=C)=O)CCC(C)(C)C(NC(=O)C=Cc2ccc(SC)s2)C1 C1(NC(C(=O)NC(C)C)=O)CN(C(=O)C=CC(N)=O)C2CCCCC12 CC1CC(C(=O)NCCNC(C2(c3cc[nH]n3)CC2)=O)C(=O)O1 C1(CNC(C(C#C)(C)C)=O)(NC(c2[nH]c(C)nc2C)=O)CCC(F)(F)CC1 C1(CC=O)CCC(C)(O)CC1.c1(CC(C)C)nc(C(=O)NC(C)CC)cs1.N N1(C(CS(=O)(=O)NCC)=O)CCC2(C1)CN(C(=O)CCCC(C)O)CC(C)O2.C c1(CC)ccc(C(=O)NC2CC(C)N(C(c3cscc3Cl)=O)C2)cc1N CCCC(C#N)C(=O)NCC1CN(C(c2[nH]nnc2C)=O)C(C)(C)C1 N=c1[nH]c(=NCc2cccc(C(N)=O)c2)[nH]c(=NCCc2c(Cl)cncc2Cl)[nH]1 c1(C(N2CC3CC2CN3C(c2cc(Cl)n[nH]2)=O)=O)ncnc(O)c1F c1(NC(C2CCN2C(c2cc([N+](=O)[O-])ccc2O)=O)=O)ncc([N+](=O)[O-])cc1Br c1(CCC(N2CCC(C)(NC(COCC=C)=O)C2)=O)c(C)nn(C)c1C c1(C(N2CC3CCCN(C(C4CCC(F)C4)=O)C3C2)=O)cnc2nccnc2c1 c1(CC)ncc(C(=O)NC2CC(C)C2)s1.c1(CC=O)ccccc1.C(=O)C C(CS(=O)(=O)NCC(=O)N)OC(C)C.C(C)CC.C(=O)C(F)=CC1CC1 C(=O)(CCCCCNC(=O)C(C)CC(N)=O)NCCOCC(C)C c1(CN(CC(=O)OC)CCN(CC=C)C(C)C)cn(CC)nn1 C12(C=O)CCCC1(C=O)C2.C1(=C(C(=O)NCC)F)CCCCC1.C1CC1 Cc1nn2c(c1C(N1CCC(CO)(NC(=O)Cc3ccon3)C1)=O)CCCC2C CC#CCCCC(=O)NCc1ccc(CNC(=O)Cc2cccc(C)c2)c(F)c1 c1(C(=O)N)ccn2nnnc2c1.N1(C(c2ccc(CC)s2)=O)CC(C)C2(CC2)C1 C(=O)(C(C)(N)C(C)(C)C)NC1(c2cccc(OC)c2)CC1 c1(C(N(C)CC2(O)CCN(C(c3cnco3)=O)C2)=O)c[nH]c2cccc(F)c12 c1(C(N(C)CC2CCCN2C(=O)Cn2cccn2)=O)cc(C#N)ccc1O N1(C(CCC#C)=O)CC(NC(=O)C(F)COC(C(C)(C)C)=O)C(C)C1 N1(C(C)C)CCCC(NC(=O)CC2COCCN2C(=O)CC2CCC(C)(C)O2)C1 CCCCCC(O)C(=O)NC(c1ccccc1)CNC(C1(OC)CCOCC1)=O CCCCCC(CC)C(=O)NCC(O)CN(C)C(C1CCC(N=[N+]=[N-])CC1)=O c1(C(=O)NCCC2CCC(NC(c3n(C)ccn3)=O)C2)cccc(C=C(F)F)c1 C1(COC)(OC)CCCN(C(C)=O)C1.c12ccc(cc1)C(=O)NC21CCC1 n1(C(CC)(C)C)nnnc1C(C1C2COCC12)(C)NCC(=O)N(C)O C1CCN(C(c2ccc(C(F)(F)F)cn2)=O)CC1O.CCS(=O)(=O)NCC(=O)N C1(C(N2CC(C)C(NC(=O)C(C)(C)C)C2)=O)Cc2ccccc2S1 n1(CCC)nccc1C(=O)N(CCC(=O)NCCCCCO)CCO C1(OC(CC2CCN(C(C)=O)C2)=O)CCCC1C(=O)NOC C(=O)(C(F)(F)CF)N(C)CC1CCCN1C(=O)CCn1cc(Cl)cn1 c1(C(=O)NCC(CO)NC(CC(CC)(C)C)=O)ccc2c(c1C)CCC2 CC1CCCCC1(CNC(=O)CC1CCCC(C#N)C1)NC(C1SCCCS1)=O C(=O)(C(CO)C(F)(F)F)N1C(C(=O)NC(C)CN2CCOC2=O)CC1C C(=O)(N(OC)C1CCOCC1)C1CN(C(c2c(CC)nn[nH]2)=O)CC(C)C1 O=C1NC(=O)c2cc(NC(C3(F)CN(c4ncnc5[nH]cc(I)c45)C3)=O)ccc21 c1(C(=O)NCCN(C(=O)CN2CCCCC2)C(C)C)cccnc1-n1cncn1 c1(CC=O)cccc(C#N)c1.c1(C(=O)NC2(C(N)=O)CC2)cc(C)on1.N C1(C(=O)NCC#CC#CCO)CN(C(=O)CC2CCCO2)CC12CCC2 C1(CNC(c2c(C)cc(F)cc2)=O)CC2(CN1C(c1cccn1C)=O)CC2(F)F C1(C(C)NC(C2CC3(CCC3)C2)=O)CCCCN1C(=O)CC1CCCC1(F)F C(=O)(C(CC)CCCCC)NC(C(CC(=O)NC(CC#C)C(=O)NC)C)(C)C C1(CC(C)C)CCCCN1C(C1(Sc2cccc(Br)c2)CC1)=O C(=O)(C(C)CC(F)F)N(C)CC1N(C(c2c(C)n(C3CC3)cc2)=O)CCC1 C(=O)(CC(C(C)C)NC(=O)CP(C)(C)=O)N(CCC)C c1(C(N(CCNC(c2ccc(SC)s2)=O)C2CC2)=O)ccn(CCO)c1C Cn1cc2ccc(C(N3CCCC(CNC(=O)C(F)(F)CF)C3)=O)cc2n1 c1(CN(C)CC)cn(CCCC(=O)NCC2(C)CC2(F)F)nn1 C#Cc1cccc(C(=O)NCC2CN(C(C3CCCO3)=O)CC23CC3)c1F c1(CCC(N2CCN(C(c3c(C)cn(C)n3)=O)CC2)=O)cc2ccccc2o1 c1(C(=O)NCC2(Nc3nc(C)cc(OC)n3)CCCCC2)ccc2cnnn2c1 C=CC1(C(=O)NCCC(C)CC)CCN(C(=O)C=CC2CCC2)C1 c1(C(CC)C(=O)N2CC(CNC(=O)CN(CC)CC)C2)c(C)noc1C.O Cc1ccc(C#N)cc1S(=O)(=O)N1CC2C(C(=O)NCC(N3CCCC3)=O)C2C1 C(=O)(C(C)(C)C(C)(C)O)NC(CC=C)CC(=O)NC1(C=C)CCCCC1 c1(SC)cccc(C(=O)NCC(O)CCNC(=O)C(O)C(F)(F)F)c1Cl c1(C(=O)Nc2ccc(Cl)c(N3CCNC3=O)c2)cc2cc(C(F)(F)F)ccc2s1 C1(NC(c2cc(-c3ccoc3)[nH]n2)=O)CCN(C(=O)CN2CCOCC2)CC1O C1(C(C)C)(C(=O)NCC2CC2(F)F)CCCN1C(=O)CCCn1cncn1 n1(CC(N2CC(C(C(=O)N(C(CF)CF)C)OC)C2)=O)cccnc1=O CC(C)C(C)CCNC(c1ocnc1C1CC1)=O.c1(C=O)cnn(C2CC2)c1 C1(C(=O)NCC2CCCN(C(C3CCCC(C)C3)=O)CC2)Cc2ccncc2C1 N(C1CCCc2ccccc21)(C(=O)NC1CCc2n(cc(C)n2)C1)CCO c1(C(=O)OC(C(=O)OCC)C)sc(=N)[nH]c1Cc1ccc(F)nc1 c1(CCC(=O)N)ccc(Cl)cc1F.C(C(F)C)NC(C1C(C(=O)OC)C1)=O c1(OCC)cccc(C(=O)N(CC(C)NC(C2CN(C(C)C)CCO2)=O)C)c1 C(=O)(C1Cc2c(Cl)cccc21)N1CC2(CN(C(C(CCC)N(C)C)=O)C2)OCC1 c1(C(=O)NCC(CNC(CN2CCC(C)(C)C2)=O)(C)O)c(O)nnc2c1CCC2 C1(NC(C2C=C(C)CS2)=O)CCCCCC1C(=O)NCCCCC1CC1 C1(C(=O)NCC2(O)CC(NC(C=CC)=O)C2)Cc2cc(Br)ccc2O1 C(=O)(C1COc2ccc(F)cc21)N(CC)CC.C1(OCC)CC(C(=O)N)C1 C1(CNC(=O)C=CCO)CCCC1NC(=O)CC(=O)NC1CC1 N1(C(c2ccc(C(=O)OC)cc2C)=O)CC2CN(C3CC3)CC2C1 C#CCC(C)(C(=O)NC1CCCCC1OC)NC(=O)Cc1ccc(C)o1 N1(C(CCNC(=O)OC)=O)CCC(NC(=O)CCC(C)c2ccccc2)C1C n1(CC(=O)NC(C(=O)OC)C2CC2)cc(CN2CCSCC2)nn1 C(CC(F)(F)F)N(C)C(c1conc1CNC(=O)CCc1ccnn1C)=O CCC(CCCC(=O)NC1CN(C(=O)C2CC2)C1)NC(C1CCC(=O)O1)=O c1(C(N2CCC(NC(C3(C=C)CC3)=O)C(O)C2)=O)cc2c(cn1)OCCO2 C1(CNC(CSC(C)C)=O)C(C)CCN1C(C1CCCN1C(N)=O)=O C1(OC)CCC2(C(=O)NCCC3CCCN3C(c3ncccc3Cl)=O)CC12 c1(C(=O)NC2CC(NC(C34CC(C)C3C4)=O)C2)cc(C(F)(F)F)ncn1 c1ccccc1C#N.C(C(O)CNC(=O)C)NC(C1(NC(C)C)CC1)=O.O C(=O)CS(=O)(=O)CCO.C1(C(=O)NCC(C)(C)OCC)CCCCS1(=O)=O C12(C(N3C4CC(NC(c5cc(C(C)(C)C)on5)=O)(C4)C3)=O)CCCCC1OCC2 C(=O)(N=c1nc(-c2cccnc2)[nH]s1)N1C(C)CCC1C C1(NC(c2cn(C)nc2)=O)CCN(C(c2nccc(F)c2Cl)=O)CC1F C(=O)(C1=CS(=O)CCC1)N1CCC(CCNC(c2c[nH]nc2-c2ccsc2)=O)C1 N1(C(C2CC(C)SCC2)=O)CCC(NC(c2cccc(CC#N)c2)=O)C(C)(C)C1 C1(C(=O)OC)CCC(CC(=O)NC2(C)CN(C(c3cnsn3)=O)C2)CC1 C=CCC(C)C(=O)NC1(C(=O)N(CCCOC)CCO)CC(O)C1 N1(C(c2n(CC=C)ccc2)=O)CCCC12CCN(C(c1cc(C)c(F)cn1)=O)C2 C1(C(=O)NCC(CC)NC(c2c(C)nc(CC)s2)=O)CC2(CCOC2)C1 N1(C(=O)CC2CCC3CC3C2)CCCC(C2CN(C(=O)CCCCF)C2)C1 CSC=CC(=O)N1CCC(CCNC(=O)C(CN(C)C)c2ccccc2)C1 C(=O)(C1CCc2nccn21)NCC(CNC(COc1c(C)ncnc1C)=O)C C1(CC(=O)NC2C(CNC(c3c(C#N)ccs3)=O)C2)CC2(CCC2)CO1 Cc1cc(CN2CC(C(=O)N=c3cc[nH]cc3)(C)C2)c(O)c(Br)c1 C1(CNC(c2cc(CC)n(C)n2)=O)CCN(C(=O)CCCCCOC)CC1C C(=O)(CCCCC(N)=O)N1C(C2(C(N(CCC3CN(C)C3)C)=O)CC2)CCC1 C=CC(CC)CC(=O)NC(CNC(c1ncoc1C(C)(C)C)=O)CCCC C(=O)(C1=CCCS1)N1C(CCNC(C2CCC23CCC3)=O)CCC1 c1(C(N2CCC(C(C)NC(CC(C)c3ccco3)=O)C2)=O)coc(C#N)c1 c1(N2C(C)CCN(C(CCNC(=O)NC)=O)CC2)ncc([N+](=O)[O-])c(C)n1 c1(C(=O)NC(C(C)NC(CCN(CCCCC)CC)=O)C)ccc(O)c(Cl)n1 c1(C(=O)NC(CCCNC(C(CC(C)C)O)=O)C)ccnc2ccc(O)cc12 c1(C=O)cc2ccc(Cl)c(F)c2o1.C1(C)(C(N(C)CCOCC)=O)CC1.N c1(CCC(N2CCCC(CNS(C)(=O)=O)C2)=O)ccc2ccccc2n1 C(C)(N=c1nc(N2CCC(C)(C)CC(C)(C)C2)c2c([nH]1)CSC2)c1n(CC)ncn1 C1(C(N2C(C(=O)NC(c3cscn3)CO)CC(OC)C2)=O)CC12CCCCC2 Cc1cccc(OCC(=O)NCC(C)NC(C2CCOC2C2CC2)=O)c1C CC1(CNC(c2cnco2)=O)CCCN(C(=O)CCN2CCNC(=O)C2)C1 c1(NC(C)C)cccc(C(=O)NC2CCC(N(C(=O)C(C)C)C)C2)c1 c1(N(CCOC)CC)ncnc2c1ncn2C1CC1.c1(C(=O)N)nnn(C)c1N N1(C(c2csnc2Cl)=O)CCC2(CC1)CC(NC(C13CC(F)C1C3)=O)CCO2 c1(C(=O)N)cccc(N=S(C)(C)=O)c1.c1(C(=O)NCCCC)nc(C)n(C)n1 N1(C(C=C(COC)C)=O)CC=CC1(C)C(=O)N(C1CCN(C2CC2)C1)C C1COCC(C)(C)C1.C(CC1CCC1)(C=O)NC(CN(C)C(=O)C1CC1)=O c1(C(NOCC(=O)NCC2N(CCC)CCC2)=O)ccc(C)n1C C(=O)(CC1=CCOCC1)N1C(CCC)CN(C(c2ccc(C)nc2NC)=O)CC1 N1(C(c2cc(C)oc2)=O)CCCC(C2CCCCN2C(=O)CC2CC(C)(C)C2)C1 C1(C(N2CC(F)(CNC(c3cc(O)nn3C)=O)C2)=O)(OC)CCC(C)C1 c1(C(C)NC(=O)Cc2ccc(F)cn2)ccc(C)cc1.C(=O)CC1CC1.N CCCC(CNC(C1CCCC2(CC2)C1)=O)C(=O)N(CCC(C)O)C C(CC(=O)N1CCOCC1C(N)=O)(C(F)F)NC(C1C(OCC)CC1)=O Cc1ccc(F)cc1C(N1CC(C(=O)NCC(C)(F)F)CC(C(F)(F)F)C1)=O C1CC2(CCC2O)C1.C(CC(=O)NCC1CC1CC=O)OCCOCC C12(CNC(CCSCC)=O)CC(CO1)N(C(c1nc(O)sc1C)=O)C2 c1(NCC(C)CN2CCCC2=O)nccc2c([N+](=O)[O-])cccc12 c1(C(N2CC(C)(C(=O)NCC3(C)C=CCCC3)C2)=O)cccc2[nH]ncc12 c1(C(=O)N)cc(F)c(F)cc1C.n1(CC)cc(CNC(C2CCCC2)=O)cn1 c1(C(=O)NCC2CCN(C(C=C(C)C)=O)C2)ccc(OCC(F)(F)F)cc1 Cc1c(Cl)ccc(C(=O)Nc2ccc(SC(F)F)nc2)c1N c1(C(C)C)c(C)cc(C(N2CCC(C3CCCN3C=O)C2)=O)cc1C.C(C)(C)C.O N1(CC)CCCCC1C(=O)NC(C(=O)N(CC(C)(CC)OC)C)C1CCCC1 C1(N(C)C(C2CC(O)CN2C(N)=O)=O)CC(N=c2[nH]nc(-c3ccccc3)s2)C1 Cc1nc2cc(C(=O)N(C3CC(NC(C4Cc5nnc(C)n5C4)=O)C3)C)[nH]c2s1 C1(NC(c2occ3c2CCC3)=O)CN(C(=O)C(O)Cc2ccccc2)CC12CC2 C1(CN(c2nccc(=NCC3CCCS3(=O)=O)[nH]2)C)COc2ccccc2O1 N1(C(c2c(C)cc[nH]2)=O)CC2CC(NC(=O)C(c3ccc(Br)cc3)O)C1C2 c1(C(=O)NCC2C3CN(C(c4nc(Cl)sc4Cl)=O)CC23)cnnc2ccccc12 C1(NC(CCC(C)O)=O)CN(C(c2c[nH]nc2C(C)(C)C)=O)Cc2nccn2C1 c1(C(N2CCC(O)(C(C)CNC(c3cc(Cl)cs3)=O)C2)=O)ccc(O)c(Cl)n1 N1(C(CSCCC)=O)CCC(N(C(c2oc(CO)cc2C)=O)CC2CC2)CC1 CC1(C)C(CC(N2C(CNC(C3(C)CSC3)=O)CC3CC23)=O)C1(C)C COn1cnc(C)c1C(N1CCOC(CNC(C2CCCCN2C)=O)C1)=O CCC(C)(C(=O)NCC(O)CC(=O)N1CC2(CC2C(=O)OC)C1)OC FCCN=C(NCC1COC1)NCC1CCN(C(N)=O)C1 C1(NC(C2CCC(CNC(C(COC)C)=O)O2)=O)CCOC(C)C1 c1(C(C(=O)NCCCF)N(C)CCn2cccn2)cc(Cl)cc(Cl)c1Br c1(C(=O)N)c(C)nsc1C.N1(C(C2C(OC(C)=O)C2)=O)CCCC1C1CC1 Cc1nn(C)cc1NC(C1(CNC(=O)Cc2ccc(F)cn2)CC1)=O C1(CC(=O)OC)CC(O)CN1C(c1cccc(NS(N)(=O)=O)n1)=O C1(N(C(=O)C=Cc2c[nH]nc2C)CC)CCCN(C(c2c(Cl)cnn2C)=O)CC1 c1(CC(=O)N(CCNC(=O)Cc2cccn2C)CC)ccc(Br)c(O)c1 N1(C(c2c(C)nc(C(C)C)s2)=O)CCC2(CCN(C(=O)C(C)(C)C#N)CC2)C1 C1(CC=O)CCOC1C(=O)NC1CCOC1CNc1ncccn1.C1CC1.N Cc1ccn(C)c1C(N1CCC(O)(CCNC(C2(C)CNC(=O)C2)=O)C1)=O C1(C(N2CCC(F)(CNC(c3ccc(C)nn3)=O)C2)=O)CC(F)(F)C1(F)F CC1CC(N(C)C(c2cc(CNC(=O)C=Cc3cnccn3)[nH]n2)=O)CCN1C CC(C)CC(C(=O)NC1CCCCC1NC(=O)CN1CCC(C)CC1)C(N)=O C1(N(C(C=C2CCC(C)C2)=O)C)CCCN(C(C2(c3ccc(F)cn3)CC2)=O)C1 N(C1CCCn2nccc21)C(C(C)NC(c1cc[nH]c(=N)n1)=O)=O C1(NC(C(C)(C)SC)=O)CC2CCC(C1)N2C(=O)CC1CCC(C)(C)O1 CCS(=O)(=O)CC(=O)N(C1CCCC(NC(=O)C(C)=C2CCC2)C1)C C1(C)(CCNC(C2CC(C)(C)C2)=O)CCN(C(c2ccc(CO)o2)=O)C1 N1(C(C(CCOC)C)=O)CC(CNC(=O)CC2CCCC2)C2(CC2)C1 c1(C(=O)N)cc(C)c(C)nn1.C1(OC)CN(C(c2ccc(C(C)C)nc2)=O)CC1 C1(O)(C(C)NC(COCC#C)=O)CCN(C(=O)CN(C2CCC2)C)CC1 c1(-c2cn(CC)c(=O)cc2)c[nH]c2ncc(C(=O)NCc3ccnc(C)c3)cc12 c1(OCC)cccc(F)c1CNCc1cnccc1C(=O)O c1(C(=O)NCCCN(C(=O)Cc2cn[nH]c2)C(C)C)ccnc(OC(F)F)c1 c1(OCC2CCN(C(Cc3cc(OC)ncn3)=O)CC2)cc(Cl)ccc1Cl N#Cc1ccc(C(N2CC3CC3(C(=O)Nc3ccc(CCF)cc3)C2)=O)s1 O=S1(=O)Cc2ccc(S(=O)(=O)Oc3ccc4c(Br)csc4c3)cc21 C1(C(=O)NC(CC)C(=O)NC)N(C(C2CN(C)CCO2)=O)CC12CCCC2 N1(C(C(C(C)C)NC(N)=O)=O)CC(C)OC(C)(C)C1.C(=O)(C1=CCCCC1)N Cc1cc(=NC2CCCC(NC(=O)Cc3cc(C(F)(F)F)n[nH]3)C2)c(C#N)c[nH]1 c1(C(=O)NC(C(CO)NC(CCSCC)=O)C)ccc2nc(Cl)nn2c1 N1(C(COC2CN(C(C3OCCN(C)C3)=O)C2)=O)CC2CCC1C(O)C2O Cc1nn(C)c(=O)c(C(N2CC(C)C(Nc3nccnc3F)C(C)C2)=O)c1C C=C(F)C1(CC(=O)NC(CNC(=O)CC(C)F)(CC)CC)CCC1 Cc1ccc(C(=O)NCCCNC(=O)C(C)CS(C)=O)cc1OC(F)F c1(C(N2C(CNC(C3(C=C)CCCC3)=O)CCC2)=O)cccn2cncc12 c1cc(C#N)ccc1C.c1(SC)nc(N2CC(O)CC2C(=O)N)cc(C(F)(F)F)n1 C1(CNC(c2ccc3c(c2)OCO3)=O)C2CCCC1N(C(=O)CC1CCSC1)C2 N1(C(Cc2c(C)nsc2)=O)CCCCC1C(=O)Nc1cnc(F)nc1 c1(OC)cc(C(=O)NC(c2cc(F)cc(Cl)c2)C)ncc1-c1cnc(F)c(C)c1 Cc1cc(CNC(=O)N(C)CC2CC=CCC2)ccn1 C(c1cccnc1)=CC(=O)NC(C)CCCNC(=O)CCC1CCC(=O)C1 c1(OCC)cc(OC)c(C(C(=O)NCC(F)F)N(c2cccc(OC)c2)C)cn1 Cc1c(Br)cc(C(=O)NC2CN(C(c3csc(Cl)n3)=O)CC2O)cc1Br N1(C(C2(C3CC3)CCCO2)=O)CC(CNc2ncnc(O)c2Br)C2(CCC2)C1 C1(CNC(C(CC)O)=O)CC2(CO1)CN(C(c1ccc(OC)nn1)=O)C2 N1(C(C=CC(C)C)=O)CC(N(C(=O)Cn2[nH]cnc2=N)C)C(C)(C)C1.CS Cc1c(Br)ccc(NC(C)CNC(=O)C(c2cccc(F)c2)C)c1[N+](=O)[O-] CC(O)CCCCCC(=O)N1CCC2CN(C(C3CC4CCC3CC4)=O)CCC12 C1(COC)CN(C(c2cn(CCO)nc2C)=O)CCN1C(=O)CCc1ncc[nH]1 c1(CN2CC(C(=O)NCCOCC#C)SCC2)c(C)cc(O)cc1C c1(CCC(=O)N(CCCNC(=O)C(C)c2cncs2)CC)ccnc(C)n1 C(=O)(C1=CCCSC1)N(C)CC1(NC(c2ccc(N3CCCC3)nn2)=O)CC1 CC1CC(C(=O)N2CCCC(N3CCN(C(=O)C(F)=CCCF)CC3)C2)=NO1 c1(CC)coc(C(N2CCCC2C2CC2)=O)c1.C(=O)CCN(C(CC)CC)C.N N1(C(CC(C)N(C)C(c2sccc2C#N)=O)=O)CCCC(C)CC1 C1(C(=O)NC(C2N(C(C3=C(C)CCC3)=O)CCC2)(C)C)CC2CCCC(C1)C2 C1(CC=C)(NC(c2cc(SC)c(C)o2)=O)CCCN(C(c2ccns2)=O)C1 c1(C(N2CCC(NC(CC(C)O)=O)C2C)=O)ccc(=O)n2c1CCC2 C1(C(=O)NCCSC(C)C)CCC2CCC1N2C(=O)CC1=CCCCC1 C1(CC)CC2CCC(C1)N2C(=O)C(C1CCCCC1)F.C1(CC=C)(C=O)CC1.N n1(C(CC)(C)C)nnnc1C(C1(CF)CC1)NCCCNC(N)=O C1(NC(Cc2c(C)non2)=O)CN(C(c2ccc(CF)cc2)=O)CC1C c1(NC(C2(C)CN(C(C3CC3(F)F)=O)C2)=O)ncccc1C(F)(F)F C1(CC)C(NC(=O)C=CC(C)(C)C)CCCN1C(c1nc(Cl)oc1C)=O c1(C(=O)NCC(CNC(C2CCCCS2)=O)OC)cc(C)cc2c[nH]nc12 c1(C(=O)NCC2CCCC(NC(C3(O)COC3)=O)C2)nccc2ccsc12 CCCCCCCCC(=O)NC1CCNCCC1CO c1(C(=O)NC(C2COCCO2)C)ccc2c(c1)OCCNC2=O C1(CCOC)CN(C(C2(F)CC2)=O)CCN1C(=O)C1=C(C)OCC1 C1(C(N2CC(NC(COC)=O)C2)=O)CN(C(=O)Cc2ccon2)CC1(F)F c1(C(=O)NCC(C(C)C)NC(c2cn(C3CCOC3)cn2)=O)cnc(S)n1C N1(C(C2CCCN(S(CC)(=O)=O)C2)=O)CCCC12CCCN(C(C1CSC1)=O)C2 C(C)(C)(CCCC(=O)NCC1(CCC)CC1)NC(C(C)OCCCC)=O C1(C(F)(F)F)(C(=O)OCC)CCCC1C.C1(=O)CN1 C#CCCCC(C)C(=O)NCC(C)(F)CNC(=O)C(C)=C1CC1 C(CC1c2ccccc2CCN1C(C1SCCS1)=O)NC(c1n(CC)ncc1)=O CCC(CC)C(F)C(=O)NCCc1n[nH]cc1C(=O)N(C)C(c1ccccn1)C N1(C(C(CC)C)=O)CCCC(C(=O)N(CC(c2ccccc2)O)C)C1 C(c1ccccc1C)=CC(N1C(C)CC(NC(CCCCC)=O)C1)=O Cc1nc(C(=O)NC2CC(NC(=O)C3=CCOC3)C2)nn1C c1(C(N(C)CC2C3CN(C(CCC)=O)CC32)=O)ccc2c(=O)cc[nH]c2c1 CCCCCC(C)CC(=O)N1CC2(CNC(=O)Cn3ccnc3C)CCC1CC2 C1(CNC(c2c(CC)c[nH]c2)=O)CCN(C(c2c(C)nn(CC)c2C)=O)CC1C C1(C(=O)NC2CC2CNC(C2CCCCNC2=O)=O)Cc2ccccc2C1 CCC(C)CCCC(=O)NCC1CC1CC(N1CCC1CC(C)C)=O C(=O)(C(=O)N)NCC.CC(C)C1CCC1.C(=O)CC.C(=O)C.C(C)=O O=C(C1=NN2CCCN=C2N1)NCC1CCOC1.c1(C(=O)N)cscc1C(F)F C=CCC(C(=O)N=c1cc2ccccn2[nH]1)NC(C1CC12CCCC2)=O CC1CN(C(=O)CCCF)CC2(CCN(C(c3c(F)cccc3Br)=O)C2)O1 N1(C(=O)OC(C)(C)C)CC(NCCCc2nccs2)C(C)(C)C1 N1(Cc2c(C(=O)OC)csc2)CCC2CCN(C(=O)CS)CC2C1.CC(F)(F)F C=CC(C)(C)CC(=O)NC(c1ccccc1)CNC(=O)C(C)CC(F)F c1(C(=O)NC2CC(NC(C3C(=C)C3)=O)C2)cc(C#N)c(O)nc1N C#CCN(OC)C(=O)CC12CCC1CN(C(=O)CN(C)C(=O)C1CC1)C2 N(C(=NCc1cc(N(C)C)ccn1)NCC1COC(=O)O1)C(COC)C c1(N2CCOCC(CNC(CSC)=O)C2)nc(-c2ccccn2)nc(C)c1C C1(C)(C(=O)NCCC2CN(C(c3n(C)nc(O)c3)=O)C2)C2Cc3ccccc3C12 C1(C)(C=O)CCS(=O)(=O)CC1.c1(CC)c(C(=O)NC)nn[nH]1.C1CCC1 C(CSC)(C(=O)NC(C)CNC(=O)CC1CCCOC1)OC c1(C(N2CC(C3(NC(C4=C(C)OCC4)=O)CC3)C2)=O)cc(=O)n2ccccc2n1 O=S(=O)(c1ccc(NC2CCCSCC2)c(Cl)c1)NCC#Cc1cccnc1 c1(C2(CNC(C3CCC(OC)C3)=O)CCC2)ccc(C)cc1 c1(C=O)cc2cccnc2[nH]1.c1(CNC(C)=O)ccc(C(=O)NCC(F)C)s1 c1(C(=O)Nc2nnc(CC)s2)ccc2oc3ccccc3c2c1 CCCC(C(=O)N1CC(=O)CC1C(=O)NC1CCCC(C2CC2)C1)C(C)C C(=O)(CCCC(=O)NCC#CCNC(c1ccccn1)=O)c1cccc(OC)c1 c1(C(N(CCC(=O)N(CC(CC)O)CC)CC)=O)cc(CO)oc1C N1(C(C(CNC(CCCOC)=O)OC)=O)CCC([N+](=O)[O-])CC1 N1(C(C(=O)O)=O)CCCC(C)C1.C(CC(C)NC(C)=O)N(C(=O)C)CC CS(=O)(=O)CCCC(=O)N1CCCCCC(NC(C2C(F)(F)C23CC3)=O)C1 c1(C(=O)NCCCN(C(COCCC#C)=O)C)ccn(C(C)C)c1C C1(NC(c2ccc(C(=O)NC)cc2)=O)CCCN(C(c2sccc2OC)=O)CC1 N1(C(c2ccc(C(C)C)o2)=O)CCC2(CC1)CC2C(=O)NC1CCC2(CCC2)C1 C1(O)(C(=O)OC)CN(C(c2cc(F)ccc2F)C(=O)NC(C)(C)C)CCC1O c1(C(=O)NC23C(CN(C(CSCCC)=O)C2)CCC3)c(F)ccc2ccncc12 c1(C(=O)NC(C(N2CCC(CCO)C2)=O)C2CCCO2)cccc2c[nH]nc12 C1(CC)C(C(=O)NCCC(C)c2cn[nH]c2)CCN1C(c1n[nH]c(O)n1)=O C1(C(=O)NCC2(OC)CN(C(CCCCCCC)=O)C2)CCn2c(C)nnc2C1 C1(C(=O)NC(CC(N2C(C=C)CCC2)=O)COC)CCOC(=O)CC1 C(C)(C(=O)N1CCC(N(C(=O)Cc2sc(C)cc2C)CC)C1)C(C)C.CC=O CCCCCC(O)CC(=O)N1CCC1CNC(=O)COC1(C)CCC1 Cn1ncc([N+](=O)[O-])c1NCC1C2CN(C(c3cccc(C4CC4)c3)=O)CC12 C1(OC)CCC2(C(=O)NCC3CCOC3C(=O)N)CC12.C1CC2CC2C1 C(=O)(CC(C(F)F)NC(c1[nH]ccc1CC)=O)NCC1(C#C)CCC1 CC1(CNC(C2(CNC(C3CCO3)=O)CCCCC2)=O)CC2CCC1C2 c1(C(N(CCC(=O)NC(CC)Cn2cncn2)CCO)=O)cn(C)nc1OC N(C(=NCCCCC(F)(F)F)NCC1CC1(F)F)C1CCN(C(=O)OCC)C1 C(=O)(C(C)CC(C)C(C)=O)N(C(CCNC(c1c(CC)occ1C)=O)C)C C(=O)(C1COc2ccc(F)cc21)NC1C(C)N(C(C2CC(F)(CO)C2)=O)CCC1 N1(C(CSC(C)C)=O)CC(NC(C2CCN(c3ccccc3)C2)=O)C(N=[N+]=[N-])C1 C1(C(N2CCN(C(c3c(C)snc3)=O)CC2C(C)C)=O)CCc2n[nH]cc2C1C C1(C(=O)NCC2(CCC)CC2)CSCCN1C(=O)Cn1cc(C)cn1 CC1=NOC(CC(=O)NCCC2CN(C(=O)CN3CCCCC3)C2)C1 N1(C(Cc2cn(CC)nc2)=O)CCC(C(F)F)(CNC(=O)C(C)SC)C1 N#Cc1cnc(NC2CC(NC(c3ccn(C4CC4)n3)=O)C23CCC3)c(Br)c1 c1(OC)ccccc1CNC(=O)C(C)CNC(=O)C=CC1CCOCC1 C=CCCCCC(=O)Nc1cccc(CNC(=O)C(C2CCOCC2)F)c1 c1(C(N(CCNC(C2CC2C2CCC2)=O)C2CC2)=O)cc2cc(F)ccc2s1 C(C1CC1)(C1CC1)=CC(=O)NC1CC1NC(=O)C(O)C1CC1 C1(F)(CNC(CCCC=C)=O)CCN(C(c2ccc(CC)cc2F)=O)CC1 C1(NC(=O)Cc2ccc(Br)cc2)CC2(CCN(C(C34CC(F)(C3)C4)=O)C2)C1 N1(C(c2ccn(C)c2)=O)CCC2CCN(C(c3cc(F)cc(Br)c3)=O)CC12 c1(C(N2CCC(CNC(C(C)(C)OCC)=O)CC2)=O)c(C)nn(CC)c1C C1(C(=O)NC(c2ccsc2)C)CC2CCC1N2C(=O)CC(=O)NC1CC1 CCCC(O)CN(C(=O)CC1CCCN1C(=O)C=C(C)C)C c1(OC)cccc(O)c1.C1(N(C(C2C(C=O)C2)=O)C(C)C)CCCCCCC1.N CCC(CC(=O)NC1CCCCCC1C(=O)NCC1(C)CCN(C)C1)C(C)C C1(CCC(=O)NCCCN(C(C)C)C)CCCN(C(C2CCOC2C2CC2)=O)C1 C(=O)(C(C)(C)S(=O)(=O)C1CC1)N1CCCC(C)(C)C1.CS(=O)CCC(=O)N.C c1(C(=O)NC(CC)(CNC(=O)C(CCO)N(C)C)CC)cnc(CO)nc1C c1(C(=O)NCCC2CCN(C(C(C)CN(C)C)=O)C2)ccc(Cl)c(Cl)c1N C(=O)(CC(C=C)CCC)N1CC(C#C)(C(=O)N(CCCC)CCOC)C1 c1(C(N2C(CNC(C(C)C(F)F)=O)CN(C)CC2)=O)csc2c1CCCC2 c1(C(=O)NC(COC)C(=O)NC2CCOCC2C)ccc(C)n1C C(=O)(C(F)CC1CCOC1)NC1(CCCNC(=O)CCC2CC2(F)F)CC1 C(=O)(CCCCC#N)N1C(CNC(C(CC)Cc2ccccc2)=O)C2CC2C1 N1(C(CCOC)=O)CCN(C(C2C(c3n[nH]c(C)n3)C2(C)C)=O)CC1C(F)F C(=O)(CCCC(F)(F)F)N(C(CNC(C(C(C)C)F)=O)C1CC1)C C(=O)(C1=CCCN(C(C2(C(=O)N(C)C)CC2)=O)C1)NC(c1ncc(C)o1)C C(=O)(C(O)C1=CCCCC1)NCC1CCCN(C(c2cnn(C)c2N)=O)C1 c1(C(N(C)CC2C3CN(C(COC(C)=O)=O)CC32)=O)cc2n(n1)CCCO2 Cc1cc(C(N2CC3(C2)SCCC3NC(=O)CC2CC2)=O)c(Cl)cc1N CC(N=c1[nH]c2ccccc2s1)C(C)(C)CNC(c1ccco1)C c1(C(=O)NCC2CCC(NC(C(C)NC(N)=O)=O)C2)ccnc(Br)c1N C1(C(=O)NCc2cncc(C)c2)CCC2(CC2)N1C(=O)CC1CCC(=O)CC1 Clc1ccc(-c2ccc(-c3nccn3Cc3ccc(OCC(F)F)cc3)s2)cc1 C(=O)(C(O)C1=CCCCC1)N1CC(C)CC(C(=O)NC2CN(C(C)C)CC2C)C1 N1(CC(=O)N(CCCC)C2CC2)CCN(C(c2ccncn2)=O)CC1 C1(CCCNC(c2n(CCN(C)C)ncc2)=O)CCN(C(C2CCCO2)=O)CC1 Cc1cc(F)cc(C(=O)NC2CC(NC(=O)C)C2)c1C.c1nnnn1C1CC1 CC(C)CCCNC(C1CC1c1ccccn1)=O.C1(C)(C(=O)N)CC(C#N)C1 C(=O)(C(O)CCC(F)(F)F)N1CC(CNC(C(C)C(F)F)=O)C(F)(F)CC1 O=C(C1=CCN(C(c2ccncc2Cl)=O)CC1)NC1CCC=CCCC1 C1(NCc2cn(CC(CC)O)nn2)CCN(C(=O)COC(C)(C)C)CC1 CN1CCn2nc(C(=O)NCCc3cnn[nH]3)cc2S1(=O)=O N1(C(c2c(C)nc(CCC)s2)=O)C2CCC1CC(CNC(C1CCC=CO1)=O)C2 c1(C(=O)OC)ccc(NC(C2CC(C)CN2Cc2ccccn2)=O)c(I)c1.O C1(N(C(CSc2nnc(C)s2)=O)C)CN(C(C2(C)CCCO2)=O)CC1(C)C c1(C(N2C(C)CC(CNC(CCC=CC)=O)C2)=O)ccc2c(c1)C(=O)CCS2 N1(C(c2ccc(C)s2)=O)C2CCC1C(C)C(NC(c1cn[nH]c1)=O)C2 C1(Nc2c(C)c(Cl)ncn2)CCC2CN(C(=O)CCc3cnccn3)CC2C1 c1(C(N2C(C(C)(C)NC(c3cnc(CC)s3)=O)CCC2)=O)nccc(OC)c1N c1(SCC(=O)NCCC(=C)CNC(c2nonc2)=O)cc(Cl)ccc1Cl.C C1(CCNC(c2c(C)con2)=O)CCN(C(=O)C(O)c2cnc[nH]2)CCC1(F)F N(C(=NCCCCl)NCC(=O)NC)CC(C1CCOCC1)OCC C(CC(F)(F)Cl)NC(C1CCCN1C(=O)CCCC1CCCO1)=O c1(SC)nc(Nc2cccnc2C(=O)Nc2nc3c(s2)CCC3)cc(C)n1 N1(C(C2C(CNC(C3C(C)(C)COC3)=O)CCO2)=O)CCc2ncncc2C1 C(C(F)(C(=O)N(OC)C(C)CC)C(C)C)NC(COCC(=O)NC)=O c1(OC)cc(O)c(CN2CC(F)(F)CC2C(=O)NC(C)CCO)cc1Br O=C(C1CCc2cc(Br)ccc21)NCc1cn(CC(F)(F)F)nn1 Cc1c(-n2cc(-c3cccc(COC(C)(C)C)n3)nn2)cccc1C1CC1 c1(C(=O)NCC2C(C(=O)NC(c3cccs3)CC)OCC2)c(C)csc1C [N-]=[N+]=Nc1ccccc1NC(=O)C(O)C1CN(C(C2CC2C2CCC2)=O)C1 C(=O)(CCC(CC)CC)N1CCC(C)(CCNC(C(CCC)F)=O)C1 C1(C(N2CC=CCC2)=O)C2C3CC4C1C1C2CC3C41.C(C)(C(=O)N)NC(C)=O c1(C(C)C(=O)NCC2CC2NC(=O)CSC2CC2)ccnn1C c1(NC(C2CN(C(c3cncc(OC)c3)=O)CC2(F)F)=O)ccc2c(c1)OCO2 c1(CN2CCN(C(c3c(CC)ncs3)=O)CC2)c[nH]c2cc(F)ccc12 Cc1ccc(S(=O)(=O)N2CCN(C(c3c(Br)ccnc3Cl)=O)CC2C#N)cc1C N1(C(C2(C)CC3CCC2C3)=O)CC2CCCC(C1)N2CCn1cccn1 N1(C(C2CCCC(C)C2)=O)CCC(C)N(C(=O)CC2CC2(C)C)CC1 C(=O)(C(C)(C)CC(=O)N1CCC(CN(C)C(c2cc(Cl)cs2)=O)CC1)OC c1(NC(C)=O)ccccc1NC(c1cc(C)on1)=O.C12CC3CC3N1C2=O C(=O)(C(C)CC(C)(F)F)NCCc1c(OC)cccc1.C1(C=O)CNC(=O)N1 c1(CCCCC(=O)NCC(C)NC(c2cnc(SC)[nH]2)=O)ccc(Cl)c(Cl)c1 C1(CNC(C(C)c2cc[nH]n2)=O)CCN(C(=O)CCC2(C)CC2)C12CCC2 C1(C(N(C(C)CCNC(C2(CF)CC2)=O)C)=O)CCc2ccccc2O1 Cc1cc2ccccc2nc1C(=O)NC1CN(C(=O)CS(=O)(=O)N(C)C)C1 c1(COC)nc(C(=O)N(CCCN(C)C(C2CC2(C)C(C)C)=O)C)co1 CCC(CN(C)C)CC(=O)N1CCC(O)C1C(N1CC(c2nc(=O)o[nH]2)C1)=O C#Cc1cccc(C(N2CCC(CC=C)(C(=O)NC3CCC(CO)CC3)C2)=O)c1 C1(C(N2CCN(C(c3c(C)sc(O)n3)=O)C(CCO)C2)=O)CCc2c[nH]nc2C1 CC1(C)CCC1CNC(=O)C.c1ccccc1.C1(CC=O)CCC(=O)N1.N Cc1cc(Br)ccc1OCC(=O)NC1CN(C(c2n[nH]cc2F)=O)C1 C=CCC(C)C(=O)N1CCC(O)(CN(C(=O)CC(C2CCC2)C2CCC2)C)C1 N1(CCO)CCc2cc(-c3ccc(N4CCCCCC4)cc3)ccc21.C1CC1 C1(CN(C(=O)Cc2cscn2)C)CN(C(c2cccc(CO)n2)=O)CCO1 CCCC(C(=O)N(CCC(C)(C)O)C)NC(=O)C=Cc1ccc(C)o1 C1(C(N(CCN(CC)C)C)=O)CC2CN(C(C3CCCC(C#N)C3)=O)CC2C1 C1(OC(Cc2n(C)cnc2)=O)CCC(C)(C)CC1 Cc1c(-n2cc(-c3cscc3Br)nn2)ccc(Br)c1C#N N1(C(Cc2c(C)cco2)=O)CCC(O)(CNC(C2CCC3CC23)=O)CC1 C(C)(C(C)C(C)C)NC(c1cn(CC=C)nn1)=O.c1(C(=O)N)ncc(F)cn1 N1(C(c2cc(C)oc2)=O)CCC(O)C1C(=O)NCC1C2CCCC12 c1(CC(N2CCC(COC)(NC(=O)C(C)CF)CC2)=O)ccc2nc(O)[nH]c2c1 CN1CC2CN(C(=O)C(O)CCCNC(=O)CSc3nc[nH]n3)CC2(C)C1 c1(SC)cn(C)nc1C(=O)NC(C)C(C)NC(=O)CSc1ccncc1 C(C(C(=O)N1CC(N2CCOC2=O)C1)C(C)C)NC(CC1C(C)CC1)=O n1(CC(=O)N(CC(C)NC(C(CC#C)(C)C)=O)C)cc([N+](=O)[O-])c(C)n1 C1(C(=O)NC2CC2NC(=O)C(Cl)=CCl)(OC)CCSC1 N1(C(C(N2CC(C)C2)C)=O)CC=C(C(C)(C)C(=O)NCC2CCC2(F)F)C1 c1(C(=O)NCC2CN(Cc3cccc(OC)n3)C2)ccnc2ncccc12 N1(C(c2cccc(OC)c2OC)=O)CC(NC(=O)C2=CCCS2)CC(C)(C)C1 N1(C(c2cnsn2)=O)CC2C(CNC(=O)C(C3CCCO3)C3CCCC3)C2C1 C(CC(C)(C)C)(C(=O)N1CC=CC(C(=O)NC(c2ccccc2)C)C1)OC C1(C(N2CC(O)(CCNC(C3CC3C3CCCC3)=O)C2)=O)CCN2CCOCC12 c1(CC=O)ccc2sccc2c1.Cc1ccn(C(C)C(=O)NC23CC(C2)C3)n1.N C1(C(N2CC(CC(=O)OC)C2)=O)CC(NC(=O)C(C)(Cl)Cl)CCO1 C1(COC)(NC(=O)C(C)O)CCN(C(c2cc(C)c(C)nn2)=O)CC1 N1(C(C(C)n2cccn2)=O)CCC(n2cc(C(C)(O)C(=O)O)nn2)CC1 C(=O)(C1CCCc2nccn21)NC(C)CCNC(=O)Cc1cccc([N+](=O)[O-])c1 C(C)(C)(CC(=O)N1CCC1(C)CCO)N(C(C1C(C)=CCS1)=O)C N1(C(N(CC(C)(C)O)CC)=O)CCC(OCc2ccccc2)C1 N1(C(CC(C)(C)C)=O)CCCC(NC(c2c(C(F)(F)F)cc[nH]c2=N)=O)CC1 C(=O)(C(F)(F)C(F)(F)OC(F)(F)F)NC(C)CCN(C)C(C1CC1F)=O C1(NC(C=C(COC)C)=O)CN(C(=O)C(c2ccc(Br)cc2)O)CC1F Cc1ccc(CNC(C2CCC2CNC(=O)CC2CCCC23CC3)=O)cn1 c1(OC)ccc(C(=O)NC(CNC(c2nn[nH]c2Cl)=O)C(C)C(C)C)cc1.O C1(NC(CC(C)CNC(C2(n3nccn3)CC2)=O)=O)COCCN(C)C1 C1(C(N(C)CC)=O)CC(C)N1C(=O)C=C(C)COC.C1(C)CC1 Cc1ncsc1CC(=O)NC(C)C.C(=O)CC1CCCC1.C(C)(C)(C)C=O N1(C(C(C)C2CCC2)=O)CCN(C(=O)CNC(=O)CC(C)(C)C)CC1C C=CCC(CNC(=O)CC1COC(=O)C1)C(=O)N1CCC(OCC(C)C)C1 C(=O)(N1CCCO1)C1CC(=C)C1.n1(C2(O)CC2)cc(Cl)cn1 CC1CCCc2cc(C(N3CCC(C(C)(C)NC(c4ccnn4C)=O)C3)=O)nn21 Cc1c(Cl)c(C(=O)NC(C)(C)CN(C(=O)CCC(N)=O)C)nn1C N1(Cc2cccc(S(N)(=O)=O)c2)CCC(S(=O)(=O)C(F)F)CC1 N1(C(Cc2c(C)ocn2)=O)CCN(C(c2cccc(F)c2)COC(F)F)CC1C C1(O)(C(N2CCC(COC)C2)=O)CCCCCC1.c1(C=O)cc(C(F)F)cs1.N c1(CCC(=O)NCCCN(C(CC2C(C)(C)C2)=O)C2CC2)ccccc1F C#CC1(C(=O)NCc2ccc(CNC(=O)CC)cc2)CCCCC1.C1CCC1 C(C(C)(C)C#CC(=O)N1CC(N(C)C)C1)NC(C1CC(C)C(=O)CC1)=O N1(C(C2C(C)N(C(=O)C3=C(Cl)CCCC3)CC2)=O)C2C=CCC1CCC2 C1(C=O)CCCC(C(N)=O)C1.N1(CC)CCCC1C(=O)NC1(C)CCC1.N C1(n2cc(COCCN(C)C)nn2)CCCN(C(CCCCC2CCCC2)=O)C1 C(N=c1cc(Cl)nc(C2CC2)[nH]1)C1C(NC(c2nnn(C(C)(C)C)n2)=O)CCCC1 c1(OC)cncnc1NC1CN(C(=O)CCNS(C)(=O)=O)CC1C c1(NC(=O)NC(c2ccccc2Cl)C(C)C)cn(C)nc1C(F)(F)F Cc1cccc(C)c1-n1nc(CCC(C)C)nc1C1CCN(C)C1C c1(CC)cc(CC(=O)NC23CC(C(=O)NCC[Si](C)(C)C)(C2)C3)on1 C1(NC(C(C)SCCCC)=O)CN(C(=O)CC(C)(C)O)CC1c1cnn(C)c1 n1(CC)nnc(CNC(=O)C(c2cccs2)NC(C2CC(C)C2)=O)n1 C(=O)(C#CC(C)(C)O)N1C(C(=O)NCC#CCC)C(C)CC1 CC(C)CC(O)CC(=O)NCc1nocc1C(=O)NCC1CC1(C)C C(C(C)CC(=O)NC1CCN(C(=O)CCC2(C#N)CCC2)CC1)OC.C1CC1.C C(CCC(C)NC(=O)C(n1cc(Cl)cn1)C)NC(C1(SC)CC1)=O CC(C)(O)C(C)(C)NC(C1CCOC1C)=O.C1(C=O)CN(C(N)=O)C1.N C12(C(N(C)CC3(O)CCN(C(c4c(C)nn(C)c4)=O)C3)=O)CCCC1CCC2 CCC(C)(C)C(=O)C(=O)NCC1CCN(C(=O)CCCN(C)C)CC1C C1(CCC)CC(C(=O)NC(C)CN(C)C(c2coc(C)c2)=O)CCO1 c1(CC(=O)NC2(CCCC)CC2)cn(C2CC2)cn1.c1(CC(=O)N)nc[nH]n1 c1(CC)ccccc1OCC(=O)N(CC(O)CNC(=O)CN1CCCC1=O)C C=C(C(=O)N1CC(NC(c2c(I)ccnc2F)=O)CC(C(F)(F)F)C1)C(F)(F)F c1(CN=c2scc(C(N3CCC(C#N)C3)=O)[nH]2)cccc([N+](=O)[O-])c1Cl c1(C(=O)OC)ccc(C(=O)NC2(C(=O)OC)CCCC3CC23)c(F)c1 c1(C(N2CC(OC)CC2C)=O)csc(S(C)(=O)=O)c1.C(=O)CCC1CC1.C C1(NC(C2(COC)CCC2)=O)CN(C(=O)CC2(O)CCCOC2)CC12CC2 CCC(CC)(C(=O)NCC(CC(=O)N1CCN(C(C)(C)C)CC1)C1CCC1)OC CCCC(C(=O)NCc1cc(C(N2C(CO)CC2C)=O)ccn1)C(C)C Cc1cc(C(N2CCN(C(c3cncn3C3CC3)=O)CC(O)C2)=O)c(Cl)cc1F C1(CN(CCNC(=O)CCCn2nnc(-c3ccccc3)n2)CC)CCCOC1 CCCCC(CO)NC(C1CC12CN(Cc1cc(Br)c(C)s1)C2)=O C(=O)(C(O)CC(N)=O)N(CCNC(=O)C=Cc1cscn1)CC C1(NC(=O)CCc2cn[nH]c2)CCN(C(C2CCCCC2F)=O)CC1 c1(C(N2CCCC(CCNC(=O)C=CC3CCC3)C2)=O)cc([N+](=O)[O-])c[nH]1 c1(-c2n(CCCOC)c(N3CC(OC)CC(O)C3)nn2)cc(C)c(C)c(Br)c1 N1(CCCC)CCN(C(C2CCCC2CNC(=O)CCCCC2CC2)=O)CC1 c1(C(=O)NCCCN(C(CSCCC)=O)CC)ccc(C)o1.c1ccccc1 n1(CC(N2CCCCC(N(C(CN(C)CC)=O)C)C2)=O)ccc2ccc(F)cc12 C1(C(N(C2CC(C(=O)OC)C2)C)=O)(CF)CCN(C(=O)CCCCC2CC2)C1 N(C1COc2ccccc21)C(C(CC(=C)Cl)NC(c1ccnnc1)=O)=O c1(C(=O)NCC(CNC(CC(n2ccc(C)n2)C)=O)O)noc2c1CCCC2 Cc1cc(C(N2CC(C(=O)N)CC(F)C2)=O)cc(C)c1C(=O)O.C(C)C(N)=O Cc1ccc(N2CCCC(C(c3ccc(Br)cc3)O)C2)nn1 c1(CNCC23C(CN(c4c(Br)cnc(CC)n4)C2)C3)c[nH]c2cccc(C)c12 N1(C(c2c(C)ccs2)=O)CCN(Cc2c(I)ccnc2Cl)C2CC12 c1(CNC(N(CCOC)Cc2ccccc2)=O)ccc(C)cc1OC c1(NC(C(N2CCC(CCC(=O)OC)C2)c2ccsc2Br)=O)ccccc1C N1(C(CC)=O)CC2(CCCO2)C1.C(c1ccc(F)cc1)=CC=O.C(CO)OC C=CCN=c1[nH]cc(C(N2CCN(CCNC(=O)CC3CCC3(C)C)CC2)=O)s1 C1(C(N(CC(C)O)C)=O)C2CC3C(C2)C13.c1(C=O)cc(=O)n(C)cn1.CO N1(CC(=O)NCC(CC)NC(c2csc(CC(F)(F)F)n2)=O)CCCCC1=O C(=O)(CC(O)CC(C)(C)C)N1CC(C(=O)N(CCCCN(C)C)C)(CC)C1 C1(C(N(CCC(C)NC(CNC(CC)=O)=O)C)=O)CC(=O)CCO1 CC1CN(C(=O)C(C)(C)NC(=O)C(F)(F)F)CCCN1C(=O)CC1=CCCCC1 C1(NC(CC(C(C)C)O)=O)CN(C(C2CCCO2)=O)C2(CCC2)C1 c1(CC(=O)NC2CC(C(C)NC(C3CC3(F)Cl)=O)C2)ccc(CO)cc1 N1(C(C(C)c2cccs2)=O)CCC2C(CCN2C(=O)C(C)(C)C(N)=O)C1 Cc1ncc(C=CC(=O)NC2CCCC23CN(C(c2ns[nH]c2=O)=O)C3)c(O)n1 C1(C(=O)NC(C#C)(C)C2CC2)CCCN(C(=O)C(CO)OC)C1 CC1CCCC(C)CN1C(C1CC12CCN(C(c1cc(C(N)=O)c[nH]1)=O)C2)=O C(C(C)(C)C(=O)N1CC(C(C)C)C1C(C)C)N(C(CCc1onc(C)n1)=O)C c1(CCNC(N2CCC(C)(c3onc(C)n3)CC2)=O)c[nH]c2ncc(F)cc12 c1(CNC(=O)CCC2CCCC(=O)N2)ccc(Cl)c(I)c1 N1(C(C=CCN(C)CC)=O)CC2(CCN(C(C3CSC3)=O)C2)C1 Cc1ncncc1C(=O)NC(C)(C)CN(C(=O)COCC(C)(C)C)C c1(C(N(C2CCN(C(=O)C(C)CC(F)F)CC2)CCOC)=O)cccc(N)c1F CC1(C)CC(NC(C2CCC2(F)F)=O)CN(C(c2cn3ccnc3cn2)=O)C1 c1(OC)nccc(C(=O)NCCCCCN(C)C(C2(S(C)(=O)=O)CC2)=O)n1 C1(CNCCS(N)(=O)=O)CC2(CCN(CC(=O)N)CC2)CO1.c1ccc(Br)cc1 C=CCCC(F)(F)C(=O)N1CCN(C(=O)CNc2ncccn2)C(CCOC)C1 c1(CCCC)cc(C(SC2=NCCS2)=O)n2ncnc2n1 c1(C(N2CC3CC(NC(C4CCCC4O)=O)C3C2)=O)ccn2ccnc2n1 c1(C(=O)NC2(C)CCN(C(C3CCCS3(=O)=O)=O)C2)cccc2nc(O)[nH]c12 C(=O)(CCCC(=O)NC1CCCCN1C(C)=O)NC1C(NC(C#C)=O)COCC1 N1(C(C2(COC)CC2)=O)CCN(c2ncnc3sccc23)CC(O)C1 N1(C(=O)Cc2ccccn2)CCN(CCn2cc(Cc3ccno3)nn2)CC1 c1(CCCC(=O)NCC2CN(C(C3SC4C=CC3CC4)=O)C2)c(F)cccc1F c1(NC(=O)Cc2cccc(Br)c2)cnc(F)cc1C(N1CCCCC1CO)=O CC1(C)CCOC(CC(N2CCC(NC(=O)Cc3cnsc3)C2)=O)C1 CC1(C)CS(=O)CCN1C(=O)C(N1CCSC(C(F)(F)F)C1)=O c1(CN2CC(N3CCN(C(=O)Cc4ccccc4)CC3)C2)cc(Br)ccc1F Nc1cc2c(cc1C(N1CCC(NC(=O)Cc3ccccc3F)C1)=O)OCO2 N1(C(=O)NCCC(C(CC)CC)N2CCOCC2)CC2CCCS(=O)(=O)C2C1 c1(C(N2CC(OC)(CNC(C3(CO)CC3)=O)C2)=O)csc2c1CCC(C)C2 c1(C(=O)NCC(CN(C)C(c2cnccc2Cl)=O)O)cc(-n2cccn2)ccn1 C1(Cn2ncc(C)c2)CCCN(C(c2csc(CC3CC3)n2)=O)C1 N1(CC23CC(OC)(C2)C3)CCCCC1.c1(CC(=O)C)cccc(C(C)=O)c1 C(=O)(C(=O)CCCOC(=O)CCc1nc(-c2cccnc2)no1)OC C=CC(C)(C)CC(=O)N1CCCC(C)(NC(=O)CCC(C)OC)C1 Cc1cc(Cl)c(C(N2CCCC(C)(NC(=O)C(F)=CCCF)C2)=O)cn1 C1(CCNC(c2nc(C)[nH]n2)=O)CCCN(C(=O)C(c2ccc(F)cc2)F)C1 Cn1cnc2cc(C(=O)NC3CC4(C3)CC4NC(c3cscn3)=O)cnc12 Cc1ncn(C)c1C(=O)NC1(CNC(=O)C(c2cccnc2)O)CCOCC1 C1(COC)(NC(=O)Cn2nnnc2C)CCCN(C(=O)CNC(C)=O)C1 N1(C(C(CCC2CCC2)NC(=O)CC2(O)CCC2)=O)CCC2C(O)CC12 CC1CCC(C(=O)NC2(C)CCCC2)S1.c1(CCC=CC(=O)N)ccccc1 c1(C(=O)NC2CCCCN(C(CCCOCC=C)=O)C2)csc2c1CCCC2 N1(C(C(=O)Nc2ccc(-n3cccn3)c(Cl)c2)=O)CC(S)CC12CCC2 C(=O)(C(=O)N=S(C)(C)=O)N1CCC(NC(C=CCN(C)CC)=O)(C)C1 N1(C(c2c(C(C)C)ccs2)=O)CCOC2CCN(C(=O)C3CC3)CC12 Cc1cnc(Br)cc1NC(C1CCCC(NC(=O)Cc2ccc(Br)cc2Br)C1)=O C(=O)(C1=CCN(C(=O)CC2CCCSC2)C1)NC1(C(N)=O)CCOCC1 CC1=C(F)CN(C(C2OCCC2CNC(c2ccncn2)=O)=O)CC1 N1(C(CCC=CC(C)C)=O)CCN(C(=O)CN2CCCCCC2)C2CC12 c1(C(=O)NCC(N2CCCC(C)C2)=O)n[nH]c2c1COC2 N1(C(C2C(CNC(C(C(C(C)C)OC)O)=O)CCC2)=O)CCc2cnccc2C1 C1(NC(C=CC=CC)=O)CN(C(c2ccns2)=O)CCC1C(F)(F)F C(=O)(C(O)CCCNC(=O)CCC(C)=O)NCC1C(C(=O)OC)C1 S(=O)(=O)(CC(=O)NC1CCN(C(=O)CC(O)Cc2ccccc2)C1C)NCC C(=O)(CCC1=NNC(=O)CC1)NCC(C)(C1CC1)NC(=O)CNC=O C1(C(=O)NC2C(NC(c3c(OC)n(C)nc3)=O)CCC2)CCc2nnc(O)n2C1 c1(CC(=O)NCCNC(C2CCO2)=O)cc(C(F)(F)F)cc(F)c1 C1(O)CCC1.C(C(C)(C)C)C(C1CCC1)=O.C1(C(NC)=O)CC1CC.C N1(C(c2scc(OC)c2)=O)CC(C)CCC1CNC(C1(CSC)CC1)=O CCCCC(=O)C(=O)N1CC=CC1(C)C(=O)NC(c1cccnc1)C O=C(C1=CCC2CCC1N2C(c1cnns1)=O)N1CC(N2CC(O)C2)C1 N1(C(C2N(C(C(C=C)CC)=O)CCSC2)=O)CCC(F)(F)C(C)C1 C1(C(N(CCC(=O)NC)C)=O)CCN(C(=O)C2=CCCSC2)O1 C1(CCOC)(NC(C2(CC(C)C)CC2)=O)CCN(C(=O)CCCC2CC2)C1 C1(NC(C2(CC)CCCC2)=O)CS(=O)(=O)CC1.c1(C=O)cccc(C)c1N.N C(N=c1nc(N2CC3CC2CC3O)c2ncccc2[nH]1)c1ccc(C)cc1F c1(C(N2CCC(CCNC(C(n3c(C)ccn3)C)=O)CC2)=O)cc(O)ccc1Cl CC(C)(CCNC(c1cnco1)=O)C(=O)NOCCCC(F)(F)F C(=O)C1=C(C#N)CCC1.c1(CC)cc(C(=O)NC2CCC(CC)C2)c(C)o1.N c1(C(=O)NCC(CNC(C(C)(C)OC)=O)C)cnc(Cl)c(F)c1N C1(CNC(c2cc(C)no2)=O)(NC(=O)Cc2cnoc2)CCOCC1 C1(NC(C2CCCCS2)=O)C2CC1N(C(=O)CCC13CCC(CC1)C3)C2 c1(NC(N(C2CC3CC2CN3)C(C)C)=O)ccc(Oc2ccc(Cl)cc2)c(F)c1 N1(C(c2n(C)ncc2)=O)CC2CCCC(C1)N2C(c1cc([N+](=O)[O-])cnc1O)=O Cc1cccc(CCC(=O)NC2CCN(C(C3CN(c4nncs4)C3)=O)CC2)c1 N1(C(CCCC(C)C)=O)CC(NC(=O)C2=C(Cl)CCC2)C2CCCC12 C1(CC(=O)N)CC2CCC1CC2.C1(C(N2C(C3CC3)CCC2)=O)CCCC(F)(F)C1 n1(CCCC)nc(CCCCN(C)C)nc1-c1oc(SC)cc1C C(=O)(C1=CCN(C(c2ncc[nH]2)=O)CC1)N(C1CCC(F)(F)C1)C N1(C(C(C)=C(CC)C)=O)CC(NC(c2nonc2N)=O)C(CC2CC2)C1 C(=O)(C(C(C)C)n1cc(C2(N(C)C)CCOC2)nn1)N(CC(N)=O)CCC CC1(C)CCN(C(C2CC(N(C)C)C2)=O)CC1CNC(=O)CCc1cscn1 c1(C(C)NC(c2ccc(F)cc2)C2CC3(C2)CC3F)ncc(F)cc1F C1(C(=O)NC2CCOCC2)C2C3CC4C1C2C34C(=O)N(CC(O)CO)CCO CCCCCCCCNC(=O)NC1CC12CCN(C(=O)CCc1ccoc1)C2 Cc1sc(O)nc1C(=O)NC1CCCC1C.C(=O)C(C)(C)C.C(=O)CC.N c1(C(N2CCN(C(C(F)=C(C)C)=O)C(CC(F)F)C2)=O)cnc2ncccn12 C#CCC(CCOC)NC(=O)NC(CCNC(=O)OC)CCO c1(C(c2nn[nH]n2)C)cccc(NC(c2conc2C2CCCC2)=O)c1 N1(C(C(CC)n2cncn2)=O)CCC(CCCCCNC(C2CC(C)(O)C2)=O)CC1 Cn1cnc2cc(C(=O)NCCN(C(c3ccsc3C#N)=O)C3CC3)ccc12 CCCCCC(C)(CC)C(=O)N(CCNC(=O)C(O)C(F)F)CCOC C(C=O)(C1CC1)NC(=O)OC(C)(C)C.c1(C=O)cnco1.CC=CC N1(C(=O)C)CC2=C(C1)CN(C(c1ccc3c(c1)COC3)=O)C2.[SH](=O)(=O)C1CC1 S(=O)(=O)(c1ccc(-c2cc(NCc3ccc(O)c(Br)c3)ccn2)cc1)NC Cc1ccc(OC(C)C(=O)NCCC(O)C)cc1.c1(C=O)cnc(C(C)C)[nH]1.N c1(C(=O)NC2C(CNC(c3ccc(C)o3)=O)CCC2)ccc(CO)c(F)c1 N1(C(c2c(CC)nn[nH]2)=O)CCC(N(C(=O)CS)C)C2(CC2)C1.c1ccccc1 N1(C(c2cccc(-c3nnc(C)o3)c2)=O)CCCCC(NC(=O)CSC2CC2)C1 c1(C(=O)OC)sc2ncccc2c1NC(=O)CC1CCCN1C(C1CCCC1)=O c1(C=O)ccc([N+](=O)[O-])[nH]1.C1CCC1.C1(C(=O)OC)CC1C=O.C(C)C CC1(CC(=O)NCC23CC(CO2)C3)CCN1C(=O)CSC1CC1 CCCCCCCCCCS(=O)(=O)NC1CCN(C(=O)COC(C)=O)C1 C1(CC(=O)OC)CCCN(C(c2noc(C)n2)C)CC1 c1(CNC(CC=C)=O)ccc(C(N2CCOCC2C2CC2)=O)cn1 C1(CC(=O)NCC2CC(O)CN2C(C2CCC23CCC3)=O)NC(=O)NC1=O N1(C(COC(C)C)=O)CC2CCC1(CNC(=O)CC1CCC(C)C1)CC2 N1(C(C2(C)CC2(F)F)=O)CC2CC(NC(c3ccccc3SCCO)=O)CC1C2 C#CC1(C(=O)NC2CCN(C3CC3)CC2)CCN(C(C2CCCC2C)=O)CC1 c1(C(=O)NCC2(C)CC(NC(=O)COC(F)F)C2)cc(Cl)cc2c1OCC2 C=C1CCC(C(=O)NCC(CC)NC(c2csc(C(F)F)c2)=O)CC1 Cc1ncc(C(=O)NC2CN(C(c3c(C)n[nH]c3C)=O)CC2(F)F)c(C)n1 CN1CC(C(=O)NC2(CNC(C3(O)COC3)=O)CCOCC2)CCC1=O N(C1COc2ccccc21)CC(c1ccc(NC(c2ccccc2)=O)cc1)N N#CC1(CC(=O)NC2C3CCC(C3)C2C(N2CC=C(CO)CC2)=O)CCOCC1 Cc1cc(C(=O)NCCC(C)C)n(C(F)F)n1.C1(C=O)CCC(C(N)=O)C1.N C1(CC(=O)NC(CC)CCCO)Cc2cc(C(F)(F)F)ccc2O1 C1(NC(CN(C)C)=O)CC(NC(C2(C)COC(=O)OC2)=O)C12CCC2 N1(C(CCC(=O)NCCC)=O)CC2CCCC1CN(C(=O)Cc1cncnc1)C2 C1(C(=O)Nc2ccc(C(C)C)cc2Cl)Cc2ccc(F)cc2O1 c1(C(N2CC(C)(NC(CC(CC)CC)=O)C2)=O)cccc2c1OC(C)C2C N1(C(C2C(C)C2)=O)CCN(C(c2cccc(-c3nnco3)c2)=O)CC1CCO c1(C(=O)NCC2N(C(C3=C(C)CC3)=O)CCCC2)cnc(C)nc1C N1(C(C2CN(C(C(CC#C)C3CC3)=O)CC2C(C)C)=O)CCc2n[nH]cc2C1 C1(N=[N+]=[N-])(C(N2C(C)CC(F)C2)=O)CCN(C(c2ncccc2N)=O)C1 c1(C(=O)NCC2(C(=O)NC3CCN(CC)C3)CCCO2)c(F)cccc1F C#CC1(O)CCN(C(C2CC(NC(=O)CCS(N)(=O)=O)C23CCC3)=O)C1 c1(C(=O)NC2CC(NC(C3(C#N)C(C)(C)C3)=O)C2)[nH]c(Cl)c(Cl)c1Br CC(C)(CC1CCCN(C(C(=O)NCC2CC2)C2CCC2)C1)C(N)=O N1(C(CCC)=O)CCC2(CCC(NC(=O)C=CC(C)CC)C2)CC1 N1(C(c2ccc(SC)cc2)=O)CCCC(C)(NC(=O)C(O)C(F)(F)F)C1 CC(C)(C(=O)NCC1CCC(C(=O)NCCc2nc[nH]n2)C1)n1cncn1 CC1CN(C(C2C3CC(F)(F)CC23)=O)CCN1C(=O)CCSCC(N)=O Cc1cc(N2CCC(CC(F)F)C2)ncc1S(=O)(=O)NCCOc1ccccc1 N1(CC=C)CC=C(CCNC(=O)C(CC)(CC)CC)CC1 c1(C(=O)N)cc2c(nn1)CCCO2.C1(F)(CNC(=O)CN2CC=CC2)CCC1 CC1(C)C2CCC1(C)C2C(=O)OCC(c1[nH]c(Cl)c(Cl)c1Br)=O C1(C(=O)NCC(C(=O)NC)O)CN(C(C2OCCC2C(C)C)=O)CCN1C C1(CNC(c2c(CC)cncc2)=O)C(C2CC2)CCN1C(c1ccncc1O)=O Cc1c(C(=O)NC2CCN(C(=O)Cc3ccc(OC(F)F)cc3)C2)cccc1O N1(C(c2ccnc(C)n2)=O)CC2(CCC(CNC(C3CCC34CCC4)=O)O2)C1 C1(C(=O)NC2(C=C)CCCC2)C2CC3C(C2NC(=O)C)C13.C1CCCC1.O c1(CN2CCC(F)(C(=O)Nc3cc(C)c(Br)nc3)C2)c(F)ccc(Br)c1Cl CCC(C(=O)NC(C(=O)NC1CC(C)(C)OC1=O)c1ccoc1)C(F)(F)F Cc1ccc(C(=O)NC2CC3COC2C3)c([N+](=O)[O-])c1.C1(C(=O)N)C2CCCC12 CC(CCC(=O)NC(C)(C)C(O)CO)NC(C1CCOC1(C)C)=O C1(C(N(CCC(=O)N)CCO)=O)CC(=O)OC1(C)C.n1(CC)nccc1C C(C1CCC(C)CC1)=C(C=O)C.c1(C(C)=O)ccc(C(=O)NC(C)CC)cc1.N N1(C(C(C)Oc2ccccn2)=O)CCC(O)C1C(N1CCN(C2CC2)CC1)=O C1(NC(CCC2(C)CN(C(C3C(C)=CCS3)=O)C2)=O)CC1C1CCCCC1 C(C)(C)(C=O)N(CCOC(C)=O)C(=O)NC(n1ccnc1C)C.C(C)C C=CCCC(C(=O)NCC1CCOC1=O)NC(c1ccnc(C)n1)=O N1(C(C(C)Cc2cnc[nH]2)=O)C2CCC1C(CNC(C1(N(C)C)CCC1)=O)C2 n1(CC=O)ccc(=O)c2ccccc12.C=C(C)C(C)(C)C(=O)NCCO.CC C1(C(C)C)(C(=O)NC2CCCC(NC(c3cnc(S)nc3)=O)C2)CNC(=O)C1 C1(N(C(c2cc(OC)no2)=O)C)CCC2CN(C(=O)C#CC(C)(C)C)CC12 N1(C(C(C)N(C(c2ccc(C=C)cc2)=O)C)=O)CCCC2CCCCC12 CC1(CNC(c2cncc(O)c2)=O)CCC(NC(=O)CO)C1.c1ccncc1 C1(C)(NC(CCC2N(C)CCC2)=O)CCCN(C(C2(O)CCCCC2)=O)C1 CC(C)CS(=O)(=O)CCC(=O)N1CCC2C(NC(c3ccn(C)c(=O)c3)=O)C12 CC(C)C(CCN(C)C(C1(C)CC1)=O)NC(c1cnc(S)n1C)=O c1(NC(CC(C)c2cnn(C)c2)=O)cccc(-n2ccnn2)c1 c1(C(C(=O)NCCCC)N(CCC(C)C)CC(C)C)cc(Cl)ccc1Cl c1ccc2c(cnn2CC)c1.c1(CNCC(CSC)O)cccc(C(=O)O)c1 C(c1cncc(O)c1)=CC(=O)NCC1(C)CCN(C(CNC(CC)=O)=O)C1 c1(C(=O)NCC2OCCC2C(=O)NOCCc2cccs2)ccc2cc[nH]c2c1 C1(CCNC(CCN(C(C)=O)C)=O)CCN(C(C2ON=C(C)C2C)=O)CC1 c1(OCC(=O)NCCC2CN(C(C(CCC)C)=O)C2)cc(C)ccc1Cl C1(NC(CCCN(CCC)CCC)=O)CCC(C)N(C(c2cnn(CC)c2)=O)C1 C(=O)(C(CCCO)c1ccccc1)NCCCC(C)NC(=O)CCS(C)=O C(C(=O)NCC1COCCN1C(=O)CCCCc1cccc(O)c1)(C(C)C)SC c1(OCC)ccc(C(=O)NC(C2(O)CN(C(=O)C(=O)NOC)C2)C)cc1 N1(C(CC(CN(C)C)O)=O)CCC2(CCN(C(c3cc(C(F)F)nn3C)=O)C2)C1 c1(C(=O)NC2C(NC(=O)CC3CC3(Cl)Cl)COCC2)cc(O)c2ccsc2c1 C(C)(CCNC(=O)C(C)N)NC(C1C(COC)C1)=O.[SH](C)(=O)=O C=C(C)CC(C(=O)N1CC(N(C(=O)CC2CC2)C)C1)OC CN1N=C(CC(=O)N2CC(=O)NCC2C(N2CCC23CC(O)C3)=O)CC1=O c1(C(=O)NC2C(C(N(C3CC(OC)C3)C)=O)CN(CC)C2)[nH]ccc(=O)c1C CCC(CNC(=O)C1CCc2nccn21)(CC)C(=O)NOCC1CCOCC1 c1(C(N2CC(CC)C(NC(C3CCC4(CC4)C3)=O)C2)=O)ccc2c(c1)OCO2 N1(C(C(C)n2ccnn2)=O)CC2CC(NC(=O)CC3CCSC3)C(C2)C1 c1(C(=O)NCCCC(C)NC(CC(CC)C)=O)ncc(C)cc1C NS(=O)(=O)c1ccc(SCC(N2CC3COCCC3(NC(=O)CCF)C2)=O)cc1 c1(C(N(C(C2N(C(C3(C=O)CC3)=O)CC(F)C2)=O)C)C)ccc(C#N)cc1 C1(NC(C)=O)CCCCN(C(=O)C(=O)NC2CC2c2ccc(OC(F)F)cc2)C1 C1(C(=O)NC2CC(CNC(=O)CCN3CCCC3=O)C2)CCC(C2CCCO2)O1 Cc1oc(NC(=O)C(N2CCC(c3cc[nH]n3)C(C)C2)C)c(C#N)c1C C1(C(=O)NCCCN2CCCC2)(NC(C2CCC2)=O)CCSC1 c1(OC)cc(C)c(CN2CC3CN(C(c4cc(O)ccc4O)=O)CC23)cc1C C1(NC(c2cc(C)c(C)o2)=O)(CNC(c2cnn[nH]2)=O)CC2CCC1CC2 Cc1cc(CCC(=O)NC2CC(C)(NC(c3cnn4c3CCC4)=O)C2)cc(C)c1 C(C(=O)OC)(C(C)SC)N(C(c1cn(CC)nc1)=O)C c1(C(N2CCC(n3cc(C(C(C)(C)C)O)nn3)CC2)=O)cncc2ccsc12 c1(C(N(C)CC2CCN(C(CC=CC)=O)C2)=O)ccc2ccc(Cl)cc2n1 Cc1cc(C)c(C(c2nnnn2-c2ccccc2)NCCc2cccnc2F)s1 N1(C(C2CC3(CCCO3)C2)=O)CC2CC(NC(C3(Cl)CC3)=O)CC1C2 c1(C(=O)NC(C)CC(C)NC(c2cnn(C3CCC3)c2)=O)ccc(C2CC2)cc1 N1(C(=O)CC(C(F)(F)F)NC(C2(O)CCC2)=O)CCC2(CCCCO2)C1 CC1(C)OC2(C(=O)NCCO)CCC1CC2.c1(C=O)ncsc1C1CC1.CC N1(C(c2cc(CC)on2)=O)CC2CCC(C1)C(NC(c1cccn(C)c1=O)=O)C2 c1(C(=O)NCC(CNC(C(CC)Sc2ccccc2)=O)O)cnc2n1CCCC2 N1(C(COC)=O)CC(NC(c2ccc(OC)cc2Br)=O)C2(CC2)C1 C1(OCC(=O)NCCN(C(=O)CO)CCC)CCCCC1.c1cccnc1 C12(CC)CC(C(=O)NC3CCCCC3)(CO1)C2.c1(CC=O)ccc(Cl)s1.C N#Cc1cnn2ccc(=Nc3ccsc3C(=O)Nc3ccc(Br)nc3)[nH]c12 CCC(CNC(=O)CC1CCC(C)CC1)(CC)C(=O)NC1(C(O)CO)CC1 c1(NC(N2CCOCC2)=O)ccc(Cl)cc1[N+](=O)[O-].[SH](=O)(=O)CC1CCC1.C C1(NC(C(C)(C)N2CCCCC2)=O)COCCN(C(C2CC3(CCCC3)C2)=O)C1 C1(NC(c2c(CC)cccc2)=O)CC(C(=O)NC(c2nncn2C)C)=CC1O c1(CC)cc(=NC(=O)C23CC(CN(C(=O)COC4CCCCC4)C2)C3)[nH]n1C Cc1cc(OCC(=O)NCC(O)CNC(=O)C(C)C(F)F)cc(C)c1Cl C1(NC(c2n(CC)nnc2)=O)CCCCN(C(C2C3CCC(F)(F)C23)=O)C1 CCC(CC)C(=O)NCC1CCCC(CNC(C2(CO)CC(F)(F)C2)=O)C1 c1(C(N2CC(NC(COCC(C)C)=O)C(C)(C)CC2)=O)ccc2ncncc2c1 CCC(C)C(C)C(=O)NC(C)(CNC(=O)Cc1cn[nH]c1)C1CC1 c1(CCC(N2CCC2)=O)ccc(C(=O)O)c(F)c1.n1(CCCOC)cc(C)nn1 C1(C(=O)NC(CNC(C2C(=C)CC2)=O)(C)C)(Cc2cnn[nH]2)CCCC1 Cc1c(C(N)=O)cccc1C(=O)NCCc1ccccc1.c1(C(=O)N)cnsc1 N1(C(Cc2cnc(C)s2)=O)CC(NC(=O)CC2CCN(C)CC2)CC1C C(CNC(=O)CCO)(CC(=O)N(C)CCN(C)C)OC.C(C)C.C(C)C C1(C(=O)OC)CCCC(C)(C)C1CN=c1[nH]nc(-c2sccc2C)o1 C12(C(=O)OCc3ccc(CC)s3)CCC(CC)(CC1)OC2 C1(C(N2CC(F)C2)=O)C2CCC(C2)S1(=O)=O.c1(C(=O)N)cnn2ncccc12 Nc1cncc(-c2nc(CCNC(c3cccc(Cl)c3)=O)no2)c1 c1(C=O)ccc([N+](=O)[O-])c(C)c1.C(CC)(C(C)C)NC(C(C)=C(CC)C)=O.N CC1Cc2cccnc2N(C(=O)N=c2cc(-c3ccc(F)cc3)o[nH]2)C1 c1(C2(C(=O)NC3CCC(CNC(c4ccncc4)=O)C3)CC2)ccccc1Br C1(C(=O)NC(CCOCC)C(=O)NCC=C2CCSCC2)CCCCNC1=O C(CC1=CCCCC1)NC(CC1CCN(C(Cc2ccc(OC)cc2)=O)CC1)=O C1(OC)CN(C(=O)C(C2CCCCC2)C)CC1.c1(C(=O)N)coc(C(C)(C)C)n1 C(=O)(C(O)CC(N)=O)NC(C)(C)CC=CC(N1CCCCC1)=O C1(OCC)CN(C(C2(C)CC2)=O)CC1CNC(=O)C(C1CC1)SC C(=O)(CCC(=O)c1ccccc1N)NC(C)CCNC(=O)C(F)C1CCC1 C1(C(N2C3(C(=O)NCCN4CC(OC)C4)CC3CC2)=O)CC(=O)C12CCC2 O1N2CCC(CC2)NC(=O)C1.c1(CCCSCC)conc1C(=O)OCC C(C1CCc2cc(Br)ccc21)NC(NC(CC)C)=NCc1cccnc1O N1(C(C2C(CC)C2)=O)CCOC(CNC(=O)C=Cc2ncc[nH]2)C1 N1(C(C2(CNC(C3C(C)CCCC3)=O)CCC2)=O)Cc2nncn2C(C)C1 c1(N(C)C(c2ccccc2OCc2cnnn2C)=O)ncc(Br)cn1 c1(CNC(C=CC)=O)ccc(C(=O)NCC(C)(CC)CO)cn1 Cc1cc(C(=O)N(CCC)C)cnc1C(F)F.c1(CC=O)cc(C2CC2)no1.N C1(NC(C2(C(N)=O)CC2)=O)CC2(C1)CN(C(=O)CC1(CO)CCOCC1)C2 C=C1CCN(C(c2[nH]ccc2CC)=O)C(C(=O)NCC(c2cn(C)cn2)O)C1 O=S(=O)(Oc1ccc(OC(F)F)cc1)c1c[nH]c2c(Br)cccc12 c1(CCC(N2CCC(NC(=O)CCC3CCCO3)C2)=O)cccc(F)c1 N1(C(C2CCC(C)O2)=O)CC2(CC2C(=O)Nc2nc(Br)cn2C)C1 C1(NC(c2c(C)nc(O)cc2)=O)CC1C1CCCN(C(=O)C2=CCC2)C1 C1(CC(=O)NCc2scc(C)n2)CN(C(=O)Cn2nccc2C)CCC1C c1(OC)c[nH]c(C(N2CCC2CNC(c2csc(S)n2)=O)=O)cc1=O C(c1ccc(Cl)s1)=CC(=O)NC(C)(CNC(=O)CC1CCCOC1)CO C12(NC(C(N3CCNC3=O)C)=O)CC1CN(C(=O)C(=Cc1cscn1)F)C2 N1(C(C2C3C(NC(C(c4ccn(C)c4)C)=O)C4C(C3)C42)=O)CC(C)CCC12CC2 C1(CC(C)NC(C2(N3CCNCC3)CC2)=O)CC(C)(C)NC1=O C12(C(N3CCC(CC=C)C3)=O)CCC(C)(CO1)C2.c1(C(=O)N)ccc(=N)[nH]c1 CC1C(NC(=O)CCOC2CN(C(=O)C(C)(Cl)Cl)C2)CCN1C c1(C(=O)NCCN(C)C(C2CCCN2C2CC2)=O)nc(Cl)sc1Br C1(CN(C(C2CC(C)C2)=O)C)CCN(C(c2ccccc2-n2cncn2)=O)CC1 CC1CC=C(C(=O)NC2(C(N3CCCSCC3C)=O)CC(O)C2)CC1 C=CCC(C)(C(=O)N1CCCCC1CNC(c1csc(C=O)c1)=O)N(C)C.O c1(CC)cnccc1C(=O)NC1CCC(NC(=O)C(O)CCSC)CC1 Cc1c(N2CCCN(C)CC2)ncnc1N1CCC(C#N)C1 N1(C(=O)C(O)CC2CCCC2)CCCC(CCO)CC1.C(C=O)C1(O)CCC1 [SH](=O)(=O)c1ccccc1N.C1(NC(C2C(C)(C)C2)=O)CCCN(C(=O)CN)C1 N1(C(C(Cc2ncn(C)c2)O)=O)CC2CC(NC(=O)C(=O)NC3CC3)C1C2 N#Cc1ccc2c(c1)CN(C(C1CC(F)CN1Cc1csc(Br)c1)=O)CC2 c1(N(C(C)=O)C(C2CC2)=O)cc(O)nc(O)c1.C(=O)C#CCCc1ccccc1 c1(OC)ccc(CCC(=O)N2CCC2CNC(=O)CO)cc1F.C1(C)CCC1 c1(C(=O)NCCC2CN(C(CCC=C)=O)CC(C)O2)ccc2nc(C)ccc2c1 C1(C(=O)NCC(C)(C2CCC2)NC(=O)Cn2cccn2)CCc2cnnn2C1 N1(C(=O)Cc2csc(Br)c2)CC2C(c3cn(CC4(O)CCSCC4)nn3)C2C1 N1(C(c2cncc(CNC(C(CCC)N(C)C)=O)c2)=O)CCCC12CCOC2=O c1(C(=O)NCCOCC(=O)NC(CN(CCCC)C)C)cc[nH]c1 c1(CNC(C(=O)NCCOC)=O)cc(CSCC(C)C)no1.CC N1(C(COCc2cc(C)no2)=O)CCN(C(=O)Cn2cc(F)ccc2=O)CC1C N1(C(=O)NC2CC(CCOCC)C2)CC2(CO)CCC2(CO)C1 CCCN=C(NCc1ccc(Br)o1)NC1CC(OCC)C12CCC2 C1(N(C(CNC(=O)OC)=O)C)CC2(CCN(C(=O)C)CC2)C1.c1cccs1.S C1(C(N2CCN(C(CS(CC)=O)=O)CC2c2cn[nH]c2)=O)CC2C=CC1C21CC1 N1(C(=O)NCc2ccns2)CCC2(Cc3ccccc3C2=O)C1 N1(C(CC(C)(C)C#N)=O)CCC(NC(=O)CC23CCC(CC2)C3)C(C)(C)C1 c1(C(=O)NCc2ccc3ccccc3n2)ccc2cnnc(O)c2c1 c1(OC(C)C(=O)OC2CCCC2O)ccc(C#N)cc1.C(=O)C(C)(C)C1CC1.N C(=O)(C(O)C(F)(F)F)NC(C)CCCNC(c1ccc(OC2CC2)cc1)=O C(N=c1[nH]c2cccc(Br)c2o1)C1(C)CCN(C(C2CCCC(=O)N2)=O)C1 C1(C(N2CC(F)(CNC(c3nocc3Cl)=O)C2)=O)(CC)CCCC1O Cc1cc(F)cc(C(N2CC3CCN(C(C4CCCN4C)=O)C3C2)=O)c1N C1(C(=O)NCCCN(C(c2sc(F)cc2Cl)=O)CC)CCn2c(cnc2C)C1 N1(C(C(C(C)C)CN(C)C)=O)CC2(CNC(c3ccns3)=O)CC1CCO2 c1(C(N2CCN(C(c3ccn(CCC)n3)=O)CC2)=O)cnc2[nH]nc(O)c2c1 CC(C)CCCNC(C1(CO)CC(C)(C)C1)=O.C(=O)C(C)(C)CC1CCC1 c1(SC2C(=O)N(c3ccc(Cl)c(Cl)c3)CCC2)ccccc1[N+](=O)[O-] C(=O)(CCCC#N)NCCCCN(C)C(C1CCC(=O)N1C1CC1)=O CC1CN(C(C2CC(N(C)C)C2)=O)CC1NC(c1cnsc1)=O C#CCCCC(=O)NC1CCN(CCCNC(=O)C(c2c(C)n[nH]c2C)C)C1 CC(CNC(c1cccc(CCO)c1)=O)S(C)(=O)=O N1(C(CC2C(C)(C)CCCO2)=O)CC2CC(NC(c3ncc[nH]3)=O)CC1C2 O=C1CC(C(N2CCN(C(c3ccc(C4CC4)o3)=O)CC2)=O)CCN1 CN1C(=O)NCC1C(=O)NCC1CCOCC1.n1(CCC=O)ccc(=N)[nH]1.N c1(OC)cc(C=O)ccc1OC(F)F.C1CC1.C(=O)C=C1CCC1.C1CC1 c1(C(N2C(C)CC(c3ccccc3)C2C)C(=O)NC)ccc([N+](=O)[O-])c(Cl)c1 N1(C(COCCCCC)=O)CC(C(=O)NCCC(C)(C)CO)CCC1(C)C N1(C(C=CCCC)=O)CC(NC(c2cc(C)sn2)=O)CC12CCOCC2 c1(C(N2CCC(CCOC)(NC(=O)CCCCC3CC3)C2)=O)ncc(F)cc1N c1(N2CC3(C)C(c4ccsc4)(C2)C3)cnn(-c2ccccc2[N+](=O)[O-])c(=O)c1Br C1(C)(C(=O)NC)CCCN(C(c2ccnc(Cl)c2O)C(=O)NCC2CC2)C1 C(C)(C(=O)Nc1nc(Cc2nn[nH]n2)cs1)(C1(C)CC1)OC C(C1=CCCOC1)NC(C(C1CN(C(c2cc(F)c[nH]2)=O)C1)OC)=O c1(C=O)cnc(=N)[nH]c1.C12(C=O)CC(C1)C2.C(=O)(C)NCCOC.N C1(C=O)CC(C)C1.C(c1ccsc1)=CC(=O)N(C1CCC1)CC=O.CC C1(C(=O)NC(C)CN(C)C(C2CCCN2C)=O)COC(C)(C)O1 c1(C(C)C)ccc(C#N)c(C(C(C)CNN2CCOCC2)=O)n1 Cn1ccc2nc(NC(c3ccc4c(c3)CN(S(=O)(=O)C3CC3)C4)=O)nc(Cl)c12 c1ccc([SH](=O)=O)c(Cl)c1.C1(CC)CCS(=O)(=O)C1.CC1(CC)CC1(F)F.N c1(C(=O)NCC(C)N(C(C(C=CC)O)=O)C)ccnc(OC2CC2)c1 CCC(C)CCCCC(=O)NCC1CC2CCC1N2C(c1cc(Cl)ncc1Cl)=O C1(NC(C2C(CC)C2)=O)CN(C(c2[nH]c(C)nc2C)=O)C(CC)(CC)C1 N1(C(=O)NC(C)C(c2ccc(Br)cc2)O)CCOC2(CCCC2)C1 Cc1nc2cc(C(=O)NC3CCN(C(=O)CCF)CC3F)cnc2[nH]1 C1(C(=O)NCCCN2CCN(C(C(C(C)C)C)=O)CC2)Cc2cncn2C(=O)N1 C1(NC(C2(N=[N+]=[N-])CC2)=O)CN(C(=O)CCSC(F)(F)F)CC1C(F)(F)F Cc1cccc2[nH]c(C(N3CC4CC(C3)N(C(=O)Cn3cc(Cl)cn3)C4)=O)cc12 CC(CN(C)C)C(=O)NCCCC1CC1.c1(C=O)csc(C(C)(F)F)n1.N CCCC(C(=O)NC1CN(C(=O)C(C)C)CC1n1cccn1)c1ccc(Cl)cc1 O(N(CC)C(=O)C(c1ccccc1)NC(=O)Cc1ccc(O)cn1)CC c1(SC)ccc2c(C)cc(N(C)Cc3c(Br)cccc3Br)nc2c1 c1(C=O)cc2cccnc2s1.c1(OC)cc(C(=O)NCC2COCC2)n(C)n1.N C(=O)(CCCC(F)(F)F)N(C(C(=O)N(CCOC)C(C)C1CC1)CC(F)F)C C(=O)(C1=CCC(F)(F)CC1)N(CC(C)O)CCNC(C(CC(C)C)O)=O C1(CNC(C(C2CC2)OC)=O)CCCCN(C(=O)C)C1.c1cccc(C)c1F.O C(CCC(=O)NCCCc1cc[nH]n1)N(C)C(c1cnn(CCO)c1)=O c1(-c2n(-c3c(OC)c(Cl)ccc3)nc(CO)n2)ccc2oc(=O)oc2c1 c1(C(=O)NC(C(C)NC(=O)Cc2cc[nH]c2)C)c(Br)cnn1C1CCC1 c1(C(N2C(C(=O)NCCCOCCCC)CCC2)=O)cc(F)c(F)c(Br)c1F C(CC(C(C)(C)C)NC(=O)CSCCC)N(C(CCCOCC=C)=O)C C1(COC)(NC(=O)CC(C)CN(C)C)CCN(C(=O)CCCC(=O)OC)CC1 c1(OC)ccc(C2CN(C3CC3)C2)nn1.C12OCCC1N(CC(C)C)C2 C(=O)(C1=CCC(C)(C)CC1)NCc1cc(C(=O)NC(C)CC(N)=O)sc1 c1(C(=O)NC2CCCCN(C(C(C)N3CCC3)=O)C2)ccc([N+](=O)[O-])c(Cl)c1 c1(C(=O)NC2C(NC(C(C)CN(C)C)=O)CCC2)cc(Cl)cc(Cl)c1[N+](=O)[O-] C1(CCNC(CC=C)=O)(C(=O)N(CC)Cc2ccn(C)n2)CCCC1 n1(CC(N2CC(C(C)NC(C3C(=C)CC3)=O)C2)=O)cc(C)cn1 CC(C(C)(C)CO)NC(C12CC(CN1C(C1(C)SCCCS1)=O)C2)=O C1(C(N2C(C(C)(C)NC(C3CC4CCC3O4)=O)CCC2)=O)CC2(C1)CC(F)C2 c1(CC(=O)NCC(CNC(c2nc(CCC)sc2)=O)O)cccnc1C C1(C(=O)NC(C)CCCCNC(=O)Cn2cnnn2)CCn2nnnc2C1 c1(C(=O)N)ccnc2c1CCO2.C1(NC(C=CCN(C)CC)=O)CC(C)C1 N1(C(c2cc(CCCCC)[nH]n2)=O)CCC2CCC(NC(=O)C=CI)C1C2 c1(C(N2C(C)CCC(NC(C3CCC(=C)CC3)=O)C2)=O)occ2c1CCOC2 Cc1cnsc1C(c1nnnn1C)NCC=C(Cl)Cl N1(C(=O)NC2CC(NC(=O)OCC)C2)CC(Cc2ccccc2)C(C)C1 c1(NC(C(N2C(CC(C)O)CCC2)=O)=O)ccc(C(=O)NC2CC2)cc1 CCC(O)CC(=O)OCC(c1cncc(F)c1)=O c1(C(=O)NC2C(NC(C(C)OCCC(C)C)=O)CCC2)ccc2ccncc2c1 N1(CC(=O)Nc2c(C)occ2)CCN(C(c2ccoc2Cl)=O)CC1 C(=O)(C(CC)CC(F)F)N1CC2(N(C(C(CCC)O)=O)CC2)C1 C(=O)(CCC1=CCCCC1)N(C1CCCC(N(C)C(c2ccccc2Cl)=O)C1)C C1(NC(C(CC)n2ccc(C3CC3)n2)=O)CCN(C(c2[nH]cnc2C)=O)CC1 N1(C(COC(C)(C)C)=O)CCCC2(CCCN2C(c2ccc(Cl)nn2)=O)CC1 N1(C(C2CCN(CC)C2)=O)CCN(C(=O)CN(C)C(c2cncn2C)=O)CC1 C1(C(C)C)CN(C(c2onc3c2CCCC3)=O)CCCN1C(=O)Cn1nccn1 c1(C(C(=O)N)C)ccc(C(F)(F)F)cc1.N1(C(C(C)OCOC)=O)CC(CO)C1 C1(NC(c2cccc3sccc23)=O)CC(NC(=O)C2=CCSC2)C12CCOCC2 c1(OC)cc(F)c(F)cc1NC(C1CCC2(CN(Cc3cccnc3Cl)C2)O1)=O Cc1ccc(C)c(NC2(CNc3cc(C(F)(F)F)cc(Cl)n3)CCCOC2)c1 CCCC(C(=O)OC)C(=O)NC(CNC(c1c(C)nn(CC)c1C)=O)CC c1(C(=O)NC2C(NC(c3ncn(C)c(=O)c3)=O)CCC2)cc(Cl)cc([N+](=O)[O-])c1 C1(NC(=O)OC(C)(C)C)CC2CCC1C1CN(C1CCc1ccccc1)CC2 Cc1ccn2ncc(C(=O)NC3CCCC3NC(c3ccnc(C)n3)=O)c2c1 CCC(CC(=O)NCC1(OCC)CN(C(C2(C)COCCO2)=O)C1)OC N1(C(CCC)=O)CCC(C(=O)NCc2ccc(C)o2)C1 C1(C(N2CCCC(C(CNC(CC)=O)(C)O)C2)=O)CCOC(C)(CC)C1 C1(CC=O)CC(C)(C)CN1C(c1ccon1)=O.C1(CC)(C)CC(C)(C)C1 C(C)(N=c1[nH]c2cccc(C)c2o1)c1ccc(OCCCC)c(OC)c1 C(C(=O)N=c1ccn(C(C)C)[nH]1)(C(C)C)NC(c1c(C)ccc(C)n1)=O Cc1nc(C2CCCO2)sc1C(=O)NC(C)(C)C1CC1.c1(C=O)cnc(O)s1 C(C(C(=O)N1CC(C(C)O)C1)C(C)(C)C)NC(COCC#C)=O C12(C(=O)N)CC(CCO1)N(C(=O)C(F)=CC1CC1)C2.Cc1cc(O)nc(C)n1 Cc1cc(C(C)C(=O)NC(C)(C)C)cc(C)c1.C(=O)C(F)(Cl)c1ccccc1.N N1(C(CSC)=O)CC2CN(C(C3C4CC3N(C=O)C4C)=O)CC2C1.C(C)(C)C.O N1(C(CC=CCC)=O)CC(NC(C2CCC(=O)N2C(C)C)=O)CC(O)C1 C(=O)(C(O)C1=CCCCC1)N1CC(N(C)C(c2ccn(CCF)n2)=O)C(C)(C)C1 C=C(C)C1CCC(C)(O)C(NC(N2CCCC2C2CCCOC2)=O)C1 N1(C(CCN(C(C(CC)C(=O)OC)=O)C)=O)CC2(CCC2)C12CCC2 c1(NC(=O)C=CCn2cncn2)ccc(CCn2ccnn2)cc1.O(C(F)F)C CC(C)C(C(=O)NCC(CO)NC(C1(n2ccnc2)CCCC1)=O)NC(N)=O c1(C(N2CC(NC(C3N(CCC)CCC3)=O)C(C)C2)=O)cc(C)ccc1OC C1(NC(c2c(C)nc(O)[nH]2)=O)CCN(C(=O)CCN2CCCCC2)C12CCCC2 C(CCCCCN(C(=O)C(C)SC(F)(F)F)C)NC(C(COC)NC(C)=O)=O C1(CNC(c2n(C(C)C)ccc2)=O)C2CN(C(=O)CC(C)(F)F)CC12 N1(C(C(C)OCCCC)=O)CC(F)(F)CC1C.C(=O)C(F)(F)c1cncs1.N c1(C(N2C3C(NC(C(C)N(C)C)=O)C(C3)C2)=O)ccc2c(c1)SCC(=O)N2 Cc1cnccc1CC(C)Nc1cc(N2CCC(C)(CO)C2)ncn1 c1(CNC(C(C)(C)CCC#N)c2n(CCC)nnn2)ccc2c(Br)cccc2c1 N1(C(C(C2CC2)OC)=O)CCC(NC(=O)CC2(C)CC2(Cl)Cl)C(C)(C)C1 C1(C(=O)NCC(C)NC(=O)CCSc2ccccc2)CCCS(=O)(=O)N1 Cc1cnc(NC(=O)CC2CCC(NC(=O)C3CC3)CC2)c(I)c1 Cc1cccc(C(=O)NCC2(C)CC2(F)F)c1F.C(=O)(C(F)n1ccnc1)N N1(C(C2(C#C)CC2)=O)CCC2(CCC2CNC(=O)CCCn2ccnc2C)CC1 C1(CC)CC(C(=O)NC2COCCN(C)C2)CCN1C(=O)Cn1ncn(C)c1=O C1(NC(c2c(C)snn2)=O)CC2CCC1N2C(c1ccc(C(C)O)cc1)=O C1(CNC(C(C)Cc2ccccc2F)=O)CN(C(c2csnn2)=O)CC12CC2 N1(C(CC)=O)CCC2CC(NC(=O)C(C)(C)c3cccnc3)CCC2C1 C(=O)(C1=CCCCCC1)NC1CCC(C)(c2cn(-c3ccn(C)n3)nn2)C1 C#CC1(OCC(=O)NC2CCCC2NC(c2occc2Br)=O)COC1 CC1(C(=O)NC2CCCC3(C2)N=N3)CC(O)CN1C(=O)Cc1cccc(O)c1 N1(C(CC(CC)O)=O)CCN(Cc2ncc(Br)cc2C)CC1CO N1(C(CCC)=O)CCC(C)C(NC(c2n[nH]c(C)c2Br)=O)C1 N1(CC(C)C)CCC(C(=O)NCCCNC(c2sccc2-c2ccccc2)=O)C1 C1(C(N2CCC(F)(F)C2)=O)Cc2ccccc2CN1C(c1cc(Cl)ccc1Br)=O C=Cc1cncc(C(=O)N(C2CCC(CNC(=O)CSC(F)(F)F)CC2)C)c1 N1(C(C(CCCC)NC(C(C=C)CC)=O)=O)CCCC2COCC12 c1(N2CCC(C(N3CC=CC3)=O)(OC)CC2)cc2ccccc2cn1 c1(-c2onc(-c3nc(C)c(C)[nH]3)n2)ccc2c(c1)CCCN2Cc1ccccc1 Oc1nc2ccc(OC(F)F)cc2s1.c12noc(n1)CO2 CC1c2nccn2CCN1C(CC1(C#N)CC1)C(=O)NCC1CCCO1 CC(C)(CO)C(c1ccccc1)NC(c1coc(C(F)F)n1)=O S(=O)(=O)(c1cccnc1N1CC2CC(C)(C)C2C1)NC(CCCC=C)C CCC(C)C(O)C(C)C(=O)N(CC(=O)NCCn1cnc(C)c1C)CCOC C1(CN(C(C=CCOC)=O)C)COCCN1C(C1CC=C(C)CC1)=O c1(SC)cccc(C(=O)NCCCC2CCCN2C(=O)CCC2CC2(C)C)c1Cl Cn1nncc1CC(N1CCC(CCC(N2CCCCC2)=O)C1)=O C1(C(=O)N)CC2(C1)C(C=O)C2(F)F.N1(C(C=CCCC)=O)CCC(CC)C1 C(=O)(C(C)(CC)CC)N1CC(NC(c2cc(COC)cn2C)=O)C(C)C1 c1(C(=O)NCc2ccc(C(CC)(C)C)cc2)cccc2c1CCCC2 C1(NC(Cc2nc(CC)sc2)=O)CCN(C(=O)C2=CCCSC2)CC1C(C)C c1(CNC(C(C=C=C)C)=O)nc2c(s1)CN(C(c1c(C)cc(C)cc1C)=O)CC2 Cc1ncnc(C)c1C(=O)NCC(CO)NC(c1ccccc1CC(F)(F)F)=O c1(C(=O)NC(CN(C(=O)CO)C)C)cnn(C)c1C1CC1.CC(F)(F)F c1(C(=O)NCC2CC(NC(CCCCC=C)=O)C2)ccc2c(c1)CC(=O)N2 Cc1ccc([N+](=O)[O-])cc1C(N1CCC(NC(=O)Cc2ccccc2)C(C)C1)=O c1(CNC(C2(CNC(CC3(C#N)CC3)=O)CC2)=O)ccc(CO)nc1 C1(O)(CC(=O)NCCCN(CCCNC(=O)C#CC2CC2)C)CCCCC1 Cc1ccc(-n2nccn2)c(C(=O)NC2CCN(C(=O)CC3CCSCC3)C2)c1 c1(CNC(CC=CCC)=O)n[nH]c2c1CN(C(=O)C(CC)C(=O)OC)CC2 C1(NC(C(c2cccnc2)N(C)C)=O)CN(C(c2nocc2Cl)=O)CC1O N1(C(C=C(C)C(C)(C)C)=O)CCC(NC(=O)CN2CC(C)(C)C2)C12CCC2 C1(C)(C=O)CCS(=O)(=O)CC1.c1nc(C(=O)N(CCC)C2CC2)c(C)o1 C1(NC(Cc2n(C)ccc2)=O)CCN(C(=O)CC(C)(F)F)CC1O C1(C)(C(=O)NCCN2CCC(C)C2)CCN(C(c2csc(Cl)c2)=O)CC1 CC1CCCC=C1C(=O)NC1C(C(=O)NC2CCN(C)C2(C)C)C1(C)C C(=O)(CCCCCCNC(C1CC12CC2)=O)N(C1CN(C)C1)C C(CN(C)C)(C(=O)N(C)Cc1cncnc1)NC(C(C)C1CC1)=O C12(NC(c3cc(C(F)F)ncn3)=O)CCCC1N(C(=O)C(Cl)=CCl)CCC2 c1(CN2CCCC(NC(c3ccc(N(CC)CC)cc3)=O)C2)cccc(F)c1C C1(F)(C(=O)NCc2nc(C)[nH]n2)CCN(C(=O)C=CC(C)C)CC1 C1(C(=O)NCCOCCCNC(C2C(C#N)CC2)=O)CC1C1CCCC1 C1(CNC(c2c(C)ncn2C)=O)CN(C(=O)CO)CC(C)(C)O1.C1CCC1 N1(CC(N2CCCC2)=O)CCC(O)CC1.C(=O)(C(C)(C)c1ccn(C)n1)NC.C C12(NC(c3cnc4scnc4c3)=O)CCC(CC1)N(C(C1CCOCC1)=O)C2 c1(C(=O)NC2C(NC(CC(=O)NCC)=O)CCCC2)cnn2c(Cl)cccc12 O=C1CCC2(CCN(N3CCC(n4nnnc4C(F)(F)F)C3)C2)N1 N1(C(C(C)SCCCC)=O)CCCC1C(C)(C)C.C1(C(=O)N)(C=O)CC1 c1(C(N(CC(N2CC(CO)CC2CO)=O)CCC)=O)cc(C#N)oc1C C1(C(=O)NC23CC(NC(C4CC5CC5C4)=O)(C2)C3)CCCS(=O)(=O)C1 C1(C(=O)NCC2CN(C(Cn3nnc(C)n3)=O)CC2C)CCc2c[nH]nc2C1 C1(C(N(CCCn2cc(C(C)(C)C(N)=O)nn2)C)=O)CCCNS1(=O)=O C(=O)(C(C1=CCCCCC1)N1CCN(c2ccccc2)CC1C)NC C1(C(=O)NC23CC(NC(=O)CN4CC5CC5C4)(C2)C3)C2CNC(=O)C12 N(C(=NCCCCl)N1CCN(CC2CCOC2)CC1)CC1CC(OC)C1 CCC(C)(COC)C(=O)N(C)CC1CCCN1C(=O)Cn1ccc(C)c1 N1(C(C(C)C2CCC2)=O)CC2(CNC(c3ccc(F)cc3)=O)CCC1CC2 Cc1nc(N2CCC(CNC(=O)CSCc3cccnc3)C2(C)C)cc(O)n1 CCC(CC(=O)NC1CCN(C(C2CCCN2C(=O)C(C)(C)F)=O)CC1)C(C)C c1(NS(C)(=O)=O)ccc(C(=O)NC2CCC(c3ccc(Br)cc3)C2)c(Cl)c1 CC1COCC(C(=O)NC2(C(=O)NCC3CCOC3(C)C)CC2)O1 c1(C(=O)NC(CC=C)C(=O)NCC2CCOC2)ccc(C#N)c(C)c1 C1(CNC(c2ncc(Cl)s2)=O)CCCC2(CCN(C(C3CCCC3)=O)CC2)O1 N1(C(CC2C(C)C2)=O)CCC2(CCCN2C(c2cn(CC3CC3)nn2)=O)C1 c1(C(N2CCC3(C(C(=O)NCCC(F)(F)F)C3)CC2)=O)cnnc2ccccc12 c1(C(=O)OCC)sc(NC(=O)CC2CN(C(c3ccccc3)=O)C2)cc1C C12(NC(c3c(Cl)cn(CCC)n3)=O)CCCC1N(C(=O)C)CC2.[SH](C)(=O)=O c1(OCC(c2ccc(OCC)cc2)C)cc(NC2CC2)nc(C)n1 CC1(CNC(C2CCCN2C(=O)CCCc2cnn[nH]2)=O)CC2CCC1C2 c1(C(=O)NCC2CC(NC(C3C(CC)OCCC3)=O)C2)cnn2ccncc12 N(C(=NCC(C)C)N(C)Cc1ccco1)C(C#C)CC1CC1 O(C=CC(=O)N1CC(N(C)C(c2ccc(-c3cccs3)[nH]2)=O)C1)CC c1(OC)cc2ccccc2cc1C(=O)NC1CC1NC(c1cccc(Cl)c1)=O C(=O)(C#CC1(C)CCCO1)NCC1(C(=O)NC2(CC=C)CCOC2)CC1 C(C1=CCCOC1)NC(=O)CCC1CCCN1C(=O)Cc1cnoc1 C1(C)(CC)CC(C(=O)NCC2CCCC2)CCO1.C(C(F)(F)F)=CC=O N1(C(CCc2nc(=N)[nH][nH]2)=O)CCC2C1CCN2C(=O)C1=NNC(=O)C1 CC(CC(=O)NC1CN(C(=O)C(O)CC)C1)n1cccn1.C(C)(C)C.C=O C1(CNC(C(CC)N(C)C)=O)CN(C(c2ccnc(Cl)c2O)=O)CCC1C N1(C(Cc2c(Cl)cn(C)n2)=O)CCCC(CCNC(=O)Cn2ccsc2=N)CC1 C1(NC(=O)CC2CC3CCC2C3)CC2CC(C1)N(C(c1csc(C3CC3)n1)=O)C2 C1(C(=O)NCC2CC(NC(C(CC)N(C)C)=O)C2)COC2COCC12 C(CC1=CCCCCC1)NCC(C(=O)OCCOC)(C)C CCCC(C)(CO)NC(C1CC(CNC(C23CC(C#N)(C2)C3)=O)C1)=O N1(C(C2CN(C(C)=O)C2)=O)C(C(N2CCCC(C#N)C2)=O)C2CC(O)C1C2 C(CNC(c1ccn(C)n1)=O)(CC(F)(F)F)NC(c1ccc(NC)cn1)=O N1(C(=O)CCCC(F)(F)F)CCCC(C2CN(C(=O)C3=CS(=O)(=O)CCC3)C2)C1 c1(C(=O)NC2CN(C(C(CC)OC)=O)CC(O)C2)cc2c(s1)CCC(C(C)C)C2 c1ccnc(Cl)n1.C1(F)(C(=O)NCCOC(C)(C)C)CCN(C(=O)C)C1.N C(=O)(C(C)(C)CCCNC(=O)C1=CCCCO1)NC(C#C)CCC C1(CNC(C(C)O)=O)CN(C(c2c[nH]c(C(F)(F)F)c2)=O)CC1(C)C Cc1cnc(C)c(C(N2CCC(C)C(NC(C3CCN(C4CC4)CC3)=O)C2)=O)c1 c1(C(=O)NCCN(C(=O)Cc2cccnc2C)CC)c(Cl)cc(C)cc1Cl c1(C(=O)OC)cc(C(=O)NCC)on1.C(=O)(CC)N.C(C)C.C(C)=O Cc1cccc2cc(C(N3CC(O)C(N=[N+]=[N-])C3)=O)sc12 C(=O)(CCCCC(F)(F)F)NCC1(C(C)NC(C(C)N2CCC2)=O)CC1 c1(CC(C)NC(c2ccc(C3CCCN3)s2)=O)c(F)cccc1F c1(CC(N2CC(NC(C34CCOCC3C4)=O)C2)=O)cc(F)c(F)cc1F C1(C(=O)NCC(=O)NC2CCCC(O)CC2)CC2CC1CC2O CCC(C(=O)NC(C)CNC(C1(C(C)(F)F)CC1)=O)c1ccccc1 N1(C(C(C=C)(C)C)=O)CC2CC(NC(=O)CCOc3ccc(F)cc3)CC2C1 C(=O)CCCC(C(=O)NC)N(C(C)C(=O)OC)C.C(C)(C)(C)OCC C(=O)(CCCCCn1cnnn1)N(CC(C)N(C(C(C=CCCC)O)=O)C)C N1(C(C(C=C)c2ccccc2)=O)CCN(C(=O)C(Br)=C(C)C)CC12CCC2 CC1CC(C(=O)N(C)CCN(C)C(c2cccc(C3(C)CC3)c2)=O)CCC1=O c1(OCC)cccc(C(=O)NCC(C)CNC(C2CCCS2(=O)=O)=O)c1 Cc1nc(C(=O)NCC2CCN(C(=O)C(C)c3ccon3)C2)c(Br)s1 C(=O)(C1=COCC1)NC1(C(=O)NCc2cn(C)nc2)CC(c2ccccc2)C1 N1(C(C2(CC)CCCCC2)=O)CCOCC(CNC(C2C=CCS2)=O)C1 c1(C(N(CCNC(=O)C)CC)=O)cc2cncc(C)c2s1.C(C)(C)CC.O CC1(C)CC(=O)N(CC(=O)NCCN(C(c2csnn2)=O)CC2CC2)O1 c1(C(N2CCC(C(C)NC(CN3CC(CC)C3)=O)C2)=O)ccnc2[nH]c(C)nc12 N1(C(C2CCC(=O)N2)=O)CCC(NC(=O)C(c2ccccc2)F)C(C(N)=O)C1 C1CCC=CCC1.CC(C)CCC=CC(=O)NC(C1CC=CCC1)C(=O)N.C1CC1 c1(OC)cnncc1C(=O)NC(C)C(C)NC(c1cccs1)=O Cc1ccc(CNC(=O)C=CC(C)NC(c2cncs2)=O)cc1 N1(C(c2cnc(OCC)nc2)=O)CC2CCC1C2.c1(C(=O)N)ccc(C)c(F)c1 c1(NCC2N(C(C(C)(C)Cc3ccccc3)=O)CCC2)ccn2nccc2n1 N1(C(C(=O)NCCSC)C2CC=CC2)CCCSc2ccc(F)cc21 N1(C(C#CC(C)(C)C)=O)CCCC2C1CCCN2C(=O)COCc1ccccn1 C(=O)(C(N)CCS(=O)(=O)NCc1cccc(C)c1N)OC C(C1C(C(=O)NCCCCN(C(=O)Cc2cccnc2)C)C1(C)C)=C(C)C N1(C(CCSCC)=O)CCC(NC(=O)C(C(C)C)n2cc(C)cn2)CC(C)(C)C1 C(=O)(C1CCCc2nncn21)N(CC(C)NC(=O)Cc1cccc(OC)c1)CC C(=O)(C1=C(C2CC2)N(C2CC2)C(=O)NC1c1c(I)ncn1C)OC C1(C(N(CCNC(c2coc(O)n2)=O)CCOCCO)=O)CCCCCC1 c1(OC)ccc(C2CN(C(=O)NCC(c3ccc(O)cc3)(C)C)CCO2)cc1 CC(C)CC(CC(C)C)C(=O)N1CCCN(C(c2cnc(S)n2C)=O)CC1 c1(NC(C(C2CCCOC2)N(C)Cc2ncco2)=O)ccc(F)cc1 C1(NC(Cn2nnc(C)n2)=O)CC(C)N(C(=O)C=CI)C1.C(=O)CC(C)(C)C Cc1cc(=O)cc(C)n1CCCC(=O)NCC1CC1.C(c1ccoc1)=CC=O CCC(C)(C)C(=O)NCC(N1CCN(C(c2cncnc2)=O)CC1)C(F)F N1(C(c2n(C)ccn2)=O)CC2(CCNC(=O)C(O)C3CCCC3)CCC1CC2 CC(CC#N)C(=O)NCCn1cnc(C(=O)Nc2cccc(CN(C)C)c2)c1 CC(CC(C)(C)C)C(=O)NCC(C)(CO)NC(=O)CCc1cc(Cl)cs1 C12CCC(C1)N(C(=O)C)C2.c1(C(=O)N)cnc(C(F)(F)F)nc1.c1ccon1 c1(OC)cccc2c1OC(C(=O)N(CC(=O)N=c1cc(C)o[nH]1)C)C2 C1(CN(C)C(C2(CF)CC2)=O)CCCN1C(=O)C(c1ccccc1)F n1(CC)cnc2c(NCC(=O)N3CCCO3)[nH]c(=NC3CC(C#N)C3)nc12 c1(CCCNCC2(C(F)F)CCC2)cc(Br)ccc1I C1(NC(C(c2ccccc2F)(C)C)=O)CCCC(NC(c2cccnn2)=O)CC1 CC1Cc2cccc(C(N3CCC(OCC4CCCO4)C3)=O)c2O1 C(=O)(C1CCCc2nccn21)NC(CC)CN(C(=O)Cc1c(C)nn(C)c1Cl)C c1(C(N2CC(CCC)N(C(C3CCNC3=O)=O)CC2)=O)n[nH]c2c(C)cccc12 c1(C(=O)NCCNC(c2cccc(Oc3ccccn3)c2)=O)ccc(O)nc1Cl c1(COC(C(C2CCC(CO)CC2)NC)=O)cc(Br)ccc1OC(F)F C1(C)COCCN(C(C2CC3(C2)CC3(F)F)=O)C1.C(C(=O)N)N(CCOC)C C1(CSCC#C)CCN(c2nnc(C3CC3)n2CCOC)CC1 C1(NC(COCCCC#C)=O)CCCCC1NC(=O)C(C)N.[SH](=O)(=O)CC c1(CCC(N2CC3CN(Cc4cc(Cl)cc(Br)c4)C3C2)=O)ccc2c(c1)OCO2 C=Cc1ccc(NCCCC(=O)NC2(n3cc(C4CCCC(C)C4)nn3)CC2)cc1 C1(C)(C(N2CC(C)C(NC(=O)CCc3nccs3)C2)=O)CC(=O)N(C)C1 C1(C)(C(N2CC(C)(NC(c3coc(Br)n3)=O)C2)=O)CNC(=O)C1 C1(C(N(CCC(=O)N(CCC(C)C)C)C)=O)CC12CCOC2 c1ccc(C(=O)N)cc1.C1(N(S(C)(=O)=O)C)CCCN(CC#N)C1.CC.CCO Cc1ccc(CC(=O)NCCCOCCN(C)C(C2CCC(C)CC2)=O)c(C)c1 C=C(C)CC(C(=O)NC(C)C(C)C(=O)OC)NC(c1cc(O)nc(C)n1)=O c1(CC(=O)NC2CC(NC(c3cc(F)cc(I)c3)=O)C2)cc(Br)ccc1O c1(CN2CC3(CC(C(=O)NC(CC=C)CO)C3)C2)cccc2[nH]ncc12 O=S(=O)(c1ccc(F)cc1Cl)NC12CC(NCc3ccc(O)cc3)(C1)C2 C1CN(C(c2ccc(C(F)(F)F)s2)=O)CC(C)(C)O1.CCC(C=O)NC(C)=O CC1CC(CNC(C2CCC(=O)O2)=O)CN1C(=O)COC.c1ccncc1 c1(C(=O)NC(CN(CC)CC)C)ccc(-c2cccc(Cl)c2)cc1 Cc1ccc(C=CC(=O)NCC2(O)CN(C(=O)C(N)=O)C2)s1 C1(CCCN(C(C)=O)CCO)(NC(=O)CC(c2c(C)noc2C)C)CCC(=O)N1 c1(C(=O)NCCCCC(C)NC(c2cnc(Cl)[nH]2)=O)ccnc2ncccc12 c1(C(N2CCCC(N(C(CC3(OC)CC3)=O)C)CC2)=O)cc2cccnc2s1 C1(C)(CC(=O)NCC(C2CC2)NC(C=CCCC)=O)CCCCC1 N1(C(c2c(OC)ncc(Br)c2)=O)CCC(NC(c2cc(C)on2)=O)C(C)(C)C1 N1(C(C(C2CCC2)OCC)=O)CC(C)CC1C(=O)NC(c1cc[nH]n1)C c1(CC(=O)NC2C(NC(=O)COC3CCOC3)C2)cn2ccsc2n1 C1(NCCC(C(=O)OC)C)CCN(CCOC)C(C)C1 C1(C(N(C2CCN(C(c3sccc3C)=O)CC2)CC)=O)CCCCN1N=O Cc1cc(N(C)C)cc(C)c1CC=O.N1(C(C)C)CCC(C(C(C)(C)C)=O)C1 c1(C(=O)NCC2CN(C(c3c(C)cns3)=O)CC2C)cc(F)c(F)c(N)c1Cl c1(-c2nccc(NCc3c(C)c(F)ccc3F)c2)ccc(C#N)c(F)c1F C1(C(=O)N)CC(=O)NC1(C)C.N1(CCNC(C2C(C)(C)CC2)=O)CCCCC1 c1(OC)ccc(CC(N2CCN(C(C3CCC(OC(F)F)C3)=O)CC2)=O)cc1 C(=O)(C#CCNC(=O)CCSC)N(CCCF)CC C(N=c1nc2scnc2c(NCC2CCCC(F)(F)CC2)[nH]1)C1(OCC)CCC1 CCC1=NOC(C(=O)NC2(CCNC(C3CCN(CC(C)C)C3)=O)CC2)C1 C(C)(C(C(=O)N1CCC12CCC2)NC(C1COCCC1C)=O)OC C1(NC(CC(COC)C)=O)CCC(O)CN(C(c2c[nH]c(=S)cn2)=O)C1 c1(CN2C(C(N(CCC#N)C3CC3)=O)CCC2)cc([N+](=O)[O-])ccc1Br N1(C(C=C(CC#C)C)=O)CCC(C)(O)C1 CC1CN(C(C23CC(CO)(C2)OC32CCC2)=O)CC2(CCN(C(=O)CO)C2)O1 N1(C(c2nc(OC)cc(OC)n2)=O)CCC2CN(C(C3CC3C)=O)CC12 C1(C(=O)NC2C(CNC(C(C)OCCCCCC)=O)CC2)(CO)CCCCC1 N1(C(C2=CCCN(C(C(OCC)OCC)=O)C2)=O)CCC2(CC1)CC2C#N N1(C(C(C)(C)SC)=O)CCN(C(C2CCCC(C)(C)O2)=O)C(C)C1 CCCCCCCCCC(=O)NC1(CF)CN(C(c2nccc3[nH]ccc23)=O)C1 C(=O)(CCCCCF)N1CC(O)(C(C)NC(c2cnc(CC(C)C)s2)=O)C1 c1(CNC(C(CCC)C)c2nnnn2CCCO)cc(F)cc(F)c1.C1CC1.C CCCC(=O)C(=O)N1CCC(C(N2CC(N)C(O)C2)=O)CC1 c1(C(N(CC(C)(C)Nc2ccc(-n3ccnc3)nn2)C)=O)ccc2nonc2c1 N1(C(c2c(C)nco2)=O)CCC2CC2(C(=O)NCC2(C)CCOCC2)CC1 CCC(C)CC(=O)C(=O)NC1(CNC(=O)CSC(C)(C)C)CC1 c1(OC)cc(C(=O)N(CC(C)NC(=O)CCC(=O)c2ccc(Cl)s2)C)cc(F)c1 Cc1ocnc1CCNC(=O)CCOCCNC(=O)C=CC(C)C N1(C(CC2(C)CC2)=O)CCC(OCCNC(=O)CCCNC2CCC2)C1 Cc1ncc(NC(C2CS(=O)(=O)N2)=O)cc1Cl C1CCN(C(c2cccs2)=O)CC1O.C1(CSCC(=O)N)C2CC3C(C2=O)C13 c1(C2C(C(=O)NC(CC)(C)CNC(C3CC(O)C3)=O)C2)ccc(Br)nc1 n1(CC)ncc(C#N)c1NC(C1CC(F)(F)CN1C)=O.c1cc(F)cc(F)c1 CC1CN(C(=O)CC2CC2(Cl)Cl)CC1NC(=O)CC(=O)NCC(F)(F)F C#Cc1c[nH]nc1C(=O)NCC(CC)NC(c1cc(C)no1)=O c1(C(=O)OC(c2ccccn2)CC#C)cc2n(n1)CCNS2(=O)=O C1(NC(C(C)OCCC=C)=O)C=CCN(C(c2cn(C(C)(C)C)nn2)=O)C1 C(CCN=C(NCCc1nccn1C)NC1CC(OC(C)(C)C)C1)OC C(=O)(CC(C)(C)CO)CC(N1CC(Cn2cc(C(C(C)C)O)nn2)C1)=O c1(CC)ncc(NC(=O)Cc2ccc(Cl)cn2)cn1 N1(C(CC(C)c2ccccc2)=O)CC2(CC(C(N3CCCOCC3)=O)CO2)C1 CC(C)CC(CNC(C1CCC12CCC2)=O)NC(c1ncccc1C(F)F)=O c1(C(=O)N)ccn(CCC(F)(F)F)n1.n1(C2(C(N(C)CC)=O)CC2)cnnn1 c1(CC)nncn1NC(=O)C1CN(C)CCN1C(=O)CC1COCC1O N1(C(C2CCCN(C(=O)C3CC3)C2)=O)CCc2cc(C(F)(F)F)[nH]c2C1 N=c1cc[nH]c(C(=O)NCC(c2nc[nH]n2)NC(C2(CO)CCC2)=O)n1 CC(CCN=c1cc[nH]cc1[N+](=O)[O-])NC(=O)Cc1ccc2n[nH]cc2c1 c1nc2nc(C)cc(C)n2n1.C1(CN(C(=O)C(=O)N)CC)COC(C)(C)O1 c1(C(N2CC(NC(CC(=O)NCC)=O)C(C)CC2)=O)ccc(Cl)c(F)c1N N1(C(C2(CC#C)CCOC2)=O)CC2CCCN(C(c3cc(O)ccc3F)=O)C2C1 C(=O)(C(C)(F)C(F)(F)F)NCC1CCCCN(C(CCCC#C)=O)C1 c1(OC)ccc(C(=O)NC23CC2CN(C(c2ccc(Cl)cc2)=O)C3)c(Cl)c1 C1(O)(C(=O)N)CCCOC1.C1(C)(C(=O)OC)CC(NC(C2CCCC2)=O)C1 C1(CNC(=O)CCOC2CCCC2)CCCN(C(c2ccc(F)s2)=O)CC1 C1CC(O)C(O)CC1C(=O)NOCC(O)CO.O=C1CC(C(=O)N)NC(=O)N1.C C=CCCCCCC(=O)NC1CCCC1NC(=O)C(C)OC1CCCCCC1 Cc1cc(C(=O)NC2CC3CCC2(NC(=O)Cc2ccoc2)C3)cc(N)c1Cl N1(C(c2ccc(OCCC#C)c(F)c2)=O)CCC2(NC(=O)C3=CCCS3)CC2C1 c1(C2C(NC(=O)NCCc3ccc4c(c3)CCC4)C2)ccnc2ccccc12 N1(C(c2nc(CNC(C3CCC(CC)O3)=O)oc2)=O)CCC(C(=O)O)C1C C1(CNC(C(CC)SC)=O)(C)CC12CCC2.C1(CC(=O)N)CC(F)(F)C1 C1(NC(=O)C(=C2CCCCC2)F)CCC2(CC1)CCN(C(=O)C1CC1)C2 C1(C(N2C3C(NC(CC(CC)C4CC4)=O)C(C3)C2)=O)COc2ccc(O)cc2O1 c1(C(N(C2CCCN(C(c3nc(C)n(C)c3)=O)C2)C)=O)cncc([N+](=O)[O-])c1 c1(C(N2CCC3(NC(c4cc(C)ncc4)=O)C(C2)C3)=O)sccc1S(N)(=O)=O N1(C(C2(C)CC2)=O)CCc2cc(F)c(F)cc21 C(=O)(CC(CO)CC(=O)O)NC(COc1cccc(C(=O)OC)c1)C N1(C(CCNC(C)=O)=O)CC(NC(c2c[nH]nc2-c2ccccc2)=O)C(C#N)C1 Cc1cc(COC(C)CCc2cnn(C)c2N)ccc1OCCO C1(C(N(CCOC)CCNC(=O)C)=O)CCCC(=O)N1C.c1ccccc1Cl C(=O)C1=C(Cl)CCC(C)C1.Cc1nn(C(C)C)c(C)c1CC(=O)NC1CC1.C CC1CN(C(=O)CC2CC2(C)C)CCC1C(=O)NC1C2CCCOC12 C1(NC(C(C)CC2CC2)=O)CC2CC1CN(C(=O)C=Cc1ccccc1)C2 c1(C(=O)NC2CC(O)C2)cncc(C#N)c1.C12(CC1)C(C)NC2=O Cc1nc(S(=O)(=O)N2CCOC3(CCSC3)C2)ccc1Br Cc1ccc(CNC(C2COCCN2C(c2ccc(NC=O)cc2)=O)=O)cc1F N1(C(COC(CC)C)=O)CCN(CCCCCNC(c2cscn2)=O)CC1 C1(C(N(C)CCN2CCCC2)=O)CC2CCCC2N1C(=O)CC1CC2C=CC1C2 C(=O)(C1=NOC(c2ccccc2)C1)N1CC(NC(c2c(C)cnnc2)=O)C(O)C1 C1(NC(C2(CC)CCN(C(C3CC4CC3CC4O)=O)C2)=O)CC(C)(O)C1(C)C C1(C(=O)NCC2CCN(C(CC(C)C)=O)C2(C)C)COC2(CCC2)CO1 C(=O)(C(C)CNC(=O)C(CO)NC(c1ccccc1)=O)OC C(=O)(C(C)(C)CC(C)C)N1CC2CC(CC)C2C1.c1(CC)nnc(N)nc1CC N1(C(C=CC(C)C)=O)CCC(O)(C2CCN(C(=O)CN3CCC(C)C3)CC2)CC1 Cc1c(Cl)ccc(C(N2CCC(NC(C3CCC(C)(C)O3)=O)C2)=O)c1N Cc1cc(SCC(=O)Nc2ccc(C)c([N+](=O)[O-])c2)n2ncc(C#N)c2n1 CC(C)C(C)C(=O)NC(c1cn(C)nn1)C(=O)N(C)C(C1CCOCC1)C C1(C(=O)NC(CCC)(C)C)COCCN(C(=O)CC2CCCN2C)C1 c1(C(=O)NC(CC)CNC(c2cc(C)nn2C)=O)ccc(C(C)C)nc1O N1(C(c2nccc(C)c2N)=O)CCC(O)(C2CCC2)CC1 c1(NC(=O)C(N2CCOCC2CC(F)(F)F)=O)nc2c(s1)COCC2 CCC(C)CC(=O)NC1(C(=O)N(C2CC(F)(F)C2)C)CCC1 N1(C(Cc2n(C(C)C)cnn2)=O)CC(NC(c2cnccn2)=O)CC1(C)C CC(C)CC(C)CC(=O)NC1CCC(C(=O)NCC2(C)CC3CCC2C3)C1 C1(C(N(C)CCOCCC)=O)CCN(C)C(=O)C1.C(=O)(C)N.CC(N)=O c1(C(=O)NC(CN(C(=O)C=CC(C)(C)C)CC)C)cc2sccc2s1 C1(NC(CCn2c(C)ncc2)=O)(C)CCCCC1.C1(CC(=O)N)CC(O)C1(C)C C1(CC)CN(C(=O)C(CC)C(C)O)CCC1NC(c1ncnn1C)=O CC(CC(=O)NC1CCN(C(C2(C)CC2)=O)C1)P(C)(C)=O c1(C(N2CCC(F)(C)C2)=O)ccc([N+](=O)[O-])nc1.C1(C=O)CC1.C1CC1.N c1(C(=O)NCC(CC)NC(c2cnc3[nH]cnc3c2)=O)cc2c(C)cccc2o1 C1(C(N2C(C(=O)NCC(CCOC)O)CCC2)=O)COC(=O)N1C C1(NC(CCCC=C)C2CC2)CCOC2(CCC2)C1 c1(C(N2CCN(C(=O)C=C3CCCCC3)C3C2C3)=O)c[nH]c2nccc-2c1 c1(NC(C2C(NC(CCC=C)=O)C2)=O)c(Cl)c(COC)nn1C c1(SCC(=O)NC2(C)CCN(C(C(CCC)C)=O)C2)nc2ccccc2[nH]1 c1(CC)cc[nH]c1C(N1CC(O)(C(F)C(=O)N(C)Cc2ccccc2)C1)=O c1(NC(C(c2ccccc2O)OC)=O)ncc(CO)cc1Br c1(OC)cccc(CC(N2CCC(C(N3CCC(C)(O)C3)=O)C2)=O)n1 Cc1c(NC(=O)Nc2ccc3c(c2)CCO3)ccc(F)c1N1C(=O)CNC1=O C1(C(=O)NC2CN(C(c3c(C)onc3)=O)CC(C)C2)CCC2(CCC2)CO1 C1(C(=O)NC2C(C)N(C(c3cnc(Cl)[nH]3)=O)CC2)Cc2ccccc2C1 C1(NC(C2CCC(C)O2)=O)CCC(C(=O)NCC(F)CO)CC1 Cn1nnc(C=CC(N2CC(O)(CNC(=O)CCc3ccccc3Cl)C2)=O)n1 N1(C(=O)CC2CCCS2(=O)=O)CCCC(C2CCN(c3ncc(O)cn3)CC2)C1 C(C(O)CC(F)(F)F)NC(C1(CC#C)CCN(C(=O)C(C)COC)C1)=O C1(CNC(C(COC)OC)=O)CN(C(c2ccc(F)cc2Cl)=O)CCCO1 C1CC2CN(C(=O)C(C)C(C)(F)F)CC12.C(CS(=O)(=O)NCC=O)OCC c1(CC(C(=O)N)=O)cccc(F)c1.CC(C)CCSCC(N1CC(CC)C1)=O n1(C2CN(Cc3ccc(CC)cc3)C2)ccc(=NC(=O)Cc2ccc(Br)cc2)[nH]1 c1(CC)cncc(C(N2CCC(NC(C3(C)COC(=O)C3)=O)C2C)=O)c1 C(=O)(C1CCCc2ccnn21)N1CCCC(CNC(COCCC(C)C)=O)CC1 c1(OC)cccc2c1C(C(=O)NCC1CN(C(c3ccns3)=O)CCO1)CC2 N1(C(CCNC(C)=O)=O)CCC2(CCCN(C(C3COC(C)C3)=O)C2)C1 N1(C(c2cc(CC)cc(N)c2)=O)CCN(C(C2CCOC2CC)=O)CC12CCC2 N1(C(C2CC3C(C)(C)C3C2)=O)CCCCC12CC(NC(=O)C=Cc1cnc[nH]1)C2 C(=O)(C1=CC(C)(C)C1)N.c1(OCC=C)ccccc1C(=O)NC(C)CCC C(c1cn[nH]c1)=CC(=O)NC1CC1CNC(=O)CN1CCCCC1 C1(CC)(CNC(c2cc[nH]n2)=O)CC(C)(C)C1.c1(C=O)cncc(C)c1.C CCCCS(=O)(=O)CC(=O)N1CC(NC(C2CC=CCO2)=O)CCC1C C1(N(C(CCOCC)=O)C)CCN(C(=O)C(CO)NC(C)=O)C1.C(N)=O CCC(CC)C(C)C(=O)NC(C)CC1CN(C(c2cnc(C3CC3)nc2O)=O)C1 c1(C(N(CC(=O)NCCCC(=C)C)CCOC)=O)ccncc1NC C(=O)(CCCC(=O)NC(C)(C)CNC(c1cc(C2CC2)on1)=O)OCC c1(CCC(=O)NCC=C(C(=O)N(C(CC)CC)CC(C)C)C)ncc(F)cn1 C(CC(C=O)NC(=O)C=CCN(C)CC)=CC.C1(CC)CC(C)(C)C1 c1(C(=O)OC)ncccc1S(=O)(=O)Cc1ccc2c(c1)C(=O)CC2 C1(F)(CNC(c2[nH]cc(C)c2)=O)CCCC1.c1(C(C(=O)N)=O)ccc(Cl)cc1 C1(CCNC(CN(C(=O)CC2(C#N)CC2)C)=O)C=NNC1=O Cc1ccc2nc(C)c(-c3nnc(N4CCOCC4)o3)cc2c1 C(=O)(C(CC(F)F)N(C(=O)CC1CC2(CC2)C1)C)NCCC1CCN(C)C1 c1(OC)cc(C(N2CCN(C(C3CCCO3)=O)C(C)C2)=O)ccc1OCC(N)=O c1(C(C(=O)NCc2ccco2)N(CC(CC)C)C)ccnc(OC)n1 C1CCCC(C(N)=O)C1.C1(C(N(C(C)C(=O)N)CC)=O)CCC(N(C)C)C1 C(=O)(CC(C)(C)N(C(=O)Cc1cnoc1)C)NC(C(C)(C)OC)C C=C(C)C(C)(O)C(=O)N1CCC1CNC(c1cncc(NCC)c1)=O N1(CCS(=O)(=O)NC(C)C)CCC(=O)N(Cc2cccc(C#N)n2)C1=O c1(NC(c2cccc(NC(CSC)=O)c2)=O)cc(F)cc(F)c1Cl C1CC2CC(C1)N(C(C1CC(=O)N(C(C)(C)C)C1)=O)C2.CC1(C=O)CCC1.N c1(C(=O)NCC2CCN(C(c3ccc(Cl)[nH]3)=O)C2)coc2c1C(=O)NCCC2 C(=O)(CS(=O)(=O)CC(=O)N1CCCCC1CN(C)C(C1CC(C)CO1)=O)OC CC(C)C(F)(CNC(=O)CNC(N)=O)C(=O)NCCC(O)CO CC(C)CN=C(NCC1CCCCC1)NCC1(C2CC2)CCC1 C1(C(C)C)CCN(C(c2cc(Cl)cn2C)=O)C(CNC(C2(C)CCCO2)=O)C1 C1(C(=O)NC2CC(O)C2)CC=CCN1C(=O)CN1CCCC1=O C1(C(=O)NC(c2ccccc2)CNC(C)C(=O)NC)CCC(=O)N2CCOCC12 N1(C(c2c(CC)nns2)=O)CC(C)(C)CC1CC(=O)NC1CC=CCC1 CC1CSCCN1C(=O)CC1CCCC(NC(c2cc(Cl)no2)=O)C1 c1(C(N2CC(C)C(CNC(c3cc(O)no3)=O)CC2)=O)nnc2ccccc2n1 C(=O)(C1=CC2(CCOC2)C1)NCC(C)N(C(=O)C(c1ccc(Cl)cc1)=O)C C(=O)(CC(C)CCC)NC(C(=O)NCC(=C)CC)(C)CSC Cc1cc(C(=O)NC(C)C(C)(C)C(=O)NC2CCS(=O)(=O)C2)cnc1C N1(C(C2C(OC)C2)=O)Cc2ccccc2C(C)C1.C(=O)(CS(=O)(=O)N(C)C)N N1(C(C2N(C)C(=O)CCC2)=O)CC2CCC1C1CN(C(C34CC(C)(C3)C4)=O)CC21 c1(C2C(C=O)C2)ccc2ccccc2c1.C(F)(C(=O)NCC1CCC1)=C(C)C C(=O)(C(C)(O)C(C)(O)C(=O)N1C(=O)NC(C)C1=O)OC.c1cc(Cl)cc(Cl)c1 CCCC(C)(C)CC(=O)NC1CCN(C(c2cnn3c2CCC3)=O)CC1CO c1(-c2nnc(N3C(CC)COCC3)n2CCC#N)cccc2cccnc12 CCC(C)CCCCC(=O)NC1(CNC(=O)CC2CCC(=O)NC2=O)CCC1 c1(CC(C(N2C(CC(N3CCC(OC)C3)=O)CCC2)=O)N(C)C)cccc(C)c1 C1(CC(=O)NCCn2c(CC)nnc2)CCCN(C(c2cncc(O)c2)=O)CC1 C(=O)(C1OCCn2ccnc21)N1CCC2(CN(C(C3OCC(C)(C)OC3)=O)C2)C1 N1(C(COCCC)=O)CCCC(C2CCN(C(=O)C(C)Cc3ccco3)CC2)C1 C#CCC(C)(C(=O)N1CCC12CN(C)C2)NC(C1CCCN1C(C)C)=O c1(N(c2c(C)ccc(C)c2)CCC#N)ccc(C)c(S(N)(=O)=O)c1 C(=O)(C(c1nccs1)N(CC(=C)C)CC)NCC=C C1(CC(=O)NC2CCC(CNC(C34CC(CO)(C3)C4)=O)C2)COCCO1 N1(C(CC(CCC)CC)=O)CCC(C2CCN(C(c3c[nH]nc3C)=O)CC2)CC1 N#CC1(C(=O)NC2CC2NC(=O)Cc2ccc(C(N)=O)nc2)CCOCC1 C1CN(C(C2CC3(CC3)C2)=O)C2(CCOC2)C1.C1(C=O)CCC(=C(F)F)CC1.N C#CCC(C)(CC)C(=O)N(CC(O)CNC(=O)COc1ccc(CO)cc1)C C1(NC(C(CC)C#N)=O)CCC2CCN(C(c3cc(C)c(C)cc3C)=O)C12 CC(CC(=O)NCC(C)CN)S(=O)(=O)c1ccc(F)cc1 N1(C(C(C)Sc2ccc(C)cc2)=O)CCCC(O)(CCNC(C2CC=CC2)=O)C1 C=C(C)CC(C(=O)N1CCC(CC)(CC)CC1)NC(=O)CCCC(OC)OC CC(F)(F)CCC(=O)NCC1(NC(C2CC23CCCOC3)=O)CCCC1 N1(C(CC2(COCC)CC2)=O)CCC2CC12.C1(C=O)CC1.C(C)C.C C(=O)(C(CNC(=O)C(C)(C)Cl)C(C)(C)C)NC(CCSC)CO c1(C(N2CCC(CCOC)(NC(=O)C(F)OC)C2)=O)cc(Cl)c(Cl)cc1N C1(NC(c2c(C(=O)OC)c(C)on2)=O)CCCN(C(=O)C2=CCCC2C)C1C CC(C)(O)C(F)(F)C(=O)NC1CCC1.c1(C=O)ccc(N)cc1.C(=O)C.C c1(CC(=O)N)nc([N+](=O)[O-])n[nH]1.CC1CCCN1CC(=O)NCCOCC c1(CC)c(C(=O)N(C)CCNC(c2ccncc2NC=O)=O)nn[nH]1.O c1(C=O)ccc(C2CC2)cc1.N1(C(C=CC(=O)N(C)C)=O)CC(CCC)C1.N CCCCC(C)(F)C(=O)N1CCN(C)C(C(N2CCC(OC)C2C)=O)C1 c1(C(=O)NCC(CC)NC(=O)CC2CCC(=O)N2)cnc(C2CC2)nc1C C(=O)(CC1=CCCC1)N(C1(C=O)CCC1)C1CC1.C(=O)(CC)NCC.C c1(CNC(C2(CC(=O)NC(C)C)CCCC2)=O)cc(O)ccc1F C1(NC(C(=O)N(c2nocc2-c2ccc(Cl)cc2)C)=O)CC2(C1)CC(C)C2 C=CC(CC)C(=O)NCC1(C(=O)NCCN2CCOC(C)C2)CC2(CC2)C1 c1(C(N2CC3C(CNC(COCC)=O)(CC3)C2)=O)cnc2sc(C)cn2c1=O Cc1cc(C(=O)NCC2(NC(C3CC4CCC34)=O)CCCC2)cn1C CC1CC(C)N(C(=O)CC2CCC2)CCN1C(=O)Cn1ncc(O)nc1=O N(C(=NCCCOC(C)C)NCC1CC1(F)F)Cc1c(C)nn(C)c1C c1(C(N2C3CC(CC3)C2)=O)cc(Cl)c(F)c(Cl)c1.C(C=O)=CC.C(C)OC.O c1(COc2cc(C)no2)nc(CCCc2ccccc2)nn1CC(N)=O c1(C(N2CCCC(CO)C2)C(=O)NC2CCCC2)cc(Br)cc(F)c1F C#CCC(C)(C)C(=O)NCC1(NC(=O)Cc2nn(C)cc2Br)CCOC1 c1(NC(CCC2N(C(CCC(=O)OC)=O)CCC2)=O)nc(C)c(Cl)cc1Cl N1(C(CCC=C)=O)CCC2(CCN(C(=O)CSC3CCCCO3)CC2)C(C)C1 n1(CC=O)ccc([N+](=O)[O-])n1.N1(C(C=C2CCC(C)C2)=O)CC2CC1(C)C2.N c1(CC(N2CCCC(C)C2)=O)ccc(S(C)=O)cc1.C1(CC=O)CC(F)(F)C1.N C(=O)(C(C)(O)C(F)(F)F)N1CCCC(CCC)C1.c1(CCC(=O)N)csc(C)n1 CC1CN(C(=O)Cn2ccnn2)CCC1CNC(=O)CCN1CCOC1=O C1(NC(C(C)SCC)=O)COCCN(C(C23CCC(F)(CC2)C3)=O)C1 C1(NC(=O)COC2CCOC2)CN(C(c2cc(=O)cc(Cl)[nH]2)=O)CCC1CO c1(OC)c(C(N2CCOC(CCCNC(=O)CSC(F)F)C2)=O)cc(F)cc1F N1(C(C2(OCC)CCC2)=O)CCCC(NC(=O)C(C)CCc2ccccc2F)C1 c1(NC(C2(CO)CN(C(CC3(C)CCC3)=O)C2)=O)cnc(O)c(C(F)(F)F)c1 C(=O)(C(C(CC)CC)OC)NC(CCCC)C(=O)NC1CCCN(O)C1=O C1(C)(NC(c2c(C#C)c[nH]n2)=O)CCN(C(C2(C)CCSCC2)=O)CC1 C(CC(=O)N)(C(C)C)OCC.C1(F)CCN(C(=O)C(N2CCNC2=O)C)CC1.C Cc1nc(N2CC(NS(=O)(=O)Cc3ccccc3)C3(CC3)C2)c2sccc2n1 c1(C(=O)NCC#CCNC(C2C(=C)C2)=O)cccc(S(=O)(=O)NC)c1 c1(OC)cc(CN2CCSCC2)ccc1-c1nc(-c2ncccn2)n[nH]1 c1(C(=O)NCC=C=C)cc(CNC(=O)C(C)N(C)C)cs1 N1(C(C2CCS(=O)(=O)CC2)C(=O)NC2(C)CC2)CC2(CCOCC2)C2CCCC12 C=CC(C)(CC)C(=O)NCC1COCCN(C(c2cccn2C2CC2)=O)C1 O=C(C1CCCn2nccc21)NCC1CCCCCN1C(c1ccc(CO)o1)=O c1(NC2C(CO)CC2)noc2c1COCC2 C=CCCCCCCNC(C1(C)CCN(C(=O)Cn2ncccc2=O)C1)=O c1(C(=O)NC(CC(C)NC(CN(C(COC)=O)C)=O)C)cc2nn[nH]c2cc1F c1(N(CCN(C)C(C2CC(F)C2)=O)C)ncnc2c1c(Br)nn2C CC1(C)COCC1C(=O)NC1(CCCNC(C2CCC2(F)F)=O)CC1 C1(C(=O)NCC(CNC(C2C(CC)C2)=O)C)CC2(C1)CC(O)C2 CCCCC(C(=O)NC1CC(CSC)C1)NC(=O)C=Cc1ccncc1 c1(CC(=O)OC)occ(C)c1C(=O)N(C)CCNC(c1csnc1C)=O N1(C(C2=CCCCC2C)=O)CCOC2(CCN(C(=O)CN(C3CCCC3)C)C2)C1 c1(C(N2CCC(C(C)C#N)CC2)=O)coc2c(Br)cccc12 CC(C)CS(=O)(=O)CC=O.C1CN(C(=O)CN(C)C=O)CC1C(F)(F)F.C c1(C(N(C2CCC(NC(c3ccc(CO)s3)=O)CC2)C)=O)ccc(O)c(Cl)n1 c1(C(=O)NC(C(OCC)OCC)C)cc(N2CCCC2)ccn1.CC CC1(C)CC(C(=O)O)N(C)C1.c1(C2CC2)ccc(OC(F)(F)F)c(OC(F)F)c1 C(C(C)(O)CNC(=O)Cc1cc(C2CC2)no1)NC(CN(C(C)C)C)=O Cc1ccc(C2(C(=O)N)CC2)c(F)c1.C(=O)(CCC(C)CN(C)C)N(C(C)C)C C(=O)(CS(=O)(=O)Cc1ccc(C#N)cc1)NCCN(C)C(c1scnc1Cl)=O C1(CNC(C2(C)CCOC2)=O)C2CN(C(c3sncc3Br)=O)CC12 c1(C(=O)NC(COCCCNC(CC(COC)C)=O)(C)C)ccc(F)cc1N CCCC(C)(O)CC(=O)NCC(C)(CC)C(=O)NCc1cc[nH]n1 CCC(CC)C(=O)NC1CC(C)(CNC(c2c(C)coc2C)=O)C1 N1(C(CCC(C)NC(C2CCCCCC2)=O)=O)CC(F)(F)CC1CO c1(C(=O)NCC2CC(C)N(C(C34CC(F)(C3)C4)=O)C2)cccc(F)c1F C(=O)(C(C)CC(=O)N1CCCC(NC(=O)CN2CC3CC3C2)C1)OC C#CCC(C)(C(=O)NOCC(C)C)NC(=O)CC(O)C(C)C N1(C(C2N(C(c3cc(C)nc(O)c3)=O)CC(=O)NC2)=O)C2CCC1CC(F)C2 C(C)(C)(C(=O)NCC=CCC(=O)NCC(c1ccco1)O)OC c1(C(=O)NC2CC(c3cn(C4CCC4)nn3)C2)ccc2[nH]c(=O)c(=O)[nH]c2c1.C C(=O)C1=NN(C)C(=O)CC1.N1(C(CC(C)C)=O)CC(F)(F)CC1CC.CC.S CCC(CC)C(=O)NCC(CC)N(C(=O)CC1CCCCC1O)C C1(CCNC(=O)Cc2ccsc2)CCCN(C(C2(C(F)(F)F)CC=CCO2)=O)C1 N1(C(C(CC)C2CC2)=O)CC(NC(c2csc(-c3ccc(C)n3C)n2)=O)C(C)C1 C1(C=O)CCOC(C)(C)C1.C#CC(CNC(c1ncoc1C)=O)CC1CC1 c1(CC(=O)N)ccc(S(N)(=O)=O)s1.n1(CC=C)cccc1C(=O)NCC CC(C)CN(Cc1ccc(C#N)cc1)N1CCOc2cc(F)ccc2C1 CC1CC(C(N2CC(O)(C3CC3)C2)=O)CN(C(C2(CO)CCCCO2)=O)C1 C(CCCCC(=O)N1CCC(O)(CNC(=O)C=CC(=O)N(C)C)C1)SC C(=O)(C(O)C(F)(F)F)NCc1ccc(C(N(C)Cc2ncco2)=O)nc1 CCC(C)(O)C(=O)NCCCNC(c1ccnc(OC2CCOC2)c1)=O CCCCC(CC(=O)NCC(C)(C)CN(C)C)NC(=O)C(C)(O)C(C)C C(CCO)(C(F)(F)F)NC(C1CCC(CNC(=O)Cn2cccc2)O1)=O C(=O)(C1CCc2c[nH]nc21)N1CCC(CCNC(=O)CSCC2CCCO2)CC1 C1(CC)CCCC2CC12.C1(C(=O)N)(CNC(CSCCC#N)=O)CC=CC1 Cc1ccc(C(N2CC(C(N)=O)C2)=O)c(N)c1.C(c1nc(C)cs1)=CC=O.C Cc1ccc(F)c(C(=O)N(CC(C)CNC(=O)C(C)CF)C)c1F C#Cc1cnc(C(=O)NCC(C)C2CC2)c(C)c1.N1(C(C(=O)N)C)CCNC1=O c1(C(=O)NC2CC(CNC(C(c3ccc(C)s3)C)=O)C2)cccnc1O N1(C(CCCc2scc(C)n2)=O)CC(C)N(C(=O)Cc2ccc(O)cc2)CC1C c1(CN2CC3CN(C(c4n(C)ncn4)=O)CC32)cc([N+](=O)[O-])cc(Br)c1O C1(C(N(CCNC(C2(C=C)CC2)=O)C)=O)(OCC)CCC(C(F)F)CC1 CC1(CNC(=O)CCCn2cc(-c3cnc(O)nc3)nn2)CCCCC1O Cc1cc(C)n(C(C)C(=O)NCC2CCCCN2C(=O)C=Cc2cncs2)n1 N1(C(c2c(C)c[nH]c2)=O)CCCC2(C1)CN(C(c1cccc(C)c1F)=O)C2 O=S(=O)(c1ccc(=NCc2ccnn2C2CCC2)[nH]c1)N1CCC2CC2C1 C(=O)(C1=CCCC1(C)C)NCC=C1CCN(C(C(C2CCCO2)OC)=O)CC1 CCC(C)C(O)C(=O)N1CCOCC1CCNC(C1(CC(F)F)CCOCC1)=O N1(C(CC2(C(=C)F)CCC2)=O)CCCCC(C)C1.N1(CC(=O)N)CCCS1(=O)=O CC1(C)OCC2CC12C(=O)NC12CC(C1)C2.c1(C=O)cc(C(F)F)ncn1 N1(C(c2nn(C)c(C(N)=O)c2)=O)CC2CCC1CN2C(c1cc(N)cc(O)n1)=O CC1=NOC(c2ccccc2)(C(N2CCC(C(F)(F)F)(CO)C2)=O)C1 N1(C(C=CS(CC)(=O)=O)=O)CCC2(CC1)CC(NC(C1CC1(C)C(C)C)=O)C2 Cc1nc(C(C)C)sc1C(=O)N.C1(C(N2CC(C(N)=O)C2)=O)CC1C1CCC1 Cc1cccc2c1OC(C(=O)NCCN(C(c1nc(Cl)cs1)=O)C(C)C)C2 c1(C(=O)NC(C2(O)CCCCC2)C(=O)NC(C)CSC(F)F)cncc(O)c1 CC1CC2CC2CC1C(N1CC(CNC(=O)Cc2ccc(F)c(F)c2)C1)=O C1(NC(C=Cc2c(C)ncs2)=O)CC2CC1N(C(C1(NC(C)C)CC1)=O)C2 c1(C(=O)NCCC(CC)(C)NC(=O)CC2CCC(C)O2)cccc2oncc12 c1(CC(=O)NC2C(C)N(C(=O)CCc3cn[nH]c3)CCC2)cnc2ncccn12 c1(C(=O)NC2C(NC(C(C)OCC=C)=O)C2)cc2cccc(F)c2s1 c1(C(=O)NCC(CN(C(CS(CCOC)(=O)=O)=O)C)C)ccnc2c1ncn2C CCCCCC(=O)N1CC(OC(=O)N(C)C)C1.c1(C(=O)O)cc(C(N)=O)co1 N1(C(C)=O)CCCC(C)(N(C(=O)C=Cc2c(C)nn(-c3ccccc3)c2C)C)C1 c1(C2(NC(N(C(c3ccccc3)C)C3CC3)=O)CC2)cc(F)cc(Cl)c1 Cc1cc(C(=O)NCC2(C)CCCC2)cnc1O.c1(C(=O)N)ccc2c(c1)CC2 C1(CC(N2CC(C)(NC(c3c(C)sc(Cl)n3)=O)C2)=O)SC2=NCCN2C1=O Nc1cc(C(=O)NC23CCN(C(C45CCC(CC4)CO5)=O)CC2C3)cnc1Cl C(=O)(C#CC1CCCC1)NC(CCNC(c1cc(SC)nn1C)=O)C C(=O)(C(F)(F)C1CC1)NC(C)CN(C)C(C1CC1C(F)(F)F)=O CC1(C)CC(C(N2CC(F)CC2CO)=O)CN1C(C1CCSC1)=O C(=O)(CCC(C)(C)O)N(C1CN(C(=O)Cc2cnco2)C1)C N1(c2c(C(=O)OC)cccc2)CCCC(NC(NS(=O)CC(F)F)=O)C1=O c1(NC2CC(F)(CNC(c3c(C)nsc3)=O)C2)nc2ccc(F)cc2o1 N1(C(CCc2onc(CC)n2)=O)CCC(NC(=O)C(C)C(O)CC)C(F)C1 c1(C(N2CCN(C(CC(CCC)(C)O)=O)CC2C)=O)cccc2c1ccn2C C(=O)(C1CCc2cccc(Cl)c21)N(C1C(C#N)CNC1)c1ncc(F)cn1 [SH](=O)(=O)c1cccc(F)c1.O=C(CCCC1CC1)NCC(CO)NC(=O)C.N CC(CCCNC(=O)C=CC(N)=O)NC(=O)CCC1CCCOC1 c1(C(=O)NC2CC2C)cccc(C2(O)COC2)c1.C1(C=O)C=CC=CC=C1 n1(CC(N2CC3C(NC(C(C)(CO)OC)=O)C3C2)=O)cnc2c(N)ncnc12 c1(NC(C2C(C(C)C)N(C(c3ccco3)=O)CC2)=O)ccc2c(c1)COC2 c1ccc2c(c1)CC2.C(CNC(=O)CCc1cn(C)cn1)(C(=O)N)N(C)C.C N1(CCC)CCC(C(N2CCCC2C(C)(C)NC(c2c[nH]nc2F)=O)=O)CC1 CC(C)C(O)C(C)C(=O)N1CCOCC(C(=O)NCCCN2CCCC2C)C1 N1(C(Cc2ccn(CC)n2)=O)CCC(CNC(c2scnc2C(C)C)=O)CC1 N1(C(CN=[N+]=[N-])=O)CC2C=CC1C(C(=O)Nc1cccc([N+](=O)[O-])c1)C2 c1(C(C2CCOC2)N(C(C)C2CC2)C)cn(C2COC2)nn1 C(c1c(Cl)cccc1Cl)=C(C)C(=O)NC(C1CCN(C(=O)CC(C)CF)C1)(C)C c1(CC(N2CCC(NC(C3(COC)CCOC3)=O)C2)=O)c(C)ncnc1C CCCC(CCC)=CC(=O)NC1CCC1C.c1(CC(C(=O)N)O)ccc(Cl)cc1 N1(C(CC(=C)C)=O)CC2CCN(C(=O)CC3CCCCC(=O)N3)CC2C1 C1(NC(c2n[nH]c(C)c2C)=O)CC2CC(NC(=O)CC3CC4CC4C3)CC12 C(=O)(C1=CCC(NC(c2cc([N+](=O)[O-])c[nH]2)=O)C1)N(C)CC1COCCO1 C=CCC(C(=O)N1CCCC(NC(=O)Cc2cn3ccsc3n2)C1)C(C)C C#CC(C)(C)C(=O)NC1CN(C(c2nc(O)sc2C)=O)CC1c1ccnn1C C1CCCN(C(c2cc(C(=O)C(F)(F)F)c[nH]2)=O)C1.C(CC)(C(=O)N)OCC C1(CNC(c2cnn(CC)n2)=O)CCN(C(C2C=CC=CC=C2)=O)C12CC2 C(=O)CC(F)(F)C(F)(F)F.N1(C(c2cnc(C(C)(F)F)s2)=O)CCC(O)(C)C1 C1(NC(c2c(OC)nsc2)=O)CCN(C(c2cc3cccn3cn2)=O)C12CCC2 N1(C(C2N(C)CCCC2)=O)CC2CC1CN2C(C1CCCC2(CC2)C1)=O N1(C(c2cc(C)n(C)c2C)=O)CCC2CCN(C(=O)CCC(CF)CF)CC12 C=CC1(O)CCN(C(=O)CCCn2cc(C3CCCOC3)nn2)C1 Cn1cnc(C(=O)NC2CC(CCNC(C3(C4(C)OCCO4)CC3)=O)C2)c1 c1(C(=O)NCC2N(C(c3c(C)ccs3)=O)CCC2)c[nH]cc(Cl)c1=O c1(CC)cc(N)c(C(=O)NC2CN(C(c3conc3C)=O)C3(CCC3)C2)cc1F N1(C(c2ccc(CC)cn2)=O)CC(NC(=O)Cc2c(C)cccc2F)C2(CC2)C1 Cc1cc(C(=O)NC2CCN(C(=O)Cc3ccoc3C)C(C)C2)cnc1O c1(N2CC(CC)OCC2)cc(N2CCOC(CC(C)(C)C)C2)nc(C(C)C)n1 O=C(NOC1CCOC1)C1=C(F)CN(C(c2ccc(O)cc2F)=O)CC1 CCCCC(=O)C(=O)N1CCC(CC(N2CC(S(C)(=N)=O)C2)=O)C1 C(=O)(C1=Cc2ccccc2C1O)NC(CN(C(c1nc(C)sc1C)=O)C)C C12(CNC(C3(NC(C)=O)CC3)=O)CCCCC1N(c1ncc(C#N)cc1Cl)CC2 C1(CC=C)(NC(c2nc(OC)ccc2C)=O)CCCN(C(C2CC(C)=NO2)=O)C1 c1(N(CCC)C=O)ccc(C)c(Cl)c1.c1c[nH]nc1-c1ccc(C(F)(F)F)s1.N N1(C(c2c(OC)c(C)cs2)=O)C2CCC1C1CC1C2.c1(CC=O)cc(C)no1.N N1(C(C(CCC)N(C)C)=O)CC(NC(C2CC2C)=O)CC2(CCC2)C1 Cc1nn(CC(=O)NC2CN(C(=O)C=Cc3cnc[nH]3)CC2C)cc1[N+](=O)[O-] C(CC)(C(=O)N1CC(OCCNC(c2coc(Br)n2)=O)C1)OCC C1(C(C)C)CN(C(=O)CC2CC2C2CC2)CCCN1C(c1cccn1C)=O N1(C(c2c(C)coc2C)=O)CC(C)CN(C(C2(S(N)(=O)=O)CCC2)=O)CC1C C(=O)(CN=c1ccc(Cl)n[nH]1)N1C2C(NC(c3c(CCC)occ3)=O)C(C2)C1 c1(C(N2CC(CNC(=O)CCOCC3CC3)C2)=O)cc(C2CC2)[nH]n1 C(=O)(C1CCc2c(Br)cccc21)NC1(CNC(CC(=O)NCC)=O)CC1 Cc1cc(O)n2ncc(C(N3CC4OCC(NC(=O)CC(C)C)C4C3)=O)c2n1 c1(C(N2CC3N(C(c4cc(C)c(Br)s4)=O)C3C2)=O)cn2c(Cl)cccc2n1 c1(C(=O)NC2CN(C(CC(C=C)CC)=O)C(C)C2)cc2cccn2cn1 N1(C(c2ncc(C)s2)=O)CC2CN(C(c3cccc(F)c3Cl)=O)CC12 C(=O)(C#CC1CCOC1)NCCCC1OCCN(C(C(N)=O)=O)C1 c1(OCC)cc(C=O)[nH]n1.c1(C=O)cnn(C(C)(C)C)c1.C1CC(CC)C1 N1(C(=O)CC2CCOC2)CCN(C(=O)CCc2nncs2)CC(CO)C1 n1(CC(C)C)ncc(C=O)c1C1CC1.C1(CC)CCCN1C(C1CCCS1)=O.N c1(C(=O)N)c[nH]nc1S(N)(=O)=O.CC1CCC1.n1(CC=O)cc(C2CC2)nn1 N1(C(C(C)C)=O)CCN(C(C2CCC(C)O2)=O)CC1CC#N c1(NC(c2nnc(C)o2)C)nc(=NCC2CCCSCC2)[nH]c2c(C)nn(C)c12 CC(C)(C)CC(C)(C)C(=O)N1CC2(C1)SCCC2NC(C1CCC(N=[N+]=[N-])C1)=O C1CCN(C(=O)CC2CC2)C1.C(CC(=O)N)OCCOCC.C(C)=O N1(C(CCCOC)=O)CC2(C1)OC1(CO)CC2C1.C1(C(=O)N)C2(CC2)C12CC2 C(=O)(C1=NN(c2ccccn2)C(=O)CC1)N(CCCNC(C1CC1)=O)CC N1(C(COC(C)=O)=O)CCC2(CC2C(=O)NCC2CCC2)C1 N1(C(C(C)(C)NCCCCl)=O)CCC(NS(C)(=O)=O)C1c1ccccc1 n1(CN(C(=O)C(=Cc2cscn2)F)C(C2CC2)=O)ccnn1.C1CCOC1.C N1(C(c2noc(CC)c2C)=O)CC(C)CN(C(c2nnc(S)n2C)=O)C(C)C1 c1(C(=O)NCCC2CCN(C(C(C)(C)N(C)C)=O)CC2)cccc2c1C(=O)CC2 CCCCCC(CC)(c1nnnn1-c1ccc(OC)cc1C)N(C1COC1)CC N1(C(c2n(C=C)nnc2)=O)CC2(C(N3CCCC(CCO)CC3)=O)CCC1CC2 c1(CC=O)ccc(O)c(O)c1.c1(C=O)cn(CCC2CC2)nn1.CC(C)C.N c1(C(=O)NCC(C)NC(=O)CC(O)CC2CC2)nccc2c1NCCC2 N1(C(C(C)NC(CC)(C)C)=O)C2CCC(C2)C1C(=O)N.c1cccc(F)c1.C N1(C(C(C)c2cccs2)=O)CCC(C)(CNC(=O)C(=O)Cc2ccccc2)C1 CC(CN(C)C)CCC(=O)NCC1CCCC1C(N1CC2CC1(C(F)F)C2)=O c1(COC(=O)Cc2ccns2)ccc(CC2CC2)s1 c1(C(N2C3CC(C3)C2)=O)ccc2ncnc(O)c2c1.CC=O.C(=O)(OCC)N c1(C(=O)NC(CCOC)CNC(C2CCC(F)(F)CC2)=O)ccc(C#N)cc1 CS(=O)CC(C(C)(C)C)NS(=O)(=O)c1ccc(Cl)s1 C1(C(=O)NCC2(C)CC(NC(CN3CC(C)(C)C3)=O)C2)CCCC1(F)F CC(C)CCCC(=O)NC(CCN(C)C(c1c(N)cccc1F)=O)c1cccs1 C1(N(C)C(c2cccnc2F)=O)CC2CCC(C1)N2C(C1CC(C)(C)C1)=O c12nccc(n1)C(=O)N2.C(C(O)CCC=C)N(C(C=CC(C)(C)CC=C)=O)C c1(N2CC(CO)(CO)C2)cc(F)c(I)c(Cl)c1 N1(C(=O)C(O)CN2CCCC2)CC2CCCC(C1)N2C(=O)CC(Cl)Cl N1(CC)CCCC1CNC(C1(CNC(c2ccc(F)s2)=O)CCCO1)=O Cc1ccc(Cl)c(C(=O)NCCCOCCNC(=O)C2=NOCC2)c1 C1(C)(C(=O)NCCOC2CCN(c3cc(C(C)=O)ncn3)C2)CCC(=O)NC1 Cc1cc(C2CC2)ncc1C=O.CCC(C)N(C(=O)CC1CC(C(F)F)C1)C.N c1(CCC(c2cccnc2)NCC(CC(C)C)OC)c[nH]c2ccccc12 C1(NC(CCn2ccc(C)n2)=O)CN(C(=O)C(C)c2cc[nH]n2)CCC1CO C1(NC(=O)NC(CC)C(=O)NCCc2ccns2)CCC(OC)CC1 CC1CN(C)C(=O)CN1C(=O)COC1CC(NC(=O)CSC(F)F)C1 C1(N(C)C(C2CCN(c3cnn(C)c3)C2=O)=O)CCCCN1C(C1CC(=O)N1)=O c1(OC)ccc(CCC(=O)NCC(F)CNC(C2CC(C#N)C2)=O)cc1OC O=S(=O)(c1ccc(NCC2(CCO)CC2)cc1Cl)NC(CCO)c1ccco1 C1(NC(c2ccoc2C(F)(F)F)=O)CCCC12CCN(C(C1(O)CCCC1)=O)C2 C(=O)(CCC(=O)NN(C)C)NCc1c(CN2CC(C)OC(C)C2)cccc1 N#Cc1ncc(Br)cc1Nc1ccn(-c2cc3ccccc3s2)c1.C1CO1.CO N1(C(CC(C)C)=O)CC2CC(C1)CN(C(=O)C=Cc1cccnc1)C2 C12(NC(c3nc(C)sc3)=O)CC1CN(C(c1ccc(C)o1)=O)C2.C1CCCC1.O N1(C(C(CCC)CNC(=O)COC(C)(C)CC)=O)CC2CCCC(O)C2C1 N1(C(C(C)=C(C)C)=O)CCC(C(=O)NC2CCOC(C)(C)C2)CC1(C)C C1(NC(C2(C)CC2)=O)CC2CCCC(C1)C2NC(=O)C1=C(Cl)CCCC1 C(CC(N)=O)(C(=O)NC1CCC2CCC1C2)NC(CNC(C(CC)C)=O)=O C1(CC(N2CC(NC(C(CSC)(C)C)=O)C(C)C2)=O)Cc2ccccc2C1 c1(C(=O)NC2CCN(C(CC(CC)SC)=O)CC2CO)cnc2[nH]nnc2c1 c1(OC(C)=O)ccc(CN2CCCC(C(C)NC(c3nccs3)=O)C2)cc1 CS(=O)(=O)CCCC(=O)N1CC2CC1CN2C(c1ncc(F)cc1F)=O C(C)(CCCC(=O)NC1C(=O)NCC1(C)C)NC(Cc1cc(C)nn1C)=O N1(C(C2(COC)CC(=C)C2)=O)C(CC(N2CCCC(O)C2)=O)C2CCCC12 Cc1c([N+](=O)[O-])cccc1S(=O)(=O)NCC1(F)CC(N)C1 CCCCCC(C)(C)CNC(=O)C(CC1CCC1)NC(C12CCC(O)C1C2)=O C=C(C)CC(C(=O)NCC(=C)CC)NC(C)=O.n1(CC=O)cc(C)cn1.N n1(CCOC)ccc(C(=O)NCC(C)C2CC2)n1.C1(C=O)COC(=O)N1.N C(CS(=O)(=O)CC(=O)NCC(C1CCCC1)NC(c1occc1C)=O)OC C1(NC(=O)CCc2cncc(O)c2)CCCCN(C(=O)C(=C2CCCCC2)F)C1 c1(C=O)ncc([N+](=O)[O-])n1C.C1(CNC(C2(C(C)C)COC2)=O)CCCC1.N C(=O)(CC(C)SC)NCC(COC)NC(=O)CN(C)C(N)=O C1(CNC(C2CC3CCC2O3)=O)C2CC1N(C(C1CC3C=CC1O3)=O)C2 C(=O)(CCC#Cc1ccccc1)N(C1CC(NC(C(C)OCC)=O)C1)C c1(NC(c2cccc(Cl)c2OC)c2n(CC)nnn2)ccc(C)c(Cl)c1 Cc1nc2cc(NC(=O)Nc3ccc(OCCO)cc3)c(F)cc2[nH]1 c1(C(N2C(CNC(CC3C(C)(C)OCC3)=O)CC2)=O)cc2ccccc2s1 C1(C#N)(C(=O)NCC(Cc2ccccc2)NC(C)=O)CCN(C)CC1 C(=O)(CCC(C(C)C)NC(=O)C=CC(F)F)N1CCCN(CC)CC1 C(=O)(C1CCc2nccn21)NCC(C)NC(c1csc(O)n1)=O C#CCC(C(=O)NC(C)C(C)(C1CC1)OC)C1CC1 C1(C(=O)NCCC(C)(C)O)CC(NC(=O)COC(C)(C)C)C12CCC2 c1(N(CC)Cc2cccc(OC)c2)cnc(C2=CCOC2)c(OC)c1 Cc1cccnc1C1(CNC(=O)NCC2CC2(Cl)Cl)CCC1 c1(C(=O)NC2CCC(NC(c3[nH]nnc3C3CC3)=O)C2)ccc2ccncc2c1 c1(OCC)ncc(C(=O)NC(C2CCN(C(c3cscn3)=O)C2)C)cc1Cl Cc1nc(C)c(CC(N2CCC(CNC(=O)C=CCN(C)C)C2)=O)s1 N1(C(=O)C=Cc2ccccc2)CCC2(CC1)CC2C(N1CCCC(CCO)C1)=O C1(CC)CCC(CNC(C2(c3cn(C(C)C(=O)O)nn3)CCCC2)=O)CC1 CC#CCCCC(=O)N(CC(=O)NCC(C)(O)C(=O)OC)C1CCC1 c1(C(C)NCC(O)CO)cc(Br)ccc1S(C)(=O)=O.c1ccc(CC(N)=O)cc1 C(=O)(C1(C)CCOc2ccccc21)NC(C)CC(C)NC(c1sccc1F)=O N1(C(C(C)(C)N2CCCC2)=O)CC2COCC2(C(=O)NCC2CC(O)C2)C1 c1(C(=O)NC2CCCN(C(C3C(CCOC)C3)=O)C2)cc(Cl)c(C)cn1 C1CCCN(C(=O)Cc2cnc[nH]2)C1.C(COC(C)C)(C(=O)N)NC(C)=O C1(CC#C)(C(=O)Nc2cnn(CC)c2)CCN(C(c2cc(OC)ns2)=O)C1 Cc1nnc2n1CCCC2C(=O)NC1CC12CC(NC(=O)CCC1CC1)C2 c1(OC)cc(OC)c(N)c(C(N2CCCN(C(C3CCCS3)=O)CC2)=O)c1 c1(C(=O)NCC2CCC(NC(CCc3onc(C)n3)=O)C2)c(Cl)ccc(C)c1N C12(NC(C(CC=CC)CC)=O)CCCCC1CN(C(=O)OC(C)(C)C)C2 c1(CC=O)ccc(F)cc1.C1(F)(CNC(COC2(C)CCC2)=O)CCC1.N N#Cc1ccc(NC(C2CC(F)CN2C(=O)C2=COCCC2)=O)cc1C#N N1(C(Cn2ncc(C#C)c2)=O)CCC(C)(C)CC1C(N1CC=C(COC)CC1)=O C1C2CN(C(=O)CCCc3nc(C(C)(C)C)no3)CC12.C(C=O)OCCOC C1(C(N(C2CCCN(C(C3(c4cc[nH]n4)CCC3)=O)C2)C)=O)CCNC(=O)C1 C1(O)(C(C(=O)NCC(CC)N(C)C)NC(c2sccc2C)=O)CCCCC1 c1(C(=O)NC2CC(CNC(C(CC)(C)CO)=O)C2)cc(C)cc2c[nH]nc12 c1(C(N2CCCC(C)C2CNC(C23CC(CO2)C3)=O)=O)[nH]nc2ncccc12 C(=O)(C1=CCC(C)CC1)N1CC(CNC(c2cc(C)sc2)=O)N(C)CC1 C1(CC(=O)N)CCCC(C)(C)O1.Cc1ccncc1CC(=O)NCC1COCC1 N1(C(C(CSC)O)=O)CC(CCNC(c2cnn(CCO)c2C)=O)C(C)C1 C1(C(C)C)CCCC1NC(=O)CCN(C(=O)CCCn1cncn1)C1CC1 N1(C(c2onc(CC)c2C)=O)CC(F)(F)CC1(C)CNC(C1CSC1)=O C1(NC(CSCC(N)=O)=O)CN(C(c2cc(N)c(F)cn2)=O)CC1C1CC1 C(CC(=O)N=c1c(Cl)c[nH]cc1Br)C1(C)CN(S(c2c(C)cc(F)cc2)(=O)=O)C1 C1(C(=O)N)CCn2nccc2C1.C1(CC)CCN(C(C2CCC2)=O)C1.C(C)(C)C C1(CNC(C2(C)CC(=C)C2)=O)CCC(C)N(C(c2ncccc2SC)=O)C1 C1(CC)CN(C(c2coc3c2CSC3)=O)CCC1NC(=O)C=CC1CC1 N1(C(c2c(C(C)C)n[nH]c2)=O)CCCC2(NC(=O)CC3CCSCC3)CC2C1 CC1CN(C(=O)CN2CC(C)(C)C2)CC(C)N(C(c2cccc3occc23)=O)C1 CC1CCC(C)(NC(C2CC(O)CN2C(C2CN3CCC2C3)=O)=O)C1 C(=O)(C(CC)CCOC)NCc1c(C(=O)NCCCOCCCC)n[nH]c1 CC(C)(C)C#CC(=O)NC1CCN(C(c2ccc(OC(F)F)cc2)=O)CC1 CC1(NC(c2[nH]ccc2CNC(c2cccnn2)=O)=O)CCOC1=O c1(C(=O)NC2CCN(C(C(F)=CC)=O)C(C)C2)ccc2snnc2c1 CC1=NOC(=O)C1CCC(=O)NCC1CC(O)C1.c1(CC=O)ccoc1.C N1(C(C2C(CC)C2)=O)CC2CCC(C1)N2C(c1coc(Br)c1)=O N1(C(C=C(CC)C)=O)CC(NC(c2cnn3c2CCCC3)=O)CC12CCOC2 C1(C(=O)NCCCC(=O)NO)(COC)C=CCN1C(C1CCC(O)CC1)=O C1(CCNC(c2ccc[nH]2)=O)CCC(n2cc(CCOc3ncccn3)nn2)C1 C1(CCCN(C(=O)OCCOCCOCCOC)C)CC1C Cc1cncc(C(=O)NCC2(C)CCC(NC(=O)CCc3ccnn3C)C2)n1 N1(C(c2c(C)n[nH]c2)=O)CC(F)(F)CC1C(N1CCC(CO)C1)=O O=S1(=O)CCC(NC(=S)NCC2CC23CC3)C1 c1(C(N2C3C(CNC(CS(N)(=O)=O)=O)C(C3)C2)=O)cc2c(F)c(F)ccc2s1 O=c1onc(-c2cccc(C(F)(F)F)c2)n1CCc1ccncc1 N1(C(C(=Cc2cccs2)C)=O)CCC2(CCN(C(=O)Cn3ccccc3=O)C2)C1 c1(C(N(C2CN(C(=O)CC3CC(F)C3)C2)C)=O)cnc(C(F)F)s1 c1(C(N2CC(NC(c3ccc(I)c(O)c3)=O)C(F)C2)=O)cnc2snnc2c1 Cc1cc([N+](=O)[O-])ccc1C(N1CC(C)CN(C(c2cnoc2C)=O)CC1C)=O C(=O)(C#CC1CCOC1)NCC(C)(C)CNC(C1CC2(CCC2)C1)=O c1(CN(C(C(=O)N(CC(F)(F)F)CC)C)CC(=O)OC)ccccc1 C1(N(C(=O)CCCC2CCC2)C)CCCC(N(C(=O)CCc2ccsc2Cl)C)C1 Cc1cc(C)c(C(=O)N(C)CC2CN(C(C3(C#N)CCC3)=O)C2)cc1Br c1(C(=O)NC2C(NC(c3c(C)nc(CO)o3)=O)COC2)cc2cccnc2s1 c1(C(N2C(C)CC(CNC(CCC(C)(C)OC)=O)C2)=O)ccc2ncn(C)c2c1 N1(CC(=O)NC2(CCCNC(C3(CC)CCOC3)=O)CC2)CCCCC1C N1(C(=O)C2=CCCC2)CCN(C(C2CCS2(=O)=O)=O)C2COCC12 c1(C(N2CC(O)(CNC(c3c(C)snn3)=O)C2)=O)c(N)ccc2nccnc12 N1(C(CC(C)c2ccco2)=O)CCCCC1CN(C(=O)C(=O)NCC(F)(F)F)C C(=O)(C(C)(C)CC(C)=O)N.N1(C(C2N(CC)C(=O)CC2)=O)CCC(C)(C)C1 C=CC1OCCC1NC(=NCc1cccc(C)c1)NCc1cccc(C(F)F)c1 C1(OC)CN(C(=O)C(F)F)CC1NC(c1ccc(CO)cc1)=O c1(C(N2CC(NC(=O)CC(O)C3CC3)CC3(C2)CC3)=O)cccc2c1OCCO2 C(=O)(C1=C(F)CN(C(C2C3COCC23)=O)CC1)N1C2(C(=O)OC)CC2CC1 Cc1cc(O)ccc1C(=O)NC1CCN(C(=O)CC2CC3(CC3)C2)CC1C c1(CC(CO)NC(=O)NCc2nc(CC)oc2)cccc(C)n1 C(=O)(C(C)CC(F)(F)F)NC1CC(C)N(C(c2cc3c(o2)CCCC3)=O)CC1 C(=O)(CCCCCC(C)(C)C)NCC(C(C)C)NC(=O)Cc1ccc(Cl)cc1F C12CC(CN1C(C1CC1c1ccccn1)=O)C2.c1(C=O)ccc(C2CC2)s1.N CS(C)(=O)=NC(=O)C(=O)N1CCC(F)C(NC(=O)Cc2ccc(F)c(F)c2)C1 Cc1ccc(C(N2CCC(CC(C)NC(C34CC(C3)C4)=O)CC2)=O)c(N)c1C CCC(O)C(C)(C)C(=O)NCCCC(O)C(=O)N1CC(CCOC)C1 c1(C(N2CCN(C(=O)C(F)C(F)(F)F)C3CCC23)=O)cc(F)c(F)c(O)c1F c1(C(N2CCC(Br)C2)=O)cc(O)c2ccc(-c3cnc(NC4CC4)nc3)cc2c1 N1(C(C2N(C(=O)NC)CCC2)=O)CCC(NC(C2CC(C#N)C2)=O)CC1 C1(C)(CCC)CCCN(C(=O)CSCCC(C)C)C1.c1cc(Br)ccc1C(=O)N C(=O)(C(CNC(=O)CS)C)NCC1(COC)CCC1.c1nc[nH]n1 N1(C(c2c(CC)nc[nH]2)=O)CC2(CNC(=O)CCc3cc[nH]n3)CC1CO2 C1(C(N2CC(F)C(F)C2)=O)CCOCCN1C(c1cnn(C2CC2)c1)=O CCCCCC(O)C(=O)NCC1C2CC1N(C(c1ccc(F)c(N)c1)=O)C2 C1(N(C(C2C(C)C2)=O)C)CCC2(CC1)CCN(C(=O)C=Cc1cccnc1)C2 C1(NC(C2C(=C)C2)=O)CC(O)CN(C(c2c(-c3ccsc3)noc2C)=O)C1 CC1CCCC1CC(=O)N(CCCNC(=O)C(C)(C)n1cnnn1)C1CC1 N1(C(c2nc(CNC(=O)Cc3ccon3)oc2)=O)CC(C2CC2(F)F)C1 c1(CN2CC3(CC(C(N(CCCCC=C)C)=O)C3)C2)cn2ccccc2n1 CC1OCCCC1C(=O)NC(C)(C)C=CC(=O)NCCC1(O)CCCCC1 Cc1ccc(F)c(-c2csc(NCc3cncc(C#N)c3)c2)c1O N(C(=NCCc1ccccc1)NCc1cccc(Cl)n1)C1C(C)CN(C2CC2)C1 C(CNC(=O)C(C)OC1CCCCC1)(CC(C)C)NC(C1(SC)CCC1)=O c1(OC)ccc(CCCC(=O)NCC(C)(C)NC(C23CCCC2CC3)=O)cc1 C1(CNC(c2nc(CCC)sc2)=O)CCCN(C(c2cccnc2F)=O)CC1 CC1CC(NC(=O)CCN2CCCCCC2)CCN1C(=O)C1=CCCS1 c1(C(=O)NCC(C)CN(C)C(c2cnn(C)c2N)=O)cccc2cccnc12 c1(C(=O)NCCCCCN(C(C23OCC(CC)(C2)C3)=O)C)n[nH]c2c1CSCC2 n1(CC)cnnc1C(=O)NCCCCNC(C1CCCC1CF)=O C1(C(N2CC(OC(C)=O)C2)=O)(CC)CCN(C(C2CC2C2CCC2)=O)C1 c1(OC)ccnc(OC)c1C(=O)NCCNC(=O)CCC1CCCN1C O=C(CC1COc2cc(O)ccc21)N1CCC(c2cn(CCCCO)nn2)C1 N1(C(c2c(C)cccc2)=O)CCCC(C)C1CNC(=O)Cn1cnc(Br)c1 Cc1ccc2nc(N3CCC(O)(C(C)NC(c4cc(Cl)sc4Cl)=O)C3)sc2n1 C1(CC(=O)N(C2CCCCCC2)CCNC(C(C)(Cl)Cl)=O)CCCC(=O)N1 CCCC(CCCNC(C1CCCCN1C)=O)NC(C1CCCCN1C)=O c1(C(C(=O)NCc2cccs2)N(CCC#N)CCOC)cc(C#N)cs1 c1(C(=O)NC(CC)CN(C(=O)CC(C)c2ccncc2)CC)c[nH]cc(C)c1=O N1(C(c2cn(CCC)nn2)=O)CCC2CC(CNC(=O)C(C)CSC)CCC2C1 N1(C(CCC=C)=O)CCC(C2CCCN2C(=O)C2=C(C)CC2)CC1 CCC(C)CC(C(=O)NCCC1CC=CC1)NC(=O)CP(C)(C)=O c1(CC(N2C(CN(C(C(C)c3ncco3)=O)C)CCC2)=O)ccc2occc2c1 C(=O)(C(O)C1=CCCCC1)NC1C2N(C(CSCCCC)=O)C(CC2)C1 N1(C(Cc2c(C)n[nH]c2)=O)CCCCC1CNC(c1cn(C2CC2)cn1)=O CC(C)(C(=O)NCC1CCCC1)c1ccncc1.C(=O)(C(C)(C)c1ccsc1)N c1(C(=O)NC(CNC(c2c(CC)ccs2)=O)CC(C)C)c(F)ccc(F)c1N c1(NC(CCNC(c2c(C)nc(Cl)cc2)=O)C(C)C)ccnc2ncnn12 c1(NC(c2scc3c2CCCC3)=O)cc(Cl)c2c(c1)OCO2 CCS(=O)(=O)c1ccc(CCC(=O)NC2CN(C(=O)C(C)OCOC)C2)cc1 C(c1ncccc1C)=CC(N1CCC(N(C(=O)CCOCC)CCC)C1)=O N(C(=NCCSC)N1CCC(O)CC(C)(C)C1)CC1CN(C(=O)OC)C1 C12(C(NNC(c3c(N(C)C)ncnc3)=O)=O)CC3CC(C1)CC(O)(C3)C2 N1(C(C2(C)CC(C)OCC2)=O)CCC2(CC1)COC(C)C2.C(=O)(C(=O)N(C)C)N N1(C(C(CCC)C)=O)CCCC2(CCN(C(=O)COc3cccc(Cl)c3)C2)C1 c1(C(N(C2CN(C(=O)C(CO)c3ccccc3)C2)C)=O)sc(N(C)C)nc1Cl C1(C(=O)NCC2C(CNC(=O)CCCc3ccccn3)C2)CCCCCCC1 N1(C(c2[nH]cc(CC)c2)=O)CC2OCCN(C(=O)COC(C)=O)C2C1 c1(C(=O)NC(C2OCCN(C(c3ccc(C)nn3)=O)C2)C)nc2c(s1)COCC2 c1(OC)cccc(C(=O)NCC2CCCCN(C(=O)CCC3CC3C)C2)c1OC CCC(CC(=O)NCCC1CC(=O)N(C)C1)NC(c1c(C)cnn1C)=O C1(C(C)C)CC(O)CN1C(C1CCC1NC(C1CC(=O)CCO1)=O)=O c1(OC(C)C(=O)NCCC2CC(NC(=O)CNC=O)C2)cccc(Cl)c1Cl C1(NC(c2nccc(OCCC)c2)=O)CN(C(=O)C)CC1(C)C.C1CCCC1.O Cc1cnc(NC2CCCCC2CNC(c2cnoc2C2CC2)=O)nc1O O=C(COC1CCC1)NOCCCC1CC1.C12CC(C1)NC2=O C(=O)(C(CC(C)(C)C)NC(=O)Cn1nnc(C)n1)N(CCC(N)=O)CC N1(C(C2CN(C)CC(C)O2)=O)CCC(NC(C23CC2C3)=O)C12CCCC2 c1(CC(N2CCOCC(NC(C34CCC3CC4)=O)C2)=O)coc2cc(O)ccc12 C12(CNC(CC3CCCC(C)C3)=O)CCCCC1N(c1nc(Cl)c(C#N)s1)CC2 Cc1csc(C(C)C(=O)NCC2(NC(=O)CCC3CC3)CC2)n1 C=Cn1ccnc1C(c1nnnn1Cc1ccco1)NC1CC(C(N)=O)C1 c1(CNc2cc(-c3cnc(OCCC)c(F)c3)ncc2)n[nH]c2ccc(C)cc12 C1(NC(CCSC)=O)CN(C(C2CC23CCCCCC3)=O)C2(CCC2)C1 N1(C(c2c(C)onc2)=O)CC(NC(=O)CSCc2cccs2)C2(CCC2)C1 CC1CC(NC(C2CCCCNC2=O)=O)CN(C(=O)Cc2c(Cl)cnn2C)C1 n1(CC)cnc2[nH]c(=NCC3CCC(O)C3)[nH]c(=NC3CCC(C4CC4)CC3)c12 c1(C(=O)NC2C3CN(C(C4(C)CC4)=O)C2C3)c[nH]c2c(C(N)=O)cccc2c1=O c1(C=O)ccc(S(N)(=O)=O)cc1.C(CC)(C(=O)NC1(C)CC1)OCC C(C(CC(C)C)C(=O)NC1CC2C(O)C(O)CC12)NC(C(CC)(C)O)=O C1(C(=O)NCC(C=C)O)CCN(C(c2cc(C)n(CC)n2)=O)C12CC2 C1(C2CCOCC2)(C(=O)NCC2(NC(C3CCCC3)=O)CCOC2)CCOCC1 CCCCC(CNC(C1CSCC(=O)N1)=O)NC(c1coc(CCO)n1)=O.C C(C)(C(C(=O)NCC(O)CC1CCC1)NC(=O)Cc1ccns1)OC C#Cc1ccc(C(N2CC3(NC(=O)C(C4(O)CCCC4)F)CC2C3)=O)c(F)c1Cl C(CCC(C)(C)C(=O)NCCC(C)CCO)NC(c1cncc(OC)c1)=O C1(C2CC2)(CNC(c2c(OC)cccn2)=O)CCN(C(=O)C(C)CC(C)C)C1 c1(C=O)cc2c(F)ccc(F)c2[nH]1.Cc1cc(CC(=O)NCC2CC2C)no1 S(=O)(=O)(C1CC2C(C1)C2(F)F)NCCN1C(=O)c2ccc(Br)cc2C1 CC(C)CC(C)C(=O)NC(C)(C)CCC1CCN(C(C2CC3CCC2O3)=O)CC1 Cc1c(C(=O)NCC2CCCCN(C(=O)CCC3CCOC3)C2)cc(N)cc1O c1(OC)cccc(C(N2CCOC(C(C)NC(c3n[nH]c(C)c3O)=O)C2)=O)c1C C1(NC(CCCSC)=O)CCN(C(=O)Cc2ccc(Cl)c(Cl)c2)C(C)C1 C1(CC#N)NC(=S)N(CC2CCCC3(CC3)C2)C1=O CC1CN(C(c2cccnc2N(C)C)=O)CCCN1C(c1csc(C(F)F)c1)=O C(c1ccc(C)cc1)=CC=O.c1(OC)oc(C)nc1C(=O)NC1CC1C c1(CCC(=O)NC2CCCCN(C(C34CCC3C4)=O)C2)cccc(F)c1F c1(C(=O)NC(C2(O)CCN(c3ccnc(Cl)n3)C2)C)cc2cccnc2[nH]1 c1(NC(N2CC(CN)OCC2)=O)ccc2c(c1)OCC(=O)N2 c1(OCC)cc(CC(=O)NCC(c2ccc(C)cc2)(C)C)ccc1C N1(C(c2c(C#N)nc[nH]2)=O)C2CCC1CN(C(=O)CN1CC=CC1)CC2 c1(CC)cncc(-c2cn(C(C)C(=O)NCc3cccnc3)nn2)c1.C(C)(C)O N1(CC)CC(C(N2CCC(C(=O)NOC(C)C)(CO)C2)=O)CC1=O C1(C(=O)NCCCN2CCN(c3ncccn3)CC2)(CN)CCC(F)(F)CC1 C(=O)(CCCCN=[N+]=[N-])N(CC(C)C)CC(=O)NC1CCCCCC1F N1(C(CCOCCCOC)=O)CC(C)OC2(CCN(c3ncc(Br)c(C)n3)C2)C1 N1(C(c2ccc(Cl)c(OC)c2)C(=O)NC)CCc2cc(Cl)c(F)cc21 c1(C(=O)NCCCC(C)NC(C2N(CC)CC2)=O)cc2n(n1)CCCC2=O Cc1ccc(Cl)c(F)c1C(=O)NCCC1(O)CCN(C(C2CCOC2C)=O)CC1 C1(CCC)CN(C(C2CC(C)=NO2)=O)CCN1C(=O)CCc1ccc(SC)cc1 C12(CNC(C3CCCCCO3)=O)CCC(F)(CC1)C2 c1(OC)cc(C#N)ccc1OCC(=O)OCC(=O)NC1(C)C=CCC1 CC1(C#CC(=O)NCC2CCCN2C(=O)C=Cc2cccc(C#N)c2)CCCO1 C12(C(=O)OCC)CN(Cc3cn(CCC(=O)OCC)nn3)CC1(C)C2 c1(CCC(=O)NC(CCN(C(c2cc(C)ns2)=O)C)(C)C)ccccc1C#N N1(C(C2OCCN(C)C2)=O)CCC2CCN(C(c3cnc4n3CCOC4)=O)CC12 C=CC1(CC(=O)N(C)Cc2ncc(C)o2)CN(C(=O)CC2CC3(CCC3)C2)C1 C1(C(=O)NC2CCC(C(=O)NC(COC)C(C)C)C2)CC(=O)CCO1 C#Cc1cc(NC(C2CC2CNC(=O)CC2CCCCCC2)=O)ccc1C N1(C(C2(CC=C)CCOCC2)=O)CC2CN(C(C34CC(CC)(C3)C4)=O)CC2C1 CC1CN(C(=O)OC(C)(C)C)CC1(c1nn[nH]n1)NCCC(N)=O CC(CC1CCCC1)C(=O)NCCN(C)C(C1(C)CC1(Cl)Cl)=O c1(C(=O)NCC=C2CCN(C(=O)C3=COCC3)CC2)ccc(F)cc1F c1(NC(N2C(C(=O)NCCc3ccccn3)CC3CC32)=O)cc(O)cc(F)c1 C1(C(=O)NCC(C(CC)CC)O)CC2CCCC2N1C(c1cnc(C)o1)=O c1(C2N(C(c3n[nH]c(C)n3)C(=O)NC)CCC2)cccc(C)c1C C(=O)(C#CC1CCCCO1)N(C1CC2CN(C(CC(CCC)(C)C)=O)C1C2)C C(=O)(C1=C(Cl)CCOC1)N1C(C)(CNC(=O)C(c2ccccc2F)O)CCC1 c1(OC)ccc(C)c(OC)c1C(N1CC(CC(C)NC(=O)C(C)CS)C1)=O C(=O)(N1Cc2ccccc2CO1)C1C(C)CN(C(c2n[nH]cc2Cl)=O)C1 CC(C)CS(=O)(=O)CCC(=O)N1CCC2CCCC(C1)N2C(=O)CC(C)N(C)C c1(C(=O)NC(C)CCN(C(=O)CC2(O)CCC2)C)cccc(P(C)(C)=O)c1 c1(NC(c2[nH]c(C)c(C(=O)NC(C3CCOC3)C)c2C)=O)ccc(C#N)cc1O c1(CNC(CSCCC)=O)cccc(NC(=O)Cn2ncn(C)c2=O)c1 c1(CC(=O)NC(C)C=CC(=O)N(CC(F)Cl)C)cc(F)ccc1F C#CCC(O)C(=O)NC1COCCC1NC(=O)Cc1c(C(F)(F)F)coc1C c1(C(N2C(CC=C)(C(=O)NCC(C)(C)C(F)F)CCC2)=O)coc2ccccc12 Cc1cn2cc(C(=O)NC3CCCN(c4cccnc4)C3)sc2n1 N1(C(C(CC)(C)C)=O)CCN(C(c2ccc(O)cc2Br)=O)C(CC#N)C1 N1(C(CN(CCC)C)=O)CCC2C(C(=O)NC(C3CCCO3)CO)C2C1 c1(NC(C(C)N(C(=O)C(C)C(F)F)C2CC2)=O)ccc2occc2c1 N1(C(c2c(C)nn[nH]2)C(=O)NCC2CC2)CCS(=O)(=O)CCC1C CCC1C(=O)Nc2ccc(C(=O)N(C(C)CNC(c3cc(F)cs3)=O)C)cc21 C1(C(=O)NCC(C)(C2CCC2)NC(C=CCC)=O)CCS(=O)CC1 c1(C(N(C2CC(NC(=O)CP(C)(C)=O)C2)C)=O)ccc(N)cc1F CC1COCCC1C(=O)NCCCNC(=O)CN(C)Cc1ccc(Cl)s1 c1(C(C)C)cccc(C(=O)NC2CCOCC2NC(=O)Cn2cnnn2)c1 C(=O)(CC(C)(C)COC)N1C(CCNC(C2C(CCC)C2)=O)COCC1 N1(C(c2c(C)cns2)=O)CCCC12CCN(C(c1cnn(C)c1Br)=O)C2 C1(C(=O)NCC(c2ccccc2)NC(c2cc(Cl)no2)=O)CC(F)C(=O)N1 C1(NC(C(c2cccc(Cl)c2)OC)=O)CC12CCN(C(=O)C(F)(F)CO)CC2 Cc1nc(C(N)=O)ccc1C(N1CCC(n2cc(CNC(N)=O)nn2)C1)=O Cn1cc(S(C)(=O)=O)cc1C(N1CCOCC1CN=c1cccn[nH]1)=O c1(NC(C)=O)ccc(C)cc1C=CC(=O)NC1CCN(C(=O)CO)CCC1CO N1(C(c2c(CNC(=O)CC3CCCC(=O)N3)noc2)=O)CCC2(CCOCC2)C1 c1(CC(N2CC3C(CNC(c4cc(C)sn4)=O)(C3)C2)=O)c(C)ncnc1C C1(CNC(=O)C(O)Cc2ccccn2)CCCN(C(=O)CSc2nc[nH]n2)C1 C(=O)(CN=c1[nH]c2ccccc2s1)N(C)CCN(C)C(C1CN2CCN1CC2)=O Cc1cc(C)c(C(=O)NC(c2ccccc2)C)[nH]1.C(=O)C(C)(C)CN(C)C.C c1(C2C(C(N(CCNC(=O)CC3(CO)CC3)C3CC3)=O)C2)ccccc1 C1(NC(C2(CSC)CC2)=O)CN(C(=O)C(C)OC(C)(C)C)CC1(C)C c1(OCC)ccc(Cl)c(C(=O)N)c1.C1(C)CCCN(C(=O)C(C#N)C2CC2)C1 Cc1c(C(=O)NC(C)CC(C)NC(=O)CCc2ccc(O)cc2)nc2sccn12 c1(CN2CC(NC(c3c(Cl)ncc(C)c3)=O)C(F)C2)cc(C#N)ccc1Cl n1(CCC)nccc1C(=O)N(CC(C)NC(C1(OC)CCCC1)=O)C O=C(CCCCCc1cccs1)NCC=CCNC(=O)C(F)(F)c1cncs1 C(CC1CCC1)(C(=O)NC(C(N1CCC(n2cccn2)C1)=O)C1CCC1)OC c1(CN2CCC(CC(=O)Nc3cc(C)n(C(C)C)n3)C2)nc2ccccn2c1C C(=O)(C1=CC(O)CCC1)N1CC(C)(C)C(C)C1.c1(C=O)cc(F)c(F)c(F)c1.N c1ccc(Cl)cc1C.n1(CC)cc(C(=O)NC2CCC2NC(=O)CCC)cn1.O Cc1nc(C)n(CC(=O)NC2CC(C)C2)n1.C(=O)(CC1(C(F)F)CC1)N C1(CNC(C2OCCN(C)C2)=O)CC(C)(C)CN1C(=O)CSC1CC1 N1(C(C)=O)CCCC1C(=O)NC(C)CCN(C(=O)COC=C)C C1(C(=O)NCC2CCN(C(c3ccncn3)=O)CC2)CCCC2CCCN12 c1(C(N2CCCC(c3n(C)ccn3)C2)=O)cncc2cccnc12 Cc1ccc(OCC(=O)NC2CCC(NC(=O)COC3CC3)C2)cc1C Cc1cc(O)cc(=O)n1CC(=O)NC1CCC1.C1(C(=O)N)CCC2CC1C2(C)C C1(CCNC(C2CCC(=O)N2)=O)CCN(C(=O)COCCF)CCC1(F)F C1(NC(Cc2ccc(OCC=C)cc2)=O)CCCCN(C(C2(F)CCC2)=O)C1 c1(NC(N(CC(C(=O)O)SC)C)=O)ccc(OCc2cccnc2)cc1 C1(Cc2cc(C)sc2C)NC(=O)N(CC2CCCC(F)C2)C1=O Cc1cccnc1CC(=O)N(C(C)CNC(c1csc(C(F)F)c1)=O)C C1(C(=O)OC)CCC(C)CN1C(=O)C=CC(=O)Nc1ccccc1C Cc1nn(C)cc1CC(=O)NC1(CN(C(=O)CCc2nnc(S)n2C)C)CC1 c1(-c2nc(N3CCCC(NC(=O)NC4CC(C)(C)C4)C3)sc2)ccc(Cl)cc1Cl c1(-c2nc(C(N3CCOC3=O)CC)on2)cccnc1C(F)(F)F c1(CN(CC(C)OCC=C)CC)ncsc1C(=O)O CCCCC(C(=O)N1CCCCC1CCO)NC(C1C(C)C1C)=O C1(OC)CC(NC(c2cnc(O)s2)=O)CN(C(=O)CCC)C1.C(=O)C1CC1.N CC(C)CC(C=O)NC(=O)C(C(C)C)NC(=O)O.c1ccccc1.C1CC1.C C1(CC(=O)NCC(N2CCN(C(=O)C3=CCSC3)CC2)C)CC(O)C12CCC2 N1(C(c2cnn(C)n2)=O)CCC(C(=O)NCCC2CCCC2O)CC1 C(=O)(CC(C(F)F)NC(=O)C=CC1CCCN1C)NC(CC(C)C)(C)C C(=O)(C(F)(F)CCc1ccccc1)NC1C(NC(=O)Cc2c[nH]nc2O)CC1 N1(C(c2nc(N(C)C)nc(O)c2)=O)CCC(C)(C2CC2)CC1 c1(CC(=O)N(CCCCNC(c2ccnc(C)n2)=O)C)sc2ccccc2c1C c1(C(C(=O)N)N(C)C(C2CC23CC3)=O)ccc(F)cc1F.C(=O)(CCC)OC Cc1ccn(C(C)C(=O)NCC2(NC(=O)C(C)n3cncn3)CCC2)n1 c1(C(C)OCCCC)nc(CCCC)nn1-c1ccc(Cl)cc1 CON=CC(=O)NC(C)(C)C=CC(=O)N(C1CSC1)C C(=O)(C(C)CCCC(C)=O)NCC(CCNC(C1CC2CC(OC)C2C1)=O)OC N1(c2cc(COC)ncn2)CCC(C)C(NC(=O)C(CO)c2ccccc2)C1 N1(C(c2cnc(C3CC3)o2)=O)CCCC(NC(c2ccccc2)=O)C1.C1CC1.O CC(CS(N)(=O)=O)NC(=O)CCO.C1(=C(C(=O)N(CC)C)F)CCCCC1 c1(N2CC(C)(CC)OCC2)nc(N2CCN(C(C)=O)CC2)nc2c1COCC2 CC(C)(CC(F)F)C(=O)N1CCC(n2cc(-c3cccc(F)c3Br)nn2)C1 c1(COC)ccccc1C(=O)NC1CCC1.c1(C=O)c(C)noc1C1CC1 CC(C)C(C)(O)C(=O)NCCCC(C)(C)NC(c1cncc(C2CC2)c1)=O O=C(CC1COCc2ccccc21)NC1CC2(CCN(C(=O)COCCF)CC2)C1 CC1CCCCN1NC(=O)c1ccc(S(=O)(=O)N(C)CCO)cc1 n1(CC(=O)NC(C2CCCN(C(C=C(C)C)=O)C2)C)cc(S(N)(=O)=O)cn1 C(N=c1[nH]c(=NCC23CCCCC2C3)[nH]c2c1SCC2)c1c(C)cn(C)n1 Cc1cc(F)cc2c1CN(C(=O)Cc1csc(Cc3ccccn3)n1)CC2 CCC(C)C(O)CC(=O)N(CC(C)(C)NC(=O)CCOC(C)C)C N1(C(c2ccc(F)s2)=O)CCC(N2CCN(C(=O)C(O)CF)CC2)CC1 N1(C(C(C)N(C)C)=O)CCN(C(c2sccc2Cl)=O)CC1CC(F)F CCC(O)C(C)C(=O)NCCN(C(C1CN(S(N)(=O)=O)C1)=O)CC O(NC(=O)C1=CCCC1)CC(N1CCC(C)(CC)C1)=O c1(N2C(C(N3CCC(NC(C)=O)C3)=O)CC(OC)C2)ncc(Br)c(C(C)C)n1 C1(CNC(C2CC3(CCC3)C2)=O)CC2(CC2)CN1C(=O)CC(Cl)Cl N1(C(CN(C)Cc2ccc(C)cc2)=O)CCN(C(=O)CO)C(CF)C1 Cc1cc(C)n2nc(C(=O)NCC3CCN(c4ccc(F)cc4)C3)nc2n1 c1(C(=O)NCC(CNC(CC(C)(F)F)=O)F)cc(O)c2ccccc2c1 C12CC(C)(C1)OC21CN(C(=O)C)C1.c1ccc(F)cc1.C=C1CC(C(=O)N)C1 c1(OC)cc2cc(NC(C3CCN(C(C)=O)C3)=O)cnc2cc1OC CCCCC(C)CCC(=O)N1CC(NC(c2conc2C)=O)C1 Cc1cncc(C)c1C(=O)NCC1CN(C(c2cncn2C)=O)C(C)(C)C1 c1(NC(c2ccc(SC)cc2)C)nc(C)cc(=NC2CCCCC2)[nH]1 c1(C(N2CCC(CNC(c3c(C)ncnc3)=O)C2(C)C)=O)cc2cc(Cl)sc2[nH]1 CN1CCC(C)(CNC(c2coc(CNC(c3ccnnc3)=O)c2)=O)C1 CCC(CC)CCC(=O)N(C1CCCN(C(=O)Cc2ccco2)C1)CC C1(CCC)(NC(c2cccc(N(C)C)c2)=O)CCCN(C(C2CC2F)=O)C1 C#Cc1cnc(C(N2CC(F)CC2C(=O)Nc2ccc(C(C)C)cc2)=O)c(C)c1 N1(C(C2CCN(CC)C2)=O)CCN(C(=O)C#CC2CC2)C(C2CC2)C1 c1(C(=O)NCCC(C)NC(c2ccc(C#C)cc2F)=O)ccc2nc(C)sc2c1 N1(C(C2CCC(C)O2)=O)CCC(CNC(c2cnsc2)=O)C12CC2 N1(C(=O)C(c2cccnc2)Nc2ccc(Cl)cc2)CCc2ccc([N+](=O)[O-])cc21 C1(C)(NC(C(CCC2CC2)NC(C(C2CC2)SC)=O)=O)CC2CCC1C2 c1(C(=O)NCC(C)CN(C)C(C2CCOC(=O)N2)=O)cn(C)c(=O)nc1O C1(CNC(CC2CCC(C)C2)=O)C2CN(C(C34CC(C)(C3)C4)=O)CC12 C1(OC)CC(CNC(=O)CCc2cnn(C)c2)N(C(C2CCCCN2C)=O)C1 N1(C(C(n2c(C)ccn2)C)=O)CCC2(CC2)CC1C(=O)NC1(CO)CC(F)C1 CC1CC(NC(=O)Cc2cccn2C)CN(C(=O)C(c2ccc(Cl)cc2Cl)O)C1 Cc1ccsc1C(=O)NC(C)(C)C=CC(=O)NCCC1CCC(C)C1 c1(-c2c(C=O)c[nH]c2)ccc(F)cc1.CC(C)C.C1(C(C)(C)O)(C=O)CC1.N C1(OC)CN(C(c2cccnc2S)=O)C(C)(CNC(=O)C)C1.[SH](C)(=O)=O C=C(C)CC(Cc1ccccc1)NC(=O)CC1(O)CCOC1 C=CCC(C)(CC)C(=O)N1CC(O)(CNC(=O)CCSCCCC)C1 C1(C(N(CCN(C(CC2(OC)CCOCC2)=O)C)C)=O)CCc2c(ncn2C)C1 CC1(C(N2CCC(C3CC3)C2)=O)CCS(=O)(=O)CC1.C1(C)(C=O)CC=CC1.C n1(C(CC)C)nc(C(N2CC=CC2CNC(=O)C(C)(C)N2CCCC2)=O)cc1C C1(Cn2cc(CN(CC)CC)nn2)CCN(C(C2CCNC2=O)=O)CC1(F)F N1(C(CC(C=C)C)=O)CC2CCN(C(c3cc(C(C)=O)cn3C)=O)CC12 C12(CNC(C(CCC)F)=O)CCCC1N(C(c1cc(Cl)ccn1)=O)CCC2 C=CC1CN(C(=O)C(Cn2cccn2)NC(c2c[nH]nc2C)=O)CCO1 c1(C(=O)CC)c(NC(=O)CCCCN(C)C)cccc1O.C(=O)(C)NCC c1(CNC(C2(OCC)CC2)=O)ccccc1C.C1(C=O)CC1C=O.N n1(CC(=O)N(C)CC)cc(CN2CCC(Oc3ccncc3)C2)nn1 c1(C2CCN(Cc3c(-c4n(C)ccc4)csc3)C2)nc2ccccc2o1 N1(C(CC(C)C2CC2)=O)CCC(C2CC2)(CNC(c2ccc(O)nc2)=O)C1 c1(C(N2C(C(=O)Nc3c(OC)c(Cl)ccc3)CNCC2)=O)c[nH]c2ncccc12 C1(CNC(C2C(C)(C)C2)=O)CN(C(=O)CS)CC12CC2.c1ccncc1.C c1(C(N2CC(NC(C3C(CC)C3)=O)C(C)C2)=O)ccc(S(C)=O)cc1 Cc1c(C(N2CCOC(C(=O)NC3CCC4(CC4)C3)C2)=O)cccc1C#N C(C)(C(=O)N(CC(CC)NC(C1CC1(Cl)Cl)=O)C)=C(CC)C CC(C(=O)NN1CCCC1C(=O)Nc1cn(C)nc1C(N)=O)c1cc[nH]n1 CCCCCC(CC)C(=O)NCC1(O)CC(NC(c2ncncc2C)=O)C1 C12(NC(CC(=O)NCC)=O)CCC(CN(C(=O)CC3CC(C)(C)C3)C1)C2 C1(CCCCC(=O)NCC(CC)NC(=O)C(C#N)C2CC2)SCC2NC(=O)NC12 C1(C(=O)NC(C=C)C2CC2)CC12CCN(C(c1ncc(F)cc1F)=O)CC2 C1(C(=O)NCc2nc(C3CC3)n[nH]2)CCC(C2CC2)N1C(c1cnco1)=O c1(NC(=O)CNC(C2CCCCC2Oc2ccccc2F)=O)cc(Br)cc(I)c1 N1(C(c2ncc(CC)o2)=O)CC(NC(C2(COC)CCCO2)=O)CC(C)C1 N1(C(C2N(C(C)C)C(=O)CC2)=O)C2CCC1CN(C(c1cc(Br)no1)=O)C2 CCCC(CNC(=O)C(C)C(C)(C)C)C(=O)Nc1ccc(C)c(C)c1 C(C)(C)(C(=O)NCC(O)CNC(C1(O)CCOC1)=O)OCC.C(C)C c1(C(N2CCC(OC)(C)C2)=O)nn(C)c2c1COCC2.C1(CC=O)C=CCC1.N N1(C(C2=C(C)CCCC2)=O)CCC(C2(O)CN(C(=O)C3=NOCC3)C2)CC1 c1(C(N(C(C)C)CCNC(=O)C(C)c2cncs2)=O)cc2ccccc2c(O)n1 C#CCC(C)(C(=O)N1CCC(C(C)CO)CC1)NC(=O)C(CC(=C)C)OC c1(C(=O)NCC2CC(NC(CCC(CC)C)=O)C2)ccc([N+](=O)[O-])c(OC)c1 CC(C)CCC=CC(=O)NCC(C1CCOC1)NC(c1cnccn1)=O c1(C(=O)NC(C2CCN(C(CCC(=O)NC)=O)C2)C)ccc2ncn(C)c2c1 C1(CNC(C(C)S)=O)CC2(CCN(C(=O)C(C)(C)Br)CC2)CO1 c1(C(N2C(C)CCC(NC(CCCOCC)=O)C2)=O)cc(Br)c(C)cc1F CC(F)(F)C(F)C(=O)NC1CCC(CNC(=O)C=C2CCOCC2)CC1 c1(C(N2CCCC(C3CC3)C2)C)cc(Cl)ccc1Cl CCCCC(CC(=O)N1CC2C=CC1CC2)NC(c1cc(OC)n(C)n1)=O Cc1ccc(C)c(C(=O)N(CC(C)N(C)C(C2CC3(CCC3)CO2)=O)C)c1N Cc1nc(C(C)C)sc1C(N1CCC(C)C1CNC(c1c(C)ncn1C)=O)=O CCC(CCC(=O)NC(c1ccnn1C)C(=O)NCC1CC(CF)C1)OC N(S(=O)(=O)N(C)C)CC(=O)N(CC)C1CC1.n1(C(C)C)cc(C=O)nn1 c1(C(N2C(CC)C(NC(=O)CO)CC2)=O)cc(C(N)=O)ccc1C.C1CC1 N1(C(CC2C(C)(C)CCCO2)=O)CCC(C2CCN(C(=O)C3=NOCC3)C2)CC1 c1(CCNC(C2C(C)C2)=O)occc1C(CC(=O)N)=O.n1(CC)cncc1 Cc1cc(NC(=O)Cc2cnn(C)c2)cc(O)c1.C1(C=O)CC2(CCO1)CC2.N S(=O)(=O)(c1cccnc1NC1CS(=O)(=O)C1)NCc1c(C)nn(C)c1C N1(C(=O)CC2CCCO2)CC(NC(=O)CCSCc2ccccc2)C2(CC2)C1 CCCC(C)(C)CC(=O)N1CC(C(F)(F)F)CC1CNC(C1(SC)CC1)=O c1(OC)ccc(C(=O)NCC2CN(C(C3CN(C)CCO3)=O)CCO2)c(F)n1 [SH](=O)(=O)c1cccc(C#N)c1.C1(C(N(C)CC)=O)CCCC1(F)F.C(=O)C.N N1(C(C2CC(C(=O)OC)C2)=O)CCC2CCC12.c1(CCC=O)c(C)noc1C.N C(CCC(=O)N)(C(C)C)NC(c1c(CC)nc(C)o1)=O.c1(C2CC2)cccnc1 N1(C(COC(CC)C)=O)CC=CC(NC(c2cnn(C(C)CC)c2C)=O)C1 Cc1ncc(C(N2CCCC2CNC(c2ccc(C#N)c(Cl)c2)=O)=O)cc1C#N N1(C(c2scc(-c3cccc(CN(C)CC)c3)c2)=O)CCc2cc(Cl)ccc2C1 C(=O)(CC(C)(C)C(=O)OCC(=O)Nc1ccccc1[N+](=O)[O-])OC C(C(CC)(CC)C(N)=O)OC.c1(C(N2CCC3(C2)C(=O)N3)=O)n[nH]c2c1COC2 C1(CNC(c2cc(C)ns2)=O)CCN(C(=O)C(F)=CCF)CC1 c1(C=O)cc([N+](=O)[O-])c[nH]1.c1(C(N(C2CCC2)C)=O)coc(CC)n1.CC.O n1(CC)ccc(CC(=O)NC(C)C(=O)NCC2(SCC)CC2)n1 N1(C(c2n(C)nc3c2COCC3)=O)CCC2CCN(c3ncc(Cl)cn3)CC2C1 N1(C(c2cnc(C)o2)=O)CCC(C(=O)N(C2CCC(=O)N(C)C2)C)C12CC2.CC C(=O)C(F)(F)C(F)(F)F.C1(C(=O)OC)CCC(C(=O)NC2CCCCC2)CC1 c1(C(=O)NC(C)CNC(c2c(Cl)cncc2Cl)=O)ccc2c(=O)n(C)cnc2c1 N1(C(c2ncc(OC)nc2)=O)CCC2CN(C(c3ccc(CO)cn3)=O)CC12 c1(CC(=O)N(CC)CC)cccc(C(F)F)c1.C(=O)C(F)Cc1ccccc1 C1(N(C(C(CCC)OC)=O)C)CCCN(C(C2(CCOCC)CC2)=O)CC1 c1(C(N2CC(NC(=O)C(O)C(F)F)C3(C2)CC3)=O)c(F)cc(F)c(F)c1F C(=O)(CCCC(F)(F)F)N1C(C)CC(CNC(COCCCC)=O)C1 N1(C(c2cc(CF)on2)=O)CC2CCCN(C(=O)C3=CS(=O)(=O)CCC3)C2C1 CCC(CCc1ccccc1)C(=O)N1CCC(NC(c2cc(O)cs2)=O)C(C)C1 Cc1[nH]c(=N)sc1C(N1CC(NC(C2C(C)C2C)=O)C(O)C1)=O c1(C(=O)NCCN(CCOC)C(c2sccc2C)=O)c(C)ncn1O.O C(C)(C(O)C(=O)NCCN(C(=O)CC1(N2CCCC2)CC1)C)OC C=Cc1cccc(NC(C2CN(C(c3cc(OC)n(C)n3)=O)CCN2C)=O)c1 C(=O)(C1c2ccccc2C2CC1C2)N1CCCCC(NC(CSCC=C)=O)C1 CCC(CC(=O)NC1CC12CCN(C(c1[nH]nnc1C1CC1)=O)CC2)C(F)F c1(C(=O)N)ccc(Cl)nc1.c1(CC)cccnc1C(=O)NC(C)CO.C1CC1 CCCCC(CC(=O)NCC1CCCN(CC)C1)NC(=O)COc1cc(C)on1 C1(C(N2C(C(C)NC(=O)COCCCF)CCC2)=O)CCCC(C)(C)C1 n1(C(C)=O)cc([N+](=O)[O-])c(NC(C2CN(C(c3n[nH]cc3C)=O)CCO2)C)n1 c1(OC)nc(C)ncc1C(N1CCC(C)(C)C1)=O.C(=O)C(C(C)C)N(C)C.N c1(C(=O)NC(CC#C)C(=O)NCC2CNC(=O)O2)ccc(C)c(C#C)c1 N1(C(=O)C=C2CC2)CC2(CCCN(C(=O)Cc3ccc(Cl)c(F)c3)C2)C1 c1(OC)cccc2[nH]c(C(=O)NC3CN(C(c4oc(C)nc4C)=O)C4CC34)cc12 C1(CN2CC(O)(CNC(Cc3cn(CC)nc3)=O)C2)CCC2CC2C1 C#Cc1cccc(C(=O)NCC(C)CNC(c2ccc(C(C)=O)cc2)=O)c1.O Cc1c(NC2(c3nnnn3C3COC3)CCC3CC23)ccc2nccn12 N1(C(c2n(C)ccn2)=O)CCC2CCCC12C(=O)NCC1(CC(N)=O)CC1 N1(C(C2(C(C)NC(C(C)C3CCC3)=O)CC2)=O)CCC2(CCCO2)C1 Cn1nc(C(c2nnnn2CC2CCOCC2)NCC2CC2(Cl)Cl)cc1I CCCC(C)CC(=O)N1CCOCC(CNC(=O)C(F)(F)CCn2cccn2)C1 c1(C(C)(C)C)ccc(C(c2nnnn2C2CCCCC2)NC2CC=CC2)s1 Cc1[nH]c2ccccc2c1CC(=O)N(CCCNC(C12CCC(CO1)C2)=O)C C1(CN(C(c2ccsc2OC)=O)CC)CCN(C(=O)CCN2CCOCC2)CC1 N1(C(C2=CCC(NC(C3CN(C)C(=O)CC3)=O)C2)=O)CCC2(CNC(=O)C2)C1 C1(CNC(C2(OC)CC2)=O)CCCC12CCN(C(=O)Cc1c[nH]nc1C)CC2 Cc1ccoc1C(N1CC(O)(C(F)C(=O)NC(c2cncn2C)CO)C1)=O C1(C(N2CC(C(C(=O)NC3(C)CCC3)OC)C2)=O)COCC1C(N)=O C(CC(=O)NC(C1CCOCC1)(C)C)(CC(C)C)NC(CC1C(C)=NNC1=O)=O N1(C(C2CN(C)C(=O)CC2)=O)CC2CCC(CNC(C3(C#N)CC3)=O)(C2)C1 C1(OC)CC(O)C1NC(C1CCCO1)=O.C(=O)(C(C)C)N(CC=O)C.C C(C(=O)N(C1CCC1)CC(C)C)(C(C)CC1CCCC1)N1CCC(OC)CC1 CC(C)CC(C)CC(=O)NCCCCCCNC(c1cc(C2CC2)nn1C)=O C#Cc1ccc(C(=O)NC(C(=O)NOCC(=O)OC)C2CCCO2)o1 c1(C(N2CC(C)C(NC(c3nonc3N)=O)CC2)=O)ccc(F)c2c1CCC2 N1(C(c2c(C)cn(C)c2)=O)CC(NC(c2nocc2C(C)C)=O)C(C2CC2)C1 N1(C(CN(CCC)C)=O)CCC(NC(=O)C(C)(C)CO)C1c1ccccc1 CCCC(CCC)C(=O)N1CCC1CNC(=O)C(F)CC(C)C N1(C(c2cc(F)nc(F)c2)=O)CCC2(CC1)CN(C(c1sccc1I)=O)C2 N1(C(C2C(C)CCC2)=O)CC2CCCN(C(=O)CC3NC(=O)NC3=O)C2C1 C(=O)(CC(C)(C)CCOC)N1CCCC(NC(c2nc(CC)oc2)=O)(CC)C1 C(CCCCC(=O)NC(CC(=O)N1CCC(n2ccnn2)C1)C(F)F)=CC CC1CC2(CCC2)CN1C(=O)C#CCNC(=O)C(C)(C)C(=O)N(C)C N1(C(C(CC)(C)C)=O)CCOC2CN(C(c3cccc(OC(F)F)n3)=O)CC12 C1(NC(=O)N(Cc2ccsc2)Cc2ccccn2)CCNC2(CCCC2)C1 N1(CC=O)CC2CCC1C2.c1(C(N(CC)CC)=O)cc(N2CCCC2)ccn1.N C1(NC(C=CS(C)=O)=O)CCC2CCN(C(=O)CCc3cn[nH]c3)C12 O=C(C1=CCC(F)(F)CC1)NC1CCN(C(c2cc(O)ccc2F)=O)C1 CCCC(C(O)C(=O)NC1COC(C(F)F)C1)NC(C1CCCSC1)=O C1CC2CC2N1C(C1CCCN1C=O)=O.C(C(C)C(=O)N)OC.C(C)(C)C c1(C(=O)NC2CC(C)N(C(=O)C=Cc3nnn(C)n3)C2)cc2c[nH]cnc-2n1 C1(NC(C(C(C)C)n2cncn2)=O)CC2CC1N(C(=O)CC13CCC(CC1)C3)C2 Cc1sc(Cl)nc1C(=O)NCCNC(c1ccc(C2CC2C)o1)=O c1(C(N2CC(C)(NC(CCCCCC#C)=O)C2)=O)cc(Br)cc2nc[nH]c12 c1(C(=O)NCCCCC(=O)NC2C(C)(O)CCC2)cccc(C#N)c1 N1(C(c2c(C)cccc2)=O)CCC2(C=C(C(=O)NCC3CCC3)C2)C1 CC1CCN(C(=O)CNC(=O)CNC(=O)C(C)C2CCCO2)CC1 C1(CNC(C(C)CF)=O)N(C(=O)C(O)Cc2cnc[nH]2)CCCC1(C)C c1(C(C(=O)NC(C(C)(C)NC(COC)=O)C)C)ccc(Br)cc1C CCCC(N)C(=O)N1CCC(c2ccc(C(=O)O)cc2)C1 c1(C(=O)NC(C)CC(=O)c2cccs2)cccc(OCC(F)(F)F)c1 N1(C(C2(NC(C(CC)CC)=O)CCN(C)C2)=O)CC(=O)N(C)CC1CC C1(C(C2CCCC2)NC(C(C(C)C)c2cccnc2)=O)CC2CCC1CC2 N1(Cc2c(OC)ccc(F)c2)CC2CCN(C(=O)CC(=O)NC3CC3)CCC2C1 c1(C(=O)NC(CN(C(C(CC(=C)C)C)=O)C)C)cccc2nc[nH]c12 Cc1c(C(=O)N(CCCCNC(C2CC23CCCOC3)=O)C)cccc1N CN=c1[nH]cc(C(=O)NC2C=CC(CC(=O)NCCc3cc(C)[nH]n3)C2)s1 C1(C(N2CC=CC2)=O)CC2(C1)NC(=O)NC2=O.c1(N(C)C)nc(C(=O)N)co1 Cc1cc(C(N2CCC(CNC(c3ccnn3CC#N)=O)C2)=O)cc(Br)c1 C(=O)(CS(=O)(=O)CC(=O)N)OC.c1(C=O)c(C)cnn1C.C1(CC)CC1.C Cc1cc(C=O)cnn1.C1(CC(N2C(C(C)C)CCC2)=O)C=CS(=O)(=O)C1.N c1(C(=O)NCC2(F)CCN(C(C(C(C)C)F)=O)C2)cc2cc([N+](=O)[O-])ccc2s1 C1CN(C(C2C3CC4C(C3)C24)=O)CC2(CCC2)C1.c1cc(C=O)on1.CCO N1(C(CCN(C(C)=O)C)=O)CCCC(C)C1CCNC(c1cnc(N)c(N)c1)=O c1(CN(c2ccc(NC(=S)NC3CC3C)cc2)C(C)=O)ccc2c(ccn2C)c1 N1(C(C2CCN(C(C(c3n(C)ncc3)O)=O)CC2)=O)CCC(CO)=C(F)C1 C(=O)(CC(C)(O)COC)NC1CN(C(CCOc2ccc(CC)cc2)=O)C(C)C1 c1(C(C(=O)NCC(=C)C)N(C2CC3CC3C2)C)csc(C)n1 C(COC(c1scnc1-c1cccc(OC)c1)=O)(C(F)(F)F)OCC C12(C=O)CCC(C)(C1)OC2.c1(CN(C(=O)C)C)cc[nH]n1.C(C)(C)C.O c1(C=O)cnc(N)c(-c2ccccc2)c1.C(CC)(C(=O)NCC(C)C)OCC.N C1(C#N)(C(=O)NCC(CNC(CC2(OC)CCCCC2)=O)O)CC12CCOCC2 C(CNC(=O)C(F)n1cccn1)(CC)(CC)NC(CCC=C)=O c1(CC)cc(C(N2CCC(CNC(=O)C(C)Oc3ccccc3)C2)=O)sc1C CCC(C)CC(=O)NC(C)(CNC(C1(CSC)CCOCC1)=O)C1CC1 c1(OC)cc(C(N2CC3CC(C)(C)C3C2)=O)cc([N+](=O)[O-])c1O C1(NC(c2n(CC)ccn2)=O)CCCC12CCN(C(C1CC1C#N)=O)CC2 C1(C(N2CCN(C)C(CNC(=O)CCCC(C)(F)F)C2)=O)CCn2nnnc2C1 C=CC1CN(C(C2(F)CCC2)=O)CC1NC(c1ccc(CCF)cc1)=O C1(C(N2C(CC=C)CCCC2)=O)CCCN(C(C23CCC(C)(C2)OC3)=O)C1C c1(OCCC)ccc(F)cc1NC(=O)N(CC)Cc1cc(Cl)cc(Cl)c1 N1(C(=O)OC(C)(C)C)CC2CCCCC2C1C(=O)NCc1ccon1 c1(C(N(CCCN(C(c2c(COC)ccs2)=O)C)C)=O)cccc2nn[nH]c12 C1(C(=O)NCC2(F)CCN(C(COCCCCC)=O)CC2)CN2CCC1(C)CC2 c1(OC)ccnc(C(N2CC(OC)CC2CNC(c2cc(C)ns2)=O)=O)n1 N1(C(c2c(N)cc(F)c(Cl)c2)=O)CCCC2(CNC(=O)C3=CCCO3)CCCC12 N(C1CN(C(c2ccc(OCCO)cc2)=O)Cc2ccccc21)C(CC=CC)=O N1(C(C(CCCCC)O)=O)CCCC(C2CN(c3ccc([N+](=O)[O-])cc3C)C2)C1 C1C(C2CC2)CCN1C(=O)Cc1[nH]cnc1C.c1(C(C(=O)N)OC)cccnc1.C CC1Cn2nccc2CN1C(C1CC2CC1CN(C(c1cc(O)cs1)=O)C2)=O c1(C(=O)NCC2CN(C(C#CC(C)(C)C)=O)C2)ccc2ncsc2c1 C(CC(C)(C)C(=O)NCCC1CCCN(C(=O)Cn2cncn2)C1)SC N1(C(C(CO)N(C)C)=O)CC(CNC(C2CC(F)C2)=O)OC(C)(C)C1 C(=O)(CC1=CCN(C(=O)C(O)CSC)CC1)NC1CC(CC)(CC)C1 C#CCCC(C(=O)NCCC1CCC(C)(C)O1)NC(=O)C(C)n1cccc1 c1(NC(C(C)OC)CC(=O)OC)ncnc2c(C)cccc12 c1(C(=O)NC2CCN(C(CNC(C)=O)=O)CC2C)cc2c(nc1O)CCCC2O c1(OC)ccc(OC)c(CN(C)C(C)C2CC2)c1.[nH]1cc(CCC(C)(C)O)nn1 C(CCC(O)C(=O)Nc1cnc(F)c(C)c1)NC(C(COCC)(C)C)=O Cc1cnc(C(=O)NC(CO)C(C)NC(C2(CO)CCCO2)=O)nc1 N1(C(CC(C(C)C)C)=O)CCC(N(C(=O)C=Cc2ccc(Cl)cc2)C)C2(CC2)C1 c1(C(=O)NCC2CC(NC(c3cc(N)c(F)cc3)=O)C2)noc2cc(Cl)ccc12 N1(C(C(OC)OC)=O)CCCC(C2(CNC(=O)CC3CCCCC3)CC2)C1.C Cc1nc(C(C)NC(=O)NC(C)C(C2CCCCC2)C)c(C)o1 c1(C(=O)NC(COC)CNC(c2c(C)ncnc2C)=O)cc(C)cc(Cl)c1.O c1(CNC(c2nnnn2CCC2CC2)(C2CCCOC2)C)ccc2[nH]ccc2c1 C1(CCCC)CCC(C(N2CC(NC(C3CC(C)OC3C)=O)C2)=O)CC1 C1(C(=O)OCC)(OC(C(CCC#C)O)=O)CCCS(=O)(=O)C1 N1(C(CCCCCC)=O)CC2CC1CN(C(C1C(Cl)(Cl)C13CC3)=O)C2 c1(CNc2nc(COC)nc(N(CC(N)=O)C)c2)cc2sc(C)cc2[nH]1 C(=O)(C(CC(C)C)NC(=O)C(C1(O)CCC1)NC(c1csnc1C)=O)NC C1(NC(C2(CCCC)CCC2)=O)CC2(C1)CC2NC(=O)CN1CCSCC1 n1(CC(=O)NC2CC3(C2)CN(C(C2CC4CC4C2)=O)C3)ccc2cc(F)ccc12 C1(CNC(c2ccn(C3CC3)n2)=O)CC(O)(C)C1.C1(C(=O)N)CCC1 C1(C(=O)NC(C)CCN(C)C(c2cnc(Br)s2)=O)CCN(C)C1=O C(CCCCCCCO)=CC(=O)NCc1ccc(CCC=C)cc1 C1(NC(CCCc2c(C)ccs2)=O)CCC(F)(CNC(=O)C(C)N2CCC2)C1 c1(C(=O)NCCCC(C)NC(=O)CCn2cc(Cl)cn2)cc([N+](=O)[O-])ccc1N C1(NC(C(C)=C2CC2)=O)CC(NC(C2(C(F)F)CCOCC2)=O)C12CCC2 c1(N(C)Cc2c(C)n(C)nc2)nc(=NC(C)C(C)C)[nH]c2c(C)nn(C)c12 c1(C(N2C3C(NC(C(CCSC)O)=O)C(C3)C2)=O)cc(F)ccc1N N1(C(C(CCC)(C)C)=O)CC2CCC(C1)N2C(c1cc(C(=O)OC)sn1)=O CCCCS(=O)(=O)NCC(=O)NC1CCCCC1C(=O)Nc1cncc(CO)c1 N1(C(C(=O)NCC(C)C)=O)CCCC(CC(=O)NCC2C=CCCC2)CC1 N1(C(CC2(C=C)CC2)=O)CCN(CCCNC(c2nccnc2SCC)=O)CC1 c1(CCC(=O)NCC(CN(C(=O)CN2CCCC2=O)C)O)ccncc1Br c1(CC)c(C(=O)NC2CC(F)(CNC(C3(C)CCC3)=O)C2)cn[nH]1.C c1(SC(C)C)nsc(NC2COCC2NC(=O)OC(C)(C)C)n1 Cc1cc2c(CC(=O)NC3CCC(C)(NC(=O)Cc4cncs4)CC3)csc2s1 S(=O)(=O)(c1cc(C=O)co1)NC.c1(CC=O)ccc(C)c(C)c1.CC#CC.N CC(C)CCC(F)C(=O)N1CC2(CC2)CC1C(=O)N(C)CC1(C)CC1 N1(C(CC=CC=C)=O)C2CCC1C(C)C(NC(c1cccn3nccc13)=O)C2 c1(CN2CC(C(=O)Nc3c(CC)cccn3)C2)cc(Br)ccc1O C(=O)(C(C)C(O)C(C)C)N1CC(C(N2CCCCC2CCO)=O)(COC)C1 C(c1ccccc1F)=CC(=O)N(C)CCOCCC.C1(C(=O)N)C2CCCC12 C1(CNC(C(N)=O)=O)CN(C(C2C3CCCCC23)=O)CCC12CCOCC2 c1(C(=O)NCC2(F)CN(C(c3[nH]cc(C(N)=O)c3)=O)C2)ccc2n[nH]cc2c1 C=C1CC2(C1)CC(C(=O)NC1CC3C1CCN3C(c1cccc(Br)c1N)=O)C2 Cc1cc(C#N)cc(C)c1C(N1CCCCC1C)=O.C(=O)(CC(C)P(C)(C)=O)N C(=O)(CC(C)C(C)(C)C)NC(CC#C)C(=O)NCc1cscc1C C1(CC)(NC(=O)CCC2CC(C)(C)CO2)CCN(C(c2cccnc2S)=O)CC1 n1(CC)cc(C(=O)C(=O)NC2(CNC(C3CC3(F)F)=O)CCC2)cn1 C=C(C)CC(C(=O)NCC(c1cccc(C)c1)C(=O)O)OC O=C1NCC(C(=O)N2CCCC2CNC(=O)C(F)(F)C2CC2)c2ccccc21 CN1CCC(OCC(=O)NCC(F)C)CC1.c1(C2C(C(=O)N)C2)cnn(C)c1 Cc1cc(F)c(O)c(NC(c2ccc(-c3ccccn3)nc2)=O)c1F N1(C(CCC(=O)NCCC)=O)CCC(c2cn(Cc3n[nH]cc3C)nn2)CC1C C(=O)(C1=COCCO1)NCC(C)(CO)NC(c1cc(C(F)F)cc(F)c1)=O Cc1cc(C(C2CC2)NC(=O)N)ccc1Br.c1(CC)ncc(C(F)(F)F)cc1Cl C1(C)(C(=O)NCCc2cc(C(=O)NCc3nnc(C)s3)no2)CCC(C)C1 CCCCC(C(=O)NCc1nc(CC)no1)NC(C1CCCSC1)=O C1(C(=O)NC(C(C)NC(C=C(CC)CC)=O)C)CCCCC1N=[N+]=[N-] S(=O)(=O)(c1cccc(=NC(C)CN2CCN(C)CC2)[nH]1)NCC(CC)(C)C CC(C)(CC(F)C(=O)N1CCN(CCO)C(=O)C1)NC(c1ccc(O)nc1)=O c1(OC)cc(C(N2CCCC(NC(c3cc4sccc4s3)=O)C2)=O)ccc1I C1(CC)CCCN(C(=O)CC2CCC(O)C2)C1C(=O)NCC(c1ccnn1C)O CC1CC(C(=O)N(CC(C)(C)C(=O)NCC(C)Cn2cccn2)C)CCO1 C1(C2CCOCC2)(C(=O)NCCC(CC)(CC)NC(C2CCC(=C)CC2)=O)CC1 c1(CCCC(N2CCCC(O)(c3ccccc3)C2)=O)csc2ccccc12 C(C1CN(C(=O)CNC=O)CC1C(=O)NC1C(C)CCC1C)=CC C1(C(=O)NC2C(F)CCN(C(CCCN(C)C)=O)C2)CCc2ncnn2C1 CC1=C(C(=O)NC(CCC(C)C)C(=O)N(C)Cc2c[nH]nc2C)CCCO1 CCCCCC(C)(CC)C(=O)N1CCCC(F)(CNC(c2ccsc2)=O)C1 N1(C(C2N(C(CCC3(C)N=N3)=O)C(C3CC3)CC2)=O)CC(F)(F)CC1CO NS(=O)(=O)CCC(=O)NCC1(F)CN(C(C2(C(F)(F)F)CCCCO2)=O)C1 N1(C(C2C(C(C)(C)C)C2)=O)CCN(C(c2scnc2Cl)=O)C(CC2CC2)C1 N(C1CCOc2ccc(Br)cc21)C(=O)Nc1ccc(N(CC)CC)nc1 c1(C(=O)NCc2snc(CC)n2)oc(C)cc1C.C1(C#N)(C=O)CC1C.N C1(CCC)CN(C(c2cc(C3CCCN3C)[nH]n2)=O)CCN1C(=O)C(N)=O c1(NC(C=CC(C)C)=O)ccc(CN2CNC(=O)C2)cc1 N1(C(=O)Cc2cccc(O)c2)CC2CCN(C(=O)C3CC3)C2C1 c1(-n2c(C3C(COC)C3)nc(-c3nccs3)n2)ccc(Cl)cc1C n1(CCC)ncc(C(=O)NCC(C(C)C)NC(=O)C(c2csc(C)n2)=O)c1C C=CCCC(F)(F)C(=O)N1CCC(C(O)CNC(=O)CN(CC)CC)CC1 C1(NC(C2(C)ON=C(C)C2)=O)CC2CN(C(=O)C=CC3CCOC3)CC2C1 CCC#CCN=c1[nH]c2c(c(=NCCCOC(=O)N(C)CC)[nH]1)CCCCC2 c1(C=O)cc(Cl)cc(Cl)c1.n1(CC)ccc(C(=O)NC(C2CCCC2)C)c1C.N c1(C(=O)NC2CCC(CNC(c3cc(C)nn3C)=O)C2)cnc2ncccn12 C1(NC(c2cccc(O)c2F)=O)CCN(C(=O)C(c2cccnc2)O)CC1F c1(C(=O)NCC(CO)NC(c2ncc(C)c(C)c2)=O)n[nH]c(C(C)C)c1[N+](=O)[O-] c1(OC)c(CN(C(=O)C=O)C)cc(Cl)cc1Br.C(CS(C)(=O)=O)C1CCC1.N C1CN(C(C2C(F)(F)C23CC3)=O)CC1O.O=C(CCC1CCCC1)NCC=O.N CCC(CCCC(=O)N1CC2CCCC12)NC(=O)C1=NNC(=O)C1 c1(CCC(=O)NCCCCCN(C(=O)CC2CCC(O)C2)C)cccc(F)c1F C(=O)(CCCn1cncn1)NC1CC(CC(=O)N(C(CC)CC)C2CC2)C1 Cc1nc(C)c(C(=O)NC2(CNC(c3cccc(CF)c3)=O)CCOCC2)s1 C(=O)(C(F)CCC)NC(C(=O)NCc1cn(CC#C)nc1)C1CCCO1 C1(NC(C2CCCN2C2CC2)=O)CCCCN(C(C2(n3cncn3)CC2)=O)CC1 C1(C(N2CC(OCCNC(c3cnc(Cl)s3)=O)C2)=O)OC2CCC1CC2 CCC(CC)CC(F)C(=O)NC(c1ccnc(F)c1)C c1(C(N2CCCC(NC(=O)NC(C)=O)C2)C(=O)NCC)cnc(Cl)n1C N1(C(c2c(C)snn2)=O)CC(O)CC1CNC(c1c(Cl)noc1C)=O C(C(N)CC(=O)N1CCCC(C(=O)Nc2nccn2C)C1)OC Cc1[nH][nH]c2ncnc(=NCc3ccccc3CNC(C3(O)CCSC3)=O)c1-2 n1(CC=O)ccc([N+](=O)[O-])n1.C1CC2(C1)CC2.c1(CC)nonc1C(=O)N C1(NC(CCC(C)(C)C)=O)CCC2(CCN(C(C3(CO)CCCC3)=O)CC2)C1 C1(CCNC(c2n(CCC)ncc2)=O)CCN(C(c2ccoc2C)=O)C(C)C1 c1(NC(c2cccc(Br)c2F)CO)snc2ccccc12 C=CCCC(C)(C)C(=O)NC(CNC(=O)C(c1ccccc1C)C)C1CC1 C(C(CNC(c1scnc1Cl)=O)C(F)(F)F)NC(COCP(C)(C)=O)=O N1(C(CC(CC=C)NC(c2ccccn2)=O)=O)CC2(C1)CN(C)CCO2 C#CCC(C)(C)CNC(=O)C(O)C1CN(C(=O)C(c2ccc(C)o2)C)C1 C1(C)(CNC(c2cn(C)c(O)n2)=O)CCN(C(=O)C(O)C(F)(F)F)CC1 c1(OC)ccc(OC(F)F)c(CNC(C2CN(C)CC2C(F)(F)F)=O)c1 Cc1cnc(NCC2(C)CC=CCC2)c(S(=O)(=O)N2CCN3CCCCC2C3)c1 Cc1ccc(I)cc1C(=O)NCC1CCC(C(=O)N(CC#N)CC#N)CC1 c1(CN2CC(CC(=O)Nc3cc(F)ccc3I)OCC2)ccnc(Cl)c1Cl N1(C(c2c(N(C)C)nccc2)=O)CC2CCN(C(=O)Cc3c[nH]nc3O)C(C2)C1 N1(C(CNC(C)=O)=O)CC2CC1CCC2NC(=O)C=CC(C)(C)C C1(CNC(c2c(CC)ocn2)=O)C(C)CCCN1C(c1cn2ccnc2s1)=O Cc1ccc(S(=O)(=O)N(C(C2CCC(O)C2O)=O)Cc2nnn(C)n2)cc1 Cc1cc(CC(=O)N(CCC(C)NC(C2CC2C(C)(C)C)=O)C)nn1C N1(C(=O)OC(C)(C)C)CC2CC(NC(c3ccc(-c4ccsc4)cc3)=O)C1C2 C1(CNC(C2(C(C)C)COC2)=O)CC2COCC2N1C(C1COC(=O)O1)=O C12(NC(CCCCOC)=O)CC(CNC(c3c(Br)cnn3C)=O)(C1)OC2C c1(SC)nc2ncnc(N3CCC(NC(c4csc(C(C)C)n4)=O)C3(C)C)c2s1 C(CCCN=c1nc2c(ncn2C)c(N(CCCn2ccnc2)C)[nH]1)=CC CC1CC(C(=O)N(CC(O)CNC(=O)CCCn2cnc(C#N)n2)C)CC(=O)N1 N1(C(C2(C=O)CCC2)=O)CCCCC2(C1)CN(C(=O)Cc1nnc(C)s1)C2.CN c1(C(=O)NCC(C)C2CC2)ccc(O)c([N+](=O)[O-])c1.C(=O)C(F)C1CC1.N C=CCC(C)(C)CC(=O)NC1C2CCC1CN(C(=O)C(C1CCCO1)C1CC1)C2 c1(C(N2CC(CNC(C(C=CC)O)=O)OCC2)=O)cc(Cl)c(F)cc1C CCCCC(CC)C(=O)NC1(C)CCOCC1.C1(C(=O)NCC)CCS(=O)CC1.N C=CC(CCC)CC(=O)N1CC(OCCC(=O)N(C)CCN2CCOCC2)C1 CC1(C(=O)Nc2cncnc2Cl)CCCN1C(c1cccnc1F)=O Cc1cccc(C(=O)NCC(C)CC(=O)N(C)CC2CCN(C)C2)c1 C(=O)(C1=NN2CCCN=C2N1)NC1CCC(NC(=O)CC2(O)CCCC2)C1 c1(CNC(=O)NCC(C)(C)n2cccn2)coc(-c2ccccc2)n1 C1(NC(c2cn3c(n2)SCC3)=O)CC12CCN(C(c1nn[nH]c1Cl)=O)CC2 c1(CC(=O)N)ccccc1.C(C(O)C)NC(COCC(C)C)=O.c1ccsc1 C1(C(=O)NCC2CCCCN2C(C23CC(CO2)C3)=O)CCS(=O)(=O)CC1 C1(CCNC(c2nc(CCC)oc2)=O)C(C)CCCN1C(=O)Cn1cnnn1 N1(C(C(C=C=C)C)=O)CCC(CNC(c2cn(CC)cn2)=O)C(F)(F)C1 Cc1c(NC2COCCOC2)ncnc1N1CCC(C(F)F)C1 N1(C(COCCC=C)=O)CCC(NC(c2cc(OCC)ns2)=O)C(C)C1 c1(C=O)ccc(N(C)C)c(F)c1.C=CCCCNC(=O)CCc1ccn(C)n1.N Cc1nnc2n1CCCC2C(=O)NC1CC2CCC1N2C(=O)Cc1ccccc1 c1(C(N2C(C)CCC(NC(CC=CCC)=O)C2)=O)nc(CC)n2ccccc12 c1(C(=O)NCCOCCNC(c2conc2C2CCCC2)=O)ccnnc1Cl c1(C(N2CCC(F)(C=O)C2)=O)ccc(C)c(C#N)c1.C(=O)(CCC(C)C)NC.N C1CN(C(C2(c3cccs3)CC2)=O)CCC1(F)F.C1(CC(=O)NC)(OC)CC1 Cc1cc(CNC(C2CN(C(=O)C(F)(F)C(F)F)CCS2)=O)ccc1I N1(C(C(C2CCC2)OCC)=O)CC=CC1(C)C(=O)NCc1cn(CC)nn1 C(=O)(C(F)CCC(C)(C)C)N(C(C)C(=O)NCc1cn(CC)nn1)CCC CN(C)S(=O)(=O)NCC=O.C1(CCC)CCCN1C(=O)CCN1CCC(F)C1.N C(CC1=CCc2ccc(OC)cc21)NC(c1ccc(OCC)cc1F)=O c1(NC)ncccc1C(=O)NC1CC(C)N(C(c2cccc(CS(C)=O)c2)=O)C1 C(=O)(C(C(C)(C)C)NC(C1CCCN(C(c2ncc(Cl)cn2)=O)C1)=O)NC n1(CC)ncc2c(N3CCC(C)=C(Br)C3)[nH]c(=NCCc3c[nH]c(=N)s3)nc12 c1(C(N2CCC3(C(NC(CC(CC)CC)=O)C3)CC2)=O)sc2ccccc2c1Cl C#Cc1cc(C(=O)N(C2CCN(C(=O)C(C)(C)c3cscn3)C2)C)ccc1Cl C(=O)(CCCNC(=O)C(CC)SCC)NC(C=C)C1CCC1 c1(N2CCC(N(CC)CC)C2)cccc(S(=O)(=O)NC)n1.c1cc(F)ccc1Br N1(C(CN(CC(C)C)C(=O)CC2C=NN(C)C2=O)=O)CCN2CC(O)CC2C1 c1(C(=O)NCC2(O)CCN(C(C3CCS3(=O)=O)=O)C2)cc2c([nH]1)CCOC2 CC1(C)CN(C(c2ccnc(O)c2F)=O)CCC1C(=O)NC1CCCC1O CC1CC(CC(N2CC3CN(c4nnc(C(C)(C)C)s4)CC3C2)=O)CC(C)(C)C1 N1(C(C2ON=C(CC)C2)=O)CC2CN(C(=O)CCOCC(F)F)CC(F)(F)C2C1 Cc1csc(=O)n1CC(=O)N.c1(C=O)cccc(C2(C)CC2)c1.C(C)C1CC1 C1(CCNC(C(CC)C)=O)CSCCN1C(=O)C(C)N=[N+]=[N-] C(=O)(C(F)(F)C(O)CC)NC(C=CC(=O)NCC(CCC)O)C C1(NC(=O)C(F)C(F)(F)F)CS(=O)(=O)C12CCN(C(C1CCCC1O)=O)CC2 CN1CCCC(N(C)C(C2(F)CCN(C(=O)C=Cc3cncn3C)C2)=O)C1 c1(C(=O)NCCCCC2CN(C(C(C)NC(N)=O)=O)C2)ccc(Br)o1 CCCCC(C)(F)C(=O)N1CCCC(O)(CCNC(c2sc(F)cc2Cl)=O)C1 c1(C=O)ccccc1.c1(CSCC)cc(C(=O)NC2CC2)no1.C(C)C c1(C(=O)NC2CN(C(C3(C)N(C(C)=O)CCC3)=O)CC2C)ccn2nccc2c1 CC(C)C(CNC(=O)CCc1ccsc1)NC(C1(Br)C(C)C1C)=O N1(C(CCNC(C)=O)=O)CC(C(=O)N(C2CCCCCC2)C)CC(C)C1 CCCCC(O)C(C)C(=O)NC(C1CCCN1C(C1CCC(O)CN1C)=O)(C)C Cc1oc(-c2nc(-c3cc(SC)ccn3)nn2CCF)cc1Cc1ccncc1 C1(NC(=O)Cc2cn[nH]c2)C2CC1N(C(C1(c3cccs3)CCCCC1)=O)C2 CCC(C(=O)N1CCC1C1CCCCC1)N(C)C(c1ccc(SC)o1)=O CS(=O)(=O)c1ncc(C(=O)NC2CCCN(C(=O)C(F)F)CCC2)s1 N(C1CN(C(c2cnc(C(F)F)s2)=O)CCc2ccccc21)C(c1ccoc1)=O C(=O)(C(C)S(C)(=O)=O)N(C(CC)C(=O)NCC(C)CC1CC1)C N1(C(c2nnn(CC)c2C)=O)C2CCC(C(=O)NCCN3CCC3)C1CC2 Cc1c(-c2nc(-c3ccccc3N3CCCC3)no2)cnn1CSc1ccco1 CCC(CC(=O)NCC1(O)CCN(C(=O)C=Cc2ccsc2)C1)C1CCC1 N1(C(C2(F)CC2)=O)CC(O)(C2(C(=O)NC)CC2)C1.C12CCCC1CC2.C C1(NC(C2(CC#N)COC2)=O)CCN(CCNC(C2C=CCC2)=O)CC1 C1(C(N2CCC(COC)C2)=O)CCOCCN1C(=O)COC1(C)CCCC1 C1(NC(CCc2c(C)n(C)nc2)=O)CN(C(=O)CC2C=CCCC2)CCC1F C1(CN(C(=O)CCCc2cccc(Cl)n2)C)CCN(C(c2c[nH]c(=N)s2)=O)CC1 C1(NC(c2cc(O)ncn2)=O)CCCC12CN(C(C1(n3cnnn3)CC1)=O)C2 c1(C(N2CC3OC(=O)N(C)C3C2)C(=O)NC)cn2c(n1)CCCCC2 Cc1cc(=NCC2CCCC(F)C2)[nH]c(=NCc2ccc(CO)cc2)[nH]1 C(=O)(CC(CCCC)NC(=O)CC(O)CC(C)C)NC(C1CCCC1)C#C CC1(NC(=O)CCn2ncc3ccc([N+](=O)[O-])cc23)CCc2ccc(Br)cc21 N1(C(C2CC(N=[N+]=[N-])C2)=O)CCCC(C2CN(c3ccn4c(Br)cnc4n3)C2)C1 c1(OC)cc(C)c2c(c1)C(NC(=O)Cc1cc(C)cc(C)c1)C(=O)N2 n1(CC)ccc(C(=O)NCCN(C(=O)CSCC(=O)O)C(C)C)n1 CCCC(C)CC(=O)NC(Cc1cnc[nH]1)C(=O)NCCC(=O)NCC c1(C(N(C2CN(C(C(CCC)F)=O)CC23CC3)C)=O)cc(C)c(C#N)c(C)c1 C1(C(N(CC(O)CO)C)=O)C2CC(O)C(C2)N1C(c1cc(C#N)cs1)=O S(=O)(=O)(c1ccccc1C(=O)O)N1C(CC)CC(C)C1 C1(NC(=O)CS(=O)C(c2ccccc2)c2ccccc2)CCC2CCCC1O2 N1(C(c2cnc(CCC)s2)=O)CCCN(C(c2cccc(CO)c2)=O)CC1C Nc1cc(C(=O)NCC2CCN(C(=O)CCC3CCCOC3)CC2O)cnc1Cl c1(C(=O)NCC(C2CC2)NC(C(C)c2ncco2)=O)cc(C2CCOCC2)no1 N1(C(c2c(CC)cco2)=O)CCCC(C(N2CCC3CC23C)=O)CC1 c1(C(N(C(CSCC)=O)CCC2CC2)=O)nc(Br)sc1C c1(C(=O)NCCCN(C(c2cc(C)n(C)c2)=O)CC)cn2c(C)nnc2cn1 N1(Cc2ncn(C)n2)CC(=O)N(C2COC(=O)C2)C1=O C=CC1(c2cn(CCO)nn2)COCCN1C(=O)CCNC(C)=O N1(C(C(CC)C)=O)CC(CNC(C2(O)CC2)=O)C(C(F)(F)F)C1 c1(C(=O)NC(C(C)NC(c2cncc(COC)c2)=O)C)cnc2ccoc2c1 C#CC1(C(=O)NC23CC(F)(C2)C3)CCN(C(c2cnc(C)cc2C)=O)C1 C1(C(N2CC(c3cn(C(C(=O)OCC)C)nn3)(O)C2)=O)C2CC(=O)CC12 c1(C(N(CC(=O)NC2CCC2)C)=O)ccc(O)cc1.C(=O)C(F)=C1CCC1 Cc1ccc2c(C(=O)NC(C3(O)CCN(C(=O)C(C)(C)CO)C3)C)onc2c1 Cn1c(=N)[nH]c2cc(C(=O)NCC(C)(C)NC(=O)C3CCc4c[nH]nc43)ccc12 N1(CCC)C(=O)CCC1C(=O)N(C1CCN(C(c2ccncc2Cl)=O)C1)C N1(C(=O)N=c2[nH]nc(-c3cccc(F)c3)s2)CCC2(CC1)COCCO2 C1(C(=O)NCCCN(C(=O)CCc2nccn2C)C)C2COCC12 C(=O)C(=O)CC(=O)c1ccsc1.C1(C(F)(F)F)(C(=O)NCCC)CCCC1.N N1(C(c2c(CC)onc2)=O)CCN(C(=O)Cn2cccc2)CC12CCC2 N1(C(=O)COC2CC=CC2)CC2(CCN(C(C34CC(O)C3C4)=O)CC2)C1 c1(C(=O)NC2(CC=C)CN(C(=O)C)C2)cc(=O)c(O)co1.C(C)(C)CC C1(NC(C=C(C)c2cccs2)=O)CCN(C(=O)C=CC=C(Cl)Cl)CC(O)C1 CC(C)CC(O)CC(=O)N1CCCOC(CNC(c2cc(C(C)(C)C)c[nH]2)=O)C1 N1(C(c2c(C(C)=O)coc2)=O)CCCC(n2cc(-c3cccnc3C)nn2)C1 CC(C)C(F)(CNC(=O)COc1ccsc1)C(=O)N1CC2COCC2O1 CC1CN(C(=O)C(F)C2CCC2)CC1CCNC(c1cnc(-c2cccs2)o1)=O c1(C=O)ccnc(S(N)(=O)=O)c1.c1(OC)csc(C(=O)NC(C)C(C)C)c1 O=C(N=c1ccnc2[nH][nH]cc1-2)C1CCN(C(=O)Cc2cc(Br)ccc2Br)C1 c1(C=O)cc([N+](=O)[O-])c(C)s1.C#CC1(C(N2CC(CC)C(C)C2)=O)CCCC1.N N1(C(c2cccc(OCCOC)c2)=O)CCCC(NC(=O)CC(C)F)C1C C(=O)(CCC(=O)OCc1cc(-c2ccccc2)on1)OC(C)C c1(C(=O)NC(C(C)NC(CC(C)F)=O)(C)C)cccc2oc(=N)[nH]c12 c1(C(N(CCCNC(C=CC)=O)C)=O)ccnc(O)c1 N1(C(c2c(C)occ2)=O)CCCC(C2CCCCN2C(c2ccc(CO)o2)=O)C1 c1(C=O)ccc(S(N)(=O)=O)cc1.N1(C(C(C)C)=O)CCCC12CC2.C(=O)(C)N C1(C(=O)OC)(COC(c2cn(Cc3ccccc3)nn2)=O)CN(CCF)C1 C1(C(=O)NCc2c(OC)cccn2)CN(C(=O)C(CO)OC)CCN1C CCC(C(=O)N1CCC(C(=O)NC2CCCC3(CCC3)C2)O1)SC C(=O)(CC(C)(C)C#N)NCC1(O)CC(C(N(CC=C)C2CC2)=O)C1 c1(C(N(CCCNC(C(C)c2cccs2)=O)C)=O)cnn2c1OCC(O)C2 C(C(=O)NCc1cccc(Cl)c1)(C(C)CC(C)C)N1CCC(O)(CCC)CC1 C1(C#N)(C=O)CC1(C)C.C1(CN(C(=O)CC2CCC2)CC#C)CCCO1 N1(C(C2CCC(=O)NC2)=O)CCC2CCN(C(=O)C=Cc3cnc[nH]3)C2C1 C(N=c1nc(O)c2cnn(C)c2[nH]1)c1c(OC)cc(N2CCCCCC2)cc1 C1(NC(C(CSC)C)=O)CCC2CN(C(=O)CCCCCCN=[N+]=[N-])CCC2C1 C1(CNC(C2CCC(F)(F)CC2)=O)CC12CCN(C(=O)C)CC2.C1CC1.C N1(C(c2csc(-c3ccc(F)cc3)n2)C(=O)NC)CCC(C)C1CC C1(C(N2CC(C(=O)NOCCF)(CC)C2)=O)CC1C1CCCC1 N1(C(C=COCC)=O)CC2CCCCN2CC1CNC(=O)C(C)(CC)CC c1(C(N2CC(N(C(CCCC=C)=O)C)C(C)(C)C2)=O)ccc2nc(O)[nH]c2n1 CS(=O)CCC(=O)NCC1CC(O)CN1C(c1ccccc1)=O.C(=O)C=NO.N N1(Cc2cc(C)sc2)CCC(O)(C(N2CCCN(C)CC2)=O)CC1 c1(CNC2(CNC(c3ccc(SC)s3)=O)CC2)ccccn1.c1ncc[nH]1 c1(N(Cc2c(OC)cccc2OC)Cc2ccccn2)cc(Br)c(C)nc1O N1(CC(=O)N)C(=O)C(=O)N(C)C1=O.Cc1cncc(C(=O)NCC(C)C)c1 C12CC(C(=O)O)CN(C1)C2=O.CC1CCC(CCC(=O)OC(C)(C)C)O1 CN=c1[nH]c(C(N2CCCCC2C2(NC(=O)C3=CCCS3)CC2)=O)cs1 N1(C(c2cc(C)c(C)[nH]2)=O)CCCCCC1C(=O)NC(c1nc[nH]n1)C1CC1 N1(C(Cc2cc(C)no2)=O)CCN(C(C2CC2C)=O)CC1C(F)F C(=O)(CCCCC(C)(C)C)NCC1C(NC(c2c(NC)c(F)ccc2)=O)C1 O=C(C#CC12CC3CC(CC(C3)C1)C2)NC1CCC(O)CN(C(C2CCO2)=O)C1 Cc1ccc2nc(NC3CN(C(C4CC5(CCOC5)C4)=O)CC3(C)C)sc2n1 Clc1ccc2[nH]c(-c3nc(-c4ccncc4)nn3C3CCOC3)cc2c1 C#Cc1cccc(C(=O)N(C)CC2(NC(=O)C(N3CCCCC3=O)C)CC2)c1F CCC(C)C(C(=O)NCc1c(C)n[nH]c1C)NC(=O)CCc1ccn(C)c1 C(=O)(CS(=O)(=O)C1CCCC1)NCC(CN(C(C1CN(C(C)=O)C1)=O)C)O N1(C(CCC(=O)NC)=O)CC2CCC1CN2C(c1ccc(Cl)cc1C(F)(F)F)=O c1(C(N2CCC(O)(C(C)NC(CC(=C)C)=O)C2)=O)cc(F)c(F)c(Cl)c1F C1(C(N2CC(CNC(C(C)C3CCC3)=O)C2)=O)CC12CC(O)C2 C(=O)(CCC(C)(C)[N+](=O)[O-])N1C(C(=O)NCC2CC(=C)C2)C(C)OCC1 N1(c2cc(C)ncn2)CCC(O)(C(N2CCC(C(C)(C)O)C2)=O)CC1 c1(CN2CCCC(C(=O)OCc3cn4ccnc4s3)C2)ccc([N+](=O)[O-])cc1Br C(=O)(C1CCCc2nnn(C)c21)NCC(CC)(CC)NC(=O)C=Cc1ncc[nH]1 C1(C2CCCN(C(C3C=CCC3)=O)C2)(NC(=O)C=Cc2cccc(Cl)c2)CC1 c1(C(CO)NC(c2cccc(NC(C(N)=O)=O)c2)=O)cccc(F)c1F C(C1=CCN(C(=O)CCCCN(C)C)CC1)NC(c1c(C)scc1)=O c1(C(=O)NC(CNC(C(C(=O)OCC)(C)F)=O)CC)cccn2ccnc12 N1(C(CC2(OCC)CCC2)=O)CCN(C(=O)C2=NOC(C)C2C)CC(O)C1 C1(O)CCC(C)(C)C1.C=C1CC(C=O)(CNC(=O)CCc2nccs2)C1.N C(=O)CN=c1[nH]c(C)cs1.N1(C(C2(OC)CS(=O)(=O)C2)=O)CCCC(C)(C)C1 CCC(CNC(C1(C(C)C)CCN(C(=O)C(C)CCOC)C1)=O)CC(C)C Cc1cc(C)c(C(=O)NC(C)(C)CNC(c2cnc(CC(C)C)[nH]2)=O)o1 c1(C(=O)NCC(C)CN(C(=O)C(C)n2cnnn2)C)ccc(F)c2ccsc12 C1(N(C(=O)CC2CSCCO2)C)CN(C(C2(Cl)CCC2)=O)CCC1O CCC(C)C(=O)NC1CC(CNC(C2(n3cccc3)CCCC2)=O)C1 c1(-c2cn(C3CC(C(N4CC(CC)C(C)C4)=O)C3)nn2)ccc(C(C)=O)c(O)c1 Cc1cc(C)nc(N2CCN(CC(=O)NCCCN3C(=O)C=CC3=O)C(=O)C2)n1 c1(CC)ncncc1C(=O)NC1CC(N(C)C(c2cc(C(F)F)ccn2)=O)C1 CCCC(CCC)C(=O)N(CC(C)C(N1CC(N=[N+]=[N-])C1)=O)C CC(C)CC(C(=O)N1CCC(C(F)F)C1)N(C)C(C1CC(O)C1)=O CCCC(C)(CC)C(=O)NCC12CC(C1)C2.c1(CC(=O)N)cc(C)ccc1C C(=O)(C(O)CC(C)(C)C)N.C1(C(=O)NCCCC)CC(C(F)(F)F)(OC)C1 N1(C(c2c(CNC(c3cnc(SC)n3C)=O)nccc2)=O)CCCC(C)C1CO c1(NC(C2CCN(C(=O)C=C(C3CC3)C3CC3)O2)=O)cccc([N+](=O)[O-])c1 Cc1cc(F)c(C(=O)NC2CCN(C(C3CCC4CCCCN34)=O)CC2)c(Cl)c1 c1(OCC)cc(C(=O)NC2CCN(CCn3cc(Cl)cn3)C2)ccn1 C1(NC(C2C(NC(c3sccc3F)=O)CCCC2)=O)CCC(C2CC2)CC1 C1(C(N)=O)(NC(C2CC(N(C(C(N3CCOC3=O)C)=O)C)C2)=O)CCCCC1 Cn1nnc(C(=O)NCC2(CNC(c3cscc3Br)=O)CCC2)c1N C(=O)C(C#N)C(C)(C)C.c1ccc(C)cc1C(N1CCC(C)CC1)=O.CCCC(C)C CCC(CCCC(=O)NC(CC1CCCC1)CO)NC(c1cnc(C)nc1)=O C(=O)(C(O)CC(F)(F)F)N1C(CNC(C2CC=C(C)CC2)=O)CCC1 c1(N2C(C(N3CC4C(C3)C4(F)F)=O)CC(OC)C2)ncnc2[nH]c(C)nc12 c1(OC)ccc2c(c1Br)CCN(C(=O)COc1ccc(S(=O)(=O)NC)c(Cl)c1)C2 c1(C(=O)NC2CC(NC(C(CC#C)C)=O)C2)cnn2c1CCCC2 c1(C(=O)NCC2N(C(C(C)O)=O)CC(C)(C)OC2)c(Cl)ccc2cccnc12 CCC(CC(=O)N(C(C)(C(=O)NCCCN1CC=CC1)C1CC1)C)OC N1(C(C(C(CC)C)O)=O)CCCC12CCCN(C(C1CC(F)(F)C1)=O)C2 c1(C(N2CC(NCc3cnc(CC)s3)C3(C2)CC3)=O)cc(Br)cc(F)c1C c1(NC2(CC=C)CCNCC2)c(C)ccc([N+](=O)[O-])c1C c1(C(N2CC(NC(c3cc(F)c(F)c(F)c3)=O)(CO)C2)=O)cccc2c1OCO2 C(=O)(CC1COc2ccccc21)NC1C(C)N(C(=O)Cc2ccccc2F)CC1 c1(NCc2scc(COC)c2)ncccc1S(=O)(=O)N1CC2C(C1)C2(C)C C1(N(CC(=O)Nc2nnc(C(CCC)C)s2)C)CCC2COC1O2 C(=O)(C(C)(C)C(C)(C)C)NC.N1(C(C)=O)CCC(C)(C(=O)N)C1.C1CC1 Cc1ccn2c(C(=O)NC3CCCCN(C(=O)CC(C)C4CC4)C3)cnc2c1 C1(CC(=O)NC(CC#C)Cc2ccccc2)(CN(C)C)CCCCC1 C1(CC)(CNC(=O)C(C)C(=O)C)CCCC1.C(C)(C)C.N(C)C=O.O N1(C(C(CC)=CC)=O)C2CCC(C2)C1CC(=O)NCC(=O)NCCO C(=O)(C#CC1CCCCC1)N1C(C)CCC(CNC(CCC(=C)Cl)=O)C1 C1(C(=O)NCC2CN(C(c3c(NC)cnnc3)=O)C2)CCc2nc(O)[nH]c2C1 N1(C(C(CCSC)O)=O)CCN(C(C2CCS(=O)(=O)N2)=O)CC1C C1(CNC(C(CC=C)(C)C)=O)CC2CCC1N(C(=O)CN1CC(C)(OC)C1)C2 c1(C(=O)N)nnn(CO)c1N.c1ccccc1.C(F)(C(=O)NCC(C)C)=CC Cc1ccc(C(=O)OCC(N2CCN(C)C(=O)C2)=O)cc1-c1cnn(C)c1 CC1CCCN(C(=O)C(N2CCC(NC(=O)CSCC3CCCCO3)C2)=O)C1 C1(C(CNC(C2(CC#C)CCC2)=O)F)CCN(C(C2CCC(CC)CC2)=O)CC1 N1(C(CSC(C)C)=O)CCC(O)(CNC(=O)CC2OCCC2C)CC1 C(C)(C(C)C(=O)NCC1(CC2CC2)CC1)NC(CCC=CC)=O C1(CNC(c2c(OC)cccc2)=O)CN(C(=O)C(C)(C)C2CCCO2)CCCO1 c1(C(=O)NCc2c(OC)ccc(C)c2)cc(C)nc2cc(C(F)(F)F)nn12 Cc1ccc(OC(C)C(=O)NCC2(O)CCN(C(C3(C)CSC3)=O)C2)cc1 C#Cc1cccc(CNC(=O)C(CCC2CC2)NC(=O)CCS(C)(=O)=O)c1 N1(C(c2c(CC)nns2)=O)CCCCC1CN(C(c1cccn1C)=O)CC c1(CC(=O)NC23C(CN(C(CCC(=C)Br)=O)C2)C3)ccc(OC)c(Cl)c1 c1(C(N2CC(N(C(=O)C(N)=O)C)C(O)C2)=O)ccc(C2CC2)c(Br)c1 c1(CC(C(=O)OCC)NC(c2ccc(OC)cc2)=O)ccc(C)cc1 Cc1cccc(C=CC(=O)NCC2C=CCN2C(c2c[nH]c(C#N)c2)=O)c1 C1(C(=O)NCCSCC(=O)NC(c2ccncn2)C)CCCCNC1=O CCCC(C#N)C(=O)N1CCN(CCNC(c2cn(C)c(C(F)F)n2)=O)CC1 N1(C(C(C)NC(C)=O)=O)CC(C(=O)NC2(C)CC(C)(C)C2)C(F)(F)C1 S(=O)(=O)(c1ccc(C#N)c(C)c1)NC(Cc1c(C)cccc1)CO c1(CNC(C)=O)ccc(S(=O)(=O)NCc2c(F)cccc2Cl)s1 Cc1cc(C(=O)NC2CN(C(=O)CCC[N+](=O)[O-])CC2C)nc(C)c1 N1(C(C2C(OCC)C2)=O)C2CCC1CN(C(c1c(C)cc(C)nc1S)=O)CC2 C1(C)(C(=O)NC(C)CCCO)C=CCN1C(=O)C=Cc1ccncc1 C=CCN=c1[nH]cc(C(=O)NC2(C)CCCC2)s1.C12(C(=O)N)CCCC1C2(F)F C1(C(=O)NC2C(NC(C3CN4CCC3CC4)=O)CC2)CCc2nnc(O)n2C1 c1(C=O)cc(C)c(C)nn1.C12(C(N(CCC)CC)=O)CCCC1(C=O)C2.N N1(C(c2c(C)coc2C2CC2)=O)CCCC(C2CCCNC2)C1 N1(C(CCN(CC)CC)=O)CCC2(CC1)CC2.C1(C=O)CC2(C1)CC2(F)F.C c1(NC(CN(CCc2ccc(F)cc2)CC)=O)coc2c(Cl)cccc12 c1(OC)ccc2c(c1)CCCC2Cn1nnnc1N1CCC(c2nncs2)CC1 C(=O)(C(C)CC(F)F)NCC(C(=O)N(CCC#C)C)(C)C C1(C(=O)NC2(C(N3CC=C(C)CC3)=O)CCCC2)CC2(CC2)CN1C C1(CNC(C(C#N)C2CC2)=O)(C)CCCCC1.C1(C=O)CC(=C2CC2)C1 c1(OC)cc2cc(C(N3CC4C(C(N)=O)C4C3)=O)[nH]c2cn1 Cc1cc(C)c2[nH]c(C(N3CC(O)CC3CNC(c3coc(C)n3)=O)=O)cc2c1 C(=O)(C(=O)NOC)N(CCOC)CCNC(c1cc(C)cs1)=O c1(C(=O)OC)cc([N+](=O)[O-])c(C)cc1NC1CCC2C(C1)C2(F)F c1(OC)ccc(OC)c2sc(=NC(C)CN(C)C(C3COC(C)C3)=O)[nH]c12 c1(CC)cc(C(N2CC(CCNC(=O)CC(C)(C)COC)C2)=O)c(C)nn1 C1(NC(=O)C(=O)NC(C2CCCCC2)C2CCC2)CC12CCC(F)(F)CC2 N1(C(c2ccnc(C(C)C)n2)=O)CCC2(CC2NC(=O)CS(C)(=O)=O)C1 N1(C(COCCC=C)=O)CCC2(CCCC2CNC(c2ocnc2C)=O)CC1 Cc1c(C(=O)NCCCCC(C)NC(=O)C(F)C2CCC2)cnn1CC(C)C C(=O)(C1CCc2c[nH]nc21)N(CCOC)CC.C1(C)(C=O)CC2(CCC2)C1.N N1(C(c2ccc(C)n2C)=O)CCC2(CCN(C(=O)C(O)CC(F)(F)F)CC2)C1 N1(C(C(C(CCC)NC(=O)C(N2CCCCC2)C)O)=O)CC2OCCN(C)C2C1 N1(C(c2c(NCC)scn2)=O)CCC(C)C1.C1(C=O)CSCCN1C(C)=O.N Cc1nc(C(F)(F)F)c(C(=O)NC2CC(C)N(C(=O)Cc3cnsc3)C2)n1O CC1CC(NC(c2ncc(F)cn2)=O)CN1C(=O)CCc1csc(=N)[nH]1 CCC(CCCC(=O)N1CC2CC1C2)NC(c1cncc(NC)n1)=O C1(C(N(CCn2cc(C3CCC3)nn2)CC)=O)CC2(CC(=O)C2)C1 C(=O)(C1=CC(O)C(NC(C2CCC3(CC2)CC3)=O)C1)NCC(C)OC CC(C)C(O)C(=O)NC(C)C(CO)NC(c1ccncn1)=O Cc1c[nH]cc(C(N2CC(C)(C)CC2CNC(=O)CC2CCNC2=O)=O)c1=O CC1CCCCC1CC(=O)NCC1CCC(N(C(=O)C(F)=C2CCCC2)C)CC1 c1(C(=O)NCC(C2CC2)NC(c2cccc(C)c2N)=O)cnn2c1OCC(F)C2 C(=O)(C#CC1(C)CCCO1)NC1C2(CN(C(Cc3c(C)ncnc3C)=O)C2)CC1 c1(CN(C2CCCN(C(c3c(OC)nsc3)=O)C2)C)nccn2ccnc12 c1(CC)ccc(C(=O)NC2CC3(C2)CC3NC(=O)C(C)CCC)c(F)c1.O c1(C(=O)N)cc2cccn2cn1.c1(CC)cccc(NC(C2(C)CC=CC2)=O)c1 c1(C(=O)NCC2CN(C(C(C=C)O)=O)C(C)(C)C2)cc([N+](=O)[O-])ccc1CC c1(OC)cccc(NC(C2OCCC2C)=O)c1O.C1(C=O)CC2(CCO1)CC2.N C1(CC=O)CC2(C1)CN(C(=O)CC1CCCC1C)C2.C1(C(=O)OC)CC1.C C1(N(c2ccc(C(N)=O)cc2)C(C)C)CCCN(C(c2ccc(Cl)s2)=O)C1=O Cn1cnc(C(N2CCC3C(NC(=O)Cc4c[nH]nc4O)CC23)=O)cc1=O C(=O)(CC(C(F)F)C(C)(C)C)N(CCCNC(C1CC(O)(C#N)C1)=O)C N1(C(Cn2nnc(C)n2)=O)CCOC(C)(CNC(=O)Cn2cc(CO)nn2)C1 c1(OC)ncnc(N2CCCC(O)(CNC(c3cccc(Cl)c3Cl)=O)C2)c1C N1(C(C(C)SC(C)C)=O)CC(C2CN(C(=O)C(C)(F)C(C)(C)F)C2)C1 C1(NC(c2c(OC)ccc(C)c2)=O)CN(C(=O)CCCC2CCC2)CC1C1CC1 C#CCC(CC(F)F)NC(=O)C=C(C)CNC(c1cncc(CO)c1)=O N1(C(c2nn(C)c(F)c2)=O)CCN(C(C2CC2(F)F)=O)C(C(C)(C)C)C1 c1(C(=O)NC2(CNC(Cc3scc(C)c3)=O)CC2)cnc2cc(C)nn2c1 CS(=O)(=O)c1ccc(-c2cn(C3CCN(C(=O)CSC4CC4)C3)nn2)cc1 N=c1nc(C(F)F)[nH]c(=NCC2CC(NC(c3nc(F)ccc3Cl)=O)C2)[nH]1 c1(CNC(C2N(C(C3(CC)CCC3)=O)CCC2)=O)ccc(Br)c(Cl)c1 C(=O)CC(C)C(F)F.C1(C(N2CCC(CO)(C)C2)=O)(COC)CC=CCC1.N CCC(CC(=O)N(C(C)CC(C)C)C)N(C(=O)CCN(C1CC1)CC)C n1(CC)cc(C(=O)NCC2(C)CCCC2NC(=O)CC=C(Cl)Cl)c(C)n1 c1(C=O)cc(C)nc(O)c1.C1(SC)CN(C(C2CC(C(C)(C)C)C2)=O)CC1.N N1(C(C2(NC(C)=O)CCC2)=O)CC2CC(O)C1C2.c1(C=O)ccc(O)cc1C.N N1(C(C=O)C)CCC(N(C(=O)CC2(C)CC2)C)CC1.C=CCNC(=O)N C=CCC(CC=C)C(=O)N1CC2(CCC(C(=O)Nc3cn(C)nc3C)O2)C1 c1(C(=O)N)cc2c(Cl)ccnc2s1.C1(NC(C2C(C=C)CC2)=O)CC2(C1)CCC2 c1(C(N2CC(C(=O)OC)CC2(C)C)C(=O)NC)cc(OC)c(OC)cc1Br c1(C(N(CCNC(=O)C(C(C)C)n2cnnc2)CC)=O)cc(F)c(N)cc1 C1(NC(C2(C)N(C)CCC2)=O)CC(F)(F)CC1NC(c1cc(N)cnc1Cl)=O N1(C(c2nc(C)sc2C)=O)CCC(CO)(NC(=O)C(C)Sc2ccccn2)CC1 Cc1cc(C(=O)N(C)CCN(C)C(C2CCN2C2CCCC2)=O)c(N)c(Cl)c1 C(=O)(C1=CCC(C)CC1)N1CCC(C(=O)Nc2c(C)nn(C)c2C)C(C)C1 c1(-c2c(C)ccs2)cccc2sc(C(=O)Nc3cc(C(=O)O)cc(C#N)c3)cc12 C(=O)(C1=CCOCC1)NCC1N(C(CCCOc2c(C)cccc2)=O)CCC1C C1(CNC(C2(N(C)C)CCCC2)=O)CCN(C(=O)C2=CCCSC2)C12CCC2 c1(C(=O)OCC(c2ccc(CC(=O)OC)s2)=O)cccc(=O)n1C C#CC1(C(N2CC(CO)(OCC)C2)=O)CCN(C(c2ccsn2)=O)C1 N1(c2cccc(NC(c3cccnc3N3CCCC3)=O)c2)CCS(=O)(=O)CC1 c1(C(c2nnnn2CC2CCOC2)NCC2(CC)CC2)ccc(F)cc1C Cc1cc(O)ncc1NC(=O)CC1CC2(C1)CN(C(=O)C(C)c1cc[nH]n1)C2 c1(C(N2CCCC(NC(c3cccc(C(F)(F)F)n3)=O)C2)=O)cc2sccc2s1 C1(CC(=O)N)CC(C)(C)CCO1.N1(C(C=C(C)C(F)F)=O)CCC(=CC)CC1 C12(NC(=O)CC3CCOC3=O)CCC(CC1)N(C(C1CCS(=O)(=O)C1)=O)C2 N1(C(Cc2ccc(CC)cc2)=O)CC(NC(=O)Cc2ccns2)CC1(C)CC N1(C(=O)CC2CCOCC2)CC(C(N2CCN(CCCO)CC2)=O)C(C2CC2)C1 N1(C(C=CCC)=O)CCC1CC(=O)N(C(C)CC1CC1)C c1(CC(N2CCC(C)C2c2cn(CCF)nn2)=O)cc(Cl)c(F)c(Cl)c1 C1(O)(CN(C(C(CC)O)=O)C)CCN(C(c2ncccc2N)=O)C1 C(=O)(CC(C)C(C)(C)NC(C1CC(N(C)C)C1)=O)NCC(CC#C)(C)CO C12(NC(C=Cc3ncn(C)c3)=O)CCN(C(c3ccc(Cl)c(O)c3)=O)CCC1C2 c1(CC)ncc(C(=O)NCC2CC(OC)CN2C(=O)C)cn1.CC(N)=O.S O(NC(=O)C1CC(=O)c2ccccc21)C(C(=O)OC)(C)C c1(CC(=O)N(C2CCN(C(C3CNC(=O)N3)=O)CC2)C)c[nH]c2ccc(Cl)cc12 C#CCCCCCC(=O)NCC(C1CCN(C(C2(C)CC2(F)F)=O)CC1)(C)O C(=O)(C(O)C1=CCCCC1)NCCC(CNC(=O)CC1CSCCO1)O C1(CNC(CC(=O)NCC#C)=O)CCC12CCC2.C(=O)C(=O)N(C)C.N Fc1cc(F)c2nccc(NC3CCc4cccnc43)c2c1 CCC(C(=O)OC)C(=O)NC(c1ccc(C)cc1)CNC(=O)CC1(C)CC1 CCCCCCC(CC)C(=O)NCC(C)(F)CNC(=O)CC1(n2ccnc2)CC1 N1(C(COCCC#C)=O)CCCC(C2CCN(C(C3(C)CCC(=O)C3)=O)CC2)C1 C#Cc1ccc(C(=O)NC2(CNC(=O)C(C3CCOCC3)C)CCC2)c(F)c1 Cc1ccc(C)c2c1CCCC2NC1CCc2nc(C(F)(F)F)cn2C1 CCC1=NOC(CNC(C2(NC(c3ccnc(O)c3)=O)CC2(C)C)=O)C1 c1(OC)nc(C)cc(=NC2CCCN(C(C3CCCC(C)C3)=O)C2)[nH]1 c1(CC)ccc2occ(C(=O)NC3CCN(C(=O)C(F)CC4CC4)CC3)c2c1 c1(C(N2CCC(C)C2C(=O)N(C2CCCCC2)CCO)=O)ccc2cncn2c1 Cn1c(C(=O)NCCC2(O)CCCN(C(=O)C(=O)N)C2)cccc1=O.CC(F)F c1(C(N2CC(C(=O)OCC)C(C(F)(F)F)C2)=O)cc2ccc(OC)cc2[nH]1 C1(C(=O)OCC)CCN(C(=O)C(=O)NC(C)C2CC2)C1 N1(C(CCC(C)NC(C23CCC(C2)C3)=O)=O)CCC2(CCCCO2)C1 CC1C(NC(C2CCOC2C)=O)CC2CCC1N2C(c1ccc2ncsc2c1)=O n1(CC)nnc2c1CCC(C(=O)NC1CCC1)C2.n1(C2(C=O)CC2)cncn1.N CC1=NS(=O)(=O)NC=C1C(=O)NC1CCCCC1.C(=O)C1=NN(C)C(=O)CC1.N c1(OC)c(-c2cnn(C)c2)cc(-c2nccn2C(CCF)C(=O)OC)cc1Cl Cc1ccc(C(N2CCC(CNC(C3CC3C)=O)CC2)=O)c(C)n1 C=C=CC(C)C(=O)NCC1CC1CC(=O)NC1CCOCC1C c1(C(=O)NC2COCCN(C(C3CC4CCCC4C3)=O)C2)n[nH]c2c1CCCC2 c1(C=O)ccc2c(c1)CCC=C2.c1(SC)cc(C)c(C(N2CC(CC)C2)=O)s1.N CCC(CNC(C1CC(N2CCCC2)C1)=O)(CC)NC(=O)CC1CC1C1CC1 n1(CC(=O)NCC2C(CNC(c3c(C)csc3)=O)C2)ccc(=O)cc1C C1(NC(Cc2ccc(OCC)cn2)=O)CCC2(CC1)CC2.C1(C=O)CCCS1.N c1(CC(=O)NC(c2cc(OC)ncc2)C)csc2nc(C)cn12 C1(N(C(C(C)SC)=O)C)CN(C(c2ccnc(C)c2)=O)CC12CC2 C=CCCC(C)(C)C(=O)NCCC(C)NC(c1ccn(C)c(=O)c1)=O C=C(C)CCC(C(=O)NCCC(=O)OCC)N1CC=CCC1 C1(C(=O)NOCC2CCC2)(CCC=C)CN(C(=O)Cc2occc2C)C1 C1(C=O)CCC(F)(F)CC1.n1(CC)cc(CCCO)nn1.CC(C)(C)OC=O.N N1(c2c(C)c(NCc3nc4c(s3)COCC4)ncn2)CCCC1C1CCCO1 C1(OCC)CCCCC1NC(=O)C#CCNC(c1sc(O)nc1C)=O CC1CCCn2c(C(N3CCC4(CCN(C(c5cc[nH]c5)=O)C4)C3)=O)cnc21 C(CCS(C)=O)(C(=O)NCCCNC(=O)C(F)(F)C(F)F)N(C)C C(=O)(C1CCCc2sccc21)OCC=CC.C1CCC(c2ccc(Cl)cc2)CN1 C1(C(=O)NC(C)CC(=O)N(CCn2cnnc2)C(C)C2CC2)CCC=CCC1 C(c1ccc(F)c(F)c1)=C(C)C(N1CCN(C(=O)CN2CCC2)CC1C)=O Cc1cc([N+](=O)[O-])ccc1C(=O)N(CC(C)NC(c1c[nH]c(C)c1)=O)C N1(C(c2c(C)ncnc2)=O)CCC(NC(=O)C=CC(=O)NC2CC2)CC1C Cn1cc(C=CC(=O)NCC(C2CCCN(C(=O)CCCC3CC3)C2)(C)O)cn1 C=CCCCCCCCCC(=O)N1CCN(C(=O)C(O)P(C)(C)=O)CC12CCC2 n1(CC(=O)NC(c2ccccc2)CNC(=O)CCn2cncn2)ncc(Br)n1 C(C)(C(CO)NC(=O)CCCc1cc(C)no1)NC(CCNC(COC)=O)=O C1(NC(CCC2CCN(C(c3c(CC)cccc3)=O)C2)=O)CCC(C#N)CC1 n1(CC)cc(Cl)cc1C(=O)NC12CC(NC(C3CC3C3CCC3)=O)(C1)C2 C1(C(=O)NC2C(NC(C(CC)SC)=O)CCCC2)CC2CCC1CC2 N1(C(CCC(=O)N(C)C)=O)CCC2(CCCN2C(=O)C=C(Cl)Cl)CC1 C1(NC(C(n2cc(C(C)CC3CCC3)nn2)C)=O)CCC2CC1CO2 C(CC(C)(C)C)(C(=O)N1CC(CSC)CC1C)NC(Cc1cn(CC)nn1)=O C(=O)(CCCCN(C)C(C1(C(=O)NC)CCC1)=O)NCc1onc(CC)n1 N(C1CSCc2ccccc21)c1cc(NCCc2cc(CC)no2)ncn1 CCCCCCCC(=O)NCC1(CC(N)=O)CCOCC1 c1(C(N2C3CC(NC(Cc4nc(C)sc4)=O)C2CC3)=O)c2c(nn1C)CCOC2 c1(C=O)cc2c(F)ccc(F)c2[nH]1.N1(C(C2C(C)(C(F)F)C2)=O)CC(F)C1.C c1(C(N(C(C)CNC(C2CCCCC2)=O)C)=O)cnc(Cl)c(N)c1 c1(N2CC(CC)(CC)S(=O)(=O)CC2)nc(=NC)[nH]c(=NCc2n[nH]c(=N)o2)[nH]1 C1(CNC(CCCC#CC)=O)CN(C(c2ccnnc2C)=O)CCC1(F)F CCCCC(CN=c1[nH]c(Cl)nc(C)c1F)NC(=O)C=Cc1ccccn1 N1(c2ncc(SC)cn2)CCC2CN(C(c3ccc(OCCO)cc3)=O)CC12 CC1C(NC(c2ccc3nn[nH]c3c2)=O)C(C)CCN1c1cc(O)nc(O)n1 Cc1cc(C(=O)NC2C3CC2N(C(c2ccc(F)o2)=O)C3)ccc1Br Cc1cc(C(=O)NCC(CC(C)C)NC(C2CCC2)=O)cc(Br)c1 c1(NC(c2ncc(OC)nc2)=O)nc2c(s1)CC(NC(=O)C(C)(C)F)CC2 C1(N(C(c2n(C=C)nnc2)=O)C)CN(C(C2CC2OC(C)=O)=O)CCC1C C1(NC(C2(C(C)C)COC2)=O)CCN(C(=O)Cc2cnn(C)n2)CC1F C1(CCC)CN(C(C23COCC2C3)=O)CCN1C(=O)CCc1ccc(O)nc1 [N-]=[N+]=NC1CN(C(C2CC2F)=O)CC1NC(C1(CC2CC2)CCC1)=O N1(C(CCc2scc(C)n2)=O)CC(NC(c2cccc(N)c2)=O)CCC1C Cc1nc2ccc(C(=O)NC3CCC(CNC(=O)CCc4cnc[nH]4)C3)cc2s1 C1(CC=C)(CCn2cc(CCCC(C3CCC3)=O)nn2)CCOCC1.CC(=O)O.S c1(CC(=O)N(C2CCN(C(=O)CSCC(C)C)CC2)CC#C)cnccc1Cl C(=O)(CCC(=O)c1ccc(Cl)cn1)NCC(CC=C)NC(C1CC2CC1C2)=O CN=c1nc(CC(=O)O)[nH]s1.c1(C2CCCC2)ccc(Cl)cc1 N1(C(c2c(OC)scc2)=O)CC(OC)CC1(C)C.C(c1csc(C)n1)=CC=O c1(C(=O)OCC)ccc(F)cc1NC(=O)CC1CCC(F)(F)CO1 N1(C(Cn2cnc(=N)[nH]2)=O)CCOC(CNC(c2scnc2C(F)F)=O)C1 C(CC(=O)N(C)C(c1cccs1)C)(C(F)(F)F)NC(C1C(OC)CCC1)=O c1(C(=O)NC(C(=O)N(C(C(=O)OC)C)C)Cc2cc[nH]n2)cnc(N)cn1 N1(C(c2cnsc2)=O)CCN(C2CCC(NC(C3(O)CCSCC3)=O)C2)CC1 C1(CC)(NC(C2C(C=C)C2)=O)CCN(C(=O)C(c2ccc(O)cc2)(C)C)C1.O c1cc(O)ccc1F.N1(C(c2[nH]cc(C(=O)OC)c2)=O)CCCC(C(=O)NC)C1 C(C(C)(C)C(=O)NCC1CCCC1O)NC(C)=O.c1ccccn1.C(=O)C.N C1(NC(C2C(OC)CN(C(=O)CCCn3ccnn3)C2)=O)CCC(=O)N(C)C1 N1(C(CC2(CNC(c3cc(CC)nn3C)=O)CC2)=O)CC2CCC(CC2)C1 C1(C)(C(N2CC(CCC)C2)=O)CCC(=O)N1.c1(C(C(=O)N)OC)cccnc1 C1(NC(COCC(C)C)=O)CCN(C(=O)C#CC2CCOC2)CCC1(F)F C1(C(=O)NCCOCCCNC(=O)CCCC2OCCO2)CCNC(=O)C1 C1(CNC(c2ccnc(C)n2)=O)CN(C(=O)C(C)C2CC2)CCC1C O(S(=O)(=O)c1cccnc1C1CC1)c1ccc(N2C(=O)OCC2)cc1 C1(OCC(Cc2c(OC)cccc2)=O)CC(=O)C12CCC2 c1(C(=O)NC(C)CN(C)C(C2(C(N)=O)CC2)=O)cnc2cnn(C)c2c1 C(=O)(C(F)(F)CF)N1CCC(OCCNC(=O)CC2CC2)C1 N1(C(C2C(C)OCCO2)=O)CCCC12CCN(C(c1cccc3ccoc13)=O)C2 N1(C(c2c(N)cc(F)cc2)=O)CC2CCC(NC(c3cccnc3O)=O)C2C1 C(=O)(C(CCOc1ccc(F)cc1)NC(=O)C(F)OC(F)(F)F)OC O=C(CC1=Cc2ccccc2C1)NC1CCC1NC(C1COC(=O)N1)=O c1(C(C(N2CCC(C(C)NC(=O)CCCc3ccsc3)C2)=O)=O)ccc(Cl)cc1 N1(C(C2C(C)(C)C2)=O)CCCCCC1CNC(c1csc2nccn12)=O C(=O)(CCCCC(=O)NC12CCN(C(=O)Cc3nonc3C)CC1C2)OC CCCC(C(=O)OC)C(=O)NC1CCCN(C(C2(c3ccccc3)CC2)=O)CC1 c1(OC)ccc(C)c(C(=O)NCC2CC2)n1.C12(C=O)CCC(F)(CC1)C2 c1(C(=O)N)nccc2ncccc12.C1(NC(C2CC(C(=O)OC)C2)=O)CCCC1 N1(C(CC)=O)CC2CC(C1)CN(C(=O)C=Cc1ccc(F)cc1)C2.C(C)OC.O C1(NC(c2c[nH]ccc2=O)=O)CN(C(C2CCCS2)=O)C2(CCCCC2)C1 c1(C(=O)NC2CCCC(NC(c3cccc(CC)n3)=O)C2)cccn2nncc12 c1(C(=O)N)c(C)c(C)cc(C)c1C.C(C)(CC(C)C)NC(CCSCCCC)=O N1(C(c2c(OC)n(C)nc2)=O)CC(CO)C2(C1)CN(C(C1CCCCS1)=O)C2 N1(C(Cc2nc(C)[nH]n2)=O)CCC2C(C1)CN2C(=O)CCc1cnc[nH]1 c1(C(=O)N)ccc(Cl)c([N+](=O)[O-])c1.C1(C(C)C)CCCN1C(C1CC2CC2C1)=O Cc1cc(C(=O)NCC(C)NC(=O)CCCC2(C)N=N2)c2ccccc2n1 c1(C(=O)NC(C2CCN(C(COCCC=C)=O)C2)C)ccc2c(c1O)CCCC2 N(C1CCc2c(Cl)cc(Cl)cc21)c1c(C#N)ccnc1 c1(C(N(CCCNC(C(C)=CC)=O)CCO)=O)cc(C2CCC2)[nH]n1 c1(C(=O)OC)ccc([SH](=O)=O)cc1.C(=O)(C(O)(c1ncnn1C)c1ncnn1C)N N1(C(c2c(C)cccc2)C(=O)NCC2CCOC2)CCCC2(C=CCO2)C1 C1(CC)(NC(=O)CC2(C)CC2)CCN(C(=O)C(C)C(C)C2CCCCC2)CC1 Cc1nc(C2CC2)nc(O)c1C=O.C1CCC12CN(C(=O)CC1CC(C)C1)C2.N N1(C(=O)CC2CCCOC2)CCN(C(=O)CCc2cccs2)C(CCO)C1 CCCCCCCC(=O)N1CCC(C)(C)C(C(=O)NCc2nccn2C(C)C)C1 C1(NC(c2cc(C)on2)=O)(CNC(C2CCCC3(CC3)C2)=O)CCCCC1C C=CC(C)(CCOC)C(=O)NCC(C)N(C)C(c1ccccc1)=O.C(N)(=O)N C1(C(=O)NCC#CCNC(=O)C(C2CC2)C2CC2)CC2CCC1C2 c1(C(=O)NCC2CC(NC(c3c(C)onc3CO)=O)C2)nnc(O)nc1O c1(C(=O)NCC(CO)NC(C(c2cccc(Cl)c2)(C)C)=O)cn2cccnc2n1 CCCCCCOCC(=O)NCC(O)CCNC(=O)Cc1csc(CSC)n1 S(=O)(=O)(c1ccc(N2CCCOCC2)c(Br)c1)N1CCC(N(CC(CC)C)C)C1 C(=O)(C#CC1CCC(=O)CC1)NCC1(OC)CN(C(c2cncnc2C)=O)C1 c1(C(C)C)ccc(C(=O)NCC(C)(C)CNC(C2(F)CC2C)=O)c(F)c1 Cc1cc(C(N2CC(CNC(c3cnn(C4CCC4)c3)=O)C(C)C2)=O)cnc1O Cc1nc(C(=O)N)c2n1CCCC2.C1(C)CC(F)(F)CN1C(C1CC1(C)Br)=O.C c1(N(CC(C)OC)C)nc2ccsc2c(=NCc2cccc3c2NC(=O)CO3)[nH]1 c1(C(=O)NCC(CC)NC(=O)C=Cc2cnc(C)s2)cnn2c1OCC(O)C2 N1(C(C2CC3(CC(=C)C3)C2)=O)CC2CCC(C1)N2C(C1CC1(Cl)Cl)=O N1(C(C(C)=C2CC2)=O)CCCC(CCNC(=O)Cn2cccc2)C1 C1(C(=O)Nc2c(Br)ccc(OC)n2)C2C(CN1C)C2(C)C.c1ccc(Br)cc1I N1(C(CN(CCOC)C)=O)CCC(NC(c2cncc(C(C)=O)c2)=O)CC1.C Cc1cc(OCCN(C)CCn2cc(CC(=O)O)nn2)no1 C1(C(=O)NC(C)CCCCNC(=O)C=CC2CCOC2)CC(=O)NC1(C)C C1(C(=O)NC(C(C)NC(c2cnc(C3CC3)nc2)=O)(C)C)CC(C2CCC2)C1 Cc1cccc(N=c2scc(-c3cnccn3)n2CC2CN(C(C)C)C2)c1 Cc1cc(F)c(Br)cc1N(C1CCNCCC1C)C(=O)C(F)(F)c1ccco1 c1(NC(C=CC(C)NC(Cc2c(C)occ2)=O)=O)cccc(C(C)F)c1 C#CCC(C)(C(=O)NC1CCC2CC1CO2)NC(c1ccc(CO)nc1)=O C(CC=O)(C(N)=O)NC(C)=O.c1(CCC=O)nc(C(C)C)no1.C1CCC1.N CCC(C)C(C)C(=O)NC(C1(C(=O)Nc2cc(F)ccc2C)CC1)C C1(C(N2CC(=C)C2)=O)CCCN(C(C2(C)CC(C)=NO2)=O)CC1 c1(NC(C2C(NC(=O)Cc3cc(F)cc(F)c3)C2)=O)cc(F)c(Br)cc1F C1(NC(=O)C=C(Cl)Cl)CN(C(c2cccc(OC(F)F)c2)=O)CC12CCOCC2 C(=O)(C(F)C(F)(F)C(F)(F)F)NC1(C)CCN(C(COC(CC)C)=O)CC1 CC(O)(C(=O)NCCCCCC(=O)N1CCC(O)C(O)C1)C(F)(F)F c1(C(N2C(C(N3CC(CC)OCC3)=O)CC(O)C2)=O)cnc2[nH]ncc2c1 N1(C(CCc2ccc(C)o2)=O)CCOCC1C(=O)NC(C)Cn1cnnc1 CC(C)(C)C#CC(=O)NCC1COCCN1C(c1ccc(NC2COC2)cc1)=O C(CC(=O)N(CC(=O)N(C)CC1CC1)CC1CC1)OCCOCC CC1CN(C(c2ccncc2-c2cn(Cc3ccc(Cl)s3)nn2)=O)CC(C)O1 O=C(C1=C2CCN=C2NC=C1)NCCCOCCNC(=O)C#CC1CCCCC1 C1(NC(C2(CCOC)CCC2)=O)CCN(C(=O)CCC(C)SC)CC1 c1(C(=O)OCCC2CCOC2=O)c(F)ccc(CO)c1F N1(C(c2ccc(CSC)cc2)C(=O)NC2CC2)CCC2(CCN(C)C2)C1 C1(NC(c2ccc(F)nc2)=O)CCC2CCN(C(=O)C(c3cccnc3)O)C1C2 Cc1[nH]c(=N)sc1C(=O)NCC(C)NC(c1ncn(C)n1)=O c1(C(N2CC(C(C)NC(=O)CC3CC3)C2)=O)cc2c(cc1[N+](=O)[O-])OCO2 n1(CCCC(=O)NC(C2CCN(C(c3cnccc3Cl)=O)C2)C)ccccc1=O C=C(C)C(C)(O)C(=O)N1CCCC(N(C)C(c2ncccc2OC)=O)CC1 C1(C(N2CC(C3CN(C(=O)C4=CCCCO4)C3)OCC2)=O)CC2(CCCCC2)C1 C1(C)(C(=O)N)CC2CCC1O2.CCCC(C(=O)N1CC(O)(CC)C1)NC(C)=O O=C(CCCC(=O)NC1CC(Cn2cc(-c3ccc(Cl)c(Cl)c3)nn2)C1)C1CC1 N1(C(C2C(C(C)C)N(C(C3CC4(CC4)C3)=O)CC2)=O)Cc2ncsc2C1 c1(OCC)ccc(Cl)nc1C(=O)NCC(CC)NC(c1cn(C)nc1)=O.O N1(C(C(C=CC)O)=O)CCC(NC(=O)C(C)(CC=C)N(C)C)C(C)C1 c1(OC)cc(C(=O)NC(C)C2CCC2)c(N)c(C)c1.c1(C=O)ncccc1Cl.N CCCC(C)CC(=O)N1CCC(C)CC1CNC(=O)CCn1ncn(C)c1=O C12(C(N3CCN(C(C(CC=C)C)=O)CC3C)=O)CCC(C)(CC1)OC2 Cc1nn(C)c(C)c1CC(=O)NC1CCCN(C(=O)Cn2cc(C#N)cn2)C1C CCC(C)(C)CCCC(=O)N1CCC(C2(NC(c3cncn3C)=O)CC2)C1 N1(C(C(CC)C)=O)CCC2(CCN(C(=O)C(C)(F)C(C)(C)F)CC2)C1 N1(C(CC2CC(=C)C2)=O)CC(C2CN(C(=O)Cc3c(Cl)ccc(O)c3Cl)C2)C1 c1(C(=O)NCC2C(NC(=O)CCc3ncc[nH]3)CCC2)coc2cc(O)ccc12 C(C(C)(O)CNC(c1nocc1Br)=O)NC(C1(C(N(C)C)=O)CC1)=O C1(N(C)C)CCCN(C(C2(C)C=CCN2C(c2cc(C3CC3)no2)=O)=O)CC1 C(=O)(COCC(=O)NCC1(CC(=O)NCC(F)Cl)CC1)NC c1cc(C)c(C=O)o1.c1(CC=O)cc(C(F)(F)F)n[nH]1.C1(CC)CC1.CC c1(C(=O)NC(CC)(C)CNC(=O)CC2CCOC2)cnc2ccncc2c1 c1(C(=O)NC2CCN(Cc3cc(OC)cc(Br)c3)C2)ccc(Br)c2ccccc12 c1(C(=O)NCC(CC)NC(c2ncoc2-c2ccon2)=O)cc(C)c(Cl)cc1C Cc1oc([N+](=O)[O-])cc1C(N1CC2CC(C1)C2NC(c1cnc(O)s1)=O)=O c1(CC(=O)Nc2ccc(CN3C(=O)CNC3=O)cc2)ncc2ccc(Br)cn12 C1(CC=C)(C(=O)NCCC(=O)NCC2COCC(C)O2)CCN(C(C)=O)C1 C1(NC(C2(C)SCCCS2)=O)CCCC(C(=O)NC2CC23CCCCC3)CC1 C(=O)(C(F)C(F)(F)F)N1CCC(CC=C)(C(=O)NCC(C)C(=O)NC)C1 CC(C)C(C)(O)C(=O)N1CCC(F)(c2cn(C3(C(N)=O)CC3)nn2)C1 CCC(CCCC(=O)N(C1CCN(OC)CC1)C)NC(=O)CC(C)n1ccnc1 NS(=O)(=O)c1cc(-c2nc(Cc3ccc(F)c(F)c3)no2)ccn1 Cc1sc(C(=O)NCC2CC(C)N(C(=O)COc3ccccc3)C2)c(C)c1C C(=O)(C1CCCn2c(C)cnc21)N(CCCNC(c1ns[nH]c1=O)=O)CC N1(C(C2N(C(Cc3ccc(OC)c(F)c3)=O)CC2)=O)CCn2nccc2C1 C1(C(=O)NCC23CC2CN(C(=O)Cc2ccc(Cl)s2)C3)CCCCC1(F)F c1(C(=O)NCC(CNC(=O)Cn2nccn2)OC)ccc(O)c(F)c1F CC1(C)COC(C(=O)NC2(CCC(=O)NC3CCC(CO)CC3)CCCC2)C1 C1(NC(C2CCN(C)C2)=O)(CO)CCN(C(c2cc(C3CC3)nc(O)c2)=O)CC1 N1(C(c2ccn[nH]2)=O)CC(C(N2CCC(N(C)C)C(C)C2)=O)CC1(C)C.CCO Cc1nc(CN2CCC(CNc3ncc(I)cn3)C2)ccc1Br S(=O)(=O)(c1cccc(C(=O)NC(CC)C(=O)O)c1)NCC(OCC)O c1(C(=O)NC(c2cn(-c3ncc(C(=O)OC)s3)nn2)C)nc2c(s1)CCCC2 c1(C(=O)NCC2N(C(c3ccc(N)cc3Cl)=O)CC=C2)ncnc2c1CCC2 N1(C(C2CCN(OC)CC2)=O)CC2CNCCC2(C(=O)O)C1 CCCCCC(O)C(C)C(=O)N1CCC(C)(C)C(CNC(=O)C=CCF)C1 Cc1ccc(C(N2CCC(C(F)C(=O)NC3(c4ccsc4)CC3)C2)=O)c(C)n1 c1(CNc2n(-c3ccccc3)nc(C)c2Cl)nc2cc(F)ccc2o1 c1(C(=O)NC2CN(C(c3c(C)scc3)=O)CC2C)cncn(C)c1=O N1(C(C(C)OCC#C)=O)CC2CC(C)N(C(=O)C=Cc3nccs3)C2C1 C1CCCC12CCN(C(=O)CC1CC(F)(F)C1)CC2.C1(OCC=O)CC1(F)F.N CC1(C)CCCC(CC(=O)NCCC2(O)CCCN(C(c3ccns3)=O)C2)CC1 N1(C(c2c(NCCCC)cccc2)=O)CCCN(C(=O)C(CCC)OC)C(C)C1 N1(C(Cc2cncc(C)c2)=O)CCN(C(=O)Cn2cnnc2)CC1CC(F)(F)F CCC(C)(C)C(O)C(=O)N1CCOC(CNC(=O)CC2CCCCC2C)C1 c1(C(N2CCCCC2)=O)cc(F)cc([N+](=O)[O-])c1.S(S(C)(=O)=O)CC=O.CC c1(N2CCC(O)(C(C)NC(=O)C3=COCCO3)C2)nc(Cl)ncc1[N+](=O)[O-] Cc1cccc(OCCC(N2CCCC(N(C(=O)C(C)C3CC3)C)C2)=O)c1C C(CCCC)(C(=O)NCCCCC1CC1C)NC(c1n(C=C)nnc1)=O CC1CCN(C(c2csc(Cl)n2)=O)CC1N(C)C(c1ccsc1)=O N1(C(C=NOC)=O)CC2CC(C1)C2NC(=O)CSC C1(NC(Cc2cc(C)[nH]n2)=O)CCC(CNC(=O)C(F)=C2CCCC2)CC1 c1(C(=O)NCCC(C)NC(CC=CC)=O)cc(=O)c2ccc(F)cc2o1 C(C(C)C)(C(O)C(=O)NC)OC.c1(C(C(N2CC(F)C2)=O)C)cccc(C)c1 N1(C(C=CC(C)NC(CSCC(C)=O)=O)=O)CC(C)CC1(C)C N1(C(C2C(C)OCC2)=O)CC(C2CCCCN(C(=O)Cc3ncncc3Cl)C2)C1 N1(C(CS(=O)(=O)NCC)=O)CC2CCN(C(=O)CC3(C)CCCO3)CC2C1 n1(CC)c(C)nn(CC(N2CCCC2CNC(C2(C)CC2(F)F)=O)=O)c1=O C1(NC(c2cc(C(C)C)no2)=O)C2CCC1N(C(C1C3CNC(=O)C13)=O)C2 c1(C=O)sc2ncnc(N)c2c1C.C1(CNC(C=C(C)C(F)F)=O)C=CCC1.N c1(CC(=O)N)cc(C(F)(F)F)cc(Cl)n1.CC1C(C(=O)N(C(C)C)C)C1C C12(CNC(c3cc(-c4ccccc4Br)no3)=O)CC(CO1)N(C)C2.c1ccccc1 CC1CN(C(c2cc(C(F)(F)F)n[nH]2)=O)C(C)CN1C(=O)CN1CCCNC1=O O=CCCCC1CCC1.C(=O)C(F)(F)F.C1(CCC)CC1.C(=O)C.C1CC1.N CC1Cc2cccc(Br)c2CN1c1nc(NC2CC3(CC3)C2)c2ncn(C)c2n1 C1(NC(CSC(C)C)=O)CCN(C(C2CN(C3CCC3)C2)=O)C1C1CC1 C1(CNC(=O)Nc2n(CC)ccn2)(CF)CC(F)(F)C1 C1(CNC(C(CC=C)OC)=O)(CO)CCCN(C(=O)Cc2csc(C)n2)C1 N1(C(CC(C=C)CC)=O)CC(N=[N+]=[N-])CC1C(=O)N(CCCO)CC C(=O)(CC(F)(F)CC)NCC(CC=C)NC(=O)CC1(O)CCCCC1 CC1(C)OCCCC1CNC(=O)CCC1CCC1.C1(C=O)CC2C=CC1CC2.N c1(C(=O)NCC2CCN(C(=O)CCCF)CC2)cc(O)cc(Br)c1 CCCCC(C)(F)C(=O)NCCC1CCCN(C(C2CCCN(C)C2)=O)C1 C1(CC(=O)NCCn2ccc(C(=O)NCC(O)C3CCC3)c2)C=CCCC1 C#CC1C(C(=O)NC(C)(C)CCNC(=O)C)C1(C)C.c1ccc(Cl)cc1.O c1(C=O)ccc(=O)n(C)n1.Cc1cc(C(=O)NC2CCCCC2)nn1C1CC1.N C12(C(=O)NC(CNC(C(F)=CCC)=O)C(C)C)CCC(C)(CC1)OC2 CC1(C)C2CCC(C2)C1NC(=O)Nc1ncc(C2CCOC2)s1 C(=O)(C(C)(C)C(C)NC(=O)CC1(C)CCOC1)Nc1ccc(SC)cc1 CCC(O)CCN=c1cc[nH]cc1S(=O)(=O)NCCC1CCN(C)C1 C1(CN(C(COC)=O)C)CCCCN1C(C1CC(c2ccccc2Br)C1)=O c1(C(N2CC3C(NC(=O)CC4CCCCO4)(C3)C2)=O)nc2cnccc2s1 C1(CC#C)(C(N2CCN(CCCNC(=O)C(O)C3CCC3)CC2)=O)CC=CCC1 C(=O)(CCC(O)C(C)(C)C)NC(C(C)C)CNC(=O)CC1CCCNC(=O)C1 N1(C(c2c[nH]nc2C2CC2)=O)CCN(C(c2cc3cccnc3o2)=O)C2CCC12 N1(c2cc(NCCCOC(=N)O)nc(COC)n2)CC(CO)OC2(CCC2)C1 N1(CC=O)CCCC2(CC2)S1(=O)=O.C1(CN2CC(CC)C2)CC(C)N(C)C1 C=C(C)CC(C(=O)Nc1ccccc1COC)NC(=O)C(F)C1CCCC1 C1(C(N(CC(C)NC(c2c(C(F)(F)F)cccc2F)=O)C)=O)CN2CCN1CC2 C(C(=O)N1CC(C)(C)C1C(=O)OC)(C(C)OC)NC(CN(CCC)C)=O Cc1n[nH]cc1CCNC(C1(N(C)C(C2CC2C)=O)CC1)=O C1(NC(c2ccc(CO)nc2)=O)CC12CCN(C(=O)C(O)c1ccsc1)C2 c1(CNC(=O)C(c2cccnc2)NC(C2CCSC2)=O)cncc(Cl)c1 C1(NC(=O)CCF)CC2CC(NC(C3CCSCC3)=O)CC12 c1(SC)ccc(C(=O)NC)c(Cl)c1.C1CC2CC2N1C(=O)C(C)=CC1CC1 C(C(C(=O)N1CC=CCO1)NC(C1C=CCCC1)=O)SCC C(=O)(C(C(C)NC(c1cc(F)cnc1O)=O)C(C)C)N(CC#C)CCOC CC1(C)CN(C(=O)CC2CSC2)CCC1C(=O)NCC(CO)C1CC1 Cc1coc2ccc(C(=O)NC(CNC(c3cccnc3O)=O)C(C)C)cc12 c1(CC(N2CC(O)(CNC(C3CCCC3)=O)C2)=O)ccc(Cl)nc1F c1(C(N2CCC(NC(CCOCCOCC)=O)C2)=O)c(O)cccc1O CC12CC1CCN2C(=O)CC1C=CC(NC(=O)CN2C(=O)CNC2=O)C1 C(=O)(C#CC1CCCOC1)NCC1C(NC(c2c(CC)nco2)=O)COC1 c1(C(=O)NC2CCC(NC(C(C(C)C)SC)=O)CC2)cc(C)nc(C)n1 Cc1nc(C2CC2)ncc1C(=O)NCC1CCCCCN1C(=O)Cc1ccoc1 C1(NC(C=C(COC)C)=O)CN(C(c2ncnn2C(C)C)=O)Cc2nccn2C1 c1(C(N2CC3CCC3(OC)C2)C(=O)NCCC)cc(Cl)cc(Cl)c1Br C(=O)(C(CCC)CCC)NC(C(=O)NC(CCCCC)C)CCCC C1(NC(c2c(C)cccc2)=O)CCN(C(c2c(Cl)cnn2C(C)C)=O)CC1C c1(C(N2CC(C(C)NC(c3n(CC)ccc3)=O)C2)=O)ccc(F)cc1N N1(c2c(C)cncn2)CCC2(CC1)CC2C(N1CCC(O)C(N(C)C)C1)=O N1(C(C2N(C(c3c(CC)noc3)=O)CCC2)=O)CCOC(c2cn(CC)nn2)C1 CC(C)C(=O)C(=O)N1CC(CC(C)NC(=O)C=C2CCCCC2)C1 C1(NC(CCn2c(C(C)C)ncc2)=O)CCCC(C)C1.C(=O)CCC1(C)CC1.N C(C)(C(=O)NCC(C)(O)C1CC1)NC(C1(C(CC)=O)CC1)=O n1(CC(=O)NC(C2CCCN(C(=O)C(C)CO)C2)C)ccc(=O)c([N+](=O)[O-])c1 C#Cc1ccc(C(=O)NC(C)(C)CO)cc1Cl.C(=O)(C(C)C)N.[SH](C)(=O)=O C1(CNC(C(CN(C)C)NC(=O)Cc2cnoc2)=O)CN2CCC1C2 N1(Cc2nc(C(C)C)on2)CCC(O)C(NCCCc2ccccc2)C1 c1(C(CSCC2CC(OC)C2)O)ccc(F)cc1C C(=O)(CC1=CCOCC1)NC.C(CC(=O)NC1CC1)(c1cccs1)NC(C)=O.C C1(NC(C=C(C)Cl)=O)CN(C(c2ccncc2F)=O)C2CC12 n1(CC=C)cc(C(=O)NCCC2CC2)cn1.n1(C(C(=O)N)C)cc(C)cn1 c1(-c2c(C(F)(F)F)ccc(Br)c2)ccc2cc(CN3CCC4(CCC4)C3)[nH]c2c1 N1(C(c2c(C)ncs2)=O)CC2CC2(NC(=O)C(C)OCc2ccc(F)cc2)C1 Cc1cc(C(N2CCC(N(C(=O)C(F)n3cccn3)CC(C)C)CC2)=O)oc1C C(=O)(CCN(CCCO)C(C1CC=CC1)=O)N(CCCN(C)C)CCC Cc1ccc(CNC(C2CCC(n3cc(C(O)C4CC4)nn3)CC2)=O)cc1 c1(C(CC)(C)C)ccccc1C(=O)NCC(C)N(C)C(C1CCCC1O)=O c1(CN(C)Cc2c(COC)cccc2)ncc(Br)cc1[N+](=O)[O-] c1(C(N(C2CCCCC2NC(C2CCOC2)=O)C)=O)cnc(S)n1C CCCCC(C(=O)N1CC(C)(OCC)C1)NC(c1cc(C)n(CC)n1)=O N1(C(C(CCC)C)=O)CC2CCCC1C2CNC(=O)CSc1ccc(F)cc1 C1(NC(=O)CCSC(F)(F)F)(CO)CCN(C(C2CC3CCC2C3)=O)C1 Cc1nn2c(CN3CCC(=O)N(CC(=O)N4CCCO4)C3=O)c(C)nc2s1 C=CCC(CC(=O)N1CCCC(=C)C1)NC(c1c(F)cccc1F)=O Cc1[nH]nc(C(=O)NCC2(CC(C)C)CCC2)c1Cl.N12CCC1C2=O C1(C(N2CC(CO)C(CO)C2)=O)CCC(C2CC2)N1C(=O)CN1CC2CC2C1 c1(C2C(CNC(c3scc(Br)c3Cl)=O)C2)cc(F)ccc1F N1(C(CNC(C)=O)=O)CCC(NC(=O)CCc2ccc(N)c(Cl)c2)C(C)C1 c1(N2CCC(COCC)CC2)nc(N2CC=C(Br)CC2)nc2c(F)cc(F)cc12 C1(C)(C=O)CC(C)(C)C1.c1(C(N(CCC)CC)=O)ccc(C2CCCCC2)s1 CC1CN(C(=O)COC2CCN(C(=O)CC(C)(C)O)C2)C(C)CO1 N1(C(C=CC=CC)=O)CCCOC(CNC(=O)C(c2nc(C)cs2)C)C1 CC(C)CC(F)C(=O)N1CC(O)(C(C)NC(c2ccc(CCF)cc2)=O)C1 c1(C(N2CCC(NC(C(CC#C)CC#C)=O)C(O)C2)=O)nn(C)c(C)c1[N+](=O)[O-] CC1(OCC(=O)NCC(C2CC2)NC(c2ccnnc2O)=O)CCOCC1 c1(C(=O)NC2CC(CC(=O)N(CCSC)C)C2)scnc1Cl C1(N(C(=O)Cc2cscc2Br)CCNC(C=CC)=O)CCCCCC1 N1(C(c2c(Cl)cc(C)s2)=O)CCN(C(C23CCC(F)(CC2)C3)=O)C(CO)C1 N1(C(c2c(C)n(C3CC3)nc2)=O)CCC(NC(c2ncncc2Cl)=O)C(CO)C1 C(CCN=c1nc(N2CCC(c3nnnn3C)(OC)CC2)cc[nH]1)OCC Cc1c[nH]c(C(=O)NC2(CCNC(=O)C(C)Cc3ccccc3)CC2)c1 C1(C)(OC)CCC(NCc2cc(-c3cccc(C(=O)N)c3)cn2C)CC1.C1CC1 C=CCCC(C(=O)NCc1cnc(C)[nH]1)NC(=O)CC1CCCC(=O)C1 C=CCCC(F)(F)C(=O)NCC1(C(=O)NCCCS(N)(=O)=O)CC1 C(CC(=O)NCCOCC(=O)N(CC(O)CF)C)OCCOCC C1CC2C(O)C(O)CC12.Cc1nc(O)sc1C(N1CCC(C=O)(C(C)C)C1)=O.N c1(C(=O)NC2CCN(C(Cc3ccc(C)o3)=O)C2)cc2c(cc1Cl)CCCC2 C(C(=O)N(CC(=O)NC)CC)SCCC.C(CC)NC(C)=O c1(C(=O)OC2C(SC(C)C)CCCC2)ccc(S(C)(=O)=O)[nH]1 Cc1cc(C(=O)NC2C3CC2N(C(c2c(Cl)noc2C)=O)C3)c(C)s1 CCC(CCC(=O)N(C(CNC(c1scc(C)c1Cl)=O)C1CC1)C)OC C1(C(=O)NC(C)(C)CF)CC2CCCC2N1C(c1csc(F)c1)=O c1(CNC(C2(NC(C)=O)CCC2)=O)cccc2c1CN(C(c1cnsc1)=O)C2 C1(C(N2CC(C)C(NC(C3COCCN3C)=O)C2)=O)CCOC(=O)CC1 n1(CC(=O)NC2CCC(N(C(c3nc(COC)oc3)=O)C)C2)cccnc1=O Cc1nnc2ccc(C(=O)OC(C)C(=O)N3CCC3)cn12 c1(C(N2CCCC(CC(N3C(C)CS(=O)CC3)=O)C2)=O)cc2cccnn2c1 c1(CC#N)cccc(C(N2CCOC(C(N3CCCC3C3CCCC3)=O)C2)=O)c1 C1(CS(C)(=O)=O)CN(C(C2CCCC2)=O)CCN1Cc1cnc(C(F)(F)F)s1 C(=O)(C(C(C)CC)NC(C1CC1(C)C(F)F)=O)NCCOCC C1CCCCCC1.c1(C(C)OC)nc(C(=O)NC(C)C2CC2)cs1.C(=O)C.N C#CCCC(C(=O)OC)NC(C1CC(O)CN1C(c1ccncc1F)=O)=O CC(C)CC(C)(C)C(=O)NC1CC1CNC(c1cccc(OC(F)F)n1)=O C1(NC(CCCOC)=O)(CO)CCN(C(=O)C=C(C)CCc2ccccc2)C1 N1(C(C(CC)N(CC)CC)=O)CC(C)(C(N2CC3CC3C3CC23)=O)CC1(C)C c1(C(=O)NCC2C(NC(=O)CCCN3CCCC3)CCC2)snc(O)c1Cl C1(C(N2C(CNC(C#CC(C)(C)C)=O)CC(F)C2)=O)CCCCC12CCC2 C1(C(CC)C)CCCCN1C(=O)CONC(c1cc(O)n(C)n1)=O Cc1cc(NC(N2CCOCC(C(C)(C)C)C2)=O)ccc1P(C)(C)=O c1(C(=O)NCC2C(NC(c3cc(C)nnc3)=O)CCC2)cncc2c1CCCC2 C1CCCCN1C(=O)C=C(C)C.C1(C(=O)OCC)CC1C(=O)NC Cc1ccc(C(=O)C(=O)NC2CCCC2C)cc1.c1(CC=O)c(C)noc1Cl.N n1(C(C)C)cc(C(=O)NC2CC(NC(C3CCC3(C)C)=O)C2)ccc1=O N1(C(C(CNC(c2c(C)nn(C)c2)=O)O)=O)CC(=O)NC(C)C1 CC(C)(CNC(=O)C=CBr)CNC(=O)C=C1CCC1 C(=O)(C(F)CCC(C)(C)C)NCc1c(C(N2CCCC(C)C2)=O)cccn1 c1(C(=O)NCC23C(CN(C(c4n(C)nnc4)=O)C2)C3)c(O)cc(Cl)cc1F C1(NC(c2ncn3cccnc23)=O)CN(C(c2cccnc2O)=O)CC2(CC2)C1 C1(C(=O)NCC2(F)CN(C(Cc3cc(CC)no3)=O)C2)CCc2ccccc2C1 c1(C(N2CCCC(C(N3CCCC(OC)CC3)=O)C2)=O)cc2cccnn2c1 N1(C(c2c(N)non2)=O)CCC2(CCOC2)C(C)C1.C12(C(=O)N)CC(F)(C1)C2 Cc1cc(C(=O)NCCC2CN(C(=O)CCCc3ccc(F)cc3)C2)cc(F)c1 Cc1nnc2n1CC(C(N1CCC(C(=O)NCCC(C)CO)CC1)=O)N(C)C2 N1(C(C2OCCN(C(C3CCCS3)=O)C2)=O)CCc2c(F)cccc2C1 C1(CNC(c2ccccn2)=O)C2CCCC1N(C(c1ccc3nonc3c1)=O)C2 C1(NC(c2cc(C(C)=O)on2)=O)CCC(NC(=O)CCO)CC1.C1CCCO1 C1(C(=O)NCc2c(OC)cc(OC)cc2O)COc2cc(F)ccc2O1 CCCCCCC(C)CC(=O)N(CCCNc1nc(C)nc2sc(C)c(C)c12)C C1(C(=O)NCC(Cl)=CCl)(NC(=O)CC2CC(F)(F)C2)CC(CO)C1 N12CCC(CC1)CN(C)C(=O)C1CCCN1C(=O)C2=O.c1(CC)cc(C)no1 N1(C(CCCC)=O)CCN(C(c2cnn(-c3cccc(F)c3)c2N)=O)C(CF)C1 N1(C(C23CC(CN(C(c4cc(=NC)[nH]cc4)=O)C2)C3)=O)CCC2CCCC2C1 CCCCS(=O)(=O)CC(=O)OCc1cnc(OC)c(C#N)c1 C(=O)(CC1=CCCCC1)NC(C(c1ccccc1)NC(CC=CC)=O)C N1(C(C(CC)CC)=O)CCC2(CCN(C(c3cc(Cl)on3)=O)CC2)C1 Cc1cc(CNC(C23CC(n4cc(CN(C)C(C)C)nn4)C2C3)=O)on1 C12CC(C13CCOCC3)N2.c1(C(CC)OC(C)(C)C)ccnn1C C(=O)(C1CCc2ccccc21)N1CCOC(C)C1C(=O)NC1C2CCCC12 C(=O)(C(C)CC(F)(F)F)NCC1CC(OC)CN1C(C1CCCC(O)C1)=O N1(C(C2N(C(C3(C)C(C)C3)=O)CC(O)C2)=O)CCC2(CCCO2)C1 C(=O)(C1=CCCC(C)(C)C1)NC12CCN(C(CCCC)=O)C1CCC2 N1(C(C2CCN(CCC#C)CC2)=O)CC(NC(=O)C2=CCCCO2)CC(C)(C)C1 c1(C(N2CC3C(CNC(c4c(C)nn[nH]4)=O)(C3)C2)=O)nccc2c(F)cccc12 N1(C(c2ccc(C)cc2C)=O)CCC(F)(F)C(C(=O)NC)C1.C1CCC(=O)NC1 C1(C(N2CCC(F)(CNC(C3CCCC(C)(C)C3)=O)C2)=O)CCCN2CCCC12 c1(NC(CC2N(S(CCOC)(=O)=O)CCC2)=O)cc2c(cc1Br)OCCO2 c1(C=O)ccc2c(c1)C(=O)NC2=O.CC1(C)C(C(=O)NC2CCCC2)C1(F)F C1(C(C)NC(=O)C(F)F)CCCN(C(=O)C=Cc2cn(C)cn2)C1 C1(C(=O)NCCCC(C)NC(C(C2CC2)OC)=O)CN(C)CCN1C c1(CC)cc(NC(C2CC2NC(=O)Cc2ccc(C#N)cc2)=O)ccc1Br c1(N2CCN(NC(c3cnn(CCC)c3C3CC3)=O)CC2)ccc(CC)cc1F N1(C(C2(CC=C)CCOC2)=O)CC2C(N(C)C(c3cc(OC)cs3)=O)C2C1 c1(-c2n(Cc3sccc3)nc(C3CCCCC3)n2)cncc2sccc12 N1(C(CCN(C)C)=O)CCCC(F)(C(=O)NOCC(O)CO)C1 N1(C(C(CC)COC)=O)C(CC(=O)N(CC)Cc2ccoc2)C2CCCC12 C1(CC(C)NC(c2cc(C)on2)=O)CCN(C(=O)CC2C=CCC2)CC1 C1(C(N2C(CNC(C(C)Sc3ncccn3)=O)CC2)=O)CCc2nnnn2C1 c1(C(=O)NC2(CO)CN(C(CC(C=C)(C)O)=O)C2)ccc([N+](=O)[O-])c(SC)c1 Cn1cc(Cl)c(CC(N2CCCC2C2(NC(=O)C)CC2)=O)n1.CC(F)(F)F.S C(C)(C)(CCC(=O)NC)OC.C1(F)CN(C(c2nnc(C(C)(C)C)s2)=O)C1 Cc1c(NC2CC2C(=O)Nc2cccc(CC=O)c2)cccc1O.C(C)(C)C.O N1(C(CSCCC(C)C)=O)CC(C(C)(C)OC(=O)CC2CCCC2)OC1=O C1(N2C(CO)CC(C)C2)CCC2(CC1)CCN(C(c1cnsn1)=O)C2 CON1CCC(C(=O)NC2(CO)CCN(C(C3CC4(C3)CC4(F)F)=O)C2)CC1 C1(C(=O)NC2CC(CC)C2)CN(C(C2(C#N)CC2)=O)CC1(C)C CC1(C)CCN(C(C2CC(=O)CS2)=O)C1C(N1CC2C=CC1CC2)=O C(=O)(C#CC1(C)CCCO1)NC(CC(C)NC(c1cc(C(C)=O)c(O)cc1)=O)C C12(C(=O)N)CC3CC(CC(C3)C1)C2.c1cc(F)c[nH]1.C1(CC)CN(CC=O)C1 c1(C=O)cnc2[nH]c(=N)sc2c1.N1(CC[SH](=O)=O)N(S(C)(=O)=O)CCCC1=O c1(C=O)c(C)nn(C)c1C(F)F.C=Cn1nncc1C(=O)NC.C1CCCC1 Cc1coc(C(C)(C)C)c1C(=O)NCC(C)(C)Cn1cc(C2CC=CCC2)nn1 N1(C(C(C)CO)=O)CC23CCCCC2(C1)CN(C(C1CCC=CCC1)=O)C3 N1(C(Cc2n(C)cnc2)=O)CCCC2(C1)CN(C(=O)C(F)(F)c1ccccn1)C2 C1(C(=O)NC(CC)(CNC(c2cn(C)c(C)n2)=O)CC)CCCCN1N=O c1(C(=O)NCCN(C(C(CC)C)=O)CCCN(C)C)sc(C(C)C)nc1C C1(O)(CCNC(=O)C=CBr)CN(C(c2cn(CC3CCCO3)nn2)=O)C1 C=CC1OCCC1C(=O)NCC1CCC(NC(=O)C(F)(F)CC)CC1 Cc1sccc1NC(N1CC(NC(C2CC2C2CC2)=O)C1)=O C1(CC)C(CO)CCCN1N(C)CC1CCN(Cc2ccccc2)C1 C1(C(N2CCC(COC)(C)C2)=O)CCC(F)(F)CC1.C1(CC=O)CCSCC1 C(=O)(C(C(C)C)c1ccncc1)N(CCNC(=O)C=C1CCC1)CC C1(CC)CCCCN1C(c1ccc(C2CCC2)nc1)=O.C1(C(N)=O)CC1C(=O)N C1(CC(=O)NC2C(CN(C(=O)C)C)CCC2)CCC(=O)N1.CSC.S N1(C(c2ccc(OCC=C)c(O)c2)=O)CC2OCC(NC(C3CCC3)=O)C2C1 C1(C(=O)NCC(C)N(C(c2c(OC)cc(N)cc2)=O)C)CCCC(C)(C)CC1 c1(C(N2CCC(CC=C)(NC(=O)C(CC)SC)CC2)=O)[nH]nc2ncccc12 N1(c2nc(C)nc(=N)[nH]2)CCC2(CCC2)C(NC(=O)C=C2CCN(C)C2)C1 c1(CN2CCC(CC(N3CCCC(OC)C3)=O)C2)csc2ccccc12 N(C(=NCCC1CC2(CCC2)C1)NCc1ccco1)CC1CC=CC1 c1(C(=O)OC)no[nH]c1=NC(=O)CC1CN(Cc2cncc(C(F)(F)F)c2)C1 Cc1sc2ncnc(NCC(=O)NCCNC(=O)CCC(C)CN(C)C)c2c1C N1(C(C2(CC(C)C)CC2)=O)CC2CCC2(NC(c2snc(O)c2Cl)=O)C1 C1(CC=C)(NC(C2CCCC2)=O)CCCN(C(c2nc(C)ncc2Br)=O)C1 c1(C(=O)NCC2N(C(C3C(C=C)C3)=O)CC(C)(C)C2)coc2c1CCCC2 Cc1cc(C(N2CCC(CNC(=O)C(C)(C)c3cc[nH]n3)C2)=O)c(Cl)cc1Cl C1(NC(C2C(C(C)NC(C3(CC)COC3)=O)C2)=O)CCn2ncnc2C1 c1(C(=O)NCC(CCNC(Cc2n(C)ncc2Cl)=O)O)cnc2cccnn12 CCC(C(C)(F)F)NC(C1CCC(NC(C2CCCN2C(C)C)=O)C1)=O c1(-c2nc(COC)nn2CCOC(C)C)cc(Cl)ccc1OC c1(OCC#C)ccc(C(=O)O)c(N=C2SCC(C)C2)c1 c1(C(N(CCCN(C)C)CC)=O)cc(Cl)cc(Cl)c1F.CC(C)CC(F)C(=O)N CC(C)CC(C)CC(=O)NC(C)(C)CCCNC(=O)CCNC(=O)CC(C)C C1(CC)(NC(=O)CCC(=O)N(C)C)CCN(C(=O)C(c2cccc(C)c2)F)CC1 c1(CC)ncc(C(=O)NC2(C(=O)NCCC(C)(C)O)CCC2)o1 c1(C(=O)NC2C(CNC(c3[nH]cc(C#N)c3)=O)C2)cccc2c1CCC(=O)N2 N1(C(C(c2cnn(C)c2)OC)=O)CCCC(C2(NC(c3n[nH]c(O)n3)=O)CC2)C1 n1(CCCOC)c(SCC2C3COCC23)nc2ccccc2c1=O N1(C(CC2(C)CC2(F)Cl)=O)CCC(NC(c2cc(C(F)F)[nH]n2)=O)C2(CCC2)C1 c1(C(N(CC(CNC(C2(C=C)CC2)=O)C)C)=O)cc(Br)c(C2CC2)s1 Cc1nnc2n1CC(C(=O)NCCCCCNC(=O)C(C)(C)C(C)O)C2 Cn1ccc2c(C(=O)NC3CC(NC(=O)Cc4ccsc4)C3)ccnc12 c1(C(N(C)CC2N(C(c3c(C)nco3)=O)CCCC2)=O)cnn(C)c1C#N C(C(=O)N1CCC(CCNC(=O)C(N2CCNC2=O)C)C1)(C(C)(C)C)SC C12(N(C(N3CCC(c4c(C)cccn4)C3)=O)C3CC3)CCC(F)(CC1)C2 O=C(C1=C(Cl)CCC1)N1CCC(N(C(=O)CCC2CCCOC2)CCO)CC1 N1(C(CC(CC)C2CC2)=O)CCC(NC(=O)CN(C)C(=O)C2CC2)C12CC2 c1(C(=O)NC(C2CCN(C(=O)CCc3cnc[nH]3)C2)C)cnc(N(C)C)s1 C1(C(=O)NCC(c2ccsc2)C)CN(C(=O)C(C)SC(C)C)CCN1C N1(C(CC2CCC(C)O2)=O)CCC(OC2CN(C(C3CC=CCO3)=O)C2)CC1 CN1CC23CCCC2(CN(C(c2csc(CCN)n2)=O)C3)C1 C(=O)(C1CCCn2ncnc21)NC(CN(C(c1c(C)oc(C)c1C)=O)C)C c1(CC(N2C(CO)CC(NC(CC(COC)C)=O)C2)=O)ccc2nc(O)[nH]c2c1 Cc1cc(CC(=O)N(C2CC(O)C2(C)C)C)cc(F)c1 c1ccc(C(C)(C)C)cc1O.C1(OCC#C)CCN(C(C2CC2NC)=O)CC1 C#Cc1ccnc(C(=O)NCC(=C)CCNC(=O)C(C)(O)COC)c1 O=C(CCC(F)(F)C(F)F)NC1COC2(C1)CN(C(=O)CC1(O)CCC1)C2 C1(NC(CCc2onc(C)n2)=O)CCCN(C(c2cc(C3CC3)[nH]n2)=O)C1C c1(C(N2CCN(C(C3(C=C)CC3)=O)CC2C2CCC2)=O)cc(S(=O)(=O)N)cs1 C1(C(N(C2CCN(C(c3cc[nH]n3)=O)C2)CCC)=O)CCCC12CCOCC2 C12CCCC1N(C(C1CCC=CO1)=O)CCC2.C(C=O)SCCN(CC)CC.N c1(C(c2nnnn2C2COC2)NC(C=C)(C)C)cnn(C)c1Cl N1(C(c2cn(CC)nc2)=O)CCC(F)(C(N2CCC(C(F)(F)F)C2)=O)C1 Cc1cc(N2CCC(O)(C(C)NC(c3ccnn3C3CCC3)=O)C2)c(C#N)cn1 C(C(C(C)(C)C)NC(C1CC2CC1CO2)=O)NC(c1cc(COC)sc1)=O N1(C(CC(=O)N)=O)CCC(F)(F)C(CNC(=O)C(F)n2ccnc2)C1.C1CC1 C1(CNC(C=CCCC)=O)CN(C(C2CCOC2CC)=O)CC1C c1(SC)cc(C(=O)NCC2CN(C(=O)Cn3cc(C#N)cn3)CC2O)ccc1F c1(C(=O)N)ccc2c(c1)OCC2.CCC(C)CCNC(=O)CC1CCC(=O)N1C Cc1ccc(C)c(C2(C(=O)Nc3cc(I)ccc3Br)CC2)c1 C12CC1CN(C(=O)C)C2.c1nncn1C1CC1.C(C)(C(=O)N)NC(CC)=O c1(C(=O)NC2CC(NCc3cccc4c3OCO4)C2)cn2c(Cl)cccc2n1 c1(N(C2CCN(C(C3CCC3)=O)CC2)C)ccnc(N2CCCC(CCO)C2)n1 CC#CCCCCNC(=O)CCC(C)NC(C1COCOC1)=O Cc1ccc2c(CC(=O)NC3CC3C)c[nH]c2c1.C1(C(=O)N)CCC(C)(O)CC1 C(CCCCCNC(c1ccsc1C(F)F)=O)N(C(C(C)Cc1cnc[nH]1)=O)C N1(C(Cn2cc(CNC(C3(OC)CC3)=O)nn2)=O)CCC12CCCOCC2 N1(C(Cc2cn(C)nc2)=O)CC2CC2(C(=O)Nc2ccsc2SC)C1 N1(C(CC2C(C)(C)CCCC2)=O)CCCCC12CC(NC(C1COC(=O)O1)=O)C2 N1(C(CCSCCCC)=O)CC2CC(NC(c3ccn4nccc4c3)=O)C(C2)C1 c1(C(=O)NCCC2N(C(C(CCCC)C)=O)CCC2)ccc(NC)c([N+](=O)[O-])c1 N1(C(C(c2cnn(C)c2)C)=O)CCC(C(C)NC(C2(CO)CCOCC2)=O)CC1 C(CC(CNC(=O)CC1CC(N(C)C)C1)NC(=O)CCCOC)OC C1(NC(c2cnn(C)c2CN2CCNCC2)=O)CNCC12CCC2 c1(CN(CCC)CC)cc(C)cc([N+](=O)[O-])c1.C1(C=O)CCS(=O)(=O)N1C c1(OC)ccc(Cl)c(CNc2ncc(-c3cnn(C4CCCCO4)c3)cn2)c1 Cc1nc(NC(=O)C(=O)NCCC(O)C2CCCC2)oc1C N1(C(C2CC(C(=O)OC)C2)=O)CCCC(C2CC2NC(=O)C=CCF)C1 Cc1cc(C#N)cc(C)c1CC(=O)NC1(C)CN(C(c2ccc(Cl)s2)=O)C1 C1(NC(CCOCC)=O)(CO)CCN(C(=O)C(C)Oc2ccccc2O)C1 c1(C(=O)OC)ccc2c(c1)CCCC2C(=O)NC1CN(Cc2ncn(C)n2)C1 Cc1cc(C(=O)NC(C)C(C(C)C)NC(c2nccnc2C)=O)n(C2CCC2)n1 N1(C(c2c(CC)[nH]c(=N)s2)=O)CC2CCN(C(C3CCC4(CCC4)O3)=O)C2C1 c1(C(=O)NCC2CCCCC2)occ2c1CCOC2.C1(C=O)CCC2(C1)N=N2.N C1(NC(c2cc(CC)on2)=O)CCN(C(c2cnc(Cl)[nH]2)=O)CC1CO N1(C(C2C(C)=CCC=C2)=O)CCC12CCN(Cc1ccc(O)c(C)c1O)CC2 Cc1ccccc1CC(=O)NC1(CNC(=O)C(c2cccnc2)C)CCCC1 c1(C(N2CC(F)CC(C(=O)Nc3cc(C)cc(Cl)n3)C2)=O)nc(C)c(C)[nH]c1=O c1(CC)c(C(N2CC(F)(CNC(C3CC4CCC3C4)=O)C2)=O)cccc1C c1(C(=O)NCC(C)NC(=O)C2CCc3ccccc32)ccc2nc(O)n(C)c2c1 c1(C(=O)NC23C(CN(C(CN(C)CC)=O)C2)C3)cc(C)c(OC)c(Cl)c1 N1(C(CSc2c(C)ccc(C)c2)=O)CCOC2(C1)CN(C(=O)CP(C)(C)=O)C2 N1(C(C=Cc2c(C)cccc2)=O)CCC2CCN(C(=O)C=Cc3cc[nH]n3)C2C1 Cc1ccc(CC=O)cn1.c1(C(N(CC)C2CC2)=O)cc(C(C)(C)C)nn1C.N N1(C(CN(S(C)(=O)=O)C)=O)CC2CCN(C(C3(F)CCCCCC3)=O)CCC2C1 N1(C(COCC=C)=O)CC(NC(=O)C(c2ccccc2Br)(F)F)C(F)C1 CC1(CNC(C2CSCCN2C(=O)C(F)OC(F)(F)F)=O)CCOCC1 CC1(C)CCN(CC(=O)NC2CC(NC(C3(c4ccsc4)CC3)=O)C2)C1 c1(-c2c(F)cc(OC(F)F)cc2)cccn2c(CCc3ccccc3)nnc12 N1(C(c2cn(CC(CC)O)nn2)=O)CC2(CCCC2NC(c2ccccc2)=O)C1 C1(CNC(c2cnc(C)nc2)=O)CCN(C(C2CCC(C)CC2)=O)CC1O C(N=C1Nc2ccccc2Sc2ccccc21)CN1c2ccc(F)cc2CC1 N1(CC=C)CC=C(CNC(c2c(F)cccc2F)=O)CC1 N1(C(c2cc(C)c(C)o2)=O)CC2CC1CN(C(=O)C(CC(C)C)NC(N)=O)C2 c1(C(=O)NCC(C)(C)NC(C2NC(=O)CC(C)C2)=O)nccc(C#N)c1F C1(OC)CN(C(c2cc[nH]c2C2CC2)=O)CC1NC(c1cc(CF)on1)=O Cc1cc(=O)c(C(=O)NCc2cc(C(=O)NC3(C)CCSC3)ccn2)c[nH]1 c1(C(=O)NC(C2CN(C(C3(O)CCC(C)CC3)=O)C2)C)cc(F)c(F)c(F)c1F c1(C2(NC(C(=O)Nc3cc(Cl)cc(Cl)c3F)=O)CC2)cc(F)c(F)c(F)c1 N1(C(c2ccc(O)nn2)C)CCC(C(=O)N)C1(C)C.c1cc(C(F)(F)F)n[nH]1.C C1(C(c2ccccc2)NC(c2cn(C)nc2)=O)CCCC2(CCOC2)O1 c1(C(N2CCN(Cc3cc(C)[nH]n3)CC2CO)=O)c(Br)cc(F)c(F)c1F N1(C(C(COCC)C)=O)CCCCC1CCC(=O)Nc1ccc(O)nc1 C(=O)(C(O)P(C)(C)=O)N(CCCC(C)C)C.C1(S(C)(=O)=O)(C(=O)N)CC1 C1(N(C(CCC)=O)C)CCC2CN(C(C3CC(O)CN3C)=O)CC12 n1(C(C)(C)C)cc(C(=O)NCC2CC2)cn1.C1(C=O)CCC1n1ccnc1 N1(C(c2c(C)cc(CC)o2)=O)C2CCCC1CN(C(C1CCSC(C)C1)=O)C2 N1(C(c2csc(C)c2N)=O)CCC2(C1)CN(C(C1CCCN1C(C)C)=O)CCO2 C1CC(C)CN(C(=O)C(C)(C)CN(C)C)C1.n1(CC)cc(CC(=O)N)cn1.C C(=O)(CC(C(C)C)NC(=O)C(O)CC)N(CC(=O)NCC)C C(=O)(C1=C(C)CCC1)N1C(CNC(CC(=C=C)C)=O)C(C)CC1 c1(OCC)ccc(CC(=O)NC23CC(C2)C3)nc1.C1(C=O)C(C)C1C.C C1(C(N2C(CNC(=O)Cc3cncnc3)CCC2)=O)CC2CCCN2C(=O)N1 N1(C(C2CCC(C)CC2)=O)CCC(CO)C(NC(=O)CC2CCCC(C)(C)C2)C1 C(=O)(CCCCN=[N+]=[N-])NC1C=CC(CC(=O)NCc2ccnc(OC)n2)C1 n1(CC)cnnc1C(=O)NCC(C)(C1CC1)NC(c1cnoc1)=O C1(NC(C(CN(CC)CC)F)=O)CCCC12CN(C(=O)CS)C2.c1cccs1 C1(CNC(c2c(CC)nco2)=O)CC(OC)CN1C(=O)C(C1CCOCC1)O C1CC2CCC1N2C(c1cn(C(F)F)cn1)=O.C(C=CC(=O)N)(CC)=CC C1(CC(=O)NCC(CC(C)C)C)CN(C(=O)C(C)NC(N)=O)CC12CC2 C1(C(=O)NCC2CCCN(C(CCC#CC)=O)C2)CCCC(C)(C)CC1 N1(C(C2C(=C)C2)=O)CC2CCC1CN2C(=O)CCc1nc(C)cs1 C1(NC(CC2(C)OCCO2)=O)CCCC12CCN(C(c1ncccc1Br)=O)C2 Cn1nc(C(=O)NC2CCCCC2NC(=O)CN=S(C)(C)=O)c2nc[nH]c(=O)c12 C1(F)(CNC(C(CCC)O)=O)CCN(C(C2CC2C(C)O)=O)CC1 N1(C(CN(CCC)C)=O)CC2CCC(C1)N2C(c1snc(C)c1N)=O C#CCCCCCCC(=O)N(C(C)CNC(c1cccc2ncccc12)=O)C c1(C(=O)NCC2CC(NC(=O)C(F)F)CC2O)ccn2nnnc2c1 N1(C(=O)NCC(F)CO)CC2COCC2(Nc2cncc(Br)c2)C1 Cc1nc(NC(C2CC3CC3N2C(c2ccc(I)cc2Br)=O)=O)c(F)c(Cl)n1 N1(C(C2(C)CCCOC2)=O)CCCCCC(N=c2[nH]c(Cl)nc3c2CCOC3)C1 c1(C(N2CC(CNC(CCC(=O)OCC)=O)C(C)CC2)=O)cc2sccc2n1C c1(C(=O)NC2C3CN(C(C(CC#C)(C)C)=O)CC32)cc2sc(Br)cc2s1 c1(NCC)ccc(C(=O)NC(C)CNC(=O)CC2CCOCC2)c(Cl)c1 n1(CC)ncc(C)c1C(=O)NC1CC2CC2N1 N1(C(c2cc(C)[nH]n2)=O)CCC2(NC(c3cc(C(F)(F)F)cc(F)c3)=O)CC2C1 Cc1nc2c(s1)CC(NC(=O)C(=O)Nc1ccc(-c3ccccc3)cc1F)CC2 C1(C(N(CCNC(c2ccc(-c3nc(C)sc3)s2)=O)C)=O)CCCCC1CN C(=O)(NN1Cc2ccccc2C1)N1CCC(CCCS(N)(=O)=O)CC1 c1(C2(C(=O)NCCN(C(=O)C=Cc3cnccn3)C)CC2)cccc(Br)c1 C(=O)(CCCCCCNC(=O)C(C#N)C(C)(C)C)NCCCCOC C1(CN(C(C=C(COC)C)=O)C)CN(C(c2cc(CCO)on2)=O)CCO1 Cc1ccc(COC(C)C(N2CC(F)CC2C)=O)cc1.c1(C=O)nonc1N.N c1(C(=O)NC(C)CO)[nH]nc([N+](=O)[O-])c1Cl.C1(C=O)CC(C(F)(F)F)C1.N N1(C(C2CC(C(C)C)OCC2)=O)CC2(CNC(=O)C3=CCCC3)CC(F)(C1)C2 c1(C(N2CCC(NC(=O)CC3CC4CC4C3)CC2)=O)cccc2nccn12 c1(CC(=O)NCC(CC)NC(C2CC(F)C2)=O)c[nH]c2ccc(Cl)cc12 Cn1cnc2cc(-c3cc(NCc4cccc(Br)c4O)ccn3)ccc12 c1(N(CC(C)C)C)nc(N(CC(F)(F)Cl)C)nc2ccccc12 N1(C(CCC)=O)CCN(N2Cc3cnc(C(C)C)nc3C2)CC1 C1(NC(C2(NC(=O)OCC)CCCC2)=O)CN(C(=O)C(C)CC)CC1.O N1(C(CC=C(C)C)=O)CCC(C)C(NC(=O)CSc2cnn(C)c2)C1 N1(C(c2ccnn2C2CNC2)=O)CCc2ccc(Br)c(F)c2C1 CC(C)(CC(=O)N1CCN(C(c2ccc(O)c(N)n2)=O)CC(O)C1)C(F)F C=Cc1cc(C(N2CCN(C(C3CCS(=O)(=O)C3)=O)CC2C(C)C)=O)cc(F)c1 Cc1nn[nH]c1C(=O)N(CC(C)N(C(=O)Cn1ccnc1C)C)C Cc1ccnc(C(=O)NC2(c3noc(C4CCS(=O)(=O)C4)n3)CCOC2)n1 N1(C(c2c(OCC=C)cc(OC)cc2)=O)CC2CCC(=O)c3cccc1c32 CCC(C(=O)N)C(C)(F)F.c1ccccc1C(N)=O.C1(O)CN(C(=O)C)C1.C C(=O)C(C)(C)CC(C)(C)C.c1(NCC)ccc(C)cc1C(=O)N.C(C)CCC Cc1cnc(C(=O)NCc2ccccc2)c(F)c1.C1(CC=O)CC2(CC2)C1.C c1(SC)cccnc1C(=O)NCC1CCN(C(C2NC(=O)CC2C)=O)C1 c1(C(=O)N)ncnc2c1CCCC2.Cc1nn(C)c(C)c1C(=O)N(CC)C1CC1 c1ccc(C(F)(F)F)cc1S(=O)(=O)N1CCC(P(C)(C)=O)C1.C(C)(C)(C)SC CCC(CC(=O)N1CCC(CNC(c2cccc(C3CCC3)c2)=O)CC1)OC CCCCCC(O)C(=O)NC1CCCCC1NC(C1(Cl)CC1)=O Cc1cc(C(=O)NCCCC2CCCCN2C(=O)CCc2ncccn2)sc1C C1(N(C(c2csnc2Cl)=O)CC)CCCN(C(=O)C(C2CC2)SC)C1 N1(C(=O)COCC2CC2)CCCC1C.C1(C2CCCO2)(C(=O)N)CCCC1 c1(C(=O)OC)ccc(C=CC=O)cn1.C1(C(N(CC)C)=O)CC2(CC2)CO1 Cc1cn(-c2ccc(Cl)cc2)[nH]c1=NC(=O)NNC(=O)NCC1CCCO1 CC1CCc2[nH]nc(C(=O)NC34CCCC3N(Cc3nncn3C)CC4)c2C1 C#CC1CC2(CC2)CN1C(=O)C(F)(CNC(=O)CCCc1cnn[nH]1)C(C)C C1(C(=O)NC(CC#C)C(=O)N(C)Cc2cccc(C)c2)CC2OC1C1CC21 N1(C(=O)C=CC2CC2)CC2CCCC1C2CNC(=O)C(F)(F)c1cccnc1 C1(C(N(CCN(C)C)C)=O)CN(Cc2c(Cl)ccc(Cl)c2Cl)CC(F)(F)C1 C(CCC(N)=O)(C(=O)N1CCC2(CC2)C1)N(C)C.C(=O)(C(C)(C)CN(C)C)N C(=O)(C(S(C)(=O)=O)C1CC1)N(CC(C)(C)NC(=O)CCCc1ccsc1)C Cc1cncc(CCNC(=O)NCC2(O)CCOC2)n1 C1(NC(c2cc(=O)cc(Cl)[nH]2)=O)CC2(C1)CN(C(=O)C=Cc1ncc[nH]1)C2 C1(CNC(c2c(SC)cccc2)=O)CCCN(C(C2(Br)CC2)=O)CC1 N1(C(CCc2nnc(C)n2C)=O)CCOCC(CNC(=O)CSS(C)(=O)=O)C1 Cc1c(Cl)ccc(C(=O)NC2CC(F)CN(C(=O)CCN3CCCC3=O)C2)c1O c1(C(=O)NCC(CCNC(=O)CC2CC=CCC2)O)ccnc2[nH]cnc12 Cc1ccc(Br)c(C(N2C3CCC2CN(C(C2Cc4nccn4C2)=O)C3)=O)c1F C1(NC(C(CC)CN(C)C)=O)CC=C(C(=O)N2CCC2CC2CCCC2)C1 N1(C(CCOC)=O)CC2(CCN(C(=O)CCCS(=O)(=O)N3CCCC3)C2)C1 c1(CC(=O)N(C2CCCCC2)CCNC(C(C)C2(O)CCC2)=O)cncnc1 c1(NC(C2CCCC2O)C)noc(=O)n1C C1(NC(CCCSC)=O)CCN(C(C2(C)CCC(C)C2)=O)CC1(C)C C1(Cl)(C(=O)NCCCN(CCCNC(C=C(C)Cl)=O)C)CC1(F)F c1(C(=O)NC2CN(C(C3(C)CC3(Cl)Cl)=O)C2)ccc2nccn2n1 c1(C(N2CCC2)=O)cc(C)n(NC(N)=O)c1C.Cc1oc(C)c(C(=O)NC)c1C CN=c1[nH]c(C(=O)NC(C)CCCNC(c2ccccc2)=O)cs1.C(C(C)C)O C(C(CC(C)C)C(=O)NCC(C)NC(c1coc(O)n1)=O)OC c1(C(=O)NC2CCCN(C(C3(C#N)CC3)=O)C2)ccc2c(c1)OCCNC2=O CC(C)C(CCC(=O)NCC1(CO)CCCO1)NC(c1ccc[n+]([O-])c1)=O c1(C(N2CC(C3OCCN(C(C(CC)OC)=O)C3)C2)=O)cccc2ccn(C)c12 C(C(C)(C)C(=O)NCCC(C)N(C(=O)CC1C(C)(C)C1(C)C)C)OC N1(C(c2cnc(C(=O)OC)s2)=O)CC(NC(=O)CCC2CCCO2)C(C)C1 N1(C(c2ccc(F)c(I)c2)C(=O)NCCC2CC2)CCC2(CCCCO2)C1 C1(C(=O)N(C)CCNC(=O)CSCCC(C)C)(CC)CCCCC1 C(=O)(CCC(=O)NCc1ccc(C(=O)N(CC(F)Cl)C)o1)NC c1(CCC(=O)N(CCC)CC)c(C)nc(O)nc1O.C1(CC(=O)N)CCCCO1 C(C(N=[N+]=[N-])C(=O)N1CCCC(C(N2CCC(OCC(N)=O)C2)=O)C1C)OCC C(C)(C)(C(=O)NCC1CCCC1NC(C1(O)COC1)=O)OC(C)C C1(N(C(CN(C(=O)OCC)C)=O)C)CCN(C(C2CC(F)(CF)C2)=O)C1 N1(C(C2CCCN(C(C)=O)C2)C(=O)NCC2CCCO2)CCC2(CC1)CC2C#N C(=O)(CCCC(C)(C)C)N1C(CC(=O)N(c2ccsc2)C)C2CCCC21 N1(C(c2c(CC)csc2)=O)CCc2c(c(C)nn2C)C1.C(=O)C(F)(F)C(C)O.N c1(C(=O)NC2CCC(C(=O)NCC3N(CC)CC3)C2)cc(C#N)ccc1N C(CCC(=O)NCC(O)CO)NC(C1C(C)CC1)=O C(=O)(C(O)C(F)(F)F)N(CC(N1CCC(CC(C)C)CC1)=O)CCC N#CC1CC=C(c2ccc3cc(C(=O)NCC4CCOC4)nn3c2)CC1 c1(CC)c[nH]cc1C(=O)NCC1CCN1C(=O)C(COC)OC C1(NC(C2CSC2)=O)CCCN(C(C2CCN(C(=O)NC3CC3)CC2)=O)C1 C(C(=O)N(C1(C(=O)NCc2cn[nH]c2)CC1)C)(C(C)C)OCC c1(C(=O)NC2CN(C(c3cncc(OC)c3)=O)CC2F)cccc2nscc12 C(=O)(CC(CC(C)C)NC(=O)CC1(C)CCOC1)NC1CC(C=C)C1 Cc1csc(=NCC(=O)N2CCCC2C2(NC(=O)COCC(C)C)CC2)[nH]1 Cc1cc(C)n(-c2ccc(NC(C3C4CC(N)CC34)=O)cn2)n1 C1(C(=O)NCC(CC)C#N)CCC2(CC2)N1C(c1c(C)cnn1CC)=O c1(OC)c(Cl)cc(C(=O)NC(C)C(C)C)cc1Cl.C(=O)(CCCc1cccs1)N C1(C(N2CCC3(N(C(CC(C)SC)=O)CCC3)C2)=O)C2Cc3cc(Cl)ccc3C12 Cc1ccc2c(c1)N(C(=O)C(C1CCN(C(=O)C(n3ccnc3C)C)C1)C)CC2 c1(NC(C)C)cc(=NC(C)c2ccc3c(c2)CCCC3)[nH]c(NCCO)n1 C1(NC(C2CCOC2)=O)CCN(C(=O)CCc2ccc(F)cc2F)CC(O)C1 N1(C(CCC#C)=O)CCC(CCOC)(C(=O)NCCc2cncn2C)CC1 CC1CC=C(C(=O)N2CC(C3(NC(C4CC5CCC4O5)=O)CC3)C2)CC1 c1(CC(N2CC(C3CN(C(C(F)=CC)=O)C3)C2)=O)ccc(S(=O)CC)cc1.O c1(C(NC)=O)ccc2c(c1)C=CS2(=O)=O.N1(C(CN(CCC)C)=O)CCCC1.C c1(C(=O)NCC2C(NC(c3n(C)ccn3)=O)CCC2)ccc2cn(C)nc2c1 N1(C(c2c(C)nns2)=O)CCC2C(C1)CN2C(C1CS(=O)(=O)C1)=O c1(C(CC)(C)C)ccc(C(N2CC(OCCNC(c3cnccn3)=O)C2)=O)cc1 N1(C(c2c(C)sc(Cl)n2)=O)CCC2(CCN(C(C34CC(C)(CO3)C4)=O)C2)C1 c1(NCCC(C(C)C)OC)ncc([SH](=O)=O)cc1Cl.C1(C)(N)CCCC(C)(C)C1 c1(C(=O)OC)ccc(Br)cc1C(=O)NC1CCCC1(C)O Cc1nc(C(=O)NC(C)C(C)NC(=O)CCSc2nccn2C)c2n1CCCC2 c1(C(=O)OC)ccccc1.N1(CC=O)C(=O)CCC1=O.C1CCC1.C(C=O)O c1(OC)ccc(NC(=O)NC(CC(=O)NC2CC2)CC2CC2)cc1O n1(CC)nc(C(=O)NCC(C(C)C)NC(=O)CC2(O)CCCCC2)ccc1=O CC(C)C(C(=O)NCC#CCNC(=O)CCC1CCCCO1)c1ccncc1 C(C(C)S(C)(=O)=O)NC(CCC1C(C)(C)C1)=O.C(c1ccc[nH]1)=CC=O.N C1(CC(N2CCCC2)=O)CCCC(C)(C)C1.c1(CC)ccc(C(=O)N(C)C)cc1 CCCCCC(O)CC(=O)N1CCCN(C(=O)C(O)C(F)(F)F)CC1CO N1(C(CCCN(C(=O)CCC2CCCCC2)C)=O)CCC(C2CCC2)C1 c1(CCC)ccccc1C(N1CCOC(C(C)NC(C2(F)CCOC2)=O)C1)=O c1(CCC(=O)NC2CC2NC(=O)CCC(F)(F)F)ccc(Br)c(F)c1 C1(CC)(NC(c2coc(C)n2)=O)CCN(C(=O)CCc2ccc(Cl)nc2)CC1 C1(COC(C2CC23CC3(F)F)=O)CCN(C2CC2)CC1 N1(C(C2(SCC)CC2)=O)CC2CCC1C2NC(C1ON=C(C)C1C)=O c1(CC)[nH]nc(C(N2CCC(CF)(NC(C3CCCC3C)=O)C2)=O)c1[N+](=O)[O-] c1(CC(=O)NC2C(C(=O)Nc3snnc3-c3ccccc3)C2)cccc(F)c1 CCC(C)CC(=O)C(=O)N1CCOCC1C(=O)NOC(c1ccccc1)C N1(C(Cc2cn(CC)nc2)=O)CCCN(C(=O)Cc2cn(C3CC3)cn2)CC1C N1(C(CCn2c(C)cc(C)n2)=O)CC2(C1)CN(C(=O)CCOC1CCC1)CCO2 C(C1=NOC2CN(C(c3cc(F)c(O)c(Cl)c3)=O)CC12)NC(CS(CC)(=O)=O)=O CC1(C)CN(CC(=O)N(C)C)CCC1NC(=O)CC1CCCOC1 c1(CC)ccc(C(=O)N(CCCOCCNC(c2c[nH]nc2Cl)=O)C)o1 C(=O)(CS(=O)(=O)CC)NC(CC)CNC(c1cnc(C(F)(F)F)s1)=O C(CCCC(=O)NCC(N1CCN(C(C2CCCC(C)C2)=O)CC1)C)OCC c1(SC)cc(C)ncn1.C1(C=O)CC(O)CN1C(c1cccnc1C(N)=O)=O.N CCCCC(O)CC(=O)NC(c1cn(C)nn1)C(N1CC2CCC(C1)C2O)=O CC1(C)CC(C(=O)NCC2CCC2NC(=O)C)CNC1=O.c1ccccn1.O c1(C(=O)NC(C(C)NC(CCNC(=O)OC)=O)C)cccc(C)c1F n1(CC(=O)NCCC(C)N(C)C(C2CCNC2=O)=O)cnc(Br)c1 C(c1cnn(C)c1C)=CC(N1CCC(N(C(=O)C2=CCSC2)CCC)C1)=O C1(C(N(C(C)C)CC)=O)CCN(C)C(=O)C1.C1(C(=O)N)CC(C)(C)CO1 CC1Cc2cc(C(=O)NCCC3CCCN(C(C4CS(=O)(=O)C4)=O)C3)ccc2O1 N1(C(c2ccc(CC)nc2)=O)CC2CC(NC(c3csc(CC)n3)=O)C(C2)C1 C(=O)(C1CN(CC)c2ccccc21)NCC(CC)NC(c1c(CCC)n[nH]c1)=O c1(C(N)=O)ccc(C(=O)NC2CCCCC2NC(=O)Cc2ccsn2)cn1 CC1(NC(=O)Cc2cnn(C3CC3)c2)CCCN(C(C2CCCCC(=O)N2)=O)C1 c1(C(C)O)ccc(C(=O)NCCC2CN(C(=O)C3=CCCS3)C2)cc1 N1(C(c2c[nH]nc2[N+](=O)[O-])=O)CCC2(CCCN2C(c2sc(F)cc2Cl)=O)C1 c1(C(=O)NC2CCC(NC(C3N(C)CC(C)(C)C3)=O)CC2)cc2c(s1)COCC2 c1(COC)cc(C(=O)N(C)CCNC(=O)Cn2cc(Cl)cn2)on1 Cc1cc(C)c(C=CC(N2CCN(C(=O)C(F)C3CC3)CC2C(C)C)=O)cc1C c1(-n2ncc(C)c2)ccc(C(=O)NCC2CC2)cc1.C(=O)C(C)C.C(=O)C N1(C(C2CN(C(C(CCOC)C)=O)CC(C)(C)C2)=O)CC2(COC(=O)N2C)C1 c1(CNC(C2CCN(C(=O)NCC=C)CC2)=O)c(C)cc(OC)cc1C C(=O)(C1CCCc2cccnc21)N1CCN(C(C(COC)(C)O)=O)CC2(C1)CC2 C(=O)(C1=COc2ccccc2O1)N1CC(C)(F)CN(C(C2(C)CC2Br)=O)CC1 N(C(=NCCc1ccns1)N1CCC(Cc2ccc(C)cc2)C1)C(C=C)C C1(C(=O)NC(C)CCCCNC(=O)C(C)(O)C2CCC2)CCC(C)(C)CC1 C(=O)(CCCS(N)(=O)=O)NC(CNC(C(C(=O)OC)OC)=O)CO C(=O)(C#CC1CCOCC1)NC1CC(C)(NC(CCCC(=O)NCCC)=O)C1 c1(C(=O)NCC(CN(C)C(C2CC(F)C2)=O)O)cc2cccc(Br)n2c1 c1(OCC)ccc(C(=O)N(C2CCCN(C(C3(O)CCC3)=O)C2)CC)cn1 CC1COCC(C(N2CC=CCC2C(=O)NC(C2CCCC2)CO)=O)O1 c1(NC(C2CC2NC(C2(O)CC2)=O)=O)cncnc1 CC(CC(C)NC(=O)C=CC1CCCC1)NC(=O)C(C)(C)n1cccn1 c1(C(C)C)conc1C(=O)NCC(C)NC(=O)C(C)(C)n1cnnn1 C1(CC)CN(C(c2cc(OC)ncc2F)=O)CCN1C(=O)CC(O)C(C)C C1(CCC)CN(C(c2sccc2C(C)=O)=O)CC1C(N1CC(C)=C(C)C1)=O CCCCC(CC)C(C(=O)NC(CC(C)C)C(=O)OC)N(C)CCN(C)C1CC1 CC(C)(CC(=O)N1CC2CCN(C(=O)CN3CCCCCC3=O)CC12)C(F)F Cc1ccc(C(=O)NC2(C)CN(C(=O)CCc3ccn(C)n3)C2)nc1O C(C(=O)N1CCCC(NC(C2CCCCS2)=O)C1)(C(C)C)OCC(C)C c1(C(=O)OC)c(NC2CCCC(CC(N)=O)C2)nc2c(OC)cccc2c1Cl c1(CNC(C2C(CCC(C)C)CCC2)=O)ccnc(Cl)c1F C1(NC(C(C)C2CCC2)=O)CN(C(=O)Cc2nc([N+](=O)[O-])n[nH]2)CC(C)(C)C1 C(=O)(CN=c1cc[nH]cc1)N1CCC(NC(CCCN(C)C)=O)C1(C)C c1(OCC(N2CCN(c3c(C)cccc3C)CC2)=O)cccn2c(C)cnc12 c1(C(=O)NC2C=CC(CNC(C(C=C)O)=O)C2)cccc(O)c1Cl N1(C(c2occ(C(=O)OC)c2)=O)CC2CCC1C(NC(C1CCCC(O)C1)=O)C2 C1(NC(C2(NC(C3CCC(C4CC4)C3)=O)CCSC2)=O)CCCN(O)C1=O C=CC1CN(C(=O)Cc2cccc(F)c2O)CC1NC(C1(F)CC1)=O c1(C(=O)Nc2c(C)c(OCCO)ccc2)c2c(nn1C)CCSC2 c1(NC(C)Cn2ccnc2)nc(N2CCCCC(CO)C2)nc2scnc12 CCCS(=O)(=O)C(C)C(=O)NC1COC2(C1)CN(C(c1ccc(F)cc1C)=O)C2 C=CC(C)(O)C(=O)NCCC(C)NC(C1(c2ccc(Cl)cc2)CCOCC1)=O c1(-n2cc(N(CCN(C(COC)=O)C)C)nn2)ccc(Br)cc1 c1(N(C)C)nc2ccc(NC(C3CCCCN3C(=O)CNC(N)=O)=O)cc2o1 C1(NC(=O)CC2CCOC2)CCC2CN(C(=O)C3=CCCS3)CCC2C1 C1(CC(=O)N(C(CC)C(=O)NCCN=[N+]=[N-])C)CCC(=O)N1C c1(C(=O)NCC(C(C)C)NC(C2(C)CC(C)C2)=O)ncc(C(N)=O)cc1Cl Cc1cc(NC(=O)NCCCOc2cccc(Cl)c2)nn1C C(=O)(CC1=CCOCC1)NC(C(C)NC(c1c(C)scc1)=O)C c1(CC)c(C(N2CCCC2CN(C(c2cnoc2C)=O)CC)=O)cnn1CC N1(C(C(C(C)NC(c2cc(CCC)on2)=O)C)=O)CC2(CCC(=O)N2)C1 c1(COC)ccccc1CC(=O)NC1(CF)CCN(C(=O)Cc2ccco2)C1 c1(C(N(C)C)=O)ccc(C=O)cc1F.c1(C(C(N)=O)C2CC2)ccc(Br)cc1 c1(C(N(CCCCCNC(c2cc(=O)cc[nH]2)=O)C)=O)cnn2ccncc12 CN=c1[nH]nc(CC(=O)NCC2C3CN(C(=O)CCn4cc(C)cn4)CC23)s1 C1(C)(C(=O)NC(C)Cc2nccn2C)CC12CCN(c1cncc(CO)n1)CC2 C1(C(C)NC(c2c(CC)ocn2)=O)CCN(C(c2ccccc2Br)=O)CC1 C(C(F)(C(=O)NC)C(C)C)NC(c1c(COC)cco1)=O.c1ccccc1F C1(NC(C(C)N(C)C)=O)CC1C1CCN(C(c2noc3cc(F)ccc23)=O)CC1 C1(OC)CC(CNC(=O)C)N(C(=O)C(F)=CCCF)C1.c1csc(C)n1.S C1(CNC(CCC#C)=O)CN(C(c2ccc(N(C)C)c(F)c2)=O)CC1(C)C Cc1ncccc1C(=O)NC(CNC(C1CCCCN1CC(F)F)=O)CO C1(N(C)C(c2ccc(CO)cn2)=O)CC2CC1N(C(=O)C=Cc1cnccn1)C2 C(=O)(C(CCC(C)C)NC(=O)CCCC(=O)C1CC1)N(CC)Cc1ncc[nH]1 N1(C(C2CC(C(=O)OC)C2)=O)CC(CNC(C2CC(F)C2)=O)C(O)C1 Cc1c(CC2CC2Cc2ccccc2Cl)nnn1-c1ccc(OC2CC2)cc1 N1(C(COCC=C)=O)CCC(CCNC(c2nnsc2N)=O)CC1C C1(NC(c2ccc(CC)o2)=O)CN(C(c2cc(Cl)ccc2O)=O)C(C)(C)C1 C1(C(=O)NCC2(O)CCC(C)C2)CCN(C(C2CC(O)C(F)C2)=O)CC1(C)C C1(NC(CC(C)F)=O)COC2C(NC(=O)COC(F)(F)F)COC12 Cc1ccc(C(N2CC3C(C(=O)Nc4cccc(C#N)n4)C3C2)=O)cc1O C1(NCc2cc(OC(CC(C)C)C)ncc2)CCC23OCCC2CC13 C(C=O)C(C)O.c1(C(N(CCCC)C)=O)cn(CCC2CC2)nn1.CC=O.N N#Cc1cc(CNc2cncc(-c3cccnc3C3CC3)n2)ccc1Br Cc1ccc(Cl)c(NC(c2cccc(NC(c3cccnc3CN)=O)c2)=O)c1 C1(C(=O)NCCNC(CC(C)N(C)C)=O)CCCS(=O)(=O)N1 N1(C(C(CCC#C)O)=O)CCC(C2(NC(=O)C=Cc3nccs3)CC2)C1 C1(C=O)CCCC2(CC2)C1.C1(C=O)CC1(C)C.C1(CCOC)(C)CCC1.N c1(N2CCC(CCOC)(NC(c3conc3C3CC3)=O)C2)nccnc1C#N C(=O)C1CCCn2nccc21.NS(=O)(=O)C1(C(=O)NC2CCCC2C)CCC1.N N1(C(Cc2c(C)non2)=O)CC2CCC(C(=O)NCCN3CCC(O)CC3)(C2)C1 C1(C(=O)NC(C2CN(C(c3cc(C)nn3C)=O)C2)C)CCCC(F)(F)C1 c1(C(=O)N)cc2c(ncn2C)[nH]1.C(=O)(C(C)N=[N+]=[N-])N1CC(COC)(C)C1 C1(NC(C2(C(F)F)CC(=C)C2)=O)CCN(C(=O)COc2ccccc2)CC1O C1(NC(C2CC=CCC2)=O)CN(C(C23CCC(CC2)OC3)=O)CC(F)(F)C1 C1(OC)CN(C(C2CC(=O)C2C(C)(C)C)=O)C1.C(=O)C(C)(O)C1CCC1 C(=O)(C1=CCCCC1C)NC(CCC)CC(=O)N(c1cccc(C#N)c1)C C#CC1COCCN1C(=O)CC1CN(C(=O)Cc2ccsc2C)CCO1 O=S1(=O)CC23CCCCC2(CN(CC(c2ccc(F)cc2F)O)C3)C1 CCCCC(C(=O)OCC)OC(=O)COC1(C#N)CC12CCC2 N1(C(C)=O)CCC2CN(c3cc(O)nc(C)n3)CC2CC1 C(=O)(C1=NOC(C)C1C)N1CCCC(C(C(=O)NCC(COC)(F)F)(C)C)C1 Cc1cc(C)nc(SCC(N2CCC3C(NC(=O)C(F)(F)C4CC4)CC23)=O)n1 CC1(C)CCCN(C(c2ccc([N+](=O)[O-])cc2)=O)C1C.c1(CC(=O)N)ccoc1 c1(-c2ccc(C)o2)nc(C)c(C(=O)NC2CCC2(C)C)s1.C(=O)CNC=O.C c1(C(=O)NC(C2(O)CCN(C(=O)CO)C2)C)cc(C(N)=O)cc2ccccc12 C(=O)(CCCCn1cc(CCS(C)(=O)=O)nn1)NC(c1ccc(Cl)cc1)(C)C N1(C(C(F)OC)=O)CCC(C)(C)C(NC(c2cnn(C(C)(C)C)c2C)=O)C1 CC(c1cnn(C)c1)=CC(N1CCC(NC(=O)C2=CCCCO2)C(C(C)C)C1)=O N1(C(C(CC)N(C)C)=O)CCCCC1CC(=O)NC(C)C.C1CC(=O)N1 C(CC(CC)C(=O)NCCOCCNC(c1ccc(N)c(N)n1)=O)=CC S(=O)(=O)(c1cc(Br)ccc1Br)N(C1C2CCC1CNC2)c1ccc(CC)cc1 c1(OC)nc(C)cc(=NC2CCOC3(CCN(C(c4cocn4)=O)CC3)C2)[nH]1 N1(C(C2C(CC(C)(C)C)C2)=O)CCC(NC(=O)CNC(N)=O)C(O)C1 C1(CNC(C(C)SC)=O)C2CCCC1N(C(=O)CC(C)SC)C2 CC(C)CC(CNC(C1(C)CCSCC1)=O)NC(C1CCC(=O)O1)=O N1(C(c2cc(COC)cn2C)=O)CCC2(NC(c3nnsc3C)=O)CC2C1 c1(C(N(CC(CC)NC(=O)CCOC2CCCCC2)C)=O)ncn2c1CCC2 C1(C(N2C3CC(C3)C2)=O)CCC(=O)N(C2CC2)C1.C(C(C)C(=O)N)OCC C1(NC(c2ncccc2Br)=O)CC2CC1CN(C(c1cnsc1)=O)C2 c1(OC)ccc(C(=O)NCC2CCCC(CNC(=O)CC(Cl)Cl)C2)cc1F N1(C(c2c(CC)cc(F)cc2)=O)CCC2(CC(NC(C3CCC(O)C3)=O)C2)C1 N1(CCNC(=O)NC2CCN(c3nc(=N)[nH][nH]3)C2)CCCC2(CCC2)C1 Cc1cc(C(N2CCCC(O)(CNC(C3CCC(O)CC3)=O)C2)=O)ccc1O C1(NC(CC(CC)O)=O)CC12CCN(Cc1cccc(F)c1I)CC2 N1(C(C2CC(OC)(OC)C2)=O)CCC(C(N2CCCCC(C)C2)=O)CC1C c1(NCC)ccc(C)cc1C(N1CCC(N(C(=O)C(COC)CC)C)CC1)=O Cc1nn(C)cc1C(=O)NCC#CCNC(c1cccnc1OCCO)=O C1(C(N(C)CC2CC2(C)C)=O)CCCN1NC(=O)C1CC2C=CC1O2 N1(C(CCCN(CCC)CCC)=O)CCN(C(=O)C2=CCCCO2)C(C(F)F)C1 C(=O)(C1=CCOCC1)NCCN(C)C(c1cc(C2CC2)ccc1F)=O c1(CC(N2CCC3C(COC)C3C2)=O)ccc(OC)c(OC)c1Cl CC1(C(=O)NCCC2CN(C(C3(C4CCCO4)CCOCC3)=O)C2)CNC(=O)C1 C1(CC)CCCCC1C(=O)NC1CCCN(C(c2csc(S)n2)=O)C1 C1(C(N(CCN(C(C=CC(C)C)=O)C)C(C)C)=O)CCC(N(C)C)CC1 C1(NC(Cc2cccc(OC)c2)=O)CCCCN(C(=O)CNC(=O)C2CC2)C1 C1(CNC(c2cc(C(F)(F)F)n[nH]2)=O)CCN(c2ncnc3ccsc23)CC1(F)F C1(CCCNC(CN(CCC#C)C)=O)CN(C(=O)C(C)c2ccco2)CCO1 N1(C(c2cnc(C)o2)=O)CC2CN(C(c3cc(Cl)c(Cl)c(Cl)c3)=O)CC2(C)C1 c1(CC)cc(C(=O)NCCCCNC(c2cc(N(C)C)nc(Cl)c2)=O)ccc1F c1(C(=O)N)csc2cncn12.N1(C(c2c(NCC)scn2)=O)C(C)CC2CC12 C1(CC)CCCCC1C(=O)NCC1CC(O)C1.C(=O)(CCC=C(C)C)N N1(C(C=C(C)C(F)F)=O)CC(N(C)C(c2ccnnc2O)=O)C(C)(C)C1 C12(CC)CN(C(C3CCC4CCC34)=O)C(C)(C1)C2.c1(C=O)ccc(N)cn1.N Cc1ccnc(N2CCC(N(C)C(C3CCCCC3C3CC3)=O)CC2)c1[N+](=O)[O-] C1(NC(COCCCOC)=O)CC(NC(=O)CCc2ncnn2C)C(O)C1 c1(C(C(=O)NC2CCC2)N(CC(F)F)CCC)cccc(SC)c1 c1(C(N2CCN(c3ccc([N+](=O)[O-])cc3)CC2)=O)cc(Br)cc([N+](=O)[O-])c1 c1(C=O)cc2cnn(C)c2s1.N1(C(CC(=O)OCC)=O)CCC(C(F)F)C1.C C1(C(=O)OC)CCCN(C(=O)C(C2CCN(C(=O)C(F)F)CC2)C)C1 C12(C(N3CCN(C4CCN(C(CC(C)F)=O)C4)CC3)=O)CCC(C)(CC1)CO2 N1(C(CCNC(=O)NC)=O)CCC2(CC1)CCN(C(=O)C(C)CS(C)=O)C2 c1(C(=O)NCCC2CC(NC(c3c[nH]ccc3=O)=O)C2)cc2c(s1)CCCCC2 C1(NC(C(COC)(C)O)=O)CN(C(c2ncc(C(F)F)s2)=O)C2CCCCC12 C12(NC(C(CCC)O)=O)CCCN(C(c3cc(Cl)c(Cl)n3C)=O)CC1C2 c1(C=O)cc(F)c(Cl)c([N+](=O)[O-])c1.Cc1ccn(C)c1C(=O)N(CC)CC NC(=O)CCC(=O)N.C1CCN(C(=O)C=CCNC2CC2)C1.c1ccccc1 C1(NC(c2cnc[nH]2)=O)CCCN(C(C2CCC=CCC2)=O)CC1F C1(CN(C(=O)CCc2ccccc2F)C)CN(C(=O)C=C2CCOCC2)CCO1 C(=O)(C(O)C(F)(F)F)NCC(C)(C)NC(C1CC1C1CC1)=O c1(CNC(C2(OC)CC2)=O)ccccc1.N1CCNC(=O)C1.n1(C)ccnn1 c1(CCNC(C(=O)Nc2c(OC)ccc(OC)c2)=O)c[nH]c2cc(Br)ccc12 C(CCCCCC(=O)NCC1C2CCCC12)NC(c1nc(C)oc1)=O C(=O)(C1CCCc2sc(C)nc21)NC(CC)(C)CNC(=O)C(C)(C)CCCOC C1(OC)CN(C(=O)OC(C)(C)C)CCC1NC(C1CCC(Br)CC1)=O c1(CC(=O)NC2(C)CCN(C(c3sc(C)c(O)n3)=O)C2)ccc2c(c1)CCCO2 N1(C(CNC(C(C)(C)C)=O)=O)CCC(O)(CCNC(=O)C(C)(Cl)Cl)C1 C(=O)(CCCCn1ccnn1)N1CC(NC(C(C)OCC(C)C)=O)C1 CC1CN(C(C2CCCN2C)=O)CCN1C(c1cc2n(n1)CCC2)=O CCCC(C(O)C(=O)NC(CCC)c1ccco1)NC(=O)CC1CC(C)(C)CO1 N1(C(c2cncc(C)c2)=O)CCN(C(c2cc3[nH]ccc3s2)=O)C2CCCCC12 c1(C(=O)NCC2=CCCN(C(CSC)=O)C2)cccc2nccn12 N1(C(C(=O)N(CCCNC(C(C)N(C(C)=O)C)=O)CCO)C)CCCCC1 C1(NC(C2N(C(c3ccccc3C)=O)CCC(CC)C2)=O)CCCCN(C)C1=O O=S(=O)(c1cnc(NC2CCCC2CCO)c(Cl)c1)N1CCCCC1C1CC1 C(=O)(C1CCSc2ccccc21)NCC(CNC(Cc1cccc(OC)c1)=O)C C12(C(=O)NCC(CCC)C)COC(C1)C(NC(c1ccn(CC)n1)=O)C2 c1(C(N2CCN(C(C=C(C)Cl)=O)C(C)CC2)=O)ccc2cnc(C)n2c1 C1(C)CCCN1C(=O)CN(C(=O)C(C)C)C.C(=O)CC(C)=C(C)C.CO C1(N(C(COCCC)=O)CCC)CCN(C(c2cnn(C)c2C)=O)CC1 C1(NC(c2c(CC)n[nH]c2)=O)CCN(C(c2cn(C)nn2)=O)CC1F N1(C(CCc2ccc(C)cn2)=O)CC2CCC1C(NC(=O)C(C)OC(C)C)C2 n1(Cc2nc(C(C)OCC)no2)ncc(Cl)c(Cl)c1=O N1(C(C2(C)CCC2)=O)CCC2CC(CNC(=O)C=CC3CCCC3)CCC2C1 N1(C(C2N(Cc3cc(C)cc(C)c3)CC2)=O)Cc2cccc(C)c2C1 N1(C(C(C)SCC)=O)CC(NC(c2cc(N)nc(Cl)c2)=O)CC(C)(C)C1 CC1N(C(=O)C(C2(O)CN(C(c3ncccc3N)=O)C2)F)CCOC1(C)C Cc1nn(C)c(-n2ccnc2C)c1NC(=O)CCN1C(=O)CCC1=O n1(C(C)C)cc(C(=O)NCC2CC2)cn1.C1CCOCC1.C(=O)(C)N(C)C C(C=O)(C(C)C)OCC(C)C.c1(C(N(CC)C(C)C)=O)ccc(Br)cc1.N C1(NC(CCCc2cc(C)sc2C)=O)CCN(C(=O)Cc2c[nH]nc2O)CC1C c1(C(=O)NCCCNC(C2CN(C(N)=O)C2)=O)cc(F)c(N)c(F)c1 c1(C(=O)NC2C(NC(CCc3n(C)ccc3)=O)COC2)nn(C)c2ccccc12 n1(CCOC)cc(C(=O)NCCCNC(=O)C(C)(C)C2CCOC2)nn1 c1(C(N2CC3(CC(NC(C4(F)C5CCCCC45)=O)C3)C2)=O)cc2cccnc2s1 C1(NC(c2c(C)onc2)=O)CN(C(c2cc3cccnc3[nH]2)=O)CC2(CCC2)C1 Cc1ccc(C(=O)NCC(C(C)(C)C)NC(=O)C(c2cncn2C)O)nn1 c1(CN(C2(c3ccc(Br)cn3)CC2)CC)ccc(F)c(C)c1Cl C(=O)(CC1C(=O)Nc2ccc(Cl)cc21)N(C)CC1(C)CC1.c1(C=O)ccsc1 Cc1ccc(N)c(C(=O)NCC2CC2)c1.c1(C=O)ccccn1.C(=O)(C)N c1(OC)cnc(C(N2CC3CC3(CNCc3ncc(Cl)s3)C2)=O)c(F)c1 N1(CC)CCCC1C(N1CC(C)(CCC(=O)NCC(C)CN2CCCC2)C1)=O Cc1c(C(=O)NCCC(C)NC(=O)C#CC2(C)CC2)cc(C(F)(F)F)cc1N c1(C=O)ccc(C(C)S(N)(=O)=O)cc1.C1(CC(=O)N(CCC)C)(OC)CCC1 Cc1cc(Br)ccc1CNc1cc(C(=O)NC(c2cc(Cl)ccc2O)C)n(C)c1 C(=O)(C1CCCn2ccnc21)N1CC2(N(C(C(C=C)(C)CC)=O)C2)C1 C1(NC(c2c(C)ccn2C)=O)CCN(C(c2snc(Cl)c2Cl)=O)CC1C N1(C(C2OCCN(CC)C2)=O)CC2CCN(C(=O)CCN(C)C(C)=O)CC2C1 c1(CNC(c2cccc(Cl)c2C(F)F)=O)c(O)nnc2c1CCCC2 C(=O)(C(CC)C(=O)NC(C)C)OCC.c1(CC=O)ccc(C2CCC2)cc1 C1(NC(CCC2(C)CC2)=O)CCN(C(c2ccoc2)=O)CC12CCC2 c1(N2C(C(CCC)C)CCC2)nc(Cl)nc2c1CCNC2 CCC(C)CC(=O)NCCC(O)CNC(C1CN(S(=O)(=O)CC)C1)=O C1(NC(c2cc(O)ncn2)=O)CCCCN(C(=O)COc2ccc(Cl)cn2)C1 c1ccc(C(N2CC3CC2C3)=O)cc1.n1(CC=O)ccnn1.C(=O)(CO)OC Cc1ccc(=O)n(CC(=O)NC2CC(C)(NC(c3c[nH]c(=N)o3)=O)C2)c1 N1(C(CC=C(C)C)=O)CCOCC1CC(=O)N(C1CCCC1(C)O)C C(=O)(CCC(C)(C)OC)N(CCNC(C(C)OCC#C)=O)CC N#CC1CC(F)(F)CN1C(c1sccc1NC(c1cccc(I)c1Cl)=O)=O N1(C(C(C)=C2CC2)=O)CCCC1(C)C(=O)NOCC1CCOC1 C(=O)(CCCC(=O)C1CC1)N1CCC(CCNC(C(C)N2CCC2)=O)CC1 CCC(C)(CNC(C1(Cl)CC1(F)F)=O)NC(C1CC(n2ccnn2)C1)=O C1(NC(C2CC2(F)F)=O)CCCC1NC(c1nncs1)=O N1(C(C2C(CC)CCC2)=O)CCCCC1C.c1(C(=O)N)cc(C(F)(F)F)ns1 Cc1cc(C(=O)NC2(CO)CCN(C(c3cccc(SCC#N)c3)=O)C2)cnn1 N1(C(C2(COCC)CCC2)=O)CCC(C(C)C(=O)N(C)C)CC1.C1CCC1 c1(C(=O)NC2(COC)CCN(C(c3oc(CC)c(C)c3)=O)C2)cc(C)ccc1Cl N1(C(C(C)CCO)=O)CCN(C(c2cc(CC3CCC3)c[nH]2)=O)CC1C N1(C(COCC=C)=O)CCCC1C(=O)NC(C1CCCN1C(C)=O)=O.O Cc1c(C(N2CCC(O)(CN(C(=O)C(C)C#N)C)CC2)=O)sc2ccccc12 C#CC(CC(C)(C)C)NC(=O)C1=CCC(NC(=O)CCC(C)OC)C1 c1(C(C)=O)cn(CC(N2CCC(C3CC3)C2CCNCC(=O)O)=O)c2ccccc12 C1(CCNC(C(CC=C)OC)=O)CN(C(c2ccnc(OC)c2F)=O)CC(C)O1 C1(CNC(c2cc(C)sc2C)=O)CC2CCC1N(C(C1CCC(C3CC3)C1)=O)C2 c1(COC)cc[nH]c1C(=O)NCC1COC(CNC(=O)C=CBr)C1 C1(CCNC(CC2CC(CC)C2)=O)CCCN(C(c2cc(CCO)on2)=O)C1 C1(NC(CSCC#C)=O)CC12CC(NC(=O)C(CCC)OCC)C2 C(C)(CCC(=O)N(C)OC)(c1n(CCOCC)nnn1)NCCS(C)=O n1(CC)ncc(Cl)c1C=O.N12CCN(CC1)Cc1ccc(cc1)C2=O.C(C)C.N CC1(C)CC(CNC(c2cnc(O)c(Cl)c2)=O)N(C(c2cnnc(O)c2)=O)C1 c1(C(N2CCCN(C(CC(C)n3cccc3)=O)CC2)=O)cncc2sccc12 N1(C(CC(COC)(C)O)=O)CCC(NC(=O)C(F)CCC(C)(C)C)C2(CCC2)C1 c1(C(N2CC(NC(C3C(C)C3(F)F)=O)C(CO)CC2)=O)cnc2c(cnn2C)c1 C1(F)(C(N2CCCC(CCNC(CC(CCC)C)=O)C2)=O)CCC(F)(F)CC1 N1(C(C(C)=CC)=O)CC(NC(c2ccc(C)cc2)=O)CC1(C)CC c1(C(C(=O)NC(c2ccccc2)C#C)NC(c2ncc[nH]2)=O)cccnc1 S(=O)(=O)(c1cnn2ccc(=NCCCCOCCO)[nH]c12)N1CCCC(C)CC1 C(CCN(C)C(C1CC1c1ccnn1C)=O)C(C)C.C(=O)(CC=O)OCC.N N1(C(CC2C(=O)NCC2)=O)CCC2(NC(C3CCCS3)=O)CCCC12 c1(C(N2CCC(N(C(=O)CN3CCC(OCC(N)=O)C3)C)C2)=O)cccnc1Cl Cc1ccc(C(=O)NC2CCN(C(=O)C#CC3CCC3)C(C)C2)c(F)c1F c1(C(=O)OCC)cccc(OCC(N2CC(C)C2)=O)c1.c1cccc(O)c1.C O=C(CCCC(F)(F)CO)NC1(CNC(c2cccc(C3CC3)c2)=O)CCOC1 c1(NC(=O)NC(C)C=O)ccc(F)cc1.C1(C)(CC=O)CCCC1.CCC.N c1(OCC(=O)Nc2coc(C=C3CCCC(C(F)(F)F)C3)c2)cnc(Cl)cn1 N1(C(C2CCC(NC(C)=O)CC2)=O)CCC(N=c2[nH]c3cc(Cl)cc(Cl)c3o2)C1 C=CCCCCCC(=O)NCC(C1CCC1)NC(=O)CC1CCCC1.C(C)=O.N N1(C(CC(C)O)=O)CCN(C2CCCN(C(C3(N(C)C)CC3)=O)C2)CC1 C1(CNC(C(C)N(C2CN(C(C3CC3C(C)(C)C)=O)C2)C)=O)CCCCC1 CCC(CC)(CC)C(=O)N1CCCC(C)(NC(=O)C2=CSCCO2)C1 C1(NC(C(C)N(C)C)=O)CC1C1CCN(C(C2CC3C=CC2C32CC2)=O)CC1 CCCCC(C)C(=O)N1CCN(C(=O)C(C)NC(=O)CSC(C)(C)C)CC1 N1(C(C(CC)C(C)C)=O)CCC(C(F)(F)F)C(N=c2ccc([N+](=O)[O-])c(O)[nH]2)C1 c1(C(=O)NC(CC(C)C)CNC(C2(C)CCC3CC3C2)=O)ccc2c(c1)COC2 C1(CNC(C(C=C)O)=O)(COC)CCN(C(=O)CNC(=O)O)C1.C C1(CNC(COC(CNC(CC=CCCCCC)=O)(C)C)=O)CCOCC1C C=CCC(CNC(=O)C(C)(F)F)C(=O)NCC1CC(=O)N(C)C1 CCCS(=O)(=O)CC(=O)NC1CCN(C(=O)CCc2ccc(C#N)cc2)CC1C c1(C(c2n(CCSC)nnn2)NCC2(CCO)CCCC2)c(C)nsc1C N1(C(c2c(C)nsc2N)=O)CCOC2(CCN(C(=O)C(C)CC3CC3)C2)C1 C(=O)(C(CCC)CCC)N.C=C(C)C1OCCC1C(=O)NCC1CC(O)(C)C1 c1(NC(C)=O)c(C(=O)NCCCN(c2cc(Cl)ncn2)C)cccc1C C1(C(=O)OC)CCC(C(N2CCCC2C(=O)NCCCCC)=O)C1.C(C)=O.N c1(C(=O)NCC(C)(C)OCC)ncccc1N.C1(CCC=O)CCCC(O)C1.N c1(C(N2C(C3CCN(c4nnc(C)s4)CC3)CCC2)=O)cccc2cccnc12 n1(C2CCCN(C(C=CC)=O)C2)cnc2c1CCN(C(=O)C(C)(C)C(C)(C)C)C2 C12CCC(CC1)NC2=O.CCC(O)C(=O)N1CC(n2ccnn2)C1.C(=O)(N)O c1(NC(c2cn(CCN3CCNC3=O)nn2)C)cc([N+](=O)[O-])n(C)n1 C1(C(=O)NC(Cc2n(C)ncc2)C(=O)O)COC(C)(C)CO1 N1(C(C=C2CCC(C)C2)=O)CCOC2CCN(C(=O)CCC3CC3)CC12 C(CN=C(NCCOC1CCSCC1)NC1CC1)c1cc(Cl)ncc1 C(=O)(C1=CCC(C)CC1)NC1CC2(CC(NC(c3cc(C)cc(Cl)c3)=O)C2)C1 N1(C(CCCCC(=O)NC)=O)CC(C)CN(C(c2cc(COC)no2)=O)C(C)C1 C1(N(C(=O)CCn2cccc2)C)CCC(NC(C2C=CCC2)=O)CC1 C1(NC(c2c(CC)nco2)=O)CCCC(CN(C(=O)C2=COCC2)C)C1 c1(OCC)ccc(CNC2CCC(C(F)C(=O)O)CC2)cc1O Cc1cncc(C(N2CC(N3CCN(C(=O)CC4COCC(C)O4)CC3)C2)=O)c1 N1(C(c2nc(C(C)(C)C)sc2)=O)CCC(NC(c2cncc(Cl)c2Cl)=O)C12CC2 N1(C(c2cc(F)cc(C)c2O)=O)CCN(C(c2cc[nH]n2)=O)CC2(CC2)C1 C1(NC(Cc2c(CC)noc2CC)=O)CC(F)CN(C(=O)C2=CCCCO2)C1 C(=O)(C(F)(F)C(F)F)NCCN(CCC)C(c1cc(C(=O)OC)sn1)=O c1(CC)cccc(C=O)c1.C(=O)(C(C)(C)CF)N(CC)CC.C(CO)O N1(C2CC(C(=O)NC(C)CNC(=O)CC(C)O)C2)CCN(C)CC1 C(C)(C(=O)N(CCC(=O)NC(c1nccs1)C)CCO)OCC(C)C CC#CCC(C(=O)NCc1cc(C)sc1C)NC(C1COCC(C)O1)=O c1(CN=C(NC(C)C)NC2CC(=O)N(CC(F)(F)F)C2)cnc2n1CCCC2 Cc1cn2cc(C(=O)NCC3(CO)CCN(C(C4CCNC4=O)=O)CC3)nc2s1 c1(C(N2CC(O)CCC2)=O)cccc2nc(O)oc12.NS(=O)(=O)C1(C(=O)N)CC1 Cc1c(F)ccc(NC(=O)C2=CCC(NC(=O)CCc3cn(C)nn3)C2)c1F C=CC1CN(C(C2CC2C=C)=O)CC1NC(=O)CC=CC(C)(C)C C(C(CC1CC1)C(=O)NCC(C)C(C)O)NC(C(C)C)=O CCC(C)(C(=O)NCCC1(C)CCN(C(=O)CCC#N)C1)OC C(CCCCCNC(=O)CCCC1CCCC1)N(C(C1C(C)CCO1)=O)C c1(OCCC)ccc(Cl)cc1CC(=O)NCCNC(=O)CCCn1cccn1 c1ccc(Cl)cc1.C1(C(=O)NC(C)CO)(COC)CN(C(=O)C(C)NC)C1 c1(C(N2CC3C(NC(c4cc(C)ncc4)=O)(C3)C2)=O)n[nH]c2c1CC1CC21 O=C1NCC(C(=O)NC(C(=O)NCCN2CCC3CC23)C2CC2)N1 c1(N(C)CC2CCCN2C(=O)CC2C=CCC2)ncn(C)c(=O)c1Br N1(Cc2cccc(C)c2C)C2CCC1CC(NC(=O)NC(C1CC1C1CC1)=O)C2 C(=O)(C1=C(C)OCCC1)NCC1CCC(NC(C(CSC)(C)C)=O)C1 c1(CNC(c2c(SC)cccc2)=O)ccc(B2OC(C)(C)C(C)(C)O2)cc1 c1(CNC(c2cc(CC)[nH]n2)=O)ncccc1C.C1(C=O)CNC(=O)C1.N c1(C(C)SCCC=C=CC)ccc(Cl)c(Cl)c1 CC(C)CC(O)C(=O)NC(c1ccccc1F)CNC(=O)C=Cc1cc[nH]n1 c1(C(=O)NC2CCN(C(C(C)NC(C)=O)=O)CC2C)cnc2ncccn12 C#Cc1ccc(C(N2CCC(O)CC2C)C(=O)NCCCN(CC)CC)cn1 C1(C(=O)NC(CC)C(C)(F)F)C(C)OCCN1C(c1occc1C)=O C12(NC(C(COCC)C)=O)CCC(C(=O)Nc3cnccc3C)(CC1)C2 C(=O)(CC(C)(C)C(F)F)NC1CC(CNC(c2scc(OC)c2)=O)C(O)C1 CCCC(CC)CC(=O)N(C1C2CN(C(c3cnoc3C)=O)CC12)C n1(CC(=O)NC(C(C)NC(=O)C(=O)NCCC(N)=O)C)nc(O)ccc1=O Nc1nc2c(cc1C(=O)NCC1(F)CCC1)CCC2.C(=O)(C)N.C(N)=O N1(C(c2cc(C)n(C(C)(C)C)n2)=O)CCC2(CC1)CC2NC(=O)C(C)CF CN1CCOC(C(N2CC3CC(NC(c4cncc(CO)c4)=O)C2C3)=O)C1=O CN1CCCCC1CC(N1CCC1CNC(=O)Cc1n[nH]c(=N)s1)=O C(=O)(C(C)(C)CC(C)(C)C)N1CCC(F)(CNC(C2CC(C)OCC2)=O)CC1 C12(CNC(c3ccc(I)cc3F)=O)CCCCC1C2(F)F C=CC1OCCCC1C(=O)N(C)CCOCCCNC(c1cncc(SC)c1)=O CC1CCC(Cl)=C(C(=O)NCC2CC(O)CN2C(c2ccc3cncn3c2)=O)C1 N(C1CCCc2ccccc21)C(N1CCOCC(CO)C1)=O c1(NC(C2N(C(C3CCCN(C)C3)=O)CC=C2)=O)ncnc2c1c(Br)cn2C C(=O)(C(C)C(C)c1ccc(F)cc1)N1CCCC1.c1(CC)[nH]ccc1C(=O)NC C(=O)(C1=C(C)OCCS1(=O)=O)NC(C1CC1)C.C1(C=O)CC2C=CC1C2.C N1(C(Cc2c(C)ocn2)=O)CC2CCCC2(NC(c2nc3sccn3c2C)=O)C1 C=CCC(CC=C)n1cc(C2CN(C(=O)C(O)Cc3ccccc3)C2)nn1 c1(C(N(CC(C)C)C(C)(C)C)=O)ccc2[nH]nc(Cl)c2c1 CC1CCN(C(=O)CCC2CC2C)C(C(=O)N(C)CC2(C)CCCO2)C1 C1(C2CCN(C(=O)CSC3CCCCO3)CC2)(NC(=O)CC2OCCO2)CC1 c1(CC=O)ccc(O)nn1.Cn1cc(CCC(=O)NCc2csc(C)c2)nn1.N c1(C(=O)NCCC2(O)CN(C(C=COCC)=O)C2)ccc(NC2CCC2)cc1 C#Cc1cccc(CCC(=O)NCC(C)N(C(=O)COC2CC2)C)c1 Cc1cccc(C(N2CC(O)(CNC(C3(O)CCCCC3)=O)C2)=O)c1 Cc1csc(C(C(=O)NC2CCOC2)N(C)Cc2cncnc2)n1 c1(C(N2CC(C)(NC(CC3C(CC)C3)=O)C2)=O)cc2scnc2[nH]1 N1(C(C(C)(C)OC)=O)CCCC(CC(=O)Nc2csc(C)c2)CC1 CC1=CCSC1C(=O)NC(C(=O)NCC1CCSCC1)C1CCC1 CC(C(C)C(=O)NC1CCC2(CC2)C1)NC(=O)CC1CCOC1(C)C CC1(C)CCCCC1CNC(=O)CCOCCNC(c1ncccc1O)=O N1(C(CNC=O)=O)CCCC(NC(c2cnn(CCC(F)(F)F)c2)=O)C(F)C1 C1(CN(C(=O)NCCc2c(C)ocn2)C)CCCN(C)C1C1CC1 C1(C(N2CC(CCOC3CC(F)(F)C3)OCC2)=O)(SCC=C)CCOCC1 C1(CCN(C(c2cnc(C(C)OC)s2)=O)C)CCCCN1C(=O)CC(C)(F)F c1(OC)cc(OC)c(N)c(C(=O)NC2CCCCC2)c1.C(=O)(C)N.CC(C)C c1(C(=O)NC2C(CNC(c3ccc(N)c(F)c3)=O)CC2)c[nH]c2nccc-2c1 C(CC(C)C(=O)NCC1C2CN(C(c3cc(CC)no3)=O)CC12)=CCC CC1(C)CC(C(N2CCSCC2)C(=O)NCCCC2CC2)CC(C)(C)C1 N1(CCCCOC)CCC(CF)(NC(=O)Cc2cncn2C)C1 N1(C(C)=O)CSCC1C(N1CC(CCCCNC(c2cnn[nH]2)=O)C1)=O C(=O)(C(CCC)c1cccc(Cl)c1)N(CCN(C(C1(C=C)CC1)=O)C)C N1(C(C=Cc2nc(C)sc2)=O)CCCN(C(c2ccncn2)=O)C(C)C1 C=C(C)C(C)(C)C(=O)NC(CCN(C)C(c1ncnc(O)c1F)=O)C(C)(C)C N1(C(C(c2ccn(C)c2)C)=O)CCCCC(NC(c2cc(CO)[nH]n2)=O)C1 C1(C(=O)NCCSCC)CC12CCN(C(=O)C(=O)NCC(C)O)C2 C1(O)(C(C)NC(C2(C#N)CC2(C)C)=O)CCN(C(=O)COCCCF)CC1 N1(C(c2ccc3c(n2)CCO3)=O)CCC2CCN(C(C3CSCCS3)=O)C2C1 c1(C(=O)NC(CCNC(C(COC)C)=O)C)coc2c1C(=O)CCC2 N1(C(CCCSC)=O)CC23CCCCC2(C1)CN(C(=O)CC1(OC)CC1)C3 Cc1cnc2n1CCCC2C(=O)NC1CN(C(=O)CNc2nccs2)CC1F Cc1nccnc1C(N1CC(C)(C)C1C1CCN(C(=O)CSC2CC2)CC1)=O S(=O)(=O)(c1ccc2nc(O)oc2c1)N1CC(C)C(NC(=O)CN2CCCCC2)C1 N1(C(C(C)=CC(C)(C)C)=O)CCCC(C(N2CC=CC2CN(C)C)=O)C1 CS(=O)(=O)C1(C(=O)NC(C2CCCCC2)CNC(c2cnc[nH]2)=O)CCC1 c1(N(CC(=O)N(C(=O)C(C2CCCCC2)O)C)C2CC2)nnnn1C c1(NCc2cc(C)nn2C)ccc(NC(c2cnnc(Cl)c2)=O)cc1F N1(C(C2CC(OC)C2)=O)CCC2(CC1)CC2NC(=O)CCC1CCCC1 C(=O)(C(CC)C(C)C)NC(CC(=O)NC)C1CC1.C12(C=O)CSCC1C2.N N1(C(C(c2cccnc2)NC(c2ncn3c2CCC3)=O)=O)CCn2nccc2C1 C1(C#N)(OC)CC(C(N2CC=CC(NC(c3cccnc3C)=O)C2)=O)C1 CC(C)(C)CC(O)CC(=O)NCC(C)(C)CNC(C1(Cl)CC1(F)F)=O c1(C(=O)NC2C(CNC(C(C=C)(F)F)=O)CCCC2)ccc2nonc2c1 C(=O)(C(O)CCC)N1CC(OCC(=O)NCCOCC#C)C1 c1(C(=O)NCCCN(C(C(C)c2ccsc2)=O)C2CC2)cccn2ccnc12 C(C(C)(O)C(C)CC)NC(C(CC#C)NC(=O)CCOC1CCC1)=O c1(CN(C(=O)NC(c2nc(O)n[nH]2)C)CC2CCCO2)ccccc1F C1(NC(=O)Cc2ccc(CO)cc2)CCCCC1CNC(c1ccc(Cl)nc1)=O N1(C(C2CCCC2O)=O)CCc2ccc(C(N3CC(CO)CC3CO)=O)nc2C1 C1(C(N2CC3(OCC(NC(c4ccco4)=O)C3)C2)=O)COc2cc(Cl)ccc2C1 N1(C(C2CCN(S(C)(=O)=O)C2)=O)CCOC(CCNC(c2ncccc2Cl)=O)C1 Cn1[nH]cnc1=NC(=O)C1CCN(C(=O)Cc2ccc(F)cc2Br)CC1O C1(CNC(C(CC=C)C)=O)N(C(=O)COc2ccsc2Cl)CCCC1(C)C C(=O)(C(C)CCCC(C)C)N1CC(C(=O)Nc2c(C)cc(F)cc2)CC12CCC2 C1(C2CC2)(C=O)CCC1.c1(C(=O)NC2CCC2C)sccc1OC(F)F.N Cc1cc(C)c(C(=O)NC(C)C(C)C(=O)NCCC(F)=C(F)F)cn1 CC(C)CC(C(=O)NC1CCOC1=O)NC(C1COCC1(C)C)=O N1(C(C(c2ccn(C)n2)C)=O)CCCCC(NC(=O)C(O)CN(C)C)C1 Cc1ccc(C=CCC(=O)NC2CCCC2NC(c2nc(Cl)ccc2N)=O)cc1 O=C1CCC(C(=O)NCC2CSCCS2)CCN1 c1(C(=O)NCC(CC(F)(F)F)NC(=O)Cc2cocn2)cn2ccc(F)cc2n1 N1(C(C2C(CNC(C(CC(=C)C)OC)=O)OCC2)=O)CCCNC(=O)CC1 C(=O)(CS(=O)(=O)CC(=O)O)N1CCC(Cn2cc(C(CC)(C)C)nn2)C1 C#CCC(C)(C)C(=O)N1CC(CC(C)NC(=O)COC)C1.c1ccc(C)cc1 Cc1sc(O)nc1C(=O)NCCC1(O)CN(C(C2C(Cl)(Cl)C23CC3)=O)C1 c1(CNC(NCC(N(OCC(=O)OC)C)=O)=NC)c(F)cc(I)cc1F c1(NC(C2C3(CN(C(c4ccc(SCC)cc4)=O)C3)C2)=O)ncc(F)cc1F c1(C2CC=CC2)nc(CN(C)C(=O)OC(C)(C)C)[nH]n1.C1(C)CCCC1.C C1(CCNC(C(C)c2ccsc2)=O)CN(C(=O)C=Cc2cc[nH]n2)CCO1 C1(C(=O)NC(CCCC)(C)C)CC2CCC1N2C(=O)C(CC)N(CC)CC C1(NC(c2n[nH]c(=N)[nH]2)=O)(CO)CCN(C(=O)Cc2ccc(O)nc2)CC1 N1(C(CNC(CNC(C)=O)=O)=O)CCCC2C1CCN2C(C1C2CCCCC12)=O C1(NC(CC=CCC)=O)CCN(C(c2cc(CO)oc2C)=O)CC1CC c1(N2CCC(CNC(c3c(CC)nc(C)[nH]3)=O)C2)snc(Cl)c1C#N N1(C(c2c(CC)ccs2)=O)C2CCC(C2)C1CC(N1CCCC(O)CC1)=O C(=O)(C1c2ccccc2CN1C(c1ccc2ccoc2c1)=O)Nc1occ(C)n1 c1(N(C2CCC2)C)ccc(CNc2cc(Br)ncn2)cc1 c1(C(C(=O)NCCc2ccns2)NC(C(C2CCC2)OC)=O)ccnn1C c1(CC)ncc(C(N2CC(NC(=O)CCc3cc[nH]n3)CCC2C)=O)c(O)n1 N1(C(C=CC=CC)=O)CC(CNC(=O)CS(C)(=O)=O)C(F)(F)C1 c1(OC)ccc(CO)cc1COCCN(C)CCc1ccccc1 C1(C)(C(NCC)=O)CN(C(=O)Cc2cncn2C)C(C)(C)C1.c1ccsc1.C C1(NC(C(C)=O)=O)CC(F)CN(C(=O)Cc2c(F)cccc2Cl)C1 c1(C(N2CC(COC)N(C(c3ns[nH]c3=O)=O)CC2)=O)ccc(F)cc1[N+](=O)[O-] c1(C(N2CC3CN(Cc4cc(Br)ccc4F)C3C2)=O)ccc2c(c1)CCCO2 N1(C(C2(CNC(=O)C(=O)N(C)C)CC(=C)C2)=O)CC2CC(C)C2C1 N1(CCCN2CCNCC2)C(=O)c2ccc(Cl)cc2S1(=O)=O c1(NC(CCNC)(C)C)nc(N2CC(CO)CC(C)C2)nc2scnc12 C1(O)(C(N2CC(NC(c3c(OCC)cncc3)=O)C2)=O)CCc2ccccc2C1 N1(C(COCCN(C)C)=O)CCCCC(C(=O)Nc2ccc(OCF)cn2)C1 c1(C(N(CC(CNC(Cc2c(C)n[nH]c2)=O)C)C)=O)coc2c(C)cccc12 C1(C(=O)Nc2c(C(C)=O)ccnc2)CCN(C(c2ccc(I)c(Cl)c2)=O)CC1O N1(C(c2[nH]cc(C#N)c2)=O)CCC(NC(C2(C3CC3)CCCO2)=O)C(F)C1 C12CCC(CC1)CO2.C(=O)CC(C)(O)C(F)F.C(C)(C(=O)NC)NC(C)=O N1(C(COCCCC#C)=O)CCC2(CCCN2C(=O)C)C1.C(=O)(C(C)(C)C)N c1(C2CCCN(C(C(CCSC)OC)=O)C2)ccc(C(F)(F)F)c(Cl)c1 C1(CNC(C(C)(C)CO)=O)CN(C(=O)C(F)=C2CCC2)CCC12CCC2 N1(C(CCCNC(=O)NCC#C)=O)CCCC(O)C1.c1(C=O)c(C)n[nH]c1C.N c1(CC)ccc(O)c(NC(=O)CC(O)C)c1.C1(CC=O)C(C)(C)C1(C)C.N n1(CC)cccc(NC(=O)C(C)CN(C(=O)COC2CCOC2)C)c1=O C1(C(N(C2CN(C(=O)C(O)CC(N)=O)CC23CC3)C)=O)CC2CSCC(C1)C2 C(c1ccc(O)cc1)=CC(N1CC=CC(NC(C(C)SC(C)C)=O)C1)=O NC(=O)CCC(=O)NC1CN(C(C2CC3CC3C2)=O)CC1n1cccn1 c1(C(=O)NC2CN(C(COCCCC(C)C)=O)CC(O)C2)cccc2c1OCO2 CCC(CC(=O)N1CCC(CCNC(C2(C(O)C(F)(F)F)CCC2)=O)CC1)OC c1(C(CC)C(=O)NCCNC(C2(c3ccno3)CCC2)=O)ccc(Cl)cc1 Cc1ccc(CC(=O)Nc2nc(-c3cnc(N(C)C)nc3)cs2)cc1F c1(C(=O)NC2CC3(CC(NC(CN(C)CC)=O)C3)C2)ccc2ncn(C)c2n1 CC(CCC(=O)NC(C)(C)CCN(C)C(C1CC(=O)N(C)C1)=O)N(C)C C(=O)(C(C)(C)NC(c1sccc1)=O)OCC.C(C1CCOC1)=CC=O.C c1(C(=O)NC2CN(C(CNC(N)=O)=O)CC2(F)F)cccc([N+](=O)[O-])c1Cl CC(C)C(C(=O)NC(C)(CNC(C1(F)CCC1)=O)CO)n1cnnn1 C(=O)(C1=CC2CCCCC12)NC1C(CNC(c2n(C)nnc2)=O)CC1 C1(C(C)NC(c2[nH]cc(COC)c2)=O)CCCN(C(=O)C(C)(F)F)C1 n1(CCCOC)c(N(C2CCCC2C#N)C)nnc1-c1cnc(-c2ccccc2)[nH]1 Cc1ccc2ncc(C(=O)NC3CCCC(NC(=O)CCc4ccon4)C3)n2c1 N1(C(C(CC=CC)NC(=O)C(C)CC#N)=O)CCC12CCCOCC2 C1(NC(C=CCCC)=O)CCC(C)(C)CC1.C12(C=O)CCC(CC1)C2(C)C.C c1(C(=O)NC(C2CCN(C(C=NOC)=O)CC2)C(C)C)cc(C)nc2ncnn12 C(=O)(N=c1cc(SC)n(C)[nH]1)C1(OC)CCN(C(=O)CCC(C)=O)C1 C1(C2CC2)(CNC(c2cc(C)c(C)nn2)=O)CCN(C(=O)C(F)=CC2CC2)C1 C12(C(N3CCC(Oc4ccc(Cl)cc4Cl)CC3)=O)CC3CC(CC(C3)O1)C2 CC(CCc1ccccc1F)C(=O)NCC1CCC1.c1(C(=O)N)cc(F)n(C)n1 C1(C(=O)NC2CC(CC)C2)CCCN1C(=O)C1CC1.c1(C=O)ccco1.N CCS(=O)(=O)c1cc(CNC(C2CCCC3(C2)N=N3)=O)cc(Cl)c1 N1(C(C(C2CCCO2)NC(c2n(C=C)nnc2)=O)=O)CCC12CN(C)C2 c1(C(=O)NC2C(NC(=O)CCN3CCCCC3)COC2)cn2ccsc2n1 c1(Cn2cc(CONC(c3cncc(C=C)c3)=O)nn2)ncn2c1CCCC2 n1(C(C)C)ncc(C(=O)NC(C)CCCNC(C2(O)CCC2)=O)c1N C1(NC(COC2(C)CN(C(C(C(C)O)N(C)C)=O)C2)=O)CCCCC1(C)C CCCC(C)CCCC(=O)N1CCCN(C(=O)COCCSC)CC1 CC1(C)CN(C(C2CCc3n[nH]cc3C2)=O)C(CNC(=O)CC2CCCC2)CO1 C(=O)(C1=CCN(C(=O)CN2C(=O)CCCC2=O)CC1)N1C(C)C(O)CC1 C1(C(=O)NC2CCCC(CNC(C3CC3F)=O)C2)CN2CCN1CC2 CCCC(CNC(=O)C(C)OCCOCC)C(=O)NC(CO)C(C)(C)C C(=O)(CCCCC(C)=O)N1CCC(=C)CC1C(=O)NC1CCNC(=O)CC1 C1(NC(Cc2ccc(C)cc2)=O)CCC(C)N(C(C2C=CC=CC=C2)=O)C1 C=CC(CC)CC(=O)N(CCC(C(C)C)NC(c1ccc(=O)n(C)n1)=O)C c1(CNC(c2cc(CC)on2)=O)nn(C)c2c1CN(C(C1CCCCC1)=O)CC2 CCCCC(CNC(c1ncccc1SC)=O)NC(=O)CC1CC(OC)C1 C1(CC(=O)NC(CO)C(=O)N2CC(OCCF)C2)CC2CC2C1 c1(NC(N(CCCCCC)CCO)=O)ccc(OC(C)C)c(C#N)c1 Cc1nc(C)n(O)c1C(N1CCC(C)(C)CC1)=O.c1(C=O)cc(O)cc(Cl)c1.N C1(C(C)NC(=O)CCN(CC(C)C(C)C)C)CCCCN1C(C1CCOCC1)=O c1(C(=O)N)ccc2nc(=N)[nH]n2c1.c1(OC)cc(C(=O)NCC)c(C)c(Br)c1 C(CCC(C(=O)NCCC(F)(F)Cl)NC(=O)C(C)CCCOC)OC C1(C)(C=O)CN(C(C2CCC3(CCC3)C2)=O)C(C)(C)C1.[SH](=O)(=O)CC.CN Cn1nc([N+](=O)[O-])cc1C(N1CCCC(C2CCC(=O)N2)C1)=O c1(C(N2CC(C)C(NC(c3cc(F)n[nH]3)=O)C2)=O)ccc(N)c(Cl)n1 N1(C(c2ccccc2)=O)CCN(C(C2(F)CCCCC2)=O)CC(O)C1 N1(C(C2(CC=C)CCCCC2)=O)CCCCC(N(C(=O)Cc2nnc(C)o2)C)C1 c1(NC(=O)NCC2CC(=O)N(c3ccccc3Br)C2)cccc(I)c1F C(=O)(N1CC(O)CCO1)C1N(C(c2c(CC)cns2)=O)CCOCC1 CC1(CNC(=O)CCc2cscn2)CCCN(C(=O)CCCc2cccs2)C1 c1(OC)ccc(C)c(CNC2CCC2NC(=O)C(=O)O)c1Br.c1ccccc1 c1(CN(c2c(C)cccc2)C(C2CC2C2CCCC2)=O)c(Cl)c(C)nn1C C(=O)(CC(C)C(C)(C)C)N1CCC(CC=C)(C(=O)NCc2noc(C)n2)C1 c1(NC(=O)CN(C(=O)CC2CC=CC2)C2CC2)ccc2ncccc2c1 C(=O)(C(C#N)(CC)CC)NCCN(C(c1ncn(CC)c1)=O)C(C)C N1(C(CC2CN(C(=O)Nc3c(OCC)cncc3)C2)=O)CCN2CCCC2C1 N1(C(c2cc(C)sc2)=O)CC2(CC2)CC1C(=O)NCc1nc(C)c(C)[nH]1 c1(COC(C(=CC2CCCC2)C)=O)cc(C(=O)O)n(C)n1.C1CCCC(C)C1 c1(CCC(=O)NCCC2CCCC2)nc(-c2ccsc2)no1.C1(O)(C=O)CC1.N C1(SC)CN(C(c2ccc(C(F)F)cc2)=O)CC1NC(=O)CC(C)CF C(C(N=[N+]=[N-])C(=O)N1CC(C)(NC(c2cc(CO)ccc2O)=O)C1)OCC C12(C(N(C3CCN(C(C4CC4)=O)C3)CC)=O)CCCCC1OCC2.C(C)C.C C1(NC(=O)CSCc2ccncc2)CC2CC1CN(C(=O)C=O)C2.C1CC1.N CCCCS(=O)(=O)NC(C)C(=O)NC1CC(F)C1.c1(C=O)cc(C)sn1.C C1(C(N2CC(NC(CCc3ccc(C)s3)=O)C2)=O)CC(=O)N(c2nccs2)C1 c1(C(=O)NC2CN(C(C3CCNC3=O)=O)CC3(CC3)C2)cc(=O)n2nccc2[nH]1 C1(OCC)CN(C(C2(CO)CCC2)=O)CC1CNC(c1ccco1)=O C1(C(N2CCN(CCN(C(C(CC(C)C)O)=O)C)CC2)=O)CCC2(CCC2)OC1 C1(C(N(C(C)C(=O)NCC2CCC(O)CC2)CCC)=O)CCCC(C)C1 CCC(CC)C(F)C(=O)N1CCCC1C(N1CC(C)=CC(C)C1)=O N1(C(C(C)Cc2cnn(C)c2)=O)CCC(N(C(=O)COCC2CC2)C)CC1 c1(CC)nccnc1C(=O)NCC1(C)CC1C(=O)OC(C)(C)C c1(OC)ccc2c(n1)NC(C(=O)NCCC(O)C1CCC1)C2 c1(OCC)ccc(CNc2ccc(Cl)c(C(N)=O)c2)cc1[N+](=O)[O-] C(=O)(CC(C(=O)OCC)C(C)=O)N(CC(=O)O)Cc1cn(CCCC)nn1 C1(C(N(C2CC(OC)C2)C)=O)CCC(CNC(=O)CC2CC(OC)C2)C1 n1(CC)cnc2c(NC3CC3C(C)C)[nH]c(=NCc3cc(C)cnc3OC)nc12 c1(C(=O)OC)ccc(OC)cc1S(=O)(=O)NCC(C(F)F)N1CCNCC1 N1(C(c2cnc(C(C)O)s2)=O)CCCC12CCN(C(c1cnccc1Cl)=O)C2 Cc1nn(C)c(NC(C2CC(O)CN2C(C2(C#N)CC2)=O)=O)c1Cl c1(C(=O)NC(C(=O)OC)Cc2ccc(Br)cc2)c[nH]c2ccc(F)nc12 S(=O)(=O)(c1c(C)n[nH]c1C)N1C(C(=O)Nc2ccc(OC)cc2C)CC(O)C1 N1(C(C2(CCOC)CCCC2)=O)CCC(C2CCN(C(=O)C(C)CF)C2)CC1 C1(C(=O)NCCC=C=C)CC(OC)CN1C(c1cnc(OC)s1)=O CC(=O)CCCC(=O)NC(CNC(C1CCCCS1)=O)C1CC1 c1(C(=O)NC2(C)CCN(C(CCC)=O)C2)ccc(Cl)c(CCC)c1 CCCCC(O)CC(=O)NC(CC1CC1)C(=O)N(C12CC(C1)C2)C c1(N2CC(CS(C)(=O)=O)OCC2)cccc(S(=O)(=O)N2CC(F)C(F)C2)n1 C(=O)(CC(CC)CC)N1CC(CCNC(C2(C=C)CC2)=O)OCC1 CC1CC(C)N(C(c2cccc(F)c2F)=O)CCN1C(=O)COC1CCCC1 Cc1cccc(C(=O)NC2CCC2CNC(=O)CCc2scnc2C)c1N Cc1cn2c(n1)CC(C(=O)NC1CCN(C(=O)C(C)(C)CC#N)CC1C)CC2 N1(C(c2ccn(C3CC3)c2)C(=O)NCCSC)CCCCCC1c1cccnc1 c1(C(=O)NCCCN(C(C2CCC3(CC3)C2)=O)CC)c(C)[nH]c2ncccc12 c1(CC(C)C)cc(C(N2CCC(F)C(NC(=O)C3=CCOCC3)C2)=O)ccc1N C(=O)(C1=Cc2ccccc2C1)N1CC(C)C(NC(c2ccc(=O)n(C)c2)=O)C1 C(CCO)(CC(C)C)NC(C(CC)N(C(=O)CN1CC2CCC1C2)C)=O c1(OC)ccc2[nH]nc(C(=O)NC3CC(F)CN(C(C4CCOC4C)=O)C3)c2c1 CCC(C)(CNC(C1(CC2CC2)CC1)=O)NC(C1CCCSC1)=O N1(C(c2c(OC)cccc2C)=O)CCC2(CC(NC(c3cnc(C)nc3)=O)C2)C1 CC1(NC(C2CNC(=O)C2)=O)CCN(C(=O)C(O)c2ccsc2)CC1 C1(SCC)CCCN(C(C2CC(OC3CC3)C2)=O)C1C=O.C1(F)CCOC1 C=CCCCCC(=O)NC1CC(CNC(c2occc2C(=O)OCC)=O)C1 c1(CC(=O)NCC(C)N(C(c2cncc(OC)c2)=O)C)cc(C)ccc1F CCC(CC)CCC(=O)NC1(C(=O)NCCc2nccs2)CCCC1 Cc1cc(CNC(C2CC2NC(c2cc(-c3ccccc3)no2)=O)=O)on1 CC(C)C(CNC(=O)C=CCCc1ccccc1)NC(C1CC2CC2C1)=O CC1=C(C(=O)NC2CC2)C(c2cc(Br)sn2)NC(=S)N1 c1(CNC(NCCC(C(=O)OCC)CC)=NCCF)ccc(S(N)(=O)=O)cc1C C(=O)(CCS(N)(=O)=O)NCC1(O)CN(C(C2OCCN(C(C)C)C2)=O)C1 Cc1nsc(NC(C2CCOC2C(C)C)=O)c1I c1(C(N(C2CC3CN(C(C(C=C)(C)C)=O)C2C3)C)=O)ccc2cnsc2c1 C(CC(=O)N1CCCC(O)(C(N)=O)C1)(C(C)C)NC(Cc1cc(C)[nH]n1)=O O=S1(=O)CCC2(CN(c3nnc(-c4cccnc4)s3)CCO2)C1 C1(NC(C(C2CCCC2)NC(C2N(C)CCC2)=O)=O)CN2CCCC1C2 C(=O)(C1CC(C)Cc2c[nH]nc21)NCC1(OC)CCCCCCC1 c1(C(=O)NC2(C)CCN(C(C3(O)CCC3)=O)CC2)cccc2cnsc12 Cc1cc(-c2nc(C3CC(O)C3(C)C)no2)c2cnn(C(C)C)c2n1 Cc1noc(C)c1CC(c1nc(-c2cnn(C)c2)nn1-c1ccc(Cl)cc1)C N1(C(C2CCC(C)(C)C2)=O)CCOCC(CNC(c2ccon2)=O)C1 N1(C(C(C)C2CCC2)=O)CCC2(C1)CN(C(c1ccc(O)c(CO)c1)=O)CCO2 C=CC1(CC(=O)N(C(C)CN(C)C(c2nn(C(F)F)cc2Cl)=O)C)CCOCC1 N1(C(COC)=O)CCC(C2(O)CCN(C(c3ccc(C(C)C)cc3)=O)C2)CC1 N1(C(CN(C2CC2)CC)=O)CCC1(C)CC(=O)NC(CO)CCC1CC1 C12(CNC(CCC=C)=O)CC(C1)CCO2.c1(C(C=O)C2CC2)ccc(C)cc1 N1(C(c2n(CCC)ccc2)=O)CC2CCCC2(NC(C2COC2)=O)C1 c1(C(C)C)cc(C(N2CCN(c3ccccc3NC(=O)C(N)=O)CC2)=O)n(C)n1 c1(C(=O)NC(CC)(C)CCO)cc(O)nc2c1CN(C(=O)CN(C)C)CC2 c1(OC)ccc(CN2CCOC(C(=O)NC)C2)cc1C(=O)O.c1cnc(Br)s1 C1(NC(Cc2c(C)cco2)=O)CCCN(C(=O)CC2(C)CCS(=O)(=O)N2)C1.C c1(OC)cc(N(C)C)ccc1C(N1CC(NC(=O)CCC(C)C)C2(CC2)C1)=O N1(C(c2ncc(OC)cn2)=O)CC2CCC1C(NC(=O)C(c1ccc(C)s1)C)C2 C1(CNC(C(CC(C)C)C)=O)CCC2(CO1)CCC2.C1(C)(CC(=O)N)CCC1 CC1(C(N2CC3C(NC(=O)CCCCCn4cnnn4)C3C2)=O)CCCC1(F)F c1(OC(C)C)cccnc1C(=O)NCC1(NC(=O)CC(C)CF)CCOC1 C1(N=[N+]=[N-])(C(=O)NCc2cc(C)ns2)CCN(C(C2OC3CCC2C3)=O)C1 c1(C(N2CCN(C(CSCc3[nH]c(=N)sc3)=O)CC2)=O)ccc2c(c1)COC2 c1(C(=O)NC2C(NC(=O)CC3CC3(Cl)Cl)C2)ccccc1.c1cccc(Cl)c1 N1(CCCC)CCC(NC(c2cc(OC)ccc2C)=O)C(C)(C)C1 C1(NC(Cc2c(C)cccc2)=O)CC2CC1N(C(c1ccoc1C1CC1)=O)C2 c1(CN2CCOCC(NC(CCSC)=O)C2)c(Cl)c[nH]c2nccc1-2 c1(CNC(C(C)N2CCCC2)=O)cnn2c1CN(C(c1cncnc1)=O)CC2 C(N=c1[nH]c2cc(Cl)cc(Cl)c2o1)C=O.CC(C)(C)OC(=O)NCCCN C(CCNC(=O)NCC(O)C1(Cl)CC1)=CCC N1(C(CCC2(NC(c3cc(CC)ncn3)=O)CCC2)=O)CCCC(F)(CO)C1 C1(NC(C(C)=C2CCCC2)=O)C2CC1CN(C(C1CC1n1cc(Cl)cn1)=O)C2 C1(CC=C)(C(=O)NCC2C=CCC2)CCN(C(c2nccs2)=O)C1 C1(C(N(C)CCNC(=O)CCC2CCCO2)=O)CCCCN1Cc1ccncc1 Cc1cc(Cl)ccc1CC(N1CCN(C(c2ccc[nH]2)=O)C(c2ncc[nH]2)C1)=O S(=O)(=O)(c1ccc(NC)cc1Cl)N1CC=CC(OC)C1.c1cc(C(C)(C)C)no1 C1(C(N2C(C)CS(=O)CC2)=O)N(C(c2cccc(O)c2F)=O)CCCC1(C)C n1(CCC(=O)NC2CCC2NC(C2CCNC(=O)C2)=O)cnccc1=O CCC(C)C(C(=O)NCCc1ccccn1)N(C)C(c1c[nH]ccc1=O)=O N1(C(CCCC(=O)OC)=O)CCC(C2(NC(=O)CCC3CCCCO3)CC2)CC1 c1(C(N2C(C(=O)NCCCOC(=N)O)CC(C)C2)=O)ccn2cncc2c1 C1(NC(C(c2n(C)cnc2)O)=O)CN(C(=O)COc2ccsn2)CC1O N1(C(CC2N(C(c3cn(CCC)nn3)=O)CC2)=O)CCCCC12CC2 C1(NC(CCC(C)O)=O)CCC2CCN(C(c3cc(N)cc(F)c3)=O)C1C2 N1(C(c2cncc(C)c2Cl)=O)CC2CC(C)N(C(c3occc3F)=O)C2C1 C1(CC=C)(C(=O)NC2CC2(C)C)CCN(C(=O)COCc2nc[nH]n2)C1 NS(=O)(=O)c1cnn(CC(=O)NCC(O)CCNC(C2CC2(F)F)=O)c1 Nc1c(Cl)ccc(F)c1C(=O)NC.C1CN(C(c2cc(C3CC3)no2)=O)CC1O C1(NC(C(=Cc2ccco2)C)=O)CCC(O)CN(C(=O)Cc2c(C)cnn2C)C1 C1(CC)OCCC1N=c1[nH]c(=NCC2(OC)CCC(F)(F)CC2)c2ccccc2[nH]1 Cc1nscc1CN1CCC(C(=O)N(C)Cc2ccco2)C1 C1(C)(NC(CCOC(C)C)=O)CCN(C(C2CCCC23CC3)=O)C1 c1(OC)ccc(C(=O)NC2C3CN(C(C4(C)CCCS4)=O)CC23)c2ccncc12 c1(C(=O)NCCC2CN(C(CC(C)c3ccco3)=O)CC2C)ccc(Cl)cc1N Cc1ccc(C(=O)NC(C2CCCN(C(=O)CCc3cccn3C)C2)C)cc1Br Cc1ccc2cnc(C(=O)NC(C(C)NC(=O)CC)C(C)C)cc2c1.C(N)=O.N n1(CC(=O)NCc2ccc(CN3CCOCC3)cc2)nc(C(F)F)c2c1CCC2 C#CCCC(=O)NCCCN(C(=O)CCc1nnc(C2CC2)o1)CCO c1(C(=O)NC2CCCC(NC(C3N(C)CC(O)CC3)=O)C2)ccn2cccc2c1 C#CCC(C)(C)C(=O)NCC1CC1CC(=O)NCC(C)(C)CCO C=CC1(C(=O)NCCOCCCC)CCN(C(=O)CN2CCOCC2)CC1 Cc1cc(C)n(CCC(=O)NCC(n2cc(CC(C)O)nn2)C)n1 N(C1CCc2sc(C(=O)O)cc21)C(c1nccc(N(C)C)c1)=O Cc1cc(C(=O)NCc2ocnc2C(=O)NCCC(C)(O)C2CC2)n[nH]1 C(C#CC(F)(F)F)NC(C1C(NC(C2CCC(CC)O2)=O)CCO1)=O C1(C(N2CCC(C(C)NC(C=C(C)Cl)=O)C2)=O)(CF)CC2(CCC2)C1 Cc1ccc2c(N3CCCC(NC(c4cc(Br)c(C)cc4C)=O)C3)ncnc2c1 C(C)(C(CC(=O)N(C1CCCC1(C)O)C)NC(=O)CC1CCOC1C)OC C1(NC(CSCC(C)C)=O)CC2(NC(c3cnc(C4CC4)o3)=O)COC1C2 c1(CC)ccccc1C(CC)NC(=O)COC(C)C.c1ccsn1.C(=O)C C12(C(N3CCC3)=O)CC(C1)C2.c1ccccc1.C(=O)(CCF)N(CC(=O)N)C N1(C(=O)NCC2C(OC)CCC2)CCN(CCOc2ccc(Cl)cc2)CC1 N1(C(C2C(COC)CC2)=O)CC2(C(=O)NOCCCOC)CC1CCO2 c1(C(N2CCC(C(N(C3CCCCC3)CCOC)=O)C2)=O)cc(OC)cnn1 C(CN=c1[nH]cncc1I)OCCNC(C1CC(C)OC(C)C1)=O c1(C(=O)NCC2(O)CN(C(CC(C)SC)=O)C2)cnc2ncnn2c1O CC1C(NC(c2ccnn2C(C)(C)C)=O)CCCN1C(=O)CC(C)(O)C1CC1 C=Cc1ccc(C(N2CCN(C)C(CNC(=O)Cc3cnc(C)[nH]3)C2)=O)cc1 C(CO)(CCCCNC(=O)CC)NC(C(c1c(C)nc(SCC)s1)CC)=O.O N1(C(c2c(C)cncn2)=O)CC(C)CCC1CNC(=O)C(F)C1CCCC1 C1(c2ccc(COCC)cc2)C(C(=O)N=c2cco[nH]2)CC(=O)N1C1CC1 N1(CC(=O)NCC(C)(O)CNC(=O)C2CC2)CCCCC1=O N1(C(Cc2cn(C(C)(C)C)nc2)=O)CCOC(C)(CNC(C2CC=CCO2)=O)C1 C(=O)(C1Cc2ccccc21)N.C(=O)(C(C)CC1CCCC1)NCCCC(=O)OC C1CC2C1CCN2C(=O)C(c1ccc(C)cc1)C1CC1.C(C(=O)N)SCC=C c1(C(=O)NCC(CNC(c2c(CC)cno2)=O)F)ccnc(C(F)(F)F)c1 N1(C(CSCC)=O)CCC(CF)(NC(=O)CC(Cl)Cl)C1 N1(C(CC(C(C)C)O)=O)CCN(C(C23CCC(C#N)(CC2)CC3)=O)CCC1C C1(CC=C)(NC(=O)C(O)C(C)(C)C)CCCN(C(c2nc(O)c(C)s2)=O)C1 CC1(CNC(c2ccn(CCF)n2)=O)CCN(C(=O)C(F)n2ccnc2)C1 C=CCC(C(=O)N(C)Cc1cc[nH]n1)NC(c1snnc1CC)=O CC(C)(C)CC(C)(C)NC(=O)CC(C(F)F)NC(c1cc[n+]([O-])cc1)=O n1(CC)cc(C)c(C(N2CCOC(c3ccc(C)s3)C2)C(=O)NC2CC2)n1 c1(COC)noc(CNC(=O)CCC2(NC(=O)C(Cl)Cl)CCC2)n1 c1(C(N2C(COC)CN(C(=O)C(C)c3cccs3)CC2)=O)nccc2n[nH]cc12 C1(NC(c2cn(C(C)C)nc2)=O)CN(C(=O)CC(O)CN(C)C)CC2(CCC2)C1 CC1(C)C(C)CCN1C(=O)CC1CCC2CC2C1.C1(C=O)C2C3CCC(C3)C12 C(c1cc(C)cc(C)c1)=CC(=O)N.N1(C(C(CC)=CC)=O)CC2(CCC2)C1 CCCCC(C(=O)N(C1CN(C(=O)C(C)CC#N)CCC1O)C)C(C)C C12(NC(CN=S(C)(C)=O)=O)CCCCC1CN(C(=O)Cc1ccc(F)c(Cl)c1)C2 c1(C(=O)NCCN2CCN(CCC#C)CC2)ccc2c(C(=O)OC)n[nH]c2c1 C1(CC)(NC(=O)Cc2cccc(F)c2)CCCN(C(=O)C(F)n2cccn2)C1 C=C(C)CC(C(=O)N1CCCC(CCCC)C1)NC(c1ccsc1OC)=O c1(C(C(=O)NC(C(=O)NC(CC)C)C)(C)C)cc(Br)ccc1OC CCCCCCCCN(c1cc(NCCC2CCC(C)O2)ncn1)C CCC1=C(C(=O)NCC2(F)CCN(C(c3ccc(C)c(F)c3)=O)C2)CCCO1 CC1(CNC(C2CCC2C(C)(C)C)=O)CCN(C(=O)C2=CCOC2)CC1 C(=O)(C(C)(C)C(N)=O)NCC(C(C)C)(C)NC(C1CCS(=O)CC1)=O CC1C(N=c2[nH]c(N(C)Cc3cscn3)nc3c2SCC3)CCN1C C1(O)(CNC(Cc2n(C)ncc2)=O)CCCN(C(c2ccc(N)c(N)n2)=O)CC1 Cc1c(Br)cc(C(=O)NC2CCCCC2c2nn[nH]n2)c(=O)n1C N1(C(C2(C)CC=CCC2)=O)CC2CC(NC(C3CCCN3C3CC3)=O)C2C1 c1(C(=O)NCCC(C)S(C)(=N)=O)cc(S(=O)(=O)N2CCCC2)ccc1Cl CCS(=O)(=O)CC(=O)NCC1CCCC1NC(c1csnc1C)=O n1(CCC#C)c(N(C)Cc2ccc(C)o2)nnc1C(C1CC(F)(F)C1)O C=CCC(C)(CC)C(=O)NCCCC(C)NC(=O)CCCc1nnc(C)n1C C(=O)(CCCC(C)(C)C)N1CCCC(C)C1CNC(c1ccncc1C(F)F)=O C1(N(C)C)(CNC(=O)COC(F)(F)F)Cc2ccccc2C1 CCN=c1ccc(C(=O)NC2(CNC(C3CCC(C)(C)C3)=O)CCCCC2)c[nH]1 C(C(COC)C(=O)NCC1(C(=O)N(C(CCO)C(F)F)C)CCCO1)OC c1(OC)cc2c(cc1O)CCN(C(=O)NCC(C)CS(C)(=O)=O)C2 C1(C(=O)NC(CC=C)C2CC2)COC2(C1)CN(C(=O)C(F)C(CC)CC)C2 c1(C(=O)NCC2CC(NC(C(C)c3ccsc3)=O)C2)ccc(P(C)(C)=O)s1 Cc1nc2cc(C(=O)NC(C)CN(C(=O)CN(C)C(N)=O)C)[nH]c2s1 C1(C(=O)NCC2(COC)CCN(C)CC2)COCC(C)(C)S1(=O)=O S(=O)(=O)(c1ccc(Br)cc1NC1COC2(CCCC2)C1)NCC1(C)CSCCO1 C1(C(=O)NCC(CC)Nc2ncccc2CCC(=O)OC)CCCCC1O C=CC1(c2c[nH]nn2)COCCN1C(=O)C(C(C)C)c1cccc(Cl)c1 C(=O)(C(C=O)C(C)C)OCC.C1(C=O)CC(C)(C)CCO1.C(C)(CC)CC.N N1(C(Cn2ncc(C#N)c2)=O)CCN(C(c2ccc(Cl)cc2)=O)C(CO)C1 C1(C(F)F)(CNC(C=COCC)=O)CCN(C(=O)CCc2ccccc2)C1 CC1(C(N2CCOCC(NC(c3[nH]cnc3C#N)=O)C2)=O)CC(C2CC2)=NO1 C=CCC(CC(C)C)C(=O)NC1CC(NC(c2c(C)noc2C2CC2)=O)C1 C(=O)(CCC(=O)CC)NC(c1cccnc1)C(=O)N(CCC#C)CCO CCCCCCCCC(=O)NCC(O)CCNC(c1nc(OC)ccc1F)=O Cc1cn2c(C(N3CCCC(C)C3CNC(c3c[nH]c(=O)cn3)=O)=O)cnc2s1 N1(C(C2N(S(CCC)(=O)=O)CCC2)=O)CCCC2C1CCN2C(C1CC(O)C1)=O c1(C(=O)NC2(CNC(C3CN(OC)C(=O)C3)=O)CC2)cc2c(nn1)CCOC2 c1(C(=O)NC(C(C)NC(=O)C(C)n2cnnn2)(C)C)[nH]nc([N+](=O)[O-])c1Cl Cc1ccc2c(c1Cl)N(C(c1cccc(C(=O)O)c1)=O)CCC2 c1(C(=O)NC(CNC(C(CC)n2cccn2)=O)CO)cc(C)nc(O)n1 Cn1c(O)nc2cc(C(=O)NCCCNC(c3cccn4nncc34)=O)ccc12 Cc1ccccc1-c1cc(NC(=O)COCC2CCC2)n(C)n1 C1(CC)CCCCN1C(c1cnc(O)o1)=O.c1(C(=O)N)cccc(C(F)(F)F)c1 N1(C(C(C2CC2)OCC)=O)CCCC2(CC=CCO2)C1 O=C1CC(C(=O)Nc2ccnc(-c3ccc(N4CCNCC4)nc3)c2)CCN1 c1(SC)ncc(C(N2CC(C(=O)Nc3ccc(OC(F)F)cn3)C2)=O)c(Cl)n1 N1(C(=O)Cc2ccc3c(c2)CCC3)CC2CCN(C(C3C=CCCC3)=O)CC2C1 CC1(C)CC(C(=O)NCCC2(O)CCN(C(=O)CCOCC(F)F)C2)CO1 CCS(=O)CC(=O)NC1(C)CC(NC(=O)C(O)C2CC2)C1 N1(c2ccc(-n3c(C)ccc3C)cn2)C(C)Cc2cc(F)ccc2C1C Cc1cc(=NC(=O)C2CN(C(c3c(C)cc(Br)cc3F)=O)CCC2O)[nH]o1 C1(CC)CN(C(=O)C=CSc2nc[nH]n2)CCC1NC(=O)C(F)(F)C1CC1 C(CC(CC)C(=O)NC1CC12CCN(C(=O)CC1CCSCC1)C2)=CC CCCCC(C(=O)Nc1cc(OC)cc(F)c1)NC(C1COCCO1)=O N1(C(c2cc(CC)no2)=O)CC(NC(=O)CSCCC(C)C)CC2(CCC2)C1 N1(C(C2CN3CCC2C3)=O)CC2(C(N3CCC(CC4CC4)CC3)=O)CC1CCO2 c1(CC(N2CCC(CN(C(=O)Cc3cnccn3)C)C2)=O)cccc2c1OCO2 C(=O)(C#CC1CCOC1)N1CCC(C(CO)NC(C(COC)(C)OC)=O)CC1 C1(OC)CC2(C1)CC2NC(=O)CC1CCN(C(=O)CC(Cl)Cl)C1 N1(C(C(C)NC(N)=O)=O)CCCN(C(c2cncc(N)n2)=O)CC1C N1(C(C(C2CN(C(C3C(C(=O)OC)COC3)=O)C2)OC)=O)CCCCCC1 c1(C(N(C2C(C)C2)C)=O)ccccc1OCC.c1cn(CCCO)nn1.C(=O)O OC(CCN=c1[nH]c2c(c(=NCC3(Cl)CC34CCC4)[nH]1)COC2)C1CC1 Cc1cc(F)c(C(=O)NCC(C)CNC(=O)CC(C)C(F)F)c(Br)c1 C(=O)CC(O)C(C)C.c1(COC)noc(C2CC2C(=O)NCC)n1.CCC N1(C(C(N2CC(CC)CC2)=O)=O)CC(C)(C)C12CCC2.C1(C)CCC(F)(F)CC1 C(c1cccc(Cl)c1)=CC(N1CC(N(C)C(C2CC2C(C)(C)O)=O)C1)=O c1(OC)cc(C(=O)NC2CC3(C2)CC3NC(c2sncc2C)=O)ccn1 C1(NC(c2cc(OC)nc(O)c2)=O)CCC2(CC1)CC2NC(=O)C(Cl)=CCl N1(C(=O)C#CC2CC2)CCCC12CCCN(C(=O)CCc1ccncc1)C2 c1(C(=O)NC2CCN(C(C3(CC=C)CCC3)=O)C2)c(F)cc(Br)cc1F N1(CC(N2CC(CCNC(CCOCC)=O)(OC)C2)=O)Cc2ccccc2C1 C1(C(N(CC(=O)NC)C)=O)CN(C(=O)CC(C)n2cccc2)CC1C(C)C N1(c2cc(OCC)nc(C)n2)CC(C)(C)CCC1C.C(=O)(C(F)C1CCC1)N C1(C(=O)NO)(C(=O)NCCCN(C(C)C)C(=O)C2CC2)CC1C C(=O)C(C)C(O)C(C)C.C1(C(=O)OC)CCCC1.c1(CC=O)cn(C)nn1.N C1(C(=O)N)CCCCCC(=O)C1.c1(CNC(c2c(C)con2)=O)cccc(C)c1 c1cc(O)cc(O)c1.c1(CC(C)C(=O)NCC2(C=O)CC2)ccc(Cl)cc1.N C(=O)(C(CC)C(F)(F)F)N(CCC(=O)NCC1CCCC1O)CC=C c1(C(N2CCC(NC(c3c(Cl)cnc(CC)n3)=O)C2)=O)coc2c1C(=O)NCC2 N1(C(c2cccc(C#C)c2)=O)Cc2ccc(-c3cc(F)c(F)c(F)c3)cc2C1 N1(C(C2CC(SC)C2)=O)CCC(C)N(C(c2nn[nH]c2Cl)=O)CC1 C(=O)(C(C)(C)C(=O)N1CC2CCC2(CNC(=O)C(O)C(C)(C)C)C1)N(C)C N1(C(C(C)(C)OC)=O)CCC2(CC(C(=O)NCC(C)O)=NO2)C1.c1ccccc1 C(=O)(C(C)(F)C(F)(F)F)N1CC2(CCC2)C1.C(=O)(CCCC(=O)N)NCCC C(=O)(CCCCC(C)C)N1CCCC1(C)C.c1(CC)nn(C)c(Cl)c1C(=O)N.C c1(CC(=O)NC2CC(CNC(C(C)OCC)=O)C2)c(C)n[nH]c1C C1(OCCC)CC(NC(=O)NCCC2(O)CCC2)C12CCC2 N1(C(C2=C(C)OCCS2)=O)CCC2(CCN(C(=O)Cn3cncc3C)C2)C1 C(=O)(CCCC(C)=O)N1C(CNC(C2(CC)CCNC2=O)=O)CC(F)C1 C(CC(O)CNC(C1CC1C(F)(F)F)=O)NC(=O)CCc1cccs1 C1CC(C)(C)CC(C)(C)C1.CC1C(=O)N(C(c2csc([N+](=O)[O-])c2)=O)CCN1C CCC(C)CCCCC(=O)NCC(C)(F)CNC(=O)C1=CCC1 c1(CC)ccc(F)c(C(=O)N(C)CCNC(C2(C)CCCNC2=O)=O)c1F C1(CCNC(C(COCC)C)=O)CCN(C(=O)Cc2csc(S)n2)CC1 C1(OC)CCC(C(=O)O)CC1.c1nocc1C(=O)NC1CC1.c1ccco1.C c1(C(=O)NC2CCC(NC(CSc3n(C)cnn3)=O)CC2)ccnc2ccnn12 c1(C(=O)NC(C2(O)CN(C(CC(CC)OC)=O)C2)C)cc2cscc2s1 Cc1cc(C)n(CC(N2CCC3CC23C(=O)N(C)CC2CC2C)=O)n1 c1(C(=O)NCC2C3CN(C(C4(C)CC=CCO4)=O)CC32)n[nH]c2nccc(Cl)c12 N1(C(C(CC)(C)C#N)=O)CCC2(CC1)CN(C(=O)C(C)(C)c1sccc1Cl)C2 C1(CC=C)(NC(c2nc(C)no2)=O)CCCN(C(=O)C(F)OC)C1 C(=O)(CCC(F)(F)C(F)F)NCCC1CCN(C(c2n(CC(C)C)ncc2)=O)C1 CCCCCC(CC)C(=O)NC1CCCCC1CNC(=O)Cc1ccsc1 CC12CC(C(=O)NC34CCN(C(=O)CC5CC5)CCC3C4)(C1)C(C)(C)O2 C1(CC=C)(C(=O)NCC(=C2CN(C(c3ccsc3OC)=O)C2)F)CCOC1 c1(C(=O)OCC(=O)NCCCOC)sc(-c2ncccn2)nc1C c1(C(=O)NCC2(C(=O)NCCCC)CC2)cc(OC(F)(F)F)cc(Br)c1 Cc1ccc(F)c(CNC(=O)CC2CCCN2C(=O)C(O)C2CCC2)c1 CC(C)CCC(F)C(=O)NC(C1(O)CCCCC1)C(=O)NC1CC(C(F)F)C1 C1CCCN(S(N)(=O)=O)C1.c1(Cc2n(CCOC)nnn2)ccc(Cl)c(N)c1.N Cc1cc(Br)c([N+](=O)[O-])cc1S(=O)(=O)NC1CCNCCC1(F)F C1(C=O)CCS(=O)(=O)C1(C)C.n1(CCC)nc(C)cc1C(=O)NC1CCC1 CCC(CCCC(=O)N1CCCC(CO)C1)NC(=O)CSc1nc[nH]n1 c1(C(=O)NC2(C3N(C(C(C(C)O)C)=O)CCC3)CC2)[nH]cc2c1CCCC2 c1(C(N2CCC(O)(C(C)NC(=O)CC3C=CCC3)C2)=O)cc(O)cc(O)c1 Cc1cnccc1-c1ccc(C(=O)NC(C)C2CC2)s1.C1(C(=O)N)CN(C)C1 C1(C)(NC(C(CC=CC)C)=O)CCCN(C(c2ccc(CC)s2)=O)C1 N1(C(C2(C#C)CC2)=O)CC(C)CN(C(c2ccc(OC)c(C(F)F)c2)=O)C(C)C1 c1(CCC(=O)OCc2ccccc2)ccc(Br)cc1 N1(C(C)=O)CCCC1CC.c1(C(C=O)N(C)C)cncn1C.C(=O)(C)OC.O C1(C(=O)NCCN(C(=O)CCOC2CCCOC2)C)OCC2CCCC1C2 Cc1ncnc(O)c1C(N1CCC(CNC(c2nccnc2Cl)=O)C1)=O N1(C(CC(C)C)=O)CCC2CN(C(C3(F)CCCC3)=O)CCC2C1 O=C(N=S(=O)(c1ccc(Br)cc1)C(F)F)c1cccn2c(O)nnc12 Cc1cc(CN2CCOCC2C(=O)Nc2cncnc2Br)c(O)c(Br)c1 N1(C(C(CC)=CC)=O)CC2CCC2(CC(=O)NC2CCC23CCCC3)C1 N1(C(C(C)OCCCC)=O)CC(C)(NC(C2CC(C)(c3ccccc3)C2)=O)C1 c1(N(C)C)ccc(C(N2CCC(NC(C3(O)CC3)=O)C2)=O)nn1 C#Cc1ccc(C(=O)NC(C)CCCNC(=O)C(C)CC(C)C)c(F)c1 c1(CC)nc(C)c(Cn2cc(C3(O)CN(C(=O)C(C)(F)CC)C3)nn2)o1 Cc1cc(C=O)c(C)n1C1CC1.C1(CC(=O)N(C(C)C)C)CCC(F)(F)C1.N c1(C(N2C(CC(=O)OC)COC(C)C2)=O)cccc(S(=O)(=O)C(C)C)c1 CC1CCN(C(c2cn(C)cn2)=O)CCN1C(c1cc(-n2cccn2)ccn1)=O c1(C(N2CC3CC2CC3C)=O)cc(C(F)(F)F)cc(Cl)c1.C1(O)(C=O)CC1 C#Cc1ccc(CCNC(=O)C(=O)NCC2CC(O)CN2C)cc1 C1(CNC(C(CSCC)NC(C2CCCCS2)=O)=O)C2CCCOC12 CCCCC(CN=c1[nH]nc(-c2ccccc2)s1)NC(=O)Cc1ccc(F)cc1 N1(C(c2ccc(CCC)s2)=O)CC2CCC1CN2C(C1(C)CC1F)=O N1(C(c2c(C)oc(C)c2C)=O)CCCC(CO)CC1.C(=O)(C(C)(C)S(C)(=O)=O)N n1(CC)ncc(C)c1C(N1CCCC(Cn2cc(CC3(O)COC3)nn2)C1)=O C(CCC(F)(F)F)NC(C(CCC)OCC)=O.c1(C=O)cnn(C)c1C1CC1.N c1(C(C)NC(C2C=CCN2C(=O)C=CC2(C)COC2)=O)cccc(F)c1 C1(C(=O)NCC(=C)C)CC(CC)CCN1C(c1cc(CCO)on1)=O CC1CCCC(C(N2CCOC(COC(C)(C)C)C2)C(=O)NC2CCCCC2)C1 c1(OC)ccc(S(=O)(=O)N(C)CC2CCCN(c3cc(C)ncn3)C2)c(F)c1 c1(CN2C(CN3C(C(C)C)C=CC3)CCC2)cccc(C(=O)O)c1 Cc1cc(C(=O)NCC2CCC2)n2ncnc2n1.c1(CCC(=O)N)cn(C)cn1 c1(C(NC)=O)ccc([SH](=O)=O)cc1.C=C(Cl)C(C)(C)C(=O)NC.C1CC1 N1(C(CC(COC)C)=O)CCC(C)N(c2nc(C)ns2)CC1 C(=O)(CCCN(C)N=O)N1CCC(N(C(C2(SCC)CC2)=O)C)CC1 C1(C(=O)NC(C(C)NC(c2coc(Cl)n2)=O)(C)C)CCN(c2ccccc2)C1=O C1(C(=O)NC(C2CCN(C(=O)Cn3cc(Cl)cn3)CC2)C)CCc2nnnn2C1 c1(C(C=O)O)ccc(C(F)(F)F)cc1.C1(C(N(CCC)CC)=O)CCCOC1.N C(=O)(C1=CCCC1C)N1CC(C)(NC(c2n(CC)cc(Br)c2)=O)C1 N1(C(C(C)NC(C2CCC2)=O)=O)CCC(NC(C2(C)CC2)=O)C1 c1(C(=O)NC2C(NC(=O)Cc3cc(C4CC4)no3)CC2)ccncc1Cl CC1(C)NC(=O)CC1C(=O)NCC(C1CCCN1c1nnc(C2CC2)s1)(C)C C1(NC(c2c(NCC)scn2)=O)CN(C(=O)C(C)=CC2CC2)CC1(C)C n1(C2(CNC(=O)NCC3CCC34CCC4)CCCCC2)ccc([N+](=O)[O-])n1 C1(NC(C=CC2(C)COC2)=O)C2CCC(C2)C1C(=O)NC1CCCCC1.C N#Cc1cncc(C(N2CCC(F)CC2C(=O)NCc2ccncn2)=O)c1 n1(CC)cc(C(=O)NC2(C=O)CC(F)(F)C2)c(C)n1.C1(CC)CCCC1.N C1(NC(c2ccc(OC)s2)=O)(CO)CCN(C(c2cc(C3CCC3)on2)=O)C1 C(=O)(C(F)CC(C)(C)NC(c1nccc(C)c1F)=O)NCC(COC)O N1(C(C2(C#C)CCCC2)=O)CC(NC(c2ccns2)=O)CC2(CC2)C1 c1(N2C(=O)CC(C(=O)NC3C4CN(C(=O)CO)CC34)C2)ccc(F)cc1F c1(C(=O)NCCCNC(c2nc(OC)oc2)=O)cccc(C(C)(C)C)n1 N1(CCC)CC(C(=O)N(CC(CO)CO)C)CC1=O.C1(C(=O)N)CC(F)C(=O)N1 n1(CC#C)cccc1C(=O)NCCC(C)(C)NC(c1ccc(Br)o1)=O c1(OCC(CNC(C2NCC23CCC3)=O)O)ccc(F)c(F)c1 c1(SC)nc2ccc(NC(=O)Nc3ccc(CS(C)(=O)=O)cc3)cc2s1 c1(-c2nc(COCC)nn2CCN2CCCCC2)ccc(C)cc1F Cn1nc(-c2ccncc2)nc1-c1cnn(OCC2CCC2)c1 C(=O)(C1CNc2ccccc21)N1CC2C(CNC(COCCC)=O)C2C1 c1(NC(C2CCCC(Cc3ccncc3)O2)=O)ccc(OC(F)F)cc1 CC1(C)OC(C)(C)C1C(=O)NCC(O)CNC(c1cnc(O)cc1O)=O C#CCC(C(=O)NCC1CCC(CO)CC1)NC(=O)Cc1ccco1 N1(C(C2(C3CCCO3)CCC2)=O)CCC(C2CN(C(C3CCOCC3)=O)C2)CC1 Cc1c(Br)sc(C(N2CC(C)C(F)(F)C2)C(=O)NCc2ccco2)c1C C1(NC(C(c2cccc(Cl)c2)OC)=O)COCCN(C(c2cccn2C)=O)C1 c1(CC=O)ccc2nsnc2c1.Cc1nn(C)c(C)c1C(C)C(=O)NC1CC1.N Cc1ccc(C(=O)N(C(C)CN(C)C(C2CCSC2)=O)C)cc1S(C)(=O)=O CC1(C)CC(C(=O)NCCCCCC(=O)NCc2nc(=O)o[nH]2)CCO1 C1(NC(C2(C)CC2(F)Cl)=O)CC1C1CCCN(c2nnc(-c3ccccc3)s2)C1 C1(CNC(C2(N(C)C)CCCOC2)=O)CN(C(=O)CC(C)(C)C)CC12CC2 C1(C(=O)N)CN2CCN1CC2C.n1(CC)nc(C(=O)NC(C)C2CC2)ccc1=O C12(C(=O)NCCC3CCN(C(C(C(C)(C)C)O)=O)CC3)CCCC1CC(=O)C2 C1(CNC(C2C(CC)C2)=O)CC2(CC2)CN1c1cc(CC2CC2)ncn1 C1(NC(CC(CC)C)=O)C2CC(O)C1N(C(=O)CCCCc1cnn[nH]1)C2 CC(C)C1=NOC(C(N2CC(CNC(=O)C#CC(C)(C)O)CC2(C)C)=O)C1 S(=O)(=O)(c1cncc(Br)c1)N1CC(CC=O)C1.c1(CC(=O)OC)ccccc1 C1(CC(=O)N(C)CCc2cccs2)CC(O)CN1C(c1cnc(C2CC2)o1)=O CCCC(C)CC(=O)N1CCN(C(c2[nH]c(C)nc2CC)=O)CC1C1CCC1 C1(NC(C2C(CCC)C2)=O)CCN(C(=O)CN2CCC(C(N)=O)CC2)C1.C C1(NC(c2c(CC)ncs2)=O)CC(NC(=O)CC)C(O)C1.CC(F)(F)F.O C1CCCN(c2ccccc2)C1=O.C1(NC(=O)OC(C)(C)C)CC(C=O)CC1O.N N1(C(c2ccc(C#N)cn2)=O)CCC2(CCC2)C(CNC(=O)C2=CCOCC2)C1 c1(C(=O)NC(CC)CN(C(=O)CCC2CCOC2)C)cc(C)c(C)nn1 C(CCCCCNC(=O)COc1cccc(F)n1)NC(C1C(C)CC1C)=O Cc1ccc2[nH]c(C(N3CCC(O)C(N(C)C(c4cnc(C)[nH]4)=O)C3)=O)cc2c1 C1(C)(NC(CSc2n(C(C)C)cnn2)=O)CCCN(C(C2CCCS2)=O)C1 C=CCC(C(=O)NCc1cc(O)ns1)NC(=O)CC(C)(C)C1CC1 c1(C(N(C)CCN(C)C(C2Cc3nncn3C2)=O)=O)cc2cccnc2o1 c1(CC)ccsc1C(=O)NCCCN(C(=O)Cc1ccsc1C)C1CC1 N1(C(CCCNS(C)(=O)=O)=O)C2CCC1CC(CCNC(=O)C#CC1CCC1)C2 C12CC(C1)CC(=O)N(C)CCO2.CC=O.CCCC.C(=O)C1CC1.CC C1(C(=O)NC(CNC(c2ccnc(C(C)C)n2)=O)CO)CC12CCCCC2 C1(CC(=O)NCC2CCN2C(c2cnsn2)=O)CCC2(CCC2)O1 C1(NC(c2cc(CC)on2)=O)C2CCCC1CC(NC(c1cn(C)nc1Cl)=O)C2 N1(C(C(CC)(C)C)=O)CCCC(NC(=O)C2=C(C)OCC2)CC1 Cc1ncnc(C)c1CC(=O)NCCOCCNC(=O)C(C)NC=O N1(C(C(CC)n2ccc(C3CC3)n2)=O)CC2(CC(NC(=O)C=CBr)CO2)C1 N1(C(CSCCN(C)C)=O)C2COCC1CC(NC(=O)Cc1ccon1)C2 C(=O)CC1=NNC(=O)C1.c1(OC(C)C)ccc(C(=O)NCC2CCCC2)cn1 c1(SC)cc(C(N2CCCCC2C(O)C(F)F)=O)cc(Cl)c1 C1(NC(c2c(C)nc(CC)o2)=O)CN(C(c2cc(O)ncc2F)=O)CC1(C)C Cc1nn(CC(=O)NCCOCC)cc1Br.n1(CC=CC(=O)N)cccn1 C(=O)C1=C(Cl)CCCC1.CC(C)(C)CCNC(c1ccccc1OCCF)=O.N C1(NC(c2c(C(C)C)con2)=O)CS(=O)(=O)CC1NC(C1(C)CSC1)=O C=CC1COCC1NC(=O)C(CCN(C)C)NC(C1CC1)=O.C(C)(=O)O C1(NC(CCC=C)=O)CC2(C1)CC2NC(=O)CC1CCCC(C2CC2)O1 c1(SC)nc(Cl)c(CN(C2CN(C(c3cn(C(C)C)nn3)=O)C2)C)c(Cl)n1 N1(C(c2c(C)n(CCO)cc2)=O)CC2(CCC2NC(=O)CC2CCCOCC2)C1 N1(C(C=C(C)Cl)=O)CCC(NC(c2scnc2C(F)(F)F)=O)CC1C1CC1 C=C1CCN(C(=O)C=CC2CCC2)C(C(=O)NC2CCOCC2C)C1 c1(C(N2C(C)C(NC(=O)CC(=O)N(C)C)CCC2)=O)cnc2cc[nH]c2c1 CCS(=O)(=O)CC(=O)N(CCC)C.C1(C(N(CC)C)=O)(CC)CNC(=O)C1 C#CCCCCC(=O)NCC1C(C(=O)NC2CC(=C)C2)C1(C)C C(c1c(Cl)cccc1Cl)=CC(=O)N(C1CCC(NC(CCSC)=O)C1)C C1(CC)CCOC1C(=O)NCCOCCOCCNC(=O)C(O)C c1(C(=O)NC2(C)CC(NC(C3CC(C)C3)=O)C2)cccc2occc12 C1(CNC(C2CC3C=CC2O3)=O)CC2CN(C(C3CSC3)=O)CC12 C1(CNC(=O)Nc2cc(CCCCC)[nH]n2)CCCNC1=O C1(C(N(CC(C)NC(C2CC2C(=O)OC)=O)CC)=O)CCCC(=O)C1 c1(C(N2CCC(NC(CCCC(C)=O)=O)C(F)C2)=O)cc2nc(C)ccc2o1 Cc1nnc2n1CCC2(C)C(=O)NCCNC(=O)C(C)OC1CCCC1 c1(N(C)CC2CCCN(C(=O)OC)C2)nc(N(CCCSC)C)c2c(n1)CSC2 C(Br)(C(=O)N1CC(CCCCNC(=O)Cn2cccn2)C1)=C(C)C C1(C(C)NC(Cc2nc(CC)sc2)=O)CN(C(=O)C(=O)NC2CC2)CCO1 Cn1ncc(C(=O)NCc2ocnc2Cn2cc(CN3CCNC3=O)nn2)c1Cl C(CCC(C)C)(C=O)NC(c1cc(COC)[nH]n1)=O.c1(CCC)ccncc1.N CC1CCOC1C(=O)NC(Cc1cn(C2CC3CC3C2)nn1)C(=O)O CCC(C)(CO)C(=O)NC(CNC(c1ccc(CO)cc1F)=O)C1CCC1 N1(C(C(C)S(N)(=O)=O)=O)CCOC2(CCC(NC(=O)CC(C)(C)C3CC3)CC2)C1 C1(NC(=O)CC2CCCCO2)CCCN(CCOc2cc(F)cc(F)c2)CC1 c1(CCC(=O)NCC(CC)NC(=O)CCc2n[nH]c(=N)s2)cnc(O)[nH]1 n1(CC=O)ccc([N+](=O)[O-])n1.C1(O)(CC)CCN(C(=O)C)C1.c1nccs1.N c1(C(N2CCCC2)=O)cc(S(N)(=O)=O)cs1.C(=O)C(F)C(C)(C)O.CCO CCCC(C)(CCC)C(=O)NCCN(CCOC)C(C1CCCC2(CCC2)C1)=O N1(S(CCC(CCOC)C)(=O)=O)CCCc2c1ccc(C)c2C c1(C(N2CC3N(C(CCC(C)O)=O)C(CC3)CC2)=O)cc2c(F)c(F)ccc2[nH]1 c1(C(=O)NC2CC(NC(C3C(C)C3)=O)C2)cnccc1C1OCCO1 C1(CC(=O)NCC(F)CNC(=O)CCc2cnc(O)[nH]2)Cn2ccnc2NC1=O C1(CNC(c2n(CC)nnn2)(C)C2COC2)COCCOC1 c1(C(=O)NC2CC(NC(C3(C#N)CCC3)=O)C2)cnc(C(F)(F)F)cn1 C(CC)(C(=O)NC(CN(C)C(C1(OC)CC(OC)C1)=O)CC)OCC C1CC2CCCC2C1.C1(C(=O)NCC)(OCCCN=[N+]=[N-])CCSC1.C1C(=O)N1 C(CC(O)C(=O)NCC(C)CN(C(=O)CC1CSC1)C)SC c1(NCC=CC)ccc(S(=O)(=O)N2CC3CC4CC3C2C4)c(Br)c1 C(CC)(CC(=O)Nc1cncc(N(C)C)c1)NC(CC=CCCCCC)=O C=CCC(CNC(c1cc(C(C)C)no1)=O)C(=O)N(CC(F)(F)CC=C)C N1(C(c2c(NC(c3ccc(Cl)cc3F)=O)c[nH]n2)=O)CCc2cc(F)ccc2C1 C(=O)(CC1(O)CCOc2ccccc21)NCCN(C(c1cncc(C)n1)=O)CC C1(C)(C(N(CCN(C(=O)Cc2ccccc2Cl)C(C)C)C)=O)CCCS1(=O)=O C(CCCCC(=O)NCC1CCC1CNC(=O)Cc1cnnn1C)OCC N1(C(CC2C(C)CCC2)=O)CC2(CCCN(C(c3ncc(Br)cn3)=O)C2)C1 N1(C(=O)OC(C)(C)C)CCCC12CCN(C(=O)CC(C)(O)CC(=O)O)C2 CC1C(NC(c2ccc(C(N)=O)s2)=O)CCCN1c1nccc(C#N)n1 c1(-n2c(C)nnn2)cc(C(N2CC(NC(=O)C(C)O)C2)=O)cc(F)c1.C1CC1 c1(C(=O)NC2CC3CC(NC(c4c(C)[nH]cc4)=O)C3C2)ncsc1S(N)(=O)=O C1(C(=O)NCC(C#C)CC2CC2)CCCCN1C(=O)CC1(C#N)CC1 N1(C(=O)C2=CSCS2)CC23CCCC2(C1)CN(C(C1CC2COCC2C1)=O)C3 CC1CN(C(c2cccnc2)=O)CCN1C(C1CCC(=O)O1)=O Cc1cc(C)c(C#N)c(NCC2CC(NC(c3n[nH]cc3Cl)=O)C2)n1 c1ccccc1Cl.C1(=C(CNC(CN(CCOC)C)=O)F)CN(C(=O)C)C1.O CC1CC(C(=O)NC23CCC2CN(C(c2cnc(C4(C)OCCO4)s2)=O)C3)=NO1 n1(CC=O)cc(C(F)(F)F)ccc1=O.Cc1sccc1C(=O)NC1CCCC1.N CN1CCCC(C(=O)NCC(=O)N)C1.c1c[nH]nn1.c1cc(C(C)(C)C)no1.C c1(C(=O)NC(C)CN(C(=O)C(C(C)(C)C)C2CCC2)C)ccn2cccc2c1 c1(C(N(C)Cc2ccc(C)c(F)c2)=O)cc(Cl)c(F)cc1Br c1(OC)cnc(C(=O)NCC(C)NC(C2(C(F)F)CC2(F)F)=O)cn1 N1(C(CCC(CC)C)=O)CC2=C(C1)CN(C(c1ccn(-c3ccncc3)n1)=O)C2 N1(C(N)=O)CCCC(NCC(F)C2CC2)C1 C(=O)(C(C(C)(C)C)NC(c1c[nH]c(=NC)s1)=O)NC(C#CC#C)(C)C c1(C(=O)NC(CC=C)C(N2CCC(C)C(C)C2)=O)ccnc(C)c1N N1(C(c2cc(C)[nH]n2)=O)CCC(O)(C(C)NC(=O)COCC(=O)NC)C1 C1(C(N2CC(F)(C(=O)NCC(c3cnn(C)c3)C)C2)=O)CCC(C2CC2)C1 CC(C)(C)C(C(=O)NCCC1CCN(C(c2cnc[nH]2)=O)C1)n1ccnn1 N1(C(C2(C#C)CCCCC2)=O)CC2(CCN(C(c3ncsc3CC)=O)C2)C1 C1(C(=O)NCCCOC=C)C=CCN1C(=O)C(C)OC N1(C(C)C(N2CCN(C(=O)C(=O)N(C)C)C(CCO)C2)=O)CCc2ccccc21 CC1CC2(CCC2)CN1C(=O)C(c1cn(C)nn1)NC(c1c[nH]c(=O)cn1)=O N1(C(C(CC)CC)=O)CCCCCC(NC(C2(Cc3ccc(O)cc3)CC2)=O)C1 N1(C(CCC#C)=O)CCN(C(c2coc(N(C)C)n2)=O)C(CCO)C1 CCC(C)C(C(=O)N(CCCNC(c1ncc(Br)cn1)=O)C(C)C)OC C1(CC)C(NC(=O)C(C)NC=O)CCCN1C(=O)C=CCN1CCCC1 c1(C(=O)NCC(CCOC)NC(C2CCCCO2)=O)sc2ccsc2c1C C1(NC(C(C)OC)=O)CN(C(c2sccc2-c2ccccc2)=O)CCC1CO c1(C(=O)NC2CC(NC(c3nc(Cl)cs3)=O)C2)cc2n(n1)CCCC2O c1(OC)ccc(CNC2CCCCN2S(=O)(=O)C2CCOCC2)c(Cl)c1OC c1(C(=O)N)ccc(F)nc1F.c1(C(=O)NCC2CC2)cc(C2CC2)cnc1Cl Cc1cc(NC(C2CCN(C(c3cnc(C)n3C)=O)C(C)(C)C2)=O)cc(C)c1F N1(C(=O)Nc2c(CC)nns2)CCCC(C(=O)NCCOC(C)C)C1 C=C1CC(C(=O)NCc2ncc(Br)s2)N(C(=O)C(C)SC)C1 C1CCCCN(C(=O)CC23COC(C)(C2)C3)C1.CN1CC=CCC1CC(=O)NC C#CCC(O)C(=O)NCC1CCC(NC(=O)CCC2CCCOC2)CC1 C1(NC(CCc2cc(C)no2)=O)CC(C(=O)NCC(O)CC(C)C)=CC1O C1(C(=O)NC(C)(C)CNC(=O)C)(OC)CCC(C)(C)C1.C1CCCOC1 c1(OC)ccc(F)c(C(=O)Nc2cccc(NC(=O)C(O)CC(C)C)c2)n1 c1(C(=O)NCC(O)CNC(C2(F)CCOC2)=O)cc(Cl)c(Cl)c(Cl)c1 C1(NC(CCCn2c(C)ncc2)=O)CCN(CC2NCCC2C)CC1 c1(OC)cc(NC(c2ncc(C(F)(F)F)cc2Cl)=O)cc(OC)c1F O=C(CCCC(F)(F)CO)NCC1(F)CC(C)C1.c1(C(C(=O)N)O)cccnc1 C(CC(=O)N1CCC12CCC2)(C(C)OC)NC(C1ON=C(CC)C1)=O N1(C(C2(CC#C)CCCO2)=O)CCN(C)C(CNC(c2cccc(C)n2)=O)C1 C1(NC(C(c2ccccc2F)C)=O)CN(C(C2C3COCC23)=O)CC1N=[N+]=[N-] c1(C(NC)=O)cccc2c[nH]nc12.c1(COC)cc(C(=O)NC2CC2)n[nH]1.C C(CCCCC(=O)NC1CC2(C1)CC2NC(c1cc(C)cc(C)c1)=O)=CC C1(C(=O)NC2C(CC(=O)NCC(C(C)(F)F)Cl)CCC2)CN2CCN1CC2 C1(C(=O)NCC2C(NC(CCN(CCCCC)CCC)=O)C2)CCN(C)CC1 Cc1oc(Br)cc1C(=O)NC1CCCCC1CNC(=O)Cc1cn(C)nn1 N1(C(C2(COCC)CC2)=O)CCCC(C)(C)C1.C1(CC=O)CCOC1C.N O=C(C#CC1CCOC1)N1CCC(N(C(=O)CC=C(Cl)Cl)CCO)C1 c1(OCC)ccc(-c2nc(-c3nn(C)nc3Br)n(-c3ccccc3)n2)cc1 N1(C(c2c(F)ccc(OC)c2)=O)CC2CC(C1)CN(C(=O)CC(C)O)C2 N1(C(CNC(C(CC)CC)=O)=O)CCC(F)C(NC(c2ncc[nH]c2=O)=O)C1 C(CC(C(=O)NCC(C)CC1CCCC1)NC(c1cnn(CC)c1)=O)OCC C1(C(N2CCC(OC)(CNC(C3CNC(=O)N3C)=O)C2)=O)Cc2ccccc2C1 C1(NC(C(COC)O)=O)CCN(C(=O)CN2CCCS2(=O)=O)C(C)C1 N1(C(C2(OCC)CCC2)=O)CC(NC(c2conc2C2CCC2)=O)C(F)C1 CCCC(C(=O)OC)C(=O)N1CCCC(C)(C)C1CNC(c1ccc(C)o1)=O c1(C(N2C(COC)CN(C(=O)C(C)=O)CC2)=O)cc2cc(Br)ccc2s1 c1(OC)ccc(NC(=O)C(CNC(=O)C(CO)C)CC2CC2)c(F)c1 C1(C(N(CCCN(C(CCc2c(OC)cccc2)=O)C)C)=O)CCN(C)S1(=O)=O C(CC(C)CC(C)(C)C)NC(C1(CCNC(C2(CC)CCC2)=O)CC1)=O c1(C(N2C(CCC)(C(=O)OC)CCC2)=O)cc(Br)ccc1N=[N+]=[N-] N1(C(C2(C)ON=C(C)C2)=O)CCC(NC(c2nc(C)ccc2F)=O)C(F)(F)CC1 C(=O)(C1=CCC(C)CC1)N1CCC(NC(c2c(C)ccnc2)=O)C1C c1(N2C(C)CCC(NC(c3snc(Cl)c3Cl)=O)C2)nc(O)c2ccccc2n1 C1(C(=O)NC2CN(C(C3(OC)CCOCC3)=O)CC2F)CCc2c[nH]nc2C1 CC1=C(C)CC(C(N2CCCCC(CNC(c3c(O)cccc3F)=O)C2)=O)CC1 C(CCCCC(=O)N1CCC(CNC(C2CN(C3CCC3)C2)=O)(O)C1)OCC Cc1[nH]c(SC(F)(F)F)cc1C(=O)NC1CCN(C(=O)C)CC1.CCN(C)C CN1CCN(C(c2cccnc2)=O)C(C(=O)NC(C(C)(C)O)C2CC2)C1 C1(NC(c2ncn(C(C)C)n2)=O)CC(C(=O)N(C)C(c2cccs2)C)=CC1O CC(C)C(CC(=O)NC1(C)CCN(C(=O)CC2SC(=N)NC2=O)C1)C(C)C Cc1cc(C(=O)NC2CN(C(C3CC34CCOC4)=O)C2)c(C)n1-c1ccn(C)n1 Cn1cc(C(N)=O)cc1C(=O)NCC(C)C1CC1.c1(CC(=O)N)cccs1 C1(C(=O)NCC2CC(NC(C(C(C)C)C#N)=O)C2)CCC2(CCC2)CO1 C1(NC(c2ccc(-c3cccnc3)cc2)=O)CC2CC1N(C(C1CCCS1)=O)C2 C1(C(=O)NCC2(NC(=O)C(C#N)C3CC3)CCCC2)(OC)CCOC1 C1(CC)CN(C(=O)C2=C(Cl)CC2)CCCO1.O=C(CCNC(c1ccoc1)=O)N N1(C(CC2CCCN(C(C(C)CC#N)=O)C2)=O)CC2(CC(CO)CO2)C1 C=CC(CC)CC(=O)NC1CCC12CN(C(C1(C(F)(F)F)CC(O)C1)=O)C2 CC1CN(C(=O)CSc2nnc(S)s2)CC(C)N(C(=O)C2=COCC2)C1 c1(C(=O)NCc2ccn(C(C)C)n2)ccc2c(c1)CCC(=O)N2 C1(C(N(C(C)CNC(=O)C(C)Cc2cnc[nH]2)C)=O)CC2COCC(C1)C2 CC1CCN(CC(=O)NCC(O)CNC(c2nccc(C(F)F)n2)=O)CC1 c1ccc(Br)cc1F.N1(C(c2cnn(C)n2)=O)CCN(C(=O)C(=O)NCCO)CC1.C C1(NC(Cc2n(C)cnc2)=O)CN(C(=O)CC(=O)NC2CC2)CC(C)(C)C1 CCC(CC)(C(=O)N1CC2(C)CC1(C(=O)NCC(O)C(C)C)C2)OC Cc1cc(C)c(CNC(=NCC2CC2)NC2CCCN(CC3CCCC3)C2)s1 c1(C(=O)NC2C(C)N(C(c3ccc(F)o3)=O)CC2)ccc([N+](=O)[O-])cc1Br N1(C(CC(C)(C)O)=O)CCC2OCCN(C(=O)CCn3ccc(O)nc3=O)C2C1 C(=O)(C1=NNC(C(F)(F)F)C1)N(CCCCCCNC(C1(C)CCN(C)C1)=O)C C1(C(N2CC3CC3C2)=O)CCS(=O)(=O)CC1.c1(C(=O)NC)ccn2ccsc12 CCC(CC(C)C)C(=O)N1CCC1C(N1CCC(n2ccnc2)C1)=O CC1CS(=O)(=O)CCCN1N1CCN(c2cccs2)CC1 C1(C(N(C(C)CNC(c2cc[nH]c2)=O)C)=O)CC2CC(O)CC(C1)C2 c1(OC)cccc(CCNC(C2CC23CN(C(c2csc(C)n2)=O)C3)=O)n1 N1(C(c2scc(OC)c2OC)=O)CCN(C(=O)C(C)n2cnnn2)C2CCC12 c1(C(c2n(-c3c(CC)cccc3)nnn2)NCCCCCF)cc(C)cc(C)c1 C#Cc1cccc(C(=O)NC2CCC(CNC(=O)CC(O)CC(C)C)CC2)c1C C(C(C)(C)C(=O)N1CCC(C)(CO)C1)N(C(=O)CCc1nccs1)C c1(C(N(CCCN(C(C(C)c2ccco2)=O)C)C)=O)nc[nH]c2ncnc1-2 C(=O)(CC1OCCc2ccsc21)N1CC(C)C(NC(=O)C(O)C(C)(C)C)C1 C(=O)(C1=CC2CCCCCC12)NCCN(C(CCCOCC)=O)CC Cc1ccc([N+](=O)[O-])cc1C(N1CCC(N(C)C(c2c[nH]c(Br)c2)=O)C1)=O c1(CC)[nH]nc(C(N2CCCCC2CN(C)C(c2c(C)nsc2C)=O)=O)c1Cl CCC(C)(CNC(=O)CC1(C(F)(F)F)CC1)NC(C1CCCO1)=O CCC(C)(C)C(C(=O)N1CCCN(C(=O)CCN(C2CCCCC2)C)CC1)OC Cc1csc(C(=O)N(C(C)(C(=O)Nc2cnc(C3CC3)nc2)C2CC2)C)c1C c1(NC(C(=O)NC2(CC=C)CCN(C)CC2)=O)ccc2nccc(C)c2c1 C=C(C)CC(C(=O)NCC1CN(C(C)C)C1)NC(c1ccc(Cl)cn1)=O C(=O)(C1=NOC(C)C1)N.C1(C(=O)NCc2cc(COC)no2)CCCC1C c1(C(=O)NC(CCOC)C(=O)N(C)Cc2ncc[nH]2)ccc(F)cc1C C(=O)(C(F)(CNC(=O)CCN(C)CC)C(C)C)N1CCOCC(=C)C1.C=O.N c1(C(=O)NCCc2c(CNC(C(CC#C)O)=O)nco2)cnn2ccc(C)cc12 C1(C(=O)NC23CC(CC(F)(F)F)(C2)C3)CCN(C=O)CC1.c1ccccc1.N C1(C(C)=O)CC(C(=O)Nc2ccc(SC(F)(F)F)nc2)=NN1c1ccc(F)cc1 c1(OC)ccc(C(=O)NC(C)CCN(C(=O)CC2CCCC23CC3)C)c(F)c1 N1(CC)C(=O)CNC1=O.C1(C(=O)N)CCOC1C=O.C1(NC(N)=O)CCC1 N1(C(C2N(C)CC(O)C2)=O)CCC(C)(C(=O)NCc2cnc3n2CCC3)CC1 c1(C(=O)NCCCN(C(C2(OCC)CCOCC2)=O)C)cnn2ccc(O)nc12 CCCC(CC(C)C)C(=O)N1CC2CC2(NC(c2cc(CC)ncn2)=O)C1 CCC(C)CCCCC(=O)N1CC(NC(=O)CCCS(=O)(=O)N2CCCC2)C1 Cn1nc(Br)cc1C(N1CCCC(CNC(c2cccc(Cl)c2)=O)C1)=O c1(C=O)cc(Cl)cnc1O.C1(OCCC(=O)NCC23CC(C2)C3)CCCOC1 c1(CN2C(C(N3C4CCC3CC4)=O)CCC2)c(Cl)cccc1B(O)O c1(C(=O)NCC2CC(NC(C3(C#N)CCCO3)=O)C2)cn2ccc(Br)cc2n1 C1(O)(CNC(C2C(C)CCO2)=O)CCN(C(C2CCCC2)=O)C1.N1CCCC1.C c1(C(N2CCN(Cc3cnc(CCC)s3)C(C(C)C)C2)=O)cc(Br)c(Cl)cc1F C1(CC=C)(C(=O)NCCc2cnn(C)c2)CCCN1C(=O)CCC(C)SC C1(C(N(CC(CNC(C(CC)CC)=O)(C)C)CC)=O)CC2CCC1C21CC1 C(C)(CCC(=O)NCC1(C)CCCN1C(c1sccc1C)=O)OC C1(NC(=O)C2=NOCC2)CCN(C(=O)C(F)(F)c2cncs2)CC1O C1(NC(C(C)CN(C(=O)Cc2cccc(O)c2)C)=O)CCCCC1(C)O N1(C(=O)C(c2cccc(Br)c2)N2CCCC2)CCc2ccc(Cl)cc21 c1(C(N(C)Cc2ccc(Br)s2)=O)cncc(C(F)(F)C(F)(F)F)c1 Cc1cc2c(CC(=O)NC3CN(C(=O)C(C)CC(C)(C)C)CCC3O)csc2s1 C(=O)(C#CC1CCCC1)N1CC(C)C(CNC(C2(C)CCNC2=O)=O)C1 c1(C(N2C(C)CN(C(=O)CCC3CCCO3)CCC2)=O)cc2ccc(Cl)cc2s1 CC1=C(C)CC(C)(C(N2CC(CNC(c3nc(Cl)sc3C)=O)C(O)C2)=O)CC1 c1(C(N2CC(O)(CNC(COCCCC(C)C)=O)C2)=O)c(N)cc(F)cc1Cl C#CCCCC(=O)NCC1C(CNC(C2(CO)CC(C)(C)C2)=O)C1(F)F C(=O)(C(C)S(=O)(=O)C(C)C)NC1(COC)CCN(C(=O)C2CC2)C1 C(=O)(C(CCN1CCOCC1)N(C(=O)CCNS(C)(=O)=O)C)OC c1(C(C)C)cccc(CNC(c2cncc(-c3ccc(C4COC4)cc3)c2)=O)c1 C(=O)(CCC=O)NC1CCC(N(C(c2n(CC#C)ccc2)=O)C)C1.C(C)(C)C N1(C(Cc2c(C)occ2)=O)CCC(C2CC2)C1CNC(C1(C2CC2)CC1)=O Cc1cc(C(C)C(=O)NCC)cc(C)c1.n1(CC(=O)N(CCC)C)ncnn1.O C1(CNC(C2(CCCC)CC2)=O)CN(CCCOC)CCCO1 CC(C)(C#N)CCC(=O)NC1CCCCC1n1cc(C2(O)CCOC2)nn1 C(=O)(C(CC1CC=CCC1)NC(=O)CCn1ccnn1)OCC c1(CC)occc1C(N1CCC(C(C)(C)C(=O)NC(C)C(=O)NO)C1)=O c1(CC)nccnc1C(=O)NC1(C(=O)NC(C)C(C)O)CCCCC1 c1(C(C=O)C)ccc(F)cc1.C1(NC(C(C)OCCC#C)=O)CC(F)(C)C1 c1(C(N2C(CNC(c3cnc(C)nc3C)=O)COCC2)=O)cccc2nscc12 C=C(C)CC(C(=O)NC(C1CCCN1C(=O)C=Cc1ccnn1C)(C)C)OC N1(C(C(C=CCCC)O)=O)CCN(C(c2cc(Cl)c(F)cc2F)=O)CC(O)C1 C1(NC(C2(CC)CCN(C(C3N(CC)CCCC3)=O)C2)=O)CCC(F)(F)CC1 c1(C(C(=O)Nc2ccc(COC)cc2)N(CC=C)CC)nc2c(n1C)CCCC2 Cc1nn(C2CC2)cc1C=O.C1(CC=O)NC(=O)NC1=O.C12CC(C1)C2.N C(CCCC(CO)NC(=O)C(CC)OCC)NC(COCCCCC)=O C1(C(N2CCC(C)(N(C)CC)C2)=O)CCC2(CC2)N1C(=O)Cc1c[nH]nc1C c1(-c2c(C)ccc(C)c2)ccc2[nH]nc(C(=O)NCc3ccc(C)nc3C)c2c1 C(CNC(c1ncoc1C)=O)(CC(F)(F)F)NC(C(OC)OC)=O C(C(C)C(F)C(=O)N1CCC(O)(CO)CC1)NC(C(C(=O)OC)C)=O c1(C(N2CC(NC(c3cc(OC)c(Cl)cc3)=O)C(C)C2)=O)cc2ccccn2c1 Cc1cccc(C(N2CCCC2CC(=O)NCC2CCC=CCCC2)=O)c1O N1(C(C(CCSC)O)=O)CCC2(CCC2CNC(c2cnc(C)cc2Cl)=O)CC1 Cc1c(C(=O)NC2CCN(C(C3(C#N)CC3C)=O)CC2)cccc1S(N)(=O)=O C(C(C)(C)C#CC(=O)NC(C1CC(F)(F)C1)C)NC(COCCCCC)=O N1(C(C23CC(NC(C4(C#N)CCC4)=O)(C2)C3)=O)CCC(n2cccn2)CC1 Cc1cccc(C(=O)NC2(C(=O)N(CC(O)CO)C)CSC2)n1 C=Cn1ncc(C(=O)NC(C2CC=CCC2)C(N2CC(=O)NC(=O)C2)=O)c1N Cc1cc(C(N2CC3CC3(C(=O)NCCC3CCOC3)C2)=O)ccc1C#N C=C(C)C(CC(=O)NCC1CCCN1C(=O)CCN1C(C)CCCC1C)OCC N1(C(c2nc(C)[nH]n2)=O)CCC(CNC(C2(F)CC=CC2)=O)C(F)(F)CC1 N1(C(CC=CC)=O)CCC2OCCN(C(=O)C(c3cccc([N+](=O)[O-])c3)C)C2C1 N1(C(COCCCC#C)=O)CC(CC)OC(C)C1.C(=O)(C(C)(C)CN(C)C)N n1(CCOC)ccc2cc(C(N3CC4CC4C3)=O)ccc12.C(=O)(C(F)C1CC1)N C(CC(C(=O)N(CC(F)(F)COC)C)NC(c1n[nH]cc1C)=O)=CC Cc1cc(C)c(C(=O)NCC#CCNC(c2ccccc2N(C)C(C)C)=O)s1 C#CCC(O)C(=O)N1CC=CC(C(=O)Nc2cnn(CC)c2CC)C1 C(CC(=O)N(C1CCC1)C)(C(F)(F)F)OC.c1(C(=O)N)cnn(-c2nccs2)c1 Cc1cc(O)ncc1C(=O)NC1CCN(C(=O)CCCN(C)C)CC1F c1(C(N2CC(NC(C3CCC(C(=O)OC)C3)=O)C2)=O)sc2nccc(C)c2c1C C(=O)(C(C)CCCC(C)C)NC(CNC(C1=C(C)CC1)=O)(C)CO C1(N(C(C(CC)Br)=O)C(c2ccccn2)c2cnc(Br)s2)CC2CC1CN2 c1(C(=O)NC2CN(C(COCCCC#C)=O)CC2C)cc(O)c(O)c(C#N)c1 S(=O)(=O)(c1ccc(Cl)cc1Cl)NC1CC(C(=O)Nc2ccnc(C3CC3)n2)C1 c1(C(C(=O)NCc2cc(C(C)C)on2)(C)C)cc(Br)ccc1F N1(C(C=CCN(C(=O)CC2CSC2)C)=O)CC(O)CC1C1CCC1 C(=O)(C(F)C(F)(F)C(F)(F)F)N.c1(CCC(=O)N(CCC)CC)cccnc1 C1(NC(c2ccc(C(F)(F)F)s2)=O)C=CCC1.c1(C=O)c[nH]nc1C(F)F CC1CCCC(CC(N2CC(C)(C)C2C2CCN(C(=O)CSC3CC3)CC2)=O)O1 S(=O)(=O)(c1c(F)cccc1F)NCc1c(C)sc(-c2ccc(CC(C)C)cc2)n1 Cc1cc(C(=O)NC(C)(C)CCCC(=O)NCC2(O)CC(O)C2)cc(C#N)c1 CCC(C)CCC(=O)NCC(C)CN(C(=O)CCC(=O)OC(C)(C)C)C C1(C(N(CC(C)SC)C)=O)CC2CC1CN(C(c1ccc(CO)cc1)=O)C2 CC1(C)CCC(CC(=O)NC(CNC(c2cc(C3(C)COC3)no2)=O)CO)O1 C1(C(N2CCC(OCC)C2)=O)(NC(=O)CC2(N(C)C)CC2)CCCC1C c1(C(N(C)C)=O)cccc(NC(=O)C(c2ccc(F)cc2)=O)c1O C(=O)(C1CCc2scnc21)NC1C2(CNC(c3c(C)nc[nH]3)=O)CCC(C1)C2 c1(CNC(=O)Nc2c(C)cnn2C)cn2cc(Cl)cc(Cl)c2n1 C1CC2(CCOC2)C1.C(C(=O)NCC1CCC(C=O)C1)(C(C)C)OCC.N C1(C(=O)Nc2cc(C)cc(C#N)c2)CCN(C(=O)C(F)C2CCC2)O1 Cc1cc(C(N2CC(NC(C3CC=CCC3)=O)C(C)C2)=O)c2sc(=N)[nH]c2n1 c1(CC(C)C(=O)N(CCCN(C(=O)CSC(F)(F)F)C)C)ccc(Cl)cc1 CC(CCN(C)C)C(=O)N1CCCC1C1(C(=O)O)CC1 c1(C(=O)NCCCN(C(c2cccs2)=O)CC)cccc(N)n1.CC(C)C.O CC1CC(NC(=O)CCc2ccccc2C#N)CCC1O C1(NC(C2N(C)CSC2)=O)CCC(N(C)C(C2CCCC(F)C2)=O)CC1 c1(OC)cc2cc(C(=O)NCC(CC(C)C)NC(C3CSC3)=O)[nH]c2cc1OC N1(C(CS(=O)(=O)NC)=O)CCC(F)(CNC(C2CCCCNC2=O)=O)CC1 C12(C(Cc3ccccc3)NC(=O)C(=O)N3CCC3CO)CC3CC(CC(C3)C1)C2 N1(CC)CCC(N(C)C(c2ccc(C(=O)NC(CN)=O)cn2)=O)CC1C.OC c1(C(c2n(CCC)nnn2)NCC2CC2)cc(C)cc(C)c1C(=O)OC S(=O)(=O)(c1c[nH]ccc1=NCCC1CC(F)(F)C1)NC(c1scc(CC)n1)C CC(C)CC(C)CC(=O)NCC1CCCCN1C(C1(S(C)(=O)=O)CCC1)=O C(=O)(C1=CCCSC1)NC(C1(C(N2CC3CC2C2CC32)=O)CC1)C c1(C(C(=O)N(C2CCC2C)C)NC(C2C(=C)C2)=O)cccnc1 N1(CC(=O)NC2(CNC(CC3C(C)CC3)=O)CCCC2)CCCCCC1 N1(C(CC2C(C)C2)=O)CCCCC(NC(c2nnc(O)nc2O)=O)C1 N1(C(CCc2n(C)ncc2)=O)CCC2(CC(NC(=O)C3=C(Cl)CCC3)CO2)C1 Cc1c(C(=O)NC(C)CO)[nH]c2c1C(=O)CCC2.c1(C=O)c[nH]nc1C(F)F.N c1(OC)cc(C)sc1C(=O)N(CCNC(C12CC(F)C1C2)=O)C1CC1 C1(C)CC(F)(F)CN1C(=O)C1=C(Cl)CCC1.CCCCCN(CCC(=O)NC)C C1(OCC)C(C(=O)NCC2CCC2)C1C.C1(C=O)CC(n2cnnc2)C1 C1(NC(C(CC)c2cccnc2)=O)CC2(C1)CN(C(c1c(F)cccc1F)=O)C2 N1(C(C2(OC)CCOC2)=O)CC2(C1)CN(C(C1CC(C3CC3)=NO1)=O)C2 CCC(F)(F)CC(=O)N(C)CCNC(=O)C(c1ccccc1OC)C Cc1[nH][nH]c(=N)c1C(=O)N(C1CCN(C(C2(C)CCSCC2)=O)CC1)C C1(C(C)C)CN(C(C2C(Cl)(Cl)C23CC3)=O)CCN1C(=O)CCCN(C)C C1(C)(C(=O)Nc2ccc(C)cc2)CN(C(c2ncsc2C)=O)C(C)(C)C1 C1(C(=O)NC(CC2CN(C(c3ccc(CCC)s3)=O)C2)C)CC(C)N(C)C1 c1(C(=O)OCCOC2CNC2)ccc(C2CC2)cc1Cl C12CC1CN(C(=O)C1=CCCC1)C2.O=CCCOC.C1(CC=O)CCCO1.N C1(NC(CC(C)CF)=O)CC12CCN(C(c1cc3cn[nH]c3cn1)=O)CC2 n1(CC(=O)NC2CN(C(CCCC(N)=O)=O)C2)ccc2ccc(Br)cc12 C12(C(N(CC(C)NC(=O)Cn3cccn3)C)=O)CCCC(C1)C(=O)N2 Cc1cc(=N)[nH]cc1C(N1CCCC1)=O.C(=O)(CCC=CC(C)C)NC1CC1 c1(CC(=O)NCC(C2CCCN2C(C2(O)CCCC2)=O)(C)C)ccccn1 N1(C(Cc2c(C)n[nH]c2C)=O)CC(CNC(c2c(N)cccc2Cl)=O)C2(CC2)C1 C1(C(C)C)CN(C(C2CN(C(C3CNC(=O)O3)=O)CC2C)=O)CC(=O)N1 N1(CC)CCC(CNC(=O)CCC2CCC2)CC1.c1(C(=O)N)cncc(Cl)c1 c1(C(=O)NC(CC)CNC(c2cnc(O)s2)=O)ccc(-n2cccn2)cc1 CC1(C2CN(C(=O)CC3CCCC3NC(C3(F)CCCC3)=O)CCO2)N=N1 c1(C(N(C)CC2OCCN(C(C(CCC)(C)O)=O)C2)=O)cc2nccn2c(O)n1 C#CCC(O)C(=O)N(CC(N1CCN(C(=O)CC23COCC(C2)C3)CC1)=O)C c1(N2CCC(Cn3c(C(C)C)nnn3)C2)nccc(=NCCN2CCCCC2)[nH]1 c1(CSCC(=O)NC2C(NC(C3C(C)C3)=O)CCC2)ccc(Br)cc1 C1(C(=O)NC23CCN(CC2)C3)CC2(CCC2)CN1C(c1cc(O)ncc1F)=O N1(C(C2CN(C(CC(C)=C(C)C)=O)CC2(C)C)=O)CCc2nc[nH]c2C1 CC(C)(C(=O)NC1CCC1)c1ccsc1.C1(CC=O)CCC(C(F)(F)F)O1.C c1(NC(C)=O)cccc(C(C(=O)Nc2ccc(CC(=O)N(C)C)cc2)C(C)C)c1 N1(C(c2n(CC)nc(C)c2)=O)CCC2(CCC(NC(c3cn(C)nn3)=O)C2)CC1 C(=O)(N=c1ccn(C)[nH]1)c1c(C(C)Nc2onc(C)c2C(=O)NC)noc1 CC(=O)CC(C)(C)CC(=O)NC1CCN(C(c2cc(C#N)ccc2Cl)=O)CC1C C1(OCC=C)CCN(C(=NCC2CCOC2)NCC2CCOCC2)C1 c1(C(C)O)n[nH]c(C(C)NC(=O)NC(C)C)n1.c1cc(-c2ccccn2)no1.C CCCCCC(C)CC(=O)NCC1CN(C(=O)CCF)CC1C(F)(F)F CN1CC(N(C)C(=S)Nc2cc(C(C)(C)C)ncn2)CC(F)(F)C1 C=CCC(CNC(=O)OC(C)(C)C)C(=O)N(C1CC1c1ccccc1)C N1(C(c2c(C(C)C)occ2)=O)C2CCC1C(CNC(=O)C(C)CC(N)=O)C2 c1(OC)cc(Br)c(C(=O)NC2CCCC2NC(=O)C(C)O)cc1F n1(CC)c(C(N2CCCCC2CCNC2(CC(F)(F)F)CC2)=O)cnc1O Cc1nn(C(C)C)c(C)c1CC(=O)NCCC(C)C.C1(C=O)CC(F)C(=O)N1 C=CC(C)(C)CC(=O)NCC(C)CN(C)C(c1cc(C(=O)OC)oc1C)=O C1(C(N(C2CN(C(C(COC)(C)C)=O)C2)C)=O)CC(c2cccnc2)=NO1 N1(C(CC=CCC)=O)CCC(C)C(CC(=O)NC)C1.c12cn(nn1)C2 C(=O)C1=C(F)CN(C(=O)C=CC)CC1.C(CC=O)OC.C(C)=O.CC.N C1(C)(N(CCCNC(=O)COC2CC=CC2)C(C)=O)OC(C)(C)OC1C C1(N(C)C)CC2(C1)CN(C(c1ccc(Nc3cnn(CCO)c3)cc1)=O)C2 C(=O)(CC(O)CC(C)C)NC1(C(N(CCCCC(C)C)C)=O)CCC1 CN1CCCC(N(CC2=NOC(c3ccccc3)C2)C(=O)OC(C)(C)C)C1 Cc1c(C=CC(=O)NC)cnn1C.C1(C)(C=O)CNC(=O)C1.C1CC(O)C1 c1(CC(C(=O)NCC2(C)COC(C)(C)O2)(C)C)cncc2ccccc12 Cc1cc(OC(C)C)ccc1NC(=O)C(c1ccc(Br)cc1)(F)F N1(C(c2c(CCC)n[nH]c2)=O)CCC(CNC(C2(F)CCCC2)=O)C(C)C1 C1(C(=O)NC(C2CN(C(CC3C(C)CCCC3)=O)C2)C)CN2CCN1CC2 c1(C(=O)NCC(N(C)C(C2CCCOC2)=O)C2CC2)cncc(-n2cnnn2)c1 C1(NC(C2C=CC=CC=C2)=O)CCSC12CN(C(C1CCC13CCOCC3)=O)C2 N1(C(c2c(CC#N)ccs2)=O)CCCC2(NC(c3ccn(C4CC4)n3)=O)CC2C1 Cc1ncnc(O)c1C(=O)NC(C1CCCN(C(c2scnc2Cl)=O)C1)C N1(C(CCC(C)OC)=O)CC2(CCN(C(C3(N(C)C)CC3)=O)C2)C1 c1(CN(CC(c2nnc(S)s2)=O)Cc2nn[nH]n2)ccccc1 C12CCC(CN(C(=O)CC3C=CS(=O)(=O)C3)C1)C2.c1(C=O)cc(C)no1 CCC(CC)C(C(=O)NCc1cc[nH]c1C(=O)NCC(N1CCOCC1)C)OC CS(=O)(=O)c1cc(C(=O)NCC(C2CCN(C(=O)C(F)F)CC2)F)cs1 c1(C(N2CC3=C(CN(C(=O)CC4CCOC4)C3)C2)=O)cc2c(Cl)c(Cl)ccc2[nH]1 CC(C)C(F)C(=O)N1CCN(C2COCC2NC(=O)CSCC(F)(F)F)CC1 S(=O)(=O)(c1cc2ccccc2s1)NC1(CC(=O)NCCCCCCO)CCC1 C1(NC(c2c(OC)n[nH]c2)=O)CCC(C)N(C(c2cc(Cl)cc(Cl)n2)=O)C1 C1(N=[N+]=[N-])(C(=O)NCC(=C)F)CCN(C(=O)CC2CCC(C)(C)O2)C1 c1(C(N2CC(NC(CC3C(OC)CC3)=O)C2)=O)nnc2ccccc2c1O Cc1[nH]nc(C(=O)NC2CN(C(=O)C(C)OCC3CCCO3)CC2C)c1O c1(CC)cc(C(=O)NCC(O)C)on1.c1(C(=O)N)c[nH]nc1-c1ccc(Cl)s1 c1(-n2ccc(C)n2)ccc(C(N2CCC(CNC(C3COC(=O)C3)=O)C2)=O)cc1 c1(C(N2C(C(N3C(C(N)=O)CCCC3)=O)CC3CC32)=O)cnc(O)c(Br)c1 CC1(C)CN(C(=O)Cn2cnnn2)CC(C)O1.c1(C(=O)N)cccc(C(F)F)n1 CCC(C)C(C)NC(=O)C=CC(C)NC(c1ccnnc1)=O N1(C(C2N(C)CCC2)=O)CCC2(CC1)CN(C(C1CCC(N(C)C)C1)=O)C2 CC1CCn2ncc(C(=O)NC3CCC4CN(c5ncnc(=N)[nH]5)CC4C3)c2C1 C1(NC(C=CCC)=O)CC2CN(C(c3ccc(Br)c(O)c3)=O)CC2C1 Cc1ccc2c(C(N3CC(CNC(c4csc(C)n4)=O)CC3(C)C)=O)onc2c1 Cc1cc(F)ncc1.c1(CC(N2CC(C)(CC=O)C2)=O)ccccc1C(C)C.N C(=O)(C(C)(F)C(=O)N(C)CC1CCCCN1C(c1c[nH]nc1Br)=O)OCC C#Cc1cc(C(N2CC(NC(=O)Cc3csc(S)n3)C(C)(C)C2)=O)ccc1C c1(CN2C3CN(C(C(C)n4cccn4)=O)C(C3)C2)c[nH]c2ccc(F)cc12 C(=O)(C(F)C(C)CNC(C1CCCCCC1)=O)N1C(C(C)C)C(C)(C)C1 CP(C)(=O)c1cncc(C(=O)NC2CC(NC(c3ccc(F)cc3C#N)=O)C2)c1 C1(C(=O)Nc2cc(C)nn2C)CN(C(c2cc(Cl)cc(Cl)c2O)=O)CCC1(F)F c1(C(=O)NC2C(NC(C3(C)CC(C)C3)=O)CCC2)c(O)ccc(Cl)c1F C=CCC(CC=C)C(=O)NCCCC(c1ccccc1)NC(=O)C(C)(C)C C1(C2CC2)(OC)CN(C(=O)CN(C(=O)C(=O)CC(C)C)C)C1 C1(CC)(CC)CC(O)CN1C(=O)CC1(N(C)C(C2CCN2C)=O)CC1 C1(C(=O)NC2(CN(C(c3c(CC)con3)=O)C)CC2)CCC(F)(F)C1O C1(C(=O)OCC)C=CCN(C(=O)CC(O)(c2ccccc2)C2CC2)C1 CC1CCCN(C(=O)C(=O)NC2CCCN(C(c3csc(C(F)F)c3)=O)C2)C1 N1(c2nc(Cl)nc(C)c2F)CCC(C2CCCN(C(=O)CCC(F)(F)F)C2)C1 Cc1c(NC(=O)CONC(C2CCC(N=[N+]=[N-])C2)=O)cccc1F Cc1cc(Cl)c(C(=O)NCCCN(C(=O)CC2COCC(C)O2)CCO)cn1 Cc1cc(S(=O)(=O)N2CC3CCOCC3C2)ccc1Cl CC1CN(N2CC(c3ccc(Br)cn3)C2)CSC1(F)F Cc1sc(O)nc1C(=O)NCC(CC1CC1)C(=O)NCC(c1cccs1)C CN1CCC(=CC(N2CC3CC3(CNC(=O)CC3CCCOCC3)C2)=O)CC1 c1(C(C)C)ncc(CNC(C2(NC(=O)CC3CC3(C)C)CCCC2)=O)[nH]1 c1(C2CCN(C(=O)Cc3cc(Cl)cs3)C2)ccc(F)nc1 C1(C(=O)NCC2CC(NC(CC(C)C3CC3)=O)C2)CCC(CO)CC1 N1(C(=O)Nc2snc(C)n2)CCC(O)(CN(CC(C)C)C)C1 c1(C(=O)NC2C3CN(C(CCc4cccc(C)c4)=O)CC32)cnc2[nH]nnc2c1 CC1(C)CC(O)CN1C(C1CCOCC1NC(c1cnccc1C#N)=O)=O C(=O)(C1CCCn2c(C)nnc21)Nc1cccc(NC(CC2(OC)CC2)=O)c1 c1(C(N2CCCC(CC)(NC(=O)CCC(C)C)C2)=O)ccc2c(=O)cc[nH]c2c1 c1(-n2c(CNC(c3sc(I)cc3Cl)=O)ncc2)ccc(F)cc1F CC(C)(C(=O)NCCCCN=[N+]=[N-])C1=CCN(C(=O)Cc2cccnc2F)C1 CCCCCC(F)C(=O)N(CC(=O)NC1CC1(C)C(F)F)C(C)C N1(C(C(C)OCCOC)=O)CCC(CCC2CCCN2C(=O)C#CC(C)C)CC1 N1(C(COC)=O)CCN(C(C2CCCN(C(c3c(OC)noc3C)=O)C2)=O)CC1 C(=O)(C1=CS(=O)(=O)CCC1)N(CCCCNC(c1c(OC)ccc(C#C)c1)=O)C C1(NC(C2(C#C)CCCC2)=O)CC2CC(NC(c3csc(O)n3)=O)CC12 C1(C(=O)NC2(C)CCC(C)C2)CC(C)(C)CN1C(=O)C(O)C(F)(F)F CCC(C)C(C)C(=O)NCC1CCN(C(C2CC(C(=O)OC)=NO2)=O)C1(C)C c1(C(N2CC(F)(C(=O)Nc3ccc(C(N)=O)cc3)C2)=O)ccnc(Br)c1Cl N1(C(c2c(C)oc(C#N)c2)=O)CC2CC(C(=O)N(CCCCO)C(C)C)C(C2)C1 c1ccc2c(=NCCC3CC3)[nH]c(=NCC3CCOCC3)[nH]c2c1 C1(NC(c2nc(C)sc2C)=O)CCCCCN(C(=O)CC2CC=CCC2)C1 C(C)(C)(CCC(=O)NCC(C)(C)C)NC(C(C)C1CCCO1)=O C1(NC(C2CC(CC(=O)OC)C2)=O)CCCCC1.c1(C=O)ccc(C)o1.N c1(CC(=O)NCC(CCOC)NC(C2CC(C)C2)=O)cc(F)ccc1Cl c1(NC(C2CN(Cc3nc(Br)cs3)C2)=O)ccc(C(F)(F)F)cc1[N+](=O)[O-] C1(CC=C)(NC(c2cn(CC)cn2)=O)CCN(C(c2cc(CF)on2)=O)C1 C1(NC(C2(COC)CC2)=O)C2CC1(C)CN2C(c1ccc(OC)cc1)=O N1(C(c2ccn(C(CC)CC)n2)=O)CCC(NC(C2CCCSS2)=O)CC1C c1(C(=O)OC(C(CC)(O)CC)(C)C)ccc([N+](=O)[O-])c(SC)c1 c1(C(=O)NC2CCCCC2n2cc(CCCCCO)nn2)ccccc1C(F)F C(CCCCC(=O)N(C)CCN(C)C(c1ncc(Cl)nc1Cl)=O)OCC c1(C(=O)NCC2CCN(S(=O)(=O)c3cncc(Br)c3)C2)ccc2[nH]nc(O)c2c1 c1(C(=O)NC(CNC(C=C(C)C)=O)C)cnn(-c2cccc(C)c2)c1C C(=O)CCCS(N)(=O)=O.CC1(C)C(C)CCN1C(=O)CN1C(=O)CNC1=O.N c1(C(N2CC(CC)(OC)C2)=O)cnc(C2CC2)nc1C.n1(CC=O)cncn1.N N1(C(c2nnn(C(C)(C)C)n2)=O)CCC2CCCCC2C1.C1(CC(=O)N)CC(F)C1 c1(CCC)cnnc(C(N2CCC(OCCNC(c3ccoc3)=O)C2)=O)c1 c1(NC(N2CC(C(=O)NC3(CO)CCOCC3)OCC2)=O)ccc2nsnc2c1 N1(C(c2cc(SC)oc2C)=O)CC2(C1)CN(C(c1ccc(F)c(C)c1)=O)C2 C(=O)(C(C(=O)NCC(C)NC(c1cnccc1C)=O)c1ccccc1)OCC Cc1nc2ccccn2c1CC(N1CC(NC(=O)C2=CCCSC2)C1)=O c1(CC=O)ccccc1.C1(C(=O)NCC2CCC2)(OC)CCCC1.C(C)C N1(C(c2nccc(C)n2)=O)CC2(C1)CN(C(=O)Cc1cccc(Br)c1C)C2 CC(C)CC(O)C(C)C(=O)NC(CCC1CC1)C(N1CC2NC(=O)OC2C1)=O c1(SCC)cccnc1C(=O)NC(CNC(=O)CCC1CC1C)C1CC1 C1CCN(C(C2CC3(CCC3)C2)=O)CC(C)(C)C1.CN1CC(C)(C)CC1C(=O)N c1(CC)c(C(=O)NC2CCCC2)nn[nH]1.C(=O)CCN(S(C)(=O)=O)C.N C1(C(=O)NC2(CNC(CC(=C)Br)=O)CCOC2)CC2CC1CC2(F)F c1(CCC(=O)NCC2(N)CC(F)(F)C2)ccc2c(c1)COCC2 c1(C(N2CCC2)=O)cnc([N+](=O)[O-])n1C.c1(C(=O)OC)cn(CC(=O)N)cn1 C1(NC(c2c(Cl)cncc2Cl)=O)CC2CCC1C2.C1(C(=O)N)CC(C2CC2)=NO1 c1(C(C)C)ccc(C(=O)NC2CN(C(c3ccncc3F)=O)CCC2C)c(O)n1 CCCCC(O)C(=O)N1CC(NC(c2[nH]cc(C)c2C)=O)CC(O)C1 CC(C)CC(CNC(c1ccnn1C)=O)NC(c1ccccc1OC(C)C)=O C1(C(N2CCC(N(C)C)C2)=O)CCCC(NC(=O)CC2(C)CCOC2)C1 c1(CC=C)ccc(OCC(=O)NCC#CCNC(=O)C(F)=C)c(OC(F)F)c1 CC(c1ccccc1)=CC(=O)Nc1cccc(NC(=O)C(C)(C)C#N)c1 CC1(C(=O)NCC2C3CC2N(C(c2ccsc2)=O)C3)C2Cc3ccccc3C12 Cc1ncnc(C)c1CC(=O)NC1CCCC1CNC(C1OCC1(C)C)=O C12(CNC(CCCOC(C)C)=O)CCC1CN(C(c1ccc([N+](=O)[O-])s1)=O)C2 C(=O)(C(C)S(=O)(=O)C(C)C)NC(C(C)NC(CNC(CC)=O)=O)CO c1(CN(CCC(=O)OC)C(=O)COC2CC2)cccc(Cl)c1 Cc1c(N)ccc(C(N2CC3CC2(C)C3)=O)c1C.C1(C(=O)N)CN(C2CCC2)C1 C1(NC(c2cccc(CO)c2)=O)C2CC(NC(c3cccc(O)n3)=O)CC12 Cc1nnc2n1CC(C(=O)NCC(C)CNC(=O)C(c1cccnc1F)(C)C)C2 Cc1cc(CCC(N2CCC(F)C(NC(C3CCCS3)=O)C2)=O)cc(C)c1 c1(C(=O)NC2CN(C(C3(C(C)(F)F)CC3)=O)CC(O)C2)ccc2c[nH]nc2c1 C(=O)(CN=c1cc[nH]cc1)N(C(CCNC(c1c(C)c(Cl)ccn1)=O)C)C N1(C(C2N(CC)CC2)=O)CCCCC(CNC(c2cnc(OC)c(Cl)c2)=O)C1 CC1CN(C(C2(C)CC2)=O)CC1NC(C1CC(=O)N(Cc2ccoc2)C1)=O C=CC1CN(C(=O)COC(c2nccn2C)C)CC1NC(=O)CCCC(C)=O c1(C(=O)NCC(CC=C)NC(=O)Cc2ccc(CC)cc2)nccc(C)c1O CN1CC(NC(C2(NC(C3CCN3C(C)(C)C)=O)CSC2)=O)C(C)(C)C1 Cc1cc(C(N2CCC(N(C)C(c3cnnc(O)c3)=O)C(C)C2)=O)cc(N)c1 N1(C(C2CC(C#C)(O)C2)=O)CCC(C(=O)Nc2cc(C)cc(Cl)c2)C1(C)C c1(C(=O)NCCC(C)NC(C23CCCCN2CCC3)=O)nccc2ccsc12 c1(OC)cccc(C)n1.C1(C(=O)N)C(C)CCN1C(c1cnn(C2CC2)c1)=O CCC(O)C(F)(F)C(=O)N1CCCCC(CNC(C2CCC2)=O)C1.C(C)=O.C c1(SCCC(=O)NCC(CNC(c2cc(C#N)[nH]c2)=O)F)nc2ccccc2s1 C(c1cn(C)nn1)=CC(=O)NC(C1N(C(CSCC=C)=O)CCC1)C c1(C(N(CCN(C(c2cc(CC)[nH]n2)=O)C)C(C)C)=O)cc(C)cnn1 c1(C(=O)N)[nH]cc2c1CCCC2.CC1OC2(CNC(C3(F)CCOC3)=O)CC1C2 c1(OC)cnc(N2C(C(=O)Nc3ncc(Br)nc3Br)CC3CC23)nc1C N1(C(C(C2CC2)OC)=O)CCC2OCCN(C(=O)C=Cc3ccc(Cl)s3)C2C1 C1(C(N(CCN(C(COCC=C)=O)C)C)=O)CCCN1CCC CC1CC(NC(=O)CCOc2ccc(F)cc2)CCN1C(c1cc(Br)co1)=O c1(C(N2CCCCC(CNC(C(C)n3cccc3)=O)C2)=O)ccnc2[nH]nnc12 c1(-c2cn(CC)nn2)ccnc(F)c1.N1(C(=O)OC(C)(C)C)CSCC1C=O.N c1(C(=O)NCC2C3CN(C(c4c(C)ccnc4O)=O)C2C3)nc2c(s1)CCCC2 c1(SC)ccc(O)c(C(=O)NC2(C)CCC2)c1.C1(CC=O)CCN(C)C1=O c1(C(N2CCC(CC)C2C)=O)cc(F)c(C)cc1F.c1(CC(=O)N)ccnn1C N1(C(CC2C(CC)C2)=O)CCC(NC(C2(c3cncnc3)CCCC2)=O)CC1 CCC(CC)C(C)C(=O)N1CCC(C)(CNC(=O)CCc2ncccc2C)CC1 c1(NC(=O)NC2CCC(=O)NC2C2CCNCC2)cc2c(cn1)OCCO2 c1(C(C(=O)N)(F)F)cccc(Cl)c1Cl.C(C)(C)(C(=O)NCC(C)(C)C)N(C)C C1(C(=O)NCC2C(NC(c3cccnc3)=O)CCC2)CCc2ccc(F)cc2O1 N1(C(C2(N3CCOCC3)CC2)=O)CCC2CCC(C1)N2C(c1nc(Cl)sc1Cl)=O C1(C(=O)NC2COC3(CCC3)C2)C2CC(O)C(C2)N1C(c1csnn1)=O c1(OC)c(C(=O)NC2CN(Cc3[nH]c(C)cc3C)CC2C#N)cccc1Cl c1(NC(=O)NC(c2c(OC)cccn2)C)cc(Cl)c(Br)cc1F C=C1CC2(C1)CC(C(=O)NCC(C(C)(C)C)NC(C1CC(C)=NO1)=O)C2 C(=O)(C1=CC2C=CC1C2)NCC(C(C)C)C(N1CCCC2OCCC12)=O C1(COC)(NC(C2CC2c2cnn(C(C)C)c2)=O)CC1(F)F C1(NC(CCC(=O)NCC)=O)CC2C1CCN2C(c1cc(C)sc1C)=O Nc1ccc(C(N2CCC(O)(CNC(c3ccc(Br)o3)=O)CC2)=O)c(F)c1 C1(C=O)CC2CCC(C1)C2.CC(CNC(=O)CNC(=O)N)C.C1CC1 C1(C(N(C)CC2CCCN2c2nnc(C(N)=O)s2)=O)CCC2(C1)CC2(F)F N1(C(c2n(CCC)ccc2)=O)CCC(NC(c2nc(C)sc2C)=O)C(F)C1 C(=O)CC(C)C.CCS(=O)(=O)NCC(=O)N.C(CC)CC.C=O.C(C)C N1(C(c2cc(C)nc(O)c2)=O)CCCCC(CNC(=O)COC2CCC2)CC1 C#Cc1ccc(CC(=O)NCC2CCCCCN2C(=O)CCCCCC)cc1 N1(C(C2(CC#C)CCC2)=O)CC2(C)CC(F)(C1)C2.c1(C(=O)N)scnc1Cl C(CCO)(CC(C)C)NC(C(C)N(C(c1cc(CC)ncn1)=O)C)=O C#CCCC(C(=O)NOCCCC1CC1)NC(C1CC(C)(C)CN1C)=O N1(C(c2c(CC)nc[nH]2)=O)CCC2(CCCN2c2nc(C)nc(Cl)c2C)C1 C(c1ccc(Cl)c([N+](=O)[O-])c1)=CC(=O)NC1CCCC1NC(c1cnn[nH]1)=O C1CCCC2(C1)N=N2.n1(CCNC(C(C2CC2)SC)=O)ccc(C(=O)N)c1 Cc1cc(=O)c(C(=O)NCC2CC2NC(C2CCC(CO)CC2)=O)cn1C CC1(C(=O)NCc2ccccc2)CCC(F)(F)CC1.C(=O)CS(=O)(=O)C1CC1 c1(C(N)=O)cc(C(=O)N)c[nH]1.C1(C=O)CC(O)(c2ccccc2)C1.C1CC1.C C(CCCCC(=O)NC(C1(O)CN(C(c2cc(C3CC3)nn2C)=O)C1)C)OC c1(C(C)C)nn(C)c2ncc(C(=O)NCc3ccc4c(c3)C(=O)NC4)cc12 C(=O)CS(=O)(=O)Cc1cccs1.N1(CC(=O)NC(C)CC)CCNC(=O)C1.N c1(OCC)ccc2nc(N3CCCOC(CNC(C4(SC)CCC4)=O)C3)sc2c1 c1(C(N2CC(F)(C(=O)Nc3cc(C)no3)C2)=O)cccc(S(C)=O)c1 N1(C(C2C(C)=C2)=O)CCCC2(NC(c3ncn4ccc(C)cc34)=O)CCCC12 C1(C(=O)OC)CCCC(C(=O)N)C1.c1(C=O)ccc(C)nc1.C1(F)CCC1.C CCC(C)C(O)CNC(=O)CCN(C(=O)C(C)NC(C)(C)CC)CCO c1(C(N2C(Cn3cc(C4(C)COC4)nn3)CCC2)=O)cccc2nc(Cl)cn12 c1(C(C2CC2)NC(C)C(=O)N(C)C)nnnn1CC(F)(F)F.c1cccs1.C N1(C(c2cnn(C)c2N)=O)CC(O)CCC1C(N1CCC(F)(F)CC1)=O C1(C(=O)NCC2CCCN2C(c2ccnn2CC)=O)(COC)C=CCC1 CC1CC(C2CN(C(=O)CCCN(C)C(C3COC(=O)N3)=O)C2)=NO1 c1(OC)ccc(NC(=O)C(C2CCC2)NC(=O)CC2CCC2)cc1C CCCC(C)(CC)C(=O)N(CCCNC(=O)C=C1CN2CCC1CC2)C C1(CN(C)C)CN(N(C)Cc2ccc(F)cc2O)CCO1 c1(OCC)cnc(C(c2nnnn2CC2CC2)NC(C)CSC)nc1 c1(C(C(=O)N(C2C(NC(c3c(C)coc3)=O)CCCC2)C)C)c(Cl)cccc1Cl c1(C(=O)NC(CNC(C2(CC)COC2)=O)C(C)(C)C)cc2n(n1)CCCO2 N1(C(C(COC)(F)F)=O)CC(C(N2CCOC(CCF)C2)=O)CC(C)(C)C1 C1(C(=O)NC(C)CCF)CC(NC(=O)C(C2CC2)C2CC2)CCO1 n1(CCC)cccc1C(=O)NCCCC(C)NC(C1(F)CC1c1ccccc1)=O Cc1cc2n(n1)CCN(C(=O)C(C)(C)NC(=O)COCC1CCC1)C2 c1(C(=O)NCCN(C)C)ccc(C(F)(F)F)nc1.c1cn(-c2ncccn2)nn1 CCCCCCC(C)(C)C(=O)N1CCC(NC(=O)C(=O)NC2CC2)C2(CCC2)C1 C1(C(=O)NC2(CC#C)CC2)CC(NC(c2cc(C3CC3)on2)=O)C1(C)C C1(C(N2CC(=CCC)C2)=O)(NC(c2oc(C)cc2C)=O)CCOCC1 c1(C(=O)NC(CCCNC(C(CC#C)O)=O)(C)C)ccc2c(C)noc2c1 N1(C(C(C)OC(=O)NCc2ccccc2)=O)CC(O)C1(C)C N1(C(c2[nH]cc(CC)c2)=O)CC(C)N(C(c2ccc(C)cc2C)=O)C(C)C1 CCC(CC)CC(=O)N1CC(C(=O)NCCc2noc(C)n2)CC(C)C1 C1(NC(CC2(CSC)CC2)=O)CCC12CCCN(C(=O)CC1=CCCCC1)C2 c1cc(-n2ccnc2)c(-c2noc(C3CC4CCC4C3)n2)cn1 C12(C(=O)NCC(=O)NC3CCCC(C)C3)CCC(CC1)CO2 C1(C=O)CCC(C)=C(C)C1.C(C)(C)(C=O)NC(=O)NCCC.C(C)CC CCCCCC(O)C(=O)NCC1C=CCN1C(c1ccc(OC)c(O)c1)=O Cc1cnn(C)c1CNC(=O)C(c1ccnn1C)NC(C1CCC2CC12)=O N1(C(c2nnc(C)s2)=O)CC(NC(c2ccc(C(F)(F)F)cc2Cl)=O)CC(C)C1 N1(C(CCC#CC)=O)CCC(C)C(N(C(=O)CNC(=O)CC(F)(F)F)C)C1 N1(C(CNC(=O)OCC=C)=O)CCC(=CC)CC1.c1(C(=O)N)sccc1C CC(CC(F)(F)F)NC(=O)C(O)CCNC(=O)CSCC(F)F C#Cc1cnc(C(N2CCCC(NC(=O)CN3CCN(C)CC3)CC2)=O)c(C)c1 N1(C(CNC(C)=O)=O)CC=CC(NC(c2nc(-c3ccco3)sc2C)=O)C1 c1(C(N2CC(O)C2)=O)cnn(CCO)c1C.C(CC1CC1)(C(=O)N(C)C)OC C1(NC(C(CC)CC)=O)CCN(C(=O)CC(C)(C)OC)CC1CC c1(C(N2CC3(NC(C(CC)OC)=O)CC2(C)C3)=O)ccc([N+](=O)[O-])cc1N.O C(=O)(CCC(=O)C(C)(C)C)N1CCCC(CC(=O)N(C2CC3CC3C2)C)C1 C=CC(C)CC(=O)NCC(C1CCN(C(=O)C=CSC)CC1)C c1(CNC(=O)Nc2ncc(C(=O)OC)cn2)cc(F)cnc1Cl C(CC(C)C)(C(=O)NC1(CO)CN(C(C2CC(=O)N(OC)C2)=O)C1)OC c1(C2(C(=O)NCC(CCNC(C(COC)OC)=O)O)CC2)ccc(F)cc1 C1(CC(=O)NC2CC(CC(=O)N(C(CO)CO)C)C2)CSCCO1 CCCS(=O)(=O)CC(=O)NCC1CON(C(=O)OC(C)(C)C)C1 C1(CC(N2CCOCC(NC(C=CCOC)=O)C2)=O)COc2ccccc2O1 N1(C(c2c(C(N)=O)coc2)=O)CC(CNC(=O)C=O)C2(CC2)C1.C1CC1 c1(C(N2CCCCC(NC(c3c[nH]nc3C3CC3)=O)C2)=O)cc2cnccc2[nH]1 C1(NC(c2ccc(CC)cc2F)=O)CC1C1CCN(C(=O)C(C)(O)C(C)C)CC1 C1(CCNC(c2ccc(CSCC)cc2)=O)CCN(C(=O)CCCF)C(C)C1 Cc1nn(C)cc1C(O)C(N1CC2C(CNC(c3ccc(=N)[nH]c3)=O)C2C1)=O C1CC2CCC(C1)N2C(c1cnn(C2COC2)c1)=O.C1(C=O)CC2(C1)CC2F.N c1(C(=O)NC(CCNC(COC(c2nccn2C)C)=O)C)csc(O)n1 C(=O)(CC(O)C(Cl)(Cl)Cl)N(C1CCN(C(C2C3(CCC3)C23CCC3)=O)C1)C c1(C(N)=O)ccc(C(=O)NCC2CCN2C(=O)Cn2cccn2)o1 C1(NC(CC2CC(OC)C2)=O)CCN(C(C)=O)CC1CO c1(C(=O)NC2CCCC(C(=O)NCCOCCC=C)C2)c(F)ccc(O)c1F N(C(=NCCCC1NC(=O)NC1=O)NC1CCOCC1)CC(C=C)(F)F Cc1cccc2c(C(N3CC4CC4(CNC(=O)C(C)CC(N)=O)C3)=O)cccc12 c1(CC(=O)NC(C2N(C(CC(C=C)CC)=O)CCC2)C)c(C)[nH]c2ccccc12 C1(NC(c2c(C(N(C)C)=O)cccc2)=O)CCCCCC1.C(=O)(CC1CCC1)N c1(C(N2CCN(C(C3CC(N(C)C)C3)=O)C(CO)C2)=O)cnc2occc2c1 c1(-c2nc(C(C)SCC)nn2-c2ccc(Cl)nc2)ncn2c1COCC2 N(C(=S)N1CCC(c2ccccc2)C1C)c1ccc(OC)c(OC(C)C)c1OC c1(C(N)=O)cccc(C(C)NC(=O)C(C)Cn2cccn2)c1.C(=O)C.CC.N c1(C(=O)NCC2CCC(NC(CCCSC)=O)CC2)ccc(=O)n(C2CC2)c1 C(=O)(C1=NN2CCC(C)N=C2N1)N1CC(NC(c2c(C)cns2)=O)(CO)C1 C(=O)(CC(C)C1CCC1)NC(C(=O)OC)(C)C.C1(C=O)C2CCC(F)C12.N N1(C(CC=C=C)=O)CCC(CNC(=O)Cc2cc(SC)nn2C)C12CC2 Cc1cnc(Cl)c(S(=O)(=O)NC2CCCC2C(=O)N)c1.c1cncc([N+](=O)[O-])c1 O=C1CCCC(CC(=O)NC2(C(=O)NCC#CC#CCO)CC(O)C2)C1 C1(C(=O)NCC=CCC(=O)N(C)CC2CCN(C)C2)COC(=O)N1C C1(C(=O)OC)CC(C)N1C(C1CCC(NC(c2cscc2C)=O)C1)=O c1(C(C)(C)C)ccnc2c(C(=O)N(CC(=O)O)Cc3sc(Cl)nc3Cl)cnn12 N1(Cc2ncn(C)n2)CCN(C(c2c(F)cccc2Br)=O)C(C(F)(F)F)C1 CN=c1nc(C(=O)NCC(C)(C2CC2)NC(C2CC3CC3C2)=O)cc(C)[nH]1 CC1CCCN(C(c2ccc(CNC(c3ncccn3)=O)cc2)=O)C1 Cc1ccccc1C(C)C(=O)N1CC(CCNC(=O)Cc2ccoc2C)C1 c1(C(N2C(CC(N3CC(=O)NCC3)=O)CCC2)=O)n[nH]c2c1CCc1ncccc1-2 C1(CNC(CCC=C)=O)CCC12CN(C(C1(S(C)(=O)=O)CC1)=O)C2 N1(C(CC2(CC)CCC2)=O)CCC2C(CCN2C(c2c[nH]c(=N)c(C)c2)=O)C1 N12CCOC(C1)N(C)C1(COC1)CC2=O.C(=O)(CCc1ncco1)N.C1CC1.C c1(CNC2CCCN(CCO)C2)cc(Br)ccc1Cl C(=O)(CCS(C)=O)NCC1(OC)CN(C(C2(c3cc[nH]n3)CCC2)=O)C1 c1(C(=O)OC)cc(C(C)C)ccc1NC(=O)CCc1ccccc1 C1(NC(c2c(C(C)C)ocn2)=O)CCCC(NC(C23CC(CO)(C2)C3)=O)C1 C1(COC)(CNC(C2CC(NC(C3CSC3)=O)CCO2)=O)CCCCC1 Cn1c(C(=O)NCCN(C(C2(CO)CCC2)=O)C2CC2)ccc1[N+](=O)[O-] c1(C(N2C(CNC(C3(OCC)CC3)=O)CCC2)=O)ccc2c(C)[nH]nc2c1 c1(NCCCC(C)NC(C23CCCCC2C3(F)F)=O)cccc(F)c1C#N C(=O)(C(C)CC(F)(F)F)N1CCC(C(NCP(OCC)(C)=O)=O)C1(C)C Cc1cc(C(=O)NC2CC(NC(c3cnc(S)n3C3CC3)=O)C2)cc(C)c1C n1(CC)cccc1C(=O)NCCNC(C1(CC(C)C)CC1)=O c1(C=O)cnc(O)nc1O.C(=O)(CCCCSC)NCCCN(C(=O)C)CC N1(CC(=O)NC(C)C(N2CC(O)(C(F)(F)F)C2)=O)C(=O)CCC1=O c1(C(=O)NC2CC(NC(C(C)Cc3ccncc3)=O)C2)c(F)cccc1Cl C(CC(C)C)(C(=O)NC)NC(C)=O.C(=O)C(F)n1cccn1.C1(CC)CC1 C1(C(N(CC=C)C)=O)(CNC(c2nccnc2OC)=O)CC2(CC2)C1 N1(C(C2CC(N(C)CC)C2)=O)CCN(C(=O)COCCOC)C2(CC2)C1 C1(CNC(C=C(C)CN2CCOCC2)=O)CC(C)N(C(C2CSC2)=O)C1 c1(CC)cc(N2CC=CC(NC(=O)COC3CCCCC3C)C2)nc(C)n1 c1(CN2C(C(=O)NCC3(C)CCOCC3)CC(C)C2)c[nH]c2cccc(O)c12 CC1CN(S(=O)(=O)c2ccc(C(F)(F)F)c(F)c2)c2ccccc2N(C)C1=O c1(C(=O)N)cc(O)nn1C.C1(C=O)CC(=O)N(C2CCCC2)C1.C(C)(C)OC c1(C(N2C3CN(C(c4cc(C)oc4)=O)C(CC3)C2)=O)cnc2c(C)cnn2c1 Cc1cnn(C2C(NC3CCN(C(=O)OC(C)C)C3)CC2O)c1 c1(C(N)=O)nc(C(F)F)c2c(n1)CCCC2.C1(CCN)CCCCC1 CC(C(=O)NC1CCN(C(c2c(N)sc3c2CCC3)=O)CC1F)C1=CCCC1 C1(C(=O)NCC(CNC(C(CC)(F)F)=O)(C)C)C2CCC(C2)C1(C)C C(=O)(C1=CCCC1C)NC1(C(=O)NC(CCC)CO)CC(F)C1 N1(C(Cc2cc(C)[nH]n2)=O)CCC(C(N2CC(CO)C(O)C2)=O)C12CCC2 c1(C(C)NC(C(C)=C(C)C)=O)nocc1C(=O)NCC1(C)CC1(F)F c1(CCCC(N2CC(CNC(=O)C3=CCC3)OCC2)=O)ccc2c(c1)CCCC2 C1(C(N2CCCC(n3cc(CNC(N(C)C)=O)nn3)C2)=O)CCc2cnnn2C1 O=C(N=c1cc(Cl)nc(Cl)[nH]1)c1csc(=NCc2ccc(Br)c(C(F)(F)F)c2)[nH]1 N1(C(c2c(C)n[nH]c2C)=O)CCC2(NC(=O)Cn3ncc(O)nc3=O)CC2C1 N(C(=NCCC(=O)N(C)C)NCC1CCOCC1)C1C(C)C1 N1(C(C(C)CNC(=O)CCc2ccncn2)=O)CCCC(CF)C1 N(C1CCSc2ccccc21)C(c1ncc(C)cc1C)c1nnnn1C1CC1 Cc1cnc(F)cc1C(=O)NC1CC(N(C)C)C12CCC2 Cn1cnc2cncc(C(N3CCCC(NC(=O)CC(C)(C)O)C3)=O)c12 n1(CCC(=O)NCCCN(C(C)C)C(c2cccnc2N)=O)cccnc1=O N1(C(C2=C(C)CCC2)=O)C(C)CN(C(c2cc3cccnn3c2)=O)CC1C C(C1Cc2ccccc21)NC(CCC(C)NC(=O)CC(=O)N(C)C)=O C1(c2nnnn2CC2CC2)(NC2(CC(=O)OCC)CCC2)CCCCC1C C=CCCC(C)(C)C(=O)N1CCC(N(C)C(c2scnc2COC)=O)CC1 CC1CC(C)CN1C(c1coc(Cl)n1)=O.C1(C(=O)N)CC(O)(c2ccccc2)C1 CC1CCCN(C(=O)CCn2cnnn2)C1CNC(=O)Cc1sccc1Cl C=CC(C)(CCOC)C(=O)N1CC(C)(C(N2C(CO)CC2C)=O)C1 CS(=O)(=NC(=O)c1c(N)cc(F)cc1Br)C1CCCC(O)C1 Cc1ccc(C=CC(=O)NCC2(F)CCCN(C(=O)C=C3CCC3)C2)nc1 C=CCC(CC=C)C(=O)N1CCC(C(C)(C)C)(CNC(=O)C(O)C=C)C1 Cn1[nH]c(=NC(=O)C(=O)NC2CCCC(C(N)=O)C2)cc1C1CC1 N1(C(CSCc2c(C)noc2C)=O)CC(C2CN(C(C3CC3[N+](=O)[O-])=O)C2)C1 N1(C(C2N(C(C)=O)CSC2)=O)C2CCC1CC(CNC(C1CC13CCC3)=O)C2 c1(C(=O)N)c(N)cc(Cl)cc1F.n1(CCCC)cc(C(=O)NCC(C)C)c(C)n1 Cc1cn2c(CC(=O)NCCOCCn3cc(-c4cscn4)nn3)csc2n1 CCCCC(C(=O)N1CCCC(O)(C)C1)NC(N)=O.C1(CC=O)CC(F)(F)C1 C(C)(CCCC(=O)NCc1cn(C2CC2)cn1)NC(COC(C)=O)=O C(=O)(C(C)(C)CC=C)NC(CC(=O)NCCCC=C)C1CC1 N1(C(C(CC)(C)OC)=O)CC(C2(NC(=O)CCCc3nc(C4CC4)no3)CC2)C1 CC1(C(=O)NCC2(O)CCN(C(=O)CCCC3CCC3)C2)CCCCC1(F)F c1(C(=O)NC2C(NC(CC(=O)NCC)=O)CC2)cccc2[nH]ncc12 C1(CNC(c2cc(C)no2)=O)CCN(C(c2cc(C)n(C3CC3)n2)=O)CC1 C(=O)(C(CNC(c1ccc(N)cn1)=O)C(C)C)N1CC(NC(COC)=O)C1 C12(C(=O)NC3CC(NC(CC4(C)CCOCC4)=O)C3)CCCCC1OSC(=O)N2 Cc1conc1CC(N1CCCC1CN(C)C(c1n[nH]c(C(C)(C)C)n1)=O)=O N1(C(CCN(C(c2c(C)nco2)=O)CC2CC2)=O)CCCC(CCCO)C1 Cc1cccc(CC(=O)NC2CCC(NC(c3cn(C(C)C)nn3)=O)CC2)c1 C1(C(=O)NC2CN(C(CCc3ccc(C)o3)=O)CC2C)CCc2ccccc2C1 c1(OC)ccc(CN2CCOCC2C(=O)Nc2nc(C)cs2)cc1C(F)(F)F C1(NC(c2n(C)ncn2)=O)CC2CN(c3ncncc3Br)CC2C1 N1(C(C(=O)NCCCC)CCCC(C)C)CCC2CS(=O)(=O)CC2C1 C1(C(C)C)CN(C(=O)CCCOC(C)(C)C)CCN1C(=O)CO.CC.CCO C1(C)(C(N(CC(C)NC(c2ccsc2)=O)C)=O)C2CC3CC(C2)CC1C3 C1(O)(CN(C)C(C2CC(F)C2)=O)CN(C(c2c[nH]nc2C(F)F)=O)C1.C Cc1cc(C(C)NC(=O)NC2(CN(C)C)CCCCCC2)ccc1F c12ccc(cc1)SC2C(=O)OC.c1(C=O)cn(CC(F)F)nc1C.C(C)(C)C N1(C(C=CCOC)=O)CCN(C(=O)Cc2nnc(S)n2C)C2CCCCC2C1 N1(C(CCCOCC=C)=O)CCC(C(=O)NCC2CCN2CC)(CF)C1 C12(NC(c3cc(C)nnc3)=O)CCC(CC1NC(c1ccc(O)c(Br)c1)=O)C2 C1(NC(=O)Cc2cnoc2)(CNC(C2(F)CC2)=O)CCC(F)(F)CC1 c1(C(C(=O)NC)N(C(C)C(C)C)CC)ccc(S(=O)(=O)C(C)C)cc1 CC(C)(C)CC(O)C(=O)NCC1C2CN(C(c3csnc3Br)=O)CC12 CC1CN(C(C2CN(c3nc4ccccc4[nH]3)C2)=O)CCc2ccccc21 c1(C(N2C(C(N3CCOCC3)=O)CCCC2)=O)ccccc1S(=O)(=O)C(F)(F)F C(=O)(C1=CCC(C)CC1)N(C1(CC(=O)NCCc2cc(C)ncc2)CC1)C N1(C(CN(C2CCC2)C)=O)CC(CNC(C2COCCO2)=O)CC12CCOCC2 C1(C(N2CCC(NC(c3c(C)nn(C)c3Cl)=O)C(O)C2)=O)CCC2(CCC2)OC1 N1(C(c2cc(C(C)C)n(C)n2)=O)CCC2(CC1)CC2CNC(C1CC1(C)C)=O N1(C(C=CCC)=O)CCN(C(c2c(NC(C)=O)c[nH]c2C)=O)C2CC12 C1(NCC(COC)(C)CO)CCCN(c2ccccc2Cl)C1=O C(CCCCCC(=O)NC(CO)C1CC1)NC(C1CCCC2CC12)=O n1(CCOC)cc(C(N2CC(NC(C3(C)CCC3)=O)CC2C)=O)c(C)n1.O CC1(C)CN(C(C2CC2F)=O)CC1NC(=O)CC(=O)Nc1ccccc1O C12(C(N3CC(F)CC(NC(=O)C4=COCCO4)C3)=O)CCCN(CC1)S2(=O)=O CC1CCC(=CC(=O)N(CC(O)CNC(=O)C(C)(C)c2ccc(Cl)s2)C)C1 C(=O)(N=c1ccn(C(C)(C)C)[nH]1)N(C)C(C1(C)COC1)=O c1(C(N2CCC(NC(C)=O)CC2)C(=O)NCC(=C)C)nc(OC)ccc1F C1(CC)CCN(C(C2CCC(=O)CC2)=O)C1C(N1CCC12CCC2)=O c1(C(=O)NCC(CNC(C2(O)CC2)=O)OC)nccn2ccnc12 C(=O)(CC1=NN(c2ccccc2)C(=O)C1)NC(CNC(C(C(CC)C)O)=O)CO CC(c1cccnc1)=CC(=O)NC1CC1C.c1(CC(=O)N)cccc(C#N)c1 C1(NC(C2CCCO2)=O)CC2CC(C1)N(CCc1ccc(F)cc1F)C2 C1(NC(=O)Cc2cncs2)CC2(C1)CN(C(=O)CCn1cc([N+](=O)[O-])cn1)C2 c1(C(=O)NCC2CCCN(c3ccnc(COC)n3)C2)ccc2ncn(C)c2n1 CCCCCC(=O)N1CC(F)CC1CNC(c1cc(C)c(C)[nH]1)=O C1(NC(c2c(C(C)C)ncs2)=O)CN(C(C2C3CCC2CC3)=O)CC1C C1(N(C)C(C2CC(CF)C2)=O)CN(C(c2cc(N)c(Cl)cn2)=O)CC12CC2 c1(N(C2CCC(N)C2)Cc2cnc(CCCC)[nH]2)cc(C(=O)O)c(C)cc1Br c1(C(=O)NCC(CNC(C23C(C)OC(CO)(C2)C3)=O)F)c(F)cc(O)cc1F c1(CC(N2C(C)CCC2)=O)ccc(Cl)cc1F.C(=O)(C(C)(C)C1(C)CC1(F)F)N C1(N(C(c2c(C)nsc2)=O)C)CCC(NC(=O)C=CC(C)C)CC1 n1(CC(=O)NC2CN(C(COC(C)C)=O)CC3C2C3)nc2ccccn2c1=O CCC1=C(C(=O)NC(C)CN(C(c2cccc(OC)c2F)=O)CC)SCCO1 C1(C(N(CC(C(N2CCCC(COC)C2)=O)C)C)=O)CC2(CC2)CN1C C#Cc1cc(C(=O)NCC2CCCCC2NC(=O)C(C)(F)F)cc(N)c1 Cc1cc(OCC(=O)NCC2C=CCN2C(=O)CCc2cnc[nH]2)cc(C)c1 C1(C(=O)NC2C(NC(CS(CC)(=O)=O)=O)C2)CC2(C1)CC(F)(F)C2 C1CC2(CCC2)CN1C(C1(C2CCCO2)CCC1)=O.Cc1coc(C(=O)NC)c1 n1(COC)nccc1C(=O)NCC1(C(=O)NCCCn2nccn2)CCCC1 N#Cc1ccc(C(N2CC3CC2(CNC(=O)CCCCC2CC2)C3)=O)[nH]1 c1(C(N2CC(NC(c3c(C)nn(C)c3)=O)C(F)C2)=O)c(F)c(F)c(F)c(F)c1F N1(C(CCc2cnc(C)o2)=O)CCC(C(F)F)(CNC(c2cn[nH]c2)=O)C1 C1(COC)(C)CCCN1C(=O)CC1CCC1(C)C.C(=O)C(=O)N(C)C.N n1(CC)nc(C(=O)NCC2CC2NC(=O)CCc2sccc2Br)cc1C Cc1ccc(C(=O)NC2CC3CN(C(C45CC(C)(CO4)C5)=O)CC23)nc1F C(=O)(C1=CC(C)CC1)N1C(C2CC2)CCC1.c1(CCCC)nc(C(=O)N)cs1.C NS(=O)(=O)CCC(=O)NCC(CNC(C12CSCC1C2)=O)CO N1(C(c2cn(C)nc2Cl)=O)CCCC(C)(C)C1.C1(C=O)CCCN1S(C)(=O)=O c1(C(N2CCC3CN(C(C4(C#C)CC4)=O)CC32)=O)ccc2c(c1)CN(C)CC2 c1(OCOC)ccc(C(=O)NC2CCCN(C(c3cccc(SC)c3)=O)C2)cc1 C1(C(C)NC(CCN(CCCCC)C)=O)CCCN(C(c2cc(C)no2)=O)C1 C(=O)(C(C(C)C)n1cc(C)cn1)NCCN(CCC)C(c1nocc1C)=O C(CCCC(=O)NC1(C)CC(C(=O)NCC(C)CC(C)O)C1)OC C1(C(N(CCc2c(C)cccc2)C)=O)CN(Cc2ccncc2)CCC1O N1(C(C=CC=CCC)=O)CCN(C(c2ncccc2C)=O)CC2(CC2)C1 C(=O)(CCS(=O)(=O)C(F)(F)F)N1CCCC1.c1(CC)c(C(=O)NC)ccn1C.C C1(OCC(N2CC(NC(C34CC(C)C3C4)=O)C(C)C2)=O)CCC(F)(F)CC1 N1(CC#N)CCN(C(C2C3CN(C(=O)C(=O)NCCCl)CC23)=O)CC1 c1(C(=O)NCCN(C)C(C23CCCCC2C3(F)F)=O)cc2c(nc1O)CCCC2 C1(C(=O)Nc2ccc(SC3CCOC3=O)cc2)COc2ccccc2C1 C1(CN(C(C2(SC)CCC2)=O)C)CN(C(=O)C(C)Cn2ccnc2)CCO1 C#CC1CCCN(C(=O)C(=O)NCc2cccc(C(=O)OC(C)(C)C)c2)C1 c1(C(=O)NCCOC2CCN(C(c3snc(C)c3N)=O)C2)ccc2nnnn2c1 CC(CNC(=O)CC1CCCOC1)CC(=O)NCc1ccc(O)nn1 C(=O)(C(CC)C=O)OCC.c1(C(N2CCC(C)(CC)C2)=O)cc(C)nc(C)c1 N1(C(C(CC=C)(C)O)=O)CC2CCCC(CNC(c3nonc3CC)=O)C2C1 N1(C(C(C(C)C)NC(C)=O)=O)CCc2sc(-c3cn(CCN(C)C)nn3)cc2C1 Cc1cc(C(=O)NC2C3CN(C(=O)C(C)CC4CCC4)CC23)cnc1C C1(CNC(C(C)N(C(=O)C(C)CC2CCCC2)CC)=O)CCCC1(C)C c1(C(N2CCN(C(=O)CC34COCC(C3)C4)C3C2C3)=O)cccc2nc(O)oc12 C(CC1=CCOCC1)NC(=O)C(Cc1ccoc1)NC(=O)C(O)C1CC1 c1(OCOC)ccc(-c2ccc(C(N3CCC(O)C(C)C3)=O)nn2)c(C)c1C C(=O)(CCS(C)(=O)=O)N1CCC(NC(CCC2(C)CC2)=O)C1c1ccccc1 N1(C(c2nc(CC)sc2)=O)CCC(OCCNC(C2(F)CC=CCC2)=O)CC1 Cc1ccc(C)c(CC(=O)NC2CC(NC(c3cccnc3C)=O)C23CCC3)c1 C1(C#N)(CNC(CNC(CNC(CC=CC(C)(C)C)=O)=O)=O)CCC1 c1(C=O)cc2scc(Cl)c2[nH]1.c1(OC)cccc(OCC(=O)NC)c1.C1CC1 N(C(=NCC(F)F)NCC(F)(F)C1CC1)CC(COC)(C)C c1(-c2nc(C(CCC)C)nn2C2CSC2)c(F)cc(O)cc1F N1(C(c2n(CCN(C)C)ncc2)=O)CC(NC(=O)Cc2cnccn2)C(O)C1 C1(C(=O)NCCCCN(C)C2CC2)CCN(C(=O)C(c2cnn(C)c2)=O)CC1 N1(C(c2cn(CCNC(CCCC#C)=O)nc2)=O)CCN2CCCCC1C2 C1(NCC2CC(=O)OC2)COC2(CCCNC2)C1 C1(NC(CSCC)=O)CCN(C(=O)C(C2CCCC2)OC)CCC1(F)F c1(N2CCCC3(C2)CC3)ccc([N+](=O)[O-])c(C)c1.C(C=CC=O)(CC)=CC.N C1(NC(CCCC(=O)N(C)C)=O)CN(C(=O)C=CCF)Cc2ccnn2C1 C(=O)(C(CO)C(F)(F)F)NCCn1ncc(C(N2CC(C#N)(F)C2)=O)c1 O=C1COc2ccc(NC(N3CCc4n[nH]cc4C3)=O)cc2N1 C1(NC(Cc2cccc(OCC=CC)c2)=O)CC2CCC1N2C(=O)CCS c1(C(N2CCN(C(=O)CCN3CCOC3=O)C3CC23)=O)ccc2c(c1)CC2 C1(CNC(C2C(C)(C)C2)=O)CCCCC1C(=O)NCCC1CCC(=O)N1 N1(C(C2(NC(=O)CSC(F)(F)F)C(C)(C)C2)=O)CCC2C(C1)C2(F)F c1(NC(C2CCN(C(=O)OCC)CC2)C)ccc([N+](=O)[O-])c(SCC)c1 C1(S(N)(=O)=O)(C(=O)NCCNC(c2nccc(C(C)(C)C)c2)=O)CCC1 c1(OC)cnc(NC2CC(C(=O)OC(c3ccccc3Br)=O)C2)nc1 c1(C(=O)NC(CN(C(=O)C(C)C2CC2)CC)C)cc2ccc(O)nc2s1 N1(C(CCOCCOC)=O)CCCC1CNC(=O)C(CC)NC(C)=O c1(CC(=O)NC2CCN(Cc3ccc(OC)cc3O)CC2)nc2ccccc2o1 C1(NC(CC(C(=O)OC)C)=O)CCCC2CN(C(=O)C(=Cc3cn[nH]c3)C)CC12 c1(C(N2CCC(NC(CC(C)OC)=O)C2)=O)ccc(C)cc1SC c1(OC)cc(OC)cc(NC(C(C)(C)CCl)c2nnnn2CCCF)c1 c1(C(N2CC(N(C(=O)CC3CC3(Cl)Cl)C)C2)=O)cc(C2CCCCC2)[nH]n1 c1(OCC2C(NC(=O)C(F)(F)c3ccncc3)CC2)ccc(Br)cc1 N1(C(c2cc(CCNC(c3c(C)cc[nH]3)=O)on2)=O)CC(=O)NCC1C(N)=O C1(NC(c2cnns2)=O)COC2(CNC(C3CCCS3(=O)=O)=O)CC1C2 c1(OC)cc(C#N)ccc1CN1CC(OC)CC1C(=O)N.c1cnc(Br)c(F)c1 C(=O)(CC1COc2cc(O)ccc21)NCCCNC(C(CCC)C)=O c1(C(C=O)(F)F)cccc(Cl)c1Cl.Cc1ncn(O)c1C(=O)NCC1CC1.N Cn1nccc1C(c1nnnn1C1CC(F)(F)C1)NCCC1CCCCO1 N1(CC(N2CC(NC(c3ccns3)=O)C(F)C2)=O)C(=O)NC2(CCOCC2)C1=O C1(C(=O)N)OC(C)(C)OC1(C)C.C1(NC(c2cnc(C(C)C)o2)=O)CCCCC1 Cc1cccc(C(=O)NCC2(C)CCC(NC(c3cccc(O)n3)=O)C2)c1C#N c1(C(=O)NC(C(C)NC(CCN(C)CC)=O)C)cccn1CC c1(CCNC(c2ccc(CC)o2)c2nnnn2CCOC)ccc(Br)nc1 c1(C(N2CC=CC(NC(c3c(C(C)(C)C)ocn3)=O)C2)=O)ccc(Cl)cc1O c1(C(=O)NCC(C)CN(C(=O)CC(C)C2CC2)C)conc1C(F)(F)F C(=O)(NN1CCCC1C(=O)NOCCC1CC1)c1n[nH]c(C)c1O c1(C(N(C(C)C)CCN(C(=O)CCC(C)(C)O)C)=O)coc2ccccc12 c1(OC)ccccc1CCNC(c1ccnc(S)c1)=O.n1(CC=O)cncn1.N C(C(C)(C)CC(=O)N1CCCC1(C)CNC(c1ccc(C)o1)=O)OC c1(C(=O)NCC2CC2)cc(Cl)cc([N+](=O)[O-])c1O.C1(C=O)CC(O)C1.C Cc1ccnnc1C(N1CCC1(C)CC(=O)NC(c1cnn[nH]1)C)=O C1(NC(c2cc(O)nc(O)c2)=O)(CNC(C2CC(F)C2)=O)CCCCCC1 c1(C(C)=O)cccc(NC(=O)COC(c2cccnc2)=O)c1.C(C)(C)(C)N C1(C(NOCC(N)=O)=O)CCC2(CC2)N1C(=O)CNC(=O)CN(C)C C1(C(N(C(C)C2CC2)C)=O)CCCN2CCCCC12.C(C(=O)N)NC(=O)NC C1(N(C(C2(C)CCN(C(c3ccncc3)=O)C2)=O)C)CS(=O)(=O)C1(C)C.CC c1(C=O)cccc(C(F)F)c1Cl.C1(NC(COCCC)=O)CCC(F)(C)C1.N c1(C(N2CC(NC(=O)CC3COCCOC3)C(O)C2)=O)cncc2c[nH]nc12 CN=S(C)(=O)c1cccc(C(N2CC(NC(c3cc4cnccc4o3)=O)C2)=O)c1 c1(OCOC)ccc(-c2cnccc2CN2CCCC2c2ccncc2)c(C)c1 CC(C(C)C(=O)NC(C)(C)CNC(c1cn(C)nn1)=O)c1ccc(Cl)cc1 C1(N(C)C(C2COCC2C(N)=O)=O)CN(C(C2CC3C=CC2CC3)=O)CC1(C)C c1(C(=O)N(c2ncc(OC(F)F)cn2)C2CNCC2(F)F)cc2ccccc2cn1 Cc1cc(C)c(C(N2CC(CN(C(=O)CC3COCC(C)(C)O3)C)C2)=O)cc1N C(=O)(C(C)(O)CCN(C)C)NCC#CC(=O)NC1C(OC)C(O)C1 c1(C(=O)NC2CCN(C(CCOC)=O)CC2C(C)C)cnn2ncccc12 C1(NC(c2n[nH]c(C)c2F)=O)CCC2CC1CN2C(=O)Cn1ccc(=O)cc1C S(=O)(=O)(c1cc(C=O)co1)NC.C(=O)(C(C)(O)C1CCC1)N(C1CCC1)C N1(C(C2C(C)(CC)C2)=O)CCCC2(CC2)C1.C1(CC=O)CC2CCC(C1)N2C C1(O)(CC)CCCN(C(C2(NC(=O)CCC(C)SC)CCCC2)=O)C1 c1(C(=O)NC(c2ccc(O)cc2)C(F)(F)F)cccc(Cl)c1O C1(CNC(c2cc(C3(O)COC3)on2)=O)CCCCC1.c1(C(=O)N)ccns1 c1(C(=O)NCCCN(C(C2C(C)(COC)C2)=O)C)ncc(Cl)c(N)c1Cl C(=O)(CCCc1ccncc1)N(CCCNC(CCNC(COC)=O)=O)C C1(C(CNC(CC(C)C)=O)C)CCN(C(=O)C(CCN(C)C)N(C)C)CC1 c1(NCc2c(C)scc2)ncc(S(=O)(=O)NC2CC3CCC2C3)cc1Cl c1(C(=O)NC23CC(NC(c4cc(C)ns4)=O)(C2)C3)ccnc(-c2ccco2)c1 C(=O)(C(O)CC(C)C)NCC(CC)NC(CNC(C(CC)C)=O)=O c1(C(N2C(CCNC(=O)C(O)C3CCCC3)CCCC2)=O)cc2c([nH]1)CCCC2 n1(CCC(=O)N)ccc2cccnc12.CC1(NC(=O)COCP(C)(C)=O)CCC1 N1(C(c2c(OC)scc2)=O)CCC2CCN(C(C3(C)CSC3)=O)CC12 C(=O)(CCC(=O)c1cccc(Cl)c1)NCCCCNC(C(CC1CC1)OC)=O N1(C(=O)CC2CC3CCC2O3)CCC2OCCN(C(c3ccco3)=O)C2C1 C1CC2(C1)CC(C)(C)C2.C(CSC)(C(=O)NC)OC.c1cn(CC=O)nn1 C1(NC(C(C)Cc2ccncc2)=O)CC2(CCN(C(=O)CC3CC3C)C2)C1 C1(NC(c2cc(CC3CC3)on2)=O)CN(C(c2cc(F)c[nH]2)=O)CC1C1CC1 C(C(O)CCNC(C1CCCN1C(C)=O)=O)NC(C1CC(SC)C1)=O C(C(C)(C)C(=O)NCC1(CC)CC1)SC.c1(CC(=O)N)ccc(Br)cn1 N1(C(C2C(C)=CCS2)=O)CCN(C(=O)CN2CC(F)(F)C2)CC(O)C1 c1(C=O)ccc(C#N)cc1F.c1(C(N(CCC)CC)=O)cc(F)c(F)c(F)c1.N C=CCC(CNC(=O)C(C)S(N)(=O)=O)C(=O)NC1CN(C(C)=O)C1 c12ccc(C)c(c1)OC2.C#CC(CC1CCCO1)NC(N1CC(O)C1)=O.C c1(C(=O)NC23CN(C(C(C(CC)C)C)=O)C(C2)C3)cc2nc[nH]c2cc1N C1(C(C)C)CN(C(c2ncccc2F)=O)CCCN1C(c1cn(C(F)F)cn1)=O c1(NC(N2CC(C(=O)OC)OC(C)(C)C2)=O)cc(N)c2nccc(SC)c2c1 N1(CC(=O)N(c2ccccn2)C(C(C)=O)=O)CCN(c2ncccn2)CC1 C1(CNC(N(CCC)C(C)C)=O)CCCCC1c1ccccc1 C1(F)(CNC(c2cc(Br)no2)=O)CC(NC(C2CCSCC2)=O)C1 C(C(C(C)(C)C)NC(=O)C=CC1CCCO1)NC(CCSc1n(C)ccn1)=O c1(C(N2CC(C)(C)C(NC(=O)COCCF)C2)=O)n[nH]c2nccc(Cl)c12 C(CCCCNC(=O)C=C1CCSCC1)N(C(C1C(OCC)C1)=O)C N1(C(C2C(C(C)C)OCC2)=O)CCCC(C)(C(N2CC=CC2CN(C)C)=O)C1 C12(C(=O)Nc3c(CC)nccc3)CCC(CC1)C2.C(=O)C(C)CCN(C)C.N O=S(=O)(c1c(F)ccc2cnc(Cl)cc12)NC1CNC2(CCOCC2)C1 N1(C(C2C(OCC)C2C)=O)CC2(C1)CN(C(=O)CC1(C)CC1)CCO2 c1(-c2nccc(C(=O)NC(CCC)CCO)c2)cc(=O)c(OC)co1 c1(C(N2CCC(N(CC#C)C(C3CC3CC)=O)C2)=O)cc[nH]c(=NCC)c1 C=C(C)CC(C(=O)NCc1ccnc(C#N)c1)NC(c1cccc(F)c1)=O N1(C(c2c(F)ccc(N)c2)=O)CCCC2(NC(=O)CC3CSCCS3)CC2C1 C1(n2cccn2)(C(N(C2CCC2)CC#C)=O)CCN(C(=O)C(COC)CC)CC1 c1(C(C(=O)OC)C)ccc(NC(c2cnc3n2CCCC3)=O)c([N+](=O)[O-])c1 c1(C(N2CCCC(N(C(C(C=C=C)C)=O)C)CC2)=O)[nH]c2ccccc2c1C#N CN1CCCC1CCN(c1nncs1)C Cc1cnc(NCC2(CC(N)=O)CC2)c(S(=O)(=O)N2Cc3ccc(Cl)cc3C2)c1 C(=O)(C(C)(C)CCCCC)N1C2CC(CC(NC(C3(C=C)CCC3)=O)C2)C1 N1(C(C(C)C)=O)CCN(C(=O)CCc2nc(O)n[nH]2)C2(CC2)C1.C(=O)OC.N c1(C(=O)NC2CCC(C)N(C(=O)CCn3cncn3)C2)ccc2[nH]nc(O)c2c1 c1(C(N2CC(NC(C(CCSC)OC)=O)C(C)C2)=O)[nH]cc2c1CCC2 C1(C(=O)NC(C)CNC(c2ccccc2Cl)=O)CC2CCC1C21CC1 c1(C(N2CC(NC(c3c(C)cc(C)nc3)=O)C(O)C2)=O)coc2cc(F)ccc12 N1(C(CC#N)=O)CC2(CC1CNC(C1CN3CCC1CC3)=O)CC2(F)F N1(C(C(C)(C)OCC)=O)CCC(C(C)NC(=O)CCN2CCC2)CC1 N1(C(CC(=O)OC)=O)CCC(NC(C2(n3cccn3)CC2)=O)CC(C)(C)C1 [nH]1cnc2cc(Br)ccc12.n1(-c2n(C)ncn2)nc(CO)nc1CN1CCCCC1 c1(SC(C)C)ccc(C(N2CC(NC(c3ccc(Br)o3)=O)C(C)C2)=O)cc1 Fc1c(NCc2ccc(Cl)cc2-n2cccn2)cccc1C(F)F C(=O)(C#CC1CCCOC1)N1C(CNC(CC(=O)NCC)=O)CC(F)(F)C1 c1(C(N(C)CC2N(C(C(C(C)(C)C)OC)=O)CCOC2)=O)ccc2cc[nH]c2n1 c1(C(=O)NC(C)CNC(=O)C=C2CCC2)cnc(Cl)cc1N c1(CC(=O)NCCN(C(C2CC2(F)Cl)=O)C2CC2)cccs1 N1(C(C(C)c2cc[nH]n2)=O)CC(F)(C(=O)NCC(O)CC2CCCC2)C1 c1(C(=O)NC(C(C)C)C(=O)NC(c2cc[nH]n2)C)cccc2cc[nH]c12 Cc1ccc(F)c(NC(=O)NC2CN(C(c3oc(C)nc3C)=O)CC2C)c1 c1(C(=O)NC2(C)CCC(NC(=O)C#CC3CCCO3)CC2)ccc2c(n1)CCC2 c1(C(N(C2CCCN(CC)C2)CC)=O)c(Cl)cccc1Cl c1(C(=O)NCC#CC(N2CCCC(C(C)O)C2)=O)cc([N+](=O)[O-])c[nH]1 CCCC(C(=O)NC(C(=O)NC1(CF)CC1)C1CCC1)NC(C)=O N1(C(C(CCC)Cl)=O)CCC2(C1)CN(C(c1cc(F)c(F)cc1I)=O)CCO2 c1(N2CCOCC(CC)C2)nc(=NCCC(O)C(C)C)[nH]c2c1cnn2C c1(-n2ncc(C(N(C3CC(NC(c4cnc[nH]4)=O)C3)C)=O)c2)ccc(F)cc1F C1(C(N(CCCC)C)=O)CCCS(=O)(=O)C1.c1(COC)csc(C=O)c1.N C(=O)(CC(O)CNC(C1CCCC(=O)N1)=O)N(C(C)CCO)C N1(C(c2c(C)c[nH]n2)=O)C2CCC1C(C)C(NC(c1ccc(C)c(C)c1)=O)C2 S(=O)(=O)(c1ccccc1Cl)N1CCC(C(=O)Nc2cn[nH]c2)C(O)C1 C1(C(=O)NC(C)CCNC(=O)Cc2ccno2)CCCCN1Cc1ccccn1 c1(OC)ncc(=NC2CCCC23CN(C(=O)C(C)CCOC)C3)[nH]c1C c1(C(N2CC3C(NC(c4cc(C)nc(C)n4)=O)(C3)C2)=O)c[nH]c2ccc(F)cc12 C1(NC(c2ccn(C)n2)=O)CC2CC1CN(C(C1CCC3(CC3)C1)=O)C2 c1(C(=O)N)ccc(N)cc1[N+](=O)[O-].C(C(C)(C)C)N(C(=O)C(F)C1CCOC1)C N1(CC)CCOCCC1C.S1(=O)(=O)CCN1 C(C1(O)CCc2ccccc21)Nc1c(SC)ccc(Br)c1 C1(NC(NCC2(C)CCC2)=NCCN2CCOCC2)CCc2ccccc2C1 C=CCC(CC(C)C)CC(=O)N1CCC(F)(CNC(C23CC(F)(C2)C3)=O)C1 c1(CNC(C=CCN(C)CC)=O)cc(C(=O)N)n(C)n1.C(C)C(F)F CC1CN(C(C2C=CCCC2)=O)CC2(CCN(C(=O)CCCC(C)(C)C)CC2)O1 N(C1c2ccccc2CCC1F)C(=O)NCC12OCC(C)(C1)C2 Cn1cc(CNC(C23CC2CCC3=O)=O)c(O)n1 c1(CC(N2CC(c3n(C)ncc3)OCC2)=O)c[nH]c2cccnc12 c1(CC(N2CCC2C2CCOCC2)=O)coc(-c2ccccc2)n1 N1(CC(=O)N(C2CCCN(C(=O)CC3(C)CCCCC3)C2)C)CCCCS1(=O)=O CC(C)(C(=O)NCCC1CC1)c1ccccn1.c1(C=O)csc(C(N)=O)n1.N c1(C(N2CC(F)(CNC(CCc3scc(C)n3)=O)C2)=O)ccccc1C CCC(C)(CNC(=O)CCc1scnc1C)NC(=O)CCC1CCCC1 c1(C(=O)NCC(C)NC(C2(C#C)CC2)=O)cccc(C(F)F)c1 C=CC1(C(=O)NOC(C)C)CCN(C(C2CC3(CC3)CO2)=O)C1 C12(CNC(c3c(C)ccn3C)=O)CCC1CN(C(c1ccoc1C1CC1)=O)C2 C1(CNC(c2c(C)con2)=O)CC2(CC(NC(=O)CS(C)(=O)=O)C2)C1 C(CN=c1cc[nH]c(C#N)n1)C1CCN(C(CCCCCCSC)=O)C1 CCCC(C(=O)NCc1csc(C(N2CCC(CC(=O)NC)C2)=O)c1)OC Cc1cc(C#N)nc(=NCC2CCN(C(=O)Cn3ccc(C(F)F)n3)CC2C)[nH]1 c1(C(CF)NC(C(n2cc(CCN3CCN(C)CC3)nn2)C)=O)cccc(Cl)c1 C1(C)(NC(C(=O)NCC)=O)CCCCC1C=O.c1(CC(C)C)ccccn1.N C(=O)(CC(C)(C)C#N)NCCC(C)CCNC(=O)CN1CCCCC1=O C(=O)(C(F)(F)C(F)(F)C(F)F)N(CC(=O)Nc1ccc([N+](=O)[O-])cc1F)C c1(OC)ccc(C(=O)NCC2CN(C(C3CCC(C)C(C)C3)=O)C2)cc1N C=C1CCN(C(=O)Cc2cc(C)cs2)C(C(=O)NC(C2CCOCC2)C)C1 C12(C(=O)NCCCc3n(C)nnn3)CCC(CC1NC(c1cc(O)cs1)=O)C2 C1(C(N2CCC2)=O)CC2CC1C1C2C1(F)F.C(CCC(=O)N)NC(=O)OC.C c1(NC(C2N(C(Cc3cnc(C)s3)=O)CC(O)C2)=O)c(O)cccc1O C1(NC(C2C3CCCC23)=O)CCCN(C(C2(C(c3ccccc3)=O)CC2)=O)CC1 c1(OC)ncc(C(=O)NC(CC2CC2)CC(=O)NCC(C)OC(F)F)cn1 N1(C(CC2C(CC)C2)=O)CCC2CC2(C(=O)NCC2CNC(=O)CO2)CC1 C1(C=O)CCC(S(C)(=O)=O)CC1.CC(C)C(C)C.C(=O)(CCC1(C)CC1)N C1(N(C(c2ccc(C)cc2C)=O)C)CCc2ccccc2N(C)C1=O N1(C(CC(=O)OC)=O)CCCC(NC(C2(c3ccnc(Cl)c3)CCC2)=O)C1 Cc1sc(C(N2CCCC2Cc2nccn2C)=O)c(Br)c1C C(CC(=O)NCC(=O)NCC(F)F)N(C(COCC#C)=O)C C1(O)(CNC(C2(C)CC(=C)C2)=O)CCN(C(c2sccc2C#N)=O)C1 N1(C(c2cnc(CC)o2)=O)CC(C(=O)Nc2cccnc2)C(C)(C)C1 CC1(C)CC(=O)N(CC(=O)NC2CCN(C(c3cc(F)ccc3F)=O)CC2O)O1 N1(C(C2(SCC)CC2)=O)CCC2CC2(NC(c2cn(C)cc2C)=O)CC1 O=C(C1=CCCN(C(C2CCC(F)(F)CC2)=O)C1)Nc1ccc(F)c(CO)c1 c1(C(=O)NC2C(NC(c3cc(CC)n(C)n3)=O)C2)cnc2cnccc2c1 N1(C(CCC(=C)C)=O)CCC2(CCCN2C(c2csc(Cl)c2)=O)C1 C1(CC)CCCN(C(=O)C(C)CN(C)C)CC1.c1(CSC)cccc(C=O)c1.N CCC(C#N)CNC(=O)C(O)C1CN(C(=O)C(c2cncnc2)C)C1 Cc1cc2cc(CNCCCc3cccc(Br)c3)oc2cc1C c1(C=O)ccc(C)c(O)n1.c1(C(C)=O)cc(C(=O)N(CCC)C2CC2)n[nH]1.N c1(C=O)cc(C)nc2ncnn12.C1(NC(CNC(C)=O)=O)CCC2(CC1)CC2.N c1(N2CCC(=CCC)C2)nc2c(c(=NC3CN4CCC3C4)[nH]1)CCCCC2 c1(OC)cccc(C(N2CCCC(NC(c3cnn(C)c3OC)=O)C2C)=O)c1F c1(C(=O)NCCC2(O)CN(C(c3scc(OC)c3)=O)C2)cnn2c1CCCC2 Cc1cccc(N)c1C(=O)NC1CCCC(NC(C2(c3ncco3)CCC2)=O)C1 c1(CC(=O)NC2(CNC(Cc3c(C)scc3)=O)CCCC2)cccc(Cl)c1 CC1(C)CC(NC(=O)C2=CCC(NC(=O)Cn3cnnn3)C2)C12CCC2 C(=O)(C(F)(CNC(C1CCO1)=O)C(C)C)NCC(C#C)(C)C Cc1c(Cl)nc[nH]c1=NCCC(C)NC(c1cnc2ccccc2c1)=O C(CC(C(=O)NCC(C)(F)C)N(C)C)N(C)C.c1(C(=O)N)cc(C2CC2)on1 C(=O)(CCCCC(N)=O)NC(C(C)C)(C)CNC(c1cc(C#N)cs1)=O N1(C(C(C)C2CCC2)=O)CCCC(CCCCNC(=O)CSc2n[nH]c(O)n2)C1 C1(CNC(C(CC=C)(C)C)=O)CCC(C)(C)CN1C(c1scnc1CC)=O c1(C(N(CC(CC)NC(=O)CC(CC)C2CCC2)C)=O)ccc(C)cn1 N1(C(CS(CC)=O)=O)CCC2(CC1)C(NC(c1ccc(Cl)cc1F)=O)CS2(=O)=O N1(C(c2ncc(CC)s2)=O)CCC2(CCCN2C(=O)CC(O)CN(C)C)C1 c1(C(=O)NC2CCN(C(C(CC)CN(C)C)=O)CC2)cccc2nn[nH]c12 C1(CC(=O)Nc2ccnn2C2CC2)CCN(C(=O)CN2CCCCC2)C1 C1(C)(C(NOCCC=C)=O)CCN(C(=O)CC2CCC(C#N)C2)CC1 C(=O)(C1=Cc2ccccc2C1)NC(CNC(C(N1CCC(O)CC1)C)=O)CO C1(C2CCC2)(C(=O)Nc2cccc(NC(c3c(N)ccc(Cl)n3)=O)c2)CC1(F)F C1(NC(C(C)C)=O)CCN(C(c2ccc3c(c2)OCC3)=O)CCC1CO Cc1cc(C(=O)NC2C=CC(C(=O)NCC3(C)CCCS3)C2)sn1 C12CC3(COCCN(C3)C(=O)N1C)C2.c1(CC(=O)OC(C)(C)C)ccsc1 Cc1ccc(F)c(CNC2CCC(CC(C)C)CC2)c1 c1(OC)cccc(CNC(c2ccccc2)=O)c1OCC1CNCCO1 C(CCSC)(C(=O)NC1COCC1C(=O)NOC1CC2CCC1C2)OC C#Cc1nc(C(=O)NC2CCCC2NC(c2ccnc(OCC)c2)=O)cs1 c1(C(=O)NCCCN(C(CCNC(=O)OCC)=O)C)snc2ccccc12 N1(C(CC2CC(C)(C)OC2)=O)CC(C2(NC(=O)CCNc3ccccn3)CC2)C1 N1(C(C(C)NC(c2ccoc2)=O)=O)CCC(C)(NC(C2CCCC3CC23)=O)C1 Cc1cccc(F)c1NC(=O)NCc1ccccc1.C1C=CCN1C(C)C.C CCC(Cc1ccc(N)cc1)C(=O)NC(C)(C)CNC(C1CCN(C)CC1)=O C1(C(N(c2ccc(Oc3ccccc3)c(F)c2)CC)=O)CN2CCC1CC2 C1(N(CC(=O)N(C)C)Cc2nc(O)n[nH]2)CCN(C(N)=O)C1 CCCC(C#N)C(=O)NC1(C)CCN(C(c2cc(C(C)C)nn2C)=O)CC1 Cc1ccc(NC(C23CC2CN(C(=O)Cc2cccc(Cl)c2F)C3)=O)c(O)c1 C1(C(=O)NCCC(F)(F)CO)CCCCCCN1C(=O)COCC(F)F c1(C(=O)NC(CNC(COCCC)=O)(C)CC(C)C)cccc2ccsc12 Cc1cc(C(=O)NCC2(C)CCCC2)n(C2CCC2)n1.C1(C=O)CCC(C)O1 C1(CC)CCN(C(=O)CCc2ncccc2C)C1CNC(=O)C(C)CSC c1(N2CC(C)C(CNC(=O)C(O)C3CCC3)CC2)nc(Cl)nc2c1CC(C)CC2 C1(NC(c2ccccc2)=O)C2CN(C(C34CCC3CC4)=O)CC12.C1(O)CCOC1 C1(CCOC)CN(C(c2ncc(F)cc2N)=O)CCN1C(=O)C(O)C(C)C N1(CC(=O)NC)CC2(CN(C(c3ccc(C(F)(F)F)cc3)=O)CCO2)C1 S(=O)(=O)(c1cccc(C(=O)NC)c1)NC.C1CCN(C(C23CCC2C3)=O)C1 N1(C(C)C)CC(C(=O)NCCCC2CCCN2CC2CC(F)(F)C2)CC1=O c1(C(=O)NC2CN(C(C(CCCC)O)=O)CC2SC)cc2n(n1)CCNC2=O C(C(=O)N(CC)OCC)=CC(C)NC(=O)NC(C)C(=O)NC c1(C(=O)NCC(N(C(C(c2cncc(F)c2)C)=O)C)C2CC2)cncc(O)c1 C(=O)(CCCC(=O)NC1CCCN(C(=O)COc2cnn(C)c2)C1)NCCC N1(C(c2ccc(Br)cc2CO)=O)CC2OCCN(C(C3(F)CCC3)=O)C2C1 Cc1cc(Cl)c(C(=O)NCC(CO)NC(=O)C(C)NC(N)=O)cc1[N+](=O)[O-] C(=O)(CC(C)C(=O)N1CC2C(CN(C)C(c3ccc(C)n3C)=O)C2C1)OC N(C(=NCc1cn(C(C)(C)C)nn1)N1CCc2cccc(Br)c2C1)C(C=C)C C#CC1(NC(=O)C(C2CCN(C(C3CCC3C#N)=O)C2)F)CC2CCCC12 CCC(COC)C(=O)N(C1CC(C#N)C1)CC(=O)NCC1CC(C)(C)C1 N1(C(C2(C)COC2)=O)CCOC(C)(CNC(c2cscc2C(N)=O)=O)C1 c1(C(N2CC(O)(CN(C(C3C(OCC)C3)=O)C)C2)=O)cc2ccccn2c1 c1(C(N2CC(NC(CCCC#C)=O)C(C)(C)C2)=O)ccc2c(c1)C(=O)CCC2 c1(C(N2CCCC(N(C)C(c3cnc(S)[nH]3)=O)CC2)=O)cc2nc(Cl)ccc2o1 CC1(C)CN(C(c2c[nH]nc2OCC(F)(F)F)=O)CCC1NCC(F)(F)F CCC(C(=O)NCC(C)CNC(c1cnc(C2CC2)o1)=O)NC(N)=O.O CC(O)(C(=O)N1CCC(NC(c2ccc(Cl)cn2)=O)CC(O)C1)C(F)(F)F C1(C(=O)NCC2OCCN(C(c3c(C(C)C)ncs3)=O)C2)CCCC2(CCC2)O1 N1(C(CCC(=C)C)=O)CCCC2(CCCN2C(=O)C(c2cccc(OC)c2)C)C1 CN1CCN(C(C2(CF)CCN(C(=O)C3=COCC3)C2)=O)CC1 N1(C(C2CC(n3ccnc3)C2)=O)CCN(C(C2(C(F)(F)F)CC2)=O)CC1CF Cc1cn2c(C(=O)NCC(C)N(C(=O)C(Cl)=CCl)C)c(Cl)nc2s1 N1(C(=O)Cc2sccc2Br)CC2CN(C(C3CCC4(CC3)CC4)=O)CC2C1 C1(CNC(Cc2cn(C)nc2)=O)C2CCCC1N(c1nnc(C(F)F)s1)C2 c1(CC)cc(C(N2CC3CC3C2)=O)nn1CCO.C1(=CC=O)CCN(C)C1.N C(C)(C)(C(N)C(=O)N(C(=O)CC1CCN(S(C)(=O)=O)C1)C)OC Cc1cc(C(=O)NC2CC(C)(NC(=O)CC3SC(=N)NC3=O)C2)cc(F)c1 CCCC(C(=O)NC(C)CCNC(=O)CC1(CC(=O)OC)CCCC1)OC c1(NCC2(CC#N)CC(F)(F)C2)ccnc(S(N)(=O)=O)c1 C(=O)(C1=NNC(=O)C1)N(C1CCN(C(CC(C)O)=O)CC1)CC1CCCO1 c1(N2CC(C)C(C(c3ccccc3)=O)C2)nc(=NCC2CSC2)[nH]c2c1SCC2 n1(CC(=O)NCCC2CC(N)C2)sc(=O)c2ccccc12 c1(C=O)ccc2c(c1)C(=O)NCCO2.C1(CNC(C2(SC)CC2)=O)CCC1 C1CN(C(c2cc(C(F)(F)F)ccc2C)=O)CC1(C)C.C1(CCC)(C(=O)N)CC1 c1(NC(=O)CC2(OCC)CCC2)ccc(CC(=O)NC(C)C=O)cc1.O N1(C(CCCOc2ccc(OC)cc2)=O)CC2CCC1CN2C(c1cocn1)=O C(O)(C(F)(F)F)C1(CC(=O)NC2CC(C(=O)NC3CCC3)C2)CCC1.C c1(C=O)c(C)coc1-c1ccccc1.C1CCCC1.C(C)(C(=O)NC)SCC c1(C(N2CC(CNC(c3c(OC)cncc3Br)=O)C2)=O)ccc2nccn2n1 N1(C(C(CNC(=O)CNC=O)OC)=O)CCC=C(F)C1 C=CCC(CC)C(=O)N1CCCC(O)(CN(C(=O)C(C)(C)N2CCOCC2)C)C1 CC1(C(=O)NCC2CCCC2C(=O)NCC#CC2CC2)CCCO1 CC(C)(C(=O)NCC1C=CCOC1)NC(=O)CC12CCCC1C2 CC1(C)CCC(CNC(c2ccc(O)nn2)=O)N(C(C2CC(CF)C2)=O)C1 CC(C)C(C)(CN=c1cc(-c2cccc(Cl)c2)nc[nH]1)NC(=O)C(C)CC(N)=O C1(O)(CC)CCN(Cc2cn(C3CC3)nn2)CC1.C(=O)CCCc1nc(CC)no1 N1(C(c2cccc(SCC)c2)=O)CC2CCC(C2)C1.C1(O)(C(=O)N)CCCCC1 C(=O)(CS(=O)(=O)C(C)(C)C)NC1C(C)CN(C(=O)C(F)(F)CO)C1 C(CO)(C(=O)NC(c1ccccc1)CNC(=O)Cn1cccc1)NC(N)=O C1(C(=O)NCC(C2CC2)NC(=O)COCC2CCC2)CNC(=O)C1 CC1CN(C(=O)CC(F)(F)F)CCC1N(C)CCc1cccc(Br)c1 CCC(C)C(C(=O)NCC1(C)CCOC1)NC(C1COCCC1C)=O N1(C(C#CC(C)C)=O)CCCC(O)(CNC(c2cnc(O)cc2O)=O)C1 Cc1nn(C)c2nc(NCc3cnn(CCF)c3)cc(Cl)c12 N1(C(C(C(=O)OCC)(C)C)=O)CCC2(CC1)OCCCC2.C(=O)C(C)C(F)F.N c1(C(N2C(C)(C(=O)NCC(=C3CCCCC3)F)CCC2)=O)cncc(C#N)c1 N1(C(CSCCN(C)C)=O)CC(C)C(F)C1.C1(CC(=O)N)CCCC1(F)F C12(NC(=O)CC3(O)CCCCC3)COC(C1)C(NC(=O)Cn1ncnn1)C2 S(=O)(=O)(CC(=O)N(CCCNC(C1CCC2CC12)=O)C)NC N1(C(C(=O)NC(CC)C)CC2CCCC(C)(C)C2)CCc2nc(C)ccc2C1 C1(CN(C(C(C)SC(C)C)=O)C)COCCN1C(c1ccccc1Br)=O c1(SCC(N)=O)ccccc1NC(=O)C(=O)N1CC(N2CCOCC2)C1 Cc1cc(C)c(C(=O)N(C)CCN(C(=O)C(CCN(C)C)N(C)C)C)c(N)c1 CCCCN=C(NCCN1CCCC(C)(C)C1)NCc1cnn2ccccc12 CC(C(=O)NCCCCC1CN(C(c2nn[nH]c2C(F)(F)F)=O)C1)C(C)(F)F N1(C(c2c[nH]c(=NCC=C)s2)=O)CC2CCN(C(c3cccc(Cl)c3)=O)CC2C1 C(=O)(CC(C)CC(C)C)N1CC(CC=C)(NC(=O)C(c2cn(C)nc2C)C)C1 N1(C(C(C)OCC)=O)CC2CN(C(=O)COCCO)CC2C1.c1ccccc1 C=CCC(CNC(c1cnn(CCO)c1)=O)NC(c1sccc1CO)=O N1(C(=O)OC(C)(C)C)CC(NC(=O)CCCC2CCOCC2)CC12CCC2 C1(NC(CNC(CC)=O)=O)CCC(N(C(=O)Cc2conc2C)CCO)C1 C=C(Cl)CC(C(=O)N(CC(C)(C)C#N)C)NC(=O)C(C(C)CC)N(C)C C1(CC=O)COCC2(CCC2)O1.N1(CCCC(=O)N(C)CC)C(=O)CNC1=O.N c1(CC(=O)NC2(C)CN(C(c3n(C(CC)C)ncc3)=O)C2)cncnc1O C(N=c1[nH]c(=NCC2C(C)C2C)[nH]c2c1SCC2)c1ccc(OC)c(C#N)c1 C(=O)(C(C)(C)Cc1cnn[nH]1)NCCN(C(CCC#C)=O)C.C1(C)CCCC1.N CCCCCC(F)C(=O)N1CC(C)C(C)(C(=O)NCC(C)C2CCC2)C1 n1(CC(=O)NCC2CCCCN(C(=O)C=C(Cl)Cl)C2)ccc2ccccc2c1=O c1(NC(C(=O)NCCc2cccnc2Cl)=O)cccnc1Oc1ccccc1F S(=O)(=O)(c1ccc(N2CCC(c3ccccc3)C2)c(F)c1)NCC(C)C#N C(=O)(C(C(C)C)N1CCCCC1)NC(C1N(C(C=CC=CC)=O)CCC1)C C(=O)(C(F)C(C)C(F)(F)F)N(CCNC(CCCC(C)C)=O)CCOCCO c1(CNC(=O)C(=O)NC2CC2)ccc(F)cc1.c1(C(=O)N)cc(Cl)ccn1 C(CCCCC(=O)NC(CNC(c1sccc1Cl)=O)(CC)CC)=CC c1(OCC)ccc(C(=O)N)cc1.c1(N2CCC(CC)C2)cc(C(C)(C)C)ncn1 c1(OC)cc(Cl)ccc1N1CCN(C(=O)NCC2(C)CCCC2(F)F)CC1 Nc1cc(F)c(C(=O)NCCOCCNC(c2n[nH]cc2F)=O)cc1F N1(C(C(COC)N(C)C)=O)CC(O)(C2(CNC(c3ccncc3Cl)=O)CC2)C1 Cc1cccc(CC(=O)NC2CCCC2C(=O)Nc2ccnc(F)c2)n1 c1(C(N2CCC(CNC(CCCC#C)=O)C2)=O)n[nH]c2ccc(C(=O)OC)cc12 Cc1nc2c([nH]1)CC(C(=O)NCc1ccc(N(C)C)s1)CC2 c1(OC)nn(C)cc1C(=O)NCC1CCN(C(c2ccc(=N)[nH]c2)=O)C1 c1(-c2cc(C)sc2C)ccc2[nH]c(C(=O)NC3CCCC(O)C3)cc2n1 CC(C)C(O)C(=O)NCC(O)CNC(c1ccccc1)=O.CCCOC(F)F.O N1(C(CCOCCN(C(CCC=C(C)C)=O)C)=O)CCC(F)(F)C1 N1(C(C(C)NC(C)(C)C)=O)CCC2(CCC2)C(C)C1.C1(C=O)(C=O)CC1 C=CC(C)CC(=O)N1CCCCC1CCCNC(=O)Cc1ccc(C(N)=O)cc1 C(CCCC(=O)NC)N(C(C1N(C(c2c(OC)ccs2)=O)CC1)=O)C c1(C(=O)NC2C(NC(c3c(C)nn[nH]3)=O)CCC2)cnn2cc(C(N)=O)cnc12 CC(C)C(CC(=O)N(C(C)CCNC(=O)CC1CCSCC1)C)C(C)C Cc1cc(C(N2CCCC2CC(=O)NCC23CCN(C2)C3)=O)cnc1Cl N1(C(C(C2CCOC2)NC(c2c(C)noc2)=O)=O)CCCC(CCO)C1 c1(C(=O)NC(CNC(CCc2n(C)ccn2)=O)(C)C)coc2c1CSC2 CC1=C(C(=O)N2CC(CC(F)C(=O)NCc3nc(O)ccc3C)C2)CCC1 CON(CCC(=O)N1CC2CC1CN2C(C)=O)C(=O)c1ncnc(O)c1F c1(C(N2CC(F)(C(N3CCCC(CC=C)C3)=O)C2)=O)cc(F)ccc1O n1(CCCN(C)C)cc(CN(C(=O)CC2CC2)CCO)nn1 C1(CC(=O)OC(CC)C(C)=O)CC2(CC2)CO1 c1(SC)cccnc1C(=O)NCC(C1CC1)N(C(=O)C(F)C1CCOC1)C C1(CC(=O)N(CC(=O)O)CC)C=CC(NC(c2cc(CO)[nH]n2)=O)C1 C1(C(=O)NCC2CC(NC(CCC(=O)NC)=O)C2)CCCC2(CCOC2)O1 C1(C(=O)NC(C(C)SC)C)CC2CCC1N2C(=O)Cc1nonc1C c1(CSCC)ccc(C(=O)N)cc1.C1(O)(CC)CCN(C(=O)C=C(Cl)Cl)C1 C1(NC(CNC(C)=O)=O)CCCC12CCN(C(=O)CCc1nc(=N)[nH][nH]1)C2 N#Cc1ccccc1CNC(C1CC(F)(F)CN1C(c1cc(Cl)ccc1F)=O)=O c1(C(=O)OC)cscc1S(=O)(=O)NC(=O)CCc1ccc(Cl)cc1Cl C#CCC(CC(F)F)C(=O)N1CCC(CCC(=O)NC(c2nnc(C)s2)C)C1 N1(C(CS(CC)(=O)=O)=O)CCC(NC(C2CCCS(=O)(=O)C2)=O)CC(O)C1 C(C(F)(C(=O)N)C(C)C)NC(c1oc(CC)c(C)c1)=O.c1(CC)ccc(O)cc1 C1(CC(N2CC(N(C(C3C(OCC)C3)=O)CC)C2)=O)CCC(=O)N1 c1(C(N(CC(CC)NC(=O)CCC(=O)OC)C)=O)cc(Cl)ccc1Br c1(NC(=O)C(N2CCCN(CCO)CC2)=O)ccc2ccccc2c1Br C1(CN(C=O)Cc2ccc(C)cc2)CC(F)(F)CC1O.C(CCO)c1ccco1.N CCCCC(C(=O)NC1CN(C(=O)CC2CN(C)C2)CCC1F)NC(N)=O C=C(C)CC(C(=O)NC(COC)CC(=O)NCC1CC(C(=O)O)C1)OC [SH](=O)(=O)c1ccccc1Cl.C(C=O)=CC=C.C(=O)(C)N(CC)C(C)C.CC c1(C(=O)NC2C(NC(C3(O)CC(C)(C)C3)=O)CCCC2)ccc2ccsc2c1 CCC(CC)C(C(=O)N(C)CC1CN(C(c2snnc2C)=O)CC12CC2)OC C=C(C)CC(C(=O)N=c1[nH]n(CCOC)cc1C)NC(c1ccccc1)=O C1CC2(CC2)CN1C(c1cscc1)=O.C1(C(=O)N)(COC)CC1(F)F.C c1(C(=O)NCC(=O)NC(Cc2cc(Cl)sc2Cl)C(=O)O)cc2ccccc2[nH]1 c1(C(N2C(CN(c3nn4cc(C)nc4s3)C)CCC2)=O)c(C)cccc1[N+](=O)[O-] CC1C(NC(c2c[nH]nc2C2CC2)=O)C(C)CCN1C(c1ccc(CO)cc1)=O CN1CC(C)(C)CC1C(N1CCCC(C)(CNC(C2(CO)CCC2)=O)C1)=O C(=O)C(C)CCC(C)(C)C.N1(C(C2CN(C(C)=O)C2)=O)CC(C)C(C)(C)C1.N C1CCCO1.c1(C(CC)NC(=O)CN(C(=O)CO)C2CC2)cc[nH]n1.C N1(CC23CCC(C(=O)OC)(CC2)OC3)CC(=O)N2CCOCC2(CO)C1 Cc1cc(C(=O)NCC2CCN(Cc3sc(Cl)nc3Cl)C2)cc(C)c1F Cc1cc(C(=O)NC(C)CN(C)C(C2CC23CCSCC3)=O)c2ncccc2c1 O=S(=O)(c1ccc(N2CCCC(OC3CCC3)C2)nc1)N1CC2CC3CC2C1C3 c1(C(N2CC(C(N)=O)C2)=O)nc(C)c(N)cc1C.Cc1csc(C(=O)NC)c1 c1(C(C(=O)NCCSC)N(C)C)cccc(-c2cnco2)c1.c1cccc(Br)c1 C1(CN(C(=O)C(C)COC)CC)CCCN(C(c2cc(C(F)F)no2)=O)C1 n1(-c2cnc(C)s2)nc(-c2cccs2)nc1C1CCCN1C C1(NC(c2cc(CC)no2)=O)CC(OC)CN(C(C2CC2F)=O)C1 C(C)(C(=O)N1CCC(C(N2CCOCC2C(=O)OC)=O)C1)(C(C)C)OC C(=O)(C1=CSCS1)NCC(C)N(C(=O)Cc1ccc(Cl)nc1)C c1(C(=O)NCC2C(NC(c3c(C)c[nH]n3)=O)CCCC2)ccc2c(c1)COB2O CC(C)CC(C)CC(=O)NCC1CC2(CC2)CN1C(=O)CCC(C)(C)C#N CC1(C)NC(=O)CC1C(=O)NC1CCCCC1C(=O)N.c1cc(F)ccc1F.C C(CC(C)(C)NC(=O)CN1CC=CC1)NC(CNC(C1C(C)C1)=O)=O N1(C(C2(C)CSC2)=O)CCC(CC(N2CCCC(CCF)C2)=O)CC1 N1(S(Cc2ccc(C)cc2)(=O)=O)CCC(NC(=O)Cc2noc(C)n2)C(F)C1 C#CC1(C(=O)NC2CC3(C2)CC(C)C3)CCN(C(C2CC2(F)Cl)=O)CC1 Cc1ccc(C(N)=O)cc1C(=O)NC1CN(C(c2cccc[n+]2[O-])=O)CC1C N1(C(=O)C=CC2CCOC2)CCC2(CCCN2C(=O)C=C2CCOCC2)C1 c1(SCC)cc(C)ccc1NC(N1CCCC2C(C(F)(F)F)C12)=O C(c1cc(Br)ccc1OC(C)C)=Cc1onc(-c2c(C)cc(C)nc2)n1 c1(C(=O)NC2CCN(C(c3c(N)c(Cl)ccc3)=O)C23CC3)nccn2nccc12 CC1c2nccn2CCN1C(=O)C(N1CCN(C)C(c2ncc[nH]2)C1)=O C(=O)(C1CCC(=O)Nc2ccccc21)N1CC(NC(c2c(OCC)scc2)=O)C1 c1(C(N2CCC(C)(C)C2)=O)coc(S(C)(=O)=O)c1.n1(CC)cc(C(=O)N)cn1 n1(CC)nncc1C(=O)NC1CC1CNC(=O)C(C)OC CC1Cc2c[nH]nc2C(C(=O)NC2(C)CCN(C(=O)COc3ccsn3)CC2)C1 c1(C(=O)NC(C2CN(c3ccc([N+](=O)[O-])cc3)C2)C)ccc2nn[nH]c2c1 N1(C(=O)NCc2c(C#C)cc(F)cc2)CCCC2(CCNC2=O)C1 CC1CCCN(CCCCNC(=O)C(=O)NC2CC(O)(CCC(C)(C)C)C2)C1 c1(N2CCC(C)C2CNC(=O)CS)cc(C#N)nc(C2CC2)n1.c1nncn1C c1(C(=O)NC2C(C)CN(C(=O)Cc3ccsc3)CC2)ccc2c(n1)CCC2 c1(C(=O)NC2CCCN(C(C(CC#C)C3CC3)=O)C2)cnn2cccnc12 c1(C(=O)NC(C(C)NC(CCN(C(C)=O)C)=O)C(C)C)cn(C)c2ccccc12 N1(C(C2CN(C(C)C)C2)=O)CCC(C)(C)C(C(N2CCC(CN(C)C)C2)=O)C1 C1(c2c(OC)cccc2)CCCCCN1C(=O)Cc1ccc(O)cc1OC C(c1cc(Cl)ccc1O)=CC(N1CCCCC(NC(C2N(CC)CC2)=O)C1)=O N1(C(C=NOC)=O)CC(CNC(=O)CCC2CC2(F)F)C(c2ccnn2C)C1 C1(C(=O)NC2CCN(CCn3cccn3)C2)CCC(C2CC2)CC1 CCC(CO)C(=O)NCC(C1CC1)N(C)C(c1ccccc1OC1CC1)=O C=CCC(CC)C(=O)N1CCC(NC(c2cnn(C)c2)=O)C1C N1(C(C2N(C)CCCC2)=O)CCCN(C(c2cccc3c2OCO3)=O)CC1CO C1(C(N2CC(O)C(F)C2)=O)(CC)CCN(C(c2cn(C)nc2C)=O)CC1 c1(C(=O)NCC(C(C)C)NC(CSCC#C)=O)cccc2nc(C)sc12 C1(C)(C(N2CC(NC(Cc3c(C)ccnc3)=O)(CO)C2)=O)CC2CCC1C2 C1(C(N2CC(OC)(C)C2)=O)CSc2ccccc2O1.C1(C=O)CC(=O)N(C)C1.N CCC(C)(CO)C(=O)NCCCC(=O)N(C1CCCCC1CO)C C(=O)(C1CCOc2ccccc21)NCC(C)NC(c1ccccc1OCC#N)=O CC(C)=CC=O.C1(CCCC)CC1.N(CCN(CC)OC)CC.OC N1(C(C2CC(=O)NC2)=O)CCC2(CCCN(Cc3cc(Cl)ncc3Br)C2)C1 N1(C(CCc2cnc(C)s2)=O)CCCC(N(C)C(C2CCN(C)C(=O)C2)=O)CC1 C(=O)(C(O)CCNC(C1CCC(=O)C1)=O)NC1(c2nc(C)[nH]n2)CC1 N1(C(c2ccc(SCC)nc2)=O)CC(NC(=O)C(C)(F)CC)CC1(C)C C1(NC(C2CC(F)C2)=O)CC(N=c2[nH]c3ccc([N+](=O)[O-])cc3s2)C1 C#CC1CCCCN1C(=O)CCC1CCCN(C(=O)CC2CCCC3CC23)C1 C1(F)(CNC(=O)C2=COCCO2)COCCN(C(=O)CCC2CCOC2)C1 C1(C(=O)NC(C(COC)C)C)C2CC3C(C2)C13.C(=O)CCCn1ccnc1.N N1(C(C2C(C)N(C(=O)Cc3cnsc3)CC2)=O)CCC(O)CC1CO C1(NC(c2n(CC#C)ccc2)=O)CCOC2(CCN(C(=O)C(O)C=C)CC2)C1 n1(C(C(=O)NC2CN(C(c3nc(C)oc3)=O)C2)C)nc(C)c([N+](=O)[O-])c1C n1(CC)nc(C(=O)N(C2(C(=O)NC3CC4CC4C3)CCC2)C2CC2)cc1O C1(C(C)NC(=O)CC)CCCN(C)C1.C(=O)(C(C)(C)c1ccno1)N(CC)C CCCCC(O)C(=O)N1CCC(O)(CC(=O)Nc2c(CO)cccc2Cl)CC1 Cc1ccc(C(N2CC(NC(=O)COC(F)(F)F)C(C)(C)C2)=O)nc1O c1(CC(=O)NC(CC)CN(C)C(c2ccsc2C(F)F)=O)ccc(C)cc1C Cc1cc(CNC(=O)COC2CCN(C(=O)C=CC(C)C)C2)cc(O)n1 CC(C)C(C(=O)NC1CCN(C(=O)CSCC2CCCO2)CC1)NC=O C1(CNS(C(C)C)(=O)=O)CN(C(C2CC=CC(n3cc(C)nn3)C2)=O)CCO1 C1CCCCN1C(=O)Cc1nnn(C(C)(C)C)n1.Cc1cc(C(=O)N(C)C)sn1 N1(C(C(C=CC)O)=O)CC(NC(c2cncc3c2CCCC3)=O)CC2(CCC2)C1 CCC(O)(CNC(=O)C(C)C(C)NC(=O)CSc1nc[nH]n1)CC N1(C(c2ccn(C(C)C)n2)=O)CC(C2CCCCN(C(=O)Cc3nccs3)C2)C1 C=CC1(C(=O)NC)CCN(C(c2cccn2C2CC2)=O)C1.C1CC1.C1CC1 CC(C)CCCC(=O)NC(C)(CNC(c1ccc(C(O)CF)cc1)=O)C1CCC1 Cc1c(C(N2CCN(C)CC2CNC(=O)CCS(C)(=O)=O)=O)cccc1Cl C(CC(C(=O)NCC(O)CCOC)NC(c1csc(F)c1)=O)=CC c1(OC)cc(=O)n(C)cc1C(N1CCC(C)C1)=O.C(c1ccccc1)=CC=O c1(CNC(C2C(OC)CN(C(C3CC34CCCC4)=O)C2)=O)ccc(F)nc1F C(CC1CCOCC1)(C(=O)NCCCC1CCOC1)NC(CSCC)=O CCCC(CC)CCC(=O)NC(CN(C)C)C(=O)N1CCC(OCC2CC2)C1 N1(C(c2c(C)cc(C)o2)=O)CC2CC(C1)C2NC(=O)C=CCCC(C)C c1(CC)ccc(C(=O)NC)cn1.C1(C)(C=O)CCCN1C(C)=O.C1CCC1 c1(OCC)ccc2cc(CSCc3nnc(O)n3C)ccc2c1 c1(C(=O)NCC(CO)NC(C(C2CC(C)(C)C2)OC)=O)ccc2nccn2c1 CCCC(C(=O)NC(CCC1CCC1)C(=O)N(CC(C)C)C)NC(N)=O.OC c1(CNC(C2(CC=C)CC2)=O)cc(C(N2CCC2(C)COC)=O)ccn1 CS(=O)c1ccc(CC(=O)Nc2cccc(NC(c3ccsc3)=O)c2)cc1 C(=O)(C1CCCc2nncn21)NC1C(CNC(c2cccc(F)c2Cl)=O)COC1 C=CC(C)(C)CC(=O)N1CCC(CCNC(C2(CC)CCCO2)=O)C1 c1(C(N2CC3N(c4cc(OC)ncn4)C3C2)=O)ccc(Cl)nc1OC c1(C(N2C(c3nc(C)c(C)[nH]3)CC(OC)C2)=O)cc2ncnc(O)c2cc1Cl CC(CS(C)(=O)=O)C(=O)N1CCC12CN(C(c1[nH]nc3ncccc13)=O)C2 C1(NC(=O)Cn2cc(CNC(c3ccc(F)cc3)=O)nn2)CC2CCCC12.C c1(C(N(CC)C(C)C)=O)n[nH]c2cccnc12.c1(CC)cc(C=O)cc(F)c1.N CC1CCCCN1CCC(=O)N.c1(C(N(CC)C2CC2)=O)ccc(C2CCOC2)s1 CCC(CCOC)C(=O)N(CCCN(C)C(C12CC3CC1C2C3)=O)C c1(CC(=O)NC2CN(C(C(CCCC)O)=O)CC(F)C2)cn(C)c2ccccc12 C1CN(C(C2CCN(C(C)=O)C2)=O)CC12CC2.C#Cc1cnn(CC(=O)NC)c1 N1(C(c2cc(C)c(F)cn2)=O)CC(C2CCCN(C(=O)C(O)CCC(C)C)C2)C1 C1(NC(CC(COC)COC)=O)CN(C(=O)CCc2ccn(C)n2)CC1C1CC1 c1(C(N(C2CN(C(=O)CC3C=CCC3)C2)C)=O)cc(F)c(F)c(Cl)c1F N1(C(c2c(CC=C)cccc2)=O)CC2(C1)CN(C(=O)CC1CCCCN1C)C2 C(CC(C(=O)N1CCC(C(C)(C)NC(=O)Cc2csc(C)c2)C1)OC)OC C1(C(=O)NCC(CNC(CCCC=C)=O)C(F)(F)F)CC2CCC(C1)S2(=O)=O N1(C(C=CCOC)=O)CCC2(C1)CN(c1nccc(-c3cnccn3)n1)C2 c1(C(=O)N)cc2cc(C)c(Cl)cc2[nH]1.C(CCCC(=O)NC(C)(C)C1CC1)SC C1(C2CC2)(C(N2CC(C)(NC(C3CCC(C)(CC)O3)=O)C2)=O)CC=CC1 CCCCC(CC)CC(CC)(c1nnnn1CC(F)F)NCc1cc(CC)on1 c1(OC)cc(C(N2CC(C)CC2(C)C)=O)cc(C2CC2)c1.C1(C=O)CN(C)C1 Cc1ccc(OCCC(=O)NC2CN(C(=O)C(C)(F)F)CCC2C)c(C)c1 C(=O)(CC1=CCN(C(=O)C(C)S(N)(=O)=O)CC1)N1CC2CC(OCC)C2C1 c1(C(N(C2CCCN(C(COCC#C)=O)CC2)CC)=O)cc(C)cc2nc[nH]c12 S(=O)(=O)(C1CC2CCC1CC2)N(C1CC2CC1C1CCCC21)C(=O)CC(O)CCO c1(CNC(=O)Cc2nccs2)ccccc1-n1cc(-c2nccs2)nn1 N1(C(C2(CC)CCCO2)=O)CCC(NC(c2cc(C)sn2)=O)CC(C)(C)C1 CC(C)(C)C1=NOC(C(N2CC(NC(=O)CO)CC2(C)C)=O)C1.c1nc[nH]n1 c1(C(N2CCC(NC(c3c(CC)cc(C)cc3)=O)C2)=O)cnc2ccc(C)cn12 C1(NC(C2(CCC=C)CN(C(=O)CCC=C(C)C)C2)=O)CN(C)NC1=O N1(C(CSCCC(C)C)=O)CCC(F)(CNC(c2nncs2)=O)CC1 C1(C)(CNC(C(C#C)(C)C)=O)CC(F)(F)CN1C(C1C=CCCC1)=O C1(C(C(=O)N(CCN(C)C)CCO)F)CCN(C(c2nccs2)=O)C1 C1(C(C)(C)C)CCN(C(C2CCCC2NC(c2c[nH]c(=S)cn2)=O)=O)CC1 c1(C(=O)NC2CCN(C(c3cc(C)c(C)s3)=O)CC2F)ncnc2sccc12 C(CN(C)C(C1CCCN1C)=O)(CO)(CO)NC(C(COC)C)=O Cn1ccc(C(=O)NC(CO)CCCNC(=O)CC2NC(=O)NC2=O)cc1=O Cc1ccc(C(C(=O)NC(C)C)N2CCC2c2cccc(Cl)c2)c2ncccc12 c1(C(N2C(C)CCC(CNC(=O)C=CC=C(Cl)Cl)C2)=O)n[nH]c2c1CSCC2 Cc1cc(C(=O)NCc2cn(CC3OCCC3C)nn2)cc(N2CCCCC2)c1 C(C(C)C(F)C(=O)NCC(=O)NC(C)(C)C)NC(COCC#C)=O c1(C(N2CC(CC(=O)Nc3c(C)c(Br)ncc3)C2)=O)c[nH]c2cc(Cl)ccc12 N1(C(C(CC)(C)OC)=O)CCC2CCC(C1)N2C(c1cnccc1C)=O c1(COC)ccnc(C(C(=O)NCC2CCOC2)N(C)Cc2ccco2)c1 CC1CC(C(N2CCN(C(C3CCSC(C)C3)=O)CC2CCO)=O)CC(C)C1 C1(C(N2CC(CNC(C3CCC3)=O)CC23CCC3)=O)CCC2(CCCC2)CC1 C(=O)(C1=Cc2ccccc2C1O)N1CCC(C)(NC(c2ccc(NC)cn2)=O)C1 C(c1ccc(F)cc1)=CCC(=O)N(CCCN(C(C1(C)C(CC)CCC1)=O)C)C C1(O)(CC(=O)NCC(C)(C2CCC2)NC(=O)CCN2CCC2)CCOCC1 CN1CC(C)(C(N2CC(NC(=O)CN=S(C)(C)=O)C2)=O)CCC1=O C1CC12CCN(C(=O)CN1CCCC1=O)C2.c1(OC)ccc(C=CC(=O)O)cc1 N1(C(COCC)=O)CC2(CCOCC2)CC1CNC(c1c[nH]c2nccc-2c1)=O C1(CC)CC(C(N2CCOC(CNC(=O)C(c3ccncc3)C)C2)=O)CCC1=O S(=O)(=O)(c1cnc(NC2CCn3nccc3C2)cc1C)NCC(CC=C)(C)CO c1(C(N(C(C)C=O)CCN(CC)CC)=O)cc(C=O)cc(C(C)C)c1 C1(CC=C)(C(=O)NC(c2ccccn2)CC)CCCN1C(c1ccncn1)=O c1(C(=O)OC)cnc(C(=O)N(C)CC2CCCN2C(=O)C=CS(C)=O)cn1 C(=O)(C1=NOC(CNC(c2cnn3c2OCC3)=O)C1)N(C(CSC)C)C C(C1CS(=O)(=O)c2ccccc21)NC(N1CCOCC1CCO)=O C1(CNC(CCC=CC(C)C)=O)CC(C(=O)NCCC2CC2C)=NO1 Cc1cnc(NCc2cc(-c3ccco3)on2)c(S(=O)(=O)NC2CCCC2O)c1 Cc1ncc(C(=O)N(C)CCOCCN(C)C(C2(Br)CC2(C)C)=O)o1 C(=O)(C1CC(=O)c2ccccc21)NC1CCN(C(c2ccc(C#C)c(F)c2)=O)C1 c1(C(N2CC=CC2)=O)cc2ccsc2s1.c1(C(=O)N)ccc(C(F)F)c(F)c1.C Cc1c(Br)cnc(NC(C2CC23CN(C(c2ccc(Cl)cn2)=O)C3)=O)c1[N+](=O)[O-] N1(Cc2c(OC)ccc(Br)c2)CCC2(CC1)CC2C(=O)Nc1ccnc(C#N)c1 C1(NC(c2n(C)ccc2)=O)CN(C(=O)Cc2cnsc2)C2(CCOCC2)C1 c1(C(N(C2CN(C(c3ns[nH]c3=O)=O)CC2(C)C)C)=O)c(O)nnc2c1CCC2 C1CS(=O)(=O)C2CN(C(C3CC3(F)F)=O)CC12.c1(C(C)(C)C)cc(C=O)[nH]n1 c1(C(=O)NC(C(CO)NC(c2nc(C)[nH]n2)=O)C)cc2ccc(Br)cc2o1 C(N=c1nc(-c2cc(Br)cc(Br)c2)[nH]o1)C1(CN)CCOCC1 C1(F)(CNC(C=CCCC)=O)CC(NC(c2cnn(C)c2)=O)C1 CCC(CC)C(F)C(=O)N1CC(C(N2CC(CO)CC2(C)C)=O)C2(CCC2)C1 c1(C(N2CC(O)(CCNC(C3CC(OC)C3)=O)C2)=O)ccc2[nH]c(C)cc2c1 N1(C(Cn2c(C)cc(C)n2)=O)CC2ON=C(CNC(c3n[nH]c(C)c3Cl)=O)C2C1 C1(COC)CN(C(=O)Cc2cc(Cl)ccc2Cl)CCN1C(C1CC(C)(F)C1)=O CC1CCN(C(c2cccc(=O)n2O)=O)C(C)C1NC(c1ccn(C)n1)=O N1(C(C(C)SCC)=O)CCC2(CCCN(C(c3cnc(Cl)cc3Cl)=O)C2)CC1 C1(C(=O)Nc2n(C(C)C)ncc2)CCC2(CN(C(c3cccc(F)c3Br)=O)C2)O1 N1(C(C(C)OC)=O)CCCC2C1CCCCN2C(c1ccc2c(c1)OCO2)=O C1(C(=O)NC(COC)COC)CCCN1NC(=O)C1CCCSC1C N1(C(C(c2cn(C)nc2)O)=O)CC=C(C(=O)NCC(CO)N(C)C)C1 N1(C(c2sccc2F)=O)CCCC(C2CCN(C(=O)C(F)(F)C3CC3)C2)C1 c1(CC(=O)NC2CCCN(c3ccc(C)cn3)C2)ccn2cncc2c1 C1(NC(=O)CC2CC2)CCc2onc(C=O)c2C1.N1(N2CCOCC2)CCCCC1 CN1C2CCC1CN(C(=O)CC1CC(NC(C34CCC(CC3)CC4)=O)C1)C2 C1(C)(C(=O)NCC)CCCN(C(c2ccc(OC(C)C)cc2)=O)C1 c1(OCC)ccc(Cl)cc1.C1(CC=O)CN(C(=O)CC(C)(C)C)CC12CC2.C N1(C(=O)Cc2coc(CNC(c3cscn3)CO)n2)CCC2CC12C(=O)O Cc1cc(C(N2CCCC(CN(C(=O)CC(C)C(C)C)C)C2)=O)cnc1C(F)F Cc1cn2ccnc(C(N3CC(NC(=O)CC4(C)CCCO4)C(C)(C)C3)=O)c2n1 N#Cc1cc(C(N2CCCCC2CNC(c2cccc(OC(F)F)n2)=O)=O)c[nH]1 c1(NC(CC(CNC(c2c(C(C)C)c[nH]c2)=O)C)=O)cncc(C#N)c1 C1(CC(=O)NC(C2CCCCS2)C)(NC(=O)CC2(O)CCC2)CCCCC1 c1(C(C)(C)C)nc(CC(=O)N(CCCNC(=O)CCc2cnco2)CCO)cs1 C(=O)(C(CC(=C)C)NC(=O)CNC(C)=O)Nc1c(C#C)c[nH]n1 C1(C(N(C)CC2(NC(CSCC)=O)CC2)=O)CCc2nc(O)[nH]c2C1 C#CCCCC(C)C(=O)NCCCN(C(=O)C=Cc1cc(Cl)sc1Cl)C N1(C(c2onc(C)c2C)=O)CC(=O)NC2CN(C(=O)C(C)n3cccn3)CCC12 CCC(CC)CCC(=O)NC1C2CCC(C2)C1C(=O)N(OCC)C(C)C c1(CCCC=C)ccc(C(=O)NCC(C)N(C(=O)COCCC)CC)cc1 C1(C(=O)NCC2CCOC2)(CNC(C2C=CC=CC=C2)=O)CC12CCC2 C(CC(C(=O)NCCCC1CCOCC1)NC(C1CC(C2CC2)C1)=O)OC Cc1cnsc1C(=O)NCCC1CCN(C(C2(C)COC2)=O)C1 C(CCC(C)N=c1[nH]c(=NC2CC3(CCOC3)C2)[nH]c2c1SCC2)=C(C)C c1(C(=O)NC2CN(C(C3(CCC)CCC3)=O)CC23CC3)cnc2ccncc2c1 N1(CCN(C(CSCCCC)=O)C)CCN(C(=O)C(F)(F)C2CC2)CC1 c1(C(=O)NCCN(C(=O)COC(C)=O)CC)ccnc(CO)c1 C(=O)(C(F)(F)CCn1cccn1)NCC(CCNC(COC(CC)C)=O)O C1(COC)CCN(C(=O)CN2CCOCC2=O)CC1.C1(N=[N+]=[N-])(C=O)CC1.C O=C(CC1=CSC2=NCCN12)N1CCc2sc(Br)cc2C1 CON=Cc1ccc(C(=O)NC2(CF)CCN(c3ccc([N+](=O)[O-])cn3)C2)cc1 c1(C(N2CC(n3cc(COCC)nn3)C(O)C2)=O)cc(C)n(C2CCOC2)c1C C1(C(C)(C)C)NC(=O)C2=C1N(CC1CC1)C(=S)NC2c1ccnc(F)c1 c1(C(=O)NC2C(C(N(CC#C)CCO)=O)CCCC2)ncn2c1CCC2 c1(C(=O)NC(CNC(C2(COC)CCC2)=O)CCOC)ccc(C)nc1 Cc1nc(C2CC2)nc(O)c1C(=O)NC1CC(C)CN(C(c2cc(Cl)cs2)=O)C1 C(=O)(C1=CS(=O)CCC1)N1CC2(CN(C(c3c(F)ccc(N(C)C)c3)=O)C2)C1 N1(C(C(CC)(C)C)=O)CCN(C(=O)C(F)=C(C)C)CC1c1nccn1C Cc1cc(C)c(C(N2CCC(N(CCO)C(c3nnc(S)n3C)=O)C2)=O)s1 CC1OC2(C)CC1C2.C12(C(=O)N)CCOC(C)(C1)C2.C(=O)C=O.CC(F)F N1(C(Cc2c(OC)ccc(C)c2)=O)CC(C)(C)OC2(C1)CN(C(=O)C(C)CO)C2 c1(C(=O)NCC2(C(C)NC(C(CC)C)=O)CC2)cccc2nccnc12 CN1CCOCC1C(N1CCC1CNC(c1sccc1-n1ccnn1)=O)=O C1(NC(Cc2ncc(C)[nH]2)=O)CN(C(c2c[nH]nc2-c2ccco2)=O)CC1(C)C c1(C2(C)CC2)ccc(C(N2CC(CC(C)NC(c3nccnc3Cl)=O)C2)=O)cc1 c1(C(N2CC(CCOC)N(C(C3C4CCCC34)=O)CC2)=O)cn(C)c(=O)nc1O N1(C(c2c(OC)c(Cl)ccc2)=O)CCC2(CC(NC(C3(F)CC3)=O)C2)C1 C1(C(=O)NCCC2CN(C(c3n[nH]c(C)c3Cl)=O)C2)CCC(C)NC1=O C1(C(=O)NC(C2CCCN2C(=O)CS)C)CCOC2(CCC2)C1.c1cscn1 N1(C(C)=O)CCCCC1CCNC(=O)Cc1nnc(C2CC2)s1 N1(C(c2n(CC)ccn2)=O)CCC(CNC(c2nc(C)nn2C)=O)C(O)C1 CCC(CC(=O)N1CC2(CCC2)CC1C(=O)NC(CC(C)C)C(=O)NC)C(C)C c1(CC)cn2c(n1)CCC(C(=O)NCC(C)(O)C)C2.c1(CC=O)ccoc1.N N1(C(=O)NC(C)CCC2CC2)CCN2C3CCC(C3)C2C1 CCC(CC)(CO)C(=O)NCC(C)CC(C)C.N1(CC(=O)N)CC(=O)N(C)C1=O c1(C(=O)NCC2N(C(C=Cc3c(C)coc3C)=O)CC2)ccn2c(O)nnc2c1 CCC(O)C(=O)NCC1CC(F)(CNC(=O)Cc2csnc2C)C1 C1(NC(c2nccc(C)n2)=O)COCCN(C(=O)C(C(C)C)n2ccnc2)C1 CCC(CN(C)C)CC(=O)N(C1CCN(C(=O)CCc2c(C)noc2C)C1)C n1(CCCOCC)c(N2CCS(=O)CC2)nnc1Cc1cccc(F)c1 C(CC(C(=O)NOC(c1ccccc1)C)NC(C1CC12CCC2)=O)=CC c1(C(=O)NCC(CC)CC)ncc(Br)cc1C(F)F.C(C)(C(C)C)=CC=O C1CCN(C(c2coc(C(F)F)c2)=O)CC1.c1(C(=O)NCCC)coc(O)n1.O C1(CN(C(c2ncc(OC)cn2)=O)C)CN(C(c2cccc(C)c2)=O)CC12CC2 CC(C)C(O)C(C)C(=O)NC1CCCC(NC(c2cncnc2C2CC2)=O)C1 C(CC(C)C(=O)NCC(CC(=O)NCCOCCC)OC)=CCC N1(C(CC)=O)CC(C)OC(C)(C)C1C.C(=O)(CC=O)N(CC=C)C.C(C)(C)C c1(N(C)Cc2c(C(C)C)cccc2)nc(N(CCCF)C)c2c(F)cccc2n1 Cc1cc2c[nH]nc2c(C(=O)N(C)CC2CCCN2C(C23CC(F)C2C3)=O)c1N C1(NC(C2C(=C)CC2)=O)CC(Nc2ncc(I)cn2)C1(C)C c1(N(CCCCCC=C)C)ncc(S(=O)(=O)NCC(CC(C)C)N(C)C)cc1Cl N1(C(Cc2c(C)cccn2)=O)CC2(CC(CNC(c3cccn3C)=O)C2)C1 c1(C(=O)NCC(CNC(C(C)(C)c2cc[nH]n2)=O)F)cccc(=O)o1 C1(CNC(CN(C)CC)=O)CCCCC1NC(=O)C(c1ccccc1)SC c1(C2C(C(=O)NC(C)(C)CCC3CCCC3)C2)cn(CCCC(=O)OC)nn1 c1(C(=O)NC2(C(=O)NC3CN(C)CC3O)CCC2)cc(O)cc(F)c1 C1(C(N(CC(CC)NC(c2cccc(Br)c2F)=O)C)=O)CCCCC(=O)N1 CC(CC(F)F)C(=O)NCCCOCCCNC(=O)Cn1cccn1 C=CCC(CC(F)F)C(=O)N1CCC(C(F)F)(CNC(c2cc(CO)on2)=O)C1 N1(C(C(CC(C)C)NC(c2cncc(Cl)c2)=O)=O)CCc2ncncc2C1 c1(C(N(CCC(C)NC(C(C(C)C)O)=O)C)=O)cc(F)cc2cnccc12 C1(CC(=O)NCCC(C)NC(CCCc2onc(C)n2)=O)CCCCCC1(F)F C1(OC)(CNC(=O)C=C2CCC2)CCN(C(c2cc(S)ccc2C)=O)CC1 c1(C(=O)NCC(CNC(C(CC)COC)=O)O)cnc2c(ccn2C)c1 N1(C(C(COC)N(C)C)=O)CCOCC(NC(c2nc(C3CC3)cs2)=O)C1 C1(C=O)CCCCC1P(C)(C)=O.c1(C(=O)NCCC)cc(C2(Cl)CC2)n(C)n1 N1(C(C=C2CCC(C)C2)=O)CC(NC(=O)C2=CCOCC2)CC2(CC2)C1 N1(C(CCC2(C)CC2)=O)CCCCC1C(=O)Nc1cn(CC2CCOCC2)nn1 N1(C(CCn2cc(C(=O)CN(CC)CC)nn2)=O)CCCCC2CCCCC12 c1ncnc2c1cnn2C(C)(C)C.CC(CNC(=O)CCO)C.CCN(C)C c1(C(=O)NCC=CC(=O)NC2C(C)CCCCC2)c[nH]c2ncccc12 Cc1cccc2[nH]cc(CC(=O)NC(CCNC(=O)C(CO)C(C)C)C(C)C)c12 CCCC(O)CC(=O)NCC(F)CNC(c1ccc(C)nn1)=O c1(C(N2CCC(CC)C2C)C(=O)NCCCSC)cc(C(F)(F)F)cc(Br)n1 C1(C(=O)N)CC12CCC2.c1ccc(CN(C)CC)o1.C(C)(C)C.C=O.C C(c1nccs1)=CC(=O)NC(C1(O)CN(C(c2cc(F)n[nH]2)=O)C1)C N1(C(C2(C#N)CC2C(F)(F)F)=O)CC2CC(NC(C3CCCO3)=O)CC2C1.C C=CCCCCCC(=O)N1CC=CC1C(=O)NC(C)Cc1cccs1 N1(C(C2(CC)CC2)=O)CCCC(C2CC2NC(=O)Cc2c(CC)n[nH]c2)C1 c1(NC(=O)NC2(C)CCN2)ccc(N2CCSCC2)c(Cl)c1 C(=O)(C1=NOC2COCC12)N.CCC(CO)(C(=O)N1CC(OCC)C1)OC.C=O c1(OC)cccc2[nH]cc(CC(=O)N(CCN3CCOCC3)Cc3ccncc3)c12 C1(N(C(c2c(CC)nccn2)=O)C)CCCCN(C(C2CCC(C)(C)CC2)=O)C1 Cc1ccc2nc(C(=O)NC3CCN(C(c4cc5ccncc5s4)=O)C3)cn2c1 C1(F)(CC)CCCN(C(c2cnc(-c3ccc(F)c(Br)c3)s2)=O)C1 CC1=NOC(C)(C(=O)NC(c2nocc2C(=O)Nc2cccc(CO)c2)C)C1 C1(CC(=O)NCCCCC2CN(C(c3cccc(Cl)c3)=O)C2)CCC12CCC2 c1(CC)cccnc1C(N1CC(F)(CNC(=O)Cc2ccc(Br)cn2)C1)=O c1(CC)cc(OC)cc(C(=O)NC2CCC2)c1.N1(CC=O)CCNC(=O)C1.C c1(C(N2CCC(N(CCC)C(c3nccn3C)=O)CC2)=O)cccc2c1CCC2 CC1(C)CC(C(=O)N2CCCC2CCNC(C2(F)CC=CC2)=O)=NO1 c1(C(=O)NC2C(NC(CC)=O)C2)cc2cc(C(=O)OC(C)C)ccc2[nH]1 C1(CNC(=O)NCC2CCC3(CC2)CC3)(CO)CC(O)C12CCC2 c1(C(=O)NCC(CC=C)NC(c2c(Cl)sc(C)c2C)=O)ccc(C)cc1Cl C1(NC(C2CCCNS2(=O)=O)=O)CCCCCN(C(=O)C2=CCCS2)C1 CC1CC(NC(=O)C(c2ccc(F)cc2)=O)CN1C(=O)CC1CCN(CC)CC1 c1cc(F)cc(F)c1.C1(NC(CN(C(C)=O)C)=O)CCC1CO.C(=O)CC N1(C(C(n2cc(CCCN3CCOCC3)nn2)C)=O)CCC2(CC1)CS(=O)(=O)C2 CN=c1nc(N2CCc3nc(C)[nH]c3C2)[nH]c(=NCC2CC(n3cncn3)C2)[nH]1 C1(C(=O)NCCC(NOCCCOC)=O)CCCCC(=O)N1 C=CCC(CNC(=O)C(CO)N(C)C)NC(C1(CO)CCOC1)=O N1(C(c2ccc(N)c(F)c2)=O)CCC2CCCN(C(c3occc3F)=O)C2C1 C1(C(=O)NCCC(C)(C)NC(c2scnc2C)=O)(OC)CCC(C)(C)CC1 C(=O)(C#CC1(C)COC1)NC1(CF)CN(C(C(CCC)(C)C)=O)C1 Cc1cccc(N(C)C(C2CC(C)CN2C(=O)C(O)CC(C)C)=O)c1C Cc1ccc2ncn(CC(=O)NC(C)(C)C(O)c3ccccc3)c2c1 c1(C(N2CCC(NC(C3(N4CCOC4=O)CC3)=O)CC2)=O)cncc2c1CCC2 C(=O)(C1CCc2ccccc21)N.Cc1cc(C(F)F)ncc1C(=O)NCC1CC1 C1(O)(C(C)NC(COCCC#C)=O)CCN(C(=O)CC=C)C1 C(c1cnccn1)=CC(=O)NCC(C)(CO)NC(=O)C(C1CCOCC1)F C(CC(O)(C(F)(F)F)c1ccccc1)NC(=NCC)NC(CC)CO c1(OCC(=O)NC2CC(CCNC(C3(C)CCC3)=O)C2)ccc(F)nc1 C1(C(=O)OC)CCC(C(N2CC=CC(NC(=O)C(c3ccnn3C)C)C2)=O)CC1 c1(CC)ccnc(C=O)c1.c1(C(N(CC)C(C)C)=O)cc(C(F)F)nn1C.N C1(CNC(C2CC(F)C2)=O)CN(C(c2c[nH]nn2)=O)CCO1.C1CCOCC1.C C1(CNC(C(C)SC(F)(F)F)=O)CC2CCC(C1)N2C(c1ccns1)=O c1(C=O)nc(=O)n(C)[nH]1.c1(C(C(=O)NCC2CC2)OC)cnn(C)c1.C CC1(C)CC(NC(=O)CCc2ccccc2)CCN(C(c2n[nH]cc2F)=O)C1 c1(C(N2CC(NC(c3c(CC)c[nH]n3)=O)C(C)C2)=O)cnc([N+](=O)[O-])n1C C1(NC(C(C)NC(C(=Cc2ccco2)C)=O)=O)C(C)(C)C1(C)C CP(C)(=O)C1CCC=C1C(=O)N1CCC(OCCNC(=O)CCn2cncn2)C1 N1(C(C2(CC)COC2)=O)CCCC(F)(CNC(c2cc(Cl)n(C)n2)=O)C1 C(C1CCCN1C)=CC(=O)N(CC(C)C(N1CCOC(CC2CC2)C1)=O)C Cc1c[nH]c(=NCCC2CCC2NC(C2CCCCC2n2cccn2)=O)nc1O C(=O)(C(C)CC(=O)NCc1csc(C(=O)NCC(C)C2CC2)c1)OC.O CC1CN(C(c2cscn2)=O)CCN(C(c2ccc(C#N)s2)=O)C1 C1(NC(CCOCCN(C(=O)CC2CCC3CC23)C)=O)CCC(O)C1 Cc1cccc(C(C)(C)C(=O)NCCC2CCCCN2C(=O)C2=COCC2)c1 Cc1cc(C(=O)NC2CC(O)CN(C(=O)C(C)C)C2)nc2ccccc12 N1(C(c2cn(C)nn2)=O)CC(NC(=O)C=Cc2ccc(F)nc2)CC(C)(C)C1 Cc1cc(Br)ccc1C(N1CCN(C(c2cc3scnc3[nH]2)=O)C(C)C1)=O N1(C(=O)NC(c2c(Br)cnn2C)C)CCC(C2(C)OCCO2)CC1 CC1(C(=O)NC(c2cccc(I)c2)CO)CC12CCN(CCCCO)CC2 c1(C(=O)NCC2(c3c(C)noc3CO)CC(=C)C2)cccnc1OCC C1(F)(CNC(c2nc(CC)sc2N)=O)CCN(C(C2CC23CCCC3)=O)CC1 Cc1ccc(C(=O)NCCCC(C)(C)CO)c(-n2cc(C3CC3)nn2)c1 c1(C(=O)NC(c2nnnn2C2CC2)C)cccc(S(=O)(=O)CC(F)F)c1 c1(C(=O)NCC23C(CN(C(CCN(CC)CC)=O)C2)CC3)cc2ccsc2n1C c1(NC(=O)Nc2c(CC)n[nH]c2)nc(C(C)C)cc(C2CCCC2)n1 c1(C(N2CCC3CN(C(C(CC)C(C)(F)F)=O)CC32)=O)ccn2ncc(C)c2n1 C1CC(C(F)(F)F)CN(C(=O)CC2(O)CC2)C1.C1(OCC=O)CC=CC1.N c1(C(N(CCNC(=O)C=Cc2ccccn2)C2CC2)=O)ccc2nn[nH]c2c1O c1(C(N2CC3(CCC(C(=O)NCCC(C)(C)O)O3)C2)=O)ccc2nccnc2c1 C(=O)(CCCCCC(=O)NC1CCC1)OCC.C12(C=O)CCC(CC1)C(C)O2.N C(=O)(C1=NNC(=O)CC1)NC1CC2CN(C(CC(C(C)C)C)=O)CC21 c1(C(=O)NC(C)CC2CN(C(=O)CCC3OCCO3)C2)cc2n(n1)CCC2 c1(C(N2CCC=C(Cl)C2)C(=O)NCC=C)cnc(OC)c(F)c1 N1(C(c2c(C)ocn2)=O)CC(NC(c2cnc(O)c(F)c2)=O)CC(O)C1 C1(CC)CCCCN(C(c2ccc(CNC(C3CCCS3)=O)nc2)=O)C1 N1(C(CCC2CCC(NC(C3CC3(Cl)Cl)=O)C2)=O)CC2(CC(O)C2)C1 C1(C(=O)NC(C(=O)NC(c2c(C)nns2)C)C2CC2)CC(=O)C12CCC2 N1(C(c2n[nH]c(CC)c2C)=O)CC(C(=O)NC2CCC2)C2(CCC2)C1 C=CCC(F)(F)C(=O)N1CC(NC(=O)COc2ccccc2CC)C(C)C1 C1(NC(c2ccn(-c3ccccc3)n2)=O)C2CC3CN(C(C4CCC4)=O)C1C3C2 N1(C(c2cc(=N)[nH]cc2)=O)CC=C(CCNC(c2ccc3c(c2)CCO3)=O)CC1 CCCCC(O)C(=O)NCC(C)(C)CNC(=O)Cc1occc1C CCCC(C)(C)C(=O)NCC1CCCCC1NC(c1ocnc1C1CC1)=O CC(CN=C(NCC1CC12CC2)NC1CCCC1)c1ccncc1 C1(CNC(C(C=C)O)=O)CCC(C)CC1.c1(C=O)cnccc1.[SH](C)(=O)=O N1(C(C(CC)(F)F)=O)CC2CCC(C1)C(NC(=O)C(C1CCCCC1)OC)C2 CC(CN=c1[nH]c2cc(F)ccc2o1)(C1CC1)NC(=O)C(=O)NCC(F)F Cc1cc(C)c(C(C)NC(=O)CCc2ncccc2C)c(C)c1 C(=O)(C1=NOC(c2ccccc2)C1)NCC1CCN(C(CP(C)(C)=O)=O)C1 c1(C(=O)NCC2(CNC(C(n3c(C)ncc3)C)=O)CCC2)ccc(O)nc1 N1(C(c2cc(C)[nH]c2)=O)CCC(C)(C)C1CC(=O)NCC1CCOC1 c1(N(C)C)cc(N2CCC(Cn3cc(CS(C)(=O)=O)nn3)C2)ncn1 Cc1ccc(Cl)c(C(=O)NC2CN(C(c3coc(N(C)C)n3)=O)CC2C)c1N C(CC(=O)NCCSC(C)(C)C)(C(C)(C)C)NC(C(C)O)=O Cc1nc(O)[nH]c1C(=O)NC(C1CN(C(c2cnc(Cl)cn2)=O)C1)C CCC(C)CC(C)C(=O)N1CCN(C(=O)CN(C)C(=O)OC)CC1CO Cc1nc(C(C)C)oc1C(N1CC(C(C)NC(c2ccncc2F)=O)C1)=O Cc1nc(NC2CC(F)(CNC(c3n[nH]cc3Cl)=O)C2)cc(Cl)n1 N1(C(=O)OC(C)(C)C)CCC2(CC2NCC2C(=O)OCC2(C)C)C1 c1(CC)cc(C(=O)NC2CN(C(=O)COc3ccsc3)CC2O)cc(O)n1 C1(CC(=O)Nc2cnc(Cl)c(Cl)c2)C2CCC1CN(Cc1cccc(F)c1Cl)C2 CN1CCN(C(c2ccc3c(c2)CC3)=O)C(CNC(C2CCC(C)(F)CC2)=O)C1 N(C1CCS(=O)(=O)c2ccccc21)C(C(N=c1cc(C(COC)(C)C)o[nH]1)=O)=O C#Cc1ccc(C(N2CCC(C)(CCNC(C3CCCCN3C)=O)C2)=O)cc1C C1(C(=O)NCCC2(C)OCCO2)(CF)CCN(C(C2CCNC2=O)=O)C1 c1(C(CCC)C)nc(-c2cn(C(C)(C)C)cn2)n(C2CCSC2)n1 C(c1cccc([N+](=O)[O-])c1)=CC=O.c1cnn(C)c1.C(=O)(C)N(C1CC1)C C(=O)C(F)(F)C(C)(C)O.c1(SC)cncc(C(=O)N(C)CCOCC)c1.N Cc1nnn(NC(=O)C(C)N(C(=O)C=C(C2CC2)C2CC2)C)c1C Cn1cccc(C(=O)NC2CCCN(C(C3(C#N)CCC3)=O)CC2)c1=O c1(C(N2CC(C)(C)C(NC(C3CC(CF)C3)=O)C2)=O)ccc2ncccc2c1 c1(CN(C)C(C2CC2NC(C2CCC(O)CC2)=O)=O)cccc2ccccc12 C=CC1CN(C(=O)CC2CCCC(=O)N2)CC1NC(c1cccc(O)n1)=O N1(C(c2ccc(CNC(C3CC(C)(CC)C3)=O)s2)=O)CCCN(CCO)CC1 Cc1ccnc(C(=O)NCCC2(NC(C3CC(C)(O)C3)=O)CCCC2)n1 C#Cc1ccc(C(N2CC(C)(CCC(=O)NC3CC(C)OC3=O)C2)=O)cc1 c1(C(=O)NCC(CC=C)NC(c2[nH]nc(OC)c2Cl)=O)nccc2ncccc12 C(CC(C)C)(C(=O)N1CCC(c2cn(C3CC(C(C)(C)C)NC3=O)nn2)C1)OC CCC(CC)CCCC(=O)N1CC(C(N2CCCC(C)(C)C2)=O)C2(CCC2)C1 c1(COCC(=O)NCC2CC2)nc2ccccc2s1.c1(C(=O)N)cnns1 c1(C(=O)NCC2CC(C)N(C(c3nnn(C)n3)=O)C2)ccccc1S(C)(=O)=O N1(C(Cc2scc(CC)n2)=O)CCCC1(CO)CNC(=O)CC(C)O C1(C)(CNC(c2c(C)ccn2C)=O)CN(C(=O)C(C)Cc2ccccn2)CC1C C1(C=O)CN(C2CC2)C(=O)N1.c1(SCC=O)nccn1Cc1ccccc1.N c1(-c2c(F)ccc(OCC)c2F)cc(C(N2CCNC(=O)C2)=O)cc2[nH]ncc12 c1(NC(c2nc(C)c(-c3cccn(C)c3=O)cc2)=O)cc(F)cc(C)c1O c1(C(=O)NC2(C3CN(C(CCOC)=O)C3)CC2)cc2ccnn2cn1 C(CC(CO)NC(c1ncoc1CNC(=O)CN(C)C)=O)SC c1(OC)ccc(-c2nnc(NCCN3CCN(S(=O)(=O)C4CC4)CC3)o2)cc1 C1(NC(c2cc3c(o2)CCCC3)=O)CN(C(C2CCCO2)=O)C2CCCCC12 N1(C(c2c(I)ncn2C)C(=O)NC(C)C)CCOc2ccncc2C1 C(=O)(C#CC1CCCCO1)NC1(C)CN(C(C(C(C)C)N2CCCCC2)=O)C1 c1ccc2nncn2c1.N1(C(c2cc(OCC)n[nH]2)=O)CCC2(CC2C(=O)N)C1 c1(OC)c(C)ccc(C(=O)NC2CCN(C(c3cc(F)n(C)n3)=O)C(C)C2)c1F C1(OC)CN(C(c2cc(Cl)c[nH]2)=O)CC1NC(c1conc1C1CCC1)=O C1(C(N)=O)OCCC1NC(c1cnn(Cc2ccccc2)c1)=O c1(N(CC(C)NC(C2(C3CC3)CCC2)=O)C)nc2c(cc1C#N)CCOC2 c1(C(=O)NC2CC2C(=O)Nc2ccc(C(F)(F)F)nn2)cc(Br)ncc1Br C1(C(N2CCC(O)(C(C)NC(c3nn(C)c(F)c3)=O)C2)=O)CCC2(CC1)N=N2 C1(CNC(c2ccc(OCCC)cc2OC(F)F)=O)Cc2ccccc2N(C)C1 Cn1ccc2ccnc(C(N3CCC4CCN(C(C5CC=CCC5)=O)C4C3)=O)c12 C1(CNC(c2ccn(CCN(C)C)n2)=O)CCC(N(C)C(C2CC2)=O)CC1 c1(C(N2CC(Cn3cc(CCOC)nn3)C2)=O)cc2c(s1)CCC(C)C2 N1(CC)CCCCC1C(=O)NCC(C)(CO)NC(c1cnn(CCN)c1C)=O CC(C)CC(C(=O)N(C(CO)C1CC1)C)NC(C1CC(=C2CCC2)C1)=O CCCCCCCCC(=O)NC1CC(CN=c2cc(C(=O)OC)nc[nH]2)C1 c1(NCC2CN(C(C(C)Cc3cnc[nH]3)=O)CC2C)nnccc1C#N N1(C(C(=O)NCCC2CCc3ccccc3C2)=O)CCCC2(C1)CC2(F)F n1(CC(=O)NC2CC(NC(CC(=C)C)=O)C23CCC3)cnc2c(cnn2C)c1=O C(=O)(CC1=Cc2ccccc2C1)OC(C(=O)Nc1c(C)ccc(Br)c1)C Cc1cc(C(N2CCC2C(N2CCN(CC3CCC3)CC2)=O)=O)ccc1I C1(C(=O)NC(CCNC(C(C)OCC(C)C)=O)C)CCC(=O)N1C C(=O)(C1CCc2c(Cl)cccc21)NC1C(NC(c2c3[nH]c(=N)oc3ccc2)=O)C1 c1(C(=O)NC(CN(C(c2cc(C)on2)=O)CC)C)ccc(-c2ccon2)cc1 N1(C(C(=O)NCCc2c(C)cc(C)cc2C)=O)CC(=O)N2CCCC2C1 c1(CC)ccc(F)c(C(=O)N(C)CCNC(C2CCCC(C)O2)=O)c1F N1(C(c2c(C)oc(CNC(C3(C#N)CC3)=O)n2)=O)CC2(C1)CC(C)(O)C2 CC(C)C(CCNC(c1ncoc1C)=O)N(C)C.C1(C(=O)N)CN2CCC1C2 N1(C(C2C(C)(C)COCC2)=O)CCC2CCN(C(=O)CC34COCC(C3)C4)CC12 N1(C(C(CC)NC(C)=O)=O)CCN(C(c2[nH]ccc2C)=O)C2CCCC12 CCCCCCCC(F)C(=O)N1CCC(CNC(c2cocc2C)=O)C1 CCCC(C)(CC)C(=O)N1CCC(CNC(c2[nH]cnc2C)=O)C1 C1(NC(C23CC(OCC)(C2)C3)=O)CCC(F)(CN)C1.C(CC=O)N C1(C(=O)NCCC(C)Nc2c(OCC)cccc2)CC12CCCCC2 N1(C(c2cn(C)nc2)C(=O)NCCOCC)CC(=O)NCC1C(C)C.C C1(CC)CCC(C)CN1C(C1CC=CCN1C(=O)CCCN1CCCC1)=O c1(C(N2CC3N(C(c4nc(C)sc4)=O)C3C2)=O)ccc2c(c1)CCCC2 Cc1cccc(C(O)C(=O)NC2CCCCC2NC(C2CC3CC3C2)=O)c1 C1(CNC(c2n(C)nnc2)=O)CN(C(=O)Cn2nccn2)CC1C(F)(F)F CCCCC(C)C(=O)N(C1CCN(C(=O)CN2CC3C=CC2C3)C1)CCC c1(C(N2CC(NC(c3ocnc3C)=O)CC(OC)C2)=O)cc(Cl)cc(Cl)c1F n1(CC(=O)NCC(CC(F)(F)F)NC(CC(COC)C)=O)cnc2ccccc12 C1(NC(c2n(C(C)C)nnc2)=O)CCCCCN(C(c2[nH]nnc2C2CC2)=O)C1 C(=O)(C1CCc2cc(F)ccc21)NC1(C)CN(C(c2c(C)c(CO)ccc2)=O)C1 C1(CNC(C(C)OCC)=O)CN(C(c2ccco2)=O)CC1(C)C.CC(C)C C#CC1(O)CC(C(=O)NC)C1.C1CCC1(C)C.c1(C=O)cc(C(C)C)oc1C C1(CC(=O)NC(CC)CNC(C2(C)CCCCCC2)=O)CCc2sccc2C1=O O(N(CC)C(=O)C(Cc1cc[nH]n1)NC(=O)C#CC1CCC1)CC c1(C(=O)NC(CNC(C(CCOC)C)=O)C2CC2)ccc(Cl)cc1[N+](=O)[O-] C1(NC(C(=C)C(F)(F)F)=O)C2COCC1CN(C(c1nccc3nc[nH]c13)=O)C2 N1(C(c2n(CC=C)ccc2)=O)CCC(C)C1CNC(C1(C)CCC1)=O N1(C(c2n(CC)ccn2)=O)CC(C(=O)NCCN2CC(OC)C2)C(C)(C)C1 c1(C(N(C2CCC(NC(C(CC)CC)=O)C2)C)=O)cnc2nc(C)oc2c1 N1(C(C(=Cc2ccco2)C)=O)CCN(C(c2cnn(C)n2)=O)CC1C1CCCC1 c1(C(N2CCCC2)=O)ccccc1.c1(CC)c[nH]nc1C(=O)NC.C(C)(C)C N1(C(=O)OC(C)(C)C)CCSCC1C(=O)OCCSc1cccc(Cl)c1 c1(CC(N2C(C)(CNC(=O)Cc3nncs3)CCC2)=O)ccnc(Cl)c1F O=C(CCCCCCCCCO)NC1CCCC(NC(c2cc(Cl)c[nH]2)=O)C1 C1(NC(=O)C(O)C2CCCC2)CCSC12CN(C(=O)CC13CCCN1CCC3)C2 c1(C(N2CCC(C)(O)C2)=O)c(-c2cnc(N3CCCC3)nc2)ccc2c1OCO2 Cc1ccc2c(c1)C=C(C(=O)NC)CO2.C12CC(C1)C2.C1(C=O)OCC1(C)C C12(NC(C3CC3(Cl)Cl)=O)CCCC1(F)CN(C(=O)CCC(CF)CF)C2 N1(C(C(n2c(C)ccn2)C)=O)CC(C)C(C)(C(=O)NCC(O)CN(C)C)C1 C1(C(=O)NC(C2N(C(c3noc(CC)c3C)=O)CCC2)C)CNC(=O)CC1(C)C C12(CCNCC1)C(=O)NOC2.c1(CC)ncsc1OCC c1(C(N(C2CN(C(=O)C(C)(C)CO)CC2(C)C)C)=O)ccc(N)cc1F c1(CC)ccc([N+](=O)[O-])cc1C(=O)NC(C)C.c1(C=O)cc2ncccn2n1.N Cc1cn2c(CC(=O)NCC(C)CNC(c3cnn(C)n3)=O)csc2n1 N1(C(C2(OCC)CCC2)=O)CCN(C(=O)CC2CCSC2)C(CO)C1 Cc1cnc(C(N2CCCC(COC(F)F)C2)C(=O)NC2CC2)c(Cl)c1 C1(NC(C2(NC(C(C)NC(C)=O)=O)CC2(C)C)=O)CCC(C2CC2)CC1 N1(C(c2c(C)ncn2C)=O)CCC(NC(C2(O)CCC2)=O)C(c2ccccc2)C1 C12(NCCn3ncc(C#N)c3)CCC(C(=O)N(C3CSC3)CCF)(CC1)C2 CC(C)CC(O)C(=O)NCC(C)(C)OCC(=O)NC1CCCC(CO)CC1 C1(C(N(CC(CCC=C)O)C)=O)CCCCC1(C)NC(C1CCCC(=O)C1)=O Cc1nc(CC(=O)NCC2CN(C(=O)C)CC2C)c(C)s1.C(=O)N.C1CC1 N1(Cc2ncn(C)n2)CCOC(C)(CNC(c2ccc(Cl)o2)=O)C1 Cc1nc(C(=O)NC(C)CCCNC(c2csc(Br)n2)=O)c(C)s1 C(C)(C)(C(C)CC(=O)NC1CC1(C)C(F)F)NC(C(C=C)C)=O CC1=C(C(=O)NCCCNC(c2cc3cnc(Cl)cc3s2)=O)S(=O)(=O)CCO1 Cc1nc(N(C(C2CSCN2C(=O)C(C)(C)C)=O)C(C)C)sc1S(N)(=O)=O C1(C(=O)NCC(CN(C(Cc2n(C(C)C)cnn2)=O)C)(C)C)CC12CCOC2 n1(CC)cc(CC(N2CCN(C(C3CC(OC)C3)=O)CC2C)=O)c2ccccc12 C(=O)(C1=CCC(C)CC1)N(C1CCN(C(c2ccc(OC)c(Cl)c2)=O)C1)C C1(C(=O)NC(CCOC)C=O)CC2(CC(=O)C2)C1.C(C)CCC=C(C)C.N Cc1ccc(C(N)=O)cc1NC(C1CC(O)CN1C(=O)Cn1ccnc1)=O N1(C(CC2CC(CC)C2)=O)CCCC1CCC(=O)NCC1CCC(C)C1 N1(C(C=Cc2n(CC)ccn2)=O)CCC=C(CNC(=O)CN2CCOCC2=O)C1 C1(NC(CC(C=C)(C)C)=O)COC2(C1)CN(C(c1ccc(C)nc1N)=O)C2 n1(CC(=O)NC2CCN(C(C3C(C(C)C)C3)=O)C2)cc(S(C)(=O)=O)cn1 CC1(C)CC(CNC(=O)C(F)(F)C2CC2)CN(C(C2Cc3ccccc3S2)=O)C1 N1(C(c2c(CC(C)C)n(C)nc2)=O)CC2(CCN(C(C3CC(F)C3)=O)C2)C1 c1(OC)ccnc(O)c1C(N1CCCC(C(C)NC(C2(CCO)CC2)=O)C1)=O c1(CN(CCNC(C)=O)C(c2ccc(O)nc2)=O)cccc(Cl)c1 c1(OCC)cc(-c2ncc(Cl)cc2C(=O)NC(C)C(N)=O)cc(C)c1 CC(C)(C(=O)N1CC(CNC(C2C3COCC23)=O)C1)c1cc[nH]n1 CCCC(CC)C(=O)NCC1CCCCC1NC(c1cnn(CC)c1Cl)=O C1(C(N(C(CN(C(C(C)SC)=O)C)C)C)=O)Cc2ccccc2C1 O=C(C1=CCCOC1)NC1CC2CC(NC(c3ccc(F)c(C(F)F)c3)=O)C2C1 C(C(CC)(CC)C(=O)NC(c1ncc(C)cn1)C)NC(c1cnc(CC)o1)=O C1(CC(=O)OC)CN(C(C2CN3CCN2CC3)=O)CC1(C)C N1(C(C2C(C)=CCS2)=O)CCOC2CN(C(c3cc(F)c(C)cc3F)=O)CC12 Cc1cc(C(N2CCOC(CNC(c3ccncc3F)=O)C2)=O)cc(C)c1 CCCCCC(O)CC(=O)NC1(C2CCCCN2C(=O)C2=CCCS2)CC1 C1(C(N2C(C(C)NC(=O)CCC(C)(F)F)CCC2)=O)CCc2cnnn2C1 c1(OC)cc(OC)c(C(=O)NC2(C)CCOC2)cc1.C(=O)CC1CCC1.N C(=O)(C(O)CC(N)=O)NCCC1(O)CCN(C(CC(=C)C)=O)C1 CC1CCN(C(C2(n3cc(C4CCCC4)nn3)CCOCC2)=O)CC1 C1(NC(C2CC3CC3C2)=O)CC=CCC1C(=O)NC(CC1CC1)CO C1(CNC(C=CC=CC)=O)CN(C(C2CC(C)(C)CN2C)=O)CC1(F)F C1(c2nnnn2Cc2ccsc2)(NC(CCC)c2ccco2)CCCCC1CC c1(C(N2C(CC)CCC2C)C(=O)NCC(=C)C)ccnc(N(C)C)c1 CC1CCCC1(C)C(=O)NCCCC1(NC(=O)Cc2ccc(Br)cc2)CC1 c1(CC(C)C(=O)N(C)CCN(C)C(C2CC3CC3C2)=O)ccc(F)cc1 c1(C(=O)N)cc2n(n1)CC(F)C2.c1(C=O)ccn(C2CC2)n1.C1(CC)CC1 N1(C(Cc2c(C)cco2)=O)CCSCC1C(=O)NCC1(OC(C)C)CC1 N1(C(c2ncc(Br)cc2F)C(=O)NC2CC2)CCCC2(CC=CCO2)C1 C1(C(=O)NCc2cc(C)no2)CCCC(NC(=O)Cc2cccc(Cl)c2)C1 NS(=O)(=O)c1cc(C(=O)NC2COCCN(C(c3cccc(F)c3F)=O)C2)cs1 C(CCC(C)(C)C(=O)N(CCO)OC)NC(C1CCC(CC)CC1)=O C(=O)(CC(C(C)(C)C)NC=O)N(CCCNC(C(CC)F)=O)C.C(C)(C)C C1(C(N(CC(C)(C)C(=O)N2CCCC2C)C)=O)CC(=O)CC12CCC2 C1(N(C(=O)CC(C)c2ccco2)CCOC)CCN(C(=O)C=C(C)C)CC1 c1(C(N2CC3C(C(=O)NCC4CC(C)C4)C(CC3)C2)=O)cn2c(Cl)cccc2n1 C1(CC=C)CN(CCOCCc2ccco2)CC1(F)F c1(OC)cc(C2CC2)ccc1C(c1nnnn1C)NCCC1COCC(C)O1 Cc1nc(C)c(C(=O)NC(c2ccccc2)CNC(=O)CC2CCOC2)[nH]1 c1(OC)cc(C)nc(N2CC3C(C2)N3C(=O)Nc2ccccc2)n1 N1(C(C2CC(OC)C2)=O)CCC(CCNC(=O)CC)CC1.c1ccc(Cl)cc1.S C1(C(N2C(C)C(NC(=O)CCc3cc(Cl)no3)CC2)=O)CCC2(CCC2)O1 C1(NC(CCCCC)=O)CC2CCC1N(C(C1CCN(C(=O)CC)C1)=O)C2 C1CCC(F)(F)CC1.c1(C(C)OCC)nc(-c2cnc(C(C)O)s2)[nH]n1.C1CC1 c1(C(N2C(C)CCC(CNC(C3CCOCC3)=O)C2)=O)ccnc2c1CC(=O)N2 C(C)(C)(CC(=O)NCC(F)(F)C(C)C)N(C(C1C(CC)CCC1)=O)C S(=O)(=O)(c1c[nH]ccc1=NCCC1CCCO1)NCc1c(C(C)(C)C)con1 C1(C(=O)NC2C(C)CN(C(=O)C3=C(Cl)CCOC3)CC2)CCC2CCCCC2C1 CC1CC(C(=O)NC2CCOCC2NC(=O)CCc2cccnc2F)CC(C)O1 C=CC(CCC)CC(=O)N1Cc2[nH]nc(C(=O)NCC3CCOC3)c2C1 C1(NC(C(C(C)C)n2cnnn2)=O)CC2CCC(C1)N2C(=O)CSC(F)F c1(OC)ccc(CC(C(=O)NC(CO)C(c2ccccc2Cl)O)OC(C)=O)cc1 c1(C(N2CCC(F)C2)C(=O)NC(CC)C)cnc(C2CCCCC2)s1 N1(C(=O)OC(C)(C)C)CCc2[nH]c(C(=O)NCC(Cl)=CCl)cc2C1 c1(C(C)C)cc(C(=O)NCCC2(C(=O)NCCCc3ncco3)CCC2)no1 CCN=c1[nH]c(C(N2CC(NC(C3CCC(F)(F)C3)=O)C(C)C2)=O)cs1 C(CC(O)C(=O)OC)SC.C1(C(C)C)C(=O)N(C)C(C)(C)CC(=O)N1 N1(CC)CCC(C(=O)NCC(O)C)C1.C1(C=O)CSCN1C(C1CCCC1)=O c1(C(N2CCCC(NC(c3[nH]cc(C)c3)=O)C2)=O)c[nH]c2cc(C#N)ccc12 C1(NC(c2cccc(F)c2Br)=O)CCC12CN(C(=O)C=C1CCCC1)C2 O(NC(=O)C1=CC2CCC(C1)C2)CC(=O)N(CC(C(=O)OC)C)C N1(Cc2c(C)con2)CCC(NC(c2ncoc2C2CCCO2)=O)CC(C)(C)C1 c1(N2CCC(CC)OCC2)nc(N2CCCC(C)(CO)C2)c2[nH]ccc2n1 O=C(C1CCc2ccccc21)N1CC2CC2(C(=O)Nc2cc(O)cc(F)c2)C1 c1(OCC(N2C(CNC(CCC=CC)=O)C(C)CC2)=O)cccc(F)c1F C1(NC(N(C(C)CCC(=O)OC(C)(C)C)C)=O)CCc2cn(C)nc2C1 C1(C(=O)NC(C(=O)N2CC(C)C2)(C)C2CCC2)CC2C=CC1C2 C(C)(c1ccco1)=CC(N1CCC(CCNC(C(CC)C)=O)C1)=O C(=O)(NNC(=O)CCC1CNC(=O)N1)Nc1cc(C(N)=O)c(C(F)(F)F)cc1 C1(C(N2CCC(NC(CC(=O)NC)=O)C2)=O)CC(=O)c2ccccc2O1.C1CC1 C1(O)(CCNC(C2CCN(C(C)=O)C2)=O)CCCN(C(=O)C)C1.CC(F)F.O CC1CCCC(O)(C(=O)NCC2(NC(=O)CCC3CCCC3)CCC2)CC1 C=CC(CCC)CC(=O)NCCCCN(C(=O)Cn1cnc(C(N)=O)n1)C c1(C(N2C(CNC(c3c(CC)[nH]cc3)=O)CCCC2)=O)cccn2nccc12 C1(CC(=O)N(C2CN(C(=O)Cc3cc(C)cs3)CC2F)C)(CC)CCOCC1 C1CC12CCc1ccccc12.C(C(F)(F)F)NCCCNC(=O)NCC(=O)N c1(CN2C(CNC(c3cscn3)=O)CCC2)c(Cl)cncc1Cl N1(C(c2c(C)oc(-c3ccccc3)n2)=O)CC(=O)Nc2ccccc2C1C n1(CC)nc(C(=O)NC2CCCC2NC(c2snc(C)c2N)=O)cc1O C#Cc1cccc(C(=O)NCC2(C)CCCCC2)c1F N1(C(Cn2c(C(C)C)nnn2)=O)CCOCC1CNC(C1(C)CC(C)(C)C1)=O C(CCC(=O)N1CCCC1CN(C)C(c1ccnn1C)=O)OC c1(C(N2CC(C(=O)Nc3c(OC)cccc3F)C2)=O)ccc2ncncc2c1 C(=O)(C(O)C)NC1CC(CCC(=O)NCCC2(COC)CCC2)C1.S C1CN(C(=O)CN2C(=O)CNC2=O)CC1(F)F.C(CC(=O)N)OCC(C)C.C Cc1cc2nc(C(N3C4CCC(C4)C3C(N3CCCSCC3)=O)=O)[nH]c2cc1C c1(OC)cccc(SCC(=O)NC2(C)CC2)c1.C1(C(=O)N)COC(=O)O1 c1(CN2C3CN(C(c4c(C)nc(C)s4)=O)C(C3)C2)cc(I)cc(I)c1O c1(OC)ccc(CC(C)C(=O)NCC23CC2CN(C(c2cncs2)=O)C3)cc1F C(CCC(=O)NC(Cc1cn[nH]c1)C=O)N(C(C)C)C.CC(C)(O)CN(C)C.N C1(NC(C2(CCC)CC2)=O)CC(C)N(C(c2cc(Br)no2)=O)C1 O=C(C1=Cc2ccccc2C1O)NC1COCCN(C(c2cnnc(O)c2)=O)C1 N1(C(C2CC(=C)C2)=O)CC2CCC(C1)N2C(c1c(I)n[nH]c1C)=O CC(C)C(C)C(=O)N(CCCNC(=O)CC1CCC(=O)NC1)CCO C1(NC(c2n(COC)ncc2)=O)CCC(C)N(C(c2n[nH]cc2C)=O)C1 Cc1cc(Cl)c(C(=O)NC(C)(C)C(C)NC(C2CN(C)C2)=O)cn1 C1(CNC(C(C)n2cccc2)=O)CC(C(=O)NCC2CC3CC2CC3O)=NO1 C1(NC(CC(=O)OC)=O)CCC(N(C)C(c2cc(C(N)=O)c[nH]2)=O)CC1 c1(C(=O)NCC2N(C(CN(CCC)C)=O)CC2)nnn(-c2ccn(C)n2)c1C C=C(Cl)CCC(=O)NC(c1ccnn1C)C(=O)NCCC(O)COC CCC(CCCO)NC(C1(CNC(=O)CC2CCCCO2)CCCCC1)=O N1(C(c2c(CC)nc(C)o2)=O)CCCCC(CCC(=O)N(CC(C)C)C)C1 Cc1cn2c(n1)CCC(C(N1CCC3(CCCN3C(=O)C(C)CO)C1)=O)C2 Cn1ccc(CNC(c2cc(C)[nH]n2)=O)cc1=O.C1(C(=O)N)CCCC(=O)N1 CCCCCC(O)CC(=O)NCCCC1CCCN1C(=O)C(C#N)C(C)(C)C Brc1coc2cccc(N3CC4OCCN(c5ccccc5)C4C3)c12 Cc1oc(CNC(c2ccnnc2)=O)nc1C(=O)N(C(C)C(C)(C)C)C Cc1ccc(-c2nc(C(=O)N(CC(C)CNC(=O)C(C)S)C)cs2)o1.C(C)C C12(CNC(C=CCOC)=O)CC(CCO1)C2.c1(C=O)ccc(Cl)cc1.N c1(C(=O)NCC2C(NC(CN(CCC)C)=O)C2)cc(C2CCCC2)no1 N1(C(Cc2nc(C)[nH]n2)=O)CCC(C(=O)NC2CCOCC2F)CC1(C)C C1(CC(=O)NC2CC(NC(c3ccn(C)c3)=O)C2)CCCC(F)(F)C1 C12(C(=O)NC3C(NC(c4cncc(C)c4)=O)CCC3)CCCN(CC1)C2 c1(C(=O)NCCN(C(=O)Cn2nccn2)C)c(C(F)(F)F)nnn1C c1(COC)noc(-c2cn(C3COCC3n3cc(C(N)=O)nn3)nn2)n1 Cc1cc(C(N2CC(NC(C3CC4CC4C3)=O)C(C)C2)=O)cc(C)c1O c1(C(=O)OC)ccc(C=CC(=O)N)o1.C1(C)(C(N(CC)C)=O)CCCC1C CCCCC(CNC(C1CC(=O)C1C)=O)NC(=O)C(F)(F)c1ccccc1 C(=O)(CCCCC(=O)NC1CCC(CNC(=O)Cc2cccc(Cl)c2)CC1)NC N1(C(C(CC)NC(N)=O)=O)CCCC1(C)C.N1(CCCC=O)C(=O)CCC1=O.N C(CN(C(=O)CNS(=O)(=O)N(C)C)C)(CO)(CO)NC(CCC#C)=O CCCS(=O)(=O)C(C)C(=O)NC1COCCN(C(C2CC(SC)C2)=O)C1 O=C(C1=CCOCC1)NC(c1cccnc1)C(=O)NCC1(F)CC(CO)C1 n1(CC)nc(C(=O)N(C)CCN(C(=O)C(c2ccc(F)cc2)O)C)ccc1=O C1(NC)CCOC1.c1(CN(CCC)CCC2CN(C(C)=O)C2)nnnn1C CCC(C)C(CC(=O)NC1(CC)CCCCC1)NC(c1[nH]cc(C)c1C)=O N1(C(=O)Cc2cc(F)cc(F)c2)CCC2CC1CN2C(=O)C#CC1CCCO1 c1(C(=O)NCC(CC)(C)NC(C2CC=CCC2)=O)ccccc1SC(F)F C(CC(C(=O)N1CC(O)CO1)NC(c1cc(OC)no1)=O)OCC c1(C(=O)NC(C2CCOC2)CNC(=O)C)ccc2c(n1)CCO2.c1ccsn1 N1(C(=O)NC(c2cn(CCOC)nc2)c2ccccc2)CCCC(C2(O)CC2)C1 CC(C)C(N=[N+]=[N-])C(=O)N1CC(C2CC2C(N2CC3CCC(C2)O3)=O)C1 C1(N(C(C(CC)C2CCOCC2)=O)CC)CCN(C(=O)CCC(N)=O)CC1 c1(OCC(=O)NC2CCCC(NC(C3C(C#N)C3)=O)C2)ccc(F)cc1Cl Cc1oc(CNC(C2NC(=O)OC2C)=O)nc1C=O.C1(CC)CCN(C)C1=O c1(C(=O)NC(C2(O)CN(C(c3n(C=C)ncc3)=O)C2)C)ccc(OC)cc1Cl c1(C=O)ccc(N)c(F)n1.N1(C(CC2C(CC)C2(F)F)=O)CC(F)CC1C.N N1(C(C(C)OCC(C)C)=O)CCCC(C)(C(=O)NC(C)(C)CCCF)C1 C(CC(C)C(=O)NCC1(C)CCCN1C(c1ccon1)=O)=CC.N1CCCC1 C(=O)(CC(CNC(c1cnn[nH]1)=O)OC)NCC(COC)(C)O CCCC(C(=O)N1CCC1CNC(=O)C(C)=CC(C)(C)C)C(C)C C(=O)(C1=CC2(CN(C(=O)C(C3CCCCC3)O)C2)OC1)N1C(C)(C)C(O)CC1 c1(C2N(C(=O)NCC3(C(=O)OCC)CCCCO3)CCC2)cc2ccccc2s1 C1(NC(c2cc(C)cc(C)c2)=O)CC2CCC(C1)N2C(=O)CC1CCCC(C)O1 C1(C(=O)Nc2c(C)ccc(F)c2)C2CCCC2CN1C(c1cc([N+](=O)[O-])n[nH]1)=O c1(NC(N(C)Cc2c(C)ccnc2)=O)cccc(F)c1C#N C1(C(=O)NC2(C(N)=O)CC2)CN(C(=O)C(C2CCOCC2)O)CCO1 C1(O)(C(=O)NCCNC(c2ccc(O)cn2)=O)CCCCC1 N1(C(C2CC2(Cl)Cl)=O)CC(C(N2CCCCC2C2(O)CC2)=O)C2(CC2)C1 N#CC1CCCC1NC(C1(NC(c2nccs2)=O)CC(CO)C1)=O C1(C#N)(NCCc2nc(N(C)C)sc2)CCCNC1 c1(CN2CC(C)CC(NC(c3cnc(C)s3)=O)C2)c[nH]c2cc(F)ccc12 CCCC(C#N)C(=O)NCCN(C(=O)CCNC(N)=O)C c1(C(N2C(COC)(C)CCC2)=O)cc2c(cn1)CCCC2.C1(C=O)CC12CC2 C1(CCC)CCC(C(C(=O)NC(C)CC)N(C(C)C(F)(F)F)C)CC1 CCC1=NOC(C(=O)N(CCC)CC)C1.c1(C=O)cn(C)nc1C(C)(F)F.N C1(CNC(C=CC(C)C)=O)CC2(CCC2O)C1.C(C(F)(F)F)=CC=O CCC(F)(F)CC(=O)NCC1CCN(C(C2CC2(C)C)=O)CC1 c1(OCC)ccc(C(C)=O)cc1.C12CCN(C1)C(=O)C(C)NC2 N1(C(CCCC#C)=O)CCCC1C1CCCN1C(=O)CC(F)(F)C(F)F C1(c2n(CCC)nnn2)(NCc2cccc(C)c2C)CCC(C2CC2)C1 N1(C(C2(C=C)CCC2)=O)CCC2CCN(C(c3c(F)cccc3F)=O)CC2C1 C(CCCCC(=O)N1CC2(NC(=O)CN3CCCCC3)CC1C2)NC(N)=O c1(C=O)cc2ccccc2nn1.CCS(=O)(=O)NCCC(=O)NC1CC1C.N c1(CC(N2CC(C)(NC(c3ncc(Cl)s3)=O)C2)=O)cn2cc(F)ccc2n1 c1(N2CC(CC=C)(NC(c3ccc(C)cc3C)=O)C2)cc(=O)n(C)c(=O)n1C C1(CNC(C(C2(C)CC2)NC(CN(C(=O)OC)C)=O)=O)CCSCC1 c1(C(N2C(CNC(=O)CCC3CC3(F)F)CC(F)C2)=O)cc2ccncc2o1 c1(OC)nccc(C(=O)NC)c1F.C1(C)CCN(C(=O)CCC2CC2(C)C)CC1 O=C(CCCCCO)NC1CN(C(c2cccn(C3CCC3)c2=O)=O)C1 c1(-n2c(C)ccn2)ccc(NC(C2(C)CCOC2)=O)cc1.C(C)(C)C.C(=O)N C1(COCC)CCCN(c2nnc(C(O)C3CC3)n2CC2CC2)C1 C1(O)(CNCc2nnc(C)o2)CCCC(C)C1 C1(N(C(C2(SC)CN(C(c3c(CC)nn(C)c3)=O)C2)=O)C)CCN(C)CC1C c1(N2CCC(C#N)C2)nc2c(c(=NCc3cn4c(n3)COCC4)[nH]1)COC2 N1(C(C2(COC)COC2)=O)CC2CCC(C(=O)NOC(CO)C(C)C)(C2)C1 Cc1cc(C)n2ccc(C(=O)NC3CC(CCNC(=O)C4=COCCC4)C3)c2n1 C1(=CC(N2C(CCCNC(CSCCCC)=O)CCCC2)=O)CCCCC1(C)C N1(C(C(CC=C)OC)=O)CCC(C(=O)N(C2CCCC2O)C)CC1(C)C C1(C(C(=O)NCC(=C)Cl)F)CCN(C(c2ccc(C)[nH]2)=O)C1 c1(C(N2CCCC(CCCO)C2)C(=O)NC2CCC2)sc(C(F)F)nc1Br c1(OC)ccc(CC(=O)NCCCCc2ccc(F)c(F)c2)cc1[N+](=O)[O-] Cc1ccc(-c2csc(NC(C3CCCO3)=O)c2)c2cccnc12 N1(C(C2(CCC=C)CN(C(c3ccc(C4CC4)o3)=O)C2)=O)CC(O)CC1C C(=O)(CCC(=O)N)NC(CNC(CSc1cnc(C)o1)=O)(C)CO.C1CCCC1 Cc1nc(NCCS(=O)(=O)N(C)C)cc(=NCc2ncccn2)[nH]1 Cc1ccc(F)c(N)c1C(N1CC(NC(=O)C(n2nccc2C)C)C2(CC2)C1)=O N1(C(CCCOC(C)(C)C)=O)CC2CC2(NC(=O)C(F)Cc2ccccc2)C1 c1(NCc2n(CCC)ccn2)cc(N2CCCOC(CCOC)C2)nc(C)n1 C1(C)(CC)C=C(C(=O)NC2CN(C(=O)CCCC(F)F)CC23CC3)C1 C=CCC(C)(C)C(=O)N1CCC(C)(CC(N2CCC(n3ccnc3)C2)=O)C1 N(C(=NCCCF)NC1CCOc2ccc(F)cc21)Cc1oc(C)c(S(C)(=O)=O)c1 C(N=c1ccc([N+](=O)[O-])c(O)[nH]1)C1CCN(C(c2sccc2F)=O)C1 N1(C(c2c(C)cn(C)c2)=O)CCCCCCC1C(=O)NC(c1cnsc1)C C(CC(C)(C)C)NC(c1cn(CCC)nc1)=O.c1(C=O)sc(C2CC2)nc1C.N N1(C(C(C)C(C)(C)C)=O)CC2C3CCC(C2C1)N(Cc1nnc(C2CC2)o1)C3 C1(NC(C2(C)CCCO2)=O)CCCCCC1NC(c1csc(Br)n1)=O C1(C(=O)NC(C2CCCC2)CNC(COCCC#C)=O)COCCC1(F)F C=C=C(C)CC(=O)N1CCC(C(C)NC(=O)C(C)c2ccco2)CC1 CC1(C)OC(C)(C)C1C(=O)NCC1CCCCN(C(=O)CC2CC2(Cl)Cl)C1 C(=O)(CCCS(=O)(=O)NC(c1cccc(Br)c1)=O)N(C1CCN(C)C1)CC CCC(C(C)CN(C)C)NC(=O)C(C)(CO)NC(=O)CCOCCOC Cc1csc(=O)n1CC(N1CCC1CNC(=O)CC1(N(C)C)COC1)=O N1(C(C(CC)c2cccnc2)=O)CCN(C(c2cc(C3CCC3)on2)=O)CC1C CCC(CC(=O)NC12CCCC1CN(C(=O)C=Cc1scnc1C)C2)C(C)(C)C Cc1cc(CNC(=O)CNC(=O)Cc2csnc2C)ccc1F C1(C(=O)NC(CC=C)CO)COCCN(C(c2cc(C)cc(O)c2)=O)C1 Clc1csc(C(c2nnnn2CSc2ccccc2)NCc2cccnc2)n1 C1(C(=O)NC2(C)CCN(C(c3c(OCC)ccs3)=O)C2)CCCC2(CC2)C1 C1(NC(c2ccc(CNC(C(C)n3ccnn3)=O)s2)=O)C=CCCCC1 C(C1=NOC2CN(C(=O)Cn3cc(Cl)cn3)CC12)NC(Cn1c(C)ncc1)=O c1(OC)nc(C(N2CCN(C(=O)C(C)O)CC2C2CC2)=O)cc(O)n1 C(=O)(C1CCCn2nccc21)NCCC(C)NC(c1c(C(F)F)cccc1F)=O c1(C=O)ccc2nc(C)oc2c1.C1(CCOC)CCN(C(=O)C(=O)N(C)C)C1.N S(=O)(=O)(c1ccc(F)c(C(N2CCC(C(F)C(=O)OC)C2)=O)c1)NCC C1(CNC(C(C)SC)=O)CN(C(=O)C(CC)n2cccn2)CC12CCOCC2 C1(NC(c2cccc(=O)o2)=O)CC2CC1CN2C(=O)CO.c1ccc(F)cc1F N1(C(C2(CC=C)COC2)=O)CCCC(O)C1.n1(CCC=O)cc([N+](=O)[O-])cn1.N N1(C(C2(C)C(C)C2)=O)CC2CN(C(c3ccc(OC(F)(F)F)cc3)=O)CC12 N1(C(c2c(C#C)c[nH]n2)=O)CCC2CN(C(=O)Cn3nnc4c3CCCC4)CC12 c1(C(=O)NCCC)cc2c(cc1Cl)NCC2.c1(C=O)cc(-c2ccn(C)n2)on1.N C(=O)(CC(C)=C(C)C)NCC1C(NC(CNS(CC)(=O)=O)=O)CC1 c1(NC(C(C2CCN(C(c3ccc(C)cn3)=O)C2)F)=O)cnc(Cl)nc1C C(CCCC(=O)N1CC=CC1C(N1CCC(O)CC1C)=O)(OC)OC N1(C(CC(C)c2ccco2)=O)CC2(C=C(C(=O)NOCCOCCO)CO2)C1 Cc1noc(CCCC(=O)N(CCNC(c2cncnc2)=O)C(C)C)n1 C1(C(=O)NC(CC#CC)CO)CNC(=O)CN1C(c1cc(COC)no1)=O N1(C(C2C(C3C(C)C3)C2)=O)CC(C)C(Nc2ncc3ncnc-3[nH]2)C(C)C1 c1(C(=O)NCC2C(NC(c3n(C)nnc3)=O)C2)c[nH]c2nccc(Br)c12 C1(CNC(c2n(C)cnc2)=O)COCCN1C(c1ccc(Cl)nc1)=O C(=O)(C#CC1CCCC1)NCC(CNC(C=C=C(C)C)=O)(C)F N1(C(Cc2c(C)n(C)nc2)=O)CC2CCN(C(=O)CC(C)C(C)C)C2C1 N1(c2ncn(C)c(=O)c2)CCC(C)(C)C(CNC(C2CC23CCSCC3)=O)C1 Cc1nc2cc(C(=O)NCC3CN(C(C4OCCCO4)=O)C3)ccc2n1C C(C(=O)NCC1CC(OC)CN1C(=O)Cc1ccno1)(C(C)C)OCC c1(C(=O)NC2CCC(CNC(CCNC(=O)OC)=O)C2)cccc(O)n1 C1(NC(C(C)(C)C2CCCC2)=O)COC2(C1)CN(C(c1cnc3n1CCC3)=O)C2 C(CCC)(CCCNC(=O)C(CC)C(C)C)NC(CC=C)=O c12cc(ccc1F)-c1noc(n1)C(=O)OCCC2.c1(C(=O)NCCO)ccco1 C1(C(N(CCC(C(C)C)NC(CCOC(C)C)=O)C)=O)CCC2C(C1)C2(F)F N1(C(CSCCC)=O)CC2CC1CCC2NC(=O)C(O)C(C)CC c1(C(=O)OCCCOCCC2CC2(F)F)ccc(OC(F)F)cc1 C1(NC(CCCC=C)=O)CN(C(C2CC(O)C2)=O)CC12CCC2 CN1CCN(C)C(C(N2CCOC(CC(=O)NCC3CCCCN3C)C2)=O)C1 C1(C)(OC)CCCN(C(=O)CCC(C)(C)NC(=O)C=C(C)C(C)C)CC1 CC(O)(C(=O)NCC1(F)CC(C)C1)C(F)(F)F.c1(C(=O)N)ccccc1 CC1CCN(C(c2ncccn2)=O)C1C(=O)NC1CC(=C2CC2)C1 C1(CC(=O)N(C)CCNC(c2ccn(C)c2)=O)CC(F)(F)C1(F)F c1(C(N2C(C(=O)NC(C3CSC3)C)CC(O)C2)=O)c(F)cncc1F c1(C(=O)NCC(C)N(C)C(C2COC(=O)N2)=O)ccc(F)cc1C(F)F C=C(C)C(C)(C)C(=O)NCC1CC(NC(=O)CC2CC(O)C2(C)C)C1 C1(NC(C2N(CC)CCC2)=O)CN(C(=O)CC2CCCCCC2)CC1C C1(C(CNCC(C2CC2)OC)O)CCCCN1C(=O)OC(C)(C)C C(CCC(F)(F)F)NC(C(Cc1ccco1)NC(c1nccs1)=O)=O C1(C(=O)NC2(CCOC)CC2)CCCCC1NC(=O)C(C)c1cc[nH]n1 CCC(C)CCC(=O)NCCC1CN(C(=O)CC2(C3CC3)CC2)CCO1 c1(NCCNC(C2CC(C)OCC2)=O)ccc([N+](=O)[O-])c(C(N)=O)c1 C1(C(CNC(c2cnc(C)[nH]2)=O)O)CCN(C(=O)C=Cc2cnc(C)s2)CC1 c1(C(c2n(CCC)nnn2)NCCCOC)cc(=O)n(C)c(=O)n1C N1(C(C(C(C)C)C)=O)CCc2nc(O)cc(C(=O)NCC(O)CF)c2C1 C1CC2(C1)CC(F)(F)C2.C1CCCS1(=O)=O.CC(C)(C)OC(=O)N.C=O CC(CC1CC1)N=c1nc2sccc2c(NCC2CCNC(=O)C2)[nH]1 C1(CC(=O)OC)Cc2ccccc2N1C(CC1CCCCO1)C(=O)NC.C1CC1 c1(C(=O)NC2CN(C(C(CC)CC)=O)C(C)(C)C2)sc2cccnc2c1Cl c1(CC(=O)N)ccc(Cl)cn1.n1(CCCC)ccc(C(=O)NCC2CCC2)n1 C1(C2CCCC2)CCC1.C(CC(=O)NCCCO)NC(COC(C)C)=O.CCCO c1(C(C(=O)OCC)N(c2ccc(OC)cc2)C)ccnc(P(C)(C)=O)c1 c1(C(N2CC3CCN(C(CC(C)NC(N)=O)=O)C3C2)=O)cccc2c1CCOC2 C(=O)(C1=Cc2ccccc2OC1C(F)F)NCC1N(C(c2cc(C)[nH]n2)=O)CC1 c1(-c2cc(Nc3nc(C)c(F)cn3)ncc2)ccc(F)cc1C(F)(F)F n1(CC(N2CC(C)(NC(C(C)OCC#C)=O)C2)=O)cnc2c1CCCC2 N1(C(CC2C(NC(COC(CC)CC)=O)CCC2)=O)CC2(C=CCO2)C1 C=CCCC(C)(C)CNC(=O)CCC(CC)NC(=O)C(C)CCN(C)C N1(C(CC2N(C(C(CC)NC(C)=O)=O)CCC2)=O)CC[Si](C)(C)CC1 C(=O)(C(F)CCC(C)C)N1C(c2c(C(=O)NC(CC#C)C(N)=O)c[nH]n2)CCCC1 N1(C(c2c(C)n(C3CCOC3)nn2)=O)CCN(C(=O)CCS(C)=O)CC2(CC2)C1 Cc1ccc(CNC(C2CCC(NC(c3cscn3)=O)C2)=O)o1 Cc1cc(F)cc(Br)c1C(N1CCOC(CNC(=O)CCOC2CC2)C1)=O Cc1nc2ncc(C(N3CC(NC(=O)CC(C)CN(C)C)C4(CC4)C3)=O)cc2o1 C(C(C)CN=C(NCc1cccc(F)c1)NC1CC1C=O)OC.C(C)(C)C.O c1(C(N2CCN(C(COCC(=C)C)=O)CC2COC)=O)ccc2nn[nH]c2c1 C=C1CCC1(C(N1CCC1)=O)NC(=O)O.c1(C=O)ccoc1.C(C)(C)C CC(C)C(CC(=O)NCC1CN(C(C2CN3CCN2CC3)=O)C1)c1ccccc1 N1(C(C2CC23CC(NC(C24CCC(CC2F)C4)=O)C3)=O)Cc2c[nH]nc2C1 c1(C(N(CCCCCCNC(C2C(CC)CCO2)=O)C)=O)ccc(N=[N+]=[N-])cc1 C(=O)(C1=CCCSC1)NC(C(C)C)C(=O)NCCCCC1CC1 c1(C(N2CCC(NC(C(CC=C)C)=O)C2)=O)oc2cc(Cl)ccc2c1C N1(C(C2(CCNC(C(CC=C)C)=O)CC2)=O)CC(C)(C)C2COCC12 N1(C(C2(CC#C)CC2)=O)CCC(CN(C(=O)C(Cc2ccccc2)CC)C)CC1 C#CC1(C(N2CC(C)(CC)C2)=O)CCN(C(=O)CC2CCSCC2)C1 CC(C)C(C)(C)C(=O)N1CCC(N(C(C2CC3CC3CC2C)=O)C(C)C)C1 Cc1cc(C(N2CCC(n3nnc(-c4ccc(Cl)cc4)n3)CC2)=O)ncc1F c1(C(=O)N)ccc(OC(F)(F)F)nc1.C1(NC(C2(C)CC2)=O)CCCC(C)C1 C1(CCC)(NC(=O)COc2ccccc2)CCN(C(=O)CCc2cnc[nH]2)CC1 c1(NC(C23CC(C(=O)NC(c4cncnc4)CC)(C2)C3)=O)cc(C)ccc1 N1(C(C2CCN(CC)C2)=O)CC2CCC(CNC(c3cscn3)=O)C2C1 c1(-n2cc(CSC)nn2)ccc(C(N2CCC(c3cnn[nH]3)C2)=O)cc1 c1ccc(C)c(C)c1.C=CC(C)(C)C(=O)N(C)CC1CCCC(NC(=O)C)C1 C1(C(N(CCC)CC)=O)CCCCCN1C(c1n[nH]cc1CC)=O CC1CN(C(=O)C(F)C2CCOC2)CCN1C(=O)CCC(=O)c1ccccn1 C1(NC(COC)=O)CC2CC1CN(C(c1ccnn1C1CCC1)=O)C2 N1(C(=O)CSC2CC2)CCC(CCC(N2CCC2)=O)C1.c1cc(C2CC2)on1.C CCCC(C(=O)NCc1nncs1)NC(C1CC(=O)C1)=O N1(C(c2c(C#N)ccnc2)=O)CCN(C(=O)Cc2cc(Br)ccc2F)C(C#N)C1 C#Cc1cc(F)c(C(=O)NCC(C)NC(c2nc(C)n3ccccc23)=O)c(F)c1 c1(C(=O)NCC2N(C(C(C)n3ccnc3)=O)CC(C)(C)C2)ccc2cnoc2c1 CCCCCCCCC(=O)NC(CNC(c1c(C(F)(F)F)cccc1O)=O)CC c1(OC)cc(C(=O)NC2CC3CCCCCC3C2)ccc1S(C)(=O)=O NS(=O)(=O)c1ccc(C=CC(N2CC34CCCCC3(COC4)C2)=O)cc1 C1(NC(C(c2ccc(C)cc2)C)=O)CN(C(=O)CSC(F)F)CC(C)(C)C1 CCC(C)C(=O)C(=O)N1CC(OCC(=O)NCc2nc(C)cc(O)n2)C1 Cc1ccc(S(=O)(=O)N2CC3CC(C2)C3NC(=O)C(F)(F)F)c(C)c1 c1(COC)ccccc1C(=O)NCC1CCCN(C(C2(C)CC(C)C2)=O)C1 C1(C(=O)NCc2ncc(C#N)o2)COCCN(C(c2ccccc2)=O)C1 C12(C(=O)NCC(C(C)C)NC(=O)CCOc3cccc(F)c3)CCCCC1C2 C1(CNC(Cc2cc(C)sc2)=O)COCCN1C(=O)C(C)C(=O)N1CCOCC1 C(CCC(=O)NC(CC1CCOCC1)C(=O)N(C)CCOCCO)=CC c1(CC(N2C(C(C)(C)NC(=O)C=CI)CCC2)=O)cccc2ncccc12 C1(NC(C2N(C)CCCC2)=O)CS(=O)(=O)C12CCN(C(=O)C(C)(C)C(F)F)CC2 C1(CNC(=O)CC2C=CCC2)CC(F)CN1C(=O)Cc1ccc(O)cn1 Cc1ccncc1C=CC(=O)NC1CCCN(C(=O)CP(C)(C)=O)C1C n1(CCC)cc(C(=O)N(C)CC2(O)CN(C(=O)CC)C2)cn1.CCN(C)C c1(C(=O)NC2CN(C(C34CC(CO3)C4)=O)C2)cccc(Br)c1Cl C(=O)(C(C)(C1CCC1)NC(=O)CN(C(=O)CCCC1CC1C)C)OC c1(CC)cc(C(=O)Nc2c(Br)csc2C(=O)OC(C)(C)C)cc(F)c1 C1(NC(CC=C)=O)CCC2(CCCN(C(=O)CNC(=O)OC)C2)C1 C(=O)(CCCC(N)=O)NC1(C)CCN(C(c2ccc(-c3ccccc3)cc2)=O)C1 C#CC1CCCCN1C(=O)CC1CN(C(C2CCC(C3CC3)C2)=O)C(C)(C)C1 Cc1cc(Br)c2cc(C(N3CCN(C)C(c4nc(C5CC5)no4)C3)=O)[nH]c2c1 n1(CCC=O)ccc(O)nc1=O.C1(CC)CCC2CC12.CC(C)(C)OC(=O)N C(=O)(CC(F)(F)Cl)NCC1CC(NC(C(C)NS(CC)(=O)=O)=O)C1 c1(CNC(C(CC)(C)O)=O)ccc(C)cc1F.C1(C=O)COCC1C(N)=O.N N1(C(CC(CCCC)O)=O)CCOC2CN(C(=O)Cc3ccc(Cl)cn3)CC12 N1(C(c2cnn(C)c2Cl)=O)C2CCC1CC(CNC(c1cc(Cl)no1)=O)C2 C(=O)(C1=CCCCC1P(C)(C)=O)NCCCN(C(=O)CS)C(C)C.C1CC1 C#CCC(C)(C(=O)NCc1ccncc1)NC(C1COC(=O)N1C)=O Cc1ccc(N)c(C(N2CC3(CCC3NC(=O)C(=O)NCC(F)F)C2)=O)c1 C1(CC(=O)NC2C(NC(CCC(C)C)=O)COC2)CCCCC(=O)N1 c1(C(C)=O)cc(C(=O)NC(CNC(=O)CC2CNC(=O)O2)CO)n(C)c1 CC1=C(C(=O)NC2(C)CC(C(N3CCC3C(=O)N(C)C)=O)C2)COCC1 c1(C(=O)NC(C(C)C)C(N)=O)ccc(Cl)c(Cc2nn[nH]n2)c1 N1(C(=O)CC(F)F)CCOC(c2ccccn2)C1 N1(C(C2=CCC(NC(C(C(C)C)N(C)C)=O)C2)=O)CC(=O)N2CCCC2C1 C1(F)(C(N2CCC(N(C(=O)COCCCF)C)C2)=O)CC=CCC1 CCCC(C)(O)C(=O)N1CC(C(=O)Nc2ccc(O)c(CO)c2)C2(CC2)C1 N1(C(C2(C)CC(F)C2)=O)CCC(CO)(NC(=O)CCc2ccon2)C1 C1(n2cc(COCC)nn2)CC2CCC1(NC(c1ccc(=O)n(C)n1)=O)C2 N1(C(C2C(OC)CCC2)=O)CCC(NC(c2csc(-c3cccs3)n2)=O)CC1 CCCCCC=CC(=O)NC(C1CCCN1C(=O)CCSc1ccccc1)(C)C c1(C(N(C2CCN(C(C3(C)C(C)C3)=O)C2)CCO)=O)cccc2c1nc(O)n2C CCCCCC(C)CC(=O)NCc1cccc(CNC(=O)CC2CCC(=O)N2)c1 C(=O)(CCCN(C)N=O)N(C1CN(C(c2cc(C)ns2)=O)CC1O)C C1(CC(=O)OC)CN(S(=O)(=O)CC2CC(C)(C)C2)C(C)(C)CO1 c1(C(=O)Nc2c(C)ccnc2C(C)C)ccc2[nH]c(=O)c(=O)[nH]c2c1 CCC(F)C(=O)N1CC(CO)(NC(C2C3CCCC23)=O)C1 C(=O)(CC1=CCCCC1)NCC1C=CC(NC(C(CC)n2nccc2C)=O)C1 Cc1cccc(F)c1C(=O)N(CC(O)CN(C(C)C(=O)NC1CCCCC1)C)C c1(OC(C)(C)C(N2CC(NC(C3CCOC3)=O)CC2(C)C)=O)ccc(C#N)cc1 C1(NC(C23CC(C)C2C3)=O)CC12CCN(C(C1CC1(F)F)=O)C2 C1(NC(CSS(C)(=O)=O)=O)CC1C1CCCN(C(=O)CC2CC3(CC3)CO2)C1 c1(-c2cn(CC(CNC(C3C4CCCC34)=O)OC)nn2)ccc(=N)[nH]c1 C1(C(N2C(C(=O)NC3CC(N(C)C)C3)CC(O)C2)=O)CCCC1C1CC1 C(C)(C(=O)N(C)CC1(CNC(=O)CCCO)CC1)(C1(C)CC1)OC C1(C(=O)Nc2cc(SC)ncc2)CCCC12CCN(C(c1cnnc(Cl)c1)=O)C2 Cc1cc(CCC(N2CCCC(CNCc3cnn(C)c3C)C2)=O)ccn1 CCC(C)C(C(=O)NCC1CCN1C(c1ccc(F)c(C)c1)=O)OC C(=O)CC(C)(C)C(F)F.C1(CC(=O)OC)(CN)CCCCC1.C1CCCC1.N CN1N=C(C(=O)NC2CN(C(=O)Cc3ccc(Cl)nc3)C3CC23)CCC1=O c1(CCC(C)O)cn(CCC2CN(C(=O)CC(=O)O)C2)nn1 N1(C(COC)=O)CCC(NC(c2cc(OC)cc(C(F)(F)F)c2)=O)C(F)C1 C1(NC(c2cc(Cl)cs2)=O)Cc2ccccc2N(C(c2ocnc2C2CC2)=O)C1 c1(OC)ccc2cnc(C(=O)NCC(F)C)cc2c1.C1(CC(=O)N)CCN(C)C1 c1(C(=O)NC2CCCCN(C(c3cc(OC)ncn3)=O)C2)c(F)ccc(F)c1O N1(C=O)CCC(C)CC1.c12nc(oc1C)C1CN(C1)C2=O.C(C)(C)C.CCN C1(C(=O)NC2(C(=O)NC3CCCC(O)C3)C(C)CCC2)C2CCC(C2)C1C C1(C(N2C3(CNC(c4c(C)csc4)=O)CC(C2)C3)=O)CC2COCC2C1 N1(C(C(C)(C)N(C)C)=O)CCN(C(c2cn3c(n2)COCC3)=O)CC12CC2 C1(C(=O)NCCC(=O)OCC)CCCCO1.C1(CC(=O)N)COCC(C)O1 C12(CNC(c3scc(C)n3)=O)CC1CN(C(=O)C(C)Cc1cccc(Br)c1)C2 C1(C(=O)NC2(CC)CCN(C(c3ccoc3C)=O)CC2)CCC2(C1)CC2(F)F N1(C(CCN(CC=C)C(c2cccc(O)n2)=O)=O)CC2(CCCO2)C1 C1(NC(C=Cc2c(C)ncs2)=O)CC2CC1CN(C(=O)CSc1ccccc1)C2 CC1OCCN(C(=O)CC2C3CN(C(C4CCCC(C#N)C4)=O)CC23)C1C Cn1nnc2c(C(=O)NC3CC4CCC3CN(C(=O)CC(C)(C)C)C4)ccnc12 C1(C(=O)NCCN(C)C(c2cc3c(nn2)CCC3)=O)CNC(=O)CC1(C)C c1(C(=O)NC2CC(NC(C(CC#C)C)=O)CC2O)cc(Br)cc(C#C)c1 C(=O)(C(F)(F)C(O)C(C)C)N1CC(CCC)C1.CCCCCC(=O)NCC(=O)N C(CCOC)(C(=O)NCc1noc(C)n1)NC(C(C=C)C)=O CC1CN(C(=O)C2=CCCSC2)CC(C)C1NC(c1ncnc2ccsc12)=O C1(NC(c2noc(CC)c2C)=O)CC2CCC1CN(C(C1CCCC1SC)=O)C2 c1(C(=O)NC(C)C(C)NC(c2cnsc2)=O)c(O)ccc(Cl)c1F c1(-n2cc(C(C)NC(=O)CCn3ccnn3)nn2)cccc(C(F)(F)F)c1 CC12CCOC(C(=O)NCCC3CCCN(C(=O)CCOC4CCC4)C3)(C1)C2 C(=O)(CC1C(=O)Nc2cc(Cl)ccc21)NC(C)CNC(c1cc(N)cnc1Cl)=O N1(C(C2(CC#C)CCC2)=O)CC2C(CNC(c3nc(C)c(C)s3)=O)C2C1 C(=O)(CC(C)COC)NCCNC(CN(CCOC)C)=O c1(OC)c(C(=O)NC)cc(Cl)cc1Cl.C1CCCCN1C(=O)Cc1cc(C)no1 CC1=C(C(=O)NC(C(=O)NCc2ccc(F)c(F)c2)c2cccs2)COCC1 C1(C)(CNC(c2ccc(C(C)C)o2)=O)CN(C(=O)CO)CCO1.c1cn[nH]c1 n1(CC=C)c(N2CCC(OCCCOC(C)=O)CC2)nnc1C(F)(F)CC c1(C(N2CCCC(CNC(C(CC)(C)CO)=O)C2)=O)c(Cl)ccc(C)c1O Cc1cc(C(=O)Nc2ccc(NC(C3COCCC3(F)F)=O)c(C)c2)c(O)nn1 c1(C(=O)OC)cc2cc(C(=O)N)sc2s1.C1(C=O)CC1(C)C.CCC1CC1 N1(C(c2c(C)nccc2)=O)CCOCC(NC(c2c[nH]nc2C2CC2)=O)C1 C1(NC(COCC)=O)C2CC1(C)CN2C(c1ccccc1C#N)=O c1(C(C)(C)O)ccc(-c2ccc(C(=O)Nc3ccc(SCC#N)nc3)cc2)cc1 C1(CC(=O)NCCC(C)NC(C2CC2)=O)SC2=NCCN2C1=O.C1CC1.C CN1CCCC2(CCN(C(=NCCCc3c[nH]nc3C(F)(F)F)NC3CC3)C2)C1 C(=O)(C1=NOC2(CCC2)C1)N.N#CC1CCCC(C(N2CC(C)C(F)(F)C2)=O)C1 c1(OC)cc(C)ccc1C.c1(C(c2nnnn2C2(C)CC2)N)nncn1C(C)C c1(C(=O)NCC(CCCC)NC(c2ccc(F)cc2)=O)cncc2nc(C)[nH]c12 c1(NC(c2ccc(SCC)cc2)C)ncccc1S(=O)(=O)N1CCC(CCO)C1 N1(C(C(COC)Cl)=O)CCC2(CCCC2C(=O)N)CC1.C(C(=O)N(C)C)C(C)C C1(C(=O)NCCOCCOC)CN(C(c2ncsc2-c2ccccn2)=O)C1 c1(C(N(C2CCN(C(=O)CC)C2)CCC)=O)coc(CC)n1.[SH](C)(=O)=O c1(C(N2CC(C)C(NC(c3ccc(O)c(N)n3)=O)C2)=O)nn(C)c2c1CCC2 c1(CC)nnc(C)cc1C(=O)NC(C)Cc1ccc(C)cc1.C(=O)CC(C)O C1(CNC(C2(OCC)CCCC2)=O)C(C)CCN1C(c1c[nH]nc1F)=O c1(NC(C2(O)CCN(Cc3c(OC)nccc3)C2)=O)nc2c(s1)CCCC2C N1(C(C2(CCC)CC2)=O)CCC2(CC(C(=O)Nc3cnsc3)C2)C1 c1(C(=O)NCC(C)NC(c2cn(C)nc2Cl)=O)ccnc(C(C)(C)C)c1 c1(C(N2C(CNC(CCCCN(C)C)=O)CCC2)=O)cc2c(ccn2C)s1 N1(C(c2c(C)c(F)cc(Br)c2)=O)CC(C2CCCN(C(=O)Cc3ccsc3)C2)C1 N1(C(C2C(C=CC)CN(C(=O)C(CC)OC)C2)=O)CCC(C2CC2)CC1 N1(C(C(CN)N)=O)CC2CCC1C(C(=O)NCC1CC1)C2 c1(C(N2CCC(C)(NC(C(CC)c3ccccc3)=O)C2)=O)cnn2c1SCC2 C1(C(N(C2CCCC(NC(c3ncncc3N)=O)C2)C)=O)C=CC=CC=C1 N1(C(COCC(=O)OC)=O)C(C(=O)NCCc2cn(C)nn2)CC2CC12 C1(C(=O)NCc2nc(C)sc2)CC(F)CCN1C(=O)CSC1CC1 CCCC(C)C(C)NC(=O)C(CNC(c1nn(C)cc1Cl)=O)N(C)C N1(C(c2ccn(C(C)(C)C)n2)=O)CCCC1C1CCCN1C(=O)CCC1CCC1 CC1=NN(C)C(=O)C1CC=O.C1(C)CN(C(=O)C(c2cccnc2)N(C)C)C1 Cc1ccc(F)c(OCC(=O)NCCC2CCN(C(c3coc(Cl)n3)=O)C2)c1 C1(NC(C(C)(C)SC)=O)CC2CCC(C1F)N2C(=O)COc1ccsn1 CC(C)(CC1CC1)CS(=O)(=O)Oc1cccc(C#N)c1 c1(OC)ccc(C(=O)NCC2CCN(C(c3cc(C)on3)=O)CC2)c(Br)c1 C(=O)(CCC1CCc2ccccc21)NCC1C2CN(C(C(C)C3CC3)=O)CC21 N1(C(CC(CNC(Cc2c(C)n(C)nc2)=O)C)=O)CCS(=N)(=O)CC1 c1(SC)ccc(C(N2CC=C(CNC(=O)CC(C)F)CC2)=O)cc1[N+](=O)[O-] C1(NC(c2cccc(C)c2)=O)CC2(CCN(C(C3CC3(C)C(F)(F)F)=O)CC2)C1 CC1(C)NC(=O)OC1C.C1(C=O)CC(O)CN1C(c1coc(C(N)=O)c1)=O n1(CCCC)cc(C(=O)NC(=O)C(c2cccs2)SC2CC2)nn1.C1CC1 C1(C(=O)OC)(C(N2CC(F)C2)=O)CC1S(C)(=O)=O.C(=O)C(C)(C)C.C c1(C(=O)NC2CC(C)N(C(=O)C(Cl)=CCl)C2)c(F)cccc1Br C(CC)(C(=O)NCCCCOCC)OCC.C(=O)(CO)N.CC c1(C(=O)N)cn2c(n1)CC(C)CC2.c1(CCC)ccc(CC(=O)NC(C)C)cc1 C#CCC(C)C(=O)N1CCN(C2CCCN(C(C3CCSCC3)=O)C2)CC1 c1(C(=O)N)ccc2c(c1)S(=O)(=O)NC2.N1(C(C2C(C=C)C2)=O)CC(C)C1 c1(C(=O)N)cncc(C(F)(F)F)c1.C1(NC(c2cocc2)=O)COCC1C C(C(F)CN=c1cc(OC)c2cc(F)ccc2[nH]1)OC c1(C(N(CCCNC(c2c(C)noc2C)=O)CC)=O)cnc2ccc(C#N)cn12 N1(C(c2ccn(C(C)(C)C)n2)=O)CCCC1(C)CNC(C1CCSC1)=O CC1CN(C(c2conc2CNC(c2n[nH]c(O)n2)=O)=O)CC1C C1CCN(C(c2c[nH]nc2C2CC2)=O)C12CC2.c1(CC(=O)NC)ccc(Cl)nc1 CCC(C)C(O)C(C)C(=O)NC.c1(C(N2CC(O)C2)=O)cc(C)n(C(C)C)c1 c1(C(=O)OC)cc(S(=O)(=O)NCC2CCC=CCC2)on1 CCC(c1ccccc1)=CC(=O)N(CCC(C)NC(C1(N(C)C)CC1)=O)C c1(OC)ncc(C)cc1-c1ccc(CNC(c2cc(F)ccc2O)=O)nc1 c1(C(=O)NC2CCCC2NC(c2ccc[nH]2)=O)ccc2cnsc2c1 c1(C(=O)NC)cccc(NC(c2csc(Cl)n2)c2nnnn2CCCF)c1C N(C(=NCCF)N1CCC(c2cccc(Cl)c2)CC1)C1C(SC(C)(C)C)CC1 C1(CC(C)C)(C(=O)NCC(C)(O)CN)CCCC1 CCCC(C#N)C(=O)NCC(C)(C)NC(C1CCCCN1C(c1ccco1)=O)=O C12(C(=O)NCC(C3CCCCC3)NC(CCSCC)=O)CC(CO1)C2 CC1CCC=C1C(=O)NC(CC(N)=O)C(=O)NC(c1nnnn1C)C c1(C(N2C(CNC(C3SCCS3)=O)CCCC2)=O)coc2c1CCCC2 N1(C(c2n[nH]c(C)c2O)=O)CCC2(CCCN(C(c3c[nH]nc3Cl)=O)C2)CC1 C(=O)(CC(C)(C)C#N)NC(CC)CNC(C1(c2cc[nH]n2)CCC1)=O N1(C(CN(CCC)C)=O)CC23CCCCC2(C1)CN(C(=O)CN1CC2CC2C1)C3 C1(COC(C)(C)C)CCN(CC(C)(C)CC2CCOC2)CC1 Cc1cnc(C(F)(F)F)c(C(=O)NC2CC3CCC2N3C(c2cc[nH]c2)=O)c1 c1(C(=O)N)csc(C)c1C.C1(CNC(C2C(OC(C)=O)C2)=O)CCCC1 N1(c2ccn(C)n2)CCC(C(=O)Nc2cc(C(=O)O)nn2CCO)C1=O Cc1nc(C(=O)NC2CCN(C(=O)CN(c3ccncc3)C)C2(C)C)cc(O)n1 CCC(C=O)C(F)(F)F.c1(C(NCC)=O)ccc(C2CC2)c(Cl)c1.C1CC1.N C1(NC(C(CCC)C)=O)CC2(CCCN(C(c3nn(C)c(C)c3N)=O)C2)C1 N1(C(C(CCC)NC(=O)CCCC(F)(F)F)=O)CC(O)CC12CCCC2 N1(C(c2nccc(OC)c2)=O)CCCC(C)(C)C1.C1(C(=O)N)CC1.C1CCC1 c1(C(N2CC3CCC2CN3C(c2[nH]cc3c2CCC3)=O)=O)noc2ncccc12 c1(C(N2CCC(C3N(C(C4C(C)(Br)C4)=O)CCC3)C2)=O)cccc(SCC#N)c1 N1(S(CC2(C#N)CCNC2)(=O)=O)CCC(Cc2cc(F)cc(F)c2)C(O)C1 c1(OC)nc(C(C(=O)NC2CCCC2)N(C)C(c2cccc(Cl)c2)C)ccc1C Cn1nc(C(=O)NC2CCCC(NC(c3ccc(C(N)=O)cc3)=O)C2)c(Cl)c1Cl n1(CC)c2ccccc2c2cc(CNCc3cc(C)no3)ccc12 C=C(C)CCCC(=O)NCC1CC(OC)CN1C(c1cccnc1)=O CC1CCN(C(c2cccc(Cl)c2)=O)C(C)C1NC(=O)C(c1ccccc1Cl)C C(=O)(C1=C(C2CCOC2)N(CCC2CC2)C(=S)NC1c1cncc(F)c1)OCC C1(NC(N2C(C#C)CCC2)=O)CC2(C1)CC(C(N1CCOCC1)=O)C2 Cc1c(Br)ccc(C(=O)N(C(C)CNC(c2cnc(Cl)s2)=O)C)c1N c1(CC)c(C(=O)NCC(C)(C)NC(C2CCC(C)S2)=O)cnn1C C(=O)(C(CNC(c1sccc1Cl)=O)C(C)(C)C)NC(C)CCc1cn[nH]c1 CCC(C(=O)N1CCN(C(C2CCCCCC2)=O)CC1c1ccnn1C)C(C)C C=CCCCCCC(=O)NCC(C(=O)NC(CC(=O)NC)C1CC1)C(C)C CC(C)C(F)C(=O)NCCN(C(=O)C(C1CCCCC1)O)CCc1ccccc1 c1(C(N2CC3C(NC(C45CC=CC(C4)OC5)=O)C3C2)=O)cnc2ncccn12 CC1CC(=O)CCC1C(=O)NCCCOCCC(=O)NOCC(N)=O c1(C(=O)NCC(C2CCC2)NC(CN(CC)CC)=O)cccc(F)c1.O c1(CC(=O)NC2C(C)N(C(c3cnccn3)=O)CCC2)csc2ccc(Cl)cc12 N1(C(CC=CCC)=O)CCn2nc(C)c(CNC(=O)C(CCOC)OC)c2C1 c1(C(N(CCC=O)CCCO)=O)cc(C)nc(C)c1.C(C)(CC)(C1CC1)OC c1(OC)ccc(NC(C2CN(C(=O)C)C2)=O)cc1.C1(CC=O)CCC1.C Cc1cc(NC(C2C3CCC(C3)N2C(c2cnc(C)s2)=O)=O)nc(Br)c1 C(=O)(C1=NOC(CNC(=O)CCn2cccc2)C1)NC(C#C)CCC C1(C(N2C(C)CC(C)(C)C2)=O)NC(=O)OC12CCC2 C1CN(C(C2CC(=O)N(O)C2)=O)C2(CCCC2)C1.c1(C=O)cc2c(s1)CCC2.N C1(C#CC(=O)NCC(=O)NCC(=O)N)(CC)COC1.C(C(F)F)N(CC)C n1(CC)ncc(C)c1C(N1CCC(C)CC1)C(=O)NCCCOCC1CC1 C1(C(N(CC(=O)NCC(C)(C)C2CCC2)CCOC)=O)CCN(C)C1=O c1(SC)cccc(F)c1C(=O)NCCC(=O)Nc1ccccn1 C1CN(C(=O)CC2(C)CCCO2)C2(CCC2)C1.c1(CC)ccc(C=O)c(O)c1.N c1(C(=O)N)ncc(F)cc1F.c1(C(=O)NC2CCC(CC)C2)cn2c(n1)SCC2 C1(CCOC)(C(=O)O)CCN(C(C2CC(=O)N(CCc3ccccc3)C2)=O)C1 C1(C(N(CCC)C2CC2)=O)CCN(C)C1=O.C1(COC)CC1C=O.C C1(OC)CC2(C1)CC(C(=O)NC1C3CCN(C(=O)C4=CCCC4C)C13)C2 N1(C(C(n2ccc(C)n2)(C)C)=O)CCC2(CCCC2NC(c2ccoc2)=O)CC1 c1(-c2c(CC)occ2)nc(-c2ccnc(-n3nc(C)cc3C)c2)nn1C1CCC1 C(=O)(C#CCNC(=O)C=CC(F)(F)F)NCCC1(COC)CC1 c1(C(=O)NCCC(C)NC(=O)C(C)Oc2ccccc2F)ccnc2ncnn12 CCCC(CC)NC(c1nocc1C(C)(C)C)c1nnnn1C C(=O)(C1CCOc2ccc(Br)cc21)NC1C(C)(C)CN(Cc2ccccc2)CC1 c1(CCSC)nc(-c2cccc3c2CCO3)n(C2CCCc3ccccc32)n1 C1(C(N2CCN(C(CS(CC)(=O)=O)=O)CC2C2CC2)=O)CCC2(CCCC2)CC1 N1(C(CNC(C)=O)=O)CCN(C(c2c(F)c(C)nn2C)=O)C2(CC2)C1 CCCC(CC)CC(=O)NC1CN(C(c2nccc(Cl)c2Cl)=O)CC12CC2 Cc1ccc(F)c(-c2cn(CCCCCCNC(C3C=CCC3)=O)nn2)n1 c1(C(=O)NC(CN(C(CCCC)=O)CC)C)cc([N+](=O)[O-])ccc1Cl N1(CC)CC(COC(C2CCC2OC(C)(C)C)=O)OC1=O C1(CN(C(=O)Cc2cscn2)C)CCCN1C(=O)CN(C1CCCC1O)C N1(C(C2C(C)CC2)=O)CCS(=O)(=O)C(CC)C1.n1(CC=O)cc([N+](=O)[O-])cn1 C1(CC(=O)NC2(COC)CN(C(=O)CCC(C)(C)F)C2)CCCCC12CC2 c1(OC)ccc(O)cc1C(=O)N.C12(C=O)CCC(F)(CC1)C2.C(CC)C(C)C C1(NC(=O)C=CCF)CN(C(C2CN3CCCC3CO2)=O)CCC12CCOCC2 N1(C(C2CC(CCC)C2)=O)CCCC(C(N2CCC(CCOC)CC2)=O)CC1 N1(C(C2N(C(C(CC=C)OC)=O)CCC=C2)=O)CC(F)(F)C(F)(F)C1 C1(CC=C)(NC(=O)C2=COCCO2)CCN(C(=O)CC2CCC(O)C2)CC1 C#CCCC(C(=O)N1CC(O)CC(O)C1)NC(C1CC2C(C1)C2(C)C)=O C(=O)(CC1C(=O)Nc2ccccc21)NCC1CCN(C(C2C(C)C2)=O)C1(C)C Cc1cnc2c(C(=O)NC(C3(O)CN(C(C4COC4)=O)C3)C)cccc2n1 C(=O)(C(C)P(C)(C)=O)N1CC(n2c(C(=O)OC)nnc2)C1 N1(C(COCCCC)=O)CC(C(N2C(CC)CCC2C)=O)CC(C)(C)C1 c1(C(=O)NC2CC(C)(NC(=O)CS(=O)(=O)CCO)C2)nc2ccccc2[nH]c1=O c1(CN2CCC(O)(C(=O)Nc3cncc(CC)c3)C2)c(O)ccc(F)c1Br S(=O)(=O)(C1CCCCC1)Nc1ccc(C(=O)Nc2cnc(C)nc2Cl)nc1 C1(NC(CNC=O)=O)CCCCC12CCCN(C(c1cccc3c1OCO3)=O)C2 Cc1ccccc1NC(=O)CNC(c1ccco1)=O C1(CNC(C(C(C)C)SCC)=O)CCN(C(c2c(Cl)cnn2C)=O)C1(C)C C=CCC(C)(C)CC(=O)N(C1CCN(C(c2ccc(F)cc2C)=O)C1)C CCC(C)CC(C(=O)N1CC(COC)C1(C)C)NC(=O)C(C)CC(F)F C(C(C)S(N)(=O)=O)N(C(C(C)OCCCC)=O)C c1(C(=O)NCC(C)N(C(C(CSC)OC)=O)C)c(C)coc1C N1(C(c2cc(N(C)C)ncc2)=O)CC(NC(=O)CCC2CCCOC2)CC(F)C1 O=C(CC(F)(F)C(F)F)NCC1CCCN(C(=O)C2=CCCO2)C1 c1(CC(=O)NC2CCCN(C(CCC(CC)C)=O)C2)ncn2c1COCC2 N1(C(c2ccn(C3CNC3)n2)=O)CC(F)CC1CN1CCC(O)CC1 c1(CC)cccc(CC)c1C(N1CC(F)(C(N2CCC(O)(CO)CC2)=O)C1)=O CC1(C)CC2(CC(CNc3nccc(=NCc4cc(Br)no4)[nH]3)C2)C1 c1(OC)ncc(C(=O)N)cc1C.C(=O)(C(F)OC(F)(F)F)N(CC(C)O)CC CC(CC(C)NC(c1cn(C)nn1)=O)NC(C1CC(C(F)(F)F)C1)=O C1(NC(CC(C)N(C)C)=O)CN(C(C2CCN(C)C2)=O)CC12CC2 Cc1cc(=NCCc2cc(C)on2)[nH]c(N2CCN(c3ccc(Cl)cn3)CC2)n1 CCCC(C(=O)NCC(C12CCC(CC1)C2)NC)C(C)C.c1cc(C)c(F)cn1 c1(C(=O)NCC2C3CN(C(CCC=C=C)=O)C2CCC3)cn2cc(C)ccc2n1 c1(C(N2CCOCC(NC(C(C(C)O)(F)F)=O)C2)=O)cc2c(n1C)CCOC2 C(=O)(C1CCc2ccc(Cl)nc21)NCCCCN1CCCCC(N)C1 N1(C(CCCC(N)=O)=O)CCC2(CCN(C(c3cnc4[nH]cnc4c3)=O)C2)C1 c1(C(=O)NCC2N(C(Cn3c(C)ccn3)=O)CC(O)C2)cc2nc(F)ccc2o1 CCCCC(O)C(=O)N(C)CCNC(=O)CN1CCOC1=O C(c1ccc(=N)[nH]c1)=CC(N1CCC(NC(C2C(CCC)C2)=O)(CF)C1)=O c1(CC)ccc2[nH]c(C(=O)NCC(C)NC(=O)CCCN3CCCC3)c(C)c2c1 CCC(C)(C(=O)NC(CO)C(C)NC(c1cc2oc(C)cc2[nH]1)=O)C(N)=O C1(CC(=O)N(CCCC(C)(C)C)CC)CCCCCC1(F)F.C1(C(=O)N)COC1 Cc1ccc(F)c(C(N2CCCC(C(N3CCC(C)(C)C3C)=O)C2)=O)n1 c1(C(=O)NC2CC(NC(c3c(CC)[nH]cc3)=O)C2)ccccc1.C(C)(C)C CCCCCC(F)C(=O)NC(CC1CC1)C(=O)NC1CN(C(=O)C2CC2)C1 C(=O)(C1=C(C)CCCC1)NC1(C)CCN(C(C2CC(C(F)F)(OC)C2)=O)CC1 N1(C(C(C)OCC=C)=O)CCN(C(c2c(C)nn(C)c2F)=O)CC(CO)C1 c1(OC)ccc(C(=O)NCc2nc(CNC(c3coc(C)n3)=O)cs2)s1 C1(C(N(CCC)C(C)C)=O)C2CCC3(COC(=O)C13)O2.C(=O)C(O)C1CCC1 C1(CC(=O)NC(C2CCN(C(CC(C)C)=O)CC2)C)Cc2ccccc2NC1=O C(=O)C1CCCc2n[nH]cc21.c1(COC)nocc1C(=O)NC1COCC1C.N N1(C(C2C(CC)C2)=O)CCCC2C(NC(c3oncc3C)=O)C(C)(C)C12 c1(C(=O)OC)cccc2nc(COC(c3nc(-c4cccc(Cl)c4)no3)=O)[nH]c12 c1(C(=O)NC(C)C(CO)NC(=O)C=CC2CCCO2)cc(C(N)=O)n(C)n1 C1(CC(=O)NCC2CCC(CC)O2)COCCN1C(=O)CCc1nccn1C C1(C(=O)NCC(CC)NC(=O)C(C)N2CCC2)CCCC12CCOCC2 C(=O)(C(O)CCCc1ccccc1)NCC1CCCN(C(C(=O)NC(C)C)=O)C1 c1(-c2nc(C)on2)ccc(NCC(=O)NC2COC(C(F)F)C2)cc1 C1(c2cn(-c3scc(C(=O)OCC)n3)nn2)CCCCN1C(=O)C(C)C(F)F C(C(C)C(F)C(=O)NCCCC(=O)N(C)C)NC(C(COC)(F)F)=O C(=O)(C(C)(C)C(N)=O)N(C)Cc1ccccc1C.C1(CC=O)OCCO1.N c1(C(=O)NCC2(C)CCCN2C(=O)COCC(F)F)ccc2cccnc2c1 N1(C(c2cc(C#C)cc(Br)c2)C(=O)NCCC)CCN2C(=O)OCC2C1 C=CC1(NC(=O)CN(C(=O)C(C)C(F)F)CCC)CCCCC1 c1(C(=O)NC2C(CNC(C(CC)O)=O)C2)c(Cl)cccc1Cl CCCCC(CNC(c1sccc1C#N)=O)NC(=O)C(C)CCC C(=O)(C1=COCC1)NC(C1CCCC1)CNC(=O)CC1OCCO1 N1(C(c2ccc(CC)cc2)=O)CC(C(=O)NCCCCCC(=O)NC)CC1(C)C CC(CS(C)(=O)=O)NC(=O)C(CC1CC1)NC(=O)CCCc1cnn[nH]1 CN1N=C(CC(=O)N2CCC2CC(=O)N(C2CCNC2=O)C)CC1=O C1(CNC(C(CC)SC)=O)CC(C)(C)CN1C(c1nc(O)c(C)s1)=O c1cccc(F)c1.c1(C(C2CC(NC(NC3C(CC)C3)=NC)C2)=O)ccc(F)cc1 C1(C2CCC2)(C=O)CCC1.CCC(C)C(=O)NCC(=O)NCC1CC(F)C1 c1(C(N(CC(O)C)C)=O)ccncc1.C1(C(=O)N)CC(CC(F)F)C1.C1CC1 c1(C(=O)NC(C)C(CO)NC(C2CCSC2)=O)nccc2ccccc12 C=CCCCCC(=O)NC(COCC)C(=O)NOCc1cccc(C)n1 C(=O)(C1CCCc2nn[nH]c21)NCC(C(C)C)NC(c1ccc(OC)nc1)=O Cc1cc(C(=O)NCC2CCC2)cc(C)c1.c1(C(=O)N)ncccc1C(F)F N1(C(CCN(C(c2cc(C)cc(F)c2)=O)CC)=O)CCC(C)(CN(C)C)CC1 CC1CCCC1N(C)CCN(S(C)(=O)=O)CC12CC(CO1)C2 CCCCC(CC)C(=O)NCC(C)(CNC(=O)Cn1ccnc1CCC)OC C12(C(=O)NCCN(C(C3(CC)CCCC3)=O)C)CCC(O)C1CC2 Cc1cc(NC(CNC(=O)CCn2cncn2)CO)n2nc(C)nc2n1 C1(NC(CCC#C)=O)CN(C(c2ccnc(C)c2C)=O)CCC1F C(C(C(C)C(C)C)NC(c1ccc(OC2CCOCC2)cc1)=O)NC(CSC)=O c1(C(=O)NC2CCN(C)C2=O)cc(O)nc2c1CN(C(c1ccccc1)=O)CC2 c1(C(N2CCC3CN(C(C(C)SCC)=O)CC32)=O)ccc2c(c1)CC(C)(C)O2 Cn1ccc(C(=O)NCCCC(C)(C)NC(c2coc(Cl)c2)=O)cc1=O C1(C2CCN(C(c3cscn3)=O)C2)CCCCN1C(=O)CCF C(=O)(C1=NOC2COCC12)N1C(C)CN(C(C23CC(C#N)(C2)C3)=O)CC1 c1(OCC)cccc(NC(=O)CC(C)NC(=O)C(C)(Cl)Cl)c1 c1(C(=O)NCCCN(C(C2(C(C)C)CC2)=O)C2CC2)ccc2nccnc2c1 Cc1nc(Cl)ncc1NC(=O)C=CCC1CCC1.C1(C=O)CCC(F)(F)C1 CC1=NS(=O)(=O)NC=C1C(=O)N1CC(NC(c2cncn(C)c2=O)=O)CCC1C CS(=O)(=NC(=O)COC1COC1)c1cnn2c1CN(C(=O)C=CI)CC2 N1(C(CC)=O)CCC2CCN(C(=O)CC3CCc4ccccc4C3)C2C1 c1(C(=O)NCC2N(C(c3n(CC)ncc3)=O)CCCC2)cc2cccc(C)n2n1 Cc1nn(CC(F)(F)F)c(C)c1CC=O.C1(CCC)CN(C(=O)CNC=O)C1 Cn1nnc2cc(C(N3CCCN(C(=O)CCS(N)(=O)=O)CC3)=O)ccc12 Cc1cc(C(=O)NC2CCCC(NC(c3ccc(C(C)C)o3)=O)C2)cc(C)c1Cl C1(C(=O)Nc2cnn(CCn3nc(C)c4cccnc34)c2)CCCN2CCSCC12 c1(C(N2CCC(N(C)C(c3cc4c[nH]nc4s3)=O)C2)=O)n[nH]c2c1CCCCC2 c1(CC(=O)NCC2(OC)CCN(C(CCCCC#C)=O)C2)c(F)cc(F)cc1F CCCN=C(NCCC1CCC(F)(F)C1)NCC(n1cc(Br)cn1)C C(=O)(C(C)CC(F)(F)F)NCCCNC(C(C(C)C)C#N)=O C1(CC)(NC(=O)C(C)OCC(C)C)CCCN(C(c2ccc(C)cc2)=O)C1.O CCC1=C(C(=O)NCC2CC3CCC2N3C(=O)C(O)CC(F)(F)F)SCCO1 C12(CNC(c3cccc(C4CCCC4)c3)=O)CN(C(C3CCO3)=O)CC1CCO2 c1(N(C)C(c2c(CNC(=O)C(O)C3CCC3)nnn2C)=O)cc(C#N)ccc1O C(C(C)(O)C(=O)NCC1(C(=O)NC2(C)CCCCC2)CC1)OC c1(OC)ccc(Cl)cc1C(C)OC(C1CC(=O)CCO1)=O N1(C(C=Cc2ccc(C)o2)=O)CC2(CCC2)C1C1CCN(Cc2ccccc2)CC1 C(CCO)(C(F)(F)F)NC(C1N(C(c2cn(CC)nc2)=O)C(C2CC2)CC1)=O c1(CC)ccc(C(N2CCC(OC3CC3)CC2)C(=O)NC2(C)CC2)cc1C C1(OCC)CC(O)C12CCN(S(=O)(=O)c1ccccc1C(F)(F)F)CC2 C1(CC(=O)NC(CNC(c2c(Br)c(C)n(C)n2)=O)C)Cc2ccccc2O1 C1(C#N)(C(N(C(c2cn(C3CCOC3)nn2)C)C)=O)CC(F)(F)C1 N1(C(C2C(COC)C2)=O)CCOCC1CN(C(=O)C(CCSC)NC=O)C C1(C(=O)NC2CCN(C(COC3CCN(C)CC3)=O)C2)CCC(=O)N(C(C)C)C1 N1(C(C(CC)F)=O)CCOC2(CCN(C(c3c(C)oc(C)c3C)=O)CC2)C1 C1(C(N(CCCNC(=O)CCC2CNC(=O)N2)C)=O)CC(=O)NC(=O)N1 c1(C(=O)NC2(CNC(C3C(C)C3C)=O)CCCCC2)c[nH]c(=O)c2ccncc12 c1(C(N2C3C(NC(c4n(C)nnc4)=O)CC(C3)C2)=O)cc2sccc2n1C c1(C(=O)NC(COC)CNC(=O)CC2NC(=O)NC2=O)cccc(C)c1Cl c1(C(N(C(C)C)CCO)=O)coc(CNC(=O)CN2CC(C)(C)C2)c1 N1(C(c2c(CC(C)C)nc(C)s2)=O)CC2CCN(C(=O)CCCS(C)(=O)=O)C2C1 c1(OCC=C)ccc(CC(=O)NCCC2CCN(C(=O)CC)CC2)cc1 O=S1(=O)CCC(CO)(NCCCn2cnnn2)CC1 C1(NC(COCC#C)=O)CN(C(=O)CCC(=O)c2cccs2)CC1C c1(C(N2C(C)C(NC(c3csc(Br)c3)=O)CC2)=O)cc(N)cc(O)c1 c1(C(=O)NC(CNC(c2cccc(C(C)C)c2N)=O)CO)cccn2ccnc12 c1(CC(N2CCC(N(C(c3ccccc3O)=O)CC)C2)=O)cc(O)nc(O)n1 C(CC(N=c1[nH]c(=NCc2cccnc2C)[nH]c2c1CC(C)CC2)C(C)C)OC CCC(O)C(=O)NCC1C(Cn2cc(CCC3CCCO3)nn2)C1(F)F C1(CC)CN(CC)CCS1(=O)=O.C1(C(=O)N)CC1CC=O.C1CC1.C=O N1(C(c2c(C)scc2)=O)CCCC(C(=O)NCC2C(C)(C)C2(F)F)C1 c1(-n2cc(Cn3c(OC)ccn3)nn2)cc(C2CCCC2)nn1C Oc1cc(F)c(CNC(=NCC2CCCO2)NCC2C=CCC2)c(F)c1 N1(C(C2C(OC)CN(C(c3cc(CO)ccn3)=O)C2)=O)CC(=O)NC(=O)C1C CC1CC=C(C(=O)N(CCCC(=O)NCCCOCCCO)C)CC1 C(=O)(C(F)CC(CC)CC)N.N1(C(C2(CC#C)CCOC2)=O)CC2(CC(C)C2)C1 Cc1cc(C(=O)N(C2CC(NC(c3cn(C4CCOC4)nn3)=O)C2)C)ccn1 C1(C(C)(F)F)CN(c2nnc(C(F)(F)F)s2)CCO1 c1(-c2n(C)c(N3CCC(N)(c4cccc(F)c4)C3)nn2)ccnc2ncccc12 N1(C(Cc2c(SCC)cccc2)=O)CCC2CCN(C(=O)CC(C)(C)F)CC12 C1(NC(C(=O)Nc2cc(C)cn3c2ncc3)=O)CCc2nc(N(C)C)ncc2C1 c1(OC)c(C(=O)N)cc([N+](=O)[O-])cc1Cl.C1C2CC1N(C(=O)CC)C2.C(C)=O c1(SCC2(CC=O)CC2)ccccc1.c1(C=O)cc(C2CC2)on1.C(C)C C1(CC)CC(C(N2CCCC(CNC(c3cnn(C)c3SC)=O)C2)=O)CCO1 Cc1ccc(C(=O)NC2CN(C(c3cscc3Cl)=O)CC2n2ccnn2)n1C c1(C(=O)NCCCCNC(CCC2CCC(C(N)=O)O2)=O)csc2nnsc12 N1(C(C(N(C)C)C2CC2)=O)CCOCC(CNC(=O)Cc2cc(F)ccc2F)C1 C1CCN(C(c2cnc(C(C)C)nc2)=O)C1(C)C.c1(OC)cc(C(=O)N)n(C)n1 c1(C(N(CCCNC(=O)CNS(N)(=O)=O)CC)=O)cnc(S)[nH]1 CN1CCN(C(C2CC3(CCC3)C2)=O)CC1CNC(=O)CC1CC=CCN1C c1(CC=CCCC)ccc2c(c1)CCCN2Cc1cn(-c2cccnc2Cl)nn1 c1(C(N2CCC(NC=O)CC2)C(=O)NCCCC)ccc(C)cc1C.C(C)C.O c1(C(N(C2CCCC2)CCNC(=O)Cc2c[nH]nc2O)=O)cc2c[nH]cnc-2n1 C12(NC(c3c(=O)ccn(C)c3)=O)CCCCCC1N(C(C1CC(=O)N1)=O)CC2 c1(CC)cc(C(=O)NCC2(C)CC23CCC3)ccn1.c1(C=O)[nH]ccc1C.N N1(C(=O)C=Cc2cn[nH]c2)CCC(O)(CNC(=O)C(O)c2ccco2)C1 c1(OCCN(CCNC(CSCC#C)=O)C(C)=O)c(CC)cccc1F CN1CC(NC(C2OCCC2NC(C2(C)C=CCC2)=O)=O)CC1(C)C C1(CC)CCN(C(C2CS(=O)C2)=O)C1CNC(C1C2CCC(=O)C12)=O CC1(C(=O)NC2CC3CC4C(C3)C24)CCCN(C(=O)Cn2ncccc2=O)C1 C1(C(C)CC(=O)O)CCCN(C(=O)CSCc2ccccc2Cl)C1 C(=O)(CCCCC1CC1)N1CCC(CNC(c2cccc(O)n2)=O)C1 c1(C(=O)OC)cnc(Nc2cccc(CNC(=O)C(C)=O)c2)nc1 c1(C(N(C2CCNCC2(C)C)c2ccnc(SC)n2)=O)cc(Cl)c(Br)c(Cl)c1 C1(NC(c2c(OC)cncc2)=O)CCN(Cc2cncc(C)c2)CC1(C)C c1(C(=O)NC2(CO)CN(C(C(c3cscn3)N(C)C)=O)C2)cc(F)c(F)cc1Cl CCCCCS(=O)(=O)CC(=O)NC1(C)CC(NC(=O)C(F)C(C)(C)O)C1 C1(NC(c2ccc(OC)cc2Cl)=O)CN(C(C2CC23CC3)=O)CC2(CCC2)C1 c1(C(N2CCC2)=O)cc(O)cc(F)c1F.c1(C(=O)N)ocnc1C(F)(F)F.C CC(CC(F)(F)F)N(C(=O)CC1CCCCN1C(=O)C(c1ccnn1C)C)C c1(C(=O)NCC(C)NC(=O)COCC2(F)CC2)ccco1 Cc1cc(F)ccc1C(N1CCOC(CNC(=O)C(n2cnc(C#N)n2)C)C1)=O C(=O)(C(F)CC1CN(C(c2ccc(CO)s2)=O)C1)N1C(COC)CC1 c1(OC(C2CC3(COC3)C2)=O)ccc2c[nH]nc2c1 C12(C=O)CC3CCC(CC(C3)C1)C2.C1CS(=O)(=O)CC1.O=CC=C1CCC1 c1(N2C3C(NC(C(C(CC)CC)C)=O)CC(CC3)C2)nc(=N)[nH]c(Cl)c1[N+](=O)[O-] c1(NC(=O)NCC2C3CN(C(C(CC)C(C)C)=O)CC32)c(C)nc2cccnn12 Cc1cc(C(=O)N(CCCNC(c2nccn2C(C)C)=O)C)c(Cl)cc1Cl C1(N(C(C2CC=CC(NC(C(CO)OC)=O)C2)=O)C)CC2CCC1CC2 Cc1cccc(C(=O)NC2COC3(C)CC2C3)c1F.C1(C)(C=O)CC(C#N)C1.N C#CCC(C(=O)NC(C)(C)CN(C)C(C1(n2cnnn2)CCOCC1)=O)C1CC1 c1(N2CCC(CNC(CNC(C=C)=O)=O)C2)ncnc2cc(OC)ccc12 CCCCS(=O)(=O)NC1CCCC1C(=O)Nc1ncccc1C C1(NC(C(CCCC)NC(c2cc(C)cc(C)n2)=O)=O)CC1C1CCCCC1 Cc1cc(C)n(C2CCCN(Cc3cnn(C)c3Br)C2)n1 Cn1ccc2cc(C(N3CC(O)(C(C)(C)C)C3)=O)cnc12.C(=O)(C(C)(C)CF)N n1(CC(N2C(C)CC(NC(c3c(O)ccc(C)c3)=O)C2)=O)cc2ccccc2n1 C1(C(N(C2C(C)C2)C)=O)CC=CCC1NC(=O)CCCC1CCCO1 c1(C(N2CC(SC)C(NC(=O)C(C)CF)C2)=O)cnc(N)c(Cl)c1 Cc1nn(C)cc1C1=NOC(C(=O)NC2CC3CCC3C2)C1.C(C)(C)C.C(=O)N C(=O)(C(C)S(N)(=O)=O)NCc1c(CN(C(C(C)CO)=O)C)cccc1 C(=O)(C1CCc2scnc21)NC1(CNC(Cn2c(C)cc(C)n2)=O)CCOC1 CC(C)CCC(=O)NC1COCC1CNC(c1ccc(N(C)C)nc1)=O CCCCC(CN=c1[nH]c(COC)nc(=N)[nH]1)NC(=O)C(C)NC(N)=O C(C)(C(C)(C)C(=O)NCCC1CCCO1)NC(C(CC=C)NC(C)=O)=O C1(CC)CCCN(C(=O)CCS(N)(=O)=O)C1C(N1CC(OCC(F)F)C1)=O C(=O)(C1=C(C)CCCC1)N(C1CCN(C(C2CC2F)=O)CC1)CCCC CC(C)(CCC#N)C(=O)N1CC(C)C2(CC2)C1.C12(C=O)CCCC1(C(N)=O)C2 C=CC(CCC)CC(=O)N1CC2CCN(C(=O)Cn3cc(Br)c(C)n3)CC12 c1(C=O)nn(C)c2c1COCC2.C(c1cocn1)=CC(=O)NCC(C)OC.N CCC(N=c1cccc(S(=O)(=O)NCCCCc2ccccc2)[nH]1)C(C)O c1(OC)cc(Nc2cccc(NC(C3(C(C)C)CCC3)=O)c2)nc(OC)n1 c1(SC)cccc(C(=O)NCC(C)CO)c1.C1(C(=O)N)OCCC1C(F)(F)F c1(COC)ccc(C(=O)N)cc1.C1(C(N2CCC2)=O)CC(=O)N(C2CC2)C1 Cn1ccc(C(=O)NCC2(CNC(c3ccc(C(F)F)o3)=O)CC2)c1 c1(C(N2C(CCNC(CCC(C)OC)=O)CSCC2)=O)sc2nnc(S)n2c1C C1(COC)N(C(=O)CC2C=CC(NC(=O)C(CCOC)O)C2)CC1(C)C C(=O)(N1CCC(C(=O)NC(CCO)C2CCCC2)O1)c1ccc(CC)[nH]1 C1(NCC2CC(NC(=O)OC(C)(C)C)C2)COc2ncccc2C1 C=CCC(C(=O)N(C1(C(=O)NC)CCC1)C1CC1)C(C)C.C1C2CCCOC12 c1(COCCCN(C(c2ccc(C)o2)C(=O)NC2CC2)C)ccc(F)c(Cl)c1 C(CC(C(=O)NCc1cc(C)ns1)NC(c1ncccc1F)=O)OC N1(C(c2cc(CNC(C3CC(=O)C3)=O)[nH]n2)=O)CCC(CO)(CO)C1 Cc1ccnc(Cl)c1C(=O)NC1CCCCC1CNC(=O)Cn1cccnc1=O S(=O)(=O)(c1cc(F)ccc1C)N1CCC(C)(C(=O)NC(CC)C(C)O)C1 C1(NC(C2CCC2)=O)CCCC2CN(c3cc(CC4CC4)ncn3)CC12.C1CC1 N1(c2nc(C)nc(-c3ccco3)c2)CCC(C2(NC(=O)C3=CCC3)CC2)C1.C1CC1 C1(F)(CNC(C2ON=C(CC)C2)=O)CCCN(C(C23CCC2CC3)=O)C1 C1(CN(C)C(C2CCC2)=O)CCCCN1C(C1CC1(Cl)Cl)=O.c1ccccc1.C O=C(C1=CCN(C(c2ccnc(O)c2)=O)CC1)NCC1(O)CCCC1 C1(NC(c2nc(OC)c(C)s2)=O)CN(C(=O)Cn2nnc(C)n2)CCC1C N1(C(C)C)CCCC(OC(C2(COc3ccc(Cl)cc3)COC2)=O)C1 C(=O)C(C)C(C)(C)c1ccccc1.C(C)(CO)NC(C1(C(=O)NC)CC1)=O c1(C(N2C3CN(C(c4c(C)[nH]cc4)=O)C(CC3)C2)=O)ccc2c(c1)NC(=O)CS2 c1(C(N2CC3CCC(NC(C45COCC4C5)=O)C3C2)=O)cnn2cccnc12 C(=O)(CC(C)(C)F)NC(C1(O)CN(C(c2ncn(C)n2)=O)C1)C CC1(C)CCN(C(C2CC(F)(CO)C2)=O)CC1C.c1(C=O)c[nH]nc1[N+](=O)[O-].N c1(C(=O)NC2C(CO)CCN(C(C3CCN(C)CC3)=O)C2)cc2n(c1)CCOC2 C1(NC(c2cncc(OCC)n2)=O)COC2(C1)CN(C(c1ccccc1Br)C)C2 c1(OC)cc(N)c(Cl)cc1C(=O)Nc1cccc2[nH]ccc12 Cc1cccc(SCC(=O)NCCCN(CCC)C)c1.c1(C(=O)N)ccn(C)c1 C1(NC(c2nccc(C)n2)=O)CCN(C(=O)C(C)C2CCC2)CC1CO C1(CN(C(=O)C=CBr)C)CCCCN1C(c1cccnc1F)=O Cc1cccc(Br)c1CC(=O)NC(C)C(c1ccc(Cl)cc1)O C1(NC(C2(CC)CCCCC2)=O)CC2CCC1C2.c1(CC(=O)N)cccc(O)c1 C(=O)(C(C(=O)N(CCC(C)NC(=O)CCn1cnnn1)C)OC)OCC C1(C#N)(C(=O)NC(C)CCNC(=O)C(F)(F)c2ncccn2)CC12CCOCC2 C(C(C(C)C)NC(=O)CC(C)(C)O)(C1CCCC1)NC(C(F)=CC)=O CC1CCCCC1C(=O)NCC1CN(C(c2cc(C(N)=O)c[nH]2)=O)C1 C1(F)CCN(C(c2ccc(C3CC3)nc2)=O)C1.CC(C(C)(C)C)=CC(=O)N.C N1(C(C=CC(CC)=CC)=O)CC(CCNC(=O)C)OC(C)C1.CC(F)F c1(C(N2CC(CNC(c3ncn4c3CCC4)=O)C2)=O)scc2c1OCCO2 c1(C=O)cc(C(F)F)no1.C1(C=O)(C(=O)N(CCC)C2CC2)CC1.CN c1(-c2c(C)csc2)c[nH]c2ncc(C(=O)Nc3c(O)ncnc3O)cc12 C(=O)(CC1=CCCC1)N1CC(CNC(c2nc(CCOCC)oc2)=O)C1 C(CCC1CC1)(C(=O)NC1CC(C)(C)C1)NC(COCC#C)=O C1(C(=O)NC(C2CCN(C(C3(CCO)CC3)=O)CC2)C)CC(O)C(F)C1 C1(CC(=O)NCCN(C(C2CC=CCO2)=O)CC2CC2)CCC=CCC1 c1(CC(=O)N(C2CCN(C(=O)CCC(C)(C)F)C2)C)csc2c(F)cccc12 C1(COC)(C)CCN(C(c2ccc(F)cc2)=O)C1.C1(O)(CC=O)CCC1.N CCCCCC=CCC(=O)N(C(C)C(=O)N(C1(COC)CC1)C)CCC Cc1ccc(C(=O)NCCC(C)N(C)C(C2CC(F)(F)CS2)=O)cc1C#N C1(C=O)CC(F)(F)C1.N1(C(C(C2CCC(=O)N2)C)=O)CC(C(N)=O)(C)C1 C(C(=O)NCC1C=CC(NC(c2c(N)cccc2Cl)=O)C1)(C(C)(C)C)OC CC1(C)CCN(c2ccc(S(=O)(=O)N3CC4CCC3C4)cc2F)CCS1(=O)=O N1(C(c2c(CC)n(-c3ccccc3Cl)nc2)=O)CCCCCC1CC(C)O N1(CC(=O)NC2CCCC(C(=O)OC)CC2)C(=O)NC2(CCCC2)C1=O CCC(CNC(c1coc(COC)n1)=O)C(C)C Cc1cc(C(=O)NCCOC2CCN(C(c3cnc(O)s3)=O)C2)cc(F)c1 C(CCC(O)C(=O)NCc1ccc(Cl)cc1)NC(C(=Cc1ccccc1)C)=O C=CC1CCCN1C(=O)C(C)(CO)NC(=O)C(C1CCCC1)OC C(=O)(C1=C(Cl)CCC1)NCC1(CNC(=O)CCC(=O)N2CCOCC2)CC1 CC(O)C(C)C(=O)NC1CCC(NC(=O)C(O)(C2CC2)C2CC2)CC1 N1(Cc2c(C)noc2C)CC2CCN(C(c3cc(Cl)ncn3)=O)C2C1 CC(C)C(CCNC(=O)C(C)CC1CCCC1)NC(=O)Cc1ccccc1O c1(OC)cc(C(N2CCN(C(c3ccncc3O)=O)CC2)=O)cc(Br)c1Cl Cc1cccc2cc(C(=O)NC(C3CCN(c4ccnc(CO)n4)C3)C)sc12 C#Cc1ccc(C(N2CC3CC(C2)C3NC(=O)C(C)OCC(C)C)=O)cc1Cl c1(C(=O)NC2CC3(C2)CC3)n[nH]c2c1COCC2.C1(C(=O)N)CC12CC(O)C2 CC1(NC(=O)C(c2cccs2)NC(C2CC2(F)Cl)=O)CC2(CC2)C1 C1(CNC(=O)COCCF)CN(C(c2ccccn2)=O)CCCO1 N1(C(c2c(C)nc(O)s2)=O)C2CCC1CC(NC(=O)CC(C)C1CCCC1)C2 CCCCC(C(=O)NC1CCN(C(=O)C=CC(=O)N(C)C)C1C(C)C)C(C)C N1(C(CCC(=C)Cl)=O)CCC2(C1)CN(C(c1ccc(COC)cc1)=O)CC(C)O2 C1(CNC(c2csc(C)c2C)=O)CN(C(=O)CCOC(C)CC(C)C)CCCO1 C1(C)(C(N2CCC(CNC(C3CCCN(CCC)C3)=O)CC2)=O)CCCNC1=O c1(C=O)ccc(F)c(Cl)c1.C1(CNC(=O)CN2CCCC2CO)CCCCC1.N C(C(CC(C)C)C(=O)NCC(C)C(F)C(=O)NCCc1ccn(C)n1)OC CC1=C(C(=O)NCC2CCCCN(C(c3cc(C(F)(F)F)c[nH]3)=O)C2)CCCC1 C(=O)(CC(C)(C)COC)N1C(CN(C(C2(CCCC)CCC2)=O)C)COCC1 Cc1nc2c(C(N3CC=CC(NC(=O)CNC(N)=O)C3)=O)cccc2o1 C#CCCCCC(=O)NCC12CCC(CN1C(=O)C(C)Sc1ccc(C)cc1)C2 N1(C(C2(CC#C)CCCC2)=O)CCC(C(=O)N2C3CSCC2C3)=C(F)C1 C1(CNC(CC(C)C2CCCO2)=O)C2CCCC1N(C(c1ncc(Cl)n1C)=O)C2 Cc1cc(CNC(C2CCN(C(=O)CO)C2)=O)cc(O)n1.c1cc(F)ccc1F C12(CNc3cn(C4CC(N)C4)nn3)CCC(CC1)CO2 C=CC1(CC(N2CC3CC2C3NC(=O)C(O)C(C)C)=O)CCOCC1 C1CCC2COCCN2C(=NCc2cnn3ccc(C4CC4)nc23)N1 C1(CC)CN(C(c2ccc(O)cc2)=O)CCN1C(c1cnc(Cl)cn1)=O CCC(C)CCC(=O)N1CCOC(CCNC(c2ncc(C)cc2Br)=O)C1 CC#CCC(C)N=c1[nH]c(NC2CC(CO)C3CC23)nc2c1CCCCCC2 N1(C(c2cc(C)nc(O)c2)=O)CCCC2C(CCCN2C(C23CC(F)(C2)C3)=O)C1 CC(C)C(F)C(=O)NC1CC(NC(=O)CCc2nnc(-c3cccc(Cl)c3)o2)C1 N1(C(C2OCC(C)C2)=O)CC23CCCC2(C1)CN(C(c1ccc(=N)[nH]c1)=O)C3 C1(NC(CSCC)=O)CCC(C)N(C(=O)Cc2cncnc2O)C1 C(=O)(CC1=CCN(C)CC1)N1C2CC(C1)C2.c1(SC(C)C(=O)NC)ccccn1 N1(C(C(F)=CCC)=O)Cc2ccccc2C1CNC(=O)CCCC(=O)N(C)C C(=O)(C(CC(C)C)C(N)=O)N(CCCCCNC(C(C)(C)OC)=O)C N(C1c2ccccc2CCC1N(C)C)C(N1CCC(OCC#C)CC1)=O C1CC(C)(C)CN1C(=O)Cc1ccccc1F.Cc1nc(C=CC(=O)N)cs1.C C1(C#CC(=O)NC2(C)CC(C(=O)N(CCS(C)(=O)=O)C)C2)(CC)COC1 C=CC(C)(O)CC(=O)NC1COCC1C(=O)NC1(C)CCSCC1 C=CCC(CC(F)F)C(=O)N(C)CC1CCCC(NC(c2csc(CO)n2)=O)C1 N1(C(C2CCCCC(C)(C)C2)=O)CCCC2(C1)CN(C(C1(C)CC1(F)F)=O)C2 C1(C)(CNC(=O)NCC2(SC)CCCC2)CCS(=O)(=O)CC1 CC1CCN(C(c2csc(CNC(=O)C(c3ccnn3C)O)c2)=O)CC1O CCCCCC(CC)C(=O)N1CCC(C(=O)NC2(C)CCC(C)(C)C2)C12CC2 CCCC(C(O)C(=O)Nc1ccc(F)cc1CO)NC(=O)CCOCCOC C(CCCCCCCO)=CC(N1CCCC(NC(C(C2CCC2)OC)=O)C1C)=O CC(C)(C)C(F)(F)CNC(=O)Cc1csc2cncn12 CN=c1cc(C(=O)NCC2CC(C)CCN2C(=O)Cc2ncc(C)s2)cc[nH]1 C1(N(C(=O)C(Cc2ccoc2)NC(=O)CC2(C)CC2)C)CCCCC1(C)C c1(C(=O)O)ccccc1C=O.C12CC1CN(c1cc(C(F)(F)F)ncn1)C2.CC C1(C)(C(=O)Nc2ccc(OC(C)C)cc2)CCCN(C(c2cccc(Br)c2)=O)C1 CC(C(=O)NCC1CCC1NC(c1ccccc1OCCF)=O)C(C)(F)F CC1Cc2cccc(C(=O)NCC(F)CNC(c3cccc4ncnn34)=O)c2O1 c1(NC)cnccc1C(N1CC(C(=O)N(CC(O)C2CCC2)C)C(C(C)C)C1)=O C1(NC(C)=O)C=C(C)CCC1.C(C)(C)(C(=O)C(n1ccnn1)O)OCCC.C c1(C(=O)NC(C2OCCN(C(COCCOC)=O)C2)C)ncc(F)cc1F O=C(C1=NOC2(CCN(Cc3ncc[nH]3)C2)C1)N(CCO)CCc1ccccc1 C(c1ccc([N+](=O)[O-])s1)=CC(=O)NC(C)C(C)NC(C1CN(C)C1)=O c1(OCC(CNCc2c(C(C)C)cccc2)O)cnc(F)cc1Cl c1(C(=O)NCCCN(C(CC(C=C)C)=O)CCO)c(CC)nn(C)c1CC C(=O)(CCC(=O)NCCCCNC(C1CCCC(OC)C1)=O)NCCC c1(C(=O)OC)cc(C(C)NCC(Cc2ccccc2)OC)on1 CC(C)CC(C(=O)NC(C)C(F)(F)F)ONC(=O)CN1CC2CC2C1 C1(NC(C(C)N(C)C)=O)CCN(C(C2(S(N)(=O)=O)CCC2)=O)CCC1CO C1(C(N(CCOC)C(C)C2CC2)=O)CC=CCC1.C(=O)CCCc1ncco1 N1(C(CCOCC)=O)CCCC12CCN(C(=O)C=Cc1ncc(C)[nH]1)C2 Cc1nc(O)nc(C)c1C(N1CC(C2(NC(C3CCC(F)C3)=O)CC2)C1)=O NS(=O)(=O)c1cnn(CC(=O)NCCC(O)CNC(c2nn[nH]c2Cl)=O)c1 N(C1CCC2(CC2(F)F)c2ccccc21)c1n(C)c(=O)nc(O)c1 C1(NC(c2ccc(-n3ccnc3)cn2)=O)CC(N=c2[nH]nc(C3CC3)o2)C12CCC2 N1(C(CC(COC)C)=O)CC(NC(c2cnc(OC(F)F)c(C)c2)=O)C2(CC2)C1 c1(NC(C2CC(C)CN2C(=O)CCc2ccc(O)cc2)=O)nc(Cl)nc(Cl)n1 N1(C(CCC=C(C)C)=O)CCC(CCNC(C2C3CCC23)=O)CC1 O=C(CCCC(F)(F)C(F)(F)F)NCCOCCNC(c1ccccn1)=O C=C=C(C)CC(=O)NCC(CC)NC(c1ccc(Cn2cc(Br)cn2)o1)=O C1(NC(=O)CC=C(Cl)Cl)COC2CN(C(C3CCOCC34CCC4)=O)CC12 Cc1cc(=NC(=O)C2(F)CN(C(c3cc(C(C)(C)C)n[nH]3)=O)C2)[nH]n1C C12(CNC(CCCOC)=O)CCC(C1)N(C(c1conc1C)=O)C2 C1(C(N2CC(c3ccon3)C2)=O)CC2(CC2)C1.CC1(C)CC(C(=O)NC)C1 c1(NC(=O)NCC)cccnc1CN(C)C(=O)NCC1CCCC1.C N(C(=NCCCCC(F)(F)F)N1CCOC(CF)C1)Cc1ncc(C(=O)OC)s1 c1(C(N2CCC(N(C(C(F)=CCC)=O)CCO)C2)=O)cccc(Br)c1F C1(F)(C(=O)NC2CC=C(C)CC2)CCCN(C(=O)CC2CCCO2)C1 C1(CNC(C(C=C)OC)=O)CCCC2CN(C(=O)COCC(=O)NC)CC12 c1(C(=O)NC2C(NC(c3c(C)cc(CO)o3)=O)CC2)csc2ccc(F)cc12 Cn1cc2c(C(=O)NCC3CCC(C)(C)NC3)cccc2n1 N1(C(CC(C)C2CC2)=O)CC(NC(=O)C)C(C)(C)C1.c1(C(=O)N)ccccn1 C(C)(C(=O)NCCN(C(=O)CO)CC1CC1)OCC.c1ccsn1 N1(C(CC(CCC)NC(=O)CCCC(=O)C2CC2)=O)CCC2(CCCCC2)C1 c1(CN2C(C(=O)NCC3CC=CCC3)CCC2)c(I)ccnc1Cl C(=O)(CC(F)(F)Cl)NC(C1CCN(C(C(C)NC=O)=O)C1)C S(=O)(=O)(c1cn(C)cn1)N(CC(N1CC(F)(C=O)C1)=O)C1CC1.CC C=CC1CCN1C(C1OCCC1NC(C1CC12CC2)=O)=O c1(C(N2CCN(CCOC(C)=O)CC2)=O)csc2c1CCC(C)(C)C2 C(CCCC(=O)NCCc1cnnn1C)NC(C(C)O)=O c1(OC)ccc(F)c(CC(=O)NC)c1.C1C(C)CCCN1C(C12CSCC1C2)=O c1(NC2(C3CN(C(=O)CN4CCCCCC4)C3)CC2)ccnc2ncnn12 C=CCC(C(=O)NC(C(c1ccccc1)NC(c1ccsc1)=O)C(C)C)N(C)C n1(CCNC(C2CC2c2ccncc2)=O)cc(CN2CCSCC2)nn1 C1(NC(C2C(C(C)C)CCO2)=O)CC2CC1CN(C(c1cnn(C(F)F)c1)=O)C2 c1(C(=O)NCC(C2CC2)NC(C2(CO)CC2)=O)cnc2c[nH]nc2c1 C1(C(=O)N)CCOC2(CCCCC2)C1.C1(C(C)(C)O)(CNC(=O)C)CCOCC1 C(=O)(C(C)(O)CC(F)F)N1CC2(CN(C(Cc3cccc(C)c3C)=O)C2)C1 N1(C(CNC(CC)=O)=O)CCC(NC(=O)C(N2CCCCC2C)=O)CC1C1CC1 C1(NC(C=CC(=O)NC(c2nc(C)[nH]n2)C)=O)CCCCC1C(N)=O C(=O)(CCCC(N)=O)N1CC(CC(C)NC(C2(OC(C)C)CCC2)=O)C1 CCCCC(C)C(=O)N1CC2C(CN(C)C(c3nccc(Cl)c3Cl)=O)C2C1 c1(N2C3CCC(NC(CC=C)=O)C(C3)C2)ncc(Cl)cc1[N+](=O)[O-] CC1CCC(C(=O)NC2CCCC2CNC(C2(O)COC2)=O)CC1 CC1(CNC(=O)CC2(C)CCN(C(=O)CCc3ccsc3)C2)CCCC1O c1(OC)ccc(NC(C2CC(O)CN2C(C2CCCC2O)=O)=O)cn1 C(=O)(C1CCSc2ccccc21)NCC(CC(C)C)(C)NC(=O)CCF C(=O)(C(C)(C)C1=CCS(=O)(=O)CC1)NCC1C(C)CCCC1.C(=O)(CCF)N N1(C(CC=CC)=O)CCC(C)C(F)(F)C1.c1(C(=O)N)nnn(C2CCOC2)c1C C(CCCCC(=O)N1CC2CC2(CNC(=O)CC2(CC)CCC2)C1)=CC N1(C(CN(C(=O)Cc2cncnc2O)CC2CC2)=O)Cc2ncsc2C1 O=C(C1=CCCOC1)NCC1(NC(c2ccc(-c3ncc[nH]3)cc2)=O)CCC1 N(C1CCOc2c(F)ccc(F)c21)C(C(NC(C)=O)=Cc1cccs1)=O C#Cc1ccc(C(N2CC=CC2(C)C(=O)NCC2CC(=O)N(C)C2)=O)nc1 N1(C(c2[nH]c(=NC)sc2)=O)CCCC(C2(NC(=O)Cc3ccc(F)cc3)CC2)C1 CCCC(C#N)C(=O)NC1CC(C(F)C(=O)NC2(CO)CCCCC2)C1 C(=O)(C(C)(C)C(F)(F)F)NC1CC(C)N(C(C2CC2(Cl)Cl)=O)C1 n1(CCCOCC(=O)NC(C(N)=O)C2CCOC2)ccnn1.C1CCCNC1.C C1CC2CCC2C1.C1(CNC(C2(C(C)(C)O)CCC2)=O)OCCC1C(=O)N c1(C(N(CCNC(C2NC(=O)OC2C)=O)CC)=O)nc(C(C)C)ncc1Br n1(CC=C)nnnc1C(CCCC1CC1)NCCNS(=O)(=O)C1CC1 c1(CC(=O)NC(CC)CNC(c2nocc2C2CC2)=O)cnc(O)nc1O C(=O)(C(C1CCc2ccccc21)NCc1cc(CC(C)C)nn1C)OC CN1CCc2c(C(N3CCOC(C(=O)NCc4cnccn4)C3)=O)cccc21 c1(C(=O)N)c[nH]c(=S)cn1.CN(S(N)(=O)=O)CC(=O)NCC1(C)CC1 C1(C(=O)NCCOC(CC)CC)(CNC(=O)CCc2cnccn2)CCCO1 c1(CC=O)ccc(C#N)cc1.c1nccn1C.C(CNC(=O)CO)(C)OC CCC(C)(CO)C(=O)NCC(C1CC1)NC(c1ccc(O)c(Cl)n1)=O N1(C(c2cccc(-c3nnco3)c2)=O)CCOC2CCNCC12 C=CCC(F)(F)C(=O)NC1CCCCCC1NC(=O)C(n1cc(Br)cn1)C C1(NC(C2(CC)CC(F)(F)C2)=O)CCCCC1.c1(CCC=O)cc(C)no1.N CC1CN(C(=O)Cc2cncc(O)c2)CCC1C.C1(C(C)(F)F)(C=O)CC1.N O(P(=O)(CCN1CC(n2cc(C(O)CC)nn2)C(C2CC2)C1)OCC)CC C1(NC(C(C(=C)Cl)(C)C)=O)COC2CN(C(c3ccn4ncccc34)=O)CC12 S(=O)(=O)(c1[nH]c(=NCCC23CC(CO2)C3)ccc1Br)NCc1cccc(C)c1C C1(C)(NC(c2c(C)cccc2C)c2n(CCCC)nnn2)Cc2ccccc2C1 N12C(CCC13CCC3)C(=O)N(C)CCCC2=O.CC(C)CC(=O)N(C)C CCC(CNC(C1CCC1C)=O)(CC)NC(=O)COCc1ccnc(O)c1 C(C(C(=O)NC1C=CCCC1)C(C)(C)C)NC(C1C(C)=CCS1)=O C1(C(N2CC(C=C)C(NC(=O)Cc3[nH]cnc3C)C2)=O)CCc2cn(C)nc2C1 c1(C(N(CC(C)O)CC)=O)noc2c1COCC2.C1(C)(C(=O)N)CC(C#N)C1 C(C(C(=O)N1CCCC1C(C)NC(=O)Cc1ccoc1)N(C)C)OC CC(C)CCCC(=O)NC1(CO)CN(C(=O)COc2ccc(CC(N)=O)cc2)C1 CC(N=[N+]=[N-])C(=O)NCC1CC(O)(CNC(=O)CO)C1.C1CCOC1 c1(C(=O)NC2CN(C(COC(CC)C)=O)CC3C2C3)cc(Br)cc([N+](=O)[O-])c1 C(=O)(C(C)CC(C)(C)C)NC(C)CCN(C(=O)Cc1ccc2c(c1)CC2)C C1(NC(=O)CCN2CCC(F)C2)CC2(CNC(=O)CO)CC1CO2 c1(N2CCC(CC)C2)ccc2cc(S(=O)(=O)N3CCCC(F)(CO)C3)ccc2n1 N1(C(c2nc(C)sc2)=O)CCCCC1CCNC(=O)CN1CCC1C N1(C(c2n(C(CC)C)ncc2)=O)CC(CO)C2(C1)CN(C(c1ccc(F)s1)=O)C2 c1(CC(=O)NC2CCN(C(C3(C=C)CC3)=O)CC2CC)noc2cc(F)ccc12 c1(CC)ccc(CNC(C2CC(NC(c3ccoc3C(C)C)=O)C2)=O)s1 Cc1cc(OS(=O)(=O)Cc2nccc(Br)c2C)cc(N2CCC(=O)NC2=O)c1 C1(C(=O)NCC2N(C(CN(CCCCCC)C)=O)CCC2)CCOCC1C Cc1ccn(C(C)CC(=O)N2CCCC2CNS(C)(=O)=O)n1 CC1CC(C(=O)N(C2(C(N3CCCCC3)=O)CC2)C2CC2)=NO1.C(N)(=O)N CC(C)C(C)C(CNC(=O)Cn1ccc(C(F)(F)F)n1)Nc1cc(F)ncn1 c1(C(=O)NC2(C)CN(C(C(COCC)C)=O)C2)ccc(F)cn1 Cc1nc(C(N2CCCC2C(C)(C)NC(=O)CC2CCCSC2)=O)sc1C c1(C(C(=O)NCCC#N)N(C2CCN(C(CC)CC)CC2)C)cc(C)ccc1Cl C1(NC(C(c2cccs2)SC)=O)CCCC(NC(=O)C=C2CCN(C)CC2)C1 C1(C(=O)NCCOCC(C)(C)O)CCCCN1C(c1cc(C(F)F)no1)=O N1(C(c2ccc(SC)cc2)=O)CC(NC(=O)CN2CSCCSC2)CCC1C C(CCN(C)C(c1cncc(C)n1)=O)(C(C)(C)C)NC(CCOCCC)=O N1(C(CC2C(C)CCO2)=O)CCn2ncc(CNC(=O)C(C)(Cl)Cl)c2C1 c1(SCC)cnc(O)c(C(N2CCC(NC(=O)C(CC)C(C)C)C(F)C2)=O)c1 CC12CC(C(=O)NC3C4CCC3N(C(c3cncs3)=O)C4)(CCO1)C2 C1(C(=O)NCC(CC(F)(F)F)NC(C=CCC)=O)CC(c2ccccc2)=NO1 c1(C(N2C(n3cc(-c4cnc(C(C)C)o4)nn3)C=CC2)=O)cc(F)cnc1O C1(NC(C2N(CC)CCC2)=O)CCCCC1C(=O)NCCC1CCCN1C C(=O)(C1CCCc2c[nH]nc21)NCC(CN(C(c1c(C)scn1)=O)C)O CC1CCCN(C(=O)Cc2nccn2C)C1CNC(c1[nH]nnc1C1CC1)=O C1(C(=O)NC(C2(O)CN(C(C(c3ccc(Cl)s3)C)=O)C2)C)CC2CCC(C1)O2 C1(CN(C(C(C)OCc2ccccc2)=O)C)CCCN(C(=O)C(C)CF)C1 N1(C(c2cc(CC)on2)=O)CC(C(=O)Nc2ccc(C)nc2C)CC(F)C1 c1(NC(C23N(C(C(CC)N(CC)CC)=O)CCC2C3)=O)ccc(C)cc1C N1(CCC)CCCCC1C(=O)NCCCCOC.c1(C(=O)N)coc(N(C)C)n1 C1(CC)C(NC(=O)CCCC2CCC2)CCCN1C(c1cnc(Cl)[nH]1)=O c1(C(=O)OC)ccc(N)c(C(N2CC(n3ccnn3)C2)=O)c1 N1(C(c2c(C)sc(O)n2)=O)CCCN(C(=O)Cc2csc3ccccc23)CC1C CC1CN(C(=O)CC2CSC2)CCN1C(c1cc(O)ccc1F)=O c1(OC)nccc(C(c2nnnn2CC2(CO)CCC2)NC2C=CCC2)c1F C1CCCN(C(=O)CCCc2cncs2)C1.C(=O)(CNC)NC(=O)NC(C)C C1(CNC(c2cscc2F)=O)CCCC2(CN(C(=O)C3Cc4ccccc43)C2)O1 C1(C(N2CCC(C)(NC(C3COC(=O)O3)=O)C2)=O)(OCC)CCOCC1 c1(OC)ccccc1-c1ncc(C(=O)NCC(C)(CO)NC(=O)CC(C)OC)[nH]1 CC1OCCC1C(=O)N(C)CC1CCCN1C(=O)COc1ccsn1 c1(OC)ccc(C(=O)NC2CCCN(CCN3CCOCC3)C2=O)cc1N CCC(CNC(c1cc2nc(C)ccc2o1)=O)N=c1cc(C(F)F)nc(SC)[nH]1 N1(C(Cc2nc(C)c(C)s2)=O)CCC(CNC(c2cccnc2)=O)C(C)C1 c1(CCC(=O)OC)ccc(C(=O)NCC)cc1.c1(C(=O)N)cc(C)c(Br)o1 N1(C(CC=C)=O)CCCC(C2CCN(C(=O)Cn3nnnc3C)CC2)CC1 Oc1ccc(-c2cccc(C3CC3CNc3cc(F)c(Br)c(F)c3)c2)c(Cl)c1Cl C(=O)(CC(C)(C)CCOC)N(CCCCCC)CCNC(=O)Cc1cnnn1C C1(CC(=O)NCC2CCN(C(c3ncc(Br)cn3)=O)C2)CCCCC1(F)F N1(C(CC2(C=C)CCC2)=O)CCC2(CO)CN(C(=O)C3=C(Cl)CC3)CC2C1 C1(CNC(CCC=C)=O)(NC(c2nn(C)nc2C)=O)CC2CCC1C2 C(=O)(C1=COCCO1)N(C)CCNC(c1cccc(N2CCCS2(=O)=O)c1)=O N1(C(CC2(C)CCC2)=O)CC(NC(=O)C(c2ccccc2)F)CC2(CC2)C1 CCC(CC(=O)N1CCC2CC12C)NC(=O)CN1CCC(=O)CC1 CCS(=O)CC(=O)NC(C)CC1CCN(c2nnc(C3CCCC3)s2)CC1 C1(C)(C(=O)NC(C)(C(=O)O)c2cccnc2)CC=CCO1 C(=O)(C(C)CC(C)(C)C)N1CCOCC(NC(c2c(OC)ccc(OC)c2)=O)C1 C(=O)(CCS(N)(=O)=O)NC(C)CCCNC(=O)Cc1ccno1 C(N=c1nc(C(F)(F)F)c2c([nH]1)CCS2)C1N(CCCC)CCCC1 C(=O)(C(F)(F)C(F)(F)F)NCCCN(c1cc(C)nc(-c2cccs2)n1)C C1(CNC(c2c(C#N)csc2)=O)CC2CCC1N(C(C1CCCC1O)=O)C2 N#Cc1c[nH]ccc1=NCC1CCC(CNC(C2CC(F)C2)=O)CC1 Cn1ncc(CC(C(=O)NC2CC3CC3C2)NC(c2sccc2CO)=O)c1O C1(CNC(C2(OCC)CCOC2)=O)CC(O)CN1C(c1nn(C)cc1C)=O C(=O)(CCCC(=O)OC)NC1(C(N(CC(=C)C)C)=O)CC1(C)C C(=O)(C1=CCOCC1)NC1C(C)CN(C(c2cnc(N3CCOCC3)s2)=O)C1 c1(C(=O)NC2(CO)CCCN(C(C(F)=C(C)C)=O)C2)cn2cccc(Cl)c2n1 N1(C(c2c(C)cc(Br)o2)=O)CC2CCC(C1)N2C(=O)COC1CCOC1 c1(C(=O)NCC2OCCN(C(C(CC=C)C)=O)C2)ccnc2c(C)c(C)ccc12 c1(CN2CCN(C(c3c(O)ccc(C(C)C)c3)=O)C3C2C3)csc2ccccc12 C1(NC(COCC(=C)C)=O)CN(C(=O)Cc2cc(C)ns2)CC1C c1(C(N(C)CC2CCN(C(C(C)CF)=O)C2)=O)ccc(CS(N)(=O)=O)cc1 C1(C(N(C2CCN(C(c3c[nH]c(Br)c3)=O)C2)C)=O)C(C#N)C1(C)C N1(C(c2ccns2)=O)CCN(Cc2cn(CC3(F)CCOC3)nn2)C(=O)C1 CCCC(CC)CC(=O)N1CC(NC(C2CCCC(O)C2)=O)C1 C1(C)(CCC=O)CN(C(=O)CN2CC3CC3C2)C1.N(CC)(C1CC1)CC Cc1c(C(N)C(=O)Nc2cncnc2C(C)C)cnn1C CN1CCN(C(=O)C(CCNC(c2cccc(O)c2F)=O)ON)CC1CO c1(-c2ccc(NC(NCCSC)=S)c(F)c2)ccc(C(F)(F)F)c2[nH]ccc12 C12(C(=O)NC(C)(CO)C3CCC3)CC1CN(C(c1nc(Cl)cs1)=O)C2 C(=O)(CC1=NN(C)C(=O)C1)N1CC2C(N(C(=O)Cc3c(F)cncc3Cl)C)C2C1 N1(C(c2ccc(OC)s2)=O)CCN(C(=O)CN2CCC2C)C(C2CCC2)C1 CC(C)C(C(=O)NCc1ncoc1CC)N(C)C.C1(C(=O)N)CCCC12CC2 C1(NC(CCCCC(C)C)=O)Cc2ccccc2C1NC(=O)CC12CCCC1C2 C1(NC(=O)Nc2c(OC)cc(F)c(Br)c2)CCCC2(C1)CC(O)C2 C1(C(N(CCC(C)(C)O)C)=O)CC12CCN(C(c1ncncc1Cl)=O)C2 C(=O)(C(F)C1=CCCCC1)N1C(CC)CN(C(c2cnn(C(C)C)c2)=O)CC1 C=CCCCCCCC(=O)NC1(CCNC(c2coc(S(N)(=O)=O)c2)=O)CCC1 c1(CN2CCC(CCNC(C(C=C)c3ccccc3)=O)C2)ccc2c(c1)CCC2 c1(C(=O)NC(CN(C(C(C)OCC=C)=O)C)C)cc(Cl)c(C)cn1 c1(C(N(C)CCNC(C2(C)CC(F)C2)=O)=O)cccc2sccc12 c1(C(N2CC(C3CN(C(CSC)=O)C3)OCC2)=O)noc2c1CCCC2 C1(c2nnnn2C2CC2)(NCC(C)Nc2ccccc2)CC2OC(C)(C)OC2C1 C1(F)CCCN(C(=O)C=Cc2cccc(F)c2)C1.Cc1nc(C(=O)N)n(C)n1.C C1(O)(CC(=O)NC(CCCNC(c2n(CCCC)ncc2)=O)C)CCOCC1 C(=O)(C1Cc2ccccc21)NC(CCCNC(C1C(OCC)C1)=O)C CP(C)(=O)c1cnn(CC(=O)N(C2COC2)C2CC2)c1.C(C)(C)C.C=O.C C(=O)(C#CC1CCC1)NCC1CC(NC(C2N(C)CCC2)=O)C1 C12(C(=O)NC3C(C)(NC(C4C(CC)CCO4)=O)CCC3)CCCC1CCC2 CC1CCN(C(=O)Cc2cscn2)CC1CC(=O)NC1CC2(CCCC2)C1 C1CN(C(=O)Cc2cc(Cl)cc(Cl)c2)C(C)(C)C1.C(=O)(C(=O)N)NCC N1(C(CC2C(C(=O)OC)C2(C)C)=O)CC2CC1CN(C(c1n[nH]c(C)c1Cl)=O)C2 c1(C=O)cc2ccccc2o1.n1(CC)ncnc1CNC(=O)CO.C1CCC1 O=[N+]([O-])c1cc2c(NC(C3CCC3)C3CC3)nccn2n1 c1(C=O)ccc2nnn(O)c2c1.Cc1cc(C(=O)NCCOCCC)c(C)s1.N C1(NC(c2cc(SC)oc2)=O)CCN(C(=O)C(N2CCCCCC2)C)CC1CO C(CCC1CCC1)(C(=O)NCCCc1ncco1)NC(c1cnncc1O)=O C1(C(=O)NCC2CN(C(=O)C=Cc3cc[nH]c3)CC2C)(OC)CCCCCC1 c1(C(=O)NC2CC3CN(C(c4scc(C)c4Cl)=O)C2C3)cccc2cncn12 C1(C(=O)NCCO)N=C(C(=O)OC)NC(C)=C1C=O.N(CC)CC.C1CC1 c1(C(N2CCC(NC(CN(C(C)=O)C)=O)C(F)C2)=O)nnn2c1C(=O)NCC2 CC(O)CC(C)(C)CNC(c1ccsc1Br)c1nnnn1CC1CCOCC1 N(C(=NC1CC1)N1CCC(CNC(N)=O)C1)C1C(CCC)C1 C(=O)(C(C(C)(C)C)n1cc(CNC(c2cnoc2C)=O)nn1)NCCC=C=C c1(C(N(C2CCN(C(C(CC#C)C)=O)C2)C)=O)ccc2c(c1)CCCCN2 c1(CC)c(NC(C2(NC(=O)CC3COC(=O)C3)CC2C)=O)cnn1C C1(C(=O)NC2CN(C(c3[n+]([O-])ccc(OC)c3)=O)C(C)C2)CCC(N=[N+]=[N-])CC1 N1(C(C(=O)NCCC)C(C2CC2)OC)CCC2CN(C)CC2C1 CC(CNC(C1CC(O)C1)=O)C(F)C(=O)N(C(C(N)=O)C1CC1)C N1(C(C2CCC(C#C)CC2)=O)CC(NC(c2cc(C(N)=O)cs2)=O)CC(C)(C)C1 C1(C(CNC(c2ncc(C)cn2)c2nnnn2C)OC)CCC(F)(F)CC1 CCC(C(=O)N1CC2CN(C(c3cc(C(C)C)on3)=O)CCC12)C(C)(F)F C(=O)(C1=CCCC(C)(C)C1)NCC1(CNC(C(C(CC)C)O)=O)CCCC1 Cc1cc(C)c(C(=O)NC2CC3CC(NC(c4nccc(C)n4)=O)CC23)c(N)c1 c1(N2C3C(CO)CC(CC3)C2)nc(NCC(C2CCCC2)C)nc2cccnc12 C1(C(=O)Nc2c(C)noc2)CSCCN1C(C1CCCCO1)=O C(=O)(C1=NNC(=O)C1)NC(C)(CNC(c1cnco1)=O)C1CC1 C1(C)(COC)CC(NC(=O)CCC)CN1C(C1CCSCC1)=O.C(C)(=O)O Cc1nn(C)c(-n2cncn2)c1C(=O)NC(c1cc(F)ccc1O)C c1(CCC)nc(C)c(C(=O)NCCC2CCCN2C(c2cnc(O)[nH]2)=O)o1.C S(=O)(=O)(c1ccc(NCC2(CC)CC2)c(Cl)c1)NC(C1CCOC1)CC N1(C(C2(C)CC3CCC2O3)=O)CCC(C2CCCOC2)CC1 C1(C(=O)NC(C)C(F)F)CCOCCN1C(c1cc(Cl)c[nH]1)=O C1(C(N2CC(OC)CC2)=O)CCCCCS1(=O)=O.N1(CC=O)C(=O)CCC1=O.N O=C1CSCC(C(=O)NCC(CC(=O)NC2CC2c2ccsc2)C2CCC2)N1 C(C1C(C=O)C1(C)C)=C(C)C.C1(CC)CN(C(C2CNC(=O)N2C)=O)CCO1.N N1(C(C(C)(O)C2CCC2)=O)CC=C(CCNC(c2cncc(C(N)=O)c2)=O)CC1 C1(OCC(=O)N(C(C)C(=O)N(C2(C)CCCC2)C2CCCC2)C)CCCCC1 c1(C(=O)NC2COCCN(C(C(CC)(C)OC)=O)C2)cccc(N=[N+]=[N-])c1 C(C(=O)N1CCC(C(C)CNC(c2cnc(S)n2C)=O)CC1)(C(C)C)OCC Cn1cc(NC(=O)CNC=O)cc1C(=O)NCCOc1ccccn1 c1(C(N2CCC(N3CCCC3)C2)C(=O)NC(CC)C)ccc(C(F)F)cn1 N1(C(CSC(C)(C)C)=O)CC2COCCC2C1.C1(C(=O)N)CNC(=O)C(C)(C)C1 c1(C(=O)NC2(CNC(C(C(COC)C)C)=O)CCC2)nnc2ccccc2c1O c1ccccc1Cl.c1(CC(N2CC(N(C(=O)CO)C)C2)=O)cn(C2CC2)cn1 C(C(C)(F)C(C)(C)F)n1cc(C2(CNC(c3cccc(C)n3)=O)CCC2)nn1 c1(C(=O)NC2C(C)CCN(C(=O)CCc3cnoc3)C2)cc2cc(Cl)ccc2s1 c1(C(=O)NCC#CCNC(C2C(C)C2)=O)cnc(S)n1-c1ccccc1 C(CCC(C)C(=O)NCCC1(C(=O)NCc2ccc(O)nc2)CCC1)OC C(C1CCCCC1)=CC(N1CCC1)=O.c1(C=O)csc(CC=O)c1.C(C)(C)C CC1CN(C(=O)CC2(c3ccon3)CC2)CC1.C(=O)C(C)(C)n1cc(Cl)cn1.N c1(OCC)nc(C)ccc1C(N1CCC(NC(c2cc(C#N)on2)=O)CC1C)=O N1(C(=O)C2CC2)CCCCC12CCCC2.C1(N(C)C=O)CC(NC(C)(C)C)C1 C1(C(N2C(C(=O)OC)CCC2)=O)CCC(NC(C2(C#N)CC(=O)C2)=O)CC1 N1(C(C#CC(=O)N(C)C)=O)CCCN(C(c2cccc(N)c2O)=O)CCC1 C1(CC(=O)N(CCCC)CCOC)C2CCC(C2)N1C(C1(O)CCC1)=O Cc1nc(C(=O)NCc2cc(C(=O)N)no2)c(C)o1.c1cnc(C(C)C)[nH]1 C(=O)(C(C)C(O)CC(C)C)N1CC2CN(C(c3ccc(C(C)C)o3)=O)CC2C1 C1(NC(=O)CSC(F)F)CCCN(C(c2ccccc2NC2COC2)=O)CC1 c1(C(=O)Nc2ncc(C(NOC)=O)s2)cc(F)cc(F)c1F c1(CN2C3C(C(=O)Nc4c(C)ncnc4C)C(C3)C2)c(F)ccc(Cl)c1Br Clc1cccc2c1CC2c1nc(C2CCCN(c3ccc(Br)cn3)C2)no1 C1(CNC(c2c(OC)cncc2)=O)CN(C(c2ccc(Cl)cc2C)=O)CCC1C c1(CC=O)nc(C2CC2)cs1.C(=O)(CCn1cccn1)N(C1CCCC1)CC.N CCCC(C)CC(=O)N1CC(NC(C2CC3(C2)CC(O)C3)=O)CC1(C)C c1(N2C(CNC(c3ccc(CCCC=C)cc3)=O)CCCC2)nc(C)ncc1F C(c1sccc1Br)=CC(=O)NCC1CC(NC(C2(SC)CC2)=O)C1 C1(C(=O)NCC2(C(N(CC(C)O)C(C)C)=O)CCCC2)CCCC(=O)C1 CC(CCN(C)C)C(=O)N1CCC1CC(=O)N(C)CC1CCOC1C C(=O)(C1=C(Cl)CCC1)NCCN(C)C(C1CC1c1ccoc1)=O C1(NC(C2(CC#C)CCC2)=O)CN(C(c2cc(C)c(C)o2)=O)C2(CCC2)C1 C1(CC(=O)N)CCCC(=O)N1.c1(C(C)NC(=O)CCOCC)ncccn1 CCC(F)(F)F.C(=O)CC(C)F.C1(C(=O)NC)CCC1.C(C)(C)C.C=O.C Cc1cc(Cl)c(Cl)cc1NC(=O)CC1CN(Cc2c(F)cncc2F)CCO1 c1(CNC(CNC(=O)NC)=O)ccccc1.N(S(N)(=O)=O)CC=O.C c1(C(N2CCN(C(c3cccc(C)c3)=O)CC(O)C2)=O)cnc2sc(C)c(C)n12 c1ccccc1.n1(CC)cc(C(F)(F)C(=O)N)cn1.N(S(N)(=O)=O)CCNC Cc1ccc(CC(N2CCC(NC(c3cccnc3NC(C)C)=O)C2)=O)cc1Cl C1(C(NNS(CC2(C)CNC2)(=O)=O)=O)CCC(N)C(F)(F)CC1 N1(C(C(C=C)(C)O)=O)CCCCCC1.C1(C=O)CC12CN(C=O)C2.C(C)(C)C.N N1(C(c2cc(C)nnc2)=O)CCCC(O)(CCNC(C23CC4CC2C3C4O)=O)C1 c1(N2C(CN(C(C(C=CC)O)=O)C)CCC2)nc(OC)ncc1Br c1(OC)c(CN2CCC(O)C(C(=O)NCCc3nccs3)C2)cc(Cl)cc1Cl N1(C(C(C=C)(C)O)=O)CCCN(C(c2ccc(C)cc2)=O)C(C)C1 c1ccc(F)cc1.c1(C2CC(C(C)NC(c3cc(OC)cs3)=O)C2)ccc(Br)cn1 c1(C(N2CC3CC(C3)C2)=O)ccc2c(c1)NCCC2.C1(C(=O)OC)CC1C=O.N C1(CNC(COCCSC)=O)CCC(F)C1.C1(C)(C=O)CC1(Cl)Cl.C CC1C(NC(c2ccnn2C2CC2)=O)CCCN1C(C1CC2CCC1CC2)=O CCCCCC(F)C(=O)N(C1CCN(C(=O)CC2CCCC2(F)F)CC1)C N1(C(=O)CN2CCOCC2)CCC(NC(C2(CO)CCCO2)=O)C(O)C1 CCCCC(C)C(=O)NC1CN(C(c2cccc(C(C)(F)F)c2)=O)CCC1CO C(CC1=CCCCC1)NC(C1(C)CCN(C(c2ccc(OC)s2)=O)C1)=O Cc1ccc(C)c2c(C)c(C(=O)N=c3ccc(-c4ccccc4F)n[nH]3)oc12 Cc1nc(C(=O)NC)cc(O)n1.C1CC2CCC1N2C(=O)C(F)(F)CN(C)C c1(C(=O)NC(C2CCOC2)C#C)c(CNC(=O)C(CC)CC)nnn1C N1(C(CC2C(CC)C2)=O)CC(NC(C2(C)CC2C)=O)C(c2cnn(C)c2)C1 [SH](=O)(=O)C(F)(F)F.CC1(CCNC(C2CC2)=O)CNC1.c1ccccc1.C c1(NC2COCCN(C(c3c(Br)c(C)n(C)n3)=O)C2)ncc2c(C)cn(C)c2n1 c1(C(N(CCCNC(c2c(C)[nH]cc2)=O)C)=O)nn(-c2ccc(F)cc2)nc1C C1(C(=O)NC(C(=O)NCCN(CCCF)C)Cc2ccco2)CCC(F)CC1 CCC(CNC(=O)C(=O)NCC1CCCC1N(C)C)CCC1CCCCC1 c1(C=O)cc2cccc(Cl)c2s1.C1(OC)CC(CC(=O)NCCC2CCC2)C1.N N1(C(C=C(CCN(C)C)Cl)=O)CCC2CCCN(C(C34CCN(CC3)C4)=O)C2C1 Cc1ccc(NC(C(=O)NC(c2noc(C3CCC3)n2)C2CCC2)=O)cc1 C(=O)(C(CCC=C)NC(=O)CCC1CCOC1)NCCOCCC=C C12(C(N3CCC(N(C)CC)CC3)=O)CC(CO1)N(C(=O)C1=CCCC1C)C2 C=CCCCCCC(=O)NCC1CN(C(c2c[nH]nc2F)=O)CCCO1 N1(C(C(Cc2ccccc2)OC)=O)CCN(C(=O)CC2(O)CCCC2)CC1 c1(OC)cc(F)c(C(=O)Nc2cccc(Cl)c2Cl)cc1OC C(C1CCN(C(=O)CC(CC)CC)CC1)=CC(=O)N(CC(C)O)CCOC Cc1cccc(CNC(C2(NC(=O)CC(C)c3ccco3)CCN(C)C2)=O)n1 N1(C(CCN(C)CC)=O)CC2=C(C1)CN(C(=O)CC(C)(C)COC)C2 c1(OC)ccc2oc(C(=O)NC(C)C(C)(C)C)cc2c1.C(=O)C(F)C(F)(F)F C1(C(=O)NCC(C)(O)C2CCCC2)(CC)CCCN(C(=O)CC2CCCN2C)C1 c1(CC(C)C(=O)NCC=CCNC(C2(C)CCOCC2)=O)ccc(F)cc1 C1(C(C(=O)NCC(F)F)N(C2(COCC)CC2)C)CCC(C)(C)CC1 CC(C(=O)NCC1CCCCN1C(=O)CCc1c(Cl)cccc1Cl)S(N)(=O)=O N1(C(c2nc(OCC)oc2)=O)CCCC(C2(NC(c3cncn3C)=O)CC2)C1 c1(C(N(C2CCN(C(=O)C(C)C(C)O)CC2)CCC)=O)cncc2nc(C)[nH]c12 c1(C(N2CC(NC(CCC(=O)OC)=O)C(O)C2)=O)ccc(F)c(C)c1Cl Cc1nc2cccc(C(=O)NC3(C)CCN(C(C4CCC(=O)N4)=O)CC3)c2[nH]1 c1(C(N(C)CC2N(C(c3cc(C)on3)=O)CCCC2)=O)cc2n(n1)CCO2 C1(C(=O)NCCCC)CN(C(C2(CCCC)CCC2)=O)CCO1 C1(NC(Cc2cccc(CC)c2)=O)CN(C(c2nnc(C)o2)C)CC1(C)C c1(C(=O)N)ccc([N+](=O)[O-])c(Cl)c1.N1(C(c2cc(SC)oc2)=O)CCC(C)CC1 O(N(CC)C(=O)C(C)(C)NC(=O)CC1CCC(=O)C1C)CC CCS(=O)(=O)CC(=O)N1CC(OC)C(NC(c2ccnc(O)c2)=O)C1 C1(C(=O)NCCC#C)CC(NC(=O)COC(C)(C)CC)CCO1 C1(C=O)CC2(CC(=C)C2)C1.n1(CC#C)cccc1C(=O)NC1COCC1.C C1(NC(C2C(C)C2)=O)CC2(CCC(CNC(c3ccc(Cl)cc3O)=O)OC2)C1 N1(C(c2cc(OC)n[nH]2)=O)CCC2C1CCCN2C(=O)C(C)n1cncn1 C1(NC(=O)CC2(O)CCC2)CN(C(C2CCCS(=O)(=O)C2)=O)CC12CCOCC2 C1(C=O)CCC(=O)N(C)C1.C1(CC)CCN(C(c2csnc2OC)=O)C1C.N N1(C(CC(C(C)C)C)=O)CC2CN(C(=O)CC3CC4(CC4)C3)CCC12 C1CC2(C1)CC2(F)F.N1(C(C2(Br)CC2)=O)CCC(COCC)CC1 CCC(C)C(=O)N1CCC(C(=O)NCc2cc(C)nc(C)c2)O1 C(=O)(C#CC1CCC1)NCC1(F)CN(C(C2C(C)(C)CO2)=O)C1 Cn1ccnc1CCC(=O)NC(C(=O)NC(CC1CC1)C1CC1)C1CCCC1 O(NC(=O)CNC(=O)CC1CCCN1C(=O)CO)C(C)C.CCCN(C)C c1(C(=O)N)cccc2c1OCCO2.C1(C)(C(N2CC(O)(CC)C2)=O)COC(=O)C1 c1(CC(=O)NCCCCC(C)NC(C2(C#C)CC2)=O)ccc2c[nH]nc2c1 C1(C(N(CC(C(=O)N2CCC(CCOC)C2)(C)C)C)=O)CN(C)CCN1C c1(CNC(C2N(C(Cc3ccc(C)s3)=O)C(C)C2)=O)ccnc(CO)c1 CC1CC(CNC(C2CCCOCC2)=O)CN1C(c1ccsc1C#N)=O c1(CCC)nc(C(=O)NCC(O)CN(C)C(C2(C3CCCO3)CC2)=O)cs1 C1(CNC(=O)C(c2ccccc2)F)C2CC1N(C(C1CC3C=CC1O3)=O)C2 C1(COC)CN(C(c2ccc(Cl)nc2F)=O)CCN1c1ncc(I)cn1 C1(NC(c2ccon2)=O)CN(C(=O)COC2CCCOC2)CC2(CC2)C1 N1(C(c2cscc2-c2cnn(C(F)F)c2)=O)CCc2nc(Cl)ccc2C1 CCCCC(O)CC(=O)N1CCN(CCNC(=O)CC(C)c2cnn(C)c2)CC1 C1(C(N2CCC(OC)CC2)=O)(CC)CCCN1C(=O)C=CC(C)(C)C N1(C(CC=CC=C)=O)C2CCC1CN(C(=O)C(c1ccc(F)cc1)CO)CC2 c1(CN2C(C)CNCCC2)ccc(F)c2ccccc12 c1(OC(C)CNC(=O)NC2(C)CC2)ccccc1CCc1ccccc1 c1(CNC(=O)NC2CCCCC2CCO)ccc2ccc(O)nc2n1 C1(C(=O)Nc2ccc(O)nc2)CCCN(C(=O)CN2C(=O)CCC2=O)CC1 C1(C(=O)NCC(C(C)C)NC(=O)CN(C)C(C)C)CCC2(CC2)C1 Cc1ncc(C(=O)NC2CN(C(=O)C(C)n3cnnn3)CC2O)cn1 C(=O)(C(C)(C)C(C)(F)F)NC(C(C)NC(c1cc(Br)no1)=O)C c1(C(=O)NC(C2CCN(C(C3CC3(C)Br)=O)CC2)C)noc2ccccc12 c1(-n2c(-c3nn(C)cc3C)nc(C(C)SCC)n2)cc(C)c(Br)c(C)c1 C(N(C)N1CCCC(c2cncn2C)C1)C1(OC)CC1 O=C(C1=COCCC1)NC1CCN(C(=O)Cn2cc(C3CC3)cn2)C(C2CC2)C1 O=C(C#CC1CCC1)NC1CCOCC1NC(=O)C(F)(F)C(F)F Cc1ccc2oc(C(N3CC(C)C(C(F)(F)F)C3)=O)cc2n1.C1(C(=O)N)CSC1 Cc1cc(CC(=O)NCC2CN(C(=O)C(C)C3CCC3)CC2(C)C)ccc1Cl C1(NC(c2ccc(C)o2)=O)CCCCCC1NC(=O)C1CC1 C1(CC)(NC(=O)CC2CCOC2C)CCN(C(=O)C(C(C)C)C2CCC2)CC1 C(=O)(C(c1ccco1)NC(=O)C(=O)N(C)C)N(CCCN(C)C)CCC CC(C)C(F)(F)CC(=O)N1CCCC(O)(CNC(=O)CCC)C1.C(=O)C1CC1 c1(N2C(CNC(C3(C)C=CCCC3)=O)CC(F)(F)C2)ncc([N+](=O)[O-])cn1 C1(NC(c2ccc(OCC)cc2)=O)C2CCN(C(=O)CCc3ccco3)CC12 Cc1nc(N2CC(C(=O)O)C(c3cccc(F)c3)C2)nc2ccccc12 N1(C(C2=NOC(C)C2)=O)CCN(C(C2CNC(=O)CC2C)=O)C2(CCC2)C1 C(=O)(C1CCc2c(Cl)cccc21)N(C1CCN(C(C2CCC=CCCC2)=O)C1)C C=CCCCCCC(=O)N(C1CCC2CN(C(=O)CCc3ccncc3)CC12)C C1(C(N2CC(CNC(C#CC(=O)N(C)C)=O)OCC2)=O)(O)CCCC(C)(C)C1 N1(C(COCC(=C)C)=O)CCCC(CC(=O)N(C)CC2(O)CCCC2)C1 CC(C)C1=NOC(C(=O)NC2COCCN(C(c3ccnc(S)c3)=O)C2)C1 c1(CC(=O)N(C(CCNC(C(CC)(F)F)=O)C)C)ccc(OC)cc1OC c1(CC(=O)NCCC(=O)NC(c2cn(C)nn2)C)cccc(F)c1 c1(C(=O)NC2CC3CC(OC)C3C2)cccn2c(C)cnc12 c1(CC)ccc(C(N2CCCCC2CCNC(=O)C(C)(COC)CC)=O)cc1N CC1(C)CCC(C(N2CCC2CC2CC2)=O)CN1C(c1cnc(Cl)s1)=O c1(SCCC)ccc(C(=O)NCCCCC)cc1.C1CCS1 C(=O)(C(C)CC(C)C)N(CCNC(Cc1ccn(CC)n1)=O)CC1CC1 Cc1nc2[nH][nH]cc-2c(=NC2CCCC2C(N2CCCC2CN(C)C)=O)n1 N1(C(COCCNC(c2occ3c2CCC3)=O)=O)CCOC2CCC12 c1(C(=O)NCCOCC(N)=O)coc(CNC(c2csc(Cl)c2)=O)n1 C(=O)(CN1C(=O)CSc2ccccc21)NCC1(C)CCO1 CCC(C)(CCC(C)C)C(=O)N1CC(NC(=O)CCc2cnc[nH]2)CC(F)(F)C1 c1(C(=O)NC23CCN(C(Cc4c(C)occ4)=O)CC2C3)cc2cn[nH]c2cn1 Cc1cc(O)cc(=O)n1C(C)C(=O)NCC(C)C.c1(C=O)ccnn1C(C)C c1(C(=O)NC2CC(C)(NC(C(CC)N(C)C)=O)C2)cc2n(n1)CC1(CC1)C2 N1(C(COC(C)C)=O)CC2CN(C(=O)C(C)NC(c3cccs3)=O)CC2C1 N1(C(Cn2cccc(C)c2=O)=O)CC(NC(c2ccncc2)=O)CC(F)(F)C1 C1(NC(c2cccc(C)c2)=O)CN(C(=O)CC2CCCCN2C)CC1N=[N+]=[N-] N1(C(C(CC)C)=O)CCCC(CNC(=O)CC2CC(O)C2)C1.c1ccccc1.C n1(CC(=O)NC(CNC(C2(OCC)CCSCC2)=O)CO)nc(C)ccc1=O C1(NC(=O)CC2(c3ccccc3)CCC2)CCCC(NC(c2cc(O)cs2)=O)C1 Cc1c(C(N2CCCC(NC(C3CCCC(=O)N3)=O)C2)=O)ccc2n[nH]cc12 C(=O)(CC(C)C(F)F)N(CCC(C(C)C)NC(C1CCCCC1)=O)C Cc1cccc(CC(=O)N(C)CC2(NC(c3cc(C)[nH]c3C)=O)CC2)c1 c1(C(=O)NC2C3CN(C(c4c(OC)ccnc4)=O)CC32)cnc2[nH]cncc1-2 O=C1CN(C(=O)CCCn2cccc2)C(C(=O)NC2(C(O)CO)CC2)CN1 Cc1cc(C(=O)NC2CCC2C(=O)N(C2CCC(C)C2)C)cc(O)n1 N1(C(C(CC(=C)C)C)=O)CC(=O)N2CCOCC2(CNC(c2csnc2C)=O)C1 c1(SCC)cnccc1C(N1CCC2C(NC(c3n[nH]cc3C)=O)C12)=O C1(NC(C(CC)COC)=O)CC12CCC(NC(=O)Cn1nccn1)CC2 c1(C(=O)NC2(CC)CCN(C(c3cc[nH]n3)=O)CC2)ccc2c(c1)CCCCS2 N1(C(C(C)SCC)=O)CCN(C(=O)CCc2cc(C(=O)OC)c(C)o2)CCC1C C1(CNC(C(c2c(C)ccnc2)(C)C)=O)CCCN(C(c2nonc2N)=O)CC1 Cc1nc(C(N2CC(O)CC2CNC(=O)CCCn2cccn2)=O)cc(O)n1 Cc1cc(C)c(NC(=O)NC2CCN(C(C)C)CC2C)c(Cl)n1 N1(C(C(C)n2cnnn2)=O)CC2(C1)CN(C(=O)CC(C)(C)F)C2 CCC(C)(C)C(O)C(=O)N1CCOC(C(C)NC(=O)C(C)N(CC(C)C)C)C1 C(CCF)(C(=O)Nc1cnn(C2CC2)c1)NC(=O)CC1CCSC1 N1(C(c2cc(CC)oc2C)=O)C2CCC1CC(N(C(=O)CN1CCC1C)C)C2 Cc1cc(Cl)cc(C(N2CCCC(CNC(c3cccn(C)c3=O)=O)C2)=O)c1O C(c1ccc(C(N)=O)cc1)=CC(=O)N.C(CCC)NC(C1(N(C)C)CC1)=O Cc1cc(C(N2CCC2CNC(c2ccn(C)n2)=O)=O)c(N)c(Cl)n1 CCCC(CC)CC(=O)N1CC(NC(c2cnc3ncccn23)=O)C(C)C1 C(=O)(C(F)(F)Cn1ccnc1)NC(C)CCCNC(c1scnc1C1CC1)=O C1(C(N(CC(CNC(c2ncc(C)cc2C)=O)C)C)=O)Cc2ccc(C)cc2S1 O=C1CCN(CC(N2CCCCC2CCNC(C2CC=CCO2)=O)=O)C(=O)N1 c1(OC)ccc(CCNC(c2nnnn2C2CCC2)c2ncc[nH]2)c(Cl)c1OC CC(CNC(=O)CCC1CCC(=O)C1)C(F)C(=O)N1CC(F)CC1C c1(CNC=O)ccc(S(=O)(=O)N2CCCCC2)s1.C1(CC(=O)O)CC=CCC1 CC1CN(C(=O)CCOC2CN(C(=O)C(C)NC=O)C2)CCN1CCO C1(CC(=O)NCCN(CCOC)C)CC(C)N(C(=O)C(O)CSC)C1 CC1CCCCC1c1nc(Cc2ccncc2)nn1-c1ccc(C(F)(F)F)cc1 CC1CC(=O)NC(C(N2CCN(C(=O)C=CC(F)(F)F)CC2C2CCCC2)=O)C1 CC1(C)CC(CNC(c2n[nH]cc2F)=O)N(C(=O)C(O)Cc2ccccc2Cl)C1 N1(CC2C(C)(C)CCC2)C(=O)CN(CCC2(F)CCC2)C1=O N1(C(C(C)(C)CC#N)=O)CCC2(CC1)CC2C(N1CCC2CCCC2C1)=O c1(C(N(CC(CC)NC(c2c(OC)cccc2F)=O)C)=O)c(F)cc(F)cc1F C12(NC(c3nc(CCCC)sc3)=O)CCN(C(c3ns[nH]c3=O)=O)CC1C2 c1(CC(=O)NC23CC(NC(C4(C(C)C)CC4)=O)(C2)C3)ccccc1Br C(=O)(C1=CCCOCC1)NC1(CC)CCN(C(=O)CC2CCCOC2)CC1 N1(C(C(CCOC)C)=O)CCCOC(CNC(C2(COC)CC2)=O)C1 N1(C(C2(F)CCN(C(c3ccn4cncc4c3)=O)C2)=O)CCCN2CCCC2C1 C1(O)(CC)CCCN(C(=O)C2=CCN(Cc3ccccc3)C2)C1 C1(NC(Cc2c(CC)con2)=O)CN(C(=O)COCCCF)CC1(C)C c1(C(=O)NC(CNC(c2ccc(N)c(N)c2)=O)C2CC2)cnc2c(F)cccn12 C(=O)(CCCC(=O)NCC1CC1C)NCC.c1(C=O)cncc(Cl)c1C.N N1(C(C=C(C)C(F)F)=O)CC2CC1CCN2C(=O)CSCC1CCCO1 Cc1cccc(NC(=O)C(=O)NCc2cncc(OC)n2)c1.C(C)CN(C)C c1(C(=O)NCC2N(C(CC(C=C)(C)C)=O)C3C(C2)C3)cc2c(s1)CCCCCC2 C(=O)(CCCCCCCCC=C)N1CC(CC#C)C1.N1(CC=O)CCCCC1=O c1(NC(=O)C(O)C(O)c2ccccc2)ccc(Br)c2ccccc12 c1(OC)cc(NC(=O)CC2CC(C=O)C2)cc(C)n1.c1(C=O)sccc1I.N Cc1[nH]nc2c1CCC(C(N1CCC(CNC(=O)C(F)(F)C(F)F)C1)=O)C2 C1(C(=O)NCC#CC(=O)N2CCCC2C2CCCC2)CC2CCC2C1 c1(OC)c(O)cc(C(N2CCC2CNC(C2(O)CCCCC2)=O)=O)cc1C#N C1(O)(C(C)NC(C=C(C)C(F)F)=O)CCN(C(c2cccnc2N(C)C)=O)C1 Cc1oc(S(N)(=O)=O)cc1C(=O)NC1C2CCN(C(=O)CCC(F)(F)F)CCC12 C1(NC(C2CCS(=O)(=O)N2)=O)CCCC12CCN(C(C1CC3CCCC13)=O)CC2 C1(NC(c2ccn(CCCC)n2)=O)C2CC1N(C(c1c(N)cccc1F)=O)C2C c1(-c2ncc(CN(C3CN(S(C)(=O)=O)C3)C)s2)ccc2c(c1)CCO2 c1(C(N2C(CNC(C(CC)N(C)C)=O)C(C)(C)CC2)=O)ccc2occ(C)c2c1 c1(OC)ccc(C(=O)NC(C)CCNC(=O)C=C(C)C(C)C)nn1 c1(C(CNC(c2nscc2Br)C)O)ccc(OCC(F)(F)F)cc1 C12(C(N3C(C4CCN(C(=O)CCF)C4)CCCC3)=O)CCC(F)(CC1)CC2 Cc1cc(C)c(S(=O)(=O)NCC2(CC(=O)O)CCC2)c(F)c1 C12(CS(N3CCC(CCC)CC3)(=O)=O)CC(C3COC3)(C1)C2 c1(C(=O)N)cnc2c(c1)NC(=O)CS2.Cc1cc(C(=O)NC2CCC2)nc(O)c1 C1(COC(C)=O)CCCCN1C(c1cccs1)C(=O)NCC(F)F.C1CC1.C c1(-n2cnnn2)ccc2nc(-c3ccc(F)cc3)sc2c1.CC1CCCC(n2cc(C)nn2)C1 C(=O)(C(=O)C(C)(C)C)N1CC(CC(=O)NC2C(OC)CC2O)(OC)C1 c1(C(=O)NC2CCCCN(C(C3NC(=O)OC3)=O)C2)coc2ccccc12 C1(C(N2C(C(N3CC(C)(N(C)C)C3)=O)(CC)CCC2)=O)CC2C(C1)C2(F)F CC1(C)CC(C(=O)NCC2C3CN(Cc4ccccc4)CC23)CNC1=O S(=O)(=O)(c1ccc(F)s1)Nc1cccc(SCCC(=O)O)c1 CCC(CC(C)C)C(=O)NC1(CN(C)C(C23CCN(CC2)CC3)=O)CC1 C1(C(N(C2CCCN(C(CCCCC#C)=O)C2)CC)=O)CCc2nc(C)[nH]c2C1 C#Cc1cncc(C(=O)NCc2cn(CCNC(=O)C(C)CCC)nn2)c1 CCC(CC(=O)NCc1nc(C2CC2)no1)N(C(=O)CC1CCC2CC12)C Cc1cc(F)cc2[nH]c(C(=O)NC3(CNC(C4CCC45CCC5)=O)CC3)cc12 C(CCC(=O)NCCC1(NC(C2(C(N)=O)CCC2)=O)CCC1)C1C(C)C1 C(=O)(CC(C)(C)C#N)NCC1OCCN(C(C#CC(C)C)=O)C1 c1(C(N2CC(CC)N(C(c3ccnc(C)c3)=O)CC2)=O)cccn2c(C)nnc12 C1(CC)CCCCCCN1C(=O)CC1COCCOC1.C12COCCN1C2=O C(=O)(C1=CCCCCC1)NC(C(CC)C)C(=O)NCC1CCC=CCCC1 C=CCCCC(C)(C)C(=O)NCC(O)CNC(C1CC1c1ccc(F)cc1)=O c1(C2(C(=O)NC3CCC(N(C(CN(C(C)C)C)=O)C)C3)CC2)c(F)cccc1Cl c1(C(=O)NCCCC)cn(C(C)C)cc1C.c1(C=O)cc(C)nn1C1CCC1.N C(CC(C)C)(C(=O)N1CC(CC(=O)N(C(C)C(C)SC)C)CC1(C)C)OC Cc1ccc2c(C(=O)NC3CC4CCC3N4C(C3(CO)CC3)=O)c[nH]c2c1 c1(OC)cccc2nc[nH]c(=NCC(C)NC(c3cc(C4CC4)nn3C)=O)c12 c1(CC)ccc(C(=O)N(C2CCCN(C(C3COC(=O)N3)=O)CC2)C)c(C)c1 C(=O)(C(C)(C)C(C)C)NC.c1(OCCOC)cccc(C=O)c1.C1CC1.N c1(C=O)cnn(C)c1-c1ccccc1.c1(CC)cc(C(=O)N)on1.CC=CC c1(C(=O)NC2CC(NC(c3c(C)cnn3C)=O)C2)ccc2nc3n(c2c1)CCC3 Cc1ccc(CN2CCC(O)(C(N3CCCC(F)C3)=O)C2)c([N+](=O)[O-])c1 c1(N2CC3(C(NC(c4cc(C)nc(Cl)c4)=O)CCS3)C2)cnc(C#N)c(C#N)n1 c1(C(N2CC(CCCNC(CCC3(C)CC3)=O)OCC2)=O)ccc(N=[N+]=[N-])cn1 C1(CC)CCC(C)N(C(c2scc(C)c2C)C(=O)NC2(C)CC2)C1 c1(C(N2CC(CC=C)(NC(=O)C(F)C3CCOC3)C2)=O)ccc(CF)cc1 Cn1cnc2ccc(C(=O)NCCOCCNC(=O)CCCC3CCC3)nc12 C1(C(=O)NCc2c(F)ccc(C#N)c2)Cc2c(Br)cccc2CN1 CCC(C)C(C)C(=O)NCC12CC(NC(=O)CCc3ccc(C)cc3)(C1)C2 CN1CCN(C(C2(C)CCCOC2)=O)CC1C(N1CC(O)C(O)C1)=O CC#CCCCC(=O)N(C1CCCC1)CCCNC(C1CSCCS1)=O N1(C(c2cnc(C)s2)=O)CCN(c2nccc(CO)n2)CC(C)(F)C1 c1(C(=O)NCC(CNC(C(CC)(F)F)=O)OC)cc([N+](=O)[O-])cc(Cl)c1Cl c1(N(CC(C)NC(=O)C(c2cccc(OC(F)F)c2)C)C)nc(Cl)c(C#N)s1 C1(C(N(C(C)C)CCN(C)C(C2CC2c2ccccn2)=O)=O)CCOCC1(C)C N1(C(c2nc(CNC(c3c(C)noc3N)=O)oc2)=O)CC(O)CC(C)(C)C1 C1(F)CCCCC1.N1(C(C)=O)CSCC1C(=O)NCC1(C(=O)NC)CC1.C c1(OCC)ncc(C(=O)NCCCN(C(=O)COC2CC2)C)cc1Cl C1(C)(CC)C=C(C(=O)NC2CN(C(c3coc(C4CCOCC4)n3)=O)C2)C1 c1(CC(=O)NCC(C)(CO)NC(=O)Cc2ccno2)cnc2ncccn12 C1(CCC=C)CCCN(C(=O)CC2CC(NC(=O)CC3NC(=O)NC3=O)C2)C1 N1(C(C)=O)CCCC(O)C1.c1(C(NC)=O)coc(C2CC2)n1.C(C)OCC.O C(=O)(C(C)(C)C(C)(C)O)N1CC(CNC(C(C)SC(C)C)=O)OCC1 C1(CC(=O)Nc2cncc(CO)c2)CCCN(C(c2cc(C(F)(F)F)c[nH]2)=O)C1 c1(C(=O)NCC(N(C(CC(CC)C)=O)C)C2CC2)cc(Cl)c(C)cc1Br C(CC(C)C)(C(=O)NCC1COCC1NC(C1CNC(=O)O1)=O)OC C(=O)(C(C1CC1C)N(CCCC)CCCC)NCC=C.C(C)CC N1(C(CCc2c(C)cccn2)=O)CC(C)(C)OCC1CNC(=O)C.CC(N)=O.S n1(C(C)C)cnnc1SCC(N1CCC(n2cc(C(C3(O)CCC3)=O)nn2)C1)=O c1(C(N(C)CCNC(=O)C(O)C2CCC2)=O)ccc2c(c1)CCCC2 Cc1ccc(C)c(NC(c2ccc(CN)c(C(F)(F)F)c2)=O)c1C C(CCO)(C(=O)NC1CCCN(C(=O)CCc2ccc(=N)[nH]c2)C1)N(C)C C1(C(N2CCCC(Oc3ccccc3)C2)=O)CCCCN1CC1CC1 Cc1nn(C)cc1CC(=O)NCC(C)C.c1(C(=O)N)ccnn1CCC(F)(F)F N1(C(C(=O)NCCCCCC)c2ccoc2)CCN(Cc2ccsc2)CC1 c1(C(N2CC(OC)C(NC(c3n[nH]cc3C)=O)C2)=O)cc2cc(F)cc(F)c2[nH]1 C=CC1(CC(=O)N(CCCCO)C)CN(C(C2(CF)CC(=O)C2)=O)C1 C=CC(C)(C)CC(=O)N(C1CCCN(C(=O)CC=C(Cl)Cl)CC1)C c1(C(C(=O)NCC(C)C)N(CCOC)C(C)C2CC2)ccc2cccnc2c1 C(C(C)(C)C#CC(=O)N(C)Cc1ccccn1)NC(CSCC)=O C1(Cl)(C(=O)NCC2(NC(C3CC(C)C3)=O)CCCCC2)CC2CCC1O2 C1(C(N2C3CN(C(C=C(c4n(C)ncc4)F)=O)C(C3)C2)=O)COC2COCC2O1 C12(NC(c3occ(C)c3)=O)CCCC(CN(C(c3cnn(C(C)C)c3C)=O)C1)C2 Cc1cc(C(N2CC(NC(c3ccc4nc[nH]c4n3)=O)C2)=O)ncc1S(N)(=O)=O C1(NC(C(c2ccccc2F)C)C)CCc2cc(Br)ccc2NC1=O C(=O)(CC(C)C(C)C)NCC1(C(=O)NCC(CO)C(C)CC)CC(=C)C1 c1(C(=O)NC)ccccc1[N+](=O)[O-].C1C2CC1N(C(=O)Cc1ccc(F)cc1)C2 C(=O)(CC(CC)CCCC)N1CCCC(C(=O)NC2(C#C)CC3CCCC23)C1 C1(CNC(C(C)CO)=O)CN(C(=O)C(C)Cc2cnc[nH]2)CCC12CCOC2 CC1CN(C(=O)C=Cc2cncs2)CCCN1C(c1cc(-c2ccoc2)on1)=O C(C1CN(C(c2csc(CO)n2)=O)CC1C(=O)NCc1nc(C)cs1)=CC C(=O)(C(F)C(=O)NC1CCCC1NC(C12CCN(CC1)C2)=O)OCC c1(C(N(C2C3CN(C(C4CC5CC5C4)=O)CC23)C)=O)cccc2nccnc12 N1(C(CC)=O)CC(NC(c2ccc(S(=O)CC#N)cc2)=O)CC12CCCCCC2 Cc1cc(C2CCC2)ncc1C(=O)NCC.C1(C=O)CCN1S(C)(=O)=O.N c1ccc2c(c1)CN(C(c1cnc(S)nc1)=O)C2.O=C(C(=O)N)NCC(F)F.C c1(C(N2CCN(C(C(CC)C)=O)C(C(C)C)C2)=O)cnn2c1CC(C)CC2 C1(C(=O)NCC2CCN(C(CCC(=C)C)=O)C2)CCc2nc(O)[nH]c2C1 C1(CCNC(c2c(COC)noc2)=O)CSCCN1C(c1nccn1C)=O CC(C)CC(O)C(=O)NCC(CO)NC(=O)C=Cc1cc[nH]n1 N1(C(C2CN(C(c3cc(C)nc(O)n3)=O)CC23CC3)=O)CC2CCC(CC2)C1 N1(C(c2c(C)scn2)=O)CCC2CCC(NC(c3occc3F)=O)C1C2 CC(C)C(CNC(=O)CCc1nccs1)C(=O)N1CC(C#N)(C(N)=O)C1 C(=O)(N=c1c(F)c[nH]cc1Br)c1c(C)nc(-c2ccc(OC)cc2F)s1 O=S(=O)(NC1CC1c1ccccc1)N1CC(F)C1 N1(CC(=O)N(CC(=O)N(C)C)CCOC)C(=O)C2CCCCC2C1=O CC1CCC(c2cccs2)N(C(=O)NC2CCCC(N3CCCC3)C2)C1 c1(C(=O)NCC=CCNC(c2ccc(C)cc2)=O)csc2c1CCC(C)C2 Cc1ccc(C(=O)NC(C)C(C)(C)NC(=O)C(F)CC2CCCC2)c2c1CCC2 c1(C(=O)NC(C)CN(C)C(c2ccnn2-c2cccnc2)=O)cnc(N)cn1 N1(CC(=O)OCc2cc(C(=O)OCC)c(C)o2)CC(=O)Nc2ccccc21 c1(C(=O)NCC(C)(C)NC(c2c(C)n(C)cn2)=O)c(O)cc(Cl)cc1Cl Cc1cc(F)cc(C)c1C(=O)NC(C)CN(C)C(C1CCc2cncn2C1)=O c1(CN(C2CN(C(c3cncc(C(C)C)c3)=O)C2)C)ccc(Br)c(F)c1 C(C(CC(C)C)C(=O)NC(CC1CCC1)C(=O)NC)OC.c1ccnc(F)c1F c1(OC)cc(CC(=O)NC2CCC(CNC(=O)C(C)C3CC3)C2)ccc1O c1(CN(c2c(C(=O)OC)cnc(N(C)C)n2)C)cc(Br)c2ccccc2c1 C1(CNC(C2C(NC(c3cnc(CC)s3)=O)CC2)=O)CCCCCC1 CCC(C(=O)NCC(CC(C)C)NC(c1scnc1C)=O)C(F)(F)F C1(C2CCC2)(CNC(C)=O)CCN(C(C2CC(C3CC3)C2)=O)CC1 C1(NC(C(C)OCC(F)(F)F)=O)CCC2(CC1)CC(NC(C1COC1)=O)C2 n1(CCC(=O)N(CCC2N(C(C)=O)CCCC2)C)ncc2c1CCCC2 C(=O)(CCCC(=O)NCC=CCNC(c1cc(Cl)ns1)=O)N(C)C Nc1cc(C(=O)NC2(C(F)F)CC(NC(C3CCCCC3F)=O)C2)ccc1F N1(C(CCC(CC)C)=O)CC2CCC1C(NC(=O)CCc1c(C)nn(C)c1C)C2 C1(C(=O)NCCC(CC)C)(CNC(=O)C(COC)COC)CC12CCC2 n1(CC(=O)NCC(C)(C)NC(c2nocc2C(C)(C)C)=O)cc(Br)cn1 C1(CNC(CC(C=C)C)=O)CN(C(c2ccc(OC)nc2)=O)C(C)(C)C1 CC1CCCC(C)N1CCC(=O)NC(C1CCN(C(=O)C=CCF)CC1)(C)C N1(C(C(CC=C)Cc2ccccc2)=O)CCCCC12CN(C(c1cnsn1)=O)C2 C1(C(N(CC(=O)Nc2ccc(CC)nc2)C(C)C)=O)CN2CCC1CC2 N1(C(c2cc(C)nnc2)=O)C2CCC1CC(NC(C1CS(=O)(=O)CC(=O)N1)=O)C2 C(=O)(CC(C)(C)C(F)(F)F)N1C(C)CN(C(c2ccc(S(N)(=O)=O)s2)=O)CCC1 N1(CC(=O)N(C(c2c(C)n[nH]c2)=O)C(C2CCCC2)=O)CCOc2ccccc21 N12CCCC1C(C)C(=O)OCC2.N(CCOC)(CC)CC N1(C(C2CCN(c3n(C)ccn3)C2)=O)CCCC(CCNC(C2CC(O)C2)=O)C1 C12(C(=O)NCCNC(c3c(C(=O)OC)c(C)on3)=O)CCOC1CCOC2 c1(C=O)ccc2occc2c1.C1(CNC(c2[nH]cc(C)c2)=O)CCC(F)(C)C1.N c1(SC)ccc2cc(C(N3CCC(CO)(NC(C)=O)C3)=O)[nH]c2c1 C1(CC)CC(C(=O)O)CN(C(=O)C(F)(F)Sc2ccc(F)cc2)C1 N1(C(C(C)O)=O)CCC2CN(C(c3ccc(I)cc3F)=O)CCC12 Cc1nc2n(n1)CC(C(=O)NC(CNC(=O)CCCCC(N)=O)C(C)C)CC2 c1ccc(C)o1.C(=O)C(C)CC1CC1.C1(CSC)CCC1.C(=O)C1CC1 Cc1cc(C(=O)NCC(O)C)c(C)n1C1CC1.C1(C=O)CC(C)(C)CN1C.N c1(C(N(c2nc(C)c(Br)cn2)CC2CCCN2)=O)cccc2c1NC(=O)C2=O N1(C(Cc2c(C#C)cccc2)=O)CCC(C(=O)NC(C)(C)CCF)CC1(C)C Cc1nc2cc(F)ccc2cc1C(N1CCCC1c1cn(CC(=O)O)nn1)=O C(=O)(C(F)C(C)C)N(C1CCN(C(=O)CC)CC1)CC.C(=O)C(C)(C)C.C C1(C)(C(N2CCCC(CCC#C)C2)=O)CCCN(C(c2cccc(O)c2C)=O)C1 Cc1cccn2cc(-c3ccc(NC(c4csc(=NC5CC5)[nH]4)=O)cc3)nc12 C1(CC)CCCN1C(=O)C(=O)N.c1(C=O)cn(-c2cnn(C)c2)cn1.C1CC1 c1(C(N2CC(CC(=O)O)(C(=O)OC)C2)C2CC2)ccnc(C#N)c1 C1(C(=O)NCC(C(=O)NCc2cc(O)ns2)N(C)C)OC2CCC1C2 C1CN(C(C2CCCC3(CC3)C2)=O)C2(CCCC2)C1.C1(C(=O)N)CC2(CCC2)C1 c1(C(=O)NC2CN(C(CCC(C)OC)=O)CC(C)(C)C2)ccc2cc[nH]c2c1F C(CN=C(NCC1(C)CCCS1)NC1CCN(CC(F)(F)F)C1)OCC=C C(=O)C1=CCCOC1.c1(NC(=O)C=NO)ccc(NC(=O)NC2CC2)cc1.N c1(C(=O)OC)ccc(C(=O)NCCCNC(c2ccc(C)nc2)=O)cc1 Cc1c(C(=O)N(CC(C)NC(C2CC2c2cnnn2C)=O)C)cnn1CCC#N c1(C(=O)NC2(C(=O)NC(C(C(C)C)OC)C)CCCCC2)ccc(F)cc1.N c1(COC)cnccc1C(=O)NCC1CCCC1.c1(C=O)ccc(Cl)cc1.N CCCC(C)CCCC(=O)NCC1(F)CCC(NC(c2cn[nH]c2)=O)C1 c1(C(N2C(CNC(c3cc(O)cs3)=O)CCC(C)C2)=O)cccc2ncnn12 C(=O)(C(F)(F)CCC=C)NC(CC#C)CC(=O)NC(C)C(=O)N(CC)CC N1(C(CCN(C(=O)C(c2ccc(C)o2)C)CC)=O)CCOC(CCO)C1 Cc1nc2ccccn2c1C(=O)NCCC(C)(C)NC(c1cn(C)c(=O)cn1)=O c1(C(CN(CC)CCO)O)cccc(OC(F)F)c1.CC(C)CC1(CO)N=N1 N1(C(C(C(C)O)NC(CCC(C)OCC)=O)=O)CC(C#N)C2(CCC2)C1 c1(C(N2CC(NC(c3cc(C)nc(O)c3)=O)C2)=O)noc2c1COCC2 CCCCC(C)C(=O)NCC1(CC(=O)NCC(O)CO)CC1 C=C1CC(C)(C(=O)NC(C2CCCN2C(c2cc(OCC)ns2)=O)C)C1 C1(CC(=O)NCCCCC2CCCN(C(=O)CC=C(C)C)C2)(CC)CCOCC1 C=CC(C)(C)CN=C(NC1CCC1)N1CCSC(CC)C1 c1(N2CC(C)(C(=O)NC3C4CC5C(C4)C35)C2)ccnc2cc(Cl)ccc12 CC1(C)CN(c2nnc(C3CCC3)n2CCCN2CCCCC2)CCS1=O C(C#Cc1ccccc1Cl)NC(C(=O)O)CCc1ccncc1 CC1Nc2ccccc2C1C(=O)NCC1(c2ccc(Br)cc2)CCCC1 C1(C(N(C2C(C)CC2)C)=O)CCCCC1(C)NC(c1cc(C)c(O)nn1)=O C1(N(C(C2CC(C(F)F)(OC)C2)=O)C)CN(C(=O)CCCN(C)C)CCC1C N1(C(C2(OC)CCOC2)=O)CCC2C(C(=O)NC3C(C)(C)C3(C)C)C2C1 Cc1c[nH]c(C(=O)NC(C(=O)N(C2CC2C)C)c2cccs2)c1 Cc1c(C(=O)NC2CN(C(=O)C=CC(F)(F)F)CCC2C)ccc(Cl)c1Cl C=C=CC(C)C(=O)N1CC(OCCNC(=O)CCC2OCCO2)C1 C(=O)(CC(C)(C)C)NC(C(=O)NCCC1(NC(CC=C=C)=O)CC1)C C1(NC(Cc2cnc(C)o2)=O)CC(NC(=O)CCC2NC(=O)NC2=O)CC1O CONS(=O)(=O)c1ccc(C(=O)NCCNC(=O)C(C(C)C)SC)cc1 C1(C(=O)NC(COC)C2CC2)(C)CC2(CC2)C1.c1(C=O)ccnnc1.N c1(-c2cccc(S(C)=O)c2)ccc2c(c1)CCN(Cc1ccc(Br)c(F)c1O)C2 C(c1cccnc1)=CC(=O)N.C1C2CN(C(=O)CC3(C(F)(F)F)CC3)CC12 CCCCCCC(=O)NCC1CCCCC1C(N1CCC(CO)CC1)=O C1(CN2CCS(=O)(=O)CC23CCC3)CCNCC1C1CCCC1 c1(OC)c(Cl)ccc(C(N2CCC(NC(C3COCCN3C)=O)C(F)C2)=O)c1N N1(C(C(C)NC=O)=O)CCC(C(=O)NCCc2cscn2)(CO)C1 c1(CNc2c(C(=O)Nc3cc(Cl)cc(Br)n3)n[nH]c2)ccc2ccccc2c1O c1(NC(CCSC)C)cc(C)c(S(=O)(=O)N2CCC(C(C)C)C2)cn1 C#CC1(OCC(=O)N(CC)C2CC2)COC1.c1(C(=O)N)ccnn1CCCC c1(C(=O)OC)cc2c(nc1N(C)CCN(C)C(c1n[nH]cc1[N+](=O)[O-])=O)CCC2 c1(-c2nccc(C(N(CCC#C)Cc3ccccc3)=O)c2)cc(Br)cnc1OC CCC(C(=O)N(C)CC)NC(c1ccoc1CNC(C1(CC)CC1)=O)=O C(=O)(CC(C)(C)CC(F)F)N1CCC(C(C)NC(=O)C=C2CCCCC2)C1 c1(C(=O)NC2CC(N(C(C3(C(C)C)CCC3)=O)C)C2)cc(O)c(F)cc1N C1(N(CC)CC)COC2(CCNCC2)C1.c1(C=O)ccc(C)o1.[SH](C)(=O)=O C(C(C(=O)N1CCC2(CC2)C1)C(C)C)NC(C1CC(C#C)(O)C1)=O c1(OC)ccc([N+](=O)[O-])c(C(=O)Nc2cc(F)ccc2C(C)=O)c1 C1(C(=O)OC)CCN(C(=O)CC2CCCC2)O1.c1(C(=O)N)cnn(C2CC2)c1 N1(CC(C)C)CC(C(N2CCCC2CNC(=O)Cc2ccccc2O)=O)CC1=O N1(C(c2c(OC)cccc2F)=O)CC2CC(NC(C3(C)CCCOC3)=O)CC1C2 c1(C(=O)NC2CC(NC(c3cncc(OC)c3C)=O)C2)cnc2c(n1)CCCC2 n1(CCC(=O)N(CCC(=O)NC2CC2)C)c(=O)oc2ccccc12 Cc1ccc(O)c(C(N2CC(C(N3CCC(C(C)(C)C)CC3)=O)C3(CC3)C2)=O)c1 CN(C[Si](C)(C)C)C(C1CCOCC1NC(=O)C(c1ccccc1)F)=O CC(C)(CCC#N)C(=O)NCC#CCNC(c1ccc(-c2cn[nH]c2)cc1)=O N1(C(=O)OC(C)(C)C)CC2CCC(NC)C2C1.C1CC2(C1)C(F)(F)C21CC1 C(=O)(C(C1=C(C)CCCC1(C)C)N(CCC#N)CC1CCOC1)NCC CS(=O)(=O)CCCC(=O)N1CCC(CO)(NC(c2cccc(C(N)=O)c2N)=O)C1 CC1(C)CC(NC(C2CC=CC2)=O)CN1C(=O)CC1CCOC1=O c1(Nc2cn(C)c(NC(=O)CCN3CCCCC3)n2)ncc2c(n1)NC(=O)C2 c1(C(=O)OCc2nnc(C3CCC3)s2)ccc(Br)c(Cl)c1Cl N1(C(CNC(C)=O)=O)CC2CCC1C(C(=O)N(CCCn1cccn1)C)C2 Cc1cccnc1C(N1CC(C)C(C)C1)=O.c1(C=O)ccn(CCN(C)C)n1.N C12(C(=O)NCC(C)N(C(c3n(CC)ncc3)=O)C)CCCC1C2Br N1(C(Cc2c(CC)n[nH]c2CC)=O)CCN(C)C(=O)C1C c1(C(C)C)cccnc1NC(C1CCCN1S(=O)(=O)C(F)(F)F)=O CC(CCNC(C1(NC(C2COC(=O)N2C)=O)CCOCC1)=O)CCO CN1C(=O)NC2(CCN(C(c3cncc(C(F)F)c3)C(=O)NCC(F)F)C2)C1=O C1(NC(c2c(C)nsc2C)=O)CC2CC1N(C(C1CN(C3CCCCC3)C1)=O)C2 C(=O)(CCC(=O)NC1CC1)N(CC(C)NC(CCc1onc(C(C)C)n1)=O)C C(=O)(C(C(=O)NC(C)(C)CC(=O)NCC1(C#N)CC1)OC)OC CC(C)C(C#N)C(=O)N.C(C)CC(F)(F)F.c1(C=O)cc(C2(Cl)CC2)n(C)n1 N1(C(COCC=C)=O)CCOC2CCN(C(=O)CC3CCC(C)(C)CO3)CC12 N1(C(CCCOC(C)(C)C)=O)CCCC(C(N2CCC(c3ncco3)C2)=O)C1 Cc1ncc(C=CC(=O)NC(C)C)c(O)n1.c1(C(C=O)(C)C)ccc(Cl)cc1 O=Cc1cccc(CN2CCSC(C(=O)NCc3cccc4nccn34)C2)c1Br Cc1cccc(SCC(=O)NCC(C)(CO)NC(=O)CC2(C)OCCO2)c1 N1(Cc2c(OCC)cc(C(F)F)cc2)CCOCC(C)(O)C1 N1(C(Cc2cn(C)nc2)=O)CC(C2CC2C(=O)NCC2CCCC2)C1 C(C)(CCC(=O)NCC(C)(CO)NC(c1oc(Br)cc1C)=O)OC C1(C(C)NC(=O)CC(=O)N(C)C)CCCN(C(c2cocn2)=O)C1.C1CC1.C c1(C(=O)NCCC(C)NC(c2ccnc(C)c2O)=O)ccc(S(C)(=O)=O)s1 C(=O)(C1=CC(C)(C)C1)NC1C(N2CCN(C(C(C=CCCC)O)=O)CC2)CCC1 c1(C(N2CC(C=C)C(NC(C34CC(C)C3C4)=O)C2)=O)ccc2c(c1)CCC2=O c1(C(=O)NCc2cccc(CNC(C(COC)C)=O)c2)cnc(N)c(N)c1 CC(C(=O)Nc1cnn(CCN2CCOCC2)c1)C(C)C(C)(C)C c1(NC(C2(C)CN(Cc3c(OC)cc(F)cc3)C2)=O)cccc2cnc(Cl)cc12 Cc1cc(CCC(N2CCCC2CNC(C2(CF)CC2(F)F)=O)=O)n[nH]1 c1(CC)cn2c(n1)CC(C(N1CCC(NC(=O)CN(C)C)C(CC)C1)=O)CC2 c1(C=O)cnc(O)n(C)c1=O.c1(CC)cc(C(N2CC(O)(C)C2)=O)cc(F)c1 C1(NC(C)=O)CCC(NCC(c2cnn(C)c2)C)CC1 C(=O)(N=c1ccn(C(F)(F)F)[nH]1)C1(C)CCCN1S(=O)(=O)c1nccs1 N1(CCNC(c2c(OC)cc(C)s2)=O)CCCN(C(c2cncnc2)=O)CC1 C1(C=O)CCN(CCO)C(=O)C1.c1(C(=O)OC)sccc1C(=O)N.C1CC1 c1(OCCC)ccc(OCCN(c2ccc(CO)cc2)C(C)C(=O)O)cc1 Cc1ccc(C#N)cc1C(N1CCCN(C(=O)CC2CCCCC2C)CCC1)=O N1(C(C2(COC)CC=CC2)=O)CCCC2(C1)CN(C(=O)C#CC1CC1)CCO2 c1(C(=O)NCCCN2CCN(C(C=CC(CC)C)=O)CC2)cnc2ccoc2c1 C1(CNC(C=C(CC)CC)=O)CN(C(C2CC3(C2)CC(CO)C3)=O)CCCO1 Cc1nc(NC(c2cc(Cl)sc2Cl)=O)sc1C(=O)Nc1ccc(O)cn1 c1(C(=O)NCC(CC)NC(=O)CC)cnn(C)c1-c1ccccn1.CC(C)C.O CCCCCC(CC)C(=O)NC(CNC(c1cc(F)c(O)c(F)c1)=O)CC(C)C N(C(=NCC(=O)NC1CC1)NCCN1CCOCC1)C(c1c(OC)nccc1)C C(=O)(C(C)(O)C(C)(C)C)N1CCCC(NC(C2CCC(NC(C)=O)CC2)=O)C1 O=C1NCCCC1C(=O)NCCC1COCCN1C(C12CC(F)(C1)C2)=O c1(NC(c2c(-c3c(C)nn(CC)c3C)cccn2)=O)c(C=O)c(C)nn1C C(CCC(C)(C)C(=O)NCc1ncc[nH]1)NC(CC1N(C)CCCC1)=O Cc1cc(C(=O)N)ncc1C(F)F.C1(C(N2CCC2)=O)COCC1C(N)=O.C N1(C(C2(NC(=O)CC3(O)CCCC3)CC(CO)C2)=O)CCC2(CC2)C1 C(=O)(C(C(C)NC(=O)COCC(F)F)C(C)C)NCCC(CC)(O)CC c1(C2(C(=O)NC(=O)NC3CC(CC(N)=O)C3)CCC2)ccc(F)cc1F C1(NC(C(CCOC)O)=O)CC2CC(C1)N(C(=O)C(CC(C)C)NC(C)=O)C2 c1(COC)ccc(C(N2CCCC(NC(=O)C(O)c3ccco3)C2)=O)cc1 N1(C(c2cc(C(C)C)no2)=O)CCC(C)C(C2CC2)C1.C(=O)(C(O)C1CCC1)N N1(C(C2CC(C)OC2)=O)CCCOC(CNC(=O)COC2CCCOC2)C1 C1(NC(c2cc(CC)nc(O)c2)=O)CCC2(CCN(C(c3ncoc3C)=O)C2)C1 N1(C(CCc2c(OC)ccc(F)c2)=O)CC2(CC(S(C)(=N)=O)C2)C1 C1(CCN(C(c2scc(C=O)c2)=O)C)CCN(C(C2CC23CCC3)=O)CC1.CO C1(C(N(CCC(N)=O)CC)=O)C=CCN(C(C2CC(F)C(=O)N2)=O)C1 C1(C(=O)NCCCNC(CSC(C)(C)C)=O)CCC2C1C2(F)F c1(C(=O)NC(COCC)C(=O)Nc2cnc(C)nc2C)cc(F)ccc1F N1(C(C(CC)n2cccn2)=O)CCCN(C(c2ccc(C(N)=O)s2)=O)CCC1 CC1=NS(=O)(=O)N(C)C=C1C(=O)NC(C)CC(C)NC(=O)C(O)CC(N)=O c1(-n2cc(CCC3(O)CN(C(C4C(C)CC4)=O)C3)nn2)ccc(N)cc1 N1(C(c2cccc(C)c2F)=O)CCCCC12CC(NC(C1CC(C)CO1)=O)C2 N1(C(c2c(C)coc2)=O)CC(C(N2CC(O)C2)=O)CC(C)(C)C1 CC(CN(C)Cc1sccc1OC(F)F)S(C)(=O)=O C1(CNC(=O)C2=C(Cl)CC2)CCCCN(C(=O)CCCCC2CC2)C1 C1(C(N2C(c3ccc(C#N)cc3)CCC2)C(=O)NC2CC2)CCOC2(CCC2)C1 c1(C(=O)Nc2sc(C)c(COc3ccc(F)cc3)n2)ccc2csnc2c1 C1(O)(C(CNC)C)CCN(C(c2cccc(OCC3CCCC3)c2)=O)C1 N1(C(C=CC(C)NC(=O)CC2C=NN(C)C2=O)=O)CCC2(CC=CCO2)C1 N1(C(c2c(NC)nccc2)=O)CC(NC(c2ccco2)=O)CC2(CCOCC2)C1 Cc1c(Cl)ccc(C(N2C3CCC2CC(NC(C2CC2C)=O)C3)=O)c1N c1(NCCNC(C(=O)NCCNCC)=O)cc(Cl)ccc1C C=C1CC2CCC(C1)N2C(C12CC1CCN2C(c1cncc(F)c1)=O)=O Cc1cccc(NC(=O)COc2ccccc2C(C)C)c1.C1(=O)CO1 N1(C(C2(COC)CCCCC2)=O)CCN(C(=O)Cc2cnn(C)n2)C(CCO)C1 c1(C(N2C(C)(C)CC(NC(C3C4CCCCCC34)=O)C2)=O)cccc2ccoc12 CCS(=O)(=O)CCn1cc(NC(c2nnnn2C2CCC2)C(C)C)cn1 C1(CC(C)C)CCCN(CCC(=O)OC)C1=O.C1(C=O)CCC(F)(F)CC1 C1(C(N2C3CCC2CC3)=O)CC(C)(C)SC(C)(C)C1.C(C(=O)N)OC(C)C C(C(=O)N(CCNC(c1nnn(C)c1N)=O)C(C)C)(C(C)(C)C)OC c1(OC)cc(CO)ccc1C(=O)N.C1(C)CCCN1C(C1CNC(=O)C1)=O.C C1(C=O)(NC(c2cc(CC)ncc2)=O)CCC(C)(C)C1.C1CCC(C#N)CC1.N N1(C(C=C(CC)CC)=O)CCC(C)(CCNC(=O)CC(=O)NC2CC2)CC1 O=C(CC1OCc2ccccc21)NCC1CN(C(=O)CNc2nccs2)CCO1 CC1CC(C)(C)CCC1NC(=O)CNc1ccc(-n2cncn2)cc1 CC1C(NC(c2occ3c2CCOC3)=O)CC2CCC1N2c1ncccc1C#N CCCCC(C(=O)NC1COCCN(c2cc(C)nc(CO)n2)C1)NC(N)=O c1(C(N2C3CN(C(c4c(C)con4)=O)C(C3)C2)=O)cc(Cl)cc(Cl)c1O O=C(CCC(=O)N1CCCC1C1CCN(C(C2CC(F)(CO)C2)=O)C1)C1CC1 Cc1onc(C(N2CC(NC(c3cc(Cl)ncc3N)=O)CC(O)C2)=O)c1[N+](=O)[O-] N1(C(c2cn(C)nn2)=O)CCOCC(CNC(C2C3CCC2CC3)=O)C1 CC(C(=O)NC(C1(C(=O)N(C)CCO)CC1)C)c1cc[nH]n1 c1(C(N2CCC(NC(c3cncc(C)n3)=O)C2)=O)cncc2ccccc12 C1(NC(C(C=C)CC)=O)C2CC3C1C3C2C(=O)NC1CC2(CCC2)C1O N1(C(C(COC)(C)O)=O)CCCC(C2CN(c3ncc(C)c(S(C)(=O)=O)n3)C2)C1 c1(C(=O)OC)cc(C(=O)NC2CC(C)C2)no1.C(=O)C(Br)=C(C)C.N Cc1cc(N2CC(NC(c3ccc4c(c3)COC4)=O)CC2C)n2nc(C)cc2n1 N1(C(C(CSC)O)=O)CCOC(CCCNC(c2sc(C)nc2C)=O)C1 C1(NC(c2ccc(F)o2)=O)CCN(C(=O)COc2ccc(F)cc2)CCC1C c1(OC)ncc(NS(=O)(=O)Cc2ccc(C#N)cc2)cc1C(N)=O N1(C(CC2(COC)CC2)=O)CCN(C(c2ccc(Br)c(N)n2)=O)C(CF)C1 c1(CN(C(CC2C(NC(CCC)=O)CCC2)=O)CC)nccc(C)n1 C(=O)(C1=CCC(F)(F)CC1)NCC(C(C)(C)C)NC(=O)CCCCCF C1(NC(C2=C(C)OCC2)=O)CCC2(CCN(C(c3cc(N)c(O)c(F)c3)=O)C2)C1 C1(CNC(CC(=C)C)=O)(CNC(=O)C(F)CC2CC2)CCOCC1 O=C1COc2ncc(C(c3nnnn3CC(F)F)NC3(CCF)CCC3)cc2N1 c1(C(N2CC(C=O)(C)C2)=O)ccc(C#N)cn1.C1(O)(COC)CCCCC1.N N1(C(C(C=C)CC)=O)CCC2CCCC12CNC(c1cc(O)nn1C)=O N1(C(C(C(=O)N(C)C)(C)C)=O)CCN(C(=O)C(c2ccccc2Cl)O)CC(O)C1 C1(CN(C)C(c2cc(Cl)ns2)=O)CCN(C(=O)C(c2ccc(F)cc2)CO)CC1 c1(C(N2CCC3(C(NC(c4ncn(C)c4)=O)C3)CC2)=O)cc2cc(F)ccc2[nH]1 CCCC(C(=O)NCCC(C(=O)NC(C)(CO)C(=O)OC)OC)N(C)C c1(OC(C)C)ccc(C(N2CCC(NC(=O)Cc3ccc(F)cn3)C2)=O)nn1 N1(C(C(CC2CCCC2)OC)=O)CC2CCC1CN2C(c1cccc(CO)n1)=O CCCCC(CC(=O)N1CC(COC)C1(C)C)NC(c1ncccc1F)=O CC(C)CC(F)C(=O)NCC1CCC(F)(C)CC1.C1(CC(=O)N)CCCCC1O N1(C(=O)NC(c2cocn2)CC)CCC(CO)(CO)CC1 N1(CC)C(=O)CC(C(=O)OCc2ccc(OC)cc2F)C1c1cnn(C)c1C c1(OC)c(C)scc1C(=O)NCC(c1ccc(Br)cc1)(C)C C1(CC=O)CCN(C(C2CC(=C3CC3)C2)=O)C1.C1(C(C)OC)CCCC1.N c1(CC)ccc(C(=O)NCC(C)(C2CCC2)NC(=O)CC(C)CO)c(F)c1 Cn1ccc2cccc(CN3CCC(C(=O)NCc4cnco4)CC3)c12 c1(C(C)NCCc2nccn2-c2ccccc2)ccc(CON)cc1 c1(OC)cc(CCC(=O)NCCC2CN(C(C3C4CCCOC34)=O)C2)ccc1O N1(C(C(C)NN(C(=O)C(C)n2cnnn2)C)=O)CCCC1CC1CC1 C1(CNC(c2cc(C)on2)=O)CN(C(C23CCC2C3)=O)CC12CCC2 C1(C(=O)NCC2OCCN(C(c3csc(C)c3C)=O)C2)CC12CCOCC2 CC1(C)C(NC(c2ncncc2N)=O)CC1CC(=O)NC1CC1 C(C1CCCN1C)=CC(=O)N.C(CC(=O)N(C1CC(C(N)=O)C1)C)SCC c1(C(N2CCCC(N(C)C(C3CCC4CC4CC3)=O)C2)=O)cccc(F)c1N C(=O)(CC(C)CC(=O)NC1CC(NC(=O)CSc2cccc(F)c2)C1)OC C1(CNC(c2ccncc2)=O)C2CCCC1N(C(C1CCc3nn[nH]c3C1)=O)C2 N1(C(c2c(CC)nc(C)[nH]2)=O)CC2(CNC(=O)C)CCC1CC2.c1cccs1 C1(CC(=O)NCC2CC(CNC(CSCC=C)=O)C2)CCCCC1C Cn1cc(C(=O)NC2CN(C(c3csc(O)n3)=O)CC23CC3)c(O)nc1=O C1(NC(C(COC)(C)O)=O)CC2CCC1N(C(C1CCC(=O)NC1)=O)C2 C(=O)(C1=NNC(C(F)(F)F)C1)NCCN(C(CCSC)=O)C1CC1 Cn1cc(C(=O)NC(C(=O)NCCN=[N+]=[N-])c2ccoc2)cn1 C(C(C)(O)C(=O)NCC1CC(NC(=O)C(C)(C)n2cccn2)CCO1)OC C1(C2CCN(C(c3c[nH]cc3C3CC3)=O)C2)CC1.c1(OCC(=O)N)cccnc1 C1(Cl)(C(=O)NC(CNC(CCCCC)=O)CC(F)(F)F)CC12CCOCC2 N1(C(CCCSC)=O)CC(NC(c2ccc(S(C)(=O)=O)o2)=O)CC12CCC2 c1(C2N(C(c3cc(C)ns3)C(=O)NCCN(C)C)CCC2)nnc2ccccn12 CC1CC(NC(=O)CCc2ccc(CO)cc2)CCN1C(=O)C1=C(Cl)CC1 C(CC1=CCCCCC1)NC(CN(C(=O)CCS(N)(=O)=O)C(C)C)=O CN1CCCCC1C(=O)NCCC1CCN(C(=O)CCc2ccc(Cl)nc2)CC1 N1(C(C2(C)CC(=C)C2)=O)CCC2CCN(C(c3cccc(C)c3Br)=O)C2C1 C1CN(C(c2cc(C)nn2C2CC2)=O)CC1N=[N+]=[N-].C(C(=O)N)SCCOC c1(-c2nc(C(=O)Nc3cccc(CNC(C)=O)c3)sc2)ccc(F)nc1C c1(N2CCC(C)(OCC)CC2)nc(=NCC2CCCC(C)O2)[nH]c2c1COCC2 Cc1cc2cc(N)ccc2cc1C(N1CC(c2nccs2)C1)=O c1(CCCNC(=NC)NCC2NC(=O)CC2(C)C)cc(Cl)cc(Cl)c1 N1(C(c2cnc(C(C)(F)F)s2)=O)CCC(NC(=O)C2=CCCC2)CC(O)C1 c1(C(C)NC(=O)NC23CC(CSC)(OC2)C3)coc2ccccc12 N1(C(c2ccccc2)=O)CCCN(C23CC(c4ccccc4)C2C3)CCOCC1 c1(CNC(CCCCC)=O)cnn2c1CN(c1cc(C)nc(S(C)(=O)=O)n1)CC2 C12(NC(C3CC(C)C3)=O)CCCC1N(Cc1ccc(F)cn1)CC2 c1(CCC(=O)NCCC(C)NC(=O)C(C)(C)c2ccns2)c[nH]c(=N)[nH]1 C(c1cnccn1)=CC(N1CCC(NC(C2CC3(C2)CC3F)=O)C1)=O c1(C(=O)NCCCCCNC(=O)COC(F)(F)F)cccc(-c2ccncc2)c1 c1(C(N2CC(N3CCN(C(C(C)SC)=O)CC3)C2)=O)ccc2cc[nH]c2n1 n1(CCC)nnnc1C(C1CCC1)NCCN(C1CCOC1)C c1(OC)ccc(C#N)cc1NC(=O)C(=O)NCC1(N2CCSCC2)CCCC1 C(=O)(CS(=O)(=O)C1CC1)NCC(CC)NC(c1c(CC)sc(=N)[nH]1)=O C(=O)(CC(C)(C)CN(C)C)N1CCC(CC(N2CCC2)=O)CC1.C(C)OC.O C(=O)(C1OCCc2ccccc21)NC1CC2(CCC(NC(C(C)CO)=O)CC2)C1 Cc1cc(C)n(NC(=O)COC(F)(F)F)c(=O)c1C(c1ccccc1)=O C=CCCC(O)CNC(C1CCCN1C(=O)C(C#N)CC)=O c1(C(=O)NCC2(CNc3c(C(C)=O)cccn3)CC2)c(C)nn(C)c1C C(=O)(C1CCCn2nccc21)NCCCCC(C)NC(c1cnn(CC)c1Cl)=O c1(NC(C2(C#C)CN(C(C3CC(CC)=NO3)=O)C2)=O)ccc(C)c(O)c1 O=S(=O)(c1csc2ccccc12)NCc1ccn(-c2c(O)cccc2F)n1 c1(C(=O)NC(CC)(C)CNC(=O)C(C2CCCCC2)O)cnc(O)cc1OC N1(C(C(CCC=C)(F)F)=O)Cc2ccccc2OC2(C1)CN(C(C1CC1F)=O)C2 CC(C)CC(O)C(C)C(=O)NC(Cc1ccoc1)C(=O)NC1CC=CCC1 Cc1ccccc1C(=O)NC(C1(O)CCN(C(c2cnoc2C2CC2)=O)C1)C c1(C(=O)NC23CC(NC(c4ncn(CC)c4)=O)C(OC2)C3)cc2occc2n1C C12CCN(C(C)C1)C2.c1(-n2cc(C(=O)NCCOC)nn2)ccc(F)cc1 CCCC(C(O)C(=O)NC1CCN(C)CC1C)NC(=O)CN1CCC(F)CC1 Cc1oc(CO)cc1C(=O)NC(CCOCCO)C(=O)NCc1ccccc1 C1(CNC(CNC(=O)OC)=O)COCCN(C(C2CC2C2CC2C)=O)C1 C=CC1(C(N2CCCC(F)CC2)=O)CCN(C(=O)C(C2CC2)OC)C1 C(=O)(C1c2ccccc2CN1Cc1cc(Br)cs1)NC(C1CCCC1)C C1(C(=O)NC2C(C)CN(C(c3cncnc3)=O)C2)CC(=O)NC1(C)C c1(C=O)nc(N)cc2ccccc12.c1(COC)nc(C)c(C(=O)NCCC)s1.N c1(C(=O)NCCC(CNC(=O)CCC2C(=O)NN=C2C)OC)cccnc1C N1(C(=O)NC)CC(C(=O)N(C2CN(C(=O)C(C3CC3)SC)C2)C)C1 c1(N2CCOCC(NC(CCS(=O)(=O)N(C)C)=O)C2)nc(Cl)nc2sccc12 N1(C(C(C)OCCC=C)=O)CC(OCC)C(CNC(c2cccs2)=O)C1 C1(C(C(=O)NCC2CCCO2)N(CCSC)C)C(C)(C)C1(C)C CCCCC(C)CCC(=O)N(C)CC1CCN(C(C2(C#N)CC2)=O)C1 CN1CCC(C(=O)NC2CC(O)C2CC(N2CCCC(CCCO)C2)=O)C1=O C(=O)(C1Cc2c(Cl)cccc21)N1CC(NC(c2cccc(C#C)c2)=O)C(OC)C1 CCC(Cc1ccccc1Br)C(=O)NC(CNC(C1(C)CC1)=O)CO C(=O)C(C)C(O)CC(C)C.C1(C(=O)N)CC(C)(C)C1.C(CC)N(CC)CC C12(C(=O)NCCCN(C(=O)C(=Cc3cscn3)F)C)CCOC1CCOC2 CC1CN(C(=O)Cn2ccccc2=O)CC1(C)CNC(=O)CC1(C)CC1 C(c1cnn(C)c1C)=CC(=O)NC(CCNC(c1cn(CC)nc1)=O)C c1(C(C(=O)N(CCCN(C(COC(C)=O)=O)C)C)(F)F)ccccc1C c1(NC(c2n(C)cc(NC(c3cc(Br)cc(Br)c3)=O)n2)=O)cc(F)cc(F)c1Br Cc1cc(F)sc1C(N1CCC(OCCNC(C2CC3(CC3)C2)=O)C1)=O N1(C(C(C(CNC(c2c(C)cccc2C)=O)C)F)=O)CC2C=CCC(C2)C1 CCS(C)(=N)=O.C(=O)C(O)CC1CCCC1.CC=O.C(=O)(CC1CC1)N c1(C(=O)NCC(C(C)C)NC(C#CC(C)C)=O)n[nH]c2c1CS(=O)(=O)CC2 CC1(CC(=O)NC(C)(C)CNC(=O)CC(O)Cc2ccccc2)CCCCC1 Cc1nc(C)c(C(=O)OCCN2CCN(C(c3ccccc3F)=O)CC2)s1 C1(NC(C(C)=C(C)C)=O)C(C)(C)CN(C(=O)C(F)n2cccn2)CC1(C)C Cc1cc(C#N)c(NC(C2CSCCN2C(c2ccc(C(C)(C)C)s2)=O)=O)s1 C(=O)(C(C)P(C)(C)=O)N1CCC(NC(C(c2ccc(OC)cc2)=O)=O)C1 C(=O)(C(O)C(C)C)NCC(C)N(C(C1ON=C(C)C1)=O)C CC1(C(=O)NC2CC(CNC(=O)CCC3CC(F)(F)C3)C2)CC1(F)Cl C12(CC)CCC(CC1)CC2.C(C(C(=O)OCC)n1cc(C2CC2)nn1)OCC Cc1ccc(C(=O)NCCN(C(=O)CCN2CCOCC2)C(C)C)c2c1CCC2 C1(C(N(CCCNC(C2CCS2(=O)=O)=O)CC)=O)CCc2nc(O)[nH]c2C1 c1(C(C(=O)NCCNC(c2c(C)c[nH]c2)=O)O)cccc(C)c1F N1(C(C2(C=C)CCOCC2)=O)CCC2(CCC2NC(=O)CC2CCOC2=O)CC1 C(=O)(C1CCCc2nc[nH]c21)N(CC(C)CNC(C1(C2CCOCC2)CC1)=O)C Cc1c(Cl)ccnc1C(c1nnnn1C1CCOC1)Nc1cccc(O)c1 C(=O)(C(C)CO)N.c1(CCC)n[nH]cc1C(=O)NCC1CCCC1.C(C)=O C1(CNC(c2cc(CC)no2)=O)(NC(=O)C)CCCCC1C.c1nccs1.N N1(C(Cc2cc(C)[nH]n2)=O)C2CCC1C(C)C(NC(=O)Cc1ccc(O)nc1)C2 C(=O)(C1=NNC(=O)C1)N1CC2C(CNC(C(C=C)(C)O)=O)(C2)C1 N1(C(C2CN(c3n(C)nnn3)C2)=O)CCC2(NC(=O)C#CC3(C)CC3)CC2C1 c1(C(=O)NC(CNC(C(CC)OCC)=O)(C)C)ccc(Cl)c(C)c1N c1(C(=O)NC2CCCC(N(C)C(c3ccncn3)=O)C2)cnc2[nH]c(=N)sc2c1 c1(CCC(=O)NCCCN(C(=O)CC)C2CC2)ncc(F)cn1.CC(F)(F)F CC(c1ccco1)=CC(=O)NCc1cccc(C(=O)N)n1.C1CNC(=O)C1.C C1(C(NCC(C)(C)C)=O)CCC(=O)N1C1CC1.C1(C=O)CC2CC2C1.C c1(C(=O)NCC(CNC(C2CCOC2)=O)OC)[nH]nc2c1COC2(C)C C12(COC)CCC(C(=O)NCCN3CCN(c4ccc(I)cc4)CC3)(CO1)C2 c1(NCCC2CCN(C(C(C(C)C)NC(C)=O)=O)CC2)cc(C)ccc1[N+](=O)[O-] c1(OC)cccc(S(=O)(=O)NC2COC(C(C)(C)C)C2)c1Br CC1CCc2sc(C(=O)NC3COCC3)cc2C1.C1(C#N)(C(=O)N)CC2(CC2)C1 C(=O)(CCC(=O)c1cccc(N)c1)NC(C)CNC(=O)C(O)CC1CCOCC1 N1(C(CSCCCC)=O)CCOCC(C(=O)NC(COC)C2CC2)C1 C1(NC(c2scc(OC)c2)=O)CCCC12CCN(C(c1csnc1OC)=O)CC2 C(=O)(C(C)C(C)NC(=O)CC(C)=C(C)C)N(CC#C)C1CC1 c1(CC(N2CC(NC(COC3CCCC(C)C3)=O)C2)=O)c[nH]c2cc(F)ccc12 C(=O)C=CS(F)(F)(F)(F)F.N1(C(CCCNS(C)(=O)=O)=O)CCCCC1C.N CC(C)C(F)(CNC(=O)COCCCN(C)C)C(=O)N1CCOC(C#N)C1 CC1CCCc2nc(C(N3CCC(O)(C)C3)=O)cn21.C1(C(=O)N)CC(F)C(=O)N1 C1(C(=O)NCCN2CCC(NC(=O)CC3CCOC3)CC2)CCCCCS1(=O)=O CC(C)C(O)C(=O)N1CCN(C(=O)CNC(C2CCCC(C)O2)=O)CC1 N1(C(C2CC(C)(C)C2)=O)CCc2n[nH]cc2C1.CC1CC1C(=O)NCC(=O)N CCC(CC(=O)NC1CN(C(c2ncccc2OC)=O)CC1C(F)(F)F)C(C)C C1(CC#C)(NC(=O)Nc2nc(C)c(C(C)=O)s2)CCCOC1 c1(CCCC2(C(=O)N(CCC=O)C)CC2)ccccc1.C(=O)C=O.CCO.N N1(C(c2c(C)nc(COC)s2)=O)CCCN(C(=O)CCS(C)=O)CC1C N1(C(c2c(C)cco2)=O)CCC(C2CC(NC(c3cn(C)c(=O)n3C)=O)C2)CC1 c1(Nc2c(OC(COC)C)ccc(Cl)c2)nc(C)nc2sc3c(c12)CCCC3 c1(C(N(C)Cc2cccnc2Br)=O)c(F)c(F)c(I)c(F)c1F c1(CCNC(CCN(CC#C)C(c2csnc2Cl)=O)=O)cnn(C)c1 N1(C(C2CCCO2)=O)CC2C(NC(c3ccccc3)C3(O)CCC3)C2C1 C1(COC)CN(C(=O)CCC(C)OC)CCN1C(=O)CCc1cscn1 C12(C(=O)NCC(C(C)C)NC(=O)CC3CCC3)CCC(F)C1CC2 C(=O)(C1CCc2c[nH]nc21)N1C(C)CCN(C(c2ccn3ncccc23)=O)CC1 C12(CC(N3CCC3)=O)CC3CC(C1)CC(F)(C3)C2.C1(C=O)CC1(C)C.CO c1(C(=O)OC)cn2c(n1)CN(C(C1CCC(C)O1)=O)CC2 C1(C(=O)N)(COC)C=CCN1C(=O)C.c1cnn(C2CC2)c1C.C1CC1 C1(NC(C(CC)N2CCCC2=O)=O)CC2(C1)CN(C(=O)Cn1cccnc1=O)C2 c1(C(=O)NC(COC)C(=O)O)cnc(CNC(c2cccc(O)n2)=O)nc1 C=C(Cl)CC(C(=O)NC(CCO)C(F)F)NC(=O)CCC(=O)N(C)C N1(C(CC=C(C)C)=O)CCCC1C(C)NC(c1ccc(C(C)C)s1)=O C(=O)(C1=CNC2=NCCC2=C1)NC1CCC(NC(Cc2n(C)cnc2)=O)C1 N1(C(C2C(NC(c3cc(C)c(=N)[nH]c3)=O)C2(C)C)=O)CC(C2CC2(F)F)C1 Cc1cccc2c(C(=O)N(C3CCCCC3NC(C3(C)CC3(C)C)=O)C)coc12 CC(C(=O)NC1(C(=O)NCC2CC(CF)C2)CC1)=CC1CC1 C1(CNC(CC(C(C)C)C)=O)C2CCCC1N(C(c1cnc3[nH]cnc3c1)=O)C2 c1(NC(CC2N(C(CSC)=O)CCOC2)=O)ncc(Cl)c(Cl)c1[N+](=O)[O-] c1(CN2CC3(C(C(=O)Nc4cnn(CC)c4C)C3)C2)cnc2cc[nH]c2c1 C1(C(=O)NC2CCN(C(C)C)C2)CCC(C)(C)N(C(C2(C)CC2)=O)C1 C(=O)(CCCC)NC(C)=O.CCC(O)CN(C)C(C1(CCOC)CC1)=O C(C(C(C)(C)C)NC(=O)CN1CC(C)(OC)C1)NC(CC(=O)OC)=O C1(OCC)CN(C(c2cc(C)on2)=O)C1.C(=O)CC.C(=O)C.C1CC1.C C12(c3nnnn3-c3ccccc3)CC1C2.C(CNCC1CCOC1)(CSC)OC C1(C(=O)NC2CCN(C)C2)CN(C(C2CCC(=O)O2)=O)CC1(C)C C1(NC(C=CC(C)NC(=O)OC)=O)CN(C(=O)CNC=O)C1 N1(C(=O)CCc2cnn[nH]2)CCCC2(CCN(C(c3cncc(Cl)c3)=O)C2)C1 C(=O)CC1=CCOCC1.Cc1c(C(=O)NCC2CCC2)cnn1CC(F)(F)F.N C(C1=NOC(CC2(O)COC2)C1)NCCC(COC)OC C1(NC(c2cc(O)cnc2Cl)=O)CC(F)CN(C(c2cnccn2)=O)C1 c1(C(N2CC3C(CNC(C(CC)C)=O)(C3)C2)=O)nc2ccccc2nc1C1CC1 c1(C(=O)NC(CC)CNC(c2nocc2C2CC2)=O)[nH]cc2c1CCC2 C1(NC(COCCC)=O)CC2C1CCN2C(c1ccc(OC(F)F)cn1)=O C(C(CNC(=O)CCc1ccccc1Cl)C(F)(F)F)NC(c1ncn(C)c1)=O C1(C(N2CCCC(NC(c3ccc(Cl)cn3)=O)C2)=O)CCCCS1(=O)=O c1(C(=O)OCC)c(C)oc(NC(=O)C(C)(C)n2ccc(C3CC3)n2)c1C#N C(=O)(CCCCCN=[N+]=[N-])N1C2CN(C(C3=CCCC3(C)C)=O)CC1CC2 C=Cc1ccc(NC(C2CN(C(c3ccc(NC4CC4)cc3)=O)C2)=O)cc1 c1(C(N2CC3CC(NC(C4(CC)CCOCC4)=O)C3C2)=O)cccc(N=[N+]=[N-])c1 CC(CC(=O)N1CCN(CC(=O)NC2CC2(F)F)CC1)CC(C)(C)C C1(C(N2C(CNC(c3ccc(-c4nc[nH]n4)cc3)=O)CCC2)=O)CCC(O)CC1 C12(NC(Cc3c(C)ncs3)=O)CCCC1CN(C(=O)CN=S(C)(C)=O)C2 CC(=O)CCCC(=O)NCC1(F)CC(NC(c2cc(Cl)ncc2O)=O)C1 N1(C(C=O)C2(C(C)C)CC2)CCCC12CC2.C(C)(C)C.C(C)SC.C=O O=C(C1=CCCC1)NCC1CC(NC(C2CC3CC3C2)=O)C(O)C1 CC(CC(=O)NC(C)C(CO)NC(c1cc(F)ccc1N(C)C)=O)CC(C)(C)C c1(NC(C)CCNC(C2COC(C)C2)=O)ncnc2sc3ccccc3c12 N1(C(Cn2c(C)c(Cl)cn2)=O)CCC2(CCN(C(=O)CCOCC(F)F)C2)C1 CC1CCN(C(c2c(F)cncc2Cl)=O)CCN1C(C1CCC(=O)N1)=O CC(CC(=O)NCC1CC2(CC2)CN1C(C1CC(CCO)C1)=O)CC(C)(C)C C(=O)(NNC(=O)C(C)Oc1ccccc1C(C)=O)c1cc(OC)ncn1 CN1CCCCC1C(N1CCCC1CC(=O)NCCc1ccnc(O)c1)=O C1(C(C)C)CN(C(=O)Cc2cn(C)nn2)CCN1C(=O)C(C)n1cccc1 N1(C(=O)CN2CCN(C(=O)COC3CCCCC3)CC2)CC2CC(O)C(C2)C1 N1(C(C=CCCC)=O)CC(F)(F)CC1(C)C.c1(CCC=O)ccc(F)c(F)c1.N CC1CN(C(c2nc(Cl)cs2)=O)CCCN1C(C1CC(F)C1)=O c1(C(NOCC(=C)C)=O)cnn(CCNC(=O)C(C)Cn2ccnc2)c1 C1(C(=O)NCC(CC)(C)Cl)C=CCN(C(C2CCCN2C2CC2)=O)C1 N1(C(C(C2CC2)OCC)=O)CCC2CN(C(=O)CCS(N)(=O)=O)CCC2C1 Cc1oc(-c2cccs2)nc1C(=O)NCCCC(C)(C)NC(C1CCOC1C)=O c1(C(CN2CCC2)=O)cc(Cl)c(Cl)c(Cl)c1.n1(CC)cc(CCC(=O)N)nn1.C C1(C(C)NC(C2(Br)CC2(C)C)=O)CCN(C(=O)O)CCC1(F)F.C(C)(C)C C1(NC(=O)Cc2ccno2)CCCCC1NC(c1nc(Cl)cs1)=O c1(CC)nc(C(=O)NCC(C(C)(C)C)NC(C2CCCN2C=O)=O)c(C)o1 C1(CNC(CN(C2(c3ccccc3)CCCC2)C)=O)CCC2COCCC2C1 N1(C(C2C=CC(NC(C3(CC#C)CCC3)=O)C2)=O)C2CCCC1CN(C)C2 C1(CNC(CCN(C(=O)CC=CCC)CC#C)=O)CC(F)(CO)C1 C(=O)(CC(C(F)F)NC(=O)COCCCC(C)C)NC1CN(CCOC)C1 C(=O)(CCCC(CC)NC(=O)C(F)C(C)(F)F)NCC(C1CCC1)OCC CC(C)C#CC(=O)N(C1CC(NC(=O)C2CC2)C1)C C=CC(C)(CC)C(=O)N(C)CC1CC(F)CN1C(c1ccn(C(C)(C)C)c1)=O CCC(C)C(O)CC(=O)NCCN1CCC(NC(C2CC3C=CC2CC3)=O)CC1 N1(C(=O)CC2CCC(F)(F)CC2)CCC2CCC(NC(C34CC(C3)C4)=O)C1C2 N1(C(=O)OC(C)(C)C)CCCCC1C1CC1.n1(CC=O)cc(C(=O)O)nn1 C1(CC)CN(C(c2ccc(Cl)c(I)c2)=O)CCN1C(C1CCC(C)O1)=O c1(C(=O)NCC2CN(C(c3c(C)csc3)=O)CC2(F)F)cccc2c1CCO2 C1(CCC(=O)N(CC(CN(C)C)(C)C)C)CCCN(C(c2cc[nH]c2)=O)C1 CC1=C(C(=O)N2CC=C(CNC(c3conc3C3CC3)=O)CC2)CCO1 CCCC(C(=O)NCCc1ccon1)NC(=O)C(C(C)O)N(C)C N1(C(C=CC(=O)N(C)C)=O)CCC2(CCC(C(=O)N)O2)CC1.C1CCC(O)CC1 N1(C(c2c(C)coc2)=O)CCC(C)CC1CNC(=O)CC1(C)CC1 c1c(Cl)cc(O)c(Cl)c1C(N1CCCC(C)C1)=O.C1(C=O)CC1C(N)=O.C C1CN(C(c2csc(S)n2)=O)C2(CCC2)C1.C1(C)(C(C)(C)C)CC(C(=O)N)C1 C1(C(=O)NC(CCC)CC)CCC(CNC(=O)C(C2CCCCC2)F)CC1 N1(C(C2(C(=O)NC)CCC2)=O)CC2CC1CN2C(c1ccnc(C)c1C)=O c1(CN(C(=O)C(=O)NCCOCCCN)C)cccc(SC)c1 c1(C(=O)NC(CN(C(c2c(C)n[nH]c2)=O)C)(C)C)cnc2n1CCCC2C C1(CC)CN(C(=O)Cc2cscn2)CCC1NC(=O)Cn1ccc(C)cc1=O C(=O)(CC(C)CNC(C1(C)CC(NC(=O)CC2CCSC2)C1)=O)NC C1(C(N2C(CNC(Cc3c(C)n[nH]c3C)=O)CC2)=O)Nc2ccccc2C1(C)C C1(CC(CO)NC(c2n(C)nc(Cl)c2)=O)CCC(F)(F)CC1 n1(CC(N2CCC3CN(C(C(CC#C)C)=O)C3C2)=O)ccc2c(F)cccc12 C1(CC)CN(C(=O)CC)C1.c1(C=O)ccco1.C(C=O)N(C1CC1)CC.N N1(C(c2cccc(C#C)c2F)=O)CCC2(CC1)CC(CNC(=O)C(O)CCC)C2 N1(C)CC(F)(F)CC1C.Cn1ncc(CCCNC(=O)N(C)CCC2CCO2)n1 C1(C(=O)NCC2CCN(C)CC2)CCCCC1(C)NC(=O)C(F)CC1CCOC1 C1CCC12CCC2.Cn1nc(C(=O)N)cc1C1CC1.C1(C=O)CC(F)(F)C1.C CC1(F)COCCN(C(=O)CC=CCNC(C2CC2C2CCCC2)=O)C1 C(=O)(C(C)(CC)CC=C)NC(CC(N1CCC(CCC#C)CC1)=O)C Cc1ccc2cc(C(=O)NC3CCC(N(C)C(c4cc(Cl)nn4C)=O)C3)nn2c1 Cc1nc(C)n(CCCC(=O)NCCC2CCN(C(=O)C(C)n3cccc3)C2)n1 c1(OC)ccc(C#N)c(NC(C2CCCN(C(c3oc(C)nc3C)=O)C2)=O)c1 C1(CNC(COCCC)=O)CCCC1NC(c1ccncn1)=O c1(C(N2CCCC(O)(CCNC(C(C)C3CCC3)=O)C2)=O)nc2ncccn2n1 Cc1c(C(=O)NCC(C)N(C(=O)CC2CC(C)C2)C)[nH]c2c1C(=O)CCC2 C1(NC(c2ccc(CC)s2)=O)CN(C(c2cc(C)c(C)[nH]2)=O)C(C)(CC)C1 n1(CCNC(C(C)c2ccco2)=O)ccc(C(=O)NCC2(F)CN(C)C2)c1 c1(C(N2C(CCOC)CN(C(c3ccon3)=O)CC2)=O)cnn2ccc(O)nc12 c1(OC)cncc(C(=O)NCC(O)CC(=O)NCC(C)(O)CSC)c1 Cc1cccc(C(=O)NC2CCCC(NC(C34CC3COC4(C)C)=O)C2)c1C C1(C(=O)NCCCCCNC(c2[nH]cc(C)c2)=O)CCCOCC1 c1(C(C)C(=O)NC2CN(CC(F)(F)C(F)F)CCC2C)cccc2ccccc12 C(CC(C(=O)NCC(C)(F)C(C)C)NC(c1ccc(CC)o1)=O)=CC c1(C=O)ccn2ccnc2c1.C(C(C(=O)NC(C)(C)C1CCC1)N(C)C)OC.N C1(C#N)(C(=O)NC(C2CN(C(c3ccn4ncnc4c3)=O)C2)C)CC12CCCC2 c1(CNC2CCN(C(c3ccc(OC)nc3Cl)=O)CC2F)cccc2ccnn12 c1(C(=O)NC(CNC(C(C=C)(C)O)=O)C(C)C)c(C)oc2ncnc(O)c12 Cc1ccc([N+](=O)[O-])cc1C(C)OC(=O)C1=CC(C)(CO)C1 C1(CC)(C(=O)NCCCOC)CCN(C)CC1.C1(C=O)CCCN1C1CC1.N C(N=c1nnn(C)[nH]1)C1(NC(CS(CC)=O)=O)COC1 n1(CC(N2CC(O)(C(C)NC(C3CC3)=O)C2)=O)cccc([N+](=O)[O-])c1=O C(=O)(C(C(F)(F)F)C(F)(F)F)NC(CCCCNC(c1onc(C)n1)=O)C c1(N2C(CNC(C3CC3C3CCCC3)=O)CCC2)ccc([N+](=O)[O-])cc1Cl N1(C(c2cc(C)cc(N)c2)=O)CCN(C(c2cnc(S)[nH]2)=O)C2CS(=O)(=O)CC12 C(=O)(C(=O)NCC(F)F)N(C(CNC(COCC)=O)C1CC1)C C(=O)(CS(=O)CCC(F)(F)F)NC1COCCN(C(CSCCOC)=O)C1 N1(C(C(C)(C)OC)=O)CC(C(=O)O)C2(C1)CN(S(=O)(=O)c1ccncc1)C2 N1(C(C2C(C(=O)OCC)C2)=O)CCC2CN(C(=O)CC(CC)C(C)C)C2C1 CCN(CC(=O)NC(C)(C)C)N1CCC(NC(C)C)C1.C1CN(C)C(=O)N1 C1(CC(C)NC(C=C(C)C(C)(C)C)=O)CCN(C(c2cccc(C)c2)=O)CC1 C12(C(N3CCC(C(C)NC(C(CC)(C)CO)=O)CC3)=O)CCCCC(F)(C1)C2 c1(C=O)ccc(C(F)F)o1.C1(C(N2CC(=C(C)F)C2)=O)CCCC1.O=CC.N N1(C(C(n2ccc(C)n2)C)=O)CCC(CNC(c2cnc(=N)[nH]c2)=O)CC1C N1(C(c2c(C)sc(Br)n2)C(=O)NCC(F)F)CCN(C2CC2)CC(C)C1 C1(OC)CC(C(N)=O)N(C(C2CC(C)N2C(=O)CCc2nncn2C)=O)C1 CC(O)(C(=O)NCC1(O)CCCN(C(c2csnn2)=O)C1)C(F)(F)F C1(CN2CC3(CCCS3)C2)CCOCC12CCCC2 C1(NC(=O)CCCn2ccnc2)CC2CC1CN(C(C1CN3CCN1CC3)=O)C2 C1(C=O)CC(C)(C)CCO1.CC(C)(F)C.CCCCOC(=O)C=CC=O.N c1(C(C)C)cc(C(=O)NCc2ccsc2C(=O)NCC2CC2C)on1 C1(C(=O)N)(NC(C(C)NC(=O)C2CC2)=O)CC(F)(F)C1.C1CCCCN1C C1(OCCOC)CC(OC)CN(N2CCC(C3CCC3)(OCC)CC2)C1.C1CO1 c1(C(N2C3CCC2CC3)=O)ccc(Cl)c(F)c1F.C(C)(C=O)NC(COC)=O.N C(CC(=O)N1CCOCC1)(C(C)C)OCC.C(c1ccnn1C)=CC(=O)N(C)C C=CCC(CC(C)C)C(=O)N1CCCC12CCNC2=O c1(NC(CN(C(=O)C2=CCOC2)C(C)=O)=O)ccc(C)cc1.Cc1cscc1 c1(C(=O)NC(CC(=O)N(C(c2cccs2)C)C)C)ccc(=N)[nH]n1 C(=O)(CCC(C)C)NCC1(CCCC)CC1.C1(CC(=O)N)CC(=O)NC1=O Cc1ccc(C(N2CC(NC(c3ccc(Cl)[nH]3)=O)CC2CO)=O)c(C)n1 n1(CC(=C)C)nnnc1C(C)(CC1CCCC1)NC1CC1CC(C)(C)C C1(NC(c2ncccn2)=O)CCCC(NC(C2CC2c2ccc(Cl)s2)=O)C1 C(=O)(C(C)CCCC(C)C)NC(CCC#C)C(=O)NCc1cnnc(C)c1C c1(CCN2CC(CCC)C(O)C2)ccc(Br)c(F)c1 Cc1cnc(C(=O)NCCCCNC(=O)CC23CCC(CC2)CC3)cc1Cl c1(C(=O)NCCCN(C)C(c2cc[nH]c2C2CC2)=O)cc2c(s1)CCCCCC2 C1CC(=O)N(C)C1.C(C)(C)(C=CC(=O)NC(C(=O)N)c1ccoc1)SC C(=O)(C(CC)C(F)(F)F)N1C(CC(=O)N(CCCC)CCO)COCC1 c1(C(=O)NC2CCN(C(C3(C(N)=O)CC3)=O)C2)ccc2nnn(O)c2c1 CC(CC(=O)NCCCOC1CCCC1)NC(C1CCSC1)=O C1(C(=O)NC2(C#C)CCCOC2)CCCCCCN1C(c1ccc(C#N)cc1)=O c1(OC2(CC(N3CC(c4ccccc4)C(F)C3)=O)CC2)ccc(F)cc1 C1(NC(C(C=C)(C)O)=O)CC2(CCCCN2C(=O)C(C)(F)C(C)(C)F)C1 N1(C(CCN(CCC)C)=O)CCOCC(NC(=O)C(c2ccccc2OC)O)C1 CCCCCC(C)CC(=O)N1CCN(CC(C)NC(c2c[nH]c(C#N)c2)=O)CC1 c1(C(N(C(C)CNC(=O)CC(C)(F)F)CC)=O)cc2ccc(Cl)cc2s1 CC1=NNC(=O)C1CC(=O)N.C1(CC)CCCCN1C(=O)CS(=O)(=O)N(C)C c1(CN2CCN(C(C(C)OCC=C)=O)C(C)C2)c(Br)ccc(F)c1F C1(C(=O)NC(C(C)C)c2nc[nH]n2)CCOCCN1C(c1cc(C2CC2)no1)=O CCC(O)C(C)C(=O)NCC1CCC(F)(C)CC1.C1(C=O)C(C)(C)C1(C)C CC1CC(CNC(=O)C2=C(Cl)CCC2)CN(C(c2c[nH]cc(Cl)c2=O)=O)C1 c1(NC(CCC2CCCN(C(CN(C)C)=O)C2)=O)cccc(N=[N+]=[N-])c1 C1(SCC(=O)NC)CCS(=O)(=O)C1.C1CCN(C(C2(F)CCCC2)=O)C1 Cc1csc(=NCC(=O)N2CCC(O)(C(C)NC(C3(O)CCOC3)=O)C2)[nH]1 CC(CCN(C)C(c1ccc[nH]1)=O)NC(=O)CSC1CC1 C(=O)(CCCS(N)(=O)=O)N(CC(CNC(C1N(CC)CCCC1)=O)C)C c1(N(C2COCC2O)C(C2C(C=O)C2)=O)nccc2c(Br)cccc12.CC(C)C.O c1(C(=O)NC(C2CCN(C(=O)C3=CCOCC3)CC2)C)cnc2c(F)cccn12 C1(O)(CN(C)Cc2n(CCC)nnn2)CCN(CC)CC1.c1(C)ccccc1 c1(C(=O)NC(CNC(c2cc(C)nnc2)=O)C2CCC2)ccc2c(c1)CCCO2 CC1CCN(C(C2(C)CC2)=O)CCN1C(c1cccc(-n2nnnc2O)c1)=O CCCC(C)(O)CC(=O)NC1CN(C(c2ccc(Cl)c(Cl)c2)=O)CC12CCC2 c12c[nH]ccc-1nc(=O)[nH]2.CC(CC(Cl)Cl)OC(C)(C)C Cn1nccc1CCC(=O)NC1CCC(CNC(C2CCC(F)C2)=O)C1 C(=O)(CS(=O)C(F)(F)F)N1CC2C(NC(CC3(C)CC3)=O)C2C1 c1(OC)cc(N2CCOC(C(N3CCOCC3)=O)C2)c(F)cc1[N+](=O)[O-] O(N(CC)C(=O)CCN(C(=O)C(O)CCSC)C)CC O=C(C1SCCc2ccccc21)NC1C2CN(C(c3cncn3C3CC3)=O)CC12 C12(OC)CCCC1(COC(c1nn(-c3ccccc3)cc1[N+](=O)[O-])=O)CCO2 N1(C(c2c(C)nc(CO)nc2)=O)CCCC2(CC2)C1.C1(C(=O)N)NC(=O)C2CC12 N1(C(C23C(CN(C(C4SCCS4)=O)C2)CCC3)=O)CCCC12CCOCC2 c1(OC)cc(C)c(C(=O)NC(C)(C)CCC(=O)O)cc1C(=O)O C1(C=O)CC(C(C)(C)C)=NO1.C#Cc1c[nH]nc1C(=O)N.C(C)(C)C1CCC1 C1(CC)C(NC(=O)C(C)C(F)F)CCCN1C(=O)CCc1ccnn1C N1(C(C(N2CCC(c3scc(C)n3)C2)=O)=O)CC23CCCCC2(C1)CN(C)C3 Cc1ccnc2ccc(C(=O)NC3C(C)CN(C(c4ccsc4)=O)CC3C)cc12 Cc1cc(C(=O)NCC(CNC(C2(CO)CC2(F)F)=O)C(F)(F)F)cnc1O c1(C(NC)=O)cn(C)c(=O)nc1O.c1(CSC)ccc(C(N2CCC2)=O)o1.C C1(NC(CNS(CC)(=O)=O)=O)CC2CCCC12.C1(C=O)(N(C)C)CCC1.N c1(C(=O)NCc2cn(CCCCOC)nn2)cccnc1NC1CCNC(=O)C1 CC(CNCCc1cccnc1)CC(F)(F)F c1(C(=O)NCC(CCNC(=O)CCc2cn(C)cn2)OC)cnc(=N)[nH]c1 C#CC(C(C)C)NC(=O)CC1CCC(NC(=O)CCCn2cccc2)C1 C1(C(=O)NCC)CCN(C)C1.c1(OC)nc(C=O)ns1.C(C)(C)C.C=O C1(CC(C)NC(C(C=C)O)=O)CCN(C(c2csc(C)c2)=O)CC1 CC(C(=O)N1CCOCCC1C(=O)NCCC(=O)N1CCCC1)S(C)(=O)=O C1(C(=O)NCC(CC(C)C)NC(c2c(C)noc2C)=O)CCC2(CCC2)CC1 N1(C(c2c(C(=O)OC)c[nH]n2)=O)CCC(C2CC2)CC1.n1(CC=O)ccnn1.N c1(NC(=O)CC2CC3(CCOCC3)C2)cc(O)nc2ccccc12 N1(C(c2c(NC)nc(C)cc2)=O)CC2COCC(C1)C2.C12(C=O)CC(C)(C1)C2 C(N=c1[nH]c(N2CCn3nncc3C2)nc2c1SCC2)C1(n2nccn2)CC1 C1(C(=O)NCC2CC2(Cl)Cl)(NC(C2C(=C)C2)=O)CCC1 C1(NC(c2cnn(CC(F)(F)F)c2)=O)CCCCC1.C1(C(=O)N)CCCC12CC2 CN1CCc2nc(C(N3CC(NC(c4ccc(Cl)cc4I)=O)C(F)C3)=O)sc2C1 c1(C(=O)N)cc(C(C)(C)C)ccc1N.C1(NC(COCCSC)=O)CCC1 C1(NC(c2nc(C)sc2Br)=O)CN(C(=O)Cc2ccn(C)n2)CCC1C N1(C(C2CN(C)C2)=O)CCC(CNC(=O)C(C)(C)c2ccn(C)n2)CC1 c1(CC=O)ccccc1.C(CC1CC1)(C(=O)N(C(C)C)C)OC.C(C)C.N c1(C(C)=O)ccc(C(=O)NC2(CCCCNC(=O)CC)CC2)[nH]1.C1CC1.O c1(CNC2CCP(C)(=O)CC2)c(Br)cc(F)cc1[N+](=O)[O-] c1(CNC(c2c(C(C)C)n[nH]c2)=O)ncccc1C.C1(C=O)CC(C)CO1.N CC(C)(C)C(CO)C(=O)N1CCC(C)(CCNC(=O)C(Cl)=CCl)C1 c1(C(c2n(CC)nnn2)NCCc2cncn2C)cccc(S(=O)(=O)C(F)F)c1 CC(C)C(CC(=O)N1CC2CCC(C1)N2C(C1CCC(F)C1)=O)C(C)C C#Cc1cc(NC(=O)CC(C)NC(=O)C=CC=CCC)cc(F)c1 C(=O)(CC(C)C(F)(F)C(F)(F)F)N1C2CCN(C(c3cccc(C)c3)=O)C(C2)C1 C1(NC(C(C)(C)C2CCCC2)=O)CN(C(c2coc(CO)c2)=O)CC2(CCC2)C1 c1(CCC(=O)NC2CCC(N(C(=O)CCC3CC3)C)C2)ccncn1 c1(CNC(C(C(C)NC(c2cccnc2O)=O)C)=O)cncc(C#N)c1 c1(C(Cc2nc(O)n[nH]2)NC(c2ncoc2C2CCCNC2)=O)cccc(Br)c1 C(=O)(CCCC(=O)N(C)C)N1CC(CNC(C2C(C(=O)OC)C2)=O)C(C)C1 CC1CN(C(c2ccc(C3CC3)cn2)=O)CCC1CNC(=O)CC1CSCCO1 C(=O)(C(C)(O)CC(F)F)N1CCCC(CNC(CCc2c(C)cccc2)=O)C1 C1(NC(CC2(C=C)CC2)=O)CC2CCC(C1)N2C(c1cc[nH]c1CC)=O CCC(C)(O)C(=O)NCCC1(O)CN(C(c2cn(CC(F)(F)F)nc2C)=O)C1 c1(C(N2CCC(F)(C(=O)N)C2)=O)ccc(C(C)C)c(Br)c1.Cc1ccc(C)cn1 c1c(C)cccc1C.c1(C(C)=O)ncc(C(=O)NCC(C)N(C(=O)CCO)C)s1 N1(C(C(C)(C2CC2)OC)=O)CCC(NC(=O)CCc2ccsc2)C(F)C1 CCCCC(F)C(=O)N1CC2(CC2)CC1CNC(c1ccc2c(c1)CC2)=O CCCC(C#N)C(=O)N(C)CCOCCC(=O)NCCC(O)(CC)CC c1(OC)ccc(CNC(C2CC(NC(C3CCC(C)C3)=O)C2)=O)cn1 C1(NC(CCCC=C)=O)CCCC12CN(C(=O)C(c1c(C)nn(C)c1C)C)C2 N1(C(CCN(CC)CC)=O)CC(n2cc(Cc3ncccc3C)nn2)C(O)C1 c1(-c2ccc(C)o2)nc(CC(F)(F)F)n(C(C)COC(C)(C)C)n1 C1(CC)CCN(C(=O)Cc2ccc(O)cn2)C1C(=O)NC1(CO)CCC1 C1(C(N(CCOCC)C)=O)CC(F)CN1C(=O)CNC=O CC1CN(C(=O)C(c2ccccc2Cl)(F)F)CC1CNC(=O)CS(C)(=O)=O Cc1cc(C(N2CCC(NC(c3c(Cl)n[nH]c3C3CC3)=O)CC2C)=O)ccc1F c1(CN2C(c3ccccc3)CCS(=O)(=O)C2)ccc2c(c1)CCCS2 C12(C(=O)OC)CCC(C(N3CC(C)C3)=O)(CC1)C2.c1ccsn1.C(=O)C.N CC(CNC(c1nc(Cl)ccc1F)=O)CN=c1[nH]ccnc1F C1(CC(=O)N(CCCC(C)O)C)CCCN(C(c2ccc(C(N)=O)o2)=O)CC1 Cc1nc(Cl)c(C)c(=NCC(CC(C)C)NC(C2CC2C)=O)[nH]1 C1(C(=O)Nc2ccc(N(C)C)cc2)OCC(=O)N(C)C1c1ccnn1C c1(C(=O)NC(C2(O)CN(C(c3cc(C)ncn3)=O)C2)C)ccc2snnc2c1 Cc1cc(C)c(NC(=O)CC2CN(S(=O)(=O)CCBr)CCO2)c(C)c1 N1(C(CCOC)C)CCC(O)C(C(=O)NCC2(CN3CCCC3)CC2)C1 Cn1ncc2c(NC3CCC3)nc(N3CCOC4(CCSC4)CC3)nc12 C(c1cccc(F)c1Cl)=CC(=O)N.C=C1CC(C)(C(N2CC(O)(C)C2)=O)C1 c1(C(=O)NC2C3(CCC(NC(C=CCC)=O)CC3)C2)cnc2c(c1)CCCO2 N1(C(Cn2ccc(C)n2)=O)CCN(C(c2cnc(Cl)[nH]2)=O)C(C)CC1C c1(CN2CC(O)(CNC(c3cccc(C)c3F)=O)C2)ccc(O)c(C)c1O CC(CNC(=O)Cc1ccns1)C(=O)NC1CCCCC1 Cc1cc(N)c(C=O)c(F)c1.C(CCN(C(=O)C=C1CCC(C)C1)C)C(C)C C1(NC(CC(CC)C(F)F)=O)CN(C(=O)CCn2cncn2)Cc2ccnn2C1 C(C(C)C(F)(F)F)NC(CC(C)C)=O.c1(C(=O)N)cccc(-c2nc(=O)o[nH]2)c1 Cc1cccc2cc(-c3ncc(Cl)cc3C(=O)Nc3nc(Cl)c(Br)cc3O)[nH]c12 C=CCC(CC(F)F)C(=O)N1CCC(CNC(=O)C(C)(C)OC)C12CC2 C1(OC)CN(C(c2ncccc2N)=O)CC1NC(c1cnc(C)s1)=O C(=O)(CS(=O)(=O)CCOC)N(C1CCCN(C(=O)COC(F)F)CC1)CC C(=O)(C(C)(C)C(=O)NC)OC.C1CCN(C(c2ocnc2C(F)(F)F)=O)CC1 C(=O)(CC(=O)N(CCNC(c1cc(Cl)ns1)=O)C1CC1)OCCC(C)C C1(OCC(=O)NCCOCCCC)CCN(C(c2ccoc2C)=O)C1 Cc1ccc(NC(C2CC(NCc3ccc(I)cc3Br)C2)=O)c(CO)n1 C(=O)(C(F)CC(C)(C)C)N(CC(C)C(=O)NCc1ccnc(O)c1)C N1(C(c2nc(C#C)sc2)=O)CCCC(O)(CNC(=O)C(O)C2CC2)C1 c1(C(=O)NCCNC(c2ccnc(S)c2)=O)csc2nccn12 C1(C(=O)NC2CC3CN(C(CC(=O)NC)=O)CC3C2)CC2CCCCCCC12 c1(C(C2CC2)OC)cn(CCNC(C2CCN(S(C)(=O)=O)C2)=O)nn1 c1(C(N2CCC(CNC(C(=Cc3cccnc3)C)=O)C2)=O)ncnc(O)c1Br CC(C)(CCC#N)C(=O)NC1CCCC1NC(C1CC1c1ccccc1)=O C1(NC(=O)Cn2cnc(Br)c2)C2CC1N(C(=O)Cc1ccns1)C2 N1(C(CNC(CC)=O)=O)CCC(C2CC2)CC1.c1(C=O)cnc(C(C)(C)C)[nH]1.N Cc1cc(C(c2nnnn2CC2CCOC2)NC2CC(C)C2)cc(Cl)c1 C(C(=O)NCC(C)(CC)NC(=O)CSc1ccncc1)(C(C)C)SCC c1(-c2ccc(NC(CCOC)=O)cc2F)ccc2c(c1)OCO2 C(CNC(c1ncoc1C)=O)(CC(F)(F)F)NC(C(C1CCC1)OC)=O C(=O)(C(C)C(C)S(C)(=O)=O)N(C1CCNCC1)CC(C)C.C1(C)CC=CC1.C C1(NC(c2c(C)[nH]c(C#N)c2)=O)CN(C(c2occc2Cl)=O)C2(CCOC2)C1 CC(F)(F)CCC(=O)NCC1(C(=O)NCCc2csnn2)CC=CC1 N1(C(C(=O)NC(C)=O)=O)CCC2(CCN(C(=O)Cc3nccs3)C2)C1.CC.O N1(CC)N=C(C(=O)N2CCC(C)(C)C2)CCC1=O.C(=O)(CC)N.CCN(C)C Cc1cc(Cl)c(C(=O)NCC2CCCC2)cc1N.C1(C(=O)N)(C(C)C)CCC1 C1(NC(C(C)C2CCCC2)=O)CCCC1NC(c1cnn(C2CCOCC2)c1)=O Cc1ccc(OCCC(=O)NC2CCCC(NC(=O)Cc3nc(=N)[nH][nH]3)C2)cc1 C1(C(=O)NCC(C)(C)OC)CCn2nnnc2C1.C(=O)CCCCC.C(N)=O.N CC(CC(=O)N1CCN(C(c2cc(N3CCCCC3)ccn2)=O)CC1C)C(F)F C1(NC(C=CC=CCC)=O)CN(C(=O)CC2CC2(Cl)Cl)CC12CCC2 c1(C(=O)NC2CC(C)(NC(c3ccc(C(C)C)nc3)=O)C2)coc2c1COC2 CC1CN(C(=O)C#CC(C)(C)C)CCN1C(c1csc(S)n1)=O C(CNC(C1(SC)CCC1)=O)(CC(C)C)NC(CNC(CC)=O)=O C1(NC(CCOC(C)C)=O)CCCC1(C)NC(c1cnn(C(C)C)n1)=O c1(NC(=O)NCC2CC3C=CC2C3)cccc2nonc12 C1(CCC)CC(C(=O)NCCCNC(=O)CC2CC(C)(C)CO2)CCO1 c1(C(=O)NC(CCCNC(CC(C=C)C)=O)C)ccccc1[N+](=O)[O-] C1(CC)CN(C(=O)CNC(=O)C)CCN1C(c1csnc1C)=O.C(C)=O.N C1(NC(c2c(C)ncs2)=O)CN(C(=O)C(Cc2ccc(O)cc2)NC)CC1(C)C N1(C(C(C(=O)OC)C)=O)CCCC2(CNC(C3(OC)CC3)=O)CCCC12 c1(C(=O)NC(CC)CNC(C2CCCC(C)(C)O2)=O)ccc([N+](=O)[O-])n1C c1(C(C)NC(c2ccn(CC)n2)=O)ccc(Br)cn1 C(C)(CCCCO)NC(CN(C(=O)CCN1CCOCC1)CC(C)C)=O c1(C(=O)NCCCNC(=O)Cc2cnccn2)cc2nc(Cl)ccc2s1 c1(C(N(CCN(C(Cc2ncc(C)o2)=O)C)C)=O)c2c(nn1C)CCC2 Cc1cc(S(=O)(=O)N2CCCC2CC(c2cnn(C)c2)O)n(CCN(C)C)n1 c1(C(=O)NC23CCC(CN(C(CC(CC)SC)=O)C2)C3)cc2c(cc1N)OCO2 C#Cc1cccc(CC(N2CC(C)CCC2C(=O)NCC2CCOC2C)=O)c1 CCS(=O)(=O)CC(=O)NCc1ccc(CNC(C2CC(C#N)C2)=O)cc1 c1(NC(=O)NC2CCC(C(=O)OCC)CC2)ncc(-c2ccccc2)cc1C C(=O)(C(C)(C)C(=O)N1CC2CC1C2NC(C1OCCN(C)C1=O)=O)OC C1(c2nc(CCCCC)nn2-c2ccc(F)cc2C)CCc2n[nH]c(C)c2C1 C12(CC(=O)NC3(CC)CCCCC3)CCC1CN(C(=O)CN1CCCCC1)C2 C#Cc1cccc(CNC2CC(NC(c3ccc(Cl)cc3C(F)(F)F)=O)C2)c1 c1(CCC)cc(C(N2CC(C)(NC(=O)CC3CC3(Cl)Cl)C2)=O)n(C)n1 C(=O)(CC(C(F)F)NC(C1CCOC1(C)C)=O)NCCCNC(C)=O C1(C2CCN(C(C3CC=CCC3C)=O)CC2)(NC(c2c(OC)ccs2)=O)CC1 C(=O)(CC(C(C)(C)C)NC(=O)CC1CCCO1)N(C)CCC1CCCC1 CN1CCc2cc(C(=O)NC3C4CN(C(C56C=CC(CC5)C6)=O)CC34)sc2C1 c1(-c2cnc(NC(=O)CN3CCCC3)s2)ccc2c(c1)CC2 C1(C(=O)NCC(CCNC(=O)CN2CCOCC2=O)O)CCCC2(CC2)C1 C1(NC(=O)OC(C)(C)C)CC(C(F)F)C1.c1(C=O)cnoc1C(F)F.N CCC(CCCC(=O)NCc1ccccc1CO)NC(=O)CCNC(=O)CO Cc1ccc(OCCC(N2CCCN(C(=O)Cn3ccc(C)n3)CC2)=O)c(Cl)c1 c1(C(N2C(C)CN(C(c3ccc(Cl)cc3Cl)=O)CC2)=O)cccc2oc(O)nc12 c1(C=O)ccc(Cl)c(C(F)F)c1.C1(CNC(=O)C(F)=CCCF)COCC1.C c1(C(=O)NCCCCCNC(c2c(C=C)cnn2C)=O)cnc2c(Cl)cccn12 CC(C)C(C(=O)NCC(O)CN(C)C(C1(N(C)C)CCCCC1)=O)n1ccnc1 Cn1c(=O)oc2cc(NC(c3cc4cc(Br)sc4s3)=O)c(F)cc12 C(CC(=O)N=c1ccn(C2CN(CC3CCCCC3)C2)[nH]1)NC(CCC(C)=O)=O C1(CC(=O)N(C)CC2CC2)(NC(c2c(OC)nccn2)=O)CCCCC1C CC(=Cn1ccnn1)C(=O)NCCC1CCN(C(c2cc[nH]c2)=O)C1 N1(C(C2C(C)C2)=O)CCC2(CCOCC2)C(CNC(=O)C(F)(F)C(F)F)C1 C=CC(CC)CC(=O)N1CCN(C(c2csc3cncn23)=O)C(C)C1 N1(C(C(CCC(=O)OC)C)C(=O)NC2CC2)CCC=C(c2ccncc2)C1 c1(C(=O)NCC=CCNC(CCNC(N)=O)=O)cncc(C(F)F)c1.C c1(C(N2CCOCC2C2CCCC2)C(=O)NCC=C)sc(C)c(C)c1C c1ccccc1.N1(C(C(=O)NC(C)C)=O)CCC(C=O)C1.C(=O)C(F)(F)F.N c1(OC)ccc(C(=O)NCC2CC3(C2)CN(C(c2c[nH]nc2C)=O)C3)cc1F C1(NC(Cc2c(OC)cccc2F)=O)CCC(O)CN(C(c2n[nH]c(C)n2)=O)C1 N1(C(c2cn(C)nc2CCC(F)(F)F)=O)C2CCC1CN(C(C1CCCS1)=O)C2 c1(CNC(C2(O)C(C)(C)C2)=O)ccc(CNC(c2ccc(F)s2)=O)cc1 C1(NC(C=Cc2scc(C)n2)=O)CN(C(C2(c3cc[nH]n3)CC2)=O)CC1C1CC1 C(C(C)(CC)C(N)=O)NC(CN1CCN(C(C2CC(C)(CC)C2)=O)CC1)=O CCCC(CCC)CC(=O)NC1(CCCNC(=O)C(c2ccccc2Cl)C)CC1 S(=O)(=O)(c1cc(F)c2ccccc2c1)NC12CC(C(=O)OC)(C1)C2 C=C(C)CC(C(=O)NC(C)CC(=O)OCC)NC(C1CCCCS1)=O C(C(C(=O)N1CCC(CC2CCC2)C1)OC(C)=O)NC(CSCC#C)=O C1(C(=O)NC2CCCC(NC(=O)CS(C)(=O)=O)C2)(CC)CC(F)(F)C1 c1(NCCCC(=O)OCCC(C(C)=O)F)ccccc1[N+](=O)[O-] c1(C(N(CCC#C)CCOC)=O)n[nH]c2c1CN(C(C1CCCN1C)=O)C2 N1(C(CC2(OCC)CC2)=O)CCC(CC)CC1.C1(=C(C(=O)N)F)CCCCC1 CC1(F)CN(C(c2ccco2)=O)CCN(C(C2C3CCC(F)(F)C23)=O)C1 C#Cc1cncc(C(=O)NC2CN(C(c3cnc(C)n3C)=O)CCC2F)c1 C1(CC)(NC(COCC(=C)C)=O)CCC1.C1(C2C(C(=O)N)C2)CCCO1 C1(NC(C2(COC)CCC2)=O)CC2CC(NC(C3(C)CCC3)=O)CC12 c1cc(C)ncn1.c1(C(=O)N)cn(CC(N2CCC(CC)C2)=O)nn1.CC(=O)N C(C(=O)NCC(C)N(C(=O)C)C)(C(C)C)NC(=O)OCC.CC(C)C C=CCC(CC)C(=O)N1CCC(C)(C(=O)NCCC2CCOC(C)C2)CC1 C1(NC(c2nnnn2C2COC2)(CC)C2CC2)C(C)CCC1C CC1C(NC(=O)C(c2ccc(Br)cc2)(F)F)CCN1C(=O)CCOC1CC1 C(CC(O)C(=O)N1CC(O)(CCNC(=O)CN2CCCCC2=O)C1)SC c1(C(N2CC(C)(NC(c3nn(C)c(F)c3)=O)C2)=O)cc(Br)c(F)cc1F Cc1cc(O)c(C(N2CCN(C(=O)CNC(=O)C(C)CO)CC2)=O)cc1F C12(NC(c3c(C)nn[nH]3)=O)CCCC(CN(C(=O)Cn3nccc3C)C1)C2 c1(C(=O)NC2CCC(NC(c3cnc(C)s3)=O)CC2)cc(C)c(C(N)=O)cn1 C(=O)(C(CC)C(=O)OC)NCC=CCC(=O)N(C(CC)C(=O)OC)C C1(C)(C(=O)N)CCC(C)(C)CC1.CC1CN(C(C2(CCF)CCC2)=O)CCC1C Cc1cc(Cl)ncc1CC(=O)NC1(CCNC(=O)Cc2[nH]cnc2C)CCC1 C1(C)(CC(=O)N(CC(CN(C)C)O)C)CC1(F)F C1(NC(c2ncc3n2CCCC3)=O)CN(C(=O)CC2CC2(Cl)Cl)C2CCCC12 CC1(C)OC(C)(C)C1C(=O)NCCCCNC(C1CCCC1O)=O Cc1csc(C=CC(N2CCC(CN(C)C(C3CCC4(CC4)C3)=O)CC2)=O)n1 c1(OC)cc(Br)ccc1C(=O)NC1CN(C(c2sc(C)nc2C)=O)CC1F C(=O)(C(C)CCCC(C)C)N(C1CCN(C(C(CCC)OC)=O)CC1C)C C1(NC(C(CC=CC)CC)=O)CC12CCN(C(c1cccc3nccn13)=O)CC2 C(=O)(C(F)CCC(C)C)NC1C(NC(c2cc(CC)no2)=O)CCC1 C(=O)C1=CCC(C)(C)CC1.Cc1nc(COCC(C)C)sc1C(N1CCC1)=O c1(C=O)cnc2c(c1)NC(=O)CO2.c1(CC)c[nH]c(C(=O)NCC2CC2)c1 Cc1cc(C(N2CCC(O)C(C(=O)NC(C3CCOC3)C)C2)=O)cc(Cl)c1 C(=O)(C#CC(C)(C)CNC(=O)CCC(=O)N(C)C)Nc1c(C)cccc1O C1(OCC(=O)NCCCCCCNC(C=CS(C)=O)=O)CCC(F)(F)CC1 C1(C(C)C)OCCCC1CNC(=O)CNC(c1ccccc1)=O.C(C)(C)C c1(CC)cc(C(=O)NCCCCN(CCCN)CCCN)c(C)nn1 c1(C(N2CCC(NC(C3(C)CCCCNC3=O)=O)C2)=O)c(F)ccc2c1OCC2 c1(CNC(C2(CSC)CCCC2)=O)cc(C(=O)NCC(C)(F)F)no1 C(C1=CCN(C(c2cc(C)ncc2C)=O)CC1)NC(C1CCC(CC)O1)=O c12c(cccc1Br)NC(=O)C1(C)CCCN1C2.c1(CC)ccccc1C(=O)O C1(C(=O)NCC(c2ccccc2)NC(C(C)(C)O)=O)CC2CSCC(C1)C2 c1(C(C=O)C)c(C)nn(C)c1C.N1(C(C)=O)CCC(C(=O)NC2CCC2)CC1.N CC(C)CC(CNC(C1(C#N)CC2CC2C1)=O)C(=O)N1CC2CCN(C)C2C1 C1(C(=O)NCc2c(CC)nco2)CC(NC(=O)CC2(O)CCCC2)CCO1 N1(C(CCC)=O)CCC2(CC1)CN(C(C13CCCCC(OC)(C1)C3)=O)C2 N1(C(c2nc(C)sc2C)=O)CCCC(NC(c2ccc(CO)c(F)c2)=O)CCC1 O=C(CS(=O)C(F)(F)F)NCC1(NC(=O)CCc2cncs2)CCOCC1 CCCC(O)CC(=O)C1CCC1.C(=O)(CNC=O)N.C(C)(C)C.C(C)N CCCC(CCC)CC(=O)N1CCC2(NC(C3CN4CCCN3CC4)=O)CC2C1 N1(C(C(CNC(c2ccc(CC)[nH]2)=O)CC2CCCC2)=O)CCSCCC1C C1(C(=O)NCCC(CNC(C(COC)C)=O)O)SC2C=CC1CC2 n1(C2CN(C(CN(C(C)=O)C)=O)C2)cc(CNC(=O)C(C)n2ccnn2)nn1 C(=O)(C1=CCN(C(=O)CN2CC3CC3C2)C1)N1CCC(O)(COC)C1 Cc1cn2c(n1)CCC(C(=O)NC1CCCC1NC(c1cn(CCF)nn1)=O)C2 N1(C(CCSCCCC)=O)CCC(C(C)NC(=O)C(C)Cc2cnn(C)c2)C1 N1(C(C2CC(C)N(C(=O)CN3CCCC3=O)CC2)=O)CCC2(CC1)CN(C)C2 N1(C(c2nc(OCC)oc2)=O)CC(C(=O)N(C2CCC2)CC)C2(CCC2)C1 N1(C(C(C2CN(C(=O)C(C)(C(C)C)O)C2)OCC)=O)C2CCC1CC(CC)C2 c1(C(N(CC(CC)NC(=O)CN2CC(C)C2)C)=O)cc(S(N)(=O)=O)c[nH]1 n1(CCC(=O)NCC(=O)NC2C(C)(C)CNC2)cc(Cl)c2cccnc12 Cc1csc(C(F)(F)C(=O)NCCN(C(=O)CN2CC=CC2)C(C)C)n1 CC(C(=O)NC1CCC(C)CC1)C(C)(F)F.n1(CC=O)ccc([N+](=O)[O-])n1.N c1(C(=O)NCCC(C)SC)ccc(CC#N)cc1.C1(=O)C(F)CC2CN1C2 C1(C(N2C(C(C)(C)O)CCC2)=O)CCCN1NC(=O)C(F)C(C)(F)F c1ccc(C#N)cc1.C1(CNC(C2(C)CC2(F)F)=O)CCCC1O.C(=O)(C)N N1(C(C2(C=C)CC2)=O)CCCC(NC(=O)C(CN2CCCC2)c2ccccc2)C1 N1(C(c2ncc(Br)cn2)=O)CCN(C(C2CC3C=CC2C3)=O)C(CCO)C1 c1(CN(C)C)ccc(C(=O)NCC#CCNC(=O)C(c2cccnc2)O)cc1 CC1N(C(C2CC3C=CC2C3)C(=O)NCc2cccs2)CCOC1(C)C C(CN=c1[nH]c(N2CC=C(C(C)(C)C)CC2)nc2c1CCC2)(N(C)C)C1CC1 CC(C)(C)C(CNC(=O)C=Cc1ccncn1)C(=O)NC.C1CC1C1CCC1 C(=O)(C1=NOC(C)C1)NCCCCCCn1cc(C(CCC)=O)nn1 c1(C(=O)NCCCN(C)C(c2cnccn2)=O)cc2scc(Br)c2s1 C1(CNC(c2ncn(CC)n2)=O)CCN(C(c2cnc(SC)s2)=O)C12CC2 CC1=C(C(=O)NC2CCCC2NC(=O)C(c2ccccc2C)C)CCO1 N1(C(C2CC(N(C)CC)C2)=O)CC=CC(NC(=O)C=C2CCSCC2)C1 c1(C(N2CC(CNC(C(C3CCC3)OC)=O)C(O)C2)=O)ccc2c(c1)OCO2 c1(CC)c(C(=O)NC(C)Cn2cc(-c3cnc(C4CC4)o3)nn2)cccc1C c1(OC)ccc(NC(=O)C(c2ccc(N(C)C)cc2)NC2CCCC2C)c(C)c1 N1(C(c2c(CC)scn2)=O)CCN(C(c2ccc(C)n2C)=O)C(C)C1 N1(C(CCC)=O)CCn2nc(C)cc2C1.C1(C2C3CCN2C3)CCOC1(C)C N1(C(C(C)SCCCC)=O)CCCC(CC(=O)N(C(C)CC2CCCCC2)C)C1 CCC(CC)CN=c1nc(N2CCC(C)(F)CC2)c2c([nH]1)COC2 C1(C(=O)NCCN(C(=O)CCS(=O)(=O)N(C)C)C)C2Cc3ccccc3C12 C(=O)(C1CCCc2ncnn21)N(CCC)CCNC(C1CCCCCCC1)=O C1(C(=O)NCC(CNC(CC(=C)C)=O)C)CC(=O)N(CC(F)(F)F)C1 c1(-c2c(CN3CC(c4ccccc4)OCC3)csc2)cccc2ccsc12 CCCC(C)C(=O)Nc1cccc(C(=O)NCCc2nccs2)c1 C1(NC(CC2N(C(C)C)CCC2)=O)CCCC(NC(=O)Cc2c[nH]ccc2=O)C1 c1(N2C3CC(C)CC2CC3)nc(N2CC3CCCC(C2)N3C)c2c(n1)CCOC2 C(=O)(CCC(CC)OC)N1CC(CCC=C)(C(=O)NC2CCSCC2)C1 N1(C(c2cccc(CC)c2)=O)CCN(C)CC1CNC(=O)CCCCOC CC1CCN(C(=O)CCN=[N+]=[N-])C1C(=O)NC1CC(CO)C2CC12 c1(C(N2CC(C)C(CNC(=O)C(C)(C)O)C2)=O)ccc(F)c(C(F)(F)F)n1 c1(C(N(C(C(=O)NC(c2ccc(C)s2)C)(C)C2CC2)C)=O)ccc(C#N)cc1C C(=O)(C(C)C1CCC1)NC(C=C)C1CC1.C1(C(=O)N)CCCN1C(N)=O c1(C(N2CCC(NC(Cc3scc(C)c3)=O)C(F)C2)=O)cnc2occc2c1 C1(N(C(C(CC)=CCCC)=O)C)CCCC(NC(c2cc(Cl)n(C)n2)=O)C1 N1(C(CSc2nc(C)[nH]n2)=O)CCCC(F)(C)C1.C1(C)(CC=O)CC1(Cl)Cl.N C(=O)(CC(C)(C)CC)NC(CC#C)C(=O)NC1CC(=O)N(C)C1 c1(CNC2CN(C(C(CC)O)=O)CC(C)C2)cc([N+](=O)[O-])ccc1O C(=O)(C(C(=O)N1CCN(c2nn[nH]n2)CC1)SCCO)OC(C)(C)C C#CC1(F)CCN(C(C2(C=C)CCN(C(=O)C=CC(=O)N(C)C)CC2)=O)CC1 Cc1ccsc1CCCC(=O)N(CC(C)NC(=O)CCN1CCC(F)C1)C CC(C)C(C)(C)C(=O)NC1C2CC(NC(=O)CC(C)(F)F)CC12 C#CC1CCN(C(c2cnc(C3CN(C(=O)OC(C)(C)C)C3)nc2)=O)CC1 CON(C)C(=O)CNC(=O)C=CC1CCCN1C(=O)C(C)=NOCC#N C1(NC(c2c(NC(C)=O)cccn2)=O)CCCC12CN(C(C1CCNC1=O)=O)C2 C12(NC(CC(=C=C)C)=O)CCN(C(=O)C(c3cccc(F)c3)F)CC1C2 c1(C(=O)NC(CNC(CC2(OCC)CC2)=O)CC)c(Cl)ccnc1C C(=O)(CC(F)(F)CS(C)(=O)=O)N1CCCCC1C.c1(COC)nc(C=O)co1 C12(CNC(C=C(c3cn(C)nc3)F)=O)CCCC1N(C(C1CCCC1)=O)CCC2 CCC(CC)(C(=O)NC1CCCC(NC(=O)C=C(Cl)Cl)C1)c1ccccc1 C12(C(=O)OC)CCCC1CN(C(C1(c3cc(C)no3)CC1)=O)C2.c1nn[nH]c1C.C N1(c2nnc(C3CC(C)C3)n2CC2CCOCC2)CCCC2(CC(=O)N(C)C2)C1 n1(CC#C)cccc1C(=O)NC(C)CCOC.c1(C(=O)N)cc(CCC)[nH]n1 Cc1cnc(NCC(O)C2(Cl)CC2)c(S(=O)(=O)NCC2CC(F)C2)c1 N1(C(c2c(C)noc2)=O)CC(C(=O)N(CCCC(F)(F)F)C)C2(CC2)C1 N1(C(C2(NC(N)=O)CC2)=O)CCN(C(C2CCS2(=O)=O)=O)CC1 Cc1cc(C(=O)NCC(CO)NC(=O)Cc2ccc(C(N)=O)cc2)cc(O)c1 c1(C(=O)NC2CC(CNC(C3(C)COCCO3)=O)C2)c(F)cc(Br)cc1F O=C1NC(=O)C2CN(C(C3CCC3CNC(C3C=CCS3)=O)=O)CC12 N1(C(c2scc(C)c2)=O)CCOC2(C1)CN(C(=O)CC(C)C(C)C(C)C)C2 C(CC(C)C)(C(=O)N1CCC1C1CCOCC1)ONC(c1c(C)cc(F)s1)=O C1(C(=O)NCC2(C(=O)NCCCCC)CC=CC2)C2CC3C(C2=O)C13.O C12CCC(C(=O)N(CC(C)C)C)(CC1)CO2.C(=O)C(C)CC(F)(F)F.COC C(=O)(CCCC(N)=O)N(C1CCCN(C(c2cc(C)sc2C)=O)C1)CC CC1CN(C(=O)CC2CCC(=O)NC2=O)CCN1C(=O)COC(F)F CN1CCCC(CNC(=O)C(F)CC2CN(C(=O)Cn3cnnn3)C2)C1=O C(=O)(C1=NN(C)C(=O)CC1)N1C(C(=O)N)C(C2CC2)CC1.Cc1cccnc1C c1(C(=O)NCC2CCCC2C=O)ccc([N+](=O)[O-])[nH]1.c1cnn(CCO)c1.N C12(C=O)CCCC1C(F)(F)C2.C(CCOCC(=O)NCCOCC)OC N1(C(c2ccsc2)=O)CCC2OCCN(C(C3CC=CCO3)=O)C2C1 Cc1cnc2cc(C(N3CCC(n4cc(CC5CCC5)nn4)C3)=O)ccn12 c1(OC)cccc(S(=O)(=O)NNC(=O)OC(C)(C)C)c1 C(=O)(CC(C)C(=O)N1C(CC(=O)NC(C)Cc2cccs2)C2CCCC12)OC c1(C(N2CC3C(CNC(c4ncccc4Cl)=O)(C3)C2)=O)noc2c1CCCCC2 N1(C(CN(C(C)=O)C)=O)CC2CCC(C)(C2)C1.C1(C(=O)N)CN(C(C)C)C1 c1(C(N2CCCN(C)CC2C)=O)ccc(Br)c([N+](=O)[O-])c1.c1(OCC)ccccc1 N1(C(C(C)OCC#C)=O)CCC(NC(=O)C(=Cc2ccco2)C)C12CC2 c1(CCC)ccc(CC(=O)NCC2CCCN(C(c3cc(=O)n(C)o3)=O)C2)cc1 C(=O)(CCC(F)(F)F)N.c1(OCC)cnc(C(=O)NC2(C)CCCC2)cn1 C(=O)(C(O)C(C)(C)C)NC(C1CN(C(C(C=C=C)C)=O)C1)C c1(NC(C23CC(c4ccccc4)(C2)C3F)=O)ccc(N2CCCS2(=O)=O)c(F)c1 C1(CC)CNC(=O)CN1C(c1ncsc1Br)C(=O)NCc1nnn(C)n1 C#CCC(CC(F)F)C(=O)N(CC(=O)NC(C)CC(=O)NC(C)C)C1CC1 c1(C(=O)NCC(C)N(C(CC(C(N)=O)NC(C)=O)=O)C)ccc2n[nH]cc2c1 N1(C(c2c(C)coc2)=O)CCCC1(C(=O)Nc1cccc(CCO)c1)C(C)C N1(C(CCN(CC)CC)=O)CC2CCC(C1)C2C.C1(C=O)CCNC(=O)C1.N c1(C(=O)NCC(C2CC2)NC(CCSC)=O)cc2ccsc2n1C CCC(CNC(c1coc(CNC(C2CCOC2C(C)C)=O)c1)=O)C(C)C N1(C(C(c2ccc(F)cc2)C)=O)CCN(C2CCC(NC(C3(O)CC3)=O)C2)CC1 c1(CSC)cccc(-n2cncn2)c1.C1CC(C(=O)NC(C)(C)C)N1C N1(CC(=O)NCC2CCN(C(=O)CCF)CC2)CCCC(C(F)(F)F)C1=O CCCCCC.[nH]1ncn(C)c1=O.C(=O)C(NC(C)=O)=Cc1cccs1.C(C)=O.C N1(C(C2(C=C)CC2)=O)CC(NC(c2c(Cl)n[nH]c2C)=O)C(O)C1 C12(C(N(C(CO)C3CC3)C)=O)CC(NC(C3CC3F)=O)(C1)C2 c1(C(N2C(C(=O)NC(CC=C)CO)C=CC2)=O)ccc([N+](=O)[O-])cc1I Cc1cccc(CCC(N2CCC(C)(NC(=O)COC3CC=CC3)C2)=O)c1 c1(C(=O)NC2CCOCC2F)cc2cccnn2c1.C12CCC1CNC2=O C1CC2(CC2)CN1C(C1CCS(=O)(=O)C1)=O.n1(CCC)cccc1C(=O)N C(C)(C)(CC(F)C(=O)NC(C)Cc1nn[nH]n1)NC(C(CC#C)C1CC1)=O C1(C)(C(=O)OC)CCN(CC2CCC(C(=O)Nc3c(C)cccc3C)C2)CC1 C1(CCC)CCc2c(sc(=O)n2Cc2c(C)sc(C)c2Br)C1 C(C(O)CC(=O)NC(C)C(C)n1cccn1)NC(COCCCOC)=O N1(C(COC(CC)C)=O)CCC2CN(C(=O)CC3(COC)CCCC3)CC12 n1(CC)cnnc1C(N1CCCC1CN(C)C(c1nsnc1O)=O)=O c1(NC(C2CCC(c3ccccc3)O2)=O)ccc2ncnc(O)c2c1 C1(C(N2C(C)(CO)CC2)=O)CCCCN1C(N)=O CC1=C(C(=O)NCC2CN(C(c3ccsc3C)=O)CCC2C(F)(F)F)CCO1 C(CC(=O)N1CC(F)CC1)(C(C)C)OCC.c1(C(NC)=O)ccoc1C1CC1 C(=O)(C#CC1CCCCC1)NCCOC1CN(C(c2nc(C)sc2C)=O)C1 c1(CC(C)NC(c2nnc(Br)n2C)c2n(C(CC)(C)C)nnn2)ccccc1C C1(C(N(CCCCO)CC)=O)C2CCCC1CN(C(=O)Cc1ccc(F)c(F)c1)C2 Cc1cc(C(=O)NC2(C)CN(C(c3ncn4ccccc34)=O)C2)c2[nH]cnc2c1 n1(CC)ncc(C(=O)NCC(C(C)(C)C)NC(c2nnc(C)s2)=O)c1Cl Cc1cc(C=CC(N2CC(NC(C3C(C)C3C)=O)C(O)C2)=O)ccc1Br C1(CCC)CCCCN1C(=O)C=Cc1cn(C)cn1.C(C(=O)N)(N(C)C)C1CC1 C1(C(=O)NC(c2nn[nH]n2)CC)CC12CCN(C(=O)C=Cc1ccccc1)CC2 c1(NC(=O)NC2CC(C)(C)C2)ccc(C(N)=O)cc1 C1(CNC(C2(C)C=CCCC2)=O)CCN(C(C2CN3CCCC2C3)=O)C12CCC2 c1(C(=O)NC(CNC(CCN(C)CC)=O)C2CC2)nccc2ccsc12 Cc1cc(=NCCC2CCN(Cc3ccccn3)C2)[nH]cn1 c1(C(=O)NC2CCC(NC(CC(C=C)C)=O)C2)c(OC)cccc1O C1(NC(Cc2ccc(C)nc2)=O)CC2CC1CN2C(c1cncc(F)c1)=O C1(C(N2CC(O)(CCC)C2)=O)C(C)CCN1C(=O)CCCCOC Cc1ccc2c(C(N3CCC(NC(c4ccn(C)c4)=O)C(F)C3)=O)n[nH]c2c1 c1(C(=O)NC(CNC(C(CC)C(=O)OC)=O)C)ccn2c(O)nnc2c1 c1(OC)ccc(NC(=O)CCC(C)(C)NC(c2nonc2C)=O)cc1F N1(Cc2cc(C)on2)CC2CCN(C(c3cc4cccnc4s3)=O)CCC2C1 Cc1ncc(Br)cc1CNC(C1(O)CCN(Cc2cc(O)ccc2Br)C1)=O C1(NC(C2CC(CC)(CC)C2)=O)CCC(C)N(C(=O)C(F)CC2CC2)C1 c1(C(N2CCC(C)(CNC(c3cc(C)[nH]c3C)=O)C2)=O)cc2c(s1)CCC2 n1(CCC(=O)NC(CNC(c2c(CCC)n(C)nn2)=O)C)ccc2cccnc12 c1(CN(C(C(C)CNC(c2nc[nH]n2)=O)=O)C)cccnc1O C(=O)(CCCC(C)(C)NC(=O)C(C)N1CCCC1)N(C1CSC1)CC#C C1(C(=O)NC2CCCC2NC(c2ccn(C(C)(C)C)c2)=O)(OC)CCOC1 C1(C(=O)NCCOCCNC(c2c(C)nc(O)s2)=O)CC2C=CC1CCC2 C1(CCC)CN(C(=O)COCC(=O)OC)CCN1C(c1ncn(CC)n1)=O N1(C(c2c(N)nccn2)=O)CC2CCCCC2(CNC(=O)C=Cc2cnc[nH]2)C1 c1(C(=O)NCC(C)(CO)NC(c2cccc(Cl)c2O)=O)cnn2c1CCC2 c1(OC)ccc2nc(C(N3CC(n4cc(C5CCN(C)C5)nn4)C3)=O)sc2c1 C(=O)(CCC(CC)NC(c1cnc(Cl)s1)=O)NC(CC=C)C CCCCC(C(=O)O)NC(Cc1ccc(C(C)(C)C)cc1)C(=O)O C(=O)(C#CC1CCCCO1)N(CC(C)(C)NC(C=C(C)C)=O)C c1(C(=O)NC2CC3(CN(C(C(F)=CC)=O)C3)OC2)cc2ccccc2n1C C(=O)(CCCC(C)NC(c1cccc(O)c1)=O)NCC(CC(C)C)C C1(C(N2C(C(=O)Nc3cn(CCOC)nc3)C=CC2)=O)CCC(F)(F)C1 c1(CC)cc(N2CCC(CO)(CO)C2)nc2ccccc12 CC1(C)CC(C(=O)N2CCC(C3(NC(c4csnc4Br)=O)CC3)C2)=NO1 C1(OCC)CCC(C(N2CC(CO)C2)=O)CC1.C1(n2ccnn2)CCCC1(C)O.O N1(C(C(C)c2ccsc2)=O)CC2CCC(C1)C2CNC(=O)CCc1ccoc1 C1(C(C)NC(C(C)OCCOC)=O)CCN(C(=O)CCC2CCCC2)CC1 N1(C(c2cc(C)ns2)=O)CC(CN(C)C(c2ccnnc2O)=O)C2(CC2)C1 S(=O)(=O)(C1CC(F)(F)C1)NC1(C)CC(N)C1 C1(OC)Cc2ccccc2N(C(C2C(c3ccccc3)C2(F)F)=O)C1C c1(CC)ccc2c(c1)C(NC(C1CCCN(CCC(=O)O)CC1)=O)C(=O)N2 N1(C(CCC#C)=O)CC=CC1(C)C(=O)NC(c1ccnn1C)C c1(OCC(=O)NCC(C2CCCC2)NC(C2C=CCC2)=O)cccc(F)c1 C1(NC(CCC)=O)C2CCN(C(c3ccc(-n4cccc4)nc3)=O)C12 c1(C(=O)NC(CCN(C(C=C(C)C(C)(C)C)=O)C)C(C)C)cc2ccsc2n1C c1(C(=O)NC2CCCN(C(C(C)(C)c3cncs3)=O)C2)nc2ccccc2[nH]1 C1(CNC(c2cnn(-c3nccs3)c2)=O)C2CN(C(c3ncncc3F)=O)CC12 C1(C(N2CC(N(C(c3cnc(OC)c(Cl)c3)=O)C)C2)=O)CCc2n[nH]cc2C1C c1(OC)ccc(NC(=O)NC2CCC(C)C2)nc1F CCC(C(=O)NC(C1CCCN1C(c1nccc2ccsc12)=O)C)C(C)(F)F N1(C(C(CC)(C)CC)=O)CC(C2CCCN(C(=O)C(C)SC(C)C)C2)C1 c1(C(=O)NCc2c(OC)cncc2)n[nH]c2c1CN(C(c1cc(F)ccc1C)=O)C2 N1(C(C(C(C)C)F)=O)CC(CNC(c2ccc(CCO)cc2)=O)CC12CCC2 C1(CCOC)(NC(=O)CSCC(C)C)CCN(C(C2CCCCC2)=O)C1.C c1(C(=O)OC)ccc(C)c(C(=O)NC(C)CC(C)NC(c2cnoc2)=O)c1 N1(C(=O)C(O)c2ccsc2)CC2CCC1CN2C(C1(CO)CCOCC1)=O N1(C(CC2(OC)CCCC2)=O)CCN(C(c2cc(C)on2)=O)C(C2CC2)C1 C1(C)(NC(c2scc(C(C)=O)c2)=O)CCN(C(=O)CCN2C(=O)CCC2=O)C1 N1(C(c2ccc(C)cc2F)C(=O)NC2COC2)CCCC2(C1)C(O)CC2O c1(C(N(C2CN(C(C(C(CC)C)O)=O)CC2(C)C)C)=O)nn(C)c2ccccc12 c1(CC)cccc(OCC(=O)N(CCCNC(=O)C(N)=O)CC)c1 c1(C(N2CCC(N(C(Cc3c(C)non3)=O)C)C2)=O)ccc(N=[N+]=[N-])cc1 c1(C(N2CCC(C(C)C(=O)NCC3CCC(F)C3)CC2)=O)ccc(CCO)cc1 N1(C(c2cncc(CC)c2)=O)CCN(C(=O)CC2C(=O)NN=C2C)CC1CCO N1(C(C2C(C=C)C2)=O)CCN(C(c2cc(-c3ccc(O)cc3)on2)=O)CC(O)C1 CC1(C)CCC(C(=O)N)O1.c1(C=O)ccc(CS(C)(=O)=O)cc1.C1CCC1.C CC(CNC(c1ccon1)=O)(CO)NC(c1ncsc1Br)=O C12(NC(CC(C)O)=O)CC(CO)(C1)OC21CN(C(=O)CCC(=O)N(C)C)C1 C(c1cn(C(C)(C)CC(=O)NC2CCN(C(C)(C)C)C2)nn1)=CC c1(CCC(=O)N(CCN(CC(=O)NC)C)C)ccc(OC)cc1 C(C(C)C(=O)NC(c1csc(C)n1)C)NC(CCSC)=O c1(CNC(C(C)CC2CCC2)=O)ccc(C)cc1.c1ccccc1.C(=O)(C)N Cc1ccccc1C.C(=O)C=CS(C)=O.C(CCC)N(C(C=CC(=O)O)=O)C.N C(CC(N)=O)(C(=O)NC(c1cnn(C)c1C)C)NC(C1CN(C(C)=O)C1)=O CC(C)C(C)CC(=O)N(CC(C)NC(=O)CCCn1cncn1)C N1(C(c2c(C)snc2)=O)CCC(NC(c2cc(C#N)cn2C)=O)CC1C c1(C(=O)NC(c2cn(CCCc3ccccc3)nn2)C)c(F)c(F)cc(F)c1F CCC(C)CCCCC(=O)NCC(C)N(C(=O)Cc1ccc(OC(F)F)cc1)C CC1(NC(c2cccc(C3CC3)c2)=O)CCN(C(=O)C=CSc2ccccc2)C1 c1(CNC(C2(C)C=CCN2C(c2cccc(CO)n2)=O)=O)cncc(C#N)c1 N1(C(=O)C2=CCN(C(C3CC34CC4)=O)C2)CCCC(O)(C2CC2)C1 c1(C(=O)NC(CCCC)CNC(=O)CC(F)(F)F)c[nH]cc(F)c1=O C(=O)(CCC(C)(C)C#N)N1CCC(OCCNC(C2C=C(C)CS2)=O)C1 c1(CC)ncncc1C(=O)NCC(C)(C)NC(C1CCC(C(N)=O)O1)=O c1(OC)ccc(Cl)c(CC(N2CC(CO)(NC(=O)CC(C)O)C2)=O)c1.C1CC1 c1(C(=O)NC2CCN(C(c3cn(C)nn3)=O)C2)nc2cc(F)ccc2s1 C1(NC(C(C)(C)OC)=O)CCCCCN(C(C23CCC(F)(CC2)C3)=O)C1 CC1CC(NC(c2ccccc2C(N)=O)=O)CN1C(=O)COC.C1CCC1 Cc1cc(C(=O)N)nn1CCO.C(=O)(C(O)CN1CCCC1)N(CC)C(C)C C1(NC(Cc2c(C)nc[nH]2)=O)CN(C(=O)C(O)CCc2ccccc2)CC1C c1(NCC)cc(I)ccc1NC(=O)NCC(C)Cc1ccc(O)cc1.CC N1(c2snc(C)n2)CCCN(C(=O)NCC(c2ccc(Cl)c(F)c2)F)CC1 c1(C(=O)NCC2C3CC2N(C(=O)Cc2c[nH]nc2O)C3)cn2c(n1)CCCC2 c1(C(=O)OC)cc(C)c(NC(=O)C(C)Oc2ccc(F)cc2Cl)nn1 c1(C(=O)NCC2(C)N(c3cc(C)nc(CO)n3)CCC2)cnc2ccccc2n1 N(C(=NCC(F)F)N(C)Cc1ccc(F)cc1C)Cc1ccc(C)cn1 C#Cc1ccc(CC(=O)NC2(C(=O)NCCCC(C)(F)F)CCCCC2)cc1 N1(CC(=O)NC2C(C(=O)NCC(C)C)CC2)CSCC1=O N1(CC)CCCC(C(N2CCCC2(C)C(=O)NC2CCCC2(C)C)=O)C1 N1(S(=O)(=O)C2CC2)CCCc2sc(Br)cc2C1.c12ccc(c(C(F)(F)F)c1)[nH]2 c1(CC(=O)NC2CCCN(C(C(CC)CCOC)=O)C2)c[nH]c2ccc(Cl)cc12 c1(OC)ccc(C(N2CCC(C(C)C(=O)NCC3CCOCC3)CC2)=O)cn1 Cn1cc2c(n1)CC(C(N1CCCC3(CCO3)CC1)=O)NC2=O N1(C(C(C)Oc2ccc(F)cc2)=O)CCCCC(NC(c2ccc(Cl)cn2)=O)C1 c1(C(N(C2CCCN(C(=O)COCCSC)C2)CC)=O)cc(Cl)ccc1O N1(C(c2[nH]c(=N)sc2)=O)CCCN(C(=O)C(O)Cc2cccc(Cl)c2)CC1CO N1(C(C(C)(O)C2CCC2)=O)CC(C2CCN(C(c3cnns3)=O)CC2)C1 C1(O)(Cn2cc(CSC)nn2)CCCN(C(c2csc(C)c2)=O)CC1 C12CCN(CC1)CCNS(=O)(=O)C2.C1(NC)CC(C(=O)OC)C1 CCCC(CNC(C1(Br)CC1)=O)NC(c1cc(C(C)C)on1)=O C1(C)(CC(=O)NCCCC2(C)CC2)CCN1C(=O)CCN1CCCCC1 CS(=O)C=CC(=O)N1CCC(C)(NC(c2c[nH]c(-c3ccccc3)c2)=O)C1 CCCCS(=O)(=O)CC(=O)N1CC(NC(c2ccc(CC)cc2F)=O)C(C)C1 N1(C(CCC)=O)C2CCC1C(CNC(c1nccc(C(F)F)n1)=O)C2 C1(NCc2cc(C)cc(F)c2)CN(C(=O)OC(C)(C)C)Cc2nccn2C1 C1(C(=O)NC2(CC)CN(C(C3(C=C)CCC3)=O)C2)CCCC(C#N)C1 N1(C(C)C(N2CC3(NC(=O)C4=CCCSC4)CCC2C3)=O)CCc2sccc2C1 Cc1nc(C(C)C)nc(O)c1C(=O)N(CCCNC(c1cn(CCO)nn1)=O)C Cc1cc(C)n(-c2ccc(-c3cccc(Oc4ccccc4)c3)nc2)n1 c1(C(=O)OC)cc(NC(=O)NCC2(O)CCCOC2)cc(C)c1F C(C1CCCO1)=CC(=O)NC(CNC(=O)CCCN1CCCCC1)C1CC1 c1(COCC)nc(C)c(C=O)s1.C(CO)CC.C1(C=O)CN(C(C)=O)C1 c1(C(=O)NCC(C)N(C(C(C2CCOCC2)OC)=O)C)ncc[nH]c1=O c1(CC(N2CC(CC=C)(NC(=O)C(CC)SC)C2)=O)cc2ccccc2nc1O Cc1ccc(NC(=O)CN2CC=CC2Cn2ccnn2)cc1.NS(N)(=O)=O.C NS(=O)(=O)c1ccnc(C(=O)NCc2cccc(F)c2)c1.C(=O)CC(F)F.C C1(C=O)CC12CCS(=O)(=O)CC2.N1(C(c2cn(CC)nn2)=O)CCC(C)C1.C C1(CNC(CNC(C(CC)C)=O)=O)CCCN(C(C2C=CC=CC=C2)=O)CC1 c1(C(N2CC(NC(CC(OCC)OCC)=O)C(C)CC2)=O)cccc(C#N)c1C C1(CCNC(CCCCOCC)=O)C(C)CCCN1C(c1oc(C)nc1CC)=O C12CC=CC(C1)OC2.c1(C(C)C)ccc(C(=O)N(CCC(=O)N)C(C)C)o1.C C(CCC(=O)NCC(C)(C)CO)N(C(C1C(C)CC1)=O)C N1(C(C(CC=C)CC=C)=O)CCN(C(c2ccoc2C)=O)C2CCCCC12 N(C1CCc2cccnc21)C(C1N(C(=O)C=CC2CCC2)CC12CCCC2)=O Cc1c(NCc2ccccc2Cl)ncnc1N1CCN(Cc2cccs2)CC1 Cc1cccc(-c2noc(C)c2C(=O)N(C)CCNC(C2(C)CCNC2=O)=O)c1 CON(C(=O)C1=CC(O)C(NC(=O)C(C)CC2CCC2)C1)C(C)C C12(CNC(c3c(CC)nco3)=O)CC(C1)C(C)(C)O2.C1(C=O)CCC1 N(C(=NCCOCC1CCOC1)N1CCN2C(=O)NCC2C1)CC(=C)C N1(C(C(C)C#N)=O)CCC(OCCCNC(=O)C=Cc2ccoc2)CC1 C1(NC(CC2(CC)CC2)=O)CCOC(C(C)(C)C)C1.N1(CC=O)CCCCC1 c1(OCC(=O)NC2CCCCC2NC(C2CC=CCO2)=O)ccc(F)nc1 c1(C(=O)NCC(CCNC(c2cocn2)=O)O)c(O)ccc(Cl)c1F C1(NC(c2ccnc(F)c2)=O)(CO)CCCN(C(=O)COC2CCCCCC2)C1 C(c1c(C)cc(C)cc1C)=CC(N1C(C)CC(NC(C(CC=C)(F)F)=O)C1)=O C1(C(=O)N)(CC)CCCN(C(c2cc(C)[nH]c2C)=O)C1.c1(CC)cc(C)n(C)n1 c1(C(N2CCC3(C(C(N4CCC(C(=O)OC)C4)=O)C3)C2)=O)c(Br)ccc(C)c1F N1(C(C(C(C)C)N(C)C)=O)CC(N(C(=O)CC2OCCO2)C)C(C)(C)C1 C(c1cccc(Cl)c1)=C(C)C(N1CC2(C1)CN(C(=O)CC(O)C1CCCC1)C2)=O C1(NC(c2cn(C)c(=O)cc2)=O)CCN(C(=O)CCC(C)(C)F)C12CCCC2 Cc1cc(C(=O)NC2(C)CCCC2)nnc1C.c1(CC=O)cn(C(C)C)nn1.N C=CCC(CC(=O)N1CC(CO)C(C)(C)C1)NC(C1CN2CCN1CC2)=O C1(F)(CNC(C=NOC)=O)CCN(C(=O)CC2CCC(=O)NC2)C1 C1(CNC(c2cc(CCC)[nH]n2)=O)C(C)CCN1C(=O)CC1CCOCC1.O Cc1ccc(F)c(C(=O)NCCCCC(N2CCCSCC2C)=O)n1 c1(C(=O)NC(C=CC(=O)OC)C)c(Cl)ccc([N+](=O)[O-])c1Cl C12(C(N3C(C)CC(NC(C4COC(=O)O4)=O)C3)=O)CC3CCC(CC(C3)C1)C2 C1(NC(c2ccn(C(CC)CC)n2)=O)C2CN(C(c3ccccc3CO)=O)CC12 n1(C(C)C)ccc(C(=O)NC2CCOC2C(=O)N(C2(C3CC3)CC2)C)n1 c1(C(=O)NCCN(C(c2cc(C)c(O)nn2)=O)C)nc(Cl)cc(N)c1Cl c1(C(=O)NCC2N(C(C(C)(C)OCC(F)(F)F)=O)CCC2)cc(N)ccc1Cl c1(C(N2CCCC(C3CCCN3C(=O)CCF)C2)=O)ncnc(O)c1Br N1(C(Cn2cc(-c3cccc(C(=O)O)n3)nn2)=O)CCCNS1(=O)=O CC1(C)CN(C(c2cc[nH]c(=N)c2N)=O)CC1NC(C1CC(F)(CO)C1)=O c1(CC)ccc(C(N2CC3C(N(C(=O)Cc4cc(C)nn4C)C)C3C2)=O)c(F)c1 c1(C(N2CCC(N(C(C(=C)C(F)(F)F)=O)C)C2)=O)cc(Cl)cc(Br)c1 C(CC(C)(C)CC(=O)N(C1(CC)CCC1)F)OC.c1(C(C(=O)N)C)ccn(C)c1 c1(CC(=O)NCC(C2CCCCC2)NC(C2C(C)CCC2)=O)c[nH]c(=N)nc1O n1(CC)ccnc1CCC(=O)N1CCC1C(=O)NC1CCN(CC2CC2)C1 c1(C(=O)NCCCN(C(c2c(C)[nH]c(C)c2C)=O)CC)noc2c1COCC2 C(=O)(CC(C)C(C)(C)NC(=O)CC(O)C(C)C)N1CCOCC(=C)C1 C1(O)(CNC(=O)Cc2cc[nH]n2)CCN(C(=O)COC2CCCC2)C1 c1(C(C)NC(c2cc(OC)nn2C)=O)cc(Cl)cc2c1OCC2 Cc1c(C=CC(=O)NCC(C)N(C)C(c2c[nH]cc(F)c2=O)=O)cnn1C N1(CC)CCC(NC(=O)C(C)C(C)NC(c2cnc(OC)s2)=O)CC1 c1(N2CCC(C)CC2)ccc(S(=O)(=O)N(C)C)cn1.c1(C(=O)N)nn(C)c(Cl)c1Cl C(=O)(C1CCCn2ncnc21)NCC1OCCN(C(Cc2cnc(C)s2)=O)C1 CC1(C)CC(CC(=O)NCC2(C)CCC2)CN1C(c1cnc(N)cn1)=O c1(OC)ccc(NC(C2CCN2S(=O)(=O)CCN2CCCCC2)=O)cc1Cl C#CCCC(C(=O)Nc1ccc(CC)cc1)NC(=O)Cn1c(C)ccc1C Cc1ncsc1C(=O)NCCOC1CN(C(c2snnc2C(C)C)=O)C1 C(=O)(C(O)Cc1cnn(C)c1)NC1CC(CCNC(COCCC)=O)C1 N1(C(C2CC(=C)C2)=O)CCN2CCN(C(=O)CCCOCCC)CC2C1 c1(C(=O)NC2CCCCN(C)C2=O)cc([N+](=O)[O-])c(F)cc1N C#Cc1ccccc1CC(=O)NC1CC2CCC1(C(=O)NCC(CCC)OC)C2 N1(C(c2ccccc2Br)=O)CCC2(CCC2)C(O)C1.CC(C)CCN(C(=O)C)CC N1(C(C2CC3C=CC2O3)=O)CCN(C(=O)C2=CCCS2)C(CC2CC2)C1 C1(C(NOC(COC)COC)=O)C=CCN1C(=O)COc1ccsc1 CC1C(NC(C2CCC(C)(C)O2)=O)CCN1C(c1ccccc1)=O.C(N)(=O)N C(N=c1cc(C(F)F)nc[nH]1)C1(F)CC(NC(=O)CC2CCCOCC2)C1 n1(CC(C)C)cc(C(=O)NCCC(C)NC(c2n[nH]c(C3CC3)n2)=O)cn1 c1(C(=O)NCC2(C)CCC2)cnc2c(F)cccc2c1.c1(C(=O)N)ccsn1 CC(CN=c1nc2[nH][nH]cc-2c(O)n1)N(C)C(c1ccc2nc(O)cn2c1)=O N1(C(C(C)N)=O)CC2CCC(C1)N2C(=O)CC(CN(C)C)C(F)F.CC(F)(F)F C(=O)(C1CCCc2n[nH]cc21)NC1CCC2CN(Cc3n(C)cc(Br)n3)CC2C1 N1(C(C(C)OCCN(C)C)=O)CCC2CN(C(=O)Cc3nnc(S)n3C)C2C1 c1(CC)ccc(C(N2CCC(C)(NC(C3CC(F)(CF)C3)=O)CC2)=O)c(C)n1 CC(C)(CCNC(C1OCC2CCCC12)=O)C(=O)NC(CC1CC1)C1CC1 c1(C(=O)NCCN(C(C(c2cccc(C)c2)O)=O)C)cc(C2CC2)ccc1F C1(C(N2C(CCCNC(CCN(C)CC)=O)CCC2)=O)CNC(=O)CC12CCC2 c1(C(N2CCC(NC(=O)NC)C2)C(=O)NC(CC)C)ccnc(F)c1C c1(SC)ccc(N)cc1C(=O)NCC(C)CO.C1(C=O)CN(S(N)(=O)=O)C1 C1CCCCN1C(C1CCC(=O)N1C1CC1)=O.c1(CC(=O)OC)cn(C)nn1 C1(NC(C2(COC)COC2)=O)CCCN(C(c2scnc2C)=O)CC1 C(=O)(C1=C(Cl)CCOC1)N1CCC(C(C(=O)NC(CC(=O)OC)C)(C)C)C1 n1(CCCC)cc(C(N2CCC(CC(F)(F)F)C2)=O)c(C)n1 C1(CNC(=O)C(c2cccc(Cl)c2)O)C2CC1N(C(c1c[nH]c(Br)c1)=O)C2 C1(c2cn(CC3CCCN3C(c3ccc(C4CC4)o3)=O)nn2)(N(C)C)CCOC1 C(=O)(CC1CCCc2oc(C)nc21)NC1CN(C(C=NOC)=O)CC1SC C1(C=O)C2C3CC4C5CC(C1C35)C24.c1(C=O)ncsc1C(C)(C)C.CC.O CCCCC(C)CCC(=O)N1CC2CC(C1)N(C(=O)C(O)C1=CCCCC1)C2 c1(CNC(C(c2ccccc2Cl)C)=O)cccc(NC(C2CCC3(CC3)C2)=O)c1 C1(N(C(=O)Cc2csnn2)C)CCCN(C(c2cccnc2-n2ccnn2)=O)C1 c1(NC(C(Cc2cc[nH]n2)NC(=O)CC2(O)CCOC2)=O)ccc2n[nH]cc2c1 C(CC(C)(C)C)(C(=O)N1CC2(CCC2)CC1C)NC(C(C)SC)=O c1(C(N2CC(F)(CNC(CC(CC)SC)=O)C2)=O)cc2c(Cl)c(Cl)ccc2[nH]1 c1(C(=O)NC2CN(C(C(CC#C)(C)C)=O)CC(C)C2)cc2c(Cl)ccnc2s1 N#Cc1ccc(C(N2CCC2c2cn(C3CC(O)C3)nn2)=O)s1 Cc1cccc(O)c1.c1(N(C(C23CC(C=O)(C2)C3)=O)C)cc(C)c(I)cn1 C1(O)(CC=O)CCCCC1.C(CNC(C1CCC1)=O)(C(C)C)OCC.C c1(NCC(=C)CC)cc(=NCc2c(Cl)cnn2C)[nH]c(C(C)C)n1 c1(C(C(=O)NCCC2CCCN(C(c3c(C)n[nH]c3)=O)C2)C)c(C)nn(C)c1C Cc1ccc(C(=O)NCC2CC3CCC2N3C(c2nnc(C)s2)=O)c(Cl)c1 c1(C(=O)N)noc2cc(Cl)ccc12.CC(C)CCCNC(=O)C(C)NC(N)=O Cc1ncc(C(=O)NC2CCCN(C(=O)CCn3c(C)ccc3C)CC2)c(O)n1 Cc1cnc(C(N2CCC(O)(CN=[N+]=[N-])CC2)C(=O)NCCCC2CC2)cc1Br Cc1nnc2n1CC(C(=O)N(C)CC1C3CN(C(=O)CSC4CC4)CC13)C2 Cc1cc(C(=O)NC(C2(C)CC2)C)sc1Cl.c1(C(CC=O)C)cccc(F)c1.N C1(N(c2nc(C)sc2)C(=O)CC2CCCC2)CC2CCC(C1)N2 CCCC(CNC(=O)C(C#N)CCC)C(=O)NCC12CCC(C1)C(=O)N2 c1(C(=O)OC)cccc(C2CCCN(C(=O)C(c3cccc(C)c3)C3CC3)C2)c1 C(=O)(C(C)(C)C(=O)N(C)C)N(C(C)C)C.c1(C=O)ccc(-c2ncon2)cc1.N C12(CNC(CCSC)=O)CCC(CCCN=c3[nH]nco3)(CC1)CO2 Cc1ccc2ncc(C(=O)NCC)n2c1.C1(C(N(CCC)C)=O)CC(C)(O)C1.O N1(C(=O)COCC2CCOCC2)CCCCC1C1CCCN1c1ccncn1 c1(C(C(=O)N2CC(CC(C)NC(c3c(C)onc3)=O)C2)(C)C)ccc(O)cc1 N1(C(Cc2ncc(C)s2)=O)CC(CNC(C2CC3CC3C2)=O)C2(CC2)C1 Cc1nn(C)c(=O)c(C(=O)NC2CCN(C(c3cc[n+]([O-])cc3)=O)CC2C)c1C C1(NC(N2CC(C)CN(C3CC3)CC2)=O)CCCCN1S(=O)(=O)N(C)C Cc1ccc2c(c1)C(C(=O)N1CCC(CO)(NC(c3nocc3Cl)=O)C1)OCC2 O=C(CC(CC1CC1)NC(c1ccc2[nH]ccc2c1)=O)NOCC(O)CO c1(OC)cccc(CSCCOc2ccccc2C(=O)O)c1C c1(C(=O)NCC(C)(C)NC(CC2C(CC)C2)=O)cc(C)c(C)nn1 c1(C(N2C(C)CC(NC(Cc3ccc(C)s3)=O)C2)=O)ccc2c(c1)CN(C)C2 Cc1cccc(C(=O)NC(C)C(C)NC(=O)C(C)(C)n2cc(Br)cn2)c1C#N C1(NC(c2cc(OC)ncc2Cl)=O)CC12CCN(C(c1cc[nH]n1)=O)CC2 c1(C(=O)N)cc2nnn(C)c2s1.CC1CN(C(C2CN(C)C(=O)N2)=O)CC1(C)C N1(C(C(C(C)(C)C)N2CCOC2=O)=O)CCC(S(C)(=O)=O)C1 C(=O)(CC(C(F)(F)F)NC(C1(F)CCCCC1)=O)N(CC)CC1CCC1 N1(C(Cc2cn(CC)nc2)=O)CCC(CCNC(C2CCCOC2C)=O)CC1 C1(CCNC(=O)CC)(OC)CN(C(=O)CC=C(C)C)C1.c1ccccc1.S C1(C(N(C2CCCCC2(C)C)C)=O)CN(C(c2cccnc2S)=O)CCC1(C)C CCCC(C(=O)N1CC(OC)CC1C)NC(C)=O.C1(C(=O)N)CC(Cl)(Cl)C1 C(=O)(CC(C)C(F)(F)F)N1C(C(=O)N)C=CC1.C1CC1.C1CC1.COC c1(C(=O)NC(CCC)CCCNC(C2(OC)CCSC2)=O)cc2ccccc2o1 C(=O)(C1Cc2c(Cl)cccc21)N1CCC2CN(C(c3cc(C)c(C)[nH]3)=O)CC1C2 c1(CS(N2CC(NC(=O)CCc3cc(Br)ccn3)C2)(=O)=O)ccc(Cl)cc1F C1(NC(=NCC(=C)C)NCC2CCN2C2CC2)CCC2(CC1)NC(=O)NC2=O c1(C(=O)NCC(CNC(C2N(CC)C(=O)CC2)=O)F)cccc(O)c1F c1(C(N2CCN(C(c3c(C)nc(CO)s3)=O)C(C)C2)=O)c[nH]c2cc(F)ccc12 N1(C(C(CC)SC)=O)CCCN(C(c2cn(C)nc2OC)=O)CC1C(C)C N1(C(C2(C)CCCC2)=O)CC2(CCCC2NC(=O)CCN2CCC(F)C2)C1 N1(C(CC(c2ccc(C)cc2)C)=O)CCCC2(C=CCO2)C1 c1(C(N2CC3C(CNC(Cc4ncc(C)s4)=O)(C3)C2)=O)ccc2ncnn2c1 CCN=c1[nH]c(C(=O)NC(C)CNC(=O)CCn2cccnc2=O)cs1 C1(CC)CN(C(c2cnn(C(C)C)c2)=O)CCC1NC(=O)Cc1ccccc1Cl O=C1CCc2cc(C(N3CC4(C3)CN(C(c3cc(O)ncn3)=O)C4)=O)ccc2N1 CCCCCCCCN(C)C(C1CCOC1CNC(=O)CCCc1ncco1)=O c1(C(=O)NCCNC(C(=O)NCC)=O)cc2c(cn1)OCO2 C=CCCCC(C(=O)OC)OC(=O)Cc1csc2ccccc12 CC1(C)CN(C(=O)CC2(CNC(C3CCCC(O)C3)=O)CC2)CC(C)(C)O1 C1(CC)CN(C(=O)CCN(C)CCO)CCC1NC(c1c[nH]c(=NC)o1)=O C1CC2(C1)CN(C(c1cc(C(C)(C)C)no1)=O)C2.CC1CC1CC(=O)NC C1(C(=O)NC(c2ccnn2C)C)CCCCCCN1C(c1cc(CO)n(C)n1)=O C1(O)CC(C)(C)C1.C(CCC(=O)NC1C=CC(C(=O)NC)C1)=CC(C)C n1(CC)ccc(C(=O)N(CCC(C(C)C)NC(C2CSC2)=O)C)c1C CC(C(C)(C)C(=O)N1CC(C(C)(C)C#N)C1)NC(=O)CC1CCCSC1 c1(C(N2C(CNC(C(C(C)O)(C)C)=O)CCC2)=O)cc(F)c(Br)cc1F C1(NC(C2ON=C(C)C2)=O)CN(C(c2c(C)noc2C(F)F)=O)CCC12CCC2 C(CCCC(=O)NC1CN(C(=O)Cn2cncn2)CC1c1cnn(C)c1)SC N1(C(C)=O)CCCCC1C(N1CCOC(c2ccoc2)C1)=O n1(C(C)C(N2CCC(O)CC2)=O)cnc2ccccc2c1=O C(=O)(C1CCCc2ncnn21)N.C1(C(=O)NCC2CC2)CC(=C2CCC2)C1 CCC(O)C(C)(C)C(=O)N1CC(OC)C(C(=O)N(C2CCCCC2O)C)C1 C1(C(=O)NCCC2(CNC(C3ON=C(C)C3)=O)CC2)CC2CCCC12 c1(C(N2CCC(C)(CCNC(C(CN(C)C)O)=O)C2)=O)cc(C(F)F)ccc1F N1(C(CCCNC(C)=O)=O)CCC(C2(NC(c3ccc(F)c(C)c3Cl)=O)CC2)C1 c1(C(=O)NCCC(C)N(C(CCc2c(C)cccc2)=O)C)c(F)cc(F)cc1F c1(C(=O)NC2C(NC(CSCCCC)=O)CCC2)c(O)cnc2ccc(F)cc12 Cc1cc(C)c(CC=O)c(C)c1.c1(C(N(CC)C2CC2)=O)cc2n(c1)CCOC2 N1(S(C2(C(C)C)CC2)(=O)=O)CCC(c2ccccc2)C1C C1(C#N)(OCC)CN(Cc2cnc(CC)o2)C1 C1(C)(C(=O)NCC)CN(C(=O)COCCSC)CCO1 c1(OC)ccc(C(N2CCCCC2CNC(c2sc(NC)nc2C)=O)=O)cc1O c1(C(=O)NCC(CC(=O)NCC2C3COCC23)OC)cn(C)ccc1=O c1(NC2(c3n(CC=C)nnn3)CC(CSC)C2)ccc2oc(CC)nc2c1 C(C(=O)N(CC)OCC)C1(C)N(C(C(COC)N(C)C)=O)CC1 c1(NC(C2CC(NC(C(CC)(C)O)=O)C2)=O)ccc2c(c1)OCCO2 N1(C(C2N(C(C)C)CCCC2)=O)CC(NC(C2CC2C)=O)CC2(CCC2)C1 Cc1cc(Cl)c(C(=O)NCC(C(C)(C)C)NC(c2c[nH]ccc2=O)=O)s1 N1(C(C(CC)F)=O)CCC2(CC1)OCCC2NC(c1sccc1Cl)=O C(CCCCCNC(C1CCNC(=O)C1)=O)N(C(C(C)C1CCC1)=O)C c1(C(=O)OC)c(C)nn(Cc2ccccc2)c1N.c12ccsc1NC2=O c1(C(N(CCC)C)=O)cc2n(n1)CCNS2(=O)=O.C=CC(O)(C=O)C(F)(F)F.N c1(NCC(N2CCN(C(C(C(C)(C)C)SC)=O)CC2)=O)cc(C)c2[nH]cnc2c1 CCCC(C(=O)NC1CCCC1CCO)NC(=O)C(O)CCSC C1(CC(=O)NCCC=CC)CN(C(=O)CC(=O)NC2CC2)CCO1 C#CC1(c2ccccc2)COCCN1C(=O)NC1CC(Nc2cccc(Cl)n2)C1 C1(NC(C2(CC#C)CCCC2)=O)C2CC3C1C3C2C(N1CC2C=CC2C1)=O C(=O)(C#CC1CC(F)(F)C1)N1C(CN(C)C(c2cc(Cl)c[nH]2)=O)CCC1 c1(C(N2C(CNC(CCC(=C)Cl)=O)CC2)=O)cc2c(nc1O)CCCC2 C(=O)(C1CCc2nccn21)N.c1(C(=O)NC2(C)CCOC2)cnc(C2CC2)nc1 N1(C(C(CCC)c2cccc(Cl)c2)=O)CC2CCC1CN2C(=O)C(CC)OCC n1(CC)nc(C(N2CCOC(C(C)NC(c3cccc(=O)o3)=O)C2)=O)ccc1=O c1(CN2CCC3(CCN(C(c4ncc(C)s4)=O)C3)C2)cc(Br)cc([N+](=O)[O-])c1O C(C(=O)N1CC(N2CC(C=O)CC2=O)C1)(C(C)(C)C)n1cc(COC)nn1.O CCC(C)(C#N)C(=O)N(C)CCN(C(=O)Cc1csc(Cc2ccccc2)n1)C CC1CCCCC1OCC(=O)NC1CCC1.c1(C=O)ccccc1C(C)(F)F.N N1(C(c2c(NC)cncc2)=O)CC2(CC2)CC1CNC(C1CC(C)CO1)=O c1(OC)cc(C(=O)NCCCCCNC(=O)C2=NOC(C)C2C)cc(F)c1F CC1=CC(C)CN(C(=O)C(C2CCN(C(=O)C(O)C(C)(C)C)CC2)C)C1 C1(NC(C(CC)F)=O)CN(C(=O)Cn2cc(C(=O)OC)cn2)CC1N=[N+]=[N-] N1(Cc2ccn(C)n2)Cc2[nH]nc(-c3ccc(OC(F)(F)F)cc3)c2C1 C(=O)(C(CCF)NC(=O)CC(C)(F)F)N1CC(COC(C)=O)C1 C(CC=CC)(C(=O)NCC(CO)C1CCC1)NC(C)=O.C#CCOCC=C Cc1cn2ccnc(C(=O)NC(CNC(=O)C(c3ccnn3C)O)C3CC3)c2n1 C1(NC(CCCCOCCC=C)=O)CC2(C1)CN(C(=O)C(CC)n1cncn1)C2 C1CC(C(=O)N(CC(C)O)CCO)C1.C1(C(=O)OCC)(C(=O)N)CC1 Cc1ccc(C(C)(F)F)cc1C(=O)NC.C1(C=O)CCCC1C.C1(CC)CC1 C(CCC(C)(C)NC(=O)CCCn1ccnn1)NC(CSCCC(C)C)=O C1(NC(CCCSC)=O)CCCC(NC(c2c[nH]nc2Br)=O)C1 Cc1cc(N(C)CCC2CCCCC2)nc(=NCCC(C)O)[nH]1 C12CCC1CN(C(=O)C(C(C)(C)C)C1CCC1)C2.C1(C(=O)N)(OC)CCC1.C Cc1ccc(-c2cncc(C(=O)NCCC(C)NC(C3CCNC3=O)=O)c2)cc1 Cc1ccc(-n2c(C3(CCCc4cccc(C)n4)CC3)nnc2C2CC2(C)C)cc1 C(CC)(C(=O)N1CCCCO1)NC(c1ccc(CC)nc1)=O c1(C(=O)NCC2N(C(C3ON=C(CC)C3)=O)CC(F)C2)cc(C)c(C#N)cn1 c1(N(C(C)=O)C)cccc(CNC2(C3CC3)COC(C3CC3)C2)c1 C1(C=O)CCC(=O)C(C)C1(C)C.N1(C(c2cnc(CC)[nH]2)=O)CCCCC1C.N N1(C(c2cnc(C)nc2C(C)C)=O)CC2CCC1C(NC(c1ccns1)=O)C2 C1(C(=O)N)CCC(N=[N+]=[N-])C1.C(CC(=O)N(CC)CC)OCCOCC C1(C)(CNC(c2n(CC(=O)OCC)nc(CN)c2)=O)CC2CCC1C2 Cc1cc(CCNC(=O)CCC(C)NC(=O)CN2CCC(F)CC2)nn1C C(C1OCCc2ccccc21)N(C(=O)NC(C)(C)C)C.C1(CC)CN(C=O)C1.O C1(NC(CC(C)c2ccncc2)=O)COC2(C1)CC1(CNC1)C2 c1(CC)cc(C(N2CCOC(Cn3cc(CCOCCO)nn3)C2)=O)cc(N)c1 C1(C=O)CC2(CO1)CC(F)(F)C2.C1(C=O)CCC(C(N)=O)CC1.CC(C)C.N c1(CC(Cc2ccccc2)NC(C(=Cc2c[nH]cn2)C)=O)ccc(Cl)cc1 C1(NC(C(C)(C)CF)=O)CCN(C(=O)Cc2cccnc2Cl)C(C2CC2)C1 c1(N2CC(C3N(CC)CCC3)(O)C2)ncnc2c1ncn2CC(O)SNC CC(C(=O)NCC1CCC2CN(C(=O)C(O)C(F)(F)F)CC12)C(F)(F)C(F)F C(C1=NOC2(CCC2)C1)NC(C(CCC)CNC(c1ccc(C(N)=O)[nH]1)=O)=O N1(C(c2ncnc3c2CCC3)=O)CC2CCN(C(c3csc(O)n3)=O)C(C2)C1 CC1CN(C(=O)N(C)C(c2ccc(I)cc2Br)=O)c2cc(C(F)(F)F)ccc2O1 CCC(CC#N)N=c1nc(N2CCNC(=O)C(F)(F)C2)c2cnn(C)c2[nH]1 c1(C(c2n(CC=C)nnn2)NCCC2CC(C)(C)CO2)cccc2nsnc12 C1(NC(c2c(SC)cccn2)=O)CCCN(C(c2coc(C)n2)=O)CC1F c1(C(=O)NC(C(C)(C)OC)C)n[nH]c2c1CN(C(c1occc1C1CC1)=O)C2 C=C(C)C1CCC(C)C(c2nnnn2CC)(NCCn2cc(Cl)c(CC)n2)C1 Cc1cc(=NCC2CC3CCC2N(C(=O)CC2CCC(F)(F)C2)C3)[nH]cc1C#N C(=O)(C(F)C(C)(C)O)NCC1C(C)CN(C(=O)CSC2CC2)C1 c1(CS(Cc2cc(C(=O)OC)no2)(=O)=O)cc(Br)ccc1[N+](=O)[O-] c1(N(CCC2N(C)CCC2)C)ccc(S(=O)(=O)N2CCCC2C(C)(C)C)c(Cl)c1 c1(-n2cc(CSC)nn2)cccc(C(=O)NCC2(C)CC=CCC2)c1 N1(S(CCOCC)(=O)=O)CCC(O)C(C(=O)Nc2cnc(C)cn2)C1 C(=O)(C1c2c[nH]nc2CN1C(=O)CCCC1CC1C)Nc1ccc(C#C)cc1 c1(CC)ccc(C(C)C(=O)NCCC(C)N(C)C(C2CC(CC)C2(C)C)=O)cc1 c1(C(=O)NCc2cc(C(=O)NC(C3CCCOC3)C)no2)ccc2n[nH]cc2c1 N1(C(C=O)C)CCSCC1.c1(C(N2CC(CC)C2)=O)cnc(CCN(C)C)s1.N C1(NC(CCSC)=O)(CNC(=O)CC2CCCCC2)CCOCC1.N(C)C.C CC1(C(=O)NC2CC(CNC(C3CC3c3cnc[nH]3)=O)C2)CCCNC1=O Cc1cn(C)nc1C(N1CCOCC1C(=O)N(C)CCn1cncn1)=O c1(OC)ccc(F)cc1CC(=O)N.c1(C(N2CCC2)=O)ccc(C(F)F)nc1.C C1(C(=O)NCCC2OCCN(C(C(C)(C)SC)=O)C2)CC(=O)C12CCCC2 S=C(NCCCNc1cccnc1)N1CCOC(C2CC(F)(F)C2)C1 C1(NC(=O)CCCF)CC2CC(NC(=O)Cc3cccnc3O)C2C1 CC1(CCNC(c2cc(Br)co2)=O)CC1(F)Cl C#CC1(C(=O)NCc2cc(C(N3CCC(OC)CC3)=O)ccn2)CC(=O)C1 c1(C(=O)NC(CNC(c2ccc3ncsc3c2)=O)C2CC2)ccc2nccn2c1 C1(COC)CN(C(C2(C)CC=CCC2)=O)CCN1C(c1cc(CO)on1)=O C1(NC(C=CSC)=O)CN(C(C2CC3(C2)CC(F)C3)=O)C2(CCOCC2)C1 C12(C(=O)Nc3cc(OC)cc(O)c3)CCCC1CCN2C(=O)Cc1cscn1 N1(C(C(CC#C)C2CC2)=O)CCC(F)(F)C(C)C1.C12C3CCN(CC13)C2=O c1(CC(=O)NC(C)CCCNC(=O)C(C)CC(F)F)ccc2cccnc2c1 O=C1CC(C(N2CCOCC2Cc2cn(CCN3CCCC3)nn2)=O)NC(=O)N1 Cc1ccc(C=CCC(N2CC(NC(=O)C#CC(=O)N(C)C)CC2C)=O)cc1 N1(C(c2c(C)[nH]nc2C(F)F)=O)CC2CCC1CN2C(c1ccc(N)c(F)n1)=O C1(C(=O)NCC2N(C(c3ccc(C(C)=O)cn3)=O)CCOC2)CCCC(=O)N1C N1(C(c2c(CC)nc[nH]2)=O)CCCN(C(C2CN(C)CCO2)=O)C(C)C1 Cc1[nH]nc(C(N2CCOC(C(=O)NCC(c3ccnn3C)O)C2)=O)c1C C1(F)(C(=O)NC(C(C)NC(=O)COCCN(C)C)CO)CCCOC1 c1(-n2cc(C3CCN(C)C3)nn2)ccccc1C(=O)NC(CN(C)C)C(F)(F)F c1(C(=O)N)cc(O)cc(Cl)c1Cl.C1(OC)CCC(C(=O)NCCC2CCC2)C1 C=CCCCCC(=O)N(CCCOC1CCCOC1)C.C1(=O)COCCN1 C(CC1=CCCCCC1)Nc1nccc(=NCc2cnc(C)s2)[nH]1 c1(OCC(=O)NCC(CC=C)NC(c2cccnc2C)=O)ccc(CC)cc1 C1(NC(CS(=O)(=O)NC)=O)CCCCN(C(C2(OC)CCS(=O)(=O)C2)=O)C1 N1(C(COCCSC)=O)CCN(C(c2cc(F)ccc2OC(F)F)=O)C(C)C1C C1(C(=O)NCCCC(=O)NC)CC(NC(=O)COC2CCC2)C12CCC2 c1(C=O)c[nH]c2nccc(Cl)c12.C1(CNC(=O)COCC2CC2)CCCC1 C1(CNC(c2ccc[n+]([O-])c2)=O)CN(C(C2(C3CCCO3)CCCC2)=O)CC1O c1(C(c2nnnn2C)NC(CCC(=C)C)C)ccc(F)c(CC)c1F N1(C(=O)NC2C(C(=O)OC(C)(C)C)CCC2)CCC(c2ccccc2Cl)C1(C)C c1(CC(=O)NC2CCC23CN(C(C2SCCCS2)=O)C3)cc2ccccc2o1 C(C)(C)(C(=O)NCc1csc(C(=O)NCCCN(C)C)c1)OC(C)=O Cc1oc(S(N)(=O)=O)cc1C(=O)N.C1(CC=O)SC(=N)NC1=O.C1CCC1 Cc1nnc(O)c(C(N2CCC(C(C)NC(=O)Cc3cccnc3Cl)C2)=O)c1C C(=O)(C1=CC(C)(C)C1)NC(CCCNC(c1c(C)n(-c2ccccc2)nc1)=O)C N1(C(c2c(C)scn2)=O)CC(CN(C)C(C2(C)CC=CCC2)=O)C2(CC2)C1 O=C1NCC(C(=O)NC2CN(C(=O)CN3CC4CC4C3)C2)O1 N1(C(C(C)(C)C(F)F)=O)CC23CCCC2(C1)CN(C(=O)C#CC1CC1)C3 Cc1nc(N2CC(NC(C3(c4ccccc4)CCOC3)=O)CC2C)cc(C#N)n1 C1(NC(=O)C2=CCC2)CN(C(c2cc3ncccc3s2)=O)C2CCCCC12 C(CCC(CCC)NC(=O)C(C)c1ccsc1)NC(c1n(CCC)nc(C)c1)=O c1(OC)ccc(C=CC(N2CCC(O)(C)C2)=O)c(C)c1.C(=O)C1=CCCS1.N C1(CNC(c2cnnc(C)c2C)=O)CN(C(C2CC(C)CCO2)=O)C2(CCC2)C1 Cc1c(C(=O)NC2CC(F)(C)C2)ccn1C.n1(CC=O)cc(C2CCC2)nn1 Cc1ccc(O)c(C(=O)NCC2CN(C(=O)CC3CCCCO3)C2)n1 C(=O)(C1=CC(O)CC1)N1C(C)(COC)C=CC1.C(=O)(CC(C)(C)C(F)F)N C1(C(C)C)(C(=O)N(C2CC(C(N)=O)C2)C)CCN(C(c2c[nH]nc2Cl)=O)C1 c1(OC)cc(C(=O)Nc2ccc(C#N)c(O)c2)cnc1C1=CCC(C#N)CC1 C1(CNC(c2c(CC)n[nH]c2)=O)CC2(CC2)CN1C(c1cccnc1O)=O C(=O)(CCCC(C)NC(=O)CN1CC(=O)NC1=O)NCC1(CC)CCCO1 C1(C(=O)Nc2c(C(=O)OCC)scc2)CCN(Cc2c(I)ccnc2F)CC1O C1(CCC)(NC(=O)COCCCF)CCCN(C(C2CC3(C2)CC3(F)F)=O)C1 c1(C(=O)OC(C)CC2CCOC2)ccnc(S)c1 c1(-n2cc(NC(N(C)CCN3CC4CC4C3)=O)nn2)cccc(Br)c1 C12(C(N3CC(C)C3)=O)CC3CC(CC(C3)O1)C2.C1(C(C=O)OC)CCCOC1.N c1(C(=O)NC(C)CCCNC(c2ncn(C)n2)=O)cc(Br)ccc1C1CC1 N1(C(C(C2CCC2)OC)=O)CCC(NC(c2oc(CC(C)C)nc2C)=O)C1(C)C Cc1oc(C(F)(F)F)nc1C(=O)NCC1CN(C(C2(C)COC2)=O)CC1O C(N=c1[nH]c(=NCc2ccc[nH]2)[nH]c2c1COC2)c1c(C)nc(C)[nH]1 Cc1cc(C(N2CC(NC(=O)Cc3c[nH]nc3O)C(C)C2)=O)c(C)nc1C N1(C(c2ccnc(Cl)c2Cl)=O)Cc2nccn2CC(NC(C2(F)CCOC2)=O)C1 c1(OC)ccc(CCNC(=O)C(c2ccccc2)O)cc1.C(=O)CP(C)(C)=O.N N1(C(Cc2c(C)nc(S)s2)=O)CCCC(NC(=O)C(c2cscn2)N(C)C)C1C C1(CC(=O)N(CCC)C)NC(=O)CNC1=O.c1(COC)ccc(C=O)o1.N CC1(C)CCCC(CNC(=O)CC2CN(C(C3(F)CCC3)=O)CCO2)O1 n1(CC)cc([N+](=O)[O-])c(C(=O)NC)n1.C1CN(C(=O)Cc2cc[nH]n2)CC1O C(CC(CC)C(=O)N1CCCC(N(C(c2cc(C)ccc2N)=O)CC)C1)=CC C1(C(=O)NC(C)CCN(C(=O)CC2CSCCS2)C)CC2(C1)CC1(CC1)C2 CCC(O)(CN=c1cc(NCCC(C)OC)nc(C)[nH]1)c1ccc(Cl)cc1 Cc1oc(C(=O)N)cc1S(N)(=O)=O.C12CC(CN1C(c1ccncc1O)=O)C2.C C(C(C)(C)C)N(C(=O)CC)CC.c1(C(C=O)C)ccc(C)s1.C1CCCC1.N c1(C(=O)NCCCN(C(c2n[nH]c3c2CCC3)=O)CC)c(F)ccc2ccoc12 CCC(CC(=O)NC1(CO)CCCN(C(=O)CCSC(F)(F)F)C1)CC(F)(F)F Cc1ccc(C(F)(F)C(=O)NC2CC(F)(CNC(c3scnc3C)=O)C2)cc1 C1(CC(=O)NC(C2CCCCC2)C(=O)NCC2CC2(F)F)CCOC1=O c1(C(=O)NC2(CF)CCN(C(C(CC)OC)=O)C2)cc2ccsc2c(O)n1 N1(C(CCN(C(CCC)C)C)=O)CC(O)(CNC(=O)C(F)CC2CCOCC2)C1 N1(C(C(C)SCCCC)=O)CCC(C)(NC(=O)C)CC1.c1c(C)occc1=O.O c1(COC(C(C(C)O)N(C)C)=O)cc(Cl)cc([N+](=O)[O-])c1 N1(C(C(C)NS(CCCC)(=O)=O)=O)CCCC12CCC2.C(=O)(CN(C)CCO)N N1(C(C2CC=CCO2)=O)CC2(C1)CN(C(C1(c3ccno3)CCC1)=O)CC2CO Cc1cc2ccc(NC(C3CC(O)CN3Cc3ccc(F)c(C#N)c3)=O)cc2[nH]1 C1(C(N2CC(C)N(C(=O)CC(C)(C)C3CC3)CCC2)=O)CCc2nccn2CC1 Cc1nc(C(=O)NCC2(F)CC(NC(c3coc(Cl)c3)=O)C2)sc1C CC1(C(=O)NC2CC(CNC(=O)CCCC3CC3)C2)CCc2ccccc2C1 Cc1cc(-n2cc(C3(F)CCN(C(c4cc(Cl)ns4)=O)CC3)nn2)cnc1Cl C(C(=O)N(C)C)(C(C)C)NC1CC(C(C)C)N(C(=O)OC(C)(C)C)C1 N1(C(C(CC)(C)C#N)=O)CCC(O)(C2(NC(c3ccc(C(F)F)o3)=O)CC2)CC1 Cc1cc(NC(c2cc(CNC(C3CCCC(C#N)C3)=O)[nH]n2)=O)ccc1Cl C1(CN(C(Cn2c(C(C)C)ncc2)=O)C)CCCN(C(=O)CC2CSC2)C1 N1(C(c2scc(Cl)c2Cl)C(=O)Nc2ccc(OC)cc2)CC2(CCC2)OCC1C C=CCCC(C(=O)N1CCN(C(C)CC)CC1)NC(c1cnc(C)cn1)=O c1ccnc(O)c1.C1(N(CC)CC)(C(=O)N)CCC1.C1CC1C(=O)NC c1(OC)ncccn1.c1(C2(C=O)CC2)ccc(Br)cc1.C12(C=O)CC(C1)C2.N C1(c2ccccc2)(CNC(=O)C(F)F)CC(NC(C2CCSC2)=O)C1 CC(C(=O)N1CSCC1C(=O)NC(CCO)C(F)(F)F)S(N)(=O)=O CC(C)C(CNC(C1CCCC2(CC2)C1)=O)C(=O)NCC1(O)CN(C)C1 Cc1cccc2[nH]c(NCCC(N3CCC(C(N4CCOCC4)C)CC3)=O)cc12 CN1CC(C(=O)NC(CC2CC2)CC(=O)NCC(CO)C2CCC2)NC1=O N1(C(C=CCN(CC#C)C)=O)CCCC1CNC(C1CC(CC)=NO1)=O C(=O)(C(C)(C)CC(C)(C)C)Nc1ccc(C2OCCN(C(=O)OC(C)C)C2)cc1 C1(C(N(C)CCNC(=O)CCCS(C)(=O)=O)=O)CCC2(CC1)CC2(F)F C(=O)(CCN(OC)C(=O)c1ccn2cncc2c1)N(C(C)COC)CC=C C1(CNC(CCc2scc(C)n2)=O)CC2CCC1N(C(=O)C(F)CC(C)C)C2 C1(C(N(C2CCCCC2)C)=O)CC12CCS(=O)(=O)CC2.C(=O)C(C)(C)C(N)=O CC1(C)CC(CNC(c2ccnc(O)c2)=O)N(C(C2OCCOC2(C)C)=O)C1 C1(O)(CNC(CC(=O)NCC)=O)CCN(C(=O)CC23CCCC2C3)C1 CC(C)CC(O)CC(=O)N1CCC2C(C1)CN2C(c1ccn(C)c1)=O N1(C(COCC)=O)CCN(C(=O)C(C)Oc2ccc(Cl)cc2Cl)C(C2CC2)C1 CC(C(CO)NC(c1cn(C2CC2)cn1)=O)NC(c1n[nH]cc1Br)=O C(C)(CCC(=O)NC12CC(C(=O)Nc3cnc(F)nc3)(C1)C2)OC c1(C(=O)N)csc(-c2ccccc2)n1.C(C)(C(=O)N(C(C)CC)C)NC(CC)=O Cc1ccc(C(=O)NC2COCCN(C(C3CCCN3C)=O)C2)c(OC(F)F)c1 N1(C(CCc2c(C)nn(C)c2)=O)C2CCC1C(NC(C1C=CC=CC=C1)=O)C2 C1(CC(=O)NC(C#C)C(C)(C)C)C2CCC(C2)N1C(c1ccc(C#N)n1C)=O C1CC(C)(C)CCO1.C(C(C)(C)C(=O)N)N(C(CNC(C1C(C)C1)=O)=O)C c1(C(C(=O)NCCOCC)N(CC(C)(C)C)CC)cc(Br)c(F)cn1 Cn1nnc2cncc(C(=O)Nc3ncc(Br)cc3N3CCCC3)c12 c1(C(N2CCC(N(C(c3nc(C(=O)OC)sc3)=O)C)C2)=O)cnc(O)n1C c1(C(N2CC(C)C(NC(=O)CCN3CCOCC3)C2)=O)cc2cccnc2[nH]1 N1(CCNC(CCC)=O)CCN(C(C2(C#N)CC2(C)C)=O)CC1 C1(CC)(NC(=O)CCn2ccnn2)CCCN(C(C2CC2C(F)F)=O)C1 C=C(C)C(CC(=O)N1CCC(NC(c2cnc(C)[nH]2)=O)C(C)C1)OCC N1(C(C2CC(CC)C2)=O)CC(CNC(c2ccn(C(C)C)n2)=O)C(F)C1 c1(OC)ccc(CN2CCSC(C(=O)Nc3cc(Br)cnc3C#N)C2)c(F)c1F C(=O)(CCC(C)(C)F)N(C(C)CNC(=O)CC1CCCCC1)C.n1(C)cnnn1 Cc1cc(CNC(C2(NC(C3CCCC(O)C3)=O)CSC2)=O)cc(C)n1 c1(NC(C2(C(=O)NC3CC(OC)C(O)C3)CCNC2=O)=O)cccc(C#N)c1 Cc1cnc(C(=O)NCC2C3CN(C(=O)C(N4CCSCC4)C)CC23)c(F)c1 C(=O)(C(C)(CC)CCC(C)C)NC1COCCN(C(CN(CCC#C)C)=O)C1 C1(CC(=O)NCC2CC(C(=O)NCC(N3CCOCC3)=O)C2)COCCO1 CCCCCC(O)CC(=O)NCC(C(=O)N1CCC(C(=O)OC)C1)C(C)(C)C N1(C(c2c(CC)[nH]cc2)=O)CC(C(N2CC(F)C(F)C2)=O)C2(CCC2)C1 C1(CNC(=NC)NCC2(CO)CC23CCOCC3)CCC(=C(F)F)CC1 N1(C(C(CC)Nc2nc3ccccc3s2)=O)CCc2cccc(OC)c2CC1 N1(C(C2C3CN(C(=O)Cc4ccc(F)cc4)C2C3)=O)CCN2CCCC2C1 CC1CN(C(C2(CO)CCC2)=O)CC1CNC(c1cccc(OC(F)F)c1)=O c1(CC(=O)NCCNC(C2C(CC(C)(C)C)C2)=O)cnc2ncccn12 c1(CC(C)C(N(OC(F)(F)F)C(C)C)=O)c[nH]c2ccc(F)cc12 C(=O)(CCCCCCNC(=O)CC(O)C1CCCC1)NC(C)COCC1CC1 Cc1nnc(N2CC(NC(c3cccc(=S)n3O)=O)C(C)(C)C2)c(C#N)c1C C12(CSC)CC(C(=O)NC3CN(C(c4ccncc4N)=O)C3)(CO1)C2 c1(OC)cc(Cl)ncc1NC(C1C=CCC1)=O.c1(C(=O)N)cnc(OCF)cn1 c1(C(=O)NC2(CC=C)CCN(C(=O)CC3CCCC3O)C2)cc2scnc2[nH]1 c1(C(=O)NCCN(C(C2CCSCC2)=O)CC)n[nH]c2ccc(Cl)cc12 C1(NC(C(C)SCCCC)=O)CCC12CCCN(C(=O)CC(C)CN(C)C)C2 C1(C)(C(=O)NCC(=O)NCCc2n(C)ncn2)CCCCC1 C(CC(O)C(F)(F)F)NC(C1C=CC(NC(=O)C(O)CC2CCCC2)C1)=O CC(C)CC(C(=O)NC(C)CCNC(=O)CC1CC1)N(C)C.c1ccccc1 c1(-c2nc(CC(C)Oc3c(C)cccc3)on2)ccc2ccccc2c1 n1(CC(=O)N(CC(CC)NC(C2CCC3CC3CC2)=O)C)ccc2ccccc12 Nc1ncc(I)cc1C(=O)NCCc1nc(CSc2ccccc2)no1 C1(NC(C2CCCC(C)(C)C2)=O)CCSC12CN(C(c1ncoc1C1CC1)=O)C2 C1(CC)CCN(C(c2cc(C)ncn2)=O)C(C(=O)NC(CO)C(C)C)C1 C1(OC)C(NC(=O)C(C)(C)NC(=O)Cn2cccn2)CC12CCC2 c1(CC)ncc(C(=O)NCCC2CCC2)[nH]1.C1(CC=O)CC(F)(F)C1.N CC(F)(F)CC(=O)NCC=CCNC(C1CC2CCC12)=O C1(CC(=O)NCC(CC)C)CCC(C)(C)CO1.c1(CCC=O)n[nH]c(=N)s1.N C1(O)(C(N)=O)CCCN(C(=O)COC2CCN(C(=O)Cc3cccnc3F)C2)C1 C1(C(N2C(CNC(CC(C)(C)O)=O)CC2)=O)CC2(CCC2)CO1 c1(-c2c(C(N(CCCCN(C(C(C)CF)=O)C)C)=O)c[nH]n2)c(F)cccc1F n1(CC(N2C(CNC(C(C)C#N)=O)CC2)=O)nc2n(c(=O)c1=O)CCC2 C(C(O)C(=O)NC1(C(=O)N(C2(C3CC3)CC2)C)CCCC1)N(C)C N1(C(c2ccnc(C)n2)=O)CCC(C)C2CNC(=O)C12 N1(C(C2(C)C=CCCC2)=O)CCC2(CCCN2C(=O)CN2CCCC2CO)C1 O=C(C1=CC2C=CC1C2)NCC1CC(CNC(C23CSCC2C3)=O)C1 N1(C(COCCC)=O)CCCC2(C1)CN(C(C1CC(SC)C1)=O)CCO2 c1(C(=O)NCC(C)NC(=O)CCOC2CC2)c(O)ccc2ccccc12 c1(CC(=O)N(C2CCN(C(CC)=O)C2)CCO)sc(C)nc1C.C(=O)NC.N c1(C(N2CCCC(CC(N3CCC(CCO)CC3)=O)C2)=O)c(I)ccnc1Cl N1(C(C2(CC)C=CCC2)=O)CCC(CO)(CNC(=O)CO)CC1.C(C)C [N-]=[N+]=NC1CC(C(N2CCCC2C(N2CC(Cc3ccco3)C2)=O)=O)C1 c1(CC(=O)NC2(C=O)CC2(C)C)ccc(O)nc1.C12(CC)CC(CO1)C2 N1(C(C2(OC)CCSC2)=O)Cc2ccccc2C(NC(=O)C(C)(C)CC(C)C)C1 Cn1cnc2c(C(=O)NC3CCCCN(C(C4CC(C)(C)C4)=O)CC3)cccc12 c1(C(=O)NC2CN(c3ccnc(C(=O)OC)n3)C(C)C2)ccc(S(N)(=O)=O)o1 N1(C(C2(OC)CC(C)C2)=O)Cc2[nH]nc(C(N3CC4(C3)CC(C)(F)C4)=O)c2C1 N1(C(CCSCC)=O)CCC2(CC1)CCN(C(=O)CC(C)c1ccncc1)CC2 N1(C(C(c2ccc(CC(C)(C)O)cc2)C)=O)CCC(O)C2(CC2)C1 CCCC(C(=O)N1CC(F)CC1CNC(=O)CC(=O)NC1CC1)OCC c1(CN2CCC(C(C)C(=O)NC3(CO)CCOCC3)CC2)cc(F)c(Cl)c(Cl)c1 c1(CCC=O)c(C)noc1C.C1C(C(N2CC(=C(F)C)C2)=O)C1C.CCO O(NC(=O)C=CCN(C)C(C1CCC(O)C1)=O)CCCOC N1(C(CC=C)=O)CCCN(C(C2SCCS2)=O)CC1C C1(C(=O)NC2CN(C(c3[nH]cc(C(N)=O)c3)=O)CC2F)Cc2cccnc2C1 Cc1cc(C#N)nc(N2CCCC(CNC(c3ccnnc3Cl)=O)C2)n1 N1(C(C(COC)NC(C)=O)=O)CCC(C)N(C(=O)CC2CCCCCC2)CC1 C=CC1(C(=O)NCCS(N)(=O)=O)CCN(C(=O)CN(C2CCC2)C)C1 c1(C=O)ccc(F)c(C2(C)CC2)c1.C1(CCCC)(C(N2CCC2C)=O)CCC1 C(=O)(C1=CC2(CCN(C(c3cnco3)=O)C2)C1)NC(C1(O)CCC1)(C)C C1(C(C)C)CN(C(=O)C=Cc2ccc(C(F)F)o2)CCCN1C(C1CC12CC2)=O c1(-c2cn(CC(N3CC(SC)C(C(F)(F)F)C3)=O)nn2)cc(Cl)ccc1F C=CCCCCCC(=O)NC(CC(=C)Cl)C(=O)N1CCCC1 C#CCC(C)(C(=O)NCCNS(N)(=O)=O)NC(=O)C=C(C)C C1(CC)(NC(c2ccc(Cl)s2)=O)CCN(C(=O)CCC2CC(OC)C2)C1 Cc1ccc(Cl)c(CN2CC(C(=O)Nc3cnccc3Br)CC(F)C2)c1F n1(CCC(=O)NC2CC(NC(C(CC)(C)OC)=O)C2)cnc2ccccc12 c1(C(=O)OC)c(C)cc(Br)c(NC(=O)N(C)CCN2CCOC2=O)c1C C1(C=O)CCN(C2CCS(=O)(=O)C2)CC1.c1(CCC(=O)OC)ccc(F)cc1.N N1(C=O)CC2(CC2)C1.C1CC(O)(C(F)(F)F)C1.CC(C)(C)OC(=O)N c1(C(=O)N)ccncc1.N#CC1CC1C(=O)NCCOCCOCCC N1(C(C2CC(C#N)(OC)C2)=O)C2CCC1CC(N(C)C(c1oc(C)nc1C)=O)C2 CCCCC(CNC(=O)COC(F)(F)F)NC(C1(CO)CC1(F)F)=O Cc1ccc(C(=O)NCC2CC(C)CCN2C(=O)Cc2csc(Cl)n2)cc1C#N C1(NC(C(C)OCCC#C)=O)COCCN(C(c2nn(C)c(N)c2C)=O)C1 c1(NC2C(SCC)CCC2)ccc(S(=O)(=O)NCc2cn(C)nc2C)cc1F Cc1csc(=O)n1CCC(=O)NCC1CC(F)CN1C(C1CC1C1CC1C)=O c1(OC)cc(C)nc(N(C2CCCN(C(=O)C=C3CCCC3)C2)C)n1 C(=O)(C1CCCc2ncnn21)NC1(C)CC(NC(c2ccc(SC)o2)=O)C1 CC1(C(=O)NCC2(C(=O)Nc3cncnc3O)CC2)CCCC1O C(=O)(CC(O)C1CCCC1)NCCN(C(C)C)C(C1CC1c1ccco1)=O c1(OC)cnc(F)cc1C(=O)NC(C1CCCN1C(c1cscc1Cl)=O)C C(=O)(C(C(C)(C)C)NC(c1cc(O)n(C)n1)=O)NC(C)Cc1ncn(C)n1 CC1(F)CCC(C(=O)NC2CC23CC(NC(c2ccccn2)=O)C3)CC1 CCCCCCCCC(=O)NC1CC2CCC(C1C)N2C(=O)CN(C)C CCC(C)(C)C(O)C(=O)NC1CC(C(=O)NC2CN(C)CC2C)=CC1O C=C(C)CC(C(=O)N1CCC(c2cnco2)C1)NC(c1cc(CO)n(C)n1)=O C(C#Cc1cccc(Cl)c1)N1CC(CO)OCC12CC2 C1(NC(C(C(C)C)SCC)=O)CN(C(c2ccc(N)cn2)=O)CCC1C c1(CC)onc(C(=O)NC(CO)C(N2CC3(CSC3)C2)=O)c1C C(=O)(CCCS(=O)(=O)N1CCCC1)N1CC(N(C(Cc2n[nH]c(=NC)s2)=O)C)C1 C(N=c1ccc(C(C)=O)c[nH]1)C1C(NC(C(COCC)N=[N+]=[N-])=O)CCCC1 N1(C(Cc2ccc(C#C)cc2)=O)CCC(C2(NC(C3CC(C)N(C)C3)=O)CC2)C1 C1(NC(CCCC#C)=O)CC(C(=O)NCC2CC=CC2)=CC1O c1(-c2ncn(-c3cn(C)nc3)c2)nc(CCC(C)(C)C)nn1CCF N1(C(C2C(OC)CC2)=O)CC2(CCN(C(c3cc(C4CC4)n(CC)n3)=O)C2)C1 C(C(=O)NC)(C(C)C)NC(C1(C(=O)NC)CCC1)=O.C1(Cl)CC1(F)F CC1C(NC(c2nsnc2O)=O)CC2CCC1N2C(c1cnc2c(c1)CCC2)=O C(C(C(C)C)NC(=O)CCC1CCCO1)NC(COCCOC)=O C(=O)(C(C)(C)COCc1ccncc1)NCC(C)(C)OC.C(C)(C)N C1(C(=O)NC2CN(C(C(OC)OC)=O)CC2O)CC12CCCCC2 CC(=Cn1ccnn1)C(=O)NC1C2CC(O)C1N(C(=O)C#CC1CCCOC1)C2 C1(NC(CSCC)=O)CC(NC(=O)Cn2cncc2C)C12CCOCC2 C1(OC)CN(C(=O)CCc2c(C)noc2C)CC1.C1(CC=O)NC(=O)NC1=O.N C(=O)(C1CCCc2cncn21)N1CC(CNC(c2c(C)cno2)=O)C(C)C1 C1(C(=O)NCC2(F)CCCN(C(=O)CC3CCC3)C2)Cc2cncn2C(=O)N1 n1(-c2ccc(C)cc2)c(C)cc(CNc2cn(C)nc2Cn2cccn2)c1C C1(C(=O)NCCCCCCNC(C(F)=C(C)C)=O)CCCCC1N=[N+]=[N-] CC1(C)C(CC(=O)NC2CC(C3CC3)C2)CCN1C(=O)CC1CC1 Cc1cc(C2CC2)ncc1C(=O)Nc1cccc(NC(c2c(Cl)cnn2C)=O)c1 C(=O)(CCC(=O)c1ccc(O)cc1)N1CCC(CCNC(=O)Cc2ccoc2)C1 c1(C(=O)N)ccc(Cl)c(Cl)c1O.C1(CNC(c2ncn(C)n2)=O)CCC12CCC2 [N-]=[N+]=NCC(C(=O)NCCCOCC1CCC1)NC(=O)CCC1CCCC1 Cc1ccc(COCC(=O)NCC2CC2)cc1.C1(C)(C=O)CCCCO1.C Cc1cc(N2CCC(C(N3CCC3CO)=O)CC2)n2nccc2n1 C1(NC(=O)CC2CC2)CC(NC(c2ncc(C3CC3)cc2F)=O)C12CCC2 c1(C=O)cn(C)nc1C(F)(F)F.Cn1ccc(C(=O)NC2CC(C)C2)n1.C N1(C(c2ccc(CC)[nH]2)=O)CC(C)N(C(=O)Cc2coc(C)n2)CC1C C1=CC(N=c2[nH]c(=NCCc3cn4c(n3)CCCC4)[nH]c3c2CCCC3)CCC1 C(C(C(=O)Nc1ccccc1)N(C1CN2CCC1C2)C)(C1CCOC1)OC C1(C(=O)NCC(CNC(c2cccc(CC)n2)=O)CO)CC2(CCCCC2)CO1 C(=O)(C(C)CC(=O)NC1CCC(C(=O)NCC2(C(C)C)CC2)C1)OC C1(C(N2C(c3cc(C)on3)CCCC2)=O)CC12CCN(C(c1ccno1)=O)CC2 C1(C(N(CCOC)C)=O)CN(C(=O)CC2OCCO2)CC12CC2 C=C1CC2CCC(C1)N2C(=O)C(CCN(C)C)NC(=O)CN(C)C N1(C(=O)NCc2cccc(C(F)F)c2)CCCN(C2CCNC2)CC1 C=Cc1cnc(NC(=O)Cc2cccc(C(=O)O)c2F)nc1 C1(C(=O)NC2C(C)CCN(C(=O)CCCc3cnn[nH]3)C2)COC2CCCCC12 C1(CC(=O)N)CC(C2CC2)C1.C(C(CCO)NC(c1occc1C)=O)N(C)C C1(NC(c2nn(CC)nc2C)=O)CCN(C(=O)CN2CCCOC2=O)C(C)C1 CC1CCCC1CC(=O)NCC(C(=O)NCCN1CCC2CC12)N(C)C N1(C(c2c(N)non2)=O)CCCC2(CCC(NC(=O)CC3CCCCCC3)C2)C1 c1(C(=O)N)cnc(O)c2ccccc12.C=C(C)CCNC(=O)CCC1CC1(C)C CN=c1nc(N2CC3CCCC(C3)C2)[nH]c(N2CCC(NC(C)=O)CC2)n1 C1(C2CCCCC2)(C(N2CC(OC)CC(NC(C(CCC#C)O)=O)C2)=O)CC1 c1(CNC(C2C(CCC)CN(C(c3sncc3C)=O)C2)=O)cccc(O)c1C Cc1ccc(C)c(C(=O)NCCCS(C)(=N)=O)c1 CCC(O)(CN(C)C(C1CCC(NC(c2c[nH][nH]c2=N)=O)CC1)=O)CC C1(C=O)CCOC(C)C1.C1(CC(=O)NCC2(C)CC2)(COC)CC1.N C(CN=c1nc(N2CCN(CC(N)=O)CC2)c2sccc2[nH]1)N(CCCC)C C1(C(=O)NC2C(C(N(C)Cc3ccncc3)=O)OCC2)C(C)(C)C1(C)C C1(C(N(C)CC2OCCN(C(CC(C)(C)OC)=O)C2)=O)CC(C(C)(C)C)=NO1 C1(NC(CC(=O)NCC)=O)CC2CCC(C1)N2c1nnc(C)s1 C#Cc1cn(C)nc1C(N1CCC(C)(CNC(=O)CCO)CC1)=O.CC(C)C C1(NC(CCSC)=O)CCC(NC(c2cc(C3CCC3)on2)=O)C1 N1(C(CNC(c2ccccc2)=O)=O)CCN(C(=O)NCCCl)CC1 C(=O)(CCCCC(=O)NCC1CC(NC(=O)CC2CC=CC2)C1)OCC N1(C(c2n(CCCC)ncc2)=O)CCC(C)(CC)C1.C(C(C)(C)C)=CC=O.N Cc1cc(O)n2ncc(C(=O)N(C(C)CNC(c3c(C)nn(C)c3N)=O)C)c2n1 CC(C)C(O)C(F)(F)C(=O)N(CCN=c1[nH]nc(-c2cccnc2)s1)C c1(N2C(C)(C(N(c3cnn(C4COC4)c3)C)=O)CC2)ncnc2c1CCCC2 CCC(C)(CNC(C1CC(NC(C2C3CCC(C3)C2C)=O)C1)=O)C(C)O c1(C(N2CCC(NC(c3c(OC)c[nH]n3)=O)C23CC3)=O)cc(Cl)c(F)c(Cl)c1 C1(C(N2CCN(C(c3c[nH]nc3C3CC3)=O)C(CCO)C2)=O)CC1C1CCCC1 Cc1cc(O)ccc1C(=O)NCC1CC(NC(C2COC3COCC23)=O)C1 c1(C=O)ccc2nccn2n1.CS(=O)(=O)C(CNC(c1ccc(O)nc1)=O)C.N c1(C(=O)NCC2N(C(c3cnc(C)s3)=O)CCCC2C)noc2c1CCCC2 C1(C(=O)NC(c2cccnc2)CC)C2CCC(C2)N1C(=O)C(F)=CC1CC1 CN1CCN(C)CC(C(N2CC(=C(F)CNC(=O)CC3CC3)C2)=O)C1 Cc1ccc(OCC(=O)NC2CCCC(CNC(=O)C(F)(F)C)C2)c(F)c1 C1(C(N2CC(C(=O)NCCn3ccnc3C)(CC)C2)=O)C2CC3C(C2)C13 CC1=C(C(=O)NC2COCC2)CCC(C)(C)C1.C12(C=O)CC(C)(C1)OC2(C)C C(=O)(C(=O)N=c1ccc(C(C)(C)C)n[nH]1)NCCc1nc(C)nc(O)c1 O(P(=O)(CCCN=C(NCC1CN(C)CCN1C)NCC(C)C)OCC)CC CC1CC2(CCN(C(=O)C(C)CNC(=O)CC3CCOC3=O)C2)CO1 CCCCC(C(=O)NC1COCC1C(N1CC(=O)NC(CC)C1)=O)C(C)C CCC(CC)(CCNC(=O)C(F)C(C)C)NC(=O)CCN1CCC(O)CC1 C=Cc1cnn(C)c1C(N1CCCCC(NC(C2CCCC2O)=O)C1)=O C1(O)(CNC(c2onc(C)c2C)=O)CCCN(C(=O)CCc2cccnc2Cl)C1 C(N=c1nc(N2CC3CS(=O)(=O)CC3C2)c2ncccc2[nH]1)c1scc(C)c1 N1(CC)CC2(CN(C(=O)C(N)Cc3nnc(-c4ccccc4F)s3)C2)C1 Cc1cc(O)nnc1C(N1CCCC1CNC(c1ccnn1C1CCCC1)=O)=O c1(C(=O)NC(C)CN(C)C(C2CC3CC3C2)=O)cc(Cl)ccc1OC(F)F N1(C(C(C)=C(C)C)=O)CC(C(N)=O)(CNC(=O)CCn2cnnn2)C1 N1(C(CC)=O)CCC2COC(CC(=O)Nc3nc(Cl)ccc3OC)C2C1 C(=O)(CS(=O)C(F)(F)F)NC1CCCN(C(c2n(CCOC)ncc2)=O)C1 c1(CCC)cc(C(N2CCOC(CNC(=O)COCC(C)C)C2)=O)c(C)o1 c1(C(N2C(CCNC(=O)CCCSc3ccccc3)CCC2)=O)cccc(=O)o1 C1(C(=O)NCCC2N(C(Cn3c(C)csc3=O)=O)CCC2)CC2(CCCC2)C1 C(C)(CCCSC)NC(C1(CNC(C=CC=CCC)=O)CC1)=O C1(C=O)CC2(C1)CC1(CC1)C2.CN1CC(C)(C(N2CCC(C)C2)=O)CC1=O.C C#Cc1ccc(NC(N2CCC(NC(C3CCCC3)=O)CC2)=O)cn1 N1(C(c2c(NC(c3noc(C)c3C)=O)cnc(Cl)c2)=O)Cc2cncnc2C1 c1(C(=O)NC(CC)CNC(c2cc(C(N)=O)cs2)=O)nc(=N)cc[nH]1 c1(NC(c2cccc(C)n2)COC)cc(NCC2CCN(C)C2)ncn1 C1CC(CC)N(C(=O)C=C2CCCCC2)C1.C(c1cn(C)nn1)=CC=O.CO N1(C(C2(C(=O)NC)CC2)=O)CC2(CCN(C(c3cnn4cc[nH]c34)=O)C2)C1 CC1ON=C(C(=O)N2CCCCC(N(C)C(C3CC4CCC3CC4)=O)C2)C1C c1(C=O)ccc(F)c(Cl)c1.CC(C)C(C)CNC(C1(CC2CC2)CC1)=O Cc1cc(CNC(=O)C(c2ccoc2)NC(c2[nH]ccc2C)=O)cc(O)c1 C1(CNC(c2ccc(OCCF)cn2)=O)CC2CCC1N2C(=O)CC(F)(F)F C(C(=O)N1CCOC(C2(C)CC2)C1)(C(C)(C)O)NC(CCSCC)=O c1(CN(C=O)C(c2scc(CC)n2)C)nc(Br)sc1C CC(C)(F)C(C)(F)C(=O)N.C1(C(F)F)CCN(C(c2ccc(C(F)F)o2)=O)C1 C1(NC(Cc2n(C)nnc2)=O)CC12CCN(C(c1ccc(F)cn1)=O)C2 C1CCS(=O)(=O)C12CN(C(C1(C)COC1)=O)C2.c1(CC)cc(C(=O)N)ncn1 Cc1ncc(C(N2CC(N(C(=O)Cc3cnc(C)s3)C)C(F)C2)=O)c(C)n1 Cc1c[nH]cc(C(=O)NC2CC(CNC(=O)CCC3(C#N)CCC3)C2)c1=O C1(C2CCCCC2)(C(=O)NCC=CCNC(=O)CC2CCCCC2O)CC1 S(=O)(=O)(c1ccc(NCc2ccccc2F)c(F)c1)N1C2CN(C)C(C2)C1 C1(C(=O)NCC(=C2CN(C(C(C(C)C)SC)=O)C2)F)CCCCNC1=O CCCCCCNC(C1CCC(C(F)(F)F)O1)=O.C(=O)C(F)(F)CC1CC1.N c1(C(N(C)C=O)=O)ccc(Cc2cccnc2)cc1.N1(CC)CCC1.C1CCC1 c1(NC(C)C)ccccc1C(=O)NC1CN(CCC2COCC2O)C1 C(CC)(CCC(=O)N(CC(O)COC)C)NC(c1c(CC)cc[nH]1)=O C(=O)(CC(C)CNC(=O)C(C1CC1)NC(C1COCC(C)O1)=O)NC CCC(C)(C)C(C)CC(=O)N1CC2C(N(C)C(c3ccc(Br)s3)=O)C2C1 c1(-c2nc(CCCCN(C)C)nn2-c2cc(Cl)nc(Cl)c2)ncc(F)cc1F c1(C(N2CCC(O)(CNC(c3c(Cl)cnc(C)n3)=O)C2)=O)c(N)ccc(F)c1C CC1COC2(C1)CN(C(C1CSCCN1C(=O)CC1CCCCC1O)=O)C2 C=CCCC(F)(F)C(=O)N1C2CCC1CC(CCNC(=O)Cc1cc[nH]n1)C2 CCC(C(=O)NCC1(O)CCN(C(C2CC(C(=O)O)C2)=O)C1)C(C)(C)CC C(CCC(C)C(=O)NCC(=C1CN(C(=O)CC(C)C(F)F)C1)F)OC C(C(C)C(=O)NC(CC1CCC1)C(=O)NC(C1CCC1)C)OC c1(NC(CS(CC)(=O)=O)=O)c(F)cnc(Cl)c1Cl c1(C(=O)NCC(c2ccc(F)cc2)NC(C2(C#C)CC2)=O)cccc(Cl)c1F c1(-c2cc(C(=O)NC3CCN(C(C4(C=C)CC4)=O)C3)n[nH]2)ccc(F)cc1 C1(NC(C2CCC(NC(C)=O)CC2)=O)CCCN(C(=O)CCCC2CCC2)C1C C1(C(N(C2CCCN(C(C3CCO3)=O)C2)CCF)=O)C2(CCC2)C12CCC2 N1(C(C(C)OCCC=C)=O)CCC2(CCOC2)C(CNC(C2CCC2=C)=O)C1 N1(C(c2cnn(CC3CCOC3)c2)C(=O)NCC(=C)C)CCSC(CC)C1.C C1(N(C(C(CC)NC(N)=O)=O)C)C2CC1N(C(=O)Cc1sc(O)nc1O)C2 C(=O)(C(CCOCCO)NC(C1CC=CCC1)=O)N(CCCCO)C CC1CN(C(C2(C)CCCN2C(=O)CCc2nc[nH]n2)=O)CC(C)(C)CO1 Cn1cc([N+](=O)[O-])c(C(=O)NC2CCN(C(C3(C)CNC(=O)C3)=O)CC2)n1.C CC1CC(NC(=O)CCN2CCOCC2=O)CN1C(=O)CCc1cocn1 C1(CNC(C2(c3ccccc3)CCC2)=O)(CC2CC2)CCOC1 N1(C(c2c(OC)scc2)=O)CCCC(C)(C(=O)NCC(C)(C)OC)C1 c1(OC)c(C)cc(C(=O)NCC(C)(O)C)cc1C.C1(C)(C=O)CC(F)(F)C1 CCCCCC(C)Cc1nc(-c2ccc(OC(F)F)cc2)nn1C(C)C(F)(F)F Cc1cc(C(=O)NC2CCC(C)N(C(c3cncc(N)c3)=O)C2)cc(C)c1Cl CC1(C)CCCC(CC(=O)NCCCCCNC(c2cn(C(C)(C)C)nn2)=O)O1 N1(C(c2c(N)ncc(C)c2)=O)CCCC2(C1)CN(C(C1CC13CC3(F)F)=O)C2 C(C)(C)(CCC(=O)N1CCC(C)(CCC)C1)NC(C=C(CCC)C)=O CCCCCCC(C)C(=O)NC(CO)C(=O)NC1CN(C)CC1(F)F c1(CNC(=O)CCc2nccs2)ccsc1C(=O)NCCN1CC2CC2C1 CCCC(C(=O)NCC1CN(C(c2cc(F)cc3c2CCC3)=O)C1)S(N)(=O)=O CC1CCN(C(c2cc(-c3cnn(C)c3)on2)=O)CC1NC(c1coc(O)n1)=O c1(C(N2CCC(NC(C3CC(CC)(CC)C3)=O)C(O)C2)=O)cnc2c(c1)CCC2 c1(C(N2CCN(CC(O)C(F)(F)F)CC2)=O)cc2c(cn1)OCCO2 C(=O)(CCC(=O)NCC1(CC)CC1)NCCOCCCCCC.c1nccs1 c1(OC)cc(C(=O)NCC(C2(O)CN(C(=O)CCC)C2)(C)C)on1.C(C)=O c1(C(C)NC2CC(C)N(Cc3ccccc3)C2)cc(Br)c2c(c1)CNCCO2 C1(C(=O)NC)(NC(=O)CCc2ccn(C)n2)CCCC1 c1(CCC)ccc(C(N2CCC(CCNC(=O)CC3CC(C)(C)C3)C2)=O)[nH]1 C(c1cccc(F)c1)=CC(N1CC(CN(C(=O)C(c2ccnn2C)O)C)C1)=O N1(C(COCCCOC)=O)CCN(C(c2cc(=O)c(OC)c[nH]2)=O)CC1CO c1(CC)c(C(=O)NC(C)CO)cnc2ncnn12.c1(C=O)ccoc1C(C)C.N N1(Cc2cnc(C)s2)CCC2(CCN(C(c3cnnn3C)=O)C2)C1 c1(C(=O)NC(CN(C(C2CCC(CCC)CC2)=O)C)C)cc(C)c(N)cc1F CCCCCCC(CC)C(=O)N1CCCC(C)C1CN=c1[nH]c2ccccc2o1 C(=O)(C(F)C(C)(C)O)N1CC2C(CNC(c3nn(C)c(C(F)F)c3)=O)C2C1 C(=O)(C#CC1CCCCO1)N.C1(CC(=O)NCC2CCCC2)C=CS(=O)(=O)C1 CC1CCCC=C1C(=O)NCC1CCCCC1NC(c1c[nH]nc1C1CCC1)=O N1(C(C(C=C)(F)F)=O)CC=C(CNC(=O)C=Cc2ccoc2)CC1 C1(C2CC2)(CNC(c2n(C)c(Cl)cn2)=O)CCN(C(=O)CC(C)(F)F)C1 N1(C(c2c(CC=C)cccc2)=O)CC(C(=O)N)C(C)(C)C1.C1CCC(C2CC2)C1 N1(C(=O)CC2CCCCO2)CCC2CN(C(c3cc4ccoc4s3)=O)CC2C1 Cc1ccoc1CC(=O)NC(C)C(c1ccccc1)NC(=O)CCn1cccn1 c1(NC(=O)COc2ccccc2F)cc(C(F)F)cc(Br)c1 C1(NC(C2N(C(Cn3cnc(C#N)n3)=O)CC=C2)=O)COCCC1(F)F CCCCC(C(C)C)N1CCOCC(C(=O)NCC2(COC)CCCC2)C1 N1(C(C(C)Oc2ccccn2)=O)CCn2cc(NCc3ncc[nH]3)nc2C1 N1(C(C(C)NC(C)=O)=O)CCC(C)(CNC(=O)C(C)(F)F)C1 c1(N2CC(CNC(C(C)(C)N(C)C)=O)C(C)(C)CC2)nc2ccc(Cl)cc2s1 c1(CNc2cn(C)c(C(=O)NCC3COC3)c2)ncc(Cl)cc1Cl C1(C=O)CCCC(=O)C1.c1(C(=O)NCC(C2CCC2)OC)cc(C)[nH]n1.N N1(C(CCCCSC)=O)CCOCC(F)(CNC(C2(CCF)CCOCC2)=O)C1 CC1(C)CC(O)CN(C(C2CCCN(C(c3ccc(O)c(F)c3)=O)CC2)=O)C1 C(c1ncccc1C)=CC(N1CCC(C)(NC(CCC=C)=O)C1)=O C1(NC(=O)Cc2cn[nH]c2)CCC2CN(C(c3ccc(Br)o3)=O)CCC2C1 CC(C)(C)S(=O)(=NC(=O)c1cc(N)cc([N+](=O)[O-])c1)C(N)=O C(CC(=O)NCC1CC(SC)C1)(C(F)F)NC(C1OCCN(CC)C1)=O N1(C(C(C)(C)CO)=O)CC(NC(c2cnc3sccn23)=O)C(S(C)(=O)=O)C1 C1(OCC)CC(C(=O)N(C)Cc2csc(C)n2)C12CCOCC2 Cc1c[nH]cc(C(=O)N(C)CC2CCCC(NC(=O)CCC3(C)CC3)C2)c1=O C=CC(CC)C(=O)NCC=C1CCN(C(C2(CCCC)CCC2)=O)CC1 N1(C(C2(SC)CCC2)=O)CCC2C(CCN2C(=O)CC2CCOCC2(C)C)C1 c1(C2CCN(C(C3CC(C(=O)OC)N3C(C)=O)=O)C2)cc(O)nc(O)n1 c1(CNC(C(C)NC(N)=O)=O)cc(C(=O)N(C2CCCC2O)C)on1 c1(NC(CC(CNC(c2cc(C)ncc2)=O)C)=O)c(C)nn(C)c1C Cc1cc(O)ncc1C(=O)NC1CCCC1NC(=O)CC(C)F c1(C(=O)NC23C(CCN(C(c4n(C)ncc4)=O)CC2)C3)cnn2cccc(Cl)c12 CCC(C)C(C(=O)NCc1cc(C(=O)N(C(C)C(C)(C)C)C)cs1)N(C)C C(=O)(C1=CCCCC1)NCC(CNC(C1(c2ccc(C)cc2)CC1)=O)O C=CCCCC(=O)N1CCCC(CNC(=O)COC2CC(F)(F)C2)C1 C1(C(=O)Nc2ncc(C)s2)Cc2nccnc2CN1C(=O)C(c1ccccn1)C C1(O)CCN(C(c2cn(CCO)nn2)=O)CC1.C(C(=O)NC)(C(C)C)OCC.C C1(NC(c2ccc(=O)n(CCO)c2)=O)CCCCN(c2ncc(Br)cn2)C1 c1(CN)ccc(OCCC(=O)NC(c2ccccn2)CO)cc1 CC1CCCC(OCC(=O)NC(C)CNc2ccc(OC3CC3)cc2)C1.O CC1(CNC(c2cnc3c(c2)CCC3)=O)CCOC2(CCC2)C1 N1(C(c2cnc(CC)o2)=O)CCC2CN(C(=O)C(F)C3CCCC3)CC12 C1(NC(Cc2ccc(C(=O)NC)cc2)=O)CCCC(NC(=O)CCOC)CC1 Cc1cc(C(=O)NCC2CCN(C(=O)CC(C)C)C2)cc(O)n1.C(=O)C(C)C C1(NC(c2ccn(C)n2)=O)CCN(C(c2cccc(C3CC3)n2)=O)CCC1(F)F c1(CCNC(C2CCC(=O)N2)=O)c(F)cc(Br)cc1F N1(C(CCCCOC)=O)CCC(C)(C)C(C)C1.C1(C=O)CC2(C1)CC(F)(F)C2.N Cc1nn(C)cc1C(=O)NC1CCCCC1CNC(c1cc(Cl)ns1)=O CCC(C)(C#N)C(=O)NCCC1CN(C(=O)C=CSC)CCO1 c1(CNC(=O)CC2CC(NCc3cc(Br)cs3)C2)cc(Br)ccn1 C=CC1(CC(=O)NC2CN(C(c3cncc(NCC)c3)=O)CC2O)CCCCC1 C(CNC(C1C(c2ccccc2)C1(C)C)=O)(C(C)(C)C)NC(CC=C=C)=O C(=O)(CCCC(C)=O)N1C(C(=O)NCc2c(OC)cccc2)CCC1C c1(C(=O)NC(C2(O)CN(C(c3ccc(F)o3)=O)C2)C)csc(-c2ccoc2)n1 CC(C)CC(C)(C)C(=O)NCC(C)(C(C)C)NC(C1CC1C(F)(F)F)=O C#Cc1ccc(C(N2CCCC(NC(c3ccnn3CCF)=O)CC2)=O)cc1C C1(C#CC(=O)N2CCC2C(=O)NCCc2ccccc2O)(CC)COC1 c1(C(=O)NC(c2cccc(O)c2)C)ccn2ncc([N+](=O)[O-])c2n1 C1(NC(COCC)=O)CCN(C(c2ccccc2-n2cccc2)=O)C(C2CC2)C1 C1(OC)CCC2(C(=O)NC(CC3CCCCO3)C(=O)O)CC12 c1(C(N2CCC(C(C)NC(C=CCOC)=O)C2)=O)cc(Br)n(C)n1 N1(C(C(C)N(CC)CC)=O)CCN(C(=O)Cc2nncn2C(C)C)C(C)C1 C=CC1CCCN(C(c2nc(C)[nH]c2Br)C(=O)NC(C)(C)C)C1 C1(CNC)CCCCN1C(C1CC(=O)N(C2CCCC2)C1)=O.C1CC2CCC1O2.C C12(C(N3C4(CNC(CCC#CC)=O)CCC3CC4)=O)CCCCC1CCC2 c1(C(=O)NCCN(CCC)C(c2ccncc2C(F)F)=O)cnc2[nH]nnc2c1 c1(C2(C(=O)NC3CN(C(=O)C(O)C4CCCC4)C3)CC2)ccc(Cl)cc1 Cc1nc(NC(C2CN(S(=O)(=O)c3ccccn3)CCC2O)=O)cnc1C#N C(CC(=O)NC(c1nncs1)C)(C(C)(C)C)NC(c1c(C)ncs1)=O c1(C(C)NC(=O)C(N2CC3CCC3(C)C2)=O)nc2c(s1)CCCC2 C#Cc1ccc(C(N2CCC(C=CC(N3CCC(C(N)=O)C3)=O)CC2)=O)cc1 C(=O)(CC1OCCc2ccccc21)NC1CN(C(C(C)(C)C)=O)CC12CC2 N1(C(c2[nH]cc(C(C(C)C)=O)c2)=O)CCC(O)(CC)C1.c1(C=O)csc(O)n1.N CC1C(NC(=O)Cn2ncccc2=O)CCCN1C(=O)CC1CCC(C)(O)CC1 Cc1nc(C)c(CNC(=O)CC2CCCN2C(=O)CCC2(C#N)CCC2)s1 c1(C=O)cnc([N+](=O)[O-])n1C.Cc1oc(C)c(C(=O)NC2CCC(C)C2)c1C.N Cc1csc(C)c1C(=O)NCc1ccccc1.c1(C(NC)=O)nc(Cl)oc1C.C N1(C(c2c(C)n[nH]c2C)=O)CCc2ccccc2C(NC(C2CCCN2C)=O)C1 C1(CC)CN(C(C23CC(C)(CCO2)C3)=O)CC(C)O1.C(=O)(C(C=O)OC)OC CC(C(C)(C)C#N)NC(C1(C(C)NC(=O)Cc2cccc(F)c2)CC1)=O Cc1cccc(SCC(=O)NCC2(CNc3ncc(Cl)cn3)CCC2)c1 c1(C(N2C3CC(NC(C(COC)N(C)C)=O)C2CC3)=O)n[nH]c2cccnc12 C12(CNC(CC=CCC)=O)CCCC1CN(C(=O)CCN(CC)CC)C2 CC(c1cccs1)=CC(N1CCC(O)(CCNC(C2(C(N)=O)CC2)=O)C1)=O Cc1cccc(F)c1CC(N1CCC(C)(NC(C2CCCCS2(=O)=O)=O)C1)=O c1(C(=O)NCc2occ(C(=O)NCC(C)C#N)c2)cc(O)ccc1F C1(CC(C)C)COCCN1C(C1CC1NC(C1CCCC1C)=O)=O O(NC(=O)C(CCCOC)NC(c1cc2ncccc2[nH]1)=O)CCCC=C c1(C(N2CCC(C(C)NC(=O)C(C)(C)c3cnco3)C2)=O)cc(N)ccn1 CC(C)CC(C(=O)N(CC(O)CNC(=O)C=Cc1cccc(C#N)c1)C)C(C)C N1(C(C2(OC)CC2)=O)CCCC2(C1)CN(C(c1nccn3ccnc13)=O)CCO2 C(=O)(N=c1[nH][nH]c2c1CN(Cc1cnc3sccn13)C2)c1c(C)[nH]c2ccccc21 C=CCC(C(=O)N(C)CC1CCCCC1)NC(=O)CC1CC1 C1(C(=O)NCCOCCCN(C(=O)CCN2CCC2)C)(CO)CCOCC1 CCC(C)(CNC(=O)C(=O)N(C)C)NC(=O)CCCn1cccn1 C(=O)(C(C)(C)CCC#N)NCC(C(C)(C)C)NC(C(C(C)C)n1ccnc1)=O c1(C(N2C(CC(=O)NCCN(C(CC)C)C)COCC2)=O)ccc(F)cc1F c1(C(C(C)O)C)nc(-c2ccc(N(C)C)cc2)nn1-c1ccnc(F)c1 C1(C(N2C(C)(CC)CC2)=O)CN(C(c2cc(C)cc(O)c2)=O)C2(CCC2)C1 Cc1cc(C(=O)N(C2CCC(NC(C3CCOCC3)=O)CC2)C)c(N)c(F)c1 C=CCN=C(NCCc1ccc(O)cc1)NCC1(c2ccccc2Cl)CCC1 Cc1ccc(C(=O)NCC2CCCN2Cc2csc(N(C)C)n2)cc1[N+](=O)[O-] C1(CCOC)(NC(=O)Cc2ccsc2)CCN(C(=O)Cc2ccccc2C)CC1 C1(NC(c2c(C)cnn2C)=O)CCCN(C(=O)Cc2ccc(C#N)cc2)CC1F c1(C(N(CC(C)C(=O)N(C)Cc2ccccc2)C)=O)cn2ccccc2n1 C(=O)(CC1OCCc2sccc21)NC1(C)CC(NC(COCCC)=O)C1 CCCC(C#N)C(=O)NC(C(=O)Nc1cnn(CC2CC2)c1)C1CC1 c1(C(=O)NCC(CCCC)NC(=O)CN(C2CCC2)C)c(C)cc(C)nc1Cl N1(C(c2c(C)nc(CCC)o2)=O)CC(C2CCCCN(C(=O)C3=CCCO3)C2)C1 C1(C2(C(=O)NC3C(CNC(c4ccc(CO)s4)=O)C3)CC2)CCCCO1 c1(C(=O)N)cccc(C2CC2)c1.c1(C(=O)OC)cnc(N2CCNCC2)o1 C(=O)(C1=C(C)CCCC1(C)C)N(CCC)CC.C1(O)(C(=O)N)CC(F)(F)C1 N1(C(C(c2ccccc2)OCC)=O)CC2CC(C1)CN(C(c1nnsc1C)=O)C2 CC1(CNC(=O)CCC2CCC2)CCCN(C(=O)CCN2CCOCC2)C1 Cc1cc(Br)cc(C(N2CC3CC2CS3=O)C(=O)Nc2ccc(Cl)cc2F)n1 C12(NC(C(CC)CC)=O)CCCCCC1N(C(c1nc3cnccc3s1)=O)CC2 C1(NC(=O)COc2ccon2)CCCC1C.C1(C2(C(=O)N)CC2)CCCO1 Cc1cc(=NCC(S(C)(=O)=O)C2CC2)[nH]c(N2Cc3[nH][nH]c(=N)c3C2)n1 c1(CCC(N2CCc3sc(C(=O)O)cc3C2)=O)cc(Br)cc2c1OCC2 CCCCC(C)(F)C(=O)NCC1(C)CC1.C1(c2ccccc2)(C=O)CCCO1.N C1C(O)CCC(=O)N1.CCCC(C)CCc1nc(CC)no1 c1(NC(CONC(C=Cc2cc(C)no2)=O)=O)ccc2c(c1)COC2 C(C(C)(C)C(=O)N(C)CCc1cc[nH]n1)NC(c1cnn(C(C)C)n1)=O N1(C(C(C(CC)C)NC(N)=O)=O)CCN(C(=O)Cc2cc(C)no2)C2COCC12 CC1CN(N2CCC3(CCC3)C(C(=O)OC(C)(C)C)C2)C(C)CCO1 N1(CC)CC(C(=O)NC2(C)CC(F)(F)C2)c2ccccc21 N1(C(C2CCN(C(C)=O)C2)=O)CC(NC(c2c(C)cccc2C)=O)C(C)(C)C1 Cc1ccc(CC(N2CC(CN=c3[nH]nc(CO)s3)(O)C2)=O)c(Cl)c1 N1(C(CCC(CC)NC(=O)C(C)=C2CCCC2)=O)CCC(CO)=C(F)C1 C=CC(C)(O)C(=O)NC(C)CC1CCN(C(=O)CC2CCC(=O)N2)CC1 c1(SCC(=O)NCC2CN(C(C=C(C)C(C)C)=O)C2)ccsc1[N+](=O)[O-] N1(C(CCCCC#N)=O)CC2(COC(CNC(=O)Cn3ncccc3=O)C2)C1 C1(NC(CC=CCC)=O)CCCCCC1C(=O)Nc1cncc(Cl)c1 N1(CC)CCCC(C(=O)NC(COC)CC(=O)Nc2c(OC)noc2C)C1 N1(C(C(CC#C)C)=O)CC2CCN(C(=O)Cc3cc(Cl)cc(Cl)c3)C2C1 c1(CC)c(C(=O)NC2CC2CNC(=O)C(N2C(C)CCC2C)C)cn[nH]1 C1(NC(CC2CC(C)(C)C2)=O)COC2(C1)CN(C(=O)C(C#N)C1CC1)C2 C12(NC(N(C(CC)Cc3ccccc3Br)C)=O)CC(C)(C1)OC21COC1 N1(C(C=CC=C)=O)CC(CC=C)C2(C1)CN(C(c1cc(I)c(C)cc1F)=O)C2.C C(C1=NOC2CN(C(c3cc4c(O)nccc4[nH]3)=O)CC12)OC C(CC(C(C)(C)C)NC(=O)Cn1cnnc1)N(C(=O)CCc1ccc(O)nn1)C C1(CCNC(C(C)C2CCC2)=O)CN(C(=O)COCP(C)(C)=O)CCCO1 CON(C)C1CN(C(C2CC(C)(C)CN2C(c2ccc([N+](=O)[O-])o2)=O)=O)C1 C1(CCNC(c2n[nH]c(C)c2O)=O)CCN(C(=O)C=Cc2cnccn2)C(C)C1 C1(NC(CC2(COC)CC2)=O)CN(C(c2csc(SC)n2)=O)C2CCCCC12 N1(C(C2CCN(Cc3c(Cl)cccc3I)CC2O)=O)CCCCC(F)(F)C1 C1(C(N(C)C)=O)CC2C(C1)C2(C)C.N1(C(Cc2nc(CC)sc2)=O)CCOCC1 Cc1cc(NC(C2CCCCO2)=O)ccc1NC(=O)CC1CCC(=O)NC1 C(C(F)(F)C(=O)O)(c1ccccc1)NCc1cccc(C(N)=O)c1 CC(C(=O)N1CC(n2cc(-c3cncs3)nn2)CO1)C1CCCOC1 c1(C(=O)NCC2(C)OCCN(C(COCCCC)=O)C2)cc(C)c2occc2c1 C12(C=O)CCC(C1)C(C)(C)O2.C(CC)N(C(C)C)C.C1CC1C(C)(C)C N1(C(c2c(C)n(C(C)C)nc2)=O)C2CC1CN(C(c1cc(C(C)C)[nH]n1)=O)C2 c1(CC)cccc(C)c1C(N1CCN(C(=O)CCF)C(CO)C1)=O C(=O)(CCC(=O)CC)NC(CCC)C(=O)NCC(O)C1(Cl)CC1 C(C(C)(C)CC(=O)N1CCCC1C(N(C)C[Si](C)(C)C)=O)OC c1(SC)c(-c2nc(CCn3ccnc3)nn2CCC(C)C)cnn1C c1(-c2nc(C(C)C3CC3)nn2CCc2cc(F)cc(Br)c2)cccc2c[nH]nc12 CCC(C)C(CNC(=O)C(Cn1cncn1)NC(C1CCOC1(C)C)=O)CO CC(C)C(CCN(C(=O)CC1CCOC1)C)NC(=O)C=C(Cl)Cl Cc1c(C(=O)NC(C)C(C)NC(c2ncc(Br)cn2)=O)ccn1C(C)C c1(OC)ccnc(C(=O)NC(C)CC(C)NC(c2ccnc(O)c2)=O)c1 Cc1ccccc1S(=O)(=O)CC(=O)NC(CNC(C1CCCOCC1)=O)C(C)C C(=O)(CC(F)(F)Cl)NCC(c1cccc(C)c1)NC(C=CC(CC)C)=O S(=O)(=O)(c1cccc(C#N)c1)NC1(COC)CCCCC1.C(C)CCN(C)C CC(CC1CCCCC1)C(=O)NC1CCC1NC(c1ccnn1C1CCC1)=O c1(OC(CNC(c2nnc(CC)s2)c2nnnn2C)C)ccccc1C C1(CNC(CC=C(C)C)=O)CCCN(C(c2cc(-c3ccccc3)no2)=O)C1 N1(C(CCOCC(C)C)=O)CC2CN(C(c3ccco3)=O)CCC2(CO)C1 C(C1c2ccccc2CN1C(c1cocc1C)=O)NC(COCCOCC#C)=O C1(C(=O)NCCCN(C(C2CCCCC(=O)C2)=O)CC)CCCCC(=O)N1 c1(N(C)CCC2CCN(C(C3COC(C)(C)C3)=O)CC2)ccc(C#N)nn1 c1(C(=O)NC2CN(Cc3ccc(F)nc3)CC2F)ccc2ncsc2c1 c1(-c2c(OC)n(C)nc2)nn(C(C)C)c(=O)n1CC CC(O)C(F)(F)C(=O)NC1CC2(C1)CC(NC(c1ccn(C)n1)=O)C2 c1(Cn2c(-c3ccc(NC(C)=O)cn3)nc(CC(CC)C)n2)ccc(Cl)cc1C c1(C(C)SCC)cccc(-c2noc(Cc3cccc(-n4cccn4)c3)n2)c1Br Cc1nn(-c2ccccc2)nc1Cn1cc(C(C)N(C)C)nn1 Cc1[nH]c2ccccc2c1CC(=O)NCC#CCNC(C1COCC(C)(C)O1)=O C1(NC(Cn2cc(C(C)=O)nn2)=O)C(C)CN(C(C2(Cl)CC2)=O)CC1C Cc1cnc(F)c(C(N2CCOCC(NC(c3ccn(C4CCC4)n3)=O)C2)=O)c1 C1(CCN(C(=O)CCCc2ncco2)C)CCCCN1C(=O)CN1CCCC1=O c1(C(=O)NC2C(F)CCN(C(C3NC(=O)OC3)=O)C2)ccnc2ncnn12 N1(C(Cc2scc(C)c2)=O)CCCC(NC(=O)Cc2cnccn2)CC1 C(=O)(C(C)(C)CC#N)NC1CC(CNC(C=CC(C)C)=O)C1 c1(C(C)(C)NC(=O)CC2(NC(C)(C)C)CC2)ccccc1 CC(C)C(O)CC(=O)N(C1CCCC1)CCCNC(=O)CN1CCCNC1=O C1(NC(NNC(=O)C2C(C)C2C)=O)CCC(P(C)(C)=O)C1 S(=O)(=O)(c1ccc(Cl)cc1F)N1CC2C(NC(c3ccc(I)cc3O)=O)C2C1 C(=O)(C(O)CCS(C)=O)N(C(C)CN(C(=O)CNS(=O)(=O)C1CC1)C)C c1(NC2C(OC)CS(=O)(=O)C2)nc2cccc(F)c2c(=NCC2CSC2)[nH]1 c1(C(=O)OC)cnc(NC2(C)CC2)c(Cl)c1.c1(C=O)cnc(O)c(C)c1.N C(C(=O)NCCO)(C1CCCC1)OC.C1(C=O)CCC1C(C)(C)C.CCC c1(N2CCC(O)(C(C)NC(C3(C)CCC(=O)N3)=O)C2)nc2ccccc2s1 CC(C)CC(CNC(c1ccc[nH]1)=O)NC(=O)CCC1CCC(=O)N1 c1(N(CCC(OC)OC)C)cc(C)c(F)c(C)c1 N1(C(CCOC(C)C)=O)CCC(C2CC2)C1.[SH](=O)(=O)c1cccs1.C(=O)(C)N c1(C(=O)NC(c2cccc(C)c2)CNC(C(CC)F)=O)c(F)ccc(F)c1F C(C(C)(C)CC(=O)Nc1cnn(CCF)c1)NC(c1c(C)con1)=O c1(C(=O)NCC2(F)CC(NC(c3csc(O)n3)=O)C2)ccc2nn[nH]c2c1 CCCCC(C)CCC(=O)N1CCCC1CNC(C1(C(F)(F)F)CC(C)(C)C1)=O Cc1cc(C(N2CC(CNC(=O)CC3CCC3C3CC3)C2)=O)nc(C)n1 N1(C(c2c(CC)ncs2)=O)CCC2(CC1)CN(C(=O)CCCC(C)C)CC(C)O2 c1(OC)cc(C(=O)NC(CNC(=O)CO)C(C)C)ccc1.c1cccnc1 C1(C(N2CC(CN(C(C3N(C(C)=O)CSC3)=O)C)C2)=O)OC(C)CC1C N1(C(C(CCCNC(c2cnc(O)o2)=O)O)=O)CCCC2COCC12 CN1CCCN(C(C2(Cc3ccccc3)CN(C(c3nnn(C)c3N)=O)C2)=O)CC1 c1(OCCC(=O)NCCCc2cn(CC(=O)OC)nn2)ccc(Cl)c(F)c1 c1(C(c2nnnn2CCCF)NCCc2n(C)ccc2)cncc(Br)c1 CC1COCCC1NC(C1C=CCCN1C(C1COC(=O)N1)=O)=O C1(C)(OC)CCCN(N2CCOC(c3cccc(C(F)(F)F)c3)C2)CC1 Cc1cc(C(N2CCC(C)(C)C2)=O)c(N)c(C)c1.C1(C=O)CC12CC(F)(F)C2 O=C(CCCN1CCCC1)NC1(CNC(C2COCCO2)=O)CCOC1 C(=O)(C(O)CC(F)(F)F)NCCC1(O)CN(C(CCCc2scc(C)n2)=O)C1 N1(C(CC2N(CC)CCOC2)=O)CC2(CCC2NC(c2cc(O)no2)=O)C1.C C12(NC(CC=CC=C)=O)CCCN(C(c3cncc4ccsc34)=O)CC1C2 c1(OC)cccc2sc(NC(=O)NC3CCC4C(CC3)C4(F)F)nc12 C=CC1(C2(C(=O)NCCC(C)N(C(=O)Cn3cccn3)C)CCC2)CCC1 C1(C)(NCc2onc(-c3n(C)cnc3)n2)CCNC(=O)C1 c1(C(CC)NC(=O)C(N2CCC(C(C)N)C2)=O)ccc(F)cc1C C(=O)C(C)(O)C=C.C(CC(=O)N(C(C)CC)C)N(CCOCCOC)C.N c1(C(N2C(CNC(CCC)=O)CCC2)=O)cnn2c1CCCC2C N1(Cc2c(OC(C)C)cccc2)CCN(C(=O)CC2COCC(C)(C)O2)C(C)C1 c1(C(=O)OC)ccc(C2CCCN2C(=O)NC2CCN(C(=O)N(C)C)C2)s1 N1(C(C2CC(C)(C)C(=O)NC2)=O)CCC2(CCCN2C(c2ccncc2Cl)=O)C1 C(C)(CNC(C1(C)CC=CC1)=O)(CO)OC.C1(CCC(=O)N)CCCN1C N1(C(c2cc3n(c2)CCC3)=O)CCN(C(=O)C(O)c2cnc[nH]2)CC(O)C1 N1(C(c2cc(OC)ncc2)=O)CC2(CC(C)C2)C1.C1(C=O)(C(F)F)CCCO1 Cc1n[nH]c(C)c1CC(=O)NCC(O)CCNC(=O)C=CC(C)(C)C C(=O)(C1=C(Cl)CCOC1)NC1CCC(CNC(CNC(=O)NC)=O)CC1 C(=O)(C1Cc2ccccc21)N1CC(n2cc(CNC(C(CC#C)C)=O)nn2)C1 N1(C(C(F)=C(C)C)=O)CCC(NC(=O)C(C)NC(=O)C2CC2)C(F)C1 Cc1ccccc1CN(C(=O)C(C)NC(=O)CSCC(N)=O)CCO C1(C(N2CCC2)=O)C(C(F)(F)F)C1[N+](=O)[O-].CC1CC(C(=O)NCC)CO1 N1(C(c2c(C)nc(C(C)OC)s2)=O)C2CCC1CC(n1cc(CN(C)C)nn1)C2 c1(CC(N2C(CNC(C3C(=C)C3)=O)CC2)=O)c(C)[nH]c2ccccc12 CC(C)CC(C(=O)NCCCCC(=O)NC1(C(F)F)CCC1)C(N)=O C(=O)(CC(CC(=O)N1CC(C)(C(=O)OC)C(C)(COC)C1)OC)OC C1(NC(C(C(C)C)O)=O)CC2(CCC(NC(c3cc4c(s3)CCC4)=O)CC2)C1 C1(C(N2C(C3(NC(C4(OC)CC4)=O)CC3)CCCC2)=O)CC(C2CCC2)C1 CN1CC(O)CCC1C(=O)N(C1CN(C(c2ccc(F)c(O)c2)=O)CCC1O)C N1(c2nccc(OCC)n2)CCN(C(c2ncc(C)cc2C)=O)CCC1C C(C)(CC(C)NC(C1CC(C)(O)C1)=O)NC(C1(OC)CCC1)=O N1(CCC#C)CCN(C(C2CC(NC(=O)CNc3ncccn3)C2)=O)CC1 c1(NC2(C)CC(NC(CC3CCCC(C)C3)=O)C2)nc(Cl)nc2c1ncn2C C#CC1CC2(CC2)CN1C(c1cccc(C(F)(F)F)c1)C(=O)NCCSC C1(C(=O)NC2C=CC(CNC(c3ccc[nH]3)=O)C2)CC2CCC(C1)C2(F)F c1(C(CNC(COC)=O)NC(c2ccn(CCN(C)C)n2)=O)ccccc1 N1(C(C2(NC(C)C)CC2)=O)CC(CNC(=O)CC2CCCC2)C(C)C1 c1(C=O)cc2c(s1)CCC(C)C2.C1(OC)(OC)CCC1C(N1CCCC1C)=O Cc1cnc2nc(C(=O)NC3CN(C(c4cccc(C(F)F)c4)=O)C3)nn2c1 c1(C(C(=O)NCCCSC)N(CC=C)CCOC)cn(C2CCCC2)nn1 N1(CCCNC(C2(C(N)=O)CCC2)=O)CCN(C(=O)CN2CCCNC2=O)CC1 C1(C(N)=O)CCCN(CC(N2CCCC(NC(C3(O)CCSCC3)=O)C2)=O)C1 C(=O)(C(C#N)C(C)(C)C)N1CCC(C)(CC(=O)NC2CC(C(C)C)OC2)C1 C(=O)(C(O)Cc1cnc[nH]1)N(CCN(C(C)C)C(c1csc(CF)n1)=O)C c1(CNC(CN(CC)CC)=O)nc2c(s1)CN(C(C1CC1C)=O)CC2 CCC(C)C(C)C(=O)NCC(N1CC2(CC(N(C)C)C2)C1)=O C1(c2ccccc2)(C(=O)NCC(C)CN(C)C(C2CC(F)C2)=O)CCOC1 c1(C(N2CCC(C3N(C(CCC#C)=O)CCC3)C2)=O)cc(COC)oc1C N1(C(CCc2n(C)ncc2)=O)CCC(F)(F)C(CNC(C2CCCN2N=O)=O)C1 Cc1csc(C(=O)NCC23CC2CN(C(=O)Cn2cc(Br)cn2)C3)c1C CCC(C)C(C)C(=O)N1CCC(NC(c2ccc(N)cc2C(C)(C)C)=O)CC1 c1(CC(N2CCC(CCC(=O)NCCc3c(C)ncs3)C2)=O)cccc(O)c1 C1(NC(=O)Cn2ncnn2)CC2CN(C(C3(n4cccc4)CCCC3)=O)CC2C1 c1(CNC(C(C)NC(=O)NC)=O)cccc(C(=O)N(CCC=O)C)n1.O c1(CC)ccc(C(N2CCC(CCNC(=O)CNC=O)C2)=O)c(O)c1.N CC1=C(C(=O)N2CCC=CC2C(=O)NCC(O)C(C)C)CCO1 n1(C(C)C)cnc2c(N3CCC(F)(CF)C3)[nH]c(=NC(C)c3ccoc3)nc12 Cc1cocc1C(=O)N(C)CC1CCCN1C(=O)CC1(C)CC1(F)Cl c1(C(=O)NC(CC)CN(C(=O)C(C)SC(C)C)CC)cc(Br)c[nH]1 C=CC(CC)C(=O)N1CCC(CO)(CNC(=O)C(C(C)C)OC)C1 c1(C(=O)NCC2(OC)CCN(C(=O)C=O)C2)cc2n(c1)CCCC2.C1CC1 C1(CC(N2CCCC2)=O)CCCC1(F)F.c1(C(N(C)C)=O)conc1C1CCC1 CC(O)C(F)(F)C(=O)N1CCCC(F)(C(=O)NCCn2ccnn2)C1 c1ccc([N+](=O)[O-])c(C#N)c1.CC1(C)CCC(C(=O)NCCC2(N)CCC2)CO1 C(C1=CCN(C(=O)CSc2ccc(Cl)cc2)CC1)NC(C(CN(C)C)O)=O Cc1nc(Br)ccc1NC1(c2nnnn2CC(F)F)CCOC(C(F)(F)F)C1 C1(NC(C2(NC(=O)C(O)Cn3cncn3)CCC2)=O)C2CCCCC12 CCCCCC(C)CC(=O)NCC1=CCN(C(C2(C(C)C)COC2)=O)CC1 C1(CC(N2C3CC(NC(c4cnc(SC)s4)=O)C2CC3)=O)Cc2ccccc2O1 C1(C(=O)NCC(C)(C(C)C)NC(Cc2c(C)n(C)nc2)=O)CCC2(CCC2)OC1 CC1CC(CNC(c2ccncc2)=O)CN1C(c1ccc(Cl)o1)=O.C1CCC1.O c1(CCC(=O)N(C(C)CNC(=O)CSC)CC)cn(C)nc1C c1(Cn2cc(CNC(C3(SC)CC(=O)C3)=O)nn2)cc2ccccc2o1 N1(CCCCC(=O)OC)CCN(C(=O)C(C(C)(C)C)C2CCCC2)CC1C C1(C(N(C(CNC(CCN(C)CC)=O)C2CC2)C)=O)CCn2nncc2C1 N1(C(C2C3CCN(C(C4(OC)CC4)=O)CC32)=O)CCCC(F)(F)CC1 N(C1CCCc2n[nH]cc21)CC1C(C)CCO1 C1(C)(NC(C(C)Cc2ccccn2)=O)CCCC1.C1(CC=O)CN(C(C)=O)C1 C(C(N=c1[nH]c(Cl)c(C#N)s1)C1CCC1)NC(C1C(C)OC(C)C1C)=O C1(CNC(CC2(COC)CC2)=O)CCN(C(=O)CCO)C12CC2.C(N)=O N1(c2nnc(C(c3ccoc3)C)n2C)CCN(c2ccc(C(C)(C)C)cc2)C(C)C1 C1(CC#C)(C(=O)NCCN(C(=O)CCCn2cccn2)C2CC2)CCCO1 N1(C(C2CCC2)=O)CCC(C)(CN=c2nc(C(C)(C)C)[nH]s2)CC1.C(=O)NC.N C(=O)(C(C)(CO)NC(=O)CC1CSCCO1)NC1C(CC=C)CCC1 CCC(CN(C)C)CC(=O)NCC(C(=O)NC(C)(CC)CCO)N(C)C c1(OC)ccc(C23CC(CC2C(N2CC(CN)CC2C)=O)C3)cc1 c1(C(=O)N=c2cc(C3CCOC3)[nH][nH]2)cc2c(C3=CCSCC3)cccc2cn1 c1(CC(=O)N(C2CC(NC(=O)CCCF)C2)C)cc2ccccc2cc1O O=C(C1=CCCSC1)NC1CC2C1CCN2C(c1ncccc1Br)=O CCCC(CNC(C1(C(N)=O)CCC1)=O)C(=O)NCc1ccc(CO)cc1 CCC(C)(CNC(c1occc1COC)=O)NC(=O)Cn1cc(Br)cn1 C1(OC)CC2CC1CN(C(=O)C(C1CCCO1)NC(=O)COC)C2 Cc1cc(CC(=O)NCC(C)(O)CNC(C2CCCN2C2CC2)=O)no1 c1(CC)cc(C(=O)NCCC(C)C)nn1CCO.N(S(N)(=O)=O)CC=O.N c1(C(=O)NCC(CC=C)NC(=O)CS)cc2c(s1)CCOC2.c1cnn(C)c1 C#CC1(O)CCN(C(=O)Nc2c(C)cnn2C(C)C2CC2)C1 C1(NC(C=C(C)C)=O)CN(C(c2cnc(Br)o2)=O)CC1(F)F Cc1ccc(C(N2CC(F)(CNC(C3(CC4CC4)CC3)=O)C2)=O)nc1 c1(C(C(F)(F)F)NC(C2CC3(CC(N)C3)C2)=O)ccc2nc(O)[nH]c2c1 C(=O)(C1=CCCCO1)NC1CCN(C(C2CCC2Cc2ccc(Cl)cc2)=O)CC1 c1(CC(N2CCC(N(C(=O)C=C(C)C)CCC)CC2)=O)ccc(Br)cc1F c1(-n2cc(CC3CCC(NC(C(COC)N(C)C)=O)C3)nn2)ccc(C)n1C c1(CC(N2CCCC(C)(CNC(CCCC(=C)C)=O)C2)=O)ccc(C)c(F)c1F N1(C(c2c(C)nc(O)[nH]2)=O)C2CCC1(CNC(c1ccnc(S)c1)=O)CC2 C(CCC(=O)N1C(C(=O)NCCC(C2CC2)C2CC2)CC1C)N(C(C)C)C C(C1CN(C(=O)CC2COCCN2C)Cc2ccccc21)NC(CSCC=C)=O N1(C(C(C)n2cnnn2)=O)CCN(C(c2ccc(Cl)cc2C(F)F)=O)CC1CO N1(Cc2cn(C)nn2)CCC(O)C(C(=O)Nc2c(O)ncnc2O)C1 c1(C(=O)NC(C2OCCN(C(CCOCC)=O)C2)C)onc2ccccc12 c1(OC)cccc(C(=O)OC)c1F.C1=CCNC1=O CCCC(CCCNC(c1cc(C2CC2)n(C)n1)=O)NC(=O)C(C)(C)CCC C1CN(C(c2cc(C(F)F)n(C)n2)=O)C2COCC2O1.CC(C(=O)NC)C1CC1 C#CCCCCCC(=O)NC1CN(C(c2n[nH]cc2Br)=O)CC1N=[N+]=[N-] c1(CN2CCN(C3CCS(=O)(=O)C3)CC2)nc(O)c2ccccc2n1 C1(NC(c2scc(C)c2)=O)C=CCN(C(C2CC2C(F)(F)F)=O)C1 c1(CN2C(C(=O)Nc3onc(C)c3Br)CC(O)C2)cccc2ccncc12 C1CCC(C)O1.C(=O)(CC)N(C1CCC1)C.C1(C(C)(C)O)(C=O)CCC1.N c1(CC)ccc(C(N2CC3C(N(C(=O)CC4CCCOCC4)C)C3C2)=O)cc1 C1(N(C(=O)COC2CCCC2)C)CCC(NC(c2cnc(C3CC3)o2)=O)C1 c1(CN2CC(C(=O)Nc3c(O)ccc(C)n3)SCC2)cc2cc(Br)ccc2[nH]1 C1(c2nc(-c3c(C)cccc3)nn2CCc2cccs2)CCc2n[nH]cc2C1C C(C)(CCCCNC(=O)Cc1csc(S)n1)NC(C(C)N(C(C)=O)C)=O Cc1nc(CO)oc1C(N1CCOC(CCNC(=O)C(C)(C)F)C1)=O Cc1cc(Cl)cc(Cl)c1OCC(=O)NCC(C(C)C)NC(C1COCCOC1)=O c1(SC)nc2ccccc2c(=NCC2CC(NC(C34CC(C)(C3)C4)=O)C2)[nH]1 Cc1cc(=O)oc(C)c1C(N1CCCN(C(c2ccsn2)=O)C(CO)C1)=O c1(CCC(N2CCC(C)C(CNC(C3CC(O)C3)=O)C2)=O)c[nH]c2ccccc12 c1(CCC(=O)NC2CCN(C(C(COC)(C)O)=O)C2)ccc(Cl)c(F)c1 O=C(NNC(=O)C1CC1)c1cncs1.c1(-c2ncc[nH]2)ccc(Cl)cc1 c1(C(N2CCN(Cc3c(C)nc(Cl)cc3)C3C2C3)=O)ccc2[nH]c(=O)ccc2c1 CC1CN(C(c2cnn(C)n2)=O)C(C)CN1C(=O)CC1CCCN(C)C1 C1(C(=O)NCC(C)N(C(C2(C)CC2)=O)CC)CCc2cnn(CC)c2C1 c1(OCC(N2CC3CC4CC3C2C4)=O)c(-c2ccccc2)cc2ccccn12 N1(C(CC(C)CF)=O)CCN(C(c2cc(Br)co2)=O)CC1C C1(NC(c2nn(C)c(F)c2)=O)COC2C(NC(=O)Cc3ncsc3Cl)COC12 CC1(NC(c2ccc(C(C)(C)C)cc2)=O)CCN(C(c2cscn2)=O)CC1 C1COC2C(NCC3(N4CCOCC4)CCCCC3)C2C1 C(=O)(CCCC(=O)N1CC2CC(NC(C3CCC(=O)N3)=O)C1C2)NC(C)C CC1CCC=C1C(=O)N1CCC(N(CCO)C(c2ccnc(N(C)C)c2)=O)CC1 c1(C(=O)NC2(CNC(C(CC)(C)COC)=O)CCCC2)ccc2nncn2c1 C#CCC(CC#C)NC(=O)C(C1CCN(C(=O)CCCC=C)C1)C N1(C(C2N=C(C)SC2)=O)CC2(C1)CN(C(=O)COCC(F)(F)F)CC2CO CCCC(C)(O)CC(=O)NC1(C)CCN(c2nnc(C(C)C)o2)CC1 c1(CC(=O)N(CCCNC(c2cncs2)=O)C(C)C)cnn2ccccc12 c1(C=O)nnn(C)c1C(F)F.C(=O)(COC1CCC1)NC(C1CC1)C N1(C(CN(c2ncccn2)C)=O)CC2CN(C(=O)C(C)(C)S(C)(=O)=O)CC(C1)O2 C1(N(C(Cc2cc(C)sc2)=O)C)CCCCC1NC(=O)C(N1CCCCC1=O)C N1(c2nnc(CC(C)C)s2)CCC2(CCCC2NC(c2ccoc2)=O)CC1 C(CCCCCNC(c1nsnc1O)=O)NC(=O)CCCF N1(C(c2c(C#C)cnn2C)=O)CCC(NC(=O)CCc2ccon2)CC(C)(C)C1 C1(C(N2CCC(N(C)C(c3cccc(CC#N)c3)=O)CC2)=O)CC2CCC(C1)O2 C1(C(=O)NCCCC(=O)N(CC(=O)NCCC)C)CCCC(C)(C)C1 c1(C(N2CC=CC(NC(c3cncc(CC)c3)=O)C2)=O)cnn2c1CC(C)CC2 C1(OC)CN(C(c2cncc(C(F)F)c2)=O)CC1NC(c1ccn(CCF)n1)=O C1(NC(c2ccoc2C)=O)CC12CCCCCC2.C12(C(=O)N)C=CC(CC1)C2 N1(C(c2c(C)c[nH]n2)=O)CC2CC2C1.c1(C(N(C)C)=O)cccc(C(C)(C)C)n1 N1(C(C2C(C=C)C2)=O)CCCCC(N(C(=O)CCOCCN(C)C)C)C1 C(=O)(C(C)CC(C)(C)C)NC(C(=O)Nc1c(OC)cc(F)cc1)C(C)C N1(C(c2c(CCC)cccc2)=O)CCC(C)CC1CNC(=O)C(CSC)OC c1(C(=O)NCC2CCCC(NC(C3(N(C)C)CC3)=O)C2)cc2ccoc2cc1F c1(N2CCCC(C(C)C)CC2)nc(N2CCC(CC(F)F)C2)nc2c1cnn2C n1(C(C)C)c(SCC2(c3nc(C(C)C)no3)CC2)nnc1C1CC1(C)C Cc1cn(CC(N2CC(N)C(C)(C)C2)=O)c(=O)nc1O C(c1cnc(OC)nc1)=CC(=O)N(CCNC(c1cnsc1C)=O)CC C1C(C)C(=O)NOCC(=O)N1.C(C(F)F)(C(C)(C)C)SC NC(=O)C(CCC(=O)O)C1CC1.C1C(=O)NOCC(=O)N1 N1(C(C2(OC)CC2)=O)CC2=C(C1)CN(C(c1cn(CCC(C)(C)C)nn1)=O)C2 C1(NC(c2cnc(C3CC3)[nH]2)=O)CCCC(NC(c2ncccc2Cl)=O)CC1 N1(c2cc(NCC(CC)C)ncn2)C2CCC1CC(CCF)C2 c1(C(N(CCCCNC(C2CC(C)OC2)=O)C)=O)ccc2c(c1)NC(=O)CN2 c1(C(=O)NCCN(CCCCCC)C(c2[nH]nnc2C)=O)cc(Cl)c(O)cc1C c1(SCC)cccnc1C(=O)NC(CNC(C1CCC(C)O1)=O)CO C12(C(=O)NC(CN(C(=O)C)CC)C)CC(C)C1C2.c1(C=O)ccoc1C N1(C(c2ncc(CC)nc2)=O)C2CCC1CN(C(c1cc(N)ccc1C)=O)CC2 c1(NC(c2ccc(OC3CCNCC3)nc2)=O)cc(-n2cccc2)ccc1Br N1(C(C2C(C)CN(C(=O)C3=CCCCO3)CC2)=O)CC(O)C(C2CC2)C1 C1(C(=O)NC(C(=O)NCCC)C)CC=CC(n2cc(-c3ccsc3)nn2)C1 Cc1noc(C(=O)NCC2CCCC2NC(=O)CC2CCNC2=O)n1 c1(C(=O)NCC(C)NC(c2cn(C)c(O)n2)=O)ccn2nncc2c1 c1(C(=O)NC(CN(C(=O)Cn2nnc(C)n2)CC)C)cc(C)cc2ccoc12 N1(CC(=O)N)CC(C(F)(F)F)CCC1=O.Cc1cc(C)c(C(=O)NCCC)[nH]1 C(=O)(C1=CCCCO1)NC1CC(C)(NC(C2CCC(Cc3ccccc3)C2)=O)C1 c1(C(=O)NC(CNC(C2(C)COCCO2)=O)C2CCC2)cc(N)c(Cl)cn1 C1(C(N2CC3C(CNC(c4cccc(Cl)c4F)=O)C3C2)=O)CC2(CCC2)CO1 c1(CCCSCC)nc(C2=S=Nc3ccccc32)n(-c2ncnn2C)n1 N1(CC=O)C(=O)NC(C)(C)C1=O.C(CCC=CC(=O)N)=C(C)C.C(C)C C=CCC(=O)NOC(CC(C)C)C(=O)N(C)CC1CC(F)(F)C1 N1(C(CSCC)=O)CCCCC1CC(=O)NCCN1CCNC(=O)C1 N1(C(C(C)=CC)=O)CCC2(CC(NC(=O)CCCCCn3cnnn3)C2)C1 c1(OC)cc(C)c(Cl)cc1C(=O)NCC(C)C.C(=O)(CCC1CC1(C)C)N S(=O)(=O)(c1ccc(C(F)F)cn1)NCc1cnc(C(C)C)[nH]1 c1(C(N2CCCC2CCC2CCCC2)C(=O)NCC2CC2)ccc(F)cc1F C1(OC)C(O)CN(C(c2cnc(SC)n2C)=O)C1CNC(c1ncoc1C)=O C1(NC(C)=O)CCC(C)(C)CC1CNC(c1cnn(C(C)C)c1Br)=O N1(C(CC(C)(F)F)=O)CC2(CC(C(N3CC4CC(CO)C(C4)C3)=O)CO2)C1 CC(C)C(C)(CNC(=O)C=CC1(C)COC1)NC(=O)CC1CC12CC2 N1(C(C(c2ncccn2)OC)=O)CC(CO)(Cc2ccccc2)C1 CC1CN(C)CC(C(=O)NCCOCC(=O)NCC2CNC(=O)O2)O1 C(C1CCc2ncnn21)OC1CCN(C(c2cnn(-c3ccccc3)c2)=O)CC1 C(=O)(C1=NOC2(CCOC2)C1)N.c1(SC(C)C(=O)NC2CC(F)C2)nncn1C Cc1ccccc1C(C)CC(N1CCN(C(=O)CNC(c2ccsn2)=O)CC1)=O c1(NC(=O)N(c2cccc(I)c2)CC2CC2)cc2oc(O)nc2cc1F Cc1ccc(O)c(C(N2CCCC2C(C)(C)NC(c2n[nH]c(C)c2F)=O)=O)n1 c1(C(=O)N)cc2c(o1)CCCC2.N1(CC)CCN(C(C23CC(F)(C2)C3)=O)CC1 C(C)(CNC(c1ccc(CCO)cc1)=O)(CC(C)C)NC(c1cncc(C)n1)=O C1(C=O)C2CCC(C2)N1C(=O)C.c1(C=O)ccccn1.C(=O)N(C)C.CO O=C(N=c1c(Br)c[nH]cc1I)C1=CCCN(C(c2ccn3ncc(I)c3n2)=O)C1 C1(C(=O)NCC(c2ccccc2)NC(C(C2CCCC2)OC)=O)CC2CC2C1 c1(C(=O)N)ccc(F)c(F)c1.C1(CC)CCCN1C(=O)C(c1ccc(Cl)cc1)=O C(=O)(C1=CC2(CCOCC2)C1)N.c1(OC)cnc(C(=O)NC(C)CC(C)C)nc1 c1(C(N2C(C)(COC)CCC2)=O)cc2c(nn1)CCOC2.c1(C(=O)N)cnc[nH]1 c1(NC(CCN(C(C=C(CC)CC)=O)C(C)C)=O)cc(Cl)ccc1C C#CCC(CC#C)NC(C1CCCCN1C(=O)C(CC)n1cncn1)=O CC1CN(C)CCC1NC(C1C(C)OCCN1C(C1CCC(O)CN1C)=O)=O N1(C(C(C2CCOCC2)OC)=O)CCCC2(C1)CN(C(=O)CN=S(C)(C)=O)C2 N1(C(=O)Nc2nccc(COC)c2)CCC(C)C(c2ccc(O)cc2)C1 c1(C(=O)NCCC2(OC)CN(C(=O)CO)C2)cc2ccc(F)cc2s1.CCO c1(CCC(N2CC(OC)C(NC(C3COC(=O)N3)=O)C2)=O)nc2ccccc2o1 C(CC(CC)C(=O)NCCC1CN(C(c2cn(C)nc2Cl)=O)C1)=CC CCCC(C(=O)N1CCC(C)C1c1cn(C2(C(N)=O)CC2)nn1)N(C)C c1(CC2CC3CN(Cc4cc(OCC)ncc4)CC3C2)c(Br)ccc2c1OCO2 N1(C(C(C)SC(C)C)=O)CC2(C)CC1(C(=O)NCC13CCCC1CCC3)C2 C(c1scnc1C)=CC(=O)N(CCCNC(c1cc(C(C)=O)sc1)=O)CCO c1(OC)nc(C(N2CCN(C(=O)CN(C)C(c3cccs3)=O)CC2)=O)cc(O)n1 C1(NC(c2ccc(SC)cc2)=O)CCN(C(=O)CC23COCC(C2)C3)CC1C C1(C(=O)NC23CCC2CN(C(=O)CN2CCCC2)C3)CCC2(CCOCC2)C1 N1(C(C2N(C(CNC(=O)Cc3ccccc3)=O)CCOC2)=O)CCC(O)C(O)C1 C1(C(N(CCCC=C)C)=O)CCN(C(=O)Cc2csc(C)n2)C1CC N1(C(C=COCC)=O)CC(NC(=O)CN2CCN(C)CC2)C(C)(C)C1 N1(C(CC2(C(=C)F)CCC2)=O)CCCCC(C(=O)NCCC(O)CC)C1 c1(OC)ccnc(CNCC2CC(C)(C)CN2)c1 Cc1ccc(C#N)cc1S(=O)(=O)N1CCN(C(=O)CN(C)C)CC1(C)C C(=O)CCCCC(F)(F)F.c1(C(=O)OC)cn(CC(=O)NC2(C)CCC2)cn1.N CCCCCS(=O)(=O)CC(=O)NCc1cccc(NC(=O)CCSCCC)c1 Cc1cc(Br)cc(C(N2CCN(C(c3c[nH]nc3F)=O)CC2)=O)c1C C1(CNC(c2ncc(CC)nc2)=O)N(C(C2COCCN2C)=O)CCCC1(C)C N1(C(C2C(C)CCCC2)=O)CCCN(C(c2cnnc(C3CC3)c2)=O)CC1 c1(C(=O)NCC(CCNC(C(CCSC)OC)=O)O)c2c(nn1C)CCC2 Cc1cccc(C)c1CC(=O)NC1CC12CC(NC(=O)Cc1cn(C)nc1C)C2 c1(NC)ccc(C(=O)NCC2CC(NC(=O)OC(C)(C)C)CO2)cc1N C(C)(CO)(C(F)F)NC(c1cc(CNC(C2CCN(C)C2)=O)[nH]n1)=O c1(C(=O)NCCC2OCCN(C(CS(=O)(=O)NC)=O)C2)ccc(C#N)c(O)c1 c1(C(=O)NCCCCC(C)NC(=O)C(C)C2CC2)cn2cccc(F)c2n1 C1(C(C)NC(c2c(C)noc2)=O)CN(C(c2c(C3CC3)noc2C)=O)CCO1 C#CC1(C(=O)NCC23CC2CN(C(C2COCCN2CC)=O)C3)CCCC1 C12(CNC(=O)CCN(C(c3ncccn3)=O)CC3CC3)CCC(CO1)C2 N1(C(C2(n3cc(-c4ccsc4)nn3)CC2)=O)CCCC1CC(F)(F)F C1(N(C(c2c(CC)con2)=O)C)CCCN(C(c2csc(CC(F)(F)F)n2)=O)C1 CCCCC(CNC(=O)C=Cc1cccnc1)NC(c1ccccn1)=O C(=O)(CC(CC)CC(C)C)NC(CCC#C)C(=O)NCCCS(C)(=O)=O C1(C(=O)NC(c2cn(Cc3ccncc3)nn2)(C)C)CC1C1CCCC1 c1(C(=O)N)cc(S(N)(=O)=O)ccc1F.CCC(C)C=CC(=O)N(CC)CC CCC(C)(C)CC(=O)N(C)CCNC(=O)C(CC1CCCC1)C(C)C N1(C(c2c(CCC)n[nH]c2)=O)CCC(NC(c2ccc(O)cc2)=O)C(C)C1 Cn1nc(NC(=O)C(=O)NCC2CCCCC2O)c2nccnc12 c1(OC)ccc(C(N2CCCC(CNC(=O)C(C)OC)CC2)=O)nc1OC c1(C(=O)O)cc(F)c(C(=O)Nc2cnc(Cl)cc2C=O)c(F)c1.c1cnc[nH]1.N C(=O)(CCCc1nc(C(C)(C)C)no1)NCCN(C(=O)C(F)C1CC1)C Cc1cc([N+](=O)[O-])cnc1C(=O)NCCCCCNC(=O)CCCN1CCCC1 C(C(COC)C(=O)N1CC(OC)CC1C(=O)NC(c1c(C)noc1C)C)OC N1(C(c2ccc(CC)o2)=O)CC2CC(NC(c3ccc(F)cc3F)=O)CC1C2 c1(CN(CC(=O)O)CCn2ccc([N+](=O)[O-])n2)cc(Br)ncc1Br c1(C(=O)NC)ccc(CNC(=O)NCc2cccnc2N2CCCCC2)cc1 C1(NC(=O)CCN2CCOCC2)CC2CN(c3nnc(-c4ccon4)s3)CC12 c1(C(C)(C)C)cc(Br)cc(CN2CCC(COCCO)C2)c1O N1(C(CCN(C(Cc2nc(C)sc2)=O)CCO)=O)CC2CC3CC2C1C3 c1(OCCC)cc(F)ccc1NC(=O)Nc1cc(Cl)nc(C2CCCO2)n1 C#CCC(C(=O)NCc1ccccc1C)C1CC1.N1(CC(=O)N)CCNC1=O C#CCC(CC(=O)NCc1conc1C(C)C)NC(=O)C=Cc1cc[nH]n1 Cc1cc(C(=O)NCC(C)N(C(=O)C(C)N(CC(F)(F)F)C)C)cc(C)c1C#N C(c1cccnc1)=C(C)C(=O)NCC(O)CNC(c1ncccc1N)=O c1(OCC)sccc1C(=O)NCCN(C)C(C1CC1(C)Br)=O N1(C(C2N(Cc3ccc(OC)cc3Cl)CC(C)C2)=O)CCc2nc[nH]c2C1 N1(C(C(C)O)=O)CCC(C2CC2NC(=O)Cc2ccsc2Cl)CC1 Cn1cncc(C(N2CCC(C(=O)NC3C4CCC3CC4)CC2)=O)c1=O C(C)(CC(=O)N1CCC2(CCO2)C1)(C(F)(F)F)N(C)C c1(C(=O)NCC(CN(C(C(C)OCC#C)=O)CC)(C)C)cnnc(C)c1 c1(C(N2CCC(NC(C(C)SCCCC)=O)(CO)CC2)=O)c(C)cc(O)nc1C c1(CC(=O)NC(CCCNC(Cc2cn(CC)nc2)=O)(C)C)ccc(O)cc1F C(=O)(C1=CC2(CCN(C(c3n[nH]cc3Cl)=O)C2)C1)NC(c1n(CC)ncc1)C c1(C(N(C(C)CNC(=O)CCc2ccnn2C)C)=O)cc(S(C)(=O)=O)ccc1Cl Fc1cc(C(F)(F)F)cc(-c2noc(C3CCCCNCC3)n2)c1 N1(CCC(CC)C)CCC(C)S(=O)(=O)CC1 C1(C(N(CC(C)CNC(c2cnco2)=O)C)=O)CC2CC2C1 C1(C2CCCC2)(C(=O)NN2CCN(Cc3ccccc3)CC2)CCNC1=O C1(N(CCOC)C(c2cnc(C)[nH]2)=O)CCN(C(=O)CC(F)F)CC1 n1(C(CC)CC)nc(C)cc1C(=O)Nc1cccc(Cc2nccn2C)c1 C1(NC(C2(C)CN(C(=O)CC3CC(=O)C3)C2)=O)CCCN(C(N)=O)C1 C1(CNC(C=C(CCC)C)=O)CCN(C(=O)CCC(N)=O)CC1(F)F c1(C(N2CC(C)C(NC(C3(Cl)CC3)=O)C2)=O)cnn2c1S(=O)(=O)N(C)CC2 C1(C(N2CCCC(C)(NC(C3CC3CF)=O)C2)=O)CCn2c(O)nnc2C1 CC1(C)CCC1C(=O)NCCOC1CCN(C(=O)CC2CC(F)C2)C1 c1(C=O)cccc(-n2cccc2)c1.CCCCN(C(=O)CCC1(C)CC1)CC.N C1(NC(c2n(CC)ncc2)=O)CC2CC(C1)N(C(c1cc(Br)cnc1N)=O)C2 CC1(NC(C2COCC2C(N)=O)=O)CC(NC(=O)Cn2cnc(=N)[nH]2)C1 N1(C(C=CC=O)=O)CCCC(N(C(C2CCC3CC23)=O)CCC)CC1.C1CC1 CCCC(C)CC(=O)N(C1CCCN(C(c2cc(C)nn2CCO)=O)C1)C c1(C(=O)NC(CN2CCN(C(c3c(C)ccs3)=O)CC2)C)ccc2ccsc2c1 CN1CCCC(CCC(=O)N(C)CCC2CCCCN2C(C23CCC2CC3)=O)C1 C1(OC)CC(O)C1NC(c1[nH]ccc1CNC(=O)C(C)(C)OC)=O C(COC(C)C)(C(=O)NCC)NC(COC)=O.c1(C(=O)N)cn[nH]c1 C(=O)(N=c1cc(-c2cncc(C)c2)o[nH]1)NCC(C)N(CC)CC c1(CCC(=O)NC2(CNC(CC(C)c3ccco3)=O)CCOC2)cccc(O)n1 C1(CNC(c2c(C)c(C3CC3)on2)=O)COC(C)(C)CN1C(C1CCCS1)=O C=CCC(C)(C(=O)NCCCC(C)NC(=O)COC1CCOC1)N(C)C C(=O)(C(C(=O)NC1CN(C(=O)CCc2ccncc2)C1)OC)OC C#Cc1cccc(NC(C2CC(NC(c3cnnc(O)c3)=O)C2(C)C)=O)c1 c1(C(=O)NCCCCNC(c2ncc(C)nc2)=O)cnc2n1C(C)CCC2 c1(OC)cccc2c(N(C)CCN(C)C(c3cnn(C)n3)=O)ncnc12 c1(OC)cc(C(=O)NC2CCC2)cc([N+](=O)[O-])c1Cl.c1(CC=O)nncn1C.C C1(N(C(C)=O)C)CCC2(CC1)CCN(C(=O)CC)C2.C(C)OCC.C(C)=O.O N1(C(C2(COCC)CC2)=O)CC=C(CCNC(C2SCCC2C)=O)CC1 n1(CC(N2CCC(NC(=O)C(c3ccc(Cl)cc3)O)CC2)=O)cnc([N+](=O)[O-])c1 CCCC(C(=O)N1CC(O)(C(C)NC(=O)CC(CC)C2CC2)C1)S(N)(=O)=O Cc1c(Cl)cc(C(N2CCC3CN(C(=O)CC4(O)CC4)CC23)=O)cc1Br C1(NC(C(CCC)N(C)C)=O)CN(C(=O)CCn2ccnc2C)C2(CCCC2)C1 C1(N(C(Cc2c(CC)noc2CC)=O)C)CCCCN(C(c2ns[nH]c2=O)=O)C1 c1(C(=O)OCC)cnccc1N1CC(CO)C1.C(=O)(CC)N.[SH](C)(=O)=O c1(CC)cc(C(=O)NCC(=O)N)no1.C1CCC(=O)O1.c1cn[nH]c1.C1CC1 c1(C(C(=O)Cn2cccn2)=O)ccc(C2CC2)o1.CCO c1(C(N(CCCN(C)C(c2ccsn2)=O)C)=O)ncc(Cl)cc1F c1(CC(=O)NCC2C(NC(Cc3c(C)non3)=O)CCC2)c(F)cccc1F c1(C(N(CCC(C)NC(c2cc(CC)c(C)s2)=O)C)=O)cccc2[nH]ncc12 N1(C(c2n(CCC)ncc2)=O)CC2(CCC(CNC(=O)C)O2)C1.C(=O)N CC(C)C(CC)NC(c1ccnn1C(C)(C)C)=O.C(c1ncc[nH]1)=CC=O.N c1(C(=O)NC(CN(C(COCC=C)=O)C)C)nc(CC)oc1C c1(C=O)ccc(C)cc1[N+](=O)[O-].C(CC(C)(C)C)NC(C(C)(C1CC1)OC)=O c1(OC)ccc2c(C(=O)NC3CC(NC(=O)C)C3)cnn2c1.c1cc(C)no1 N1(C(C(N(C(C2(OC)CCSC2)=O)C)C2CC2)=O)CCC2CC1C(=O)N2C N1(C(=O)OCC)CCCC(N(c2nnc(CC(C)C)n2C)C)C1.c1ccn(C)n1 C(=O)(C1=C(c2ccc(Cl)cc2F)N(C2CC2C)C(=S)NC1c1nc(Cl)cs1)OC C1(C(N2CCC(NC(CC(CC=C)(C)C)=O)CC2)=O)CC2(CCCCC2)CO1 C(=O)(CCC1=CCCCC1)N1CC(NC(C2CCC(CCCC)CC2)=O)C(C)C1 C1(OC)CN(C(=O)Nc2ncc(C)c(O)n2)C2COCC12 c1(CC(=O)NC2C(NC(CCNC(=O)OCC)=O)CC2)cnccn1 C1(CC)CN(C(=O)CC23COC(C)(C2)C3)CCC1N=c1[nH]c(Cl)ncc1C(C)=O n1(CC(=O)N(CCC2CN(C)C2)C)cc(Cn2cncn2)nn1 C(=O)(C1CCCc2scnc21)NCC1CCN(C(c2cn(C)nn2)=O)CC1O C(=O)(CC(C(F)F)n1cccn1)NC(CCNC(COCC(=O)NC)=O)C C1(C(OC)OC)CCCCN1C(=O)Cc1ccc(Br)cc1 c1(C(=O)NC(CNC(c2c(C)ncnc2O)=O)C)cn(C)c(C)cc1=O C=C1CC(C(=O)NCC(C)OCCO)(CNC(=O)C(c2ccnn2C)C)C1 Cc1sc(C(c2nnnn2C2(C)CC2)NC(c2ccc(Br)cc2)C(N)=O)cc1Br c1(CCC)occc1C(N1CC(F)(CNC(c2cnc(CC)s2)=O)C1)=O C1(NC(=O)C=CC(F)F)CCCC1NC(=O)CNC(=O)C1CC1 C1COC(C)(C)CN1C(=O)C=Cc1cocn1.CC1=NNC(=O)C1CC(=O)N CC(CF)CC(=O)N(CC(N1CCN(C(=O)CSCc2ccncc2)CC1)=O)C C(=O)(C#CC1CCCC1)NC(C(N1C(C)C(O)CC1)=O)(C)C1CCC1 C1(O)(C=O)Cc2ccccc2C1.CC1(C)C(C(N2CCC2C)=O)CCS1(=O)=O.N c1(C(N2CC(NC(c3n(C)ncc3)=O)C(F)C2)=O)ccc2c(c1O)CCCC2 C1(CC)(CC)Oc2ccc(NC(=O)CN3CCN(CCCF)CC3)cc2O1 C(CCCCCC)(C(=O)OC)CNC(CNC(COCCC=C)=O)=O c1(C(N2CC(C(=O)O)C(c3cn(CCCCO)nn3)C2)=O)cccc(I)c1 N1(C(=O)CC2CCCCO2)CCC2(CCCN2C(=O)C(F)C2CC2)CC1 N1(C(COCCCCC)=O)CC(O)C(O)C1CNC(=O)CC1CC=CCC1 c1(C(=O)NC(CNC(CC(=O)NCC#C)=O)CO)ccc(C=NOC)cc1 N1(C(C(OCC)OCC)=O)CCC(O)CC1C(N1CCCCC1C(=O)O)=O C12(C(=O)NC3CC4CN(C(c5nc(C)n(C)c5C)=O)C3C4)CCC(CC1)C(C)O2 c1(CC)cc(F)ccc1C(=O)NC1COCCN(C(=O)CCc2cnoc2)C1 CCC(CC)(C(=O)NC1CC2(C1)CC2C(=O)NC1CCCC2(C1)N=N2)OC C1(O)(CN2CCCC(CS(C)(=O)=O)CC2)CCNC2(CC2)C1 N1(C(CSC(C)(C)C)=O)CC2COCC(C1)C2NC(C1C2CCCCCC12)=O C(=O)(C(O)C(F)(F)F)N(CCNC(CC1(C#N)CC1)=O)CC1CC1 C1(NC(C2C(C)C2)=O)C2CC3CN(C(C4CCCC4c4nc(S)n[nH]4)=O)C1C3C2 c1(C(=O)NCC(CC)(C)NC(=O)CCCO)ccc(C)c([N+](=O)[O-])c1.CC CC1(CO)CC2(CCN2S(=O)(=O)CCC2(C)N=N2)C1 C(=O)(CC(C)(O)C(F)(F)F)N1CCOCC(NC(C(C(C)(C)F)(C)F)=O)C1 C1Cc2cc(Br)ccc2O1.N1(CCNC(=O)NC)CC2(C1)CN(C1CCC1)C2 C1(NC(CSCCOC)=O)COCCC1.c1(C(=O)N)cccnc1-n1cncn1 c1(CNC(C2CNC(=O)N2)=O)ccc(C(N2CCCC(CCF)C2)=O)cc1 C1(N(C)C(C2CC2CF)=O)CN(C(c2cc(C(F)(F)F)cs2)=O)CC12CC2 c1cccc(Cl)c1C.C(=O)(CCC1(C)CC1)NCCN(CC=O)CCOC c1(CN2CCCC(C)(C(=O)NCCc3ccccc3F)C2)nc2ccccc2[nH]1 N1(C(CCC=C)=O)CC(C(=O)N(C(CC)CO)C)CCC1(C)C C1(C(C(=O)NC(CSC)C)NC(=O)C(F)n2ccnc2)CCCCC1 C1(CNC(CNC(C)=O)=O)(NC(=O)Cc2cn[nH]c2)CC(F)(F)C1 c1(C(=O)NCC(CNC(CCC(CC)OC)=O)(C)O)ccn2cncc2c1 C=Cc1ccc(C(N2CCC(NC(c3ccc(CSC)o3)=O)C3CC23)=O)cc1 CN1CCCCC1CCC(=O)NCCCNC(C1CCCN(C(=O)N(C)C)C1)=O N1(CC(=O)NCC(C)N(C(=O)C2=CCSC2)C)CCC(OCC(F)F)CC1 c1(OC)ccc(NCC2COC3(C)CC2C3)cc1S(=O)(=O)N(C)C C#CC1(C(N2CCCOC(C(C)C)C2)=O)CCN(C(=O)Cc2ccc(C)nc2)C1 CC(C)CC(CN(C)C)NC(=O)CC(C)NC(=O)CCCn1ccnn1 C1(c2ncc(C(N3CC(O)(CCNC(CCC#C)=O)C3)=O)[nH]2)CCCN(C)C1 CC1OCCC1(C)C(=O)Nc1cccc(NC(=O)CCc2ccccc2O)c1 N1(C(c2cc(C)no2)=O)CCC(F)(C)C1.C1(C(=O)N)CC(C)(C(C)(C)C)C1 C(CC(C)C)(C(=O)N)NC(C1C(C(=O)OCC)C1)=O.c1cc(O)ncn1 Cc1ccc(CCC(=O)NCC(C)CNC(C2(CCF)CCC2)=O)cc1 c1(CC(=O)Nc2n(C)c(=O)ccn2)cc(F)ccc1Br c1(OC)ccc(CC(N2CCC(OCC)C2)=O)cc1F.C(=O)C(C)CN(C)C.N c1(C(N2CCN(C(C(C3CCC3)OCC)=O)CC2)=O)ccnc(C)c1O Cc1ocnc1CCNC(=O)CC1CC(NC(=O)CN2CC=CC2)C1 C1(F)(CNC(=O)C(C2CCCCC2)O)CCN(C(C2Cc3nccn3C2)=O)CC1 C#Cc1ccc(C(=O)NC23CCN(C(=O)CNc4cccnc4)CC2C3)cc1 C1(CNC(c2c(C)[nH]nc2CO)=O)CCN(C(=O)COC2CCOC2)CC1O N1(C(c2ccc(OC)cc2Cl)=O)CCC2(CC1)OCCC2NC(=O)C1=CCCC1 C(=O)(C(F)C(F)(F)F)N1CCC(NC(c2cccc(OC)n2)=O)C1C N1(C(c2c(C)c(Cl)ccc2)=O)CC(C)C(N=c2ccnc(Cl)[nH]2)C1 CCC(C(C)(C)O)NC(C1COCC1NC(C12CCN(CC1)C2)=O)=O C#CC1(C(=O)NCC2CNC(=O)C2)CCN(C(=O)CCCCCC#N)CC1 C1(O)(CCNC(C(C)Cc2cnc[nH]2)=O)CCN(C(=O)CCc2cncs2)C1 c1(C(N2CC(F)CC(NC(C(COC)(C)C)=O)C2)=O)cc([N+](=O)[O-])cc(C)n1 c1(NC(N2C(CNC(=O)Cc3ccco3)CC2)=O)cc(Cl)ncc1Cl C#CC1CN(C(c2cc(CNC(=O)C(C)CC3CCC3)[nH]n2)=O)CCN1C c1(CCC)cc(C(=O)NCCC2CN(C(C3(C)CC3)=O)C2)n[nH]1.C1CCC1 CC(C)CCC(O)C(=O)N1CCC(=CCNC(C2(c3ccccc3)CC2)=O)CC1 c1(C(N(C)CC2N(C(C(=Cc3cn[nH]c3)C)=O)CCC2)=O)csc(C)c1N c1(C(N2C(CN(C(C3N(C(C)=O)CCC3)=O)C)CCCC2)=O)ccc(C)c(N)c1 C1(C(N(C2C(OC)COC2)C)=O)CN(C(=O)C(C)=CC2CC2)CC1C C(=O)(CC1=NNC(=O)C1)OCC(C(C)C)C(=O)OC(C)(C)C c1(C(C=O)(F)F)ccc(F)cc1C.C(CC)N(C(C1CC1)=O)CC.C(C)=O C(C(C)(CO)CO)N(C)C(C1(CNC(C2CCC2C)=O)CCCC1)=O c1(C(=O)NC2C(CNC(C(COC)C)=O)CCC2)cccc(SC)n1 c1(C(N2C(C)C(NC(C3(C)CC3(F)F)=O)CC2)=O)cc([N+](=O)[O-])cn1C Cc1nc(C)n(O)c1C(N1CCCC1CN(C)C(c1cnnc(O)c1)=O)=O CC1CCc2ccccc2N1CCO.C123CCN(CCCC1C2)CC3=O CC(CC(=O)NC1CC2CN(C(C3CC4CC4CC3C)=O)CC12)C(F)F CC#CCCC(=O)N1CC2CC2(NC(c2cnn(-c3ccccn3)c2N)=O)C1 N1(C(C2(C=O)CC2C)=O)CCC2(C1)CN(C(=O)CS(=O)(=O)C(C)C)CCO2.C C1(NC(CC2(C=C)CCCCC2)=O)CN(C(=O)C(C)CF)CC(C)(C)C1 c1(NC(c2scc(C)n2)=O)ccc2c(c1)CN(c1ncnc3c1CCCC3)C2 Cc1c(C(=O)N)cccc1C#N.C1(N(C(C23CC(C2)C3)=O)C)CCC2(CC1)CC2 c1(OC)ccc2c(ccn2CC(=O)NC2CN(C(=O)C(O)C3CC3)CC2O)c1 n1(CC(=O)NCC2(NC(c3[nH]cc(C)c3)=O)CCC2)cnc([N+](=O)[O-])c1 C1(C(=O)NC2(C3N(C(C(C)C4CCCC4)=O)CCC3)CC2)CCC2CC1C2(C)C N1(C(CC)(C)C)CCN(C(C2CC=CCC2)C(=O)NC2CCOCC2)CC1 c1(CC=O)coc2ccc(C)cc12.C1(COC)(C)CN(C(c2ccsc2)=O)C1 c1(C(=O)NC2CCC(CCNC(CCCC#C)=O)C2)ccc(Br)cc1O CC#CCC(C(=O)NC(C(=O)OC)C1CC1)NC(=O)CCCOCC C12(NC(c3cnc(Cl)s3)=O)CCN(C(c3nn(C(F)F)cc3Cl)=O)CC1C2 C1(NC(CSCC#C)=O)CN(C(=O)C(C)OCCN(C)C)CC12CCOCC2 c1(C(C(=O)N(CCCN(C(C(C2CCC2)OC)=O)C)C)O)cccc(C)c1 CCC(N)(C(=O)NC(Cc1ccccc1)C(=O)N1CCCCC1)c1ccccc1 CC1CCC(N=c2[nH]c3c(c(=NCC4(n5ccnn5)CC4)[nH]2)CCC3)CC1 N1(C(C(CC)CC2CCCC2)=O)CCN(C(c2cc(OC)n(C)n2)=O)CC(C)(C)C1 c1(C(=O)NC(CCCNC(CCN(C)CC)=O)C)cc(F)c(F)c(OC)c1F C=CCC(C)(CNC1(c2nnnn2CC2CCCO2)CC(C)(CO)C1)CO C1(COCC)CCCN(C(C2(C)CCN(C(=O)C=C(C)CO)C2)=O)C1 CC1(C)OCC2CC12C(=O)NCC1CCCC1NC(c1cnco1)=O Cc1ccc(-c2nc(COCc3ccccc3)nn2CCN2CCCCC2)n1C c1(OC)ccnc(OC)c1C(N1CCC(C)C(C)C1)=O.C(=O)(CCC(F)(F)F)N Cc1coc2c(C(=O)NC3CC(N(C(=O)Cn4cnnn4)C)C3)cccc12 N1(C(Cn2nnc(C)n2)=O)CCc2nc(CNC(c3cnn(C)c3F)=O)sc2C1 Cc1ccc(C(N2CC(NC(c3cnc(C(C)C)[nH]3)=O)CCC2C)=O)c(N)c1 C(C(C)(C)C=C=C(C)C)(c1nnnn1CC(F)F)NC(CCC)C(N)=O N(C1CCOc2ccc(Br)cc21)C(c1c(Cl)ccc(C(C)C)c1)=O c1(C(=O)NC(C)(C)C=CC(=O)NCc2ccncn2)c[nH]nc1Cl C(C)(C)(CC(=O)NC1CCN(CCO)CC1)N(C(=O)Cn1cnc(C#N)n1)C CCC(O)C(F)(F)C(=O)N1CCC(CCNC(=O)CCC(C)(C)C)C1 c1(C(N2CCC2(C)C)C(=O)Nc2cccc(OC)c2)ccc([Si](C)(C)C)cc1.C C(CC1=CCN(C(=O)C(C)(C)CCCO)CC1)NC(Cc1c(C)nccc1)=O C=CCCCC(C(=O)N1CCC1C(C)C)NC(c1ccc(O)c(C)c1)=O CCCCC(O)CNC(=O)CN(C(=O)C(C1CC1)C1CC1)C1CCC1 C1(F)(C(N2CC(CC)C2)=O)CCN(C(=O)C(C)OC)C1 c1(C(=O)NC2C(CNC(c3cc(C)nnc3)=O)CC2)ccc(C#N)c(F)c1 N1(C(c2cccc(C#N)c2)=O)CC(NC(=O)CCc2cscn2)C2CCCCC12 c1(OCC)ccc(OC)cc1C.C1(c2nnnn2CC)C(C)(C)OCCN1 C1(C=O)CS(=O)(=O)CC12CC2.Cc1ccnnc1C(=O)NC.C1(C)CCCC1 O=C(C1CCCc2ncccc21)NC12CCC1CN(C(=O)CCc1ncc[nH]1)C2 c1(N2CCN(C(C3C(C)=CCC=C3)=O)CC2)ncc(C(F)(F)F)cc1Cl CC(F)(C=O)C(C)C.C1(CCC)(C(=O)N)CC(=O)C1.C(C(C)(C)O)C1CC1 N1(C(c2cc(C)no2)=O)CC2CC(NC(C3CCN(CC(F)F)CC3)=O)C1C2 c1(NC(C(C)(C)NC(=O)C2=NOCC2)=O)cnc2ccccc2c1 N1(C(Cc2c(C)noc2C)=O)CCC2(CC(C(=O)N)C2)C1.C1(C(N)=O)CCOC1 CN1CCS(=O)(=O)CC1CC(=O)NC1CN(C(c2ccc(Cl)cn2)=O)CC12CC2 C1(NC(CCN(CC=C)C(C2CC2F)=O)=O)CCC(CCO)CC1 C1CC2(C1)CC(C)(C)C2.Cc1cn(C)nc1C(=O)NC(CN(C)C)C=O.N c1(CC)ncncc1C(=O)NC(CNC(c1oc(CC(C)C)nc1C)=O)CO c1(C(N2C(C(N(CCCCC)CCO)=O)C(C)C2)=O)cc2ncccc2[nH]1 C1(CCNC(CC2ON=C(C)C2)=O)CCN(C(=O)CCc2cnn[nH]2)CC1(F)F Cc1cnc(C)c(C(=O)NC(C)CN(C)C(C2(O)CCOC2)=O)c1 CON(C(=O)c1csc2nc(C)cn12)C1CCCOc2cc(C)ccc21 c1(OC)c(-c2csc(NC(=O)Nc3cnnc(O)c3)n2)cc(F)cc1F Cc1ccc(-n2cc(C(CC(N)=O)NC(C3(C)CC3(C)C)=O)nn2)cc1N N1(CCNC(Cc2cc(CC)no2)=O)CCN(C(=O)C(c2ccccc2)F)CC1 C(=O)(CC(C(F)(F)F)N(C)C)N1CCC(N)(COC)C1 C(CC(C(=O)NC1COCCC1)NC(N)=O)SC.c1(C=O)c[nH]cc1C1CC1 N1(C(C2CCCN(C)C2)=O)CCOCC(C(N2CCSC2(C)C)=O)C1 N(C(=NCC1CCCS(=O)(=O)C1)N1CCN(S(C)(=O)=O)CC1)Cc1cc(C)on1 c1(C(N2CC(n3cc(CCN(C)C)nn3)(C(=O)OC)C2)=O)nn(C)cc1C CC(C)(CC(=O)NC1CCN(C(c2cnn(C3CC3(F)F)c2)=O)CC1)C(F)F N1(C(=O)C2=CCCC2)CCC2C(CCCN2C(=O)CCc2cnn[nH]2)C1 Cc1ccc(C(N2CCCC2C(=O)NCCCCNC(N)=O)=O)c(F)c1 C1(C(C)(C)C)COCCN1C(=O)CCO.c1(C(N2CCC2)=O)cn(C(F)F)cn1 C(=O)(C1=NOC2(CCC2)C1)NCC1N(C)CCN(C(=O)C(O)c2ccco2)C1 Cc1noc(C)c1CC(=O)NCCCCNC(c1ccc(C2CC2)s1)=O C1CCCN(C(c2csc(C(N)=O)n2)=O)C1.c1(CN(C)C)ccsc1C(=O)N CN1C(=O)CN(CC(=O)NS(=O)(=O)Cc2ccn(C)n2)C1=O N1(C(C(CC(CC)C)C)=O)CCC2(CC1)OCCC2NC(c1n[nH]c(C)c1C)=O C(=O)(NNc1ccc(F)c(Br)c1)NC(C)Cn1ccc(=O)cc1 N1(C(C(C(CC)C)O)=O)CC2CCC1CC2NC(c1ncc(F)cn1)=O CC1=C(CNc2ccc([N+](=O)[O-])cc2C(=O)N(C)C(C)C)S(=O)(=O)CCO1 C1(C(=O)Nc2cncc(Cl)c2)(NC(=O)CCOC2CCCC2)CC(F)(F)C1 N1(C(COCCC#C)=O)CCC(C(=O)NC(C)C(C)(C)CC)CC1 CON(C)C(=O)CNC(=O)CC1C=CCC1.C1(C=O)CCC(C(N)=O)C1.N CC(C(C(=O)NC1CCOCC1)N(C1CCCCC1C)C)C1CCCCC1 C=C(C)CC(C(=O)NC(COC(C)C)C(=O)NCC(n1cccn1)C)OC CC1CCCCCN1C(=O)COC1CC(NC(C2(C#N)CCOC2)=O)C1 C1(NC(Cc2nc(C(C)C)sc2)=O)CCCC12CN(C(=O)CN(C)C(C)C)C2 N1(C(Cc2cc(C)no2)=O)CCN(CC(N2CCCC2CC(C)O)=O)CC1 C(=O)(C(CC)C(C)C)N1CCC(OCC(C)C)C1.C1(C#N)(CC(=O)N)CC1 c1(C(=O)NC2(C#N)CCN(C(C(C(C)C)O)=O)C2)cc2cc[nH]c2cc1Cl CCCCCCC(=O)NCCCCCN(C(=O)Cc1cccnc1OC)C(C)C CC1OCCC1(c1nnnn1C1CC1)Nc1cncc(CN(C)C)c1 c1(OCC)ccc(C(N2CCCC2CNC(C2CCOCC2)=O)=O)cc1 c1(C(=O)NCC(C)C)c(NC(N)=O)cccc1F.C1(C)(C(=O)N)CCOC1 C1(COCC(N2CC(N(C(=O)CC3CC(F)C3)C)C2)=O)CCCOC1 C(=O)(C1CCCc2c[nH]nc21)NC1C=CC(CNC(c2ncccc2Br)=O)C1 C1(C)(CC)CCN(C(=O)C)C1.C(F)(C(=O)N)=CCC.C(=O)C.C(C)=O c1(C(=O)NC(CO)C(=O)NC(CC2CCCC2)CO)cccc(CO)c1 S(=O)(=O)(c1sc(C)c(C(=O)O)c1O)N1CCC(C(c2c(C)cccc2)O)CC1 N1(C(CONC(C(C)c2cnn(C)c2)=O)=O)CCCC2(CC2)C1 C1(CS(=O)(=O)NCc2ccc3cc[nH]c3c2)CCC2(CCOCC2)CO1 C(N=c1[nH]c(Cl)ncc1Br)C1(CNC(=O)C2=CCC2)CC12CCC2 C1(C(=O)NC2CN(C(c3csc(C4CCCCC4)n3)=O)C2)CC(O)C(F)C1 N1(C(c2c(F)ccc(NS(C)=O)c2)=O)CCN(C(=O)Cc2cnoc2)C2(CC2)C1 O=C1CC2(CCN(C(=O)CCC3(NC(C4CC45CCCC5)=O)CCCC3)C2)CN1 C1CN(C(=O)C=CC(C)(C)C)CC1(C)C.c1(C(C)C(=O)N)ccc(Cl)c(Cl)c1 C(=O)(C1COc2ccccc21)NCC1C(NC(=O)CCc2cccnc2Cl)C1 c1(C(N2CC(CN(C(=O)C=C3CCCC3)C)OCC2)=O)ccc(Cl)c(C#N)c1 c1(C(=O)NC2C(CCOC)C2)cc(CNC(=O)Cc2cnnn2C)cs1 C1(C(N2C(C)(C)C(NC(=O)CCC(N)=O)CC2)=O)CC2(CO1)CC(F)(F)C2 C=CCCCCC(=O)N(C)CC1(O)CCN(C(=O)CC2CC(C(C)(C)C)C2)C1 N1(C(Cc2c(C)noc2)=O)CC(NC(c2c(C)[nH]c(C)c2C)=O)CC(F)C1 O=C(C1=CCSC1)NCC1(F)CCN(C(C2CCO2)=O)C1 N1(CC)CC(C(N2CCC(OCC)C2)=O)CC1=O.c1(C(C(=O)N)O)ccccn1 c1(C(N2CC(OC)(C)C2)=O)cc(C2CC2)ccn1.C(C1CCC1)=CC=O.N N1(C(C(C(C)C)NC(C)=O)=O)CCN(C)CC1CNC(c1cnc(Cl)s1)=O N1(C(c2cncc(C(C)C)c2)=O)CC(CO)C2(C1)CN(C(c1cc(F)cs1)=O)C2 c1(CC)c(C(=O)NC2(C(=O)OC)CCSC2)cnn1C1CCCC1 C(c1ccccc1Cl)=CC(=O)NCC1CCCCC1NC(c1n[nH]cc1F)=O C(=O)(C(C)C(F)(F)C(F)F)NCCCN(C(Cc1c(C(C)C)con1)=O)C C1(C=O)Cc2cncn2C(=O)N1.C(=O)(C(C)CC(=O)N1CCC(C)(C)C1)OC.N C1(CC=C)(NC(c2cc(CCN)on2)=O)CCOCC1 CCC(CC)(CCNC(C1CCN(C)C1)=O)NC(c1ccc(COC)cc1)=O c1(NC(=O)OCC)ccc(Cl)c(C(=O)NC2CN(C)C(=O)O2)c1 C1(NC(c2ncc(OC)cn2)=O)CN(C(c2cc(C)co2)=O)Cc2ccnn2C1 N1(C(CC(CC)CC)=O)CC2CC(CNC(=O)C(C)CCOC)CC1C2 C(CCC(C(=O)N(C1CCCC1C#N)C)NC(=O)C(=O)NC(C)C)OC N#CC1(C(N2CCCCC(CNC(C3C4CCCC34)=O)C2)=O)CC2(CC2)C1 c1(C(N2CC(OCCNC(C(C)OCC)=O)C2)=O)cc(C)c(Br)cc1C Cc1nc(-c2ccccn2)sc1C(=O)OC(C)CNC(=O)Nc1ccccc1 C(=O)(C(O)CC(C)C)N(CCCCC)C.C1(C)(C(=O)OCC)CC1C(=O)N C=C1CCN(C(C2CC23CCC3)=O)C(C(=O)N(C)Cc2ccccn2)C1 C(=O)(CC(F)(F)C(F)F)N1CCOC(C(F)(F)F)C1.Cc1c[nH]nc1C(=O)N.C N1(C(C(C)(C)c2nn[nH]n2)=O)CC(C)(C(=O)O)C(F)(F)C1 C1(C(=O)NCC(CN(C(=O)CO)C)O)CCCN(CCc2ccccc2)C1 C1(NC(CC(CCC)O)=O)CC2(CCC(CNC(=O)C(=O)N)CC2)C1.C1CC1 C1(c2nnnn2C2COC2)(NC(CCC)c2ccco2)CCCCCC1 N1(C(c2ncnc(C)c2C)=O)CC2(CC(C(=O)NCCC3(C)CCCO3)CO2)C1 C=C(C)CCCC(=O)N(CC(CO)(CO)NC(c1cc(Cl)cs1)=O)C CC(C)CC(O)C(C)C(=O)N(CCCCC(N1CC2CCC(C1)O2)=O)C n1(CC#C)cnnc1C(=O)NCC#CC(=O)NCCCNC(=O)CC CCCC(C)C(=O)NCC1CCC(NC(C2CCC(CCO)CC2)=O)CC1 C1(C(c2ccccc2)CC)CCC(=O)N(CCCc2ccccc2C)C1=O c1(C(c2n(CCC3(C)CC3)nnn2)NCCCC(F)F)ccc(C#N)s1 N1(C(C(C)CBr)=O)CCC12CCN(C(c1ccc3cc[nH]c3c1)=O)CC2 C#CCC(C(=O)NCc1nnn(C)c1C(=O)NC)C1CC1.c1nnc(O)o1 c1(OC)cccc(CC(=O)NCCCCC(C)NC(C2OCCOC2C)=O)c1 C1(C(=O)O)CC2(CC(N(CC#N)CCO)CCS2)C1 Cc1[nH]nc(C(=O)NCC2CN(C(c3ncn(C)n3)=O)CC2C)c1[N+](=O)[O-] c1(C(=O)NC(CO)CO)cc(F)cc(Br)c1O c1(OCC)cc(F)ccc1Cn1cc(-c2ncc(OC)c(=N)[nH]2)nn1 c1(C(=O)NC(CNC(CSC)=O)CO)cc(C)cn2ccnc12 C(CCN(C)C(c1sc(Br)nc1C)=O)(C(C)C)NC(C1N(CC)CC1)=O C1(C)CCC(=O)N1C.C1(OC)CC(C(=O)Nc2cc[nH]n2)N(C(=O)C(Cl)Cl)C1 Cn1nnc2c1CC(C(N1CCCC(NC(c3csc(C(F)F)c3)=O)C1)=O)CC2 c1(C(N2CC(O)CC(NC(c3cc(OC)no3)=O)C2)=O)cccn2cc(C)nc12 Cc1scc(C(=O)Nc2cccc(N3CCN(C4CC4)CC3)c2)c1C1CC1 N1(C(c2cccc(OC)c2)=O)CCCCC2C1CCCN2C(=O)CSCC(C)C C(=O)(C(O)(CN(C)C)C(F)(F)F)NCC(CNC(C=NOC)=O)F C(=O)(C(F)C(F)(F)F)NC(CN(C)C)C(N1CCC(N2CCC2)CC1)=O c1(NC)snc(C)c1C(=O)NC1CCN(C(c2cn(C3CCCC3)nn2)=O)C1 N1(C(CC2(C)CCN(C(c3cnc(C)n3C)=O)C2)=O)CCC2C(C(N)=O)C2C1 N1(C(CC(COC)C)=O)CC2CC1CCN2C(=O)Cc1cnn(C)c1C Cc1cc(Cl)cc(Cl)c1OCC(=O)NCCCC(C)NC(=O)C(F)F c1(N(C(C(N2CCC(OCCO)C2)=O)=O)C)cc(Br)c(Br)o1.Cc1cnco1 N1(C(Cn2c(=N)scc2)=O)CCC2CCC(NC(=O)Cc3c(F)cccc3Cl)C1C2 N1(C(C2CC(O)(CC#C)C2)=O)CCC(C#C)(C(N2CCCC(C=C)C2)=O)C1 N1(C(C(C2CC2)NC(CCC(C)OCC)=O)=O)CC2CC(CO)C(C2)C1 c1(NC(C(CCOC)NC(c2ncccn2)=O)=O)cc(C)cnc1C C=CC1CN(C(=O)C(C)(C)SC)CC1NC(c1ncoc1C(C)(C)C)=O C1(C(=O)NCc2n(C)ncc2)CCN(C(c2ccc([N+](=O)[O-])o2)=O)CC1O CC1CN(C(C2CCCC(F)C2)=O)CCC1NC(c1cn(C)cn1)=O c1(CC(=O)NCCC2CC(NC(=O)C(O)C(F)F)C2)ccc([N+](=O)[O-])cc1Cl CC1(C)OC2(C(=O)NC3CN(C(c4ccc([N+](=O)[O-])o4)=O)CC3O)CC1C2 C=CC(C)C(C)C(=O)NCCCN(C(c1cnccn1)=O)C1CC1 N1(C(c2cnc(SC)n2C)C(=O)NC2CCOC2)CC(C)OC(C)(C)C1C C(c1ccc(C#N)cc1)=CC(=O)NCC(CNC(C(CCC)N(C)C)=O)C C(=O)(NN=c1[nH]c2cc(Cl)ccc2nc1Cl)C1(F)C(C)(C)C1(C)C c1(C(=O)NCC(CC=C)NC(=O)C(C(CC)CC)OC)ncn2ccccc12 C(c1nc2ccccc2s1)=CC(=O)NC(CC=C)CO N1(C(C2CCN(OC)CC2)=O)C2CCCC1CN(C(=O)C(C)CC1CCCC1)C2 c1(SCC(=O)NC2CCN(C(c3c(CC)ocn3)=O)C2C)ccsc1[N+](=O)[O-] c1(C(=O)NC2CC3C(NC(CC(C)c4ccco4)=O)C3C2)cc([N+](=O)[O-])c[nH]1 CC1CC(CNC(=O)CC23CCCN2CCC3)CN(C(=O)CC(C)(C)C2CC2)C1 N1(C(c2c(C)csc2)=O)CC2CC2C1C(N1CC(C)(C)C1C(C)C)=O CCCC(F)(F)F.c1(C=O)c(C)nn(C)c1C.C1(C(=O)N)(COC)C=CCC1 C1(C(=O)NCC2(NC(C3CCOC3)=O)CCCCC2)CCCC2(CCC2)O1 N1(C(C=CCN(C)C)=O)CCN(C(c2cccc(O)n2)=O)C2CC12 C1(C(=O)NCCC(C)NC(Cc2c(C)nc[nH]2)=O)CCN(CP(C)(C)=O)CC1 C12(C(=O)N)CCCC1CCN2C(=O)C=Cc1ccc[nH]1.c1(CC)ccc(C)nc1 CC(CCN=c1nn[nH]n1C)NC(c1c[nH]nc1S(N)(=O)=O)=O C(=O)(C1=CCS(=O)(=O)C1)N1CCCC(N(C(C(CCC)NC(C)=O)=O)C)C1 C(=O)(CCCCC(=O)OC)NC1CCN(C(C(CCOC)OC)=O)C1C c1(C(c2scc(CC)n2)c2nnnn2CC)ccc(N2CCCCCC2)cc1 N12CCCC1C2=O.c1ccccc1.S(S(C)(=O)=O)CC(=O)N(C1CC1)C.C c1(N(CC(=O)NC)C)[nH]c(=NC(C)c2nc(=N)[nH][nH]2)nc2sccc12 CCCCC(O)CC(=O)N(C)CC1COCCN1C(C1C=CCS1)=O C1(C(=O)NCc2cnn(-c3ccc(F)c(Cl)c3)c2)CCCNC12CCC2 c1(C(=O)NCC(CC=C)C(=O)N(C)CC2(OC)CCC2)cnc2ccccn12 Cc1cc(C(N2CCC(C(C)NC(c3snnc3C)=O)C2)=O)cc(C)c1O C(c1ccc(O)cc1)=CC(=O)NCCC1CCCN(C(=O)CC2OCCCO2)C1 c1(C(C(N2C(CNC(CC=C(C)C)=O)CC2)=O)O)ccccc1 c1(CCC(=O)NC(CNC(=O)CC2CCC(=O)N2)C2CC2)cccc(Br)c1 Cc1ccc(NC(=O)C(=O)NC2CCCC2)cc1.c1(C=O)cn(C)c(O)n1.C Cc1cc(C(F)F)oc1C(=O)NCC1CCCC1NC(=O)CC1CCOC1 C1(NC(C2C(CCC)C2)=O)CCC(C)CC1.C(=O)(C(O)CC1CCCCC1)N C1(C(=O)Nc2cn(C(C)C3CC3)nc2)CC2CCC(C1)N2C C1(F)CCCN(C(c2c[nH]nc2C2CCC2)=O)C1.C(C1CCCO1)=CC(=O)NC C1(N(C(c2cc(C3CC3)on2)=O)CC)CCCN(C(C2(F)CCCCC2)=O)CC1 c1(OC)nccc(C(=O)NCC2(F)CCC2)n1.c1(C(C=O)=O)cnn(C)c1 C1(CCNC(C2CCSC2)=O)(OC)CN(C(=O)C(C)CS)C1.c1ccccc1 N1(c2n(CC=CCl)nnn2)CC2C=CC1C(c1nc(C3CC3)no1)C2 C(CCCCCCCO)NC(C1C(NC(c2ccc(OC)c(C)c2)=O)C1)=O C(N=c1[nH]c(=NC)[nH]c(=NCCn2cc(Cl)cn2)[nH]1)C1(CCOC)CC1 c1(N2CC3(C(NC(CCCN=[N+]=[N-])=O)CCS3)C2)ncnc2sc3c(c12)CCC3 C(C(C)(C)C(=O)NC1CCN(C(c2cccc(C(=O)OC)n2)=O)C1)OCC O(N=C1CCCCCC1)CC(=O)NC1COCC1NC(C1(C2CCCO2)CC1)=O Cc1ccc(C(=O)NC2COCC2NC(C2(CC(C)C)CCC2)=O)c(N)c1 N1(C(=O)CO)CCn2nccc2C1.c1(-c2cn(C(C)C=O)nn2)ccc(F)c(Br)c1 C1(C(=O)N)CCc2cn(C)nc2C1.C(c1cncn1C)=CC(=O)N(C(C)C)CC C1(CC(=O)NC(C)CN(C(=O)C2=COCC2)C)CCC(C)(C)CO1 C12(C(=O)Nc3cc(C)ns3)C3CC1C1C(C(N4CCCC(O)CC4)=O)C3C21 N1(CC)CC(C(=O)N(CCCNC(C2C3CCCC23)=O)C(C)C)CCC1=O C1(NC(c2cc(C)c(O)nc2)=O)CN(C(c2cccc(=O)o2)=O)CC1N=[N+]=[N-] c1(C(N2CCC(N(C(=O)CCc3cnn(C)c3)C)C2)=O)cccc2ccnn12 C1CCCCN1C(=O)CC1CC(C)=NO1.C(=O)(C(=O)NC)NCCOC.C c1(NC(=O)NCC)csc(C(=O)OCC2CCCSC2)n1 C12(C=O)CC3CCC(CC(C3)C1)C2.c1(CC)nnsc1C(N1CC(O)C1)=O.C N1(C(CCc2nc(=N)[nH][nH]2)=O)CC2CCC1C(NC(=O)CSCc1cscn1)C2 C(=O)(C(C)C(C)C)NCC(CC(=O)OC)O.c1(CCC(=O)N)cc(C)[nH]n1 C1(CC=C)(C(=O)Nc2cncnc2O)CCCN1C(C1CC2CC2C1)=O Cc1cc(C)c(NC(C2CN(C(C3CCC(=O)N(C)C3)=O)CC23CC3)=O)c(C)c1 Cc1ccc2c(c1)C=C(C(=O)NC(C)CNC(c1cnn(C(C)C)n1)=O)CO2 CC(CNC(c1cc(C(N)=O)c[nH]1)=O)CC(=O)NC1CC(CO)(CO)C1 CC(C)CC(C)(C(N)=O)NC(C1CC(C)CN1C(c1cn(C(C)C)cn1)=O)=O C1(C(=O)NCC(N2CCOCC2)=O)CN(C(c2csnn2)=O)C2(CCC2)C1 CCCC(C)(C)C(=O)N1CC2CC2(CNC(c2coc(-c3ccccc3)n2)=O)C1 c1(C(=O)NC2C=CCN(C(c3ccc[n+]([O-])c3)=O)C2)cccc(O)c1Br C(=O)(CCC(C)(F)F)NC1(CNC(C2C(c3n(C)cnc3)C2)=O)CC1 Cc1oc(Cl)nc1C(N1CCC(N(C)C(c2cnn(C)c2)=O)C1)=O c1(C(=O)NC2C(NC(=O)Cc3cc(F)ccc3O)C2)ccc2nc(O)sc2c1 N1(C(c2ccc(C(C)=O)nn2)=O)CC(C)N(C(=O)CC2CCC(=O)NC2)CC1C C1(C=O)(OC)CCC(C(F)F)CC1.CC(C)CN(C(=O)CCc1ncco1)C.N c1(C(=O)N)cc(C2CC2)n(C)n1.C1(C(N2CC(CC)C2)=O)CCC(F)(F)C1 c1(C(N2C(C)CC(CNC(c3cc(Cl)c(Cl)n3C)=O)C2)=O)nnn2ccccc12 c1(OC)nc(NC(C2(C)CCCN(C(c3ccc(O)c(F)c3)=O)C2)=O)cc(O)n1 N1(C(c2cnc(OCC)s2)=O)CC(NC(=O)CC)C(CC(C)(C)C)C1 C1(CNC(CCCC#C)=O)CCC(C)CN1C(=O)CC1CC2(CCO1)CC2 C1(C(=O)NCCN(OC)C)CCCN(C(=O)CCC2CCC(=O)C2)C1 NC1C2CC3CC(C2)CC1(CNC(=O)Cn1nnc2ccccc12)C3 C1(CC)COCC1N=c1[nH]c(=NC)[nH]c(=NCc2cn3cc(Cl)cc(Cl)c3n2)[nH]1 C1(O)(C(=O)NCC2C(C)CN(c3ncncc3I)CC2)CCC(C)(C)CC1 C(C1CN(C(c2cc(Cl)cn2C)=O)CC1C(=O)NCCC)=CC.C(C)(=O)N Cn1cc(C(=O)NCC2CC2C)ncc1=O.c1ccc(F)cc1.C(=O)CC.N C(N=c1cc(Cl)nc(C(C)OC)[nH]1)C1(NC(CC(CC)OCC)=O)COC1 c1(CC)nc(C)c(CNC(C2(CC)CCCC2)=O)o1.c1(C=O)ccc(C)o1 c1ccccc1.C(=O)(C(C)OC)NCCN(C(=O)Cn1cccn1)CCC c1(OC)cc(C)c(C(N2CCC(NC(=O)Cn3cnnc3O)CC2)=O)c(F)c1 C1(NC(CC=CCC)=O)CCN(C(=O)CC(C)C(C)(C)C)C12CCC2 Cc1cc(C(=O)NCCN(C)C(C2CCS2(=O)=O)=O)cn1C(C)C C1(CC(=O)NC(c2ccnn2C)C(=O)NC(C)Cc2cccs2)CCCCCC1 N1(C(=O)NCC(C)(O)CC2CCCCC2)CCC2(C=CC2)CC1 c1(CC=C)ccccc1C(N1CC2CC2(NC(=O)CC(F)(F)F)C1)=O c1(C(=O)NCCC23CN(C(C(COC)C)=O)C(CC2)C3)cc([N+](=O)[O-])nn1C C1(CNCCOCCC(C)=O)CCC12CCOCC2 c1(-n2c(Cn3ncc(C)c3)nc(-c3cnn(CCO)c3)n2)cc(Cl)ccc1C C1(NC(C(C)(C)C)=O)CC(NC(c2cccc(N3CCOC3=O)c2)=O)C12CCC2 CC1CC(C(N2CC(O)(CNC(c3csc4nccn34)=O)C2)=O)CCN1C C1(N(C(=O)CC(C2CC2)C2CC2)C)CCCCN(C(=O)C(O)P(C)(C)=O)C1 C1(OC)(CNC(C2CCCC2)=O)CCOC1.c1(C=O)coc(C(N)=O)c1.N C1(C(=O)NCC(C)NC(=O)COCCN(C)C)CC(=O)N(C)C1 CCC(CC(=O)NCC(O)CNC(c1nn(C)c2ccccc12)=O)CC(F)(F)F C1(NC(Cc2n(C)nnc2)=O)CN(C(=O)C=Cc2ncc[nH]2)CC12CCOCC2 c1(C(C2CC2)NC(C(=O)NCCOC)=O)cnccc1.C(C)(C)C.O C1(CCCNC(C)=O)CCN(C(C)=O)CC1 Cc1ccccc1NC(=O)C(O)C1CN(C(c2cccs2)=O)C1 c1(C=O)ccc(S(N)(=O)=O)s1.N1(C(COCCOC)=O)CC(CC)C1.N c1(OCC)ccc(Cl)cc1S(=O)(=O)N1CCN(C2CCOC2)C(=O)C1 C(=O)(C(C)(C)CC(=O)NC(C)C(=O)NC1CC2C(C1)C2(F)F)OC c1(C(N2CCC(n3c(=N)nc(C)[nH]3)CC2)=O)cc2cc(Cl)sc2[nH]1 Cc1cc(Cl)ccc1C(=O)NCC1CN(C(=O)C(C)Cn2ccnc2)CC1(C)C c1(CC)c(C(N2CC(NC(C3CSC(C)=N3)=O)C(C)C2)=O)nnn1CC C#CCCCC(=O)N(C)CCNC(c1csnc1-c1ccccc1)=O c1(C(=O)NC2CN(C(C3CC(OC)C3)=O)CC2C(F)F)ccc(O)cc1Cl CCCC(CCCNC(C1(C)CC2CC2C1)=O)NC(c1ccsc1Cl)=O Cc1ncnc(O)c1CCC(=O)N(CCCCN(c1nccnc1C#N)C)C N1(C(c2ccn(CC)n2)=O)CC(NC(=O)CC2OCCC2(C)C)CC1C N1(C(CC(CC)(C)C)=O)CCC(n2cc(-c3cc(N)ccc3C)nn2)C(C)(C)C1 c1(C(N2CCN(C(CC(C)O)=O)C3C2COC3)=O)ccc2cc(O)ccc2c1 CC1CN(C(=O)Cc2cnns2)CCCN1C(c1cscc1C#N)=O CC1=CCC(C(=O)NCCCN(CCCCNC(c2nc(Cl)sc2C)=O)C)CC1 CC1CCN(C(C2(C)CC(C)(C)C2)=O)CCN1C(c1ccc(Br)c(O)c1)=O c1(-c2nc(C(C)O)nn2CC2CCCC2(F)F)cc2ccoc2cc1F Cc1ccc(C(N2CC(NC(c3ocnc3C3CC3)=O)CCC2C)=O)c(N)c1F c1(C(N2C(OC)COCC2)=O)cnc(-c2ccc(OC)cc2COC)c(OC)c1 c1(C=O)cc(C2(Cl)CC2)n(C)n1.c1(C(=O)OC)cc(C=O)no1.C1CCC1 c1(C(=O)N)cc2c(=O)[nH]c(C)cn2n1.c1(C(=O)NCC(CC)C)ccc(C)nc1 c1(C(N2C(C)CC(NC(=O)CCC(F)F)CC2)=O)cc2c(s1)C(C)(C)CCC2 CC1N(C(C2CCCN(C(=O)C(=O)Nc3cc(F)ccc3N)C2)=O)CCC1(C)C C1(NC(C(CSC)O)=O)COC2C(NC(c3ncsc3Br)=O)COC12 c1(CC)ccc(F)c(C(=O)NC2CC(F)C2)c1.C1(C=O)CCCS1(=O)=O.C N1(CC(=O)Nc2c(-n3c(C)cc(C)n3)cccc2)CCNC(=O)C1(C)C c1(C(=O)NCCCN(C(c2cc(C)nn2C(F)F)=O)C)cnc2n1CCC(C)C2 C(=O)(C(CCCC=C)NC(=O)C(F)C(=O)OCC)NC1(CC#C)CC1 C(=O)(C1=NOC(C)C1C)N1CC(C)CC(NC(Cc2cccc(C)c2C)=O)C1 C1(C(=O)NC2C(N(C)C)COC2)CC2CC1CC2.C1(C(=O)N)CC1.C1CCC1 C1(CNC(c2csc(-c3ccco3)n2)=O)CCN(C(c2cc[nH]c2)=O)CC1 CC1CCC(OCC(=O)NC2CCN(C(c3cc(=O)cc[nH]3)=O)C2)CC1 c1(NC(=O)NC(c2cc(Cl)cc(Cl)c2)(C)C)ccc2c(ccn2CCO)c1 c1(C(N2CC(CC)SCC2)=O)coc2c1CN(C(c1c[nH]nc1Cl)=O)C2 c1(C(=O)NC2(CNC(CCCOC)=O)CCOC2)cncc(N2CCCC2)n1 Cn1cc(C(=O)NCC2CC2C)c(Cl)n1.C(=O)(C(C)(C)c1cccs1)N C1CC2(CCCO2)C1.N1(C(C(C2CCCC2)NC(=O)C)=O)CCCC(CF)C1 C1(C(N(CC(CC)C)C)=O)CNC(=O)CN1C(C1CC(C)(C)CCO1)=O N1(C(c2c(C(C)C)cnn2C)=O)CCC(C2CC(NC(=O)C=CBr)C2)CC1 n1(CC(=O)Nc2nc(OC)sc2)cc([N+](=O)[O-])c(C(F)(F)F)n1 CCC(C)(C)C(O)C(=O)NCC(C)(O)CNC(c1c[nH]ccc1=O)=O N1(C(CSSC)=O)CCCC1(C)CNC(=O)COC1CCCOC1 C1(C(=O)NCc2cccc(OCCC=C)c2)(CN)CC2CCC1C2 NS(=O)(=O)c1scnc1C(=O)NCCC.C1(C(=O)N)COCCN1C1CCCC1 C1(C(=O)NCc2cccc(O)n2)COC2(C1)CN(C(C1C3CCCCCC13)=O)C2 c1(C(=O)NC(CC)CN(C)C(C23CC(C2)C3)=O)ccc(CN(C)C)o1 N1(C(c2c(C)cc(C)cc2C)C(=O)NCC(F)F)CCCC(C2CCCC2)C1 C1(CC(=O)NCCn2cc(-c3c(C)c[nH]n3)nn2)CCC(C)C(C)C1 c1(NC(N2C(SCC)CCCC2)=O)ccc(N2C(=O)CNC2=O)cc1C C1(C(=O)NC(CC=C)CNC(=O)Cc2cnn(CC)c2)CC2CCC(C1)S2 C(C#Cc1ccc(Cl)cc1)N1CCCC(NC(Cc2c(OC)cccc2)=O)C1C C1(NC(COC(CC)C)=O)CC2CCC1CN(C(c1c(N)ccc(C)c1F)=O)C2 c1(OC)ccc2[nH]cc(C(N3CCCC(C)CC3)=O)c2n1 N1(C(c2n(CC)ncn2)=O)CCC(C2CC2)C1CNC(C1CC1(Cl)Cl)=O C(CCCC(C)NC(c1cc(C)c(C)s1)=O)NC(C(C)SCC)=O c1(C(=O)NCC(C)(C)NC(C2N(C(CCCC)=O)CSC2)=O)ccc(N)cn1 N1(C(c2cc(CC)ncn2)=O)CCN(C(c2occc2Cl)=O)CC1CC N1(C(CC2C(OC)CC2)=O)CCC(C)(CNC(c2nn(C)cc2C)=O)CC1 c1(C(=O)NC2C(CNC(CC(C=C)CC)=O)CC2)ccc2cncn2c1C C1(C(C)C)COCCN(C(=O)C(O)CCCNC(=O)COc2cnn(C)c2)C1 C(=O)CCC(C)(C)[N+](=O)[O-].c1(SC(C)C(=O)NC2CCC(C)C2)ccccc1.N c1(C(N2CC(CCNC(C(CC)F)=O)(OC)C2)=O)ccc(Br)c(F)c1OC C1CC(C=O)C12CCC2.n1(CC(=O)N(CC)C2CC2)ccc(C)cc1=O.CO C#CCCC(C(=O)OC)NC(=O)CC(CNC(=O)CSCC)C1CCC1 C=CC(C)(C)C(=O)N(C(C)CNC(c1ccccc1SCCO)=O)C N1(C(C(CN(C)C)O)=O)CC2CCCN(C(C3Cc4ccccc4CO3)=O)C2C1 CC(N=c1[nH]c2ccccc2o1)C1CCN(C(=O)CCC(C)N(C)C)CC1 C12(CCNC(c3c(C)cco3)=O)CCC1CN(C(=O)CCc1ncc(F)cn1)C2 Cn1ncc(C(N)=O)c1NC(C1(F)CCN(C(=O)C=CCBr)C1)=O C(=O)(CC(CNC(=O)C(N1CCC12CN(CC)C2)=O)CC(C)C)OCCC C1(C(=O)NC(CN(C)C(c2nccc3n[nH]cc23)=O)(C)C)CCCCC(F)(F)C1 C=C(C)CC(C)C(=O)N1CCN(C(C2CCC3(CC2)CC3)=O)CC1CC(F)(F)F c1(CNC(CC=CCNC(C(C)SC)=O)=O)cccc(F)c1F N1(C(CCC=C)=O)CC(NC(c2cc(Cl)c(Br)cn2)=O)C2CCCC2C1 c1(C(N2CCC(C)(CCNC(C=C=C(C)C)=O)C2)=O)ccc(O)c(Cl)n1 C1CS(=O)(=O)CC1.c1(C=O)cnn(CC(F)F)c1.C1(C=O)(C=O)CC1.C C(=O)(C#CC(C)(C)CNC(=O)C=Cc1cscn1)NC(c1ccnc(C)n1)C c1(C(C)C)ccc(C(=O)NC2(C3CCCN3C(c3nnn(C)n3)=O)CC2)nc1 c1(OC(C)C(=O)N(C2CCCN(c3cnn(C)c3)C2)C)cccc(Br)c1 C(=O)(C(CCC=C)NC(=O)COc1ccn(C)n1)NC(CCC=C)C c1(C(N2CCCC(NC(c3csc(C(F)F)n3)=O)C2)=O)ccc(O)cc1Cl C12(CNC(C3CCC(C)C3)=O)CC(C1)C(C)O2.N1(CCC=O)CCCCC1=O Cc1c(NC(c2nncs2)C)ncnc1N(C)CCN1CCCCC1 C1(N(C(C(CC)NC(C)=O)=O)C)CCCCN(C(=O)COc2ccc(F)nc2)C1 C1(CNC(C2C(OC)CCC2)=O)CCCCC1NC(=O)CC1CCCOC1 Cc1[nH]c(C)c(C(=O)NCC(O)C(=O)NC(C(N)=O)C2CC2)c1C C(=O)(C(C)C(C)C(C)(C)C)N1CC(c2cn(-c3cccc(OC)c3C)nn2)(F)C1 N1(C(C(C)(C)OC)=O)CCC2CN(C(c3c(F)cccc3I)=O)CC12 CC(CCC(C)(C)C)C(=O)NC1CC(CNC(=O)CCCC#N)C1 C1(NC(c2nn(C)c(F)c2)=O)CN(C(c2coc(C(F)F)n2)=O)CC1(C)C c1(NC(CCc2c(OC)ccc(F)c2)=O)cnc2c(c1)CCN2 C1(NC(C(C)NC(N)=O)=O)CC12CC(NC(c1ccccc1)=O)C2 C(=O)(C1=C(C)OCCS1)NC(CN(C(C(C(=C)C)(C)O)=O)C)(CO)CO c1(C(N(C(C)CNC(=O)CC2CCC(=O)N2)C)=O)n[nH]c2c1COCC2 C1(SC)CN(C(=O)CCCCNC(=N)N)CC(C)(O)C1 CCC(C)(CO)C(=O)NCC1CCN(C(=O)CC2CC(F)(F)C2)CC1O c1ccc(Cl)c(F)c1.C1(NC(C=CC(=O)N(C)C)=O)CN(C(=O)CF)CC1O N1(C(c2ccc(C)o2)C(=O)NCC)CCC(c2ccc(C)cc2)CC1 CC1CN(C(C2CCN2C(=O)Nc2n[nH]cc2[N+](=O)[O-])=O)Cc2ccc(Cl)cc21 C(=O)(C(C)CC1CC1)NC(C1CC(F)(F)C1)C.C1(C(=O)N)CCCCC1 c1(C(N2CC(NC(=O)CCc3ccco3)C(F)C2)=O)c(F)cc(Br)cc1Cl c1(C(=O)NCCC2CN(C(C3C(OC)CC3)=O)C2)cccc(N(C)C)c1 N1(C(C2(C)CCCCC2)=O)CC2CCC1CN2C(=O)Cc1ccc2n[nH]cc2c1 C(=O)(C(O)CCS(C)=O)NCCN(C(c1cnc(C(F)(F)F)cn1)=O)CC C1(F)(C(=O)O)CN(C(=O)C=O)CC1(C)C(F)(F)F.C(C=C(Cl)Cl)NCC Cc1coc(C(C)C)c1C(N1CCC(N(C(=O)CCOC2CCC2)C)C1)=O c1(C(=O)NCCC(=C)CNC(C2CC23CC3)=O)c(Cl)sc(Cl)c1C N1(C(C(C=C)(C)O)=O)CCC2CCC(NC(=O)Cc3ccc4c[nH]nc4c3)C1C2 N1(C(CN2CC(=O)NCC2)=O)CCCC2(NC(=O)C(F)(F)C3(O)CCC3)CC2C1 C=CC(CC)CC(=O)NC(C1CCN(C(=O)COC2CC(F)(F)C2)CC1)CO CC(CCC(=O)N1CC(C(C)(C)C#N)C1)NC(C1CC(=O)CS1)=O C1(NC(C)=O)CCC(C=O)CC1.c1(C=O)nnn(C)n1.C(C)(C)C1CCC1.N C(=O)(C(C)(C)C(C)(F)F)N1CCCC(N(C)C(c2ncc(C(F)F)s2)=O)CC1 N1(C(C2(C)CCN(C)C2)=O)CCOC(C(N2CCC(C(F)(F)F)C2)=O)CC1 c1(C=O)ccc([N+](=O)[O-])cc1.CN1CCCC(C)(C(=O)NCC2(O)CCC2)C1 c1(C(N2CC(O)CC(NC(CCCSC)=O)C2)=O)c(F)ccc(C(F)(F)F)c1F CN=c1cc(C(N2CCCCC2C(=O)NCc2cn(C3CC3)cn2)=O)cc[nH]1 CC1CCC(=CC(N2CC(NC(C3(C)CCCOC3)=O)C(O)C2)=O)CC1 CN1CCCC(F)(C(N2CCC(CO)C(NC(=O)C=CC3CC3)C2)=O)C1 c1(CCNCc2c(C)oc(=O)o2)cc(C(F)(F)F)cc(S(C)(=O)=O)c1 C1(NC(=O)NCC(=O)NCC)COC2(CCN(C(=O)CCC=O)C2)C1.O CCC(C)C(O)CC(=O)NC1(C)CC(NC(C2(C)CCS(=O)(=O)CC2)=O)C1 C(C(C(=O)NCCC1(O)CN(C(C2(C(F)F)CCC2)=O)C1)N(C)C)OC c1(NC(C(CSCC)NC(=O)OC(C)(C)C)=O)cnn2c1OCC(C)C2 Cc1cc(C(=O)NCC#CCNC(=O)CC(C)CF)c2ccccc2n1 C(CC(CNC(C1(O)CCCC1)=O)NC(C1(c2ccno2)CCC1)=O)OC C1(NC(C2C(CC)C2)=O)CN(C(C2CC23CC(O)C3)=O)C2CCCCC12 C1(NC(COC(C)(C)CNC(=O)C(C2CCOCC2)F)=O)CC2CCCC2C1 c1(CC(C)C)nc(-c2ccc(OC(C)(C)C)cn2)nn1CCc1ccccn1 c1(C(=O)NCC(C)NC(c2nc(C)oc2C)=O)cccc(Cl)c1F n1(CC(N2CC(SC)C(n3cc(C4CCOC4)nn3)C2)=O)cnc2c1CCCC2 CN1CC2OCCN(CC3CCN(CCc4ccccc4)C3)C2C1 C(=O)(CC(CC)C(F)F)NC(CC=CC(N1CCC(OCC#C)C1)=O)(C)C C1(C(=O)NC(C)C(C)n2cccn2)CCCN1NC(=O)c1ccsc1 c1(C(=O)OC)c(NC(=O)CC2(N(C)C)CC2)sc2c1CCOC2 N1(C(c2ccc(C#N)s2)=O)C(C(N2CCn3nccc3C2)=O)CC2CCCCC12 CC1N(C(=O)C(N2CCC(N3CCN(C)CC3)CC2)=O)CCC1(C)C CCC(C)CCCCC(=O)N1CCCCC(NC(=O)C(C)O)C1 c1(C(=O)NC2CN(C(c3n(CCOC)ncc3)=O)C(C)C2)cc(Cl)ncc1O C#CCC(C)(C)C(c1nnnn1C1CCC1)NC1CCCN(c2cccnc2)C1 Cc1cc(NC(=O)C=Cc2cn[nH]c2)ccc1.c1(C=O)ccoc1CC(N)=O.N c1(OC)ccccc1CCC(=O)NC(C1CCN(C(C2(O)CCOC2)=O)C1)C c1(C(c2n(CCCF)nnn2)NCCC2(OC)CCC2)ccc(Cl)c(C(F)F)c1 CCC(C(=O)NC1CC2(C1)CC(NC(=O)Cn1cc(Br)c(=N)[nH]1)C2)C(C)C CCC(F)(F)CC(=O)N1CC(NC(c2ccoc2Cl)=O)CC(O)C1 c1(OC)ccc2[nH]c(C(=O)NC(C)CC)cc2n1.c1(CC(=O)N)csc(=N)[nH]1 C1(C(=O)N)CCCCCC1.CC1OCCC1C(=O)N(C1CC(NC(=O)CC)C1)C C(C(=O)N1CCC(C(C)(C)O)CC1)(C(C)(C)C)NC(C1CN(C)C(=O)C1)=O C(=O)(CC(C)P(C)(C)=O)N1CC(CCC)N(C(=O)C=Cc2nc(C)cs2)CC1 C(=O)(CCC(=O)c1ccc[nH]1)NCC1C(NC(c2c(C)coc2)=O)CC1 N1(C(C=C(C)C(F)F)=O)CCCC1.c1(CCC(=O)NC2CC2)cnc(C)o1.C c1(C=O)ccc(F)cc1.C1(CC(=O)NCC2C(CCOC)C2)CCC1.N C1(NC(C(C)NS(CCCC)(=O)=O)=O)CN(C(C2(F)CC2)=O)CC12CC2 C1(NC(C=NOC)=O)CCC2(CCCN(C(c3cc4cc(F)ccc4o3)=O)C2)C1 C(=O)(C(C)(C)C(=O)NC1CCN(C(c2csc(C)c2)=O)CC1C(N)=O)OC c1(C=O)cc(O)nc2ccc(Cl)cc12.C(C)(C)(CC(=O)NC1CC1C)OC.N N1(C(C(=O)NC(CC)(C)C)C2CC2c2cccs2)CC=CCC12CCCCC2 Cc1cc(C)c(C(=O)NC2CCN(C(=O)CCc3cnn(C)n3)C2C)c(C)c1 c1(CC)ccccc1OCC=O.c1(C(N(CCC)C(C)C)=O)cc(=N)[nH]n1C C1(NC(CCCN(C(C)C)C)=O)CN(C(C2C=CCCC2)=O)C2(CCCCC2)C1 c1cccc(C#N)c1.CC(CNC(C1(CCF)CC1)=O)C1CC1.C(=O)(C)N CC1(C)COCC(NC(C2C3CC2N(C(C2(CO)CCOC2)=O)C3)=O)C1 c1(C(=O)NC2C(C)CN(C(c3cc4ncsc4[nH]3)=O)C2)c(Cl)ccc(F)c1Cl C1(COC)(NC(=O)CNC(=O)O)CCN(C(=O)CCc2csnn2)C1 c1(C(=O)NC2CC(NC(c3cnsc3)=O)C23CCC3)c(F)ccc(F)c1O N1(C(C(C(C)(C)C)OC)=O)CCC2(C1)CN(C(C1(CC3CC3)CC1)=O)C2 N1(C(CCCC(C)C)=O)CCCN(C(C2CCC2(F)F)=O)CC1C C1(NC(CSC)=O)CN(C(=O)CCc2ccc(N)cn2)CC12CC2 C1(NC(C(=O)NCC)=O)CC1C1CCN(C(C2CC(O)C2)=O)CC1 CCC(CNC(=O)C(C1(O)CN(C(c2coc(N(C)C)n2)=O)C1)F)(CC)CO c1(C(=O)NC2CCC(NC(CCC)=O)C2)cc(C)n(-c2ccc(Cl)cc2)n1 C1(CNC(COCCOC)=O)CCCN(C(=O)C)C1.C1CCOC1.NC.O N1(C(CCC=C)=O)CC(NC(c2ncnc(O)c2Cl)=O)C(C2CC2)C1 CC(C)CC(O)C(=O)NCC(O)CNC(c1ccc(NCC(N)=O)cc1)=O C1(NC(C2(C)C(C)(C)C2(C)C)=O)CCCC(N=c2[nH]c3ccc(N)cc3s2)C1 C1(C(N(C2CCC(NC(C3CCCC(=O)N3)=O)CC2)C)=O)CCN(C)C1=O c1(C(=O)NCC2(F)CC(Nc3cc4nncn4cn3)C2)cc2ccc(O)nc2s1 C1(C(CC)C)CN(C(C2(C(C)NC(C3CCC3C)=O)CC2)=O)C1 c1(C(=O)N)cnc2c(F)c(F)ccc2c1.C(CC(=O)NC1CCC1)OCC(C)C N1(C(c2occ(C)c2)=O)CCCCC1CN(C(=O)CCN(CC(F)(F)F)C)C c1(C(=O)NCCC(C)NC(C2(C)CCC2)=O)cc(-c2ccc(Cl)s2)[nH]n1 O=C(C1=CCN(C(C2CC23CCC3)=O)C1)N1CC(Cn2ccnn2)C1 Cc1ccc2c(c1)C(C(=O)NC1CCN(C(=O)C=Cc3sccc3Br)C1)C2 c1(C(=O)NC(CC(C)NC(C=C(CC)CC)=O)C)cc(Cl)c(Cl)n1C N1(C(C2CC(F)C2)=O)CCN(C(C2CC2c2ccncc2)=O)CC(CO)C1 Cn1cnc2cccc(C(=O)NCCC3CN(C(C4CC45CC5)=O)C3)c12 CCC(C)(COC)C(=O)NC1CCC(C)C1.c1(C(C=O)=O)cc(F)ccc1C.N CCC(CC)C(C(=O)NCC1COCCN1C(c1coc(C(C)(C)C)n1)=O)OC CCCCC(C(=O)NCC1(C)CCCN1C(c1ccc(OC)cc1F)=O)ON N1(C(C(CC)OC)=O)CC2CC1CCN2C(=O)CCc1ccnn1C C1(C(N(CCCNC(=O)CSC(F)(F)F)C2CC2)=O)CCC1(F)F C1(NC(=O)C(O)C2CN(C(=O)C#CC3CCOC3)C2)CCc2nncn2C1 C1(C(N2CC(CNC(c3n(CC)ccn3)=O)(C)C2)=O)CC1C1CCCC1.O c1(C(=O)NCC2C(NC(C(C)SC)=O)C2)ccc2ncncc2c1 C(=O)(C(C)(C)C1=CCN(C(C2CCCCC2F)=O)C1)N1C(CC=C)CCCC1 Cc1nn(C)c(C(=O)NC(C2CCCN(Cc3cccc(F)c3Br)C2)C)c1F c1(C(N2CCC(NC(=O)NC)C2)C(=O)NCCCSC)cc(F)cc(F)c1 c1(C(=O)NC(C)C(C)NC(c2cn(CC(=O)N(C)C)nn2)=O)ccncn1 Cc1ncc(C(N2CCC(CC(=O)NCC3CCOCC3C)CC2)=O)cc1C#N c1(C(=O)NCC2(C)CCCC2(F)F)nc2cc(F)c(Br)cc2[nH]1 C(C(C)(C)C(=O)N1CCC(N(C(=O)Cc2cncs2)CC2CC2)CC1)SC C(=O)(C1CCCc2scnc21)NC(C1CCN(C(c2ccc(F)cn2)=O)C1)(C)C C1(C(=O)OC)CC(C(=O)OC)CN(Cc2ccc(C)n2C)C1 C(=O)(CCC=CBr)NCC(C)(C)NC(c1cn(CC2CCOC2)nn1)=O c1(C(N2C3CCC(NC(CSCC#C)=O)(C3)C2)=O)cc(Cl)cc(Cl)c1OC N1(C(COCCSC)=O)CC(F)(F)CC1CCNC(C1CC(O)C1)=O C(=O)(C(Cc1ccsc1)c1ccccc1)NCC(N1CCCC1)=O.c1ccccc1.C CC1(C)CC(CC(=O)NCCCNC(=O)C=CCN2CCOCC2)CCO1 C1(n2cc(CC(C)(C)OC)nn2)CC2CCC(C1)N2C(C1CC1C=O)=O.O CCC(CC(=O)NCCc1cc(C(=O)NC2CC(O)C2OC)no1)C(C)C c1(CCC(=O)NCCN(CCOC)C(C2CC(F)C2)=O)cncc(C)c1 c1(C(=O)NCCO)ccc(OC(F)(F)C(F)F)cn1 CC1=C(C(=O)NCCC)C(=O)OC1(C)C.[SH](=O)(=O)c1cccs1.C(=O)CC.N c1(C(=O)NCCCC(C)NC(c2n(CC)ccc2)=O)c(F)cc(N)cc1F C1CC2CCCC12.C1(C(=O)OC)CC=CCC1C(N1CCC(O)C1C(=O)N)=O c1(C(=O)NCC(C)N(C(=O)CC2(O)CCC2)C)ccn2c(Br)cnc2c1 CC1C(NC(c2cc(O)nn2C)=O)CCCN1C(=O)C(C#N)CC1CC1 Cc1nccnc1C(=O)NC1(CNC(=O)C(F)C2CCCC2)CCOCC1 C#CCCCC(C)C(=O)NCC1CC2CC2N1C(c1cccnc1)=O c1(NC(c2n(C)cc(NC(c3c(C)nsc3)=O)n2)=O)cc(F)cc(F)c1 c1(C(=O)NC2(CO)CCCN(C(=O)CCn3cncn3)C2)cc2cccn2cn1 Cc1cc(C#N)ccc1C(N1CCOC(CC(=O)Nc2ncccc2C#N)C1)=O C(=O)(C1=CC(O)C(NC(=O)C=CC)C1)NCc1c(C)nc(CC)o1 N1(C(c2cnc(SC)s2)=O)CCCC(C2CCCCN2C(=O)C(C)C(C)O)C1 c1(C=O)cn(C)c2ccc(Cl)cc12.N1(CC(=O)N(CC(O)C)C)CC(C)(C)C1 Cc1nc(Cl)ccc1C(N1CC(c2cn(CC3CCCO3)nn2)C(O)C1)=O Cc1cc(OC(C)C(=O)N(CC(C)(C)NC(=O)C=CS(C)=O)C)ccc1Cl C1(C(=O)NC2CCCN(C(c3c(Cl)cnc(CC)n3)=O)C2)CCCC(F)(F)CC1 N1(C(CS(C)(=O)=O)=O)C2CCCC1CC(NC(=O)CCCn1cnc(C#N)n1)C2 N1(C(c2c(CC)ncs2)=O)CCC2C(C1)CN2C(=O)CCC1CC1(Cl)Cl CC(C)CC(C)CC(=O)NCCCC(C)(C)C(=O)NCCc1csnn1 C(C)(CCCC(=O)N(CCC1CC1)CC)NC(c1nccc(CC)c1)=O c1(C(N2CC(C)C(n3cc(-c4cc[nH]n4)nn3)C2)=O)sccc1S(N)(=O)=O c1(C(=O)NC(CCCCNC(c2n(CCC)ncc2)=O)C)ccc(OC)cc1Cl CCC(C)CCCC(=O)N1CC=CC(NC(c2cncs2)=O)C1 c1(C(=O)NC2C(CNC(C(C)(C)CF)=O)C2)cccc2c1OCCO2 C(c1ccc(F)cc1)=CCN(C(C(=O)OCC)C)CCNC CC1CN(C(=O)CCCN(C)C)CC1(C)C(=O)NOCC1CCCCC1 C1(N=[N+]=[N-])(C(=O)NCc2cnc(CC)[nH]2)CCN(C(=O)CS(=O)(=O)CC)C1 C(=O)(C(C)(CC)C(=O)N1CCC2(CC2)C1)OCC.c1(C=O)cnc(S)nc1.N C(=O)CCC(CF)CF.C1(C(N(C)CC2CC2)=O)CCCN1S(C)(=O)=O.C C(=O)(C(C)(C)c1ccsc1)N.C(=O)(C(C)=C1CCC1)N(CCOC)CC C1(C(N(CCC#C)C)=O)CCC(O)CN1C(c1cnc(S)nc1)=O Cc1ccc(C(=O)NCC2CC(NC(=O)C3=COCC3)C2)c(Cl)c1C C(=O)(C1=CCCN(C(=O)C(C)Cn2cccn2)C1)N1CCCC(CCC)C1 C(=O)(C(C)(C(C)(C)C)NC=O)Nc1ccc(C)cc1.C(C)(C)C.C1CCC1 CS(=O)(=O)CCCNC(C1(CNC(=O)CC2CCC(O)C2)CC1)=O C1(CNC(C2(C(C)C)CC2)=O)CC2(C1)CN(C(C1CC(F)(F)CS1)=O)C2 c1(CCC(=O)N(CCCNC(C(CC)(C)CC)=O)C(C)C)nc2cnccc2[nH]1 c1(CC)occ(C)c1C(=O)NCC(CCOC)NC(c1cnn(C)c1)=O C#CC1(C)CCCN(C(c2ncccc2F)C(=O)NCCC#N)C1 N1(C(=O)CSc2cn[nH]c2)CC2CC(C(=O)NCC3C4COCC34)(C2)C1 C1(NC(CCCNC(=O)OC)=O)CC(C(=O)NC2C(C)CCC2C)C12CCC2 c1(C(=O)NCC(CCCC)NC(=O)COCC)nn(C)c(C(F)(F)F)c1Br C1(CNC(c2cscc2F)=O)CCC2(CCC2)C1NC(c1nsnc1O)=O C1(OC)CC2(CCC(C(=O)NCC(C)(C)NC(c3cccnc3)=O)CC2)C1.C N1(C(=O)C(F)(F)c2nccs2)CCCC(CNC(C2(c3cc[nH]n3)CC2)=O)CC1 C#Cc1ccc(CCC(=O)NC(C2CCCN(C(=O)CC(C)(C)C#N)C2)C)cc1 c1(C(N2CC(CNC(C(F)OC)=O)(O)C2)=O)cnn2c1NCCC2C(C)(C)C c1(C(=O)NCC2CC(C)N(C(c3cn4c(n3)CCC4)=O)C2)ccc(Cl)c(Cl)c1 C1(CC(=O)NCCCC(C)NC(Cc2cc(C)ns2)=O)CCCCC12CC2 CCCCCC(O)C(=O)NC(CC)(CC)CCNC(c1cc(C)n(C(F)F)n1)=O C1(C(N2CC3(C2)CN(C(C2(F)CC2)=O)C3)=O)CC2C=CC1CCC2 N1(C(c2ccc(OC)cc2)=O)CCC(NC(C2NC(=O)OC2(C)C)=O)C(C)C1 C1(C(N2CC(CCC)C2)=O)CC(F)CN1C(c1cc(CO)n(C)n1)=O CN1C(=O)CC(C(=O)NCCCOCCS(N)(=O)=O)C1c1ccnn1C C1(CC(N2CCC(N(C(=O)CCCNC(C)=O)C)C2)=O)(COC)CCCC1 Cc1cc(CC(=O)NCCC2CCN(C(=O)CC34CC(C3)C4)C2)c(C)s1 C1(N(C(c2ccc(C)s2)=O)C)CN(C(=O)COc2ccsc2)CC1(C)C C1(CCC)(NC(c2cn(CCCC)nn2)=O)CCCN(C(=O)C(C)S(C)(=O)=O)C1 N1(C(CC(=O)N(C)C)=O)CCC(CNC(C2CC(C)(F)C2)=O)C(F)(F)C1 C1(N(C(C2C3(CCC3)C2)=O)C)CCOC(C)(C)C1.CC(=NOCC#N)C(=O)N c1(C(=O)NCCC(c2ccccc2)C)cn2cc(CN)ccc2n1 CCC(C)(CNC(c1[nH]ccc(=O)c1C)=O)C(=O)NC1C=CC(CO)C1 C(=O)(C#CC1CCOC1)NCC(CC)NC(=O)C(F)(F)O.c1cc(Cl)cc(Cl)c1 C1(C(N(C)CCn2cc(-c3cn(C)nc3C(F)F)nn2)=O)CC1C1CCC1 c1(CC(=O)NC2C3CN(C(CCOC)=O)CC32)cc(OC)ccc1Br N1(C(CC(C(C)C)O)=O)CCC2CN(C(c3c[nH]c4nc(Cl)ccc34)=O)CC2C1 C(C(=O)NCc1ccccn1)(C(C)(C)C)NC(C(C1CC1)OC)=O C1(CN(C)C)CC(N=c2cc[nH]cc2S(=O)(=O)NC2CC3CSCC3C2)C1 c1(NCC2N(C(C(C)NC(C)=O)=O)CCCC2)cc(OC(F)F)ccc1[N+](=O)[O-] c1(CCCC(=O)NC2CCC3CC23C(=O)O)c(F)cccc1F CCCCCCNC(c1occc1C(C)C)=O.C1(C)(CCC=O)CCC(=O)N1.N C=CCC(F)(F)C(=O)N1CC2CC1C2NC(=O)CC1CCC2CC12 c1(OCCOC)ccc(CC(=O)Nc2cn[nH]c2)cc1.C12CC(O)C1O2 Cc1[nH]c2ccccc2c1CC(=O)NC(C)(CNc1cnc(C#N)cn1)C1CC1 CC(C)CC(C)CC(=O)N1CC(NC(c2cccnc2O)=O)C1 C#CC1CCCN(C(c2n[nH]cc2CNC(c2ccoc2)=O)=O)C1 Cc1sc(C)c2sc(CN3CC(n4cc(CCCS(N)(=O)=O)nn4)C3)cc12 n1(CCCC)nnnc1C(CC)(CC)NC1(CCO)COC1 c1(CN2CCCN(C(c3cccc(OC)c3C)=O)CC2)ccc(O)c(C)c1O c1(C(N(CCNC(CCSc2nc(C)[nH]n2)=O)C)=O)cnc2occc2c1 C1(NC(c2ccc(N(C)C)cc2F)C)CN(C(=O)OC(C)(C)C)CC12CC2 C(C1c2ccccc2CCN1c1cc(C)ncn1)NC(CC(COC)(C)O)=O c1(CC(=O)NC(CCNC(c2n(CCC)nc(C)c2)=O)C)ccc(O)cc1Cl c1(C(N2CCC(N3C(C(N(C(CC)C)C)=O)CCC3)CC2)=O)ccnc(F)c1OC CCCC(C)CC(=O)N1CCN(C(c2cc(CC)no2)=O)CC1C(C)C Cc1cc2cc[nH]c2cc1NC(c1ccc(CNC2(C)CCC(C)(C)C2)cc1)=O c1(CC=C)ccccc1C(=O)NCC1(NC(c2oc(CO)nc2C)=O)CC1 C1(NC(Cc2cc(C)no2)=O)CCCCN(C(=O)C(C)Cc2ccccc2)CC1 c1(CNC(C2C(CCOC)C2)=O)cc(C(N2CC(F)C2)=O)cs1 c1(CNC(C)=O)ccccc1C(N1CCCC1C)=O.c1(C(=O)N)ccnc(S)c1 N1(C(C=C(COC)C)=O)CC(CCNC(=O)CC2C=CCCC2)C(C)C1 c1(C(N2CCC3CC3C2)C(=O)NCCOC)nc2c(s1)CCCC2 N1(C(c2c(CC)nc[nH]2)=O)CC2CCC1C(NC(c1ccnc(C)n1)=O)C2 c1(OCC(=O)NC(C)CCNC(=O)CSC2CC2)ccccc1F C1(NC(CCN(CCCCC)C)=O)CC2(CCN2C(C2CC=CCC2C)=O)C1 C#Cc1cccc(C(N2CCN(C(C3C4COCC34)=O)C(CF)C2)=O)c1 CCC(CN(C)C)C(=O)NC1CCC(C(=O)NC2C3CCCCC23)C1 c1(CC)[nH]nc(C(=O)NCC(C)CN(C)C(c2nocc2C)=O)c1Cl C1(CNC(C(C2CCOCC2)C)=O)C2CN(C(c3ccccc3)=O)CC12.CC#N.S C(=O)(CCC(C)CN(C)C)NCC1N(C(c2c(C)occ2)=O)CCCC1 CCCC(C#N)C(=O)N1CCC(C(=O)NC(CO)C2CC2)C1(C)C CC(C(=O)N1CCC(CO)(NC(=O)CSC2CC2)CC1)C(C)S(C)(=O)=O c1(C(C)O)ccc(C(=O)NCC(CNC(c2ccccc2C2CC2)=O)CO)cc1 N1(C(C2CC(=C)C2)=O)CC2CCCC(NC(c3cnc(C)n3C)=O)C2C1 C1(C(=O)NCCC(C)(C)C)CCC2(CC1)CC2.C1(CC=O)CC(O)C12CCC2 C=C1CC2CCC(C1)N2C(=O)CC1CCCN(C(c2occc2C)=O)CC1 C(CC(C(=O)NC(C)CCCCO)NC(=O)C=Cc1cc[nH]n1)OCC c1(C(C)C)ncc2c(n1)CN(C(c1n[nH]cc1Br)C(=O)NC1CCOC1)C2 c1(C(C(=O)NCCC)N(C2CCCC2)CCOC)cccc(C(=O)OC)c1 c1(C(N2C(CC)C(C(=O)NCC3(CCO)CC3)CC2)=O)cc(C#N)cn1C C(C(O)(C(F)(F)F)c1ccccc1)NC(=O)NCC1(c2ccncc2)CCC1 CCC(CCC(=O)NC1(C(=O)NCC(C)(O)C(=O)OC)CC(CO)C1)OC c1(C(N(C)CCNC(C2CC=CCO2)=O)=O)noc2c1CCCC2 C1(CC(=O)NC(C2CCN(C(c3ccn(C)c3)=O)CC2)C)CC2CCC1O2 c1(C(c2n(CCCOC)c(N(C)CC3CCOC3)nn2)C)c(F)cccc1F c1(CC)ccc2c(n1)CN(C(C(=O)NCc1ccc(OC)cc1)C1CC1)CC2 c1(CC(=O)NCC=CCNC(Cc2c(C)ocn2)=O)cc(O)ccc1Br Cc1cc(C(N2CC(NC(=O)C3=NOCC3)C(C3CC3)C2)=O)ccc1S(N)(=O)=O c1(C(N(CCCN(C)C(c2cn(CCC)cn2)=O)C)=O)cc(F)c(F)c(N)c1Cl C1(C)(C(=O)NC)CCN(C(c2ccn(C(C)C)c2)C(=O)NC)C1.C1CCOC1 Cc1c(C(=O)NCC(C)(CO)NC(C2CC=CCC2)=O)nnn1C Cn1ccc(C(=O)NC2(C(=O)NC3(C(O)CO)CC3)CC(F)C2)cc1=O C(c1cc(F)cc(F)c1)=CC=O.N1(C(COC2(C)CCC2)=O)CC2(CCC2)C1 C1(CC=C)(NC(=O)C(COC)CC)CCN(C(=O)C=CSC)C1 Cc1cc(N(C)Cc2c[nH]c3cccnc23)nc(=NCCCc2ccco2)[nH]1 C(=O)(C(C)C(CC)CC)NC1C=CCN(C(c2c(C)nc(CCC)o2)=O)C1 N(C(=NCCF)NCc1ccc(OC)c(F)c1)CC1N(CCOC)CC1 C1(CNC(c2ccc(-c3ccncc3)cc2)=O)CCN(C(C2COC2)=O)C12CC2 C1(C(=O)NCCCSCC)CC2CC1CN(C(=O)C(C)(C)n1cncn1)C2 c1(CC(=O)N(CCCCNC(=O)COC)C)cn(C)nc1Cl.c1cccnc1 C(=O)(C(O)CC(C)C)NCC(CNC(CCn1c(C)ccc1C)=O)(C)C N#CC1(c2ccccc2)CCCN(N2CCC3(CCCNC3=O)CC2)C1 C1(CCNC(CNC(C)=O)=O)CN(C(=O)CCc2ccncn2)CC1C C1(F)(CNC(C(C2CCOC2)NC(c2csc(F)c2)=O)=O)CC(CO)C1 c1(NCc2nc(C)sc2)cccc(C(=O)Nc2ccccc2)c1 c1(C(N(C)CC2(O)CN(C(C3CCC3(F)F)=O)C2)=O)ccc(=O)n(C)c1 N1(C(C2C(C)C2)=O)CCOCC(NC(c2c[nH]nc2C2CCC2)=O)C1 c1(C(=O)NC(CN(C(=O)CCC2CCCO2)CC)C)cc(O)ncn1 C1CC(O)CN1C(C1CCN(c2ccncc2)C1)=O.C(CC(=O)NC)NC(C)=O N1(C(CN(CC(C)(C)C)C)=O)CCC2CCCC12CNC(c1cnc[nH]1)=O C1(CC(C)C)CCN(C(=O)CC2(C#N)CC2)CC1.C1(N(CC=O)C)CCSC1.N Cc1c(C(=O)NC2CC(O)C2CC(=O)NC2CCCC2N=[N+]=[N-])cccc1F N1(C(CCC=CC)=O)CCC2CCC(C1)N2C(c1cnc(NCC)c(Cl)c1)=O C=CC(CC(=O)NCC1CC(NC(c2oc(CC)cc2C)=O)C1)c1ccccc1 C1(COCCOC)CCN(C(=NCc2cc(C)co2)NC2CCCCC2)C1 c1(C(NOCCOC)=O)cn(CCNC(c2cccn2C2CC2)=O)nn1 C(CCCC(=O)N1CCCC1C=CC(=O)NCCn1ccnc1C)OC C1(C(=O)NCC(CCNC(c2c(C)nsc2)=O)O)CCc2cnc(C)n2C1 CN=C(NCc1ccc2nccc(N)c2c1)N1CCCC(CN2CCOCC2)C1 c1(CN(CCCN(C(CC2C(OCC)COCC2)=O)C)C)ccc(F)nc1F C1(NC(CCCC=C)=O)CN(C(c2cccc(O)n2)=O)CCC1(C)C C(C(CCC(F)(F)F)NC(=O)NC1CC(O)C(F)C1)OC C1(NC(c2c(C(C)(C)C)cccn2)=O)CC2(CCN(C(c3cnn[nH]3)=O)CC2)C1 N1(C(c2ncn(C)c(=O)c2)=O)CC(C(=O)NC(CCO)C2CCC2)CC(C)(C)C1 N1(C(CN(C(=O)C(F)CC2CCOC2)CCOC)=O)CCN(C)C(CO)C1 N1(C(C(c2c(C)noc2C)CC)=O)CC(CNC(C2CCC2)=O)OC(C)(C)C1 Cc1ccc(CCNC(=O)CNC(c2cnc(C)s2)=O)cc1.C(=O)C(C)O CC(C)(CNC(=O)CC1CC(CF)C1)C.C1(C=O)CCCN1c1ccccc1 CCCCCC(O)C(=O)NCC12CCC(NC(=O)Cc3csc(C)c3)(CO1)C2 c1(C(N2CC(C)C(NC(=O)COCC(F)(F)F)C2)=O)cc2ccc(Cl)cc2s1 CC1CCCC1C(=O)NCC(C)(C)NC(=O)CCCc1csc(=N)[nH]1 C1(NC(C=CCNC(C2N(CC)CC2)=O)=O)CC2CCC1(CO)C2 c1(C(N2CCOCC(F)(CNC(C(C)C(F)F)=O)C2)=O)ccnc2ccccc12 c1(OC)ccc2cc(C(=O)NCCC3CN(C(=O)C(C)C#N)CCO3)ccc2n1 C1(N(C(c2cccnc2)=O)CC)CCC2CN(C(=O)COC3CCOCC3)CC12 c1(C(N2C(C(=O)NCc3cc(C)[nH]n3)C(C)CC2)=O)ccc2cccnn12 Cn1cc(-c2cc(C(N3CC(NC(=O)CCN4CCC(F)C4)C3)=O)no2)nn1 N1(C(c2cc(CC)n(CCO)n2)=O)CCC(C)CC1.c1(C(=O)N)nc(O)c(C)s1 c1(C(=O)OC)cccc2oc(=NCCC3CCN(C(c4ns[nH]c4=O)=O)C3)[nH]c12 C#CCCC(C(=O)NCC1CCCOC1(C)C)NC(C1CCCC(C)(C)C1)=O c1(C(=O)NCC(C2CCCN2C(=O)C(F)F)(C)C)ccc2cccnc2n1 c1(OC)n[nH]c(C(=O)NC(C)CC2CCN(c3cc(C(F)F)ncn3)CC2)c1Cl C1(C)(CC)CC(NC(=O)CCNC(c2cccs2)=O)CN1C(=O)C(C)C CC1C(C)N(C(c2cscc2Br)=O)CCN1C(=O)COC(C)(C)C c1(CC)cc(=NC(=O)c2cc(CNC(C3CCC(=O)CC3C)=O)no2)[nH]n1C c1(N(C)CC2CC2(C)C)ccc(S(=O)(=O)N2CCCCS2(=O)=O)c(Br)c1 CCCC(C(=O)NC1(CNC(C2(C#N)CCCO2)=O)CC2CCC1CC2)C(C)C c1(C(N(CC(CC)NC(C2CCC2C(=O)O)=O)C)=O)ccc([N+](=O)[O-])n1C N1(C(C2CCC(C)C2)C(=O)NC(C)C)CCc2c(cc(F)c(F)c2F)C1 CC(C)(C)C(CCC1CCCC1)NCC(C(F)(F)F)c1ccon1 N1(C(C(=O)N(C2CCCOC2)CC)=O)CCCC(OC2CCC2)C1 c1(C(=O)NCCCN(C(=O)CC(O)C2CCCC2)C2CC2)ccc(Cl)c(F)c1 N(C(=NCC#Cc1ccccc1)NCC1CC=CCC1)CCNS(C)(=O)=O CC1C(NC(=O)C2=CCCC2)CC2CCC1N2C(c1c[nH]nc1C(C)(C)C)=O c1(OCC)cc(C(=O)NC2CC(C)C2)ccc1.C1(C=O)COCC1(C)C.N C(C(F)(F)F)(C(C)(C)C(=O)O)N(C)Cc1cc(C(F)(F)F)cc(F)c1 C1(C(N2CC3C(NC(C4(O)CCC4)=O)C3C2)=O)COc2cc(Cl)ccc2C1 Cc1nc2c(o1)CCCC2CC(=O)NC1CC2CCC(C1)N2C(C1(F)CCC1)=O C1(OCC)CN(C(=O)C(C)SS(C)(=O)=O)CC1.c1(C(=O)N)ccco1 c1(CNC(COc2cn(C)nc2)=O)ncccc1C(=O)NC.C1CC(O)C1 c1(C(=O)NCC2C(NC(C(CC#C)C)=O)CC2)cc(C(C)C)n2ncnc2n1 c1(C(N(C2CCN(C(C34CC5CC3C4C5)=O)C2)CC)=O)n[nH]c2c1COCC2 c1(C(C)NC(c2ccc(C(=O)NC)cc2)c2n(CCC)nnn2)c[nH]ccc1=O C1(NC(Cc2c(C)nc[nH]2)=O)CN(C(=O)C(C)C2CC2)CC2(CC2)C1 C(=O)(N=c1[nH]cc(Br)nc1S(N)(=O)=O)c1c2ccc(OC)cc2oc1 N#CCCCC(N)C(=O)N1CCC(C(O)CO)CC1 c1(C(N(CC(CNC(c2c(CC)con2)=O)(C)C)C)=O)cc(C)c(C)o1 c1(C(=O)NCC2CCN(C(CC)C)C2)cccc2[nH]ccc12 N(C)(C(=NCCC1CCCO1)NC(CS(C)(=O)=O)C(C)(C)C)CCCCOC N1(C(C2(C(C)C)CCC2)=O)CCN(C(=O)CN2CCCCCC2)C(C)C1 c1(CC)cccc(C(=O)N(CCC)C2CC2)c1N.C12(C(=O)N)CC(CCO1)C2 c1(C(=O)NC(C)CCCNC(C2CCCC3CC23)=O)cnn2c1CCCN2 N1(C(c2cn(CC)nc2C2CC2)=O)CCS(=O)(=O)C(CC)C1.C(=O)CC.N Cn1ccc(C(N2CCCC(CCNC(C3(Br)CC3)=O)C2)=O)c1C1CCC1 C1(C)(C=O)CN(C(=O)CC2(NC)CCC2)C(C)(C)C1.n1(C(C)C)cccn1 c1(C(=O)Nc2ccc(C(=O)C(F)F)cc2)c[nH]c2cc(Br)ccc12 N1(C(Cc2ccn(C)n2)=O)CC(C(=O)Nc2cnc(Br)c(Cl)n2)CC(F)(F)C1 C1(F)(CNC(C2CC2C(F)(F)F)=O)CCN(C(C2(CO)COC2)=O)C1 C1(CN2CC(CC=C)C2)CS(=O)(=O)CC(=O)N1.C(=O)C(C)Cc1cnc[nH]1 C(=O)(C1(C)CCc2ccccc21)N1CCC(NC(c2n(C)nnc2)=O)CC(O)C1 S(=O)(=O)(c1cccc2c1CCN(N1CCC(F)(C#N)C1)C2)NC(C)C c1(N(C(c2ccccc2I)C=O)CCN(C)C)cc(C)ccc1F.C(CC)SC.N c1(C(N2CCC(CC)C2)=O)ccccn1.C12(C(=O)N)CC(C)(C1)C2.N(C)C C12(CCNC(c3cc(CC)sn3)=O)CCC(CC1)C2.N1(CC=O)CCCC1C CC1CC(C(=O)N(CCNC(=O)CNS(N)(=O)=O)C(C)C)CC(=O)N1 N1(C(Cc2ccc(OC)cn2)=O)CCCC1C1CCCCN1C(=O)C#CC1CC1 Cc1coc(C(C)C)c1C(=O)N(C1CC(NC(=O)Cc2ncncc2Cl)C1)C c1(NC(C)=O)cccc(F)c1C(=O)NC1(CF)CCN(C(=O)CCCCCO)C1 C1(NC(C2CC3(C2)CC3F)=O)C=CCN(C(c2c[nH]nc2-c2ccncc2)=O)C1 c1(C(=O)NCC2CC(C)N(C(=O)CCCc3cnn[nH]3)C2)cc(F)c(F)c(F)c1 Cc1cc(C)c(C(=O)NCC2CC2)cc1N.c1(C=O)ccc(C(C)C)c(F)c1 c1(CNC(c2n(CC=C)nnn2)CSc2ccc(Br)cc2)ccc2c(c1)CCC2 c1(C(=O)NC(C2(O)CCN(C(c3ccccc3)=O)C2)C)c2ccccc2nn1C C1(C(=O)NCC2CCC2NC(=O)CC#N)(NC(C)=O)CCCc2ccccc21 C1(C(=O)N(C(C)CC2CC2)C)(NC(C(C)C2(O)CCC2)=O)CCN(C)C1 S(=O)(=O)(c1cccnc1NC)NC(C)COCC1CC1.c1coc(Br)n1 c1(CNC2CCCC(C(=O)Nc3cnn(CC)c3C)C2)ncc(Cl)cc1F c1(C(=O)NC2(C(N(C(C3CCCC3)C)C)=O)CC2(C)C)ccc(=N)[nH]n1 n1(CC)cnnc1C(=O)N.C1(F)CCC1.c1(C=O)c[nH]nc1C(C)(C)C.C c1(OCC)ccc(C(=O)N)cc1.C(C)CC.C1(N2CCCC2)(CC=O)COC1 c1(NC(c2cnn(-c3ccc(F)cc3)c2)=O)cc(I)ccc1-n1cnnn1 C1(CC(NOCCC)=O)CN(C(=O)C(CN(C)C)N(C)C)CC12CC2 n1(CC(=O)N(C2CCN(C(C3CC(CF)C3)=O)C2)C)nc2n(c1=O)CCOC2 C1(NC(C2(SCC)CC2)=O)C=CCN(C(c2cc(Br)c[nH]2)=O)C1 C1(c2c(Oc3cccc(C#N)c3)cccc2)CCCN(N2CC(OCCO)C2)C1 c1(SC)cccc(CC(=O)NCC2CCCN2C(=O)C(C)n2cnnn2)c1 c1(C(=O)NCCOCCCN)cc(=O)cc(Cl)[nH]1 c1(C(=O)NCC(CNC(=O)Cc2cncnc2)O)[nH]cc2c1CCC2 CC1CN(C(=O)CN2CCC2C)CCC1NC(=O)CCCCN(C)C c1(CC)ccccc1C(F)(F)C(=O)NCC1CC(NC(=O)C(C)C)C1 c1(CC)ccc(NC(=O)C(=O)NC2C=CCCC2)cc1S(N)(=O)=O N1(C(CCc2c(C)noc2)=O)CCC(F)(C(=O)NCC2(C)CC(C)(C)C2)C1 c1(C(=O)NC(C2(Cc3ccc(F)cc3)CCCC2O)CC)cc(Br)c(NC)cc1C O=C(N=c1cc(-c2ccc(Cl)cc2Cl)[nH][nH]1)NC1CC(n2cccn2)C1 N=c1ccc(C(N2CC3C(CNC(C4CC(=O)N4)=O)C3C2)=O)c[nH]1 N1(C(CC(C=C)(C)O)=O)CC2CC(C)N(C(c3nnn4c3CSCC4)=O)C2C1 C12(NC(c3cc(C)[nH]c3)=O)CCCCCC1N(C(=O)C1=NOC(C)C1)CC2 N1(C(CCC(=C)Br)=O)CCC(O)CC1Cn1cc(-c2cccc(N)n2)nn1 N1(C(CCCC(=C)C)=O)Cc2ccccc2C(CNC(C2(CC(C)C)CC2)=O)C1 CCC(CC)CC(=O)N1CCC(CNC(c2cc(C(C)(F)F)n[nH]2)=O)C12CC2 CC(CNC(=O)CC1CCCCCC1)C(F)C(=O)NCC1CCC(C)(C)O1 c1(C(C)C)ccc(Cl)c(C(=O)OCc2cnc(C3CC3)nc2)c1 C1(C=O)CC2(CCCC2)CO1.c1(SCCC(=O)NCC2CCC2)ccccn1.N N1(C(CCOCC(C)(C)C)=O)CCN(c2ccc(C(=O)N)cn2)CC1.C1(C)CC1 C=Cn1nccc1C(N1CCC(NC(=O)CO)C1C(C)C)=O.c1cnn(C)c1 C(CCCCC(=O)NCC1CCN1C(=O)C(C)(Cl)Cl)c1ccc(OC)cc1 N1(C(C#CCNC(C(C(=O)OCC)F)=O)=O)CC2(COC(=O)C2)C1 c1(C(=O)NCC2CN(C(C=CSC)=O)C(C)C2)c(N)cccc1F C1(O)(CN(C)C(c2cc(CO)n(C)n2)=O)CCCN(C(c2cnn[nH]2)=O)C1 C1(C(=O)NC(CC(C)C)CO)CCN(C(c2ccc(I)c(O)c2)=O)CC1O N#Cc1cc(Br)c[nH]c1=NCCC1CC(N(C2CC23CC3)C(c2ccccc2)=O)C1 N1(C(C(C(CC)C)c2ccccc2)=O)CCc2[nH]nc(C(=O)NC(C)(C)C)c2C1 C1(C(=O)NC2CC3(CN(C(C(C4CC4)OC)=O)C3)C2)(C)CC2C=CC1CC2 C1(C(=O)NCC(CO)NC(c2c(C)c(Br)cs2)=O)CC12CCOCC2 C1(CN(CCOCC)C(C)C)CCCC(N)C1 C1(NC(C2(C)CCC2)=O)C2CCC1CN(C(c1ccc([N+](=O)[O-])o1)=O)C2 C(=O)(C(C)(F)C(C)(C)F)N(CCCCCC(=O)NC1CC(CO)C1)C N1(C(CC2N(C(C3CNC(=O)C3)=O)C3C2CCC3)=O)CC2(CCNC(=O)O2)C1.C c1(SC)ccsc1C(=O)NCC(C1CCC1)NC(c1cnccn1)=O C(=O)(CC(C)C(F)F)NCCCCCN1CCN(C(COC(CC)C)=O)CC1 C1(NC(CN(C)C)=O)CCC12CCN(C(C1CCOC1c1nccn1C)=O)CC2 n1(CC(=O)N(C(CN(C(C2(CC#C)CCOC2)=O)C)C)C)c(C)csc1=O c1(C(N(CC(C(=O)NCC2CC(OCC)C2)C)C)=O)cncc(OC)c1 N1(C(c2c(C)n(C)c3c2cccc3)=O)CCCC(C2CCN(C(=O)C(N)=O)C2)C1 N1(C(COCCCN=[N+]=[N-])=O)CC2CCCC2(C(=O)NCC2Cc3nccn3C2)C1 C(C(COC)C(=O)N1CCCC1CC(=O)N(CCCF)C)OC Cc1nc2c(s1)CC(NC(=O)C(Cc1ccc(O)cc1)CC(C)(C)C)CC2 C(C(=O)NC1CN2CCC1CC2)(C(C)(C)O)NC(C(C)n1ccnn1)=O C(=O)(C#CC1(C)CCCO1)NC(CCN(C)C)C(=O)NCCC(F)(F)CO Cc1cccc(C)c1C(O)C(=O)NC(C)CC1CCN(C(=O)CP(C)(C)=O)CC1 N1(C(c2cc(C)nc(C)c2)=O)CC2CN(C(=O)C(O)CC(F)(F)F)CC(C1)O2 c1(CC(=O)N(CCCNC(C2CCOCC2)=O)CC)csc2nc(C)cn12.O C12(C=O)CC(CCO1)N(C(=O)CC=CC(C)(C)C)C2.CC(C)NCC.C n1(CC(=O)N(C(C)Cc2ccco2)C2CC2)cc(CCC(C)(C)O)nn1 c1(CN(CC(CC)C)C=O)cc2ccccc2nc1O N1(C(C(COC)OC)=O)CC(C(=O)NCC2(O)CC3CCC2O3)CC1(C)C Cc1cc(O)ccc1CC(N1CC(CCCC)C1)=O.C1(CC(=O)N)CCC(C)(C)C1 c1(-c2cc(N(C)C)ncc2)c(C(N2CC3CC3C2)=O)nc2ccccn12 C(CNC(=O)C(C)CN(C)C)(CCNC(C1CCN(C)C1)=O)OC N(C1CCc2ccccc21)C(C1(C)CC(C)(C)N(C(C2OC3CCC2C3)=O)C1)=O c1(N2CCC(N(C(=O)CC3CC3)CCC)CC2)cc(Cl)nc(C(=O)OC)n1 N1(C(CSc2c(OC)cccc2)=O)CC2CCN(C(c3[nH]nnc3C)=O)C2C1 Cn1cc2cccc(C(N3CCCC3CCNC(C3(F)CCCOC3)=O)=O)c2n1 Cc1ccn(CC(=O)NCC2CCCCN2C(c2cnc(C)[nH]c2=N)=O)c(=O)c1 N1(C(=O)C(F)C(F)(F)F)CCC2CCN(C(c3cc(Cl)nnc3O)=O)C2C1 N1(C(CCC=C=C)=O)CC2CCN(C(=O)C=CCN3CCOCC3)CC2C1 CC1CN(C(=O)CC2CCC3CC3C2)CCN1C(=O)CNc1ccccc1 N1(C(C2CC(C)OC2=O)=O)CCN(C(=O)C(C)(C)C)CCC1C C(=O)(CC(C(C)C)c1ccccc1)NCC1CN(C(C2(SC)CCC2)=O)C1 N1(C(c2c(CC)occ2C)=O)CCC(C(=O)NC2CCN(C)C2)CC1(C)C C1(N(C(=O)C(=O)Nc2cnc(Cl)c(Br)c2)C)CCN2CCOC1C2 c1(C(=O)NC2C(NC(C(C)CC(C)(C)C)=O)COC2)cc(Cl)cc2ccncc12 C1(C(N(CC)C2CC2)=O)CN(C)C(=O)CCO1.c1(OC)ccc(C(=O)N)s1 N1(C(CC(=O)NCC#C)=O)CCC(C)(NC(=O)C(CCC)OCC)C1 Cc1cc(C(=O)NCC2CC(C)(C)CN2c2cc(Cl)nc(C)n2)c2c(c1)CCO2 C1(NC(c2nc(CCCCC)sc2)=O)CC(F)CN(C(C2(N(C)C)CCC2)=O)C1 c1(C2C(C(=O)NCC3N(C(c4ccn(C)c4)=O)CCC3)CCO2)ccc(F)cc1 N1(C(c2cnns2)=O)CCC2CN(C(=O)C(c3cccc(F)n3)(F)F)CCC2C1 C(=O)(C1=CCCC1C)NCc1nc(C(N2CCC(OC)C2)=O)c(C)s1 [N-]=[N+]=Nc1cncc(C(=O)NC2(C)CCOCC2)c1.c1(C(=O)N)cc(Cl)c(Cl)[nH]1 C1(C(N(CCC(F)(F)F)CC)=O)CC(NC(=O)CCCSC)CCO1 c1(CN2CCC(N(C(=O)CC3CCCC(=O)N3)C)C2)nnc(S(C)(=O)=O)s1 C1(CC)CN(C(c2c(I)n[nH]c2C)=O)CCN1C(=O)C(C)CC N1(CC=O)CCN(C(C23CCN(CC2)C3)=O)CC1.C(=O)(OCC)NCC N1(C(CC(C)O)=O)CCCCC(CCC(=O)NCCc2ccc(F)nc2)C1 C(C(C(=O)NCc1cc(C)on1)C(C)C)NC(C(C(=O)OCC)F)=O C1(C(N2CC(OC)C2)=O)CC2(CC(NC(=O)CC)C2)C1.C(=O)C1CC1.N CCC(C)C(C)(O)CNC(=O)C(C)N(C(=O)Cc1cccnc1O)C1CC1 c1(C(N2CCN(C(C3CN(C)C(=O)C3)=O)C(CO)C2)=O)cccc2nc(O)oc12 N1(C(C)C)CCN(CCC(N2CC(NC(c3cncn3C)=O)C3CC23)=O)CC1 c1(C(=O)NC(CCNC(C(C)(C)OCCOC)=O)C)ccccc1.CC#N N1(C(CCNC(COC)=O)=O)CCN(C(C2CCC(OCCN)CC2)=O)CC1C C1(NC(C(c2nnc(C)s2)N(C)CCOC(F)F)=O)CCC(F)(F)CC1 CC(CCCC(=O)Nc1cccn(C(F)F)c1=O)NC(=O)C1=CCCC1 CCC=O.C(=O)CC.C1(N(CC=O)C(C)(C)C)CCCC1.C(=O)C1CC1 N(C(=NCCC1CC1C1CC1)N1CCCC(CC(N)=O)C1)CC(C)C c1(C(=O)NCC(C(C)C)NC(CCNC(=O)OC)=O)cc(C)ncc1C c1(CN(C=O)CC2(Br)CC2)cnn[nH]1 C(=O)(C(C)S(N)(=O)=O)N(C)CC1N(c2nccc(SC)n2)CCC1 C=CC(C)(O)CC(=O)N(C1CCN(C(c2cccc(Cl)c2C)=O)CC1)CCO C1(NC(c2cc(C)c(F)cc2N)=O)CN(C(C2CC2[N+](=O)[O-])=O)C2(CCCC2)C1 CC1CCN(C(=O)OC(C)(C)C)C1C(N1CCCC1c1ccc(Br)cc1)=O C1(CN(C(C(C)OCC#C)=O)C)CCCN1C(=O)CCCO.c1cccnc1 c1(C(N(CC(CC)NC(c2cnc(O)cc2OC)=O)CC)=O)cnc2sccn12 c1(C=O)cc2cc(Cl)sc2[nH]1.c1(OC)ccnc(NCC(=O)N(C(C)C)C)n1.N C#Cc1cccc(C(N2CC=CC2CNC(=O)CC23COCC(C2)C3)=O)c1 C1(NC(CSC)=O)C(C)CN(C(=O)CCCc2ccncc2)CC1C Cc1[nH]nc2c(C(=O)NC)cccc12.C1(C)CC(F)(F)CN1C(=O)C(F)C(C)C C(=O)(C(C)(C)C(O)C(C)C)NCCC1(O)CN(C(COC)=O)C1 c1(C(N2CC(C)C(NC(C3(C)CCN(C)C3=O)=O)C2)=O)c(F)ccc2ccoc12 Cc1cccc(CNC(=O)C(Cc2ccoc2)NC(c2snc(C)c2N)=O)c1O c1(NC(C)=O)ccc(Cl)c(CN2CC(NC(=O)C)C(F)C2)c1.c1cccnc1 C1(CC(=O)NCCC(=O)N(C)C)C2CN(C(c3ccc(O)nn3)=O)CC12 c1(NC(N2CCN(CC3CCCSC3)CC2)=O)ccc(Br)cc1Cl c1(CC)c(C(=O)NCCCN(C(=O)C)C2CC2)cnn1C.c1ccccc1.O c1(OC)ccccc1OCC(=O)NC1CN(C(c2c[nH]c(=N)s2)=O)C2CC12 C1(C(=O)OCc2cccc(OC(F)F)n2)CC2CCCCCCC12 CC1c2cc(F)ccc2CCN1C(CCCC(C)(F)F)C(=O)NCCCF C1(C(=O)NC2C(CNC(CN(C)CC)=O)C2)CSc2ccccc2O1 Cc1cc(C(=O)NC2CC3CC2CN3C(=O)CCc2nc(O)n[nH]2)cc(C)c1Cl C1(C(=O)NC(C2CN(C(CN(C)CC)=O)C2)C)CCC(C)(C)OC1 CCC(CC(F)(F)F)C(=O)NCC1CCCC1.C1(CC(=O)N)SC(=N)NC1=O C(=O)(CC(C)(C)C1CCCCC1)N(C1CCN(C(C2CCC(=O)C2)=O)C1)CC N1(C(C2N(CC)CCC2)=O)CC(NC(=O)CCC(N)=O)C(n2cccn2)C1 N1(C(CC2(OCC)CCC2)=O)CC=CCC1C(=O)NCCC(C)(C)CC c1(CNC(CN2C(C)CCC2)=O)cccc2c1CN(C(C1CC3C=CC1O3)=O)C2 c1(C(=O)NC2C(NC(C3C(C#C)C3)=O)CCCC2)ccc(C(=O)OC)cc1Cl CC1(C)CN(C(=O)C2CC2)C(CNC(=O)C)CO1.C(=O)CCO.C(N)=O c1(CC)ccc(C(=O)NCCC(C)(C)NC(=O)Cc2conc2C)cn1 c1(CCN(C)C(c2ccc3ccoc3c2)=O)ccc2ccccc2c1 c1(C(N2CC(SC)C(NC(c3cc(C#N)c[nH]3)=O)C2)=O)c(F)ccc2c1OCO2 C1(NC(C(C(=O)OCC)(C)C)=O)C2Cc3ccc(Br)cc3C12 CCC(CCCC(=O)NC(CN(C)C)CCO)NC(=O)Cc1ccns1 C1(C(=O)NCC(C)(CC(C)C)NC(c2c(C)cco2)=O)CC(C2CCCC2)C1 c1(OC(C)(C)C)ccc(CCNCCc2ccc(OC3CCCC3)cc2)cc1Cl n1(C2CN(C(=O)CCc3nccs3)C2)cc(CNC(C2(F)CCC2)=O)nn1 C1CN(C(c2cccnc2)=O)C2(CCC2)C1.C1(C(=O)NC)CCC(C(F)F)CC1 C(c1ccccc1)=CC(=O)N(CCOCCNC(C1CC(=C)C1)=O)C.S C1(O)(CCNC(CN(c2ccccc2)C)=O)CCCN(C(=O)CC2=CCCC2)C1 c1(CNC(CC=C(C)C)=O)ccc(C(=O)NCC(C)OCCO)s1 C1(C(N(CCNC(C2C(C(=O)OC)C2(F)F)=O)C)=O)OCC2CCCCC12 c1(-c2cnc(NC(c3ncccc3F)=O)s2)cncc(C(F)(F)F)c1 c1(CSC)cccc(CN)c1.C12CCCCN1C2.c1cnn(C2CCCCO2)n1 CCCCCCC(O)CCC(=O)NC(C1CCCN1C(=O)C(F)CC)(C)C CC(C)C#CC(=O)NC(C1CC=CCC1)C(=O)N1CC(CF)C1 c1(CC(=O)N(C(C)CCNC(C2CC(O)CN2C)=O)C)cc2ccccc2s1 Cc1cc2cc[nH]c2cc1NC(=O)C(N1CCC(C)C(CO)C1)=O Cc1cc(C(=O)NCC2CCC2NC(=O)C(C)(C)CC#N)ccc1Br Cc1ccc(NNC(=O)c2c(C)cnnc2O)c(Cl)c1 C(=O)(CC(O)(CCC)CCC)N1CC(NC(CCCC#CC)=O)C(SC)C1 C1(F)(C(=O)NC(C2N(C(c3c(C)oc(Cl)n3)=O)CCC2)C)CCS(=O)(=O)C1 C#Cc1ccc(CC(=O)NC2CC2CNC(=O)Cc2cnc[nH]2)cc1 CC(CNC(=O)Cn1cc(-c2ccc(C(F)F)cc2)nn1)C(F)(F)F C=CCC(C(=O)OCC)NC(=O)C(=O)NC1CC(C#N)C1 c1(OC)cc(NC(N2CCC(C)(C)C(CO)C2)=O)ccc1S(C)(=O)=O Cc1ccc2cc(C(=O)N(C3CCC(NC(c4ccsn4)=O)CC3)C)[nH]c2c1 CC1CC(NC(c2ccoc2CC(N)=O)=O)CN(C(=O)CN2CC3CC3C2)C1 CC(C)C(CCC(=O)N1Cc2ncsc2C1)NC(c1ccccn1)=O Cn1cc(C(O)C(=O)N)cn1.C1CCCN1C(C1(CS(C)(=O)=O)CCC1)=O.C c1(CC)nccnc1C(=O)N(C1CCCN(C(C2C3CCN2CC3)=O)C1)CCO Cc1cc(C2CC2)cnc1C(=O)NC1CC(CNC(=O)CC)C1.C1COC1 C1(O)(C(=O)NCCC)CCCC(C)(C)C1.c1(C(C=O)(F)F)ccc(Cl)c(Cl)c1 CC(c1nc(C(c2cccc(C)n2)C)no1)=CC(C)(C)C C1(N(C(=O)C(F)C(F)(F)F)C)CC2CCC(C1)N2C(c1cccc2nncn12)=O C1(C2CCN(C(C(CC3CC3)OC)=O)C2)CCCCN1C(=O)C=CCO c1(C(=O)NCC(N(C(CCOCCCOC)=O)C)C2CC2)cccc(F)c1 c1(CNC(CN(CCC)C)=O)cccc2c1CN(C(C1(CC)COC1)=O)C2 Cc1sc(C(N2CCCC(CCNC(=O)C3=NOCC3)C2)=O)cc1Br N1(C(C2C(F)(C=O)C2)=O)CC(C2CC2)C1.C1(=CC=O)CCC(C)C1.C Cc1csc(CC(C)NC2CC2c2ccnn2C)n1 C1(C(N2C3CN(C(c4c(C)nn(C)c4C)=O)C(C3)C2)=O)CC2CC(C1C)C2(C)C C(CC(C(=O)N1CCCC(CC(N)=O)C1)NC(=O)C(C)C1(O)CCC1)OCC C(=O)(C(=O)CC(C)C)NC(C(=O)NCc1n(CC)c(C)nc1)C1CCCC1 C(=O)(C1=COCCO1)NCCOC1CN(C(CC2(C)CCOCC2)=O)C1 C(=O)(CS(=O)(=O)C1CCCC1)NC(C(C)C)CC.C(=O)(C(F)(F)c1cscn1)N C1(NC(COCCCOC)=O)C=CCN(C(C2CCC=CCC2)=O)C1 c1(OCC(N2CCC(NC(C(C)c3ccsn3)=O)(CF)C2)=O)ccccc1C#N Cc1cccc(CNC(=O)C(C2CCCC2)NC(c2ccnn2CCF)=O)c1F c1(C(=O)NC(C(C)NC(Cc2cccc(C)c2)=O)C(C)C)ccn2ncnc2c1 Cc1cc(CNC2C3CCC2CN(C(C2(Br)CC2)=O)C3)c(O)c(Br)c1 C#CC1CN(C(c2cnn(CC)c2)=O)CCN1C(c1cc(C2CC2C)on1)=O C(c1ccccc1Cl)=CC(N1CCC(OCCNC(CCOCC#C)=O)C1)=O N1(C(C)=O)CC2CCN(C(=O)C=Cc3ccc(O)c(O)c3)C2C1 C(=O)(C(CNC(=O)Cn1cnnc1)CC(C)C)NC(CC)(C)C(=O)OC C1(CC)CN(C(=O)CN2CCN(C)CC2)CCC1.c1(C(=O)N)ccc(=O)n(C)c1 Cc1cccc(O)c1C(=O)NC1CCCCC1NC(c1cc(O)nc(Cl)c1)=O c1(C(=O)NCCCN(C(c2ccnc(Cl)c2N)=O)CC)cc(F)c(F)cc1Cl C#Cc1cccc(NC(C2(C#C)CCN(C(c3cc(C)nnc3O)=O)C2)=O)c1 c1(C(=O)NCC2CN(C(C(C)c3ncco3)=O)C2)ccn(CC(F)(F)F)n1 C#CC1(O)CCN(C(C23CC(CN2C(C2CCCCC2O)=O)C3)=O)C1 C(=O)(CCCS(C)(=O)=O)NC(CC(C)NC(C(c1scc(C)n1)(F)F)=O)C c1(C(=O)NCC(C(=O)NC2(CC)CC2)(C)CC)cnn2ccc(Cl)c(F)c12 C(C)(C)(CC(=O)OC)NC(C(C1CN(C(C(C=CC)O)=O)C1)OC)=O C=C(C)CN=C(NCc1cc(CC)ccn1)NC1CCOC(CC(C)C)C1 C1(C(N(C(C)CCNC(=O)CCc2cnoc2)C)=O)C2CCC1(c1ccco1)C2 N1(C(C(CC)F)=O)CC2CN(C(=O)C(c3ccc(NC(C)=O)cc3)=O)CC2C1 c1(C(N2C3CC(CNC(C(C#C)(C)C)=O)C2CC3)=O)[nH]c2c(Cl)cccc2c1C N1(C(=O)C(F)(F)CO)CC2(C(=O)NCC34CCCC3CCO4)CC1CO2 C#CC1(NC(C2CCN2C(c2cc(N)ccc2Br)=O)=O)CCOCC1 Cc1cc(Cl)cc(C(=O)NC2CN(C(=O)CCCNC(N)=O)CCC2CO)c1C C1(C(=O)NCc2ccc3c(c2)CCNC3)CC(c2cccnc2)=NO1 c1(C(=O)NCC(CN(C(CCOC)=O)C)C)cnoc1-c1cccs1 C(=O)(C1=COCCC1)N1CCCC(CC(=O)NCC2C(=O)NC(=O)N2)C1 CCC1=C(C(=O)N2CCC(O)(C(C)NC(=O)C(=O)NC3CC3)CC2)CCCO1 c1(C(=O)NC2CCC(NC(c3c(CC)scc3)=O)CC2)ccc(N)c(N)n1 N1(C(C2CC(O)(CC#C)C2)=O)CCN(C(=O)C(C)n2ccnc2)CC1CO c1(C(N(CCCCNC(=O)CC2CCC(=O)N2)C)=O)ccc(CCO)cc1 C1(CNC(c2c(F)ccc(C)n2)=O)CN(C(C2CCOC2C)=O)CC12CCC2 N1(C(C(c2ccc(C)cc2)O)=O)CCN(C(=O)CCc2cnc[nH]2)C(CCO)C1 N1(C(C(CCC)NC(C)=O)=O)CCC2(C(=O)N(CC(C)(C)COC)C)CCCC12 C(=O)(C(CCC)O)NCC(C1N(C(C2CC(O)(CC#C)C2)=O)CCC1)(C)C C1(CC(=O)O)CCCCN1C(=O)COc1nn(-c2cccc(F)c2)cc1O c1(C(=O)OC)ccc(C(=O)NC2CCN(C(c3cnn(C)c3)=O)C2)nc1 c1cc(Cl)ccc1Cl.C1(CNC(C(COC)NC(C)=O)=O)CC(C)N(C)C1 N1(CC)CCCC1C(=O)N(CCC(=O)NC1(C(N)=O)CCC1)C C(=O)(C1=CCCC(C)(C)C1)N(CC(C)(C)CNC(c1cccnn1)=O)CC C(=O)(CCC(C)NC(=O)CC1C=CCC1)NC(CCC)CO C(=O)(C(C)CC(=O)N1CCOCC1CNC(=O)CNS(C)(=O)=O)OC c1(C(=O)NC2CCC(NCc3cc(C)cc(O)c3)C2)cnc2cc(C)nn2c1 c1(CC(=O)NCC2C(C)CCN(C(C(CC)COC)=O)C2)ccc2nn[nH]c2c1 c1(C(=O)NCCNC(=O)COc2cncc(Br)c2)cc2ccccc2s1 Cc1cc(C#N)sc1C(N1CCCC1C(C)(C)C)=O.C1(CC(=O)N)CCCSC1 C(CC(C)(C)CBr)(c1nnnn1CC1CCCO1)NC1(CC)CCCC1 C(CC(C)C)(C(=O)Nc1cnn(C(C)C)c1)N(C(C1CCCC(OC)C1)=O)C Cc1c(O)ccc(C(=O)N(C2CN(C(=O)C3=CCCC3)CC2(C)C)C)c1C CCCC(O)(CCC)CC(=O)N(C)CCC1CCCCN1C(=O)CS(=O)CC c1(SCC(=O)NC(CC)CNC(=O)C(C)C#N)ccc(Cl)cc1[N+](=O)[O-] C12(NC(C(CCC)=CCC)=O)CCC(CNC(c3ccoc3)=O)(CC1)OC2 C=CCCN=C(NCc1ncccc1C)N1CC(C)CC(C)C1 c1(C(N2CC(C)(CNC(C3C(=C)CC3)=O)C(C)C2)=O)cc2[nH]nnc2cc1OC C(C)(C(C)(C)C(=O)N1CCC(C#N)C1)NC(C(SC)SC)=O N1(CC(=O)NCCC2(C(=O)O)CCCC2)C(=O)C2C3CCC(O3)C2C1=O N1(C(C2CCC(CC)O2)=O)CCC2(CCCN2C(=O)Cc2cnnn2C)C1 C=C(C)CCCC(=O)N1CCCC(NC(c2ccc(N)c(O)c2)=O)C1 Cc1oc(CO)cc1C(=O)NC(C1(C(=O)NC(C)CC(F)(F)F)CC1)C C(=O)(C1=CCCC(C)(C)C1)NC1CC2CN(C(c3cn(C)nc3C3CC3)=O)C1C2 CCC(CC)C(C(=O)Nc1cc(Cl)ccc1OC)OC n1(CC(=O)NCC(CC)N(C(=O)C(O)CC)C)cnc(=N)[nH]1 Cc1cc(C)n(CC(=O)N(CCCN(C)C(c2ncc(F)cc2N)=O)C)c(=O)n1 c1(OCC(=O)N(C)C)ccc(NC(c2ncsc2C(F)(F)F)=O)cc1 C1(C(=O)NCC2C(C(N3CC(O)(C(C)C)C3)=O)OCC2)CC=CCC1C N1(C(C(C)NS(CC)(=O)=O)=O)CCC(C2CCN(C(C3CC34CC4)=O)CC2)CC1 C(CCCC(C)NC(C1CCCN(C)C1)=O)NC(CC(C)C1CCCCC1)=O CCC(COC)C(=O)NCCCN(C(=O)C=Cc1ccccc1)C Cc1nc(O)ccc1C(=O)NOCC(=O)NC(C)(CO)CCF c1(C=O)ccc2c(c1)nnn2C.C(=O)(C(C)(C)C)NCCC(=O)NCCCC CCCCCC(O)C(=O)NC1CCN(C(=O)CC2CCOCC2)C1 C(=O)(C1=Cc2ccccc2C1)N1CC(C)C(NC(c2snc(O)c2Cl)=O)CC1 C(=O)(C1CCCc2cncn21)NCCCC1CCN(C(C(CC#C)(C)C)=O)CC1 C#Cc1cc(C(N2CCN(C(=O)C(COC)NC(C)=O)CC2C)=O)cc(F)c1 C1(C2CCN(C(c3nccc(C(F)F)n3)=O)C2)CC1.c1(SC)ccc(C(=O)N)o1 N1(C(C2CC(CC)C2)=O)CC(C)(OCC(N2CCC(C(F)(F)F)C2)=O)C1 c1(C(=O)OC)cn2cc(CNC(C3CC4CCCCN4C3)=O)ccc2n1 Cc1cc(C)n(CC(=O)NC2(CNC(=O)C(C)(C)C)CCOC2)n1 c1(C(=O)NCCC(C)CCNC(=O)Cn2cc(C#N)cn2)nc2cnccc2s1 c1(C(N(CCCN(C(CCC(C)OCC)=O)C)C)=O)c(C)ccc2nsnc12 CCCC(C(O)C(=O)N(CC)CC1CCOCC1)NC(c1cnc(C)s1)=O N(C(=NCCCOC(C)(C)C)NCCCN1CCCC1)C(C1(O)CCOC1)C C(=O)(CS(=O)(=O)CC)NCCCCCN(C(C(CCC)NC(N)=O)=O)CC S(=O)(=O)(c1cccnc1NCc1csc2ccccc12)N1C(COC)COCC1 C1(NCc2c(CC)cccn2)CCC2(CCNCC2)C1 c1(C(=O)NC(C)CNC(=O)CN(C)C)ccc(I)nc1 Cc1cnn(C)c1C(N1CC(NC(c2cncn2C(C)C)=O)C(F)C1)=O N1(C(C23CC(C(C)(C)C)(C2)C3)=O)CCOC(C)(C)C1.c1(C=O)cnccn1.N CC1(C)CC(C(N2CCOCC(F)(F)C2)=O)CCN1C(=O)CCc1cncs1 C1CC(F)(F)C1.c1(C=O)cc(C2CC2)ns1.C(CCNC(=O)CO)OC C1(NC(=O)CN(C(=O)CC2CCCOC2)C2CC2)CN2CCC1C2 c1(C(=O)NC(C)C)ccc(CCC(=O)NCc2nn[nH]n2)[nH]1 C#Cc1cccc(C(=O)NC2CN(C(=O)C=CC=CCCCCC)CCC2F)c1Cl c1(CC)cc(Br)cnc1NC(N1CCCC(n2nc(C)nc2C)C1)=O CC1(C)CN(Cc2ccc(Br)s2)CC1NC(=O)CCC1CCCOC1 C1(CNC(C=CC=CC)=O)CCN(C(=O)C(O)C)C1.c1ccccc1.O C(=O)(C(C(C)O)N(C)C)N.C1(C(=O)NC(c2ccnn2C)C)(CC)CCCC1 C1(NC(c2cn(CCC=C)nn2)=O)C(C)CN(C(C2CC3(CCC3)C2)=O)CC1C c1(C(N2CCCC2)=O)cc2ccc(C(C)=O)cc2[nH]1.C(C(C(=O)NC)OC)OC N1(C(Cc2c(OC)cccc2)=O)CCOC2CCN(C(C3CC3C#N)=O)CC12 C1(OCCCCC)CCC(C(N2CC(N(C3CCC(=O)NC3)CC)C2)=O)CC1 CC1(C)CCCN1C(=O)C.c1(C(=O)N)cccc(CS(N)(=O)=O)c1.C1CC1 c1(C(=O)NC2CC(C)N(C(=O)C(F)=CC3CC3)C2)ccc(Br)cc1O N1(C(C2CC3CCCC3C2)=O)CC2CCC(C1)N2C(=O)COC1CCOCC1 C1(C2CCN(C(c3cnc(C(F)F)s3)=O)C2)(NC(c2ccc[nH]2)=O)CC1 C1(C(N(C)Cc2ccccc2)=O)CN(S(N)(=O)=O)C1.C(=O)C(CO)N(C)C c1(C(N2CCCC(NC(c3c(C)occ3)=O)C2C)=O)ccc2ccccc2n1 C1(CNC(C2OCC(C)(C)C2)=O)CC2(CC2)CN1C(=O)CCC1CCCCC1 Cc1cc(Cl)ccc1C(=O)NCC(C(C)(C)C)NC(C1(C)CNC(=O)C1)=O CC1CN(C(c2c[nH]nc2-c2ccnn2C)=O)CC1CNC(c1nnn(C)n1)=O c1(C(N2CCN(C(c3cnc(C)[nH]c3=N)=O)CC2)=O)cn2ccc(CO)cc2n1 c1(CNC(CSCC#C)=O)ccsc1C(=O)N.C1CCOC1C(C)C.C c1(C(N(C(C)C)CC)=O)c(F)cc(N)cc1F.C1CCC(C)CC1.C(=O)C.N c1(C(=O)NC(C(C)NC(C2(CF)CCOCC2)=O)CO)[nH]nc([N+](=O)[O-])c1Cl c1(C(N(CC(C)NC(=O)C2=COCCC2)C)=O)cc2n(n1)CCO2 C1(C(C(=O)NC(c2ncn(C)n2)C)C)CCN(C(=O)C)C1.CCN(C)C.O N1(C(CCc2c(C)nn(C)c2)=O)CCOC(C)(C)C1.C1(CC(C)C)(C(=O)N)CC1 c1(C(=O)NCCC(C)(C)NC(=O)C(F)=CCCF)cccc(C(F)F)c1F N(C1CS(=O)(=O)c2ccccc21)Cc1c2ccc([N+](=O)[O-])cc2sn1 CC1(C)C2CCC1(C(N1CCC3(CNC(c4n[nH]cc4Cl)=O)CCCC13)=O)CC2 C1(C(=O)NCC2CCCOC2)(NC(C(C)c2ccsc2)=O)CCCCC1 C#CC1CCCN(C(=O)CC2CC(O)CN2C(C2CC3(CC3)CO2)=O)CC1 c1(SC(C)C)ccccc1C(=O)NCCCCF.c1(C(C=O)F)ccccc1 N1(C(c2cn(CC)nc2)=O)CCC(N(C)Cc2cccc(Cl)c2)CC1 c1(OC)cc(C(=O)NC2CCN(C(c3c(F)cccc3Br)=O)CC2F)cc(C)c1 C(CC(C)(C)C(=O)NC(C)Cc1ncn(C)n1)NC(c1cc(C)ncn1)=O S(=O)(=O)(c1ccc(CCC(N2CCCCC2CNC(=O)CCO)=O)cc1)NC CC1(NC(=O)C=CC2CCN(C(C3CCOC(=O)CC3)=O)CC2)CC2CCC1C2 O=C(C1SCc2cccnc21)NC1CCCN(C(C2CC(CF)C2)=O)C1 c1(C(=O)NC(CNC(Cc2cc(OC)no2)=O)C(C)C)oc(SC)cc1C C(CNC(=O)CCCN(C)C)(CC(=O)N1CCC(C)(C(N)=O)C1)OC c1(C(=O)NCCOCC(N2CCC(O)CC2)=O)ccc(Cl)c(Cl)c1.C1CC1F Cc1cn2cc(C(N3CC(NC(c4cc(C)c(C)s4)=O)CC(O)C3)=O)nc2s1 C12CC3CC(CC1C3)C2.C(CC(C(=O)N)NC(=O)C(N1CCCCC1)C)OCC C(=O)(C#CC1(C)COC1)N1CCN(C(Cn2cccc(C)c2=O)=O)CC1C1CC1 C1CCS(=O)(=O)C12CN(C(c1cncs1)=O)C2.C(C1CC1)(C1CC1)=CC=O.N CN=c1[nH]cc(C(N2CCC(N(C)CCOCC(O)C(=O)OC)CC2)=O)o1 C(=O)(CC(C)P(C)(C)=O)N(CC(C)O)CCNC(=O)C=C1CCCCC1 c1(C(N2CCC2)=O)cccc(S(=O)(=O)C(F)F)c1.CC(CF)CC(=O)NCC.O Cc1cc(O)n2ncc(C(=O)NC3(CCNC(C4CC4CF)=O)CC3)c2n1 N1(C(c2ccc(C(C)=O)[nH]2)=O)CC(NC(=O)C(c2ccccc2Cl)O)CC(C)C1 N1(C(Cc2c(C)cccn2)=O)CC(C2(NC(=O)CN(C)C)CC2)C1 c1(C(=O)NCC(CCCC)NC(c2cc(F)c[nH]2)=O)cc2occ(Br)c2[nH]1 CC(C)C(=O)COC(c1cc(-c2ccc(Cl)s2)[nH]n1)=O C1(NC(C2C(C)N(C)CC2)=O)CCC12CN(C(=O)CC(C)(C)C)C2 c1(OCC)oc(C)nc1C(=O)Nc1ccccc1.C1(Cl)(C=O)CC1(C)C.N CC1CCOCCN1C(=O)COC1(C)CN(C(c2csnc2Cl)=O)C1 c1cncc(C(C)(C)C)c1.n1(CCOCC)nnnc1C(C1CCSC1)N.C c1(C(=O)N)ccc2c(n1)OCCO2.C(C(C)C(C)C)NC(CCSCC(C)C)=O C1CCCCC1.c1(N(C)C)sccc1C(=O)NCCNC(=O)CC1CC=CC1 C12(NC(c3cccc(CC)c3)=O)CCCN(C(C3(COC)CCC3)=O)CC1C2 C=C1CC(C)(C(=O)NCCCOCCCNC(C2CCCN2C)=O)C1 N1(C(CCc2ccc(N(C)C)nc2)=O)CCN(C(=O)CCc2cscn2)C2CC12 Cc1nn(C)c(C)c1C(=O)C(N1CCCC(NC(c2ncc(Br)cn2)=O)C1)=O c1(C(N(CC(C)NC(CCCNC(C)=O)=O)C)=O)ccccc1.CC(N)=O.S C(N=c1[nH]c(N2CCC(CO)C(F)(F)C2)nc2c1SCC2)c1nccc(C)c1F Cc1cc(NC(C2CC3CC3C2)=O)ccc1NC(c1cc(C)c(C)o1)=O C1(C2CCC2)(C(N2C3CC(CNC(c4nccs4)=O)(OC3)C2)=O)CC1(F)F C1(NC(C(CCCC)NC(c2sc(O)nc2C)=O)=O)CCCCCC1(C)C C(C)(CCC(=O)NC1CCC(C(=O)NCCC(F)=C(F)F)CC1)SC C(=O)(CS(=O)(=O)C(C)C)N1C(CCNC(Cc2cc(C)c(O)cc2)=O)CCCC1 c1(CC(=O)NC(c2ccnn2C)C(N2C(C(=O)NC)CC2)=O)cn[nH]c1.C C1(OC)CCC2(C(=O)N(CCCCCCNC(=O)Cc3nnc(C)o3)C)CC12 c1(OC)cc(C=O)ccc1.C1(CC(F)F)(C(N(CC)C)=O)CCC1.C(C)C.N C(=O)(C(CCC1CCC1)NC(=O)Cc1cscn1)NCC(CCOC)O C(CCCCCC(=O)N1CCC(F)(CF)CC1)NC(C1(C#C)CC1)=O C(C=O)(C(C)C)NC(C)=O.c1(C(C(=O)N(CC)C)=O)cnn(C)c1.CC.N C1(NC(C2(C#C)CCC2)=O)CC2(C1)CCC2.C1(CC=O)CCCC1.C(=O)C C1(NCC(c2ccsc2)OC)CCCCC1(OC)OC Cc1cc(Br)c(C(=O)NC(C)CC(C)NC(=O)CSC2CC2)nc1C c1(C(N2C(C(=O)N(CCCC(O)CO)C)(CC)CCC2)=O)cccc(C#N)c1 c1(C(=O)NCC2C(C)CCN2C(C2(O)CCCC2)=O)ccn(CCO)c(=O)c1 S(=O)(=O)(c1cc(Cl)c(Br)cc1F)N1CCCC(C(N2CCC(F)C2)=O)C1 C1(NC(CCOC(C)C)=O)CC2CCCC2C1.C(=O)(C(C)(C)Cc1cnn[nH]1)N Cc1cc([N+](=O)[O-])cnc1C(N1CCN(C(C2CC(O)CN2C)=O)CC1)=O c1(C2(C(N(CC(CC)NC(CN(CCC#C)C)=O)C)=O)CC2)ccc(Cl)nc1 CCCCCC(CC)C(=O)N1CCC(O)(CNC(=O)C(C)CCO)CC1 N1(C(c2ccc(C)s2)=O)CC2CCCC(C1)N2C(c1cnc(C(N)=O)cn1)=O C1(C)(CNC(C(C)O)=O)COCCN(C(=O)Cc2cc(F)cc(F)c2)C1 C1(NC(CCC#CC)=O)CN(C(c2n[nH]c3c2CCOC3)=O)CC12CCOCC2 C1(C(=O)NC(CCC=C)C)CN(C(C2(CC)CCCO2)=O)CC1NC CCCC(C)CC(=O)NCC1CCC(C(=O)NCc2nncn2C2CC2)C1 N1(C(=O)OC(C)(C)C)CCCC2CC(NC(=O)C3SCc4cccnc43)CCC12 Cc1nn(C)c(C)c1OCC(=O)NCC1CCN1C(c1ccccc1O)=O S(=O)(=O)(c1[nH]c(=NCC2(CC#N)CC2)ccc1Br)NCC(C(C)O)(C)C N1(C(c2ncn(C)c2)=O)CCCC2CCN(C(c3ccc4c[nH]nc4n3)=O)CC12 C1(NC(C2(O)CCC2)=O)CCCC(NC(C2CC(O)C2)=O)CC1 c1(N2CCC(N(C(=O)C=CC3CCC3)C)CC2)ncnc(Cl)c1[N+](=O)[O-] C1(C(=O)NCCC2CCN(C(C3CC3C3CCC3)=O)CC2)Cc2ccccc2O1 N1(C(COCCOC)=O)CCOC2CN(C(C3(C)CCN(C)C3=O)=O)CC12 C1(NC(CC(C)c2ccco2)=O)CC2(CCCN(C(=O)CCCF)C2)C1 C1(NC(C2C=C(C)CS2)=O)CCCCCC1C(=O)NC(C)CC(C)(C)O c1(C(=O)NC2C(C=C)CN(C(=O)Cc3c[nH]nc3C)C2)ccc([N+](=O)[O-])cc1 N1(C(c2cccc(F)c2OC)C(=O)NCCOC)CC2CN(C3CCC3)CC2C1 Cc1cc(=O)n(C)cc1C(=O)NC1CC(C(C)NC(=O)CCC2CCC2)C1 N1(C(C2N(C)CCC2)=O)CC(NC(c2cnn(Cc3ccccc3)c2)=O)C(O)C1 N1(C(CNC(CCC)=O)=O)CCC(C2CC2)C1C(=O)NCC(O)CC(F)(F)F N1(C(CC2C(OC)COCC2)=O)CC(C)(CO)C(C)(CO)C1 C1(C(=O)NC(C2CCOC2)C)CC(C)CN1c1ccnc(C2CC2)n1 Cc1nc(C)c(CN=C(NC2CCC2)NC2CCN(CC=CC=O)CC2)c(C)n1 Cc1ccnc2c(C(=O)NC3CCN(C(=O)C=CCO)CC3O)cnn12 c1(OC)ccccc1C(O)C(N1CCC(O)(CNC(=O)C(O)CCSC)C1)=O C(=O)(C1=C(Cl)CCOC1)NC1(C2N(C(c3n(CC#N)ncc3)=O)CCCC2)CC1 c1(C(=O)NCC2(NC(C(CSC)O)=O)CCC2)ccc2[nH]c(=O)cnc2c1 c1(NC(=O)CCC2CCCC2=O)ccnc2c(I)cccc12 N1(C(C(CC(F)F)N(C(=O)C(O)CN2CCCC2)C)=O)CC2CCC(CC2)C1 N1(C(C=CC=CC)=O)CC2CN(C(=O)C(C)CC(C)(C)C)CC2C1 CCC(CC(F)(F)F)NC(C1CN(C(C2CCCCC2O)=O)CC1(F)F)=O N1(C(C2(CC#C)CC2)=O)CC2(CCC(C)O2)C1.C1(C=O)CCCC2(CCC2)O1 C(C(=O)NC1CCCCN(C(C2(C)CC=CCO2)=O)C1)(c1ccccc1)=C(C)C C(=O)(CCS(N)(=O)=O)NC(CN(C(=O)CC12CCC(CC1)C2)CC)C N1(C(CCCC(C)NC(c2cc(C)c(C)s2)=O)=O)CCC2(CCOC2=O)C1 Cc1c(C(=O)N(C2CCC(NC(C3CC3C)=O)CC2)C)cnn1C(C)C(C)C N1(C(C(N2CC(C)C2)C)=O)CCN(C(=O)Cc2ccc(Cl)cc2)CC1C1CC1 C=CCCCC(C(=O)NC1CCn2cnnc2C1)NC(=O)CCC1CCCCC1 c1(N2C(C3CCCN(C(C(C(C)(C)O)F)=O)C3)CCCC2)ncnc2scnc12 c1(C(=O)NC2(C(=O)OCC)CC2(C)C)c(-c2ccccc2)nn(C)c1Cl c1(C(=O)NC2CC(C)(NC(c3nc(C)sc3C)=O)C2)cc2n(n1)CC(F)C2 C(CC(=O)O)(C(=O)N1CC2(CC2)CC1C(N1CCC(C(=O)NC)CC1)=O)NC c1(C(N2CCN(C(C=CCCC)=O)CC2CCOC)=O)cc(C)cc([N+](=O)[O-])c1 C1(NC(C(CC)SC)=O)CC1C1CCCN(C(=O)CCCS(C)(=O)=O)C1 C(=O)(C(O)CCCNC(C1(F)CCCC1)=O)N(C1COCC1O)C c1(C(N2CC(CNC(C(C(C)C)O)=O)C(C)CC2)=O)ccc2oc(O)nc2n1 C1(C(C)C)CN(C(C2CCS(=O)(=O)CC2)=O)CCC1NC(=O)Cn1cccc1 c1(C=O)cc(C)nc(C)c1.c1(C(C)=O)ncc(C(=O)NC2CC(O)(C)C2)s1 c1(C(N2CCN(C(c3cc(SC)oc3)=O)CC2C)=O)cccn2cnnc12 C1(CCCC)CN(C(c2cccc(C)c2C)=O)CCN1C(c1cc(C)co1)=O c1(C(=O)NC2CC(CNC(c3nc(C)oc3)=O)C2)cnn(CCO)c1N c1(C=O)cc(Cl)cc2c1OCC2.C(C(C)(C)C)N(C(C1CNC(=O)C1)=O)CC N1(C(C(COC)CC(C)C)=O)CCC2CN(C(c3sccc3OCC#N)=O)CCC12 c1(CC)cc(C)ccc1NC(=O)CC1CC2(C1)CN(C(C1CCSC1)=O)C2 C(C(=O)N(C)CC1CCCN(C(C2(C(F)F)CCOCC2)=O)C1)(C(C)C)OC N1(C(c2ccc(CO)s2)=O)CCC2CCN(C(C34CCN(CC3)C4)=O)CC2C1 C1(OCCNC(C2CC=CCC2)=O)CCN(C(C2(CF)CC2)=O)C1 N1(CC(=O)Nc2ccc(C)cc2)CC=C(CNC(C2CCC(=O)N2C)=O)CC1 C1(C(C)NC(c2coc(Cl)c2)=O)CN(C(c2ccc(F)cn2)=O)CCO1 C12(C(N(CC(C)O)C)=O)C3C4C1C1C2C3C41C.c1(CC)occc1C(=O)N CCC(CC(=O)NC(C)COC)N(C(=O)C(C)C#N)C Cc1cccn(CC(=O)NC(C(C)(C)O)C2CC2)c1=O c1(C(c2n(CC=C)nnn2)NCC(N2CCOCC2)C)cccc2c1CCOC2 C1(C(=O)NC(C2CCOCC2)C)C2CC(F)C(C2)N1C(c1c(F)cccc1F)=O CCCC(CCC)CC(=O)NC1CN(C(C2CCN(C(=O)OC)CC2)=O)CC1C C1(C(=O)NC23C(CN(C(CCC4(C)CC4)=O)C2)CC3)Cc2ccccc2S1(=O)=O C(CCOCCO)(C(=O)NC1C(O)CC1O)NC(CCc1onc(C)n1)=O c1(CN2CCN(CCCNC(c3n[nH]cc3I)=O)CC2)cc2ccoc2cn1 C1(NC(C(C)Oc2ccc(F)cc2)=O)CN(C(C2CC(O)C2)=O)C(C)(C)C1 CC1CCc2[nH]c(=NCc3cccc(F)c3)nc(N3CCSC(C)(C)CC3)c2C1 Cc1cc(C)n(CC(=O)NC2COCC2)c(=O)n1.c1(C(=O)N)cnc(O)c(F)c1 Cn1c(C(N2CC3C(C(=O)Nc4ccc(Br)c(Cl)c4)C3C2)=O)cccc1=O O=C(C(CC(F)F)NC(=O)C(F)n1ccnc1)NCCCN1CCCCC1 CCC(CC(C)C)C(=O)N1CC2CCC2(CNC(c2cnc3n2CCCC3)=O)C1 c1(C(N(C)CC2(CNC(CCc3cnc(C)o3)=O)CC2)=O)cncnc1C CC(C1CCCCC1)=CC(=O)NC1COCCN(C(c2n[nH]c(C)c2O)=O)C1 C1(OC)CC(CNC(=O)C(C(C)C)c2cccc(Cl)c2)N(C(=O)C)C1.CCF CC(O)C(C)(C)C(=O)N1CCOC(C(=O)NCC2CCCCN(C)C2)C1 C1(OC)(CNC(=O)Cc2cccs2)CN(C(=O)Cn2cc(Br)cn2)C1.S N1(C(C2CN(C)C(=O)CC2)=O)CC2(CC(C(=O)N(CCO)CCO)CO2)C1 C1(NC(N2CCCCCC2c2ccco2)=O)CNCC12CCOCC2 C1CCC(F)(F)CC1.C(C(CO)NC(C1(C(=O)NC)CC1)=O)N(C(C)C)C.C C(=O)(C1=CN=C2N=CNN2C1)N1CCCCC(NC(C(C)(C)C2CCCO2)=O)C1 Cc1c(C=O)oc2c(Cl)cccc12.C(=O)(C(C)CC1CCC1)N(CC(C)C)C.N c1(C(=O)NC2CCC(NC(=O)CC3CCCOCC3)C2)ccc2scnc2c1 Cc1cc(N)c(C(=O)NC2C(C)CN(C(=O)Cn3ccnc3C)CC2C)nc1C C1(NC(C(c2cccc(Cl)c2)C)=O)CC2(C1)CC2NC(=O)OC(C)(C)C c1(CCC(=O)NC(CC)=O)cc(F)ccc1NCCSC C(=O)(C1=CC(C)(C)C1)N.C1(NC(C2(COC)CCC2)=O)CCC(C)C1 c1(CCC(N2C3CC(NC(c4nc(C)c(C)s4)=O)(C3)C2)=O)csc2ccccc12 C1(CN(C(=O)CSc2cccs2)C)CCCCN1C(c1ncccn1)=O Cc1ncc(C(=O)N(CC(C)(C)NC(=O)Cc2ccsc2Cl)C)[nH]1 c1(COC)nc2ccccn2c1C(N1CCC(NC(=O)CC=C(Cl)Cl)CC1)=O CCCCCCOC(C)C(=O)NCC1(CC)CC1.c1(C(=O)N)cc(C)sn1 C1(NC(C2CN(S(CC)(=O)=O)C2)=O)CCC(O)C1.C(=O)C.C(C)(C)C.N Cc1cc(C(=O)NC2CCCC(CNC(c3csc(O)n3)=O)C2)cn1C Cc1noc(C)c1CC(=O)NCc1cc(C(=O)NCCCC=O)n[nH]1.C1CC1 C=CC1(CC(=O)NCC(C)(C2CC2)NC(C23CCCC2C3)=O)CCOCC1 C1(C=O)CCc2nn(C)cc2C1.n1(C(C)C)ccnc1C(=O)NC(C)C1CC1.N C(=O)(C1=CC2(CCOC2)C1)N1CCCCC(NC(c2ccnc(C3CC3)n2)=O)C1 CC1CS(=O)CCN1C(C1(CNC(=O)CCc2nccs2)CCCCC1)=O C12(NC(=O)Cc3cc[nH]c3)CCOCC1CN(C(c1ccn3nccc3n1)=O)C2 CC1CCCCC1(CNC(=O)C(F)(F)CO)NC(c1ccnn1CCF)=O CCCCCCCCNC(N1CCCC1CN1CCCCC1)=O C1(C(=O)NCCC(C)NC(=O)C(F)=C2CCC2)CCS(=O)(=O)N1C C(COC)(CC(=O)NC1CC(O)C1O)NC(C=CC=CC)=O Cc1ccccc1C(=O)NC1CN(C(C2CC2[N+](=O)[O-])=O)CC1CC1CC1 N1(C(CCC#C)=O)CCN(C(c2ccc(Cl)cn2)=O)C(COC)C1 C1(NC(C(=O)NC(c2ccncc2)C(C)C)=O)CCOC2(CCSCC2)C1 c1ccc(Cl)cc1.c1(OC)sccc1C(=O)NC1CC(CCNC(=O)C)C1 CCCCC(O)CC(=O)N1CC2C(NC(C3C=C(C)CS3)=O)C2C1 c1(NC)cc(Cl)ccc1C(=O)N(C)CC1CCN(C(=O)CC2CN(C)C2)C1 CC(CCO)N=c1[nH]c2c(c(=NC(C)Cc3cccc(Br)c3)[nH]1)CSC2 c1(C(N2CCCC(N(C(c3cc[nH]n3)=O)CC)C2)=O)nc(C)oc1OC C(C(C)(C)CC(=O)N(C)CCN(C)C(C1(N(C)C)CCOCC1)=O)OC c1(CC(C=O)C)cccc(F)c1.C(C)(C)(C)NC(CC1(CSC)CC1)=O C(=O)(C1=CS(=O)CCC1)NC1CC(NC(=O)CNC(c2ccncc2)=O)C1 C(=O)(CC(C)(C)CNC(c1csc(F)c1)=O)NC12C(CN(C)C1)C2 c1(C(=O)NCCCNC(CC=C)=O)c(C)nn(C(C)C)c1C c1(OCC)cccc(CNC(=O)NC2CCCC2NC(=O)CCC)c1.O N1(C(CC2CC(=C)C2)=O)CCN(C(c2ccn(C)c2)=O)C2CS(=O)(=O)CC12 N1(C(Cc2ccc(C)nc2)=O)CC2(CC2)CC1C(=O)NCc1ccc(O)nn1 c1(OC)cc(C(N2CC(NC(=O)CC3CCOC3)C(C)C2)=O)cc(OC)c1O c1(C2(C(N(CCC)C)=O)CCC2)ccccc1.C1(C=O)(COC)CCC1.N C(CC(C)(C)CC(=O)N1CCC1(C)CC(N1CC2CCC1(CO)C2)=O)OC N1(C(CCCCCSC)=O)CC(C)CN(C(=O)C#CC2CCC2)CC1C n1(CCSC)nnnc1C(c1cscc1Cl)NCc1noc(-c2ccccn2)n1 N1(C(c2occ(C)c2)=O)CC(NC(c2cc(C(C)(C)C)oc2C)=O)CC(C)C1 C(=O)(C(CN=[N+]=[N-])NC(=O)Cc1cccn1C)NCC(C)C(F)F C1(NC(c2ccc(OC)c(OCC(=O)O)c2)=O)CC2CCC1(C)C2(C)C N1(C(c2c(C)sc(O)n2)=O)CCN(C(=O)Cc2cc(Br)cs2)CC(C)(F)C1 c1(C=O)c(C)nc2sc(C)nn12.Cc1c[nH]c(C(=O)NCC2CC(C)CO2)c1 N1(C(C(CCC)(C)C)=O)CCC2(CC1)CN(C(c1cnc(OC)s1)=O)CC(C)O2 C(=O)(C(CC(C)C)N(C)C(C1CCN(S(=O)(=O)c2cccs2)C1)=O)OC C1(C(=O)NCC2CN(C(CCC3N(C)CCCC3)=O)C2)Cc2nnsc2S1 Cc1cncc(C(=O)NCCOC2CCN(C(C3(C)CCCO3)=O)C2)c1Cl c1(C(c2nnnn2C2CC(F)(F)C2)NC(C(C)C)C)ccnn1C C(CC(C(C)(C)C)NC(=O)C(C1CCCCCC1)O)N(C)C(c1cnsc1)=O c1(C(=O)NCC(C2CC2)NC(CN(CCCCCC)C)=O)ccc2ccsc2c1 N1(C(C2(CC#C)CCCO2)=O)CCN(C(=O)CCCCCSC)CC1C CC(C(C)C(=O)NOCC=CCl)NC(C1CC2(CCC2O)C1)=O C(c1ccncc1)=CC(=O)N.C1(O)(CC)CCN(C(=O)CC2CC(=O)C2)C1 CCC(CNC(C1(CNC(C2(C#N)CCCC2)=O)CC1)=O)C(C)C CC(C)C(CNC(c1cccn1C1CC1)=O)C(=O)N(C1CCOCC1C)C N1(C(c2cc(CCOC)on2)=O)CC2CCC1C2NC(c1csnc1C)=O N1(C(c2nccc(C(C)(C)C)c2)=O)CCCN(C(C2(C)CCCCO2)=O)CCC1 Cc1nc(S)nc(C)c1CCC(=O)NC(C)(C)C(C)NC(=O)CS.C(C)C C1(NC(C2CC(C(=O)OCC)C2)=O)CC2(C1)CN(C(C1CC1C)=O)C2 N1(C(CNC=O)=O)CCc2cc(CNC(=O)C)ccc2C1.C(C)(C)C(F)(F)F CCCCC(O)CC(=O)N1CCCC(C)(CNC(c2occc2COC)=O)C1 CC1C(NC(=O)CCC2CCCO2)CCCN1C(c1ccc(CO)cc1)=O C1(NC(C(C(C)C)F)=O)CCCCN(C(c2cn(CCN(C)C)nn2)=O)C1 CCC(C(=O)N1CC(O)(CCNC(=O)C(C)(C)N(C)C)C1)NC(C)=O C1(O)(CCCNC(C2C(NC(CC3(COC)CC3)=O)C2)=O)CCC1 c1(C(N2CC(O)C2)=O)occ2c1CCCC2.C1(CC(=O)N)(COC)CCCC1.C C(=O)(C(C)(C)CC(F)(F)F)NCC1CCC(N(C(C2C(C)C2)=O)C)CC1 c1(C(=O)N)cc(C2CCCCC2)[nH]n1.C(CC(=O)N1CC(C)C1)OCCCOC c1(C(=O)NC(CC2CN(C(c3cc(C(CC)CC)no3)=O)C2)C)cccnc1S c1(SCC)cc(-c2nc(C(C)C)nn2Cc2ccccc2Br)ccn1 C1(C(=O)NCc2nc(C(C)C)on2)CC2CCN(C(C)CN3CCCCC3)CC12 C1(CNC(c2cscn2)=O)CCN(C(C2CCNC2=O)=O)CC1(F)F N1(C(c2ccc(C(=O)OC)s2)=O)CC(N(C)C(c2cnnc(C)c2)=O)C(F)C1 c1(C(=O)NCC(C)NC(C2(C(=O)OC)CC2)=O)c(C)n[nH]c1C CC1C(NC(C2(S(C)(=O)=O)CCC2)=O)CCCN1C(c1cc(N)ccc1Cl)=O Cc1cc(N)c(C(=O)NC2CCCCC2NC(C23CCCC2C3(F)F)=O)cc1C c1(C(=O)Nc2c(C(C)O)cccc2)cc2cc(-c3ccccc3)ccc2oc1=O C(=O)(C(O)C(F)(F)F)N.C1(C(N(C(C)C(C)(C)C)C)=O)(C)CC(C)(C)C1 c1(-n2cc(C(CCC)NC(=O)CC)nn2)cc(OC)c(OC)c(OC)c1 Cc1cc(O)c(Cl)cc1C(N1CCC(CF)(NC(c2coc(Cl)c2)=O)C1)=O C1(C(=O)NC2CN(C(C3(C(F)F)CCCCC3)=O)CC2O)(OC)CCC12CCC2 CC(C)CCCO.C1(O)(C=O)CN(C(=O)C=CC(N2CCOCC2)=O)C1.CC C1(C(N(c2ccc(F)cc2)C)=O)C=CCN(C(=O)CN2CCCC2=O)C1 c1(C=O)ccc(N2CCCC2)nn1.C(C)(C)(C(=O)NCC1CCCC1)N(C)C.N C1(C(N2CC=CC(NC(c3oc(C)cc3C)=O)C2)=O)(CC)CNC(=O)C1 C1(C)(C(=O)NC(c2ccccc2)CNC(c2nc(C)n(C)c2)=O)CCNC(=O)C1 C1(CNC(CCOC(C)C)C)CCOC1C(C)(C)C C1(CC)CN(C(C2(F)CCOC2)=O)CCC1NC(c1ocnc1C1CC1)=O C1(N(C(=O)CC2(CO)CC2)C)CCC2CN(C(c3ccc(N=[N+]=[N-])cc3)=O)CC12 C=CC1(c2cn(CC(=O)OCC)nn2)COCCN1C(c1nccc(Cl)c1Cl)=O c1(OC)nc(N(C2CNCC2F)C(=O)CC2CCCCO2)nc2[nH]cnc12 C1(C=O)COCC(C)(C)CN1C(=O)C1CC1.C1(C=O)CCC1.C(C)(C)C.C Cc1scc(C(=O)NC(C)CN(C)C(C2CC2CN(C)C)=O)c1C C#CC1(NC(C2CC(C)(C)CCN2C(=O)C(C)COC)=O)CCC(C)(C)C1 c1ccccc1.C1(NC(C(C)NC)=O)CCCC1CNC(=O)C.C1CCC1.O N1(C(CN(C(C(C)C)CO)C)=O)CCOCC1CC(N)=O CCCCCC(=O)NC(CC1CCOCC1)C(=O)NCCC(=O)NCC c1(CNC(C(=O)OC)CO)cc2cc(C)ccc2o1 c1(C(N2C(C)CCN(C(C3C(CC)C3)=O)CC2)=O)ccc2nc(O)cn2c1 C1(CNC(C(c2ccn(C)n2)(C)C)=O)CN(C(=O)CO)CC1O.c1nc[nH]n1 C1(C(N(C2(n3cccn3)CC2)C)=O)CCN(C(=O)CN=[N+]=[N-])C1 Cc1cccc(C2(C(=O)NC3CCC3)CC2(F)F)c1.c1(C(=O)N)csc(C)c1C CC1CCC(O)(C(=O)NCCOC2CCN(C(=O)C(=O)C(C)(C)C)C2)CC1 C1(NC(C2C(=C)C2)=O)CC(C)N(C(c2cc(C3CCCN3C)[nH]n2)=O)C1 C1(C=O)CC2CCC(C1)C2(F)F.C1(NC(C2CC(OC)C2)=O)CC12CCC2.N n1(CC2(F)CC2)c(N2CCC(c3cccc(Cl)c3)C2)nnc1C1CC1 c1(C(=O)NCC(CO)NC(C2(F)CC=CC2)=O)cc(O)nc(Cl)c1 c1(NC(C2C(NC(=O)Cc3ccc(F)cn3)C2)=O)ccc(Cl)c(Br)c1 Cc1ccc(C(C)(F)F)cc1C(=O)NC1(C)CN(C(c2coc(C#N)c2)=O)C1 C1(NC(=O)CCc2cnco2)CCCC1NC(=O)CCC1CNC(=O)N1 CC1(O)CCC(C(=O)NC(C(=O)NCCCSC(F)F)c2ccco2)CC1 C1(C)(C(=O)NC2CCN(C(c3nnc(C)s3)=O)CC2)CC(c2ccccc2)=NO1 CCC(C)C(CNC(=O)C(N1CCN(c2ccsc2C#N)CC1)=O)OC c1(N(CC(=O)Nc2cccc(Br)c2)C)nc(N(C)C)c2[nH]ccc2n1 N1(C(C)=O)C2CCC(C(=O)NC3(CN(C)C)Cc4ccccc4C3)C1CC2 c1(C(=O)NC(CC)CN(C)C(C2(C)CC3CCC2O3)=O)cnc2c(c1)CCCC2 c1(C(=O)NCCN(C(=O)CCOC)CCOC)ccnc2[nH]c(C)nc12.O c1(OC)cc(-c2csc(-c3nc(C(C)C)nn3-c3ccc(F)cc3)c2)ccc1F C(=O)(C(C#N)C(C)(C)C)N1C(C(C)C)C(C(=O)NC2CC=CC2)CC1 Cc1ccc(F)c(CC(=O)NCCCC(C)NC(C2CN(C3CCOC3)C2)=O)c1 c1(C(C)(C)C)ccc(C(=O)NCCC(C)(C)C)cn1.CC(F)(F)F.C(=O)C.N C1(C(=O)NCC(C#C)OC)CC2(CCN(C(=O)CCC(=O)CC)C2)C1 c1(C(N2CCC(NC(C3(C)CC3)=O)C(C)(C)C2)=O)ccc(F)c2ccncc12 c1(C(N2C(C)(C(=O)NCc3c(C)nccn3)CCC2)=O)cnc(O)c(F)c1 Cc1cc(C)c(C(=O)NC(CNC(=O)Cc2cccnc2Br)C(C)C)cn1 C1(C(=O)OC)CCC(C(F)F)(NC(=O)NCC2CCCC(C)O2)CC1 C(C(CO)C(F)(F)F)NC(c1n(CCOC)nnn1)c1nnn(C)n1 c1(CNC2CC(C(NC3CCN(CC)C3)=O)C2)c(F)cncc1F C1(C(N(CC(CC)NC(=O)C(C)=CCO)C)=O)CCCCC1 N1(C(c2c(CC)cno2)=O)CC(OC)C(C(=O)N(CCC(O)CO)C)C1 c1(NC(C(C)N(C(CC)=O)C)=O)ccc(Cl)c(S(=O)(=O)N2CCN(C)CC2)c1 C1(C(=O)NC(c2ncccc2C)CC)CC2CCN(C(C)Cc3ccsc3)CC12 c1(C(N2CCC(C)(CC)C2)C(=O)NCCOC)cccc2ccoc12 N1(CC(=O)NCC(CC)NC(C2CCCN(C)C2)=O)CCCCS1(=O)=O C12(C(=O)OCC)CCCCC1N(C(=O)C(=O)NC1CCCC1CN)CC2 N1(C(CCCC)=O)CCC(NC(c2cc(F)ccc2OC(C)C)=O)C(C)C1 C(=O)(C(CNC(c1nscc1C)=O)CC1CCCC1)NCC(CCC)C c1(C(N(CC(C)NC(c2cc(C)c(C)nc2)=O)C)=O)nc(=N)[nH]c2ccccc12 Cc1cc(O)ncc1C(=O)NC1CC1C.N1(CC=O)OC(C)(C)CC1=O.N c1(CC)nn(C)c(CC(=O)N(C2CCC(NC(=O)CCCF)C2)C)c1Cl N1(C(C2C(C=CC)CN(C(=O)C(F)CC3CCOC3)C2)=O)CCCC12CCOC2=O C(C(C)(CO)NC(=O)Cc1cc(OC)no1)NC(CCC)=O c1(C(=O)NC(CNC(C(n2cnc(C#N)n2)C)=O)CO)ccc(C(F)(F)F)nn1 CCC(C)C(C)(O)CNC(C1C2CCN(C(c3ccon3)=O)CC12)=O C1(NC(CC(C)C2CCCO2)=O)CCN(C(=O)CO)CC12CCC2 Cc1cccc(CC(=O)NC(C)CNC(c2cc(-c3ccns3)on2)=O)c1 c1(NC(c2ccc(NC(c3c(OC)nccn3)=O)cn2)=O)cc(C)ccc1Cl C1(CC(=O)N(CC(C)OC)CC)C2CCCC2N1C(C1CCOC1(C)C)=O c1(C(=O)NCC(COC)C)ccc(CNC(c2cnc[nH]c2=N)=O)cn1 S(=O)(=O)(CC(=O)N1CC(C(C)NC(c2ccnn2CCF)=O)C1)NC C1(CC(=O)NCC2C(CC(N3C(C(C)O)CC3)=O)C2)CCCC(=O)C1 Cc1nc(C(=O)NCC(C)N(C)C(c2ccc(OCF)cc2)=O)c(C)n1C1CC1 c1(-c2nc(C(C)OC)nn2CC(C)(C)CO)ccc2c(O)n[nH]c2c1 C1(NC(C2ON=C(CC)C2)=O)CCN(C(=O)Cc2cncs2)CC1F C1(NC(c2cnn(CC)c2C)=O)CC2CC(NC(=O)CC(C)OC)CC2C1 c1(C(=O)NCc2ccc(-n3cccn3)cc2)cnc2c(c1)CCOC2 Cc1ccc(C(=O)O)cc1-n1nnnc1CNC1CCC2NCCC12 N1(C(=O)CC(F)(F)F)CCC2(CCC(N3CCN(C4CCOCC4)CC3)CC2)C1 c1(COC(C)C)ccc(CNC(=O)NCCCc2cnccn2)cc1 N1(C2CCCN(C(CCOCC#C)=O)C2)CCN(C(C2(O)CC2(C)C)=O)CC1=O C1(C2CCOCC2)(C(=O)OCCCOCc2ccccc2)CCOCC1 CC(C)C(C(=O)NC(C)C)NC(=O)C(C)(C)C.c1(C=O)nn(C)cc1Cl.N C1(CC(=O)NCCC(C)N(C(=O)COC2COC2)C)CCC(C)C1 c1(-c2n(C(CC)C)nc(-c3ccc(C)c(F)c3)n2)cccc2c[nH]nc12 c1(OCC=C)ccc(C(=O)NC2CCN(C(c3ccc(CCF)cc3)=O)C2)cc1 Cc1cc(C(=O)NC23CC2CN(C(c2ocnc2C)=O)C3)sc1Br C(=O)(CC(O)C(C)CC)N(C(C)C(N1CCn2ncnc2C1)=O)CCC C1(O)(CNC(=O)Nc2cccc(C)c2)CCCN(Cc2cnc(Cl)nc2Cl)C1 C(CC)(C(=O)NC(C)(CNC(=O)C=CCOCC)CC)=CCCC C(=O)C1CCC(=O)c2cccn21.C1(NC(=O)CSc2nc[nH]n2)CC(F)(C)C1 C(CCCC(=O)NC(C)(C)Cn1cccn1)OCC.C1(C(=O)N)CC1(F)F C1(C(C)(C)C)(COC)CCN(C(=O)COC2CCCC2)C1 c1(OC)ccc(C(=O)NC2(C)CC(NC(=O)Cc3ccsn3)C2)cn1 CC1(C)CCC(C(=O)NCCCOCCCNC(C2(Cl)CC2)=O)OC1 c1(C(C(C)NC(=O)COC(F)F)NC(=O)COC(F)(F)F)ccccc1 CC1CN(C(=O)CC2CC(C(F)F)C2)CCC1NC(C1COC2COCC12)=O CN=c1nc(C(=O)NC(C)(C)CN(C)C(c2cc(F)ncc2)=O)cc(C)[nH]1.O CN=c1cc(C(=O)NC(C2CCOC2)CNC(=O)C(C)(C)C(F)F)cc[nH]1 C1(NC(COCc2cc(C)on2)=O)CC(O)CN(C(=O)C(O)C(C)C)C1 c1(N2CCCC(COCC)C2)nc(Cl)nc2[nH]cnc12.C12(CCOCC1)C(=O)N2 c1(C(N2C3CC(NC(c4cc(C)c(O)nn4)=O)C(C3)C2)=O)ccc2nonc2c1 O=C1CCC(CC(N2CC(F)CC2CNC(c2cnncc2O)=O)=O)C(=O)N1 c1(CC(=O)NC(COC)C#N)cc([N+](=O)[O-])ccc1F Cc1ccc(C2CCN(C3CCN(c4ccc(Cl)cn4)CC3)C2)c(C)c1 CN=c1[nH]cc(C(=O)NC2CC(C)(NC(c3ccc(-n4cnnn4)cc3)=O)C2)o1 C1(NC(C2(C(C)C)CCN(C(C3CCCCC3)=O)C2)=O)CCCCCC1F C(=O)(C(C)(C)C1=CCSCC1)NC1C2CN(C(C(C)CC3CC3)=O)CC21 C1(C(=O)N)CC(=O)NC(=O)C1.C1(CC=C)CCCCN1C(=O)CC(C)C1CCC1 C1(CNC(C=C(CCC)C)=O)CCN(C(=O)CS(=O)(=O)CC)C1(C)C C#CCC(C)(C)C(=O)N1CCC(NC(c2ccc(C(=O)OC)n2C)=O)CC1 C(C(C(=O)NC(CN1CCCC1)CO)NC(=O)Cc1ncc(C)o1)OCC C1(C(=O)OC2CC(SC)C2)COc2cc(F)ccc2O1 C1CN(C(=O)Cn2nnc(C)n2)CCC1(C)C.c1(CC)cc(C(=O)NC)sc1C n1(C(C)C)cccc1C(=O)NCC(C)N(C(=O)C(C)CSc1ccccc1)C C(=O)(CCC(C)NC(c1cnnn1C)=O)N1CCC(OC)C1 C1(C(N2CCC(C(=O)Nc3ccccc3)C2)C(=O)NC)CC2CC(OC)C2C1 C#CC1(OCC(=O)NCC(C)(O)CNC(=O)C(C)OCOC)COC1 c1nc(C)cnc1C#N.c1ccnc(C=O)c1.C1(C(=O)OC)CC1C(=O)NC c1(C2C(C=O)C2)cccc(Cl)c1.c1(OC)cscc1C(=O)NCC1CCC1 c1(C(=O)NC(CNC(c2ccc(C(C)C)cn2)=O)C)cc(Cl)cc(Br)c1 C1(N(c2c(CC(=O)OCC)cccc2)C(=O)C(O)C(C)C)CCNCC12CC2 N1(C(C(CC2CCC2)NC(c2cc(CC)ncc2)=O)=O)CCC(C)(CCO)CC1 c1(C(N)=O)nccnc1NC(=O)C(=O)NCC.c1(C[SH](=O)=O)ccccc1 n1(C(C)C)ncc2c(NC3CC(F)C3)[nH]c(=NCCC(=O)Nc3ncc[nH]3)nc12 CC1CC(NC(=O)CCc2ccccc2)CN1C(=O)C(F)n1cccn1 CCC(C)(CO)NC(=O)NCC(c1cccs1)OC N1(C(C(=O)Nc2ccc(C#N)cn2)=O)CCCC2(C1)OCc1ccccc12 CCC(CC)CC(F)C(=O)NC1(COC)CCN(C(=O)CCC2(C)CC2)CC1 Cc1nn(C)c(-n2cccn2)c1C(=O)NC(C)CCN(C)C(C1C=CCC1)=O C(=O)(C1CCCc2nncn21)N1CC2C(NC(c3ccccc3OC(F)F)=O)(C2)C1 CCCC(C=O)NC(=O)C.C1CCN(C(=O)CN2CC3CC3C2)C1.C(C)=O.O c1(CNC2C(O)CCC(C(=O)OCC)C2)cc(-c2sccc2C)c2cc[nH]c2c1 n1(CC)ccc(CN(C)Cc2cc(CO)on2)c1 C=CCN=c1[nH]c(C(=O)NCCC2CCCCN2C(=O)CCc2cnc[nH]2)cs1 C1(C(=O)OC)N(C(=O)C(C(C)(C)C)N2CCNC2=O)CC12CC2(F)F Cc1cncc(C=CC(=O)N(C)CC2CCN(C(=O)CS(C)(=O)=O)CC2)c1 CC1=NOC(=O)C1CCC(=O)NC(C)CN(C(=O)C(C)C(C)C)C C(=O)(C(=O)N=c1cc(C)o[nH]1)NCC12N(C(CCSC)=O)CCC1CCC2 CCCC(CC)CC(=O)NC1CC(CNC(c2cnn(C3CC3(F)F)c2)=O)C1 C1(CC=O)CCS(=O)(=O)C1.C#CC1(C(N2CC(C(N)=O)C2)=O)CCC1.C c1(CC(=O)NCCC2CCCN(C(CC(C)C)=O)CC2)c[nH]c2cnccc12 Cc1c(Br)cnc(O)c1C(=O)NCC1CC1NC(C1CCCCC(=O)N1)=O C(=O)(CCC(CC)(CC)[N+](=O)[O-])NC1(C)CCN(C(C2CC3(CC(=C)C3)C2)=O)C1 c1(C(=O)NC(CCNC(c2c(CC)cco2)=O)C)nccn2c(C)nnc12 c1(CNC(CC2CC(NC(=O)COC3CCOC3)C2)=O)ncc(Cl)cn1 C1(CNC(=O)CC(=O)NC2CC2)CN(C(c2ccccc2)=O)CCC12CCOC2 c1(OCC=C)cccc(C(c2nnnn2CCCCCC)NCC(CO)C(C)C)c1 N1(C(CN(CCCCCC)C)=O)CCN(C(c2cc(Br)no2)=O)CC1CO c1(C(=O)NCC(N(C(C2CCCN(CC)C2)=O)C)C2CC2)ccc(F)cc1O C12(C(=O)NC3(C(C)(F)F)CC3)CC(CN1C(C1CC13CCC3)=O)C2 CCCC(C)(O)C(=O)N1CC(O)(CNC(c2cccc(SC(F)(F)F)c2)=O)C1 C1(CCNC(c2c(CC)nc(C)[nH]2)=O)CCCN(c2ccc(C(C)=O)cn2)CC1 CC1CN(C(C2CC(C)(C)CN2C)=O)CC1(C)CNC(c1cc(C#N)cn1C)=O C(=O)(C(Cc1ccccc1)NC(=O)CCc1ncc(C(=O)O)[nH]1)OCC N#Cc1ccc(OCCCc2cccc(C(F)(F)F)c2)cc1 c1(CCNC(=O)Nc2n(C)ncc2)cccc(NS(=O)(=O)C(F)F)c1 CC1CN(C)CCC1NC(=O)C(C1CCCC1)NC(=O)CC1CCCSC1 c1(C(N(C(C)C(N2CC(CO)C(O)C2)=O)CC)=O)cccc(F)c1N Cn1cc(C(=O)NC2CS(=O)(=O)CC2NC(=O)CO)c2cccnc12 C1(NC(CN2CC(C)(C)C2)=O)CC(C2CCN(C(=O)Cn3cnnc3O)CC2)C1 N1(C(c2ncc(Cl)s2)C(=O)NC(CC)C)CCCCC1P(C)(C)=O CCC(CC(=O)N(C1CN(C(=O)Cc2ccc(SC3CC3)cc2)C1)CC)OC N1(C(C2CN(S(N)(=O)=O)C2)=O)CCCC2(C1)CN(C(=O)CC(F)F)C2 c1(OC)n[nH]cc1C(=O)NCC(C1CCCN1C(=O)CC1CC1C1CC1)(C)C C1(C(N2CCC(CC=O)C2)=O)C2CCC(C2)N1C(=O)CCc1nncn1C.CN N1(CCOC(CC2CCN(C(C)(C)C)C2)=O)C(=O)NC2(CCCC2)C1=O c1(C(N2CC(=C(CNC(c3nc(C)c(C)[nH]3)=O)F)C2)=O)cc(C2CC2)nnc1O c1(N2CCN(C)C(=O)C2)ccc2nc(SCc3ccccc3Cl)sc2c1 C1(C(N(C2CCSC2)C)=O)CCN(C(C2(C)CCOCC2)=O)C(C)(C)C1 C1(CN(C)C(c2cnccc2Cl)=O)CCCN(C(C2CCCSC2)=O)C1 C1(CC)CN(C(c2csc(CC3CC3)n2)=O)CCN1C(=O)C(C1CCOCC1)O c1(C(N2CCC(NC(CS(=O)(=O)NC)=O)CC2C)=O)ccc2cc(O)ccc2c1 C1(NC(C=C(CCC)CCC)=O)CC2CCCC(C1)N2C(=O)C=Cc1cnc[nH]1 N1(C(CCC(c2cc(C)sc2C)=O)=O)CCN(C(C2CC3CC3C2)=O)CC1CF N1(C(CCSCC(C)C)=O)CCC(N(C(=O)CC2C=CCCC2)C)CC1 C1(CC)(CC)CC(NC(C2(CCO)CC2)=O)CN1C(=O)CCn1ccnn1 C(C1=NOC2CCCC12)NC(CN(C(c1c(C)csn1)=O)C(C)C)=O N1(C(C(C(C)C)NC(COC)=O)=O)CC2(C1)CN(C(=O)CC1CCCC1C)C2 Cc1cc([N+](=O)[O-])c(Cl)cc1NC(C1CCCC1NCc1c(Cl)cccc1I)=O N1(C(CC2(OC)CCC2)=O)CC(C(=O)NCCCCCCC2CC2)C(C2CC2)C1 CC(C(C)(C)C(=O)N1CC(c2ncccn2)C1)NC(=O)C=Cc1cncn1C CC1(C)CC(CNC(=O)CCC2CCOCC2)CN1C(c1cn(CCF)nn1)=O C1(NC(Cc2n(C)nc(C3CC3)c2)=O)CCN(C(=O)Cc2cn[nH]c2)CC1(C)C c1(C(=O)NCC2N(c3nccc(OCC)n3)CCOC2)ccc(F)c(F)c1C C1(C2CCN(C(=O)CCCC)CC2)(NC(C2CC(O)(CC#C)C2)=O)CC1 C1(C(C(C(=O)NC(C)C)N2CCC(CC=C)C2)C)CCC(F)(F)CC1 c1(C(=O)NC(CCN(C(CCCOC)=O)C)C)ccc2snnc2c1 C=Cc1cncc(-c2noc(-c3c(CNC(=O)OC(C)(C)C)c[nH]c3)n2)c1.C N1(C(C2C(C(C)NC(c3cc4n(n3)CCC4)=O)C2)=O)CCC(CO)CC1C Cc1ccnnc1C(=O)NCC1C2CN(C(=O)CCC3(C#N)CCC3)CC12 c1(C(=O)Nc2c(C)cc(C)nc2Cl)ccc2c(c1)ncn2CCc1ccccc1 CCC(C)CCC(=O)N1CCN(C(=O)C(C)(C)CO)CC1c1ccccc1 c1(C=O)ncccc1.C1(C(=O)NCC(=O)NC2CC2)CCCC1.C1CC1.C C1(NC(CN(C(=O)C(O)C=C)CC#C)=O)CC2CC(OCC)C2C1 C1(CC(=O)NCCCN(C(=O)CO)CCO)CC2(CC2)CO1.C1CCOCC1 CS(=O)C=CC(=O)N1CCCC(NC(=O)CSCc2ncc[nH]2)C1 C(C(=O)NOCc1nc[nH]n1)N(C(=O)CC1CC2(CC2)C1)C C(=O)(C(CNC(=O)CC1CCCCN1C)(CC)CC)N1CCCC(C#C)C1 c1(NC(CN(C(c2c(CCC)n[nH]c2)=O)CC)=O)cn(C)nc1CC N1(C(C=CSC)=O)CCCCC1Cc1cn(C2COCC2n2cccn2)nn1 C1(NC(c2c(C)scn2)=O)C2CC3C(C2)C13C(=O)NCC(Cl)C(C)(F)F c1(C(N2CCCC(C(N(C3CCC3)CC)=O)C2C)=O)ccc2cncn2c1 C1(CNC(c2c(CCC)[nH]cc2)=O)(OC)CCN(C(=O)C(C)(C)CO)C1 Cc1ccccc1CC(N1CCOC(CN(C(=O)C(C)C2CCCC2)C)C1)=O N1(Cc2cc3c(cc2)OC(C)(C)C3)CCCC2(CCCCCC2)C1 CC(C)C(CC(=O)NCC(C)(C(C)C)NC(=O)CCC1CCC1)C(C)C C(=O)(C(C)(C)CC#N)NCC(C)(C)OCC(=O)NCC(c1ccco1)O Cc1cc(Cl)cc(C)c1C(=O)NC1CC(C)(NC(c2ccnnc2C)=O)C1 N1(C(COCCSC)=O)CC2C=CC1C(C(=O)NCCCN1CCCC1C)C2 C(=O)(C(CNC(=O)CC1CCSCC1)C(C)(C)C)N(C)Cc1cn[nH]c1 C(=O)(C(C1=CCCCCCC1)N(C1CCC(C)CC1)C)NC(C(=O)OC)C CCS(=O)(=O)c1ccc(C(N2CCC(O)(Cc3nn[nH]n3)C2)C)cc1 C1(OCC)CC2CN(C(=O)C(COC(C)C)NC(C3CCC3C)=O)CC12 c1(C(N(C)CC2N(C(CSCC#C)=O)CCCC2)=O)ccc(OC)c2cn[nH]c12 C1(C(N(CC(=C)C)CC)=O)CCC(C)(C)N(C(=O)C=C(CC)CC)C1 C1(C(=O)NCC2(c3ccccc3F)CCC2)(OC)CCN(C(=O)C2CC2)C1 c1(C=O)cnc[nH]c1=N.c1(CNC(C)=O)ccc(C(=O)NC2CC2C)o1 C(CCC(C)(C)NC(=O)CCC1CCCCO1)NC(CNS(NC)(=O)=O)=O O=C1CCC(C(=O)NCCOCCNC(c2cnns2)=O)=NN1 CCCCCC(O)C(=O)N1CC(NC(c2cnc(C)nc2C)=O)CC1(C)C C1(CC(=O)NCC(C)N(c2ncc(Cl)cn2)C)OCCCC1(C)C CCCC(CNC(=O)C(C)C(C)(C)C)C(=O)N(C(C)C(N)=O)C CC1(C#CC(=O)N2CC(CC(F)C(N3CCC(C)(C4CC4)C3)=O)C2)CCCO1 C1(CCC=O)CCCOC1.C1(=C(C)F)CN(C(=O)C)C1.C(=O)(C)N.C1CCC1 Cc1ncc(CC(=O)N(C)CC2(C)CC2)s1.C(=O)C=CC.C(C)(C)C C1(n2cc(-c3n(CC)ncc3)nn2)CN(C(=O)C(C)COC)C(C)(C)C1 CCC(C)C(CC(=O)N(C)Cc1cc(C)nn1C)NC(=O)CC(O)CC c1(C(N(CCC(C)NC(c2cccnn2)=O)C)=O)ccn2ncccc12 N1(C(C(CCCC)C)=O)C2CCC1CC(N(C(=O)C(c1cc(C)oc1C)C)C)C2 c1(N2C(C(N3C(C)CCC3CO)=O)CC3CC32)ccc(I)cc1C(F)(F)F C(C)(C(C)C(=O)NOCC(=O)NC)NC(C1C(=C)C1C(=O)OC)=O c1(C(=O)NC(c2nc(C(F)(F)F)cs2)C)ccc(O)c2c1CCCC2 C12(NC(C(CC)NC(C)=O)=O)CC1CN(C(C1(C)CCC(=O)N1)=O)C2 CCCCCNC(=O)CN(C)CCOCCOCC.C(=O)(N(C)C)N CCCC(O)C(=O)N(CCNC(=O)C(CO)NC(=O)O)CC.C(C)(C)C c1(C(=O)NC(CCNC(CN(C2CC2)CC)=O)C)cc(F)c(Br)c(F)c1N n1(CCOC)ccc2cc(NC(=O)C(N3CCC(CCC(=O)OC)C3)=O)ccc12 Cn1ccc(CC(N2CC(CF)(NC(=O)CC3CCCCC3)C2)=O)n1 CC1(C)CN(CC(=O)NC2(C(=O)NCc3ncco3)CC(F)C2)C1 C=C(C)CC(C)C(=O)N1CCN(C(c2cc(C)ccc2OC)=O)C(C2CC2)C1 N1(C(CC(C)C)C(=O)NCCN(C)C=O)CC2CCC(C1)C(=O)N2.C(C)(C)C c1(C(C)C)ccc(C(=O)N(C2CCN(C(c3ncn(C)n3)=O)C2)C)o1 C1(O)(CNC(Cc2c(C)nc(C)s2)=O)CCCN(C(=O)CC(C)C)C1.C(N)=O C=CC(C)(CCOC)C(=O)N1CCC(C)(NC(c2cnc(OC)nc2)=O)C1 c1(C(=O)NC2CCC(NC(C(C(C)C)C)=O)CC2)ncnc2c1CCC2 c1(C(N(CC(CN(C(C(CCCC)C)=O)C)O)C)=O)coc2cc(F)cc(F)c12 C1(C)(C(=O)OCc2c(C)ocn2)C=CCCC1 c1(C(=O)NC(CCOC)C(=O)NCC2(C)CCC(O)CC2)ccc(O)cc1F S(=O)(=O)(c1c[nH]c(C(N2CCC2)=O)c1)NCC.[nH]1cc(CC(CO)CO)nn1.C N1(C(COC(C)C)=O)CC(NC(=O)Cc2ccc(Cl)s2)C2CCCC12 N1(C(c2c(CNC(C3C(C#N)C3)=O)nccc2)=O)CC2CCCCC2C1 C(N=c1[nH]cnc2ccc(F)cc12)C1CCN(C(=O)C=CC2CCCO2)C1 Cc1cc(C)n2ccc(C(N3CCC(NC(c4cnoc4C)=O)C(O)C3)=O)c2n1 N1(C(Cn2ncn(C)c2=O)=O)CC(NC(c2ncoc2C(C)(C)C)=O)CC(F)C1 Cc1[nH]cc(C(N2CC3CC(NC(C4C(C)(C)C4(C)C)=O)CC2C3)=O)c(=O)c1Cl c1(N2CCCC(C)(C)CC2)ncnc2c(Cl)c(Cl)ccc12 Cc1ncc(CCC(=O)NCC2C3CN(C(=O)CCc4ccon4)CC23)c(O)n1 c1(CC(=O)NC2(CCO)CN(C(c3c(C)nco3)=O)C2)ccc2sccc2c1 Cc1cc(C(N2CCC(O)C2)=O)n(C(C)(C)C)n1.C(c1ncc[nH]1)=CC=O.C Cc1ccc(C(=O)NC2CCN(C(=O)CC3(C#N)CCC3)C2C)nn1 Cc1[nH]c2ccnn2c(=O)c1CC(=O)NCC(C)N(C)C(c1csc(C#N)c1)=O c1(C(N2CCN(CCNC(c3cnns3)=O)CC2)=O)ccc(C2CC2)c(F)c1 N1(C(C(CCC)O)=O)CCC(F)C(NC(c2cc(OC)ncc2F)=O)C1 c1(C(C)NC(C(C)OCCCC)=O)nocc1C(=O)NCC.c1ccncc1 C1(C(=O)NC(c2nncs2)C)OCCC1NC(C1CC(CF)C1)=O C1(NC(C2CC=CCC2)=O)CC2CN(C(C3(C(F)(F)F)CCCC3)=O)CC2C1 Cc1c(I)ccc(NC(=O)CSCC2CCCCO2)c1C N1(C(C2N(C(CCC)=O)CC2)=O)CC2CCOCC2(C(=O)O)C1 c1(C(N(C)CC2N(C(C3CC(C)OC3)=O)CCC2)=O)cncc(N)c1 Cc1nccc(-n2cc(-c3nc(Cn4cncn4)no3)cn2)n1 N1(C(c2cncc(C(C)C)c2)=O)C2CCC1CN(C(=O)C1=C(Cl)CCOC1)C2 Cc1c(C(=O)NC2CN(C(=O)CCC3CCCCO3)CC2O)cnn1CC(F)F N(C(=NCCN1CCc2sccc2C1)N1CCCC(C)C1)CCOCC C1(C(N(C2CCN(C(c3[nH]nnc3C)=O)C2)CC)=O)Cc2cc(C)c(C)cc2O1 c1(C(N(CCCNC(CNC(CCC)=O)=O)CC)=O)csc(C2CCCCC2)n1 Cc1cc(N2CC3C(C2)C3(C)C)ncc1S(=O)(=O)N(CC(C)CO)C C(=O)(C(O)C(F)(F)F)NC1(CNC(C(OC)OC)=O)CC1 c1(C(=O)NCCC(C)C)ccnc(N2CCCC2)c1.C1(C=O)CC(N(C)C)C1.N C1(NC(C2(OC)CCSCC2)=O)CC2CC(C1)N(C(=O)Cc1ccn(C)n1)C2 Cc1scc(C(=O)NC(CNC(=O)CSc2cnn(C)c2)CO)c1C C1(NC(c2cc(CNC(C=CC(CC)C)=O)ncc2)=O)CCOC(C)(C)C1 O=C(C1=C2CCCN=C2NN1)NCC1CC(CNC(=O)C(F)C2CCC2)C1 C(=O)(C1Cc2c(Cl)cccc21)N(CCCN(C(CC(CCC)O)=O)C)C CCCC(C(=O)NC1COCC1NC(=O)CCCOC(C)C)OC N1(C(C(COCC)n2cc(CCC3CC3)nn2)=O)C(CN(C)C)CC2CC12 C1CN(C(=O)CCC2CC2(F)F)CC2(CCC2)C1.c1(C=O)ccoc1C1CC1.N C1(CC)CN(C(C2CC2(F)F)=O)CC1C(N1CC(F)(CO)C1)=O c1(C(N2CC(OCCNC(C(C)C3CCOC3)=O)C2)=O)cc(Br)cs1 n1(CCC(=O)NC2CC2NC(c2cc[nH]c3nccc2-3)=O)ccc2ccccc12 c1(C(N2CCC(C)(NC(CN3C(C)CC3)=O)C2)=O)nc(OC(C)C)ccc1Cl Cc1ccc(F)cc1C(=O)N(C)CC1CCN(C(=O)C(C)C(C)(C)C)C1 C1(CN2CCN(C(=O)OC)CC2)CC2(CCCN(C(=O)OC(C)(C)C)C2)C1 CN1CCC2CCN(C(C3(CNC(=O)C(C#N)C(C)(C)C)CC=CC3)=O)C2C1 c1(CC(=O)NC2CCCCN(C(c3coc(O)n3)=O)C2)ccc(Br)c(F)c1 C(=O)(C1=NOC(C)C1)N1CCC2C(NC(c3c(C)sc(-c4nc[nH]n4)n3)=O)C21 N1(C(CCC2C(C)C2)=O)CC2(CCC2C)C1.c1(C=O)csc(C(C)(C)C)n1.N C1(C(C)(C)C)CCCN1C(=O)CC1CCCO1.C(=O)(C)C(=O)C.CCCF.N N1(C(C2CCN(C(C)=O)C2)=O)CCCC(C)(NC(c2cn(CCCF)nn2)=O)C1 C1(NC(c2c(C(C)C)csc2)=O)CCCCC1CNC(C1CCCO1)=O C1(COC)CN(C(C2(O)COC2)=O)CCN1C(c1ccc(C)c(Br)c1)=O CC(C)C(C)C(CNC(c1cccn(C)c1=O)=O)NC(=O)CCS(C)(=O)=O C1(CC=C)(C(=O)Nc2cscc2CC)CCN(C(=O)C=C2CC2)C1 Cn1cc(CCC(=O)NC2CCC(C(=O)NCCCNC(N)=O)C2)cn1 Cc1[nH]nc2c1CC(C(=O)NCC1CCC1NC(=O)Cc1ccsn1)CC2 C1(NC(C(c2n(C)ncc2)(F)F)=O)CCCCC1N=c1nc(C2CC2)[nH]s1 Cc1cc(C)c(C(=O)NCC2CCOC2)cn1.C1(CC=O)NC(=O)NC1=O.N C1(C(=O)NCC2N(C(C(C(C)O)N(C)C)=O)CCCC2)CCCCC1(F)F N1(C(C(C=C)O)=O)CCCC2(CCN(C(c3cc([N+](=O)[O-])c(C)cc3C)=O)C2)C1 N1(C(CC(CC)(F)F)=O)CCc2ccc(C(=O)NC(C)CC(C)C)nc2C1 Cn1cnn(CC(N2CCCC2(C)CNC(C2CC3CCC2O3)=O)=O)c1=O CCS(=O)c1ccccc1C(=O)NC1CC(F)(CNC(C2CC2(Cl)Cl)=O)C1 C(=O)(C1=NOC2(CCC2)C1)NC1(CO)CCN(C(C(C)C2CC2)=O)C1 C1(C#N)(C(=O)NCC2N(C(Cn3c(C)csc3=O)=O)CCC2)CC12CCOCC2 C1(CC)CCOC1C(N1CC(n2cc(C)nn2)C1)=O.c1(C(=O)N)cnc(O)s1 c1(OC)cc(F)ccc1C(=O)NCC(CC(C)C)NC(=O)C(C1CC1)SC Cc1cc(C(F)(F)F)ccc1C(F)F.N12CCC(C1)C(=O)N1CCC(C1)C2 C1(CSC)CCN(C(=O)C(C)NC(C2(C)CC=CC2)=O)C1 CCCC(C(=O)NCC1(CCCO)CC1)NC(c1csnn1)=O c1(OC)ccc(F)c(C(=O)N(C)CC)c1.c1(CC(=O)N)ccc(C(F)F)cc1 C(C1=CCN(C(=O)C(c2cc(F)ccc2C)=O)CC1)NC(C1(C)ON=C(C)C1)=O N1(C(C=O)C)C2CCC1CCC2.C1(C(=O)N)CCC(=O)N1C.CC(C)C.C(N)=O C(=O)(C1=NOCC1)NC(C)C(C)NC(=O)CCc1cscn1 C1(OC)CN(C(=O)CC(C)CN(C)C)CC1C(=O)NCCCF c1(CC(N2CCC(NC(c3c(C)noc3N)=O)C2C)=O)ccc2cccnc2c1 C1(NC(C(C)OCC=C)=O)CC2CCC1CC2.c1(C=O)cn(C2CC2)nn1.N N1(c2cc(C)c([N+](=O)[O-])cn2)CCC2(CCCN(C(C3(C(C)(F)F)CC3)=O)C2)C1 C1(NC(CCC(C)NC(=O)CCS(N)(=O)=O)=O)CCn2nnnc2C1 c1(C(C)(C)OC)nc(=NCC(C(C)(C)C)NC(=O)C(O)C2CCC2)s[nH]1 CCCC(C(=O)N(C1CCCC(NC(=O)CSCC(C)C)C1)C)NC(N)=O N1(C(C(CC=C)C(=C)C)=O)CCc2[nH]nc(-c3ccc(SC)cc3)c2C1 Cc1cccc(C(F)(F)C(=O)N(C)CC2CC2)c1.c1(CCC(=O)N)scnc1C CC1(C)C2CCC13CCN(Cc1c(F)cc(F)cc1F)C3C2 c1(C(=O)NCC2N(C(c3c(C)nc(Br)s3)=O)CCC2)cc2ccccc2cc1O Cc1cccc(-c2nc(CC=O)cs2)c1.N12CC1C(O)C2.CC(=O)C1CC1 C1(CNC(C(F)OC)=O)CC12CCN(C(c1cccc3cnsc13)=O)CC2 Cc1nc(N2CC=C(CNC(=O)Cn3ncc4ncccc34)CC2)c(C)c(Cl)n1 C1CCC12CCN(C(C1CN(S(N)(=O)=O)C1)=O)CC2.C(C=O)C1CC1.CCO c1(C(=O)OC)ccc(C(=O)NCC2CCN(C(C3(F)CCCCC3)=O)C2)nc1 N1(C(CCC2C(C)C2)=O)CCCC12CCN(C(C1CCC(C)(C)OC1)=O)C2 c1(NCC2OCCN(C(C3(C4CCCO4)CCOCC3)=O)C2)cc(O)ncn1 CN=c1[nH]cc(C(N2CCCC2CCNC(C23CC(C)C2C3)=O)=O)o1 S(=O)(=O)(c1ccc(OC(C)C)cc1)N1CCCC(C(=O)NC(C=C)CO)C1 N1(c2ccc(OC)c(OC)c2)CCC(C)N(C(=O)C(C)N)CC1 c1(OC)ccc2c(C(=O)NCC3CC(C)N(C(c4ccoc4Br)=O)C3)cnn2c1 CCC(C)C(O)C(=O)NCC1(NC(c2cnn(C3COC3)c2)=O)CCOC1 C1(C(=O)NCCN(C(=O)COCC(C)C)CCC)CC(C)=NO1 N1(C(c2coc(C(F)F)n2)=O)CCN(C(=O)C2=COCCC2)C2COCC12 C1(NC(C(F)=C(C)C)=O)CN(C(=O)C(C(C)C)n2cccc2)Cc2ccnn2C1 N1(C(CCC(=C)Cl)=O)CC2CCOC2(CNC(=O)CCC(=O)NCCCOC)C1 CCC(CCC(=O)OC)NC(C1CCN1C(c1sccc1F)=O)=O C1(NC(c2cc(OCC)ncc2)=O)CN(C(=O)Cc2nocc2C)C2CCCC12 C1(NC(COCCC)=O)CCC2(CCN(C(C3(C(F)F)CC(O)C3)=O)C2)C1 C(=O)(C(C)C(C)COC)N1CCN(C(C2(C(=O)NC)CCC2)=O)CC1 N1(C(=O)CC2CCCN2C(C2CC2(F)Cl)=O)CCCN(C2CC2)CC1 c1(OC)c[nH]c(=NCCCN2C(=O)CCCC2=O)c(C)c1O Cn1cc(C(=O)NCC2(NC(=O)Cc3ccc(Cl)nc3)CCCC2)c(=N)[nH]1 C(CN=[N+]=[N-])(C(=O)NCC1=CCCCC1)NC(C(CCC)OCC)=O C(CC(C)C(=O)NCC1(O)CCN(C(c2nc[nH]c2C(C)(C)C)=O)C1)OC CCC(CC)C(C(=O)N1CC2(CC2)CC1CC(=O)NCc1ccco1)OC C1(NC(c2ncn(CC)n2)=O)CCN(C(c2ccccn2)=O)C1C(C)(C)C.O N1(C(c2cc(OC)n[nH]2)=O)CC2CC3CC2C1C3NC(=O)CCc1cc(Cl)no1 c1(C(=O)NCC(C)NC(c2ccc(SC)s2)=O)cnc(-c2ccoc2)[nH]c1=N n12cc(c(O)nc1=O)C2.c1(C2CN(C(=O)OC(C)(C)C)C2)nc(C2CC2)no1 c1(C(=O)NCC(C)NC(C(CC)C2CCOCC2)=O)cnc2nccn2c1 C1(SC)CN(C(=O)Cc2ccoc2)CC1C(=O)NCCc1nnc(C)n1C c1(C(=O)NCC2ON=C(C(=O)NCCc3nnc(O)o3)C2)cc2ccccc2[nH]1 Cc1cc(C(=O)N)cc(Cl)c1.C(c1nnc(C(C)C)o1)=CC=O.CC(C)(O)C c1(OC)cc(CO)ccc1-c1cncc(C(=O)N(CCCO)CCCO)n1 c1(C(N(CC(=O)NC(C)C(C)(C)OC)CCC)=O)cc(C#N)[nH]c1C N1(C(c2cc(CNC(CSCCC(C)C)=O)oc2)=O)Cc2ccncc2C1 c1(CN2C(C(=O)Nc3cc(C)c(Br)cc3)CC2)ccc(Cl)cc1[N+](=O)[O-] C1(O)(CC(=O)NCC(CC)C(=O)O)CCCN(C(=O)OC(C)(C)C)C1 c1(OCC)nc(N2CCC(NC(c3ccc(Br)cc3O)=O)C(F)C2)ncc1C CC1(CNC(=O)C=CC2CC2)CCN(C(=O)C=CBr)C1 C1(N(C(c2cc(C(C)C)n(C)n2)=O)C)CCCN(C(=O)CCC2CC2(Cl)Cl)CC1 C1(C(=O)NCC(CNC(c2cnc(CC)[nH]2)=O)(C)OC)(CO)CCCCO1 C1(CC)CCC(O)(C(=O)NC)C1.C1(C(F)F)CCN(C(c2ccsc2Cl)=O)C1 CCC(CC(=O)N(C)CC1CCCCCC1)NC(=O)CC1CCC(C)(C)O1 C(=O)(C1=NOC2(CCC2)C1)NCC(CNC(Cc1c(SC)cccc1)=O)F Cc1cc(C(N2C(C(=O)NCCCF)CCC2C2CC2)=O)cnc1C N1(C(C(CC=C)OC)=O)CCN(C(C2CC2c2ccco2)=O)C2(CCC2)C1 c1(C(N2CCC(CC)C2)=O)cc(S(N)(=O)=O)c(Cl)o1.c1oncc1C=O.CC c1(C(N2CCCC(NC(C3C(OC)CCCC3)=O)C2)=O)c(F)cc(Cl)cc1Cl N1(CCOC)CCN(C(c2cc(C)co2)C(=O)NCCC#N)CC1 C(CCN=C(NCCN1CCC2CCCCC2C1)N1CCC(F)(C#N)C1)OC C#CCC(C)(C(=O)Nc1cc(C)cnc1O)NC(c1cnnc(O)c1)=O c1(NC(c2ccnn2C)C)nccc(N(C)Cc2nnc(CO)n2C)n1 c1(C(=O)NC(CC)CNC(C2(C3CCC3)CC2)=O)cnn2c1CC(F)(F)C2 N1CCCC2(CC2)C1.C1(C(NOCC(=O)C(=O)C)=O)CCOCC1 CCCC(C(=O)N(C)CC1C2CN(C(c3cc(N)nc(Cl)c3)=O)CC12)C(C)C n1(CC(=O)NCCCCNC(CC2ON=C(CC)C2)=O)cccc([N+](=O)[O-])c1=O C1(NC(c2n(C)nc([N+](=O)[O-])c2)=O)CCCC(N=c2[nH]c3cc(F)cc(F)c3o2)C1 c1(C(=O)NC2CCC(NC(C3C(=C)CC3)=O)CC2)sccc1S(N)(=O)=O C(=O)(C1=CCCCC1)N1C(CCNC(C2(CC)CC2)=O)CC(OC)C1 C1(C(N2CCC(F)(CNC(C(C)NC(N)=O)=O)CC2)=O)CCc2nncn2CC1 c1cc(C(=O)O)nc2ccccc12.C1(C(=O)N)CCC2(CN(C(=O)C3CC3)C2)O1 c1(OCC(F)F)cc(Br)cnc1NCC1CCC2(CC1)CC2 C(CNC(=O)C(O)C1CCCC1)(CNC(C1(SC)CC1)=O)OC c1(C(c2nnnn2C2COC2)NC(CC)C)c(Br)sc2ccccc12 Cc1c(C2(C(=O)NCCCC)CC2)cccc1F.C(=O)C(CN(C)C)N(C)C.N c1(NCc2cccc(CCC(=O)OC)c2)c(F)ccc(C(=O)OC)c1F C1(C(CNC(=O)Cn2cc(Cl)cn2)F)CCN(C(=O)CC2CC(=O)NC2=O)CC1 CC1CCC(C)(C(=O)NC2C3CC4C2C4C3C(=O)NC2CCCC2(F)F)CC1 Cc1nc(C)c(C(=O)NC2CCCC2O)c(C)n1.c1(C(=O)N)cccn1C(C)C CC1(C)C(C(N2CC(CNC(c3ccoc3)=O)C2)=O)C1(F)F c1(C(N2C(CN(C(CC3N(CC)CCOC3)=O)C)CCC2)=O)ccn2ccsc12 c1(C(=O)NCC2CCC(C)CN2C(c2cc(O)n(C)n2)=O)c(F)cc(F)cc1F CS(=O)(=O)CCCCCCCC(=O)NC1CCN(C(=O)Cn2cccc2)CC1O C=CCC(CC)C(=O)N1CCC(C(=O)N2CCCc3ccnn32)O1 C(=O)(CC(C)P(C)(C)=O)NC(COC)CNC(c1ccoc1Cl)=O N1(C(Cc2nc(CC)sc2)=O)CC(C)OC(C)(C)C1.C(=O)(CCc1cscn1)N c1(CNc2cccc(C3CCN(C)CC3)c2)c[nH]c2ccc(OC3CCC3)cc12 N1(C(c2c(OC)cc(F)cc2)=O)CCCC2(C1)CN(C(c1csc(C)c1)=O)C2 N1(C(C2(OC)CCCC2)=O)CCC(C(F)CNC(=O)C(C)C2CCC2)CC1 c1(C(N2CC(C)(C)C2C2CCN(C(=O)C(N)=O)CC2)=O)cc2n(n1)CCC2 N1(C(c2ccc(C(C)O)cc2)=O)CC2OCCN(C(c3ccc(=O)oc3)=O)C2C1 N1(C(=O)CC=C(Cl)Cl)CC(O)(C2CCN(C(=O)C3=COCCO3)CC2)C1 O=C(C1=COCCC1)NC1C2CC3C(C2)C13C(=O)NCC1CC1[N+](=O)[O-] C#CC1(O)CC(C(=O)NCCC(O)CNC(C2CC2(C)C)=O)C1 c1(C(N(C(CNC(CSCC#C)=O)C)C)=O)cc2cc(Br)cn2cn1 C1(NC(c2c(C)csc2)=O)C2CC3CN(C(=O)C(N4CCCC(C)C4)=O)C1C3C2 c1(C(=O)NC(c2ncccn2)C2CC2)cnc2[nH]c(O)nc2c1 N1(C(CCOC)=O)CC2CCC1CN2Cc1ccc(O)cc1OC(F)(F)F N1(Cc2snc(C(C)(C)C)n2)CCNc2ccccc2C1 C1(NCCc2ccc(OCCCCC)cc2)CCC(O)C2(CCCC2)C1 CC1=C(C(=O)NCC2(F)CCC2)C(C)(C)CCC1.C1(C=O)CC1C(F)F n1(CC(N2CCC2)=O)ccc([N+](=O)[O-])n1.c1(C(C)=O)cccc(C(=O)N)c1.C CC(C(=O)NC1CN(C(=O)C=Cc2cccnc2)CC1n1cccn1)C(C)O C1(CC(=O)N)C(=O)NN=C1C.c1(CC(=O)N(CCC)CC)nc(C)sc1Cl C=CCC(CNC(c1ccsc1C(F)F)=O)NC(=O)Cc1cnc[nH]1 N1(CCNC(CCSCC)=O)CCCN(C(=O)CCCC(=O)OC)CC1 N1(C(C(=O)N(C)C)=O)CC(CNC(=O)CC2CCC(=O)N2)C2(CC2)C1 C(=O)(CC1OCc2cc(Cl)ccc21)N.C1(NC(=O)CSC(F)(F)F)CC2(C1)CC2 C(=O)(C(C(C)(C)C)NC(c1ncccn1)=O)Nc1c(OC)cccc1 c1cccc(-c2cnco2)c1.C1(O)(CC(=O)N)CN(C(C2(C(=O)O)CC2)=O)C1 N1(C(C)=O)CSCC1C(=O)NCCCNC(C1CC12CC2)=O c1(CNC2CCCC(NC(C3CCN(CC(F)F)CC3)=O)C2)cc2n(n1)CCC2 Cc1c(C(=O)NC23CC(C(N4CC5C(C4)C5(F)F)=O)(C2)C3)cccc1C#N C1(C(C(=O)N(CCCCC=C)C)C)CCCN(C(c2cc[nH]c2)=O)C1 N1(C(C2CC(=C3CC3)C2)=O)CC2(C1)CN(C(C13COCC1C3)=O)C2 c1(C(C)NC(C(CN(CC)CC)F)=O)ccccc1.C(=O)C(F)=C1CCC1 CC1OC2(C)CC1(C(=O)NCC(O)CNC(c1c(Cl)cncc1Cl)=O)C2 c1(C(N2CCC(O)(C(C)NC(C(n3ncc(C)c3)C)=O)C2)=O)cc(C)c(C)nn1 CC1(C)CC2(CC(c3nnnn3CC(F)F)(NCc3ccc4sccc4c3)C2)C1 N1(C(C(C2CCCCC2)C)=O)CC(O)(C(F)C(N2CCC(n3cncn3)C2)=O)C1 C(C)(CC(=O)N1CCC2C(NC(c3cccc(O)n3)=O)C12)(C(F)F)N(C)C c1(C(=O)NCC2OCCC(NC(c3c(CC)nc[nH]3)=O)C2)ccc(N)cc1C Cc1cc(C(N2CCCC(C(C)NC(c3coc(C)c3)=O)C2)=O)nc(N(C)C)n1 c1(C(N2C(CC)C(NC(=O)CC3CSC3)CCC2)=O)ccnc2ncnn12 C1(NC(C(OC)OC)=O)COCCC1NC(c1cnnc(O)c1)=O c1(CC=O)cc[nH]c(=N)c1.n1(CCC=C)cc(C(=O)NCC=CC)nn1.N C=CC(CC)CC(=O)NCc1ccc(C(=O)N(CCCC(C)O)C)cn1 CC1(C)CC(NC(=O)C=Cc2nccs2)CN1C(=O)COCC(F)F C1(NC(C(C)NC(C)=O)=O)CC2(CCN(C(=O)C(F)(F)CC3CC3)C2)C1 c1(C(N2C(C(C)NC(c3csc(Cl)c3)=O)CCC2)=O)cnn2ccc(Cl)c(F)c12 C1(CNC(C2N(C(C)C)CCC2)=O)CCCN(C(=O)CC2CCCC2)CC1 C1(C)(CNC(CCNS(CC)(=O)=O)=O)COCCN(C(=O)C(C)O)C1 C1(CNC(CN(CC)CC)=O)CC(F)CN1C(c1ncc[nH]c1=O)=O N1(CC(=O)Nc2cnc(-c3nn[nH]n3)c(Br)c2)CCc2ccccc2C1 c1(CNC(N2CCC(CN3CCCC3=O)CC2)=O)ccc(Cl)cc1I Cc1c(C(=O)N(CCCCCCNC(c2cn(C)nc2O)=O)C)noc1C1CC1 C(=O)(CCC(=O)NCC(C)N(C(=O)C(C)(C)c1sccc1Cl)CC)NCCC C(=O)(N1CC(O)CCO1)C1C2(CCN(C(c3cncc(O)c3)=O)C2)C1 N1(C(c2cnc(S(C)(=O)=O)s2)=O)CC(CO)C2(C1)CN(C(C1CCCS1)=O)C2 c1(OCC)cccc(C=CC=O)c1.C(=O)C=CS(C)=O.C1(CC)CCCC1.N c1(OC)ncc(F)cc1C(N1CC(NC(C2(O)CC2)=O)C(C#N)C1)=O C1(CNC(CCC(C)NC(COCC#C)=O)=O)CCC(=O)NC1C C1(C(=O)N)CC2CCC1NC2=O.c1(C(=O)NCCOCC)cc2cccnc2[nH]1 CCCC(O)CC(=O)NC12CCC(CC1NC(C1C3CC4C(C3=O)C14)=O)C2 c1(C2(C(=O)N)CC2)cc(Cl)cc(Br)c1.N1(C(c2cccnn2)=O)CCOC(C)C1 C1(NC(C(C)CC(F)F)=O)CCN(C(c2ccc(N)c(F)c2)=O)C12CCC2 C(=O)(C1=NNC(=O)CC1)NCC(C(C)(C)C)NC(C(COC)C)=O C1(C(N(CC=O)C2CCC2)=O)CC2(CCCO2)C1.CC(C)CC1CCOC1.N N1(C(c2ccc(CSC)o2)=O)CC(C)C(C)(C)C1.C(=O)(CC(C)C(C)C)N c1(CC(=O)NC(CCCC)CNC(=O)C(O)c2ccsc2)cccc2nsnc12 c1(CC(=O)N(CCNC(c2ncc(C)c(C)c2)=O)C2CC2)cccc2ccsc12 n1(C(C)C)ccnc1C(N1CCC(C2CCCN2C(=O)C(C)N(C)C)C1)=O N1(C(C2(C#N)CCCC2)=O)CC(NC(c2csc3ccccc23)=O)C2(CCC2)C1 Cc1nc2cc(C(=O)NCC3CC(NC(C4CCCCC4(F)F)=O)C3)ccc2o1 N1(C(CCCC=C)=O)CCCC(O)(CNC(C2CCC2(F)F)=O)C1 C1(COC)CCN(C(=O)C(C)CS(C)=O)CC1.c1(C=O)cnn(CC(F)F)n1.N C1(OC)CCCCC1CN(C)C(c1ccc(C(=O)O)s1)=O C1(NC(CN(C(C(C)SCCCC)=O)CC(C)C)=O)CCN(C)CC1(C)C c1(N(C2CC(N)C2)C(c2coc3ccccc23)=O)ncnc2c(Br)cccc12 C1(F)(C=O)CS(=O)(=O)CC12CCC2.CC(C)(C)C(C)(O)C(=O)N.C1CCC1 N1(C(c2c(C)nc[nH]2)=O)CCC(C(F)(F)F)CC1.c1(C(=O)N)n[nH]cc1C(C)C N1(C(C2CC(C)(C)C2)=O)CC2CCC2(CNC(C2CC2)=O)C1.c1ccccc1 c1(CN2C(CCC)COCC2)cc2cc(Cl)ccc2s1 CCC(C)C(C(=O)NC(C1CC(NC(=O)CC(=O)OC)C1)C)N(C)C c1(C(N2CCC(CNC(C3CC=CCC3)=O)C2)=O)cc(Cl)c(O)cc1F CC(C)(C)C(CNC(C1CC1C(=O)NC1CC=CC1)=O)CO N1(C(C2(CCC=C)CN(C(c3coc(C(N)=O)c3)=O)C2)=O)CC(O)CC(F)C1 C1(NC(C2(C)C(C)(C)C2)=O)CCCCN(C(C2(C)CC2c2ccccc2)=O)C1 C1(C(=O)NCCCN(C(c2c[nH]cc(Br)c2=N)=O)CC)CCC12CCCO2 CN1CC(C(=O)NC2CCCC(C(=O)NC3C(=O)OCC3(C)C)CC2)CCC1=O C1(CNCCCc2onc(C)n2)CCCN1NC(=O)C(C)SC(C)C C#CCC(C(=O)NC(CC1CCCC1)C(=O)Nc1cccnc1)C1CC1 CCC(CC)C(C)C(=O)NCCC(C)NC(c1sc2sccc2c1Cl)=O C1CN(C(=O)C(C)(C)O)CCC1C(F)(F)F.Cc1onc(C2CC2)c1C(=O)N C1(NCc2cc(C)cc(F)c2)CCCC2CN(C(c3ccnnc3)=O)CC12 C=C1COc2c(C(=O)NC3(CNC(=O)C(C)(F)F)CCCCC3)cnn2C1 C(CCC)(C(=O)NCCNC(=O)CCn1cccnc1=O)=CCC.C1CC1.C N1(CC(C)C)CCN(C(C2(C)CN(C(c3ccnc(Cl)c3)=O)C2)=O)CC1 c1(N2CC(COC)OC(C)(C)C2)cccc(S(=O)(=O)NCCC(C)C(F)F)n1 n1(CC(=C)C)nnnc1C(c1csnc1C(F)F)NC1CCC(C(=O)O)C1 N1(C(CC2CN(C(C(C)SC)=O)C(C)(C)C2)=O)C2C=CCC1CCC2 C(=O)(CCC(=O)N1CCCCC1CN(C(=O)CCC(C)=O)C)OCC c1(NC(C2Cc3c(C)scc3CC2)=O)ccc2c(c1)CCCN2CC(=O)N(C)C c1(SC)cnc(N2CCC(C(C(F)(F)F)NC(c3ncccc3Cl)=O)CC2)nc1 C1(CC#C)(C(=O)N(CCOC)CC)CCN(C(=O)CCc2ccncc2)C1.O N1(C(C)(C)C)CCCC(C)(C(=O)NCC(Cl)Cl)S1(=O)=O C1(CNC(c2c(C)onc2)=O)CN(C(C2(c3cncs3)CC2)=O)CCC1C c1(C(N(CCCN(C(C2OCCN(C)C2)=O)C)C)=O)cnc2[nH]nnc2c1 C=CC1CCN(C(C2CC(C)N2C(C2(COCC)CCC2)=O)=O)CC1 C(=O)(CC(O)CC(C)(C)C)NC(COC)C(=O)NC1(c2noc(C)n2)CC1 C1(NC(C(CC)=CCCC)=O)(CF)CCN(C(C2CC(F)(F)C2)=O)C1 N1(C(C(CC)CC(C)C)C(=O)NCC(F)F)CCc2c([nH]c3ccc(F)cc23)C1 C1(CN(C(c2nnc(C)s2)=O)C)CN(C(=O)C(O)C(F)F)CCO1 C(=O)(CC(O)CC(C)C)NC(CNC(c1c(OCC)c(F)ccc1)=O)C(C)C c1(C(=O)NC2CN(C(c3nc(C)[nH]n3)=O)CC2F)ccn2nncc2c1 N1(C(C)=O)CCOCC1C(N1CCCC(C(=O)Nc2ccnc(C)n2)C1)=O N1(C(C(C)C2(O)CCC2)=O)CCC2(C1)CN(C(=O)CC13CCCC1C3)C2 c1(C(C(N2CCC(CNC(C(C=C)(C)O)=O)(O)C2)=O)=O)ccc(F)c(F)c1 Cc1oc(C(=O)NCC2(CN(C)C(c3cccnn3)=O)CC2)cc1CO c1(NC(CCc2ccc(C(=O)NC3CC(=O)OC3)[nH]2)=O)cccc(O)c1O C(=O)(CC(O)CC(C)(C)C)NC1(CO)CCN(C(CC(C)c2ccco2)=O)CC1 C1CCS(=O)(=O)C12CN(C(C1(N(C)C)CC1)=O)C2.C(=O)CCCC=O.CC.N c1(C(=O)NC2CCC(N(C)C(C3CCC4(C3)N=N4)=O)CC2)ccc2[nH]ccc2n1 C(=O)(C1CCCn2cnnc21)N1CCN(C)CC1CNC(C1CCC2(C1)N=N2)=O c1(NC(CCC2CCCN(C(C(C)NC=O)=O)C2)=O)ccc2occc2c1 Cc1nn(C)c(C)c1C(=O)NC1C=CC(C(=O)NC(C)C(C)F)C1 N1(C(C2C(C#N)C2)=O)CCC(O)(CNC(c2ccc(-c3cc[nH]n3)cc2)=O)CC1 N1(C(c2ccc(OC(C)C)cc2)=O)CCCC(C)(C)C1.c1(C(=O)N)cc(Cl)cs1 C(C(O)CN=c1cccc(S(=O)(=O)N2CCC3(CCCO3)C2)[nH]1)OC C(CC1CCCC1)(C(=O)NOCCCO)NC(c1c(OC)ccnc1)=O c1(C(=O)NC2(C)CN(C(c3c(COC)nn[nH]3)=O)C2)cc2sc(C)cc2s1 CC(CN=c1[nH]c(=NC(C)c2cn(C)nn2)[nH]c2ccsc12)c1ccsc1 c1(OC)ncc(C(c2nnnn2CC)NCC(c2cccc(F)c2)(C)C)cc1Br c1(C(N2CC(OC)(CNC(C3COC(=O)N3)=O)C2)=O)cccc2oncc12 c1(C(N2C(C)(C)CC(NC(C3CC3(C)C)=O)C2)=O)cc2cc(F)ccc2o1 C(CCC(=O)NCCCn1ccnc1)(C(C)C)NC(c1c(OC)ccnc1)=O c1(OC)cccc(S(=O)(=O)N2C(C(N3CCC(F)(F)CC3)=O)CC3CC23)c1 c1(C(=O)Nc2c(C)nc(Br)cc2)cc(-c2c(F)cc(F)cc2F)c2cn[nH]c2c1 c1(C(=O)NCC2(C)CC(NC(C(CC=C)(F)F)=O)C2)cnc2ccsc2c1 c1(C(=O)NCCN2CCN(C(C(C(COC)C)C)=O)CC2)cnn2ccncc12 S(=O)(=O)(c1c(Cl)cc(Cl)cc1Cl)NCC(=O)NC1c2cccc(C)c2OC1 C1(C(=O)NCCn2cc(C(=O)NC3CC(OC)C3)nc2)CCCC1C1CC1 CC1(C)OC(C(N2C3CCC2CC(NC(c2ccsc2)=O)C3)=O)C(C)(C)O1 c1(OC)ccc(CNC(=O)NCC2(Sc3ccccc3F)CC2)cc1 C(=O)(CC1=CCCCC1)N1CCC(CC#C)(C(=O)NC(C)CC#CC)C1 CON(C(=O)C(O)CNC(=O)CCC1CCCN1C)C(C)C C(CC(C(=O)NC1(C(O)CO)CC1)NC(c1cncnc1)=O)OCC Cc1ccc(C(C)C)c(CNC2CCOCC2C(C)C)c1 Cc1ccc(C(N2CCC(CCNC(=O)CC3CCC(=O)N3C)C2)=O)c(O)c1C N(C1CCCn2cnnc21)C(C(CO)NC(C1CCC(C)(O)CC1)=O)=O CC1CCC=C1C(=O)N1CC=CC(C(=O)N(C)CC2CCCOC2)C1 CC(O)C(F)(F)C(=O)NC1CC2CCC2C1.c1(C(=O)N)cnc(S)n1C1CC1 CC#CCCC(=O)NC(c1ccccc1)C(=O)NC1CCCC1(F)F C1(CNC(c2cc(C)c(Cl)cc2)=O)CC2CC(C1)N(C(c1cc(Cl)ccn1)=O)C2 C1(C(N(C)CCN(c2ncc(Br)c(O)n2)C)=O)CCCC(F)(F)C1 c1(OC)c(F)ccc(C(N2CCC(C(C)NC(C3(C#N)CCCC3)=O)C2)=O)c1F c1(CC(=O)NC(CC)CN(C)C(C2(CC)CCOC2)=O)ccc(C(C)C)cc1 C(C)(CCC(=O)N(C(C)CCNC(c1cncc(C(C)(C)C)c1)=O)C)SC C1(NC(c2cnc3cnccc3c2)=O)CC2(C1)CC2N=c1nc[nH]s1 N1(C(c2nc(CC)oc2)=O)CC(F)(F)CC1C(=O)NCC(C)CC(=O)OC Cc1cc(C)n(CC(=O)NC2CC(N(C)C(c3ccc(O)cc3C)=O)C2)c(=O)n1 C1(NC(CC(=O)N)=O)CN(C(c2cnc(S)n2C2CC2)=O)CC1F.C1CC1.C C1(C(C)C)CCC(C(N2CC(CCNC(=O)CC=C(Cl)Cl)C2)=O)CC1 Cc1cnc2ccccc2c1C(=O)N(C1CCN(C(C2CCCC2C)=O)CC1)C C(=O)(N=S(=O)(CCN)CCO)c1cc(OC(C)C)c(Br)cc1 C1(NC(c2n(CCC)ccc2)=O)CN(C(c2c(C)oc(C)c2C)=O)CC(C)(C)C1 CC1(C)CC(C(=O)NC(C2CCCCC2)CNC(=O)Cc2cccs2)CNC1=O C1(C(N(CCCN(C)C)C)=O)CCN(C(=O)CN2CCOCC2)O1 c1(CNC2CC(C(N(C)Cc3ccccn3)=O)C2)c(F)c(F)cc(F)c1F C1(NC(C(COCC)NC(=O)CCn2ccnc2)=O)CC2(CCC2)C1O N1C2CCC1CN(C(=O)CC1C3CCC(C3)N1C(=O)CN1CC3CC3C1)C2.CC CN1C(=O)C(CC(=O)Nc2cnn(CCN(C)C)c2)c2ccccc21 CC1CN(C(c2ccccc2CNC)=O)CC(C)O1.c1cc(C(=O)O)cc(Br)c1 c1(NC(C2CC(C)CN2C(=O)C(CO)c2ccccc2)=O)ccc(O)c(F)c1 C1(CC(=O)NC2(C(=O)NC(c3ccns3)C)CCC2)CCCC12CC2 C(=O)(CCC(=O)NCCCCC(C)NC(=O)C(C)O)NCC.c1ccc(Cl)cc1 N1(C(C2(COC)CC=CC2)=O)CCC(NC(C23COCC(C2)C3)=O)CC1.C c1(CN2CCC(O)(C(N3CC4CC3CO4)=O)C2)nc(Br)ccc1F c1(C(=O)NCC2CCN2C(c2cnccn2)=O)ncn2cc(Cl)ccc12 C1(C(N2CCC(C(=O)OC)CC2)=O)CC12CCN(C(c1cccc(C)c1)=O)C2 Cc1cc(-c2csc(NC(C3CCC(NC(N)=O)CC3)=O)n2)c(C)n1C c1(CCC(=O)NC(CC=C)CNC(=O)COC2CCC2)c(F)cccc1F CC1=C(C(=O)NC(C2CCCN(C(=O)CCC3CCN(C)CC3)C2)C)CCO1 CN1CCN(C(c2nccn2C)=O)C(CNC(=O)CC2CC(F)C2)C1 N1(C(c2nn(C)c(Cl)c2Cl)=O)CCC2(CC1)CC2CNC(=O)C(C)(C)CF Cc1[nH]c(=O)c(C)nc1NC1CCC(=O)N(c2cccc(F)c2)C1 C(=O)(C(F)C(C)(C)O)NCC(C)NC(Cc1ncc(CC)[nH]1)=O Cc1cc(C)c(C(=O)NCC2CC(NC(=O)C(C)(C)N(C)C)C2)[nH]1 C1(C)CCN(C(C2C(Cl)(Cl)C23CC3)=O)C1.c1(CC(C)C)ncc(C(=O)N)s1 C1(C(=O)N)CCC2(CCC2)OC1.Cc1[nH]c(C(C)(C)C)cc1C(=O)N(CCC)C N1(C(C2(C=C)CCN(C(c3snnc3CC)=O)C2)=O)CCOC(C)(C)CC1 c1(C(N2C(C)(CNC(Cc3c(C)nc[nH]3)=O)CCC2)=O)ccc2c(n1)CCCN2 C(=O)(C1c2ccccc2CN1C(c1cnccc1C#N)=O)NCC1(C)OCCO1 C(C=O)C(C)C.C1(CC)CCN(C(C2CC3(CCC3)C2)=O)CC1.C(=O)(OC)N Cc1ccc(SCC(=O)NC2(C)CCN(c3cc(=O)n(C)cn3)C2)c(Br)c1 c1(CC)n[nH]cc1C(=O)NC1(C(N2CCC(CSC)C2)=O)CCSC1 N1(C(c2ccc(OC)cn2)=O)CC(C(=O)NCCc2ncoc2C)CC12CCC2 c1(C(N2CCCC(C)C2CNC(C2OCCCO2)=O)=O)cc(F)c(Cl)cc1F N1(C(C(C)(Cl)Cl)=O)CC2(C1)CN(C(c1cncc(CO)c1)=O)CCO2 Cc1cc(C(N2CCCC(O)(CNC(=O)CCCC(F)(F)F)C2)=O)cc(F)c1C c1(CC(N2CCC(O)C2)=O)cnc2c(C)cccn12.C(C(=O)NC)NC(C)=O c1(CC(=O)NCC2CCCCN(C(c3csc(Cl)c3)=O)C2)cccc(F)c1O N1(C(C2C(C)(CC)C2)=O)CC2(CCCN(C(C3CC(O)C3)=O)C2)C1 c1(C(N(CCC(=O)NCCn2ccnn2)C(C)C)=O)cc([N+](=O)[O-])n[nH]1 C(=O)(CC(C(C)OC)NC(=O)CC1CSCCO1)N1CCC(O)(CC)C1 c1(NC(CC2N(C(C=CC3(C)COC3)=O)CCOC2)=O)ccc2c(c1)CCO2 CCC(CC(=O)NCCC(C)CCNC(c1nn(C)c(C)c1Br)=O)C(F)F C1(NC(c2cc(CCOC)on2)=O)CCCC(NC(C2(CF)CCC2)=O)CC1 C1(C(=O)NC2(C)C(C)CCC2)CN(C(c2cccc(O)n2)=O)CC1(F)F C1(NC(=O)C(C2CCOCC2)F)CN(C(C23CCC(CC2)CC3)=O)CC1C1CC1 C12(CNC(CN(C(=O)C(C)C3CC3)CC#C)=O)COC(C1)C(O)C2 c1(CNC(CCCOCC=C)c2nnnn2C)c(OC)cccc1OC CC(C)(C)C(C#N)C(=O)N1CC(O)(C(F)C(N2CCOCC(CO)C2)=O)C1 C1(NC(c2ccon2)=O)COCCN(C(=O)C=CCBr)C1 c1(C(=O)NC2CN(C(CC)=O)C2)coc2c1CN(C(=O)CC1C=CCCC1)C2 Cc1c(C(=O)NC2CC(C(=O)Nc3c(Cl)cnnc3Cl)C2)cc(Br)cc1F C1(NC(CC(C)C(F)F)=O)CC2(CCCCN2C(=O)CC2CC2(Cl)Cl)C1 c1(C(=O)NC(C2CCN(C(C(C)=C3CCCC3)=O)C2)C)cn2c(n1)CCC2 c1(C(N2CCC(NC(c3c(OC)cnc(Cl)c3)=O)C2)=O)cccc2c(C)[nH]nc12 c1(C(=O)Nc2onc(C)c2Cl)cnc2c(c1)CCN(C(C1CC1C)=O)C2 CC(CC(=O)NC1COCCC1NC(=O)CCc1nnc(C(F)F)o1)C(F)F Cc1c(C(=O)NCCCN(C(=O)CCc2cnco2)C)cnn1C(C)C CCC(CC(=O)NCCCC(O)CO)NC(C1CC1(Cl)Cl)=O C1(CNC(CCN(C)CC)=O)CCN(C(C2CCCOC2)=O)C1 C(=O)(CCCS(C)(=O)=O)N(C1CCN(C(=O)C(C)C#N)CC1)CCOC C1(CC)C(C(=O)NCCN2CCC(OC)C2)CCN1C(c1cc(OC)no1)=O N1(C(c2cncc(N)c2)=O)CC2CCC(CNC(c3csc(Cl)n3)=O)C2C1 C1(C(N(CC(C)C)CCC)=O)CC2(C1)CN(C(c1cc3sccc3s1)=O)C2 C1(NC(C2CC(=O)NC2)=O)CC2CC(C1)N(C(=O)Cn1nnnc1C1CC1)C2 Cc1ccc2[nH]nc(C(=O)NC(C)CCNC(=O)CCOC3COC3)c2c1 C(C)(CCCC(=O)N(C1CCOC1)CCO)NC(Cc1c(C)nccc1)=O C(c1cccc(C)c1)=C.CCC(CO)N(CCC(=O)N(C)C)CC=C(C)C C1(C2CCC2)(CNC(C2CCCS2)=O)CCN(C(=O)CCn2cccc2)CC1 N1(C(C2C3C(NC(CC(CC)CN(C)C)=O)C4C(C3)C42)=O)CCC(C2CCCC2)C1 C1(CN(C)C(c2ccnn2-c2ccncc2)=O)C2CN(C(C3SCCS3)=O)CC12 c1(C=O)ccc(Cl)c2cccnc12.C1(C(=O)NC)(OCC)CCCC1.C1CC1 C1(CC(=O)NCCCCCN(C(=O)CCOC2CCC2)C)CCCC(C)(C)O1 CC1(C)CN(C(C2C3CCC(F)C23)=O)CCC1C(=O)NC1(C2CC2)CCOC1 Cc1oc(C2CC2)nc1C(=O)NC(C)(C)CC.C1CCN(C)CC1.C(=O)C.N C(=O)(C(C(=O)OCC)C(C)C)NC(CC1CCN(C(CC=CC=C)=O)CC1)C C(=O)(C(C)(C)CCF)NC(COC)CNC(=O)CC(C)C1CCCCC1 CC1CC(C(=O)NCCc2ccco2)N1C(=O)CNC(N)=O c1(CC(CSC)C(=O)N2CCN(c3ncc(F)cn3)CC2)ccc(F)cc1F c1(OC)cccc(Cl)c1C1CC1C(N1CCN(C(=O)CS(=O)(=O)OC)CC1C)=O c1(C(=O)NC2(CNC(c3c(C)ccs3)=O)CC2)cc2cc(Cl)ccc2s1 N1(C(CC(C=C)CC)=O)CC2CCCC(C1)N2C(=O)COC1CC=CC1 CCCC(CC)CCC(=O)N(C1CN(C(c2coc(OCC)n2)=O)CC1(C)C)C C1(C=O)CS(=O)(=O)CC(=O)N1.C1(N(C)C(c2cnn(C)n2)=O)CCCCC1.N C(C)(c1ccccc1Cl)=CC(=O)N.N1(C(CNC(C)=O)=O)CC(C)CCC1C c1(C(=O)NCCCNC(C2CC(C)CC(C)C2)=O)cnc2c(c1)nnn2C CC1Cc2cc(NC(c3nn(-c4ccccc4)ccc3=O)=O)ccc2O1 C1(SC)CCC(NCc2cccc(C)n2)CC1 C1(NC(c2c(C)nn[nH]2)=O)CCCN(C(=O)C(C2CCCCCCC2)O)C1C c1(C(N(C)CC2CCCN2C(=O)Cc2cnccn2)=O)ccc(O)nn1 N1(C(C2CC3(OC)CC2C3)=O)CCCC1(C)CNC(C1CCC(=O)C1)=O C(=O)(CC(C(F)(F)F)NC(C1CCC=CCC1)=O)NC(C(=O)NC)C c1(C(=O)NCC2N(C(C3CN(CC)C(=O)N3)=O)CC2)ccc2ncsc2c1 C(C1CCN(C(C2CCCC(C#N)C2)=O)CC1)=CC(=O)NC(CC)(C)CO N1(C(CCn2c(C)cc(C)n2)=O)CC(F)(F)CC1.C1(C=O)CC1C(C)(F)F.C Cc1cc(C(=O)NC(CO)C(C)NC(=O)CC2CCCC2)nc2ccccc12 CCN=c1ccc(C(=O)NC(C)CNC(c2ccnn2C2CCOCC2)=O)c[nH]1 C1(C(N2C(C(=O)NC)CC(O)C2)=O)CCN(C(=O)C(C)CCN(C)C)C(C)C1 C=CC1COCC1NC(C1CCCC1CNC(c1nc(C)sc1C)=O)=O N1(C(C(CCC)NC(N)=O)=O)CCCC(C2CN(C(c3sc(F)cc3Cl)=O)C2)C1 CCC(C)(C)CC.C1(C(=O)N)CN(C(c2cc(C(C)=O)c[nH]2)=O)CC1C(C)C Cc1nscc1NC(=O)C(c1ccccc1)NC(C1(C)CC1(F)F)=O N1(C(C2CNC(=O)N2)=O)CCc2[nH]nc(CNC(C3CC3C(F)F)=O)c2C1 C(=O)(C(C)(C)CN(C)C)NC(C(C)NC(CCCOC)=O)C C(=O)(CN=S(C)(C)=O)N(CCCCCNC(c1cnn(C2CCCCC2)c1)=O)C N1(C(C2CN(C)C2)=O)CCCC(CC(=O)NC2CC2F)CC1 C1(CNC(C(CCC)C)=O)CN(C(C2CCCCCC2)=O)CCCO1 C1(NC(CC2(N(C(C(C)SC(C)C)=O)C)CC2)=O)CC(O)(CO)C1 CC(C)C(C)(C(N)=O)NC(C1CN(C(=O)C(C)N=[N+]=[N-])CC1F)=O N1(C(C=Cc2n(C)ncc2)=O)CCC2(CCCN(C(C3CNC(=O)N3)=O)C2)C1 Cc1cc(Cl)c2c(c1)CCN(C(C(=O)NCc1ccco1)c1cc[nH]n1)C2 N1(C(Cn2nnc(C)n2)=O)CC(NC(c2cnc3ccoc3c2)=O)C2(CCC2)C1 C1CCN(C(=O)CC(C)(C)C)CCC1(F)F.C=C1CC(C(=O)NC)C1.C(N)=O c1(C(N(C(CN(C(c2c(OC)noc2C)=O)C)C)C)=O)cc(C)nc(O)n1 C=CC(F)(F)C(=O)N1CC(O)(C(F)C(=O)NCc2csc(C)c2)C1 N1(C(CC(CNC(=O)OC(C)(C)C)OCC)=O)CCC2(CC1)OCCC2O CC1CC2CN(C(=O)C(C)(C)CF)CC2N1C(C1CCN(C)S1(=O)=O)=O CCC(CCC(=O)NCCOCCCNC(C1CC(O)CN1C)=O)OC c1(-c2nc(COC(C)C)nn2C2(C)CCS(=O)(=O)C2)ccc2c(c1)CCCO2 C1(OC)(CNC(C2CCCC(O)C2)=O)CCN(C(=O)CO)C1.c1ccccc1 CC(N=[N+]=[N-])C(=O)N1CCCCC1c1noc(C(C)(C)C)n1 N1(C(Cn2c(C)cc(C)n2)=O)CC(CNC(=O)Cc2ccsn2)C2(CCC2)C1 Cc1ccc(C(=O)NCC2CCN(C(C3(C)CCCCO3)=O)C2)cc1C C1(NC(C(C)C)=O)CN(C(c2csc(=N)[nH]2)=O)C2CCCC12 N1(C(C2(C#N)CC(C)C2)=O)CCCC(C2CC2NC(c2nn(C)c(Cl)c2Cl)=O)C1 CC1CC(C#N)(C(=O)NC2CN(C(=O)C(C)C=Cc3ccccc3)C2)C1 C1(C(=O)NCC2(NC(C=CCCC(C)C)=O)CCOC2)C(C#N)C1(C)C C1(C(=O)NC(CNC(c2n(C)[nH]c(=N)c2)=O)C(C)(C)C)CCc2c[nH]nc2C1 C(=O)(CCC(C)(C)OC)NC(CSC)(C)C(=O)N1CCC(OC(C)=O)C1 C(=O)(C(=O)NNc1ccc(Cl)c(Br)c1)c1c[nH]c2ccc(C)cc21 CC(C(CO)NC(=O)Cn1nccc1-c1ccccc1)NC(C1(F)CC1)=O N1(C(C(c2ccccc2)C)=O)CCC(N2CCCCC2CO)C(C)CC1 c1(C(=O)NC2C(CNC(CCCOCC)=O)CCCC2)c(F)ccc(Cl)c1N Nc1c(F)c(F)cc(C(N2CCC2CNC(c2cn3ccccc3n2)=O)=O)c1Cl CC1=C(C(=O)NCC2(C)CCCC2)CCCO1.C1(CCC=O)CC(F)(F)C1.N C1C2CC3CN(C(=O)C=Cc4cncs4)C1C3C2.O=C1CC(CC(=O)N)C(=O)N1 CC1C(NC(c2cn(C(C)(C)C)nn2)=O)CCCN1C(C1CC12CC2)=O Cc1[nH]nc2c1CCC(C(=O)NC1CC(NC(c3cnn4ccccc34)=O)C1)C2 C=CC(O)C(=O)NCCN(C(=O)C(Cc1cccnc1)C1CCCC1)CCC N1(C(CN(C(=O)CC2CCCC23CC3)CC)=O)CC(OC)CC(C)(C)C1 c1(C(=O)NC2C(NC(C=C(COC)C)=O)CCC2)ccc2c(c1)CCC=C2 c1(CCCOC)nc(-c2coc(C(C)C)n2)n(-c2ccnc(Br)c2)n1 C(=O)(CCC(C)OC)N(C1CCN(C(C2(OCC)CCCCC2)=O)C1)CCC Cc1c(Br)ccc(C(=O)NC2CCCCC2NC(=O)C(C)(C)C2CC2)c1F C1(C(=O)NCCCNC(C2(F)CCCOC2)=O)CC2CCC(C1)C2(F)F c1(C(=O)NCCCNC(CC(=O)NC(C)(C)C)=O)cc(N)cnc1Cl c1(C(=O)NC2CCN(C(c3cc(OC)cc(Cl)c3)=O)C2)cnc2ncc(Cl)cn12 C1(CNC(c2ccc(=N)[nH]c2)=O)CC2CN(C(C3CC3c3cn[nH]c3)=O)CC12 c1(C(=O)NCCC(=O)NC2COCC2NC(c2cnsn2)=O)ccc(Cl)cc1 O=NN1CCCCC1C(=O)NCc1ccc(CCNC(C2CC2F)=O)cc1 C1(CN(C(=O)C(c2cccc(Cl)c2)O)C)CCCN(C(C2OCCCO2)=O)C1 CC(CNC(=O)C(c1ccco1)NC(C1CCN1C)=O)CC(F)(F)F CC(C)C(O)CC(=O)NC(c1cccnc1)C(=O)NC(CC1CC1)C1CC1 c1(C(=O)NC2CN(C(c3ccc(C(C)=O)[nH]3)=O)C2)n[nH]c2cc(C)ccc12 CC1(C)CCCC(C(=O)NCC2(C)CCN(C(=O)Cc3ccc(O)cc3)C2)CC1 C(=O)(C1CCCc2scnc21)N1CCCC(N(c2nc(C)c([N+](=O)[O-])cc2)C)C1 CN1CCOC(C(=O)NCCC2(NC(c3ccc(C4CCCC4)o3)=O)CCC2)C1 N1(C(Cc2ccc(C)o2)=O)CCCC(CC(=O)N(CC(C)C(C)(C)C)C)C1 C12(NC(CNC(=O)OC)=O)CCCC1CN(C(=O)C(C1(O)CCCC1)F)C2 C(=O)(CC(C)C(=O)NCC(O)CC(=O)N1CCC(c2nn[nH]n2)C1)OC Cc1[nH]nc(C(=O)NCCCCN(C(=O)CN(CC(=O)N)C)C)c1O.C1CC1 c1(NC(CC=C)CC)cc(Br)ccc1S(=O)(=O)NCCN1CC=CC1 N1(C(CCn2c(C)cc(C)n2)=O)CC(C)N(C(c2cc(Cl)c(Cl)n2C)=O)CC1C C(C)(CCC(=O)NCC1C(Cn2cc(C(CC)OC)nn2)C1(F)F)OCC C1(C(=O)NCc2cnc(C)[nH]2)C(C)CCN1C(C1CCOC1(C)C)=O c1(C(N2C3CCC2CC3)=O)cc(Cl)cc([N+](=O)[O-])c1.c1(CC)cc(C(=O)N)no1 C(=O)(C1CCCc2n[nH]cc21)NCC(C)N(C(=O)C=CC(=O)NC1CC1)C N1(C(=O)OC(C)(C)C)CC2CC1CN(N1CCC(C3CCOCC3)C1)C2 C(=O)(CC(C)P(C)(C)=O)N(CC(C)N(C(=O)CN(C1CCCC1)C)C)C N1(C(c2cc(CCCC)oc2C)=O)CCC2(CCN(C(=O)CC(C)N(C)C)C2)C1 N1(C(=O)NC2CCN(CC)C2)CCC(C2CCN(C)C2)C1 c1(C=O)ccc(Br)c([N+](=O)[O-])c1.C1(C(=O)NCCNC(=O)N)CCCC1 CC1(C)CC(CC(N2CCCC2c2ncc(C(=O)NC3CC3)s2)=O)CO1 N#Cc1cccc(C(=O)NCC(CC2CCCC2)C(=O)O)c1Br N1(C(C(CCCCC)O)=O)CC2CCCC(CNC(c3ccc(C#N)s3)=O)(C2)C1 CC1CN(C(C2CCCC2F)=O)CC1NC(=O)CN1CSCC1=O C(C(F)(F)C(F)F)NC(=O)CCOCCNC(C1(C2CC2)CC1)=O C(C)(C)(CCC(=O)NCC1COCCN1C(C1CC1C#N)=O)OC C1(NC(c2c(C)n(C)nc2)=O)CCCN(C(C2(CO)CCCC2)=O)CCC1 c1(C(C(=O)NC2CC(F)(F)C2)N(C)Cc2n(CC)ccn2)nc(C)c(C)s1 CCC(F)(F)C(=O)NCCC1(O)CN(C(c2cc(-c3cccc(C)c3)no2)=O)C1 c1(C(N2C3C(NC(C4CC4CF)=O)(CCC3)CC2)=O)cc(F)c2ncccc2c1 C12(C(N(C3CCCN(C(C(C)c4ccco4)=O)C3)C)=O)C3C4C1C1C2C3C41C c1(CC)cc(N)ccc1C(=O)NCC1CCC1.N1(CC=O)CC2CC2C1.N c1(C(N2C(CNC(CCCCOC)=O)C(C)CC2)=O)nc(O)[nH]c(=O)n1 C1(CNC(C2(CC)COC2)=O)CN(C(C2CCn3ncnc3C2)=O)CCC1(C)C C1(CNC(C(C)c2ccsc2)=O)CCC(NC(=O)C(F)(F)c2nccn2C)C1 C1(N=[N+]=[N-])(C(N(C2(C#C)CC2)C)=O)CCN(C(=O)Cc2cc(C)cs2)C1 Cc1cc(C)cc(S(=O)(=O)N2CC3(CCN(C(=O)CCC4CCOC4)CC3)C2)c1 c1(OC)ccnc(CNC(C2(F)CCN(C(C3CC=CCO3)=O)C2)=O)c1 C(=O)(C1CCc2cccc(=O)n21)NC1CCCCN(C(C2(C#N)CC2)=O)C1 C1(NC(C=CC(CC)=CC)=O)(C)CCCN(C(c2nc(O)c(C)s2)=O)C1 C1(C(N2C(CN=[N+]=[N-])CCC2)=O)N(C(=O)C(N)=O)CC12CCCC2 C12(C(N3CCC(C)C3)=O)CCC(CC1=O)C2.C1(CC(=O)N)(NC(C)=O)CC1 Cc1cc(CNC(C2(C)CC(O)CN2C(c2ccsc2C)=O)=O)cnc1Cl c1(OC)c(C(=O)NC2CN(C(=O)CN3C(=O)CCCC3=O)CC2C)c(C)nn1C C1(C)(C(=O)NC(C)Cc2nncn2C)C=CCN1C(c1cc(C(N)=O)c[nH]1)=O N1(C(C2C(CCOC)C2)=O)CC23CCCC2(C1)CN(C(c1cc(C)nn1C)=O)C3 CC12CC(C(N3CCCC3CC)=O)(CCO1)C2.C1(CC(=O)N)CCCS1(=O)=O C(=O)(C1=CC2C=CC(C1)C2)N1CC(CC(C(=O)NC2CCCSC2)F)C1 N1(C(c2ccc(F)cc2)C(=O)NC(CC)C)CCOC2(COC(C)(C)C2)C1 Cc1cnc(C(N2CCC2C(=O)NCC2CC3(CCC3)C2)=O)cn1 c1(C(=O)NCC(C)Cc2ccc(C(C)(C)C)cc2)c(O)nnc2c1CCC2 C1(C(N2CC(O)(CN(C)C(C3(C(F)(F)F)CC3)=O)C2)=O)C2CCN1CC2 N1(C(=O)CC2CC3CC3C2)CC2CC1CN2C(C1(c2ccncc2)CC1)=O C(=O)(C(COC)C(F)(F)F)NC(CC)(C)CNC(c1ccncc1NC)=O C1(OCC)CN(C(C2(CC)CC(F)(F)C2)=O)CC1.n1(CC=O)cnnn1.C C1CC2CCC(C1)N2C(=O)C=Cc1cc[nH]c1.CC(C)(C(=O)N)c1cccs1.C N1(C(c2c(OC)ccnc2F)=O)CCC2(CC1)CCN(C(C1CCC(F)C1)=O)C2 c1(CC(=O)N(CC)C)cccc(O)c1.C1(C)(COC)CC1C=O.CC.N C=Cc1cc(C(=O)N)cc(F)c1.C1(C(N2C(CC)CCC2)=O)CCS(=O)(=O)N1C C1(CC(=O)N(C)C)CC(O)CN1C(c1cc(F)n(C)n1)=O.C1CCCC1(C)C CCS(=O)CCC(=O)N1CC2CC1CC2NC(=O)Cc1ccncc1 CC1CC(C(=O)NC2CCC(F)(CNC(=O)C=Cc3cccs3)C2)CN1C C=C(Br)CC(C)(C)C(=O)NCCCNC(c1ccc(C(=O)N(C)C)cc1)=O C1(N(C(C(CC2CC2)OC)=O)C)CCCN(C(c2cncc(F)c2)=O)CC1 N1(C(C(CCOC)C)=O)CC(NC(c2nc(OC)ccc2F)=O)C2(CCC2)C1 c1(C(=O)NCC#CC)cn2c(n1)CCN(CC(=O)N(C)Cc1ccccc1)CC2 c1(C(N2CC=CC(C(=O)NC(C#C)C(C)OC)C2)=O)cnccc1C#N Cc1cc(Br)c(C(=O)NCC2=NOC3COCC23)cc1N c1(CC)cncc(C(N2CCC2CNC(=O)CSc2ccccc2)=O)c1.O C(=O)(C1Cc2ccc(F)cc21)NC1C(CNC(CCCC(C)=O)=O)C1 CC(C)CCCC(=O)N1CSCC1C(=O)NC1(C)CCSC1 C(=O)(C1=CC(O)CCC1)NCCCC(C)NC(c1ccnc(C(C)(C)C)c1)=O c1(N2CCC(NC(C=CC(C)C)=O)CC2C)cc(C(C)C)nc2ncnn12 c1(OC)cccc(CNC(c2nnnn2C2CCOC2)C2(C)CC2)c1OC N1(C(C2C(C)(C)C2)=O)CC(NC(c2ccc(CO)c(Cl)c2)=O)CC2(CCC2)C1 c1(CC(=O)NCC23CC2CN(C(c2ncccc2O)=O)C3)nc2c([nH]1)CCCC2 C(c1ccc(=N)[nH]c1)=CC(N1CCC(C)C1CNC(C1(C)CC=CC1)=O)=O O(NC(=O)CN=c1cc(NCCCCN2CCCCC2C)nc(C(C)C)[nH]1)CC C1CC(C)(C)CN1C(=O)CN(C1CCSC1)C.C=C(F)C1(CC(=O)N)CCC1 c1(NC(C2CN(C(=O)OCC)CC2CC)=O)cc(C)cc(OC)c1N C1(C(=O)NC2C(C)CN(C(c3ccc4c(c3)CC4)=O)CC2)CCCC(F)(F)CC1 c1(C(=O)NC(CCN(C(CCC=CC)=O)C)C)cc(C)n(C)n1 C(=O)(C1=C(C)CCC1)NCC(CNC(c1cn(CCOCC)nc1)=O)O c1(C(C)C(=O)NC2CC(NC(C3CC=CC3)=O)C2)ccc(C(F)F)cc1 C(=O)(CS(=O)(=O)CC)NC(C1CCN(C(CC(CC)C)=O)C1)C N1(C(C2CC2)=O)CC(C2CC2)C1.c1(C=O)csc(-c2ccco2)n1.NC(=O)N C1(CNC(C=CC=CC)=O)C(C)CCN1C(=O)C1=NOCC1 c1(CC)cccc(C(N2CCOCC2CN(C(=O)C(C(C)C)OC)C)=O)c1N Cc1cc(F)c(N)cc1C(N1CCCC(O)(CCNC(c2cc(Cl)no2)=O)C1)=O c1(C=O)cc2cc[nH]c2cn1.CC1OC2CCC1(C(=O)NCCC1(C)CC1)C2.N N1(C(c2c(CCC)n(C)nn2)=O)CCN(C(=O)C(C)(F)F)C(C(C)C)C1 CC1(C)CCCNC1C(=O)Nc1ccc(OC(F)F)c(OC(F)F)c1 C12(C(=O)NC(CNC(CCCC)=O)CC(F)(F)F)CCOC1CC(=O)NC2 C=CCCCCCC(=O)NCc1ncoc1CCNC(C1NC(=O)OC1C)=O Nc1cc(C(N2CCCOC(CNC(=O)C)C2)=O)cc(Cl)n1.C(=O)C1CC1.N C(C(=O)C(C)(C)C)c1nc(NCc2n(C(C)C)ncc2)sc1 Cc1cc(Cl)c(C(=O)NCC2CC3CC3N2C(C2CC2C)=O)c(Cl)c1 c1(C(=O)Nc2c(C#N)c(O)cs2)nc2ccc(-c3ccco3)cc2s1 c1(CCC(=O)N)ccccc1O.c1(OCC)nc(C(=O)NC(C)C(C)C)co1 C1(O)(CNC(=O)CN2CC=CC2)CN(C(=O)CCOc2cccnc2)C1 c1(C(=O)NC(CNC(CCCC#C)=O)CC(F)(F)F)c(F)ccc(F)c1N c1(N(C2CC3CNC2C3)C(c2c(C)noc2)=O)ccc2ccoc2c1 c1(NC(CCNC(CCC)C)=O)nc2ccccc2s1 N1(C(C(C)(C2CCC2)NC(c2n(CC)ccc2)=O)=O)CCCC(C)(F)C1 N1(C(C2CC(O)(CC#C)C2)=O)CCCCC(CNC(c2ccc(N)cc2O)=O)C1 CC(C(=O)N1CC(NC(c2cccnc2)=O)CC1(C)C)S(C)(=O)=O.N(C)(C)C C(=O)(C1CCCc2nn(C)cc21)N1CCCC(C2(NC(CCCC#C)=O)CC2)C1 CCC(C)(C)C(C)CC(=O)NCC1CC(O)CN1C(=O)C1=CCCOCC1 c1ccc2c(c1)C1CC2N(c2nnc(C3CCCCO3)n2CCC2CC2)C1.C1CC1 c1(CNC(COCCNC(C(C)OCCC(C)C)=O)=O)ncccn1 N1(C(c2c(CC)ocn2)=O)CCC(O)CC1C(=O)NCc1cccnc1C C(=O)(C(F)CCC(C)C)N(C(C(=O)NCc1cc(C)ncn1)C)C1CC1 CCC(O)CC(=O)N(CCCCCCNC(C1CCN1S(C)(=O)=O)=O)C c1(C(N(CCCC)C)=O)cc(S(N)(=O)=O)cs1.C(c1sccc1C)=CC=O N1(Cc2c(NC(C(N3C(C)CNCC3)=O)=O)cccc2)CCS(=O)(=O)CC1 C(=O)(CC(C)C(C)(C)NC(c1ccc(F)c(C)c1)=O)NC(c1ccc(C)cc1)C CCCC(C)(CCC)C(=O)NCC1CCCCC1NC(c1cncc(O)c1)=O O(NC(=O)C(C)(C)C1CCN(C(c2ccc([N+](=O)[O-])[nH]2)=O)C1)CC(C)O c1(OC)cccc(COCCN(C2CCN(C(=O)Nc3ccns3)C2)C)c1 C(=O)(CCS(=O)(=O)C(F)(F)F)N1CCCCC(NC(C(C(C)(C)O)F)=O)C1 c1ncc(C)c(C)n1.c1(SC)ccc(CC(=O)Nc2cc(C)sc2C(=O)N)cc1 C(=O)C(C)CC(F)F.C1(OC)CC(C)N(C(c2ccc(C(F)(F)F)o2)=O)C1.N N1(C(=O)CC2CCCCO2)CCc2ccc(-c3nn[nH]n3)cc21 O=C(N1CC(O)CCO1)C1CN(C(=O)CN2CC=CC2)CCO1 N1(C(C2(C)COC2)=O)CC(O)(C(F)C(=O)NCCC#CCO)C1 N1(C(CCC=C)=O)CC(NC(c2ccc(=O)n(CCCC)n2)=O)C2CCCC2C1 C(CC(=O)N(C1CC1C1CC1)C)(C1CC1)NC(C(C)NC(=O)NC)=O C12(CNC(C(CNC(c3c[nH]c(=N)o3)=O)N(C)C)=O)CCC(CO1)C2 C1(CNC(C)=O)CCC2(CCC2)C1NC(=O)C=Cc1cccc(Cl)c1Cl N1(C(CC(=O)NC)=O)Cc2nccn2CC(NC(C2(C)CNC(=O)C2)=O)C1 C=CCC(CNC(=O)CC1CCOC1)C(=O)NCc1[nH]nnc1CC c1(OCC(=O)OC)ccc(C(=O)NC)cc1.C1CCOCC1.C(=O)C(C)O c1(C(N2CCCC2)=O)ccc([N+](=O)[O-])c(Cl)c1.C1(CNC)CC1C(F)(F)F Cc1cccc(C(=O)NC2CC2CNC(=O)C(c2ccccc2)O)c1O c1(CC)n[nH]c(=NCC(C2CC2)N(C)C(c2cnnc(Cl)c2)=O)s1 CCC(C)C(C(=O)NCC1CCCC1CF)N(C)C(c1cncnc1)=O C1(CCCC)CCCN(C(=O)C(CC)NC(=O)C(c2ccc(F)cc2)(F)F)C1 C(CC(C)(C)CO)NC(C(C1(C)CC1)NC(C(C)C1CCCC1)=O)=O C12(NC(C(C(C)C)NS(N)(=O)=O)=O)CCC(CC1)OC2.c1(C=O)cnns1.C N1(C(c2c(C)ccs2)=O)CCCC(C2CCCN2C(c2ccc(F)cc2)=O)C1 c1(CC(=O)NC2C(NC(c3cn(CCOC)nc3)=O)CCC2)cnccc1C N1(C(C(C)N(C(C2(C)CC2(C)C)=O)C2CC2)=O)CC2C3CCC(O3)C2C1 Cc1cc(C(=O)NCC2CC2)c(C)n1-c1ccon1.c1(C=O)sccc1Cl.C Cc1ccc(N(C2COC2)C(c2cn(CCN(C)C)nc2C)=O)cc1 Cc1ccc(CC(=O)NC(C)CN(C)C(C2CC2c2ccccn2)=O)o1 N1(C(CCC2CC(OC)C2)=O)CCC(C2CC2NC(=O)CCC(C)(C)C)CC1 Cc1c(NC(c2cccc(C#N)n2)c2nnnn2C(C)C)cccc1CO C(CC(CO)NC(=O)CCn1cc(C(C2CCCN2CC(F)(F)F)=O)nn1)SC Cc1ccc(OCCC(=O)NCC(C2CC2)NC(=O)C(O)CF)cc1C C(=O)(C1CCCc2ccccc21)NCC12CC(NC(C3(C)COC3)=O)(C1)C2 C1(NC(=O)CCF)CCC2(CCCN(C(c3scnc3C3CC3)=O)C2)C1 C(O)(CN=C1NCC(C(F)(F)F)CN1)c1c(OC)cccc1F C1(NC(c2c(CNC(C(CC)n3ccnc3)=O)c[nH]n2)=O)CC2CCC1C2 N1(C(CCC(=O)OC)=O)CC2CCC1CN2C(=O)C(=Cc1ccc(C)cc1)C C(=O)(N=c1cc2n([nH]1)CCO2)c1c(SCC)cc(C(F)(F)F)cc1 c1(C(N(CCC(C)NC(=O)Cc2csnn2)C)=O)ncn2c1CCC2 c1(OC)oc(C)nc1C(=O)NC.C1CCOCC1.c1(C=O)ccc(C2CC2)o1 C1(C(C)(C)NC(C2CCCS2)=O)CCCN1C(=O)CC1OCCO1 C(=O)(C1CCCn2ccnc21)NC(C1CN(c2snc(C)c2C#N)C1)C c1(C2(CN(CC(C3CCOC3)OCC)C)CC2)cccc(Cl)c1 C(=O)(CC(C)CC(F)(F)F)N1CCCC(CCC)(NC(=O)CCc2cnc[nH]2)C1 CN1CCN(CC(C)(C)C(=O)NCC2(F)CCCC2)CC1.c1(C(=O)N)ccon1 C1(C(NOC)=O)CCC(O)CN1C(c1cnc(O)c(F)c1)=O c1(C(=O)NC2(c3cn(Cc4cnc(C)nc4)nn3)CCC2)cc(C)c(N)cc1F c1(N2C3C(NC(=O)C=CC=C(Cl)Cl)(CCC3)CC2)ccc([N+](=O)[O-])cc1C(F)F N(C(=NCCN(CC(F)(F)F)C)NCC1COCCN1C)C(CC)C C=C1CC(C(=O)N(CCCN=[N+]=[N-])C)(CNC(C23CSCC2C3)=O)C1 c1(C(=O)OC)cn(Cc2cn(CC(C)(C)C)nn2)cn1.C(=O)(C(F)(F)F)N Cc1ccnc(CCNC(=O)CCN(C(=O)CCc2cnc(C)o2)C(C)C)n1 N1(C(C2N(C(c3c(OC)cccc3)=O)CCCCC2)=O)CC2CC3CC2C1C3 c1(C(=O)NCC2C(NC(=O)CC3C=CCC3)COC2)ncn2ccccc12 c1(CC)c(C(=O)N(C2CN(C(C3C4CCCOC34)=O)CC2O)C)nnn1C C1(C)(CN(C(C(COCC)C)=O)C)CCCC1NC(c1cscc1S)=O c1(OC)nc(C)cc(=NCCCN(C(=O)CN2C(=O)NC(C)(C)C2=O)C)[nH]1 CC(=O)C(C)CC(C)C(=O)N1CCCC2(NC(c3ccnc(S)c3)=O)CCCC12 N1(C(C(=Cc2cn[nH]c2)C)=O)CCC(C(N2CC(CN=[N+]=[N-])C2)=O)C(O)C1 N1(C(CCc2n(C)cnn2)=O)C2CCC1CC(NC(C1CCCOC1)=O)C2 C1(C)(C=O)CCNC(=O)C1.C1(C)(C(N(C)CCOCCC)=O)CCCCC1.N N1(C(CN(C(C)C)C(C2CC2(C)C(F)F)=O)=O)CCC(O)CC12CC2 c1(N(CC(=O)NC)C)nc(NC2CCC3CCC23)nc2ccc(Cl)cc12 c1(CNC(C(CC#C)O)=O)ccc2c(c1)CCN(C(=O)C1=CCOC1)C2 C=C(Cl)CC(C(=O)NCC=C(Cl)Cl)NC(=O)C=CC1CCCN1C C(CC(C)(C)CC(=O)NC1CCCC1NC(c1ncncc1Br)=O)OC C1(O)(CC(=O)NCCCC)CCCN(C)C1.c1(C(=O)N)cc(C(C)C)ccc1O N1(C(C(CCC#C)NC(c2csnc2OC)=O)=O)CC2CCCCC2C1C CC1(CNC(C2CC2)=O)CN(C(=O)CS(=O)(=O)Cc2cccs2)CCO1.C C1(C(=O)NCC2=CCCCC2)(CC)CCCN1C(c1cc(O)nn1C)=O C1(NC(C(C)=C2CCCC2)=O)C=CC(C(=O)NC(c2cc(C)on2)C)C1 c1(CCNCC(C)CN2CCOCC2)cnn(C)c1C(F)(F)F CCC(CC(=O)NC(c1cn(C)nn1)C(=O)N(CC(C)(CO)CO)C)SC Cc1c(C(=O)NC2C=CCN(C(c3cc(CF)on3)=O)C2)[nH]c2c(C)cccc12 C1(N(C(C=COCC)=O)CCOC)CCN(C(=O)CC(C)C=C)CC1 c1(N2CC(C)=C(C)CC2)ncc(S(=O)(=O)NC(C2CCCCO2)C)cc1Cl c1(OC)ccc(CNC(=O)C(c2c(I)ncn2C)N(C2COCC2(C)C)C)cc1 CC1=C(F)CN(C(c2sccc2CNC(=O)C(C)S(C)(=O)=O)=O)CC1 N1(C(=O)CN2CCCC2)CC2C3CCC(C2C1)N(CCC1CC1)C3 C1(C(=O)NC)CC2CC1CN(C(=O)CC1CC3(CC3)C1)C2.C1(O)CC=CC1 C(CCC)(CCC)=CC(=O)N(C(C)(CSC1CC1)CO)C1C(=C)C1 C1(NC(c2n(C)nnc2)=O)CN(C(c2cncc(-n3cccn3)n2)=O)C(C)(C)C1 c1(C(N2CCC(NC(C(CCC)(C)C)=O)C(F)C2)=O)cccc2ncnn12 c1(C(N(C2CCCN(C(C3CC4(C3)CC4(F)F)=O)CC2)C)=O)c(F)ccnc1F N1(c2ccnc(C)n2)CC2CCC1C(NC(c1cc(C)n(C)c1C)=O)C2 c1(CC(=O)NC2(c3ccccc3)CN(C(=O)Cc3cscn3)C2)ccccc1 c1(C(=O)NC2C(NC(C=C3CCN(C)CC3)=O)C2)ccc2c(c1)COC2(C)C c1(OCC(=O)NCC#CCNC(C2(CF)CCC2)=O)ccc(Br)cn1 C1(C(=O)NCC(C)CNC(C2(CCN(C)C)CC2)=O)CC1C1CC1 N1(C(C2(C#C)CCOCC2)=O)CC2CCN(C(=O)CCCCSC)C(C2)C1 c1(C(=O)NCC2CN(C(COC)=O)C(C)C2)sc2[nH]c(C)nc(=O)c2c1C C12(C(N(CC)Cc3ccccn3)=O)COCC1CN(C1CCNC(=O)CC1)C2 C1(c2nnnn2C2COC2)(NCC(c2ccccn2)C)CCCSCC1 C(=O)(CS(=O)C(F)(F)F)N(C)CCOCC.C1(CC=O)CCCC12CC2.N C(=O)(CCCCCN(C)C)N(C(C)C(=O)NCCC1CCCC12CC2)C1CC1 Cn1cc(C(=O)NC2CCC(NC(c3ccc(-n4cccc4)nc3)=O)C2)c(Cl)n1 C(=O)(C(C(C)C)c1ccncc1)O.C(=O)(C(Cn1ccnc1)NC(=O)C)OC C(=O)(CC1CC(=O)Nc2ccccc21)N1C2CCC(NC(CN(C)C)=O)(C2)C1 C1(C(C)C)CCOC1C(=O)NC1(CC(N2CCC2(C)C)=O)CC1 CC(CC(C)(c1nnnn1C)NCCOC(c1ccccc1)C)C(F)F CCCC(CCCNC(=O)C=C(Cl)Cl)NC(c1n[nH]cc1-c1ccncc1)=O C(=O)(C(CC(F)F)N(C(=O)COc1ccccc1)C)N(C)Cc1ncco1 C(=O)(C1CCCc2nc(C)[nH]c21)NC(CSc1ccc(C)cc1)C c1(OC)ccncc1NC(c1c(CNC(C2(C)C=CCC2)=O)cnn1C)=O N1(C(C2CC=C(C)CC2)=O)CC2CCN(C(c3cnsc3C)=O)CC2C1 C(=O)(C(C)(C)CC(=O)N1CCC2(CNC(C3CC3(Cl)Cl)=O)CCCC12)OC c1(C(=O)NC(Cn2cc(C(CC(C)C)(C)O)nn2)C)nn(C)cc1S(C)(=O)=O c1(CCc2nc(COCC)nn2-c2ncnn2C)cc(Cl)cc(Cl)c1 C(=O)(C1=CCN(C(=O)CCNC(=O)CC(C)C)C1)NC(CC)Cn1cncn1 O(NC(=O)C(C)(CO)NC(C1CCC(=O)N(C)C1)=O)CC(=O)OCC c1cc(C)ccc1I.N1(C(C(CC)NC(C)=O)=O)CCCC1(C(=O)O)COC Cc1nc(CC(N2CC(F)(CNC(C3CCC(O)C3)=O)C2)=O)n[nH]1 c1(C2C(CN3CC(O)(C(C)(C)C)C3)C2)ccc(Cl)cc1.C1(F)(C=O)CCOC1 N1(C(C(CC)SC)=O)CC(NC(c2ccc(OC(F)(F)F)cc2)=O)C2(CC2)C1 c1(NC(N2CCC(C)C2C(=O)O)=O)cc(C(C)(C)C)cc(C(C)(C)C)c1 C1(CC)CC(F)(F)CN1C(c1ccc(C(F)F)o1)=O.c1(CC)ncc(C=O)s1 c1(CNC(c2nnnn2C2(C)CC2)CCOC)ccc(C)c(Br)c1C C(=O)(CC(C)(C)C(F)F)NCCCN(C(C(C)=CC1CC1)=O)CCO c1(SCC(=O)NCCC2CCN(C(c3c(C)ccs3)=O)C2)cccc(F)c1 c1(C(N(CC(C)NC(C2CCC(C)(CC)O2)=O)C)=O)cc(F)cc2ccoc12 Cc1ccc(CC(=O)N(CCC(N2CCCC(F)C2)=O)CC2CC2)cc1 N1(C(c2cc(C)[nH]n2)=O)CC2CCOCC2(NC(=O)C=C2CCN(C)C2)C1 C(C(C(=O)N=c1cc2ccccn2[nH]1)NC(=O)CCC(=O)N(C)C)SCC C(=O)(CCCC(=O)NC1(c2ccccc2)CN(C(c2ccc(C)[nH]2)=O)C1)NC C1(C(=O)NC2(CC=C)CCN(C(c3cnns3)=O)C2)CCCCC1(F)F C1(CNC(c2c(NC)cccc2)=O)CC(C(=O)N2CCC(CCO)CC2)=NO1 N1(C(c2cc3scc(C)c3[nH]2)=O)CCC2(CCCN2C(=O)C(N)=O)C1 c1(C(C)(C)C)ccnc(C(N2CCC(C)(NC(=O)CN3CCCNC3=O)C2)=O)c1 C=CC(C)C(C)C(=O)N(C1CCN(C(=O)CCC2CC2)CC1)CCOC CC1(CNC(c2csc(Cc3ccccc3)c2)=O)CCCO1 c1(OC)cc(CNC(c2nc(O)n[nH]2)C)c([N+](=O)[O-])cc1OCC(F)F c1(C(=O)NCC2(F)CCN(C(C(CC(C)(C)C)O)=O)C2)nccc2ccccc12 CCC1=NOC(CC(=O)NCCOC2CN(C(=O)C=CSc3nc[nH]n3)C2)C1 c1(C(N(CC(CNC(c2cc(C)sn2)=O)(C)C)C)=O)ccc(O)c(C)c1 c1(C(N(CCCNC(c2ccnn2C)=O)C)=O)ccc2c(c1)COCO2 N1(C(C2CN(C(C(CC)COC)=O)C(C)(C)C2)=O)CCn2c(cnc2C)C1 C1(C(N2CC(C)C(C)(C)C2)=O)(OC)CCCCCCC1.C(=O)C(C#N)C1CC1.N C1(C(=O)NCC2C(NC(c3c(C(C)C)ocn3)=O)CCC2)CCc2nc[nH]c2C1 C1(CNC(=O)CC2CC=CCC2)CCN(C(=O)C=Cc2cscn2)C12CC2 n1(CC(N)=O)nc(C2OCCc3ccccc32)nc1-c1ncnc2sccc12 C(=O)(CC(C)CNC(=O)C=CC(C)(C)C)NCc1n(CCC)ncn1 CCC(C)CC(C(=O)NOC(C)C(=O)OC)NC(c1cnc(O)cc1C)=O C(=O)(CCCCCCCC1CC1)N1C(CNC(C(C)N(C)C)=O)CC2(CC2)C1 c1(C(N2CCC(O)(CC)CC2)=O)c(C)[nH]c2ccc(O)cc12.C(C(=O)N)OCC CC1C(NC(=O)Cc2cncnc2O)CCCN1C(=O)C(=O)C1CCCC1 O=S(=O)(c1c[nH]c2ncccc12)NC1CCC2CCCC2C1 CC(C)C(C(=O)N1CC(C(N)=O)(CNC(c2cnc(S)n2C)=O)C1)N(C)C CC(CC(=O)NCCOCCCN(C(=O)CC(C)(F)F)C)CC(C)(C)C N1(C(c2ncc[nH]c2=O)=O)CCC2(C1)CN(C(C1CCCS1(=O)=O)=O)CCO2 C(C(=O)N=c1cccn[nH]1)N(C(=O)OC(C)(C)C)C1CC1 C1(n2cccc2)(CC(=O)N(CCNC(C=CC)=O)C)CCOCC1 Cc1cc(CN2CCNC(=O)C2CC(=O)N(C)C)nc2ccccc12 c1(N2CCN(C(c3cccc(SCCC)c3)=O)CC2)ccc2nc[nH]c2c1 c1(C(=O)NC2CC(NC(COc3c(C)cccc3)=O)C(O)C2)ccc(O)c(F)c1 C(=O)(CC(C)CC(C)(C)C)N.C1(C(=O)NC2CCCCC2)(COC)CCCOC1 Cc1cc2nccnc2cc1C(N1CC2C(CNC(C3CCNC3=O)=O)C2C1)=O Cc1ccn(C)c(=O)c1NC(=O)CCC1(C)CN(C(C2CCCC(=O)C2)=O)C1 N1(c2nccc(C(=O)OC)c2)C2CCC1CN(C(=O)C(F)(F)CO)C2 C1(NC(c2cc(C)n(CCN)n2)=O)Cc2ccc(Cl)cc2C1 N1(C(C2(CNC(C(CC)C)=O)CC3(CC3)C2)=O)CCC2(CC1)CSC2 C(CC(C)N=c1[nH]c2c(c(=NCC3CC3(Cl)Cl)[nH]1)CCC2)SC CC1c2cccnc2CCCN1C(c1ccc(Cl)c2occc12)=O c1(C(N)=O)ccc(C(=O)NCC2CN(C(=O)C=CSc3nc[nH]n3)C2)cc1Cl C1(C(=O)OC)CCc2ccccc2N(C(c2cc3c(cc2[N+](=O)[O-])OCO3)=O)C1 N1(C(C2C(C#C)C2)=O)CC(C2CC2)C1.c1(CCC(=O)N)ccccc1.C(C)=O C1(C(N2CCC(C)C2CNC(c2cccnn2)=O)=O)CC(S(C)(=O)=O)C1 CC1CN(C)CCCN1C(C1(C)CN(C(c2ccoc2Cl)=O)C(C)(C)C1)=O CCCCCCC(C)C(=O)N1CC(NC(C2CC2(C)C)=O)CC2(CC2)C1 C1(C(N2CCN(CC(C3CCCOC3C)=O)CC2)C)COc2ccccc2O1 CC1CN(C(=O)C(F)CC2CCOC2)C1C(=O)NC1(CC(N)=O)CC1 N1(C(CCc2scc(C)n2)=O)CC(NC(=O)Cc2conc2C)CC(C)(C)C1 C1(CC)(NC(=O)Cc2ccc(O)c(O)c2)CCCN(C(c2cn(C)cn2)=O)C1 N1(C(=O)CSCC(F)F)CCC(CCCNC(C2CN3CCC2C3)=O)CC1 O=S(=O)(c1ccc(N2CCC(CCO)CC2)cc1Br)N1CCc2cnccc2C1 C1(n2cc(C(C)SC3CC3)nn2)CCN(C(c2nccc(C(F)F)n2)=O)CC1 c1(C(N(CCNC(c2c(C)n(C3CCC3)nc2)=O)C)=O)coc2c1COC2 c1(CNC(C(N2CC(C)(C)CC2)=O)=O)cccc2c1OCCO2.C1(C=O)CC1.N Cc1cn(C(C)C)cc1C(=O)N(C)CC1(O)CCN(C(=O)C(C)C(F)F)C1 N1(C(C2C(OCC)C2C)=O)CC(NC(=O)CC2CCCCC2)C(C)(C)C1 CCCCC(C(=O)NOC(C)C(=O)OC)NC(=O)CC1C(C)(C)C1(C)C C1(NC(C2C(C)(C)CCO2)=O)CCC2(CCN(C(c3cnn4c3OCC4)=O)C2)C1 n1(CCOCC)cc(C(=O)N)cn1.C(=O)(C(C)Cc1ccccc1)N1CCC1 C1(C(=O)NCCN(CCC)C(c2csc(C)c2)=O)CCC2(CCOCC2)C1 c1(C(=O)NC2(CCO)CN(C(c3c(C)ccc(F)c3)=O)C2)cccn2nccc12 C1(C(=O)NCC2CCC2)CN(Cc2sccc2Cl)CCS1 C(=O)(CCC(C)(C)NC(=O)C(C)C1CC1)N1CCC(OC(C)C)CC1 C12(NC(c3cccc(NC(C)=O)n3)=O)CCN(C(C3CC=CC3)=O)CC1C2 CCCCC(C)(F)C(=O)NC1COCC1CNC(c1cnc(OC)c(C)c1)=O N1(C(CC2CCCC(=O)N2)=O)CC(CO)C2(C1)CN(C(C1COC(=O)C1)=O)C2 N1(C(CCCN(C(Cn2nc(C)oc2=O)=O)C)=O)CCC2C(CCN2C)C1 Cc1noc(C(C)C)c1C(=O)NC1CCCCC1NC(c1cnn[nH]1)=O N1(C(c2c(CCCC)ccs2)C(=O)NC2CCOC2)CCc2c[nH]nc2C1 N1(C(CC=C(C)C)=O)CC(NC(c2cc(-c3ccn(C)c3)[nH]n2)=O)CC(C)C1 C=CC(CCC)CC(=O)NCCN(C(=O)C(C)C(C)C)CCOC C(=O)(C(CO)C(C)(C)C)N1CC(C(C)NC(C(CC)CCOC)=O)C1 c1(C(=O)OCC)c(C)[nH]c(C(=O)N)c1C.C1CN(C(c2csnn2)=O)CC1O N1(C(c2ccn(CCCC)n2)=O)CCC(O)(CC)C1.C(c1cn[nH]c1)=CC(=O)N C(=O)(CCCCC(F)F)N1CC2(C(NC(c3cccc(OC)n3)=O)CC2)C1 c1(CCC)ccc(C(=O)NC(C)CNC(C2CCCN2C(=O)CC)=O)s1 C12(C=O)CC(C)(CN1C(C1(C(N)=O)CC1)=O)C2.c1(CCC)ncccn1.N Cn1cc(-c2cc(C(=O)NC(CNC(=O)CC3CC3)C3CC3)n[nH]2)cn1 c1(CNC(c2ccc(CN=[N+]=[N-])o2)=O)ccccc1.C1(C=O)CCC(F)CC1.N C1(C(=O)NC(C2(O)CN(C(C3CCC(=O)N3)=O)C2)C)CC1C1CC1C N1(C(CC#N)=O)CCCC(CCNC(C2CCN(c3ccccc3F)C2)=O)CC1 C=CC(C)(C)CC(=O)N1CCC(C)C(C)C1.c1(C(=O)N)cc(C(C)C)nc(O)c1 C(=O)(CC(C)C(C)C(C)C)N1CCC(N(C(=O)CCc2ncccn2)CC)C1 c1(C(N(CC)CC2CCN(C(=O)CN3CCC3C)CC2)=O)cc2cnccc2o1 Cc1c(C(N2CC(F)(F)CC2CNC(=O)CC)=O)oc2ccccc12.C(N)=O C1(NC(c2n(CCC)nc(C)c2)=O)CN(C(C2(C)COCCO2)=O)CC1C1CC1 c1(C(=O)NC(CN(C(=O)C=Cc2ccoc2)CC)C)nc(C2CC2)cs1 N1(C(c2c(C)nncc2)=O)CCC2(COC(CNC(c3ccncc3)=O)C2)C1 C(=O)(C1CCc2nccn21)NCC1(NC(C(CC=C)C)=O)CCCCCC1 C1(NC(C(=C(C)C2CC2)F)=O)C=CCN(C(C2(c3cccs3)CC2)=O)C1 N1(C(CC(C)(F)F)=O)CCN(C(=O)C=Cc2cccc(F)c2)CC1CO c1(OCC)ncc(C(=O)NC2CC(NC(=O)C(N3CCCCCC3)C)C2)cc1Cl c1(OC)ccc(C=CC(=O)NOc2ccc(C(N)=O)cc2)cc1 C1(NC(C2(OCC)CCOC2)=O)CN(C(c2cncnc2)=O)CC1C(F)F c1(C(=O)NC(CCNC(C2(CC#C)CCCC2)=O)C)nccc(N)n1 C1(C(C)C)CCC(C(=O)N(C)CC2CN(C(=O)CC3CCC3)CCO2)CC1 C1(NC(C2(C#C)CC2)=O)CC1C1CCCN(C(C2CCC(C)=C(C)C2)=O)C1 CC1(C)CN(C(C2CCN(C(c3ccc(Cl)cn3)=O)C2(C)C)=O)CCS1 N1(C(c2ccn(CCCC)n2)=O)CC(C)N(C(=O)C=Cc2cccnc2)CC1C N1(C(c2nnc(-c3ccncc3)o2)=O)CCc2cnccc21 CC(C)C(CNC(C1SCCS1)=O)C(=O)NCC1(C(N)=O)CC1 N1(C(CC2C(C)CCCC2)=O)CC2(CC(NC(c3ncc[nH]3)=O)CO2)C1 N1(C(C(C)OCCC=C)=O)CCCC(NC(C2CC2F)=O)CC1 S(=O)(=O)(c1ccc(C)cc1C)NCC(CC)Oc1cccc(Cl)c1 N1(C(c2c(C)nn[nH]2)=O)CC(S(=O)(=O)N2CCN(Cc3cc(C)n(C)n3)CC2)C1 C1(NC(=O)COC2CCCCC2)COC2C(NC(=O)CO)COC12.C1CCC1 c1(C(N2CCC(NC(C3CN(C(C)C)C3)=O)(CF)C2)=O)cc(Cl)c(Cl)cc1O C1(C(N(CCC)C)=O)COCCN(C(c2ccnn2CC)=O)C1 C1CCCCN(C(=O)CCN(C2CCCCC2)C)C1.CC(C(=O)N)NS(C)(=O)=O CC(CC(=O)N1CC(C2(NC(C3C4CC5C(C4)C35)=O)CC2)C1)C(F)F S(=O)(=O)(c1cccnc1NCC1CC(F)(F)CO1)NCC1CC(C#N)C1 C1(NC(c2cn(C(C)(C)C)nc2)=O)CN(C(c2ccon2)=O)CC(F)(F)C1 N1(C(C2C(C)C2)=O)CC(F)(CNC(c2ccoc2Br)=O)C1 c1(CN2CC3CN(C(=O)CNc4ccccc4)CC32)cc(F)c(F)cc1F C#Cc1ccc(C(N2CC(CNC(=O)C(C)=C3CCCC3)CC(C)C2)=O)cc1F C=CCCCCC(=O)NC1CN(C(=O)COc2ccc(F)cn2)C1 c1(C(C(N2CC(C(=O)NC(c3ccccn3)C)C2)=O)n2cccc2)ccccc1 N1(C(c2onc(CC)n2)=O)CC(C2CCCN(C(c3ccc(C)o3)=O)C2)C1 C1(C(N(CCCNC(c2c(OC)csc2)=O)C(C)C)=O)CCCCC1F O(NC(=O)C(CC1CCC1)NC(=O)CC1CCC1)C(C)CO N1(C(C(CC)NC)=O)CCC12CCCN(C(c1ccncn1)=O)C2 N1(C(CC2CC(=C)C2)=O)CCCC2CCN(C(=O)CCCCCF)CC12 Cc1cc(C(=O)NC2(CO)CN(C(C3CCO3)=O)C2)cc2cccnc12 C(CC(C)C(=O)N1CC(O)(C(F)C(=O)N(C2CC2C)C)C1)=CC N1(C(c2ccc(N3CCC(C)CC3)nc2)=O)CC(NC(=O)CNC=O)CC(O)C1 c1(CC(=O)NC2C(NC(COCC)=O)CCCC2)ccc2oc(O)nc2c1 c1(CNC(c2cncc(NC(C(CC)C)=O)c2)=O)ccc(Cl)nc1OC n1(CC(=O)NCC=C)c(N(CC)Cc2ccco2)nnc1-c1cccnc1 c1(C(=O)NC(CN(CCC)CC)C)cc(O)nc2c1CNCC2 C1CC2CCC1N(C(C1C3CCCCC13)=O)C2.C(=O)(CC(=O)N)OC(C)(C)C.C CC1(C(=O)NCCC2CCCC2)COC(=O)N1.N1(CC(=O)N)CCC(O)CC1 C1(C(=O)N)(N(C)C)CCCCC1.Cn1ccc(-c2cc(C(=O)NCCCO)n[nH]2)c1 C1(CC=C)(NC(=O)C=Cc2cccs2)CCN(C(c2cocc2C)=O)C1 Cc1[nH]nc(C(=O)NCC2C3CN(C(c4cnc[nH]c4=N)=O)CC23)c1C CN1CCC(NC(=O)C(C)C2CCC2)C1(C)C.C1(C(=O)N)CC2(C1)CC21CC1 N1(C(C2C(C=C)C2)=O)CC2(C1)SCCC2NC(c1cnc(CC(C)C)[nH]1)=O C(C)(C(C(C)C)NC(C1CC(Cl)(Cl)C1)=O)NC(c1cnc(C)s1)=O N1(C(CN(C2CC2)CC)=O)CC(C(=O)NCCC(F)CN=[N+]=[N-])C(C2CC2)C1 N1(C(CCC2CCC(NC(C(CC(=O)OC)C)=O)C2)=O)CCC2(CCCO2)C1 N1(C(C2CCC(CNC)O2)=O)CCC(CC(C)NC(c2cnn(C)c2)=O)CC1 c1(C(N(CC(CNC(CCOCC)=O)C)C)=O)cc(OC)ccn1 c1(CC(N2CCC(C)C(NC(=O)CCCN=[N+]=[N-])C2)=O)ccc2ccoc2c1 C(=O)(CC1=Cc2ccccc2C1)N1CC(N(C)C(c2n[nH]cc2Cl)=O)C(F)C1 C1(NC(C(C)N(C)C(C2CN3CCC2C3)=O)=O)CCc2ncnn2C1 C1(C(N2C3C(NC(C4CCC(=O)NC4)=O)C(C3)C2)=O)CC2CCCC(C1)C2=O N1(C(C(CSC)(C)C)=O)CC(C)C(NC(=O)CCC(=O)c2cccnc2)C(C)C1 Cc1sc(C)c(C(=O)NC)c1C#N.C1C(C2CC2)CCN1C(c1cc(Cl)on1)=O c1(OC)ccc(C(C)(C)C(=O)NC(CC)C(C)C)cc1.C1(C)(C=O)CC1C.N C(=O)(C1=CCCSC1)Nc1nccc(CN2C(C)CC(N3CCOCC3)C2)c1 C1(C(=O)NC(C)(C)CNC(C2CCCC3(CC3)C2)=O)OCC2COCCC12 c1(NCCC(CCC)C)nc2ccccc2nc1NC(C)COC c1(NC(C2C(Nc3c(C)cncn3)CCCC2)=O)nc2cc(Cl)ccn2n1 c1(C(=O)N)nc2c(s1)COCC2.C1(CCOC)CCN(C(=O)C=O)C1.C1CC1 C(=O)(CC(C)P(C)(C)=O)NCC1(OC)CN(C(c2c[nH]nc2C)=O)C1 N1(C(C(C=C)CC)=O)CCN(C(=O)C(C#N)CC)CC1C1CCC1 C(=O)(CC1C(=O)Nc2ccc(Cl)cc21)NCCCCCNC(CN(CC)CC)=O N1(C(c2ccc(SC)s2)=O)CCC(C)(C)C(C)C1.c1(CC(=O)N)cnccc1C C(=O)(C(CCCCCC)NC(=O)OC(C)(C)C)N1CC(C=C)(O)C1 N1(C(C2CC(OC)C23CCC3)=O)CCc2cc(F)cc(F)c2C1 c1(OC)ccncc1C(=O)NC1CCC(C(=O)NCCc2ccncc2C)CC1 Cc1cc(CNC2CN(C(=O)Cc3ccsc3)CC2C)cnc1F N1(C(C=C(C)C(C)C)=O)CC=C(CC(=O)N(C)Cc2nnc(C)o2)CC1 c1(C(=O)NC2C(NC(CCN(C(C)=O)C)=O)CC2)cnc2ccsc2c1 c1(C(N2CCC(C)(CNC(C3CCCN3N=O)=O)C2)=O)cnc2occc2c1 CCCCCN(CCC(=O)NCC(C)NC(=O)Cn1ccnn1)CC CC(C)CCCC(C)C(=O)N1CCN(C(C2CNC(=O)C2)=O)C(C)C1 C(N=c1[nH]c(Cl)ncc1F)C1N(C(C2CCC(=C)CC2)=O)CCCC1C C(CCCCC(=O)NC1(C)CC(NC(C2CC=CCC2)=O)C1)OCC CCC(C)CCCC(=O)N(CCCCN(C)C(c1ccc(C(C)=O)cc1F)=O)C CCC(C)(CCC(C)C)C(=O)N1CCC(CN(C(=O)CC2CNC(=O)C2)C)C1 c1(C(N2CCC(C)(NC(C3C=CCC3)=O)C2)=O)cc2scc(Cl)c2[nH]1 O=C(CS(=O)(=O)C1CC1)NCC1C=CC(NC(=O)C(F)(F)CO)C1 n1(CC)nc(C)c(CNCC2CC23CC3(F)F)c1C C1(C)(C=O)CCS(=O)(=O)CC1.C1(CNC(C(C)C2(O)CCC2)=O)CCCC1 N1(C(c2cc(CC)on2)=O)CCC(C2CN(Cc3ccc(Br)cc3)C2)CC1 N1(CC(N2CC(C=C)C(NC(C3CC3)=O)C2)=O)CCCCC(C(C)=O)C1=O.C c1(CN2CCC(C(=O)Nc3c(C(C)=O)ccc(F)n3)C2)cc2ccccc2n1C N1(Cc2onc(C)n2)CCCCC(NC(=O)NC2CC23CCOCC3)C1=O c1(NC2CCC(C(=O)NCCCN3CCNCC3)CC2)ncc2c(n1)CCCC2 N1(C(C(CC)F)=O)CCN(C(c2nncn2CC)=O)CC1CO Cc1cc(N)c(C(N2CC(O)(C3CCCN3C(C3CC4CC4C3)=O)C2)=O)cc1F CCCCCCC(CC)(CC)C(=O)NCC1CC(NC(c2cccnc2O)=O)C1 CC1CCC(CNC(=O)C=Cc2cccc(CO)c2)N(C(c2ccnn2C)=O)C1 C(=O)(C(O)CC[S+](C)C)NC1CC(NC(COc2cn(C)nc2)=O)C1 CC1CC(NC(C2(C3CCCCO3)CC2)=O)CN1C(c1ccc(CN=[N+]=[N-])o1)=O c1(OC)cccc(C(=O)NCC(CCOC)NC(=O)C=Cc2nccs2)c1 N1(C(c2cncc(Br)c2)C(=O)NC(C)(C)C)CCc2ccc(Cl)cc21 Cc1nc(C2CC2)ccc1C(=O)NCCN1CCCN(C(=O)C(Cl)=CCl)CC1 CCCCC(O)C(=O)NC1C=CC(CNC(C2(C)CC2)=O)C1 Cc1cnccc1CCNC(=O)CC1CCCCC1NC(c1nccnc1C)=O c1(N2C3C(CNC(c4ccn(C)n4)=O)C(CCC3)C2)c(C#N)cccc1[N+](=O)[O-] C1(CC#C)CCCCN1C(=O)C(Cc1cn[nH]c1)NC(=O)CO.C1CCC1.C Cc1nc2c([nH]1)C(C(=O)NCC1CC1NC(=O)C)CCC2.CCN(C)C c1(NC(C2CC3CC3N2C(c2cccc(O)c2Cl)=O)=O)ccc2cccnc2c1 c1(C(N)C(=O)NC2CC(O)C2)cc(Cl)cc(Cl)c1 c1(C(=O)NC2CN(C(c3cc(C)nn3C)=O)C(C)C2)cn2cc(Cl)cnc2n1 c1(CC)cnc(Cl)[nH]c1=NC(CNC(c1cc(S(N)(=O)=O)c[nH]1)=O)C(C)C c1(C(N(CCC(=O)NCC2CCC(F)C2)CC)=O)[nH]nnc1C N1(C(=O)CSc2nc(C3CCCO3)n[nH]2)CC(O)CC1C(=O)O C1(NC(c2c(C(C)C)cco2)=O)CN(C(=O)COc2ccccc2O)CC1(C)C C1(C(N2C(CCCNC(CCCCC)=O)CCC2)=O)Cc2ccc(OC)nc2N1 N1(C(C2(F)CCCN(C(c3c(C)ccnc3)=O)C2)=O)CCOC2(CCC2)C1 N1(C(CCC)=O)CC2(CCN(C(c3sc(CO)nc3C)=O)CC2)C1C(C)C C=Cc1cncc(C(=O)NC2CCCC(NC(C3(CC)CCCC3)=O)C2)c1 N1(C(C)C)CCC(NC(=O)C(c2ccccc2)NC(=O)CCc2cccs2)C1=O C1(NC(C(C2CCCC2)OCC)=O)CCN(C(c2cn[nH]c2)=O)CCC1(F)F CN1C(=O)CCCC1C(=O)NCCC1(NC(c2nc(Br)c[nH]2)=O)CC1 Nc1nc2ncccc2cc1C(=O)NC1CC(O)CN(C(c2csc(O)n2)=O)C1 c1(SC)ccc(CCC(=O)NCC(C)N(C(=O)C(CC)n2nccc2C)C)cc1 C(=O)(N1CCC(C(N2CCCC(F)(CO)C2)=O)O1)C1(OC)CCCC1 N1(C(C2(C)CC(=C)C2)=O)CC2(C1)CN(C(=O)CC(CC)CC(C)C)CC2CO c1(C(=O)NC2CCC(C)N(C(=O)C=CBr)C2)cccc2sccc12 Cc1c(Br)ccc(O)c1C(N1CC2CC2(NC(=O)C(C)SC(C)C)C1)=O c1(CC(N2CCN(C(CC(=C=C)C)=O)CC(O)C2)=O)ccc(S(N)(=O)=O)cc1 C=CCC(=C)C(=O)NC1CCC(c2ccc(Cl)cc2)C1 C1(N(c2ccccc2)C(c2cccc(CN(CC)CC)c2)=O)CCC(=O)NC1C N1(C(C(C(=O)OCC)OC)=O)CCC(C)C12CC2.c1cc(C)on1.C(=O)C O=C(C1=NOC2(CCN(c3ncc(C4CC4)cn3)C2)C1)Nc1cc(Br)ccc1I c1(CC)cc(C)ccc1C(N1CCC(O)C1)=O.C(=O)CCN(S(C)(=O)=O)C Cc1cc(=NCCC2(C)CCC2)[nH]cc1S(=O)(=O)N1CCOC(C)C1 c1(C(=O)N)csc2cncn12.C1(C(=O)OC)C(C(=O)NC(C)CC)C1(C)C c1(CNC(CC(C)F)=O)cnn2c1CN(C(c1ccc(C(C)(C)C)[nH]1)=O)CC2 N1(C(c2c(CC)oc(C)c2)=O)CCC(NC(=O)C(C)OCCC(C)C)C(C)C1 c1(SCC#C)cccc(C(=O)Nc2csc(Br)c2)c1 c1(C(N2C3CN(C(C(CCOC)(C)C)=O)C(C3)C2)=O)cc2c(cc1O)OCO2 CCCCC(CNC(c1ccc(OC)nc1)=O)NC(c1cn(C)c(O)n1)=O N1(C(C(CC#C)C2CC2)=O)CCOCC(C(=O)NCC2OCC3CCC2C3)C1 C1(CNC(C2CCC(C(=O)OC)C2)=O)(C)CCN(C(c2cscc2Cl)=O)C1 C1(C(=O)NC(C=CC(=O)NC(C(C)(C)OC)C)C)CCOC1(C)C c1(CC=O)noc2ccc(F)cc12.C1(O)(CC#C)CC(C(=O)NCC(C)C)C1 C12CCC(C1)C(=O)N2.c1(CNC(=O)Cn2ncnn2)cncc(C(=O)N)c1 Cc1nc(C2CC2)nc(S)c1C(N1CCCCC1)=O.C1(CC(=O)N)CNC(=O)C1 C1(C2CCN(C(c3c4c(nn3C(C)C)CCCC4)=O)CC2)(C(=O)OC)CC1 C(CN=c1nc2sccc2c(NCCc2ccc(Br)cc2)[nH]1)c1c(C)noc1C c1(C(=O)NCC2OCCN(Cc3nnc(CC)s3)C2)c(Cl)nc2ccccn12 C(=O)(C(C)(C)C(C)(C)O)N(CC)CC.[SH](=O)(=O)C1CC1.C(=O)(C)N N1(C(c2ccc(C3CCCO3)nn2)=O)CC(NC(C2(O)CCC2)=O)C2CC2C1 Cn1ncc2c(N3CCC4(CCC(O)C4)CC3)nc(=NCC(F)C3CCC3)[nH]c12 Cc1nc(-c2ccsc2)ccc1C(=O)NC1CCCCC1NC(C1CCCC1)=O C=CCCCCCCC(=O)NCC(C(=O)Nc1ccc(CO)c(F)c1)C(C)C CC1CCC(C)(C(N2CCC(O)C(NC(=O)CCCCc3cnc[nH]3)C2)=O)CC1 CC1(C)C=CCCC1.C1(C=O)CCCN1C(=O)C1CC1.C1(C=O)(CC)CC1 C(CCCC(=O)N1CCC(F)(CF)C1)N(C(CN1C(C)CCC1)=O)C c1(OC)cc(Br)c(NCc2ccncc2-c2cnc(O)c(C)c2)c([N+](=O)[O-])c1 CCCC(O)(CNC(=O)NC(c1ccccc1)C1CCC(C)C1)CCC C(C)(CC(C(=O)NC(C)C)N(C)Cc1ccccc1Br)SC c1(C(=O)OCCC)sc(NC(c2ncc(Cl)cn2)=O)cc1C C(=O)(C1=NNC(=O)C1)NC(CC(C)C)CNC(C1(Cl)CC12CCC2)=O Cc1nc(C(=O)NC(c2cnn(C)c2)C(=O)N)c(C)s1.C(CC1CCCC1)CO c1(C(=O)NC(CC#C)C(=O)NC(C)CCCO)cc(O)nc(C)n1 n1(CC(N2CC(C(C)NC(=O)CC(=O)N(C)C)C2)=O)ccc([N+](=O)[O-])n1 Cc1c(C(N2CC(CF)(NC(=O)Cn3cc(C(C)O)nn3)C2)=O)cccc1F N1(C(CC=CC=C)=O)CC(F)(F)CC1(C)CNC(c1cc2c[nH]nc2s1)=O c1(C(=O)NC(C)CC2CCN(C(=O)CCc3cnc[nH]3)CC2)cc(O)ccc1N CCCC(C)C(C)N(C(C1CC(=O)N(c2cnn(C)c2)C1)=O)CC C1(CC(=O)NCCN2CCCN(C(CS(C)(=O)=O)=O)CC2)CC2(CCCC2)CO1 Cc1nc2c(N3CCN(C)CC3CNC(=O)CCC3CCOC3)ncnc2s1 C1(C(=O)N)CC2CCC1C2.c1(C(C(=O)N2CC(C)C2)NC(CC)=O)ccccc1 c1(C(N2CC(CC)C2)=O)cn(C)c(=O)n(C)c1=O.c1(CC=O)ccoc1.CO CC1C2CC(C(=O)OC(C)(C)C)(C2)N1CC(=O)Nc1ccc(F)cc1F O=C(C1=CCOCC1)NCC1CCCC(NC(=O)CSCC(F)(F)F)C1 C(=O)(CS(=O)(=O)CCC(F)(F)F)NC(C)C(C)NC(=O)C(C)(C)C(N)=O C1(C(=O)NC2C(C(N(CC)CC3(O)CCC3)=O)OCC2)CCOC1(C)C c1(NC(C)CN(C)C(C2(Cc3cccc(Cl)c3)CCC2)=O)ncc(Cl)cn1 c1(CN(C(c2cscc2OC)C(=O)NCC2CC2)CCCC)ccccc1 c1(CNC(Cn2c(C)nc(C)n2)=O)cc(O)nc(C)n1.c1(C=O)ccsc1Cl.N Cc1cnn(CC(=O)NCCC(O)C)c1.C1(C=O)CCCN1C(=O)C(F)(F)F.N CCCCC(C(=O)NCCC1(NC(=O)COc2ccccc2F)CC1)N(C)C c1(OC)cccc(N(C)CC2CCN(C(c3cc(Cl)on3)=O)C2)c1[N+](=O)[O-] N1(C(C(CC)C#N)=O)CC2CCC1C(NC(c1c(Cl)n[nH]c1C)=O)C2 c1(OC)cncc(CNCc2ccc(OC(C)C)cc2)c1 Cc1ccc(N)c(C(=O)NCC(C2CC2)N(C)C(c2oc(C)nc2C)=O)c1 C(=O)(CCCC(=O)O)NC(CCOC)C(=O)N(C1CC(F)(F)C1)C.C(C)(C)C C(C)(CC1CCC1)(C(=O)NC(C)CN(C(=O)Cc1cn(C)nn1)C)OC CC1CCC(C)N1CC(=O)NCCC(N1CC(C)(NC(N)=O)C1)=O.C1CC1 CC(CCCCNC(=O)C(=Cc1cn(C)cn1)F)NC(C1CCCN1C)=O N1(C(C=CC=CCC)=O)CCC2CCC(NC(c3cn(C)cn3)=O)C1C2 c1(C(N(C)CC2CCCN2C(=O)CCc2ccc(F)nc2)=O)ccc(O)c(N)n1 N1(S(C(C)C)(=O)=O)CCC(C(=O)NC2CCCC(C)C2)C(C)(C)C1.C(C)C.C CC1=C(C(=O)N2CC3(CC(NC(c4c[nH]c(C(N)=O)c4)=O)C3)C2)CCO1 C1(CC#C)(C(=O)NC2CN(C(c3cnn(C)c3CCC)=O)CC2C)CCCCO1 c1(C(=O)NCC(CCOC)NC(c2ccoc2C(C)C)=O)cnnc(O)c1 c1(NC(c2ccc(SCC)nc2)=O)ccccc1C.c1(C=O)cc(C)c(C)[nH]1.N C1(CNC(COC(CC)C)=O)CCN(C(c2c[nH]c(=N)s2)=O)C1(C)C C1(C(C(=O)NC2(C(C)=O)CC2)C)CCCN(C(c2csc(CO)n2)=O)C1 CC1(C)CCN(C(=O)Cc2cccnc2)CC1NC(=O)CC1CC=CCC1 c1(C(C)C)cc(O)ccc1C(=O)NCc1cc(O)cc(O)c1 c1(-c2nc(CNC(C3CCn4nccc4C3)=O)on2)cnc2cc(C)ccc2c1 C12(C(=O)NCC3COCCN(C(c4ccc[nH]4)=O)C3)CC1COC21CCC1 N1(C(c2c(CC)noc2)=O)CCOCC(F)(C)C1.c1(C(=O)N)c(C)oc(C)c1C C(=O)(CCCCNC(C)C)NCC(C(C)C)OC c1(-n2c(C3C(CCC)C3)nc(-c3ccc(Cl)cn3)n2)c(C)cccc1C C1(NC(c2c(C)cccc2)=O)CCOC2(CCN(C(=O)C(F)Br)CC2)C1 Cc1cc(N2CC3C(NC(C4CCCC(O)C4)=O)C3C2)n2nc(C)cc2n1 C(=O)(C1=CCCC(C)(C)C1)N.N1(C(c2c(C)cc(SC)o2)=O)CCC(CO)CC1 C(CC(C)(C)CNC(=O)C(CC1CCC1)NC(=O)CC(C)n1cccc1)OC C1(C(=O)NCC(C)NC(C2COC(C)(C)CO2)=O)CC(C)(C)OC(C)(C)C1 c1(C(=O)N)cncc([N+](=O)[O-])c1.C1(NC(C(c2cn(C)nc2)O)=O)C2CCCC12 c1(OC)cc(C(N2CCCC2C(C)C)=O)on1.C(=O)(CC)N.C(=O)C1CC1 C(=O)CC(F)(F)C(C)C.C(C(=O)NC1CCC1)(C(C)C)NC(CC(C)C)=O.N C(=O)(CCCCCC(C)(C)C)NCCCCCCNC(c1c(CC)cncc1)=O c1(C(N2CCCC(CCNC(C(C(=O)OC)C)=O)C2)=O)ncc(N)nc1C c1(CC)ccc(C(=O)NCC2(C)CCN(C(C3(C)CCC3)=O)C2)c(F)c1 c1(C(=O)NCC(C)C)ccc(C#N)cc1.C1(C(=O)N)CCC(C(C)(C)C)CC1 Cc1cccc(C(=O)NC(c2c(C)cccc2Br)C(=O)N(C2CSC2)C)c1O CC1(C(=O)NCC2(F)CC(NC(C3CCCC3)=O)C2)CCCS1(=O)=O.C C1(NCCN(C(C)C)C)CCN(c2cc(NC3CC(CF)C3)ncn2)CC1 N1(C(C(COC)OC)=O)C2CCC1C1CC1(NC(C1CC=CC1)=O)C2 C(C(F)(C(=O)NCC(=O)NC(C)C)C(C)C)NC(c1n(CC)nnc1)=O N1(C(c2c(C(N)=O)cccc2)=O)CCC(F)C(NC(=O)CCCC2CCCC2)C1 CC1(C)CN(C(C2CC2(C)Br)=O)CC1NC(=O)CCC1(C)CCC(=O)N1 C(N=c1[nH]cnc(NCc2ncoc2C(C)C)c1C)c1c(OC)nn(C)c1 C1(CC)CN(C(=O)C(N2CCCC(C)C2)=O)CCC1NC(=O)C(C)(C)CCF C1(C2CCCO2)(C(N2CCC(CN(C(C3CCCO3)=O)CC)CC2)=O)CCCO1 C1(C(N2CCC(F)(CNC(C(C)OC)=O)CC2)=O)CCc2cnn(C)c2C1 C(=O)(CCC[S+](C)(C)C)N(C1COC1)C C(C)(CNC(N1CCN(CCCn2ccnc2)CC1)=O)(C(F)(F)F)OC c1(C(N2CC(C)CC(NC(COCCCC)=O)C2)=O)c2c(nn1CC)CCCC2 c1(C(N2CCCC(NC(CCCC(C)C)=O)C2)=O)cc2cc(F)c(F)cc2[nH]1 Cc1nc2ccc(C(N3CCCc4ccccc43)=O)cc2s1 N#Cc1c[nH]c(C(N2CC3CC2C3NC(c2cc(CCO)on2)=O)=O)c1 C#Cc1ccc(C(=O)NCC2CCN(C(=O)CNc3ccccn3)CC2C)cc1 C1(C(=O)NCCNC(c2csc(C3CC3)n2)=O)CCN(C2COC2)CC1 N1(C(CC(CC)(C)C)=O)CC(NC(=O)C(F)(F)c2ncccn2)CC2(CCC2)C1 N1(C(CC(C)OC)=O)CCCC(N(C)C(c2nnn(C)c2C(F)F)=O)CC1 CCCCCC(O)CC(=O)N1CC2OCCN(C(=O)C(F)(F)C3CCCC3)C2C1 CC(CC(=O)NC1CC(O)(CNC(=O)CCc2nncn2C)C1)c1ccncc1 CCCC(C(=O)NCCC1CC(F)(F)C1)NC(=O)C(C)(O)C1CCC1 CCCC(CC)CC(=O)NC12CCC1CN(C(c1cc(N)c(Cl)c(O)c1)=O)C2 C(N=c1ccc(C#N)c[nH]1)C1CN(C(C2(CC#C)CCCO2)=O)CC1C(F)(F)F N1(CCN(C)C)CC(C(=O)N(C)CCNC(c2cnc(Cl)[nH]2)=O)CC1=O Cn1[nH]c(C(=O)NC2CN(C(C3CC3c3ccc(F)cc3)=O)C2)nc1=O N1(C(C(CC)N2CCCC2=O)=O)CC2CC2(CNC(=O)Cn2cc(C#N)cn2)C1 C1(C(=O)N)CC2CC1CC2.C1(C=O)CC2(CCC2)CO1.C(C)(C(F)(F)F)OC CC1(C)C(CNC(c2ncc(Cl)cc2Cl)=O)CCN1C(=O)CC1(C#N)CCC1 CC(C(=O)NCCO)Nc1ccoc1.C1(CC(=O)N(CCC)C)CC1(Cl)Cl CCC(O)CC(=O)NC(Cc1cn[nH]c1)C(N1CCC(C)(CCO)C1)=O N1(C(c2cccc(C)c2N)=O)CC(NC(C2(F)CCCOC2)=O)CC2(CC2)C1 c1(C(N2CCC(F)(F)CC2)=O)cc2c3c(ccc2[nH]1)N(C(c1cnon1)=O)CC3 C#Cc1ccc(F)c(C(=O)N(C)CCN(C(=O)Cc2cc(C)ccc2C)C)c1 CN1CCC(CC(N2CCC(OCC)C2)=O)C1=O.C1(CC=O)CCCS1(=O)=O.N N1(C(C23CCC(C=O)(C2)C3)=O)CC2CC1CN2C(=O)C(N1CCSCC1)C.CO c1(-c2cn(CC(=O)O)nn2)ccc(C(=O)NCc2cncc(CO)c2)nc1 N1(C(CC)=O)CC2(NC(=O)CCSCc3cccc(OC)c3)CCC1CC2 C1(NC(C2CC(=O)NC2)=O)COCCN(C(=O)CSc2ccc(Br)cc2)C1 N1(C(c2cccc(N)n2)=O)CCCCC(NC(C2CCCCS2(=O)=O)=O)C1 c1(C(=O)NCCCOCCN(C(C(CC=C)C)=O)C)ccc([N+](=O)[O-])[nH]1 C1(NC(C2CC2[N+](=O)[O-])=O)C=CCN(C(c2cscc2C(F)(F)F)=O)C1 C(=O)(C(COC)OC)NC1(C(NOCC(=C)Cl)=O)CC1 N1(C(CC(C=C)CC)=O)CC2(C(=O)NC3CC(C)CCC3O)CCC1CC2 c1c(C)cccc1C.c1(COC)ccc(Cn2cc(CNC(=O)N)nn2)nc1 c1(OC)cc(Cl)ccc1C(C)(C)NC(=O)C(Cn1cccn1)OC N1(C(C(C2CCCCC2)C)=O)CCCC(C2CN(C(=O)CSCC(F)F)C2)C1 C(=O)(C1=CCOC1)N(CC(CN(C(c1c(C(C)C)ccs1)=O)C)O)C N1(C(CCCCCC)=O)CCc2nc(CNC(C3CCC4(CCC4)C3)=O)sc2C1 Cc1cncc(CCC(=O)NC(C2(O)CCN(c3nnc(C(C)C)o3)C2)C)c1 C1(O)(CNC(C2(C)CC(=C)C2)=O)CCN(C(c2ccc(O)cn2)=O)CC1 CC1CC(NC(c2ncoc2C2CCCO2)=O)CCN1C(=O)Cc1ccccn1 c1(N(C(C)CCNC(=O)CN2C(=O)CCC2=O)C)cc(O)nc(O)n1 c1(SCC)ccc(C(N2CCC(CNC(=O)C(O)c3cnc[nH]3)C2)=O)cc1 N1(S(c2ccc(OC)cc2Cl)(=O)=O)Cc2ccc(F)cc2CC1C C(=O)(C1=NNC(=O)C1)N(CCCCC(N1CC2C(CC)(C2)C1)=O)C c1(C(N2C(C(=O)NC(CC=C)CO)CCCC2)=O)cc(C)nc(O)c1 N1(C(=O)CCc2ccc(O)cc2)CC2(CCN(C(=O)CSc3cn[nH]c3)CC2)C1 C1(N(C(C(C)N2CCC2)=O)C)CCCC2CN(C(=O)CCCC(F)(F)F)CC12 C#CCC(CC(F)F)C(=O)N1CCC(C(=O)NCC2(CN=[N+]=[N-])CC2)O1 c1(C(N2CC=CC(C(=O)NCC(COC)OC)C2)=O)cccc(F)c1O N1(C(CNC(CCC)=O)=O)CCN(C(=O)CC2OCCC2(C)C)CC1CO C1(COC)CCN(C(=O)C(c2cnn(C)c2)NC(=O)C(C)SC)C1 c1(CN(CCNC(c2cc(F)n[nH]2)=O)CCOCCO)ccccc1 c1(OC)ccc(CC(=O)NC(C2CCCN2C(=O)C(C)(C2CC2)OC)C)cc1Cl CCC(C)C(CC(=O)Nc1ccccc1OC)NC(C12CC(C#N)(C1)C2)=O c1(C(C2CC(=C3CCC3)C2)N(C(C2CCC2)=O)CC)cnc(Cl)c(C)c1 C1(C(N(CCOC)CC2CC2)=O)CCC2(CC2)N1C(=O)CCCSC C(=O)(C(C)CCCC(C)C)N(C(C(=O)NC(C#C)C(C)OC)C(C)CC)C c1(CCC(N2C(CN(C(C)=O)C3CC3)CCC2)=O)ccc(O)nc1 C(=O)(CCN=c1[nH]ccs1)CC1N(C(C2CC(C)(C)CN2c2cc(O)ncn2)=O)CC1 c1(OC)ccc(C(=O)NC2CN(C(c3ccsc3C)=O)CCC2C)c(OC)c1 C1(C(=O)NC2CCCC(CNC(CC=C=C)=O)C2)CCCC1C1CC1 CC1CCN(C(c2ccncc2)=O)CC1CC(=O)N(CCC(=O)NC1CC1)C c1(C(C)C)nsc(CNC(c2nscc2Br)c2nnnn2C2COC2)n1 C(C#N)(C(=O)C(C)(F)F)=C1CN(C=O)C1.CC(C)C.CC=CC=CC N1(C2CC(N)CC2O)CCC(S(=O)(=O)c2ccccc2)C1 S(=O)(=O)(CCC(=O)NCCCCC1CN(C(=O)CC2COCC(C)O2)C1)NC n1(CCC(N2C(C)CCC2)=O)cnc([N+](=O)[O-])c1.Cc1nc[nH]c1CC(=O)NC c1(OC)cccc(NC(=O)NCC2CC2C2CC2C)c1C C=Cc1cc(C(N2CCN(C(c3[nH]c(=N)ccc3C)=O)C(CC)C2)=O)cc(F)c1 C(=O)(C(C)CC(F)F)N(C(CNC(CCc1nc(C)c(C)o1)=O)C)C C(=O)(C(CC(C)C)C(N)=O)N1CC(OC)CC1.C1(C(=O)N)CSCN1C(C)=O c1(CC)noc(C)c1C=O.C12(CCC3CC3)CC1CN(C(=O)C(C)(F)F)C2 CCC(CC)CCC(=O)NC1CC(C)CN(C(c2cc(C(C)(C)C)nn2C)=O)C1 N1(C(C2(C)CC=CC2)=O)CC2CCC(CNC(=O)CS(=O)(=O)CCO)C2C1 C(=O)(C(O)C(F)(F)c1ccccc1)N1CCC(CNC(C(C)(C)C2CC2)=O)CC1 c1(N(CC=C(C)C)C2CC2)nc2c(c(=NCCC(C)O)[nH]1)COCC2.C(C)(C)C N1(C(C(C(C)C)NC(c2cnn(C)c2)=O)=O)CCC(O)(C(F)(F)F)CC1 n1(CC)cc(C(=O)NC23CC2CN(C(=O)CC2CC(O)C2)C3)c(O)nc1=O c1(C(=O)N)cc(Cl)ncc1N.Cc1ncn(C)c1C(N1CCC(C(F)F)(C)C1)=O C=CCC(CC(C)C)C(=O)N(CCCC(=O)NCC(C)(C)C(C)C)C C(=O)(C1=CCCCC1C)NC1CN(C(CN(C(C)=O)C)=O)C(C)CC1 C1(NC(CCC2CCN(C(c3nc(C)sc3)=O)C2)=O)CCCC1C1CC1 C1(CC=O)CC2C=CC1CC2.C1(NC(C(C)OCCN(C)C)=O)CC(F)C1 C(CCCC(CO)NC(=O)C(F)(F)c1ccccn1)NC(=O)Cc1ccccn1 c1(C=O)cc(C2CC2)[nH]n1.C(CCCNC(=O)CC1CC1)OCCCC.C c1(CC(=O)NCC2N(C)CCC2)cc2cc(Cl)ccc2[nH]1 C(CN=c1[nH]c2ccccc2[nH]1)NC1(c2nnnn2C)C(CC)CCCC1 N1(C(C2N(CC)CCOC2)=O)CCC(CO)C(NC(=O)COC(C)=O)C1 S(=O)(=O)(c1ccccc1Cl)N1CCC2(C(C(=O)Nc3cc(C)nn3CCO)C2)CC1 C1(CC#C)(C(=O)NC(CO)C(C)NC(c2n[nH]cc2CC)=O)CC=CCC1 C(c1ccccc1[N+](=O)[O-])=CC(=O)NCC1CN(C(=O)CCCn2cncn2)C1 c1(CC(N2CC(NC(C(C)O)=O)C3(C2)CC3)=O)ccc2[nH]ccc2c1 N1(C(c2c(C)cc[nH]2)=O)CC(C)OC2(CCC2)C1.c1(C(=O)N)coc(N(C)C)n1 c1(CNC(c2nc(C)ccc2OC)c2n(CC)nnn2)cc(OC)ccc1F CON(CCC(=O)NCCc1cccc(F)n1)C(=O)COC1CCOC1 c1(CC)c[nH]cc1C(=O)NCCCN(C(=O)C(C)c1ccsn1)CC c1(-c2cccc(C3C(C(=O)NC(CCCN)CO)C3)c2)cnc2[nH]cnc2c1 c1(C(N2CCC(NC(=O)COC3CCCCC3)C2)=O)ccnc2c1OCO2 CCC(CC(=O)NCc1cn(CC(N2CCC3CC23C)=O)nn1)C(C)(C)C C=C(C)CC(C(=O)N(CC(C)C(C)C)C)NC(=O)CC1(N(C)C)CC1 c1(N2C(CN(C(CCC3C(C)C3)C(=O)NC3CCCCC3)C)CCC2)cccc(F)c1 N1(C(C(C)N(C)C(C2CCN(C)C(=O)C2)=O)=O)CCC12CC(C(N)=O)C2 c1(CC)nc(C)c(C(N2CCC2)=O)o1.C1(C(=O)N)C2CCC1(c1ccccc1)C2 CCCC(CCCNC(c1cccnc1S)=O)NC(C1CC1Sc1ccccc1)=O CC(CC(F)F)C(=O)NCc1cnn(C)c1C(=O)NC(c1cccnc1)C CCC(C)(CNC(c1ocnc1C)=O)C(=O)NCC(C)(O)CN(C)C C1(CNC(=O)CCc2ccncc2)CC(C(=O)NC2CCOC2=O)=NO1 C(=O)(C1CCOc2ccc(Br)cc21)N1CC(NC(C(=O)N(C)C)=O)C(F)C1 N1(C(c2scc(C)c2C)=O)CC2CN(C(=O)C(F)n3ccnc3)CC2C1 N1(C(CNC(C)(C)C)=O)CCC2C(CCCN2C(C2CCc3ccoc3C2)=O)C1 C#Cc1cc(F)c(C(=O)NCC2CCC2)cc1F.C(c1cccnc1)=CC=O.N C1(C(C)NC(C2CC2[N+](=O)[O-])=O)CCCCN1C(=O)CO.C1(C)CCOCC1 C1(OC)CCCC(CNC(c2cccnc2)=O)C1.n1(CC=O)ccc(C)n1.C c1(C(N(C2CCCC(N(C)C(c3occc3F)=O)C2)C)=O)cncc(Cl)c1 c1(C(=O)OCc2onc(-c3c(C)ccs3)n2)oc(C2CCCN(C)C2)nc1C c1(C(=O)NC2CCN(C(Cc3c(C)ocn3)=O)CC2C)cnc2ncnn2c1O Cc1ccc(=O)n(CC(N2CCC(NC(C34CCC(C3)C4)=O)CC2C)=O)c1 c1(CNC(CC2N(C(c3c(CC)ncs3)=O)CCC2)=O)cccc(OC)c1O c1(C(=O)Nc2c(-c3cccc(C)c3)cccn2)cc(Cl)cc(Cl)c1OC(F)F C1(NC(C(CC)=CC)=O)CC2CCC1N(C(c1cc(N)ccc1Cl)=O)C2 N1(C(CSc2c(C)noc2C)=O)CCC2(NC(c3cnsc3C)=O)CCCC12 CC(C)C(C(=O)NCC1CCC1)c1cnn(C)c1.C1(=CC=O)CCOCC1.N C(CCNC(C1CCCS1)=O)(C(=O)NC1(c2noc(C)n2)CC1)OC Cc1ccn2nc(C(=O)NC3CCN(C(=O)C=C4CCN(C)C4)C(C)C3)nc2n1 C1(CC)CC(C)CN(C(=O)CC(C(C)C)NC(=O)CCCCC=CC(C)C)C1 c1(C(=O)NCC2CN(C(c3cnn(CC)c3C)=O)CC2C)ccc2cnnn2c1 O=C(C1CCCc2nn[nH]c21)NCC1CN(C(c2ccc(Cl)c(O)c2)=O)CCO1 N1(C(=O)NC(C)(C)C)CCCC(C(N2CCCCCC2CO)=O)CC1 N1(C(C2(CC#C)CCCCO2)=O)CCN(C(=O)C=CI)CC12CCC2 c1(CC(N)=O)ccc(S(=O)(=O)N2CCCC2C(=O)O)cc1.c1ccc(O)cc1.C c1(C(N(C)CCN(C)C(c2cnsc2)=O)=O)ccc(F)c2ccoc12 Cc1cccc(-n2nc(-c3ccco3)nc2-c2ccoc2Br)c1 N1(C(C2CC3CCC2CC3)=O)CC2CCC(C1)N2C(C1CCCNC1=O)=O c1(OC)ncc(C(=O)NC2CCC(CN(C)C(c3csc(Cl)c3)=O)CC2)cn1 C1(C)(CNC(CC(C)NC(c2cc[nH]c2C2CC2)=O)=O)CCCC1O Cc1cc2[nH]c(O)nc2cc1S(=O)(=O)N1CCCC1c1ccc2c(c1)OCCO2 C1(C)(C(=O)NC(CN(C(=O)CCCCN2CCOCC2)CC)C)CCNC(=O)C1 c1(OC)c(C(=O)NC(C)(C)C)cccc1[N+](=O)[O-].c1(C=O)csc2nnsc12.N C(CC(C)(C)C)(C(=O)NCC#CCCO)NC(C1CCCN(C)C1)=O C12(C(N(C)CC3CC3(F)F)=O)CC1CN(C(=O)C#CC1CC1)C2 c1(C(=O)OCC)ccc(CNC(=O)C(=O)N)cc1.CC=O.C(C)(C)C C(CC(C(=O)NCc1cc(C)sc1C)NC(=O)CC(CC)OC)=CC c1(OC)c(C(=O)NCC(CO)NC(=O)Cn2cccn2)cc(Br)cc1F C1(NC(C(C)n2cccn2)=O)CC2(C1)CC2NC(=O)COC(C)(C)C C(C1=CCCN(C(C2(S(C)(=O)=O)CC2)=O)C1)NC(c1cc(C)nn1C)=O c1(CC(N2CCC(NC(CC(=O)OC)=O)CC2C)=O)csc2cc(Cl)ccc12 c1(C(N(CCNC(c2cnc(N3CCOCC3)s2)=O)CC)=O)cc(Cl)ccc1F CCN=C(NCC1CCC(CC(=O)OCC)CC1)NCC1CCOC(C)C1 Cc1oc(-c2cccs2)nc1CC(=O)NC1CN(C(=O)C(C)c2cc[nH]n2)C1 C1(NC(Cc2nc(COC)sc2)=O)CN(C(C2(OC)CCSC2)=O)CC1F N1(C(C2C(C=CC)CN(C(=O)C(CC)CCOC)C2)=O)CCCN(C)C(=O)C1 c1(CC(N2CCC2)=O)ccc(S(C)=O)cc1.C12COC(C=O)(C1)C2.COC c1(C(=O)NC2C(CC)N(C(=O)C=CC=CCC)CCC2)cccc2[nH]ncc12 c1(C(=O)NC(CNC(CSCC=C)=O)CC)nc(C)oc1C C#Cc1ccc(C(=O)NCC(O)CNC(=O)C(c2ccc(Cl)cc2)(C)O)cc1 NC(=O)CCCCC(=O)NC(C(=O)NC12CC1COC21CCC1)c1ccoc1 c1(OC)nscc1C(=O)NC1(c2cn(CC3CCC(=O)O3)nn2)CCOC1 Cc1cnc(C(=O)NC2CC(NC(=O)Cn3ccnn3)C23CCC3)c(C)c1 C(C1=NOC2C3CCC(C3)C12)NC(N1C(C#C)C2CCC1C2)=O c1(C(N2C(CN(C(C(C)C3(O)CCC3)=O)C)CC(F)C2)=O)cnn2cnnc2c1 c1(C(N2C3CN(C(=O)CC4CCC45CCC5)CC2CC3)=O)ccc2nc(O)[nH]c2c1 CC1CC(NC(c2cccc(N3C(=O)CCC3=O)c2)=O)CN(C(=O)C(C)(F)F)C1 CC1CN(C(C2(C)CCC(=O)N2)=O)CC1NC(=O)Cn1cc(C#N)cn1 Cc1cc(C(N2CC(N(C)C(c3ccc(=N)[nH]c3)=O)C2)=O)c(F)cc1Cl c1(C(=O)NCC(C)NC(C2CCC23CCC3)=O)cc2cccc(O)c2n1C C(=O)(C1CCc2nccn21)NC1(CC(=O)NCc2cnc[nH]2)CCC1 C(CCC(=O)NC1CC(N2CCCC2)C1)N(C(=O)CCc1cscn1)C c1(CN(CCC)CC2CC(OC(C)(C)C)C2)cc(Cl)ccc1F c1(C2(C(N(CCC)CCNC(=O)C(O)C3CC3)=O)CCCO2)ccccc1Br CCCC(CNC)CCO.c12cn(nn1)C(C(=O)OC)COC2 C#Cc1cc(C(N2CC(Cn3cc(CCC(C)O)nn3)C2)=O)ccc1C N#Cc1nc[nH]c1C(=O)N(CCC)C1CC1.c1(CC(C=O)O)ccc(Cl)cc1.N Nc1cc(Cl)nc(C(=O)NC2CCCC2NC(c2ncc(C(F)F)s2)=O)c1Cl c1(C(=O)NCC2(O)CN(C(C3CC(C)C3)=O)C2)cc(Br)cn2ccnc12 C(=O)(C(C)(C)C)NC(C(=O)N(C(C)CNC(=O)CC1CN(C)C1)C)C CC(O)(C(=O)N1CC(NC(=O)CCC2CC2)C(O)C1)C(F)(F)F c1(C(C(=O)NC)N(C(C)Cc2ccccc2Cl)C)cc(OC)c(OC)cc1F CC1CCC(NC(=O)Cc2cccnc2)CN1C(c1n[nH]cc1Cl)=O c1(C(=O)NCCC(C)N(C(C(C(C)(C)C)SC)=O)C)c(O)nnc2c1CCCC2 CCC(C)C(C(=O)N1CC2COCC2C1)NC(c1cc(C)ns1)=O C12(C(=O)NCC(CNC(=O)C(C)O)OC)CC(C(C)C)(C1)C2 c1(C(=O)NC(C)CNC(C2COC2)=O)ccc(C(F)(F)F)c(Cl)c1Cl N1(C(=O)CCN(C2CNC2)CC2CCCO2)CCC2(CCOC2)C1 N1(C(c2cc(OC)ns2)=O)CC(NC(c2cc(C(F)(F)F)n[nH]2)=O)C(C)C1 N1(C(C=C2CCC(C)CC2)=O)CC(NC(c2cccc(F)c2Cl)=O)CCC(O)C1 Cn1nc(C2CCC2)cc1C(N1C(C)CC2CC12)=O.C1(C2CC2)(C=O)CC1.N C12(C(=O)NC(CCCCNC(c3ncc[nH]c3=O)=O)CO)CCCCN1CCC2 N1(C(CC=CC)=O)CC(=O)NC2CN(C(=O)CCS(N)(=O)=O)CCC12 N1(C(Cc2nc(COC)sc2)=O)CC(CNC(C2OCCCO2)=O)C(C)C1 C(C1CN(C(=O)CCC(C)SC)CC1C(=O)Nc1cccc(F)c1F)=CC N1(C(CCc2c(OC)cccc2)=O)CCCC2CCN(C(=O)COCCF)CC12 C(=O)(C1=CCC(C)CC1)N1CCC(NC(C(C(CC)C)OC)=O)CC1 CC1CC(CNC(=O)CCN(C(=O)C=Cc2cncs2)C)=NO1.C1CC1 CCCCC(CC(=O)NC(CN1CCCC1)CC)NC(c1ccnc(C)c1C)=O N1(C(C(C)(C)C#N)=O)CCC2(CCC(NC(c3c[nH]c4ccccc34)=O)CC2)C1 C1(NC(C(N2CCCCC2=O)C)=O)CCC2(CC1)CC(NC(=O)CNC=O)C2 CC(C)CC(C)CNC(=O)C=Cc1cccnc1.C1(C=O)CC(F)C(=O)N1.N C(=O)(CCCCCF)NC1(CNC(CCN2CCC(C)CC2)=O)CC1 c1(C(N(CCN(C(C2C(CC)CCC2)=O)C)C(C)C)=O)cc(C#N)c[nH]1 c1(C(=O)NCC(CNC(c2cncc(C)c2)=O)F)ccc(C)c(Br)c1C C(=O)(CCC(O)C(C)(C)C)N.C(C(=O)NCCCCc1ccccc1)(C(C)C)OC C1(F)(C(=O)NC(CN(CCCC)C)C)CCN(C(=O)CCC(C)(F)F)CC1 c1(C(c2nnnn2C2CC2)NCC(CC)n2cccn2)ncc(C(C)C)s1 c1(C(N2CCOCC(CNC(C3(C)CCNC3=O)=O)C2)=O)cn2cccnc2n1 C(=O)(CCC(F)(F)F)NC(C)C(C)(C)NC(=O)C=CC1CC1 N1(C(C(C(C)C)O)=O)CCC(C)CC1CNC(=O)CC(C)(C)C c1(C(N2CC(CNC(C3(C)CC=CC3)=O)OCC2)=O)ccc(=O)n2c1COCC2 N1(CC)CCC(Sc2ccccc2)C1=O.C12(CCC1)C(=O)NC2 C1(C(=O)NCC2(NC(C3(OC(C)C)CCC3)=O)CCC2)CCCCN1C c1(OC)ccnc(C(=O)NC(C2(O)CN(C(c3csc(C)c3)=O)C2)C)c1F Cc1cn2c(=O)cc(CN3CC(OC(C4CCc5ncnn5C4)=O)C3)nc2s1 CC1(CNS(=O)(=O)Cc2ccc(Cl)cn2)CCCCC1(F)F CCCC(C(O)C(=O)NCc1cccc(C#N)c1)NC(=O)C(=O)CC(C)C N1(C(c2nc(OC)c(F)cn2)=O)CCN(C(=O)CN2CCC(C)(O)C2)CCC1C CC1=C(C(=O)NC2(CNC(C3CCCC3(C)C)=O)CCOC2)CCS1(=O)=O N1(C(c2scc(C#N)c2)=O)CCCC12CCN(C(c1cnnc(C3CC3)c1)=O)C2 NC(=O)CCCCC(=O)N1CCOC(CNC(c2nc(Cl)cc(N)c2Cl)=O)C1 CCCN=C(NCc1nc(-c2ccncc2)n[nH]1)NCC(N1CCCCC1)(C)C c1(OC)ccc(C(=O)C(=O)NC2CC2NC(C2CC(C)CCO2)=O)cc1Cl C1(CC=C)COCC1NC(=O)CCC1CCN(C(c2c[nH]nc2C(F)F)=O)C1 CC1CC(C(=O)NC2(C(F)F)CC(NC(C3SCCCS3)=O)C2)CCS1 c1(SC)ccc(N2CC(C(=O)NCC3CC4(CCC4)C3)CC2=O)cc1 CCCC(C=O)NC(=O)OC(C)(C)C.C(C)CCC.C(=O)C(F)CN(C)C CC(C)CC(C)CC(=O)NCC(O)CNC(c1ncnn1C(C)C)=O c1(OC(C)C)ccc(Cl)nc1C(N1CCC1CNC(=O)CCC#N)=O Cc1nc(NNC(=O)NCC23CCCCC2NCCC3)nc(O)c1C c1(OCC#C)cccc(C(=O)NCCN(C)C(c2ccc(OC)cc2)C)c1 C1(C(C(=O)NC2CC(F)(F)C2)N(c2c(OC)cccc2)C)CC(C)CC(C)C1 CCCC(CC(C)C)C(=O)N1CCC(C(N2CC(O)CC2C(=O)NC)=O)(CC)CC1 c1(C(=O)NC2CC(CNC(CCC(N)=O)=O)C2)cc(Cl)c2c(c1)OCO2 N1(C(CCSCC)=O)CCCC(C)C1CCNC(=O)C(c1cccn1C)=O CC(C)C(CCN(C)C(C1CC2CC1CO2)=O)NC(=O)CCC.[SH](C)(=O)=O.N S(=O)(=O)(C=Cc1ccccc1)N1CC2CCN(Cc3cc(C#N)ncc3)C2CC1 C#CCCCC(C)C(=O)NC1CCCC(C(N2CCC(F)(C#C)CC2)=O)C1 N1(C(CCC(=O)NCC2CC(NC(C3C(C)C3)=O)C2)=O)CCc2sccc2C1 c1(OC)nsc(OC)c1C(=O)N(C)CCOCCNC(=O)CC(C)(C)C N1(CC(N)=O)CCN(C(=NC2CCOCC2)NCC(C2CC2)C2CC2)CC1=O N1(C(=O)OC(C)(C)C)CCSC1C(=O)NC1CC1.c1(C=O)ccc(Cl)o1 c1(OC)ccc2c(c1)C(C(=O)N1CCN(C(c3occ(C)c3C)=O)C(C)C1)CC2 C1(=CNC(c2n(C)nnc2)=O)CCN(C(=O)CC2CCN(CCF)CC2)CC1 c1(NC(C2C(NC(c3coc(Cl)n3)=O)CCC2)=O)ccc([N+](=O)[O-])c(Cl)c1 C1(C(C)C)CCC(N=c2ccc(Br)c(S(=O)(=O)N(C)CCF)[nH]2)CC1 N1(C(C(C=C)C)=O)CCN(C(c2cc([N+](=O)[O-])c[nH]2)=O)CC1CO c1(CC)ccc(C(=O)NCCC2(C)CC2)cc1.C1(CC=O)COC2CC1C2 c1(C(N(CCN(C(C2C(C)CCCC2)=O)C)C)=O)cc2c(s1)CCC2=O N1(C(C(CO)OC)=O)CCCCC1CCNC(=O)CCCF Cc1cccc(C(N2CCC(NC(C3CC(CF)C3)=O)C(F)C2)=O)c1F c1(C(=O)OC)cc(NC(=O)CC2CCCN(Cc3cccc(Br)c3)C2)n(C)n1 N1(C(C(CCC)F)=O)CCCC2C(NC(c3cnn(C(C)C)c3)=O)C(C)(C)C12 c1(C(N2CC(N(C)C(c3ccc(-c4ccncc4)s3)=O)C2)=O)cccc(=O)n1C c1(C(N(C)CC2CCN(C(CC(C)C3CC3)=O)C2)=O)cn(C)ccc1=O C1(C(=O)N)(NC(c2ccc(OC)o2)=O)CCC(C)(C)C1.c1nc(C)c(C)s1 C1(CNC(C=C(CCC)C)=O)CCN(C(=O)C(F)F)CC1(F)F C(=O)(N=c1nc(Cc2ccccc2)[nH]s1)N1CC(C)N(CC(F)(F)F)CC1 CC(C(=O)NCC1(NC(c2n[nH]c3cccnc23)=O)CC1)C(C)S(C)(=O)=O C1(O)(CC(=O)NC2CCCC2NC(C2CC23CC3)=O)CCCC1 N1(C(=O)NCCc2ccccc2OC(F)(F)F)CCc2ccccc2C1 N1(C(c2ccc[nH]2)=O)CC(O)(C2(CNC(C34CSCC3C4)=O)CC2)C1 c1(CC(N2CC(N)(CC)C2)=O)ccc2cncn2c1 c1(NC(Cc2cccc(OC)n2)=O)ccc2c(n1)OCCO2 CC1(C#CC(=O)N2CC(CNC(c3ncccc3Cl)=O)C3CC23)CC1 N1(C(C(C)SC)=O)CCCC2(C1)CN(C(c1ncc(C)cn1)=O)CCO2 C1(OCCC(=O)N(CCC)C)CCCCC1C(C)(C)C.c1(C=O)cnccn1.N N1(C(CCCOC(C)C)=O)CCCC1(C)CNC(=O)CC(C)O.C(=O)C1CC1 C1(NC(c2ccnc3[nH]ncc23)=O)CCCC12CN(C(C1CSC1)=O)C2 C1(N(C(c2n[nH]cc2Br)=O)CC)CCCN(C(=O)COCC(F)F)C1 N1(C(Cc2nc(C)sc2Cl)=O)CCN(C(c2ccn(C(C)C)c2C)=O)C2CC12 C1(NC(C(c2ccccc2)OC)=O)CCCN(c2cc(=O)n(C)cn2)CC1 c1(C(N(CCOC)CCNC(=O)CC2CC2(C)C)=O)cn2ccncc2n1 C(=O)(CCCCCn1cc(-c2ccc(Cl)cc2)nn1)N1CC(C)C(N(C)C)C1 O=S(=O)(c1csc2ccccc12)N1C2CC1CN(Cc1ccc3[nH]ccc3c1)C2 C1(C(N2C3CC(NC(=O)COC4CC4)C3CC2)=O)C2Cc3c(Br)cccc3C12 C(C(=O)N1CCCC2(CC2)C1)(C(C)CC)N(C(c1ccc(CC)s1)=O)C C(=O)(C(C(C)CC)N(C)C)N1C2(C(=O)NC3(CCC)CCOC3)CC(C1)C2 C1(NC(c2ccc(C)c(C)c2)=O)CC2CC(NC(C3(C)CSC3)=O)CC2C1 N1(C(C(CC)C)=O)CC2(CC2)CC1C(=O)Nc1ccc(C)c(Br)c1 C1(CNC(CC(=O)NCC#C)=O)CCCCN(C(=O)C)C1.C(=O)C1CC1 Cc1cc(C(=O)NC(C)CO)ccc1S(N)(=O)=O.C1(C=O)C(F)(F)C12CCC2 c1(C(N(C)CCOc2ncc(C(F)(F)F)cc2Cl)=O)ccc2cc[nH]c2c1 CC(C)(C#CC(=O)N1CCCC1CCO)CNC(=O)C=CCO N1(C(C=CC(C)=O)=O)CCC(C2CCCN(C(C3(C)CCNC(=O)C3)=O)C2)C1 N1(C(C(C2CC2)OCC)=O)CCC2(CC1)CN(CC1CCC3CC3C1)CCO2 C1(CNC(C(=O)NCC=CCCOC)=O)CCCC(C)CC1 N1(CC(C)C(F)(F)F)CC2CCCCC2(CNC(=O)OC(C)(C)C)C1 CC1(F)CN(C(=O)CCn2cccnc2=O)CCN(C(C2CC2F)=O)C1 C(=O)(C(C)(C)CCCC(=O)N1CCCOC(CNC(=O)C(C)C(C)(C)C)C1)OC C(=O)(CN=c1ccc(Cl)n[nH]1)N1CCC(CCOC)(NC(C2CC=CC2)=O)C1 c1(C(C)NC(c2cccc(C)c2)C(C)C)c[nH]c2ccc(F)cc12 C#CC1(C(N2CCCC(CC)C2)=O)CCN(C(=O)CCC(C)=O)CC1 C(=O)(CS(N)(=O)=O)NCCCC(C)NC(=O)Cc1cnoc1 C1(C(N2CC3C(NC(c4cccc(Cl)c4)=O)C3C2)=O)CC(c2ccncc2)=NO1 CC(F)(F)CCC(=O)N1CCN(C(=O)C(c2cccc(C#N)c2)(C)C)CC1 C#Cc1ccc(C(N2CCC(NC(=O)Cn3ncn(C)c3=O)C2C)=O)cc1F Cc1ncc(Cl)c(C(=O)NC2CC(NC(=O)CCCCN3CCCC3)CC2O)n1 C1(C=O)CC(C)(C)CCO1.C(C(=O)OC)N(C(=O)C=CCC)CC=C c1(CC(=O)NC2CCC(N(C)C(c3ccc(Cl)o3)=O)C2)sc(O)nc1O c1(C(=O)NC(C)CN(C)C(C2(C(N)=O)CC2)=O)ncc2n1CCCC2 CC1=C(C(=O)NCC2CCC2C(=O)N=c2ccn(CC(C)C)[nH]2)SCCO1 c1(CC(=O)NC(CC)CNC(C2CC2C(F)(F)F)=O)n[nH]c2c1CCCC2 c1(C2C(CN(C)C(C3(NC(c4nnn(C)n4)=O)CC3)=O)C2)cccnc1 c1(C(=O)NC(C2OCCN(C(C3(OC)CC3)=O)C2)C)cccc2nncn12 C(=O)(CCC(=O)NCC)N(C(C)CNC(=O)C(C)(F)F)CC C1(C(=O)NCC(C)(CO)NC(C2C(C)(C)C2(C)C)=O)CCOC2(CCC2)C1 C1(C(=O)Nc2c(CC)n(C)nc2)CC2(CC2)CN1C(=O)CCCSC c1(CC=O)c(C)cc(C)cc1C.C1(CC=C)(C(=O)NC)CC=CC1.C1CC1 Cc1c(C(N2CCCC3(CNC(=O)CCC4CC4)CC23)=O)[nH]c2ccccc12 N1(C(C)C)CCOC(C(=O)NCC2CCN2C(=O)CN(C2CCC2)C)C1 c1(C(=O)NC(C(=O)NC(C=C)(C)C)CCOC)[nH]ccc(=O)c1C N1(C(c2ccc3ncn(C)c3c2)=O)CCC2(CCN(c3ncc(F)cn3)CC2)C1 N1(C(c2cn[nH]c2)=O)CCCC(C(=O)NC2CC2)C1.C(C=O)OCC#C.N C1(C(=O)OCCOC)CCCC(C(=O)O)N1.c12ccnc(c1)NC2 CC12CCC1(C)CN(C(=O)CC1CN(C(=O)Cc3ccccn3)CCO1)C2 N1(C(C(C)C(C)(F)F)=O)CC2CCCC2(NC(=O)CSCc2ccccn2)C1 C1(C(N(C2CC(NC(C3CCCSC3)=O)C2)C)=O)CCc2nnnn2C1 c1(NC2CN(C(=O)CS(=O)(=O)C3CC3)C2)cc(-c2nn[nH]n2)ccn1 C#CCN(OC)C(=O)C(CCOC)NC(=O)CC(C)CCC CC1(C)CC1(C#N)C(=O)NOCC(=O)NCCOCCN(C)C N1(C(C2(CC)CCCC2)=O)CCOCC(CNC(=O)Cc2occc2C)C1 C1(CC(=O)NCCC(=O)NCC)CCCCN1C(c1ncc(F)cn1)=O c1(CC)ccc(C(=O)NC(C)C=CC(=O)Nc2cnc(C)nc2)cc1 c1(C(=O)N)cc(F)c(F)c(O)c1F.CC1CN(C(=O)C=C2CCN(C)CC2)CC1 Cc1cnnc(O)c1C(=O)NCCC(O)CNC(c1nc[nH]c1C(F)(F)F)=O Cc1cc(C(N2CCN(C(C3CCOC3)=O)CC2c2ccncc2)=O)cc(C)n1 CCC(C(=O)NC1CCC1NC(c1n[nH]c(C)c1C)=O)C(C)(C)CC N1(C(c2n(CC)ccc2)=O)CCC(C)C(CNC(=O)C(F)=C(C)C)C1 C#Cc1cnn(C)c1C(N1CCC(F)(C(=O)NCCC(=O)N2CCCC2)C1)=O C(S(=O)CC(O)CC(=O)Nc1cnc(Br)c(Br)c1)c1ccn(C)n1 N1(C(C(c2ccc(F)c(F)c2)C)=O)CC2(CCN(C(c3ccc[nH]3)=O)CC2)C1 c1(C(=O)NC2CCN(C(c3n(CC)cnn3)=O)CC2)ccc2c(c1)CCN2 C(N=c1[nH]c(N2C3CCC2CC(CO)C3)nc2cc(C)ccc12)c1occ(C)c1 Cc1noc(-c2ccc(Br)cc2)c1C(=O)NC1CN(S(=O)(=O)C(F)(F)F)CC1F N1(C(c2nc(C)[nH]c2C(F)(F)F)=O)CCN(C(=O)C(O)CF)CC1C C1(CNC(CCOC)=O)CCCC2(CCN(C(C3(C#N)CC4CC4C3)=O)CC2)O1 c1(C(N2CC(CC)C(NC(c3ccn(CC)n3)=O)CC2)=O)onc2c1CCCC2 CN1CCC(NC(c2[nH]ccc2CNC(=O)C=CCO)=O)C(C)(C)C1 Cc1cc(C(N2CCCC(NC(=O)C(CN(C)C)N(C)C)C2)=O)ccc1O N1(C(Cc2cc(C)no2)=O)CC2CC(NC(c3cnc(C(C)(F)F)s3)=O)C1C2 C=CCCCCCCC(=O)N1CC(C)(NC(C2CNC(=O)C(C)(C)C2)=O)C1 N1(C(CCOCC#C)=O)CC2CC1C2NC(c1cc(Br)c(C)o1)=O N1(C(c2nc(OCC)oc2)=O)CC2CCC(N(C)C(C3CCCOC3)=O)C2C1 CCC(C)CC(CC)(c1nnnn1-c1ccc(OC)cc1)Nc1csnc1OC C1(C(=O)NC2CCC(NC(c3cc(C4CC4)ns3)=O)CC2)SC2C=CC1CC2 C(=O)(C(F)CCC(C)C)NC1C2CC(C(=O)NC3CCCC(C=C)C3)C(C2)C1 N1(CC(=O)NCC2CCN2C(=O)C)C(=O)C2CC=CCC2C1=O.C1CC1.S C1(C(=O)NCc2nccc(CC)c2)CCN(C(=O)C(O)C(F)(F)F)C(C)C1 c1(C(=O)N)cn(C)nc1-c1ccccc1.C1(C(=O)NCCC)(COC)CC1 c1(C(=O)NC2C(NC(C(CC)O)=O)C2)cc2cc([N+](=O)[O-])ccc2n1C C#Cc1cncc(NC(c2ccc(CNC(=O)Cc3cncs3)cc2)=O)c1 C(=O)(C(F)(F)C(O)c1ccccc1)NCC1(C)N(C(C(C)(C)SC)=O)CCC1 Cc1nc(N(C)C)sc1C(=O)NC(C(C)NC(C1CCC=CO1)=O)C(C)C CCC1=C(C(=O)N2CCC(F)(CNC(=O)CC3CCCC3(F)F)C2)CCCO1 c1(C(N2CCC(OC)(CNC(c3cccs3)=O)C2)=O)cc(N)cc(O)c1C S(=O)(=O)(c1ccc(C(=O)Nc2ccc3c(n2)CCC3)cc1)N1CCCC(C#N)C1 N1(C(C(=O)NC(C2CCCOC2)COC)=O)CCCc2c(cnn2C)C1 C1(C(=O)NC2CCN(C(C3CN(C(N)=O)C3)=O)CC2)CCCCC(F)(F)C1 O=S(=O)(c1ccc(=NCCOCCO)[nH]c1)NC1CC2C=CC1C2 c1(CCC)c(C(N2CC(CC(C)NC(c3cn[nH]c3)=O)C2)=O)nnn1C c1(C(=O)NCCC2CCC(NC(C(F)OC)=O)C2)cccc2ccn(C)c12 c1(N2C(C(=O)NCC3(C)CC3)CC(O)C2)ncc2[nH]cc(I)c2n1 C1(C(N2CCN(C(C(C=C)c3ccccc3)=O)C(C)C2)=O)CC(=O)CC12CCC2 Cc1cccn2nc(C(N3CCC(NC(=O)Cn4cncn4)C(CO)C3)=O)cc12 c1(C(N2CC(OC)C(NC(C)=O)C2)=O)csc2cc(C)ccc12 c1(C(=O)NC2CN(C(=O)CCOCC(F)F)CCC2F)ccnc2ccncc12 N1(C(C(COC)COC)=O)CC2(CCC2NC(=O)C=Cc2ccccn2)C1 N1(C(C2(CC=C)CN(C(=O)CCSC)C2)=O)CCN2C(=O)OCC2C1 O=C(CC(CNC(C1(O)CCOCC1)=O)C1CCC1)N1CC2CC2(CO)C1 C1(NC(c2cc(COC)no2)=O)CC2CCC1C2.N1(CC=O)CSCC1=O.C CCCCC(C)C(=O)N1CC(O)(CN(C)C(c2cc(O)ccc2C)=O)C1 C1(C(=O)NCC(C)(C)CC2CN(C(=O)C(=O)N)C2)CCCCCC1.C1CC1 C(=O)CC(C)C(F)F.C1CCCCC1.C(=O)(C(=O)N)NCCOCCOC c1(C(=O)NC2C(C)CN(C(c3cnc(S)[nH]3)=O)C2)ccc2c(c1)COC2=O c1(C(=O)NC(CN(C(c2c(C)ncs2)=O)C)C)cccc(C(F)(F)F)c1N C(=O)(C1=CCC(NC(=O)CCc2ccncc2)C1)N(CC(CC)(C)OC)C N1(C(Cc2c(C)cccn2)=O)CC2CCN(C(C34CCC(F)C3CC4)=O)CC12 N1(C(c2c(CCC)cccc2)=O)CCN(C(=O)C2=CC(C)(CC)C2)CC(C)(C)C1 N1(C(Cn2c(C)cc(C)n2)=O)CCC(NC(C2CC(n3ccnn3)C2)=O)C12CC2 c1(C(=O)NC2(C#N)CCN(C(=O)CN3CCOCC3)C2)ccc2cccnc2c1 C1(C(=O)Nc2ccc(N3CCC(C)C3)cc2)CC12CC(C)(C)C2 C(=O)(C#CC1CCCOC1)N1CCC(C)CC1.C1(C(N(C)C)=O)(C(=O)NC)CC1 c1(C(N2CC(NC(C(CC)CCOC)=O)C(F)CC2)=O)ccnc2ccnn12 c1(C(=O)NCC2(O)CCN(C(C3(C)COCCO3)=O)C2)ccc(F)cc1F C(=O)(C(C)C(=O)N1CCC1CC(=O)Nc1cnn(CC(C)C)c1)OC Cc1ccc(C2(C(=O)N)CC2)cc1.c1(C(N2CC(CCC)C2)=O)c(C)nsc1C C1(C)CCN(C(=O)C(C)(C)C2CCCCO2)C1.CCS(=O)(=O)NC(C)C(=O)N N1(C(CCCC=C)=O)CC2(CCN(C(=O)C(c3cccc(O)c3)C)CC2)CC1C c1(COC)cccc(CC(=O)NCC2CC(C)N(C(=O)CCC#N)C2)c1 CC1=C(C(=O)NCC2COCCN(C(=O)CC(C)F)C2)CCS1(=O)=O C(=O)(C(CNC(=O)CN=[N+]=[N-])CC1CCCC1)N(C(C1(C)CC1)C)C C(CC(C)(C)C(=O)NCCC(C)C(F)(F)F)NC(C1CC(O)(CC#C)C1)=O N1(C(CCC2CCN(C(c3ccoc3)=O)CC2)=O)CC2CC(CO)C(C2)C1 C1(NC(C2CCC(C)(C)OC2)=O)CCCCCCC1NC(=O)C=Cc1cnc[nH]1 N1(C(C2C(NC(CCCN(C)C)=O)CCOC2)=O)CCc2ncccc2C1 C1(c2ccon2)(CC=O)CS(=O)(=O)C1.C1(C)CC1C(=O)N(CCCC)C N1(C(C(C)Cn2ccnc2)=O)CC2CC2(CNC(=O)C(c2cccn2C)=O)C1 C1(C)(C(=O)N)CC(C)(C)C1.C1(CC)CCN(C(=O)CC2CCCC(O)C2)CC1 C1(Nc2cc(NCc3n(C)nnc3)ncn2)C2Cc3cc(F)ccc3C12 C(=O)(C1=CCC(C)(C)CC1)N1CCCCC(NC(CC(CCC)C)=O)C1 N1(C2CCN(C(C(F)=C(C)C)=O)C2)CCN(C(C2CC2C2CC2)=O)CC1 N1(C(Cn2c(C)nc(C)n2)=O)CCN(C(=O)COc2cc(F)cc(F)c2)CC1C c1(N2CCCC(NC(C(CC)CC3CCCC3)=O)CC2)ncc([N+](=O)[O-])c(C)n1 CC1CC(C(=O)NC2CCC(NC(=O)COc3cn[nH]c3)C2)Cc2nn[nH]c21 N1(C(CC2(C#N)CC2)=O)CCCC2(CCC(NC(c3coc(C(N)=O)c3)=O)C2)C1 N1(C(CSCC(=O)OC)=O)CCn2ncc(C)c2C1.C1(C(=O)N)COCCN1C Cc1ccc2[nH]c(C(N3CCN(C(C4CCS(=O)(=O)N4)=O)C(C)C3)=O)cc2c1 c1(C(=O)NCC(C)NC(c2cn(C)nc2Br)=O)cc(F)cc2c1NCCC2 c1(CNC(CONC(c2[nH]cc(C)c2)=O)=O)cc(C)c(C)o1 C1(C(N(C)C)=O)CCN(N2CCCN(Cc3cscn3)CC2)C1 Cc1ccc(C(C)C(N2CCN(Cc3cc(C)on3)CC2)=O)cc1 N1(C(CC2CC(OC)C2)=O)CC=CC1(C(=O)N)COC.c1cnn(C)c1.C N1(C(CC2CN(C(C(CC=C)CC)=O)C(C)(C)C2)=O)CCn2cnnc2C1 C1(NC(=O)CC2(CNC(=O)C(C3CCOCC3)F)CC2)COC(C2CC2)C1 c1(OC)csc(C(N2CCC(N(C)C(c3cnn(C)c3N)=O)C2)=O)c1OC c1(SCC(=O)NC2CC(C)CN(C(C3C4COCC34)=O)C2)ccccc1[N+](=O)[O-] C1(C(N(CCOC)C)=O)CC1C1CN(C(c2ncc(C)cc2F)=O)C1 CC1CC(NC(=O)CCc2cnc[nH]2)CC(C)C1.C(c1cn(C)cn1)=CC=O.N C1(C(=O)NCC(C)(C)CNC(=O)CCc2ccsc2)CCCC12OCCO2 C(=O)(C(O)C1=CCCCC1)N1CC(C)(C)C(C(N2CCC3CCCC3CC2)=O)CC1 C1(C(N2C(CNC(c3cc(C)c(Cl)s3)=O)CC(O)C2)=O)CNC(=O)C(C)(C)C1 C(=O)(C1CCc2nccn21)N1CCC(C)(C(=O)NCC2(F)CCC2)CC1 O=[N+]([O-])c1ccc2[nH]nc(CN3CC(NS(=O)(=O)c4cc(F)ccc4F)C3)c2c1 c1(NC(c2ccc(-c3c(C)nccc3)cn2)=O)cc(Cl)c(O)c(Cl)c1 O=C(C1CCCn2ccnc21)NCC1CCCCN1C(c1ccc(O)cc1F)=O C1(C(=O)NC(c2ccccn2)COC)Cc2cscc2C1 CC(C#N)CCC(=O)NCC1CCN(C(C2CCCN(C)C2)=O)CC1 C1(OC)CCCC(C(=O)NC2(CCCNC(=O)CCn3ccnc3C)CC2)C1 c1(C(NNC(=O)NCCC(=O)NCCC(=O)OC)=O)cc(Cl)ccc1Cl c1(C(=O)NCCN(C2CCC(C)C2)C)cccc(-c2nn[nH]n2)n1 Cc1cccc(C(N2CCC(C(C)C(N3CCC(C)(C)CC3)=O)C2)=O)c1F C(=O)(C1CSc2ccccc21)NC(C(C)C)CNC(c1nnc(O)cc1O)=O C1(C(=O)NCC2C(C(N3CC(C)SCC3)=O)CCCC2)CCCCCN1C CCC(C)(C(=O)NCC1C2CC1N(C(=O)CC(O)C(C)C)C2)C(N)=O C1(CNC(=O)CCCc2nccs2)CN(C(C2CC(O)C2)=O)C2CCCCC12 C(=O)(CN=S(C)(C)=O)NCC(C1CCN(C(c2sc(C)c(O)n2)=O)CC1)C C(COc1ccccc1)(C(=O)NC1CC1)OC.C1(C=O)CN(C(C)=O)C1 Cc1c(C(=O)NCCCCCCNC(C2(O)CC2(C)C)=O)ccn1C1CC1 C#Cc1c[nH]nc1C(=O)NC1CCCC1C(=O)N(C(C)CC#C)C C1(C(=O)NC2CC(C(C)(C)C)C2)C2CN(C(c3ccc(CO)nc3)=O)CC12 O=C1Nc2ncc(Br)cc2C12CCC(NCc1nnc3n1CCOC3)CC2 CCC(F)(C(=O)OC)C(=O)NCCCCCN(C)C(c1cnc2c[nH]nc2c1)=O c1(OC)cnc(Cl)c(NC(C2(C)CCN(Cc3cc(F)cc(Cl)c3)C2)=O)c1 C1(C#N)(CN(C(=O)Nc2nc(-c3cccc(OC)c3)no2)CC)CCOCC1 C12(C(N3CC4C(CN(C(C#CC(C)C)=O)C)C4C3)=O)CC3CC1C2C3(F)F N1(C(CCC(=C)C)=O)CCCC(C)C1CNC(=O)Cn1cc(CC)cn1 c1(C(=O)OC)cccc(C(=O)NC(C)(CNC(c2ccccn2)=O)CO)c1 Cc1cc2cc(C(=O)NCC(C(C)C(C)C)NC(c3ccoc3)=O)c(Cl)cc2[nH]1 Cc1cn2cc(C(=O)NCCNC(C3(C)CCOC(C)C3)=O)sc2n1 CC(C)(C)CCC(=O)NCC1CN(C(C2CCCN2C2CCCC2)=O)CCCO1 O=[N+]([O-])c1cc(Br)ccc1CNCCc1ccc(Br)c(Cl)c1 C1(CC=O)CC(=O)NC(=O)C1.CC1(C(=O)NC2CCC(CC)C2)CCCO1.N C1(NC(c2c(C)nc(CC)s2)=O)CCNC(C)C1.c1ccc(C(F)(F)F)cc1.C c1(C=O)cn(-c2cccc(F)c2)nc1C.C(C)(C(=O)N(CCC)C(C)C)OC.N C1(OCC)(CNC(=O)N)CCCS(=O)(=O)C1.C1(C)CCCC(F)(F)C1 c1(C(=O)NCC2(F)CCCN(C(C3OCCN(C)C3)=O)C2)c(F)cc(Cl)cc1F CON1CCC(C(=O)NC2CCCCN(C(c3ccc(F)c(CO)c3)=O)C2)CC1 CCCCC#CC(C)(C)NC(=O)C(C1CCOC1)NC(c1n[nH]cc1Cl)=O C1(C(N(CC(C)O)C(C)C)=O)CC(C23CC(C2)C3)CN1.c1(CC)ccccc1 N1(C(c2c(C)nc[nH]2)=O)CCC2(CCCN(C(c3cccc(=O)n3O)=O)C2)C1 C1(N(CC(=O)N(CCCC)CCCC)C)CCN(CC2CCC2)C1 c1(C(=O)NC2C(NC(C(c3cccc(C)c3)O)=O)C2)cnn2c(C)ccnc12 C1(COC)(C)CCCN1C(=O)CC1CC(C)(C)C1.c1(C=O)cccnn1.N C1(C(=O)NC2C(C(N3CC(OC)C3)=O)COC2)CC2CCC1C2 C(=O)(CC(O)(CCC)CCC)N1CC(CNC(C2(CC=C)CCC2)=O)N(C)CC1 C1(C(=O)NCCc2cc(C(=O)N)no2)(OC)CC(C)C1.CC=O.C(C)C N1(CCC(=O)N)C(=O)CCC1=O.C1(OC)(OC)CCC1C(=O)NC1CC1 C(=O)(N=c1[nH][nH]cc1C)c1cc(OC)c(-c2ccc(C(F)(F)F)cn2)nc1 C1(CNC(C(C(CC)C)O)=O)CN(C(=O)CC(C)(C)C)CCC12CCOCC2 c1(OC)cccc(C(N2CCC(CNC(c3cc(CO)n(C)n3)=O)CC2)=O)n1 CC(C)C(C)CC(=O)NC(C1CCN(C(C2(Br)CC2)=O)CC1)C(C)C C(=O)(C(CC1CCCC1)OC)NCC(CN(C(COCCCCC)=O)C)C C(C)(C(=O)NCC1(CN(C(=O)CSC(F)F)C)CC1)(C1CC1)OC C1(N(C(=O)CCc2ccccc2)C)CCCCC1S(C)(=O)=O Cc1c(CCNC(=O)NC(C(C)(C)C)C(F)(F)F)ccc(Cl)c1Cl C12(COC(c3cc(C(F)(F)F)cc(C4CC4)c3)=O)COCC1C2(F)F N1(CCC(C)F)CCCOC(CNC(c2ccccc2Cl)=O)C1 C(=O)(C1=C(C2CCC2)N(CCC(C)C)C(=S)NC1c1ccc(Cl)cc1Br)OC N(C(=NCC(C)CC(C)C)N1CCN2C(=O)CCC2C1)C(CC)CC c1(C(=O)NC2CCN(C(c3cnc(O)s3)=O)C2)cncc2ccsc12 c1(N2C(CCNC(=O)C(C3CCCCC3)O)CCCC2)ncc([N+](=O)[O-])cc1Cl O=S(=O)(c1ccc(NCC2(CCO)CC2)cc1Br)NC1(CC2CC2)CC1 N1(C(c2ccc(C)[nH]2)=O)CC2(C(N3CC(O)CC3CO)=O)CCC1CC2 c1(CCC(=O)N(C2CN(C(C=CCC)=O)CC23CC3)C)ccc(F)c(F)c1F C(=O)(C(C(=O)NCC(=O)NCC(=O)N(C1CC(S)C1(C)C)C)OC)OC c1(OC)ccc(C2CC2CC(=O)NC2CCC2)cc1.C(=O)CCC1CCCC1.N CC(C)C(O)C(C)C(=O)N1CC(NC(=O)C=C(Cl)Cl)CC(C)C1 C1(CCC(=O)NCC2CCN(C(=O)CCc3ccoc3)C2)NC(=O)NC1=O C1(N(C(C(C)N=[N+]=[N-])=O)C)CN(C(c2ncn3c2CCC3)=O)CC12CC2 C1(C(=O)NCC(C)NC(C23CCC(F)(CC2)C3)=O)OCCOC12CCC2 c1(NC)cc(-c2cccc(C(N3CCCCC3C(N)=O)=O)c2)cc(F)c1 N1(C(C2C(C)(C)N(C(c3ncncc3Cl)=O)CC2)=O)CC2COCC2(C)C1 c1(C(=O)OCC(C)(C)OC(C)=O)nc(-c2ccccn2)n(-c2ccccc2C)n1 C1(C(N(C)CCNC(=O)CCNC(=O)CO)=O)CCOC(c2ccccc2)O1 N1(C(CC)C)CCC(NC(=O)Nc2cc(-c3ccco3)nn2C)CC1 C1(O)(CNC(CSCCOC)=O)CCN(C(=O)C(C)(C)O)C1.C(C)C c1(C(C(N2CC(CC=C)(NC(=O)CC(C)CF)C2)=O)C)cc(F)cc(F)c1 Cc1cc(C(=O)N(CC(C)CNC(c2c(C)nsc2C)=O)C)c2cnn(C)c2n1 c1(CC)ncncc1C(=O)NCCC1COCCN1C(C1CC(F)(F)CS1)=O Cc1cncnc1C(=O)NC1CN(C(=O)CC2CC=CCC2)CC1O c1(C(N2C(CNC(C3C(C)C3)=O)CCC2)=O)ccc2c(c1)CC(C)O2 CCCC(CC)CC(=O)N1CCC2(NC(C3CCCC4(CC4)C3)=O)CCCC12 C1(CNC(c2c(C)onc2Br)=O)CN(C(C2CCC(O)CC2)=O)CCN1C C1(C(=O)NC2(CNC(c3c(N)cccn3)=O)CC2)CC2(CCC2O)C1 N1(C(CCc2c(C)ncs2)=O)CCN(C(=O)CCOC2CCOC2)CCC1C C1(C(=O)NCCOC(=N)O)CCC(O)CN1C(c1ncn2c1CCC2)=O Cc1cc(NC(=O)C(Cc2cc[nH]n2)NC(=O)CCOCC(F)F)ccc1Cl CC1(C(=O)NC2CNC(=O)OC2)CC(O)CN1C(c1cc(C#N)c[nH]1)=O Cc1oncc1C(=O)OC(C)C(=O)Nc1n[nH]cc1C1CC1 c1(C(=O)N)cn2nc(C)sc2n1.C1(C)(CC(=O)N(CCC)CC)CC1(F)F N(C(=NCCc1ccc(Cl)cc1Cl)N1CCC2(C)C(C1)C2(Cl)Cl)CCOCC=C C1(CNC(c2cscn2)=O)CC2(CC2)CN1C(C1CCC2(CCC2)C1)=O C1(C)(CNC(C2C(C)CCCC2)=O)CCN(C(=O)C(F)(F)c2cncs2)CC1 c1(C(=O)NC2CN(C(C3CCC(C(F)(F)F)CC3)=O)CC2O)ncc(Br)cc1F c1(SCC)cccc(CC(=O)NC2CCCC(C)C2)c1.c1(C=O)csc(=N)[nH]1 N1(C(C(CCCC)O)=O)CCC(C2CCN(C(=O)C(CC)OCC)CC2)C1 C=C(C)C(C)(O)C(=O)N1CC(CNC(=O)C(C)NC(=O)OC)C1 Cc1cc(C(=O)NCC(CC(C)C)NC(=O)Cc2ccsn2)c(C)n1NC(N)=O Cc1cc(C(=O)N(C2CCC(NC(c3ccc(N)cn3)=O)C2)C)nc(C)c1 CCC(CC(=O)N(C)CC1(O)CN(C(=O)C(C2CCC(O)CC2)(C)C)C1)C1CC1 CC1CN(C(C2(CO)CCOCC2)=O)CC(C)CN1C(=O)CC1COC(=O)N1 C1(C(=O)NC(CCNC(c2c(C)ccnc2)=O)C)CCCCNC1=O C(=O)(C1=CCCC1C)NC(C1(C(=O)NC2C(C)COCC2)CC1)C C(=O)(C(C(C)CC)c1ccccc1)NCCOCCCN(C(C=CCC)=O)C c1(C(N2CCSC3CCC23)C(=O)NCCC)cccc(Br)c1Cl C1(CNC(CCC=CC)=O)CCC12CCN(C(c1ccnn1CC(F)F)=O)CC2 c1(C=O)ccc(S(N)(=O)=O)s1.Cc1noc(C(=O)NC2CCC2(C)C)c1C.C c1(OC)cc(F)ccc1C(=O)NC1CC1C(=O)NCCc1cccc(Br)c1 Cc1ccc2c(CC(N3CC(NC(c4scnc4Cl)=O)C4(CC4)C3)=O)c[nH]c2c1 CCC(C)C(=O)N(C(C)(C(=O)NCCOCC1CC1)OC)C CCCC(O)CC(=O)N1CCN(C(=O)C=Cc2ccccc2)C(CC)C1 C1(CC)CN(C(=O)COC(F)(F)F)CC(C)O1.c1(C(C)C)ncc(C(=O)N)cn1 C=CCC(C)(C)C(=O)NC(CC(=O)NCC(O)CC(C)(C)C)C1CC1 c1(C(=O)NCC=CCNC(CCCOCC=C)=O)cnn(C2CCC2)c1C C1(NC(c2cc(CCC)on2)=O)(CNC(=O)C(C)C#N)CCCCC1 C1(CC)(NC(c2cccc(C(N)=O)n2)=O)CCCN(C(C2(SC)CCC2)=O)C1 c1(C(N2CCOCC2C2CCC2)=O)cccc(OC(F)F)c1F c1(C(=O)NCCCCNC(=O)CCc2ccc(Cl)nc2)cn2c(n1)SCC2 C=C(C)CC(C(=O)NC(CCN(C)C)C(=O)N(CC(C)(C)COC)C)OC c1(OC)cc(NC)nc(C(F)(F)F)n1.c1(C(N2CCC2)=O)ccc(C)c(F)c1 c1(C(C(=O)NCCNC(CC(CC)C)=O)=O)cc(Cl)cc(Cl)c1 C1(NC(CC(COC)C)=O)CC2CCC1CC2NC(c1ccc(F)c(C)c1N)=O c1(N(C(=O)NCCC2CC2C(F)(F)F)CC)ccc(Cl)cc1 N1(C(C(C2CCOC2)OC)=O)CCOC2(CCN(C(=O)C3=CCCS3)CC2)C1 c1(C(=O)NC2C(CC)N(C(=O)C(C3CC3)OC)CC2)cccc2ccoc12 c1(SCC)ccc(Cl)cc1C(=O)Nc1ccc(C2CCC2(C)C)cc1 C(=O)(CC(O)CNC(=O)CCOCC(F)F)N(CCC(C)(C)C)CC c12cccc(n1)OC(=O)C2(F)F.CCS(=O)(=O)N.C1CO1 N1(C(CCC#CC)=O)CC(F)(F)CC1CCNC(c1cc(C(F)F)cs1)=O C12(C=O)CCC(C)(C(=O)O1)C2(C)C.Cc1nccnc1C(N1CCC(C)C1)=O.N C1(N(C(C(n2cc(Cl)cn2)C)=O)C)CC2CC1N(C(c1cc(CF)on1)=O)C2 C1(C(=O)NCC2(C)CCN(C(c3cc[n+]([O-])cc3)=O)C2)Cc2cc(F)ccc2O1 C1(NC(C(C)(C)C2CCCCC2)=O)CCCN(C(=O)C=CC2CC2)C1 C(CCC(C)CO)NC(C(c1cccnc1)NC(C(C)C#N)=O)=O c1(NCC2C(C)C2)ncc(C(F)(F)F)cc1Cl N1(C(C(N2CCCCCC2)C)=O)CCN(C(=O)Oc2cc[n+]([O-])cc2)CC1 c1(C(=O)OCC2CCC(C(CC)(C)C)CC2)ccc(F)cc1C(=O)N(C)CC N1(C(C(F)=CC)=O)CCCC2(CCN(C(c3cnc4c(=O)[nH]ccc4c3)=O)C2)C1 c1(CC)nc(C)c(C(=O)NC(C)CCC)c(C)n1.C12(C=O)CCC(CC1)C2.N CC1CCCC(CC(=O)NC2CCCCC2CNC(c2ccc(CO)o2)=O)C1 Cc1cc(-c2ccccc2)nc(N2CCC(NC(C3CCCSC3)=O)CC2)n1 c1(C(C)=O)ccsc1C(=O)NC1CCC1.c1(C2C(C)(C=O)C2)ccccc1.N C#Cc1ccc(CCN(C)CC2COC(C)(C)O2)cc1 C1(NC(CCCCN(C)C)=O)CC2CCC(C1)N2C(C1CCCCN(C)C1=O)=O C=CC(C)(C)C(=O)NCC(C)CNC(=O)CC1CCC(=O)N1CC c1(N2CC3(OCC(C)C3)C2)cc(Br)ccc1S(=O)(=O)N1Cc2ccc(Cl)cc2C1 N1(C(C2N(C(=O)C(CC)CCC)CCC(=C)C2)=O)C2CCC1CN(C)C2 N1(C(C2(CN(C)C)CC2)=O)CC(NC(C2(C)COC(=O)C2)=O)CC1(C)C N1(C(C2C(C(=O)OCC)C2)=O)Cc2[nH]nc(C(N3CCCC(O)C3C)=O)c2C1 c1(OCC(=O)NCCC(C)C)ccc(O)cc1.C(C1CCOC1)=CC(=O)N c1(OC)ccc(C2(C(=O)NC3CC(C)C3)CCCC2)cc1.C1(C(=O)N)CSC1 CC(C)CCCC(C)C(=O)N1CCC(C(=O)Nn2cnnc2)O1 C1(CC)CN(C(c2cc(F)ccc2OC)=O)CCN1C(=O)C=Cc1cnccn1 c1(NC(c2c(OC(C)C)scn2)=O)ccc(N(C)C)nc1 C(CCO)(C(C)(C)O)NC(c1c(C)ncn1O)=O c1(CC(=O)NCCN(C(c2c(Cl)cnn2C)=O)CC)ccc2nc[nH]c2c1.C N1(C(C(CC)OCC)=O)CC2(CCC2NC(c2[nH]cnc2CC)=O)C1 Nc1cc2c(cc1C(=O)NCCCCNC(=O)Cc1ccns1)CCCC2 c1(C(=O)NC(C)CC2CN(C(C3CCCN3C=O)=O)C2)ncn2c1CCC2 c1(C(=O)NC23CC(CNC(C(C)c4ccsc4)=O)(C2)C3)ccncc1Cl C1(CNC(c2ncc(Cl)s2)=O)CN(C(c2cnccn2)=O)CCO1 c1(C(=O)NC2C(C)CN(C(c3c(Cl)cnn3C)=O)C2)ccc2c(C#N)c[nH]c2c1 CCCCC(O)CNC(=O)C(C)N(C(=O)C(O)CC)C1CC1 C1(CCC)CN(C(=O)C(C)CSC)CCN1C(=O)CSc1ccc(OC)cc1 N1(C(C2C(OCC)C2)=O)CCC(C(F)(F)F)CC1.CC(C)(C)C.C(=O)C O=C(C1=CCOCC1)NCCC1CCN(C(C2CC2c2ccsc2)=O)C1 C(C(C(=O)NC1(c2ccsc2)CC1)n1cc(C2(n3ccnc3)CC2)nn1)SC C1(NC(c2cc(CSC)c(C)s2)=O)(CO)CCN(C(c2cnsn2)=O)CC1 C(C)(CN=C(NCc1cnc(-c2ccccc2)o1)NC1CC1)OC Cc1cc(Br)cc(S(=O)(=O)N2CCNC(C(N3CCC4(CC3)CC4(F)F)=O)C2)c1 C(C(O)C(=O)N1CC(NC(c2c[nH]nc2-c2ccncc2)=O)C1)=CCCC N1(C(C(CC)OCC)=O)CCCC(C(=O)Nc2ccc(C)nc2CC)CC1 C(=O)(C(O)C(F)(F)c1ccccc1)N1CCC(O)C1.C#CCCOCC(=O)N.C C1(CC(=O)O)(COC(CCC=C(C)C)=O)CCCN(C(=O)O)C1.C(C)(C)C C1(O)(C(CNC(C2(SC)CC2)=O)C)CCN(C(c2snc(C)c2N)=O)C1 C=CC1(CO)CCN(C(c2cncn2-c2cccnc2)=O)CC1 C(C(CC(C)C)NC(C1CCC=CO1)=O)NC(c1c(OC)nsc1)=O C1(CC(=O)NCc2ncc(CC)s2)CN(C(C2CN(C)C2)=O)CC1C C1(C(=O)NC2(C)CCN(C(c3c(C)n(C)cc3)=O)CC2)CCCC2(CCC2)C1 C=CC(CC)CC(=O)NNC(=O)CNS(=O)(=O)c1ccc(Cl)cc1 c1(C(N2C(CNC(CC=C)=O)CC2)=O)[nH]cnc1C(C)=O c1(OC)cncc(C(=O)NCC(C)(C)NC(=O)Cc2ccn(C)n2)c1 c1(CC(N2CC3C(C3)C2)=O)cc(F)cc(Cl)c1.c1(C(=O)N)coc(C(F)F)c1 N1(S(c2ncn(C)c2)(=O)=O)CCC2C(CCN2C(c2nc(C(=O)O)cs2)=O)C1 c1(C(=O)N)cnn2c(=O)cc[nH]c12.C1(C=O)C(F)(F)C12CC2.CCC1CC1 c1(N(CCCCC=C)C)nc2cccnc2c(=NCC2N(C)CCCC2(C)C)[nH]1 CN1CC2CCC1C(NC(=O)C(F)(F)CCn1cc(CC(=O)O)nn1)C2 N1(C(CN(C(=O)COCCCN=[N+]=[N-])C(C)C)=O)CCOCC(C2CC2)C1 c1(C(=O)N)cc2c(nc1N)CCC2.CC(C(=O)NCC1C=CCC1)P(C)(C)=O c1(CC(=O)NC23CCC2CN(C(=O)C(=O)NCC(F)F)C3)ccccc1[N+](=O)[O-] C(C1=CCN(C)CC1)N1CCN(CCC(C)C(F)F)CC1 CC(CC(=O)NC1(C)CN(C(=O)CCc2cccc(F)c2)C1)C(C)(C)C N1(C(CCNC(COC)=O)=O)C(C(=O)N(CCC(C)O)C)CCC1C(C)C C#CCC(CC#C)NC(=O)CN(C1CCC1)C(C1CC2CCC2C1)=O CC(CC(N)=O)C(=O)N(C(C)CNC(c1ccnc(F)c1Cl)=O)C Cc1onc(Br)c1C(=O)NC(CNC(=O)CCC1CC1)C(C)C.C1CC1 N1(C(C=CCC)=O)CC(CNC(c2c[nH]nc2C(C)C)=O)C2CC12 C1(CCC(N2CCC(OCCO)C2)=O)CCN(C(=O)CC2CC2)CC1 C#Cc1cccc(C(=O)NC2CC(C)(NC(=O)CCCc3ccncc3)C2)c1Cl N1(C(c2csc(O)n2)=O)CCCN(CC(F)(F)F)CC1 CN1CCCC(F)(C(N2CC(CNC(=O)CC(O)c3ccccc3)C2)=O)C1 Cc1ccc(C)c(C(N2CCCN(C(=O)C(O)CC3CCOCC3)CC2)=O)c1 C1(CCNC(C(C2CCOC2)OC)=O)CCCN(C(=O)CCn2cncn2)CC1 C(=O)(C1=CCCCC1C)NCC=CCNC(c1c(C)cco1)=O c1(OC)cc(F)ccc1C(=O)N(CC(C)C)C.c1(C(C(=O)N)C)c(C)n[nH]c1C n1(CC(=O)NC2(C3N(C(C(C)C4CCC4)=O)CCC3)CC2)cc2ccccc2n1 C1(C(N2CCCCC2C)=O)CCCC2C1C2(F)F.C1(OCC)CC(CC(=O)N)C1 C1(C(F)F)(CNC(Cc2n(C)ccn2)=O)CCN(C(c2cn[nH]c2)=O)C1 CCC1=C(C(=O)NCCCC(=O)NC(C)(CC)C2CC2)CCCO1 c1(C(N2CCCC(C)(NC(=O)COCC3CCCC3)C2)=O)ccnc2cc[nH]c12 N1(C(CCC=C)=O)CCC(C)C1c1cn(Cc2ccnc(OC)c2)nn1 C#CCC(C)C(=O)N1CCC(CNC(C2(F)CC2)=O)(OC)C1 C1(C)(C(=O)NCC(CCNC(c2c(CC)con2)=O)OC)CC(C)=NO1 C(=O)(C1CCCc2cccnc21)N1CCCCC(NC(C2=CC(C)(CC)C2)=O)C1 C#CC1CCCN(C(=O)C(C2(C)CC2)NC(c2ccc(C)nc2C)=O)C1 c1(C(C(=O)NC(C(C)NC(CCC(C)C)=O)(C)C)C)ccc(Cl)c(Cl)c1 N1(C(c2c(CC)nco2)=O)CC(F)(F)CC1CNC(=O)C(C)(CC)CC c1(C(=O)NCC(O)CNC(C2CCC2(F)F)=O)ccc(Cl)c(Cl)c1 c1(OC)ccc2cc(C(=O)N)cnc2c1.C1(C=O)CC(=O)N(O)C1.CC=CC C1(NC(c2n(CCC)ncc2)=O)CC2CC1CN2C(c1ccc(F)cc1F)=O C1(NC(=O)CC2COCCOC2)(CO)CCN(C(=O)C=CC=C(Cl)Cl)CC1 CCC(C)(C)CC(=O)N1CCC(NC(c2nc(Cl)ccc2N)=O)CC1C N1(C(C(C)OCC(C)C)=O)CC2CC1CN2CC(c1ccccc1)O C1(C(=O)NC2CCN(C(c3nc(C(C)C)oc3)=O)C23CC3)CCc2nnnn2C1 N1(C(C2C(C)OCCC2)=O)CCCN(C(=O)C(N2CCCC2)C2CC2)CC1 c1(CC(N2CCC(C(C)NC(C(C(=O)OC)C)=O)CC2)=O)c(C)n[nH]c1C.C c1(CC(=O)Nc2nc(C)sc2)cc(-c2cncc(CN(C)C)c2)ccn1 N1(C(C=C(C)C)=O)CCOC2(CCN(C(C3CCCS3(=O)=O)=O)C2)C1 c1(C(=O)N)ccc(Cl)nc1O.c1(C(=O)NCC2CCCCC2)ccc(F)c(O)c1 N1(C(CCC)=O)CCC2(NC(=O)C=Cc3ccccc3OC)CCCCCC12 N1(C(C(CCCCC)O)=O)CCC(NC(c2ccon2)=O)C12CCCC2 O=C(CN=c1cc[nH]cc1)NC1CC=C(C(=O)N2CC3(C2)CC3(F)F)C1 C1(NC(c2cc(O)ncn2)=O)CC2CN(C(C3CC4(C3)CC(O)C4)=O)CC12 c1(C(=O)NC(c2occ(C(N(CC(C)OC)C)=O)n2)C)ccc2cc[nH]c2c1 c1(OCC)cccc(CC(=O)N(CC(C)NC(c2cccs2)=O)C)c1.C1CC1 C1(NC(COCC(C)(C)C)=O)CN(C(=O)C(F)Cc2ccccc2)CCC1C N=c1nc2c(c[nH]1)CC(NC(=O)NC(c1ccc(F)c(Cl)c1)C(F)(F)F)CC2 c1(Cn2cc(CCCNCCC3CCC(=O)N3)nn2)ccc(O)nn1 c1(C(=O)NC(CN(C(C(CC)(C)C)=O)C)C)cnn2cc(C#N)cnc12 c1(CC(N2CCN(C(C(CCC)O)=O)C(C(F)F)C2)=O)cnc2c(C)cccn12 Cc1cc(Cl)c2ccc(C(=O)NC3CC(C(=O)NCC(C)O)C3)cc2n1 C(C1CCN(C(C2(SC)CC2)=O)CC1)=CC(=O)Nc1c(CC)noc1 N1(C(CCCC2C(C)C2)=O)C2CCC1(CNC(C1(O)CCSC1)=O)CC2 N1(C(C=Cc2n(CC)ncc2)=O)CCN(C(c2cc(O)cc(=O)o2)=O)C2CCC12 c1(CCC(=O)NC2CC(C(C(N)=O)C3CCC3)C23CCC3)ccc([N+](=O)[O-])cc1 c1(C(N(C(C)C)CCNC(=O)CC(C)F)=O)ccc(F)cc1 n1(CC(=O)NCCN(C(C(C)(C2CC2)OC)=O)C)sc2ccccc2c1=O C1CN(C(=O)CC2(O)CC2)C2(CCOCC2)C1.C1(CC(=O)N)CC(=O)NC1=O CC1C(C(=O)NCC2CC(NC(C3CCC(CO)CC3)=O)C2)=Cc2ccccc21 Cc1ccn(CCC=O)n1.c1(C(N(CCC)C(C)C)=O)cc(C(C)(C)C)n[nH]1.N C1(NC(=O)Cc2ncn3c2CCC3)CCN(C(C2(CO)CCCO2)=O)CC12CCC2 c1(CC)ccccc1OCCC=O.C1CCN(C(C2CCN2S(C)(=O)=O)=O)C1 c1(CNC(c2c(NCC)scn2)=O)c(Cl)cccc1[N+](=O)[O-] c1(CC(=O)NCC(CCNC(c2cnnc(C)c2)=O)OC)cc(C)ccc1F C(C#Cc1cn(Cc2cccc(F)c2)nn1)NC(c1ccc(F)c(Cl)c1F)=O C(C(C)(C)C#CC(=O)NC1CCCC1CN(C)C)NC(c1csc(C)c1C)=O C1(NC(c2n[nH]c(CC)c2Cl)=O)CCN(C(c2nc(Cl)sc2C)=O)CC1F N1(C(c2cc(N3C(CC)CCC3C)ncn2)=O)CCC2(CCOCC2)C1 c1(C(=O)NCC(CCC(C)C)(C)O)ccc(N)c2cnccc12 C1(NC(C(OC)OC)=O)C=CC(CC(=O)NCC2(CCO)CCCC2)C1 C1(C(NOCCOC)=O)CCCN(C(c2cc(C)sn2)=O)C1C c1(CC)cc(C(=O)NC(C2CCCN2C(=O)C(OC)OC)(C)C)cc(C)c1 c1(CC)nc(C)c(C(=O)NC2CC(C(=O)NC(C)CCO)C2)o1 CC1CN(C(=O)CN2CCC(O)CC2)CCCN1C(=O)CCc1cnccn1 C(C(=O)NC(CO)CCCO)(C(C)C)NC(COC(CC)CC)=O C1(C(=O)N)CC2CC1CC2O.C=CC1(C(=O)NCC2(C)CCOCC2)CCCC1 c1(CC(=O)N(CC(O)CNC(c2cn(CCO)nn2)=O)C)cc(Cl)n(C)n1 N1(c2n(CC(C(=O)NCC)(C)C)c(C(C)C)nn2)CCC(=O)N2CCCC12 C(=O)(C1=CCS(=O)(=O)C1)N.Cc1occc1CC(=O)N(C)CC1(C)CC1 c1(C(=O)NC(C2CCCN2C(C2CC3C(C2)C3(F)F)=O)C)ccn2cccc2c1 C(=O)(CC(O)CC(C)(C)C)NCC(C)CNC(c1cccc2cccnc12)=O C#CCC(O)C(=O)NC1CN(C(C2(C(N3CCOCC3)=O)CC2)=O)CC1SC N1(C(C2CC2c2ccsc2)=O)CCC2C(C1)CN2C(C1CC2(CCC2)C1)=O Cn1nc2c(c1C(=O)NCC1(C)CCN(C(c3cncc(Cl)c3)=O)C1)COCC2 C1(C(N2C3CN(c4ncnc(C)c4Br)C(C3)C2)=O)CCOC2(CCCCC2)C1 c1(C(=O)NCCOCC(=O)NC(C2CCCC2)C)ccsc1C#N CCC(C(=O)NCC(C1CCCC1)NC(=O)C1=CCOCC1)C(C)(C)CC O=C(C1=CC2C=CC(C1)C2)NCC1C2CN(C(C3CN4CCN3CC4)=O)CC12 CC1OCCN(C(c2ncccc2N)=O)C1C(=O)NCc1nncs1 CC1(C(=O)NC2C=CCN(C(=O)CCc3cc(Cl)cc(Cl)c3)C2)CC2(CCC2)C1 c1(N(CC)Cc2nc(F)ccc2F)ccc2nc(O)[nH]c2c1 C1(C(=O)NCC(CNC(c2scc(C)c2)=O)(C)F)CC(O)C(F)C1 C1(C(N2CC(C)(CC)C2)=O)CC2C=CC1N(C(=O)CCn1ccnc1)C2 C1(C(N2CC(CNC(C(CCC)=CCC)=O)C2)=O)CCS(=O)(=O)C(C)C1 c1(C(=O)NCC(C)CO)cc(P(C)(C)=O)ccn1.c1(C=O)ccoc1C1CC1 N1(C(c2cc(N)c(N)nc2)=O)CC2(CC(NC(=O)CC(F)F)c3nccn32)C1 c1(C(=O)NC(CC=C)CNC(=O)CCc2cc(OC)no2)cccc(F)c1N c1(OC)cc(C(=O)N(C2CCC(NC(c3oncc3C)=O)C2)C)on1 C1(NC(C2CC23CC3)=O)C=CCN(C(=O)C=CCF)C1 c1(C(=O)NCC(C)(C)NC(C2CC(C)SCC2)=O)nn2cccnc2c1Cl N1(C(c2cc(OCC)ncc2)=O)Cc2ccnn2CC(NC(c2cnco2)=O)C1 C1(C(N(C)CC2N(C(c3cc(C)ncc3)=O)CCCC2)=O)CCC(C)(C)CC1 C1(C(=O)NC(c2ccc(C(F)(F)F)cc2)C)CC2CC2N1.c1ccc(O)cc1.C C12(C(N(OC)CC3CC3)=O)CCC(CC1)N(C(c1cc(C)c(C)nn1)=O)C2 C1(NC(CCSCC)=O)CN(C(=O)CCO)CC1C1CC1.c1cc(C)cc(C)c1 c1(C(N2CC(CN3CCCC(N4CCOCC4)C3)C2)=O)c(O)cc(O)cc1O C(=O)(C1=CCCN(C(c2cc(C)cs2)=O)C1)NCc1onc(CC)n1 c1(C(=O)NC(CC)CN(C(=O)CC(=O)N(C)C)C)cc(Cl)c2ccncc2n1 c1(C(C)C)cnc2cc(C(=O)NCC(O)CNC(C3(CO)CCCO3)=O)[nH]c2c1 c1(C(=O)NCC(CNC(c2nnn(CC)c2C)=O)F)ccc(O)nc1Cl N1(C(C2(C=C)CCN(C(=O)C(=Cc3ccco3)C)C2)=O)CCC(OC)C(C)(C)C1 c1(OC)ccc2[nH]cc(C(N3CC4(CCN4S(=O)(=O)c4ccc(C)cc4)C3)=O)c2n1 C1(OC)CN(C(C2CCC(O)CN2C)=O)CCC1NC(C1C=CC=CC=C1)=O c1(OCC(=O)Nc2cc(C(C)C)cc(F)c2)c(Cl)cc(Cl)cc1Cl C=CC1CN(C(c2[nH]ccc2CNC(c2cnccn2)=O)=O)CCO1 C=CC1OCCCC1C(=O)NC(CNC(=O)C=CSc1ccccc1)CC(C)C c1(C(=O)NCC(C2CCC2)NC(=O)C(C2CCCCC2)O)ncc2[nH]ncc2n1 c1(C(=O)NCC2(C(C)(C)O)CN(C(=O)C)C2)cnc2cnccc2c1.C1CC1 N1(C(c2c(CC)nco2)=O)CC(C)CN(C(=O)C(C)SC)C(C)C1 C(=O)(C(CO)C(F)(F)F)NC(C1CN(C(C(C)OCc2ccccc2)=O)C1)C N1(C(C(C)NC(C)=O)=O)CC2(C(=O)NCC(C)(O)CN(C)C)CCC1CC2 CCC(C(=O)N1CC(CNC(=O)CC2CCC2)(SC)C1)Nc1nc(C)cs1 CC1(F)CN(C(=O)COc2cccc(F)c2)CCN(c2ncc([N+](=O)[O-])cn2)C1 N1(C(C)C)CCC(N(C)C(C2CCCN2C(C2CCCN2C2CC2)=O)=O)C1 C=C=C(C)CC(=O)N1CCCC1C(C)C.c1(CC=O)cc(C(F)(F)F)n(C)n1 C1(C(N(C)CCNC(c2nc[nH]c2C(C)(C)C)=O)=O)CSCN1C(N)=O c1(OC)cccc(CN2CCC(CC(=O)NCC3CNCCO3)C2)c1O N1(C(c2c(CC)nco2)C(=O)NCc2ccco2)CC(C(=O)OC)CC(C)C1 C1(C(=O)NCC(O)CC(=O)NC)(CC)CC(C)(C)C1.C1(C)CCC(=O)N1 c1(C(=O)NC2C(NC(c3cnc(OC)s3)=O)COCC2)cccc(OC)c1O n1(CC(=O)N(C)C)c(=N)[nH]c2cc(Br)ccc12.c12ccccc1CC2 C(CC(F)F)(C(=O)N1CCCCCC1C)N(C(c1c(C)nncc1)=O)C Cc1ccc(C=CC(=O)Nc2ccc(C(N3CCC(O)(CO)CC3)=O)nc2)cc1 c1(C(=O)NC(C)CNC(=O)C(O)C2CCC2)cnn2c1CCC2 C(CC(C)C(=O)N1CC2CC2C1C(=O)NCC1CN2CCC1C2)=CCC CC(C)(CCN=c1nc2c(c[nH]1)COC2)NC(c1cc(F)cc2nccnc12)=O c1(OC)cc(Br)cc2[nH]c(C(=O)NC(C)C(CO)NC(=O)C(C)O)cc12 CCCC(C)(C)C(=O)NC1CN(C(c2cc(F)cn2C)=O)CC1(F)F N1(C(CCS(CC)=O)=O)CCC2(CCOCC2C(N2CCN(C)C(=O)C2)=O)CC1 c1(CS(=O)(=O)N2CCC2Cc2nnc(C(F)(F)F)o2)ccccc1Cl C1(NC(CCCCC=CC)=O)CC2CCC(C1)N2C(C1CCCN1C=O)=O c1(CNc2c(C(C)(C)C)cccc2)c[nH]c2nccc(O)c12 c1(C(N2CCCC(C)C2CNC(C2(C#N)CCCC2)=O)=O)cccc2ncsc12 CCCC(C(=O)N1CCOC(CN(C(=O)Cc2cnnn2C)C)C1)OCC c1(C(=O)NC2CSC(C(F)(F)F)C2)ccc(Br)cc1 c1(C(=O)NCC2C(NC(c3c(C)ncnc3)=O)C2)coc2ccc(F)cc12 c1(SCC)ccc(CC(=O)NC2CCCC2O)cc1.C(C1CCCO1)=CC=O.N c1(C(=O)NC2C(NC(C3CCC(C(N)=O)O3)=O)CCC2)ccc(C2CC2)nc1 C(=O)(CCCC(=O)N1CCC(O)(CC)C1)OCC.c1(CC=O)cccc(C)c1.N Cc1cc(NC(=O)CC2CCCC2NC(C2(C)CCCCC2C)=O)cnc1Cl c1(OC)cc(C(=O)NC2CCCC2CC(N2CCCCC2C(C)C)=O)n(C)n1 C1(N(C(C(F)=CC)=O)C)CCCCN(C(=O)Cc2ccc(C)c(O)c2)C1 C(=O)(C(O)CCC(C)C)N(CC(=O)NCCc1cncn1C)CC CCC(C)C(C(=O)NCCC1CCC1)NC(C1CC(O)C(F)C1)=O c1(C(=O)NCCCCC2CN(C(C(C)O)=O)C2)cn2c(n1)CCC(C)C2 Cc1ccc(Cl)c(CN2CC(C(N3CCC(C#N)C3)=O)CC(F)(F)C2)c1F C1(NC(c2c(C(C)C)noc2)=O)CN(C(=O)CC2CCCCCC2)CC2CC12 C1(C)(NC(CCN(CCCCC)CCC)=O)CCN(C(=O)CC)C1.[SH](C)(=O)=O CCCC(C)(C)CC(=O)N(CC(C)(C)NC(c1cn(C(C)(C)C)cn1)=O)C CCC(CCC(=O)N1CC(C(C)(C)O)(CO)C1)NC(=O)C(F)(F)c1nccs1 N1(C(CSC(C)(C)C)=O)CCCC(C2CN(C(=O)Cc3ccccc3O)C2)C1 c1(C(=O)NC2CC(NC(c3cc(F)cs3)=O)C2)cccn2cnnc12 Nc1cccnc1C(=O)NC1CC1NC(c1ccc(Oc2ccccc2)cn1)=O Cc1nc(C2CC2)oc1C(=O)NC1CN(C(=O)CCN2CCCCCC2)CC1C N1(C(CC(COC)C)=O)CC2(C1)CN(C(=O)CCC(C)SC)C2 c1(OCC(C)C)ccc(CNC(C23CCC(CN)(C2)C3)=O)cc1 Cc1cc(C(=O)NC2C3CN(C(=O)C(C)c4cccs4)CC23)nn1C c1(NCC(CO)OCC)cc(Br)ccc1S(=O)(=O)NC1CCS(=O)(=O)C1 COn1cnc(C)c1C(=O)N(C)CCOCCC.C1(C(=O)N)CCC(C)NC1=O Cc1ncc(CCC(=O)NCC(CO)NC(C2CC(n3ccnn3)C2)=O)c(O)n1 CCCCCC(CC)C(=O)NC1(C(=O)NCCC(O)CCO)CC1C c1(NCC2C(CC)C2)[nH]c(=NCC2(C3CC3)CCCO2)nc2sccc12 c1(C(=O)NC2C(C(=O)OCC)CCC2)ccc(OC)cc1C(F)(F)F c1(C(N2CCC(C)CC2)C(=O)NCc2cccs2)sc([N+](=O)[O-])cc1Cl C1(N(C=O)Cc2sc(-c3ccccc3)cc2Br)CCC1C1CC1 CCCC(C)(O)C(=O)NCc1ccnc(C(N2CCCC(CC=CC)C2)=O)c1 c1(OC)cc(C(N2CCCC(NC(C3CCS3(=O)=O)=O)C2C)=O)cc(Cl)c1 C1(C(=O)NC2CN(C(=O)CCCC3CCCO3)CC23CC3)Cc2ccccc2O1 N1(C(CC(=O)NCC(F)(F)F)=O)CCC(NC(C2(O)CCOCC2)=O)C(CO)C1 CCC(CC(=O)NCc1cc(C(=O)NC(c2ccccc2)CF)on1)C(C)(C)C c1(CN2CCC(CNC(c3sccc3F)=O)C2)c[nH]c2nccc(Cl)c12 C1(NC(CSc2ccc(C)cc2)=O)CCCC12CCN(C(=O)CNS(N)(=O)=O)C2 c1(NC(N2CC(O)CC(NC(N)=O)C2)=O)cc(F)ccc1O.c1ccccc1.C c1(C(N2CCC(CNC(C(C=C)(F)F)=O)CC2)=O)c(Cl)sc(Cl)c1C C1(NC(C(CC#C)(C)NC(=O)CCc2conc2C)=O)CC2CC1CC21CC1 C(=O)C1=NNC(=O)CC1.N1(CC(=O)NCC2(C)CCC2)C(=O)CNC1=O.N c1(C(C(=O)NCc2ccccc2)N(C)Cc2nc(C)on2)n[nH]c(C)c1Br O=S(=O)(c1ccc(Br)c2nsnc12)N1CCC(O)(c2cnn[nH]2)C1 CC(C)C(C)(O)C(=O)NC1CC(F)CN(C(c2cc(C3CC3)n(C)n2)=O)C1 c1(C(N2CCC(C)C(NC(=O)C(=O)NCC(F)F)C2)=O)cccc2c1CCCN2 c1(C(=O)NC2C(CNC(C(C)(C)SC)=O)COC2)cc2cccc(Cl)c2[nH]1 c1(C(=O)NCCN2CCN(C(CC=C)=O)CC2)cn2ccc(F)c(C)c2n1 N1(C(c2n(C(C)C)cnc2)=O)C2CCC1C(C(=O)NCC(N1CCOCC1)=O)C2 c1(C(=O)NC2(CNC(c3c(C)[nH]cc3)=O)CCOC2)cccc2cnnc(O)c12 C1(C(N(C2CCN(C(C3CCC(C)(C)OC3)=O)CC2)C)=O)CC2C=CC1CCC2 c1(N(CC(F)F)C)nc2c(c(=NC3CCN(C4CCOC4)CC3)[nH]1)COC2 CC(C)CC(C)(O)CNC(=O)C(CC1CC1)NC(c1csc(O)n1)=O C(=O)(CCC(N)=O)N1CCCC(C(C(CSC)OC)=O)CN1C N1(C(CCCCCN(C)C(c2ccncc2F)=O)=O)CCN2CC(F)CC2C1 C#Cc1ccnc(C(=O)NC(C2CCCN2C(c2csc(C)c2N)=O)C)c1 C1(CNC(=O)CC2(O)CCCN(CCC3CC(=O)NN3)C2)CCc2nc[nH]c2C1 c1(N2CC(C(=C)C)OCC2)nc(=NC(CC)c2cccs2)[nH]c2c1COC2 C1(C(=O)NCC(C)C(=O)NC2(C)CCOC2)CCC(=O)N(C)C1 C1(C(N2CC(C(C)NC(C(COC)C)=O)C2)=O)CC2CCCCCCC12 N1(C(c2cn(C)c(=O)cc2)=O)CC2CCCC1(CNC(=O)CC1C=CCC1)C2 c1(C(=O)NCCC(C)NC(c2cccc(C)c2Cl)=O)c(F)ccc2cnn(C)c12 c1(N(C(N(C2CCCC2)CCOC)=O)CC2CSC2)cc2c(s1)CCC2 c1(C(CC)C)nccc(=NCC2(NC(c3ccc(C)c(F)c3F)=O)CCOCC2)[nH]1 CC1C(NC(=O)C(CCO)N(C)C)CCN1C(=O)CC1(C)CCC1 C(=O)(C(CC(C)C)C(N)=O)NCCCN(C(C1CNC(=O)N1C)=O)CC C(=O)(CCCC(F)(F)C(F)(F)F)N1CCCC2(CN(C(C(C)C(C)(C)O)=O)C2)C1 C1(O)(CCNC(C2CCN(C)C2=O)=O)CCN(C(C23CCC(CC2)O3)=O)CC1 c1(C(=O)N)cc2n(n1)CCO2.N1(C(C(C)NC(=O)OC)=O)CC(C)CC1C c1(CNC(c2c(C)ccc(-c3nn[nH]n3)c2)=O)c[nH]c2nccc(Br)c12 Cc1nc(C#N)cc(=NCC23CCC(NC(=O)CC4CCCC4(F)F)(CO2)C3)[nH]1 c1(CC)nc2ccccn2c1C(=O)NC1CN(C(=O)C(C)C)C2(CCC2)C1 c1(CC(=O)N(C(CNC(C2C(C)OCC2)=O)C2CC2)C)csc2ccccc12 C=CCCCCCCC(=O)NCC(CC(=O)NCC(CC)CCCC)OC C1(CC(=O)NCCc2nc(C)[nH]n2)CCC1(C)C.C(=O)(CCCC)N.C(N)=O Cc1cccc2cc(C(=O)NC(C)(C)CNC(c3cccs3)=O)nn12.C1CC1 N1(C(C(C)NC(C)=O)=O)CCN(C(C2CN3CCN2C(C)C3)=O)CC2(CC2)C1 Cc1cc(NC(C2CCN2C(C2CC(O)C2)=O)=O)sn1 C(CN=C(NC(C)CC(F)(F)F)NC1CCC1)N1CCC(C)C1 c1(OC)cccc(-n2nnnc2C(c2ncoc2C(F)F)NCCF)c1 N1(C(c2ncc(OC)nc2)=O)CCCC(O)(CNC(C2CCCCCCC2)=O)C1 C1(CCC=C)CN(C(C2(CC(C)=O)CC2)=O)CCN1 C#Cc1cnc(C(N2CCN(C(=O)C(O)C=C)CCC2C)=O)c(C)c1 C(=O)(C1=NNC(=O)C1)NCC(c1ccccc1)NC(C1C(CCC)C1)=O c1(C(C)C)nc(NCCc2ccc(F)cc2Cl)cc(=NCC2(C)CCCOC2)[nH]1 c1(C(=O)NCC2CN(C(c3c(CCC)cccc3)=O)CC2C)nccc(Cl)c1F N1(CC2CCC(CCC)CC2)CC(CO)CC(C)(C)C1 CCCC(C)(O)CC(=O)NC(C)Cn1cc(-c2cnc(OC)c(F)c2)nn1 c1(C(N(C2C3CN(C(C4(Cl)CC4)=O)CC23)C)=O)cc2c[nH]cnc-2n1 c1(C(N(C2(C(N3C(C)(C(=O)OC)CC3)=O)CC2)C)=O)cccc(F)c1O C1(NC(C(C)Sc2ccncc2)=O)CCN(C(=O)CC23COC(C)(C2)C3)CC1O c1(C(=O)N)csc(CC(F)(F)F)n1.C(C1CCC1)=CC(=O)N(CC)CC C1(NC(C(CCOC)C)=O)CC2CC1N(C(C1CC(=C(F)F)C1)=O)C2 c1(C(N2CCCC(CNC(C3C=CCC3)=O)CC2)=O)cc(Cl)cc([N+](=O)[O-])c1 Cc1sc(C(=O)NC2CCC3CCC23)nc1O O(NC(=O)CCCN(C(=O)C(C)(C)N(C)C)C)C(C(C)C)CO CCCN=[N+]=[N-].C1(N(CCC)CC)CC(C(=O)NCCS)C1.C(=O)C.C C1(NC(C(CC)F)=O)COCCN(C(=O)CCCCN(CCO)CCO)C1 N1(C(C(C)(C)C#N)=O)CCCCC(C(=O)N(CCCO)CCCO)C1 C(=O)(C(C)C(C)C)NC1(C)CC(NC(CC(=C)C)=O)C1 N1(C(c2n[nH]cc2Cl)=O)CCN(C(c2ccc3nccn3c2)=O)CC(O)C1 N1(C(c2n(C(C)C)ncc2)=O)CC2(C1)CN(C(c1cnsn1)=O)CCO2 Cn1ccc(C(=O)NCCCNC(=O)CC2CCCN2C(C)C)c(O)c1=O c1(OC)ccc2[nH]c(C(=O)N(CC(C)NC(=O)C(F)(F)CO)C)cc2c1 CC1(CNC(c2cc(-c3ccc(Cl)s3)[nH]n2)=O)CCN(C(c2ccncc2)=O)C1 C(=O)(C1CNC(=O)c2ccnn21)NCC1(NC(=O)CS(=O)(=O)C2CC2)CC1 c1(CC)ccc(C)cc1C(=O)NCC(C(C)C)NC(c1n[nH]cc1[N+](=O)[O-])=O CC(C)C(O)C(C)(C)C(=O)NCC(C1CCCC1)NC(c1ccsn1)=O O(NC(=O)CCCN(C)C(c1cc(CC)no1)=O)CC=CC c1(OC)cccc(-c2cc(CNC(=O)NCC(c3ccncc3)O)c(C)o2)c1 C1(NC(C(CCF)NC(Cc2c(CC)con2)=O)=O)CCN(C)CC1C C1(CC(=O)N(C)CCNc2cccc(F)c2)CC(C)(C)CCO1 CC(O)CCCCCC(=O)N(CC(O)CNC(=O)Cn1cc2ncccc2n1)C c1(C(N2CCCC(COCC)C2)C(=O)NCCCC2CC2)ccc(OC)cc1F CC1CCCC1C(=O)NCC1(O)CN(C(=O)COc2cn[nH]c2)C1 C=CCC(CC(C)C)C(=O)N1CC(NC(c2cc(Cl)c3n[nH]cc3c2)=O)C(C)C1 Cc1ccc(-c2nc(C(=O)NOCC(=O)NCC3CCCC3)cs2)cn1 c1(C(N2CC(C(C)NC(C3(OC)CCCCC3)=O)C2)=O)cc(Cl)ccc1O c1(C(N(C)CC2CN(C(C3(c4cccnc4)CCC3)=O)C2)=O)ccc(O)cc1F C=C(CNC(=O)C(C)c1ccsc1)CCNC(=O)CCCOC C1(C(=O)NCCNC(=O)C(F)=CCCF)(Oc2ccccc2)CCCCC1 C1(C(=O)NCCOCC)COCCN1C(=O)CC1CC2(CC2)CO1 N(C1CCC(NC(=O)C(C)N2CCC2)c2ccccc21)c1nc(C(C)=O)c(C)s1 c1(OCC#C)cc(CNC2CCCC2C(C)(C)C#N)cc(Br)c1 c1(-c2cn(CCC(=O)NC(c3ccc[nH]3)C)nn2)ccccc1N(C)C C(c1sc2ccccc2c1Cl)=CC(N1CCC(NC(CC(C)(C)C)=O)C1)=O C(CCCCCC(=O)NCCCc1cn(Cc2n[nH]cc2C)nn1)SC N1(C(c2ccc(COC)[nH]2)=O)CC23CCCC2(C1)CN(C(C12CCCC1C2)=O)C3 C1(C(=O)NCC(CN(C(=O)C(F)=CC2CC2)C)O)CC1C1CCOCC1 S(=O)(=O)(c1nc(N(CC(C)C2CC2)C)ccc1Br)NCC(CCC)O N1(C(c2ccc(CC)o2)=O)CCCC(C(N2CCC2CF)=O)C1CC Cc1[nH]c(C(N2CCC(N(C)C)C2)=O)c(C)c1C(=O)NCC.[SH](C)(=O)=O C1(C(=O)NC2CC(c3cn(CC4CCCCC4)nn3)C2)(OC)CCOCC1 CCCCC(CC)CN=c1nc(N2CCC(C)(CCO)C2)c2c([nH]1)CSC2 CC(C)C(C)N=c1[nH]c(=NC2CCCC2n2cccn2)c2c(ncn2C)[nH]1 N1(C(CSC)=O)CCC2(CCN(C(=O)CS(=O)(=O)CC3CCCO3)CC2)C1 O=C(C1=CC2(CCN(C(=O)CC3CCC(=O)N3)C2)C1)N.c1nnnn1C1CC1 N1(C(C2(N(C(C(CCC)CC)=O)C)CC2)=O)CCCC(C2CC2)CC1 c1(C(N2CCN(C(CCC(CC)C)=O)C(C)C2)=O)cnc2ncnn2c1O C(=O)(CCC1CCc2ccccc21)NC1COCCN(C(C(C)(C)C2CC2)=O)C1 C1(NC(c2cnn(CC)c2C)=O)CC2CN(C(=O)Cc3cccnc3N)CC2C1 CN1CC2(CCN(C(=O)CC3CCN3C(c3cncc4[nH]ccc34)=O)C2)C1 c1(C(=O)NC2(C)CCCN(C(c3c[nH]ccc3=N)=O)C2)cc2scc(Cl)c2[nH]1 c1(NC(C(C2CC(=C)C2)N(C(C)CN(C)C)C)=O)ccccc1OCC Cc1nnn(C)c1C(=O)NC1CCC(NC(=O)CCNC(=O)CO)C1 N1(C(CCOCC(C)C)=O)CCOC(CC(=O)NCCCc2nnnn2C)C1 CCCC(CC(=O)N(CC(=O)OC)C)NC(=O)C(C)OCC(C)C C1(NC(=NCC)NCc2cc(C)on2)Cc2n[nH]cc2C(C(F)(F)F)C1 C1(NC(=O)C(F)=CCCF)CCN(C(C2CC(F)(CO)C2)=O)CC1O C(C)(C)(C(=O)NCC(C)N(C(c1cc(C(N)=O)co1)=O)CC)OCC CCC(CCC(=O)NC1(C(=O)N(C)CCN2CCOC2=O)CCC(C)(C)C1)OC C1(C(NOCCNc2ccc(Br)nc2)=O)CC2CCC1N2C(=O)OC(C)(C)C CCCC(C)C(C)N=c1nc2ncn(C)c2c(NCCCN(CC)CC)[nH]1 C1(SCC)CCCCN(C(c2cc(Br)co2)C(=O)NCC2CCCO2)C1 C1(NC(c2c(CCC)nco2)=O)CC2CCC1N(c1ccncc1[N+](=O)[O-])C2 c1(C(=O)NC2CN(C(CC(CCSC)O)=O)CC(C)C2)ccc2nc(O)[nH]c2c1 Cc1cc(C(=O)NC2CCN(C(=O)C=Cc3cn(C)cn3)C(C)C2)nc(O)c1 Cc1cc(NC(c2cccc(I)n2)=O)cc(C)c1S(N)(=O)=O C(=O)(C(C)CC(=O)NC(c1ccccc1)C(N1CCC(C)(C)CC1)=O)OC c1(C(=O)NCCCN(CCN(C)C)C)ccnc2c1ncn2C C1(CNC(c2cn(C)nc2)=O)CN(C(=O)C(N)=O)CCC12CCOC2 CCC(CCOC)C(=O)NCC(C)NC(c1cc(-c2cccs2)[nH]n1)=O C=CCCC(O)CNC(=O)CC1CCCN(C(C2CCC(O)C2)=O)C1 C1(C(C)(C)C)COCCN1C(=O)CC1C(NC(=O)CCc2nc(O)n[nH]2)CC1O C1(CCCNC(c2n(CC)ncc2)=O)CCCCN1C(=O)C(c1cnccn1)C c1(OC)cc(N)ccc1C(N1CCCC(O)C1)=O.c1(C(=O)N)ncoc1C(C)C c1(OC)cc(C(=O)Nc2c(F)cccc2F)cc(Cl)c1 C1(NC(C2CN(C(C)=O)C2)=O)CCN(C(c2ccc(Cl)cn2)=O)CCC1CO CC(C(C)C(=O)N1CC(O)(CO)C1)NC(=O)C(C1CCOCC1)=O c1(CCCNC(=O)NCCC(C)N(C)C2CC2)ccnc2ccccc12 CC(C)(C)CC(O)CC(=O)NC(Cc1ccco1)C(N1CC2C(CO)C2C1)=O c1(C(=O)NC(C(=O)NCc2cnns2)c2ccco2)ccnn1CCF N1(C(CCC=CC)=O)CCC(O)(CCNC(c2cc(CC3CC3)on2)=O)C1 c1(CC(=O)N(CC(CC)NC(c2sc(C)nc2C)=O)C)ccc(C)c(F)c1F N1(C(C2CCN(C(CC)=O)C2)=O)CC2CC1(CNC(=O)C(c1ccnn1C)O)C2 C1(CCNC(=O)Cn2cccn2)CSCCN1c1ncc(I)cn1 C(=O)(C(C)C(O)C(C)CC)NC(CC#C)(C)C(=O)N(C1CC(C)CC(C)C1)C C(CC(F)F)(C(=O)NC1CCC2(CCC2)C1)N(C(c1c(C)cccc1)=O)C C1(CNC(C(C(C)O)NC(C(C(C)C)SC)=O)=O)CC2(CCO1)CC2 c1(C(N2C(CC(=O)Nc3ccnc([N+](=O)[O-])c3)CCC2)=O)cc2cc(Br)ccn2n1 CC(C)C(O)CC(=O)NCC(CC(=O)NCCC(C)O)C1CCC1 N1(CNc2cc(CC)nn2C)CCC(O)(CC#N)CC1 c1(OC)ccccc1CCC1CCN(C(=O)NCC(c2cccc(C)c2)O)CC1 N1(C(C2(OCC)CC2)=O)CCCC1.c1cccc(Cl)c1.C(C)(C)C.C=O.C c1(C(N(C2CCC(NC(C3(P(C)(C)=O)CC3)=O)CC2)C)=O)snc(Cl)c1Cl N1(C(c2c(C(C)C)ncnc2)=O)CC2(CC(NC(C3CC3(C)C)=O)C2)C1 C1(CNC(C=CSC)=O)CC(C)N(C(=O)Cc2cccc(Br)c2)C1 c1(C(=O)NC(CCCNC(c2ccc(SC)cc2)=O)C)cc(C)n(C)c1C c1(COC(c2cccc(=O)o2)=O)ccc(OC(F)F)cc1F N1(C(C=C(CCC)C)=O)CC=C(CC(=O)N2CCC(C(=O)NC)C2)CC1 C12(CNC(=O)Cc3nc(Cl)cs3)CC1CN(C(=O)Cc1sc(Br)nc1Br)C2 c1(C(=O)NC(CC)CNC(c2cnn(CC)c2)=O)ccc(Cl)c(Cl)c1N C(=O)(C1CCCn2cnnc21)N1CC2CC(NC(CC3(C)CC3)=O)C2C1 C1(C)(C(=O)NCC2(F)CCN(C(c3ncc(NC)nc3)=O)C2)CCN(C)CC1 c1(OC)ccnc(C(N2CC(CNC(=O)C(C)C3CC3)CC(C)C2)=O)c1F.O Cc1ccc(C(=O)NCC2(C(=O)NCCCC(F)(F)F)CCC2)c(O)n1 C1(C(C2CC2)OCC(=O)NCC2CC(C)(C)C2)COc2ccccc2O1 C(=O)(C1CCc2snnc21)NCC(CNC(c1cc(C)cc(C)c1)=O)O C1(CC)(CC)CCCN1C(c1cnc(S)nc1)=O.c1(C(C=O)=O)csc(C)n1.N C1(COC)CN(S(=O)(=O)N2CCNC(=O)C2C(C)(C)C)CCO1 c1(C(N2CC(F)CC(NC(CP(C)(C)=O)=O)C2)=O)cnc(O)c2cnccc12 c1(CC(N2CCCCC2)=O)nn(C)cc1[N+](=O)[O-].C1(OCC)CC(CC=O)C1.N C1(c2ccccc2)(CNC(C2C(c3c(OC)c[nH]n3)C2)=O)CC2(CC2)C1 O(NC(=O)C(C)(C)C(C)(C)O)C(CC(C)C)C(=O)NC(C)CC(C)C N1(C(COCc2n(C)ncn2)=O)CCC(CNC(=O)C)C(O)C1.C(N)=O C1CN(C(C2CCC(F)(F)C2)=O)CC12CC2.Cc1cc(COCC(=O)N)on1 CC(O)(C(=O)NCC1CC1)c1ccccc1.C1(CC=O)CS(=O)(=O)C1.C N1(C(c2nc(C)c(C)s2)=O)CC2CCC(C1)N2C(C1C(C#N)C1(C)C)=O Cc1cnc(CNC(C2COC(CNC(=O)CCc3nccn3C)C2)=O)o1 Cc1ccc(OCCCC(=O)NC(C2CCCO2)C2CCC2)cc1 C(=O)(C1=Cc2ccccc2C1)NC(C(=O)NC1CC(C(F)F)C1)O C(CC(C)C)(C(=O)N1CC2CC2C1)NC(=O)OC.c1(C=O)cc(Cl)cn1C.C C1(C(N2C(C)CNC(=O)C2)=O)CN(C(c2ccns2)=O)CC(C)(C)C1 c1(OC)ccc(C)c(C(=O)NCC2CCN2C(C2(O)CCOC2)=O)c1 c1(C(N(C2CCN(C(CCC(=O)NC)=O)C2)C)=O)c[nH]c2cc(Br)ccc12 Ic1cc(CNCc2c[nH]nc2C2CCC2)cc(I)c1 Cn1ncc2c(NCC(C)(F)C(C)(C)F)nc(N3CCNC(=O)C3)nc12 C(=O)(CCCCc1ccccc1)N1CCC(NC(C2(CCC)CC2)=O)C1 c1(C(C)F)cccc(NC(C2(NC(C3COCC(C)O3)=O)CCN(C)C2)=O)c1 C=CCC(F)(F)C(=O)NC(CO)C(C)NC(C1CCCCN1C1CCCC1)=O c1(NCc2cc(COC)no2)[nH]c(=NCC(C)(C)C2CCCO2)nc2c1cnn2C CC(C)C(CN1CCCC1)NC(=O)Cc1ccnn1C.C1(CC(=O)N)CCSC1 c1(C(N2CC(C)CN(C(CN(C)CC)=O)CC2C)=O)cc2c(C)ccc(F)c2o1 C1(C(=O)NC(C(N2CCC(C#C)C2)=O)CC2CC2)CCOCC1(C)C CC1CCCCC1CC(=O)NCCC1(O)CN(C(=O)CCc2cnco2)C1 c1(C(N2CC(NC(COCCC(C)C)=O)C(O)C2)=O)coc(S(N)(=O)=O)c1 CC(C)C(O)C(F)(F)C(=O)NC1CC2CCC(C1)N2C(=O)Cc1cocn1 C(c1cnccn1)=CC(=O)NC(CC)CNC(=O)C(C)(C)c1cscc1Cl C(C(F)(F)C(F)F)NC(C1N(C(C(CSC)C)=O)CCC1)=O N1(c2ncnc(SC)n2)CC2(CN(C(=O)COC3(c4ccccc4)COC3)C2)C1 C1(C(N(CCCC=C)CC)=O)CCC(C)(C)N(C(=O)C(C)(C)CCCF)C1 N1(C(C2CCN(CC)CC2)=O)CCN(C)CC1C(N1CC(=O)NCC1CC)=O C1(NC(CCC=C(C)C)=O)CN(C(=O)C=C(C2CC2)C2CC2)CCC1C N1(C(c2c(C)cncc2)=O)CCC=C(CNC(=O)C(C(C)C)C2CCC2)C1 C1(CC)CCC(C)N(C(=O)C(=O)NC2CCN(c3ncncc3Cl)C2)C1 c1(C(N2CC(F)CC(NC(c3c(C)cccc3)=O)C2)=O)ccnc2c1CCC2 c1(CC)cccc2c(CN(C)Cc3c(C)nn(Cc4ccccc4)c3C)c[nH]c12 C(C(=O)NC1(C)CC(NC(=O)CCc2cccs2)C1)(C(C)C)SCC N1(C(CCCC)=O)CCC(C(C)NC(C2CC2CCC)=O)CC1 N1(C(C)=O)CCC(NC(=O)C(C)CNC(=O)C(F)F)C1 c1(OC)nn(C)cc1C(=O)N.c1(C=O)noc(C2CC2)c1C.C12CC(C1)C2 c1(C(N(C(CNC(C(CCOC)(C)C)=O)C2CC2)C)=O)cc2c(o1)CCCC2 N1(C(C(CC=C)CC=C)=O)Cc2nccn2CC(NC(=O)CCCC(C)(C)C)C1 CC1CN(C(C2CCC(C)(C)C2)=O)CCN1C(=O)C1=CCCSC1 N1(C(CSCC(C)=O)=O)CCC(NC(=O)C=Cc2scnc2C)C(F)C1 Cc1cc(F)c(C(=O)N)c(F)c1.C1CN(C(=O)CN(C)C2CC2)C2(CCC2)C1 C1(C(CNC(C=CC(C)C)=O)(C)C)CCCN1C(C1CCN(C)C1)=O c1(C(N(CCNC(C(C)OCC)=O)C)=O)cncc(N2CCOCC2)c1 c1(NC(C)=O)c(C(=O)NC2CCC2)cccc1C.c1(C(=O)N)cccc(F)c1F c1(C(=O)NC2CC2C)c(F)cc(Cl)cc1F.C1(C=O)CCCC1c1nc[nH]n1 c1(CC(=O)NCC(CNC(c2cnc(SC)[nH]2)=O)C)ccc(O)cn1 c1(C(N2CC3N(C(C(CC)(C)O)=O)C3C2)=O)ccc2cc(C)[nH]c2c1 CC1CN(C(=O)C(O)CC(N)=O)CCC1C(=O)NCC1(C)CCCCCC1 CC1CC(NC(=O)CC(C)(O)c2ccccc2)CN1C(=O)CN(C)S(N)(=O)=O CCC(CC(=O)NCC)C(F)F.c1(C(N(CCC)C)=O)cc(C)nn1C1CC1.O C1(CC(=O)N(C2CCN(C(c3cncnc3)=O)C2)C)CC(=O)NC1=O CCCCCC(O)C(C)C(=O)NC1CN(C(=O)CCCCCC(C)C)C(C)(C)C1 C1CCC(=C2CCC2)CC1.N1(C(CC)=O)CCC(C)(NC(=O)CC2CCCCC2)C1 O=C1NCC2CN(c3nc(N4CCCC(O)CC4)c4ncsc4n3)CCN12 C(=O)(C(COCC)N=[N+]=[N-])NC(C(=O)NCC(=C)F)C1(C)CC1 Nc1cc(F)c(C(=O)NC2CC3CC(C2)N(C(C2(CCF)CC2)=O)C3)c(F)c1 C1(NC(C(C(C)C)(C)O)=O)COC2C(NC(=O)CCOc3ccccc3)COC12 c1(CC)cc(N)c(C(N2CC(C3CN(C(=O)C=CCF)C3)C2)=O)cc1F c1(NC(C(C(C)C)C)CNC(C2(C(F)F)CCCC2)=O)ncc([N+](=O)[O-])cn1 C(c1cn(C)c2ccccc12)=CC(N1CC(OCCNC(CC(C)CF)=O)C1)=O CCC(C)(C)C(=O)C(=O)NCCCc1cccc(C)c1 c1(C(=O)NCC(=C)CCNC(C2CCCS2(=O)=O)=O)cc2ccccc2[nH]1.O N1(C(C(CC)COC)=O)Cc2occ(C(=O)NCCC(C)C(=O)OC)c2C1 CC1CCC(C(=O)NC2CC(C)(C)C2)N(C(=O)C(F)F)C1 CC(C)C(O)CC(=O)N1CCOC(C(=O)N(C(C(N)=O)C2CC2)C)CC1 N(C1CC2(CN(C(=O)CC3CC(F)(F)C3)C2)n2ccnc21)C(C(CCCC)O)=O CC#CCCCC(=O)N1CCC(C)C1C(=O)Nc1ccc(OC)c(O)c1 CCC(C#N)(CC)C(=O)N1C2CCC(C(=O)Nc3cc(O)cc(F)c3)C1CC2 c1(C(N2CC3C(C(N4CCCC(OC)C4)=O)(C3)C2)=O)ccc2nc(Br)sc2c1 C1(F)(CNC(c2c(NC)snc2C)=O)CCCN(C(C2CC(F)C2)=O)C1 c1(C(=O)OC)coc(S(=O)(=O)NC(C2CCCCC(=O)N2)=O)c1 c1(CNC(C2N(C(C3(N(C)C)CCCC3)=O)CCC2)=O)cccc(O)c1 N1(C(C2N(C(C)C)CCC2)=O)CCOC2(CCN(C(c3sc(F)cc3Cl)=O)C2)C1 c1(OC)cnc(Br)cc1C(=O)NCCC1CCCN1C(=O)C1=CCCCO1 N1(C(c2ncc(CC)s2)=O)CCCC(C)C1CNC(=O)Cc1cnn(C)c1 C1(C(N2CC(C(=O)NCC(O)C(=O)OC)(CC)C2)=O)CC2CCC1CC2 c1(C(N(CCNC(C(C)CO)=O)C)=O)ccc(N2CCCC2)nc1 C1(NC(C2(CC)CC2)=O)CC(C)N(C(C2CCC(C(=O)OC)CC2)=O)C1 C1(NC(Cc2n(C)ccn2)=O)CC2(C1)CN(C(C1CC1(c1ccccc1)C)=O)C2 c1(C(=O)NC2C(CC)CN(C(=O)Cc3csc(C)c3)CC2)ccc2c(c1)CCO2 C(=O)(C1=CC2CCCCCC12)NCC1C(C)CCN(C(c2nccc(C)c2)=O)C1 C1(C(N2C3(CNC(CCc4c(C)cccc4)=O)CC(C2)C3)=O)CC(C)OC(C)C1 c1(NC)ncccc1C(=O)NCC1(C(=O)NCC2CC23CCC3)CC1 Cn1nc(C(F)F)cc1C(=O)NC(C)(CNC(C1(CCF)CCC1)=O)CO c1(C(N(C(C)CN(C(=O)CCC2CC2(C)C)C)C)=O)cccc2c1CCCC2 C1(NC(CCCCSC)=O)CC2CC(NC(=O)C(C)NC(C)=O)CC12 c1(NC(C2CN(C(C(C)OCc3ccncc3N)=O)CC2C)=O)ccc(F)cc1 CS(=O)(=NC(=O)C1(O)CCOC1)c1cnn2c1CN(C(=O)C=CC=C(Cl)Cl)CC2 C=C(Cl)CC(C(=O)N1CCC(C(C)C#N)CC1)NC(=O)Cn1cnnn1 CCC(C)CC(C)C(=O)N(C1CC2CCC(C1)N2C(c1cnsn1)=O)C c1(NC(C)=O)ccc(C(=O)N)cc1Cl.C1(CC=O)CCC(C)CO1.C(C)(C)C C(=O)(C1=Cc2cc(Cl)ccc2OC1)N1CCN(C(C2C(OCC)C2)=O)C2(C1)CC2 c1(CNCC2(C(=O)Nc3c(C)cc(Cl)nc3)CC2)cc(F)cc(F)c1O N1(C(C2(CC=C)CCN(C(c3cncnc3)=O)C2)=O)CCc2n[nH]cc2C1 Cc1cn2c(n1)CC(C(N1CC3CC(NC(c4snc(O)c4Cl)=O)C1C3)=O)CC2 C(=O)C1CCc2c[nH]nc21.C(C(=O)N)(C(C)C)NC(=O)OCC.CCC(C)C C1(c2ccccc2)(NC(C2CCC(F)CC2)C)CCNCC1 n1(C(C)C)nccc1C(N1CCC(C2CCCN2C(=O)CCc2cnc[nH]2)C1)=O Cc1nc(C(N2CCCC2(C)CNC(c2cc(CO)oc2C)=O)=O)c(C)o1 C1(C(=O)NC(c2nc(C)[nH]n2)CO)N(C(=O)C(C2(O)CCCC2)F)CCC1(C)C c1(C(N2CC(C#N)C(NC(c3cc(Cl)cc(I)c3)=O)C2)=O)cc2n(n1)CCCC2 C1(NC(Cc2c(C)noc2Cl)=O)Cc2ccccc2C1N=c1[nH]nco1 CCC(COC)C(=O)N(CC(N1CCN(C(=O)C(F)CN(CC)C)CC1)=O)C C(=O)(C(C)(C)C(F)(F)F)N1CCC(C)CC1.Cc1cn(C(C)C)cc1C(=O)N.C C1CCN(C(=O)CC2CC(=O)NC(=O)C2)C(C)C1.c1(OC)cc(C=O)ncn1.N N1(C(CCCSC)=O)CCN(C(C2CN3CCN2CC3)=O)C2CCCC12 Cc1ccc(CCC(=O)NC2CN(C(c3c[nH]c(=N)o3)=O)CC2C)cc1Cl CC1CCC(CNC(C2SCCS2)=O)N(C(C2CCC2(F)F)=O)C1 C(=O)(CCCCCC(C)(C)C)N(CC(O)(C(F)(F)F)c1ccccc1Cl)C Cc1cc(N)ccc1C(N1CCCN(C(=O)C(c2ccccc2)C)CC1)=O c1(C(N2CC(NC(c3cc4n(n3)CCC4)=O)C3C2C3)=O)nccc2ncccc12 C(=O)(C(C)(CO)NC(=O)C(O)CC1CCCC1)N(C)Cc1onc(C)n1 c1(CC)cc(NC(C2CC=CC(NC(C3(C)CCCO3)=O)C2)=O)cc(F)c1 c1(C2(CC(=O)NC(C)C=CC(=O)O)CC2)ccccc1 C(=O)(C1=CCC(C)(C)CC1)N1CCC(C(N2CCCC(C)C2)=O)(CC)CC1 N1(C(C23N(C(C4CCC(CC)CC4)=O)CC(C2)C3)=O)CCCC2(CC2)C1 c1(C(=O)NCC(CC)NC(c2cnc3scc(C)n23)=O)nc(C)n2ccccc12 CCC(CNC(=O)OC(C)(C)C)C(=O)NCc1cnc(C(C)C)s1 C1(c2cccc(Br)c2)(CNC(=O)CCOC2CCCCC2)CCCCC1 Cc1cc(C(=O)NCCC2CCN(C(c3c(C)cccc3O)=O)CC2)cc(O)n1 CCCCC(=O)C(=O)NCC1(C(=O)NCC(CC)C(C)(F)F)CCCCC1 Cc1ccc(C#N)cc1C(=O)NCC1CC(NC(c2cnsn2)=O)CCO1 c1(CC)ncc(C(=O)NC2CCC2NC(=O)CCNC(N)=O)c(O)n1 C1(C)(C(=O)OC(c2ccc(C)c(F)c2)C)CCC(F)(F)CC1 c1(C(=O)NCCC(=O)OCC)cc(OC)ncc1N.c1ccc(O)cc1C.C C(=O)C1=CC2C=CC(C1)C2.c1(C(=O)NC(c2ccccn2)C)occc1C.N CCCCCC(F)C(=O)N(CCCC(=O)NCCc1noc(CC)n1)C O=C1CN(N2CCN(c3ccccn3)CC2)C(c2ccccc2)CO1 N1(C(C2(CC)CCN(C(=O)COC(C)=O)C2)=O)CCC(C)(C)C1C C1(C(=O)N)(CC)CC(F)(F)C1.C1(C(N(C2CCCC2)CCC)=O)CCOC1C Cc1ccn2cc(C(=O)NC3(C4CCN(C(=O)CC(C)O)CC4)CC3)nc2c1 c1(OC)c(CNC(=O)NCC(C)(C)C(N)=O)ccc2ccccc12 C1(CNC2(c3n(CC)nnn3)CC(C)(CBr)C2)CC2CCC(C1)N2C N1(C(c2cc(C)ns2)=O)CCC(CO)C(NC(=O)Cn2ccnc2C)C1 CC1CNC(C)(C)CN1C(=O)Cc1c(F)cc(F)cc1Br C(=O)(C(O)C1=CCCCC1)N1CCOCC(NC(c2cc(C)on2)=O)C1 N1(C(c2c(CC)c(F)ccc2)=O)CC(NC(=O)CSC)CC2(CC2)C1 c1(CC(=O)N(C2CCN(C(C(C)Cc3cnc[nH]3)=O)C2)CCO)ccc(O)cc1 CC1C(C)N(C(=O)Nc2cccc(C(N3CCCC3)=O)c2)CCN1C c1(C(N2CCCC(C)C2C=O)C(=O)NCC)cc(Cl)nc(Cl)c1.C(C)(C)C CC(CC(=O)N1CCC(C(=O)N(CCCN=[N+]=[N-])C)C1(C)C)C(F)(F)F c1(C(C)C)nc(C(=O)NC2CC(CC(=O)NC(c3cccnc3)C)C2)co1 c1(C(=O)NC2CC(CNC(=O)C(=CC3CCCCC3)F)C2)ccc2n[nH]cc2n1 C(CNC(=O)CCc1cnoc1)(C(C)C)NC(C=C(C)I)=O C1(CNC(CCc2n(CC)ccn2)=O)CCC2(CCC2)C1.C1(C=O)CC(O)C1 C1(C(=O)NCC2CC(NC(c3n(C(C)C)ccc3)=O)C2)CCC2CC2CC1 C1CN(C(C2CCCN2S(C)(=O)=O)=O)CCN1C(c1cc(F)cc(Cl)c1)=O.C Cc1ccc(Cl)cc1C(=O)NC1(C)CCCC1NC(=O)C(C)OCCC(C)C C1(NC(c2ccc(COC)s2)=O)CCS(=O)(=O)C12CN(C(=O)C(C)O)C2 Cc1cc(=O)oc(C)c1C(N1CC2CCC(C2)C1)=O.C1(C(=O)N)CSCC(=O)N1 Cc1cc(C(N2CC3CC(C2)C3NC(c2cnc(C3CC3)s2)=O)=O)nc(O)c1 N1(C(CSC(C)C)=O)CCOC2(CCN(C(c3ccc(OC(F)F)nc3)=O)C2)C1 CCC(C)CC(=O)NC(C1(O)CCCCC1)C(=O)N(CC(O)C1CCC1)C c1(C(N2CC(NC(C3(n4cc(Br)cn4)CC3)=O)C2)=O)ccccc1.C(CO)S C1(C(C(=O)NCc2cccs2)N(CC=C)C2CC2)CCC2(CC2)C1 C1(NC(c2ncc(OC)cn2)=O)COCCN(C(c2n[nH]c3c2CCC3)=O)C1 c1(CN2CCCC(CN(C)C(c3c(Br)cnn3C)=O)C2)nc2ccccc2o1 c1(CNCC(c2cccc(Br)c2)C(=O)O)csc2ccc(F)cc12 c1(C(N2CCCC23CCC3)=O)ccc2nnc(S)n2c1.CC(C(=O)N)NC(N)=O C1(CCN(C(=O)C(c2ccccc2Cl)O)C)CCN(C(C2CNC(=O)C2)=O)CC1 C1(C(NOCC)=O)CCOCCN1C(=O)C(N1CCCCC1)C N1(C(c2c(C(C)(C)C)con2)=O)CCCCC(NC(=O)CN2CCC(C)(O)C2)C1 c1(N2CCC3(CN(C)C3)C2)ccc(S(=O)(=O)NC(c2cccs2)C2CC2)cc1Br C(=O)(CCCC(=O)N)N(CC)CC.C1CC(O)CN1C(C1CCN(C)C1=O)=O C1(C)(C(=O)NCC2(NC(c3cccs3)=O)C(C)CCCC2)CCC(F)(F)CC1 C(=O)(CC1=CCOCC1)N1CC(CNC(C(C)n2ccnn2)=O)CC1(C)C C1(C(C)NC(=O)CC2(N(C)C)CC2)CCCN1C(=O)CCc1cnn[nH]1 C1(CC(N2CC(CC(=O)NCC(CC)OC)(OC)C2)=O)CCCNC1=O S(=O)(=O)(CCC(=O)Nc1ccccc1)NC.C12(CCC(=O)N)CCC(CC1)C2 C(=O)(C1=CCN(C(=O)C(C)Cn2ccnc2)CC1)NCCCCCC=C Cc1cc(N)cnc1C(=O)N.c1(C2(C=O)CCC2)cc(Cl)ccc1F.CC=CC CCCCC(C)C(=O)NC(Cc1cn[nH]c1)C(=O)NCCCc1nncn1C c1(C(=O)NC(CCNC(c2c(C)onc2Cl)=O)(C)C)cccc(F)c1O N1(CCNC(CCCNC(c2c(CC)noc2)=O)=O)CCOCC1=O C1(NC(CS(=O)(=O)N(C)C)=O)CCC2CCN(C(c3ccc(Cl)nc3N)=O)C1C2 C(C(C)(C)C#CC(=O)NC(CO)(CO)CO)NC(c1cn(CCC)nn1)=O C(C(C)S(N)(=O)=O)Nc1ncc(CC)o1 c1(C(=O)NC2C3CCN(C(CC(=C)C)=O)CCC32)ccc2ccccc2c1F c1(CCC(N2CC(N(C(c3cc(CCC)on3)=O)C)C2)=O)ccc2ncsc2c1 N1(C(c2[nH]cc(C)c2)=O)CCC2(NC(c3ccc(O)cc3C)=O)CC2C1 Cn1c(COCC(=O)N)nnc1S.C1(CC)CCCN(C(C2(C#N)CCC2)=O)C1 c1(C2N(C(C#CC)=O)CCC2)cc(=NC(=O)C2(Br)CC2)[nH][nH]1 Cc1c(Cl)ccc(COC(=O)C(O)(C(F)(F)F)c2cn[nH]c2)c1Cl C12(CNC(c3c(C)nn[nH]3)=O)CCCC1N(C(=O)COC(C)(C)C)CCC2 c1(CC(=O)N(CC(=O)N(CCC)CC2CC2)C2CC2)cc[nH]c1 c1(C(=O)NC(CC)CN(C)C(C2CC(=O)N(OC)C2)=O)ccc(OC)c(Cl)c1F C12(NC(c3ccc(C)cc3Br)=O)CCC(CN(C(c3ccnn3C)=O)C1)C2 Cc1cnc(Cl)[nH]c1=NC1CCC2CN(C(c3cn(C)cn3)=O)CC12 C1(c2nnnn2C2CCOC2)(Nc2ccc(OCC)s2)CCCC1OC c1(C(=O)NC2CCCCC2NC(C2(F)CCOC2)=O)coc2c1CSC2 c1(C(=O)NCC2COCCN(C(C(CC)OC)=O)C2)cc2ccccc2n1CC CC1(C(N2CC(c3ccc(O)cc3)C2)=O)CCN(C(C2CCNC2=O)=O)CC1 Cc1ccc(C(=O)NCC(CO)NC(=O)CC2CCC(C)CO2)c2c1CCCN2 NS(=O)(=O)C1(C(=O)NC2CCC2)CCC1.c1(C=O)cc(-c2ccoc2)[nH]n1.N C(=O)(C1=NOCC1)C(=O)CSC1CCCC1.c1(OCC)cccc(N)c1.C C(=O)(C(C)CC1CCC1)N(CCC(=O)NC(CC)C)C c1(C(=O)NCC(CN(C(C2C(=C)C2)=O)C)C)ccc([N+](=O)[O-])cc1[N+](=O)[O-] c1(C(N2CC3C(CNC(C4CN(CC)C(=O)C4)=O)(C3)C2)=O)nc2ncccn2n1 c1(C(N2CC(NC(CCCn3ncc(C)c3)=O)C(C)C2)=O)sc2cncn2c1C C1(C(=O)NCC(=C)CCNC(c2nc(C)sc2C)=O)CCc2ncnc(C)c2C1 C(C)(C)(C(C)CC(=O)NC1(C)CC1)NC(C(C)NC(=O)NC)=O S(=O)(=O)(c1c(F)ccc(F)c1F)N1C(C(=O)OC)CCc2n[nH]cc21 Cc1nn(C(C)C)c(C)c1CN(C)C(C1(c2ccc(Cl)cc2Cl)CCOCC1)=O C(=O)(CCCCCCC(=O)NCCCC(C)(C)NC(C1C2CCCC12)=O)OC c1(C=O)ccc(Cl)cc1-c1ccsc1.Cc1scnc1C(=O)NCC1CC1.C c1(C(=O)NC(C#C)CC(C)C)n[nH]c2c1CN(C(c1c(O)cccc1F)=O)C2 C(=O)(C(O)C(CCC)NC(c1ncsc1C)=O)N1C(CC#C)CC1 C(C(=O)N1OC2CC1C(O)C2O)Sc1c([N+](=O)[O-])cccc1 Cc1cc(C(=O)NC(C)C=CC(=O)NC2CCCC2(F)F)c(O)nn1 N1(C(C23CCC(OC)C2C3)=O)CCC(NC(c2ccc(Cl)c(F)c2)=O)C1(C)C CC1(C)CN(C(C2CC(F)(CO)C2)=O)CCO1.C(=O)C(C)C.CC(F)(F)F.C CCC(COC)C(=O)N(CCCCNC(C1CCC=CCC1)=O)C N1(C(C2CC(C#N)(OC)C2)=O)CCCC12CCN(C(=O)CC1CC13CC3)CC2 c1(NC(C2CCCCO2)C)nccc(=NCc2cc(O)ncn2)[nH]1 C#CC1(C(=O)NC2CC(C)(NC(=O)C(=O)N(C)C)C2)CCCC1 N1(C(c2cnco2)=O)CCC(C2CCN(C(C3(n4cncn4)CC3)=O)C2)CC1 C1(CCNC(c2c(C)cn(C)n2)=O)C(C)CCCN1C(c1ncc(Cl)cc1Cl)=O C(c1ccc(I)o1)=CCOC(C(C=C)OC)=O CC(C)(C)CCC(=O)NC1(CO)CCN(C(C2CCC23CCC3)=O)CC1 N1(C(=O)OC(C)(C)C)CC2CC(C(=O)Nc3ccnn3C3CCCCC3)C2C1 CC1(C(=O)NC2CCNCC2O)CCCN(C(c2ccc(Br)cc2)=O)C1 C1CC(C2CCN(C(=O)C3=CCS(=O)(=O)C3)C2)C1.CC(C(C)(C)C)=CC=O.N C(=O)(CC(C(C)OC)NC(c1cnc(O)c(F)c1)=O)N1C(CC)C(O)CC1 C1(C(=O)NCCC(O)COCc2ccccc2)CCn2nccc2C1 N1(C(C2CCC(CC)O2)=O)CCC2C(C1)CN2C(c1cc[nH]n1)=O CC(N=c1nc(C2CCOCC2)[nH]s1)C1CCN(C(=O)C(N)=O)C1 C1(NC(CC2CCC(NC(C3(C(C)C)CC3)=O)CC2)=O)CN(C)C2(CCC2)C1 C1(C(=O)NC2C3C(C)N(C(c4cc[nH]n4)=O)C2C3)CCOCC12CCCC2 C1(C(N2CC(F)=C(C)CC2)=O)CC(N=[N+]=[N-])CN1C(=O)C(O)C(C)C N1(C(c2ccc(C#N)cc2O)=O)CC(NC(=O)C(O)C2CC2)C2(CCCC2)C1 C(CCC(=O)NCC1CCCC1NC(C1CCC(C)C1)=O)N(C(=O)OC)C C(C(C)C(F)C(=O)N1CC(C)(CO)C1)NC(c1n(C=C)nnc1)=O Cn1cc(C(=O)NC2(C)CC(NC(=O)C)C2)c(C2CC2)n1.c1cn[nH]c1.O C1(CNC(C=C(C)C)=O)CC2(CCOCC2)CN1C(C1C(C#N)C1(C)C)=O CC(C(=O)N1CCC(CN(C)C(c2cc(C(C)(C)C)ccn2)=O)C1)C1=CCCC1 N1(C(C2(CC)CCCN(C(c3cccc(=O)o3)=O)C2)=O)CC2CCC(O)C2C1 C(=O)(C(C)(C)C(=O)OCC)Nc1cccc(NC(C(CC=C)C)=O)c1 N#Cc1cnc(N2CCCCC(NC(C3COC4COCC34)=O)C2)c(Cl)c1 N1(C(C(CC)SC)=O)CCOC(CNC(=O)CCCc2cc(C)no2)C1 c1(C(=O)N)ccc2c(c1)CCS2(=O)=O.c1(SC)ccc(C(=O)NC(C)C)s1 c1(N2CCN(CCOC)CC2)nc(N2CCC(OC(C)C)C2)c2ncccc2n1 O=C(C#CC1CC1)N1CCC(C(N2CCCC(CCO)C2)=O)C1 N1(C(c2c(OC(CC)C)cccc2)=O)CC2(CCC2NC(c2conc2C)=O)C1 C(=O)(C1=NNC(=O)CC1)N1CC(C#N)C(NC(c2cccc(OC(F)F)c2)=O)C1 N1(C(C2(CC)CC2(F)F)=O)CCC(NC(C2(C#N)CC23CCC3)=O)C(C)C1 N1(C(c2nc(C)nn2C)=O)CCCC(NC(c2ccn(C3CCCC3)n2)=O)C1C Cc1nc(CCC(N2CC3C(CNC(=O)C(n4ccnc4C)C)C3C2)=O)oc1C N1(C(C(C)C)Cc2nccn2C)CC2CN(C(=O)OC(C)(C)C)CCC2(CO)C1 C=C1CCN(C(=O)Cn2ncccc2=O)C(C(N2CC3CC3(C(=O)OC)C2)=O)C1 c1(CN2CCCCC(N(C)C)C2)cc(Br)c(Cl)c(Br)c1O C1(C(N2CC(C)C(NC(=O)CC(O)C3CCCC3)C2)=O)CC12CC(C)(C)C2 N1(C(C2CCC(CNC(C3(C4(C)CC4)CC3)=O)C2)=O)CCC(F)(F)C(F)C1 CC(CC(=O)N(C)CC)CC(C)(C)C.C1(=CC(=O)N)CCC(C(C)(C)C)CC1 c1(OC)ncc(-c2cncc(NC(c3csc(Cl)n3)=O)c2)cn1 c1(C(N2CCC(F)(CNC(C(CC=C)(C)CC)=O)C2)=O)cc2ccnc(Cl)c2s1 N1(C(CCC2C(C)C2)=O)CCN(C)CC1CNC(=O)C(=O)NCC1CC1 CCCC(C)C(=O)NCCN(C(C1CCOC1(C)C)=O)C1CC1 N1(C(C(C)=C(CC)C)=O)CC(NC(c2ccc3c(c2)NCC3)=O)CC12CCOC2 C(=O)(CC1OCCc2ccsc21)NCCN(C(CSCCOC)=O)C c1(C(=O)Nc2ncc(F)c(N3CCN(CC)CC3C)n2)cc(Cl)cc2nc[nH]c12 c1(C(=O)NC2(CCCO)CCC(F)(F)CC2)nc2ncc(Br)cc2s1 C1(CN(C(=O)CC2CCOC2)CC)CCN(C(c2ncsc2C)=O)CC1 Cc1[nH]nc(C(=O)NCC(CNC(=O)CSCc2cscn2)CO)c1O N(C(=NCCC1CC1(Cl)Cl)NCC(F)F)CC(C1CCOCC1)(C)C Cc1nc(C(C)(C)C)sc1C(N1CC(C)CC1C)=O.C1(C(=O)N)COC(=O)C1 c1(N2C3(CNC(C4CCC(C)C4)=O)CC(C2)C3)nc(Cl)ncc1C(F)(F)F CCC(C)(CNC(=O)CC1CC1Cc1ccccc1)CO CC1CC(CNC(=O)C=CCN(C)C(c2nc[nH]n2)=O)CCO1 Cc1cc(Cl)c(C(=O)NCC(C)(CO)NC(=O)Cc2cccnc2C)cn1 c1(C(=O)NCC2(O)CCN(C(COCCC#C)=O)C2)cnc(OC)c(Cl)c1 CC(C)CC(CNC(c1cc(F)cc(F)c1)=O)C(=O)N1CC2CC2C1 C1(CC)CCN(C(C2SCCS2)=O)C(C(=O)NC(C2CC2C(=O)OC)C)C1 c1(CN(C(c2nocc2Cl)=O)C(c2cccs2)C2CC2)ccccc1F C#CC1CN(C(=O)CC2CCCS2(=O)=O)CCN1C(C1CCC(=O)N1CCC)=O C(=O)(CC(CCNC(C)(C(C)OC)c1nnnn1C1(C)CC1)C(F)(F)F)OC C1(NC(=O)C2=COCCO2)CCCN(C(=O)C(F)C2CCOC2)CCC1 C#Cc1cc(C(=O)NC2(C(F)(F)F)CCC(C)(C)CC2)ccc1C C1(CC)CC(C(=O)NCc2ccc(O)cc2F)CCN1C(c1cncc(Cl)c1)=O C(=O)(C1=CCCCO1)NC(C)(C)C(=O)NC1CC2CCC1O2 C(=O)(C(O)CC(C)(C)C)NC(C(=O)N(CCC1=CCCCC1)C)CO c1(CC(N2CCC(O)(C(CNC(CCCC#C)=O)C)C2)=O)ccc2c(c1)COC2 Cc1ccc(CNC(C)CC2CCSCC2)cc1O C1(CN(C(=O)Cc2cncs2)C)CCCC(NC(=O)CCCC2CCCO2)C1 C(CCC(=O)NCCCN1CCC(NC(=O)CC(C)O)C1)OCC=C C1(C(=O)NCC(c2cc(F)cc(Cl)c2)NC(C)=O)CCCCC1(F)F C(=O)(C1=C(Cl)CCCC1)N1C2CC(NC(COc3c(C)cc(N)cc3)=O)(C2)C1 c1(C(=O)N)ccc2nc(N(C)C)[nH]c2c1.CC(CNC(=O)C(C)c1ccsc1)C C1(C)(C(=O)NC(CC)CO)CCN1C(c1csc(COC)n1)=O c1(CC)ncc(C(=O)N(C(C)C(=O)NCC(C)N=[N+]=[N-])C)cn1 c1(N(C(CCc2c(C)cccc2)=O)C2CNC2)ncc2ccn(C)c2n1 C(CC(=O)N1CCC1C(N)=O)(CC(C)C)NC(CCCNC(=O)OC)=O c1(C(N(CCCN(C(C2C(OC)CCC2)=O)C)C)=O)ccnc(-c2cc[nH]n2)c1 N1(C(Cc2n(C)cnc2)=O)CCOC2CN(C(C3CCCCO3)=O)CC12 C(=O)(C(C#N)C(C)(C)C)NCc1nccc(C(=O)Nc2ccc(C)c(O)c2)c1 c1(OC)cc(N)c(C(=O)NCCCCCNC(=O)CCCn2ccnc2)cc1F N#CC1CN(Cc2cncs2)CCN1C(=O)C(Cl)(Cl)Cl c1(C(=O)NC2CC(C(=O)NCc3nc(C)oc3)OCC2)c(C)oc(C)c1C c1(OCCCNC(CN(C)C(c2cc(F)ccc2F)=O)=O)cnc(F)cc1Cl Cc1ccc(C(C)C)cc1NC(=O)NCC1C(C)(C)C1(C)C c1(C(N2CCCC(CC)(NC(=O)Cc3cncnc3)C2)=O)c(C)cc(F)cc1C N1(C(c2c(C)nc(CCC)s2)=O)CC2CCC2(CCNC(c2cnsc2)=O)C1 c1(C(=O)NC(C2CN(C(C3OCCN(C)C3=O)=O)C2)C)ccc(F)c(N)c1 C#Cc1ccc(C(=O)NC(CNC(c2cc(F)cnc2O)=O)C(C)C(C)C)cc1 N1(C(c2nc(CNC(C(C3CCC(=O)N3)C)=O)oc2)=O)CCC(C#N)C1 C(=O)(C(F)(CNC(=O)Cn1cnnn1)C(C)C)N(CCCC#C)C N1(C(COCc2cc(C)on2)=O)CCC2CCC(C1)N2C(=O)CCS(C)(=O)=O C1(NC(C=C(CCC)C)=O)CCC2CC1CN2C(c1cnc(CC(C)(C)C)o1)=O C1(C(=O)NCC(CC)C#N)C2CCC(C2)C1NC(c1c[nH]nc1C(C)C)=O C1(N(C)C(C2CNC(=O)O2)=O)CN(C(=O)C2=NNC(=O)C2)CC1(C)C c1(C(N2CC(CC(=O)OCC)C2)=O)cccc(CS(C)(=O)=O)c1 n1(-c2cn(C)nc2)cc(NC(=O)NC(C2CCC(F)(F)CC2)CCO)ccc1=O N(C(=NCCCc1ccc(Cl)cc1Cl)NCCSCCC(F)(F)F)C(COC)C N1(C(CCc2scc(C)n2)=O)CCC(NC(=O)Cc2c[nH]ccc2=O)CC1C c1cccc(C#N)c1.C(=O)(CC=O)NCC#C.CCCN(C(=O)CNC)C.N Cc1ccc(NC(=O)CC2C=CCC2)cc1OCC1CCC1 N1(C(C2C(C)CCC2)=O)CCN(C(c2cccc3ccccc23)=O)C2(CCC2)C1 C(CC(C(=O)N1CC(COC)C1)NC(=O)COCC)OCC c1(OC)ccnc(F)c1C(=O)NC(C1CCCN(C(C2CC23CCC3)=O)C1)C c1(C(C=O)(C)C)ccc(F)cc1.C(CO)(C(=O)N1CCC(CC)C1)NC(C)=O.N C=CCCCC(C1CC1)NC(=O)NC1(CCCCO)CC1 c1(C(N(CCC)C)=O)ccc(SCC)cc1.c1(C=O)n[nH]cc1Cl.C(N)(=O)N O=C1Nc2ccc(C(=O)NCC34CCC(CC3)C4)cc2CO1 C1(C(C)C)CN(C(=O)C=Cc2ccco2)CCC1NC(C1(Cl)CC1)=O c1(C(N(C(c2cn(-c3ccc(C(F)(F)F)cc3)nn2)C)C)=O)cc(I)ccc1F N1(C(=O)NCCc2c(C)ccc(Cl)c2)CC2C(C(=O)O)(C1)CS2(=O)=O C(=O)C1=C(C)OCC1.c1(CSC)ccc(C(=O)NCC2CCCO2)cc1.C C=CCC(CC(C)C)C(=O)NCC1(OC)CN(C(=O)C(C)CC)C1 c1(-c2cn(CCOCCNC(C3(c4nccs4)CC3)=O)nn2)cccc(F)n1 CC1CC=CCC1C(=O)NCCC(O)CNC(=O)C.c1(C(=O)N)ccncc1 c1(OCCn2cc(CC3N(C(c4c(C)nn[nH]4)=O)CCC3)nn2)ccc(F)cc1 c1(C(N2CC3C(NC(c4ccc(CC)c(Cl)c4)=O)C3C2)=O)c(C)cc(C)nc1S O=C1CC2(CCCN(C(c3csc(Cl)c3)C(=O)NCCCF)CC2)CN1 S(=O)(=O)(c1nc(N2CCC(C)CC2)ccc1Br)NC(c1cc(C)cc(C)c1)CO Cc1ccc(CCC(=O)NCCC2(NC(=O)C(O)CC3CC3)CC2)c(C)c1 Cc1cc(C)c(C(=O)NC(C)CC(C)NC(c2ccns2)=O)o1 N1(C(c2c(C#C)c[nH]n2)=O)CCC(O)C(NC(c2ccccc2OC(C)C)=O)C1 c1(C(N(C(C)CCNC(C2C3COCC23)=O)C)=O)ccncc1Cl C=C(Cl)C(C)(C)C(=O)NCC1CN(C(C2(C)CC2C(F)(F)F)=O)C1 c1(N2CCCC(NC(C(C)C(=O)N3CCOCC3)=O)C2)cc(=O)n(C)c(O)n1 C1(C(=O)NCC2(c3ccccc3)CC2)CCNCCC1(F)F C(=O)C(C)(C)CN1CCOCC1.C1(CC(=O)N)CCS(=O)(=O)C1.C=CCCC c1(C(C)N(CC(C)C)C)cc(C(C)(C)C)cc(C(C)(C)C)c1.Cc1ccnn1C C#CC1CCCN1C(C1C=CCN(C(=O)CNC(=O)CC(C)C)C1)=O C(C(C)CN=c1nc(Cl)[nH]c(C)c1C#N)NC(C(CCC)C(C)C)=O c1(CCOC)nc(C23CC2CN(C(C)=O)C3)n(-c2ccc(OC(F)(F)F)cc2)n1 c1(C(=O)NCCN(C(C=C(C)C(C)C)=O)C2CC2)c(Cl)cccc1[N+](=O)[O-] N1(C(c2cc(C)c(C)nn2)=O)C2CCC1CC(NC(C1CCCC13CCC3)=O)C2 c1(C=O)ccc2cc[nH]c2n1.C(=O)(CCCCC1CC1)NCC(C)(C)OCC.N C1(NC(Cc2cc(OC)no2)=O)CN(C(=O)C(C)(C)CF)CC1C c1(C(N2CC(C)C(CNC(C3(O)CC4CCC3C4)=O)C2)=O)cnc2[nH]cncc1-2 Cn1cc(C#CCN=c2[nH]c(=NCC3CC34CC4)c3cccc(F)c3[nH]2)cn1 N1(C(c2occ(C)c2)=O)CC(N(C(=O)Cc2cncn2C2CC2)C)C(O)C1 N1(C(c2c(C)ncn2C)=O)CC(NC(c2cc(C(N)=O)ccn2)=O)CC(F)C1 c1(C(N2C(CC#N)CN(C(c3csc(Cl)n3)=O)CC2)=O)cc2ccccc2cn1 C1(CC(=O)NCCC2CCN(C(C(CSC)OC)=O)C2)CC2(CCO1)CC2 C#Cc1ccc(C(=O)NC2(C(=O)NC(CC)CO)CC2)cn1 Cc1cc(C)c(C(N2CCC(C)(C)C(CNC(c3ccncn3)=O)C2)=O)cc1N c1(C(CC(=O)N(CCNC(C2(C(CC)=O)CC2)=O)CC)O)cccc(F)c1 C1CCN(C(=O)C(C)(C)C2CCC2)CC1.C(c1cnn(C)c1)=CC(=O)N(C)C CCC(C)(CNC(=O)CC(=O)NC1CC1)NC(=O)CC1(C)CCCC1 C1(NC(c2c(CC)nns2)=O)CN(C(=O)C(C)Cc2cccc(F)c2)CCC1C C(c1ccccc1)=CC(=O)NCC(C1CC1)NC(=O)Cc1cn[nH]c1 c1(C(N2CC3CN(C(c4cocn4)=O)C3C2)=O)cc(Br)nc(Br)c1 CC(C)(C(=O)NCCCc1ccccc1)NC=O.c1(C(=O)N)cn(C2CC2)nn1 c1(-c2cn(CC(C)NC(=O)C(C)(O)C3CCCCC3)nn2)cnc2ccccn12 C(C1=CCN(C(=O)C(Cl)=CCl)CC1)NC(C1CCC(CCC)CC1)=O C1(N(C)C)(C(=O)NCC(C)(CO)NC(c2cncs2)=O)CCCSC1 C=Cc1cncc(C(=O)N(C(C)CCNC(=O)Cc2cccnc2O)C)c1 CCC(C)(C)C(=O)NC1CC1CNC(=O)C(F)(F)Oc1ccccc1 C1(CNC(c2cnc(CC)[nH]2)=O)COCCN1C(=O)COCCOC CC1(C)Cc2cc(C(=O)NC3CCCC3C)ccc2O1.C(=O)(CCP(C)(C)=O)N c1(C(=O)NC2CC(NC(Cc3c(C)nsc3)=O)C2)cc(N)ccc1Cl N1(C(c2cnc(SC)s2)=O)CC23CCCC2(C1)CN(C(=O)Cc1nncs1)C3 Nc1cc2ccccc2c(C(N2CC3(C2)SCCC3NC(c2cncs2)=O)=O)n1 C1(CNC(Cn2c(C(C)C)nnn2)=O)(NC(c2ccsc2)=O)CC2CCC1CC2 C(=O)(CCCC(=O)N1CC2CC(NC(=O)Cc3ccn(C)n3)C2C1)NC C1(CCNC(C2N(CC)CC2)=O)CCN(C(=O)C2=CCCCO2)CCC1(F)F c1(C(N(C2CCN(C(c3ncccn3)=O)C2)CC)=O)ccc([N+](=O)[O-])cc1Cl Cc1cc(CN2CCCCC2C(=O)NCC(F)CO)cc(C)n1 Cc1onc(C2CC2)c1C(=O)NCCN(C1CCCCCC1)C(=O)CC(C)F c1(C(N2CC3CCCC(NC(C(C)=CC)=O)C3C2)=O)cncc2c(O)nccc12 C1(C(C)NC(c2csc(F)c2)=O)CCCCN1C(C1CC(n2cnnc2)C1)=O C(CCCCC(=O)N1CCCC1CNC(c1cc(=O)n(C)cn1)=O)OCC N1(C(CCCCN(C(c2c(CC)ccs2)=O)C)=O)CC2(C1)CN(C(C)C)C2 N1(C(c2c(C)cns2)=O)CCC(C(F)(F)F)CC1CNC(c1cccnc1N)=O c1(C(=O)NCC2N(C(C(CCC)C)=O)CCCC2)cc(C)cc(F)c1F CON(Cc1ccc(C)o1)C(=O)C(CC(F)F)N(C(=O)CCC1CC(C)C1)C c1(CC(N2C3C(NC(Cc4nc(C)[nH]n4)=O)C(C3)C2)=O)c[nH]c2c(C)cccc12 N1(C(C23C4C5C(C(=O)O)C(C2C4)C53)=O)CCCC(O)(C2CC2)C1.c1cccnc1.N CC(C)(CC(=O)N1CCCOC(CCNC(c2ccc(F)cc2F)=O)C1)C(F)F N1(C(C(CC)N(C)C)=O)CCC(C)C1CNC(c1cnn(CCF)c1)=O C(=O)(CC1=CCCC1)NCC(CC(=O)NC(C)Cc1ccncc1)O c1(C(=O)NC2CN(C(C(C3CCC3)OC)=O)CC2O)cc2c(nc1O)CCOC2 C1(CC)CN(C)CCCN1C(C1CC1(C)C)=O.c1(C(=O)N)cc(C(N)=O)[nH]n1 C(=O)(C#CC1CCCC1)N.c1(C(CC(=O)NC2CC2)NC(C)=O)ccc(Cl)cc1 c1(C(N2CCCC(C3(C)COC(=O)N3)C2)=O)cc(Cl)cc2c1OCC2 c1(OC)cccc2c1C(C(=O)N1CCCN(C(c3cccc[n+]3[O-])=O)CC1)CC2 C1(CC(=O)NCCC)COC(C)(C)CO1.C1(C(C)(C)C)(C(=O)N)CCCC1 c1(OC)ccc(NC(C2(C)CCCN(C(C3CC3C)=O)C2)=O)cc1C c1(C(=O)Nc2scc(CC(=O)Nc3cc(OC)n[nH]3)n2)ccc(O)c(O)c1O c1(OC(C)C)cc(C(=O)NCC2C3CN(C(C4CC4(C)C)=O)CC23)ccn1 C1(OC)CN(C(=O)Cc2scnc2C)CC1NC(C1CC1CF)=O CC1(C(N2CC3CC(C2)N(C(=O)COC(F)F)C3)=O)CC(C(F)(F)F)=NO1 c1(C(=O)NCC2C(NC(CCc3c(C#N)cccc3)=O)C2)ncn2c1CCCC2 c1(C(=O)NCC(C)(C)NC(c2csc(C(F)F)c2)=O)[nH]nc2ncccc12 c1(C=O)ccc(C=O)cn1.C1(C(N(C(C)C2CC2)C)=O)CSCC(=O)N1.CO N1(C(C(CSCC)NC(=O)Cc2ccno2)=O)CC(F)(F)C1C1CC1.C N1(C(C(C)(CSC)NC(CCCCC=CC)=O)=O)CC(C)OC(C)(C)C1 n1(CC)nc(C)c2cc(C(N3CC(NC(=O)C4=CSCS4)C4(CCC4)C3)=O)sc12 N1(c2cc(N(C3CC4CNC3C4)C)ncn2)CCn2c(cc3c(Cl)cccc23)C1 c1(C(=O)NC(CNC(COc2ccc(OCC)cc2)=O)C)ccc(C)cc1C C1(NC(CC2(OC)CCC2)=O)CCN(C(c2ccc(F)cc2SC)=O)C12CC2 C1CC(O)C(O)C1.C1(CCC=C)(C(=O)N)CN(C(c2cn(C3CC3)cn2)=O)C1 c1(NC(CCCC(C)NC(C(C2CCC2)OC)=O)=O)cnc2[nH]cnc2c1 O=C(C1CNc2ccccc21)NCC1CCN1C(C1CSCC(=O)N1)=O C1(CC=O)CCCC(F)(F)C1.Cc1cn(C(C)(C)C(=O)NC2CCC2)cn1.C N1(C(C(C)c2ccsc2)=O)CC2(CNC(=O)Cc3cnnn3C)CC1CO2 N1(C(C)=O)CCCCC1CC(=O)NCCN(C(C1CCC(=O)O1)=O)C1CC1 C(C)(C(C(=O)N)C(C)C)NC(c1cc(C)cc(O)c1)=O.c1cnn(CC(N)=O)c1 c1(N2CCN(C(c3cscn3)=O)CC2CCO)ncnc2[nH]c3ccccc3c12 c1(NC(CC)CCOC)[nH]c(=NCCOC2CCOCC2)nc2c1ncn2C CC(CN1CCOC1=O)CN=C(NCC1COC(C)(C)OC1)NC1CC1 C(c1ccn(C)c1)=CC(N1CC(C)C1C(=O)NCCC1C=CCC1)=O C(=O)(C1=CCS(=O)(=O)C1)N1C(CC)CSCC1.N1(C(C)C)C(=O)CCC1C=O c1(C(=O)NCC(C2CCC2)NC(=O)CO)csc([N+](=O)[O-])c1 CC(O)(C(=O)NCCNC(C1C=CCCC1)=O)C1CC1 C(c1nnc(C(C)C)o1)=CC(N1C(CNC(C(COC)C)=O)CCC1)=O C(=O)(C(C)(C)CCCF)NCCC(C(=O)NCC1CC(C(=O)OC)C1)O C1(CNC(c2ccc(CC)[nH]2)=O)C2CN(C(C3CC4CC4C3)=O)CC12 c1(N2CC(NC(=O)CCc3ccccn3)C(F)CC2)ncc2c(Cl)cccc2n1 CCC(CNC(=O)CC1C2CN(C(=O)CNC(C)=O)CC12)CCO N1(C(c2c[nH]nc2C)C(=O)NC(CC)C)CCC(Oc2ccccc2)CC1 C1CC2(C1)CC(C(=O)N(C(C)C)C)C2.c1(C=O)ccccc1C(C)(C)C.C Cc1nc(C(N2CCC(N(C(=O)C(c3ccccc3)N(C)C)CCO)C2)=O)cs1 c1(C(N2C(CNC(=O)C(C)(C)C)CCC(C)C2)=O)cc2c(s1)CCCNC2=O C(=O)(C1=CC2(CCN(C(c3sc(C)nc3C)=O)C2)C1)NCC(COC)(C)O c1(CC)nc(C(=O)NCC(O)CNC(=O)Cc2ccsn2)co1 c1(C(=O)NCC(CNC(Cn2ncc(C#C)c2)=O)O)cccn2nnnc12 CC(C)C(O)C(C)C(=O)N1CCCC(NC(c2ccc(C(F)(F)F)cc2)=O)CC1 c1(C(=O)NC2CCC(N(C(c3n(CCC)ccc3)=O)C)C2)cccc2[nH]ccc12 C1(NC(c2n(C)cnn2)c2nnnn2C2CCOCC2)C2CCCOC12 C12(C=O)CC(C)(CCO1)C2.c1(SC)cc(C(=O)NC2CCCCC2)c(C)o1.C c1(C(=O)NC2C3CN(C(c4scc(OC)c4)=O)CC32)c(Cl)ccc(OC)c1N C1(NC(C=NOC)=O)CCCOC1C1CCN(C(c2cc(O)n(C)n2)=O)CC1 c1(CN(CCC(N2CCCCC2)=O)C)c(N)cccc1F.c12cncc(c1)NC2 C1(CC#C)CCN(C(C2CC(OC)CN2C(C2CC3(CC3)CO2)=O)=O)CC1 c1(C(=O)NCC(CCNC(C(C)(C)c2cc[nH]n2)=O)O)ccc2occc2c1 c1(OC)cnc(CNC(=O)CCN(C)C(c2scnc2Cl)=O)cn1 C1(NC(CCNC(COC)=O)=O)CCC2(CC1)CN(C(c1ccoc1)=O)CCO2 CC1CN(C(C2CCC2)=O)CC1(C)CNC(=O)CC1CCCCN1C C(C(C)(CC)CO)NC(COCCNC(c1c(CC)cco1)=O)=O C12(C(N(C)CCNC(c3ncnn3C3CCOCC3)=O)=O)CCC(C)(C1)OC2 c1(C=O)ccc(S(C)(=O)=O)s1.C1(C(N2CC(CC=C)C2)=O)OCCN(C)C1=O N1(C(C(CC)N(CC)CC)=O)CC(CNC(C2(CC)CCOCC2)=O)C(O)C1 N1(C(C23CCC(OC)C2C3)=O)CCC(C(=O)N(C2CC3CCC2CC3)C)=C(F)C1 c1(OC)cc(C(=O)N(CC(=O)NCC)C(C)C)[nH]n1.C(=O)(C1CC1)N C1(CC(=O)NCCC(C)NC(=O)Cn2ccccc2=O)CC(O)C12CCC2 C(=O)(C(C)(C)CC(=O)NCC)OCC.C1(c2ccccc2)(C=O)CCCO1.N C1(CC(=O)N(C2(C(=O)NCCCc3ncn(C)n3)CC2)C)CCC=CCC1 N1(CC(N2CCC(N(C)C(c3ccccc3CO)=O)C2)=O)CCS(=O)(=O)CC1 c1(C(N2CCC(O)(Cn3cc(C4C5CCCCC45)nn3)C2)=O)cnc2ccsc2c1 C(=O)(C(C)C(C)S(C)(=O)=O)N1CCC(NC(c2c(SC)ccs2)=O)C(C)C1 Cc1cc(S(C)(=O)=O)cnc1NCC(F)(F)Sc1ccc(Br)cc1 C1(CC(N2CCOCC2)=O)CCCC(F)(F)C1.c1(OC)nc(C(=O)NC)sc1C N1(C(C2C=C(C)CS2)=O)CC(C)CCC1C(=O)NCCC1CC(C)(C)CO1 N1(C(C(=O)NCC)=O)CC(OC)CC1(C)C.C(C(C)(C)C)N(CC=O)C C(CC(C(=O)NCc1cscc1C)NC(=O)C(C)CN(C)C)=CC N1(C(C=C(C)C(F)F)=O)C(C)CC2CN(C(c3conc3C3(C)COC3)=O)CC12 c1(C(=O)NCc2c(CNC(C(C)C3CCC3)=O)cccc2)cccc2oncc12 S(=O)(=O)(c1ccc(CBr)cc1)NC1C(C(N2CCC(C#C)CC2)=O)C1 c1(C(=O)NC2C(NC(C3CC(C)(O)C3)=O)CCCC2)cnn2c1CCC2 NS(=O)(=O)CCC(=O)N(C1CCCCC1)CCNC(=O)C(=O)NCC(F)F c1(NC(C2CCCN(C(c3c(Cl)cccc3I)=O)C2)=O)cc(Cl)cnc1O c1(CC(=O)NC(C)CCNC(c2cc3ccsc3s2)=O)ccccc1S(C)=O c1(C(CC)C)nccc(N2CCC(C)C2CNC(=O)CCc2nnc(C)n2C)n1 c1(C(=O)NC2(COC)CCN(C(=O)C(C)C(C)C)CC2)cc2cncc(C)c2s1 C1(CC)CCC(CNC(C2(N(C(=O)Cc3csc(C)c3)C)CC2)=O)CC1 CC1(C)CC(NC(=O)Cc2ccc3c(c2)OCO3)CN(C(c2cc(F)n[nH]2)=O)C1 N1(C(C(CCCC)NC(=O)CCn2ccnc2C)=O)C2C=CCC1CCC2 O=C1CN(CC2=CCOCC2)C(=O)N1Cc1cc(C(F)(F)F)co1 C1(C(=O)NCC2(COC)CCCC2)CCC(C)CC1.c1(C=O)cnsn1.N c1(OCCOC)ccc(NC(=O)Nc2ccc(CC(F)(F)F)cc2F)cc1F n1(CC)cc(Br)c(C(c2nnnn2C2(C)CC2)N)n1.C1CC(n2cncn2)C1 N1(C(C(C)N(C(=O)CC2(C)OCCO2)CCC)=O)CCSC(C)CC1 CCN=c1[nH]c(C(N2CCC(N(C(=O)C=CC3CCOC3)C)C2)=O)cs1 n1(CC(=O)NCCCNC(=O)Cc2ccsc2)cnc2sccc2c1=O C(F)(F)C(F)(F)F.C(C(O)C)N(C(COCC(=O)OC)=O)C.C(=O)C c1(C(=O)NCC(OCC)OCC)cnc(Br)s1 Cc1[nH]nc(C(=O)NC(C2CCCN2C(c2cccc(=O)o2)=O)(C)C)c1O C1(NC(CN(C)C(=O)C2CC2)=O)CCCCN(C(=O)CC2CCCCC2)CC1.S CC1(C)CC(=O)NCC1C(=O)NC12CC(C1)C2.C1(C=O)CCC=CCCC1.C c1(C(=O)NCc2ccnn2CC(F)F)cc2c(s1)CNCC2 Cc1c(C(N2CC(CCCCNC(=O)CCc3cnoc3)C2)=O)ccn1C C1(C(N2CCC(C)C2CNC(c2cn(C)c(=O)n2C)=O)=O)CCCC(=O)N1C c1(C(N2CCC(N(C(c3nc(C)[nH]n3)=O)C)C2)=O)ccn(CC2CC2)c1C C#CCC(CC#C)C(=O)N1CCC(C)(C)C(C)C1.C(c1cc(C)no1)=CC(=O)N C1(C(=O)NCCC2(CO)CC2)CC12CCN(C(c1cccc3c1CCC3)=O)CC2 N1(CC)CC(C(=O)NC2CCC(NC(=O)CO)C2)CCC1=O.CC(C)(C)C C1(OC)CCCC(c2nnnn2C2CCCCC2)(NCC2CC3(CC3)C2)CC1 C1(CCOC)(NC(=O)C(c2ccccc2)C2CC2)CCN(CCF)CC1 c1(C(=O)NCCN(C(CCC2CCC(C)O2)=O)C2CCCC2)cn2ccsc2n1 C(=O)(C1CCSc2ccccc21)NCC(CNC(c1c(C)cc[nH]1)=O)C N1(C(CCC=C=C)=O)CCCC2CN(C(c3ccnc4ncnn34)=O)CCC12 CC1(C)CN(C(C2CCCOCC2)=O)CC1NC(c1ccc(Cl)cn1)=O CS(=O)(=O)c1ccc(C(=O)NCC2CC2NC(c2ccc(O)nc2)=O)s1 C(=O)C1c2c[nH]nc2CCC1C.c1(CCN(CCC)CC)c[nH]c2ccc(C)cc12 N1(C(CNC(CC(C)C)=O)=O)CCCC(F)(C(=O)NC23CC=CC(C2)OC3)C1 C1(CC)CC(C(=O)Nc2cnc(Cl)cc2C)CCN1C(C1CC1C(N)=O)=O Cc1cc(C)c(CC(=O)Nc2ccc(C(=O)N=c3[nH]nco3)cn2)c(C)c1 C(CC(C)C)(C=O)NC(=O)OC.C1(S(C)(=O)=O)(C=O)CCC1.C1CCC1 CC(C)(O)C(F)C(=O)NCc1ccsc1C(N1CCOC(C2CC2)C1)=O c1(NC2C(F)CCN(C(CCN(C(C)=O)C)=O)C2)ncc2c(C)cn(C)c2n1 N1(C(C(=O)NCCCSCC)c2cnsc2)CCC(OC)C1C1CC1 N1(C(C2C(C)CC=CC2)=O)CCCCCC(NC(C2CC3C=CC2C32CC2)=O)C1 C1(CCC(=O)N(CCO)Cc2ccsc2)NCC2CNCC1C2 C1(O)(C(C)NC(c2coc(Br)n2)=O)CCN(C(c2ccncc2N)=O)C1 c1(C(=O)OC)nc(C2CCCN2C(=O)CCC2CC2(C)C)sc1C C1(C(N2CC(SC)C2)=O)CC12CC(NC(=O)CCN1CCCC1=O)C2 C1(C(=O)N)CC(=O)NC(C)C1.C(CCCCC)N(C(c1nc(COC)oc1)=O)C CCC(C)(C(=O)N1CCC(NC(c2cc(OC)ccn2)=O)C(CO)C1)C(N)=O C1(OC)CCCN(C(=O)C=CCN(C)C(c2ccnnc2O)=O)C1 C1(C(=O)NC(CC)C(C)(C)O)N(C(c2c[nH][nH]c2=N)=O)CCC1(C)C N1(C(C(C)SCC)=O)CCC2(CCC(NC(=O)C#CC3CCOCC3)C2)C1 C=CC1CN(C(C2CCOCC2NC(=O)C(C)c2ccco2)=O)CCO1 c1(NC(C)=O)ccc(C)c(C(=O)NC2CC(O)CN(Cc3ncc[nH]c3=O)C2)c1 C1(C(NOCC(=C)Cl)=O)C2CC3C(C2NC(C2CCCCNC2=O)=O)C13 C1(CC(=O)N)CCS(=O)(=O)C1.C(=O)(CCc1cn(-c2ccccc2)nn1)OC N1(C(C2(OC)CCOC2)=O)CCC(N=[N+]=[N-])C1.C12(CC(=O)N)COC(C1)C2 CCC(CC1CCCC1)C(=O)N(C1CCC(NC(c2cc(OC)no2)=O)CC1)C C1(C(=O)NC2CCC(N(C(c3n(CC#C)cnn3)=O)C)CC2)CCCC(C)(C)C1 CCC(=O)CCC(=O)N1CC(C(=O)NCc2ccncc2F)C(F)(F)C1 C1(CNC(C2N(CC)CC2)=O)CCC2CN(C(c3cc(O)ccc3C)=O)CC12 c1(N2CCC(N(CC(F)F)CC)CC2)nc(N2CCC=C(C)C2)cc(C)n1 C(=O)(C1=CCOCC1)NCC(c1cccnc1)N(C)C C1(C(=O)NC(CCC)C(=O)OC)CCN(C(=O)CC(C)F)O1 Cc1cc(C(=O)NC2CC(C)(NC(c3cccnc3N)=O)C2)ccn1 CC(C)CC(C(N)=O)NC(C1CCCN(C(=O)CCOC2CCC2)CC1)=O N1(C(CSCC)=O)CCC(CNC(=O)CCc2ccc(O)c(F)c2)C(C)C1 C1(C(=O)NC(c2ncccn2)C)CC2(C1)CN(C(C1(CO)CCCCC1)=O)C2 Cc1nc([N+](=O)[O-])cn1CC(N1CC(NC(C2CC2C)=O)C(C)C1)=O CCCC(C(=O)NC1CCC(CCNC(=O)CNC=O)C1)NC(N)=O Cc1ocnc1CC(=O)NCC1CC1CNC(C1(CO)COC1)=O c1(OC)ccc(OC)c(C(=O)NC2CC2C)c1.c1(C=O)cn2c(n1)SCC2 C(=O)(CS(=O)(=O)CCO)NCc1[nH]nc(C(N(CCCC)CC)=O)c1C CCN=c1ccc(C(=O)NC2CCOCC2NC(C2CC2CC)=O)c[nH]1 C#Cc1ccc(C(=O)NC2CN(C(c3ccc(N)c(Cl)n3)=O)CCC2F)cc1C c1(N2CCC(C)(C)C(CO)C2)nc(=N)[nH]c(=NC2CCCCC2CCO)[nH]1 CCCCCS(=O)(=O)CC(=O)N1CCN(C(C23CC(C)C2C3)=O)CC1C c1(CC)cc(C(=O)NC2CCC2)nn1C(C)(C)C.C(=O)CC.C(C)(C)C C1(C(N(CC(CO)(CO)NC(C2CC2(C)C)=O)C)=O)CC1C1(C)COC1 N1(C(C(C=C)(C)O)=O)C2CCCC1CN(C(c1c(-c3cccs3)noc1C)=O)C2 N1(C(C2CC(N=[N+]=[N-])C2)=O)CCC2(CCC2)C(NC(=O)CCCC(F)(F)F)C1 c1(C(=O)NCC(CNC(C(CCC)NC(C)=O)=O)C)ccc(Br)c(O)n1 C1(CC(N2C(CNC(C(C)OCCC=C)=O)CC2)=O)COCCN1CC c1(C(N2CCC(C)(NC(CC3C(C)OCC3)=O)CC2)=O)cc2cnc(Cl)cc2s1 N1(C(=O)CCc2cn[nH]c2)CCC(O)(C(=O)N(C2CC2)Cc2ccncc2)CC1 c1(C(N(CC=O)CC(C)C)=O)cc([N+](=O)[O-])n[nH]1.CCC.C(=O)(OC)N c1(SC)cc(C)ccc1C(=O)NC1CC(CC)C1.c1(C=O)ccc(O)nc1Cl.N C1(CC=O)N(C(C2CCCCC(=O)N2)=O)CCC1(C)C.n1(CC)cc(C)cn1.N CC(=O)CCCC(C)C(=O)NC1(CC(=O)NCCc2cn[nH]c2)CC1 C1(C(N2CCC(C(C)C)C2)=O)Cc2cccc(F)c2C(=O)O1 C(CC(O)C(=O)NCC(Cc1ccccc1)SC)SC c1(C=O)c(F)cccc1F.c1(C(=O)NCC(C)C)ccc(CC2CCC2)cc1.N C1(C(=O)NCCc2c(C)ocn2)CCOCCN1C(C1CCS1(=O)=O)=O CC(C(=O)NC(C1CCN(C(c2cnc[nH]2)=O)CC1)(C)C)P(C)(C)=O c1(C(N)=O)ccc(NCc2cc(-c3ccccc3Cl)on2)nc1 c1(CNC2CC(CC(=O)Nc3nc(C)c(Cl)s3)C2)cc(Cl)c(Cl)cc1Cl N1(C(C(C(=O)OC)(C)C)=O)CCCCNC(=O)C(F)(F)C1 C1(C)(OCC)CCN(C(c2c(CNC(=O)C(C)(C)SC)nnn2C)=O)CC1 c1(C(=O)NC2C(NC(c3cccc(C)c3F)=O)CCC2)cnc2c(c1)CCCC2 C1CCC(C)CN1C(=O)Cc1cnn(C)c1C.c1(CC)sc(=N)[nH]c1C(=O)N c1(C(N2CCN(C(=O)C=Cc3nccs3)C(C3CC3)C2)=O)cnn2ncccc12 c1(C(N(CCCCN(C(=O)C(CO)NC(N)=O)C)C)=O)cccc2ncccc12 Cc1cc(S(=O)(=O)N2CC(O)CC2C(=O)Nc2cc(F)ccn2)c(C)cc1Cl C1(C(N2CCC(C(C(=O)OCC)C#N)CC2)=O)CCc2ccccc2C1 Cc1ccc(C(N2CCCCC(NC(C3CC34CC4)=O)C2)=O)c(O)c1C c1(C(C=O)(F)F)cccc(Cl)c1.N1(C(CN(CCOC)C)=O)CC=CC1C.N C1(CC(=O)N(CC(C)NC(C2N(C(C)=O)CSC2)=O)C)CCC(F)(F)C1 C(=O)(C(C)CCC(C)(C)C)N1CCCCC1.c1(C(N(CC)C)=O)cc(C)cnc1Cl C(=O)(CCC1CCc2ccccc21)NCCCC(C)NC(c1ccc(C)o1)=O C(C1c2ccsc2CCN1C(=O)C=CC(F)(F)F)NC(C(CC=CCC)C)=O C1(NC(c2cccc[n+]2[O-])=O)CN(C(c2csnc2Br)=O)CC1F N1(C(c2ccc(CN(C)C)[nH]2)=O)CCC(O)CC1.C(=O)C(C)(C)CN(C)C.N C1(C(=O)OC)(NC(=O)C(C(C)C)n2cncn2)CCCCC1.C1C(=O)N1.CC C#CCC(C)(CNC(=O)CN(C(=O)CC(C)COC)C)CO C1(C)(C(=O)OCC)CCCN(C(c2sccc2-c2cc(F)ccc2F)=O)C1 C1(NC)CCCN(C(=O)CCOCCN(C)C(C2CC(C(C)C)C2)=O)C1 c1(C(N2C3CC(CNC(C(CCC)C)=O)CC2CC3)=O)ccc2c(c1)CN(C)C2 CCC(CC(=O)NC(C1CCN(C(=O)C=Cc2cn[nH]c2)CC1)C(C)C)C1CC1 C1(C(=O)NC2CCN(C(C3CC(N(C)C)C3)=O)CC2)CCc2cc(F)ccc2O1 C1(CC)CN(C(=O)C2CC2)CCC1NCc1cn(-c2cnnc(O)c2Br)nn1 C12(CC)CN(C(=O)CC3CCCO3)C(C1)C2.c1(C=O)[nH]nnc1C1CC1.C CCC(C#N)(CC)C(=O)N1CC(OC)C(NC(=O)Cc2csc(Cl)n2)C1 c1(C(=O)NCC2N(C)CCN(C(CC(CCC)O)=O)C2)cc2c(Cl)cccc2[nH]1 N1(C(C(C)OC(=O)OCC)=O)CCCC(F)C1.C(=O)(C(F)=C(C)C)N C(CC(C)CCNC(=O)C=C(C)I)NC(CC1CC(=C)C1)=O O=C(N1OC2C=CC1CC2)C1CCC2(CC2)N1C(=O)CSC1CC1 C1(C)(CC(=O)NCCCC#C)CCN(C(C2CC(N(C)CC)C2)=O)C1 N1(C(c2ccnc(C)n2)=O)CC2(CCN2C(=O)C(C(C)(C)C)N(C)C)C1 C1(C2CN(C(C3CC3(F)F)=O)C2)(NC(c2cc(C(=O)OC)[nH]c2)=O)CC1 n1(CC)c(C(=O)NC2CCC2NC(c2cnc(SC)n2C)=O)cc2ccccc12 C1(NC(c2ccc3c(c2)CC3)=O)CCSC12CN(C(C1CC3(CCCC3)C1)=O)C2 C(=O)(CC(C)(C)CNC(C12CCCCC1C2)=O)Nc1c(C(C)C)n(C)nc1 c1(C(=O)OC2CC(N(CCC)CC)C2(C)C)cc(C(N)=O)cc([N+](=O)[O-])c1 CC(CC(F)(F)F)C(=O)N1CCCC(C)(CNC(=O)Cc2cccs2)C1 C1(C(=O)OC)CCCN(C(=O)CC(c2ccc(F)cc2)NC(C2CCCO2)=O)C1 N1(C(c2c(N)ccc(N(C)C)c2)=O)CCC2CN(C(C3(O)CCC3)=O)CCC2C1 N1(C(C2(C(=O)OCC)CCCOC2)=O)CCc2cc(OC)c(OC)cc21 Cc1cc(C(=O)NCCC(C)(C)NC(=O)CC(C)O)ccc1C#N C1(CN(C(COCCCC#C)=O)C)CCCC(NC(c2csc(Cl)c2)=O)C1.O CC(C)CC(C)C(=O)NCC1(NC(=O)C=Cc2ccc(F)cc2)CCOC1 N1(C(c2scc(CNC(CCOC)=O)c2)=O)CCS(=O)C(C)C1 Cc1ccc(CN2CCCC(CNC(C3CCCCO3)=O)C2)cc1Br C1(NC(c2cc(Cl)nc(Cl)c2)=O)CCC2CN(C(=O)CC3(O)CCC3)CC2C1 C1(C(=O)NCCn2c(C)nc(C)n2)CCCN(C(=O)C=Cc2ccccc2)CC1 c1(OCC(=O)NC2CCCCC2NC(c2nccnc2Cl)=O)ccc(Br)nc1 C1(NC(c2ccncc2)C)COc2ccc(F)cc2C1 N1(C2CC2)CCOC(CCCNC(c2ccn(CCOC)n2)=O)C1.C1(C)CC1 CCCC(C)NC(C1(C=O)CC=CC1)=O.C1(C=O)CC=CCC1.C(C)(C)C.O N1(C(C2C(c3nc(C)[nH]n3)C2(C)C)=O)CCC(CO)(NC(=O)C2=CCC2)CC1 Cc1sc2ncnc(N3CCN(C(C4CN(C)CCO4)=O)CC(O)C3)c2c1C C(F)(F)(C(=O)NCCC(C)(C)NC(=O)CCc1ccccn1)C1(OC)CCC1 c1ccc(S(=O)(=O)CC)cc1.N1(C(C23CC(N)(C2)C3)=O)CCCC(F)(F)CC1 c1(C(=O)NCCC2OCCN(C(C3(OC)CC3)=O)C2)c(F)ccc2n[nH]cc12 O=C(CCCCC1CC1)OCc1csc(C(F)(F)F)c1 c1(N(C(c2nc(C(C)OCC)sc2)=O)C)cccc(S(F)(F)(F)(F)F)c1 c1(C(=O)NCC2CC(NC(C(CC)(F)F)=O)C2)cnc2c(Cl)cccn12 N1(C(c2occ(C)n2)C(=O)NCSc2ccccc2)CCOc2cccc(Br)c2C1 N1(C(C(CCOC)C)=O)CC2(CCCN(C(=O)CC34COC(C)(C3)C4)C2)C1 N1(C(C(C(C)C)F)=O)CC2(CC(CNC(=O)C=C3CCC3)C2)C1 C1(C(N2CC(C)(NC(=O)Cn3cnc(Br)n3)C2)=O)(C(F)F)CCCCC1 CCCC(C(O)C(=O)NC(C)COC)NC(=O)Cn1ccccc1=O C1(CNC(C(=O)NC(c2c(OC)ccc(F)c2)C)=O)CCC12CCOCC2 C(=O)(CCCCC(N)=O)N1CC(CC(=O)NC2(C=C)CCC2)C(C)CC1 c1(C(=O)N)c(C)cc(Cl)cc1C.N1(C(CNC(C(CC)C)=O)=O)CCC(C)(C)C1 N1(C(c2c(CC)c[nH]n2)=O)CCN(C(=O)CC2CCSCC2)C2CCCC12 C(=O)(C1=CCCCC1)NC(C(C1CCCCC1)NC(Cn1c(C)csc1=O)=O)C Cc1cc(C(=O)N(CC(C)N(C(=O)Cc2ccno2)C)C)nn1CCO N1(C(c2c(C)sc(O)n2)=O)CCN(C(=O)C(C)(C)c2ccccc2)CC2(CC2)C1 C1(NC(CCC2CC(N)C2)=O)CNCCS(=O)(=O)C1 C1(C(=O)NC2CCOCC2O)CN(c2nnc(C3CC3)o2)CCC1O C1(NC(=O)Cn2cc(Cl)cn2)CC2CC(C1)N(C(=O)C1=CS(=O)CCC1)C2 c1(C2C(C(=O)NC(C)CNC(c3cccn3C)=O)C2)ccc(Cl)cc1 C1(CC(=O)NCCNC(=O)CS(=O)(=O)CCO)CCC2(CCOCC2)CO1 c1(OCC)ccc(CNC(c2ccc(-c3nnc(C4CC4)o3)cc2)=O)cc1 Nc1c(C(=O)NCCC2CCN(C(=O)C(F)=CC3CC3)CC2)ccc(Cl)c1Cl N1(C(c2n(C=C)nnc2)=O)CCC(C)C(CC(=O)Nc2c(O)cccc2Cl)C1 C1(C(=O)NC(C(CC)O)C)CC12CCCCCC2 C=Cc1ccc(C(=O)NC2CCN(C(C3CC(SC)C3)=O)C2(C)C)cc1 C1(CCC)CC(=O)N(Cc2ccc(C(=O)NC)nc2)C(=O)N1 C#CCC(C(=O)NCC)C1CC1.n1(CC(=O)N)cc(C2CC2)nn1.C1CC1 C1(NC(CSC)=O)CCN(C(C2CCC2c2nc[nH]n2)=O)C1C1CC1 C1(C(=O)NCC(C)O)C2CC2CN1C(=O)C(O)CN1CCCC1 N1(C(C(CC)C(C)C)=O)CC(C)CN(C(C2(O)COC2)=O)CC1C N1(C(C2C(CCC)C2)=O)CCC(F)(CNC(c2cc[nH]c2CC)=O)CC1 N1(C(c2c(OC)nc(-c3cnc(F)c(F)c3)cc2)=O)CCCC2CCCCC12 c1(C(N(CCCCCNC(C2(CSC)CCC2)=O)C)=O)cc2n(n1)CCCO2 CC1(NC(c2[nH]nnc2C2CC2)=O)CCCC1.n1(CC=O)nnc(C2CC2)n1 c1(OC)ncc(C(N2CC(C)C(C)(C)C2)=O)nc1C.c1(C=O)c[nH]c(C#N)c1.N CC1CC2(CCO1)CC2C(N1CC(O)(C(C)NC(c2csnn2)=O)C1)=O Cc1cc(C(N2CC3C(CNC(c4ccnn4C)=O)C3C2)=O)cnc1C c1(C(CF)NC2CNCC(N(C)C)C2)ccc(C#N)cc1 C1(N(C(=O)CSS(C)(=O)=O)C)CCCN(C(=O)C2=CCOCC2)CC1 c1(NC(C2C(NC(=O)C=Cc3cnccn3)C2)=O)n[nH]c2ncc(Br)cc12 c1(C(N(CCN(c2ncc(C(C)=O)cc2C)C)C)=O)ncc2ccccn12 N1(C(c2cc(OC)ns2)=O)CCC(NC(=O)Cc2ccon2)C1c1ccccc1 CC(C)P(=O)(CC(=O)N1CC2CCN(C(c3cncc(O)c3)=O)C(C2)C1)C(C)C CCCC(CCCNC(c1ccc[nH]1)=O)NC(c1ccn(CC(F)F)n1)=O Cc1c(Cl)ccc(C(N2CC(NCc3cc(Cl)cc(C)c3O)C3(CC3)C2)=O)c1Cl N1(C(c2c(C)nn(C)c2)=O)CCC2(CCN(c3ncnn4c(Br)ccc34)C2)C1 C1(C(=O)NC2CC(F)(CNC(C3(C)C(C)C3)=O)C2)CC2CCC1CC2 c1(C(=O)N)cc(S(N)(=O)=O)cs1.Nc1ccnc(C(N2CC3C(C)C3C2)=O)c1 Cc1c[nH]cc1C(=O)NCc1occc1C(=O)N.C1(CC2CCC2)CCC1 C(=O)(CC(CC)CCC)N(C1CCCN(C(C2CCC(=C)CC2)=O)C1)CCO C(CC(=O)NCc1cccc(O)c1F)(C(C)C)NC(Cc1c(C)n(C)nc1)=O CC1CN(C(C2(C)CCCOC2)=O)CCC1C(=O)NC1CN(C)CCC1O C1(CNC(c2ncn(C)c2)=O)CCN(C(=O)CC2CCCC23CC3)CC1C1CC1 N1(C(C=CC2(C)COC2)=O)CC(NC(C2CCn3cncc3C2)=O)C2(CCC2)C1 CC1CN(C(=O)CC(O)CNC(=O)Cc2ccnn2C)CC1N(C)C N1(C(c2c(C)oc(C(C)C)n2)=O)CCC2CCC(NC(C3CC34CC4)=O)C12 C1(CNC(CSCCC)=O)(CO)CCN(C(C2CC2CN(C)C)=O)C1 C(=O)(C#CC1CCCO1)NC1CCN(C(c2cc(C(C)(C)F)c(F)cc2)=O)CC1 c1(C(=O)NC2CCCC(CNC(c3cn(C)nc3)=O)C2)ccc2ccoc2c1 C(=O)(CC(C)C(C)(C)NC(c1csc(F)c1)=O)NCCc1c(C)noc1C c1(-c2nc(C3(CC)CCCCC3)on2)c(F)ccc(F)c1Cl C1(NC(C(CC)F)=O)CN(C(c2ccnn2C(F)F)=O)CC12CC2 C1(C(N2C(COC)CCCC2)=O)CC12CCN(Cc1nc(Br)ccc1OC)C2 C1CC(CC)N(C(=O)C=Cc2cccs2)C1.c1(C=O)cc(C(N)=O)cs1.CO N(C1CCCc2ccoc21)C(CCC(CC)NC(c1cc(C)n(C)c1C)=O)=O O=C1CCC(c2cn(CC3C=CCN3C(c3cn(CC4CC4)nn3)=O)nn2)CC1 c1(C(=O)NC(C)CNC(C2CC=CCC2)=O)cn(C)nc1C(F)F C=Cc1ccc(C(=O)NC2C=CCN(C(=O)Cc3cnc(C)s3)C2)cc1 N1(C(C2(C)CC(F)(F)C2)=O)CC2(C(=O)NCC3(C)CCOCC3)CCC1CC2 c1(C(=O)NCCC(C)NC(C2OCCN(C)C2=O)=O)cccc2c1CCO2 N1(C(c2ccc(C3CC3(Cl)Cl)cc2)=O)CCN(C(=O)C(F)(F)C2CC2)CC12CC2 c1(C(=O)NCCN(CC(C)O)C(c2c(CC)occ2)=O)ccc(C)cn1 C(=O)(C1=NN(CC(C)C)C(=O)CC1)NC(C1CCN(C(C(CC)C(C)O)=O)C1)C Cc1nnc2n1CC(C(=O)NC13COC(C)(C1)C3)C2.C(=O)C(C)CC(N)=O.N c1(C(N2CCC(NC(=O)Cc3cc[nH]n3)C23CCC3)=O)cc2nccn2c(O)n1 CC(CC(=O)N1CCCC(C2CC2NC(=O)CCC(F)(F)F)C1)CC(F)(F)F C1(O)(C(N2C3CC(C2)C3)=O)CCC(C)(C)CC1.C(=O)C(O)C(C)C.COC CC1CN(C(c2ccn(C)n2)=O)CC(C)N1C(C1CCc2nnnn2C1)=O C1(N(CCC)C(c2nocc2CC)=O)CCN(C(=O)CCc2cnc(C)s2)CC1 C(Cc1ccccc1)(C(=O)OCC1(C(C)(C)C)CCNC1)NC(C)=O CC1(C)CCC(C)(NC(C2CC(O)CN2C(C2CS(=O)C2)=O)=O)C1 c1(C(N2CCc3[nH]nc(CO)c3C2)=O)cc2c(Br)cnn2cn1 N1(C(c2c(OC)csc2)=O)C2CCC1CC(C(N1CCCCC1C#N)=O)C2 CC(C)CCCCC(=O)N1CCC(CC(C)NC(C2NC(=O)OC2C)=O)CC1 c1(C(N(C2CCN(C(c3ccc(=N)[nH]c3)=O)C2)CCC)=O)occ2c1CCOC2 C1(C(N(C)CC2(O)CN(C(c3ccc(CO)nc3)=O)C2)=O)CCCC(F)(F)C1 CCC(C)C(C(=O)N1CC2(CNC(=O)CC(Cl)Cl)CC1CO2)N(C)C C1(NC(CN(C)C(=O)C2CC2)=O)CCN(C(c2ccccc2C(F)F)=O)C1 N1(C(C(=O)NCCSCC(=O)O)=O)CCCC1CO c1(OC)cc(Cl)ccc1C(=O)N(C)C.c1(C(N2CC(O)C2)=O)ccc(F)cc1F Cc1ncc(C(=O)N(C(C)CNC(C2(C)CCCCO2)=O)C)cn1 N1(C(C2CCCC(NC(C(C)(C)N=[N+]=[N-])=O)C2)=O)CCCC2(C=CCO2)C1 C1(NC(C(CC)N(C)C(c2cccnc2C)=O)=O)CC(CO)C2CC12 c1(C(=O)NC2CC(CNC(Cc3n(C)ccn3)=O)C2)cn(C)c2ccccc12 c1(C(=O)NC2CN(C(CC=C=C)=O)CC2CC(C)(C)C)ccc2nc(O)[nH]c2n1 C(CC(CC)C(=O)NC1C=CC(C(=O)NC2CCC23CCCC3)C1)=CC N1(C(c2cnc(C)s2)=O)CCC(C)(C)C1CC(=O)NCC1CCC=CCC1 C1(C(=O)NCC(C)(CC(C)C)NC(CC(=C=C)C)=O)COc2ccccc2O1 N1(C(C(CC(C)C)NC(c2cc(OCC)no2)=O)=O)CCC(O)CC(C)C1 C1(N(C(C(CC)C)=O)CC)CCN(C(C2CCOC2c2cccc(C)c2)=O)CC1 C(=O)(CCCCCCCCC1CC1)NC1CN(C(C=C(C)C(F)F)=O)CC1O CCC(CCCC(=O)N1CC2CC2C1)NC(=O)C1=C(C)OCC1 c1(C(C=O)N(CCN(C)C)CCN(C)C)cc(Br)c(F)cc1F.C=CC.N Cc1nc(C(N2CCOC(C(C)NC(=O)CCS(N)(=O)=O)C2)=O)c2ccnc-2[nH]1 C1(C(=O)NC2COCC(C)(C)C2)CCCCCCN1C(c1ns[nH]c1=O)=O N#Cc1ccc(C(=O)NC2CC(CC(N3CCC4COCC4C3)=O)C2)cc1[N+](=O)[O-] C1(NC(c2c(C)cc(O)nc2)=O)CCCN(C(c2oncc2C)=O)CCC1 N1(C(c2c(CC)cccc2)=O)CC(NC(=O)Cc2ccccc2)CC12CCOC2 c1(CSC)cccc(C(N2CC(N(C)C(c3cc(CCCO)on3)=O)C2)=O)c1 C1CCOC(C(C)C)C1.n1(CCNC(C=C(COC)C)=O)cnc(C=O)c1.N C(=O)(C(CCSC)OC)N(CC(CC)NC(C1CC(Cl)(Cl)C1)=O)C C1(C)(C(N2CC=CC(C(N(C(C=C)C)C)=O)C2)=O)CCN(C)CC1 C#Cc1cc(F)c(C(=O)NCc2c[nH]nc2C2CCN(C(=O)CCC)C2)cc1F c1(C=O)ccc2nn(C)cc2c1.S(=O)(=O)(CC(=O)NC1CCC1C)NC.N c1(CC(=O)NCC(CN(C(C(CC)n2cncn2)=O)C)O)ccc(C#N)cc1 C1(NC(C=CC(C)(C)SC)=O)CN(C(=O)Cn2ccnn2)CC(C)(C)C1 N1(C(C(CO)OC)=O)CCCC(CCNC(c2cc(C)oc2C)=O)CC1 C1(NC(CCCc2onc(CC)n2)=O)CCC(N(C)C(c2scnc2C)=O)CC1 C(=O)(CC1OCc2ccccc21)N(CC(C)CNC(=O)CC1CCC(O)C1)C C1(C(N2CCC(O)CC2)C(=O)NCCCCCC)CC2(C1)CC(OC)(OC)C2 CC(C(=O)N1CCC(N(C)C(c2cccc(N)c2O)=O)C1)C(F)(F)C(F)F C1(CNCc2cccc(C)c2Br)CCN(C(=O)OC(C)(C)C)C2C1C2(F)F c1(NCc2c(OCC)ccc(Cl)c2)nccc(=NCCOc2ccccc2Cl)[nH]1 C(=O)(C(C)(C)C(=O)NC1CCC(N2CCN(C(C)C)CC2)C1)NC n1(CCN(c2ccccc2)CC2CN(C(C)=O)CC2(C)C)ccc(Br)cc1=O C1(C(N2CCN(CC=C)CC2)=O)CCCC(NC(c2ncc(C)cc2F)=O)CC1 C(C(CC(C)C)C(=O)N1CC(NC(=O)CSc2nnnn2C)CC(F)C1)OC C(CC)(C(=O)N(CC(=O)N(CCC(F)(F)F)C)CC1CC1)=CC Cc1ccc(CC(N2CC(NC(c3ccn(C(C)C)n3)=O)C(C#N)C2)=O)cc1C C=CCCCC(C(=O)NC1(CCCC)CC1)NC(C1CCCCNC1=O)=O C1(CC)CN(C(=O)CN2CCCCS2(=O)=O)CCC1NC(c1cccc(N)c1)=O C(CO)(CCF)NC(C1(CNC(=O)C(c2ccccc2)F)CCCO1)=O C(=O)CN=c1ccc(Cl)n[nH]1.CCC(C(=O)NCC1(O)CCC1)NC(N)=O.C N1(C(CN(S(C)(=O)=O)C)=O)CC2COCC(C1)C2.C1(C)C(F)(F)C12CCC2 C(=O)(CC(CN(C)C)C(F)F)N(C1CCCN(C(c2cnc(C)[nH]c2=N)=O)C1)C n1(CC)ncc(C(=O)NC(CNC(=O)C(C)CSC)C(C)C)c1Cl C1(C(N2CCC(CC3CCC3)C2)=O)CCCCN1C(=O)CN1CCOCC1=O C(=O)(C(CCC(=O)Nc1ccc(NC(=O)CC(C)(O)C)cc1)C(F)(F)F)OC c1(NC)ccc(C(=O)NCCC2CCN(C(=O)C(C)(C)C3CCC3)CC2)nc1 C(=O)(C(C)CS(C)=O)N.c1(NCC)cccc(C(=O)NC2CC(CC)C2)c1 c1(CNc2c(C(=O)NC(C(C)C)CO)cc(Cl)nc2)ccc(F)c(F)c1F C1(NC(CCOCCC)=O)CCCN(C(C2CCN(C(=O)CC(C)C)CC2)=O)C1 C=C(C)CCCC(=O)NC(C1CN(C(c2ccc(N)c(OC(F)(F)F)c2)=O)C1)C S(=O)(=O)(c1cn(C)nn1)NCC(C(CC)C)O c1(C=O)cccn2cnnc12.C(=O)(CC(C)(C)C)NC(C)C(=O)N1CC(C)C1.N c1(C(C(=O)NC(CC)CNC(C2CCC(C)(C)O2)=O)OC)c(F)cccc1F C1(NC(c2cc(CCC)on2)=O)CC12CCN(C(C1CC1C1(C)COC1)=O)CC2 c1(CC(=O)NCC2(NC(C3CC(C)C3)=O)CCOCC2)ccc2ncccc2c1 c1(C(=O)NCC2(C)CCCN2C(=O)CO)cc([N+](=O)[O-])cc2c1OCCO2 c1(C=O)cc[nH]c2nccc1-2.C1(CC=C)CCN(C(=O)COC(C)(C)C)C1.N N1(C(c2cnc(CCCC)s2)=O)CCC(O)(CN(C)C(C2CCC23CCC3)=O)C1 C#CC1CCC(C(N2CCC(O)(C)C2)=O)CC1.C(=O)(C=CC(=O)N(C)C)N c1(C(N2CCCN(C(C3C(C#C)C3(C)C)=O)CC2)=O)cccc2ccsc12 CC1CN(C(C2CC3C=CC2CC3)=O)CCN1C(c1ccoc1)=O N1(C(C2(CC=C)CC2)=O)CCC2CN(C(c3cnn(CC(F)F)n3)=O)CC12 C1(C(C(=O)OC(c2cc(Cl)sc2Cl)C(=O)OC)O)COC(C)(C)O1 c1(NC2C(OCC)CCCC2)nc[nH]c(=NCC(C2CCC2)SCC)c1C c1(OC)cccc(CC(C)C(=O)NC(c2ccccc2C(F)(F)F)C#N)c1 C(=O)(C1=CCN(C(=O)CC2NC(=O)NC2=O)CC1)NC(CCC(=O)OC)C C1(O)(C(N(CC(C)(C)C)CC)=O)CCN(C(c2cn(C(C)C)nn2)=O)C1 c1(SC)ccc(F)c(-c2ccc(NCc3ccc(F)c(O)c3)cn2)c1F O=C1CN(C(=O)C(CCF)NC(C2C=CCC2)=O)CCCN1 CC1CN(C(C2(CC3CC3)CC2)=O)CC1CCNC(=O)Cc1cc[nH]n1 C(CC(=O)NCC1(S)CCC1)(C(F)(F)F)NC(C(C(C)C)OCC)=O C1(CC)(C=O)CCCC1.C(=O)(CCCc1csc(C)n1)N(CC)C1CC1.CO C(=O)(C(CCCC)C(C)C)N(CCCN(C(C(C=C=C)C)=O)C)C C1(C2CCOCC2)(C(=O)NC(CC=C)CNC(c2ccccn2)=O)CC1(F)F c1(C(N2C(CNC(CCc3cn(C)nn3)=O)CC(F)C2)=O)ccc(Cl)nc1O Cc1cc(C(N2CCC(CC(=O)O)C2)=O)cnc1OC(F)F N1(C(CC=CC=C)=O)CCN(C(c2nc(C)n(C)n2)=O)C(C)CC1C N1(C(C2N(C(C3CC4(CC(C)C4)C3)=O)CCC2)=O)CCn2ccnc2C1C C(=O)(C(C)C(O)C(C)C)N(CCCCCC)CCNC(=O)C(CC)OC N1(C(=O)C(=CC2CCCCC2)F)CCC(NC(C2(CO)CCOCC2)=O)C(O)C1 C(=O)(CCC(C)(C)C)NCCCN(C)C(C1(Cl)CC1(C)C)=O CC1=C(C(=O)NC(CC(C)(C)C)C(=O)NCC2CC(O)C23CCC3)CCCO1 CC1=CCC(C(=O)N(C2CN(C(C3C(c4ccccc4)C3(F)F)=O)C2)C)CC1 N=c1[nH]c(=NCCC2CCCN2)[nH]c(=NCC(CO)C(F)(F)F)[nH]1 C(=O)(C1CCc2nccn21)NCC(C)(C)NC(C1C(=C)CC1)=O CC1(C)C(CNC(c2nnsc2C(F)F)=O)CCN1C(c1cccnc1)=O CC1CCC(CNC(=O)CC2(C)CCC2)N(C(=O)CCc2ccccc2)C1 C1(COC)(NC(=O)Cn2ccc(=O)cc2)CCN(C(=O)C(CO)C)CC1 c1(OCCC(=O)NCC(C)NC(=O)CN2CCC(C)C2)ccccc1F c1(CNC(C(C)N(CCC)C(C23CCC(C2)C3)=O)=O)nn(C)c(=O)o1 N1(C(C2C(CC)CCCN2C(c2ncsc2C)=O)=O)CCC2(C1)CC2(F)F c1(C(N2CC(C)(NC(=O)CC3(C#N)CC3)C2)=O)ccc2nnc(C(F)F)n2c1 c1ccc(C(=O)Cc2nc(-c3ccc(F)cc3)n[nH]2)cc1.C(C)(CC#N)NCC C1(NC(C2C(OCC)C2)=O)CCN(C(=O)C(c2ccc(Cl)cc2)OC)CC1 C(c1cccc(Cl)c1)=CC(=O)NCCC1(C)CCN(C(C(CC)C#N)=O)C1 N1(CC)CCC(C(=O)NCCNC(=O)Cc2ccc(O)nc2)CC1.C1CC1 c1(C(=O)NC(C2N(C(c3ccc(C)nn3)=O)CCCC2)C)cc(Cl)cc(Cl)c1 C(=O)CC(F)(F)C(C)C.c1(OCC)cccnc1C(=O)NC.C1(F)CCC1 c1(C(=O)NC2CC3CN(C(C4CCCCCC4)=O)CC23)ccc(Cl)c(F)c1F N(C(=NCCN1CCCC1)NC1CCN(S(C)(=O)=O)CC1)C(C)CC(F)F N1(C(C(C)SCC)=O)CCCC(c2cn(Cc3ncoc3C3CCC3)nn2)C1 CC(=NOCC#N)C(=O)NCCO.c1(C(C(c2ccccc2)N)=O)ccccc1 c1(COC)nc(C(C)NC(=O)N(C2CCN(Cc3ccccn3)C2)C)no1 N1(C(C(C)SCCCC)=O)CCCC(C)(C(N2CC(C)(C)C23CCC3)=O)C1 c1(NC(c2c(-c3cc(OCC)ncc3)c[nH]n2)=O)cc(C)ccc1OC C1(C(N(CCC#C)CC)=O)N(C(=O)CCCc2ncco2)CCC1(C)C c1(C(=O)NC(CNC(C(C)OCCC#C)=O)CC)cc(C2CC2)n(C)n1 C1(C)(C(=O)NC2C(NC(c3cc(CC)n(C)n3)=O)CC2)CC(C2CC2)=NO1 S(=O)(=O)(c1cn(C)c2ccccc12)N(CC)Cc1ccccc1CN(C)C C(=O)(C1=CC2CCCCCC12)NCCCCCCNC(Cc1n(C)ccn1)=O CC1(C)CCN(C(=O)Cn2ncnn2)C1CNC(=O)CC1(C)CCC1 N1(C(CC(C=C)C)=O)CC2(CNC(c3ccc(CC(C)(C)C)cc3)=O)CC1CO2 Cc1cc(C2(C(=O)NCC3CCCC(C)C3)CC2)ccc1F.C(=O)(C(C)O)N c1(C(=O)N)cc(C)cc(O)n1.N1(C(C)=O)CC(O)CC1C(=O)NC1CCCC1 CCC(CC(=O)N1CCC(NC(=O)C(C)(C)n2ccnn2)C1)c1ccc(C)cc1 c1(CC(=O)NC2C(NC(CC(CCC)(C)O)=O)CCC2)oc2ccccc2c1C Cc1ocnc1CC(=O)NC1(CC(=O)NCCCC(=O)N(C)C)CCC1 C=CC1(C(=O)NCC2CCCOC2(C)C)CCN(C(=O)C(C2CCCCC2)C)C1 Cc1ccc(CC(=O)NCC(C2CC2)N(C(=O)C(F)C(F)(F)F)C)c(Cl)n1 C(=O)(C1=NNC(=O)CC1)N1CC(CC(C)NC(C(C=C)CC)=O)C1 N1(C(c2n(CC#C)ccc2)=O)CC(NC(=O)CSCCO)CC2(CC2)C1 C(CC(F)F)C(=O)O.c1(CC(N2CCC2Cn2cc(CN)nn2)=O)cnccn1 Cc1ccc(F)cc1C(=O)NCC(F)C.c1(C(C=CC=O)=O)ccc(F)cc1 c1(C(=O)NCC(C)N(C(C(CC)COC)=O)CC)cnc2nccn2c1 c1(OC)ncc(C(=O)NCC2CC2)cn1.c1(C=O)cc(C(C)(C)C)oc1C N1(C(c2cccn(C)c2=O)=O)CCCC2(CC(NC(C3(C)CCCC3)=O)CO2)C1 c1(OC)ccc(C(N2CCC(CC)C2)=O)cc1.C1(C=O)CCCN1S(C)(=O)=O C1(OC(C)C)(CNC(=O)C(n2cc(CN3CCNC3=O)nn2)C)CCOCC1 N1(C(CC(CC)CN(C)C)=O)CCOC2(CCN(C(c3ccc(OC)s3)=O)C2)C1 c1(C(N2C(C)CC(NC(=O)CC(O)C3CC3)C2)=O)ccc2ccncc2n1 c1(C(N2C(CC(=O)NC3CCC(N(C)C)C3)CC(O)C2)=O)cn(C)c(=O)n1C C1(O)CCCN(C(=O)CN2C(=O)CN(C)C2=O)C1.c1(CC)ccoc1C(=O)N N=c1[nH]c(=NCC2(c3ccsc3)CC2)[nH]c(=NCCN2CCn3nccc3C2)[nH]1 c1(C(=O)NC(C2CCN(C(C3(C)CCC(=O)NC3)=O)C2)C)cc2cccnc2[nH]1 C1(CCNC(c2c(C)c[nH]n2)=O)CC(F)(F)CN1C(=O)C.c1(CC)cccs1 C1(CC(=O)NCCN(CCC)C(c2cc(Cl)c(Cl)[nH]2)=O)OCCC1(C)C c1(C(N2C(C)CC(NC(c3cc(CC)nc(O)c3)=O)C2)=O)cnc2nccn2c1 c1(C(N2CC3CC2(CNC(C2CC2)=O)C3)=O)c[nH]c2c(F)cccc2c1=O.C C(=O)(C(CO)C(C)(C)C)N(CCCC(C)(C)C)C.c1(CC(=O)N)cccc(O)c1 Cn1c(C(=O)NCCCCC2CN(C(c3cc(Cl)on3)=O)C2)cccc1=O c1(N2CCN(CCC)CC2)ccc(NC(C2CC2c2cccc(Cl)c2)=O)cc1C N1(C(C(CC)N(C)C)=O)C(CNC(=O)COC2COC2)CC2COCC12 Cc1c(NC(C2(NC(=O)CCCn3ccnc3)CCCC2C)=O)cccc1Cl c1(C(=O)OC)cc(Cl)cc(S(=O)(=O)NCC2CC2C(F)(F)F)c1 N1(C(CC2(CC)CCOCC2)=O)CC(NC(=O)CNC=O)C(N=[N+]=[N-])C1 c1(CCC(=O)NC2C(NC(CC(=C)C)=O)COC2)csc2nc(C3CC3)cn12 CC1CC(CNC(c2c(Cl)cnn2C)=O)CN1C(=O)Cc1csc(Cl)c1 c1(C(=O)NCC2C(NC(c3snc(Cl)c3Cl)=O)C2)csc2ncnc(O)c12 c1(C(=O)NCC2(Nc3cc(C4CC4)ncn3)CCCC2)ccc2nc[nH]c2n1 c1(OC)c(C(N2CC(NC(C3CC3CC(C)(C)C)=O)C(C)C2)=O)csc1C C1(CCCCNC(CCCSC)=O)CCCN(C(=O)C(c2cccn2C)=O)C1 C1(CC(=O)NC2CSCC2C)(OC)CN(C(=O)CN2CC3CC3C2)C1 Cc1ccc(CNC(C2CCC(C3CC3)N2C(C2CCCC2F)=O)=O)cc1F N1(C(CCCSC)=O)C2COCC1CC(NC(=O)CC1CCC(C)(C)C1)C2 c1(C(N(C(C)CNC(=O)CC2CCCNC(=O)C2)C)=O)csc2c1CCCC2 Cc1nnsc1CNC(=O)C(C1CC=CCC1)NC(c1sccc1CO)=O C1(C(=O)NCC2CC(NC(C=CC=CC)=O)C2)CC2CC1C1CC21 Cc1cc(O)c(C(=O)NCC2CCC(NC(c3cc(Cl)ccc3Cl)=O)C2)nn1 N1(CC=O)CCC(C)CC1.C12CCC(C1)C(=O)N2.C1(CC(=O)OC)CCC1 O=C(Cc1csc(-c2ccc(O)cc2)n1)NNC(CF)CO N1(C(C2C(C)C2C)=O)Cc2ccccc2CC1CNC(=O)C1=C(Cl)CCC(C)C1 N1(C(C(C)SCC)=O)C2CCC1CC(CNC(c1ccnc(Cl)c1)=O)C2 C1(C(C(=O)NC2CC3(C(NC(Cc4c(C)non4)=O)C3)C2)C)CCC(C)(C)CC1 n1(CC=O)c(C)cc(C=O)c1C.c1(C(N(CC)C(C)C)=O)coc(C)n1 N1(C(C(c2cn(C)nn2)NC(CN(C)C)=O)=O)CCC(C2OCCO2)C1 C1(NC(C2C(C#N)C2)=O)(CNC(=O)CCC2CCCC2)CC2CCC1CC2 C1(NC(c2c(CN(C)C)cco2)=O)CN(C(C2CCCN2C2CC2)=O)CC1O CCC(C)C(C(=O)O)NC(c1sc(-c2cccc(-c3nn[nH]n3)c2)nc1C)=O n1(CCNC(C(c2cn(C)nn2)NC(COC)=O)=O)nc(C)nc1C N1(C(C(C)CC2CC2)=O)CCC(NC(c2coc(C3CC3)n2)=O)C(F)(F)CC1 C1(OC)CC(C(N2CCC(N(C(=O)CCc3ncc(F)cn3)C)C2)=O)CC1OC CC1(C)CC2(CC2C(=O)NC)C1.C1CC12CCC2.c1(C=O)ccc(=N)[nH]c1 Cc1c(C(=O)NCCN(C(=O)C2=NOCC2)C2CC2)oc2cc(Cl)ccc12 C(=O)(C1=CCCSC1)N1C(C)CC(CC(=O)NCc2ncc(C)o2)C1 c1(-c2nc(-c3cn(CC)c(=O)nc3O)on2)ccc2cc(OC)ccc2c1 CC1CN(C(c2cnccn2)=O)CCC1CNC(=O)CCc1cn[nH]c1 N1(C(CCCC)=O)CCC(CNC(C2CCc3ccnn3C2)=O)C(F)(F)C1 C(=O)(C1CCCc2c1ncn2C)NC1C=CCN(C(Cn2ncc(C)c2)=O)C1 n1(CC)cc(CC(=O)N(CC(C)C)C)nn1.c1(C(=O)N)cc(C(C)(F)F)on1 C(=O)(CC(C)C(C)(C)C)N1CC(C(C(=O)NCC=CC)OC)C1 C1(C(=O)NC2(C)CCN(C(CC(C)OC)=O)C2)CC2CCCCCCC12 c1(C=O)cnn2c1OCC2.C1(CC(=O)NC2(C(COC)O)CC2)CCC1(C)C c1(C(N2C(C(=O)NCC(CC)N=CC(C)(C)C)CCC2)=O)ccc(OC)cc1 C(=O)(CS(=O)(=O)C(C)(C)C)N.c1(CC)cc(C(=O)NC(C)C(C)C)on1 Cc1onc(-c2cccc(F)c2)c1C(=O)NCC(F)C.C1(C(=O)N)OCC1(C)C c1(C(N2C(CN(C)C(C3CC34CCC4)=O)COCC2)=O)cc2sccc2[nH]1 Cc1cccc(F)c1C(=O)NCC1(C)CCCN1C(=O)C(c1cnn(C)c1)=O c1(CC)nc2n(n1)CC(NC(=O)NCC(N1CC(C)OC(C)C1)C)CC2 Cc1cc(Cl)c(C(=O)NC)s1.C1(C=O)CCCN1C(=O)C1CC1.C1CCC1 CCC(F)(F)CC(=O)NCC(CNC(=O)C(c1ccccc1)=O)C(F)(F)F CON1CC(C(=O)NCC(C)(C(C)C)NC(c2cnc(S)n2C)=O)CC1=O CCCCCCCCC(=O)NCCOC1CN(C(c2cccn3cnnc23)=O)C1 c1(C(=O)OC)ccc(C=CC(N2CCCN(C(C3CCOC3C)=O)CC2)=O)cc1 C1(C(=O)N)CC2(C1)CC2(F)F.CCC(CO)C(=O)N1CCC(C(C)(C)C)(C)C1 CCC(C)CCCCC(=O)N(CC(O)CN(C)C(c1c(C)csc1Cl)=O)C c1(CC(N2CC3CN(Cc4ccnc(Cl)c4)C3C2)=O)cc(F)c(F)cc1F CC(C)CC(O)C(=O)NCC1(C(=O)NCC(c2ccnn2C)O)CC12CCC2 C1(NC(C(C)NC(CCc2ccc(C)o2)C)=O)CC2CC3CC(C2)CC1C3 c1(CN2CCCC(C(N3CCN(CCCOC)CC3)=O)C2)cc(Cl)c(F)cc1O CCC(CCC(=O)NC1(C)CCC(C)C1)NC(c1cn(C)c(C)n1)=O CC(C)C(F)C(=O)N1CCSCC1CCNC(=O)COCCOCCO c1(OC)ccc(C=CC(=O)N)cc1F.C(=O)(C1=CCCSC1)N1CC(O)(CC)C1 C1(CCOC(c2cc(C(N)=O)oc2)=O)NC(=O)c2ccccc2O1 C12(C(N3CC(C)N(C(=O)C=Cc4cccc(F)c4)CC3)=O)C3CC(CC13)C2(F)F N1(C(c2c(C)cccc2F)=O)CCC(C)N(C(=O)CS)CC1.C1CCS(=O)(=O)C1 c1(C(N2CC(CCC)C(C(N3CCSC(C)(C)C3)=O)C2)=O)cccc(O)c1F N1(C(COCC#C)=O)CC(OC)C(C(=O)OC)C1.c1(CN)cc(OC)n[nH]1 N1(C(c2c(CC)c[nH]n2)=O)CC(=O)NCC1C(=O)NCCN=[N+]=[N-] Cc1cccc(C(N2CCC(CNC(=O)C(C)Cc3cnc[nH]3)CC2C)=O)c1O Cc1cc(O)n2ncc(C(N3CCC(C(C(C)C)NC(=O)C(C)O)CC3)=O)c2n1 C1(C=O)CCC(=O)N(C2CC2)C1.c1(C(=O)NC(C2CC2)C)cc[n+]([O-])cc1 c1(C(=O)NC2C(NC(C(C)(C)Cc3cnn[nH]3)=O)CCC2)onc2c1CCCC2 C1(COCC)NC(=O)N(Cc2oc(CSc3ccccc3)nc2C)C1=O C1(C(N(CCC)C(C)C)=O)CCC(NC(=O)CN2CCCC2=O)CO1 CC(CF)CC(=O)N(C)CC1CN(C(C23CC(CC(F)F)(C2)C3)=O)CCO1 C12(NC(c3ccc(C(C)C)s3)=O)CN(C(=O)C#CC3CC3)CC1CS(=O)(=O)C2 S(=O)(=O)(c1c(F)ccc(F)c1)NC(C(=O)OC)CC(=O)OC(C)(C)C.O Cc1cccn(CC(N2CCC(NC(c3ccc(Cl)c(F)c3)=O)C2(C)C)=O)c1=O C1(C(N2CC3CC(NC(=O)COC(F)(F)F)C3C2)=O)CCC(C2CCCO2)O1 C1(C(=O)N)CCN(CCO)C(=O)C1.Cc1c(C(=O)NCC2COCC2)nnn1C C#Cc1cccc(C(=O)NCC2(F)CCCN(C(=O)CCOCC(C)C)C2)c1C N#CC1CCC(C(=O)NC2CC(C(=O)NCC3CC(C(N)=O)=NO3)C2)CC1 O=C(C(O)CCC(F)(F)F)NC1CC(NC(C2CCC([N+](=O)[O-])CC2)=O)C(O)C1 c1(OC)ccc(CCC(C)NC(C2CCC23CCC3)=O)c(C)c1 C(=O)(C(C)C(C)n1cccn1)NCCCN(C(=O)C1=CCSC1)CC Cc1cc(F)ccc1S(=O)(=O)NC1CCCN(C(c2c[nH]nc2C)=O)C1 CC(C)(C)CCC(F)C(=O)N1CCC(F)(C(=O)NCC(C)(O)C(C)(C)C)CC1 C(=O)(C(F)CNC(C1CCN(C(C2CNC(=O)N2)=O)C1)=O)OC C12CC1CN(C(C1(C)CS(=O)(=O)C1)=O)C2.C1(C(=O)NC)(C=O)CC1.N CN1N=C(CC(=O)N2CCC3C(C2)CN3C(C2CCC(C(F)(F)F)O2)=O)CC1=O CCCC(F)C(=O)N1CCCC1CCC(N1CC(C)(CC)C1)=O CCCC(C)CC(=O)NC(CCC)CCCNC(C12CC(C(=O)OC)(C1)C2)=O C1(C(N2CCC(NC(Cc3n(C)nc(CC)c3Cl)=O)C2)=O)CNc2ccnn2C1 c1(CC)ccc(NC(=O)CNC(=O)COC2CCCCC2)cn1 C1(CNC(CCCc2nc(C)sc2)=O)C2CN(C(C3CC(F)C3)=O)CC12 c1(NCC(=O)NCC(N2CC(=C)C2)=O)cccnc1 c1(CN2C(C(=O)NCc3c(Br)ccc(OC)n3)CCCC2)cc(C)c(C)cc1C c1(C(=O)NCC2(C(C)(C)O)CN(C(C(CC)F)=O)C2)ccc(C2CC2)cc1 N1(C(Cc2c(C)ccc(C)c2)=O)CCC(C)N(c2nc(C3CC3)ns2)CC1 N1(C(c2c(C)cco2)=O)CCC(C2CC2)(NC(=O)C(O)CC(F)(F)F)C1 C1(NC(C2CCCN(CCC)C2)=O)CCC2CCN(C(c3cccc(C)n3)=O)C12 N1(C(c2ccc(OC)o2)=O)CCC2CCN(C(c3ccn(C(C)C)c3C)=O)C2C1 C(=O)(C(C#N)C(C)(C)C)N1CC=CC(C(=O)Nc2ccc(C)nc2O)C1 C1(N(C(CCCc2cc(C)no2)=O)CCO)CCN(C(C2CCOCC2)=O)CC1 c1(C(=O)OCC)cc2c(=NC3CCN(C)C3)nc[nH]c2s1 C=CC(C)C(C)C(=O)N(C1CCC(CNC(=O)CCOC2CCC2)CC1)C CCCCC(CC)CC(=O)NC1(CF)CCN(C(=O)CC2COC(=O)N2)C1 CC1C2C(CCN2C(=O)C(=O)N=S(C)(C)=O)CN1C(=O)CSc1nc[nH]n1 N1(C(CN(C)S(N)(=O)=O)=O)CC2(CCC2NC(=O)C=CCO)C1 N1(C(CC)=O)CCC2(CCCN(C(=O)C3=C(C)CCC3)C2)CC1 C(=O)(C1=CCN(C(C2CC(=O)NC(C)C2)=O)CC1)NCC(CCCCC)O N1(C(C2(CC(=O)OC)CC2)=O)CCCOC(CNC(=O)C2=CCCOC2)C1 c1(C(=O)NC(C2CCN(C(COCC=C)=O)C2)C)ccnc(S)c1.C1CC1 C(=O)(N=c1cc[nH]cc1)c1ccc(C2(C(=O)O)CCC2)c(Cl)c1 c1(CN(C)CC)cn(CCCCCNC(C2CC2C2CCCO2)=O)nn1 c1(C(=O)NC(CCNC(CC2(C(=C)F)CCC2)=O)C)c(F)ccc(C)c1O C1(O)(CC(=O)N(C(C)C(=O)NC(C)(C)C)CC)CCCCCC1 c1(C(=O)NCC(C)CN(C(=O)C)C)ccc(S(N)(=O)=O)cc1N.CCCF.O C(=O)(CC(C(F)F)n1cccn1)N(CCCNC(=O)CN1CCCC1=O)C1CC1 N1(C(CNC(c2ccccn2)=O)=O)CCCC(SC(F)F)C1 c1(C(=O)OC)cccc(C(=O)NC2CC2)n1.C1(C)(CC(=O)N)CCCCC1 NS(=O)(=O)C1CCN(C(=O)NCCNC(=O)Nc2ccc(F)cc2)C1 C1(C(N2CCCC(NC(c3c(CC)cno3)=O)C2)=O)CCc2nc(=N)[nH]cc2C1 c1(CC)cc(C(=O)NCCOCC)cc(F)c1.C1(C)(C(=O)N)CCCC1C C1(C(=O)NCCC2CC(C(N(CC=C)C(C)C)=O)C2)COC(=O)N1C c1(C(=O)NCC2(OC)CCCC(C)(C)C2)cn(C)c2c(Cl)nccc12 C1(NC(Cc2c(C)ccs2)=O)C(C)CN(C(c2cnoc2C(C)C)=O)CC1C N1(C(Cn2c(C)ncc2)=O)CCCC(CC(=O)NCCC2CC=CC2)C1 CCC(CC)(CO)C(=O)N1CCC(C2(NC(=O)C=C3CCSCC3)CC2)C1 N1(C(C2(CC=C)CC2)=O)CCC(C(=O)NCCO)C(C)C1.CCN(C)C C1(C(=O)N)CCN(C2CC2)CC1.C1(NC(CCNC(C)=O)=O)CCC(CC)C1 CCCC(C(=O)N1CCC(=CCNC(=O)C(C)(C)C(N)=O)CC1)C(C)C N1(CCCOC)C2CCC1CN(C(c1cnc(C)cn1)=O)C2 CCCCCCCCCCCC(=O)N1CCCC(C(=O)O)C1c1ccccc1 c1(COC)cc(C(N2CC(NC(c3cnn(C(C)C)c3F)=O)C2)=O)c(C)o1 N1(C(c2ccc(NC)cn2)=O)CCC(CNC(C2(C)CCCN2C)=O)C12CCC2 C(=O)(C(C)(C)CC#N)NC1C(C(N(CCOCCO)CC)=O)OCC1 C1(O)(C(C)NC(C2OC3CCC2C3)=O)CCN(C(C2(N3CCCC3)CC2)=O)C1 N1(C(C)=O)CCC(n2ccnn2)C1.c1(C=O)coc(C(N)=O)c1.C(=O)(OC)N C1(NC(C(CC)C(=O)OC)=O)CCCCCN(C(c2cc3sc(Cl)cc3[nH]2)=O)C1 c1ccc(S(=O)(=O)N2CCCCCC2)cc1.CC(C)(C)OC1CC1NC(=O)N C(C)(C)(CC(=O)NCC(C1CCCC1)O)N(C(=O)CC1CCCN1C)C c1(C(N2CC3CN(Cc4ccc(F)c(C)c4F)C3C2)=O)ccc(S(C)(=O)=O)cn1 C=CC1CCCN(C(=O)CCN(C(=O)C(CC)SCC)CC2CC2)C1 N1(C(C2C(C)CCC2)=O)CC(NC(c2cccc(F)c2F)=O)C(C#N)C1 CCCC(O)CNC(C1(NC(C)=O)CN(C(=O)CC(C)n2cccn2)C1)=O C1(NC(CCSC)=O)CCN(C(c2nc(C3CC3)cs2)=O)CC1C(C)C CC1(C)OCCC1CC(=O)NC1CCCN(C(C2(C(C)(C)C)CCCC2)=O)C1 C1(NC(C(C)SC(C)C)=O)CCN(C(=O)CN(C)C(C)C)CC1O N1(C(C2C3CCCCC23)=O)CCN(C(C2CC(CC3CC3)C2)=O)C2(CC2)C1 N1(C(C2C(NC(CC(COC)(C)C)=O)C2(C)C)=O)Cc2nc(C)sc2C1 C1(c2nc(-c3ccccn3)nn2CC2CCCO2)CCn2nncc2C1 N1(C(CCC#C)=O)CCC(C(C)C(=O)N(CCC(=O)OC)C)CC1 c1(C(N2C(C)(C)C(NC(c3cncn3C3CC3)=O)CC2)=O)ccc2n[nH]cc2c1 C1(CC(=O)NCC(CNC(CN(CC)CC)=O)OC)CC2CC2C1 c1(C(N(CC(CNC(Cc2cc(C)on2)=O)C)C)=O)cnc(C(C)C)nc1 C1(F)(CNC(C2CC(C)C2)=O)CCC(CNC(c2ccn(C)c2)=O)C1 Cc1nc2ccccn2c1CC(=O)NC12CCCCC1N(C(=O)C=CBr)CC2 c12ncc(C)cc1-n1ccnc1-c1cc-2cs1.C(C(C)(C)O)OC CC(C)CCC(=O)NC1CCC1CNC(=O)C.c1(C(=O)N)ccc(Cl)cc1 N1(C(COCCCC)=O)CCCC2(CC(NC(=O)C(C)CCOC)C2)C1 C(=O)(CCNC(=O)C(F)OC(F)(F)F)NCCN(CCO)CC C1(C(=O)NCC2CCOC2)CCCC12CCN(C(=O)Cc1cccc(Cl)c1)C2 c1(C(N2CCC(C)(CCNC(C(C)=C(C)C)=O)C2)=O)ccc2ncccc2n1 c1(NC(CCCCNC(=O)C=CC2CC2)=O)ccc2nncn2c1 C1(OC)CN(N2Cc3ccccc3C(CO)C2)CCO1 C1(S2=C(COC)C(C)=N2)(c2nn[nH]n2)C=CCN1C(C1CSCC1C)=O N1(S(C)(=O)=O)CCCC1C(N1CCC(NC(c2ccc[nH]2)=O)C1)=O.C1CCC1 CC(C)C(C)C(C)CC(=O)NCC1(F)CC(C)C1.C(=O)C=C1CCC1.N Cc1cc(C(=O)NCC2CC(F)CN2C(c2cncs2)=O)cnc1C.C1CC1.N C(N=c1[nH]c(Cl)ncc1F)C1CN(C(CC2(C)CC2)=O)CC1(C)C C1(CNC(c2cc(OC)no2)=O)CN(C(c2cccc(Cl)c2)=O)CC1(F)F c1(C(=O)NC23C(CN(C(C=CC=CC)=O)C2)C3)cccc2ccccc12 C1(NC(C(C(C)O)C)=O)CCN(C(=O)CCn2ccccc2=O)CC1C C1(c2nnnn2CC(F)F)(NC(c2cc(C)on2)C)CC2(CCCCO2)C1 c1(NCC2(COC)COC2)ccc(OC(=O)CCc2cocn2)cc1 c1(CNC(N2CC(C(=O)OCC)OCC2)=O)ccc(Cl)cc1F CC1CN(C(c2ccc(C#N)cn2)=O)CCC1CNC(C1CCCCCC1)=O CC1CC(C(N2CCC(NC(=O)CC3CC(CF)C3)CC2)=O)CC(C)(C)C1 c1(CNc2ccc(C(N3CC(N4CCCC4=O)C3)=O)cc2)ccnc(Br)c1F c1(C(=O)NCCN(C(C(CSC)C)=O)CC(C)O)n[nH]c(-c2ccccc2)c1C N1(C(C2N(C(c3nc(CC)oc3C)=O)C(C)CC2)=O)CCCC(C)(C#N)C1 Cc1[nH]nc(CO)c1C(N1CC(O)(C(F)C(=O)NCCc2ncccn2)C1)=O c1(-n2cc(CCOC(c3occ(C(N)=O)c3)=O)nn2)ccc(Cl)c(Cl)c1 C(=O)(CCCCC(F)(F)F)N1CCOCC(CNC(C(C)(C)S(C)(=O)=O)=O)C1 N1(C(C=CC=CC)=O)CCN(C(c2sccc2C#N)=O)C(CC)C1 c1(N2CCC(=CCC)C2)cc(=NC2CCOCC2OC)[nH]c(C(F)(F)F)n1 C1(CNC(CCCOC)=O)CCN(C(c2cc(C)[nH]c2C)=O)CC1 c1(C(N2CCC3(NC(Cc4c(C)ocn4)=O)C(C2)C3)=O)cc2sccc2n1C c1(NCC(C)NC(=O)OC(C)(C)C)ccc(F)cc1.c1(S)cccc(N)c1 c1(CCNC(=NC)NCC2CCCCN2C2CC2)cccc(S(C)(=O)=O)c1 C(=O)(C1CCc2ccccc21)N1C(C)(C)CC(NC(C2(C3CCC3)CC2)=O)C1 C1(C)(CNC(C)(CCc2ccncc2)c2nnnn2C2CCOC2)CC(F)(F)C1 CCCCC(C)C(=O)NCC1C2CC1N(C(C1Cc3nncn3C1)=O)C2 N1(C(C(C)(C)COC2CCCC2)=O)CCCC(O)C1.N1(CC(=O)N)CCCC1=O N1(C(C(CSC)O)=O)CCOC(C(=O)N(CC(C)C(C)(C)C)C)CC1 C1(N(C)C)CN(C(=O)C(=O)N(C2CC2)CC2CC(O)C2)CC12CC2 N1(C(C(CC(=O)OC)C)=O)CCC2(CC1)CC2C(=O)N(C(CC1CC1)CO)C CC1CNCC(C(N2CCOC(c3ccc(Br)cc3)C2)=O)C1 c1(C(N(C(C)CNC(=O)C)CC)=O)c2c(nn1C)CCC2.C1CCOC1=O N1(C(C(CC2CC2)NC(c2scc(C)c2)=O)=O)CCc2oc(C)nc2C1 N(C1CC2(CCC2)Oc2ccccc21)C1(c2n(CC=C)nnn2)CC2COCC12 CCC(CNC(=O)CCC1CCC(=O)N1)CC.c1(C(=O)N)c[nH]nc1C1CC1 C1(C(N(CCCC(=O)OC(C)(C)C)C)=O)CC12CCNC2.c1ccc(Br)c(F)c1 CCCC(C)(CC)C(=O)NC1C=CCN(C(c2nccc(Cl)c2O)=O)C1 Cc1cc(=NC(=O)CC2CCCC2NC(=O)CC2CCC(=O)C2)[nH]n1C1CC1 c1(C(N2C(C)CCC(NC(=O)COC3CC(CF)C3)C2)=O)cccn2cncc12 C1(CNC(C(F)=CC)=O)CN(C(=O)CCc2cncc(Br)c2)CCC1(C)C C(=O)(CCN=C(NCc1cc(C2CC2)on1)NCC1C(F)(F)C12CC2)NC N1(C(c2cnn(C(C)C)c2N)=O)CC(NC(=O)C=C2CC2)CC(C)C1 CN1CC=CCC1CC(=O)NC(CO)C(=O)NCCOCCN(C)C C(=O)(C(C)(CC(F)(F)F)c1ccccc1)N(C1C2CN(C(C3COC3)=O)CC12)C C1(C(=O)NCC2C(C)(C)OCC2)CCCCN(C(c2cscc2Cl)=O)C1 C(c1cn(C(COCC)C(=O)NCC2CC(Cl)(Cl)C2)nn1)=CC c1(CC(C)C)c(C(=O)NCC(C)(C)NC(C2CCC(=O)N2C)=O)cnn1C C(=O)(C(C)(C)F)NCC(CN(C(C(=O)NCCOCCCC)=O)C)C C(=O)(CCCCCO)N(C1CCN(C(c2cccc(NC(C)=O)n2)=O)C1)C c1(C(N2CC3C(CNC(=O)C(O)C4CCC4)(CC3)C2)=O)cc([N+](=O)[O-])ccc1Cl C=CC(O)C(C)(C)C(=O)N1CC2(CCCC2CC(=O)NCc2ccccn2)C1 N1(C(C2(SC)CC2)=O)CCC(CNC(=O)C(C)CC(F)F)C(C2CC2)C1 CON(CCC(=O)N1CC(C(N)=O)C(C)C1)C(=O)C1CCC(=O)CC1 N1(C(c2c(CNC(c3nsnc3O)=O)ccs2)=O)CCC(F)(F)C1 N1(c2c(C)ncc([N+](=O)[O-])c2)CCc2c(F)cc(Cl)cc2C1 c1(CN2CCN(CC(N3CC(C)(O)C3)=O)CC2)ccc(F)cc1NC1CC1 CCC(CC)CC(=O)N1CC(CNC(C2CCCOC2C)=O)C(C(F)(F)F)C1 N1(C(c2ccn(C)c2)=O)CCN(C(=O)CC2CCCCCC2)C(CC(F)F)C1 C1(CN(C)C(=O)Nc2cc(Cl)nc(C(C)(C)C)n2)CNC(=O)C(C)(C)C1 C1CC2(CCN(C(=O)CC3C=CS(=O)(=O)C3)CC2)C1.C=C1CC(CC=O)C1.N C1(C(=O)NCC2CCC(CC)O2)CN(C(=O)C(O)CC)CCN1C C=Cn1nncc1C(=O)NCCCC(=O)NC(C)(C(=O)OC)C1CC1 C1(=O)C(C(C)(C)C)N1.C(C(C1CC1)NC(=O)CSC1CC1)OC N1(C(c2c(CC)nc[nH]2)=O)CCOCC(NC(=O)CCc2ccc(Cl)c(F)c2)C1 C(=O)(C1=C(Cl)CCCC1)NCC1C(NC(CCc2c(C)cccn2)=O)C1 c1(N2C(C)c3cc(O)ccc3CC2)ncc(Br)c2cc([N+](=O)[O-])ccc12 c1(C(N2CC(CNC(c3n(CC)ccn3)=O)OCC2)=O)cc2c(Cl)ccnc2s1 CCCC(C)CCCC(=O)N1CC(OC)CC(NC(c2cnc(C)cc2C)=O)C1 C1(C(=O)NC(c2nc(CC)[nH]n2)C)CCN(C(=O)C=C=C(C)C)CC1(C)C C(=O)(C(F)(F)C(F)F)N1C2C(CNC(CCC=C(C)C)=O)C(C2)C1 c1(SC)ccccc1CC(=O)NC1CCC(C)(C)C1.c1(C=O)cc(C)nn1C.N CC(C)C(CCNC(C1CCC(F)CC1)=O)NC(=O)C=C1CCC(C)C1 N1(C(c2cncc(COC)c2)=O)CCCC(NC(=O)Cc2n[nH]cc2Br)CC1 C1(CCNC(CCN(C)CC)=O)CC2CCC(C1)N2C(C1(C#N)CC1)=O CCCCCCC(CN(C)C(=O)OCc1ccc(Br)cc1)CC c1(C(N(CC(CC)NC(CC(C=C)CC)=O)C)=O)cc2sc(C)nc2[nH]1 O(NC(=O)C(CCC)NC(=O)C(CC)n1ccnc1)CCCCC CS(=O)(=O)CCCC(=O)N1CCOCC(CNC(C2CC3C(C2)C3(F)F)=O)C1 C1(NC(c2ccc(COC)o2)=O)CN(C(c2ccc(=N)[nH]n2)=O)CC1OC Cc1[nH]nc(C(=O)N(C2CC(C#N)C2)CC(=O)N(C(C)C(F)F)C)c1O n1(C(COC)C)nc(-c2cccc(C)c2)nc1-c1cn(C)c(C(F)F)n1 N1(C(CCc2ccn(C)c2)=O)CCOC(CC(N2CCC3(CC3)C2)=O)C1 c1(C(=O)NC2CCN(C(CSCC)=O)CC2C)ccccc1N=[N+]=[N-] N1(C(=O)CO)CCC2CCCC(C1)N2C(C1CC2C=CC1CCC2)=O C1(CN=C(NC2CCN(CC=C)CC2)NCC(C)C)COCC12OCCO2 N1(C(c2c(C)cccn2)=O)CCC2(C1)CN(C(C1(CO)CC(F)(F)C1)=O)CCO2 C1(CNC(C(C2CCN(C(CCSCC)=O)C2)C)=O)CCCC(OC)C1 C(CCC(C)C(=O)NC(C(=O)N(C)Cc1cnc(C)s1)C(C)C)OC CC1(C)CN(C(c2nnsc2N)=O)CCC1NC(=O)CC1CNC(=O)O1 C(CCCC(=O)NC1CCOC(CO)C1)NC(C(C)(C)C)=O S(=O)(=O)(c1cc(C)c(-c2ccc(C#N)cc2)cc1C)NCCc1cccc(C)c1 C(=O)(C1=CC2C=CC1C2)N1CC(CNC(C2C(CC)OCC2)=O)CC1(C)C C1(C)(NC2C(C)(C(=O)OC)C2)CN(C(=O)OC(C)(C)C)C(C)(C)C1 C1(C(N2CC(C(C(=O)NC3C=CC(CO)C3)OC)C2)=O)COC(=O)N1C c1(C(=O)NCC(=O)NC)[nH]c(C)c(C(=O)Nc2cnc(O)nc2O)c1C c1(C2C(C(NCC)=O)C2)ccc(Cl)cc1.C1CC1.C(=O)C=C(C)Cl.C CC1(C)CC2(CC(C=O)C2)C1.CC(C)S(C)(=O)=O.n1(CC=O)cnnc1O.N C(CCC(C(=O)N1CCN(CCO)CC1)NC(c1cccc(O)c1C)=O)OC Cc1cc(Cl)c(C(=O)NC2CC(C)CN(C(=O)C(C(C)C)n3cncn3)C2)cn1 CC(=NOCC#N)C(=O)NCC1(NC(c2ccnnc2O)=O)CC1 Cc1c(F)cc(C(=O)N(C2CCN(C(C3CCNC(=O)C3)=O)C2)C)cc1F c1(CC)cccc(C(=O)NC2CC(CCNC(c3ccncc3Br)=O)C2)c1 N1(C(C=CCCC)=O)CCOCC(C(=O)N(C(C)C(F)F)C)C1 c1(C(N(c2c(C)[nH]nc2)C2CC2)=O)ccc(OC(C)C)nc1C.c1ccccc1.C C1(NC(C2CC(NC(C=CCOC)=O)C2)=O)CC=CCC1 C1(NC(C(C=C)(F)F)=O)CN(C(c2cc(C)nnc2CC)=O)CCC1C CCC(CCCC(=O)NCC1(C)CSC1)NC(c1ccccc1Cl)=O N1(C(C(c2cc(C)sc2)(C)C)=O)CCOCC(CNC(c2ccccn2)=O)C1 c1(C=O)ccc(=O)n(C)n1.N1(CC#C)CCC(C(=O)NC2CCC(C)C2)CC1 c1(OC)ccc(C(C)=CC(=O)NC2(CO)CCN(C(=O)C3=CCCS3)C2)cc1 c1(OCC(=O)N(CCCNC(c2cc[nH]n2)=O)CCO)cccc(O)c1 N#CC1CCCN(C(=O)C(Cn2ccnn2)NC(C2CCNC(=O)C2)=O)C1 N1(C(Cc2c(C)n[nH]c2C)=O)CCC2(COCCN2C(=O)C=CC2CC2)C1 N1(C(C2C(C)CC(=O)NC2)=O)CCC2(CCCN2c2nc(Cl)nc3[nH]ccc23)C1 N1(C(c2cccc(C)c2O)=O)CC2ON=C(CNC(c3sccc3F)=O)C2C1 Cc1nc2cc(C(=O)NC(CO)C(C)NC(=O)CC3CC(F)C3)ccc2n1C C1(NC(C(CC)n2cncn2)=O)CCSC12CN(C(C1CC(=O)NC1(C)C)=O)C2 CS(=O)(=O)CCC(=O)N1CC2CC2(C)C1.c1(C=O)cnn(CC(F)(F)F)c1N.N C1(CC)(NC(=O)CC(F)(F)Cl)CCCN(C(=O)CC2CCC(OC)CC2)C1 c1(C(N2C(C3CCN(C(C4(C)CC4(F)Cl)=O)C3)CCC2)=O)cc(=O)cc[nH]1 N1(C(C2(CC)CC2(F)F)=O)CCC2CC(C1)CN(C(c1cncc(C)c1)=O)C2 C1(CC(=O)N(CCC=C)CC)CCCN(C(=O)C(CCC)N(C)C)C1 N1(C(C(CC=C)(C)CC)=O)CCC2(CCCN(C(c3cc(C)c(CC)o3)=O)C2)C1 C(C)(CC(C)C)NC(COC(CC)(C)C)=O.c1(C(=O)N)cscc1C(N)=O c1(CC(=O)NC2CN(C(c3coc(C(F)F)n3)=O)CC2F)ccc(F)cn1 C12(CNC(=O)Cc3ccc(O)cn3)CCC(CN(C(c3ncc[nH]c3=O)=O)C1)C2 C(C(=O)N1CC(OCCC(=O)N(c2csnc2C)C)C1)(C(C)C)OC CCCC(CCCNC(C1CCC(CC)CC1)=O)NC(c1cnn2c1CCC2)=O N1(CCC(=O)NC(c2cn(Cc3cnns3)nn2)C)CCC(F)C1 c1(C(C(=O)Nc2ccccc2)N(CCC#N)CC=C)cccc(F)c1I C(=O)(CCCCC(F)(F)F)NCC(C(C)C)NC(c1ccc2c(n1)NCC2)=O c1(C(N2CC(n3cc(C(C4CC4)OC)nn3)C(C)C2)=O)c(F)ccc(Cl)c1Br C(CC(C)C)(C(=O)N)NC(=O)OC.C1CC(O)CN1C(c1c[nH]c(Br)c1)=O c1(OCC)ccnc(NC2CCC(CNC(=O)C(c3cnn(C)c3)C)C2)n1 S(=O)(=O)(c1nc(N(CC(C)OC)C)ccc1Br)N1CCC(CCC=C)C1 n1(CC(=O)NCCCC2(NC(C(C)c3ccco3)=O)CC2)cc(Cl)cn1 C(C)(C)(C(=O)NCCC1CC1)OC(C)C.n1(CC=CC=O)cncn1 c1(C(c2n(CCC(=O)OCC)nnn2)N)ncc(F)cc1C.C1CCC(=O)O1 CCCCC(C)C(=O)NC(C)C(=O)NCCC1(CO)CC1 Cc1ccc(Oc2cc(NC(=O)C(=O)NC(C(=O)O)C(C)O)ccn2)c(C)c1 C1(C(N2CCC2)=O)CC(c2cccnc2)=NO1.C1(CC#C)(C(=O)NC)CCOC1 N1(C(c2n(CC)cc(Cl)c2)=O)CC(C)OC2(CCN(C(=O)C(C)N(C)C)CC2)C1 C(CC(C)C)(C(=O)NCC1(F)CC(NC(=O)CCn2ccnc2)C1)OC N1(C(c2cc(C)c(C)nc2C)=O)CCCC1C1CCCN1C(=O)CCC(C)(C)F C(=O)(C(C(=O)NC1CCCCC1NC(C1CC(O)C1)=O)OC)OCC O=S(=O)(c1cnc(O)s1)N1CCCC(O)(C(F)(F)F)CC1 C#CCCN=C(NCc1cc(CC)ccn1)NCC1CCN(C(=O)C(C)(C)C)C1 C1CCCCN1C(=O)C(O)Cc1cnn(C)c1.c1(C(N(C)C)=O)c[nH]c(=O)cn1 C(=O)(C1=CCCOC1)NC1CCCC(CN(C(=O)Cc2cccc(SC)c2)C)C1 CC1(C)C(NC(=O)CCCn2cncn2)CCN1C(c1ncc[nH]c1=O)=O O=C(C1=CCC(NC(c2nc(Cl)cs2)=O)C1)NCc1cc(O)cc(F)c1 CC(C)(C)CC(O)CC(=O)NCC#CCNC(c1cc(O)ccc1Br)=O N1(C(C=C(CC)CC)=O)CCC2(CC2C(=O)NC2CC(n3ccnn3)C2)C1 C(=O)(CC(C)(C)CCC)NC(C(C#C)NC(C1CC(NC(C)=O)CCO1)=O)C C1(N(C(=O)CSc2ccccn2)C)CCCC(NC(C2(F)CCCC2)=O)C1 c1(C(=O)NCC(C2CC2)NC(C2N(CC)CCC2)=O)cc(N)ccc1Br C(=O)(C(C)Cc1cnn(C)c1)N(CCC)C.C1(C=O)CC(CC(F)(F)F)C1.N CC(C)CC(C)CNC(=O)CC1CCC(NC(C2CC=CCO2)=O)C1 CCCCCCCCCC(=O)N1CC(NC(=O)CC2(N3CCCC3)CC2)C(F)C1 Cc1cc(=NC(=O)C2CCN(C(C3CCC3C)=O)C2C(C)C)[nH]n1C1CC1 C(=O)(CC(C)(C)C)NC(CNC(=O)OC)C.C1(C(=O)N)OCCCC1(C)C N1(C(=O)Cc2csc(C(F)(F)F)n2)CC2(C1)CN(C(=O)CC1CCOCC1)C2 C(=O)(C(CCC)NC(c1cc(Cl)n[nH]1)=O)N1C(=C)CCC1 N1(C(C2(NC(c3ccc(C)cn3)=O)CC(F)C2)=O)CCCC(C)(C)C1 Cc1c(Br)ccnc1C(N1CCC(NC(=O)C(O)C(C)C)C1C)=O Cc1cc(F)ccc1C(O)C(=O)NCCC1CC1.C1(O)(CC(=O)N)CCC1 CC1CN(C(C2CCOCC2(C)C)=O)CCC1C(=O)Nc1csnc1C1CC1 C(CN=C(NCc1cc(Br)ccc1F)N1CC2C(C1)C2(C)C)OC CC1CC=C(C(=O)NCC2CCCC(NC(c3cc4c[nH]cnc-4n3)=O)C2)CC1 C(=O)(C(C)S(=O)(=O)C(C)C)NC(CC)(C)CNC(=O)C1=CSCCO1 c1(C(N2CCC(NC(C3(CC)CCC3)=O)C2)=O)ccc(S(=O)CC#N)cc1 CC1CC(N=c2[nH]c3ccccc3s2)CN1C(c1cncc2ccsc12)=O Cc1cc(C)c(C(=O)NC2CCOC(CNC(=O)C=CC3CCC3)C2)cn1 C(=O)(C1=C(SC)CCCC1)NCCC(=C)C.c1(CC(=O)N)ccc2c(c1)COC2 c1(C(=O)NC(CNC(C(CSC)C)=O)(C)CC(C)C)cc2c(ncn2C)[nH]1 CCC(C)(C)C(=O)NC1CCCC1C(C)C CCC(CC(C)C)C(=O)N(C)CCN(C(=O)CC1Cc2ccccc2N1)C c1(C(N(CC(C)NC(C2N(CC)CCOC2)=O)C)=O)cc2sc(C)nc2[nH]1 n1(CC)nc(C)c(C(=O)NCC2(C)CCC2)c1Cl.c1(C=O)c[nH]c(=N)o1 N1(C(CCN(c2ccc(Br)cn2)C)=O)CCCCC(C2CCOC2)C1 N1(C(c2c(Cl)cn(C)n2)=O)CCC2(CCCN2C(=O)CC2CCCC(O)C2)CC1 C1(CCNC(CN(C(C(C)CO)=O)C2CCC2)=O)CCCN(C)C1 CN1CC2(CC2)CC1C(=O)NC1CN(C(=O)Cc2ccccc2)CC1C(F)F C1(C(=O)NC(CCOCCO)C=O)CC2(CCC2O)C1.C1CC2(CC2)CO1.N C(=O)(C(O)CC(F)(F)F)NCC(C)(C(C)C)NC(Cc1scc(C)c1)=O N1(C(C2C(C)C2)=O)CCC(C2(O)CN(C(C3(n4cnnn4)CC3)=O)C2)CC1.C CCC(O)C(C)C(=O)NCCN(C(=O)Cc1ncc(C)s1)CC N1(C(CCc2c(C)nccc2)=O)CCCC(NC(=O)COC2CC2(F)F)CC1 c1(CC)cccc(F)c1C(=O)NCCC1CCCN(C(C2CC3CC3C2)=O)C1 N1(C(CCSCCCC)=O)CCCCC(NC(c2cc(OC)no2)=O)CC1 C(CCC(=O)NC1(C2CCCN2C(C2CCCC2C)=O)CC1)=CCC=C N1(CCN)CCCC1C1CC1(F)F Cc1cc(C(c2nnnn2CC(F)F)NC(c2ccccc2C)C)c(C)o1 c1(C(=O)NC2(CNC(Cc3cc(OC)no3)=O)CC2)ccccc1F.CCF C1(CNC(C2N(C)CCC2)=O)CC2(CCC2)CN1C(=O)CCC(CF)CF CC1(C)CN(C(=O)CCC2CCCC2)CCC1C(=O)NC1CC2CCCC(C1)C2 C(=O)(C1CCCc2c[nH]nc21)N1C2C(NC(C3CCCO3)=O)(CCCCC2)CC1 c1(NCC2(NC(=O)Cn3cc([N+](=O)[O-])cn3)COC2)ncnc2[nH]cc(I)c12 Cc1csc(CC(=O)NCC2(C)CCC2)c1.c1(C(=O)N)cnc(C(C)O)s1 C1(c2cn(Cc3c(C)nn[nH]3)nn2)CN(C(=O)C(O)CC(C)C)CCN1C Cc1cc(C)c(NC(=O)Nc2cccc(C(c3cccc(C#N)c3)=O)c2)c(C)n1 C1(CNC(C2(CC#C)CCCOC2)=O)CCN(C(=O)C(C)C)C1(C)C C1(NC(CC(=O)NCC#C)=O)CCCN(C(C2(C)CC(=C)C2)=O)C1 C1(CNC(C(CC)N(C)C)=O)C2CCCC1N(C(=O)CCNc1ccccc1)C2 c1(OC)ncc(F)cc1C(=O)N(C1CCN(C(=O)CCNC(=O)C=CCl)C1)C N1(CC2(O)CC3CC(CC(=O)C3)C2)CC2(CC2)c2ccccc21 C1(O)(CCNC(C2(C#C)CCC2)=O)CCN(C(c2ncc(CC)cn2)=O)CC1 C=CC(C)(O)CC(=O)NC1(CN(C(=O)CCn2cnnn2)C)CC1 N1(C(Cc2ccc(OCC=C)cc2)=O)CC(NC(c2nnc(C)s2)=O)CC(F)C1 C=CC(CC)CC(=O)N1CCCC(N(CCF)C(c2cccc(C3CC3)c2)=O)C1 CCCC(CCC)C(=O)NCC1(CCNC(=O)C(CC)C(F)(F)F)CC1 C#Cc1cc(C(N2CCC3C(NC(=O)CSCCC(F)(F)F)CC23)=O)ccc1C CC(CC(=O)N1CCC(C(C)(C)NC(c2cn(C)nn2)=O)C1)NC(N)=O C(c1c(Cl)cccc1Cl)=C(C(N1CC(NC(C(CCC)(C)O)=O)C(C)C1)=O)C C1(C(N(CCC#C)CC)=O)CCCCN(C(=O)CC2(N(C)C)CC2)C1 C1(CC(=O)NC2CCC2)CCC(F)(F)CO1.c1(C(=O)N)csc(-c2nc[nH]n2)n1 c1(C(=O)NC(CNC(CC2CC(SC)C2)=O)C)cc2ccc(Cl)cc2o1 CCCCCCCC(=O)N1CCC(F)(C(=O)NOCC(O)C(C)C)C1 c1(CCC(=O)NC2C(NC(C3CN(C)C3)=O)CC2)nc(-c2ccncc2)no1 Cc1ccncc1-n1cc(C(CC(N)=O)NC(C2CCCN2C(C)C)=O)nn1 Cc1ccc(Br)c(CC(=O)NC2CN(C(c3nnn(C)c3N)=O)CC2C)c1 C=CC(C)(CC)C(=O)NCCCC(C)NC(=O)CSCC(=O)OC c1(C=O)cnc(C)n1C.N1(S(CC)(=O)=O)CCCC1C(=O)NCC1CC1.N c1(CC)cncc(F)c1.C(CCOCC(=O)NCC1(C(=O)N)CC1)OC C#Cc1cncc(C(=O)N(C)CC2CCCC(NC(=O)COCC)C2)c1 c1(C(=O)NC2CCN(CC(Cl)=CCl)CC2)cc2n(n1)CCO2 n1(CCC(=O)NCCC2(NC(C(CC)C)=O)CCC2)cc([N+](=O)[O-])nc1C c1(C(N2CC(N(C(C3C(C)(C(C)C)C3)=O)C)C2)=O)cccc2ncn(C)c12 c1(C(=O)NCC2COCC2NC(c2csnc2Br)=O)cc2ccncc2[nH]1 c1(C(N(CCC(=O)NCc2cn(C)nn2)CCCO)=O)cc(CO)n(C)n1 C1(NC(C2CN(C(C)=O)C2)=O)CCCC1(C)NC(=O)CCCC1CCC1 CC1C(=O)CCCN1Cc1ccc(C(F)(F)F)c(Cl)c1 CC(CS(C)(=O)=O)C(=O)N1CCOC(CN(C)C(c2cc(Cl)ccc2Cl)=O)C1 Cc1ccc2[nH]cc(CC(=O)NC3CCC(NC(c4cnc(C)s4)=O)C3)c2c1 C1(N(C2CC3CNC2C3)C(c2cc[n+]([O-])cc2)=O)CCc2nncn2C1 Cc1cccc(Br)c1C(=O)NCC#CCNC(=O)C(C)C1CCOC1 C1(C(c2nnnn2C2CC2)NCc2cc(C(C)(C)C)on2)CC2(CCCO2)C1 C(=O)C(C(C)C)c1ccc(Cl)cc1.C1(CNC(C2(OC)CC2)=O)CCC1.N C1(NC(c2nc(C)sc2)=O)CCOC(CNC(C2(C#N)CC2)=O)C1 C1(NC(C(C)CN(C)C(C2CCOC2(C)C)=O)=O)CC(C)(C)OC1=O N1(C(C(C=C)CC)=O)CCC2(CC2C(=O)NC2(C(=O)OCC)CC2)C1 N1(C(CCCC)=O)CCCC1(C)CNC(C1CCCN1c1ccncn1)=O c1(C(=O)NCC2(F)CCC(NC(C(CC)SC)=O)C2)ccn2ccccc12 Cc1ccc(Cl)c(C(=O)NCC2COCCN2C(C2CN(c3nncs3)C2)=O)c1 O=C1CC(CC(=O)NC2CCCC(CC(=O)N)C2)C(=O)N1.N1(CC)CCC2CC12 c1(C(N2CCCC2)CNC(=O)NCCNOC)c(F)cccc1F C1(OC)CC(NC(c2cnc(C)[nH]2)=O)CN(C(c2cnc(C(C)=O)s2)=O)C1 C1(CNC(CC(=C=C)C)=O)CCC2(CCC2)C1.C1(C(=O)N)CC2(CCO1)CC2 CC1(C)CCN(C(=O)CC2CCCO2)C(C(=O)NCCCCCCCO)C1 c12cncc(c1)CNC(=O)C1CCN(C1)C2=O.c1(CSC)cncc(O)c1 N1(C(c2cc(CC)oc2C)=O)CCC=C(C(=O)NC2CN(C(=O)CC)C2)C1 C1(NC(c2c(OC)oc(C)n2)=O)CN(C(C2CCOC2C2CC2)=O)CC1(C)C N1(C(C(=O)NCCCC(=O)OCC)C2CC(C(C)C)C2)CCC(C)CC1 Cc1[nH]c2ccc(F)cc2c1C(=O)NCCC12CCCC1C2 CC1CCCc2ncc(C(=O)NCC(C)(CO)NC(=O)COc3ccccc3)n21 c1(C(CC)(C)C)ccc(C(=O)N)cc1.c1(C=O)cc(C(C)=O)cs1.C1CC1.C Cc1n[nH]c2nc(O)c(C(=O)NCC3(C)CCC3)cc12.c1(C(=O)N)cncnc1 n1(CC)nc(C)c(CC(N2CCCC(C)C2)=O)c1C.C12(C(=O)N)C=CC(CC1)C2 N1(Cc2c(OC)nn(C)c2)CCC(CC(=O)NCc2ccccc2C#N)C(C)C1 C1(C(=O)NCCC2(C(=O)NC(C(C)C)CO)CCCC2)CC12CCCC2 CN(NC(=O)C1CCC(n2cc(CNc3ncccn3)nn2)C1)c1ccccc1 C(CCCCC(=O)N1CCC(C)C(NC(=O)CC(=O)NCC2CC2)C1)OC C1(C)(C(=O)NC(CC)CNC(=O)CCc2ccccc2OC)CCC(OC)CC1 C1(C(C)OC)CCN(C(=O)CCC2CCCN2C(=O)C(C(C)C)C2CCC2)CC1 N1(C(CC(C)CC(C)(C)C)=O)CCCC(C2CN(C(=O)CC3(CO)CCC3)C2)C1 C1(C2CC2)CC1(C)C.C(C(=O)C1CC1)N(C)C(N)=O.C1(CC=O)CC1.N c1(OC)ncc(C(N2CCC(CO)C(NC(=O)Cc3ccn(C)c3)C2)=O)nc1C N1(CCOC)CCCC(CN=C(NCC2CC3CC2C3)NC2CCC2)C1 c1(C(=O)NC2CCCC(N(C(CC=C=C)=O)C)C2)cc(F)c(F)c(O)c1F Cc1cc(C)c(C)c(C(=O)NCCN(C)C(c2cnn(C3CCC3)c2)=O)c1C C#Cc1cccc(CC(=O)NCc2nc(C(=O)NCc3nc(C)cs3)co2)c1 N1(C(C(C(C)(C)O)F)=O)CCC2(CC1)CN(C(c1ccc(Cl)s1)=O)C1COCC21 c1(CC(N2CC(NC(CS(=O)(=O)NCC)=O)C(F)C2)=O)ccccc1[N+](=O)[O-] C1(C)(CNC(CSCC=C)=O)CCN(C(=O)CC2CCC(C3CC3)O2)C1 c1(C(=O)NCCC(C)CCNC(=O)C(F)(F)c2cscn2)c(F)ccc(F)c1F CC(Cn1cccn1)C(=O)NNc1cc(F)c(C#N)cc1F Cc1cccc(C(C(=O)O)NC(=O)CC2(C(=O)O)CCCCC2)c1 c1(CNC(CN2CCN(C(CC=C)=O)CC2=O)=O)ccc([N+](=O)[O-])cc1F c1(C(=O)NC2CC3(CN(C(c4nc(OC)c(C)s4)=O)C3)C2)ccn2ccnc2c1 Cc1cn2cc(C(N3CCN(C(=O)C(C)(C)C)C(C)C3)=O)ccc2n1 C1(CC(C(=O)O)NCc2scc(C)c2C)CCC([N+](=O)[O-])CC1 c1(NC(c2cc(C)c(-c3cn(C)nc3C)cn2)=O)cc(Cl)c(Cl)cc1C#N C(CC(CNC(=O)Cc1cnnn1C)NC(c1ccc(-c2cccs2)[nH]1)=O)OC c1(N(CC(=O)OCC)CCC)cnc2c(ccn2CC(=O)OCC)n1 N1(C(c2c(C)nc(CC)o2)=O)CCC(CO)C(NC(=O)Cc2scnc2C)C1 N1(C(C2CCC(C)=CC2C)C(=O)NCC)CCOc2c(F)cccc21 c1(C(=O)NC2(COC)CN(C(C(CC=C)C)=O)C2)ccc2nc(O)cc(O)c2c1 c1(C(=O)NC(C(=O)NC(c2nccc(C)n2)C)C)ncnc(C)c1C N1(C(c2c(C(C)=O)ccs2)=O)CC2(C)CC(F)(C1)C2.C(=O)C(O)C(F)(F)F N1(C(COc2cc(C)on2)=O)CCC2(CCN(C(=O)CCC3CCCOC3)C2)C1 C(=O)(CC(C)P(C)(C)=O)N1CCN(C(CNC(c2ccc(C)cc2)=O)=O)CC1C c1(SCC)cnc(O)c(C(=O)N(C2CN(C(C3CCC4CC4C3)=O)C2)C)c1 C1(CN(C(C=C(C)C(C)C)=O)C)CN(C(=O)CC(O)C2CC2)CCO1 CCC(C)CCC(O)CC(=O)NCC(C)(C)NC(=O)CC1(C)CCCCC1 C=CCCCC(C(=O)NCc1ocnc1CC)NC(C1CCC(C)(C)C1)=O C12(C(=O)NCC(C)(C)OCC)CC(CN1C(c1cccc(O)n1)=O)C2 Cc1cc(=O)n(C)nc1C(=O)NCC12CCCC1N(C(=O)C(C)C)CC2 c1(C(=O)NC(CC)CC(=O)NC2CC(n3cccn3)C2)ccc(C#N)cc1 c1(C(N2CC(N(C(C(C)=CC)=O)C)C(C)(C)C2)=O)ccc(C#N)nc1O c1(C(=O)NCC2CN(C(CCCOCC)=O)C(C)C2)ccc(F)c(O)c1 CCC(C)(CN=c1[nH]c(=NCCCC(C)CO)[nH]c2ccc(Cl)cc12)OC N1(C(CC=CCC)=O)CCC(N2CCC(NC(=O)C=C3CCOCC3)CC2)CC1 C(=O)C(CC(C)C)N(C(=O)C=Cc1cc[nH]n1)C.C(=O)(CC1CC1)NC.N C12(C(N3CC(O)(CC)C3)=O)CCC(CC1)CO2.c1(CCC(=O)N)cc(Cl)cs1 Cc1cc(C)c(C)s1.C1(CC=O)NC(=O)NC1=O.C(=O)(CCc1cc[nH]n1)N c1(C2(C(=O)NC3C(NC(C(C)(C)O)=O)CCC3)CC2)ccccc1C#N CC(O)CCC(=O)N1CC(N(C)C(C2CC(O)(c3ccccc3)C2)=O)C1 N1(C(c2c(SC)ccs2)=O)CCN(C(c2c[nH]nc2C)=O)C(C)C1C N1(C(CS(CC)=O)=O)CCCC2(C1)CN(C(c1ccc(OCC(=O)OC)cc1)=O)C2 N1(C(C2N(C)CCC2)=O)CCN(CCCCCNC(C2CC2C(N)=O)=O)CC1 N1(C(CC(C)N(C)C(C2CC3(CCC3)CO2)=O)=O)CCC(F)(F)C(F)C1 CCCCC(C(=O)Nc1cccc(O)c1)NC(=O)CC1COCC1O C1(CNC(CSC)=O)CC2(C1)CN(C(C1CCC(F)(F)CC1)=O)C2 c1(C(C)C(=O)NC2CCN(C(c3cc(C4(C)CC4)on3)=O)C2)ccc(F)c(F)c1 c1(C(N2CCCC(N(C(C(CC)(C)O)=O)C)CC2)=O)c(C)ccc(C)c1O C1(CCC)(C(N2CC(NC(=O)CC(c3c(C)noc3C)C)C2)=O)CCNC1=O O=C(CS(=O)(=O)C1CCCC1)NCC(O)CNC(c1cncc([N+](=O)[O-])c1)=O CC(C)C(=O)NCC(C)NC(=O)C(C)C1CCC1 CCC(CC(=O)N1CCCC(COC)(NC(=O)CC(F)(F)C(F)F)C1)C(C)(C)C C1(C)(C(=O)OC(C)C(=O)NC2CC2)CCCN(C)C1 N1(C(c2cc(SC)c(F)cc2)=O)CCCC(NC(=O)Cn2ccnn2)C(F)C1 C(=O)(C(O)CC(=O)OC(C)(C)C)N1CC(NC(C(CC)C)=O)C(OC)C1 c1(CC(=O)N)ccc(Cl)c(F)c1.CC(O)(C)C.c1(C2C(C=O)C2)ccccn1 C1(C(=O)OCC(c2ncc[nH]2)C)CCCCN(C(=O)OC(C)(C)C)CC1 N1(C(c2c(C)scn2)=O)CCCC12CCCN(C(C1CCC(=O)C1)=O)C2 CC(C)CC(C(=O)NCC(O)C(=O)N1CCC(OC2CCC2)C1)C(N)=O c1(C(N(CC(C)(C)C)C)=O)ccc2cnnc(O)c2c1.C(CC)(C(=O)N)OCC C=CCC(CC=C)C(=O)NCCC1CSCCN1C(=O)CC(=C)Br c1(NC(C(=O)NC2CC(C)NCC2)=O)ccc(F)c(S(N)(=O)=O)c1 c1(OC)ccc(C)cc1C(=O)NC1CCC(N(C)C(c2cnc(C)n2C)=O)CC1 c1(NC2CCC(NC(C=CC=CC)=O)CC2)ncc(Br)c(O)n1 Cc1c(C(=O)NCC(C)(O)CNC(C2CCC(CO)CC2)=O)cnc2ccnn12 CCC(CC)C(c1nnnn1C1CCOCC1)NCc1cc(Cl)n(C)n1 N1(C(Cc2c(C)ocn2)=O)CCC2(CCCN(C(c3ccc(N)cc3Cl)=O)C2)C1 C1(OC(C(C)(C)C2(O)CCNC2)=O)CCC2CC1OC2=O C(C1CCCC1)=C(C)C(=O)NC1CCCC1C.c1(C(=O)N)c[nH]nc1C1CC1 C(=O)(CC(C)(C)C#N)NC(C(=O)NC1C(CC=C)CCC1)COCC CN1CCc2nc(NC(C3(C)CCCN(Cc4cccc(F)c4O)C3)=O)sc2C1 c1(C(=O)NC(COC)C=O)cc(CO)ccn1.C12CC(OC)(C1)NC2=O.O N1(C(c2c(C)noc2)=O)CCOC(CNC(c2cnc(C(N)=O)cn2)=O)C1 N1(CC(=O)NCC=C)C2CCC1C(C(=O)OC)C2C(=O)OC C(=O)C1Cc2ccccc21.c1(C(=O)NC2CC2)ccc(S(=O)(=O)N2CCC2)o1 N1(CC(=O)NC2CN(C(c3c(CC)cno3)=O)C2)CCSC2CCCCC12 C=CC1(C(=O)NC2CN(C(C3CCOCC3C)=O)C2)CCOCC1 CN1CCN(C(=O)Cc2cc[nH]n2)CC1c1cn(CCCN2CCSCC2)nn1 C(N=c1[nH]cc(-c2c[nH]c3ncccc23)cc1C)c1nc(CC)sc1 c1(-c2c(OC)n[nH]c2)nc(-c2cccc(N)n2)nn1CCc1ccccc1 C1(CNC(COC(CC)C)=O)CN(C(=O)CCP(C)(C)=O)CCN1C c1(N2CCCC(COC)C2)nc(=NCc2cc(Br)cs2)[nH]c2ccc(OC)cc12 CC1(C)CC(NC(=O)CNC(C2CC3CC2CC3=O)=O)C(C)(C)O1 c1(C(=O)NC(C)(C)CCNC(C2CC3CCC3C2)=O)ncn2c1COCC2 c1(NC(c2cc(-c3ccc(-c4cn(C)nc4)cc3)on2)=O)cnn2c1CCCC2 N1(Cc2onc(CC)n2)CCC(CNC(=O)C(C)=C(C)C)C(C)C1 N1(C(c2c(CC)nn[nH]2)=O)CC2CC(C)N(C(C3CC34CCOCC4)=O)C2C1 c1(C(N2CC3N(C(c4ccc(C)cc4)=O)C3C2)=O)cncc(C)c1C CC1(C(N2CCC(=CCNC(=O)CC3CCSCC3)CC2)=O)CCC(=O)C1 C1(C(=O)N)CC(c2ccccn2)=NO1.C12CC1CN(C(C13CC(F)(C1)C3)=O)C2 N1(C(C2(CCC=C)CC2)=O)CC2(CNC(=O)Cc3ccccc3)CCC1CC2 N1(CC(=O)NC2(C)CC(NC(CCSCC)=O)C2)C(=O)CNC1=O c1(CC)onc(C)c1C(N1CCC(C(=O)NC(c2cccnc2F)C)C1C)=O c1(-c2ccc(C3(C(N(C)C4CC4)=O)CC3)cc2)cccc2cnn(C)c12 CCCC(CCCNC(c1nnn(C)n1)=O)NC(=O)C(CC)CCOC N1(C(CCCSC)=O)CCC(C)(C)C(NC(c2cccc(CO)c2)=O)C1 c1(OC)ccc(C=CC(=O)N(C)C)cc1S(=O)(=O)N1CCCCC1C(F)F c1(C(N2C(CNC(C(=Cc3cnc[nH]3)C)=O)CC(F)C2)=O)ccc(N)c(F)c1 CC(C(=O)NNS(=O)(=O)Cc1ccnc(Cl)c1)c1ccc(F)cc1F c1(C(N2C3CCCC2C3)=O)cc(I)ccc1Cl N1(C(Cc2c(F)ccc(C)c2)=O)CC2CCC1CN2C(=O)CCCCC(C)C C(=O)C(CN(C)C)C(C)C.C1(NC(CSc2nc(C)[nH]n2)=O)CCCCC1C C(=O)(C1OCCc2ccccc21)NC1CC(NC(C2CCc3nnnn3C2)=O)C1 CC1(C)CCN(C(=O)CCSCC(N)=O)CC1NC(=O)CCCc1cccs1 Cn1c(CCC(=O)NC2(C)CCOC2)nnc1S.c1(C(=O)N)cocc1C(N)=O N1(CC)CCCC(N=c2ccnc(NCC3CC(OCC)C3(C)C)[nH]2)CC1 Cc1cccc(C2CC2C(=O)NC2COCC2NC(c2cc(CF)on2)=O)c1 Cn1nccc1C(N1CCCC1C(C)(C)NC(c1ccoc1Br)=O)=O C(C(C(C)(C)C)NC(c1scnc1Cl)=O)NC(C1OCC(C)C1)=O c1(N2C(CC(=O)NCc3cc(Br)cc(Br)c3)CCC2)ncnc2c(Br)cccc12 c1(C(=O)NC2(C)CC(NC(c3ccc(O)cn3)=O)C2)nn2cccnc2c1Cl C1(C(=O)NC2CN(C(c3c(C)coc3C)=O)CC2O)CCOCC12CCC2 N1(CC(CC)O)CCN(C(=O)NCC(O)C(O)CSC)CC1 N1(C(C)C)CCC(C(=O)NC2CN(C(C3CC3c3ccc(Cl)s3)=O)CC2F)CC1 CCCC(C(C)(C)C)NC(=O)C=CC(C)NC(=O)C(CN(C)C)N(C)C c1(-c2ccc(CC(=O)NCCC)c(F)c2)cc(F)cc(Cl)c1O N1(C(C(Br)=C(C)C)=O)CCN(C(=O)C(=O)Cc2ccccc2)CC1C1CC1 Cc1cc(Br)cc(C(=O)NCC2(C)CCN(C(c3cnccn3)=O)C2)c1C Cc1nnc2n1CCC(C(=O)NCc1ocnc1Cn1cc(C3(O)CC3)nn1)C2 N1(C(CC2(COC)CCCC2)=O)CCN(C(=O)C=CSC)CC1C N1(C(C(C)c2cc[nH]n2)=O)CCC(C(C)(C)NC(=O)C=C2CCC2)C1 CS(C)(=O)=NCCNC(c1ccoc1CNC(=O)Cn1cnnn1)=O c1(CC)cc(C(=O)NCCCOC)c(C)o1.c1(C(=O)N)cc(C(C)C)no1 CCCC(CCC)CC(=O)N(CC(=O)NC1CCN(C(=O)CC(C)COC)C1)C C1(C(=O)NCC(CC=C)NC(c2cncc(N(C)C)c2)=O)CCC(C)(O)CC1 CC(C)CC(C)CC(=O)NC1CN(C(=O)CC2CCCC(C)C2)CC2(CC2)C1 C(=O)(C1c2c[nH]nc2CN1C(c1cccc(CO)n1)=O)NCC1OCCN(C)C1 N1(C(c2cc(C)c(N)cn2)=O)CC2(C=C(C(=O)NC3CC=CCC3)CO2)C1 n1(CC)ncn(NC(=O)C23CC(CO)(CN2C(=O)C(O)C2CC2)C3)c1=O C(=O)(CCC(=O)NC(C1CCCC1)C)N(CC)CC.c1(C=O)cnc(Cl)n1C CCC(F)(F)CC(=O)N1CCC(C)(NC(c2c[nH]cc(C)c2=O)=O)C1 c1(C(=O)NCC23CC2CN(C(C2CCCS2(=O)=O)=O)C3)c(O)cccc1F CC1(C)C(CC(N2CCCCC2c2cc[nH]n2)=O)CC1O N1(C(C)=O)CCN2CCN(C(c3cc4c(s3)C(C)(C)CC4)=O)CC2C1 C1(C(N2CCC(N(C(C3CCCN3C=O)=O)CC)CC2)=O)CCN(OC)CC1 C(C)(C)(CCCNC(=O)CC(F)(F)Cl)NC(c1cc(C(C)C)[nH]n1)=O CC1(C)CN(C(=O)COCc2nc[nH]n2)CC1.c1(C=O)cc(CCO)on1.C c1(CC)ccccc1OCC(=O)NC(C)(C)C1CC1.C(=O)(CC=C(Cl)Cl)N CC#CCCCC(=O)NCCNC(c1cn(-c2ccc(F)cc2)nc1C)=O C(C(CO)NC(=O)CC1CC(F)C1)NC(C1C(CCOC)C1)=O C1(C(=O)NC(c2cnn(C)c2)CC)CCN(C(c2sccc2C#N)=O)C1C C1(NC(C=CC)=O)C2CC1N(C(=O)COCCO)C2.C1CCC(C)CC1 C(=O)(CCCCCN=[N+]=[N-])NCC1(NC(C(C)NC(N)=O)=O)CC1 N1(C(C(C(C)C)NC(=O)COC2(C)CCCC2)=O)CC(=O)NC(C2CC2)C1 C1(c2nnc(N3CCCC(C(=O)OC)C3)n2C)Cc2c(F)cccc2N1 c1(C(N2C(CNC(C=Cc3c(C)ccnc3)=O)CCC2)=O)cccc(C#N)c1F C1(NC(c2ncc(OC)cn2)=O)CCCN(C(c2cn(C)[nH]c2=N)=O)CC1 c1(C(C)(F)C(=O)NCCOC2CCN(C(c3ccncn3)=O)C2)ccc(F)cc1 c1(C(=O)NCC2CC(NC(=O)CC3(O)CCOCC3)C2)n[nH]c2c1CCCC2 c1(C(=O)NC2CCCC(NC(c3cccnc3)=O)CC2)n[nH]c2ccccc12 C(C(C(=O)N1CCOCC1)N(C)C)NC(C)=O.c12cn(nn1)CC(=O)NCC2 N1(C(C=CC=CC)=O)CCSCC1CCNC(=O)Cc1ncc(C)s1 c1(C(=O)OCC(OC)OC)cc(S(N)(=O)=O)c2ccccc2c1O C1CCN(C(=O)C=Cc2scnc2C)C(C)C1.c1(C(=O)OCC)cccnc1N C1(C=O)CCCCN1C(=O)CCCCC1CC1.C1(C(=O)OCC)(C)CC1.N c1(CC)ncnc(CC)c1C(=O)NC1CCCC1.C1(C)(C(=O)N)CC2CC2C1 c1(C=O)ccnn1-c1ccccc1.CC(C)(C)OCC=CC(=O)N.C1CC1 N1(C(C2CCN(C)CC2)=O)Cc2cccc(CNC(=O)CCF)c2C1 Cc1ocnc1C(=O)NCC(C(C)C)NC(=O)CC(=O)OCCC(C)C Cc1n[nH]c(C)c1CCNC(=O)C(C1CCCN(C(=O)C=Cc2ccoc2)C1)C N1(C(CC=C=C)=O)CCC(C(F)(F)F)C(NC(c2c(Br)cnn2CC)=O)C1 CCC(C)CC(C)C(=O)N1CCCC1CNC(c1cccnn1)=O N1(C(C2CCCCC2O)=O)CC(CO)C2(C1)CN(C(C1CCC=CO1)=O)C2 N1(CC)CC(Sc2ccc(-c3nccn3C3CC3)cc2-c2ccoc2)C(C#N)C1 N1(C(CC2CCC(=O)NC2)=O)CCC2CN(C(C3CCS(=O)CC3)=O)CC12 C(=O)(CCS(C)(=O)=O)N1C(C(N2CC3(C(C(=O)OC)C3)C2)=O)CC2CC21 C(C(=O)N1CCC(C(N2CC3CCC3(CO)C2)=O)O1)c1c(C)non1 C1(NC(c2nncs2)=O)(CO)CCN(C(c2csc(-c3cccs3)n2)=O)CC1 CC1CN(C(=O)CN(C2CCCC2)C)CC1C(=O)NC1CC(n2cccn2)C1 C1CN(C(C2CC(=C3CCC3)C2)=O)C2CC12.C(C=O)N(S(C)(=O)=O)C.N C(c1cnc(O)nc1O)=CC(=O)NC1CC(NC(C2(C)CCC2)=O)C12CCC2 CC1CCC(C(N2CCC(=CCNC(=O)C(C)(C)N(C)C)CC2)=O)CC1C C(=O)(C1=CCOCC1)N1CCC(NC(Cc2cc(C)on2)=O)C1 C1(OC)CC(CNC(=O)CCN2CCOC2=O)N(C(C2CCNC(=O)C2)=O)C1 c1(C(=O)NC(CC)CNC(C2(n3cc(Cl)cn3)CC2)=O)ccc(O)nn1 N1(CC#C)CCN(C(c2cc(C)ns2)C(=O)NCc2nnn(C)n2)CC1=O CCCC(C(=O)NCC1(O)CCSC1)NC(=O)CCC(N)=O CC1(C)CCC=C1C(=O)N1CC=CC1C(=O)O C(=O)(C1COc2ccc(F)cc21)NC1C(C)N(C(c2nccc(Cl)c2F)=O)CC1 c1(C(=O)NCC(CNC(CCc2cc(C)on2)=O)CO)ccnc(C(C)(C)C)c1 Cc1ccnn1C(C)C(=O)NCC1CCCC1NC(=O)C(C)(C)c1cnco1 c1(C(N2CC(C)(NC(C3CCS(=O)CC3)=O)C2)=O)cncc2cccnc12 Cc1cccc2c(C(=O)NC3CC(C)CN(C(C45COCC4C5)=O)C3)c[nH]c12 C(=O)(C1=CCOC1)NCCCN(C)C(c1cncn1-c1ccc(F)cc1)=O c1(CC)cc(C(N2CCCCC2)=O)c(C)nn1.C(=O)(CC)NC.[SH](C)(=O)=O.C c1(C=O)ccc2c(n1)CCC(C)C2.CCCCN(C(=O)CSCCN(C)C)C c1(CCC(=O)N(CCN(C(C2CN(CC)C(=O)N2)=O)C)C)ccc2[nH]ccc2c1 C1(C(N2C(C(N3CCC(O)(CC(C)C)C3)=O)(CC)CCC2)=O)CC2(CC2)CN1C Cc1nn(C)c(C)c1C(=O)NCCC1CC1.C(=O)C(O)Cc1ccccn1.C C1(CN(C(CCOCCCNC(CNC=O)=O)=O)C2CC2)CCCOC1 C1(CNC(CCC(N)=O)=O)CN(C(C2CC3CCC2CC3)=O)CCC12CCC2 CC1(C)CC(NC(=O)Cc2ccccc2Cl)CCN(C(C2CCC2(F)F)=O)C1 N1(C(C(c2ccc(Cl)cc2)OC)=O)CCC(NC(=O)CCC(C)=O)C(F)C1 C(=O)(CN=c1cc[nH]cc1)NCC(=O)NCC(=O)NCC(CCCC=C)(C)C Cc1cc(C(=O)NC(CNC(=O)C(C)(C)C(N)=O)CO)nc(C(F)F)n1 C1(CC)CCCN(C(c2cc(N(C)C)ccn2)=O)C1.c1(C(=O)N)nc(O)c(C)s1 N(C(=NCCCCl)N1CCC(C(F)F)CC1)CCCO Cc1cnn2cc(C(=O)NC(C)(CNC(=O)C(F)n3cccn3)C(C)C)cnc12 c1(NC(CCC=C)C)ccc(S(=O)(=O)NC(c2ccccc2OC)CO)c(Br)c1 n1(CCC)nc(C)c(C(=O)NC2CCN(c3nnc(C)o3)CC2O)c1C c1(C(N(CCCCN(C)C(c2ccccn2)=O)C)=O)cc(Br)c(F)cc1O c1(C(=O)NCC2(NC(CC=CC)=O)CCOC2)cnn2c(C)c(C)ccc12 C(CCCC(=O)N1CC(OCCNC(=O)CC2CCS(=O)(=O)C2)C1)SC c1(CNC2(C(=O)OC)CC2)cc(F)ccc1Cl.C1CCO1 c1(CNC(Cc2nc(C(C)C)sc2)=O)ccc2c(c1)C(=O)N(C)C2 N1(C(CCc2onc(CCC)n2)=O)CCC(NC(c2ncoc2C)=O)C(CC)C1 C1(C(N2CC(C(C)OC)C2)=O)COC(CNC(C2CC2(C)C(F)F)=O)C1 N1(C(c2nc(C)sc2)=O)CC(NC(=O)C=C2CCN(C)C2)C(n2ccnn2)C1 c1(CCNC(C=C(C)C)=O)cc(C(=O)NC(C2CCOC2)C)no1 C1(NS(CCOCC)(=O)=O)C2CCC1CN(Cc1cc(F)cc(F)c1Br)C2 C1(NC(=O)C#CCNC(c2[nH]ccc2C2CC2)=O)C2CCCCCC12 c1(C(=O)NCC(C)NC(C=Cc2c(C)noc2C)=O)cc2c(Cl)cccc2s1 c1(NC(C(N2C(CC(=O)NC)CCC2)=O)=O)ccc(Cn2cccn2)cc1 C1(C(N2C3C(NC(Cc4ccc(C)s4)=O)C(C3)C2)=O)COc2ccc(F)cc2C1 N1(C(CC(c2cccc(F)c2)C)=O)CCC(NC(C2CCC(C)(C)C2)=O)CC1 C(=O)(C(C)C(C)O)N(CCCNC(=O)C(=O)NCCC(N)=O)CC CCC(C(=O)NCC1CC1CNC(=O)C(C)(C)n1cnnn1)C(F)(F)F C(=O)(CCC(C)(C)F)N1CCC(C(N(CC=C)CC)=O)(CC=C)C1 c1(OCC(CC(=O)N2CCC(C(=O)OC)C2)N)ccc(Br)cc1Br C1(CCC)CN(C(c2ccc(Br)o2)=O)CCN1C(C1CCNC(=O)C1)=O C1(C(=O)OC(c2nc3cc(Cl)ccc3n2C)C)C2CC(C(O)C2O)S1(=O)=O O=C(N=c1[nH][nH]c2ncccc12)C1CC(O)CN1C(c1cc(Cl)ccc1Cl)=O N1(C(c2cc(C(=O)OC)cc(C)c2)=O)C2CCC1CN(C(C1CCCC1C)=O)C2 n1(CC(=O)NC2CCC(NC(CC3C(C)(C)C3)=O)C2)ccc(O)nc1=O N1(C(Cn2c(C)ccc2C)=O)CCC2CCCC12C(=O)NCC1C2CCCCC12 C(C1c2ccccc2CCN1)NC(C(C)OCCOC)=O.c1coc(C2CC2)n1.C N1(C(CCC)=O)CC(C)(C)CCC1CNC(=O)C(CC)SC N1(C(CCC(C)SC)=O)CCN(C(=O)CCc2ncccn2)CC1C C1(NC(Cc2cn(C)nn2)=O)CC(NC(=O)C(O)c2ccsc2)C(O)C1 CCC(CC)C(C)C(=O)NCc1cc(C(=O)NCc2ccc(O)c(C)c2)co1 N1(Cc2cccn(CC#C)c2=O)Cc2ccc(Br)cc2C(C#N)C1 C1(NC(CCCC)=O)CC2(CCCN(C(=O)Cn3cc(Cl)c(C)n3)C2)C1 C1(NC(C(C)c2ccsc2)=O)CCC(CNC(=O)C)CC1.CCCN(C)C.O N1(C(c2cc(OCC)ns2)=O)CCCC(C2CN(C(C3C=CCC3)=O)C2)C1 C(=O)(C1CC(O)c2ccccc21)N1CCC(NC(=O)C(F)=CC2CC2)C1 C1(NC(C2(NC(C3C(CCC)C3)=O)CC(F)C2)=O)CC(C)CC(C)(C)C1 c1(CC)nn(C)c(C(=O)NCC(F)CNC(=O)C)c1Cl.c1cc(C)ccc1F Cc1cc(C(N)=O)cc(C(=O)NCC2(F)CCN(C(C3C=CCCC3)=O)C2)c1 N1(C(c2ncn(C)c2)=O)CCCN(C(=O)Cc2csc(C3CCOCC3)n2)CC1 c1(C(=O)NCC2CCCC(NC(=O)Cc3ccco3)C2)cnc2ccncc2c1 N1(C(C(C(C)C)O)=O)CCCN(CCNC(=O)C=Cc2cocn2)CC1 C(=O)(CC(C(F)(F)F)NC(=O)C(C)(C)c1ccno1)NCC(=O)N(C)C C1(c2onc(C(c3ccc(Cl)cc3)CCCOC)n2)CCC(C)CO1 c1(OC)cc(C(=O)Nc2cccc(NC(=O)C(CCO)N(C)C)c2)cc(C)n1 c1(C(N(C)CCNC(c2cccc3oncc23)=O)=O)cc(=O)c2ccncc2o1 CCCC(C)C(=O)NC(C1CCN(C(C2CSC(C)=N2)=O)CC1)(C)C c1(N(c2cnn(CCc3ccc(F)cc3)c2)CC)ccc2cc(Br)ccc2n1 C(=O)(C1=CC2C=CC1C2)N1C(C(=O)NC2CC(C(C)O)C2)C(C)CC1 N1(C(CC(=O)NCC)=O)CC2CCCC(NC(=O)CC(C)P(C)(C)=O)C2C1 C(CC(CC)C(=O)NCC(O)CNC(=O)C(=CC1CCCC1)C)=CC C(=O)(CC(C)CCC=C(C)C)N(CC(C)NC(c1ccc(N)cn1)=O)CC Cc1nc(C(=O)NC(CNC(=O)CC(O)C2CC2)C(C)(C)C)ccc1C#N C1(NC(C=Cc2n(C)cnc2)=O)CCN(C(C2OCCCC2(C)C)=O)CC(O)C1 CC(C)(CCS(N)(=O)=O)NC(=O)CCCn1cc(C2CCCC23CC3)nn1 C(=O)(C(C)(CO)NC(=O)C(C)CC1CCCC1)N(CCCCC=C)C c1(C(=O)NCC2C(NC(c3c(C)onc3)=O)CCC2)nccc(Br)c1O c1(C=O)ncnc(O)c1F.C1(COC)CCCC1.C(=O)CC1CC1.C1CC1.N C12(NC(C=NOC)=O)CCN(C(=O)CC3CCC3C)CC1C2 c1cc([N+](=O)[O-])cc([N+](=O)[O-])c1.c1(C(=O)OC)ccc(CCNC=O)cc1.N C(=O)(C1Cc2ccccc21)NC1CN(C(c2c(N)cc(Cl)cc2)=O)CC(F)C1 CCCCC(C)(F)C(=O)NCCNC(c1nocc1CC)=O c1(CC)ccc(S(=O)(=O)N(C)C)cc1.C(CC(N)=O)C1CCCCC1.C(=O)CN.N Cc1oc(S(N)(=O)=O)cc1C=O.C(C)CC(C)C.c1(C=O)cc(Cl)n(C)n1.N CC(C(=O)NN1CCCC1C(=O)NC1(c2cccnc2)CC1)=C1CC1 C1(NC(c2cc(CNC(c3cccnc3S)=O)no2)=O)CNC(=O)C12CC2 Cc1cc(C(N2CC=CC(C(=O)NCC(C)(C)N(C)C)C2)=O)[nH]c1C N1(C(C2(CCC)CC2)=O)CCC2(NC(C3CCC(C)(C)CC3)=O)CC2C1 CC1CC(C(=O)N2CCC2CNC(c2cc(N)nc(Br)c2)=O)=NO1 C1(CN(C(C(c2ccccc2)C)=O)C)CCCN1C(=O)C(C)Oc1ccncc1 N1(C(CC(CC)O)=O)CCC(C)(C)CC1C(=O)N(C)Cc1cscn1 Cc1cc(C(=O)NC(CNC(=O)C(C)O)C2CCC2)n2nccc2n1 c1(C(=O)NCC(CNC(=O)CN2CCCC2=O)F)cccnc1C(F)F C1(C(N(C(C2CCC2)C)C)=O)OCCO1 C1(N(C(Cc2ccc(C)s2)=O)C)CN(C(c2ccc(C#N)s2)=O)CC1F C(=O)(C(C)(O)C(C)C)N1CCC(C=O)C1.c1(C(C)C)cc(C(=O)N)on1.CC C=C(Cl)CC(C(=O)NC1CCCCC1C#N)NC(c1ccc(C)cc1F)=O C1(CCC=C)(NC(c2ncnn2CCCC)c2nnnn2CC2CC2)CCCC1 N1(C(CCCCC)=O)CCCC(NC(c2ccc(C3CCCOC3)cc2)=O)C1C CC1(C)CCCN1C(C1CC(=C2CC2)C1)=O.c1cccc(F)c1.C(=O)CC.N N1(C(C(c2cccc(Br)c2)C)=O)CCC(C2CCOCC2)C1 c1(C=O)cnc(C2CC2)[nH]c1=N.CC(C)C.C1(C(=O)N)CN(CC(F)(F)F)C1 CC(C)C(C(=O)N1CCCC1CF)NC(=O)CN1CSCC1=O C1(NC(=O)C=C2CCSCC2)CCOC12CCN(C(C1CC3CCC1O3)=O)CC2 C(=O)(C1=CC2(CCOC2)C1)NC(C(C)C)C(=O)NCCC1CC1.C1CC1.C C1(OC)CCCC(CC(=O)N(CCC(C(C)C)NC(c2nccnc2C)=O)C)C1 c1(NC(=O)NC2CC(C)(CC)C2)nc2cc(Cl)cnc2n1CC C#Cc1cccc(C(N2CC(NC(c3nnc(O)nc3O)=O)C3(CC3)C2)=O)c1 C1(C)(C(=O)NC(c2cn(C)nc2)C(N2CCCC(CCCO)C2)=O)CCCCO1 c1(C(=O)NCCC(C)NC(C2CSCCS2)=O)ccnc2c1nnn2C N1(Cc2c(OC)nc(Br)cc2)CC2(CCC(C(=O)NCC)O2)C1.C(C)=O.N Cc1noc(C)c1C(N1CCC1C(N1CCC(N2CCCCC2)CC1)=O)=O c1(C(=O)NC2CCN(C(CCN(C)CCO)=O)C2)ccc2nc(O)cc(O)c2c1 N1(C(c2c(CC)occ2)=O)CCN(c2nccc(C#N)n2)CC(O)C1 C=CCC(C(=O)NCC(O)CC(=O)OC)NC(=O)C(C=C)OC n1(CC=C)ncc2c(O)nc(N3CC4C(NC(=O)Cn5ccnc5C)C4C3)nc12 Cc1ccn2cc(C(N3CC(C)(NC(=O)Cc4ccoc4C)C3)=O)nc2c1 C(=O)(CCCC(C)(C)C)NCC(C1CCCCC1)NC(c1ccn(CC)c1C)=O C(CCO)(C(=O)N1CC(O)CC1CNC(C1CC1c1cn[nH]c1)=O)N(C)C N1(C(C(CC)C(C)C)=O)CCCC(C)(C)C1CNC(=O)CN1CCC(C)(C)C1 C(=O)(C(c1ncco1)N(CC(F)(F)F)CC(=O)OC)NC(CC)C CC(N=c1[nH]c(N(C)Cc2ncc(-c3ccccc3)o2)nc(=N)[nH]1)c1ccco1 C(=O)(C(CCC)C(C)C)N1CC(NC(CC(CCC)O)=O)C(O)CC1 C1(N(C(C)=O)C)CN(C(c2cc(C(N)=O)co2)=O)CC1F.Cc1cc(CO)no1 c1(C(N(C(C)C)CC)=O)cc2nccn2c(O)n1.n1(CC=O)ncn(C)c1=O.N N1(C(=O)Cc2csc(-c3ccccc3)n2)CCC2(CCC(O)C2)CC1 N1(C(COC)=O)CCC2C(CCN2C(c2csc3ccc(C(F)(F)F)cc23)=O)C1 CCC(CC(C)CO)N=c1ccn2ncc(S(=O)(=O)NCc3ccc(Cl)s3)c2[nH]1 Cc1cccc(CC(=O)NCC2(NC(c3nocc3Cl)=O)CCCC2)c1C c1(C(CN(C)CC2CC(F)(F)CO2)O)ccc(F)cc1F C1(CC(=O)NC2C(NC(C(C)=C3CC3)=O)CCOC2)CC2CCC(C1)N2C Cc1cc(=NC(=O)C(=O)NC2(CCNC(C3CCC(F)CC3)=O)CCCC2)[nH]o1 c1(N2CC(C)C(O)C(C)C2)nc(N2CCN(CCF)CC2)c2cccc(F)c2n1 CC1CCC(C)N1C(C)C(N1CCCC1C1(NC(=O)CO)CC1)=O Cc1ccc(CC(C)C(=O)N(C2CN(C(c3cnn(CC(C)C)c3)=O)C2)C)cc1 c1(NCc2cnc(CCC)s2)cc(C)cc(-c2nccn2C)c1F Cc1c(C(=O)NC2CCN(C(=O)CC3=CCCCC3)C(C)C2)cnc2ncnn12 C1(C(=O)N)CCCCC1(C)C.C1(CCC(=O)NCC(C)OC)CC(F)(F)C1 C(=O)(C1=CCc2ccccc21)NC1CC(F)(CNC(=O)CC2COCCO2)C1 c1(C(=O)NC2(CCCNC(=O)CSc3ccncc3)CC2)cncc(O)c1 Cc1cn2cccc(C(=O)NCC3C(C)CCN3C(c3cc(F)n(C)n3)=O)c2n1 C(=O)(CCCCN=[N+]=[N-])N1CCC(NC(CCOCCC)=O)C12CC2 CCC(C(=O)N(CCC(=O)NCc1cc(OC)no1)CCCO)N(CC)CC Cc1snnc1C(N1CCCC1CNC(=O)CSCC1CCCO1)=O N1(C(C(C2CC2)OC)=O)CCCN(C(=O)CCC(C)(C)N2CCOCC2)C(C)C1 C1(C(=O)NC2CC(F)(CNC(c3cccs3)=O)C2)CC2CCC(C1)C2 C1(NC(COCCCCC)=O)CCCC(NC(=O)Cc2csnc2C)CC1 c1(C(N2CCCC2CC(c2cccs2)O)C(=O)NCCCF)cccc(Br)c1 Cc1cnn(CCC(=O)NCCN(C(=O)CC2CS(=O)(=O)C2)C(C)C)c1 C=CC(C)C(C)C(=O)N1CC(OCC)C1.c1(C(=O)N)cc(C)ccc1C1CC1 C1(C(N(CC(C)N(C(=O)CCCNC(=O)C2CC2)C)C)=O)SCCCS1 c1(OC)c(C)cc(NC(=O)CC2CCN(C(=O)C=Cc3ccoc3)C2)cc1C C1(CC(=O)N)CCCC(C)(C)C1.C(C)(CC)OC.C(=O)C(F)CC1CCOC1 C1(CC)CCCC(NC(=O)CN2CCN(C(=O)Cc3cc[nH]c(=N)c3)CC2)CC1 CC1(C(=O)NCC2CCN(C(C3CC(N=[N+]=[N-])C3)=O)C2)CCCOC1 N1(C(CC(=C)C)=O)CCC(F)(CNC(=O)CC(C)COC)C1 S(=O)(=O)(c1ccc(Br)cc1NC1CCOCC1C)N1CCC(CSC)C1 C1(N(C(C2CC(CC)(CC)C2)=O)C)CCCN(C(=O)C(c2ccc(C)cc2)=O)C1 N1(C(CCOCCC)=O)CCN(C(=O)CN(C)C(C2CCCC(CF)C2)=O)CC1 c1(OCc2onc(NS(C)(=O)=O)n2)cc(Br)cc([N+](=O)[O-])c1 CCCC(CCC)(c1nnnn1CC(F)F)NCC1(OC(C)C)CCC1 C1(O)CCN(C(=O)C(CC=O)N(C)C)CC1.C1(C)(CC)CC(C(=O)NC)C1 CC1(C)COCC(CC(=O)NC2CC(C)C2)O1.C(c1ccccc1)=CCC(=O)N c1(OC)ccc(C(N2CCN(C(=O)C(CSC)OC)C(CO)C2)=O)cc1OC c1(NCCC(=C)C)[nH]c(=NCCC2COCC(C)O2)nc2c1ncn2C N1(C(CC2CC(CC)OCC2)=O)CCC(C2(NC(c3nccn3C)=O)CC2)CC1 c1(OC)cncc(CNC(c2ccc(C)nc2)=O)c1.C1(C=O)CC12CCC2.N N1(C(C2(COC)CC=CC2)=O)CCC2(C=C(C=O)C2)C1.C1(C)CCOC1=O.N c1(C(N2CCC(O)(CNC(=O)CC3CCC3)C2)=O)cnc2[nH]ccnc1-2 CCCCC(C)C(=O)NCC(C1CCN(C(=O)CC2(OC)CCC2)CC1)C N1(C(C2OCCN(C(c3nn(CC)c(O)c3)=O)C2)=O)CCCC(C)(F)C1 C=C(C)C(O)CC(=O)NC1CCN(C(c2ccncc2)=O)C1C(C)C Cc1cc(NC(C2CCC(O)CN2C(=O)CCc2csnn2)=O)cnc1O N(C1=NCC(C2CC2)N1C)CCSCC c1(C(=O)NC(C)C2CCC2)c[nH]ccc1=O.N1(C2CC(C(=O)N)C2)CCOCC1 C1(NC(c2cccnn2)=O)CN(C(c2csc(-c3nc[nH]n3)n2)=O)CC1C1CC1 Cc1cc(OCC=O)cc(C)c1.CCC(C)(C)C.C1(C(C)(C)O)(C=O)CC1.N C#CCCCC(C)C(=O)NC(C)CC1CN(C(c2cncc(C(N)=O)c2)=O)C1 CC1CN(C(C2CCCCO2)=O)CC(C(=O)NCCCN(C)C)O1 C(CCCC(CO)NC(=O)Cn1cncc1C)NC(C1(CCC)CCC1)=O C=CCC(C)(CC)C(=O)N1CC2CC2(C)C1.c1(C=O)cc(C(=O)C(C)C)c[nH]1.N C#CC1(C(=O)NC2C3CC2N(C(=O)CC2CCC4CC4C2)C3)CCCC1 C(=O)(CC(CC)C(F)F)NCc1c(C(=O)NCC2(CCC)CCC2)scc1 C1(CNC(c2ccc(CC)nc2)=O)C2CCC(C2)N1C(C1CCCCC1)=O.O N1(C(C(C(=O)OC)(C)C)=O)CC2CCC(NC(=O)C(F)C3CCCC3)C2C1 CC(CN(C)C)CC(=O)NCc1ccsc1C(=O)NC1(CO)CC(O)C1 N1(C(c2ccc(CCC)cc2)=O)C2CCC1C(F)C(NC(=O)CC(CC)OC)C2 c1(CC(=O)NC2CCN(C(CC(CCC)O)=O)C2C)cn2cc(C)sc2n1 c1(OC)cc(CCNC(=O)C(=O)N(C(C)C)Cc2cnccn2)ccn1 C(N=c1nc(C)nc2[nH][nH]cc1-2)C1CN(C(CC(CCC=C(C)C)C)=O)C(C)C1 CC(C)CC(C)CC(=O)NC1C2CCC(C2)C1C(N1CC2CCC2(CO)C1)=O c1(SC)nc(Cl)c(CN2C(C(=O)Nc3ncc(C)c(Cl)n3)CC3CC23)c(Cl)n1 N12CC3CC(C1)CN(C3)C(=O)C1(CC1)CNCC(C)C2=O.c1ccccc1.C C1(C(=O)OCCC2CN3CCC2CC3)COc2ccccc2C1 c1(C(N2CCN(C(CNC(CNC(CC)=O)=O)C)CC2)=O)cc2n(c1)CCCC2 Cc1cc(C#N)cc(C)c1CC(=O)NC(C)CN(C(=O)CCC(F)F)C c1(CC(=O)NCC(C)NC(C(CC)SC)=O)cccc([N+](=O)[O-])c1 c1(C(N2C(CNC(=O)C#CC(C)C)CC(OC)C2)=O)ccc(O)c(C)c1C c1(C(=O)NC(C)CNC(C2(CO)CCCO2)=O)cc(Cl)ccc1N c1(C(N(C)CCNC(=O)CCc2ncc[nH]2)=O)cnn2cccnc12 CCCCC(CNC(C1CC(O)C1)=O)NC(c1oc(C)nc1CC)=O c1(C(=O)NC2CN(C(c3n(CC)ccn3)=O)C2)cccc(-n2cncn2)c1 C1(C2CCN(C(=O)Cc3ncc(C)s3)C2)(NC(C=C(C)c2cccnc2)=O)CC1 C(=O)(C1=NOC(C(N2CCC(NC(c3ccc(F)c(F)c3)=O)CC2C)=O)C1)OC c1(C(=O)NCCN(C(c2n(CC#C)ccc2)=O)C)cc(C2CC2)cc(F)c1 N1(C(C=CC=CC)=O)CCC2CCC(C1)N2C(c1cc(C(C)C)on1)=O C(C)(C)(C(C)C)NC(C1N(C(CCC)=O)CCC1)=O.c1(C=O)ccc(O)nc1.N Cc1cccc(NC(C2CN(C(=O)NC3CCCS3)C2)=O)c1F C1(CNC(C2C=CCC2)=O)CC2COCC2N1C(c1cc[nH]n1)=O c1(C(=O)NCC)noc2ccc(Cl)cc12.C1CN(C(=O)CC2CC(F)C2)C1.O N1(Cc2cccc(Br)c2)CCc2c(-c3ccccc3)cccc21 N1(C(c2n(CC)cc(Cl)c2)=O)CC2CC(NC(c3ccc(O)nn3)=O)C1C2 N1(C(c2c(C)cc(OC)nc2)=O)CCCN(C(c2c[nH]nc2C)=O)CC1C(C)C c1(N2CCC(CC)(CO)C2)nc(=NCC2(F)CCC2)[nH]c2ccccc12 c1(C(C)O)ccc(C(=O)NCC2CCCCN2C(C2CCC(=O)N2)=O)cc1 c1(CC)nc(CCc2ccc(Cl)s2)n(-c2cccc(Br)c2)n1 N1(C(CCC(CCCC)C)=O)CC=C(C(C)(C)C(=O)N2CC(CCOC)C2)C1 N1(C(C(C(C)NC(c2nc(OCC)oc2)=O)(C)C)=O)CC2CCC(C2)C1.C c1(OC)ccccc1C(C)=CC(=O)NCC(O)CCNC(C1CC2CC2C1)=O C1(C=O)CN(C(=O)CC2CCC(=O)C2C)CC1(F)F.c1(OC)ccccc1C.N c1(N2CC(C(C)NC(=O)C=Cc3cccs3)OCC2)ccc([N+](=O)[O-])c(C#N)c1 N1(C(c2c(CC)occ2C)=O)CCC(N(C(=O)Cc2cnc(C)o2)C)C(C)C1 c1(C(=O)NCCCC(C)NC(C2C(C=C)CC2)=O)c(Br)ccc(F)c1N c1(N(C(C(CC=C)=C)=O)C(C)C(=O)OCC)ccc(C=C)cc1 O=C1Cc2ccc(C(N3CCN(C(=O)C(C#N)C4CC4)C(C(F)F)C3)=O)cc2N1 Cc1cn2nc(C(N3CC(O)(C(C)NC(C4CCCSC4)=O)C3)=O)cc(C)c2n1 c1(C(=O)NCC2CC(NC(=O)C#CC3CCC3)C(O)C2)cccc2c1C(=O)NC2 N1(C(=O)NC2CCCC(SCC)C2)CCCC2(C1)N=N2 N1(C(C(C)C)=O)CCC(C)(C)C1C(=O)NCC(F)Cl C12(NC(C(OC)OC)=O)CC1CN(C(=O)C(C1CCOCC1)O)C2 c1(CC)cc(NC(C2(F)CCN(C(C3(C(=O)CC)CC3)=O)C2)=O)cc(C)c1 c1(CC(=O)NC2CCC(NC(C3CCC(CC)O3)=O)C2)cccc(F)c1Cl Cc1cccc2cc(OC(c3c(OC(=O)C(C)(C)C)cnn3C)=O)ccc12 c1(C(N2CCC(CNS(CCC(=O)OC)(=O)=O)C2)=O)cnc2ccc(F)cn12 N1(C(c2cc(C)n(C(C)C)n2)=O)CC(NC(=O)CC2(O)CCC2)CCC1C C(=O)(C(CNC(=O)Cc1ccoc1C)CC(C)C)N(CC)CC1CCCO1 CC(C(C)(C)CO)NC(=O)C=CCNC(=O)COc1ccccc1 C(=O)(C1=C(C#N)CCC1)N1CCC(NC(=O)CC2CC(C)(C)OC2=O)C1.CC c1(C(N(CC(CNC(C(CC)C(C)C)=O)O)C)=O)cccc2ccccc12 C(C(C)(C(=O)NCCCCCN(C)C)NC(=O)C=Cc1ccoc1)SC c1(C(N2C3CC(NC(CSS(C)(=O)=O)=O)(C3)C2)=O)cnc2ccnn2c1 NC(=O)CCCCC(=O)N1CCCN(C(=O)CCc2ccc(O)cc2)CC1CO C=C(Cl)CC(C(=O)NCC1(OC)CC1)NC(=O)C=CC1(C)COC1 CCC(C)(C(=O)NC1CC(F)CN(C(c2ccc(F)cc2)=O)C1)C(N)=O c1(COCC)nc(N(CCCNC(c2nc(C)oc2C)=O)CC)cc(C)n1 c1(C(N(CC(CN(C(CC(CC)O)=O)C)O)C)=O)ccc(Cl)cc1C(F)(F)F C1(CN(C)C(c2csc(-c3cccs3)n2)=O)CCN(C(C2(C)CC2)=O)C1 Cc1sc2cncn2c1CNC(=O)Cc1cc(=O)n(C2CCS(=O)(=O)C2)[nH]1 N1(C(COC(C)=O)=O)CCCC(C(=O)N(C)Cc2nc(C)cs2)C1 C1(C(=O)NCCNC(C)=O)CC(NC(C2CC=CC2)=O)C1(C)C O(P(=O)(OCC)C1(NC(=O)CCc2ccc(O)cc2)CCNCC1)CC c1(C(C)C)conc1CC(=O)N(C)C.C1CCN(C(=O)C(C2CC2)N(C)C)C1 C(C(C(C)(C)C)NC(C1CCN(C)C1)=O)N(C)C.C(=O)CCC1CC1(F)F.N Cc1ccc(Br)cc1C(C)NC(=O)NC1CC2COCC2C1 N1(C(C=C(C)Cl)=O)CC2C(CN(C(=O)CCn3cccn3)C)C2C1 C1(C(=O)NCc2c(C)ocn2)(Cc2ccc(C(F)(F)F)cc2)CCOCC1 N1(C(CCC2(C)N=N2)=O)CC2(CC(C(N3CCOC(C(C)(C)C)C3)=O)CO2)C1 CC1=CCC(C(N2CCC(CC(=O)N(C)Cc3c[nH]nc3C)CC2)=O)CC1 C1(CNC(=O)CO)CCCC(NC(c2ccncc2C(F)(F)F)=O)C1 C#CCCCC(C)C(=O)N1CC2(CCCC2NC(=O)CNC=O)C1 C(=O)(C(CC1C=CCC1)N(CC(F)Cl)C)NC(CC)C Cc1ccc(C(=O)NCCOCCC)c(C)c1.C1(C)(CC=O)CC1(F)Cl.N C(C1=NOC2CCCC12)NC(CN(C(c1c(CC)occ1)=O)C)=O CC(CC(=O)NC1CC2CC(C1)N(C(c1ccc(C#N)s1)=O)C2)C(C)(C)C CC1CCCCC1(C)C(=O)N(C)CCN(C)C(c1nc(Cl)sc1Cl)=O c1(C(N(C2CCN(C(=O)C(C#N)C(C)C)C2)CC)=O)nnc(O)c2c1CCCC2 C1(CNC(CCCSC)=O)CCC(C)N(C(=O)C=Cc2cnn(C)c2C)C1 c1(C(=O)NCCCCN(C(CCN(CC)CC)=O)C)cccnc1S Cc1nc(NC(=O)C(N2CCC3CNC3C2)=O)c2ccccn12 C(=O)(C(C)(C)S(C)(=O)=O)N1CC(F)(CNC(C(C(COC)C)C)=O)C1 C12(C(N3C(OC)C(Br)CCC3C(=O)O)=O)CC(C(=O)O)(C1)OC21CCC1 C1(C(=O)NCC=CCNC(CCN(CC)CC)=O)CCOCC1(C)C Cc1cccc(Br)c1C(C(=O)NCc1ccsc1)NC(C1CC2CCC1CC2)=O N1(C(CC(C)C2CC2)=O)CC(C2CCCN(C(c3cnc(S)n3C)=O)C2)C1 CCCCC(C(=O)N(C)CC1(C)CC1)NC(C1CC2(C1)CC(O)C2)=O c1(C(C)NC(CCNC)C)cnc(-c2ccncc2)s1.CCS C1(O)(C(CNC(C2C(=C)C2)=O)(C)C)CN(C(C2(SC)CCC2)=O)C1 N1(C(C2CC(C#C)(O)C2)=O)CCCN(C(c2csc3nccn23)=O)CC1C C1(NCc2nc(C)n(C(F)F)c2)CCN(C(=O)OC(C)(C)C)CC(C)C1 C1(C(N(CCCO)CC#C)=O)CCCCCCN1C(c1ccc2[nH]ccc2n1)=O c1(C(N2CCC(F)(CNC(C3(Cl)CC34CCC4)=O)CC2)=O)nccc2n[nH]cc12 N1(C(CC2CN(C(C)=O)C2)=O)CCC(F)(F)C(NC(c2ccsn2)=O)C1 Cc1sc(O)nc1C(=O)NCC1(O)CC(C)C1.C1(C=O)CCC(C)(C)O1 C=C(C)CC(C(=O)NCC(C)N(C)C)NC(c1cccc(NC)n1)=O.C1CC1 N#CC1CCCC1NC(=O)CCC1(NC(=O)C=CCN2CCC2)CCC1 C(C)(C(O)C(C)C)NC(CCN(C(=O)C(N)=O)CC#C)=O C1(C(N(C)CC2(NC(C3CC3F)=O)CC2)=O)CC(=O)NC1(C)C c1(C=O)ccc(-n2cccc2)c(F)c1.C(C(=O)N)(C1CC1)OCC.CC(F)C CC1CCc2c(C(=O)NC3CCN(C(=O)C(F)F)CC3F)csc2C1 N1(C(C2CC(=O)NCC2)=O)CC(C(=O)NCCO)C(F)(F)C1.C1CCCC1.C CCC(C(=O)NCCCNC(c1cn(CCO)nn1)=O)Oc1ccccc1 N1(C(=O)CN2CC3C=CC2C3)CC2CC(NC(=O)C3=COCC3)C2C1 C(CC(C)C)(C(=O)NCC(C)S(C)(=O)=O)OC.C1(Cl)(C(=O)N)CC1(F)F C(=O)(C(F)C(F)(F)F)N1C(C(N(CCC)CC2CC2)=O)C=CC1 C(=O)(C(F)(F)C(F)(F)F)NCCC1(O)CN(C(=O)CCc2ccccc2Cl)C1 c1(C(=O)NCCNC(=O)CC2CCC3(CC3)CO2)cc2cc(Cl)cnc2o1 O=C(CCCC(F)F)NCCC1CN(C(c2cnn(C3CCOCC3)c2)=O)C1 c1(CNC(=O)NC2C(C)(C(=O)OCC)CCCC2)c(Cl)cnc(Cl)c1Cl c1(C(=O)NCC2N(C(CC(C)CF)=O)CCOC2)cc(Cl)cc2ccncc12 Cc1cn(C)nc1C=O.C(C(C)(C)C)N(CC(C)C)C(C1(CC)CC1)=O.N N1(C(C2CCC(C(=O)O)O2)=O)CC(=O)NC(c2cn[nH]c2)C1 c1ccc2c(c1)CN(C(c1c(C)noc1C)=O)C2.C1(CC(=O)NC)(OC)CCC1 S(=O)(=O)(c1cnccc1N1CCCC(c2ncco2)C1)NCC(CS(C)(=O)=O)O S(=O)(=O)(c1cccc(=NCC(C)C(=O)OC)[nH]1)NC(CCN(CC)CC)CO c1(OC)ccccc1C(C)CC(=O)NCC1CCOC1.c1(C=O)cn(C)nn1.N CC1(C#CC(=O)N2CCOC(C(=O)NCC3(C4(O)CCC4)CC3)C2)CCCO1 c1(NC(CCOC2CN(C(C(CO)NC(N)=O)=O)C2)=O)cccc2ccoc12 N1(C(C(=O)NCc2ccccc2)CCc2ccsc2)CCN2CCC1C2 C(C(C)(CC(C)C)NC(c1conc1C)=O)NC(c1ncc(OC)cn1)=O c1(CC(=O)NCC23CCCN(C(c4cccnn4)=O)C2C3)ccc2nc[nH]c2c1 C1(n2c(-c3cccc(-c4nccc(=NC)[nH]4)c3)ncc2)CCN(C)CC1C#N Cc1cc(C(=O)NCCC(C)N(C(=O)CC2CCC(=O)N2)C)c(C)nc1C C1(NC(c2nc(C(C)C)oc2)=O)COCCN(C(C2CCC(C)C(C)C2)=O)C1 C(=O)(CC(C)(O)C(F)(F)F)N(CCCCNC(c1ccc(C(C)C)o1)=O)C c1(C(=O)OC)cc(C)nn1CC(=O)NCCCC(C)NC(=O)C(C)(C)CO N1(C(COCCCOC)=O)CCC2(CC2)CC1C(=O)NC1CCN(CCF)C1 C(=O)(C1=NNC(=O)CC1)NCC(n1cc(-c2ccc(OC)nc2)nn1)C c1(C(N(CC(C)NC(=O)CC(C)OC)CC)=O)cnc2c(cnn2C)c1OC c1(C(c2ccccn2)NC(CC2CCC(C)CO2)=O)ccc(Cl)c(Cl)c1 N1(C(C=CCOC)=O)CCN(C(=O)C(F)(F)CN(C)C)CC1CC(C)(C)C c1(C(N2CC(OCC(N3CC(CC(=O)OC)C3)=O)C2)=O)ccc(F)cc1 C1(NC(C(=CC2CCCC2)C)=O)CCC(O)CN(C(C2CCN(C)C(=O)C2)=O)C1 C12(C=O)CCC(CC1)C2.c1(CC)nonc1C(=O)NCC12CC(C1)C2 CC(C)CC(C(=O)N1CC(CC(=O)NC2CCC(CO)CC2)CC1(C)C)N(C)C c1(C(=O)NC2C(O)CCN(C(C(C)C3CCC3)=O)C2)csc2ccccc12 N1(C(c2c(COC)cccn2)=O)CC2=C(C1)CN(C(C1(CF)CC1)=O)C2 C(=O)(CCS(=O)(=O)c1ccccc1)NCC1C(NC(C=CSC)=O)CC1 N1(C(C2CC(=O)OC2)=O)CCC2CN(C(=O)C(F)(F)C3(O)CCC3)CC2C1 c1(C(=O)NC2CN(C(C=CC)=O)C(C)(CC)C2)cc(Cl)c(OC)c2cccnc12 C1(CC)CN(C(=O)CC2CCC3CC23)CCO1.C1(C(=O)N)(COC)CCCC1 c1(CC(=O)NC(CNC(C(=O)NC(C)C)=O)C)ccc(S(C)=O)cc1 CCCC(CCCNC(c1ccc(C(O)CF)cc1)=O)N=c1[nH]nc(C)s1 C1(NC(c2cccc(C)c2F)=O)CN(C(c2cnsc2)=O)CC2(CCOCC2)C1 c1(-n2c(CC(c3cccc(Cl)c3)C)nc(COC)n2)ccc(C)c(F)c1 C(=O)C(C)(C)CS(C)(=O)=O.C1(C)(CNC(CN2C(C)CCC2)=O)CCCCC1 C#CCC(CC(=O)N1CCOC(C)CC1)NC(=O)CCN=[N+]=[N-] C1(C(=O)N)C2CCC(C2)S1(=O)=O.Cc1ccnc(C(N2CC(O)(C)C2)=O)c1N CC1CCCCC1(CNC(c1cc(N)c(F)cn1)=O)NC(=O)CCCCCF N1(C(C(=O)NCC2(NC(C=CC)=O)CCC2)=O)CC(O)(CO)C1 N1(C(C2CC(OC)C2)=O)C2CCC1CC(F)(CNC(C)=O)C2 N1(C(COCCC)=O)CCCC(NC(c2ccccc2C2CCOC2)=O)CCC1 C(=O)(CC(C(F)F)NC(=O)CN1C(=O)CCCC1=O)NC1(C)CCSC1 C1(C(=O)NCc2c(C)cco2)C(C2CC2)CCN1C(c1cc2cccn2cn1)=O Cc1cncc(C(=O)NCC(C)(C)CCNC(c2cn(C(C)(C)C)nn2)=O)n1 n1(CC)nc(C(=O)NCCC(C)C)c(C)n1.C(=O)C(O)Cc1cnn(C)c1.N c1(COC)ncsc1C(=O)NCCC(C)N(C(=O)CC(C)C1CCCCC1)C n1(-c2cc(NC3(C(=O)OC)CC(C(F)F)C3)ncn2)nc(C)c(Br)c1C CC(C)(CCNC(C1CC1F)=O)C(=O)N1CC(C)(C)C1C1CC1 CC(C)CCC(C(=O)NCC1(C)CC1(F)F)NC(c1n[nH]c2c1CCC2)=O CC1(C)CC(CC(=O)NOCC2CCC2)N(C(C2(O)CCOC2(C)C)=O)C1 CCC(c1ccccc1)=CC(=O)NCC(CCOC)NC(C1CCCSC1)=O C(C(C)(C)C(=O)NC1CCCC(NC(=O)C(C)NC(N)=O)C1)SC c1(NC(C2(C)CCN(C(CCOC)=O)C2)=O)c(I)cccc1C#N c1(C(N2CC3N(C(C(CC)(C)C)=O)C(CC3)C2)=O)cnc2c(c1)NC(=O)CN2C C1(NC(Cc2c(C)cccc2)=O)CC(F)CN(C(C2CC3CC3C2)=O)C1 c1(C(N2CCCC(NC(COc3cc(C)on3)=O)CC2)=O)cc(F)c(C)cc1N c1(C(=O)NCC(CC)NC(=O)CSS(C)(=O)=O)cn(CCO)c(=O)nc1O c1(NC(=O)CC2CC(NC(c3ccc(O)cc3)=O)C2)cc2ccccc2c(Cl)n1 c1(CC2CN(CC(n3cc(C4CCCCC4O)nn3)C)C2)ccc(P(C)(C)=O)s1 C1(C(N2CCC(CNC(c3cscn3)=O)C2)=O)(COC)CCCOC1 C=Cc1ccc(C(=O)NC2C3CCN(C(=O)C(CC4CC4)OC)CC23)cc1 c1(C(=O)NCC(C)N(C(=O)CCn2c(C)ccc2C)CC)ccnc(Cl)c1 N1(C(c2[nH]cc(C)c2C)=O)CC(C(=O)NCCn2ncnn2)C2(CC2)C1 C1(CC(=O)N(CC(C)N(C(CC2CCC2)=O)C)C)CC(F)(F)C1.CCO N1(C(c2scc(OC)c2)=O)CCCC(CCNC(c2cnccc2OC)=O)CC1 c1(C(=O)NCC=CC(=O)NCCC(C)C2CC2)cc(O)ncn1 c1(CC)ccc(C=O)c(C)c1.C1(CC(=O)N(C2CCC2)C)CC(C)(C)CO1.N CCCCC(CNC(C1(SC)CC1)=O)NC(=O)CNS(=O)(=O)CCCC C(C(CC)N=c1nn[nH]n1C)NC(c1c(COC)noc1)=O C#CC12C3C4C1C1C2C3C41C(N1CC(C)(NC(=O)C(CC)NC)C1)=O C1(C(=O)NCC=C2CCN(C(C=C3CCN(C)C3)=O)CC2)CCCCCS1(=O)=O c1(CC)ncc(C(=O)NCCN(C(=O)C(C)(C)C#N)C)cn1 c1(CC(C)C)ccc(S(=O)(=O)NCC2CC3CC3C2)cc1 N1(C(c2cc(OC)ns2)=O)CCC(NC(c2cn(C(C)(C)C)nn2)=O)C1(C)C CC(C(=O)N1CCOCC1)C(=O)N1CCC(NC(=O)C)C1.[SH](=O)(=O)C1CC1.N c1(C(N2CC(NC(C3(CC)CCCC3)=O)C3C2C3)=O)nc2cc(O)ccc2[nH]1 C(CC(O)C(=O)N1CC(O)(CCNC(=O)CCN2CCCS2(=O)=O)C1)SC C(=O)(C(C)(C)C(C)O)N1CC(C=O)C1.N1(C(C)C(=O)NCC)CCNC1=O.N c1(COC(c2cn(CC3CCOC3)nn2)=O)nc2cc(Br)ccc2s1 C1(C)(CNC(C2(C(C)(F)F)CC2)=O)CCCN1C(C1CCC(=O)O1)=O CC(C)CC(CC(=O)NCC1CCCOCC1)NC(=O)CC1CCC(=O)C1C N#Cc1ccc2c(c1)CCCC2NC(C1CCN(C2COC2)C1)=O n1(CCN(CC)CC)cc(C2(NC(c3cnoc3C)=O)CCC2)nn1 Cc1cccc(C(N)CNC(=O)CC2COC3CC2C3)c1 C(CC(C)(C)C)(C(=O)N1CCC(C)(CNC(=O)CCCC#N)CC1)OC c1(-c2cn(C(C)C)nn2)ccc(C(=O)O)c(Cl)c1.c1(C=O)ccc(C(C)(C)C)[nH]1 C(=O)(C(C)(C)CC(F)(F)F)N1CC2C(CNC(CC(CC)C(C)C)=O)(C2)C1 c1(CC)cccnc1C(=O)NC(C)CN(C(=O)CCc1ccc(Cl)cc1)C c1(C(=O)NCC(c2ccccc2F)NC(C2CCCC2)=O)ccn2ccsc12 Cc1cc(F)c(C(=O)NCCCN(CCO)C(c2cnsc2C)=O)cc1F N1(C(C2SCCCS2)=O)CC2CC1CN2C(C12CCCC(C1)OC2)=O C=C(C)C(O)CC(=O)NCCCNC(=O)Cn1c(-c2cccs2)nnc1S c1(C(C)NC(C(N2CC(CNC(C)=O)OCC2)=O)=O)c(C)cccc1C N1(C(c2c(CC)nn[nH]2)=O)CC2C(C(=O)NCC(C3CCCC3)O)C2C1 N1(C(CCC2CCN(C(c3occ(C)c3)=O)C2)=O)CCC2(CC1)CN(C)C2 C1(C(CNC(CC2(C=C)CC2)=O)(C)C)CCCCN1C(=O)COC(F)(F)F c1(OC)ccc(NC(=O)Cn2cc(I)cn2)cc1Br c1(C(N(CCN(C(C)C)C(C2CC2(F)Cl)=O)C)=O)cncc2sccc12 C(=O)(C(CC(F)F)N(C(=O)CS)C)NCC(C)Cn1ccnc1.C(C)(C)C C1(C(=O)NCC2(NC(C(C)=C(CC)C)=O)CC2)CCN(CC(C)C)C1 N1(C(C2OCCN(CC)C2)=O)CC(CC(=O)Nc2cncc(Cl)c2)C2(CC2)C1 C(c1ncc[nH]1)=CC(=O)NCc1csc(CNC(c2ccccn2)=O)n1 n1(CC)nc(C)cc1C(=O)NCC1CN(C(=O)C(C)C(=O)OC)CCO1 N1(C(C(CC(=C)C)C)=O)CCC2C1CCCN2C(=O)CC1=NNC(=O)C1 N1(C(c2n[nH]c(CC)c2Cl)=O)CCN(C(=O)CC2C(C)C2(F)F)C2(CCC2)C1 C(=O)(N=c1cc[nH]c2cc[nH]c12)C1N(Cc2ccc(C)c(C#N)c2)CCSC1 c1(NC(C2(C)CCN(C(c3cnc(O)[nH]3)=O)C2)=O)nc(Cl)c(Cl)nc1CO C#CC(CNC(=O)C(c1cccs1)NC(=O)CCc1nncs1)CC C1(NC(CCc2cn(C)nc2)=O)CCSC12CN(C(=O)C=Cc1cccs1)C2 N(C(=NCCc1ccn(C)n1)NC1CCC(=O)NC1)C(C=C)C N1(C(c2cn(C(C)C)nc2)=O)CC=C(CC(=O)NC2C3CCCOC23)CC1 C1(NC(C2(C)CCNC(=O)C2)=O)CN(C(C2(CCF)CC2)=O)C2CCCCC12 c1(OCC)cc(CNC(=O)CCNC(C2C=C(C)CS2)=O)on1 C1(NC(CC2CCCC(C)(C)O2)=O)CC2CCC1CN(C(C1(C)CCCO1)=O)C2 N1(C(COCC(=C)C)=O)CCCN(CCNC(=O)CC2CC3COCC23)CC1 Cc1cc(C2(C(=O)NC3CCC(C)N(C(=O)C#CC(C)C)C3)CC2)cc(C)c1 C1(CC(=O)NC(CN(C(c2ncsc2Br)=O)CC)C)C=CCCC1 c1(OC)cccc(Br)c1C(N1CC2(NC(=O)C(C)C(C)O)CCC1C2)=O C1(C(CO)NC(C2CC(=C)C2)=O)CCN(C(=O)C(c2ccccc2)N(C)C)CC1 CC1C(NC(C23CC(C)(C2)OC3C)=O)CCCN1C(=O)CSc1ccccc1O c1(C(=O)NC(C(C)OC)CC(=O)NCc2[nH]c(C)nc2C)c[nH]c2nccc-2c1 C1(NC(c2c(C)cn(C)c2)=O)CCSC12CN(C(C1(C)CC(C3CC3)=NO1)=O)C2 Cc1nccn1CCC(=O)NCCOC(C)(C)C.C1(C)(C=O)CC(C)C1.N CCC(C)(CCNC(=O)CC1CCC2CC12)NC(c1ccc(CO)s1)=O c1(CC)nn(Cc2ccccc2)cc1C(=O)N.C1CN(C(=O)C2=COCC2)CC1O CC1(C)CC(NC(C2CC(=O)CN2C(C2(C#N)CCOCC2)=O)=O)C(C)(C)O1 c1(N2CCC(C=O)C2)ccc(Cl)c(F)c1.CC(O)(C)C.C1(C=O)CCS1(=O)=O c1(C(=O)Nc2ccc(-c3cnc(C)s3)s2)c(C#N)cnn1C N1(C(C(C#C)(C)C)=O)CCCN(C(c2sc(C(C)OC)nc2C)=O)CCC1 c1(NC(C(=O)N(C)Cc2cn(CC#C)nc2)=O)ccc2c(C)nn(C)c2c1 C#Cc1ccccc1CC(N1CCC(NC(=O)C(O)C(C)CC)C1(C)C)=O CC1CN(C(=O)CC23CCCC2C3)CCCN1C(c1c(Cl)cnn1C)=O c1(OC)ccc(C(c2nnnn2C(C)C)NCCC2CC(C)(C)CO2)cn1 C#CC1CN(C(c2cnco2)=O)CCN1C(C1CC2C=CC1CC2)=O Cc1cncc(NC(C2CC3CNC2C3)=O)c1C C12(C(N(CC)CC)=O)CC=CCN1CCC2.C1(C=O)CCC(C(N)=O)O1.CO CC1CCCCC1(CNC(c1ccc(Cl)c(N)c1)=O)NC(c1ncc[nH]c1=O)=O C1(N(C(C(N2CCCCC2=O)C)=O)C)CCCCN(C(C2(CC(F)F)CC2)=O)C1 CCCC(CC)CCC(=O)N(CC(=O)NC(CO)CCF)C C(=O)(C1SCCc2ccccc21)NC(C)CNC(=O)CC1CCC=CCC1 c1(C(N2CCN(C(C(SC)SC)=O)C(C(C)C)C2)=O)ncn2ccccc12 N1(C(=O)C=CCCc2ccccc2)CC2CCN(C(=O)Cn3ccnn3)C2C1 c1(C(N(CC(C)(C)NC(C=C(C)C)=O)C)=O)c(C)cc(O)nc1C CC1(C)CCN(C(=O)Cn2ncc(C#N)c2N)C1CNC(=O)CCCC(N)=O C(=O)(C1CCc2c[nH]nc21)N1CCC(NC(C(C)C)=O)C(CO)C1 CC1(CCC(N2CCN(C(=O)C)CC2)=O)CCC(=O)N1.N1(CC(=O)N)CC=CC1 c1ccc2cc(F)cc(Br)c2n1.c1(COCC)nc(C2(COC)CC2)n(C)n1 c1(C(=O)NC2CC2CNC(C23CC(C2)C3)=O)cc(Br)c2[nH]nnc2c1 N1(C(CC(=O)NCC)=O)CC(NC(c2cnn(CC(C)C)c2)=O)C(C)C1.C Cc1cc(F)ccc1-n1nc(-c2ccccc2Cl)nc1C1(C)CCCN1 C(=O)(C1=NN(CC)C(=O)CC1)N(CC(CC)NC(=O)C(F)n1cccn1)C c1(CSCCNC(C2(C(C)C)COC2)=O)cn(C2C=CCCC2)nn1 C1CC(CC)N(C(c2cc(C(C)=O)c[nH]2)=O)C1.C(=O)CC(C)(C)C1CC1.CO c1(C(C)C)ccc(C(N2C3CN(S(=O)(=O)c4cccs4)CC23)=O)cc1Br C(=O)(C(O)CC(F)(F)F)NCC(=O)NCC(=O)N(C)Cc1ccco1 c1(C(=O)NC2CN(C(c3cccc(C#C)c3)=O)C(CO)C2)cc2cccnc2[nH]1 n1(C(C(=O)NCCN(C(=O)C=CC2CCCC2)C)C)ccc(Br)n1 c1(N2C(COC)(CNC(=O)CCCC3CCCC3)CCC2)ccnc2ncnn12 N1(C(CCC(=C)C)=O)CC(C)OC2(CCN(C(C3(CF)COC3)=O)C2)C1 CCCCC(C)C(=O)NCCC1CC(NC(=O)C(=Cc2cccnc2)F)C1 c1(OC)cccc2ccc(C(=O)NC(C)CCN(C)C(C3(C#N)CCC3)=O)nc12 N1(C(c2cncc(C)c2)=O)CCCC2CN(C(C3(C)CCC(C)C3(C)C)=O)CC12 Cc1c(Cl)ccc(C(N2CC(N(C)C(c3cc(Cl)cn3C)=O)C2)=O)c1Cl c1(CC)nc(C(N2CCCC2C(C)NC(C2CC=CCC2)=O)=O)co1 C#CCCCCCCC(=O)N1CCC(NC(c2n[nH]c(C)c2O)=O)C(CC)C1 C(=O)(C#CC1(C)CCCO1)N1CCN(C(CN(C)C(C2CC2(C)C)=O)=O)CC1 C1(NC(c2ccc(C)s2)=O)CC2CC1N(C(c1cnc(-c3ccoc3)s1)=O)C2 C(=O)(C(C)C(C)NC(C1(F)CC=CCC1)=O)N(CCOCCOC)C c1(C(N2CC(C(=O)NC(C#C)CCC)(SC)C2)=O)ccncc1OCC C1(NC(N)=O)CCCN(C(c2ccn(CC(F)F)n2)=O)C1 N1(C(C=CC)=O)CCC(C2(NC(c3nc(OC)c(C)s3)=O)CC2)C1 C1(C)(N(CCC)C(=O)CC)CCCCC1.C(=O)C.C1CC1.[SH](C)(=O)=O CC1CN(C(c2ccc(C#N)o2)=O)CCCN1C(c1ccnc(OCCO)c1)=O C(C)(CCC(=O)N1CCCC1C(C)NC(=O)CCOCC(F)(F)F)SC C(=O)(CC(CC)CC(C)C)NC1(CNC(C(CCC=C)(C)C)=O)CC(F)(F)C1 C1(NC(CCC(=O)N(CCC)CCC)=O)CCN(C(=O)C2CC2)CC1C C1(NC(C2(C)CC(=C)C2)=O)CCN(C(=O)CC2CCC2C)CC1C(N)=O C1(NC(Cn2nc(C)oc2=O)=O)CCCN(C(c2ccc(C)o2)=O)CCC1 c1(C(=O)NC2(CF)CCN(C(C=CC(CC)C)=O)C2)cnn2ccc(C)cc12 N1(C(CC2(OC)CC2)=O)CC2CC1C2C(=O)NCCOc1ccccc1F C1(CNC(C(C=C)(C)C)=O)CCCCN(C(c2cn(-c3cccnc3)nn2)=O)C1 c1(N2CCC(C)(F)C2)ccc(S(=O)(=O)N2CCCC(OC3CCC3)C2)cc1F c1(C(=O)NCC(CC)(C)C(=O)NCCOc2ccccc2)cncc2[nH]ccc12 C1(NC(C(CCC)NC(=O)C(O)Cn2cncn2)=O)Cc2ccccc2C1 CCC#CC(C)(C)NC(C1(C(C)NC(=O)C(C(C)C)OCC)CC1)=O C(=O)(C(C#N)C(C)(C)C)N1CC(NC(c2oc(C)c(Br)c2)=O)C(O)C1 C1(C(C)C)C(C(C)C)CN1C(=O)CC1CCN(C(c2cccnn2)=O)C1 N1(CCC(=O)NCCCN(C(=O)C(CCC)=CCC)CC#C)CCC(O)CC1 S(=O)(=O)(c1ccc(Cl)cc1F)Nc1ccc(C(C)C)cc1F C(CC(CC)C(=O)N1CCCC(O)(CNC(c2ccc(C)c(F)c2)=O)C1)=CC C1(NC(C2(NC(CC3C(C)OCC3)=O)CCC2)=O)CCC(C)(C)C(C)C1 c1(CC)ncnc(CC)c1C(=O)NCCCCC(C)NC(c1cnc(C)s1)=O C1(CC)CN(C(c2ccn(C)c2)=O)CCN1C(=O)CCN1CCN(C(C)C)CC1 N1(C(CCC(=C)Cl)=O)CC2CC(NC(C3(C)CC(O)CN3C)=O)CC(C2)C1 c1(C(N(C(c2ccc(Br)s2)C(=O)OC)C)=O)ccccc1CS(C)(=O)=O C(=O)(C1=NOC2COCC12)NCC1(NC(C=C(C)C(F)F)=O)CCC1 N1(CC)CC(NC(C2(C(C)C)CCN(C(=O)C(C)N(C)C)C2)=O)C(C)C1 N1(C(CC2(C)CCCC2)=O)CC2(CC(NC(c3ccn4cnnc4c3)=O)CO2)C1 C1(O)CCN(C(C2CC2c2cccnc2)=O)CC1.CC1(C)CCC(C(=O)NC)O1 Cc1c(C(N2CC(NC(=O)CCc3cnn[nH]3)CC(C)C2)=O)ccc2cncn12 Cc1cccc(NCC(=O)NCC2COCCN2C(=O)C(CCO)N(C)C)c1C CCCCCCCNC(=O)CC1CN(C(=O)O)C1.C(=O)C(N)=O.C(C)(C)C C(CC(CO)C(C)C)NC(C1(CNC(=O)C2=C(Cl)CC2)CC(=C)C1)=O C(=O)(C(F)CCC(C)C)N1C2C(NC(c3c(CCC)nco3)=O)CC(C2)C1 CCC(C)(CC)C(=O)NCC1CC(F)CN1C(c1cccc(C(F)(F)F)c1)=O N1(C(c2nncc(C)c2)=O)CC(CO)C2(C1)CN(C(C1CC3CCC1CC3)=O)C2 N(C(=NCC)N1CCC(c2ncccn2)CC1)C(C=C)C.N1(C=O)CCCCC1 C1(NC(C(COC)COC)=O)COC2(C1)CN(C(=O)Cc1ccc(Cl)cc1Cl)C2 N1(CCNC(C(C)(CC)OC)c2n(CC)nnn2)Cc2ccccc2C1 c1(OC)ccc(CN2CCCC(C(C)NC(c3cncc(O)c3)=O)C2)c(Br)c1 c1(C(=O)NCC2CCCC(CNC(C(CC)SC)=O)C2)c(Cl)c(C)nn1C CCCCC(O)CCC(=O)N1CC2CN(C(C3CC4(C3)CC(F)C4)=O)CC2C1 N1(C(CCS(C)=O)=O)C2CCC1CC(CNC(=O)CCC1CCCCO1)C2 CC1CCOCC1C(=O)NC1CC2(C1)CC2C(=O)NCC1CC1 C(C)(C(=O)NCCC1CN(C(=O)C(C)CC2CCC2)C1)(C1CC1)OC c1(C(N2CCC(C(C)NC(COCc3ncc(C)o3)=O)C2)=O)csc(C)c1C c1(SC)ccc(N)cc1C(N1CCC(CNC(C2CC(F)C(=O)N2)=O)C1)=O c1(C(N2CC(C(C)NC(c3ccc(OC)c(Cl)n3)=O)C2)=O)scc2c1CCCC2 C=Cn1ncc(C(=O)NCCOCC(=O)NC2CCCN(C)CC2)c1N Cc1cc(F)cc(NC(C2CC(C)CN2C(c2ccno2)=O)=O)c1O c1(C(N2CC3C(NC(c4nc(C)nn4C)=O)(C3)C2)=O)cccc(O)c1Cl c1(C(N2CCCC(C(=O)Nc3nc(Cl)ccc3F)C2)=O)c(F)c(F)cc(F)c1F C1CN(C(=O)Cc2cccc(C)c2F)CCCO1.C1(C(=O)NC)(OC)CC(C)C1 C1(COCC(=O)NCCOCCC)CCCO1.C1(CC(=O)N)CCCO1 C12CC(N(C(=O)Cc3nc[nH]n3)C1)C(=O)N2.C1CCCC1.O=CCC1CC1.N Cn1nnc2c(C(=O)NCC3CN(C(c4ccnnc4S)=O)CCO3)ccnc12 C1(CC(=O)N)CC2(C1)CN(C(=O)CC1CNC(=O)O1)C2.C1CC2(CCC2)C1 C(=O)(C1=C(CC)OCCS1)N(CC1N(C(C2(CC#C)CCCC2)=O)CCC1)C CCC(CC)CC(=O)N1CCCC(CCCCNC(c2nnc(O)nc2O)=O)C1 CC(CCCNC(c1cn(C(C)(C)C)nn1)=O)NC(C1(CF)COC1)=O C1(NC(CCSCC)=O)CN(C(=O)COC2CCCOC2)CC(C)(C)C1 c1(C(=O)NCCCCC(=O)N(C)CC2CC2(C)C)cc2ncccc2[nH]1 C1(NC(=O)Nc2cccc(C3CCCC3)c2)CCc2ccccc2C1 C1(C(=O)OC)CN(C(=O)NNC(=O)c2c(C)coc2C)CCC1C(=O)O c12cc(C)c3ccc(cc3n1)S2.C(=O)(CCN(C)CCN(C)C1CC1)OCC C(=O)(CC(C)(C)C(=O)NCC(C)(C)OCCNC(c1cscn1)=O)OC Cc1cnc2[nH]cc(CNC3CC3C(=O)Nc3nc(C(F)(F)F)ccc3Br)c2c1 C(CCCCCC(=O)NCCCn1cnnc1)NC(c1c(CC)cccc1)=O N1(C(C(C)NC(CC)(C)C)=O)CCC(CC)(NC(C2CCCN2C)=O)CC1 c1(CN(C2C(OC)COC2)C=O)cc(CO)cc(C)c1 c1(C(=O)OC)cc(NC(C2(C)CCN(C(=O)CCCN(C)C)C2)=O)ccc1Cl C(=O)(C1=COCCC1)NCC(C(C)C)NC(=O)Cn1ncc(C#N)c1N C(CC(C(=O)NC(C)COCC)NC(=O)C(C)n1ccnn1)OCC.O c1(CN2CC(CC#N)N(C(c3ccc(S)cc3)=O)CC2)ccccc1[N+](=O)[O-] c1(C(C)C)ccc(C(N2CC(C(O)C(=O)NCCCC(N)=O)C2)=O)o1 C1(C(=O)NCC(C)(C)CN)COC2(CCN(C(c3ccc(O)c(Cl)c3)=O)CC2)C1 n1(C(C)C)nc(C2CCC(C(C)(C)C)CC2)nc1-c1cc(O)ncn1 C(C)(C)(CC(=O)NCc1occc1C(=O)NC(c1ccccc1F)C)OC N1(C(c2cnc(C)s2)=O)CC2CC2(NC(=O)Cc2cn(C)nc2C)C1 C1(CNC(C2(C(=O)OC)CC2C)=O)CCCCNC1 c1(C(=O)N)ccnc2ncccc12.C1(NC(C2CC(C#N)C2)=O)CS(=O)(=O)CC1 n1(CC(=O)N(CC(C)O)Cc2ccc(OC)cc2)nnc2ccccc12 c1(C(=O)NC2CC(NC(C3OCCN(C)C3)=O)C2)ccc(C(F)F)nc1O c1(NC(C2CCN(C(Cc3cc(C)no3)=O)C2)C)cc(=O)n(C)c(=O)n1C c1(N2CCCC3(NC(c4ncc(C)c(Cl)c4)=O)C(C2)C3)ncc2c(n1)CCOC2 C12(CC(N(C)OCC(F)(F)F)=O)CCC1CN(C(C1(c3cccs3)CC1)=O)C2 c1(OC)ncc(CNC2CC(F)CN(C(c3cccnc3C(N)=O)=O)C2)cc1C CC1CCC(NC(C2(C)CCCN2C(=O)CC2OCCO2)=O)CC1 c1(C(=O)OC)c(C(=O)N(CC(O)CN(C)C(c2cc(C)sn2)=O)C)cnn1C C1CN(C(C2(n3cccn3)CC2)=O)CCC1(F)F.C1(SC)CC(C(=O)NC)C1 c1(OCC(=O)NC)ccc(C(F)(F)F)nc1.C1CCSCC1.C1CC(C=O)C1 C1(C(=O)NC(C)Cc2nn[nH]n2)(NC(C(C=C)C)=O)CCC(C)(C)C1 C1(C(CNC(C(C=C)O)=O)(C)C)CCCCN1C(c1cccc(C(F)(F)F)n1)=O c1(C(=O)OCC)cc(=NCC2CCC(NC(=O)CC3CC3)C2)[nH]c(C)n1 c1(NC(C2CCCCN2S(=O)(=O)CCCCl)=O)cc(Br)ccc1I C1(NC(CC(CC#C)NC(=O)CCC2CCOC2)=O)CCn2nnnc2C1 N1(C(C(C)CC(C)(C)C)=O)CC(NC(c2ccnc(O)c2)=O)CC12CCOCC2 S(=O)(=O)(c1csc2ccccc12)N1CCC2(C(C(N3C(C(N)=O)CCC3)=O)C2)C1 C1(CC)CN(C(c2cc(OC)cs2)=O)CCC1NC(=O)C(=O)NOC c1(COC)nc(O)cc(NC2CCCC(NC(=O)C(=O)NC(C)C)C2)n1 n1(CC(C)C)ncc(C(N2CC(NC(=O)C(C)CF)C(O)C2)=O)c1C1CC1 C(=O)(C1=NOC2(CCC2)C1)NC.N1(C(c2scc(COC)c2)=O)CCOCC1.C N1(C(COC)=O)CCC(CN(C)C(C2CCCC(OCC)C2)=O)CC1 C(=O)(CC(C1=CCCC1)OC)NC1C2N(C(CC=C)=O)C(CC2)C1 C1(N(C(C2CN(CCOC)C(=O)C2)=O)Cc2cccs2)CCc2n[nH]cc2C1 C1(NC(CNS(NC)(=O)=O)=O)CCCC(CNC(=O)CC(C)n2cccn2)C1 C1(CC)(NC(=O)C(CCO)N(C)C)CCCN(C(=O)CSc2nnnn2C)C1 CC1(C)CCOC1C1(NC(C2C(c3ccccc3)C2(F)F)=O)CC1 N1(C(=O)C2CC2)CCCCC1.C1(C(=O)O)CCCCC1n1cccc1 C1(N(C(C2N(C(Cc3ccc(C)s3)=O)CC2)=O)C)CCCC1(F)F N1(C(c2cc(CC)n(C)n2)=O)CC2(CCN(C(c3ccccn3)=O)CC2)CC1C C1(CNC(C(F)OC)=O)CCCCN(C(=O)COc2cnn(C(C)C)c2)C1 C(=O)(C1=C(C)OCC1)N1C(Cc2onc(C3(C(=O)OC)CCC3)n2)CCC1 c1(OCCCCC)ccc(NCc2ccc(C(F)F)nc2)cc1 N1(C(c2cc(C)cc(O)c2)=O)CC2CCC(CNC(=O)C3=CCCC3)(C2)C1 c1(OC)ccc(C(=O)NC(C)CC(C)C)c(C)n1.c1(C=O)ccc(C#N)n1C.N n1(CC(N2C(CCCNC(C(C)SCC)=O)CCC2)=O)c(C)ccc1C N1(C(c2n[nH]c(C)c2O)=O)CC2CC3CC2C1C3NC(=O)CS(=O)(=O)C(C)C N1(C(c2cncc(C(C)=O)c2)=O)CCC2CN(C(=O)C(C)N)CCC12.[SH](C)(=O)=O C1(OC)CCCC1C(=O)NCCCOCCNC(=O)CC1(C)CCCC1 Cc1nc2nccc(N3CCN(C(=O)C(C)C4CCC4)CC3C)n2n1 N1(C(CCc2nc(C)sc2)=O)CCC2CCCN(C(c3ccncc3N)=O)C2C1 Cc1cnn(CCNC(C2(NC(=O)C(C)n3ccnc3)CC(CO)C2)=O)c1 N#Cc1cc(F)c(Br)cc1NC(=O)Cc1cc(C2CC2)on1 CN1N=C(C(=O)N2CCCC2C(=O)NCC2CCC3(CC2)CC3)CCC1=O C(=O)(C#Cc1ccc(F)c(F)c1)N1CCCC(C)(C(=O)OC)C1 c1(C(N2CCC3CN(C(c4cnco4)=O)CC3C2)=O)cc2ccccc2nc1O C1(NC(c2nc(OC)oc2)=O)CC(NC(c2cnc(C(C)C)s2)=O)CC1O c1(C(=O)NC(c2ccccc2OCC(=O)NC)CC)cccc(S(C)=O)c1 c1(C(N2CCC(C)(C(=O)OC)CC2)C(=O)NCCSC)cc2cccc(Br)c2o1 C(=O)(C(F)C(F)(F)F)N1CC(CCC)C(C(=O)NCC(C)(Cl)CC)C1 C(=O)(C(F)C(F)(F)F)NCC1(C(N)=O)CN(C(c2ccns2)=O)C1 c1(CC)cccc(C(=O)N(C2CCCCC2N(C(=O)CCC(C)OC)C)C)c1C C(=O)(CC(C=O)N(C)C)OC.C1(C=O)C(C)(C)C1(C)C.C(C)(C)C.CC N1(C(CC2C(C)CCO2)=O)CCCC2(CCN(C(c3cc(F)cc(F)c3)=O)C2)C1 Cc1ncc(C(N2CC(O)(CNC(c3cccn(O)c3=O)=O)C2)=O)cc1N N1(C(CC(=O)NCC)=O)CCC(C(F)F)C1.C1(C=O)CCC(N(C)C)CC1.N N1(C(C=C(C)C(C)C)=O)CCCCC(N(C)C(c2ccc(NC(C)C)nc2)=O)C1 C(=O)(CC(C)(C)CC(F)F)NCCC(C(C)C)NC(c1ccnc2[nH]ncc12)=O C1(C(=O)OC(c2nn[nH]n2)C)CN(C)CCN1CC(C)(C)C c1(C(=O)OC)sc(C2(NC(C)CN(C)C)CCOC2)nc1C N1(C(C)=O)CSCC1C(=O)NC1(CCCC)CC1.N1(CC=O)CCC(C)C1.N CC1CN=C(N2CCN(C(c3ccc4c(c3)OCCO4)=O)CC2)S1 C(=O)(CCCCCCS(N)(=O)=O)N1C(CN(C(CC2CC(C)C2)=O)C)CCCC1 c1(CC)sc(C(=O)NC(CO)C(C)NC(=O)C(C)C2CC2)cc1C C1(C=O)CCC2(CCC2)C1.c1(CC)c[nH]c(C(=O)NCC2CC2)cc1=O.C N1(C(C(C)c2cc[nH]n2)=O)CCC(C(O)CNC(C2CCCC2F)=O)CC1 c1(NCC=C(CSC)C)ccc(C(F)(F)F)c(Cl)c1Cl C(=O)(C1=C2CCCN=C2NN1)NC(CC(C)NC(=O)CCCCCF)C c1(CC)ccc2cc(C(=O)NCC(C)NC(C3CS(=O)(=O)C3)=O)[nH]c2c1 N1(C(CCCN(C(C(C)c2cc[nH]n2)=O)C)=O)CC2CCC(C1)O2 C1(C(=O)NCCC(=O)OCC#C)CCC(=O)C(CC)C1 c1(N2CCC(N(CC#C)C(c3ccn(C4CC4)n3)=O)CC2)ncc(Cl)c(CC)n1 C(=O)(CS(=O)CCC(F)(F)F)N(CC(C(=O)OCC)C)C c1(C(=O)NC2CC(N(C(=O)C(C)(O)C3CCOC3)C)C2)cc2c(n1C)CCOC2 CCCCC(CNC(c1ccc(C(C)O)cc1)=O)NC(C1CCCC1)=O N1(C(C2(C)CCN(C)C2=O)=O)CCc2sc(CNC(=O)C3=COCCC3)nc2C1 c1(NC(=O)NC)cccc(C(=O)NC(C)CCC)c1.c1(C(=O)N)cncnc1 CC(C)(C(=O)N)S(=O)(=O)C1CC1.C1CC2CC(C1)N(C(C1(O)CCSC1)=O)C2 C1(CC)CN(C(C2C3CC4C(C3=O)C24)=O)CCN1C(c1n[nH]c(C)c1F)=O C1(C(N(CC(C2CCCCC2)O)C)=O)CN(C(=O)Cn2ncnn2)CCC1(C)C N1(c2nc(C)nc(C#N)c2)CCC2(CCOC2)C(CNC(C2CC3(CC3)C2)=O)C1 C(=O)(C(F)(F)CC1CCCO1)N(CC(C)NC(=O)CC1(C2CC2)CC1)C Cc1cc(C(=O)NC(C)C(C)C(=O)NCC2CC(F)(F)C2)c(C)nn1 C12(CNC(c3ccsc3)=O)COCCN1CCN(C(C1COCCO1)=O)C2 C12(CCCCC1)C(=O)OCC(=O)N2.C1(COCC=C)CC1(Cl)Cl Cn1nc(C(N2CC(NC(=O)C(O)C3CCC3)C(O)C2)=O)cc1O CN=c1[nH]cc(C(=O)NCc2cccc(C(=O)NC(C)C(F)F)n2)s1 CC1CCOCC1C(=O)NC(CC1CCOCC1)C(=O)NCC1(C)COCCO1 C1(CNC(c2[nH]n(C)c(=O)n2)=O)COCCN(C(=O)CCc2csc(=N)[nH]2)C1 n1(C(C)C)ncc2cc(C(=O)NCC3CCN(C(=O)Cc4ccon4)C3)cnc12 c1(C(=O)NC2C(NC(C(CC)(C)O)=O)CCOC2)cncc2nnn(C)c12 C(CC(=O)N(CC)CC1CCCO1)(C(F)(F)F)NC(CNC(CC)=O)=O CC1CC2(CN1C(c1ncc(Br)s1)C(=O)NC1CCCC1)CC(F)(F)C2 N(C(=NCCC(=O)Nc1ccc(F)cc1Cl)NC(C)C1CC1)CC1CC(=C)C1 c1(C(=O)NCC2CCCC(NC(C3C(=C)C3)=O)C2)c(F)ccc(C)c1F CCC(C)(C)C(=O)N(CC(CO)(CO)NC(C1CCOCC1)=O)C c1(C(=O)NC(CNC(CC(CC)OC)=O)C(C)C)ncc2ccccc2c1O c1(C(=O)NCCC(C)NC(=O)CC2CC3CC3C2)cc(C(F)(F)F)ncc1Cl Cc1ccc(-c2cn(CCc3nnc(CO)s3)nn2)cc1Cl Cc1ccc(F)c(Oc2ccccc2-c2ccccc2)c1 O=C(C1=CC(O)CC1)NCc1ccn(C2CC2)n1.C(=O)(C1=NNC(=O)C1)N Cc1[nH]c(C#N)cc1C(=O)NC(CNC(=O)C(C)C1CCCC1)CC(F)(F)F c1ccccc1.C12(C(NC3CC3)=O)CC1CN(S(=O)(=O)CC1CC1)C2.C C(=O)(C(C)CC(C)(C)C)N1C(CN(C(CCOC(CC(C)C)C)=O)C)CCCC1 c1(CC(C(=O)NC(C)CNC(C2CC(Cl)(Cl)C2)=O)OC)ccc(F)cc1 CN1CCC(C2CCN(C(c3cccc(C4(C)COC(=O)N4)c3)=O)CC2)C1 C12(NC(c3cc(C)ncc3)=O)CCC(CNC(c3csc(O)n3)=O)(C1)OC2 Cc1sc(Br)cc1C(=O)NC1CCC(n2cc(-c3ccsc3)nn2)CC1 Cc1nc(CC(F)(F)F)sc1C(=O)NC.C1(C)CCCN1C(=O)C.C1CC1 CCC(C)(C)C(C(=O)N1CCC(CN(C)C(c2cc(=O)cc[nH]2)=O)C1)OC c1(C(c2n(CCCC)nnn2)NCC2(CO)CC=CC2)cc(C)c(F)c(C)c1 n1(CC)ncc(C(=O)NCC2CC(C)N(C(=O)C(CC3CCC3)O)C2)c1C CCCCC(O)C(=O)N1CC(NC(C2(C(=O)NC)CC2)=O)CC(F)C1 C1(CNC(C(CC)O)=O)CC2(CCOCC2)CN1C(=O)Cc1c[nH]nc1O N1(c2nnn(C)n2)CCCC2C(NC(c3cc4c(F)cccc4[nH]3)=O)C(C)(C)C12 c1(CC)cccc2ccc(C(=O)NCCN(C(c3ccsc3C)=O)CC)nc12 Cc1nc(C(C)NC(c2ccon2)=O)sc1C(=O)O c1(C(N2CC(C(O)C(=O)NC)C2)=O)cc(CO)ccn1.n1(C2CC2)cccn1 c1(C(N(CC(O)CO)C(=O)OCC)C)ccccc1.C1C(CO)N1 C1(C(=O)NC2CN(C(C(CCC)OCC)=O)C(C)CC2)Cc2ccccc2N1C C1(C(=O)NCC2(OC)CCCCC2)CCCCCN1C(c1cccnc1C)=O C1(CCNC2(CCC)CC2)CCCCCC1 Cc1ccc(C)s1.c12ccc(s1)CNC2.C1(C(=O)NC(C)(C)C)CC1 C=CCC(F)(F)C(=O)NC12COC(C1)C(NC(=O)CSCCOC)C2 c1(N2CC3CC3C2)ncc(Br)c(C(F)(F)F)n1.c1(CC)ccnc(C(=O)N)c1.C C#Cc1nc(C(=O)NCC2CC(NC(c3cnccc3C(F)F)=O)C2)cs1 O=S(=O)(c1ccc2nc(O)oc2c1)N1CC2CN(Cc3ccnc(Cl)c3Br)C2C1 c1(C=O)cnc(C2CC2)nc1O.CC1OC(C)CC1C(=O)NCCC1CC1.C c1(C(N(C(C(=O)NCCS)c2cnn[nH]2)CC)C)ccccc1C(F)(F)F C1(NC(Cc2nc(C)sc2)=O)CCSC12CN(C(=O)CC1OCCC1(C)C)C2 N1(C(C(CN(CC)CC)F)=O)CC2CC(N(C(=O)CCN3CCOCC3)C)C1C2 C(=O)(C(O)CC(N)=O)NC1C(N2CCN(C(CC(C)(C)C)=O)CC2)CCC1 c1(NC(CN(C(CCSCCC)=O)CCC)=O)ccc(O)nc1 c1(C(c2n(CC(=C)C)nnn2)NC(CC(N)=O)c2ccccc2)cc(C)c(Br)s1 C1(C(=O)NC2CC(NC(C3CC34CC4)=O)C2)Cc2nnsc2S1 CCC(CC(C)C)C(=O)N1CCC(F)C(NC(c2cccc(C(=O)NC)c2)=O)C1 C(=O)(C1=NN(C)C(=O)CC1)NC(C1CCCN1C(=O)C(c1ccccc1)C)C c1(C(=O)NC2(CCCNC(Cn3c(C)cc(C)n3)=O)CC2)cc2ncccc2s1 N1(C(c2cc(OCC)no2)=O)CC(NC(=O)CCn2cc(Cl)cn2)C(O)C1 c1(OCc2onc(-c3c(I)csc3)n2)ccccc1I C=CCCC(C)(C)C(=O)NCC1(NC(C2CCCOCC2)=O)CCOC1 C12(CC(=O)NCCSCC(=O)NCCN(C(C)C)C)CCCC1C2 N1(C(c2n[nH]c(C)c2Cl)=O)CCC2CN(c3ncnc4c(C)csc34)CC2CC1 CC1CN(C)C(C)CC1NC(C1(NC(c2coc(C3CC3)n2)=O)CC1)=O N1(C(=O)NCC(c2cccc(C)c2)N2CCOCC2)CCC(O)C12CCSC2 c1(C(N2CC(NC(C3(OC)CCC(C)(C)C3)=O)C(O)C2)=O)ccc(F)c(F)c1N C1(C(N(C2CCN(C(Cn3ccc(C)cc3=O)=O)C2)C)=O)CC2(C1)CC(C)(C)C2 Cc1ccc(C(=O)N(C)CC2CCN(C(c3ocnc3C3CCC3)=O)C2)o1 C1(NC(c2scc(OC)c2O)=O)COCCN(C(=O)CC2CC3(COC3)C2)C1 C(=O)(C=C1SCC(=O)N1C)N1C(C)CC(CNC(CCCOCCOC)=O)C1 Cc1cc(=NC(=O)C(=O)NC23CC2CN(C(c2c(Cl)ccc(C)c2N)=O)C3)[nH]o1 C(=O)(CS(=O)c1ccc(Cl)cc1)NC(C)CN(C)C(c1cscc1F)=O N(C1CCNC(=O)c2[nH]ccc21)C(C(N1C(C#C)C2CCC1C2)=O)=O C1(NC(C2CCC(C)(C)OC2)=O)CN(C(=O)C(C)(C)O)CC(F)(F)C1 Cc1ccc2occ(C(=O)N(C3CC(NC(=O)C=C4CCC(C)CC4)C3)C)c2c1 C(=O)(C=C=C(C)C)NC(COC)C(=O)NC1CCC(F)CC1 n1(CC)cccc1C(=O)NC(C1CCCN1C(=O)CO)(C)C.c1ncnn1C CC(CCCNC(C1(c2cccnc2)CC1)=O)NC(C1CCOC1C)=O C(=O)(C(C)CCN(C)C)N.C(C(F)(F)CN(C(=O)CCC1CCC1)C)OC C#Cc1ccc(C(=O)N(C(CNC(=O)CC2CC(C)OC2C)C2CC2)C)cc1 C1(C(N2CC(O)(CNC(C(CSC)(C)C)=O)C2)=O)CCc2nnc(O)cc2C1 c1(C(=O)NC(C(C)NC(COC(C)C)=O)C)nc2c(cc1Br)OCCO2 C1(C(C)NC(Cc2nc(CC)sc2)=O)CN(C(C2CC(C)(O)C2)=O)CCO1 C(c1ccc2occc2c1)=CC(N1C(CNC(=O)CCCC2CCCC2)CC1)=O C=C1COCCN(C(=O)CN(C(c2nn(CC)nc2C)=O)CC2CC2)C1 N1(C(c2c(NC)nc(C)cc2)=O)CC(n2cc(CNC=O)nn2)CCC1(C)C N1(C(C2(OC)CCOC2)=O)CCC2(CC1)CCN(C(C1CCCSC1)=O)C2 c1(C(=O)NCC(CNC(CC2C(C)C(=O)CC2)=O)(C)O)cn2ccnc2cn1 C1(CCS(=O)(=O)NC2CCOC2CC2CC2)CCCCC1(F)F C1(C(=O)NCC(CNC(=O)CNC=O)OC)CCN(C)S1(=O)=O C1(C(N2CC3C(C(=O)NC(CC)CC)C3C2)=O)CCC(=O)N(C)C1 c1(C(=O)NCCCCNC(C2(C)CCCCC2)=O)cccn(O)c1=O N1(C(C(CC(C)C)F)=O)CCC2CCN(C(c3cc4n(n3)CCO4)=O)C2C1 N1(C(C(N2CCCOC(CCS)C2)=O)=O)CCc2c(C(F)(F)F)cccc21 C1(CNC(=O)CC(O)c2ccccc2)C2CN(C(c3ccc(Br)cn3)=O)CC12 C(CC1=CCCCC1)N(C(c1c(C)oc(CNC(=O)C(N)=O)n1)=O)C C1(C(=O)NC2C(NC(=O)C(F)=CCCF)CCC2)Cc2cc(F)ccc2O1 N1(CC(N2C(CNC(c3[nH]cc(CC)c3)=O)CCC2)=O)C(=O)CNC1=O CCC(C)C(C(=O)NC(C1CN(CC2CCC(=O)N2)C1)C)c1ccccc1 C1(NC(C(CC)N(C)C)=O)CC(C(=O)NCC2CC(O)C23CCC3)=CC1O CCC(C)(C(=O)N1CC(N(C)C(c2ccnc(OC)c2)=O)C(O)C1)OC c1(NC(C2N(C(c3cn(CC)nn3)=O)CCCC2)=O)c(O)cccc1Cl C1(CC)CC(C(=O)NC(CCNC(=O)CC2CCC3CC23)C(C)C)CCO1 CC1C2C(CCN2C(=O)Cc2ccnn2C)CN1C(c1cc(=N)[nH]c(Cl)n1)=O C(C(N=c1ccc(=N)[nH][nH]1)c1ccccc1Cl)NC=O.C1CCCCC1 CCCCC(C)N(C(c1ccsc1Cl)C(=O)NCCCF)C c1(C(N2CCC(N(C)C(c3cnc(N4CCOCC4)s3)=O)C2)=O)cccc[n+]1[O-] N1(C(c2cccc(OC)c2)=O)CC(NC(=O)CCN2CCCS2(=O)=O)CCC1C CC(C)(C)C(CNC(C1CC(C2CC2)C1)=O)NC(=O)C(Cl)=CCl N1(C(C(NOC)=O)=O)CCN(C(c2cc(O)cc(Cl)c2)=O)CC(C)C1 c1(CCC(=O)N(CC(CC)NC(C2CC2(Cl)Cl)=O)C)ncccn1 C1(CC)(NC(=O)C(CC2CCC2)NC(=O)CC(C)C(F)F)CCCCCC1 C1(C(N2CCC(OC)C2C)=O)C(C2CC2)CCN1C(c1coc(SC)c1)=O c1(CC)n[nH]c(CC)c1CC(=O)NC(C)CN(C)C(c1ccc(C)o1)=O.C C1(NC(c2cnc(CCC)s2)=O)CCCCC1C.c1(CC(=O)N)ncc(Cl)s1 Cc1c(C(N2CCCN(C(c3csnc3Cl)=O)CC2)=O)oc2c1C(=O)CCC2 c1(CN2CCCN(C(C3=C(C)OCC3)=O)C(C)C2)cc([N+](=O)[O-])c(F)cc1Cl c1(C(N2CCCC(C(C)NC(c3c(C)cnnc3)=O)C2)=O)c(N)cc(F)cc1F c12cccc(c1)NC(=O)C(=O)N2.c1(NC)cc(C(=O)OC)sn1 CC1(C)CC(NC(=O)CCc2ccoc2)CCN(C(=O)Cc2cnoc2)C1 c1(C(N(CCCN(C(Cn2c(C)cnc2)=O)C)C)=O)cccc(C2CC2(F)F)c1 c1(N2C3CN(C(Cc4c(C)cc(Br)cc4)=O)C(CC3)C2)ncnc2ccccc12 C12(NC(=O)NOC3C(=O)OCC3CO)CC3CC(CC(C3)C1)C2 n1(C(C(N2CC(C#C)(O)C2)=O)C)cc2ccccc2n1 Cc1ccc(C(=O)C(=O)NCC2CC2NC(=O)Cc2cccc(C)c2)cc1 C1(C(=O)NCC(N(C(c2c(C)noc2C)=O)C)C2CC2)CCc2nncn2CC1 N12CCC(C1(C)C)CNC2=O.Cc1cc(C2CCCN2Cc2ccccc2)on1 c1(C=O)cccc(F)c1Cl.c1(CN(CCC)C)ccc(C(=O)NC2CC2)o1.C S(=O)(=O)(c1ccc(-c2ccc(NC(C3CC3C3CC3)=O)s2)cc1F)NCC N1(C(C2C(C(C)(C)C)C2)=O)CCCCC1C(=O)NCCn1ccnn1 c1(C(=O)NCCC(C)NC(Cc2cn(CC)nn2)=O)csc2c(OC)cccc12 C=CC1(C(=O)NC2CCC2CNC(=O)COc2ccccc2)CCOCC1 CC1(C)CCC(F)(F)CC1NC(=O)NCC1CCN(c2ccc(F)c(F)c2)C1 C(=O)(C(CN(C)C)C(C)C)N(C(C)C(=O)N(C)CCn1cncn1)CCC NS(=O)(=O)c1ccc(C(N2CCOCC2C(=O)NCC2(O)CCCCC2)=O)cc1 CC1CC2(CCN(C(=O)NC3CC3C(C)O)CC2)C(=O)N1 Cc1c(Br)c(C(=O)N(C2CCCN(C(c3cc(=O)n(C)o3)=O)C2)C)nn1C c1(OC)cc(C(=O)N(CC(C)(C)NC(=O)C(C2CCC2)OC)C)ccc1F CC(C)CCCC(C)NC(=O)CSCC(N1CCC1c1ccc(Cl)cc1)=O CS(=O)(=O)C1CCN(C(c2cccc(I)c2)C(=O)NCSc2ccccc2)C1 c1(CCC(=O)NC(CNC(C(C)NC(c2cccs2)=O)=O)CO)ccn(C)n1 S(=O)(=O)(c1ccc(C#N)c(N(CCCOC)C)c1)NCC(CC=C)(C)CO c1(CCCC)ccc(C(=O)NCCCC(C)NC(=O)CS(C)(=O)=O)cc1[N+](=O)[O-] C1(CNC(=O)C=CCn2cncn2)CCCCC1.C(=O)(CCc1cnco1)N c1(C(=O)Nc2scc(-c3ccc(OC)cc3F)n2)nc2ccccc2[nH]1 C1(CCCNC(C2C(C(=O)OC)C2)=O)CN(C(=O)CC)CCO1.C1CCCC1 c1(C(=O)NC2CCN(C(=O)COC(F)F)CC2)ccc(Cl)cc1I c1(CC(=O)N)ccc2c[nH]nc2c1.N1(C(c2cc(C(N)=O)oc2)=O)CCCCC1C CCC(C#N)C(=O)NCC=CCC(N1CCC(C)(CC)C1)=O CCC(C)C(C)C(=O)NCC1CN(C(C2(CC(F)F)CCC2)=O)CC1C C#Cc1ccc(C(N2CCC(F)(C(N3CC(N(CC(C)C)C)C3)=O)CC2)=O)nc1 CN1CC2(CN(C(=O)NCc3csnn3)C2)OC1=O C(=O)(CCCC(F)(F)F)N1C(C(C)C)CCC1C(=O)NCC(N1CCCCC1)C CCC(C)C(C(=O)NCC1CC2CCCC2C1)N(C(=O)Cc1coc(C)n1)C N1(C(c2c(C)ccnc2)=O)CCN(C(C2CNC(=O)N2)=O)C(CF)C1 c1(C(N(CCN(C(c2c(Cl)ncs2)=O)C(C)C)C)=O)cncn(C)c1=O.C c1(C(C)=O)cc(C(=O)NC2(C)CCC2)oc1C.c1(C=O)cccnc1N(C)C CN=c1[nH]nc(CC(N2CC(CNC(c3ccon3)=O)C3CC23)=O)s1 C1(C(NOCC(C)C)=O)CCc2nc[nH]c2C1 C#CC(CNC(=O)CC1(C)CCN1C(=O)C(F)C1CCCC1)CC1CC1 N1(C(CC2CC(OC)C2)=O)CCC(C)C1(C)C.C1(CC(=O)N)CN2CCN1CC2 C1(NC(CCCCSC)=O)C2CC1CN(C(C1(C)CCOCC1)=O)C2 C=C(C)CCCC(=O)NC1CCCC1NC(=O)COCc1nnc(C)s1 CCCCCCC(CC)C(=O)N1CC2CC(NC(c3cc(F)cs3)=O)CC1C2 N1(C(c2ccc(-c3cc(N4CCCC4)nc(F)c3)cn2)=O)CCC12CCCCC2 N1(C(c2n(CC#C)cnn2)=O)CC(NC(C2CCC2C=C)=O)C(CCC)C1 N1(C(CC=C(C)C)=O)CCN(C(=O)CCCc2ccc(O)cc2)C(CC(F)F)C1 C1(C(=O)NCC(C)S(C)(=O)=O)COCCN(C(=O)CCc2nccs2)C1 N1(C(C2(CC=C)CCN(C(C3CC(=O)C3(C)C)=O)C2)=O)CCC2(CCC2)C1 CC(C)CC(F)(F)C(=O)NCCCC(C)(C)NC(c1ccc(C(C)C)cc1O)=O c1(CCC(C)O)cn(CC(F)CCNC(=O)CCOc2ccccc2)nn1 C1(C)(CC=O)CCCCC1.C1CCCC1.C1(C(=O)OCC)CC1CC(=O)N C1(NC(CCc2c(OC)cccc2)=O)CCCN(C(=O)CCC#N)CC1F Cc1cccc2ncc(C(N3CCN(C(=O)CCC4(C)CC4)C4CC34)=O)n12 C1(CC=O)OCCCC1(C)C.CC(CN(C)C)CC(=O)NCC1(C)CC1.N Cc1cn2cc(C(=O)NC3CCC(NC(=O)C(F)(F)C(C)O)C3)ccc2n1 C1CC2CCCC(C1)N2C(C1CCC(F)CC1)=O.c1(COC)ccoc1C(=O)N O=C1CC2(CN1)CN(C(=O)CCC1CCN(C(C34C=CC(CC3)C4)=O)CC1)C2 N#CC1CCN(C(C2CC2CNC(c2cc(C3CC3)[nH]n2)=O)=O)CC1 CCC(C)(CC)C(=O)N1CCN(C(c2cc(C(C)(F)F)on2)=O)C(CO)C1 C1(C(C)C)CC(CC(=O)NCCCOCCNC(c2cscn2)=O)CCO1 CCC1=NOC(C(N2CCC(N(C(c3cnn(CC4CC4)c3)=O)CC)C2)=O)C1 S(=O)(=O)(c1cccc(=NCCS(=O)c2ccccc2)[nH]1)NC1C(SCC)CCC1 C12(C(=O)NCCCN(C(C3CC(C)SCC3)=O)C3CC3)CCC(F)(CC1)C2 n1(CC)cc(Br)cc1C(N1CC(NC(=O)C(C)(O)COC)C(C)C1)=O N1(C(C2(CC)CC2)=O)CCCCC1CNC(C1CCN(C)CC1)=O.C1CC1 C1(C(=O)NCC)CN(C(=O)CN(C(C2CC2F)=O)C2CC2)C1 N1(C(c2nc(COC)oc2)=O)CCN(C(=O)CCn2cnc(=N)[nH]2)CC1 CCC(C)C(C(=O)N1CCC(C(=O)N(C2CCN(C)C2)C)CC1C)N(C)C CCCCC(C(=O)N1CC(OC(=O)NCC)C1)NC(=O)CCNC(N)=O N1(C(C2(CC=C)CC2)=O)CCCC(CCNC(c2ncc(Cl)s2)=O)C1 c1(C(C)C)conc1C(=O)N(CCCCNC(=O)COCC1CCCOC1)C c1(C=O)c[nH]nn1.c1(CN(C(=O)C(C)N(C)C)CCOC)noc(C)n1 C12(C(=O)OC)CCC(CC1NCCNC(N)=O)C2(C)C N1(C2CC3CN(C(C(C)Cc4ccccn4)=O)C2C3)CCn2nncc2C1 N1(C(c2cccc(NCC#C)c2)=O)CCCC12CCN(C(C1CCCC1)=O)C2 c1(C(N2C3CN(C(C=CC(=O)N(C)C)=O)C(C3)C2)=O)c2ccccc2nn1C N1(C(C(C)S(N)(=O)=O)=O)CCc2nc[nH]c2C12CCN(C(=O)CCCCC#N)C2 C1(C)(NC(c2nc(CCC)oc2)=O)CCCN(C(C2(N3CCCC3)CCC2)=O)C1 c1(C(NC)=O)cc(N)c(F)cn1.c1(CNC(c2nc(C)oc2)=O)ccccc1.C CCCCCCC(CC)C(=O)NC1CCCN(C(c2nc(C3CC3)no2)C)C1C N1(C(c2c(OC)cc(C)cc2)=O)CC2(C1)CN(C(=O)C(C)(C)CCC#N)CCO2 C1(C)(C(=O)NCCCC(C)C)CC2CCC1C2.N1(CCC=O)C(=O)CCC1=O.N c1(C(=O)N)cc2ccc(F)cc2s1.C(c1cccnc1)=C(C(=O)NCC1CC1)F C=CC(C)(O)C(=O)N1CC(C)(C(=O)NCC23CC(CN2C)C3)C1 Cc1nc(C(F)(F)F)c(C(N2CCCC2)=O)n1O.C1(C(=O)N)(C(N)=O)CCC1 c1(C(=O)NCCCNC(C(C(CC)O)C)=O)ccc2c(c1)N(C)CC2 C1(C(=O)NC2CC(F)(C)C2)CCC(F)(F)CC1.C(=O)C(F)(F)C1CC1.N c1(C(N(C2CCCN(C(c3cnn(CC)n3)=O)C2)C)=O)c[nH]c2nccc-2c1 n1(CCC(N2CC(NC(C(c3ccc(C)s3)C)=O)C2)=O)c(C)c(C)sc1=O N1(C(c2c(C(=O)OC)scc2)=O)CCN(C(c2nn(C)c(N)c2C)=O)C(C)C1 c1(C(=O)NCCCC=C)cc(C)c(O)c([N+](=O)[O-])c1.C1(C=O)CC2(CCC2)C1 N1(C(CCC(C)SC)=O)CCC2(CC1)OCCCC2NC(C1CCCC(O)C1)=O N1(C(c2c(CNC(COC)=O)noc2)=O)CC2(COC(C)C2)C1 C1(CC)C(NC(=O)Cc2ccc(O)nc2)CCCN1C(=O)C(C)CC(F)F C1(CNC(C(C)CO)=O)COC(C)(C)CN1C(c1cc(C#N)ccc1Cl)=O c1(C(=O)NC2C(F)CCN(C(COCC#C)=O)C2)cn2c(Br)cccc2n1 c1(NC(N2CCC(O)C2)=O)ccc(Cc2nn[nH]n2)c(F)c1.C1CCCC=C1Br.C C1(NC(C(CCC)OC)=O)C2CCCC1CC(NC(c1ccc(C)c(N)c1)=O)C2 Cc1nc(CC(N2CCC(F)(CNC(C3CC34CC4)=O)C2)=O)oc1C c1(C(C)C)c(C(=O)OCC(=O)NC2(C)CCCCC2)cnn1C c1(C(=O)NCC2N(C(c3ccn(C)c3)=O)CC3(CC3)C2)cc2ccc(Cl)cc2[nH]1 c1(C(N(CCCNC(c2c(C)c(F)c(F)cc2)=O)C)=O)cnc2cnccc2c1 CC(N=c1[nH]c(NCC(N2CCCC2)=O)nc2cc[nH]c12)c1ccc(F)c(F)c1 c1(C(=O)NC2CN(C(CC3C(OC)CC3)=O)CC2C)cc(C)n(C2CC2)c1C N1(C(C2C(NC(C3ON=C(CC)C3)=O)C2(C)C)=O)CCC(O)CC(C)C1 Cc1nn(C)c(Cl)c1S(=O)(=O)NC1(COC(C)(C)C)CC1 C(=O)(CCC(=O)NC(C)CC(C)NC(c1noc(C)c1CC)=O)NCCC C(CCCCC(=O)NCCOC1CCCC1)NC(C(CC)n1cncn1)=O C(=O)(CCCC(=O)NCC1CC1NC(c1cccc(SC)c1)=O)NCC N1(C(C2CCC(=C)CC2)=O)CCC2(CC(NC(C3(Cl)CC3(C)C)=O)C2)C1 c1(NC(c2nc(C)[nH]n2)=O)cnc(Cl)cc1C(=O)N.c1(C2CC2)ccc(F)cc1 CC(F)(F)C(C)(C)CC(=O)NC1(C2CCCN2C(c2cc[nH]c2)=O)CC1 C=CC(CC)CC(=O)N(C)CCOCCCNC(=O)Cc1nc(=N)[nH][nH]1 c1(NC(c2c(CNC(C(C(C)C)n3cncn3)=O)ocn2)=O)ccc(F)cc1O N1(C(C(C)Cn2cccn2)=O)CC(O)C(O)C1CNC(=O)CCc1cnoc1 CCCCCCC(C)C(=O)NC1CC2CC(NC(=O)C(=O)NC(C)C)C2C1 Cc1ccc(S(=O)(=O)N(CC(C(=O)OC(C)(C)C)C2CC2)C)cc1C c1(C(N(CC(C)NC(CC=C(C)C)=O)C)=O)c(C)c2cnccn2c1C C(=O)(C(F)(F)C(C)(C)O)NCC(C)NC(c1ccnn1C)=O C1(CC)C(C(=O)NCCCC(F)(F)F)CCN1C(=O)C(C(C)C)C1CCC1 N1(C(COC)=O)CCCC(NC(=O)CCCc2ccc(F)cc2)C1 C1(NC(Cc2cc(C)[nH]n2)=O)CC(C2CCN(C(=O)C(C)(C)CC(F)F)C2)C1 C=C(C)C1CN(C(C2(F)CN(C(C3CC=CCC3C)=O)C2)=O)CCO1 c1(C(=O)NCC(CC)CC)cc(C)c2nc(C)cn2c1.C1(C=O)C(C)C1(F)F.N c1(CN(C)C(=O)NCCCO)csc(-c2ccccc2)n1 Cc1cc(CC(=O)NC(C)CCNC(c2ccnn2CC(F)(F)F)=O)no1 N1(C(c2c(C(=O)OC)cccc2)=O)CCC(O)(NC(c2cc(O)no2)=O)CC1 N1(C(CSCC=C)=O)CC2C=CC1C(C(=O)NCCN1CC3CC3C1)C2 C12(NC(Cc3ccc(C)o3)=O)CCN(C(c3cnc(C)nc3C(C)C)=O)CC1C2 C#Cc1ccnc(C(=O)NCCN(C(=O)C(CO)N(C)C)C)c1 N#CC1=C(C(=O)NC(C(N2CC3(CCOC3=O)C2)=O)C2CC2)CCC1 CC1=C(C(=O)NC2CC23CCN(C(c2c[nH]c4nccc-4c2)=O)CC3)COCC1 c1(CC(N2CC(CC(=O)NC(c3n(CC)ncc3)C)C2)=O)ccc(O)cn1 N1(C(C)=O)CCCC(C(N2CC(NC(=O)CCN3CCNC(=O)C3)C(O)C2)=O)C1 C(C)(CN=c1[nH]c2cccc(C)c2s1)NC(c1ccc2cc(C)cn2c1)=O Cc1ncccc1CC(=O)NCC=CCNC(c1cnn(C(F)(F)F)c1)=O Cc1nc(O)[nH]c1C(=O)N(CCCCNC(c1c[nH]nc1C1CCC1)=O)C O=C1Cc2c(C(=O)NCC3CC(F)CN3C(=O)CC3CCCCC3)cccc2N1 CCCC(CNC(=O)C(C(C)C)OCC)C(=O)NCC1(O)CCN(C)C1 c1(C(=O)OC)c[nH]ccc1=NCC1(NC(=O)CCc2cc(Cl)cs2)CCCC1 c1(C(N2CCC2)=O)cnc2c(cnn2C)c1.C1(OC)CC(CC(=O)NC)C1(C)C N1(C(c2nn(CCCC)c(=O)cc2)=O)CCC(C2CC2)C1.C(=O)(CC1(C)CC1)N c1(CC(=O)NCCC)ccc([SH](=O)=O)cc1.c1(C(=O)N)ccccc1.CC#N C(C(C)N=c1[nH]c(Cl)ncc1Br)N(C(c1c(Cl)cnc(CC)n1)=O)C Cn1nc(C(=O)NCCCn2cc(-c3ccnc(C(F)(F)F)c3)nn2)c(Cl)c1Cl C1(CC(=O)N(CC(C)O)CCNC(C(C)C)=O)CSc2ccccc2NC1=O C1(CC(=O)NCc2c(C)nns2)CN(C(c2cn(C)c(=O)cn2)=O)CCC1C C1(C(=O)NC2C(CNC(c3nc(C)sc3)=O)CCC2)CC2CCC1C21CC1 C1(C)CCCCC1C(=O)N(C1CCN(C)C1)CCO.C(C)(C(=O)N)SC(C)C C1(C(N(CC(=O)NCCC2CC2C)CC#C)=O)CNC(=O)C1 C(CCCCC(=O)NCC(n1ccnn1)C)NC(CCc1c(C)noc1)=O C1(C)(C(=O)Nc2ccc(CC)cc2)CN(C(=O)CCc2ccoc2)CC1C c1(NC(C)=O)cccnc1C(=O)NC1CC1.C1(C(NC)=O)CC(C)CO1.C c1(C(=O)NC2CN(C(CCC(=C)C)=O)CC(O)CC2)cc(F)cc(S(N)(=O)=O)c1 C1(NC(=O)CN2CCOCC2=O)CC(CNC(=O)CCc2cnoc2)C12CCC2 c1(C(=O)NC(C2N(C(CCC#C)=O)CCC2)C)cc2c(=O)[nH]c(C)cn2n1 c1(C(=O)NCC(C(=O)NC(C)Cc2nc[nH]n2)C)c[nH]c(C#N)c1 C1(c2cn(CC)nc2)OCCCC1C(=O)NCCC.c1(CC=O)cc(C)[nH]n1.N C(CCCCC(=O)NC1CC(CNC(c2scnc2Cl)=O)C1(C)C)NC(C)=O c1(CC)ncccc1C(=O)NCC(C1CCOC1)NC(=O)CC(F)F Cc1cc(Cl)cc(C)c1C(=O)NC1COC2(C1)CN(C(c1cc(Cl)sc1Cl)=O)C2 Cc1cc(CNC(C2CC2C(C)NC(=O)CN2CCCC2=O)=O)ncn1 C(=O)(C(Cc1cn(CCNC(=O)C(C)CF)nn1)C1CC1)OC C=C(C)C1OCCC1CNC(=O)CCNC(=O)CCn1cnc(=N)[nH]1 C1(O)(C(N2C3(c4cn(CCOCC)nn4)CCC2CC3)=O)CN2CCC1CC2 C1(C(N2CCC(C)(NC(c3cc(OC)ns3)=O)C2)=O)CC(C2CC2)=NO1 c1(C(N2CCC=C(F)C2)C(=O)NCC(C)C)cc(F)c2c(c1)CCC2 CCC(CC(=O)NC1COCCN(C(c2cc(Cl)c(N)cc2F)=O)C1)C(F)F C(=O)(CC(C)(C)C(=O)O)NCCC(C(=O)Nc1c(CC)nn(C)c1)(C)C N1(C(c2cc(OC)n[nH]2)=O)CCC=CC1C(N1CCCC(NC(C)=O)C1)=O c1(NC(N2C3CC(=C)C(C3)C2)=O)cnn2c(-c3cccs3)ccnc12 C1(NC(C(C)OCCC=C)=O)CCCCC1.c1(C=O)c(C)noc1C1CC1.N c1(C(N2C(CNC(=O)COC3CC3)CCC2)=O)ccc(-n2ccnc2O)cc1 C1(CC(=O)NCCCCCNC(C2(O)C(C)(C)C2)=O)CCCCC1(F)F C(C(CCC)C(=O)NCC(C)(C)C(N)=O)NC(CSCC=C)=O Cc1cc(F)c(C(=O)NCCC(C)(C)C)cc1Br.C1(C(=O)N)C2CC3C(C2)C13 c1(C(N2CCN(C(Cn3c(C)ncc3)=O)CC2)=O)ccc(Br)c2c1OCCC2 N#CCCCC(=O)NC1(C(=O)NC2CCCCC2O)CCOCC1 N1(C(c2cc(C)on2)=O)CC2CC1CC2CNC(C12CC(F)(C1)C2)=O CC(CN=c1nc2c(cnn2C)c(NCCC(C)N(C)C)[nH]1)c1nccs1 CCC(CCC(=O)NC(c1nnnn1C)C)NC(c1cncn(C)c1=O)=O c1(OCC(=O)NCC2CCCC(NC(C3CCC3)=O)C2)ccccc1Cl Cc1ccoc1CNC(=O)C(CO)NC(C1CC1CC(C)C)=O O=C1COc2cc(C(=O)NCCCCNC(=O)CCOCC3CC3)ccc2N1 Cc1cc2ccc(C(N3CC(NC(=O)CC4CSC4)CC(C)(C)C3)=O)cn2c1 N1(C(CC(C(=C)C)OCC)=O)CC2CCCN(C(=O)CCc3n[nH]c(=N)s3)C2C1 CC(CC(=O)NCC1(O)CN(C(c2ccoc2Cl)=O)C1)C(=O)c1ccccc1 C1(NC(C2N(CCC)CCC2)=O)CC2(CCN(C(=O)C(C)CC(C)(C)C)C2)C1 Cc1ncc(C(C)NC(C2(NC(=O)CC3C=CCC3)CCCC2)=O)s1 CC1(C)C2CCC(C)(C2)C1NC(c1sc(C2(C)OCCO2)cc1Br)=O C1(NC(CC(=O)NCC#C)=O)CC(NC(=O)C=NOC)CC1O c1(C(C)NC(=O)C(=O)NC2CCN(C)C2)cccc(Cn2cccn2)c1 C1CC2(CCN(C(C3(c4ccc(Cl)nc4)CC3)=O)CC2)C1.C1(C=O)CC1(F)F.N C(CC)(C(=O)N(CC(C)(C)C)CCO)OC.C1(C(C)(F)F)(C(=O)N)CC1 c1(C(N(C(CNC(CCOC)=O)C2CC2)C)=O)cncc(C(C)(C)C)c1 C1(CC=C)(C(=O)NC2(CF)CCN(C(=O)CC(C)COC)C2)CCCCC1 c1(OCC)ncc(C(=O)NC2CC(N(C(=O)CN(C3CCC3)C)C)C2)s1 C(C(C)C(C)C(=O)N)OC.c1(C(N2CC(C(C)(C)O)C2)=O)cnc(Cl)c(Cl)c1 C(N=c1[nH]cnc(Cl)c1F)C1CCCN(C(C2C(C)OC(C)C2C)=O)C1 C(=O)(C#CC1CCCOC1)N1CC2(CC(NC(c3cn4c(n3)CCCC4)=O)C2)C1 C1(NC(CC=CCC)=O)CC2CCC1N2C(=O)C=CCN1CCOCC1 N1(CC(=O)NCC(c2ccc(C(C)C)cc2)N)CCCCCCC1=O C#CCC(C)(C)C(=O)NCC(CC(F)(F)F)NC(c1ccc(C(C)=O)[nH]1)=O CC(c1ccccc1C)=CC(=O)N.C1(O)(CC(=O)N(CC(C)O)CC)CCCC1 C1(NC(COCCOCC#C)=O)CCCCC1.C1(C=O)(C=O)CCC1.N CCC(CC)C(C(=O)NC1CN(C(=O)Cc2nc[nH]n2)CC1C)OC CC(C(=O)OCC(=O)N(C)Cc1ccccc1Br)S(N)(=O)=O C(CC(C(=O)NCC1CCOC1(C)C)NC(=O)CC1CCCCCC1)=CC n1(CC(c2cc(C)cc(Br)c2)N2CC3CC2CN3C)nnc2ccccc12 N1(C(c2occ(C)c2)=O)CC(NC(c2cn(C(C)(C)C)nc2C)=O)CC(O)C1 N1(C(c2cc(CC)n(C)n2)=O)CCCC2(NC(c3cc(Cl)cc(Cl)c3)=O)CC2C1 c1(C=O)cc(Cl)cc(Cl)c1.C1(C(=O)OC)CC(F)(C(=O)NC(C)CC)C1 Cc1ccc2c(c1)C(N(C1CC1)CC1CCC3(COC3)OC1)CC2 C1(n2cc(NC(=O)OCC)nn2)CCN(C(=O)NCCS)CC1.C(C)C Cc1nc(N2C(C(=O)Nc3c(C=O)c(C)nn3C)CC3CC23)c2ccccc2n1 C1(C(C(=O)OCC)C)CCN(C(c2nnc(C)o2)C(=O)NCCCF)CC1 N1(C(C(CC)COC)=O)CCN(C)C(CNC(c2cc(=O)n(C)o2)=O)C1 C1(C(=O)Nc2n(C(C)C3CC3)ncc2)Cc2cccnc2C1 N1(C(C2CNC(=O)N2)=O)CCCC(NC(c2occc2-c2ccccc2)=O)C1 C(CC(C)C)(C(=O)N1CC(O)CC1C(=O)NC1CC2(CCC2)C1O)OC CCS(=O)(=O)CC(=O)NC(CO)C(C)NC(=O)CC1SC(=N)NC1=O CCCC(CNC(C1CN(C(=O)C(CC)NC(C)=O)CC1(F)F)=O)CCC C(=O)(CC(F)(F)C(F)F)N1CCC(CNC(C(Cc2c(C)n[nH]c2C)C)=O)CC1 C1(CNC(c2n(CC)cnn2)=O)(CO)CCN(C(C2C3CCCC23)=O)CC1 CN1CC(C(N2CC(O)(C)C2)=O)C(C(F)(F)F)C1.C1(C)(C=O)CCCOC1.N c1(OC)cc(C(N2CC3CC2(CNC(C2CCNC2=O)=O)C3)=O)c(O)cc1Cl Cc1cc(Br)cc(CN2CCC(C)(CNC(=O)Cc3cccnc3)CC2)c1O CC(CCP(C)(C)=O)(c1nnnn1C1CCCC1)NC1CC12CCCCC2 c1(C(N2CCC(F)(CNC(C3C(C)CC3)=O)CC2)=O)nccc2c1CNC2=O C#Cc1ccc(C(=O)NC(C(=O)NCC2CCCC2(C)C)C2CCC2)cc1C Cc1noc(CCC(=O)NC(C(=O)NCC2CCOCC2)C2CCCC2)n1 C1(NC(C(C2N(C(c3ccc(OC)o3)=O)CCC2)(C)C)=O)COC(C)(C)C1 Cc1ccc(F)c(CC(=O)N(C)CC2(O)CCN(C(C3CCC3)=O)C2)c1 Cc1cc(Cl)ncc1S(=O)(=O)NC1CCCN(C(=O)C(C)S)C1 c1(C(=O)NCC)ccc(-c2ccc(C)c(CO)c2)nc1C C1CCN(C(=O)Cc2cnn(C)c2C)CC1.c1(OCC)sccc1C(=O)NC.C N1(C(C(c2ccoc2)NC(c2c(COC)cco2)=O)=O)CCOCC(C)(C)C1 Cc1nc(Br)oc1C(N1CCC(C)C1CNC(C1CC(N(C)C)C1)=O)=O N1(C(C2(C(F)(F)F)CC=CCO2)=O)CCOCCC12CC2 c1(CC)nnc(=NCC(C)(C(C)C)NC(c2ccnc(OC)c2)=O)[nH]c1CC C(C1CN(C(C2CC2CC(C)(C)C)=O)CC1C(N1CCCC(F)CC1)=O)=CC C1(N(CC#C)C(C2CC3(C2)CC3F)=O)CCN(C(=O)CO)CC1.C1CCCC1 C#CCCCCCCC(=O)NC1CC=C(C(=O)N2CCSCC2CO)C1 c1(C(=O)NCC2(F)CC(CNC(C(CC)C(C)O)=O)C2)cccc2ncsc12 CC1=C(C(=O)N2CCC(C(F)CNC(C3CCCC3(F)F)=O)CC2)CCCO1 c1(CNC(=O)CC2CCCN(C(c3ccnc(F)c3)=O)C2)ccc2nc[nH]c2c1 C(C(=O)NOCC1CCCO1)(C1CC=CCC1)NC(CC1CC(OCC)C1)=O n1(CC)c(O)nc(N2C3CCC2CC(CNC(=O)C(C)(C)CSC)C3)cc1=O C(=O)(C1CCCc2ccnn21)NCCCC(c1ccccc1)NC(C(C)(C)F)=O C1(C)(NC(c2c(CC)non2)=O)CCCN(C(c2sccc2C(C)(C)C)=O)C1 C1(F)(C(=O)NC(C)CN(C)C(c2ccc(-c3ccccc3)s2)=O)CCCOC1 C(CCC(=O)NC1CC(OCC(=O)NC(c2ncnn2C)C)C1)OC(C)=O N1(C(c2n[nH]c(CC)c2I)=O)CC2CC(NC(C3CC4(CCC4)C3)=O)C2C1 C1(NC(C(C)OC(C)(C)C)=O)CCN(C(C2CC2F)=O)C1 C1(C)(CNC(CCC=C=C)=O)CN(C(=O)CSc2ccccn2)C(C)(C)C1 c1(OC)nc(Nc2cccc(F)c2C(=O)Nc2cccnc2F)ncc1Br C(C(C)(C)C(=O)N1CCC(F)(CNC(=O)C(CO)N(C)C)C1)SC N1(C(c2nc(C)oc2)=O)CC(NC(c2sc3nccn3c2C)=O)C2CCCC2C1 N1(C(Cc2n(C)ccn2)=O)CCOC(CCCNC(c2cc(C3CC3)cs2)=O)C1 CC1CN(C(=O)Cc2ccns2)CC(CCNC(=O)C(=O)C(C)(C)C)O1 N1(C(CCSCCC)=O)CCC(C2CC2)(CNC(=O)C(CCS)N(C)C)C1 c1(C(=O)NCC(=O)NC2C(NC(CCC=C)=O)CCC2)cc(C)ccc1F Cc1conc1CC(=O)NCC1CCC(C(=O)NCc2nc(CO)n[nH]2)O1 N1(C(C2N(C(CCn3c(C)ncc3)=O)CCC=C2)=O)CCN(C)C(=O)C1C c1(C(N(CCOCCOCCCC)CCC)=O)cnn(C)c1Br c1(OC)cc(C(=O)NC(C2CN(C(c3occc3F)=O)CCO2)C)c(O)c(Cl)c1 c1(CC(C)C(=O)NC(C2CN(C(C3(C(F)F)CCCO3)=O)C2)C)ccccc1Cl C1(Nc2ccc(NC(C(C)(C)C)=O)cc2)COC2(CCNC2)C1 c1(NCc2nnn(CC)n2)nc2ccccc2nc1NCC(C)C(F)(F)F C(=O)(CCCCC(N)=O)N1CCCC(NC(COc2cccc(C)c2)=O)CC1 CCCCC(C)CCC(=O)N1CC2=C(C1)CN(C(=O)C=CSc1nc[nH]n1)C2 Cn1cc(C(=O)NC2CN(C(c3cc(C4CC4)ccc3F)=O)C2)c2cccnc12 C1CC2(CC2)S(=O)(=O)N1.C1(C)(CC(C)(C)NC(=O)N)NC(=O)NC1=O N1(C(C2C(C(C)C)OCC2)=O)CCC(CNC(=O)CCCN=[N+]=[N-])C(O)C1 C1(C(N2CCC(NC(=O)C(C3CCOCC3)O)CC2)=O)CCn2nnnc2C1 CCCCCCCCC(C(=O)NC(C)CC)N(CCC#N)CCc1ccccc1 c1(-c2cn(C(C)(C)C(=O)O)nn2)ccccc1C(=O)Nc1csnc1C(N)=O C1(NC(c2c(CCC)occ2)=O)CCCCCC1NC(C1CC(C)(C)CO1)=O c1(C(N2CCC(NC(c3cc(C)ncn3)=O)C(C)C2)=O)cccc2c1NCCC2 Cc1cc([N+](=O)[O-])ccc1C(=O)NCC(C)(CO)N(C)C N1(C(CSCCCC)=O)CCC(C)C(NC(C2(C)CCN(C)C2=O)=O)C1C c1(N2CCC(Oc3cc(C)ncn3)CC2)cnc(C#N)c(C#N)n1 C1(C=O)CS(=O)(=O)CC(=O)N1.CC(C)C(C)C.C1(C(=O)N)CCS(=O)CC1 N1(C(C2(C)CC(F)(F)C2)=O)CCN(C(=O)C=CSc2nc[nH]n2)CC(C)(F)C1 c1(C(=O)NCc2oc(C(N3C(C=C)CC3)=O)c(C)n2)ccc2[nH]nc(Cl)c2c1 C(C)(c1ccccc1)=CC(=O)N(CCC)C.c1nc(C)c(C=O)s1.COC N1(C(C(CC)SC)=O)CC(C(N2CCc3ccncc32)=O)CC(C)(C)C1 C1(C(=O)N)C2C3CC4C1C2C34C(N1CCC(C2(C)N=N2)CC1)=O.CC(C)C C1(=CCNC(C(N2CCCC(O)C2)C)=O)CCN(C(=O)Cc2nccn2C)CC1 C(C)(CCC(C)C)N(C(C(c1ccco1)NC(c1cc(C)no1)=O)=O)C Cc1nc(C2CC2)nc(O)c1C(=O)NC(C)CC(C)Nc1nccnc1C#N C(CCC(C)C)OC.C1(O)(C(C(=O)N)F)CN(C(c2ccc(C(N)=O)[nH]2)=O)C1 Cc1cncc(C(=O)NC2CC23CC(NC(C2C(C)(C)C2(F)F)=O)C3)n1 c1(C(N2CCC(C=O)C2)C(=O)NCCCSCC)ccc(C(F)F)cn1.N CCCCCC(=O)NCC=CCC(=O)NCC1(CO)CC12CCC2 N1(C(C(CC)C)=O)CC(=O)NCC1C(=O)NCC1CN(C)CCN1C C#CC1(C(N2CCCC(CC=C)C2)=O)CCN(C(C2CC(=O)N(OC)C2)=O)CC1 C(=O)C1=CCC(C)(C)CC1.N1(C(C(C(C)C)OCC(C)C)=O)CC2(CCC2)C1 c1(C(N2CCN(C(C3(C=C)CCOCC3)=O)CC2CC)=O)cc2n(n1)CCOC2 n1(CCC)cn[nH]c1=NC(=O)N1CCC(NC(N2CCCC2)=O)CC1 C1(C)(C(N(CC(O)CO)C)=O)CCCN1C(C1CC1[N+](=O)[O-])=O C(=O)(C(C)(C)C(=O)NCCC1(O)CCN(C(c2cc(Cl)cn2C)=O)C1)N(C)C c1(CS(=O)(=O)C2CC2c2ccccc2)c(F)ccc(F)c1Cl C(C1=NOC2CN(C(c3ccccc3S(=O)CC)=O)CC12)NC(CCC)=O c1(NC(Cc2c(C)nn(CC)c2C)=O)c(C(=O)O)sc2c1COCC2 n1(CC)cc(Cl)cc1C(N1CCC(NC(=O)Cc2cccc(CO)c2)C1)=O c1(C(N(C(CCNC(C2(COCC)CC2)=O)C)C)=O)ncc(F)cc1N c1(C2C(C(=O)NCC34C(CN(C(C(C)CO)=O)C3)C4)C2)ccc2ccccc2c1 C(=O)(CC(C)(C)C=O)OCC.c1(CC=O)ccnn1C(C)C.C(C)CC.N C1(n2cc(Sc3ccc(C)nc3)nn2)CC2CCC1(CN1CCCC1C)C2 c1(C(N2CCC(N(C(CN(C3CCSC3)C)=O)C)C2)=O)cc(C2CC2)nn1C c1(C(=O)NC(C2CN(C(c3cc(C4CC4)[nH]n3)=O)C2)C)ccon1.C1CC1 C1(NC(C(C)SCC)=O)CCN(C2CCN(C(=O)C3=CCC3)C2)CC1 C#CCC(C)(CC)C(=O)NCC1CN(C(c2ccc(CCC)cc2)=O)CC12CC2 C1(CNC(COCCC=C)=O)CCCC1NC(=O)CCSc1nccn1C c1(C(=O)NCCC2CC(OC)CN2C(C2OCCO2)=O)ccc2nc(C)[nH]c2c1 CC(C)CS(=O)(=O)CC(=O)NC(C)CC(C)NC(C12CCC(CC1)OC2)=O.C N1(CCc2cn(C(C)C(=O)N(CCSC(F)(F)F)C3CC3)nn2)CCC(O)CC1 C=CCCCCCC(=O)NCC1(COC)CCN(C(c2[nH]ccc(=O)c2C)=O)C1 C(=O)(C1Cc2ccccc21)N(C(CC(=O)N(CCN(CC=C)C)CC)CC)C C1(C(C)C)CN(C(c2cc(Cl)no2)=O)CCN1C(=O)CNC(C1CCC1)=O CCC(C)CC(C(=O)N(C)Cc1cnc[nH]1)NC(=O)CCC1CCCCC1 CC(c1ccccc1F)=CC(=O)N(CC(C)(C)NC(=O)CC1CC2CC2C1)C c1(C(=O)OCCOc2cc(Cl)ccc2Cl)c(F)ccc(F)c1Br C1(NC(CCSCC)=O)C(C)CN(C(c2ccnc(O)c2)=O)CC1C c1(C(=O)NCC=CCNC(=O)Cc2cscn2)ccc2cnoc2c1 C(=O)(C(C)CC(=C)C)N1CCC(CN(C(C(C=C)c2ccccc2)=O)CC)CC1 CC1(C)COCC1CC(=O)N(CCCNC(=O)C(N)=O)CC1CCCC1 C(CCC(C)(C)NC(=O)CNC(=O)NCC)NC(C1(C#C)CCC1)=O C(c1ccc(F)cc1)=C(C)C(N1CCCC(C)C1)=O.C1(C)(C=O)CS(=O)(=O)C1 c1(C=O)c(F)cncc1Cl.c1(NC(C)=O)nc(C(=O)NC(C)C2CCC2)cs1 C1(C(=O)NC(CC(C)C)CO)CCC2(CN(C(c3cccc4c[nH]nc34)=O)C2)O1 C(=O)C(C)(C)S(C)(=O)=O.C1(CNC(C(F)=C(C)C)=O)CCCC(C)C1 c1(OC)ccc(CCC(=O)NCCCNC(=O)CCCCC2CCCCC2)cc1 C(CC(CO)C(C)C)NC(C(C)N(C(c1cc(C(C)C)[nH]n1)=O)C1CC1)=O CC(C)C(=O)C(=O)N1CC(C)(C(=O)NCC(C)(O)C2(C)CC2)C1 C(=O)(N=S1(=O)CCCC2(C1)OCCO2)c1cnn(C)c1C(F)(F)F C=CCC(CNC(C1CC(OC2CC2)C1)=O)C(=O)NC1CC(C)(C)C1 c1(CC(C(=O)N(CCCc2c(C)ncs2)C)C)ccc(Cl)cc1 C1(NC(C(C)OC)=O)CCN(Cc2ncccn2)CC1C C1(CNC(c2c(C)c[nH]n2)=O)COC(C)(C)CN1C(=O)C=CC(F)F N1(C(c2c(CC)noc2)=O)CC2CN(C(=O)C(F)(F)C(C)O)CC2C1 c1(CC(=O)NCC(CNC(CCCCC=C)=O)C)cnn2c1CCCC2 Brc1cccc(CNC2(c3ccc(Br)cn3)CCC2)c1 c1(CC)cc(C(=O)N(C)C)c(C)nn1.c1(C(C(N2CCC2)=O)C)c(C)n[nH]c1C C1(NC(=O)NCC(C2CC3C=CC2C3)(C)O)CCS(=O)(=O)C(C)(C)C1 Cc1cc(C(N2CCC(C(C)NC(c3ccsc3Cl)=O)CC2)=O)c2c(c1)CCO2 c1(C(N(CCC(C)NC(=O)C)C)=O)cc2n(n1)CCO2.N1(C(C)C)CCCC1.O C1(CNC(c2cc(COC)no2)=O)COCCN(C(C2CCC3CC23)=O)C1 c1(C(C)NCc2ccc(NC)c(F)c2)ccc2c(c1)OCO2 N1(C(COc2c(CC)cccc2)=O)CCCCC(NC(=O)C)C1.CC(F)(F)F.S CC(C)C(C(=O)N1CCC1(C)C(C)C)NC(C1COC(C)C1)=O c1(C(=O)NC(CNC(CSCCC(C)C)=O)C)coc(C2CCOCC2)n1 c1(C(=O)NC(CC(C)NC(C(CC)SC)=O)C)cnc2c(c1)CCOC2 N1(C(C=Cc2ccc(OC)cc2)=O)CC2CCC(C1)C2N1CCC2CCOC2C1 C1(O)(C(=O)NC2CCC(c3cn(CCCOC)nn3)CC2)CC2CCC1C2 C(=O)(C(O)C1=CCCCC1)NCCOCC(=O)NCC(C(=O)NC)C c1(NCCOC(C)(C)C)cc(=NC2CC2C2CCCC2)[nH]c(C(F)(F)F)n1 C1(NC(=O)NCCCCC#C)CC2CC1CC2NC CCCCC(=O)N1CSCC1C(=O)NC1CC(NC(=O)C(F)(F)c2cscn2)C1 C(=O)(C(F)(F)C(O)CC)NC1CCC(NC(CC(C(=C)C)OCC)=O)C1 N1(C(CC(CC)C)=O)CCC2(CCCN2C(c2cccc(Cl)c2N)=O)C1 N1(C(C(C)SCC)=O)CC(NC(C2(C3CCOCC3)CC2)=O)CC12CCC2 C=C(C)CCC(C)(c1nnnn1CC)Nc1cnn(CCOC(C)=O)c1 C(CC(C(=O)NC(C1CCOCC1)C)NC(c1conc1C)=O)SC c1(N2CC(NC(C3(CC)CCC3)=O)C(C)C2)c(Cl)cc([N+](=O)[O-])cc1Cl C1(NC(C(CNC(c2c(C)ncs2)=O)(C)C)=O)CCCCC1N=[N+]=[N-] C(=O)(C=CSc1ccccc1)N1CC(CC(C)NC(C2CC2[N+](=O)[O-])=O)C1 N1(C(C)=O)c2ccccc2CC1CNC1C(NC(=O)CCC2CCC2)CCC1 c1(CCC(=O)NCC(C)(C)C)ccc(O)c(Cl)c1.C1(C=O)CCC(=O)NC1.N O=C(C#CC1CCOC1)NCC1CC2CC2N1C(c1coc(Br)n1)=O C1(CNC(C2CS(=O)(=O)C2)=O)CC12CCN(C(C1COCCO1)=O)CC2.C C1(NC(C(Cc2ccc(C)cc2)C)=O)CC(N=c2[nH]nc(C(C)(C)C)o2)C1 C1(C(=O)NC2CC(OC)C2)(NC(C(C2CC2)OC)=O)CCN(C)C1 CCC(C)CC(=O)N1CC(N2CC(NC(c3cc(C(F)(F)F)on3)=O)CC2=O)C1 CC1CN(C(C2CCN(C(C3CCC(C(=O)O)C3)=O)C2)=O)CC(C)O1 N1(C(c2ccc(CCC)[nH]2)=O)CC(NC(=O)C(O)Cc2ccccc2)CC(C)C1 C1(C)(C(=O)NC2CN(CCC)C(=O)C2)CN(C(=O)C(C)N(C)C(C)=O)CC1C N1(C(c2c(C)csc2)=O)CC2CCN(C(c3cccc(Cl)c3I)=O)C2C1 c1(C(N2C(C3(O)CN(C(Cc4cccc(C)c4)=O)C3)CCC2)=O)cc(C)cc(Cl)c1 c1(OC)cc(C)c(C(N2CC(NC(=O)CCSC(F)(F)F)CCC2C)=O)cn1 C1(N(C(C(Cc2ccccc2)OC)=O)c2nc(C)ns2)COC2(CCNCC2)C1 O=C(C1=CS(=O)(=O)CCC1)NC1CCCN(C(C2C3CCC4C(C3)CC24)=O)C1 c1ccc(F)cc1.Cc1cocc1C(=O)NC(C1CCCN1C(=O)CSC)C C1(NC(Nc2ccc(F)cc2)=S)CCCCCCC1 CC1CCCCN1CC(N1CCC(CC(=O)Nc2cncc(Br)c2)C1)=O c1(OC)ccc(CNC(=O)C(=O)NC(c2cccs2)C2CC2)cc1 C(c1ccncc1)=C(C)C(=O)NCC1CCC1(C)C.C(=O)(CCc1ccoc1)N N1(C(c2ncn(C)n2)=O)CC(NC(c2c(Cl)csc2Cl)=O)C2CCCCC12 Cc1ccc(C(=O)NC2CCC(C(N3CC(C#N)(CCF)C3)=O)C2)c(C)n1 c1(C(N(C)CC2CCCN(C(CCC(=O)NC)=O)C2)=O)cc(C)ccc1O CCCC(C)C(=O)NCC1(C(N)=O)CN(C(=O)CCc2cnn[nH]2)C1 c1(C(=O)N)c(F)ccc(F)c1F.c1(C(=O)NCCC)ccnc(OC(F)(F)F)c1 c1(-c2ncc(C(=O)NC(C3CN(C(C4C=CCC4)=O)C3)C)s2)ccccc1Cl C1(N(C(=O)CC2(O)CCC2)C)CCN(C(=O)CCc2ccc(O)cc2)CC12CC2 C=CCN=C(NCC1CCC(c2ccccc2)C1)N1CCCC2(CC2)C1 c1(C(=O)OC)sc(=NC2CC(C)N(C(C3CC4CCC3CC4)=O)C2)[nH]c1Cl C1(N(C(Cc2nc(C)sc2C)=O)C)CC2CC1N(C(c1cc(C(N)=O)c[nH]1)=O)C2 CC1CCN(C(=O)Cc2cccc(C(N)=O)c2)CC1NC(C1(O)CCOC1)=O C1(NC(c2n(CC)ncc2)=O)CC(C)N(C(C2CCN(C3CC3)C2=O)=O)C1 C(C(=O)NC1(CO)CCN(C(=O)CC(O)C(C)C)CC1)(C(C)(C)C)c1ccc(C)o1 N1(Cc2ccc(OCC#C)cc2)CC2CCC1CN2C(=O)Cc1ccccc1F C1(OCC)CCCC(C(CC)=O)C1.C(=O)(C)NCC.C(=O)NCC.CC CS(=O)c1ccccc1C(=O)NCC(CNC(=O)C(F)=CC1CC1)CO c1(CC)nc(=N)[nH]cc1C(N1CCC2(NC(=O)CC3(O)CCCC3)CC2C1)=O n1(CC)nc(C(N2CCC(NC(c3cc(C)[nH]n3)=O)C(OC)C2)=O)ccc1=O c1(C(N2CC(O)(C)C2)=O)ccc(C(F)(F)F)[nH]1.C1(C=O)(C(=O)O)CC1 C1(NC(CCC2C(C)(C)C2)=O)CCC2(CC1)CCN(C(=O)CNC(N)=O)C2 C1(C)(CNC(CCCC2C(C)C2)=O)COCCN(C(=O)CCc2nccs2)C1 c1(C(N2CC(C)C(CNC(=O)Cc3ccc(Cl)cn3)C2)=O)cc2ccsc2[nH]1 c1(NC(C(c2cccnc2)NC(c2c(CC)c[nH]n2)=O)=O)cc(C)cc(C)c1 C1(CC(=O)NCC(=O)OCC=C)CCCCC1.C(CCN)N.C(C)=O CC(C)(C)S(=O)(=O)CC(=O)NC(CO)CCCC.C1(C=O)C(C(F)F)C1(C)C CCC(CN=c1cc(NCC2(N(C)C)CC2)nc(C)[nH]1)N(C)C N1(C(COC(CC)C)=O)CC2(C1)CN(C(=O)C=Cc1ccco1)CC(C)(C)O2 C1(C(N(CC(c2ccccc2)O)C)=O)C2CC1N(CCN1CCCCC1=O)C2 c1(CC=O)cc(F)ccc1C.C1(COC)CCC(C(=O)NC)C1.C1CCCC1 c1(NC(C)C2=CCN(C)CC2)ccc(S(=O)(=O)N2C3C=CCC2CC3)c(Br)c1 C(CC(=O)NCC=CC)(C(F)(F)F)OC.c1(C=O)cnn(C2CCC2)c1.N c1(C(N2C(C3(NC(=O)CSC4CCCC4)CC3)CCC2)=O)ccnc(S)c1 C(c1cnc[nH]1)=CC(=O)N(C(C)CCNC(=O)CCc1cscn1)C c1(C(=O)NC2CN(C(c3nnc(C(C)C)s3)=O)C(C)CC2)ccc2nncn2c1 c1(C(=O)NCC(CNC(C2C(C(N)=O)C2)=O)F)cc2cnc(Cl)cc2s1 N1(C(C2C(OCC)CC2)=O)CC(OC)CC1C.c1nccn1C.C(=O)(C)N O=C(C(O)C(F)(F)F)NC(C(=O)NCc1nnnn1C1CC1)c1ccco1 C1(C(=O)NC2CC(C)(NC(c3c(NC)cnnc3)=O)C2)OCCCC1(C)C c1(CNC(C2CCC2c2ccccc2Cl)=O)ccc(Br)cc1Br c1(C(C)C)ccc(C(=O)N)c(O)c1.C1(CC)CCN(C(=O)C=Cc2cnc[nH]2)C1 CC(CC(N)=O)C(=O)NC1CC1CNC(c1ccc(OC(F)(F)F)cn1)=O C1(O)(C(C)NC(=O)Cn2cc(Br)cn2)CCN(C(=O)C2=CSCS2)C1 C1(CCC)CCCC1C(N1CCCC1Cn1cc(-c2nc(C)cs2)nn1)=O C1(C)(C(=O)NC2C(C)N(Cc3ccccc3)C(=O)C2)Cc2ccccc2C1 C1(NC(C(N2CCCC(C(N)=O)C2)c2cccnc2)=O)CCOC2(CCC2)C1 C(C1=CCCN(C(C2(N(C)C)CC2)=O)C1)NC(Cc1ccc(C)cc1)=O C1(C(N2C(CNC(C3(OC)CCCCCC3)=O)CCC2)=O)CCn2nncc2C1 c1(C(=O)NCC2CN(C(=O)CCc3cc[nH]n3)CCO2)nc[nH]c2ncnc1-2 c1(CC)ccc(C(C)OC2CCOCC2)o1.C1(C)(C)CCN1 N1(C(C2CCC(C#N)C2)=O)CC2(CC2)CC1CNC(=O)CN1CCCC1=O N1(C=O)CCN(C2CN(C(=O)CC3CS(=O)(=O)C3)C2)CC1.c1c[nH]cn1.C C1(C(=O)NCCCCC#C)CCC(NC(=O)C(C(C)C)NC(C)C)CO1 N#Cc1cc(NC(=O)CC2CN(C(c3ccc(O)c(O)c3)=O)C2)ccc1F C1(C)(CC)NC(=O)N(CC(=O)OC2CC3CCC2O3)C1=O c1(C(=O)N)c(C)noc1C.c1(C(C(N2CC(OC)(C)C2)=O)CO)ccc(F)cc1 C#Cc1cccc(C(N2CC3C(NC(c4c(C)nsc4)=O)C3C2)=O)c1.C1CC1.N C(=O)(C1Cc2c(Cl)cccc21)N1CCCC(N(C)C(c2cccn2C)=O)C1 Cc1ncc(N)cc1C(N1CCN(C(c2ccn(C(F)F)n2)=O)C(C2CC2)C1)=O S(=O)(=O)(c1ccc(N2CCOC3(CCCC3)C2)nc1)NC1CCS(=O)(=O)C1 c1(C(N2C(CC(=O)NC(C3CCCCC3)CC)CCC2)=O)nc(=N)cc[nH]1 c1(CC(=O)NC2C(C)N(C(c3cccnn3)=O)CCC2)csc2ccccc12 c1(CNC(=NCCCOCC)NCC(C)CC)cc(C#N)ccc1F N1(C(C2(CNC(CC=C=C)=O)CC2)=O)CCCCCC1C c1(OC)ccc2c(c1)CCC(C(=O)N)C2.C(=O)(C(C)(C)C(F)F)N1CC(O)C1 C(=O)(C1CCCn2cnnc21)N1CC(NC(c2ccco2)=O)CC2(C1)CCC2 N1(C(C2C(NC(c3occ4c3CCC4)=O)COC2)=O)CCc2nocc2C1 Cc1ccc2c(c1)CC(C(=O)NC(C1CCCCC1)C)N2 O=C(CCN=c1[nH]c(=NCCC(O)C2CC2)c2cc(F)cc(F)c2[nH]1)NC1CC1 c1(OC)ncccc1CC(=O)N(C)CC1CCN(C(C2CCOCC2C)=O)CC1 c1(C(=O)NCC2N(C(C3CC(OC)C3)=O)CC(C)CC2)c(Cl)ccc(Cl)c1O C1(CCNC(c2ncc(-c3ccc(Br)cc3)[nH]2)C)CC2CCC1CC2 CC(C(=O)NO)NC(C1CCCN1C(=O)COCc1nc[nH]n1)=O C1(C(=O)NCC(C)NC(C2Cc3ccncc3N2)=O)CCc2nn[nH]c2C1 C(CC(N=c1ccnc(NCC(C)(C)C)[nH]1)c1cccnc1)N(C)C c1(C(N2CCN(C(C(CC)C)=O)CC(C)(F)C2)=O)cccc(S(C)(=O)=O)c1F c1(C(N2CC(C(C)NC(C3CC3C#N)=O)OCC2)=O)ccc2nccnc2c1 Cc1cc(C(N2CCN(C(=O)CCP(C)(C)=O)CC2C2CC2)=O)nc(C)c1 c1(NC2C(C(N3CCCC(F)(F)CC3)=O)C2)ncc2c(Cl)cccc2n1 N1(C(c2nc(C)oc2)=O)CC2N(C(=O)C(O)CCC(C)C)CCC2(C)C1 C1(CC(=O)NCCCN2CCN(C(C(C)n3cncn3)=O)CC2)COCC(C)(C)O1 c1(OC)c(C(N2CC(CNC(C3(C(F)F)CC3)=O)C2)=O)oc2ccccc12 C1(CC(=O)NCc2cnccc2Cl)CCN(C(C2CC(O)C2)=O)CC1 CC(CF)CC(=O)N1CCCCC1CN(C)C(c1ccnn1C)=O N1(C(c2ncn(C)c2)=O)CC2(COC(CNC(C34CC(F)(C3)C4)=O)C2)C1 N1(C(C(CC)OC)=O)CCCN(C(=O)C(=Cc2ccc(Cl)cc2)C)C(C)C1 N1(C(CCC=CCC=C)=O)CC2CC2(CNC(=O)CNc2cccnc2)C1 c1(C(N2CC(CCCNC(C(C)C3CC3)=O)OCC2)=O)sc2sccc2c1Cl O=C(C1=CC(O)CCC1)NCC1CCCN1C(c1cn(CC2CC2)nn1)=O c1(C2C(C(=O)NC(CNC(CCCC)=O)CC)C2)cc(Br)ccc1C N1(C(C(C)(C)O)=O)CCCN(C(C2CCC3(CCC3)O2)=O)CCC1 c1(C(N2CCN(C(c3n(CC)ccn3)=O)CC2CF)=O)ccc2nn[nH]c2c1O CC1CC(NC(=O)C(CN(C)C)N(C)C)CCN1C(C12COCC1C2)=O N1(C(C2CN(CC(C)C)C2)=O)CCCC1C(C)NC(=O)CN(C)C c1(OC)cc(OC)c(C(=O)NC2CC(C)C2)cn1.C1(C=O)CC1.N(C)C C(N1C(=O)Cc2ccccc21)n1c(N2C(C)(C)CSCC2)nnc1SC1CC1 CCC(CC)(CC)C(=O)N(CCC(C)NC(c1ccc(CNC(C)=O)s1)=O)C C1(CC(=O)NCCCOCCCO)CCCN(C(=O)CCC2CCCCC2)CC1 CC1(C(=O)NC2CN(C(C3(c4cnn(CC(F)F)c4)CC3)=O)C2)CC2CC2C1 c1(CN2CC(C(=O)OC)C2)ccnn1-c1ccccc1 N1(C(C2OCCC2C(F)(F)F)=O)CC2CCC(C1)N2Cc1cc2n(n1)CCCO2 C(c1ccccc1Cl)=CC(N1CCC(C(C)NC(C2(C)CC3CC3C2)=O)CC1)=O N1(C(C=CCN(CC#C)C)=O)CCC(C)C(NC(c2cc(O)cnn2)=O)C1C c1(C(N2CCCC(NC(C3CCC(C(N)=O)CC3)=O)C2)=O)cc(F)c(F)cc1I c1(C(=O)O)ccc(C(=O)NC2COCC2n2cc(C3CCOC3)nn2)o1 N1(C(C(N2CCC(O)CC2)C)=O)CCCC(CO)(NC(=O)C(F)C(C)(C)O)C1 C(=O)(C1=CCCOCC1)N1CCC(NC(C(C)NC(C2CCC2)=O)=O)(CO)CC1 c1(C(C)=O)cnc(F)c(NC2CCC(CNC(=O)OC(C)(C)C)C2)c1 CCC(CCC(=O)NCC(O)CCOC)NC(=O)COCC1CC1 c1(CC)cnsc1C(N1CCCC1CC(=O)NCC1CCC(O)C1)=O C1(NC(CCC(=O)NC)=O)CCCN(C(=O)CCn2ccc(O)nc2=O)C1C c1(SC(C)C(=O)NCCCOCCN(C(=O)CCS)C)ccccn1.CCO C1(C)(CC)CC(NC(c2sccc2F)=O)CN1C(c1cccnc1)=O.N(C)C.C c1(-c2n(CCNC(C)=O)ccn2)ccc(-c2nc(N3CCOCC3)n[nH]2)cc1 c1(NC(CCC2CCCN(C(C3CN(C(C)=O)C3)=O)C2)=O)cnc(C)c(C)c1C c1(C(C(=O)N2CC(OCC(N)=O)C2)NC(C)=O)ccccc1 C1(CC=O)CC(=O)NC(=O)C1.C1(C=O)(C(=O)N(CCCC)C)C=CCC1.C O=C1CC(CNC(=O)C(c2ccoc2)NC(=O)CC2OCCO2)CCN1 C(=O)(C#CC1CCOCC1)N(CCC(=O)N(C1CC(C)OC(C)C1)C)C c1(C(=O)NCc2ccc(CCC(=O)OC)o2)ccc(N=[N+]=[N-])cc1 C1CC2CCC(C1)O2.C(C1CCC1)=CC(=O)NCCOCC.CC.CC.O C(=O)C1=CCS(=O)(=O)C1.N1(CC(C)C)CC(C(N2CCC(C)C2)=O)CC1=O.N c1(OC)cc(Br)cnc1C(N1CC(C)(NC(C2CC(C)=NO2)=O)C1)=O N1(C(C=O)=O)CCN(C(c2ccc(C(C)(C)C)c(Cl)c2)=O)C(C(C)C)C1.CC C1(NC(CC2C(C)(C)CCN2C(c2cscc2Cl)=O)=O)CC2COCC(C1)C2 CC1=NNC(=O)C1CCC(N1CCCC1Cc1cn(CCCO)nn1)=O Cc1cc(O)nc(C)c1C(=O)NCCCN1CCN(Cc2ncccn2)CC1 CC1(C)CC(C(=O)NCC2(C)CCCC2)C1.C1(C#N)(CC=O)CCC1.N CC1(C)CCC(CNC(C2CCC(=O)N2)=O)N(c2ncncc2Br)C1 N1(C(C2CC(C#N)(OC)C2)=O)CC2CC1CN(C(c1cc(CO)[nH]n1)=O)C2 C1(CCC)(C(N2CC3CC2(CNC(=O)CC(C)n2ccnc2)C3)=O)CCNC1=O Nc1cc(C(NC2CCc3ccsc32)=O)c(F)c(C(F)(F)F)c1 C1(C)(C(=O)NCC2CN(C(C(CO)NC(C)=O)=O)C2)COC(C)CO1 C1(O)(CC(N2C(CNC(C(c3ccc(F)cc3)(C)F)=O)CCC2)=O)CCOCC1 C1(CNC(C(C=C)c2ccccc2)=O)CN(C(C2CC23CC3)=O)CCCO1 C12(NC(C=CCOC)=O)CCOCC1CN(C(=O)CC1CCSCC1)C2 CCCC(CCC)CC(=O)N1CCCC(C(=O)NCC(F)(F)F)(CC)C1 c1(-c2ccc(NCCN3CCC(Oc4cn(C)nc4Cl)C3)s2)cccc(F)c1C#N N1(C(c2c(F)ccc(OC)n2)=O)C2CCC1CC(F)(CNC(=O)CC(C)S)C2 c1(OCC)ccc(CNC(c2cnc(-c3ccsc3)s2)=O)c(C)c1 NS(=O)(=O)c1cc(C(=O)NCCCNC(C2COC(=O)N2)=O)cc(F)c1 c1(C(N2CCCC(N(C(c3ccnnc3)=O)CC)C2)=O)cnc(OC)c(C)n1 C(=O)(C(O)CCCc1ccccc1)N(CCCCNC(C(C)C1CCC1)=O)C N1(C(C(C2CC2)OC)=O)CCC(C(N2CCC(CC3CC3)CC2)=O)C1(C)C c1(OC)ccc2oc(C(N3CCCN(C(c4cc(C)sn4)=O)CCC3)=O)cc2c1 N1(C(c2c(C)ccs2)=O)CCC(C)C12CCC2.N1(CC=O)C(=O)CN(C)C1=O.N C1(OC)CC(CNC(=O)CC(C)O)N(C(c2ccc(C3SCCCS3)cc2)=O)C1 C=CCC(C(=O)NCC1CCN1C(=O)CC(C1=CCCC1)OCC)C(C)C C(C)(C)(CC(C)NC(=O)C(CCF)NC(=O)Cn1cc(C)cn1)OC C1(C(=O)OCC)(C(C)C)CCCN(C(=O)NCC2CC=C(C)CC2)C1 CC(C)C(O)C(=O)Nc1cccc(NC(=O)C(F)(F)c2nccn2C)c1 Cc1cc(Br)cc(CN=c2[nH]cc(-c3cnn(CC#N)c3)s2)c1O c1(C(=O)NCCn2cc(CNC(C)=O)nn2)c(F)ccc(C)c1O C1(OC)(CNC(C2CC(=O)N(C)C2)=O)CCN(C(=O)CC2CSC2)C1 c1(C(N2CCN(C(c3c(C)nc(C)o3)=O)C3C2C3)=O)ccc2nccnc2c1 CC(c1cccnc1)=CC(=O)NCC1(C)CCN(C(=O)CCC2CCCOC2)C1 C1(CC=C)(C=O)CCCC1.c1(CC)n[nH]cc1C(=O)N(C(C=C)C1CC1)C.N C1(OCc2cccc(OC)c2)CC2(C1)CC(NC1CCC(=O)C(C=O)C1)C2 N1(C(COCCOCCOC)=O)CC2CCC1C2.c1(C(=O)N)cn(C)nn1 N(C(=NCC(O)c1cccc(Cl)c1)NCc1nc(COC)n[nH]1)C(CC)C C1(n2cc(C3CCN(C)C3)nn2)CC(C)(C)OC1(C)C.C12(O)CCN(CC1)CC2 c1(C(c2n(CCSC)nnn2)NC2CS(=O)(=O)C2)c(C)cc(Cl)cc1C C(C(=O)N1CCC(C(=O)NC2CC(c3n[nH]c(C)n3)C2)O1)N(C(C)=O)C N1(C(c2c(CC)ncs2)=O)CCC2(CC(NC(c3c[nH]nn3)=O)C2)C1.C1CC1 c1(OC)cccc(CN2CC(C(=O)Nc3ccnc(C(N)=O)c3)CC(F)C2)c1C C1(N(C)C(C2CC23CCSCC3)=O)CC2CC(NC(=O)C(=O)N)C1C2.C1CC1 Cc1cnc(C(N2CC(C)CCC2C(N2CCCN(C)CC2)=O)=O)cc1C N1(C(c2ncc(Br)cc2F)C(=O)NC2(C)CC2)CCn2cccc2C1 N1(C(COCCCC)=O)CCC2(CCCC2C)CC1.C(=O)(C(C)(C)C1CCC1)N c1(CCC(=O)NC2CCN(C(C=CCC)=O)CC2C)c(O)nc(=N)[nH]c1C C#CCCC1C(=O)N1.C(=O)(CCC(C)OC)N1CC(C(=O)OC)(CC=C)C1 C1(CC)CN(C)CCN1C(=O)CCN(C(=O)C)CCO.C1(C(=O)N)CC1C C1(OC)CCN(C(C2CC2CNC(=O)CCO)=O)C(C)C1.C1CCC1.C O=C1NC(Cc2cscn2)C(=O)N1Cc1ccc(-n2cncn2)nc1 CC1(NC(=O)Cn2cccc2)CCCCC1C(N1CC(F)(F)C1C1CC1)=O N1(C(c2ccc(OC)cc2F)=O)CCN(C(=O)C(O)C2CCC2)CCC1C C1(C2(O)CN(C(C3CN4CCC3(C)C4)=O)C2)CC1.Cc1snnc1C(=O)NC CC1Cc2sc(C(=O)NCC3(C)CC3)cc2C(C)C1.C1(F)(C=O)CC=CC1 CCCCC(CC)C(=O)NCC1COC(C)(C)CN1C(=O)C=Cc1cc[nH]n1 c1(C(=O)NCC(C)CNC(=O)CC2CCC2)ccc(I)c(O)c1 c1(C(N2C(C)CC(NC(C3(F)CCCC3)=O)CC2)=O)cnc2c(c1)COCC2 Cc1[nH]nc(Cl)c1C(=O)NCCC(O)CNC(c1cnn(C)c1CC(C)C)=O O=C1CCC(C(=O)N2CCn3c(CC(F)(F)F)nnc3C2)c2ccccc21 C(=O)(C1CCc2c[nH]nc21)N1CC(NC(CC(CN(C)C)(C)C)=O)C2C1CCC2 C1CCCCC1.n1(CC)cnc(C(=O)NC)n1.C(=O)(C(C)SC(F)(F)F)NC c1(C=O)ncnc(O)c1F.C1(C(=O)NC(C23CC(CO2)C3)C)(C)CC=CC1 Cc1nn(C)cc1C(=O)NCC(C)C.C(=O)(C(C)C)N.C(C)(C)C.C=O C(c1ccc(F)c(Cl)c1)=CC(N1CCN(C(C(N)=O)=O)C(CC(F)F)C1)=O N1(C(CNC(CCC)=O)=O)CCC(CO)(NC(C2CCC3CC3CC2)=O)CC1 n1(CC=C)c(N(CC(C)(C)C)C)nnc1-c1ccc(OC(F)F)cc1 C1(CC=C)(NC(c2ccc(C)c(F)n2)=O)CCN(C(c2ccno2)=O)CC1 CC1CN(C(c2cnn(C)c2C2CC2)=O)CCCN1C(=O)C1=CCS(=O)(=O)C1 N1(C(C2(C(F)(F)F)CCC2)=O)CCCC(n2cc(Cc3cnn[nH]3)nn2)C1 C(C(=O)NCC1CN(C(c2ccccc2C)=O)CCO1)(C(C)C)n1ncc(C)c1 C12(CNC(C(CC(C)C)N3CC(F)(F)CC3C)=O)CC3CC(CC(C3)C1)C2 CCCCC(C)(F)C(=O)NCC(COC)NC(C1CCCCN(C)C1=O)=O C(C(O)(CO)CO)NC(C(C1CN(C(C2C(OC)CCC2)=O)C1)OC)=O c1(C(N2CCC(C)(NC(Cn3c(C(C)C)nnn3)=O)C2)=O)csc2nccn12 C1(CCNCC(=O)NC(C(=O)N(CCCN(C)C)CCN)=O)CCCC1 CCC(CCC(=O)NCCCC(C)NC(=O)CCc1c(C)n[nH]c1C)OC c1(CN(CCN(CC)CC)C=O)ccc2ccc(Cl)cc2n1.C(C)(C)C.O N1(C(C(c2ccncc2)C)=O)CC2OCCC2C1.C1CCOC1.C(=O)(CO)N.C C1(CN=[N+]=[N-])CCN1C(C(=O)NCc1cccs1)c1nc[nH]n1 C1(NC(c2ccn(CCOC)n2)=O)CCCCN(C(c2cc(C)c(C)o2)=O)CC1 c1(CC)nnc(C)cc1C(=O)NCC(C)N(C(=O)C(C)N1CCC1)C C(=O)(C(CC)CCCCC)NC(CC(=C)C)C(=O)NCCc1noc(CC)n1 N(C1CC(C)n2ncnc21)C(c1nnn(-c2cccc(C)c2)c1C)=O C1(C(=O)NC(C)CC2(O)CCC2)CCC(O)CN1C(c1ccoc1)=O CONC(=O)C(=O)NCCc1ocnc1CNC(C1CC2CC2C1)=O C=CC(CC)CC(=O)NCC1C2CCC(C2)N1C(=O)Cn1ccnn1 c1(C(=O)NC2CN(C(C(=O)OCC)=O)CC2O)ccc2c(c1)OCCO2 N1(C(CCOC)=O)CCCC(N(C)C(C2CC(C3CC3)=NO2)=O)CC1 N1(C(C(C)SC)=O)CCCC(N(C(=O)C(N2CCC(C)CC2)=O)C)CC1 C(CC)(C(=O)NCc1cnc[nH]1)NC(COCC(=C)C)=O c1(OC)cc(C(=O)NCC(C(C)C)c2ccccc2)cc(Cl)c1O c1(-c2cn(Cc3cc(NC4(CC(=O)OC)CC4)on3)nn2)cccc(C)c1Cl CCC(C)(O)C(=O)N1CCC(CC(=O)Nc2nc(C3CC3)cs2)C1 N1(C(c2cnn(CCO)c2)C(=O)NCC)Cc2ccccc2C(C)C1 N12CCCC(O)(CC1)CNC2=O.c1(SCC(=O)OCC)n[nH]c(O)n1 CCCCCCC(C(=O)NC1CN(C(c2nc(C)c(C)[nH]c2=O)=O)C1)NC(C)=O C1(CNC(c2ccc(C#C)cn2)=O)C2CCCC1N(C(C1CC=CCC1)=O)C2 Cc1cc(Br)cc(Cl)c1C(=O)NC(CNC(=O)CC(O)CN(C)C)CO c1(NC(c2ccccc2)CF)ccc2nccnc2n1 C=C1CCC(C(=O)NCCC2CCCC2)CC1.c1(C(=O)N)cnn(C2CC2)c1C CC(O)CC(C)(C)CN(CC(=O)N(C)Cc1ccccc1)Cc1ccc(Br)cc1 C(=O)(C(C(C)(C)C)NC(c1cn(C)ccc1=O)=O)NCC(CSC)(C)C c1(C(=O)NCC(C)NC(c2cc(C)cc(Br)c2F)=O)ccc2ncccc2c1 C(C(COC)CC(=O)N1CC(C=O)C1)OC.C1(Cl)(C=O)CC12CCC2.CC.N C1(CC(=O)NC(C(=O)OC)CC)CC(F)CN1C(=O)OC(C)(C)C Cc1nc(C)n(CC(=O)NC(c2ccccc2)C(C)NC(c2ccsc2Cl)=O)n1 N1(C(C2OCC(C)C2)=O)CCCCC(NC(c2ccccc2N2CCCC2)=O)C1 C1(NC(c2c(CC)ccs2)=O)CCCCCN(C(=O)CCOCCOC)C1 C(=O)(CS(C)(=O)=O)N1C(CCNC(C(C)CN(C)C)=O)CCC1 CCC(CNC(=O)C=CSC)(CC)NC(c1cc(Br)c(C)o1)=O CC(CNC(c1ccc(CNC(=O)CCN2CCOC2=O)o1)=O)C(C)O c1(OC)ccc(F)cc1C(N1CCSCC1c1cnn(C)c1)=O c1(C(=O)NC2CC(CCNC(C(CCC)O)=O)C2)cc2cccnn2c1 N1(C(c2nn(C(CC)C)c(C)c2)=O)CC2CCC1C2NC(c1ccc(F)s1)=O N1(C(CC2CC(CC)OCC2)=O)CCC2(CC1)CN(C(C1(F)CC=CC1)=O)C2 C1(NC(C(C)N(C2CCCCCC2)C)=O)CC2CCC(C1)N2C(=O)C1CC1 c1(CC)cc(C(=O)NCc2ocnc2C(=O)NCc2cnc(C)o2)ns1 CCC(C)CC(C)N(C)C(C1(NC(c2cnn(C)c2CC)=O)CSC1)=O C(=O)(CCC1=CCc2ccccc21)OCCOC1CCCC(C)C1 C1(C(=O)NCCCOCCC(=O)Nc2cn(CCC)nc2)CC(C2CC2)C1 C=CC(C)CN=C(NCc1ccncc1Cl)NC1CC1C.C(C)(C)C.C(=O)N C1(C(N2CCC(CCNC(C3CCCSC3)=O)C2)=O)(COC)CCCC1 c1(NC(c2nc(C)c(C)s2)c2n(CC)nnn2)ccccc1OCCCCCO c1(C(N2CCCC(NC(=O)CN3CSCCSC3)C2)=O)cc2n(n1)CCCO2 n1(CCCCC)cc(C#CC(C)(C)c2ccoc2)nn1 n1(CC(=O)NC(CNC(C(C)(C)CCC#N)=O)CO)ccc2ccccc2c1=O c1(SC)cn(C)nc1C(=O)NC(C)(CNC(=O)C(C)CC1CC1)CO Cc1ncc(C(N2CC(CNC(=O)CC(C)n3ccnc3)C(C)C2)=O)cc1C#N N1(C(C(C)c2ccco2)=O)CCCC1(C)CNC(=O)Cc1ccc(Br)nc1 c1(C(=O)OC)cccc(S(=O)(=O)Nc2cc(C(=O)OC)ccc2C)c1C Cc1cc(CNCCC2CC(F)C2)cc(C)c1OCC(=O)O c1(N(C)CC2CCOC2)ccc(Br)c(S(=O)(=O)NCC(c2cncs2)O)n1 n1(CC=C)cc(NC(=O)NC(C(F)(F)F)c2nc(C(C)(C)C)n[nH]2)nn1 c1(SC(C(=O)NC(CNC(C(c2ccccc2)C)=O)(C)C)C)ccccn1 CC1(C(N2CCCC(O)C2)=O)CCCN(C(C2CCCC(C(F)(F)F)C2)=O)C1 CCC(CC(=O)NCCC1CN(C(=O)C(C)(F)F)CCCO1)C(=O)O.C(C)(C)C N1(C(c2ncc(C)nc2)=O)CCC(C)(C)C(NC(=O)C#CC2CCC2)C1 CCCC(C(=O)N(C1CCCCN(C(c2cc(CC)on2)=O)C1)C)C(C)C C(=O)(C(C)(C)S(=O)(=O)C1CC1)N.N1(C(CC(C)(C)C#N)=O)CCCC(CO)CC1 N1(C(c2cc(F)nc(F)c2F)C(=O)NC(C)C)CC2(CCOCC2)CC1C C(=O)(C(C1CN(C(c2cnsc2)=O)C1)OC)NCC=CCSC C1(C#N)(C(N2CCC(CN(C(C=Cc3c(C)ccs3)=O)C)C2)=O)CCOCC1 c1(NC(CC2CCN(S(CC=C)(=O)=O)CC2)=O)cc(C(N)=O)c2ccccc2n1 C1(CC(=O)N(CCCC)CCCC)CN(C(c2cc(C)sn2)=O)CC12CC2 O=C1CCN(Cc2ccccc2[N+](=O)[O-])C(=O)N1CC1CCS1(=O)=O CCCC(C(=O)NCCNC(=O)OCC)NC(C1CCCC1)=O Cc1cscc1C(=O)NC1(C)CN(C(c2cnc(S)[nH]2)=O)C1 C(C)(C)(C(C)CC(=O)NC1CC(C)(CO)C1)NC(CCn1ccc(C)n1)=O C1(C(=O)NCC2CCCCN(C(c3nc(C)[nH]n3)=O)C2)COc2ccccc2C1 c1(CC)ccc(O)c(C(=O)NCC2CCCN2C(=O)CC2CCC2(C)C)c1 Cc1cc(F)ccc1CNC(=O)C1=NOC(C)C1.C(=O)(C(C)c1ccsc1)N C(C)(C(C)(C)C(=O)NCC(C)(C)OC)NC(COCC)=O C1(n2cc(C(C)(C)NC(N)=O)nn2)CON(C(=O)CCc2cc(O)nc(O)n2)C1 C#Cc1ccc(NC(=O)C(C2CC2)NC(c2cc(CO)ccn2)=O)cn1 N1(C(C2CN(C(C)=O)C2)=O)CCC(NC(=O)CC(C)n2ccnc2)C12CCC2 C(CC(C)(C)C)(C(=O)NC(C(=O)N)C1CCOC1)OC.c1nn[nH]c1C1CC1 CC(=O)CCCC(=O)NCCCC(C)(C)NC(=O)C(F)C1CCOC1 Cc1cc(C(=O)NC2CC(O)CN(C(c3cocn3)=O)C2)cc(S(N)(=O)=O)c1C c1(-c2ccc(C)cc2)nc(Cl)cc(=NCCC2CCCC2(F)F)[nH]1 C1(CCC)CCC(NC(=O)CCN(C)C(c2c[nH]c(=NC)s2)=O)CC1 N1(C(c2cnc(C)n2C)=O)CC(N(C)C(c2c[nH]c(Br)c2)=O)C2(CC2)C1 N1(C(CCOC(C)C)=O)CCC(C)N(C(C2CCc3ccnn3C2)=O)CC1 C#Cc1c[nH]nc1C(=O)N.C1(=CC)CCN(C(=O)CCC2CC2)CC1.C1CC1 c1(CC)ccccc1C(=O)NC(Cn1cncn1)C(=O)NC(C)C(F)(F)F Cc1c(C(N2CCOCC2CN(C)C(C2(O)CCSC2)=O)=O)cncc1Cl N1(C(C(C)=O)=O)CCCCC1C.c1(CC(=O)N)ccccc1.C(=O)C(F)(F)F Cc1nc2ncccn2c1C(N1CC2CC1CC2NC(c1cc(C)n(C)n1)=O)=O c1(CC)cccc(NC(=O)NC(c2ncco2)Cc2ccccn2)c1 N1(C(=O)C=Cc2ccc(C(F)F)o2)CC23CCCC2(C1)CN(c1ncccn1)C3 CC1CN(C(=O)CNS(=O)(=O)N(C)C)CCN(C(C2C=CCCC2)=O)C1 c1(C(N2C(CNC(=O)Cc3csc(S)n3)C3CCC2C3)=O)occ2c1CCCC2 C1(NC(CN(C(COC)=O)C)=O)CC(F)CN(C(=O)CCC)C1.C(C)(C)C.O C1(C(N2CC(C#C)(C(=O)NCc3ncc(C)o3)C2)=O)CC2C(C1)C2(F)F Cc1cn2c(n1)CCC(C(=O)NCCC)C2.C1(C(=O)N)CC(=O)N(C(C)C)C1 C(=O)(CCC(C)(C)[N+](=O)[O-])NC(C(=O)NC(CC#C)C)Cc1cnn(C)c1O N1(C(Cc2c(OC)cccc2)=O)CC(C)C(C)(C)C1.C(=O)CN(C)C(N)=O CC1CCN(C(=O)CCC2CCCOC2)CC1N(C(=O)CCC1CCC1)C Cc1cnc(NCc2ncccc2C)c(S(=O)(=O)N(C)CC2CCCN(C)C2)c1 C(=O)(C(C)(C)CC1CC1)NCC(C1CCOC1)NC(COCC=C)=O O=C(O)CC(CNC(C1CNC1)=O)C1CCCCCC1 CCCCC(C(=O)NC(C)C(C)NC(c1ccns1)=O)ON=C(C)C Cc1ncc(C(N2C3CCC2C(CNC(=O)C2CC2)C3)=O)c(O)n1 N1(C(c2cnc(C)s2)=O)CCCCC1CNC(C1(O)CC(c2ccccc2)C1)=O C=CCCCCCCC(=O)NC1CC(NC(c2cnns2)=O)C12CCC2 CC1Oc2ccc(C(=O)NC3(CNC(c4ccc(F)o4)=O)CCCC3)cc2C1C C1(CN(C(=O)C)C)CN(C(C2CC2C#N)=O)CCO1.c1(CC)ccc(Cl)s1.O c1(OC)cccnc1CNC1CCC(C(=O)Nc2csc(C)n2)CC1 C=CC1(CC(=O)NC2CCCCC2COC)CN(C(c2cn(CC)nc2C)=O)C1 OCC(CC1CC1)CN=c1ccnc(NCc2cccc(Cl)n2)[nH]1 N1(C(C(CCC)OCC)=O)CC(NC(=O)CCOCC(C)C)C2(CC2)C1 N1(C(c2c(C)n[nH]c2)=O)CCC(C)(C)C(C(=O)NC2CC=CCC2)C1 C(CCCC(CO)NC(c1ncc(F)cc1F)=O)NC(CC(C)CF)=O C1(C(=O)NC2CC(NC(c3cn(CC)nc3)=O)C2)CS(=O)(=O)CC12CC2 N1(C(C(CC)=CC)=O)CCC(C2CN(C(=O)Cc3cc(C)ccc3C)C2)CC1 CCC(O)C(=O)NC(C1CCCCC1)CNC(c1cc(C(N)=O)c[nH]1)=O C1(CC(C)NC(c2cc(F)n[nH]2)=O)CCN(C(c2cn(C3CC3)nn2)=O)CC1 N1(C(c2c(C)nn(C(C)(C)C)c2)=O)CC(NC(=O)CC(C)C)CC(C)C1 N1(C(C2(CNC(C(CCC)C)=O)CC3(CC3)C2)=O)CC2CSCC2(C)C1 C(=O)(CCS(=O)(=O)N1CCOCC1)NCCNC(c1c(C(C)C)c[nH]c1)=O C(C(C)(C)C(=O)NCC1(NC(C2CCOC(C)C2)=O)CCOCC1)OC CC(C)CS(=O)(=O)CC(=O)NCCC(C)N(C)C(c1nccc(N)c1Cl)=O CCC(CC(C)C)C(=O)NC(CNC(C1CC2(CSC2)C1)=O)CO N1(C(CN(C2CCCC2)C)=O)CCCC(N(C)C(C2C3CCC23)=O)C1 C1(n2cc(C(C(C(=O)OCC)O)C)nn2)CON(C(=O)CCSC2CCCC2)C1 c1(NC(c2nccc(-c3cnc(OC)nc3)c2)=O)cc2c(C)snc2s1 c1(N2CCN(C(=O)NC(C(C)(C)C)CCO)CC2)ncnn2cccc12 c1(CC)oncc1C(=O)NCC1C=CCN1C(c1coc(Cl)n1)=O N1(C(C(=Cc2cccs2)C)=O)CC2CCCC2(NC(=O)CC2CNC(=O)C2)C1 C1(CNC(C=C(C)Cl)=O)CN(C(c2ncccc2OC(C)C)=O)CCCO1 N1(C(c2c(C(C)NC(C(C(C)C)SC)=O)noc2)=O)CC2(CCN(C)CC2)C1 C12(CNC(=O)C=Cc3cocn3)CC1CN(C(c1cnco1)=O)C2 Cc1ccc(C(N2CCC(N(CCO)C(c3cc(C)nc(C)n3)=O)C2)=O)c(C)c1 N1(CCNC(CCOCC#C)=O)CCCCC1.c1(C(C(=O)N)O)ccc(F)cc1 C1(CC=C)(C(=O)N(CCCC)CCO)CCN(C(c2cccn2C)=O)C1 C#Cc1ccc(C(=O)NC(C)(C)CCCNC(=O)CC2CCCCC2)cc1F c1(OC)ccc(O)c(Sc2cccc(CN(CC(=O)O)C)c2)c1.c1ccccc1 C1(NC(c2cc(C3CC3)on2)=O)COCC1NC(C1(O)CC1)=O N1(Cc2c(C(=O)OC)n[nH]c2)CCN(C(C2(c3cccs3)CC2)=O)C2CC12 C(=O)(C(C(=O)NCC1(Cc2ccc(Cl)cc2)CC1)c1ccccc1)OCC Cc1cnc(NC2CCCCC2N(C)C)c(S(=O)(=O)NCc2cn(C)nn2)c1 c1(C(=O)NCC2N(C)CCN(C(C(CSC)C)=O)C2)cc2nccnc2cc1C C(=O)(C1=CC(c2ccccc2)NC(=O)N1)N(C)CC1N(C(C2C(C)C2)=O)CCC1 C(=O)(CCCCC(C)CC)NC1(C(=O)Nc2ccc(CC)cc2)CSC1 C1CN(C(=O)Cc2csc(NC=O)n2)CCO1.N1(C(C)=O)CC(C(=O)NC)C1 c1(OC)cc(O)ncc1C(N1CCCC1C)=O.c1(CC(=O)N)c(F)cccc1F Cc1cc(C)c(C(=O)NC2CC(F)CN(C(=O)C(C)(C)CF)C2)c(C)c1 Cc1cc(C(=O)NCCCCCNC(=O)CCc2cncn2C)n(C2CCC2)n1 c1(C(=O)NCCC(CNC(c2[nH]c(=NCC)sc2)=O)(C)C)cnc2sc(C)cn12 c1(C2(C)CC2(F)F)ccc(C(=O)NCC(O)CC)cc1.c1(C(=O)N)csc(Cl)n1 C1(C(N2CC(C(=O)NC3CCC4(CC4)C3)(SC)C2)=O)CC2CC1CC2O c1(C(N(CCC)CC)=O)ccc2c(c1)SCCN2.C1(CC(=O)N)CCCC(O)C1 CCCCC(C(=O)NC1C2CC3C(C2)C13C(=O)N(C1CC1)C)NC(N)=O c1(NCC(CNC(c2cn(C)nc2)=O)O)nc(C2CC2)nc2c1CCC2 C1(C(=O)NC2CC(NC(C(CCC)CC)=O)C2)CCn2nccc2C1 c1(CC=O)cccc(F)c1F.c1(CC)cnn(CC(=O)NCC2(O)CCC2)c1 C1(NC(c2c(C)nc(C)o2)=O)CCN(C(=O)CC2CN(C)C2)CCC1CO C(=O)(CC1OCCc2ccsc21)NC(C)C(C)(C)NC(=O)CCC1CC(F)(F)C1 c1(C(C)C)ccccc1C(=O)NC1(CO)CCN(C(=O)C)C1.CCN(C)C.S O=C(CC1CCc2ccc(O)cc21)NCC1CC(NC(c2cc(Cl)no2)=O)C1 N1(C(CCCc2ccc(SCC)cc2)=O)CC(NC(=O)COC)CC2(CCC2)C1 C=CCC(CC=C)C(=O)N1CCC(=CCNC(c2cccnc2)=O)CC1 C(=O)(C(CCC)NC(c1ccc(Cl)o1)=O)NC1(C)CC(=C)C1 C(=O)(CN=S(C)(C)=O)N(CCCCCNC(=O)CSc1ccc(F)cc1)C C(=O)(CCC(C)(C)O)NCC1N(C(C(C)CF)=O)CCC1 C1(CC(=O)NC(C(=O)NCCc2n(C)cnn2)Cc2cc[nH]n2)CCCNC1=O C(c1cccnc1)=CCNC(c1c(CNC(COCCC=C)=O)cc[nH]1)=O CC(CCNC(=O)C(O)CCNC(=O)C(C)CO)C(F)(F)F C(C(=O)NC1CCCCC1F)(C(C)O)NC(Cc1c(C)non1)=O c1(OC)cccnc1C(N1CC(NC(C2(F)CCOC2)=O)C(O)C1)=O C(=O)(C(O)CCCNC(C1(CC)CCC1)=O)NC1CN(CC)C1 C(CCC(C)C(=O)N1CC(NC(c2scnc2C2CCCC2)=O)C1)OC CC(CN=c1ccnc(C2CCC2)[nH]1)NC(=O)CC1CCC(=O)NC1 CC(C)CC(CC(C)C)NC(c1cc(F)c(F)cc1Br)c1nnnn1C1(C)CC1 C12(C(NOC(C(=O)OC(C)(C)C)(C)C)=O)CNCC1CS(=O)(=O)C2 N=c1nc2c(c[nH]1)CC(C(N1CCC(NC(C3COCCOC3)=O)CC1)=O)CC2 S(=O)(=O)(c1ccc(N2CCCc3occc3C2)c(F)c1)NC(C=C)C1CC1 c1(OC)ccc(C(=O)NCCC(C)NC(C2CC23CCCC3)=O)c(N)c1F N1(C(c2c(C)c(Cl)cnc2)=O)CCC2CN(C(=O)Cc3ccsc3)CC2C1 N1(CCC2CCC(C)C2)CCN(C(c2ccc(C(=O)OCF)cn2)=O)CC1 C(N=c1ccn(CCCO)[nH]1)(c1cccc(C#N)n1)c1nnnn1CCCF c1(CNC(C(CCC)NC(=O)Cn2cnnn2)=O)cccc(C)c1C C(C)(C)(CC(=O)NCCOC1CCN(C(=O)CCC)CC1)OC.C(N)(=O)N c1(SC)ccc2c(c1)C(NCC)CCC2.C1(C=O)CCC(C(F)F)CC1 S(=O)(=O)(c1ccc(-n2cnnn2)cc1)NC1CC(C)(C(=O)OC)C1 C1(NC(C2C(C)OCCC2)=O)C(C)CCN(C(C2CC(F)(CO)C2)=O)C1C N1(C(c2[nH]c(=N)sc2)=O)C2CCC1CN(C(C13CC(C(F)(F)F)(C1)C3)=O)C2 C1(N=[N+]=[N-])(C(=O)NC(CC)(C)CC)CCN(C(c2cc(C)c(O)nn2)=O)C1 C12(NC(C3C(C)(C)C3)=O)CCCC(NC(=O)CCc3csc(=N)[nH]3)(C1)C2 c1(CC(N2CC(CNC(C3(C)CCC(=O)C3)=O)OCC2)=O)c(F)cccc1Cl O(N=C1CCCCCC1)CC(N1CCN(C(=O)Cn2cnnn2)CC(O)C1)=O C1(NC(Cc2c(C)cccc2C)=O)CCCC12CN(C(=O)CO)C2 N1(C(C(C)SCC)=O)CCCC(O)(CN(C)C(C2(C)CCCCCC2)=O)C1 CC1(C)CCOC(C(=O)NCCC2CN(C(c3c[nH]c(=N)s3)=O)CCCO2)C1 c1(C(=O)NC(CNC(C#CC(C)C)=O)CC(C)C)ccc2c(c1)COCC2 N1(C(C2CCN(C(CCC=C)=O)C(C)C2)=O)CCC(F)(F)C(C)C1 CCCCN=C(NCc1cc(Cl)cc(Cl)c1O)NCC(C)S(C)(=O)=O N1(C(=O)CCCC(F)F)CC23CCCCC2(C1)CN(C(=O)COC1CCCC1)C3 CC1(C)CCN(C(c2cccc(C#N)c2)=O)CC1NC(C1C(C)(C)C1(F)F)=O C(=O)(C(C)CC(C)(C)C)N(C1CCN(C(c2cnn(C(C)C)c2N)=O)C1)CCC c1(CC)oc2ccccc2c1C(N1CC(NC(=O)CS(C)(=O)=O)C2(CC2)C1)=O CCC(CC)(CC)C(=O)NCCOCCNC(C1CC1C1CCCC1)=O c1(CCC(=O)NC2C(NC(c3n(C)nnc3Br)=O)CCC2)ccccc1C#N C1(C)(C(=O)NC(COCC)C(=O)NCCOCCO)CC(C)=NO1 N1(C(C(CCC)NC(=O)CN2CSCC2=O)=O)CCCC(N=[N+]=[N-])C1 C(=O)(CCC1=CCc2ccccc21)N(CC(C)O)CC.C(=O)(C1=CC(C)(C)C1)N c1(CC)ccc(COC(C2(C(=O)N)CC2(C)C)=O)cc1.C1(F)CCC1.C C(=O)(CC(C)(C)CC(F)F)N1CC(C)C(C(=O)NOC)C1.c1c(O)ncnc1O c1(CCC)cc(C(=O)NC2CN(C(C3CCCCCC3)=O)C3CC23)cc(O)n1 c1(CNC(C)CCCCCl)cc2n(n1)CC(C)(C)CO2 C(=O)(C(F)CC(C)(C)NC(=O)C(O)CN1CCCC1)Nc1cc(C)ncc1 c1(NC(CN(C(=O)CCCN=[N+]=[N-])CCOC)=O)cnc(C)c(C#N)c1 CCCC(C)(O)CC(=O)NCCN(C(=O)C(c1ccc(F)cc1)CC)C1CCCC1 c1(C(=O)NC(CNC(c2c(F)cc(N)c(Cl)c2)=O)CO)cnc(O)c2ccsc12 C(C(CC)(CC)NC(=O)CC1CCC(C#N)C1)NC(CC=CCC)=O C(=O)(CC(C(=O)NC(C)CNC(C1(C(F)F)CCC1)=O)N(C)C)OC CC1N(C(C2(NC(C34C(=O)C5CC3C4C5)=O)CCC2)=O)CCCC12CCC2.C N1(C(CCC#CC)=O)CCCC(CCC)(NC(=O)COCC2CCCCO2)C1 C12(C(=O)Nc3c(SC)cc(O)cc3)CCCCC(=O)N1CCC2 C1(NC(c2cn3c(n2)SCC3)=O)CC(O)CN(C(=O)Cc2ccc(F)cn2)C1 Cc1nsc(Br)c1C(=O)NC1CCC(NC(=O)Cc2ccsn2)CC1 N1(C(c2cc(C(C)C)on2)=O)CCC(NC(=O)CC2COC3CC2C3)C(O)C1 C#CC1(C(=O)NCc2ncc(C)s2)CN(C(=O)CC(=O)Nc2nccs2)C1 CC1CN(C(c2ccc(C#N)o2)=O)CCC1NC(c1c(Br)cnn1C)=O C1(CNC(c2cnn(CC)n2)=O)CC(F)(F)CN1C(c1cc[nH]c1)=O c1(CNCC(CNC(C2(SCC)CC2)=O)F)cc2c(cn1)OCCO2 N1(C(Cc2c(COC)cccc2)=O)C2CCC1CC2.n1(CC(=O)N)cc(C)cn1 CC1C(NC(c2cc(C3(Cl)CC3)n(C)n2)=O)CCCN1C(c1ccc(O)nn1)=O S(=O)(=O)(c1nc(N2CCC(OCCCO)CC2)ccc1Br)N(C)Cc1ccns1 C1(C(N2CCN(C(c3ccc[nH]3)=O)CC2C2CCC2)=O)CC2CC(O)CC(C1)C2 c1ccc(Cl)c(O)c1.c1(CCN(C(=O)NC(c2cccnc2)C)C)ccccc1 CN1CCOCC1C(=O)NC1(C(=O)NCCCc2nccs2)CC1 C1(NC(c2c[nH]c(-c3ccccc3)c2)=O)CCN(C(C2(C(F)(F)F)CC2)=O)C1 c1(C(=O)NCC2(OC)CCSCC2)cc(Cl)c2ccncc2n1 N1(C(CCC2CCCN(C(=O)OC(C)(C)C)C2)=O)CC2CCC(C1)O2 c1(C(N2C(CCNC(c3coc(Cl)c3)=O)CCCC2)=O)c(O)cccc1O c1(OC)ncccc1C(N1CCCC(CNC(C2CC2c2cccs2)=O)C1)=O CCCCC(CC(=O)NCC(F)(F)COC)NC(=O)CN(C(=O)COC)C C(=O)(CCCCSC)N(C1CCN(C(=O)C(O)CC2CCCCC2)C1)CC N1(C(CCCCCOCC)=O)CCN2CCN(C(=O)CC3CCCCC3)CC2C1 C1(C(=O)NCC(COCC)C)CCN(C(=O)C(C)O)C(C)(C)C1 C#CC(C)(C)C(=O)NCC(CC=C)NC(=O)C(c1cccc(Br)n1)(F)F C1(C(N2CCC(NC(=O)NC)C2)=O)CCCCN(C(c2cnn(CCF)c2)=O)C1 N1(C(COCc2ccc(C)s2)=O)CCCC(N(C)CCC2CCC(=O)N2)C1C C1(NC(C2CC3CCC2C3)=O)CCCC12CN(C(c1cc(Cl)ncc1O)=O)C2 C1(CC(=O)N(CCCC=C)CC)CC(NC(c2ncccc2F)=O)C1(C)C c1(OC)ccc(CC#N)cc1NC(=O)Cc1ncccc1F Cc1cc(C(N2CCC(N(c3ncccn3)CCO)CC2)=O)cc2c[nH]nc12 C#CCC(CC(F)F)C(=O)N1CCC(C)(CC(N2CCC(CO)CC2)=O)C1 CCCCC(C)C(=O)NCC(CCNC(c1cc2n(n1)CCO2)=O)OC C(=O)(C(C)(C)C(F)(F)CC)NCCC(C)NC(C(CCC)C)=O C1(C(=O)NC(CC)C(C)(F)F)CCN(C(C2CC=C(C)CC2)=O)CCO1 c1(C(=O)NC(CCNC(c2cc(C)cc(C)c2N)=O)C)csc2c(Cl)cccc12 N1(C(COCC#C)=O)CCCC1(C)CNC(=O)COCc1ccccc1 [SH](=O)(=O)c1ccc(Br)cc1N(CCC(O)C(C)(C)C)C.C1(CC)(C)CCOC1.N C(=O)(C(C)(F)C(C)(C)F)NCC(C)NC(c1c(C)cns1)=O C1(NC(C2(C)CCC3CC3C2)=O)CCCCCCC1NC(c1cc(CO)on1)=O C=CC1CCCC(NC(C2(C)CCCN2C(=O)CCc2cscn2)=O)C1 C(C(C)(O)C(=O)N1CC2CC1(C)C2)OC.C1(C=O)(C(=O)N(C)C)CC1.N N(C(=NCCC(C)=O)N1CCS(=O)(=O)CC1)CCC1CC(OC)C1 Cc1c(C(=O)NCC2CC2)noc1C1CC1.C1(C=O)CC(n2cnnc2)C1 Cc1c([N+](=O)[O-])c(C(=O)NCC2CC(F)(F)CN2C(=O)C2=CCCS2)nn1C C1(NC(C=C(C)C)=O)CC12CCN(C(c1ccccc1C1(C)CC1)=O)CC2 n1(CC)nc(C(N2CCN(C(C3CC3(C)CC)=O)CC2C)=O)ccc1=O c1(NC(CC2(O)CCN(C(c3scc(C)c3)=O)CC2)=O)nc[nH]c2ncc(I)c1-2 C1(N(C(=O)CNC2CCCO2)Cc2ccc(-c3cccs3)s2)CCC(O)CC1 C1(CC#C)(C=O)CC=CCC1.C12CC(CN1C(=O)CC1(C=O)CC1)C2.N C1(NC(=O)COC2CCC2)CCN(C(C2CC(Cl)(Cl)C2)=O)C1 C=CCC(C(=O)N1CCN(C(c2cc(OC)no2)=O)C(CC)C1)C(C)C C(C(=O)N1CCC(C)CC1)(C(C)(C)C)NC(C)=O.C12(C=O)CC(C1)C(C)O2 C(=O)(C(O)C1=CCCCC1)N(C)CCN(C)C(C1CC1c1cccc(F)c1F)=O N1(C(CNC(=O)Cc2ccccc2)=O)CCN(C(C2CCCSC2)=O)C2CCC12 CC1(C)CC(C(=O)NCCOCCNC(C2CCC23CCC3)=O)CNC1=O N1(C(C(=O)NC)C)CC(C(C)(C)C)CCC1C(N1CCC(NC(C)=O)CC1)=O N1(C(C(CC2CCCCC2)OC)=O)CC2(CCCN(C(C3CCOC3)=O)C2)C1 C1(C2CC2)(NC(CN2CC(C)CC(C)C2)=O)CCC(=O)CC1 C1(C(N2CCC(NCc3ccc(O)cc3Br)C2)=O)CCC2CCC(=O)N2C1 c1(C(=O)NC23CC(NC(c4cc5ccccn5n4)=O)(C2)C3)ccc2nn[nH]c2c1 CCCC(CNC(C1CCCCNC1=O)=O)C(=O)NCCC(=O)NC(C)(C)C c1(CNC(=NC)NCC2(C(F)(F)F)CCC(=O)NC2)ccc(F)c(SC)c1 N1(C(C(COCC)(C)C)=O)CC2CC(NC(c3cn4ccsc4n3)=O)C1C2 CC1CCCC1(C)C(N1CCC(NCc2ccc(OC(=O)N(C)C)cc2)CC1)=O Cc1ccc(C(=O)CN2CCC(=CC(N3CCC3)=O)CC2)cc1.CC1CC1 CC1=NOC(=O)C1CC(=O)NCCCCCN(C(=O)C(c1ccccc1)F)C CCC(O)CN(C)C(C1CC(CCNC(=O)Cc2ccns2)C1)=O C(=O)(CC(C)CC(C)C)N1CCC(C(N(CC#C)CC2CC2)=O)(OC)C1 N1(C(CSCC(C)C)=O)CC(NC(=O)C=Cc2cccnc2)CC12CCCC2 C1(NC(c2ccccc2)=O)CCCCC12CCN(C(C1CC3(CC3)CO1)=O)CC2 Cc1cc(=NCc2cn(C3CCOC3)nn2)[nH]c(NC2CC3CCCCCC23)n1 N1(C(C2C(=C)C2)=O)CC(NC(c2ccc(Sc3ccccn3)cc2)=O)C(C)C1 N1(C(C2C(=C)C2)=O)CCS(=O)(=O)CC1(C)OC(F)(F)F c1(C(=O)NC(CNC(COCC(=O)NC)=O)CO)ccc2[nH]c(=N)[nH]c2c1 n1(C(C(=O)NC(C)COC(F)F)C)cc(CCC2(CCO)OCCO2)nn1 C1(NC(CC=C)=O)CCN(C(=O)CCc2ccc(Cl)s2)C(C2CC2)C1 CC1CCC(N(C)C(c2cn(CCNC(=O)C=CC3CCCN3C)nn2)=O)CC1 N1(CCC(=O)NCC(CN(C(C(CO)OC)=O)C)O)CCC(C)CC1 c1(C(C(=O)NCCC2CN(C(C=CSC)=O)CC2C)O)c(C)cccc1C N1(C(CC(c2ccc(C)cc2)NC(N)=O)=O)CCc2cc(O)c(O)cc2C1 N1(C(C2C(C)(C)C(=O)C2)=O)CCC(NC(=O)Cn2cnnc2)C12CCCC2 C1(NC(c2ccc(F)c(Br)c2)=O)CCN(C(c2cccs2)=O)CC1F n1(CC(N2CCC(NC(C(CCCC)O)=O)C2C)=O)nc2c(n1)CCCC2 c1(C(=O)NCC(C)C)ccc(S(=O)(=O)C2CC2)cc1.C12(C=O)CC(C1)C2 N1(C(C)(C)C)CCCC(C)(C(N2CC(C3(NC4CC4)CC3)C2)=O)S1(=O)=O CCC1=NOC(CC(=O)NC(C)CNC(=O)CCc2ccc(N(C)C)cc2)C1 C(CCC(C)C(=O)N1CCCCC1C(C)(C)CNC(=O)CCOC1CC1)OC CC(C)(C)CC(O)C(=O)N1CCC(CO)(CNC(=O)C(C2CCOCC2)F)C1 c1(C(=O)NCC(C)NC(=O)CC2CCC3CC23)cc(O)nc(N(C)C)n1 CC1CC(C)CN(C(C2CC3(C2)CN(C(=O)C=CCBr)C3)=O)C1 c1(CC=O)c(F)ccc(Br)c1F.CC1CC2(C(=O)NCC3CC3C)CC12 c1(C(N2C(C(N(C)Cc3n(CC)cnn3)=O)CC(C)C2)=O)ccc(C)c(O)c1 Cc1ccc(CC(N2CCC3(NC(C4CC(CF)C4)=O)CC3C2)=O)cc1[N+](=O)[O-] C#Cc1cc(F)c(C(=O)NCCC2CC2)c(F)c1.C1(C=O)CC(C2CCC2)C1 c1(C(=O)N)ccc2nc(C(F)(F)F)cn2c1.CCC(C)CNC(c1cccs1)=O c1(C(=O)NCCn2cncn2)nccc(-c2ccccc2F)n1 c1(C(NO)=O)ccc(CNC(C23COC(C2)C3)=O)cn1.C(C)(C)(C)NC.C c1(CCNC(C(c2ccccc2)C)=O)cccc(C(C)C)c1.C1(O)(C=O)CC1.N N1(C(C2(C=C)CCC2)=O)CCC(O)(C2(NC(=O)C(C)NC=O)CC2)CC1.N C1(CNC(c2ccn(C(C)C)n2)=O)CC(C(=O)N2CCCC(C(N)=O)C2)=NO1 c1cccc(F)c1.C1(C(C(=O)N)N(CC(C)(C)C)CC(C)C)CCCC1(C)C.C CC1(C)C(C=O)C1C(F)F.c1(C(N(CC)C)=O)cc(-c2ccco2)on1 CCC(C)CC(=O)C(=O)N1C2CCC1CC(CNC(=O)C=Cc1cnn(C)c1)C2 c1(NC(C2C(NS(CCC)(=O)=O)C2)=O)cc(OC)c(OC)cc1C(=O)O N1(CC(N2CCC(CCNC(C(C)CO)=O)C2)=O)C(=O)c2ccccc2C1=O Cc1ccc(C(=O)Nc2cccc(NC(C3(C)C=CCC3)=O)c2)c(C)n1 N(C1CCc2c(C(=O)O)cccc21)Cc1c(C)nn(C2CC2)c1 C1(NC(C(C)(C)C2CCCO2)=O)Cc2ccccc2C1NC(=O)CC1(CO)CC1 CCC(CCC(=O)NC1C2CC1CN(C(C1(NC(C)=O)CCCCC1)=O)C2)OC Cc1cc(=O)c(C(=O)NC)cn1C.C1(C)CCCN(C(=O)CN(C)C2CC2)C1 C(=O)(CC1CCc2ccccc21)NC(CC)CNC(c1cnn2ccn(C)c12)=O N1(C(c2c(CNC(C3C(OC)CCC3)=O)nccc2)=O)CC2CCC1C(CO)C2 CC(C)(O)C(C)(C)C(=O)NCC(O)CNC(=O)C(c1cccnc1F)(C)C N1(C(c2cc(C)ns2)=O)CCCC(NC(C2(C)CC2)=O)CC1 N1(C(C(C(C)C)SCC)=O)CC2CC1CCN2C(=O)COCCC(C)C N1(C(CC(CC=C)(C)C)=O)CC(C)CN(C(c2cnc3[nH]cnc3c2)=O)CC1C Cn1cnc2c(N3CCOC(CF)C3)nc(=NCc3cc(Cl)cc(Cl)n3)[nH]c12 Cc1cc(C(=O)NCC2CCN(C(=O)CC3CN(C)C3)CC2C)c(C)cc1Cl C1(CNC(c2cc(OC)cc(Br)c2)=O)C2Cc3ccccc3C12 C1(C)(C=O)CCCCC1.C=CCCCNC(C1(C(=O)OCC)CCC1)=O.N S(=O)(=O)(c1cc(F)cc(Br)c1)N1CC(C)(CC(=O)NC(C)CN(C)C)C1 N1(C(C(CC)Sc2nc(=N)[nH][nH]2)=O)CC(C2(NC(=O)CC3CCCC3)CC2)C1 c1(C(=O)OCCC(C)C(F)F)nc2ccccc2[nH]1 c1(C(N2CCCCC(NC(C=CCCC)=O)C2)=O)cc2n(n1)CCCO2 CCC(C(=O)NCC1CCCN1C)NC(C1CCCC1)=O Cc1cccc(Cl)c1S(=O)(=O)N1CCCCC1C(=O)Nc1c(C)ncnc1C Cc1ccc(C(=O)NCC(N2CCC(NC(c3cc(=O)n(C)o3)=O)C2)=O)cc1 CC1=C(C(=O)NC(C2CCCN2C(C2CC2C)=O)C)CCC1 C#CC(C)CN=C(NC1CCCC1)N1CCC2(CC1)CNC(=O)O2 C1(CC)OCCC1C(N1CC(N(C)C(c2cn(C)cn2)=O)C1)=O N1(C(c2ncc(C)cc2Br)=O)CCCC1C1CCCN1C(c1cc[nH]c1)=O c1(C(=O)NC2(COC)CCN(C(C3(C)CC=CCC3)=O)C2)ccc2n[nH]cc2c1 C1(CC(N2CCC(C(C)NC(=O)Cn3cc(Cl)cn3)C2)=O)CCCCC1O C(=O)(C(CCC(C)(C)C)N1CCC(C(O)C(N)=O)CC1)Nc1cccc(OC)c1 C(CC(C(=O)NC(COC)CC)NC(c1coc(C(N)=O)c1)=O)=CC N1(C(C(C)OC)=O)CCCC(O)(CN(C)C(c2cnc(CC(C)C)[nH]2)=O)C1 c1(OCCC(N2CC(NC(c3c(C)occ3)=O)C(C)C2)=O)ccc(Cl)cc1Cl Cc1csc(Cl)c1C(=O)NCCCC(CO)NC(=O)C(C)(C)c1ccccn1 S(=O)(=O)(c1cc(Br)c(Br)s1)N1CC(F)CC(NC(=O)CCCn2ccnc2)C1 N1(C(Cc2c(C)ncs2)=O)CC=C(CC(=O)NC(c2ccccc2O)C)CC1 CC(C)(C(=O)NCCNC(=O)Cn1cnc(Br)n1)n1ccc(C2CC2)n1 C1(C(=O)NCCOCC)CCOCCN1C(=O)CC1COC(=O)C1 C(CC(C)(C)C(=O)N(C1(C(=O)NC(C2CCCCC2)C)CC1)C)OC c1(C(=O)NC(c2ccc(OCC)cc2)CCC)c(C(F)(F)F)coc1C N1(C(c2c(C)ccs2)=O)CC2C(C1)N2C(C1CCCN1C1CCCC1)=O c1(C(=O)NC(CC)CN(C(=O)Cc2ccc(C)o2)C)ccc2c(c1)OCCO2 C(=O)(C(C#N)C(C)C)N1CCC(C(N2CC(N(CCOC)C)C2)=O)C1 Cc1csc2cc(C(=O)NC3CC(CNC(=O)C(CCO)N(C)C)C3)[nH]c12 C1(NC(CN(CCC#C)C)=O)CCCC12CN(C(C1CC3(CC(OC)C3)C1)=O)C2 CS(=O)(=O)c1ccsc1C(=O)NC1CC1NC(=O)Cc1ccc(F)cc1 [N-]=[N+]=NCCCCC(=O)NCC(O)CC(=O)NCC(c1ccsc1)O C1(N(CC(C)C)C(=O)C)CCN(C(C2CCOC2)=O)CC1.C1CC(F)(F)C1.O C(=O)(CC1OCc2ccccc21)NCC(C)NC(c1ccc([N+](=O)[O-])cn1)=O C1(C2CCN(C(c3[nH]c(C)c(C(C)=O)c3)=O)C2)CC1.C(C=O)OCC#C.N C1(CNC(c2onc(C)c2C)=O)CC2(CCC2)CN1C(=O)C#CC1(C)CC1 n1(CC)cnnc1C(=O)NCC1CCC(NC(=O)CC2(O)CCCC2)C1 N1(CC=C)C(=O)NC(c2sccc2S(N)(=O)=O)C(C(=O)OCC)=C1CC c1(CC)ccc(C(C)=CC=O)cc1.C(=O)(C(C)(C)CC(C)C)N(CCCC)C.N C(C)(CNC(=O)CCc1cnoc1)(CC(C)C)NC(CC1(OC)CCCC1)=O C(CN=c1[nH]c2cccc(Br)c2o1)C1CCC(NC(c2ccco2)=O)C1 c1(N2C(C(=O)OC(C)(C)C)CCCC2)c(F)cc(Br)cc1[N+](=O)[O-] C(=O)(CC1CCCc2oc(C)nc21)N(C)Cc1cccc(OC)n1 c1ccc(C(C)(C)C)cc1.C1(C=O)CCCC1.C1(N(C(=O)C)C)(C)CC1.N C1(C(N2C(CN(C(=O)CC3(O)CCCC3)C)CCC2)=O)CC1C1CCCCC1 C1(CCOC)(NC2(c3n(CC(=C)C)nnn3)CCSCC2)CCC(O)CC1 Cc1cc(C(=O)NC2CN(C(=O)CSC(F)(F)F)C(C)(C)C2)c(C)n1C C1(C(=O)NCc2scc(C#N)n2)CC(F)(F)CN1C(=O)C(C1(O)CCCC1)F C#Cc1cc(C(=O)NC2CCC(CCNC(=O)CC3=CCCC3)C2)ccc1C c1(Nc2cc(NCCCC(=O)N3CCOCC3)ncn2)cc2c(s1)CCC2 N(C(=S)N1CCNC(=O)C1C)c1ccc(C)cc1 C(=O)(C(CC)NC(=O)Nc1ccccc1)N1CC(NC(C=CCC)=O)C1 c1(C(=O)NC(CNC(C2CC(CC)(CC)C2)=O)CO)cc(C(C)C)ccc1C N1(C(C(C)C2CCC2)=O)CCC(C(N2CCC(CO)C2)=O)C12CC2 C(C)(C=O)(C(=O)N)OC.C12CC1CN(C(=O)Cc1cnoc1)C2.C(C)(C)C Cc1ccnc2sc(C(=O)NC(C)C(C)C)c(C)c12.C1(C=O)CC1.N(C)C.N N#Cc1ccc(C(=O)NCC2(F)CC(NC(=O)CC3CCCCC3O)C2)cc1 c1(C(N(CC(CC)NC(C2CC2O)=O)C)=O)cc2cc(OC)cc(OC)c2[nH]1 c1(COC)cc(NC(C2CCN(C(c3cc(C(C)C)on3)=O)C2)C)ncn1 C1(CC)CCN(C(c2cnc(C)[nH]c2=N)=O)C(C(=O)NCCCc2cccs2)C1 c1(C(N(C2CCN(C(C)C)C2)CCC)=O)ncoc1Cc1ccn(C(C)C)n1 N1(C(C2CC(=C)C2)=O)CCC(C2(O)CCN(C(C3CC34CCCC4)=O)C2)CC1 c1(OC)cncc(Br)c1C(N1CC(NC(=O)CSCC(C)C)C(O)C1)=O C(=O)(CC(C)N1CCCC1=O)NCCCN(C(=O)C(C)c1ccsc1)C(C)C CCCC(C)(O)CC(=O)NCC(C(=O)N1CC(n2cnnc2)C1)OC N1(C(C(C)OCCCCCC)=O)CC(CO)C2(C1)CN(C(=O)C1=CC(C)(C)C1)C2 c1(NC(=O)CC2CCCCC2NC(C23CCC(CC2)C3)=O)cccc2c1CCC2 CN1CCN(c2ccc(CN3CCN(C(=O)C=CCBr)CC3)cc2)CC1 C1(C(=O)NC(C2CN(c3nc(CC)nc(C)c3)C2)C)CCc2nc(O)[nH]c2C1 C(=O)(CC1OCc2ccccc21)NCC(C1CCC1)NC(c1cc(CC)on1)=O C1(NC(CCCSC)=O)CC2CC(NC(c3cc4n(n3)CCC4)=O)CC12 C1(NC(CCCOCC)=O)CC(C(=O)NCC2(OC)CCCC2)CC1O N1(C(C(C)(C)c2cnco2)=O)CC2(C1)SCCC2NC(=O)Cc1cccs1 Cc1cc(N2CC3CCCC2C3CNC(C2(C)C=CCC2)=O)ncc1C#N N1(C(C2CN(CC=C)C(=O)C2)=O)CCC2CC(C(N3CCCC3CC)=O)C2C1 O=C(C1CCc2ccccc21)NC12CC(C(N3CCCC3c3nn[nH]n3)=O)(C1)C2 c1(CC=O)ccc2c(c1)CCC2.C1(OCC(=O)N)CC(F)(F)C1.C1CCC1 C1(C)(C(=O)NCC(c2ccccc2)NC(CCCC#C)=O)CCC(OC)CC1 N1(C(C(c2c(C)ccnc2)(C)C)=O)CC(NC(c2cnn(C)c2)=O)CC(C)C1 C(C(C)N=c1[nH]nc(-c2ccccc2)o1)NC(c1ccc(C2(OC)CC2)cc1)=O N1(C(CCOCC)=O)CCCN(C(c2cccc(OC(C)C)c2F)=O)C(CO)C1 c1(C(=O)NC(C)C(N2CC3CC2(c2ccnn2C)C3)=O)ccc(Cl)cc1 CC1(C)CC(NCc2cn(C3CC(N4CCOCC4)C3)nn2)C(C)(C)O1 CC1(NC(=O)C2CC2)CC(NC(c2cnn(CC3CCC3)c2)=O)C1 Cc1[nH]c2ccc(Cl)cc2c1CCN(C=O)Cc1cc(C(F)(F)F)n[nH]1 C1(NC(c2c(CC)nn[nH]2)=O)CC2(C1)CC2.C(C1CCCC1)=C(C(=O)N)C C1(C(N2CCC(=CCNC(c3c(O)cccc3O)=O)CC2)=O)CCCC12CCC2 C1(c2n(Cc3occc3)nnn2)(NC2CC3CCC2C3)CCCSC1 C(CC(C)(C)CC=O)OC.C1(C(N(CC(C)C)C)=O)CCN(S(C)(=O)=O)C1.N c1(-c2ccc(C(N3C(C(=O)OC)C(C)CC3)=O)s2)c(F)cccc1F Cc1nn(CC(=O)N(C2CCC(NC(c3cc(Cl)no3)=O)C2)C)c(C)c1Cl c1(OC)ccc2[nH]cc(C(=O)N(CC(C)N(C(=O)C(O)CCSC)C)C)c2c1 CC(C)CC(C)CC(=O)NCC(C)N(C)C(c1cccnc1-c1cnn(C)c1)=O Cc1oc(S(=O)(=O)N(C)C)cc1C(=O)N.C1COCC1n1cc(C(=O)O)nn1 c1(C(N2C(C)CC(CNC(c3c(CCC)occ3)=O)C2)=O)cnn2c1CCC2 N1(C(C(C=C=C)C)=O)CC2CCC1C(CNC(=O)CCCSC)C2.C(C)(=O)N C=CC1(C(=O)N(CC2CCCCC2)OC)CCN(C(c2coc3c2COC3)=O)CC1 N1(C(C(F)=CC)=O)CCC(C(F)(F)F)C(C)C1.C(c1cncn1C)=CC=O N1(C(C2CCCN(CCC)C2)=O)CCN(C(C2CC(C#N)C2)=O)C2COCC12 c1(C=O)cc(F)ccc1Cl.C(C)(C(=O)N(C1CCCC1)CCC)OCC(C)C.N Cc1coc(C(=O)NCCCN(CCCCNC(=O)CC2CCCO2)C)c1C c1(C(=O)OC)cncc(NC(C2(O)CCN(Cc3cncnc3)C2)=O)c1 C(=O)(C1=CCN(C(=O)C(N2CCNC2=O)C)CC1)Nc1c(C)n(C)nc1 C=CCN=c1[nH]cc(C(=O)NC2CC(N(C(=O)C(C)CF)CC)C2)s1 Cn1ccc2c(C(=O)NCC(O)CNC(c3cnccc3Cl)=O)ncnc12 N1(C(C2C(C)(C)C2(C)C)=O)CCCC(F)(CNC(c2cnc[nH]2)=O)C1 C(C)(CNC(=O)CS(N)(=O)=O)(CC(C)C)NC(C(c1ccc(C)s1)C)=O C1(C(N2CCC(C)(CC)CC2)=O)CN(C(C2(CC)CC2)=O)CCC1(C)C c1(C(=O)NCC2(NC(CCC(C)SC)=O)CCC2)cc(F)cc(F)c1 C(CN=C(NCC(C)(C)C)NCC1CCOC1c1cnn(C)c1)NS(NC)(=O)=O c1(N(CC(=O)NCCOC)C)nc2c(c(=NC(C)CC(C)C)[nH]1)SCC2 Cc1ccc(NC(c2n[nH]cc2CNC(=O)CC2CCCCO2)=O)cc1Cl n1(CC(=O)NC(C)C)cc(NC(c2cn(C3CCOC3)nn2)=O)cn1 CC1(C)CC(C)(NC(=O)C2=CCN(C(c3ncc(F)cc3N)=O)C2)C(=O)O1 c1(OCC(=O)NC2CCCN(C(C=C)=O)C2)c(C)nn(C)c1C c1(OC)cc(C)c(NC(C2(F)CCN(Cc3cc(F)ccc3F)C2)=O)cc1Br c1(C(N2C(CNC(c3sccc3C)=O)CC(OC)C2)=O)ccn2ncccc12 CCCC(CCCS(C)(=O)=O)C(=O)N1CCC(NC(=O)CNC(=O)O)C(F)C1 c1(C(=O)NC2CC(CC(=O)OC)C2)n[nH]c(=NCC2(CO)CCC2)s1 N1(C(C(C)C2CC2)=O)CCC2(CCN(C(c3cc4ncccc4o3)=O)C2)C1 C1(CNC(C(=O)N(C)C)=O)CN(C(=O)CCO)CC(C)(C)C1.C1CC1.C N1(C(C2CCCCC2)=O)CCN(C(N)=O)CC2(CC2)C1.CC(C)(C)OC(=O)N c1(CC(CNC(c2c(Cl)cnc(CC)n2)=O)OC)c[nH]c2ccccc12 c1(C(N(C(C)CNC(=O)CC(C)C2CCCO2)C)=O)ccc2c(c1)NC(=O)NC2 C#CC(C)(C)C(=O)NCCC1CCC1.c1(C(=O)N)ccc(OC(F)(F)Cl)cc1 c1(COCC)nnc(COC2CCCCO2)n1C1CCCC1 CS(=O)CCCN=c1cc[nH]c(=NCCCc2cccnc2)[nH]1 N1(C(c2c(C)nccc2)=O)Cc2occ(C(=O)N(C)OCC(F)(F)F)c2C1 N1(C(c2n(C)c(Cl)nc2)=O)CCC2(CCC2)C(NC(=O)CCCn2cncn2)C1 C1(SC)CCCCN(C(C23CC(CN(C(=O)CCCOC(C)=O)C2)C3)=O)C1 C1(CC=C)CCN(C(C2CCCN(S(=O)(=O)CC)C2)=O)CC1.C(=O)(C(O)CC)N N1(C(C2C(CC)CCN2C(c2ncccc2O)=O)=O)CC(O)C2(CCCC2)C1 c1(C(N2CCC(NC(C=C(C)C(F)F)=O)(CF)C2)=O)cc([N+](=O)[O-])ccn1 CCCCCC(O)CC(=O)N1CCC1(C)CC(=O)N(CCO)CCOC c1(C(N(CC(C)C)CC)=O)[nH]ccc1CNC(=O)C=Cc1ccsc1 N1(C(CNc2ccc(N3CC(C)OC(C)C3)cc2)=O)CCC(C)C(F)(F)CC1 C(C)(CO)(C(=O)NC(CO)C(N)=O)NC(CCCOC)=O c1(CCC(=O)N(C(CNC(C(F)OC)=O)C)C)ccc(C(N)=O)cc1 CC(CC(=O)N1CC(CC(F)C(=O)NCC2(C)CSC2)C1)C(C)(C)C CC(C)CC(C)CNC(C1C(C)(C)C1(F)F)=O.C1(N(CC=O)C)CCCC1 CCCC(CCOC(C)CCCN(C)Cc1ccccc1)NC c1(C(N2CCCC(F)(C(N3C(C)CC3)=O)C2)=O)cccc2c[nH]nc12 CC(C)C(F)C(=O)N1CCOCC1CCNC(C1(C(F)F)CC(F)(F)C1)=O c1(C(N2CC(N(C(C(C)C3CC3)=O)C)C2)=O)ccc2oc(N(C)C)nc2c1.CO Cc1cc2n(n1)CC(C)CN2C(C1CCC=CCCC1)=O C(=O)(C(CO)C(C)(C)C)N1CC(CNC(c2c(F)ccc(C)n2)=O)N(C)CC1 C1(CC#N)CN(C(C2CNC(=O)C2)=O)CCN1C(=O)CCCCCl N1(C(c2cn(CCNC(c3c(C)nn[nH]3)=O)nn2)=O)C(C)CCCC1C c1(C(N2C(C)(C)C(NC(=O)Cc3ccco3)CC2)=O)cnc2[nH]cnc2c1 C1(NC(CCOCCC)=O)CN(C(c2ccc(C(C)(F)F)cn2)=O)C2CC12 c1(Sc2cccc(C)c2)ccc(NC(=O)CN(C(C)C)C2CC2)c(Br)c1 C1(CC=C)(C(N2CC(n3cccn3)C2)=O)CCCN1C(=O)CCCn1cncn1 N1(C(C2OCCN(C(C3C(C)(C)CCCO3)=O)CC2)=O)Cc2cccc(O)c2C1 c1(C(N2CCN(c3ccc(S(=O)(=O)NCC)o3)CC2)=O)cc2c(C)n[nH]c2cn1 O=C(C1=NOC2COCC12)NCCC1CC(NC(C2CC3C=CCC(C2)C3)=O)C1 Cc1nc(CS(=O)(=O)NC(c2cn(C(C)C)nn2)=O)no1 C1(N(C(c2cnn(-c3cccc(C)c3)c2C)=O)CCO)CCC(C)CC1C C1(NC(C(P(C)(C)=O)O)=O)CC2CCC(C1)N2C(=O)CSc1nc[nH]n1 c1(C(N2CC(NC(C3CCC(C)(C)C3)=O)C3(C2)CC3)=O)c(Cl)nc2ccccn12 C(C(C(=O)N1CC(n2ccnn2)C1)OC)OC.c1(C2C(C=O)C2)ccn(C)n1.N C1(CCCC)CCCN(C(=O)COC2CCN(C(c3cccs3)=O)C2)C1 N1(C(C2C(F)CCN(C(=O)OC(C)(C)C)C2)=O)CC(CO)OC2(CCC2)C1 CC(CCC(=O)N(C1CCCOC1)C)NC(C1(c2ccno2)CC1)=O C1(CCC)(NC(=O)C(c2cc(C)cc(C)c2)C)CCCN(C(=O)COC)C1 N1(C(C(CC)(C)O)=O)CC2CCCC2(NC(c2ccn(C(F)F)n2)=O)C1 c1(C(C)=O)cccc(SC(C2CCCCO2)C)c1 c1(C(=O)NCCCC(C)NC(C23CCCC2CCC3)=O)cnnc2ccccc12 N1(C(C(F)=CC)=O)CCCC1CCNC(=O)CNC(=O)N.C1CC1 N1(Cc2cc(OC)ncn2)CCC(NC(C2(F)CCCCC2)=O)CC1C N1(C(C2N(C(C(C)SC)=O)CC=C2)=O)CCCC(C)C1 c1(C(N(C(CNC(CCSCC(C)C)=O)C)C)=O)cnc(C2CCOCC2)s1 N1(C(c2c(C)nns2)=O)CC2(C1)CN(C(C1CCCN1N=O)=O)CCO2 Cc1c(C(N2CCCC(NC(C3CC4C(C3)C4(C)C)=O)C2)=O)sc2nnc(S)n12 c1(CC)cc(C(=O)NCC2C(C=O)C2(C)C)n(C)n1.CCCOC(=N)O c1(N(C)CC2CC2(C)C)nccc(N2CC3CC3C2)n1.c12noc(n1)C2 Cc1nccc(C(=O)NC2CC(NC(=O)C=Cc3cscn3)CC2O)n1 N1(C(c2ns[nH]c2=O)=O)CC2CN(C(=O)CC3CCC(C4CC4)O3)CC2C1 Cc1c(C(=O)NC2(CNC(=O)C3=CS(=O)CCC3)CC2)cnc2nncn12 N1(C(C2(C(C)C)N(C(CCC(=C)Cl)=O)CCC2)=O)CCC(=O)N(C)CC1 c1(C(N2CCN(C(C(C(=C)C)(C)C)=O)CC2C2CC2)=O)cc(C)[nH]c(=NC)n1 N1(C(CN(CCCCCC)C)=O)CC2C(N(C(=O)CC(=O)NCC)C)C2C1 C(CC(C(=O)NOCC1CCCCC1)NC(=O)C(F)C1CCCC1)=CC N1(C(=O)N)CC2CCCN(C(=O)C)C2C1.C1CCCC1.CC(C)(C)OC(=O)C C1(C(=O)NC2C(NC(c3ccn(C)c3)=O)CCOC2)CC(=O)NC(=O)C1 C1(COC)CC2(CCN2C(=O)NCCCc2nc(-c3ccncc3)cs2)C1 Nc1nccnc1-c1nc(CCC(F)(F)F)nn1-c1cccc(C(F)(F)F)c1 C1(N(C(C(C2CN(C(C(C)NC(CC)(C)C)=O)C2)OC)=O)C)CCC(CO)CC1 Cc1ccc(C(=O)NC(C)CNC(c2cccc(-c3ccncc3)n2)=O)c(C)c1 CCC(C(=O)NC(CNC(c1ccc2c(ccn2C)c1)=O)CO)C(C)(C)CC C1(CC(N2CC(CCC)C2)=O)CC1C1CC1.C1(CC=O)CC(C)C1.CC(C)C N1(Cc2ncn(C)n2)CCc2c(C(=O)Nc3oncc3C#N)n[nH]c2C1 N1(C(C)=O)CCCCC1CCC(N1CCCC1CF)=O C(=O)(C1=NN2CCCN=C2N1)N1CCC(=CCNC(CSS(C)(=O)=O)=O)CC1 N1(C(CSC(C)=O)=O)CCC(C)(NC(C2CCC(C(F)(F)F)CC2)=O)C1 Cc1cncc(NNC(=O)NNC(=O)C2CCOC2C(C)(C)C)c1 c1(C(N2C(C)CC(NC(c3c(Cl)nn(C)c3Cl)=O)C2)=O)nnc2ccccc2n1 C1(CC(N2CC3CC3C2)=O)COCCN1Cc1sccc1Cl CC1(NC(=O)Nc2ccc(-n3cccn3)cn2)COc2ccccc21 C1(C(=O)NC2CN(C(C3CC(=O)NCC3)=O)C2)Cc2ccccc2CO1 C1(C(=O)NC2C(C)CN(C(c3cnc(Cl)cn3)=O)C2)CCCNS1(=O)=O C1(C(N2C(C)CC(NC(c3c(C)nc(CC)o3)=O)C2)=O)CC(=O)NC(=O)C1 C=CCC(CNC(=O)Cn1ncnn1)C(=O)NCc1cc(OC)ccn1 N1(C(C2CCN(CCC#C)CC2)=O)CCN(C)CC1CNC(C1COC1)=O c1(C(C(=O)NCC)N(C)Cc2nc(CC)sc2)cc(C)n(C)n1.C1CC1.O C1(F)COCCN(C(c2n[nH]cc2C(C)C)=O)C1.C(C(=O)N)N(CC)CC.C CC(CC(=O)NCCC1CC(NC(=O)C(C)SC(C)C)C1)N1CCCC1=O N1(c2cc(NCC3(CC)CCOC3)ncn2)CCN2C(=O)C(C)CC2C1 C(=O)(C(CC)(CC)OC)N1CC(NC(C(CCC)NC(N)=O)=O)C(F)C1 C(=O)(CC(C)C(F)F)NC1C(NC(CC2(OC)CCCCC2)=O)COC1 c1(C(=O)NC2CC(C(NOCCCC#C)=O)OCC2)cc(F)ccc1O C1(C(N(C)CCNC(=O)COC2CC2(F)F)=O)(C(F)F)CCCCC1 N1(C(CCCCC#N)=O)CCCC2(CCC(O)C2)C1 CN1CCCN(C(=O)Cc2cnc(-c3ccccn3)nc2O)c2cc(Cl)ccc21 N1(C(c2ccc3ocnc3c2)=O)CCCC(C2CC2NC(=O)C(F)(F)C(F)F)C1 Cc1ccc(OCC(=O)NCC2(F)CC(C)C2)cc1.C1(CC=O)CCCO1 CC1CCCCN1CC(N1CCOCC1C(=O)NC1CC(=O)N(O)C1)=O C(=O)(C1SCCc2ccccc21)N1C2CC(CNC(C3(OC)CCC3)=O)C(C2)C1 C1(C(N2CCC(C)(NC(=O)C(=C3CCCCC3)F)C2)=O)Cc2cc(F)ccc2O1 c1(OC)ccc(-c2ccc3c(c2C(=O)Nc2nccnc2OC)CC3)cc1C#N Cc1cc(C)c(C(=O)NC(C)CNC(C2(F)CCC(=O)CC2)=O)c(C)c1 c1(C(=O)NC2CCN(C(C3CCC(C)C3)=O)C2)ccc(C(=O)N(C)C)cc1 Cc1nn2c(C)cccc2c1C(=O)N(C)CC1CC1.c1(C(=O)N)ccc(C)n1C C1(NC(C(CC)(C)CC)=O)CC2CCC(C1)N2C(c1cccc(C#N)c1Br)=O C1(C(=O)NCCCNC(C(C)(C)c2ncco2)=O)CC(=O)NC(=O)N1 N1(C(C(C)OCCC(C)C)=O)CC2CN(C(c3cnn4c3N(C)CC4)=O)CC2C1 N1(C(C(C)C2CCCC2)=O)CC(C)(CNC(=O)C#CC(=O)N(C)C)CC1(C)C c1(C(N2CCCC(C(C)NC(c3[nH]nc(OC)c3Cl)=O)C2)=O)csc2nccn12 C(c1ccoc1)=CC=O.C(=O)(CC)N(CC)CC.C(=O)(C=CCC)N N1(C(C(F)=CCC)=O)CC2(C=C(C(=O)NCc3coc(C)n3)CO2)C1 N1(C(CC(n2c(CC)ncc2)C)=O)CCC(NC(=O)CCO)C(O)C1.C(N)=O.N Cc1ccc(CCCNC2CC(O)C2n2cccn2)cc1 C12(C(=O)NCC(n3ccnn3)C)CC(CO1)N(C(C1CCCC(O)C1)=O)C2 C(=O)(CC(F)(F)C(F)(F)F)N1CC(CCC)N(C(C2CCOC(CC)C2)=O)CC1 c1(C(=O)OCC)nnc(S(=O)(=O)N2CCOC(CO)C2)s1 c1(C(=O)NCC2(NC(c3cc(F)ccc3F)=O)CC2)cc2c(o1)CCCC2 C(C1CCCCC1)=CC(=O)NCCC1CCOC1.C1(CC=O)CS(=O)(=O)C1 c1(CC(=O)NC2C(NC(C3(OCC)CCC3)=O)C2)nccn1C c1(OC)ccc(C(=O)NCC2CCCN(C(c3cccnc3F)=O)C2)c(F)c1 c1(C(=O)NCC23OCC(NC(C4(C)CC4)=O)C(C2)C3)ncc2ccccn12 c1(N(CC(C(=O)NC)C)C)nnc(-c2c[nH]nc2C)n1CCc1ccccc1 N1(C(C(N2CCCC(C)C2)=O)=O)CC2CN(C(c3cc(F)n[nH]3)=O)CC2C1CO N1(C(c2ccoc2)=O)CCN(C(=O)CC23CC(C2)C3)C(CO)C1 c1(C(=O)NC(C2CN(Cc3ncc(C(C)(C)C)o3)C2)C)cc2ncccc2[nH]1 N1(C(CC2N(CC)CCC2)=O)CCC(C2(NC(C3CC(O)C3)=O)CC2)C1 c1(OC)cccc(C(C)C=O)c1.C12(C=O)CC(CC(F)F)(C1)C2.C1CCC1.N c1(CNC(C2C(CC)C2)=O)ccc2c(c1)CCC2NC(c1nnc(C)s1)=O CC(C)(C)CCC(=O)N(C(C(=O)N)C1CC1)C1CC1.C(C1CC1)C1CC1 C(=O)(C(C)(C)C(C)(C)O)N1CC(OC)(CNC(c2coc(Cl)n2)=O)C1 C1(NC(c2cn(CC)nn2)=O)CC2(C1)CC2C(=O)NCCc1nccs1 C(=O)(C1c2c[nH]nc2CCC1C)NCC1CC(NC(C2CN(CC)C(=O)C2)=O)C1 C1(CN(C)C(c2cncn2C)=O)CN(C(C2CCCCS2)=O)CCO1 Cc1c(F)ccc(C(N2CCC(CO)(CNC(=O)C(C)(C)O)C2)=O)c1C C1(=CC(=O)NC2CCCC(F)(F)C2)OC(=O)N2CCCCC12 N1(C(c2ccccc2)=O)CCOC2(C1)CN(C(=O)Cc1cc[nH]c1)C2.CCOC C#Cc1cccc(C(=O)NCC(F)CNC(C2(C3CCC3)CC2)=O)c1Cl C1(C(N(CCC(C)NC(=O)CC23CCCC2C3)C)=O)CC(=O)C1C C=C1COc2c(C(N3CCC(C)(CNC(C4(O)CCSC4)=O)C3)=O)cnn2C1 CC1CCN(C(=O)C(C2CCCCC2)O)CC1NC(=O)C1=NOC(C)C1 CC1(C)C2CCC(NC(C3(F)CCN(C(C4CC4(Cl)Cl)=O)C3)=O)C1C2 C1(c2cn(CC(C)NC(=O)OC)nn2)CCCN(C(c2cncc(Cl)c2)=O)C1 c1(N2CCC(N(C(=O)CC)CC#C)CC2)cc(C)nc(C(C)(C)C)n1.C(N)=O C(=O)(C(N=[N+]=[N-])C(C)C)N1C(CNC(C(CCOC)C)=O)CCCCC1 c1(OC)cc(CCC(=O)NC2CCC2CNC(c2cnn(C)c2)=O)ccc1F CCC(CC)C(C(=O)NCC1(C)CCN(C(=O)C(C)(C)O)CC1)OC c1(N(C)Cc2nnnn2Cc2ccccc2)nnc2c(c1C#N)CCC2 N1(C(C(COC)OC)=O)CCCC(C)(NC(c2ccc(OC)cn2)=O)C1 c12ccc(cc1Cl)NC2.CC(CO)C(CNc1nccs1)C1CCC1.C1C(=O)N1 N1(CC2CN(C(c3nn[nH]n3)C)C2(C)C)CCN(c2cccc(C(N)=O)c2)CC1 C1CN(C(=O)Cc2ccc(F)cn2)CC1C(F)(F)F.C(F)(C(=O)NC)OC c1(C(=O)NC2C(NC(c3nc(CCCCC)sc3)=O)CCC2)cccc(SC)c1 Nc1ncc(C(=O)NCC2CCC(CNC(c3cncs3)=O)CC2)cc1O N1(C(C(=O)N(C)C)=O)CCCCC(NC(=O)C(C2(O)CCOCC2)(F)F)C1 N1(C(C(n2ncc(C)c2)C)=O)CC2(CCC(NC(c3ccccc3O)=O)CC2)C1 C(=O)(CC(C)(C)CS(C)(=O)=O)NCCCNC(c1n(C)nc(C)c1Br)=O C1(C(N2CCC(NC(=O)NC)C2)=O)(C=O)CC2(CC2)C1.C1CCCC(O)C1 Cc1cc(Cl)cc(C)c1OCC(N1CCCN(C(C2CCC(=O)O2)=O)C(C)C1)=O c1(OC)cc(C(N2CCCC(C)C2)=O)c(F)cn1.c1(C(=O)N)cc(N)c(Cl)cn1 C1(C(=O)NCC(CC)(C)NC(c2cncc(OC)n2)=O)CC(=O)N(C)C1 C#Cc1cnc(C(N2CCC(NC(c3oc(CC)cc3C)=O)C2C)=O)c(C)c1 CC(C)C(O)C(C)C(=O)N1CC(N(C)C(c2cnc3ccsc3c2)=O)C1 N1(C(COc2c(OC)cccc2)=O)CCN(C(=O)CN(C)C2CC2)C(C)CC1C c1(CCC(=O)OCc2cc(Br)nn2Cc2ccccc2)c(Br)nc2n1CCCC2 Cc1cc(NC(C2(C)CCCN2C(c2ccnc([N+](=O)[O-])c2)=O)=O)cc(Br)c1C C1(NC(c2c(SC)csc2)=O)CC(C)N(C(c2ccccc2N2CCCC2)=O)C1 C1(NC(C2(C)CCN(C)C2)=O)CC2CC1N(C(=O)CCc1nc(=N)[nH][nH]1)C2 n1(C(C(=O)NCC(CC=C)NC(=O)CC=O)C)c(C)cc(O)cc1=O.C1CC1 c1(C(=O)NCC2N(CC(CC)OC)CCCC2)cc(=O)c(OC)c[nH]1 c1(OCC=C)c(C(=O)NC2CCC(CNC(=O)C(C)CO)C2)cccc1C c1(CCC(N2CC3C(N(C(C=COCC)=O)C)C3C2)=O)cc(C)cc(C)c1 C(=O)(C#CC1CC1)NC(C)CC(C)NC(=O)CNC(N1CCCC1)=O c1(OC)ccc(OC)c(CCNCCCc2cnn(C)c2)c1 C(=O)(C1CCCc2sccc21)NC1CC(CNC(=O)COc2ccon2)C1 C1(C(N2C(CC)CCC2C)=O)CC2CC1CN(C(=O)COCCSC)C2 c1(CCC(=O)NC(CNC(c2ccc(COC)[nH]2)=O)C)c(C)nn(C)c1C C1(CCNC(=O)C(=O)NC(C)C)(OC)CN(C(C2CCC(C)C2)=O)C1 c1(C(N2CCN(C(C3C(=C)C3)=O)CC2C)=O)cc(=O)n2ccccc2n1 Cc1cc(N2CC(C)(NC(c3oc(C(F)F)cc3C)=O)C2)nc(-c2cccs2)n1 C1(C(=O)NCC(CNC(C(C)=C2CCC2)=O)O)CC(=O)CC(=O)C1 c1(N2CCCC(C)(NC(COCCC)=O)C2)ncc2c(Br)cccc2n1 c1(C(=O)Nc2cc(C(C)C)on2)ccc(C(=O)N(C)C)cc1 N1(C(C=C(CC)CC)=O)CC(=O)CC1C(=O)NCc1ccncn1 N1(C(COCCC#C)=O)CCCN(C(c2cnc(Cl)cc2N)=O)C(CO)C1 C1(CC(=O)NC2(CCNC(CN(CC)CC)=O)CC2)CSCCS1 C1(C(=O)NCC#C)CCCN(C(c2ccc(OCC)nc2)=O)C1 C1(C(=O)NCC2CCC(NC(C3C(=C)C3)=O)CC2)CCn2cc(C)nc2C1 c1(C(=O)NC(CNC(CCSCCCC)=O)(C)CSC)cc(O)ncc1F c1(OC)cnc(C(=O)NC(CNC(=O)CCOC)CO)nc1.C1CCCO1 c1(C(CO)NCc2ccc(C(C)(C)C)cn2)ccc(Cl)cc1F c1(NC(=O)NCC(c2cc(F)cc(F)c2)C)ncc2c(n1)CNC2=O C1(CC)C(NC(c2cccc(C#N)c2)=O)CCCN1C(=O)CN1CCCCC1C C(C)(C)(CC(=O)NCC(C)(CO)NC(=O)CCC(=O)c1cnn(C)c1)SC C=C(C)CC(C(=O)N1CC(F)C(F)C1)NC(C1CCCN(CC)C1)=O C(CCC1CC1)(C(=O)NCC1(CO)CCOC1)NC(=O)Cn1cc(Cl)cn1 N1(C(C(CC2CC2)OC)=O)CC2C(NC(c3csnn3)=O)CS(=O)(=O)C2C1 CC1CC(NC(c2cc[nH]n2)=O)CCN1C(c1ccc(OCCF)cn1)=O C1(NC(C=CCC)=O)C2CC3C(C2)C13C(N1CCC(C)(CCO)CC1)=O C1(N(CCC)C(c2cnn(C)n2)=O)CCN(C(=O)C(C)=CCN(C)C)C1 Cc1cc(N)cnc1C(=O)NC1CCCC(N(C(=O)CCCn2ccnn2)C)C1 Cc1cncc(C(=O)NC2CC2NC(=O)C(C)CN2CCCCC2)c1C n1(CCC(=O)N)ccc(O)nc1=O.C1(C(=O)NCC(O)C)(COC)COC1 N1(C(CCC(=O)NCCC)=O)CC(C)(C(N2CCCC(C(F)F)C2)=O)CC1(C)C Cc1cccc(C2C(C)CN2CC(=O)N(C2CCNCC2)C2CC2)c1 Cc1cc(C2CC2)ncc1C(=O)NC.C1(F)CCN(C(c2cnc(S)nc2)=O)C1 CC(C#N)C(=O)NC(C(=O)NCCCn1cccn1)C1(O)CCC1 Cc1ccc(S(=O)(=O)N(CC(=O)NCCC(N2CCS(=O)CC2)=O)C)cc1 C(=O)(C(F)(F)C(C)(C)O)N1CCC(CCCNC(CSc2n(C)nnn2)=O)CC1 c1(CC)nc(C)oc1C(N1CCCC1C(=O)NCc1nccn1C1CC1)=O C1(NC(CCCN(CCC)CCC)=O)CCN(C(C2(C(=O)NC)CC2)=O)CC1F c1(C(N2C(CN(C(=O)C3=CCC3)C3CC3)CCC2)=O)cnc2ncccn12 C#Cc1cc(C(=O)NC2C=CCN(C(c3cc(OC)cc(F)c3)=O)C2)ccc1C n1(CC)nc(C(=O)NC23CCCN(C(C4CC(C)C4)=O)C2C3)ccc1=O C(=O)(NNC(=O)C(C)NS(=O)(=O)c1cccs1)N1C(CCC)(CO)CCC1 CCC(C)C(=O)N(C(C)C(=O)NCc1nccn1C)CC C1(CNC(=O)C=C2CCCCC2)CN(C(=O)CC2COCCO2)CC12CCC2 c1(C(=O)NCC(CCOC)NC(CC(C=C)(C)O)=O)cc(C)cc2c1OCC2 Cc1nn(C)cc1C(=O)Nc1ccccc1.C12(C(=O)N)CCCC1(C(N)=O)C2 Cc1nc2c(o1)CCCC2CC(=O)NC12COC(CNC(=O)C3=COCC3)(C1)C2 C1(C2CCC2)(C(N(CCC)C)=O)CCC1.C(C(=O)NCC(=O)N)NC(C)=O c1(C(N2CCN(C(c3c(CC)[nH]nc3Cl)=O)C3C2C3)=O)onc2ccccc12 C1(NC(CCN(C)CCO)=O)COC2(C1)CN(C(=O)CC1COC(=O)C1)C2 C1(NC(Cn2ccc(C)n2)=O)C2CCC(C2)C1C(=O)N(C)Cc1cc(C)on1 c1(OC2CC(C(=O)OC)(CF)C2)ccc(-n2nnnc2C2CC2)cc1 C1(C(C)(C)C)(CNC(c2nncs2)=O)CCN(C(C2CCC3CC3C2)=O)C1 c1(C(=O)Nc2c(C(=O)Nc3ccnnc3O)scc2)n[nH]c2c(F)cccc12 Cc1ccc(C)n1CCC(=O)N(C1CN(C(=O)CC2(C)CCCC2)C1)C C1(NC(CCC2(C)CC2)=O)CCN(Cc2cn(C(C)C(=O)N3CCCC3)nn2)CC1 c1(-c2n(C(C=C)C)nc(COCC)n2)nccc2c(Br)cccc12 Cc1ccc(NC(=O)C(=O)ON2CCOCC2)cc1.c12sccc1C(=O)O2 C1(NC(C(c2cccc(C)c2)C)=O)CC12CCN(C(=O)CC(C)C(F)F)C2 N1(C(CC(C=C)(C)C)=O)CCC2(CC1)COC(C)O2 c1(OC)ccn2ncc(C(=O)NC(C)C(n3cc(C)cn3)C)c2c1 N1(C(=O)NCCN2CCC(O)CC2)CCC(C2CCCC2)C1 N1(C(Cc2cn(C(C)C)nc2)=O)CC(N(C(=O)Cn2[nH]cnc2=N)C)C(C)(C)C1 Cc1ccc(C(=O)NC(C)CCCCNC(c2cncc(C3CC3)c2)=O)c(F)c1 c1(OC)ccc(CC(=O)NC(C)C2CC2)c(F)c1.C(=O)(C(O)C(F)(F)F)N C1(C(=O)NCC2(CC)CC2)CCC(C)(C)N(C(c2ccc(Cl)o2)=O)C1 c1(C(N2CCCC(N(C)C(C3CC(F)C(=O)N3)=O)CC2)=O)cccc2nncn12 CCCC(CNC(C1(COC)CN(C(=O)Cc2ccn(C)n2)C1)=O)OC N1(C(C(CCOC)C)=O)CCCCC(N(C(=O)CCc2nc(C(C)C)no2)C)C1 Cn1cc2c(C(=O)NC3CN(C(=O)CCC(F)(F)F)CC34CC4)cc(F)cc2n1 C(c1cnccn1)=CC=O.C(=O)(CCOC(C)C)N(CCCC)CCOC C1(NC(CC2CCCC(=O)N2)=O)CCCC12CN(C(=O)C(=O)NCC1CC1)C2 C=CCCCC(C(=O)N1CC(C(C)(C)O)C1)NC(c1nonc1C)=O C1(N(C(C(F)=CC)=O)CC)CCN(C(C2(C)CC=CC2)=O)CC1 c1(C(=O)NC(CC=C)CNC(=O)CSCC(N)=O)onc(OC)c1Br c1(C(CCC)C)nc(C(F)CC)n(-c2ccccc2C(F)(F)F)n1 C1(NC(CC(CCC)C)=O)CC2(CCN(C(c3cncc(O)c3)=O)C2)C1 c1(C(C)=O)c(NCC2CCC(NC(c3ccc(F)s3)=O)C2)ncnc1Cl c1(N(C)C)ccc(C(N2CCC(CNC(C34CCC3C4)=O)C2)=O)cc1F c1(OC)ccnc(-c2nc(Cc3cc(C(C)C)no3)n(CC3CCCOC3)n2)c1 C1(NC(CCC2CC(NC(CCC(=O)NCCC)=O)C2)=O)CC(C)CCC1O c1(C(=O)NCC2C(C)CCN(C(c3ccc(O)cc3)=O)C2)cn2ccncc2n1 CCC(CCCC(=O)N(CCOC)C1CC1)NC(c1ccc(C)c(O)n1)=O CC(CCC(C)(C)C)C(=O)N1CCC2C(NC(=O)C(O)c3ccsc3)C2C1 c1(C(=O)NC2C(NC(c3cccc(C#N)c3)=O)C2)[nH]cc2c1CCS2(=O)=O c1(C(=O)N)ccccc1.c1(OCC)ncc(C(=O)NC(C)C)s1.CC(C)C c1(C(N2CC3C(C3)C2)=O)c(C(F)(F)F)nn(C)c1C.CCC1=NOC(C(=O)N)C1 N1(C(C2CCC(C(=O)OC)C2)=O)CCCC(C)C1.c1(C=O)ccc(Cl)c(Br)c1.N CC(C)CCC(F)C(=O)NC1CC(O)C1CC(=O)NC(C)(C)CC(N)=O Cc1cnn2ccc(C(=O)N(CC(O)CNC(=O)CS)C)nc12.c1n[nH]c(O)n1 c1(C(=O)NC(CN(C(CCCC(CC)C)=O)CC)C)ccc(SC)c([N+](=O)[O-])c1 c1(C(=O)NCCC2CCN(C(C(C)O)=O)C2)ccc2ccccc2c1 C1(F)(CNC(C2(CC=C)CCOC2)=O)COCCN(C(=O)C(N)=O)C1 N1(C(c2cnc(SC)[nH]2)=O)Cc2cccc(CNC(=O)CSC3CC3)c2C1 C1(CSC)CCC(NC(=O)CC2CC(NC(=O)OC(C)(C)C)C2)C1 c1(C(N(CCC)CC)=O)cc(C)nc(Cl)c1N.C1(C(=O)N)CCOC1C(C)C C(=O)(C(F)C(C)(F)F)N1C(CC)C(C(=O)NCc2ccc(C)s2)CC1 C1(C(N(CC(O)CF)C)=O)CC2(CC(NC(=O)CCc3cn(C)cn3)C2)C1 N1(C(c2scc(C)c2C)=O)CCCN(C(C2CC(CC(F)F)C2)=O)CC1C c1(C(N2CCC(F)(CNC(c3nc(C)sc3)=O)CC2)=O)ccnc2cc[nH]c12 Cc1cc(C(C)C(=O)NCC2CCC(NC(c3ccno3)=O)CC2)c(C)o1.C C1(O)(CCNC(C2(C)C=CCCC2)=O)CCCN(C(c2ccc(=O)oc2)=O)C1 N1(C(Cc2ccn(C)c2)=O)CCC(C(=O)NC2CC(CO)C2)(CO)C1 c1(NC(c2cncc(-c3cn(CS(C)(=O)=O)nc3)n2)=O)ccc(Br)cc1OCBr Cc1ccc(C)c(NC(C2CC2)=O)n1.c1cccc(C2(C(F)(F)F)CC2)c1.C C1(CN(CC(C)C)C)CCCN1C(=O)C(C)(C)C.C1(C=O)CC1.C1CC1 CN1CCCCN(C(C2(n3cc(CC4CCCCC4O)nn3)CC2)=O)CC1 Cc1c(C=O)cnn1C(C)C.C1(C(N(CC)C(C)C)=O)C(C)(C)C1(F)F N1(C(C=C(C)c2ccsc2)=O)CCCCCC(NC(c2cnc(S)n2C)=O)C1 c1(C(N(CCC(C)NC(=O)C(N2CCN(C)CC2)C)C)=O)nc(=N)cc[nH]1 c1(OCC(=O)NCC2CCCCN2C(C2CCCSC2)=O)ccc(F)cc1O C1COC(C)(C)CN1C(C1C(C)C1C)=O.c1(CCC)nc(C)c(C(=O)N)s1.C N1(C(c2cc(COC)on2)=O)CCN(C)CC1C.c1(C=O)c(C)ncnc1O.N CCCC(O)(CCC)CC(=O)N1CC(NC(C2CCCN2N=O)=O)CC1C Cc1c(C(=O)NC(C2CC2C(=O)NC2CN(C)CC2C)C)nnn1C N1(C(C(F)=CCC)=O)CCC(NC(C2CN(C)C2)=O)C(F)(F)CC1 CC1CCCCCC1N=c1[nH]c(=N)[nH]c(=NCc2cccc(F)c2Br)[nH]1 C(=O)(CCC(F)(F)Cn1cc(CCC#N)nn1)N(C)Cc1ccc(OC)cn1 C(=O)(C(C)(CO)CO)N.c1(OC(C)C)ccc(NC(=O)Cc2ccccc2)cn1 C1(NC(CSCc2nc(C)sc2)=O)CCOCC1.c1(C(C(=O)N)=O)cccn1C N1(C(C(=O)OCC)=O)CC2CCC1CN(C(c1csc(=N)[nH]1)=O)C2 CCC(CC)C(=O)NCC1CCCC(NC(c2[nH]ncc2C#N)=O)C1 CCCC(F)C(=O)NCC(C(=O)NC1CCS(=O)(=O)C1)N(C)C C1(NC(c2cnc(OC)nc2)=O)CC2CCC(C1C)N2C(c1cccc(C)c1)=O c1(OC)cncc(C(=O)NC(C)C(C)C)n1.C(=O)CCC(=O)N(C)C(C)C.N C1(CC(=O)NCCC2CCCC2O)CCCCN1C(c1ncoc1CO)=O c1(OC)cc2cc(-c3nc(CCO)nn3-c3c(C)noc3C)sc2cc1OC c1(C(N2CCOCC2)=O)cccn2c(O)nnc12.C1(C(=O)NC)(SCC)CC1 C(=O)(C1=CCCOC1)NC12CC(CNC(C3C(C)CCCC3)=O)(OC1)C2 C1(CNC(CCC)=O)CC(NC(c2cc(C(N)=O)no2)=O)CCO1 C1(NC(c2ccc(C#C)cc2)=O)CN(C(C2(CC)CCCC2)=O)CC1N=[N+]=[N-] C1(C)(OC)CCCN(C(=O)C(C)(C2CC2)N(C(=O)C(F)C2CCCC2)C)CC1 Cc1oc2ccccc2c1C(N1CCN(C(C2CCCC(=O)N2)=O)CC(O)C1)=O C1(CCC)(NC(C2CC2C(F)(F)F)=O)CCCN(C(c2snnc2)=O)C1.C CC(C)C(CC1CCCC1)C(=O)N1CCCCC(NC(C2CC23CC3)=O)C1 C=CC(CC)CC(=O)N(CC)CC1CCCCN1C(=O)CCc1cccnc1 CCC(CCCC(=O)NOCCO)NC(c1c[nH]c(=NC)o1)=O c1(C(C(=O)NC(C)CN(C(=O)CNC=O)C)O)ccc(F)c(Cl)c1F C1(C(N2CCC(C)(NC(Cc3c(C)noc3C)=O)CC2)=O)CCc2nccn2C1 N1(C(CC(C)c2cccnc2)=O)CC(CN(C)C(c2cnns2)=O)C2(CC2)C1 c1(NC(CNC(C(C2CCOC2)OC)=O)C(C)C(C)C)nc2c(C)cccc2o1 C(CC(C(F)(F)F)N(C)C)NC(C1N(CC)CCC1)=O CCC(C)C(C=O)NC(N)=O.C12(CC=O)CNC(=O)C(C1)C2.C1CCC1.N C#CCC(C(N)=O)NC(=O)CCCC1(NC(=O)C(C)CCOC)CCC1 C(=O)(C#CC1CCC1)N1CCN(CCN(C)C(C2CC2C2CCCC2)=O)CC1 C12(NC(C(=O)NCC)=O)CCC1CN(C(C1CCOC1)=O)C2 Cc1nc(C)oc1C(=O)N(C1(C)CCSC1)CCO.c1(C(C=O)=O)cccn1C Cc1cc(F)ccc1CNC(c1c[nH]nc1C)=O.C1(C=O)CN2CCC1CC2.N Cc1cc(Cl)c(C(=O)N(CC(C)(C)NC(c2nc(Cl)cs2)=O)C)s1 C1(C(=O)N)CC12CCCC2.C1(CC(=O)N(CCC(C)C)C(C)C)COCC1(C)C N1(C(C(C)CC#N)=O)CC(C(=O)N(CC(C)(C)CN(C)C)C)CC1(C)C C(=O)(C(O)CCCNC(=O)C(=O)C(C)(C)C)N1C(COCC#C)CCC1 CC(C)(C(=O)NCC1(CC)CC1)C(F)(F)F.C1(C(=O)N)CCC12CCCO2 c1(C(=O)NC2CCC(CNC(CC=CCC)=O)C2)c(C)cncc1C N1(CC(=O)N(C2CCN(C(=O)CC(C)N(C)CC)C2)CCC)C(=O)CCC1=O c1(C2CC(NC(=O)Cc3sccc3-c3nn[nH]n3)C2)ccc(Cl)cc1 N1(C(C2(CC#C)CC2)=O)CC(C2CCCCN(C(=O)CN3CCOCC3=O)C2)C1 N1(C(c2ccn3ccnc3c2)C(=O)NC)CCCC(C2CC2)CC1 c1(C(=O)NC2CC(NC(C3CCC(=O)O3)=O)C2)cc(OC(F)(F)F)ccc1F Cc1ncccc1NC(C1CC(O)CN1C(=O)CCc1cccc(O)c1)=O N1(C(c2cn(CC)nc2C)=O)CCCCC(C(=O)Nc2ccc(F)nc2)C1 Cc1cc(C(=O)NCC(CC(=O)NC2CCCCC23CC3)C2CCC2)cc(C)n1 C(=O)(C1=C(Cl)CCOC1)NCC(c1ccccc1)N(C(C(F)=C(C)C)=O)C C(=O)(C1=CCCN(C(=O)C#CC2(C)COC2)C1)NCC1CCC(CC)O1 N1(C(c2cc(C(F)(F)F)cs2)C)CCN(C)C2CC12 CC(C(=O)NC1CC1NC(=O)C(c1ccc(Cl)cc1)=O)C(F)F C1(NC(CC(CC)C2CCC2)=O)CN(C(=O)CC2C=CCC2)CC12CCOCC2 CC1CN(c2ncc(Cl)cc2O)CC(c2ccccc2)O1 C#CCCCCC(=O)N1CCC(O)(CNC(=O)Cc2ncc(C)o2)CC1 CCCC(CC)CCN(C(CCO)c1cccs1)C=O C(=O)(C1CCc2nccn21)NCC(C)NC(=O)C=Cc1ccc([N+](=O)[O-])s1 N1(C(C(CC)F)=O)CCC2CCC(C1)N2C(c1csc(S(C)(=O)=O)c1)=O C(=O)(C1=CCCCCC1)NCC1OCCCN(C(C2(C)CC(F)(F)C2)=O)C1 C1(NC(C=NOC)=O)CCN(C(c2ccc(C)s2)=O)C1c1ccccc1 C1(C(N2CCC(NC(CCCC=C)=O)C2)=O)Cc2cccc(OC)c2O1 C1(C(C#C)C)CCN(C(=O)C(C)(C2CC2)N(C(=O)CC2CCC(=O)CC2)C)CC1 N1(C(CC(C)N(C)C)=O)CC2CCC(N(C)C(C34CC3CNC4=O)=O)C2C1 Cc1cc2c(N3CCCC4C3CCN4C(C3CC3(F)F)=O)ncnc2[nH]1 C1(NC(Cc2ccc(C)s2)=O)CCC(NC(c2csc(C(F)(F)F)n2)=O)CC1 C1(N(C(=O)C(C)O)CCC)CCN(C(=O)CC(c2ccccc2)C2CC2)C1.C c1(C(=O)NC23CCN(C(=O)Cc4ccsc4)CCC2C3)nc2cc(F)ccc2s1 CCC(CC)CCC(=O)N1CC2CCC1CN2C(C1(C(N)=O)CC1)=O CC1CN(C(=O)C(=O)NCC2CCCn3ccnc32)CC2(CCCOC2)O1 C1(CNC(C2CC2CF)=O)CC2(CCN(C(C3CC3F)=O)CC2)CO1 C(C)(C(C(C)C)NC(=O)CCCn1ccnc1)NC(c1c(OC)nsc1)=O Cc1cc(CNC(C2CCOCCN2C(c2ccc(C(F)F)o2)=O)=O)ccc1F N1(C(CCCN(C(C2C(C)SCCC2)=O)C)=O)CCC2(CNC(=O)N2)C1 C1(NC(c2ccccc2C2CCC2)=O)CCCN(C(c2cccnc2O)=O)CC1 C1(F)(C(N2CC3C(NCc4c(C)nc(F)cc4)C3C2)=O)CCCCC1(F)F N1(C(C2(C#C)CC2)=O)CCN(C(C2CCSC(C)C2)=O)CC1CO c1(OC)ccc(C(=O)NCC2(O)CCCN(C(c3csnn3)=O)C2)cc1N CCC(C)(C)C(O)C(=O)N1CCC(CCCNC(=O)Cc2ccsc2)CC1 C1(CCOC)(C(=O)N(CC(C)NC(C2CNC(=O)C2)=O)C)CCCC1 c1(C(=O)NCC(N2CC(C)OC(C)C2)C)cncc([N+](=O)[O-])c1 Cc1ncc([N+](=O)[O-])cc1C(=O)NC(C)CO.C1(CCC(=O)N)CCC(=O)N1 C#Cc1ccccc1CC(=O)NC1CCN(C(c2ncsc2C(F)(F)F)=O)C1 C(C(C)C(C)C)NC(C1(COC)CCC1)=O.C(=O)CN(C1CCC1)C.N N1(C(c2ccc(C#C)cc2F)C(=O)NCC(=C)C)CCCCC1C1CCCO1 c1(C(N2CCC(N(C(c3ccc(Cl)o3)=O)CC)C2)=O)n[nH]c2c1CC(F)(F)CC2 c1(CC)nn(C)c(CC)c1C(=O)N.C(=O)(C(F)C(C)(C)O)N1CCCC1.C C(CC(C(=O)N1CC(CO)C1(C)C)NC(=O)C(c1ccccc1)C)=CC C1(NC(C=COCC)=O)CCC(C)N(C(c2nocc2CC)=O)C1 C=C(C)CN=C(NCC1CC1C)NC1CCC(C(F)F)CC1 C12(CNC(CC3CCC(C)C3)=O)CCC(CC1)N2C(c1ccc(F)c(F)c1)=O Cc1nc(C)n(CC2CCCN2CC(C2CCN(C(=O)OC(C)(C)C)CC2)C)n1 N1(C(C(CCC)C#N)=O)CC2CC(C1)CN(C(c1cc3ccccc3[nH]1)=O)C2 c1(C(=O)NC(CCCC)CNC(C2(C#N)CCCC2)=O)cnc2scnc2c1 C(N=c1nc(N(C)Cc2nnc3ccccn23)c2c([nH]1)CSC2)C1(CSC)CC1 c1(C(=O)OC)cc(C(=O)NC2CCN(Cc3[nH]c(C)nc3C)C2)ccc1Br N1(CC)CC2CN(C(=O)CCN3C(=O)C=CC3=O)C2C1.c1(C(=O)N)cnccn1 c1(CN2C(C(=O)Nc3ncc(Br)s3)CC(O)C2)cn2ccccc2n1 N1(C(c2ccc(OC)c(Cl)c2)=O)CCN(C(=O)C=C(Cl)Cl)CC(C)(F)C1 c1(C(=O)NCCC(C)N(C(=O)C(O)C2CC2)C)ccc2c(c1)nnn2C C1(OC)CC2CC(C(=O)NCC3CCOCC3)CC12.c1(C=O)ccc[n+]([O-])c1.N C(C(=O)N)(C(C)C)OCC.C1CCCCC1.C(=O)CC1(C(F)(F)F)CC1 S(=O)(=O)(c1scnc1C(=O)O)NC1CCN(S(C(C)C)(=O)=O)CC1C C1(CC=O)CCC(C)CC1.C(=O)(C(C)N(C)C)N(CC)Cc1ncc[nH]1.N C#CC1(NC(C2CCC(C)CN2C(C2CCCC(=O)C2)=O)=O)CCCOC1 C(=O)(C1=Cc2ccccc2C1O)NCC(CN(C(C(C)c1ccco1)=O)C)(C)C C1(NC(c2ccn(CC)n2)=O)CC2CC1CC2C(=O)N.C1CCCN1C(C)C C1(C)(C(=O)N)CCCCC1C.c1(C(C)NC(=O)CNC(=O)C)nnnn1C CCCCC(CNC(=O)CC(c1cccc(C(F)(F)F)c1)C)NC(=O)C1CC1 CC1c2ccccc2CC(C)(C)N1C(C1CCN(C2CCN(C)CC2)C1=O)=O C(C(=O)N(CCC(=O)NC(C1CCCC1)C)C(C)C)(C1CCC1)OC CCC(C)C(O)CC(=O)N1CC(CNC(=O)OC(C)(C)C)(O)C1.C(C)C c1(CN2CC(NC(=O)Cn3nccn3)CC(F)(F)C2)cc(F)cc([N+](=O)[O-])c1 C1(N(CC=O)C)CCS(=O)(=O)C1.CC(C)CC.c1(C=O)sccc1C1CC1 C(C1=CCCN(C(c2cnc(C(F)F)nc2)=O)C1)NC(C(C1CC1)SC)=O Cc1ccc2n1CCN(C(C1(C)CCCN(CC(C)O)C1)=O)C2C Cc1ccc(C(=O)NCC2CC2CNC(c2ccc(O)nn2)=O)c(F)c1Br Cc1c(C(N2CCCC2C(=O)NCCCCCN(C)C)=O)c[nH]c1C#N C(N=c1[nH]c(=NCC(F)c2ccccc2)[nH]c2c1COCC2)c1c(SC)ccnc1 N1(C(C(c2n(C)ccc2)=O)=O)CC2CCN(C(c3ccn4ncccc34)=O)CC12 c1(C(=O)NCC(CNC(CC2CCC(C)C2)=O)C)cccc2nccn12 c1(C(=O)NC(CNC(c2cc(C#N)on2)=O)C2CC2)cc(Cl)nc(Cl)c1 c1(C(=O)OCC(=O)N(C2CCS(=O)(=O)C2)CC(C)C)ccc2n[nH]cc2c1 C(=O)(C(C(=O)N1CCC1CNC(c1ccc(C)[nH]1)=O)C(C)C)OCC c1(C=O)c(Cl)cnn1C(C)C.C1(CCNC(CC2(C#N)CC2)=O)CCCC1.N c1(C(N2CCN(C(C3CN(C(N)=O)C3)=O)C3C2C3)=O)nnc2n1CCCCC2 C#CC1(O)CCN(C(C2CN(C(=O)C(O)C=CC)CCC2(C)C)=O)CC1 N1(C(Cc2cnc(C)[nH]2)=O)CCC2CC(C1)CN(C(=O)C(c1cnn(C)c1)O)C2 C1(NC(Cn2c(C)nnn2)=O)CCN(CCNC(=O)C2=CCC2)CC1 C1(C(=O)NC2(C)CC(NC(C(CC)(C)C#N)=O)C2)CC2(CCOCC2)CO1 CCCCC(CNC(c1nc(C2CC2)oc1C)=O)NC(C1(C=O)CCC1)=O.N N1(C(c2cc(C)c(C)[nH]2)=O)CC2CC(NC(C3CC4CC4CC3C)=O)CC2C1 C1(CNC)C(=O)NCCC(=O)N1.c1(CC2(C(=O)OC)CC2)ccccc1 C12(C(=O)OC)CC(CN1C(c1cn(CC)nn1)=O)C2.C(=O)CC.C(C)=O n1(CC(=O)NC(CNC(c2c(C)nccc2)=O)C2CCC2)ncc2ccccc12 C=C=CC(C)C(=O)NCCCN(C(=O)C(c1ccc(Br)s1)=O)C1CC1 N1(C(C(=O)NCCCC)c2cnc[nH]2)CCOC2(CC2)C1 C1(NC(C2CC(OCC)C2)=O)CCN(c2ncncc2I)CC1F C=CCCC(C(=O)N)NC(=O)OC(C)(C)C.c1(C=O)cnnc(Cl)c1.CCC Cc1ccc(C#N)cc1C(N1CCN(C(C2CC2C)=O)C(C2CCC2)C1)=O S(=O)(=O)(CC(=O)N1CC(C(C)NC(c2cc(OC)n(C)n2)=O)C1)NC C(=O)(C(C)(CC)CCC)N1CCC(CNC(CCOCCC)=O)(OC)C1 C1(NC(C(COC)COC)=O)CCCN(C(c2cc3ccccc3[nH]2)=O)CC1F N1(C(c2c(OC)c(Cl)ncc2)=O)CC2(CCC2)CC1C.n1(CC(=O)N)cncn1 c1(C(=O)NC2CCC(NC(C3(c4c(C)c[nH]n4)CC3)=O)C2)nc(Cl)sc1C N1(c2cc(C)nc(CO)n2)CC2(CN(C(=O)C=CC=C(Cl)Cl)CCO2)C1 N1(C(C(c2c(C)nn(C)c2)O)=O)CCC(CO)(NC(=O)CC#N)CC1 c1(C(=O)OC)cccc(C)c1F.N1(C(C(=O)N)=O)CCC(C(O)C(F)(F)F)CC1 C1(C(=O)NCCCSCC)CCCC1C1CCN(C(=O)NCC2CC2)CC1 c1(C(N2CC(CC(C)NC(C(n3cc(C)nc3)(C)C)=O)C2)=O)c(C)cccc1Cl N1(C(=O)NCc2ccc(CN(CC)CC)cc2)CC2(CC(=O)NCC2O)C1 C1(CNC(C(C)(C)CO)=O)CN(C(C2CCC2(F)F)=O)CCC12CCC2 C1(NC(C(COC)C)=O)CN(CCC2CCCC(C)C2)CC1(C)C C1(C(=O)NCCCCCNC(C(C)OCC#C)=O)CCCN(c2cnccn2)C1 Cc1cc(C(N2CC(CN(c3ccnc(C)n3)C)C2)=O)n(C2CCC2)n1 c1(C(C(=O)NC2COC2)N(CCCC)C(C)CC)cn(C)nc1I O=S(=O)(C1(Cl)CC12CCNCC2)N1CCCC1c1cccnc1 C1(C(=O)NC2C(NC(c3c(C(C)C)cco3)=O)CC2)CN2CCN1CC2 C1(NC(C(COC)(C)C)=O)CCCCN(C(=O)C(N2C(C)CCC2C)C)C1 C1(C(=O)NC2CCN(C(C=C(C)C3CC3)=O)CC2C)C2CCC1(C)C2(C)C C1(OC)CCC2(C=O)CC12.c1(CC)cccc(C)n1.C(C)(C)CC=CC=O.N C(C#Cc1ccccc1)NC(C(=O)Nc1c(Br)ccc(C(=O)OC)c1)=O c1(C(=O)NC(CC)CNC(=O)C(C)C(=O)OC)cncc(Cl)c1.CC(C)C.O N1(C(Cc2scc(C)c2)=O)CCCN(CCNC(=O)C=Cc2cc[nH]n2)CC1 c1(C(=O)OCC2COC3CCCC3O2)cccc2ccccc12 Cc1cc(C(N2CC(NC(=O)COC(F)(F)F)CC(C)C2)=O)ncc1C#N Cc1cccc(N(C)C(c2ccccc2C(N2CCOC(C)C2)=O)=O)n1 C(CC1CC1)(C(=O)N)OC.C1(C=O)CC(C)(C(C)(C)C)C1.CCC.CC C(=O)(C(F)C(C)CNC(=O)C(C)(C)CO)NCCn1c(C)nc(C)n1 N1(C(C=C(C)CNC(c2cc(CCO)on2)=O)=O)CCC(O)C(F)C1 N1(C(C2C(C(=O)OC)CCCC2)=O)CCCN(C(c2ccccc2I)=O)CC1C c1(C(N(CCNC(c2ccc(-c3nc(C)sc3)s2)=O)C)=O)c(C)ccnc1C N1(C(C2CC(CC(F)F)C2)=O)CC2(CCCCN2C(c2cc(Cl)nnc2O)=O)C1 n1(CC)nnnc1C(c1cccs1)NCCC(=O)NCCOC c1(CC)cc(C(=O)NC(CO)CCCNC(=O)C(C)=C(C)C)n(C)n1 N1(CC(c2cn(C)nc2)=O)CCC(SCCC2CNC2)CC1 C1(C(N(CC(CC)NC(c2sccc2F)=O)C)=O)CCN(c2ccccc2)C1=O c1(CC(=O)NCCN(C(=O)CN2C(C)CCC2C)C(C)C)cccc(F)c1Cl C(=O)(C1CCCc2ccccc21)NC(C1(O)CCN(C(C(CC=C)C)=O)C1)C C(=O)(C(F)CC1CCCCC1)N(C1CCN(Cc2cc(C)on2)C1)CCC c1(C(=O)NCC(CO)NC(C2CCN(OC)CC2)=O)cccc2nc(Cl)cn12 c1(C(N2CC(N(C(=O)C=CCF)C)C3(C2)CC3)=O)cc(Cl)cc2c1OCC2 CC(C)C(O)C(C)C(=O)N1CC(OCCC(N2CC(O)(c3nn[nH]n3)C2)=O)C1 CN1CC(C(=O)NCC2CN(Cc3nncn3C)C2)CC1=O c1(C(N(C(C)(C(N2CC3C(N(C)C)C3C2)=O)C2CC2)C)=O)nnn(C)c1N C1(CN(C(=O)CCC2CC(NC(c3csnc3Cl)=O)C2)C)CCCC1O C=C1CCC(C(=O)NCC2CN(C(=O)Cc3cc(OC)no3)CCO2)CC1 N1(C(C(CC#C)C)=O)CCN(C(c2cn[nH]c2)=O)C2CS(=O)(=O)CC12 N1(C(Cc2c(C)cccn2)=O)CC2CCC1C(NC(c1ccc(F)c(O)c1)=O)C2 C1(C(=O)NCCCC(C)CO)COCCN(C(c2ccn(C(F)F)n2)=O)C1 C(CCN=c1nc(N2CCCCCC2)cc[nH]1)N1CC(C)CC(C)C1 N1(C(CC2ON=C(C)C2)=O)CC2(CCC2NC(c2cc(C)c(Br)o2)=O)C1 C1(CC)CCOCCN1C(C1CCCC1NC(=O)C(c1ccn(C)n1)C)=O CC1CN(C(C2CCCCN2C(C23COCC2C3)=O)=O)CCS1=O c1(-c2ccc(OC)cc2)cc[nH]c(=NCCC(COC)OC)n1 c1(-c2c(C)nc(OC(C)C)cc2)ccc2cc(C(=O)NC3CCCOC3)[nH]c2n1 Cc1ccc(CC(=O)NC2CC(NCc3ccnc(OC(F)(F)F)c3)C2)cc1 c1(C(N2CC(O)CC(NC(C3CCC4CC4CC3)=O)C2)=O)cccn2cnnc12 c1(C(C)(C)C(=O)N2CCC(NC(=O)CCNC(=O)CO)C2)ccc(Cl)cc1F Cc1c(C(=O)NC2CC(NC(c3sccc3Br)=O)C2)c(Cl)nn1C c1(C(N(CCC(C)(C)NC(CNC(C)=O)=O)C)=O)cccc2occc12 Cc1cnnc(O)c1C(=O)NC(C1CCCN(C(=O)Cc2cnoc2)C1)C C1(N(C(=O)CN2CCCNC2=O)C)CCN(C(=O)COC2CCCCC2)CC1C c1(C(=O)NC(CC)CNC(c2cncn2C)=O)cc2c(OC)ccc(OC)c2[nH]1 CC1OC2(CO)CC1(C(=O)NC1COCCN(C(c3cc(O)ccc3F)=O)C1)C2 C(=O)(C1CCc2c[nH]nc21)NC1(CO)CCCN(C(C(C)OCC)=O)C1 N1(C(c2ccc(C#C)cc2)=O)CC2CCN(C(C3(C(F)F)CC(F)(F)C3)=O)CC12 C1CCCCN(C(=O)C=C)C1.c1(C(=O)OC)coc(C(=O)NC)c1.N1CCCC1 c1(OC)ccc2cc(C(=O)NC34CCCC3N(C(=O)C(C)C)CCC4)[nH]c2c1 N1(C(C2(C)CCCS2)=O)CCC2(CC1)OCCC2NC(c1cnn(C2CC2)c1)=O c1(C(N2C(C)CC(CO)C2)C(=O)Nc2cccc(F)c2)ccc2[nH]nc(Cl)c2c1 C(=O)(N1OC2C=CC1CC2)C1C=CCN(C(C2C(C(C)C)OCC2)=O)C1 N(C1CCc2cccnc21)C(=O)NC1CC(c2cn(C)nc2)S(=O)(=O)CC1 C=CC(C)(O)C(=O)NCC(C(C)(C)C)NC(=O)C(C)(C)c1nncn1C C1(N(C(c2nc(CC)sc2)=O)CC)CCCN(C(=O)CCc2ccc(O)nc2)C1 c1(C=O)cc(C2CC2)ncn1.C1(C(=O)NCCC2CCCC2)(SC)CCC1.N C1(C=O)C2CCC1(c1ccccc1)C2.C(C(C)C(=O)N1CC(OCC)C1)OC.N N1(C(CNC(CCC)=O)=O)CC2(C1)CN(C(=O)CCn1cncn1)CCO2 c1(C(N2CC(C)(NC(Cc3nc(C)sc3C)=O)C2)=O)ccc(Br)cc1N CC12CSCC1(C)CN(C(=O)NC1CC(=O)N(c3c(F)cccc3F)C1)C2 c1(C(=O)NCC2(C(N)=O)CN(C(=O)C)C2)ccc(F)cn1.c1ccccn1.S O(NC(=O)C1=CCCC1)CC(=O)NC(CC#C)C(=O)NC(C)=O C(c1cnccn1)=CC(N1CCCC(N(C(=O)Cn2cnnc2O)CCO)C1)=O C(c1ccco1)=CC(=O)N(C1CCN(C(C2(C)CC2(F)F)=O)C1)CC CCN=C(NCCS(=O)(=O)NC(C)(C)C)N1CCC(c2ccccn2)C1 CCC(C)(CNC(C1CC(C)(C)CN1C(=O)CCCN=[N+]=[N-])=O)C(N)=O N1(C(c2cc(CC)ncc2)=O)CC(C)(C)CC1CNC(C1CC(C#N)C1)=O CC(C)C(O)C(=O)N(C1CCCC1)C(C)C.N1(C(CNC(C)=O)=O)CCCC1=O c1(C2(C=O)CC2)ccccc1Cl.C1(CC(=O)N(CC)CC)CCC1(C)C.CO N1(C(Cn2ccc(=N)[nH]2)=O)CCC(F)(CNC(=O)COc2ccon2)CC1 c1(C(N2CC(NC(c3scc(C)c3)=O)C(C)C2)=O)cc2cnc(Cl)cc2s1 c1ccc(C)c(C)c1.C1(CC=C)(NC(C2CCC3CC23)=O)CCN(C(=O)C)C1 c1(C(N2C(c3cn(Cc4nnc(C)o4)nn3)CCC2)=O)cc(F)cc(Cl)c1N C#CCC(O)C(=O)N1CCCC1CNC(c1ccc[nH]1)=O C(C)(C(=O)NOCCOCCO)(C1CC1)NC(CC1CCC(C)C1)=O N1(C(C=Cc2ccc(SC)s2)=O)CC2CCC1C2.C1(C)(C=O)CC2(CCC2)C1 N1(C(C2(C(=O)NC)CC2)=O)CCCC1(C)C.c1(C(=O)N)ccccn1.CCF N1(C(c2c(C)cc(C)s2)=O)CCN(C(c2cccn2C2CC2)=O)CC(C)C1 c1(C(=O)OC)cnn(CC(=O)NC2CC2NC(=O)C)c1.CCCC(C)C.O c1(NC(C(=O)OCC)=O)cccc(CCCOCCCCCN)c1 Cc1cc(C(=O)NCC2CC2C2CC2C)c2c(n1)CCCC2=O c1(C(=O)NCC2(OC)CCN(C(C3SCCS3)=O)CC2)ccnc2[nH]c(O)nc12 C#CCCCC(C)C(=O)NC(CO)C(=O)NC(COCC)C(C)C CC1(C)Cc2ccc(C(=O)NC3CCN(C(C4(C)CCOC4)=O)C3)cc2C1 N1(CCC(=O)Nc2n(C(CC(C)C)C)ncc2)CCCCC(C)(C)C1 CCC(C)(O)C(=O)NCC(C)(C1CC1)NC(=O)C=Cc1ccc(Br)s1 O=C(C(F)CC1CCC1)NCCCCNC(C1(O)CCCC1)=O C12(CN)CCC(CC1)C2.C1(NC(=O)OC(C)(C)C)C(=O)NC2CC12 c1(C(=O)NCCC)ccccc1Cl.C(=O)CCC1CC1(F)F.C(=O)C1CC1.N c1(C(=O)NCC(C)NC(C2(O)CC2)=O)cccc2c1C(C#N)C2 c1(C(=O)NCC2CC(Nc3c(C#N)c(Cl)ns3)C2)cccc2cnnn12 N1(C(C(C)=CC2CC2)=O)CC(S(=O)(=O)NC2CC2)C1 CC(C)=C=CC(=O)NCc1cc(C(=O)NCC2COCCO2)n[nH]1 c1(CC(C(=O)NC2CCNC2=O)NC(CC2(C)CCCC2)=O)ccc(Cl)cc1Cl C1(C(N(C)CC)=O)CCCCN1C(=O)CC1CCCOCC1 c1(C(C(=O)N(C2CCC(NC(=O)C(N)=O)C2)C)(F)F)cccc(Br)n1 C(C(C)(O)CC=O)OC.C(C)(C)Cn1cccn1.C1(C=O)(C(C)C)CCC1.N C1(C(=O)NC(C#C)C(C)OC)CNC(=O)CN1C(=O)CC=CC=C c1(OC)cccc(C(F)(F)C(=O)NCC(O)CNC(=O)Cc2ccon2)n1 C(CC(=O)N1CC=CC(NC(c2ccnn2C)=O)C1)(C(F)(F)F)OC.C1CC1 c1(C(=O)NCC2CCN(C(CCCCCCC)=O)C2)c(OC)ccc2[nH]ccc12 CCCCC(C(=O)N(C)Cc1cccc(C)c1)N(C)C.C(=O)C(O)CC1CC1.N N1(C(N(CC=C)Cc2cccnc2)=O)CCN(C(C)C)CC1 Cc1nc(C)c(C(N2CCC(n3cccn3)CC2)C(=O)NC2CCC2)s1 c1(COC)cc(C(=O)NCC2CCCC2NC(c2csc(Cl)c2)=O)n[nH]1 c1(C(=O)NCC2(Nc3ncc(C#N)cc3F)CCCC2)ccc2c(c1)CCOC2 C1(NC2(c3n(CC)nnn3)COCCOC2)CCc2ncccc2C1 c1(SC)ccncc1NC(=O)CC(C)NC(=O)CCC1(C)COC1 Cc1cc(C(=O)N)cc(C)c1O.C(C)(C)C1CCC1.C1(C=O)(C(N)=O)CCC1 N1(C(C(CC)COC)=O)CCC(C2CC2NC(C23COC(CF)(C2)C3)=O)CC1 C1(NC(C(C)CO)=O)CCN(C(c2csc(-c3cccs3)n2)=O)C1C(C)(C)C N1(C(C2(C)CNC(=O)C2)=O)CC2CC(NC(c3cncc(F)n3)=O)CC2C1 N1(C(C2CC3CC3C2)=O)CCC(O)(CNC(C2(C(F)(F)F)CC2)=O)C1 Cc1cc(C(=O)NC2(C)CC(NC(=O)CC3CC4COCC34)C2)n(C)n1 Cc1cnc2cc(C(=O)NC3CN(C(C4(C)CCC(C)CC4)=O)CC3C)nn2c1 N1(C(C(COCC)C)=O)CCC(C)C(CC(N2CCCOCC2)=O)C1 Cc1cncc(C(=O)NCC2CCOC2C(=O)NOCC(C)C)c1 Cc1nc(Cl)ccc1C(=O)NC1CCCC1NC(c1cc(Br)nn1C)=O C=CC(CC)C(=O)N1CC=CC(C(=O)N(CC(N)=O)CC(C)C)C1 C(=O)(C(Cc1ccccc1)C(C)C)N.C1(NC(CN(CC)CC)=O)CCCC1 c1(CCC)occc1C(=O)N(CC(C)O)CCNC(C1CC12CCC2)=O Cc1ccccc1C(F)(F)C(=O)NCCN(c1nccnc1F)C1CC1 C(=O)(C(O)C(C)(C)C)N1CC(CC)(OC)C1.C1(C=O)CCN(C)C1C(C)C N1(C(CCC)=O)CC(CO)(NC(c2ccc(SC(F)(F)F)s2)=O)C1 CCC(C)(C(=O)NC(C)Cc1cn(CCC(=O)OC(C)C)nn1)C(F)F CCCCC(O)C(=O)NCC12CCC1CN(C(=O)C=Cc1cocn1)C2 C1(CNC(C(n2cc(Cl)cn2)C)=O)COCCN1C(C1CC(CF)C1)=O N1(C(C(C2N(C(c3cc(CC)sn3)=O)CCC2)(C)C)=O)CC2CCCC1C2CO N1(C(C2C(C(=O)OC)C2)=O)CC2CN(C(c3cc(C4CCC4)no3)=O)CCC12 CC1CN(C)CC(C=O)O1.c1cc(C(=O)N(CC(N)=O)CC(N)=O)n(C)n1.N C(C(C)(CC(C)C)NC(c1cc(-c2cc[nH]n2)ccc1F)=O)NC(COC)=O S(=O)(=O)(c1cccc(N2CCC3(CCCCC3)C2)n1)N1CC(C)(C)C(O)CC1 N1(C(C2(N)CCC2)=O)CCCC1CS(N)(=O)=O n1(CC)ncc(C(N2CCN(CCN(C)C(C3(C)CC3F)=O)CC2)=O)c1C C1(O)(CNC(C2CC=CCC2)=O)CC(C(N2CCC2C2CCCC2)=O)C1 c1(C(=O)NC(CC)C(O)CC)ccnc(Cl)c1Cl N1(C(=O)NCCCCC(=O)N(C)C)CC2CCCC2C1 c1(C(N2CC=CC(NC(C(C)=C(C)C)=O)C2)=O)cnc2cnccc2c1 C=C=CC(C)C(=O)NCCSCc1ccccc1.c1(CC=O)c(C)noc1Cl N#Cc1ccc(F)c(C(=O)OCC(N2CCc3ccccc32)=O)c1 N1(C(c2cc(C)cc(O)n2)=O)CCC(C(=O)NC2CC3(CCOC3)C2)=C(F)C1 CN1CC(NC(=O)CC2(CNC(=O)C(O)CC(N)=O)CC2)C(C)(C)C1 c1(OC)ccc(C(=O)NC2CC2NC(c2cc(C3CC3)no2)=O)c(O)c1 N1(C(C(CC#C)C)=O)CCN(C(C2(c3c(C)cccc3C)CC2)=O)CC1CCO c1(C(N(CC(=O)O)CCOC)=O)cc(-c2cn[nH]c2)cs1 C1(CNC(c2cc(C)c(F)cn2)=O)CN(C(c2cc[n+]([O-])cc2)=O)CCC1(F)F N1(C(Cc2c(C)nsc2)=O)CC(NC(=O)COC2CC(F)(F)C2)CC1C C1(NC(c2ncn(C)n2)=O)C2CCN(C(C3CC(C)(C)C3)=O)C2C1(C)C Cc1ccc(OC(C)C)c(S(=O)(=O)N2CCC3(C)C(C2)C3(Cl)Cl)c1 Cc1cccc(C(=O)NC(CO)C(=O)NCCC2OCCC2C)c1C#N N1(C(C2(NC(C(C)n3cnnn3)=O)CC(F)(F)C2)=O)CCc2ccncc2C1 C1(CNC(=O)CC2CCC(=O)N2)CCC2(CN(C(=O)COCCO)C2)O1 Cc1cccnc1C(C)NC(=O)CCOC(C)C.C(=O)(C(F)C1CCCC1)N CC(C)CCCCC(=O)NCC1(NC(c2cc(F)cc(F)c2O)=O)CCOCC1 C(=O)(C(C)Cn1ccc(C)n1)N.C(C)(CO)NC(C1(CC(C)=O)CC1)=O N1(C(C(CC=CC)C)=O)CC(O)CC1(C)C(=O)NOCCCCCC1CC1 CC1CN(C(C2(C)CCCS2(=O)=O)=O)CC(C)CN1C(=O)Cn1cnnc1 CC1CN2CCN1CC2C(=O)NC1CC2CC(C1)N(C(c1c[nH]ccc1=O)=O)C2 C1(NC(c2cnn(C)c2C#N)=O)CCCC2CN(C(c3cc(C#N)c[nH]3)=O)CC12 Cc1nnc2n1CC(CN=C(NC1CC1)NC1CCc3c(nnn3C)C1)CC2 c1(C(N(CC(CN(C(C2CC=CC2)=O)C)O)C)=O)cc2ncccc2s1.COC c1(OC)ccccc1C(C)=CC(=O)NCC1CCCN(C(=O)C(CO)N(C)C)C1 Cn1cnc2cc(C(N3CC4CC4(CNCc4c[nH]ccc4=N)C3)=O)ccc12 c1(CN(CC=C)CCc2ccc(Cl)s2)nc2ccccc2n1C(C)C c1(C(=O)NC2C(C)CN(CCc3c(F)cccc3Cl)CC2)scc2c1OCCO2 C1(NC(CC2(C)CCOC2)=O)C2CC3C1C3C2C(=O)NCCn1cnnc1 Cc1[nH]c2ccnn2c(=O)c1CC(=O)NCC1CC1.C1(CC=O)CC2CC2C1 c1(CN=C(NC(C)C)NCc2cn(C(C)(C)C)nn2)cc(C)cc(C)c1 CC1CC(C(=O)NCCOCC(=O)NCC2CCSCC2)CCS1 c1(C(=O)NC(C(=O)NCCS(CC)=O)CCN(C)C)cc(C#N)[nH]c1C CC(C)(CNC(=O)Cn1cc(C2CC2)nn1)CCNC(C1CC1(C)C)=O N1(C(C(C)(C)N(C)C)=O)CCC2(CCCO2)C1.c1(C(=O)N)cc(C(N)=O)cn1C Cc1cc(C)c(NC(C2CCCN2C(=O)CSCC(N)=O)=O)cc1O C1(NC(=O)CSC2CC2)CN(c2ncc3c(Br)cccc3n2)CC12CCOCC2 C1(NC(CC(=C)C)=O)CN(C(=O)COC2(C)CCCC2)CCC1c1ccccc1 Cc1cc(C(=O)NC(CNC(=O)CCCCC2CC2)CO)c(C)cn1 c1(C(N2CCC(CC(=O)N)C2)=O)cccc2[nH]ncc12.C(CC(=O)N)C1CC1 Cc1ccc(C(=O)NC(C)(C)C)cc1C(F)(F)F.c1(C(=O)N)c[nH]ccc1=O C(=O)(CCC(C)(C)[N+](=O)[O-])N.C1(CN(C(=O)C(F)OC(F)(F)F)C)CCC1 C#CCC(O)C(=O)NC(C(N1CCC(NC)C1)=O)C1CC1 C1(CNC(C=CSC)=O)(COC)CCCN1C(c1cnn(C2CCCC2)c1)=O C1CCCCC1.c1(C=O)ccnn1CCN(C)C.CCCN(C(=O)CO)C.C C(=O)(C(C)(C)C(=O)NCc1ccc(C(N2CCC(C)C2)=O)s1)OCC c1(C(N(CC(C)NC(=O)CCCCCSC)CC)=O)cc2n(n1)CC(C)NC2=O C1(C(N2CCN(C(=O)Cn3cccc3)C(CF)C2)=O)CC2CCCCCC12 Cc1cc(C(=O)NCC2(CCNC(=O)C)CC2)c(C)nc1C.c1ccon1 c1(CC)cc(CC(=O)NCC2COCCN2C(=O)C(O)COC)n(C)n1 C1(Br)(C(=O)NCC(C)NC(C2(CC(C)C)COC2)=O)CC1(F)F C(=O)C(C)C(O)C(C)C.Cc1ccc(F)c(C(N2CC(C(N)=O)(C)C2)=O)c1.N Cc1ccc(CCNC(C2CCCCN2C(C2CCC2C#N)=O)=O)cc1 N1(C(c2c(OC)n[nH]c2)=O)CCC(CNC(c2cccc(N(C)C)c2)=O)CC1C C1(C(=O)NC2(C)CCSC2)COCCN(C(c2cnc(O)o2)=O)C1 C1(CNC(c2c(C)n(C)nc2)=O)CC2CCC1N2c1ccnc(Cl)n1 C1(CC(=O)NCCCC2CCC2)C2CN(C(C3CCO3)=O)CC12 C1(CNC(=O)Cn2ncc(O)nc2=O)CC2COCC2N1C(C1CCCS1)=O c1(C(=O)OCC)cc(C(=O)N)[nH]c1C.n1(CCC=O)cc(Cl)cn1.C(C)C C1(NC(C=Cc2nc(C)c(C)[nH]2)=O)COC2C(NC(c3ccncn3)=O)COC12 c1(C(=O)NCCC(C)NC(C(CC)C)=O)cnc(N)c(O)c1 CCCCCCC(C)C(=O)NCC1(C)CN(C(=O)COCCC)C(C)(C)C1 c1(C(=O)NC2CC3CC(NC(CC(CN(C)C)O)=O)CC32)ccnc2ncnn12 C1(CNC(CN2CCC(C)CC2)=O)CC2CCC(C1)N2C(=O)Cc1cncnc1 S(=O)(=O)(c1ccc(NCC2CC(C)C2)c(Cl)c1)N1C(COC)CCCC1.C c1(C(=O)N)c[nH]c2cccc([N+](=O)[O-])c12.CC(C)(F)C(=O)NCCC1CCCC1 N1(C(CCCSC)=O)CCC2(CC1)CC2NC(C1(N=[N+]=[N-])CC1)=O N1(C(C(CC=C)CNC(C2CCCC23CCC3)=O)=O)CC2(CCC(C)OC2)C1 O=C(CN1CCN(Cc2cccc(F)c2O)CC1)N=c1cc(Cl)cn[nH]1 N1(C(C2C(=C)C2)=O)CCC2(CCCN2C(c2cnn3c2CN(C)CC3)=O)CC1 C1(OC)CC(NC(=O)CC2=CCCC2)CN(C(c2coc(C3CC3)n2)=O)C1 C12(C(=O)NCCC#C)CCN(C(c3cnc(OC)s3)=O)CCC1C2 c1(C(=O)NC2CC(C)(C)N(C(=O)Cc3ccoc3)C2)ccc2ccncc2c1 C(S(=O)(=O)CC(=O)N1CC(CNC(c2cccc(F)c2N)=O)C1)c1cn(C)nc1 N1(C(c2[nH]c(=N)sc2)=O)CCCC(CO)(NC(C2CC3(CCC3O)C2)=O)C1 C(C(C(C)(C)C)OC)NC(CCC1CC(NC(COC)=O)C1)=O c1(SC)ccc([N+](=O)[O-])cc1C(=O)N.C1(C)(C=O)CCOC1.C(C)C1CCC1 C1(CC)CN(C(=O)C(C)C(=O)OC(C)(C)C)CCN1C(=O)CS(N)(=O)=O c1(C(=O)NCC2C(NC(c3csc(Br)c3)=O)C2)ccc2nsnc2c1 N1(C(C(COC)O)=O)CC(C)C(C)(CNC(c2ccnc(C3CC3)n2)=O)C1 Cc1occc1C(N1CCCC1C1CCCN(C(=O)C(O)CN(C)C)C1)=O.CO C12(C(N3CCCC(N4CCN(C(C5C(C)=C5)=O)CC4)C3)=O)CC1COC2(C)C c1(C(CNC(COCCCC)=O)NC(c2scnc2CC)=O)ccccc1Cl Cc1ccc(C(N2CCC(CNC(c3cocc3Br)=O)CC2)=O)nn1 Cc1cc(F)cc(NC(C2CCCN2C(=O)CCOc2ccccc2)=O)c1C Cc1c(C(=O)NC2CC(NC(=O)Cn3nnnc3C)C2)cnn1CC(F)(F)F c1(CC)ocnc1C(=O)NCC1CC(C(=O)NC2(CO)CCC2)CO1.C C1(NC(C(C)OCC=C)=O)CCC(N(C(=O)C(C)=C(C)C)C)CC1 c1(CCNC(CC=CCC)=O)ccc(N(C)C)cc1.C(=O)C(C)n1cncn1.N C(=O)(C1COc2ccccc21)N1CCCC(NC(c2ccncn2)=O)(CO)C1 C1(CC)(NC(c2cc(C3CC3)ns2)=O)CCCN(C(=O)C(c2ccccc2)F)C1 c1(C(=O)Nc2cc(CN)c(Cl)cc2)cc(F)ccc1N1CCCCC1 CC(C)C(CNC(C1CCCC1C)=O)NC(c1nc(C(C)(C)C)no1)=O C1CCN(C(c2cc(C)ccc2C)=O)C(C)C1.C1(CCOCC)(C=O)CCC1.N N1(C(C(C)(C)OCCC)=O)CC2CC(C(=O)N(C)Cc3scnc3C)C(C2)C1 N1(C(C(C(CC)CC)C)=O)CC2CCN(C(C3(O)CCCC3)=O)CC2C1 c1(C(=O)NCCCCNC(c2c(OC)c[nH]n2)=O)cc(OC)ccn1 C(C(C)N=c1[nH]c(=NC)[nH]c(=NC(CN2CCCC2)C2CC2)[nH]1)NC(=O)OC C#CC1(CNC(C2CCC(NC(=O)C(O)C=C)C2)=O)CCCC1 C(=O)CCC1CCc2ccccc21.CC(C(C)C)NC(=O)COCC1CCCC1.N N1(C(C(C2(O)CCC2)NC(C2CC2(F)Cl)=O)=O)CC2CC=CC1C2 N1(C(C2CC(N(C)C)C2)=O)CC2(C(N3CC(CO)C(C)(C)C3)=O)CCC1CC2 c1(C(N2CC(C)N(C(c3ccc4sncc4c3)=O)CC2)=O)ncc2ccccn12 C(Cc1ccc(Cl)cc1)(C(=O)NNC(C)=O)OC n1(CC)cc(NC(=O)CN(C(=O)C(C)NC=O)CCOC)c(C#N)n1 C(=O)(C1=NOC(C)C1)NCCN(C)C(C12CCCN1CCC2)=O.C1(O)COC1 N1(C(=O)CC2CSC2)CCC(C2CCCN2C(c2coc(Cl)c2)=O)C1 C1(NC(C2=CC(C)(CC)C2)=O)CCOC2(CCSCC2)C1 N1(C(c2cnc(OC)nc2)=O)CCN(C(=O)CCc2nccn2C)C(C)C1C C(=O)(CC(C)(C)C)NCC1(OC)CN(C(=O)Cc2ccc(Cl)nc2C)C1.S c1(C(C(=O)NC)N(C)C(c2ccc(C)cc2)C)nc(C(F)(F)F)cc(C)n1 Cc1cccc(C=O)c1.C1(C=O)C2CC(F)(F)CC12.[SH](C)(=O)=O.C1CC1.N Cc1ccc2c(C(=O)NCC3CN(C(C4CC45CC5)=O)C(C)(C)C3)csc2c1 C1(C(=O)NCC(CCC)OC)CCCC(NC(c2c[nH]nc2OCC)=O)CC1 c1(OC)cc(C(=O)NCCn2cc(C3C4COCC34)nn2)n(C)n1 CCN=c1[nH]cc(C(=O)NC2CCN(C(C3CC4CCCCC34)=O)CC2)s1 CC(C)CC(C)(O)C(=O)N(CC(C)NC(C1(F)CCC1)=O)C C(=O)(C(C)(C)NC(=O)C(C)N(C(=O)COCC1CCCO1)C)OC c1(C(=O)OC(c2cccc(OC)c2)C(=O)OC)c[nH]c2cc(Br)ccc12 C(=O)(CC(CC)C(C)C)NC1CC2CC(NC(c3c(CC)occ3C)=O)CC21 N1(C(c2n(C)ccn2)=O)CCC2(CC1)C(NC(=O)Cc1cnsc1)CS2(=O)=O c1(CNC(=O)CN2CCN(C(c3cncc(O)c3)=O)CC2)ccc([N+](=O)[O-])nc1 c1(C(=O)N)cc(C)c(F)cc1F.c1(OC)ccc(CC(=O)NC2CC2C)cc1 C(=O)(CS(=O)(=O)CC(C)C)NCC(C)NC(CCCCCC)=O C1(CC)CN(C(C2CC23CCCC3)=O)CCC1NC(c1c(C)oc(C)c1C)=O C12(CNC(CC(C)n3ccnc3)=O)CN(C(C3CCC(=O)O3)=O)CC(F)(C1)C2 C(CCC(C(=O)NCC1Cc2nccn2C1)NC(=O)C(O)CC(C)C)OC Cc1cncc(C)c1C(=O)NC(CC(=O)NC1CC1c1cncs1)C(F)F c1(CC)scnc1C(=O)NCCC1CN(C(C2CC2OC)=O)C1 C1(NC(c2ncc(CC)s2)=O)CS(=O)(=O)C12CCN(C(=O)C=CI)CC2 c1(CC(=O)N(CCOC)CCNC(=O)C(C)S)cc(C)on1.C(C)C N#Cc1ccc(NC(c2cnn(CC(F)(F)F)c2)=O)c2ccccc12 C1(CC)CCCCC1C(C(=O)NC1CCCCC1)N(C)Cc1nccn1C C1(NC(C2C(C=C)C2)=O)CCC12CCN(C(c1ncsc1Br)=O)CC2 N1(C(C2C(C)CC3CC3C2)=O)CC2CCN(C(=O)CCCCNC(N)=O)CC12 N1(C(CCSCCC)=O)CCCC2(CCCN2C(c2cc(CC)nc(O)c2)=O)C1 N1(C(C(CC=C)C)=O)CCCN(C(c2nc(OC)ccc2C)=O)CC1C C(C(CO)C(C)C)NC(C(Cc1cn[nH]c1)NC(c1ccc(C)o1)=O)=O Cc1cc(C(=O)N(C)CC2(C)CCCC2NC(=O)Cc2cnnn2C)c(C)s1 c1(C(N2CC(C)N(C(C)C)C(C)C2)C(=O)NCC=C)nc2cc(Br)ccc2o1 Cc1c(Cl)c(C(N2CCN(C(c3c[nH]c(=N)s3)=O)C(CC(F)F)C2)=O)nn1C CC1CN(C(c2cc(CO)[nH]n2)=O)CCC1NC(=O)CCN1CCOCC1 c1(CC)ccc(C(N2CCOCC2)=O)cc1.C1(C(=O)OC)(CO)CC1 C1(F)(C(=O)NCCC2CCN(C)C2)CCN(C(=O)CC2CCC(=O)NC2)CC1 C(=O)(CCCn1cc(CN2CCCC2)nn1)NCCC(C)OC c1(C(=O)NC2CC3CN(C(Cc4nc(=N)[nH][nH]4)=O)C2C3)cc2cccc(Cl)c2o1 c1(OC)cc(SC)ccc1C(=O)NCC(C1CCCC1)NC(=O)CO c1(C(CC)O)nc(-c2ccccc2OC(C)C)n(-c2cccnc2)n1 c1(CSCC(=O)NC2C(NC(C(c3cccnc3)C)=O)C2)ccncc1 N1(C(c2ccc(COC)s2)=O)CC(C)CCC1CNC(c1ncsc1C)=O c1ccc(S(N)(=O)=O)cc1N(C(=O)C(F)CC(C)(C)N)C1CCN(C)CC1.CO C(=O)(C(C)(C)C(F)(F)F)N1CCCC(O)(CCNC(C(CC)(C)F)=O)C1 C1(CC(=O)NCC2OCCN(C(CCc3ccc(C)s3)=O)C2)CCCCC1(C)C C(=O)(C(C)(C)CCCF)NC(C)CCC(=O)NCC(O)CC(F)(F)F C1(CC(=O)NCCNC(c2nn(CC(F)(F)F)cc2Cl)=O)CCCC1(F)F C1(CNC(c2cnc3sccn23)=O)C(C2CC2)CCN1C(=O)CCc1nncs1 C1(CNC(CC2(C)CC2(Cl)Cl)=O)CC2(CCN(C(c3ccsn3)=O)CC2)C1 CC1c2ccc(C#N)n2CCN1C(=O)C(O)(CN(C)C)C(F)(F)F N1(C(c2nc(C)oc2)=O)CCCC(NC(=O)C(O)Cc2[nH]cnc2C)C1C C1(C(=O)NCC(=O)NC)(C)CCCN(C(C2(c3ccccc3C)CCC2)=O)C1 c1cc(S(C)(=O)=O)ncn1.N1(C(C2N(C(C)(C)C)CC2)=O)CCC(C)(C)C1.N C1(C(N(C2CCN(C(CSCc3nc(C)sc3)=O)C2)CCO)=O)CC(C)CCO1 c1(C(C)S(N)(=O)=O)ccc(C(=O)NC2CCCC2)cc1.C(=O)(C)N.C1CC1 CCCCC(O)CC(=O)N1CCCCCCC1C(N1CCC(O)(C(F)F)C1)=O C1(C(=O)NC2C3CN(C(C4CCSCC4)=O)CC23)(OC)CCCC(C)(C)C1 N1(C(CC(=O)OC)=O)CCC2CCN(C(=O)Cc3cc(O)nnc3O)CC2C1 c1(C(c2nnnn2CCCF)NCC=C=C)cc(Br)c(F)cc1[N+](=O)[O-] c1(COCC(=O)NCC(CNC(COC(C)C)=O)C)cnn(C)c1 C1(C(c2nnnn2C2(C)CC2)NCC2CC(C)OCC2)C2CC3CC(C2)CC1C3 C(=O)(C(C)(C)C(=O)N1CCCCC1)OCC.C(=O)(C(F)CC1CCCC1)NC C(c1cnc2ccccc2c1)=CC(=O)NCC(c1ccc(Br)cn1)=O Cc1ccc(CNC(=O)Cn2ccnn2)cc1.C1(C=O)COC(=O)N1.CC.C C1(NC(c2cncc(OC)c2C)=O)COC2CN(C(=O)C(C#N)CC3CC3)CC12 C1(OC)CCCCN(CC(N2CCC(O)(CNC(=O)Cn3ncnn3)C2)=O)C1=O C1(C(=O)NCCC2(COC)CC2)C=CCN1C(=O)CCc1cncnc1 c1(-c2ncn(C)c2CN2CCC2c2ccccc2)ccc(Cl)cc1Cl CC(CC(=O)NC1CC2CCC1C(NC(=O)C1=COCC1)C2)C(F)(F)F c1(NC(c2cc(CNC(c3cncc(OC)c3)=O)ncc2)=O)nccc(C)c1Br N1(C(C(COC)(C)OC)=O)CCC2C(C(N3CCC(C)(C(=O)OC)C3)=O)C2C1 C(=O)(C1=CC(O)C(NC(c2nccnc2CC)=O)C1)N1CCCC(CCC)C1 c1(C(C(=O)NCC(F)F)N(CCC(=O)OCC)C)c(Cl)c(C)nn1CC C12(C(=O)NC(C)CCCNC(=O)CCS(C)=O)CCCN(CC1)C2 N1(CC(=O)N(C)C)CCC2(CCN(C(c3scnc3C(C)(C)C)=O)CC2)CC1 C1CN(C(C2CCC(C(N)=O)CC2)=O)CCC1(C)C.C(C(=O)NC)NC(C)=O c1(CC)c(C(=O)NC(C)(CNC(C2CCNC2=O)=O)C2CCC2)csc1C C=CC(CCC)CC(=O)NCC1(C(=O)NC)CC(=C)C1.c1[nH]ccc(=O)c1O C1(CNC(=O)CC(F)F)CC2(CCN(C(c3ccon3)=O)CC2)CO1 c1(CC)cnoc1C(=O)NC(C1CC1C(=O)N(C)Cc1ccoc1)C c1(-c2cc(C)sc2)ccccc1SC1CCCCC1 Cc1ccnc(C(=O)NCC23CC(NC(C4CC4(F)F)=O)(CO2)C3)c1 c1(NC)cc(C(=O)NC2CCCCC2)cc(Cl)n1.n1(CC(=O)N)nc(C)cc1C C(=O)(CS(=O)(=O)C1CCCC1)NC(CNC(C(CC)(F)F)=O)CO C1CC2CCC1N(C(C1C(C#N)C1(C)C)=O)C2.CC(C)CCCOCC(=O)N.C C1(NC(c2c(CC)c[nH]c2)=O)CCOCC1NC(C1CCN(CC)C1)=O CCCC(C(O)C(=O)NC(C)CC(C)C(F)F)NC(=O)Cc1cncnc1O N1(Cc2ccc(C(=O)OC)cc2)CCCC(C(=O)Nc2ccc(I)c(C)c2)CC1 C1(O)(CN(C(=O)CCN2CCC2)C)CCN(C(C2(C3CC3)CC2)=O)C1 N1(C(CSCCCC)=O)CCC2CC(NC(c3[nH]nnc3C3CC3)=O)CCC2C1 C1(NC(c2nc(OC)c(C)s2)=O)CN(C(C2C(C)C2C)=O)CC12CC2 N1(C(C(CCSC)O)=O)CC2(CC(CC(=O)N)C2)C1.c1cnn(CCN(C)C)c1 C1(C(C)C)CCC(C)CC1C(N1CC(C)(C)CC1CNC(C1CCOC1)=O)=O c1(C(N(CCCCCNC(c2cnc(C)nc2)=O)C)=O)ccn2nccc2n1 c1(C(C(C)NC(=O)C(O)C(C)C)NC(CC)=O)ccc(Cl)cc1Cl CCCCC(C(=O)NCCC(C)(C)O)NC(=O)C(CO)N(C)C c1(C=O)cc(F)cc2nn(C)cc12.C(CC(=O)NC)NC(=O)NC.C1CC1 N1(C(CSc2c(OC)cccc2)=O)CCN(C(=O)C=CC2CCC2)CC(C)(F)C1 C(Cc1cnc[nH]1)(C(=O)NCC1(O)CCCC1)NC(C=C(C)C1CC1)=O C1(C(N(C2CCN(C(c3ccn(CC#N)n3)=O)CC2)CCC)=O)CCC(F)(F)C1 C(=O)(CC(CC)C(C)(C)C)N.c1(C(=O)NC(CC=C)C2CC2)cc(C)ccn1 c1(C(=O)NCC2(CCNC(c3cc(C)ns3)=O)CC2)ccc(C#N)o1 C(=O)(CC(C)(O)C(F)(F)F)N1C(CNC(c2nc(COC)oc2)=O)CC1 C1(CCCCNC(CCOCC#C)=O)CCN(C(c2cn(C)nc2SC)=O)CC1 C1(C)(NC(c2cc(CC)n(C)n2)=O)CCC(NC(=O)CC(CC)OC)CC1 CC(C)C(O)CC(=O)N1CCC2CC12Cc1ccc(C2CCC3(CCC3)C2)cc1 S(=O)(=O)(c1cnc(Cl)n1C)N(C(C)Cc1ccc(F)cc1)C C1(CNC(CCC(=O)OCC)=O)CN(C(c2scnc2C)=O)CC12CC2 N1(C(CC(C=C)(C)C)=O)CC(NC(C2NC(=O)CC2C)=O)CC12CCOCC2 C[S+](C)CCC(O)C(=O)NCCCC1(NC(c2ccc(F)c(O)c2)=O)CC1 C(=O)(C(O)CC(C)C)N(CC(=O)NCCCC(=O)N(C)C1CC1)CC CC1CCC(Nc2ccc(O)cc2Br)CN1C(=O)OC(C)(C)C S(=O)(=O)(c1cccnc1N1CC2CC2(CO)C1)NCC(CSC)OC Cc1ccc(C(F)(F)F)cc1CN1CCOCC(Nc2ncc(C3CC3)cn2)C1 c1(C=O)nsc2ccccc12.c1(C(=O)NCC2CCOC2)cc(O)cc(=O)o1.N C#CCC(C(=O)OC)NC(=O)CN(C(c1cc(C)co1)=O)C(C)C C#CC1(C(=O)NCC2CCCC2NC(=O)CC2(C)CCCC2)CCOCC1 C1(CN(C(CC=C)=O)CC)CCC(C)CN1C(=O)COCc1ccccc1C CCCCCCC(C)NC(C1C=CCN(C(=O)CCc2nc(O)n[nH]2)C1)=O CSC=CC(=O)NCC(C)(C)NC(=O)CC1CCC1.C(C)(C)C.C(=O)O N1(C(=O)OC(C)(C)C)CC2(C1)CN(C(C1CCCN1C=O)=O)CC2C(=O)O N1(C(C2(F)CCC(C)CC2)=O)CCC2(CCN(C(C3(C)COC(=O)C3)=O)CC2)C1 N1(C(C2C(=C)CC2)=O)CC2(CC2)CC1CNC(C1CC(=C2CC2)C1)=O C=CCCCC(C)(C)C(=O)NCCCNC(c1ccccc1-c1ncnn1C)=O c1(NC2C(OCC)COC2)nc2c(c(=NCc3c[nH]nc3C)[nH]1)COCC2 Cc1cccc(CN(CCO)C(=O)NC2C3CN(CC(F)F)CC23)c1 c1(C(N2C(CCNC(C(CC#C)O)=O)CSCC2)=O)cc2ccc(O)cc2[nH]1 C#CC1(C(=O)NCCc2cc(O)ncn2)CCN(C(c2cncn2C)=O)C1 N(C(=NCCN=c1ccc(F)c[nH]1)NC1CC2(C1)CC(F)(F)C2)CC(C)C C(c1cnccc1C)=CC(=O)NC(CN(C(c1ccc(C)n1C)=O)CC)C C1(C(N(C)CC2N(C(c3c(C(C)C)ocn3)=O)CCCC2)=O)CCCCC(=O)N1 N1(C(C(CC)N2CCCC2=O)=O)CCN(C(c2nc(Cl)c(Cl)s2)=O)CC12CCC2 c1(SC)ccc(C(=O)NCC2CC2C)cc1.C(=O)C(C)Cc1ccncc1 Cc1ncnc(C)c1C(N1CC2(CCN2C(c2cc(C(C)C)n(C)c2C)=O)C1)=O C1(C(N2C(CNC(C3(C)CCOCC3)=O)CCCC2)=O)CN2CCN1CC2 C(=O)(C(C1=C(C)C=CCC1(C)C)N1CC2CC(C(=O)OC)C2C1)NC.C1CN1 C(CN=c1nc(NCc2ccc[nH]2)c2c([nH]1)CCOC2)(c1ccccc1Cl)OC c1(CC(=O)NC2C(N(C(C(=O)NCC)=O)C)CCCC2)ccc(OC)cc1 N1(CC(=O)N(C(C)C)C)C(=O)CCC1=O.c1(C(=O)N)csc(-c2ccccc2)c1 Cc1nnc(CN(C)C(C2C(NC(=O)CCC3CCCCO3)C2(C)C)=O)o1 Cc1nc(Br)c2ccc(C(=O)N(C)Cc3cn(CC4CCOC4)nn3)cn12 C(=O)(C1CCCc2nccn21)NC1(CC)CCN(C(c2cnsn2)=O)CC1 C1(N(C(C(C)=C(CC)C)=O)C)CC2CC1N(C(c1c(Cl)c(CC)nn1C)=O)C2 N1(C(C)=O)CCOCC(C(=O)NCC2CCC(=O)NC2)C1 C1(NC(CN(CCC)C)=O)C2CCN(C(=O)C(O)CSC)C12 c1(CNC(C2(C(C)C)COC2)=O)ccoc1C(=O)NC1CCC2CC12 C12(NC(C3CCN(S(CCC)(=O)=O)CC3)=O)CCC1CN(C(c1cn[nH]c1)=O)C2 Cc1ncc(C(=O)NCC2CCCN2C(c2cc(F)n(C)n2)=O)cc1C#N N1(C(C(C)CC#N)=O)CC2(CCC2)CCC1CNC(=O)Cn1ccnn1 C12(C(N(CCNC(=O)C(c3ccccn3)(F)F)CC)=O)CC1COC2(C)C c1(C(=O)N)cnn2cccc2c1.C=C(C)CCCCNC(=O)COC(C)(C)C c1(C(N2CC(CC)C(NC(C3CC3(Cl)Cl)=O)CC2)=O)ccc2nccnc2c1 c1(CNC(c2cnc(CC)[nH]2)=O)ccc2c(c1)CN(C(=O)CCCCCC#N)C2 Cc1ccc(S(=O)(=O)CC(C)N2CCC3(CC2)OCCCO3)cc1 C1(CC(=O)NCC2CCCN2C(=O)Cc2cnsc2)CCC2(CC1)CC2 C1(C(N2CC(O)(C(C)NC(CN(C(C)C)C)=O)C2)=O)CCOCC1(C)C C1(N2CC(OC)C(F)C2)CC2(CCN(Cc3ncn4ccccc34)CC2)C1 c1(C(C)C(=O)NC2(C)CN(C(=O)C=CCn3cncn3)C2)cc2ccccc2o1 C1(NC(c2n(CC)nc(C)c2)=O)CN(C(=O)COC2CCOC2)CC1(C)C c1(SC)c(C(N2CCOCC2CNC(=O)C(C)Cc2cnc[nH]2)=O)cccc1F Cc1c(CN2CC3(CCCN3C(c3cn[nH]c3)=O)C2)[nH]c2ccccc12 C1(NC(CCN(CC#C)C(c2csc(=N)[nH]2)=O)=O)CCCC(CC)C1 N1(C(CCC2N(C(Cn3cnc(=N)[nH]3)=O)CCC2)=O)CCS(=O)CC1 N1(C(c2c(C)nc(C)[nH]2)=O)CCCC2C(NC(c3ccncc3Cl)=O)C(C)(C)C12 CC1CC(NC(C2(N(C)C(c3nccn3C)=O)CC2)=O)CC(C)(C)C1 N(C1CCCc2ccoc21)C(C1CN(C(C(C(C)C)(C)C)=O)CC1F)=O N1(C(c2ccc(N(CC)CC)c(Br)c2)=O)CC2CN(C3CCC3)CC2C1 C1(C(=O)NCC2C(C)(C)CC2)CN2CCCN1CC2.c1(C(=O)N)snc(O)c1Cl Cn1c(C(=O)NCC2(C)CCN(C(C3(C)COC(=O)C3)=O)CC2)cccc1=O CC(C(=O)N(CCCCCNC(=O)CC1(C)CC(F)(F)C1)C)C(F)F C1(C(N2CCCC(NC(CCC#C)=O)CCC2)=O)CCCCN1S(N)(=O)=O c1(COCC(=O)N(C2C3CN(C(C)=O)CC32)C)cccc(C2CC2)c1Cl N1(C(CC2COCC(C)(C)O2)=O)CC2(NC(=O)Cc3n[nH]c(=N)s3)CCC1CC2 CC1OCCCC1C(=O)NC1C2CC(NC(c3cc(Cl)c[nH]3)=O)CC12 C1(CNC(c2ncc(OC)cn2)=O)CCCCCN1C(=O)C=CC1CCOC1 C12(NC(c3ccco3)=O)CCCC1(F)CN(C(=O)CC1COCC1O)C2 Cc1nc(C2CC2)ccc1C(N1CC2CC1CN2C(C12CCC1C2)=O)=O c1(C(=O)NC2(C3CCCO3)CCC2)cnn2ncccc12 C(=O)(CCS(=O)(=O)c1ccc(Cl)cc1)N(C)CC1(NC(CCC#C)=O)CC1 CC(C)S(C)(=O)=O.C(C1C(C=O)C1(C)C)=C(C)C.CC(C)(C)C.C(=O)C c1(N(C)Cc2c(CNC(C(C(COC)C)C)=O)cccc2)nc(C)nc(O)c1C C1(O)(CNC(c2cn(CCC)nc2)=O)CCN(C(=O)COCCSC)C1 C1(CC(=O)N)CC2C=CC1C2.c1(C(N(C2CCC(O)C2)C)=O)cn(CC)cn1 C(=O)(CC(C)(O)C)NCC1(C(N)=O)CN(c2cc(C(=O)OC)ncn2)C1 C(=O)(C(F)(F)CNC(=O)C(C)C1CCC1)N1CCC(CC(=O)NC)C1 c1(C(=O)OC)ccc(C(N2CC(C(C)NC(=O)C(c3ccccc3)O)C2)=O)[nH]1 c1(C(N(CCNC(C(C)C2CCCO2)=O)C2CC2)=O)cc2ncn(C)c2cn1 C1(CCCNC(C2(N(C(C3CC3(F)Cl)=O)C3CC3)CCC2)=O)CCOCC1 N1(C(c2n(CC#C)cnn2)=O)CCC2(NC(=O)CC3CC3)CCCCCC12 c1(CC(=O)NCC(CNC(CC(CCCC)O)=O)OC)c[nH]c2ccc(C)cc12 c1(C(N2CCCCC2CNCc2ccn(CCF)n2)=O)sc(Br)cc1Br N1(c2c(C)cnc(C)n2)CC2CCC1C1CN(C(=O)C3=CCCO3)CC21 CCCC(C(=O)OC)C(=O)N1CCCC(CC)C1C(=O)N(CC(C)(O)C1CC1)C n1(CC)nc(C)c(C(N2CCC(CO)C(NC(C3COCCO3)=O)C2)=O)c1Cl CCC(C(=O)N1CC(CNC(c2cnn[nH]2)=O)C2(CCC2)C1)C(C)(C)CC C1(C(=O)OCC)CN(CC(c2ccc3nnc(C)n3n2)=O)CCC12OCCO2 C1(C2CC2)(CNC(CN2C(C)CC2)=O)CCN(C(c2cn(C)nn2)=O)C1 C=CCC(CC)C(=O)NCCC1(C)CCN(C(=O)C(O)c2ccsc2)CC1 c1(OC)c(C(=O)NCC2CC23CCSCC3)ccnc1F C1(CC(=O)NC2(CNC(CCCOC(C)=O)=O)CCCC2)CCOC1(C)C N1(C(=O)Nc2ccc(OC)cc2F)CC2CN(C3COC3)CC2C1 Cc1cc(C(=O)NCC2(CC(=O)NOCC(F)(F)F)CC2)cc(C#N)c1 C1(C)CC(F)(F)CN1C(=O)CC1CCCO1.C1(N(C)C)CC(C(=O)NC)C1 c1(CC)cc(CC)c(S(=O)(=O)NCC(c2cc(Cl)ccc2Cl)O)c(CC)c1 N1(C(C(C2CCOC2)NC(C=C(C)C)=O)=O)Cc2cccc(C#N)c2C1 CC(CC(=O)N1CC=CC1CNC(C1CCC(C(F)F)CC1)=O)C(F)(F)F c1(C(N2CCC(C#N)C2)=O)cccc2ccn(C)c12.C(=O)(CNC=O)OCC C(=O)(CCCCC1CC1)N1CC(C(=O)NCCN2CCOCC2=O)(CC)C1 CC1CCN(C(=O)COCC2(N)CC2)CC1CO C(=O)(CCCC(C)(C)C#N)NC1CC(C(C)NC(C(n2ncc(C)c2)C)=O)C1 n1(CC)cc(C(=O)NC)c2ccccc12.C1(C(N2CCC2)=O)CCC2(CCC2)C1 C1(CNC(CC(C=C)C)=O)CCCCCN1C(=O)CC(C)(C)C CC(N=c1nc2c(ncn2C)c(NCc2cnc3n2CCCC3)[nH]1)c1cc[nH]n1 C1(C(=O)NCC(c2nncn2C)C)CC12CCC2.C(=O)C=CC(=O)N(C)C c1(CC)nn(C)c(NC2CN(C(c3ccnn3CC)=O)CC2C)c1[N+](=O)[O-] c1(CC(N2CC(F)CC(NC(C3C(=C)CC3)=O)C2)=O)c(C)[nH]c2ccnn2c1=O C1(CNC(c2scc(C)c2Cl)=O)CN(C(=O)CCc2ccnn2C)C2(CCC2)C1 N1(C(Cc2c(C)ccs2)=O)CC(O)CC1C(=O)NCCNC(C1CCC1)=O CC(CN=c1[nH]c(N2CCCC(n3cccn3)C2)nc2c1CCCCC2)C(F)F c1(CC(=O)NC(C)(C)C)ccc(CNC)cc1.c1ncccc1-c1ccccc1 Cc1ccc2ncc(C(N3CC(CNC(c4cnns4)=O)CC3C)=O)cc2c1 C=CC(CC)CC(=O)NC1CN(C(=O)C=Cc2cn(C)cn2)CC1F c1(C(N2C(CCNC(C(c3ccc(C)s3)C)=O)CCCC2)=O)ccc(N)c(O)c1 CC1CN(C(c2ccc(-c3ccc(F)cc3)cc2)=O)C(C)CN1C C(=O)(C(C(C)(C)C)NC(c1cn(C)nn1)=O)NC1CC(CC)OCC1 CCCC(C)CC(=O)N(C(C)CN(C)C(c1ccc(OC)nc1F)=O)C C(=O)(C(CO)N(C)C)NCC(CNC(=O)Cc1cccs1)OC Cc1cnc(C(=O)NCCCCCN(C(=O)Cc2sc(C3CC3)nc2C)C)nc1 c1(C(=O)OCC)ccc(N2CCC(C)C2C)nc1.C12(C=O)CC(CO1)C2.N CC(CC(=O)N1CC(F)(CNC(c2csc(Br)c2)=O)C1)P(C)(C)=O C1(CCC)CCCN(C(=O)COC(F)F)C1 c1cccc2ccccc12.C12(C(=O)OC)COC(CNC(=O)N)(C1)C2.CC c1(CC(=O)NC(C)CNC(C23CCC2C3)=O)ccc(O)cn1 N1(C(=O)CC2CCC(O)C2)CCCC(C(N2CCC(c3cc[nH]n3)C2)=O)CC1 C12CCC(CC1)C2.c1(CC(C(=O)N)N(C)C)ccc(O)cc1.C(=O)C=CCO c1(C(=O)NCC(CNC(c2cnc(C)o2)=O)CO)cc(F)cc2cc[nH]c12 N1(c2nccc(OC)n2)CCC(C(=O)Nc2cnc(Cl)c(Br)c2)C(O)C1 c1(C(=O)NC(C(C)NC(=O)COCCCF)C)noc2c1COCC2 N1(C(c2nc(Br)cs2)C(=O)NCCCSC)CCOC(c2cccnc2)C1 C=CCC(C(=O)N1CCC(C(N2CCCC2CC)=O)O1)OC Cc1ccc(CN2CCC2CNC(=O)Cc2c(F)cccc2Cl)c(C)c1 N1(C(CCc2cc(C)sc2C)=O)CC2CCN(C(=O)C=Cc3ccnn3C)C2C1 C1(NC(C(C)(C)OCC)=O)CC1C1CCN(C(=O)CC2CSCCS2)CC1 C(C(C)(O)C(=O)NCC1CCCN(C(c2cc(C(F)F)ccn2)=O)C1)OC C1(C(N(C)CC2(C)CC2)=O)CCC(CNC(=O)CCC2CCCN2C)O1 N1(C(COC(C)C)=O)CC(NC(C2CCC3(CCC3)CC2)=O)CCC(O)C1 Cn1cnc(CCNC(=O)C(O)C2CN(C(=O)CC3CSCCO3)C2)c1 c1(C(N2CCCC(NC(C3CCC34CCC4)=O)C2)=O)cc2ccncc2cc1F c1(CCC)nc(NC(=O)NCCOCCOC2(C)CCC2)sc1CC CC(CC(F)(F)F)C(=O)N1CCC2(NC(c3cncc(Cl)c3Cl)=O)CCCC12 C12(NC(=O)COCC(F)F)CCCN(C(C3CSC3)=O)CC1C2 C=C1CCN(C(c2cc(C(N)=O)[nH]n2)=O)C(C(=O)N)C1.C(C(C)C)c1ncc[nH]1 c1(OC)cccc(C(=O)NCC2C(C)CCN2C(c2cc(Br)co2)=O)c1F C1(C(=O)NCC(Cn2cc(CN(C)CCO)nn2)OC)CCCC1C C1(CNC(C(N2CCC(NC(=O)NC)C2)=O)=O)CC(=O)NC(C)C1 c1(C(=O)NC(C)(C)CCNC(=O)C(O)CC(F)(F)F)ccnc2c(F)cccc12 N1(C(C(C)CN(C(=O)CC(=O)NC2CC2)C)=O)CCC(C)(CO)CC1 CCC(CC(=O)N(CCC(C(C)C)NC(=O)C(O)CC1CCCC1)C)OC c1(N2CCC(C(C)(C)C)(CO)C2)ncccc1S(=O)(=O)NCCCN1CC=CC1 C1(NC(N2CCC(C3C(C(=O)OC)CCO3)CC2)=O)CC2(C1)CS(=O)(=O)C2 c1(N(CCC)C)ncc(C)cc1S(=O)(=O)NC1(C)CCCCC1C N1(C(C2C(OCC)CC2)=O)CC(C2CCCN(C(=O)C=CBr)C2)C1 c1(OC)ccc(C(C(F)(F)F)OC(c2ccncc2Cl)=O)cc1 c1(OC)ccc(C=CC(=O)NCCC)c(C)c1.c1(C=O)ccc(C#N)nc1O.N c1(CC(N2CC(C)(NC(=O)CC(O)c3ccccc3)C2)=O)ccc2nonc2c1 CN1CCC2(CC1)CN(C(=O)C(C)(C)C1CCCN1C(=O)CC1CCCCC1)C2 C(=O)(CCC(CF)CF)NC(C(N1CC(C)C(N(C)C)CC1)=O)(C)CO c1(C(=O)NC2CC3(C(C(NOC(CC)C)=O)C3)C2)cc(C#N)[nH]c1C Cc1ccc(CC(=O)NC2CC(C(=O)Nc3ncc(CCO)s3)C2)cn1 CCCCC(CNC(=O)CCC1CCN(C(=O)C(F)=C(C)C)C1)CC c1(OC)cc(C(=O)NC2CCCC(N(C)C(c3cc(CO)oc3C)=O)C2)nn1C Cc1cc(F)cnc1C(=O)NC1CCN(C(c2ccc(C3CCOC3)s2)=O)CC1 c1(C(=O)NC(CC#C)C(N)=O)cc(-c2ccncc2)nc2ccc(Br)cc12 c1(C(=O)NC(C)Cn2cc(-c3csnn3)nn2)ccc(OC(F)F)nc1 CCC(C)C(O)C(=O)N1CC(NC(c2cc(C)ncc2C)=O)CC1(CC)CC CCC(CCC(=O)Nc1ccc(OC)cc1)NC(c1ncc(C)cc1C)=O CCC(O)C(=O)NCC(C)(F)CNC(c1cc[nH]c1C1CC1)=O c1(C(N2CCC(C(C)NC(C3(C)CC3(F)Cl)=O)CC2)=O)c(O)cc(O)cc1O N1(C(C2CCCCC2)=O)CC2(C1)CN(C(=O)CC(C)C1CC1)C2.C(=O)(OC)N C1(C(=O)NCCN(C(CC)=O)CC(C)O)CCCC(N(C)C)C1 c1(NC(C2CN(C(c3cccc(F)n3)=O)C2)=O)cccc2c1CCO2 n1(CC(=O)N(CCCNC(C2(OC)CC2)=O)CC)cccc(C)c1=O C(=O)C(O)CC(C)C.Cc1[nH]nc(C(F)F)c1C(=O)NCc1ccc(C)cc1 n1(C(C(=O)N)C)cc2c(n1)CCCC2.C(C(O)CC)NC(CC1(CC)CCC1)=O C(=O)(C1CCc2cccc(=O)n21)N1C(CNC(CCNC(COC)=O)=O)CC1 CCCC(C)(O)CC(=O)NC1CCN(C(c2c[nH]c(=N)nc2C)=O)CC1F C(=O)(C(CC)C(=O)NC1CCCN(C(c2cc(Cl)n(C)n2)=O)CC1)OCC C1(CNC(C(C)Cc2cnn(C)c2)=O)CN(C)CCO1 C1(C)(C(=O)NC2CC(CC)OCC2)CC=C(C(C)C)CC1 C(=O)(CC(C)C(C)C)NC(CNC(c1nc(C)n(C)n1)=O)(C)C CCC(CC(=O)NCC1CN(C)CCN1C(c1n[nH]cc1C)=O)C(C)C Cc1cccc(OCC(=O)NC2CCN(C(=O)C(O)CN(C)C)C2)c1C C1(CCC)(NC(=O)C(=O)N)CCCN(C(C2CCCC(=O)N2C)=O)C1.C1CC1 N(C(=NCC1CCCOC1C(C)(C)C)NC)CC(c1cn(C)nc1)(C)O.C1CC1 n1(CC)c(SCC(c2ccccc2)=O)nc2c(F)cccc12 CCC(CC)(CC)C(=O)NC1CN(C(=O)CN(S(=O)(=O)c2ccccc2)C)C1 C1(CCC)CN(C(=O)Cc2ccccc2O)CC1C(=O)NCCC1CC1C N1(C(c2cc(OC)c(O)cc2)=O)CCC2OCCN(C(=O)CSC(F)(F)F)C2C1 C1(OC)CCCN(NC(=O)C(F)(F)c2ccnc(C)c2)CC1 n1(C2CC(C(N3C(CC(C)(C)C)CC3)=O)C2)cc(Cn2ccnc2)nn1 C1(C)(C(=O)OC)CCN1C(=O)C(C)CNC(=O)C(O)c1ccsc1 C(=O)(C(CNC(C1(C)CC(C)C1)=O)C(C)(C)C)NC(c1c(C)ncs1)C C1(c2cn(C(C)CO)nn2)CCN(C(=O)C(C)(O)C2CCC2)CC1.C1CCC1 N1(C(C=C2CCN(C)C2)=O)CCCC2(CCCCC2NC(=O)CCCCCO)C1 C1(C(N2CC(O)(CN(C)C)C2)=O)(C(F)F)CCOCC1 c1(C(=O)NC(Cn2cncn2)C(=O)NCCC2CC2)cn2ccccc2n1.C CC1CCCC(NC(=O)CCC2CC(NC(c3ccc(C#N)n3C)=O)C2)CC1 CC1CCC(NC(c2cccnc2S)=O)CN1C(=O)CC1(N(C)C)CC1 CC(C)(C(=O)NC1CCCC1NC(C1CC1C(F)(F)F)=O)c1cc[nH]n1 c1(CC(N2CC(CC=C)C2)=O)sc(CCC)nc1C.C1(C=O)CC1(C)C(C)C C(=O)(C1=NOC2(CCC2)C1)N1CC(C(=O)N)C2(C1)CCC2.CC1(C)CCCC1(O)C C1(C(=O)NCCN(CCC)C(c2ccc(N)cc2F)=O)CCCC(C)(C)C1 C1(NC(=O)COCCc2cccs2)CN(c2ncc(Cl)cn2)CC2(CCC2)C1 C1(C(=O)NC2CC(CCNC(C(C)c3cccs3)=O)C2)CC(C)(C)C1 C1(CNC(c2cnc(SC)[nH]2)=O)CC2CCCCC2N1C(c1cc(CO)[nH]n1)=O C#CCC(CC(=O)N1CC2C=CC2C1)NC(C1(COC)CC1)=O CC(C)(COCC(F)F)C(=O)NC1CCCC1.C1(C=O)CC2(CC2)CO1.C Nc1cccc(Cl)c1C(=O)NC1CCCC1CNC(=O)C#CC1CC1 C1(NC(C=CCCC)=O)CCC2(CC1)CN(C(=O)C(C(C)CC)OC)CCO2 C(=O)(C1=CC(C)CC1)N1CC=CC(NC(c2c(C)nsc2)=O)C1 c1(C(N2CC(CNC(C=NOC)=O)N(C)CC2)=O)nnc2ccccn12 c1(C(N2C(C)CCC(NC(c3csc(C)c3N)=O)C2)=O)cc(P(C)(C)=O)ccn1 N1(C(C=COCC)=O)CC2CC(NC(c3n[nH]c4c3CSCC4)=O)C(C2)C1 c1(OC)cc(NC(C2CCC(NC(C3CC(O)C3)=O)CO2)=O)ccc1C C1(C(=O)OCC)CC=CC(NCC2CCCN2Cc2cc(C)sc2C)C1 N1(C(CCS(N)(=O)=O)=O)CC(NC(=O)CC2CCCSC2)C2CCCC12 c1(OC)ccccc1CNC(=O)C(N1CCSCC1C)c1sccc1Br N1(C(C2C(NC(c3[nH]cc(C)c3C)=O)CCOC2)=O)CCC(F)(CO)CC1 C12(NC(CCC(N)=O)=O)CCN(C(c3cnc(O)n(C4CC4)c3=O)=O)CCC1C2 N1(C(CCOCCN(C(C(C)CC2CCC2)=O)C)=O)CCC(C)(N(C)C)CC1 N1(C(C)C)CCCC1C(=O)NC1CCC(C(=O)NCC(c2cccs2)O)C1 C1CC(C)(C)CCC1.n1(CC=O)ncn(C)c1=O.CC(C(F)F)=CC(=O)N.C c1(C(=O)NCCCNC(c2ncnc3c2CCC3)=O)cccc(C#CCO)c1 C(=O)(C(C)(C)C(=O)N1CCOCCC1)OC.C1(C(=O)N)CC(O)CN1C(C)=O c1(OC)cncnc1C(=O)NCC1(NC(=O)C(=Cc2ccco2)C)CCC1 N1(C(CC(CC)C(C)C)=O)CC(C2CCN(C(=O)C(C(C)(C)C)N(C)C)CC2)C1 N1(C(CCN(CC)CC)=O)CC(C)OC(C)(C)C1.C1(C(=O)N)CCC(=O)N1 CC1C(C(=O)N2CCCCCCC2C(=O)NC2CC3(C2)CC(O)C3)=NOC1C N1(C(C(C)n2ccnc2)=O)CCN(C(C2CCC(C)(C)OC2)=O)CC12CCC2 c1(C(=O)Nc2c(F)ccc(Br)c2F)cc2cc(-c3ccnc(F)c3F)ccc2o1 c1(C(=O)NC2CCCCCN(C(C=COCC)=O)C2)ccc2c(c1)NC(=O)CO2 CCC(C)(C)C(O)C(=O)NC(C1CN(C(=O)CCC2CCCC(=O)N2)C1)C C=C=CCN=c1[nH]c(=NC(C)c2cnn(C)c2C)c2ccc(C)cc2[nH]1 c1(C(N2CC(CN=c3cc(C)nc[nH]3)C(C)CC2)=O)cnc2c(n1)CCCC2 c1(C(C=O)N(CCC(N)=O)C(C)(C)C)cc(C(C)(C)O)on1.C(C)OC C=CCC(CNC(c1ccc(C(N)=O)[nH]1)=O)C(=O)N.C1CC(C(N)=O)=NO1 c1(C(N2CCC(n3ccnn3)C2)=O)cc(C)c(C)nn1.C(C(C)C(=O)NC)SC C(=O)(C(O)CCCNC(=O)CC1CCCC(=O)N1)N1C(CC)(CC)CCC1 C1(NC(c2cccc(CC)n2)=O)CCC(O)CN(C(C2OCC2(C)C)=O)C1 N=c1nc2ccc(C(=O)NC3CC34CC(NC(c3ccns3)=O)C4)cn2[nH]1 c1(NC2CCN(C(C(CCCC)O)=O)CC2)ncnc2[nH]cc(CC)c12 C1(NC(CC(C)c2ccccc2)=O)CS(=O)(=O)CC1N CCC(=O)CCC(=O)NC(C(=O)NC1CC(=O)N(C)C1=O)C(C)OC CCC(F)(C(=O)OC)C(=O)NC1CC(N(C(=O)Cc2ccc(F)c(F)c2)C)C1 c1(CNC(C2C(=C)C2)=O)cccc(C)c1.c1(C(C(=O)N)C)c(C)noc1C C1(CC(=O)N(C(C(=O)N(CCOC)CC)C)C2CC2)CCCN(C)C1 C1(N(CC#C)C(C2OCCC2C)=O)CCN(C(=O)CC(C)(C)OC)CC1 C1CCN(C)CC1.C(C1CCCO1)=CC(=O)N(C)CCOCC.C(=O)C.N C1(C(N(CCN(C(=O)C)CC)CC)=O)CCCC1O.C(=O)(C1CC1)N C1(CCCNC(C2(CC=C)CCCC2)=O)CN(C(=O)CC(C)OC)CCO1 c1(C(=O)NCC2(C)CCCN2C(C2CC(=C3CCC3)C2)=O)ccc(F)cc1Cl C1(C(N2CC(CNC(CN(S(CC)(=O)=O)C)=O)C(O)C2)=O)CCc2nncn2C1 C#CCC(C(=O)N1CCC(COCC)C1)NC(=O)CC(CC)OC C1(C(=O)NCCC(C)N(C(=O)COC2CCCCCC2)C)CCC2(CC1)N=N2 CN1CCC(C(=O)N(CCCNC(C2CCS2(=O)=O)=O)C)C1.c1ccccc1 c1(OC)ccnc(NCC(=O)NCCCCC(C)NC(c2n[nH]c(C)c2F)=O)n1 N1(C(c2cc(CC)on2)=O)CC2CC1(C(=O)N(C)C(c1cnn(C)c1)C)C2.C C(CC(C)C(=O)N(CC(C)NC(c1cccc(C2CCCC2)c1)=O)C)OC N1(C(C2(C)COC2)=O)CCCC(C2CN(Cc3c(F)ccc4occc34)C2)C1 c1(C=O)cc2c([nH]1)CCC2.c1(CS(C)(=O)=O)nc(CN2CCC(CC)C2)cs1 CC1(C)CCCCC1C(=O)NC1CCOC1c1ccc(O)nc1 C1(NC(C(CC#C)C)=O)CCCCN(C(=O)CSc2nccn2C)CC1 C1(C(=O)NC(C2CCN(C(CCC#C)=O)C2)(C)C)CN2CCCC1C2 c1(C(=O)NC(C(C)NC(c2nc(OC)c(C)s2)=O)(C)C)cc(C)ccc1C C1(CC(=O)N(CC(=O)NCC(C)C2CCC2)C2CC2)CCC(=O)C1C c1(OC)cc(S(=O)(=O)N(C2CN(S(=O)(=O)C3CCC(=O)CC3)C2)C)ccc1Br N1(C(c2cc(CC)on2)=O)CC(F)CC1C(=O)O Cc1cc(C)c(C(=O)NCC2CCC(NC(c3cnc(=N)[nH]c3)=O)CC2)cc1C c1(C(C=O)(C)C)ccc(F)c(F)c1F.CC1(C(=O)NC2CC2)CCC(=O)C1.C N1(C(C23CC(C)(C2)C3)=O)CCC(NC(C2CCC(=O)N2)=O)C(C)(C)C1 C1(NC(=O)CC2CC3CC3C2)CCN(C(c2nocc2Cl)=O)CC1 C1(NC(CCn2ncc(C)c2)=O)CCC2CN(C(=O)CSCC(N)=O)CCC2C1 c1(C(=O)NCC2C(C)(C)CN(C(c3ccoc3Cl)=O)C2)cc2cccnc2cn1 c1(OCC=C)cccnc1C(N1CC2C(CNC(=O)C(C)S)C2C1)=O.C N1(C(COc2ccc(C)cc2)=O)CC(NC(c2nnc(O)cc2O)=O)CC(C)C1 C12(NC(C(C)OCC)=O)CCOC(C1)C2.c1(C=O)cnn(C)c1C(F)F Cc1ccc(F)c2oc(C(=O)NC3CN(C(C4CC4C(F)F)=O)CC3O)cc12 C1CS(=O)(=O)CC1C(F)(F)F.C1(NC=O)CCCC1Nc1ccccn1.N N1(C(C(COC)(F)F)=O)CC2CC(C(=O)NCCc3ccc(F)nc3)C(C2)C1 C1(O)(C(=O)OC(=O)C=CCNC(=O)OC(C)C)CCCC1 Cc1cc(NC(=O)CCCC2CCCC2)ccc1NC(=O)CCSC(F)(F)F C=CCCCCC(=O)NC1CCC1CNC(c1ccc(C(F)F)c(F)c1)=O Cc1cc(Cl)c(C(N2CC=CC2CNC(C2CC3(CC3)CO2)=O)=O)cc1C CC1c2c[nH]nc2CCC1C(N1CC(CNC(c2cncc(F)c2)=O)C(C)C1)=O O(NC(=O)C(c1c(C)cnn1C)N(C)Cc1ccccc1)CC(CC)O c1(CC(=O)NC2CN(C(=O)OC)C2)c[nH]c2cnccc12.C12CCCN(C1)C2=O C1(NC(c2c[nH]nc2C(F)(F)F)=O)CCN(C(c2oc(C)nc2C)=O)CC1.CC Cc1cc(C(N2CC(C)(C(N3CCC(CC(N)=O)CC3)=O)C2)=O)cc(F)c1 c1(C(=O)N)ccc2c(c1)C(=O)CCO2.c1(CC(=O)NC(C)C2CC2)cccs1 c1(C(=O)N(C2CCCC(N(C(=O)C#CC3(C)CC3)C)C2)C)ccc(=O)n(C)c1 c1(C(N2CCCC(C)(NC(C3CCC(C)O3)=O)C2)=O)ccc2c(c1)NC(=O)CC2 C(=O)(CCCCCNC(C1CC(=O)C1(C)C)=O)NC1(C)CC(O)(CO)C1 C12(OC)CCC(C(=O)N)(CC1)C2.C1(CC)CCCN(C(C2CCC(C)CC2)=O)C1 C1(C(=O)NC(COCC)C(C)C)CN(C(c2ncc(C)cc2F)=O)CCN1C n1(CC)c(C(=O)NC2CC(C)(NC(=O)C3=COCC3)C2)cnc1O c1(-n2cc(CCC3N(C(c4nc(CC)sc4)=O)CCC3)nn2)cccc(F)n1 NS(=O)(=O)c1ncccc1NC(c1sc(Cl)cc1I)=O CCC(C)(COC)CN=c1nc(N2CC(=O)N(C)C(=O)C2)c2c(F)cccc2[nH]1 Cc1ccc2c(c1)C=C(C(=O)N1CC(C(C)NC(C3CCS3(=O)=O)=O)C1)CO2 C1(N(C(=O)CCc2cnc[nH]2)CC)CCN(C(=O)CC2CCNC2=O)C1 c1(C(=O)NC(CC(C)C)CNC(=O)C(c2cncnc2)C)cccc2c[nH]nc12 c1(OC)ccc(C(O)C(=O)NCC2(NC(c3sncc3C)=O)CC2)cc1 N1(C(C(=Cc2ccccn2)C)=O)CCN(C(c2ccc(C)nc2C)=O)CC1C c1(C(N2CCCC(C)(NC(c3cscc3Cl)=O)C2)=O)nccc2cc[nH]c12 c1(NC)ncccc1CCCNC(C)C(=O)NCc1ccccc1 c1(C(N2CC(CNC(C3CC(N(C)CC)C3)=O)C2)=O)cc(Cl)c[nH]1 C1(NC(CC(CCC)(C)C)=O)CCC2(CC1)CN(C(=O)CC(C)C(F)F)CCO2 C1(CC(=O)Nc2c(C(N)=O)n[nH]c2)CCCN(C(c2cc(=O)cco2)=O)C1 c1(C(=O)N)[nH]c2ccccc2c1Cl.N1(C(C(C)NS(C)(=O)=O)=O)CC=C(C)CC1 N1(C(CCCC#C)=O)CC(C)N(C(c2nn(C(C)(C)C)cc2Br)=O)CC1C C(=O)(C1=NOC(C)(C)C1)NCCCCOC.C1(C=O)CCS(=O)(=O)C1(C)C N1(C(COC(C)C)=O)CCOC2CCN(C(=O)C(O)C(F)(F)F)CC12 C=CC1(CNC(=O)N(C(CC)CO)C)CCOCC1 C1(CNC(C2(CCNC(CNC(N)=O)=O)CCC2)=O)CC12CC2(F)F c1(C(=O)NC2CCCC(C(=O)NCc3ccc(C)s3)CC2)ccc2c(c1)CCC2 C1(N(C(C(CO)OC)=O)C)CCN(C(=O)CC2COCCOC2)CC1C c1(OC)cccn2ncc(C(N3CC(NC(c4cccnc4C)=O)C(O)C3)=O)c12 N1(C(C(C)(C)O)=O)CCC(C2CCN(C(c3cnsc3)=O)C2)C1 c1(OC(C)CON)ccccc1OC(=O)C(C)(C)C C(N=c1[nH]c(=NCc2nncn2C)[nH]c2ccc(Cl)cc12)c1c(C)nccc1 CC(CC(C)NC(=O)CC1CCC1)NC(c1cc(F)c[nH]1)=O Cc1cc(C(N2CC(NC(=O)C=Cc3ccc(C)s3)C3CC23)=O)c(C)cn1 C1(NC(CC=CC=C)=O)CN(C(=O)CC(C)c2ccccc2)CC1(C)C c1(OC)cc(CNC(c2nc(-c3cccnc3)no2)C)cc(C(F)(F)F)c1 c1(C=O)coc(S(C)(=O)=O)c1.C1(C(=O)NCCCC)CC(S(C)(=O)=O)C1 N1(C(=O)Nc2cn(CC(=O)OC)nc2)CCCCC1c1ccccc1 CCC(C)CC(C(=O)N1CCC(O)(CC)C1)NC(=O)C(O)CC1CCCC1 C1(N(C(c2ccc(CCC)s2)=O)C)CCCC(NC(=O)CC2COCCOC2)C1 CC1CCCN(C(=O)C(CNC(c2ccn(C)c2)=O)CC2CC2)CC1 C=CCC(CC(=O)N1CC=CC(OC)C1)NC(c1n[nH]cc1Cl)=O C1(C(=O)NC(c2onc(C)n2)C)(CNC(C2CCC2(F)F)=O)CCCCC1 C(=O)(C(CC(F)F)C1CCC1)NC1CC(C)(NC(C(C)Cc2ccncc2)=O)C1 C1(NC(C2N(C3CCN(C(CCCNC)=O)CC3)CCC2)=O)CS(=O)(=O)CC1O N1(c2c(C#N)nccn2)CCn2ncc(CNC(C3(n4cncn4)CC3)=O)c2C1 N1(C(c2c(C#C)c[nH]n2)=O)CCN(C(=O)Cc2cc(C)nc(O)c2)CC1CCC CCCCN(OC)C(=O)NC(c1ccc2cc[nH]c2c1)C C1(CN(C(=O)Cc2cc(C3CC3)on2)C)CCCN(C(C2CCC2)=O)C1 Cc1cnc(N(C)Cc2cccs2)c(S(=O)(=O)N2CCOC(CCF)C2)c1 c1(OC)nn(C)cc1C(N1CCCC1CCNC(c1coc(Cl)n1)=O)=O C1(CNC(c2ncsc2Br)=O)CCCCC1(F)F C1CCN(C(=O)CCN2CCCS2(=O)=O)CC1.C(C(=O)N)NC(=O)OCC c1(SCC)cccc(C(=O)N)c1.C1C=CCC1.C(=O)C=O.CC(F)(F)F.C C(C)(CCCCNC(=O)CC1C=CCCC1)NC(COCCCC(C)C)=O N1(C(C(CCC)OCC)=O)CC(N=[N+]=[N-])CC1C(=O)NC1CC2(CCCCO2)C1 c1(C(=O)OC)c(F)cccc1NN1CCC(N(CCO)C(=O)OC(C)(C)C)CC1 C1(NC(CCSCCCC)=O)CCC(C#N)C1 CCCC(F)(F)C(=O)NCC1CCC(C(N2CCC(N(C)C)C2C)=O)CC1 C1(CC=O)CCCC2(CCC2)O1.c1(CC)ccc(F)cc1C(=O)N.C(C)(C)C CC(CC(=O)NC1CCCC1)NC(C1(C(N)=O)CC1)=O c1(C(N2CC(NC(c3c(C)ccnn3)=O)C(C)CC2)=O)cc2cccc(Cl)c2[nH]1 C(C(C)C(F)C(=O)NCCC(=O)N1CC(C(C)(C)C)C1)NC(COC)=O C(CCCCCNC(=O)C(O)C(C)OC)NC(c1c(CC)cno1)=O C1(NC(C=Cc2ccc(C)s2)=O)CCC(C)N(C(=O)CC2(O)CCC2)C1 C(CCCCCCCCO)NC(=O)C(F)(F)C1CCNC1 N1(C(c2cccc(C)c2)=O)CCC(C)C(NC(=O)CC2CC3CCC2C3)C1C CCC(CC(F)F)C(=O)NCC1CC2CN(C(c3nccc4[nH]ccc34)=O)CC12 c1(OC)cc2ncnc(NC3CCC(SC(C)C)C3)c2cc1OC c1(CCC)cccc(C(N2CCN(Cc3ncc(C)s3)C2)=O)c1 c1(NC(C)CCNC(=O)CC2CCS(=O)(=O)CC2)c(Cl)cccc1[N+](=O)[O-] N1(C(c2ccc(N)cc2)=O)CC2(CCCC2NC(C2CCOCC2)=O)C1 n1(CCC)c(C)cc(C=CC(N2CC(NC(c3ncn(C)c3C)=O)C2)=O)c1C c1(NCC(=O)NCCCN(C(CC)CO)CC)ccccc1OC n1(CC(=O)NCCC2(CCCO)CC2)cc(COc2ccccc2)nn1 Cc1ccc(C(=O)NC2CCN(CCC3CCNC(C)C3)CC2)cc1 c1(C(C(N2CCOCC(NC(C(CC)O)=O)C2)=O)=O)cc(S(N)(=O)=O)cn1C N1(C(C2N(C)C(=O)OC2)=O)CC(C2CCCN(C(C3CC4CCC3CC4)=O)C2)C1 C1(NC(C(CC)N(C)Cc2ccccc2)=O)CCCN(C(C2CC(OC)C2)=O)CC1 CCC(CC(=O)N1CC(C)(C)C1)N(C(=O)CCC(C)OC)C c1(C(=O)OC)cc(C#N)cnc1N1CCC(O)(C(C)NC(c2ccoc2Cl)=O)C1 CCCCCCCCCCCC(O)C(=O)NC(COC)C1CC1 C(=O)(CCCCCCCC1CC1)N(CC(C)(C)NC(=O)CC1CCC(C#N)C1)C N1(C(COC2CC(NC(c3ccccc3)=O)C2)=O)CC2(CCC2O)C1 CC(C)CC(O)C(=O)NCCC1CCC(NC(c2ccc(O)nn2)=O)C1 c1(N2CCC(C(=O)NC(CNC(C(C)C)=O)C(C)(C)C)CC2)ccccc1C#N C(CCCCC(=O)N1CCCC1C(C)NC(C1(C)CC=CCC1)=O)SC C#CCCCC(=O)NC1CCCCC1NC(=O)C(c1cccc(Cl)c1)N(C)C c1(C(=O)NC2CCCN(C(CC(=C=C)C)=O)C2)coc2c1C(=O)NCC2 C(CCCC(=O)NC(C)C)NC(C(=O)N(c1nc(C(C)N)[nH]n1)C)=O N1(C(C(C)N(C)C)=O)CC(NC(=O)C(C)N(CC(F)(F)F)C)C(C)(C)C1 c1(SC)cccc(NC(=O)CC2CCCN(C(C34CCC(CC3)C4)=O)C2)c1 N1(C(=O)Nc2ccc(Oc3c(C)cccc3)cc2)CCC(C2CCCNC2)C1 C(=O)(C(C(C)C)OC)N1CCC(C(C(=O)NCC(CC)CC)(C)C)C1 C1(CNC(=O)C2=COCC2)CCCN(C(C2CC3(C2)CC3(F)F)=O)CC1 n1(CCNC(CNC(CC)=O)=O)cc(C(=O)NCC2CCCN2C)cn1 C1(NC(c2cc(C3CC3)[nH]n2)=O)(CO)CCCN(C(=O)Cc2c[nH]ccc2=O)C1 c1(C=O)ccc(C(C)C)cc1F.C1(COC)CN(C(=O)Cn2cc(C)cn2)C1 c1(C(N2CC(C)(C)C2c2ccccc2)=O)cc2cc(N)ccc2o1 C1(C=O)CCCC12CC2.c1(C(N(CC)CC)=O)ccccc1N(C)C(C)C.N CCCC(C)CC(=O)NC1CCN(C(=O)C=Cc2cncc(O)c2)C(C)C1 c1(SCCC(=O)NCC(CC)NC(C2CCCCO2)=O)cc(F)ccc1F n1(CC2CCCN(CC3CCS(=O)(=O)C3)C2)cnc2ccccc12 c1(C(=O)NCCCNC(C2(CC)CCCC2)=O)ccnc2[nH]c(O)nc12 N1(C(c2cc(C)sc2C)=O)CCC2CCC12CNC(=O)C(C)(C)CF Cc1cc(CCC(N2CCC(N(C)C(c3cnsc3C)=O)C2)=O)n[nH]1 C(CO)(C(C)(C)CO)NC(C(Cc1ccoc1)NC(c1[nH]cc(C)c1C)=O)=O N1(C(Cc2cccc(C#C)c2)=O)CCC2CCCN(C(=O)C=C(C)CCC)C2C1 C(CCCCC)N(C(CN(C1CC1)CC)=O)C.C1(C(=O)N)CCC1n1cccn1 CCC(CC)C(F)C(=O)N(C)CC1(O)CN(C(=O)Cn2ccc(C3CC3)n2)C1 N1(C(CC2(C=C)CN(C(=O)C=CC3CCOC3)C2)=O)CC2(CNC(=O)N2)C1 C(=O)(C1CCCc2cnn(C)c21)NCC(C(CC)C)OC N1(C(CC(C)SC)=O)CCCN(C(=O)CCC2CC2)CC1CO C(CO)(C(=O)NCC1CN(C(c2cscc2Br)=O)C1)N(C)C C1(COC)CN(C(=O)C(C2CN(C(=O)OC(C)(C)C)C2)OC)CCO1 C(=O)(C(=O)N(CC)CC)NCC.C1C(C)=CC(=O)N1 c1(OC)cc(F)c(C(=O)NCC(CO)NC(=O)Cc2cc(C)ccc2C)cc1N n1(CC)nc(C(=O)NC(C)CCN(C)C(c2ccnn2CC(F)F)=O)cc1O N1(C(Cc2cc(OC)no2)=O)CC=CC(NC(c2ccnnc2)=O)C1.C(C)(C)O c1(C(=O)NCCC(C)CC)cc(S(N)(=O)=O)co1.C1(C(=O)N)CC2CCC1O2 N1(C(c2ccc(=N)[nH]n2)=O)CCCC(NC(=O)CCCOC2CCOCC2)CC1 C(C(C(C)(C)C)NC(C1CCCC(C(N)=O)C1)=O)NC(CC(=O)OC)=O c1(NC(C)CNC(c2ccc(=O)n(O)c2)=O)cc(C#N)c(F)cc1[N+](=O)[O-] c1(OC)ccc(C(N2CC(CNC(c3csc(C)c3C3CC3)=O)C2)=O)nc1 c1(-c2cn(C(C)C(=O)N(C)Cc3cc(C(C)(C)C)n[nH]3)nn2)ncccc1C#N c1(C(=O)NCC(C)NC(=O)CS(=O)(=O)C2CC2)csc2ncnc(O)c12 C1(C(C)C)(C(=O)NCCn2cnc(CO)c2)CCN(C(C2CC(F)C2)=O)C1 C(CCCCCNC(=O)CC1CCCCC1NC(=O)C(C)C)OC.C(C)=O.O c1(-c2cc(C(=O)OCC3CC34CC4)n[nH]2)ccc(Cl)cc1 c1(C(N(CCC)C)=O)cc2c(s1)CN(C)CC2.CCC(C)C(=O)NCC(=O)N Cc1ccc(C(=O)NCCCCC(C)NC(C2CCC(=O)NC2)=O)c(N)n1 C1(NC(COCc2nnc(C)s2)=O)CCN(C(c2cccc(C#N)n2)=O)C(C)C1 C1(CC=O)C=CS(=O)(=O)C1.c1(C=O)cc(C(=O)C(C)C)c[nH]1.CCCC.N C12(C(=O)NCC(CC)CC)CC1CCN2C(C1CC(OC)(OC)C1)=O C1(NC(C2(CCC)CCC2)=O)CCN(C(C2CCC2)=O)CC1C.C(C)(C)(C)O c1(C(=O)NC2CCC(C)N(C(=O)CC3=CCCCC3)C2)cnn2ccccc12 C12(C(=O)NC(c3cnn(C)c3)CC)CCCC1CCN2C(=O)C1=CCCOC1 C1(C(=O)NCC2(NC(c3n(CC)ccc3)=O)CCC2)CN(C)CC(C)O1 N1(C(C(CC)=CCC)=O)CCC(C)C(CC(=O)NC)C1.n1(C2CC2)cccn1 Cc1nn(CC(=O)NC(c2ccnn2C)C(=O)NC(c2csnn2)C)c(=O)o1 CC1CC2(CO1)CN(C(c1ccc(Cn3cc(CCC(N)=O)nn3)cc1)=O)C2 C1CN(C(C2CC2(C)C(F)F)=O)CC1N(C)C.c1(CC)cc(C(=O)N)n[nH]1 c1(C(=O)NCC2C(NC(Cc3c(OC)cccc3)=O)C2)cc(N)nc(Cl)c1 C1(C(=O)NC(C2(O)CCCCC2)C(=O)N(C2CC2)C)CC(=O)C1(C)C.C c1(C(N(CC(C)C)CC(=O)NCCc2ncnn2C)=O)ccc(F)c(O)c1 c1(C(=O)Nc2ccc(NC(CCC#C)=O)nc2)cc(F)c(F)c(O)c1F C1(C(=O)NCC2N(C(C=Cc3n(CC)ccn3)=O)CC2)CCCC(C)(C)O1 C1(S(C)(=O)=O)(C(N(CCCC)C)=O)CCOCC1.c1(CCC=O)cnc(O)[nH]1.N C(=O)(CCC(C)(F)F)N1C(C(C)(C)NC(c2c(CC)c[nH]c2)=O)CCC1 C(=O)(C(C)(O)C(F)(F)F)N(C1CCN(Cc2ncc(C)c(Br)c2)C1)C C(c1cccc(O)c1)=CC(=O)N(CCC)C.c1(C(=O)N)ccc(C2CCOC2)s1 N1(C(COCCCN(C)C)=O)CC(C2CCN(C(C3(C4CC4)CC3)=O)CC2)C1 c1(OC)nn(C)cc1C(=O)NC1CC(F)(F)C1.C1(C=O)COCC(C)O1.C C1(C)(C=O)CCCCC1C.c1(C(N(CC(COCC)O)C)=O)cc(C)cs1.N N#Cc1ccc(S(=O)(=O)N2CCC3(CC2)CC3NC(=O)CCc2ccoc2)cc1 C1(C)(OC)CC(NC(=N)NCc2cc(C3CC3)on2)C1(C)C c1(CC(=O)NCC(C2CC2)NC(C(CC=C)(F)F)=O)cccc2sccc12 N1(CC)CCCC1C(N1CCC(N(C(=O)Cc2ccsc2C)CC)C1)=O C(CCCNC(=O)CCN(C(=O)CCC1CC1)CC1CC1)OC(C)C c1(COC)nc(NCC2CCOCC2)cc(=NC2CCCc3sccc32)[nH]1 N1(CC(=O)N(CCC(N2CCC(C3CCCO3)C2)=O)CC=C)C(=O)CCCC1=O c1(C(N2C(CC(=O)NCCC3CCCOC3)CC2)=O)cn2ccccc2n1 c1(C(=O)NC2CCN(Cc3ncc(CC)o3)CC2C)c(C)[nH]c2ccccc12 C1(NC(C(N2CCOCC2)C)=O)CC2CC(C1)N(C(C1(O)CCCCC1)=O)C2 C(=O)(C(C)(C)NC(c1cnn(C)c1)=O)NCCC1C(C)C1 C12(NC(C)=O)CCN(C=O)CCC1C2.C(C[Si](C)(C)C)OCC.CC.CC.O CC(C)CCC(=O)C(=O)NCC1(C(=O)NCC(C)(C)C(C)(F)F)CC=CC1 c1(C(=O)NCC2(O)CCN(C(c3c[nH]c(=N)o3)=O)C2)cncc2ccsc12 NS(=O)(=O)c1ccc(C(N2CC(NC(=O)C(O)C(F)F)C3(CCC3)C2)=O)cc1F c1(C(=O)OC2CCC(OC)C2)cc(C)n(-c2nc(C)cs2)c1C N1(C(CC(C)n2ccnc2)=O)CC(NC(=O)C(F)(F)C(C)O)CC12CCOCC2 N1(C(C(Cc2cn[nH]c2)NC(C(CC)OC)=O)=O)C2CCC1CC1(CC1)C2 N1(C(C2(C(=O)OCC)CC2)=O)CCN(C(c2cnn3c2OCCC3)=O)C(C)C1C Cc1cccc(C2CCCN2C(=O)NCc2ccccc2N2CCN(C)CC2)c1 CCCC(C)(O)C(=O)N1CC(CNC(=O)CC(C)(C)COC)C(F)(F)C1 C1CCS(=O)(=O)C2(C1)CCC2.c1(C(C)=O)ccccc1.CC(C)(C)OC(=O)N c1(C(N(c2cc(C)c(Cl)cc2)c2ccccc2)=O)ccn2ncnc2c1 c1(C=O)c(C)cc(=O)oc1C.N1(C(C(C)NS(CC)(=O)=O)=O)CCC(C)C1.C n1(CCCOC)nc(C(=O)NC2(CF)CCN(C(=O)C)C2)ccc1=O.C1CC1 c1(OC)csc(C(=O)NCC2(F)CCC(NC(C3C4CCCC34)=O)C2)c1 C1(Cn2c(-c3n[nH]c(C)c3Cl)nc(CCOC)n2)CCC(F)(F)CC1 n1(C(C(=O)N(C(C)C)CCN(C(=O)CS)C)C)cnc2ccccc12.C1CC1 CCC(C(=O)NCCOCCn1ccnn1)NC(C)=O.C(C)C(=O)O.C Cc1cc(C(N2CCCCC2CNC(=O)C=CC=C(Cl)Cl)=O)n(C(F)F)n1 CCN=c1cc(C)nc(NCC2CCCC2N2CCN(C)CC2)[nH]1 C(=O)(C(CNC(c1cc(OC)n[nH]1)=O)CCC)NCCCCCC CCC(CC(C)O)NC(C1(CCNC(=O)CSc2nc[nH]n2)CCC1)=O C1(C(=O)NC2CC(C(=O)NCCCOCC)C2)CCC(N=[N+]=[N-])C1 CC(C)(CNC(C1(CCNC(C2(C)C=CCC2)=O)CC1)=O)CO C1(NC(C(c2cnn(C)c2)NC(C2C(C)C2C)=O)=O)CC2CC(O)C1C2 C=CCC(C)C(=O)N1CCCC1CN(C(c1cn(C)cc1C)=O)C1CC1 C1(CNC(CCCc2cc(C)no2)=O)C2CCCC1N(C(=O)C(C)(F)F)C2 c1(OC)cc([N+](=O)[O-])c(Cl)cc1S(=O)(=O)Nc1cc(Br)cc([N+](=O)[O-])c1 N1(C(C(CC=CCC)C)=O)CC(NC(c2cccc(OC(F)F)n2)=O)C(C)(C)C1 N1(C(CC2(OC)CCCCC2)=O)CCC2CC1CN(C(=O)Nc1cnoc1C)C2 C1(C(=O)NCC2COCCN(C(CSC)=O)C2)COc2ccc(Cl)cc2C1 C1(CC)CCOC1C(=O)N(CCCC(=O)NCCn1ncnn1)C C1(CCC)CN(C(C2C3CCCOC23)=O)CC1NC(C1(C)CCCOC1)=O N1(C(C2CCCOCC2)=O)CC2OCCN(C(C3CC3[N+](=O)[O-])=O)C2C1 C(=O)(C(C)S(N)(=O)=O)N1C(C(N(C)CC2(OC)CCC2)=O)CC(C)C1 C(C)(CC)(C(N)=O)NC(CCCNC(CC1CC(CC)C1)=O)=O N1(C(C2(C)COCCO2)=O)CC2CN(C(c3cc4occc4s3)=O)CC2C1 Cc1cc(C(N2CC(CC)OC(C)C2)=O)c(N)c(Cl)c1.N1(CC(=O)N)CC=CC1 c1(C(C)NC(C2(CF)CC2)=O)cccc(NC(=O)CC2COCCO2)c1 CC1(C)CC(=O)NC1CNCc1nc(-c2cccnc2)cs1 C(=O)(C(C)c1ccco1)NCC=CC(=O)NCC(=O)NCC(C)C C1(C(N2CC(O)(CNC(C=CC=CC)=O)C2)=O)Cc2cccc(F)c2O1 CN1CCc2nc(O)c(C(=O)NC34CC3CN(C(=O)CNC=O)C4)cc2C1 C(C(C)(CC(C)C)NC(c1ccc(C(F)F)cn1)=O)NC(CCN(C)CC)=O c1(C(=O)OC)ccc(S(=O)(=O)N2CCC(c3ccn(C)n3)CC2)cc1Cl c1(N(C(CNC(C2C(CC)CCC2)=O)C)C)ncnc2cccc(F)c12 C1CN(C(c2cnn(C3CCC3)c2)=O)CC(C)(C)C1.CN1C(=O)CCC1C(=O)N CC(CNC(c1cnc(S)[nH]1)=O)(CO)NC(c1cc(F)c[nH]1)=O Cc1cc(C(=O)NCC(C)NC(C2CC23CC(O)C3)=O)c(F)cc1Cl N1(C(C(C(C)C)O)=O)C2CCC1CC(N(C)C(c1cn(C)c(=O)cn1)=O)C2 N1(C(CCC#C)=O)CC2CCCN(C(c3ncccc3Cl)=O)C2C1 C(c1ccccc1F)=CC(=O)NC(CNC(=O)C(O)C1CC1)C1CCC1 c1cnn2c1CN(C(=O)C=Cc1cc[nH]n1)CC2.C(C(=O)NC)N(C1CCC1)C N1(C(CNC(c2ccccc2)=O)=O)CCC(O)C(C(N2CC3CCC2CO3)=O)C1 C1(NC(C2C(C)C2)=O)CCN(C(=O)C=Cc2ccnn2C)CC1F C(C)(CC(C)(C)OC)(c1n(CCCC)nnn1)NC1CC2C(C1)C2(F)F c1(N2CCCC(CC(N)=O)C2)[nH]c(=NCC(Cl)(Cl)Cl)nc2scnc12 N1(C(C2CC(NC)C2)=O)CCC(C=CC=O)CC1.C1(C(N)=O)CCOC1.CC C=CC1CN(C(=O)Cc2cnn(C)c2C)CC1NC(=O)CC(C)C1CCCCC1 N1(C(C)=O)CCC(C)(NC(C2COCCC2)=O)CC1.C(=O)(C(F)=CC1CC1)N O=C1OC(C(N2CCC(OC=O)CC2)=O)Cc2ccc(F)cc21.C12CCCN1CCC2.N C1(NC(Cc2nc(C)oc2)=O)CC=CCC1C(=O)NC12CC(C1)C2 C1(C(C)(C)C)CN(C(=O)C2=COCCC2)CCN1C(=O)C=Cc1cccc(O)c1 C(=O)(C(CNC(=O)C(OC)OC)N(C)C)N(CC=C)CC1CC1 C1(NC(C2(NC(C3(CCOC)CC3)=O)CC(F)C2)=O)CC2CCC1C2 c1(C(N(C(C)C(N2CCCC(C)C2CO)=O)CCC)=O)nnc(O)nc1O C(=O)(CCCCCC#N)N1CC(N(C(=O)COCP(C)(C)=O)C)C2(C1)CC2 C1(C(N2CC(CNC(C3(OC)CCC3)=O)C(O)C2)=O)CCC2(CCOCC2)CO1 c1(C(N2CC(C(=O)NC(C)C)(CO)C2)=O)ccc2ccnn2c1.C1CCCC1(C)C C1(C(NOC(CC)C)=O)CN(C(c2cn(Cc3ncccc3C)nn2)=O)CCO1 C(=O)(CC(C)CC(F)(F)F)NC1CN(C(CCOCCOC)=O)C(C)C1 c1(C(=O)NCC2OCCC(NC(c3cc[nH]n3)=O)C2)cccc(Cl)c1F Cc1cc(=NCC(C)NC(c2cnn3c2OCCC3)=O)[nH]cn1 Cc1c[nH]nc1C(=O)N(C)CCOCCCC.C(=O)(CC(C)c1ccncc1)N c1(N(C)Cc2ccc(C)s2)nnc(-c2cccn2C)n1CC(C)(O)c1ccco1 CCCCCS(=O)(=O)CC(=O)N1CC(N(C)C(C23CCCC2(C(N)=O)C3)=O)C1 CC1CCCCN1CCC(=O)Nc1cccc(C(C)(C)C(=O)N(C)C)c1 C(C1CCCN1C(=O)CC1CC1)=CC(=O)NCC1CC2CCC1O2 c1(C(N2CC(CCNC(CCN3CCN(C)CC3)=O)C2)=O)cccc2c1CCC2 S(=O)(=O)(c1ccncc1)NC1CCC(C(N2C(CCOC)CCCC2)=O)OC1 c1(CC)ccc2cc(C(=O)NC3C(NC(c4cc5sccc5s4)=O)C3)ccc2c1 C1(CNC(C(=O)NCC(C2CCC2)OCC)=O)CC(OC)C(OC)C1 c1(C(=O)NC2C(NC(C(C)(C)OCC)=O)CCCC2)nn(C)c(=O)cc1C N1(C(c2ncc(Br)cc2F)C(=O)NCC(=C)C)CC(C)NC(=O)C1(C)C N1(C(C=CSC)=O)CCC(O)(C(C)NC(=O)CC(C)n2ccnc2)C1 C(=O)(C1=CCC(C)(C)CC1)N1CC(N(C)Cc2cn[nH]c2)C1.C1CC(F)(F)C1 c1(CCCNC(C(C)NC(COC(CC)CC)=O)=O)ncn(C)n1 Cc1cc(C(=O)OC(C)C(F)(F)F)c(C)c(C)c1 C1(O)(C(CNC(C(F)=C(C)C)=O)C)CCN(C(=O)C(c2ccccc2F)F)C1 CC1(C)CCCC(CN(C=O)CC2CC3(CCCO3)C2)C1 c1(C(=O)NCC(=O)Nc2cc[nH]n2)ccc(=NCc2ccc3nncn3c2)[nH]c1 Cc1coc(C)c1C=CC(N1CC(NC(c2cc(N)ccc2Cl)=O)C(C)C1)=O C1(C(=O)Nc2c(I)ccc(C)c2)CCC2(CN(C(c3cc(C)ccc3Br)=O)C2)O1 CC1CCCC=C1C(=O)NCC1CN(C(=O)C(c2ccn(C)n2)C)CC1(F)CO C(=O)(C1=C(C)CCOC1)NC1C(C(=O)NCC(C(CC)C)CO)C1(C)C Cc1sc(C(F)(F)F)nc1C(=O)N(C)CC1CCN(C(C2(C)CCC2)=O)CC1 C(C)(CNC(c1nc(-c2nc[nH]n2)sc1C)=O)(C(C)C)NC(CC(=C)C)=O c1(C(C)NC(C(N2CC(CCOC)OCC2)=O)=O)ccc(Br)cc1Br c1(C(=O)NC2C(NC(=O)C=CCO)CCCC2)cc2c(Br)[nH]nc2s1 n1(C(C)C(=O)N(C2CCCC2)C)cc(Cn2cnc(-c3ccccc3)n2)nn1 c1(NCC(CC)Oc2ccccc2)cc(S(=O)(=O)NC(C)C(C)CO)ccc1C#N N1(C(C2C(C)CC(=O)CC2)=O)CCCC(C2CC2NC(=O)C=Cc2ncc[nH]2)C1 c1ccccc1.CCC(CN(C(=O)CSC)CC)NC(C1CC(O)C1)=O.C CCC(C)C(O)C(C)C(=O)N(C1CC(C(N2CCOC(CCO)C2)=O)C1)C C(=O)(CC(C)C(=O)N(C1(CC(=O)NCCCSC(F)F)CC1)C)OC Cc1c(CCC(=O)NC2CC(C)N(C(=O)Cc3cscn3)C2)cnn1C c1(C(=O)NC23CC2CN(C(=O)CC24CCCC2C4)C3)cc(Cl)cnc1O N1(C(CC(C)(C)NCC(=O)O)=O)CC(CC(=O)O)OCC1(C)C C1(NC(C2CC(CN(C)C)C2)=O)CCCN(C(C2CC3CC3C2)=O)C1 c1(CC(CN(C(C)C)Cc2cnc(C3CC3)nc2)O)cccc(O)c1 c1(OC)ccc(C2(C(=O)NCC(C)Oc3cccc(F)c3)CC2(Cl)Cl)cc1 S(=O)(=O)(c1ccc(C#N)cc1)N1CC2(N(C(c3c(CC)cc(Br)cc3)=O)CC2)C1 N1(C(C(Cn2ccnn2)NC(c2ccc(C)nn2)=O)=O)CC(O)CC(C)(C)C1 C(=O)(C1CCCc2nccn21)OCC1C(CC)=NN(c2ccccc2OC)C1=O C1(CNC(C(C=C)(C)O)=O)CC2(CC2)CN1C(=O)CCc1cccs1 CC(C)C(C)CC(=O)N(C(C)(C(=O)NC1(c2cc[nH]n2)CC1)C1CC1)C CC(C)C(=O)C(=O)N1CC(NC(=O)CCNC(=O)CO)C(O)C1 CC1(CNC(C2CCCCC2)=O)CCCN1C(=O)CCn1ccnc1 N1(C(c2c(SC)ccs2)=O)CCC2(CC1)CN(C(=O)C1=CCOCC1)C2 CCCC(C(=O)N1CCN(C(c2ccc(O)c(F)c2)=O)CC(O)C1)S(N)(=O)=O C12(CNC(C3CCOC3)=O)CCC(CN(C(=O)CCc3ccco3)C1)C2 N1(C(COCCC#C)=O)CC2CC(NC(c3nncn3CC)=O)CC1C2 N1(C(C(C)SCCCC)=O)CCCN(C(=O)CCOCC(C)C)C(C)C1 Cc1cc(O)ncc1C(N1CC(CNC(C2CCC(C)CC2)=O)CC(C)C1)=O c1(CC)ccc(C(=O)NC2C=CC(CNC(c3snc(O)c3Cl)=O)C2)cn1 C=C(Cl)CC(C(=O)N(C1CCN(CC)C1)C)NC(=O)C(CC)CCC N1(C(c2c(CNC(=O)CCc3cnccn3)nccc2)=O)CCC2(C=CCO2)C1 C(=O)(C#CC1CCC1)NCCC(C)N(C)C(c1ccnc(OC2CC2)c1)=O c1(C(=O)NCCCn2cc(C3(O)CSC3)nn2)nccc2cc[nH]c12 N1(C(CC2(NC(c3c(CC)cno3)=O)CC2)=O)CCn2c(C)cnc2C1 c1(C(N2C(C(C)(C)NC(CCN(C)CC)=O)CCC2)=O)cc(C)n(C)n1 CC1(C2CC2)CCN(c2ccnc(NCC3CC(O)C34CCC4)n2)C1 C(=O)(CCC(C)(C)C(=O)N1CCCC(c2cn(CC(F)(F)F)nn2)C1)OC C1(C(N(CC(C)OC)CC)=O)C2CCC(C2)C1NC(c1ccc(O)s1)=O C1(C)(C(=O)NC(CCCCNC(CN(C)CC)=O)C)CC=C(C)CC1 c1(CC)ncnc(N(C2CN(C(c3[nH]nnc3C3CC3)=O)C2)C)c1F c1(SC(C(=O)NCCCCCN(C(CCC(C)OC)=O)C)C)ccc(C#N)cc1 C(CC(C)CCNC(=O)Cn1ncc(Cl)c1C)NC(CC(C)OC)=O c1(NC(c2scc(CNC(CCNC(N)=O)=O)c2)=O)cccc(Cl)c1 C1(NC(C=C(C)C2CC2)=O)CCCC(NC(=O)COCC2CCCCO2)C1 C(=O)(CCC(C)(C)c1ccccc1)N(CC(CC)NC(=O)CC(=O)N(C)C)C C1(C(N(CCCNC(c2cn3c(n2)SCC3)=O)C)=O)CCN2CCCC2C1 N1(C(C(C(C)C)N2CCN(C)CC2)=O)CC2(CCN(C(=O)CCF)C2)C1 CC1=NOC(=O)C1CCC(=O)NCCOCCC.c1(C(=O)N)cc(C)sc1C N1(C(=O)Nc2c(C)n(C3CCN(C)CC3)nc2)CCCN(CC(F)F)CC1 c1(C(=O)OC)ccc(NC(N2CCC23CC(C(N)=O)C3)=O)cc1Cl C1(C(=O)NCC(CCCC)NC(c2cnc(F)c(C)c2)=O)CC(C)(C)CN1C C1(C=O)CC2C(C1)C2(F)F.c1(C=O)nc[nH]c1C(F)(F)F.CC=CC.N Cn1ncnc1CC(C(N)=O)NC(c1cnn(C2CC2(F)F)c1)=O N1(C(c2nc(N(C)C)oc2)=O)CCN(C(C2(O)CCCCC2)=O)CC1CC(F)F c1(CC)ccc(C(=O)NC2CCCCC2NC(=O)Cc2ncc(Cl)s2)cc1F N1(C(CSCC)=O)CCN(C)CC1CNC(C1CCN(C)C(C)C1)=O c1(CC(N2CC(O)(CNC(CC3CCC(C)C3)=O)C2)=O)cccc(F)c1F c1(C(N(CC(C)N(C)C(c2nc(O)nc(O)c2F)=O)C)=O)ccc2oncc2c1 N1(C(C(CC)SC)=O)CC(CNC(=O)CCc2cnoc2)C(C)(C)C1 C=CC1(O)CCN(C(=O)C(C(C)OC)C2CCC2)C1 c1(C(=O)NCCCCC(=O)N(C)CCc2cnccn2)cc(F)ccc1F c1(C(N2CCCC(CN(C)C(c3cc(O)ncn3)=O)C2)=O)ncc(Cl)cc1Cl c1(C(N2CC(NC(C(CCSC)O)=O)C(CO)C2)=O)cc2ccc(C)cn2n1 CCCCC(C(=O)NC)NC(C1CCCN(C(=O)CCC2CCCC2)CC1)=O N1(C(c2nc(C(C)C)sc2)=O)CCN(C(=O)CC2(O)CC2)C(C)C1 Cc1nc2c([nH]1)CC(C(=O)NCC(O)CNC(c1ccc(C#N)cc1F)=O)CC2 c1(C(=O)N)ccc2c(c1)OC(F)(F)O2.CC(C)C(O)C(=O)NCCC1CCC1 c1(CN2CC(CNC(C3CC(C)OC3)=O)C2)ccc(F)c(F)c1 N1(C(c2cn(C)nn2)=O)CC2CCN(C(c3cnn4c3CCCC4)=O)CC2C1 C1(NC(c2ccc(N)c(O)c2)=O)CCCC2CN(C(C3CC3(F)F)=O)CC12 O=C(CC1OC(=O)c2ccccc21)NCc1ccncc1Cl C(C(O)CC(=O)N)NC(C1(CCNC(CC(=O)NCC#C)=O)CC1)=O Cc1cn(C)c(C(C(=O)Nc2ccccc2C)N(C)CC2(CC(C)C)CC2)n1 Cc1ccc(COC(=O)CCC(C)(F)F)c(F)c1F c1(C(C)C)cnn(C)c1NC(N1CCC(Cc2ccc(Cl)cc2)C1)=O n1(CCCCC)cc(CNCC2CC(C)(C)CN2)c(C)n1 C(=O)(C(C(C)(C)C)C1CCCC1)N1CC(CNC(C(CSC)C)=O)C1 Cc1csc(C(O)CC(=O)NCC2CN(C(C3CC3c3ccccc3)=O)C2)c1 N1(C(C(COC)NC(C)=O)=O)CCOCC1.C(=O)C(C)Cn1ccc(C)n1.C c1(CC(N2CC(CCNC(C3(C)CC(F)C3)=O)C2)=O)ccc2occc2c1 C1(CNC(CCNC(N)=O)=O)CN(C(=O)CC2CCC(=O)NC2)CCCO1 Cc1c(C(=O)Nc2cnc3cc[nH]c3c2)oc2ccc(F)cc12 CC(C)C(O)CC(=O)NC1(CCNC(=O)C(c2ccc(F)cc2)O)CCCC1 C1(C(=O)NCc2c(C)noc2C)CN(C(C2CC2F)=O)CCC1(F)F C1(NC(CCCC2C(C)C2)=O)CC2C(NC(c3ccc(CCF)cc3)=O)C2C1 C1(CN=[N+]=[N-])CN(C(c2cc(CNC(C3(F)CC=CC3)=O)cs2)=O)CCO1 Cc1cc(O)c(C(N2CCOC(C(C)NC(=O)CCc3ccccc3)C2)=O)nn1 C#Cc1cccc(C(=O)NCCCCC2(NC(C)(C)C)CC2)c1Cl S(=O)(=O)(c1ccc(OC(=O)COC)c(-c2cccc3ccsc23)c1)NCCC N1(CC(Cc2c(C)n(C)nc2)CN)C(C)CC(CC(F)(F)F)C1C C1(CC(=O)NCC2(OC)CCC2)CCCCN1C(C1CC(N=[N+]=[N-])C1)=O c1(C(=O)OC)ccc(C(=O)NC2CCCCN(C(C3(C)COC3)=O)C2)c(F)c1 C1(CCC(F)(F)F)CCCN(CCC2CC2(Cl)Cl)C1 C(N=c1[nH]cnc2cc(C)[nH]c12)C1N(C(c2cc(C)cc3c2OCC3)=O)CCC1 C(=O)(CC(C)C(F)(F)F)N1C(C)CCC(NC(c2c[nH]cc2Br)=O)C1 c1(C(N2CC3CSCC3(C)C2)C(=O)NC(C)C)cc(S(N)(=O)=O)cs1 C#Cc1ccc(C(N2CCC=C(CNC(C3(COC)CCC3)=O)C2)=O)cc1 C1(NC(C2(CC)CC2(F)F)=O)CN(C(c2cccc(C)n2)=O)CCC1C c1(C(=O)NC2(CNC(CN(c3ccccc3)C)=O)CC2)cnccn1 N1(C(CCCSC)=O)CCC(C(C)(C)NC(=O)C(c2cccc(C)c2)C)CC1 C1(NC(CCN2CCN(C(C)C)CC2)=O)CCCN(C(C2CNC(=O)N2)=O)C1C c1(C(=O)NCC(C)(C)NC(=O)CCc2cncs2)ccc(C#N)cc1 C1(C)(CCCCCc2onc(C3CCN(C)C3)n2)CCN(C(=O)C(C)(C)CO)C1 C1(CC=C)(NC(=O)Cc2ncc(C)s2)CCCN(C(=O)C(C)CCN(C)C)C1 c1(C(N(C(C)C)CCN(C(=O)C(F)C2CCOC2)C)=O)n[nH]c2c1CSCC2 c1(C(N(CCNC(C2CC(OC)C2)=O)C(C)C)=O)cc(Cl)ccc1F C1(F)(CNC(CC(C)F)=O)CCC(CNC(=O)C(N)=O)C1 C(=O)(C(CC(C)CC)NC(=O)COCC(F)F)Nc1cccc(C#C)c1 C1(NCC(C(C)C)(C)O)CCCC2CCCCC12 C1(CC=O)CCC(C)(C)C1.C(CCC(=O)N)OCCOCC.C1CCOC1 N1(C(C(C)OCCOCC)=O)CCSCC1CCNC(c1ccccc1)=O CCC(O)C(F)(F)C(=O)NC(C)CNC(=O)C(C(=O)O)OC.C(C)(C)C CCC(C(=O)NCCCCNC(=O)CC1CC(C)(C)OC1=O)C(C)(F)F C1(C2CCOCC2)(C(N(C(C)CCNC(=O)CC2OCCCO2)C)=O)CC1 C(N=c1[nH]c(=NCC2CCCN(C)C2)[nH]c2cccnc12)c1c(C)nccn1 C(CC(=O)NOCC1CCCO1)=CCNC(C1C(C(C)(F)F)C1)=O C1(C(=O)NCC2(NC(CC3N(C)C(=O)CC3)=O)CC2)COC(C)(C)CO1 c1(NC(C2C(C)C2)=O)cnc(Cl)cc1C(=O)Nc1ncc(F)cn1 N1(C(c2[nH]cc(CC)n2)=O)CCC(N(C(=O)C(=O)NC(C)C)C)CC1 C(=O)(CCC1=CCc2ccccc21)NCC1(NC(COC)=O)CCCCC1C c1(C(N2CCC(C(=O)NCC(CC3CC3)OC)C2)=O)cnc(Cl)n1C C(=O)(C(C)(C)C(C)(C)O)NC(CC(=O)NC(CC(C)C)C)C(C)C c1(C(=O)NC2CCC(NC(c3c(C)csc3)=O)C2)oc(CC2CC2)nc1C C=CCCCCCCCC(=O)NC(C)CN(C(=O)C(C)CC(C)(C)C)C Cn1cnc(N2CCC(C3CC3)C2CNC(=O)CCN2CCOCC2)c(Br)c1=O C=Cn1nncc1C(=O)NCC(N1CCN(C(=O)C(C)CC2CC2)CC1)C(F)F CCC(CC)C(C)C(=O)N1CCOC(CNC(c2cnn(CCOC)c2)=O)C1 C1(NC(c2cc(CC)n(C)n2)=O)COC2CN(C(c3cc(C)ccc3N)=O)CC12 c1(CNc2ccc(-c3nccc(C)n3)cc2)n[nH]c2c1CCCC2 CC1CCCc2cc(C(=O)N(C)CCOCCN(C)C(c3cc(F)c[nH]3)=O)nn21 N1(C(c2ccc(OC)o2)=O)CC(NC(c2sncc2Br)=O)C(C)C1 C1(NC(C2CC(=O)N(C3CC3)C2)=O)CN(c2ccncn2)CC2(CC2)C1 CCC(C)(CC)C(=O)NC(C)CCCC(=O)N(CC(C)(C)O)C N1(C(CCOCCN(C(=O)C=CC2CCOC2)C)=O)CCCC12CCOCC2 c1(NC2CCCN(C(C(c3n(C)cnc3)O)=O)C2)cc(O)nc(O)n1 Cc1ccc(NC(=O)CCNC(=O)CC(N)C(C)O)c(Cl)c1 C1(NC(C(C(C)C)NC(C)=O)=O)C2CCC(C2)C1C=O.C1CC2CCCCC12 C1(C(N(C)Cc2c(C)ncs2)=O)COCCN(C(=O)C(O)C2CCC2)C1 C1(CC#C)(C(=O)NC2CN(C(C3CC3(C)C(F)F)=O)C2)CCCCC1 C1(NC(C(COC)C)=O)CCCC(NC(c2cc(C(N)=O)cn2C)=O)C1 C1(CC(=O)N)CC2(CC2)CO1.c1(C(C(N2CCC2)=O)C2CC2)ccc(F)cc1 N1(C(Cc2c(C(=O)OC)cccc2)=O)CCC(C2CC2)(C)C1.C1(C=O)CCCS1 Cc1ccc2c(C(=O)NC(CNC(=O)CCc3ccncc3)CO)c[nH]c2c1 c1(CC)ccc(CNC(=NCC2CC2(C)C)NC(C)COC(F)F)cc1 Cc1cc(NC(=O)C(C)(C)CN(C(=O)C(C)n2cncn2)C)c(C)cc1F c1(OC)cc(Br)ccc1CS(=O)CC(=O)NC(C)C(=O)N1CCCC1 c1(CNc2c(CC)cccn2)c(C)nn(C2CCS(=O)(=O)C2)c1C C1(NC(CCc2nc(C)c(C)[nH]2)=O)CCN(C(c2cc(Br)co2)=O)CCC1CO c1(NC(C)=O)ccc(C(=O)NCC(CNC(=O)C(C)N2CCC2)OC)s1 c1(C(=O)NCCCN2CCN(C(C3(C)C=CCCC3)=O)CC2)cc2c(s1)CCC2 c1(OC)c(F)c(C(N2CCN(C(=O)C(C)(C)CCl)C(C)C2)=O)cc(F)c1F C(=O)(C(C)(C)CC)NCc1scc(CC)n1.C1(CC=O)CCC(=O)NC1.N C1(C(F)F)CCN(C(C2CC(C)(C)C2)C=O)C1.N1(CC2(C)CC2)CCOCC1 c1(C(=O)NC(C2CCN(C(C(C)(C)OC)=O)C2)C)cnc2nc(C)[nH]n2c1=O CN1CCN(C(c2cc3n(n2)CCO3)=O)C(C(=O)NCC(C)(C)C(C)(C)O)C1 CN1CCC(C(N2CCC(O)(C(F)F)C2)=O)(NC(c2cnsn2)=O)C1 C1(C(N2CC(C(C)NC(c3cc(Cl)on3)=O)OCC2)=O)CC1C1CCCCC1 C(CN=c1cc(C(C)=O)nc[nH]1)N(C(c1cccc2cnnn12)=O)CC c1(CCC(=O)N(CCOC)CC2CC2)ccccc1C(=O)NOC1CC1 c1(C(C(=O)N(C)CC2CCN(C(=O)CN3CC=CC3)C2)SC)cccc(Cl)c1 CCC(C)(CCNC(=O)Cc1cn(C)nc1C)NC(c1cc(CO)[nH]n1)=O c1(C(=O)NCC(C)N(C(CCCCOC)=O)C)cn2c(n1)CCCC2 CN1CC(O)CCC1C(=O)NC1(C(=O)NCCCC(C)(F)F)CCC1 C1(NC(Cc2ccc(C)s2)=O)CCC2CC1CN2C(=O)C(O)C(C)(C)C C#CC1CCCN1C(=O)CCCC1(NC(=O)CC2CCOC2=O)CCC1 c1(C(=O)NCCN(CC(C)O)C(c2cc(C)oc2)=O)cncc2[nH]ccc12 C1(C(=O)OCC)OCCNCC1N(c1cn(C)cn1)C(c1cccs1)=O c1(C(=O)Nc2c(C#N)nc(Cl)cn2)cccc2[nH]nc(-c3cnn(CCF)c3)c12 C1(NC(C#CC2(C)CC2)=O)CN(C(c2cccc(F)c2)=O)C2(CCCOC2)C1 C=CC(CC)CC(=O)NCC12CC(NC(=O)CCCCSC)(CCO1)C2 c1(OCC)ncnc2c1CN(Cc1c(F)cc(O)cc1F)CC2 c1(NC(C2(C)CCN(c3cc(OC)ncn3)C2)=O)cc(Br)cnc1I c1(C(N2CCC(C)C2CNC(=O)C2=CCOCC2)=O)c(F)cccc1F c1(C(CNC(COCCCCC)=O)NC(C2CC(CCC)C2)=O)ccccc1 C(C)(CCC(=O)NCc1ocnc1C(=O)N(C(CO)CO)CC)OCC c1(OC)cc(OC)c(-c2ccc(F)cc2F)cc1CN1CC1CC1CCOC1 C1(C=O)Cc2ccccc2C(=O)O1.C1(F)CCC1.C(C(C)=CC(=O)NC)OC N1(C(CC2CCC(C)(C)O2)=O)CCCC2(CNC(c3cccc[n+]3[O-])=O)CCCC12 C1(CN(C(=O)C=Cc2ccncc2)C)CCCCN1C(c1cn[nH]c1)=O N1(CC)CCC1C(=O)NC(C(=O)NCCCc1nccs1)C1CC1 c1(C(CNC(=O)Cn2ccnc2C)NC(C(C)OCC=C)=O)ccccc1 c1(N(C)C)nc(C(=O)NC2CN(C(C3CCCN3N=O)=O)CC2(C)C)cc(O)n1 C=CC(C)(O)C(=O)NCc1ccc(C(=O)NCc2ncnn2C)cc1 CS(=O)(=O)c1cc(C#N)ccc1CNC1CC(C(=O)N)C1.C1CCCOC1.C N1(C(c2cc(Cl)cnc2O)=O)CCCN(C(c2ccc(Cl)c(F)c2)=O)C(CO)C1 CCCC(O)C(=O)NC(c1ccc(C)cc1)CNC(=O)Cc1csc(Cl)n1 N1(c2nc(C(=O)OC)c(C)s2)CC(NC(C2CCCN2C(C)=O)=O)CCC1C C1(NC(C2C(C#N)C2)=O)CN(C(=O)C=CC(=O)NC2CC2)CC1C1CC1 Cc1c(OCC(N2CC3C(NC(C4(C)CCC4)=O)C3C2)=O)cccc1Cl C(CCC(C)Cc1nc(C2CC2)nn1C)=C(C)C C1(N(C(c2c(C)ncs2)=O)C)CCCC(N(C)C(c2cnn(C)c2N)=O)C1 N1(C(c2c(C)c(Br)cnc2)=O)CC2(CCN(S(=O)(=O)c3nccs3)CC2)C1 C(=O)(C(CNC(c1cnc(C)cn1)=O)CC=C)NC(CC=C)(C)C Cc1cnc(S(=O)(=O)NCCCCC(C)(F)F)c(C)c1 c1(CC(=O)NC(CCNC(C23CC(OC)C2C3)=O)C)cc2ccccc2s1 C1(C(=O)OC)CCC(C(N2CCC(NC(=O)Cc3ccsn3)C2)=O)CC1 C(=O)(CCC(F)(F)F)N(C(CC)CC(=O)N1CCCC(NC(C)=O)C1)C n1(C2CN(C(=O)CC3COC3)C2)cc(Cc2ncccn2)nn1 C1(NC(c2cncc(C)n2)=O)CCCCN(C(=O)CCC2CCC(C)O2)C1 Cc1cccn2c(C(=O)NCC34CC(C3)C4)cnc12.C(=O)C=C1CC1.N N1(C(c2c(C)ccc(C)n2)=O)CC(NC(c2ccc(C(C)C)o2)=O)CC(C)(C)C1 Cc1cc(C(N2CCC(CCC(=O)NC3CC(=O)N(C4CC4)C3)C2)=O)cnn1 N1(C(c2n(C)ncc2)=O)CC2(CCC2)CC1CNC(c1coc(N(C)C)n1)=O N1(C(C(C)=CC)=O)CCCCCC1CNC(=O)C(C)(COC)CC Cc1cnc(C(C)Nc2cc(N(C)CC3CCC(=O)NC3)nc(C)n2)c(Br)c1 c1(C=O)cccc(C)c1[N+](=O)[O-].c1(OCC=C)cccnc1C(=O)NC1CC1 C(=O)(C(C)(C)C(N)=O)NC1CCC(NC(c2c(C)c(C3CC3)on2)=O)CC1 Cc1ccc(C=CC(=O)NCCC2CCC2)s1.C(C1CCCO1)=CC(=O)N n1(CC=C)cccc1C(=O)NC(C1CCCN1C(c1csc(C)n1)=O)(C)C CC1CN(C(C2(c3cccc(F)c3)CCOCC2)=O)CC1NC(C1CCCC1)=O N1(C(C23CC4CC(CC(NC(CC)=O)(C4)C2)C3)=O)CCC2(CCCN(CC)C2)C1 CN=c1[nH]cc(C(N2CC(CNC(=O)C=CC3CCOC3)CC2C)=O)o1 C(=O)(C1=C2CCN=C2NC=C1)N1C(C)CCC1.n1(CC)nc(C(=O)NC)cc1O C1(NC(CC2CCN(C(C(CC3CC3)OC)=O)CC2)=O)C(O)C2CCOC12 Cc1nc(C(C)(C)C)sc1C(=O)NCC1CC(C)N(C(C2CSC2)=O)C1 Cc1c(C(=O)NCC2CCCC2NC(c2csc3cncn23)=O)cc(N)cc1O C(N=c1[nH]c(N2CCC(N(C)C)C2)nc2c1CCC2)c1c(C)c(Br)ccc1 C(CN=c1[nH]c(=NCC2CCOC2)c2cccc(F)c2[nH]1)N(CCC)CC c1(CNC(=O)NC(CCCOC)(C)C)ccc(-c2noc(C3CC3)n2)cc1 C(C)(C(C(=O)N1CCC2C(C(N)=O)C2C1)C(C)C)NC(CCCC=C)=O N1(C(c2c(CCC)occ2)=O)CCC(N(C)C(c2cc(C)n(C)c2)=O)C(C)C1 N1(CC(=O)NCC(=C)CCNC(c2coc(Br)n2)=O)CCCC(CC)C1 CC1c2ccccc2CCN1C(C1(C)CN(C(=O)CC2NC(=O)NC2=O)C1)=O c1(C(=O)NCC(CO)NC(CSCC=C)=O)cccc(C(F)(F)F)c1F C1(CC=C)(C(=O)NC(C)C(O)C(F)F)CCCN1C(c1ccsn1)=O C(CCCCCCCO)=CC(=O)N(CCC(C(C)(C)C)NC(CC(C)F)=O)C N1(C(C2(C#N)CC23CCC3)=O)CC2CCCN(C(c3cnccc3Cl)=O)C2C1 c1(C(N2CC3C(CNC(C4CC(SC)C4)=O)C3C2)=O)ncc(C)cc1F C1(N(C(CCC#C)=O)C)CCCCN(C(=O)CC2CCNC(=O)C2)C1 C1(C(N2CC(CCC)C(CO)C2)=O)CCOCCN1C(=O)C(N1CCNC1=O)C C(=O)(C1CCc2cc(Cl)ccc21)N(C)CC1N(C(CCOC(C)C)=O)CCC1 c1(C(N2CC=CC(NC(c3sc(F)cc3Cl)=O)C2)=O)cc2cccnn2c1 CC1C(NC(C2(F)CCOC2)=O)CCN1C(=O)CCC1CCCCO1 N1(C(c2c(C)cnn2C(C)C)=O)CC2CCC1C2.C1(C(=O)N)CCN(C)C(=O)C1 c1(C(N(CC(C)N(C(CCC(CC)C)=O)C)C)=O)coc2c1N(C)C(=O)CCC2 CN1CCC(NC(c2cnc(CC(C)(C)C)s2)=O)C12CCCN(C(=O)C1CC1)C2 C(=O)(CCCC(F)(F)C(F)(F)F)NCC(C(C)C(C)C)NC(CCCCC#C)=O C1(OC)CN(C(=O)Cn2cnnc2O)CC1NC(=O)C(C)(F)c1ccccc1 CC#CCCC(=O)N1CC(CNC(c2sccc2CN(C)C)=O)C(O)C1 N1(C(c2cc(OC)nn2C)=O)CCCC2(CCC2)C1.C(=O)(CCCS(C)(=O)=O)N Cc1cc(NC(c2oc(CNC(C3CCCSC3)=O)nc2C)=O)c(C)c(C)c1 CCC(C)C(=O)C(=O)NC(CNC(c1cc(C(C)C)[nH]n1)=O)C1CCC1 c1(CC)c(C(=O)NC2COCC2)ccn1C.c1(C2C(C(=O)N)C2)ccn(C)n1 C1(CC(=O)NC(c2nc[nH]n2)C)CN(C(=O)C(C)(C)N(C)C)CC12CC2 c1(CC(=O)NC2CCC(N(C(C(CCC)O)=O)C)CC2)cc(F)c(F)cc1F CC(C)CCC(O)C(=O)N1CCCOC(CCNC(=O)C=CC(C)(C)C)C1 C1(C)(C(N2CCC(C(=O)OC)C2C)=O)CC(O)CN1C(=O)C(C)C(F)F n1(CC=O)ncc2ncccc12.CN(C)S(=O)(=O)NCC(=O)N.C1(CC)CC1 c1(CN2CC(n3ncc(NC(c4ccn(CC)n4)=O)c3)C2)cc(Br)cnc1C C1(NC(C(C)(C)C2CCN(C(=O)CCC3CCCO3)C2)=O)CC2(CCCO2)C1 S(=O)(=O)(c1cc(C2CC2)nn1C)NCC(CC(C)(C)C)OC C1(C(=O)NC(C)CCNC(c2ccc(C(F)F)cc2)=O)CCC(C2CCCO2)O1 Cc1cc(C)c(C(=O)NCC2CC(C)CO2)c(O)n1.C1(C)(C=O)CCC1.N c1(C(=O)NC2CCN(C(=O)COC3CCOCC3)CC2O)cccc2nn[nH]c12 C1(CNC(C2C(C)C2C)=O)CN(C(=O)COC2CC=CC2)CCC1C C1(C)(C(=O)NC(CC=C)CNC(=O)CCn2cccc2)CCC2CC2C1 N(C)(S(=O)(=O)NCC(O)CCN)C(C=C)C c1(C(=O)NC2C(NC(CC3N(C)C(=O)CC3)=O)CCC2)cc(C#N)cn1C C1(CC(N2C(CNC(CCCOCC)=O)C=CC2)=O)CCCCC1(C)C N1(C(C(C)Cn2ccnc2)=O)CCCN(C(=O)C(C)N2CCC2)CC1 C(=O)(CCS(N)(=O)=O)N(C1CCN(C(C2CC2Cc2ccccc2)=O)CC1)C N1(C(CN(C(=O)CC2CCCO2)CC#C)=O)CC(C)(OCCOC)C1.O CCCCCCCCC(=O)N1CC2CCC(C(N3CCC(CF)C3)=O)(C2)C1 N1(C(C2ON=C(CC)C2)=O)CCN(C(C2CSC2)=O)C(C2CC2)C1 C=CC1(CC(=O)N(C)CC2CCCN2C(=O)C(F)C(C)(C)O)CCOCC1 C#CC1CCCN(C(C2CCCCC2NC(=O)Cn2ccc(C)c2)=O)CC1 CC(c1ccccc1)=CC(=O)NCC1CN(C)CCN1C(c1sccc1C#N)=O N1(C(C(C)N(C)C)=O)CC23CCCC2(C1)CN(C(c1nnc(S)n1C)=O)C3 c1(C(N2CC(CNC(=O)C(F)(F)c3nccs3)C(O)C2)=O)ncccc1Cl Cc1cc(=NCC2CCC(CO)CC2)[nH]c(N2CCC(P(C)(C)=O)C2)n1 C(C)(C1OCCc2sccc21)NC(c1c(O)ccc(C(C)=O)c1)=O C#CCCCCCCC(=O)NC1CCOC(C(=O)NCC2CCOC2C(=C)C)C1 c1cc(F)cc(F)c1.CC(O)C(C)C(=O)N1CCC(O)(C(C)NC(=O)CO)C1 C1(CC(=O)NCC(CC=C)NC(c2cc(C)ccn2)=O)CCC(=O)C1C C(=O)(C1=CCC(C)(C)CC1)NC(C1CCN(C(=O)C)C1)C.C1CC(F)(F)C1 C(=O)(C(F)C(F)(F)C(F)(F)F)NCC1C(C)C1 C(=O)(CC(C)P(C)(C)=O)N1C(C2(NC(C3C(OC)C3)=O)CC2)CCCC1 CC1CC(NC(C23CC(c4ccccc4)(C2)C3F)=O)CC(C)N1 C(=O)(C(CO)C(C)(C)C)N1CC(C)(CCC(N2CC3(CCCO3)C2)=O)C1 Cc1cccc(F)c1C(=O)NCC(CO)NC(=O)C(F)CC1CCCC1 c1(C(N2CCC(C3CCC3)C2)C(=O)NCC=C)cc2cc(Cl)cnc2o1 N1(C(C(=O)N(C)C)=O)CC2(CNC(C3CC34CCC4)=O)CCC1C2 c1(Sc2nc(N3CCC(NC(=O)CC4(CO)CC4)C3)sn2)cccc[n+]1[O-] O=C(C1=COCCC1)NCCC1CCC(NC(c2conc2C2CCC2)=O)C1 c1(C(CC(=O)NC2CC2)NC(C)=O)ccc(Cl)cc1.c1(C=O)ccc(C)s1.C c1(NCC2C(C)CN(C(c3csnn3)=O)CC2)ncnc2scc(Br)c12 Cc1cc(CCC(=O)NCC2CCN(C(=O)C(C)C)CC2C)ccc1Cl N1(C(CC2(CNC(C3(CC)CCC3)=O)CC2)=O)CCOCC(C)(F)C1 n1(C(C(=O)NCCC(C)N(C(COCCCOC)=O)C)C)cc(C)cn1 O=C(C(CO)C(F)(F)F)NC12CCC(CN(C(C3CC4(C3)CC43CC3)=O)C1)C2 C1(C(N2CCC2(C)CC)=O)(NC(CNC(CC)=O)=O)CC(C)C1 c1(C(N(C2CC(NC(CCc3ccc(C)s3)=O)C2)C)=O)cccc2oc(C)nc12 C1(NC(C2CC(CC)OCC2)=O)CCCCN(C(=O)CN2CC3CC3C2)C1 C12(C(=O)NCC(COC)O)CCC(CC1)N(C(=O)C(CO)N(C)C)C2 c1(C(=O)NCCC(C)N(C(=O)CCC(N)=O)C)sc(Br)cc1F C1(N(C)C)CN(C(C2CCC2(F)F)=O)CC1CNC(c1cccc(=O)o1)=O C1(C(=O)NC(CC)C)CC2CC2N1C(c1ccccc1)=O c1(C(N(CCC(C)C)C)=O)cc2cnccc2[nH]1.CCS(=O)(=O)N(CC(=O)N)C C(CCCCC(=O)NCC(C1CCC1)OC)NC(c1cc(COC)no1)=O c1(OC)ccc(-c2ccnc(CN(CC(C)N(C)OC)C)n2)cc1Br N#CC1(C(=O)N)CCS(=O)(=O)CC1.C1CN(C(C2CNC(=O)C2)=O)CCCO1.C Cc1ccc(C(=O)NC2CC2)cn1.CC(F)(F)F.C(=O)C.C(=O)C1CC1.C c1(C(N2CC(C(C)NC(=O)C(C)Cc3ccco3)OCC2)=O)c[nH]c(=N)nc1O C1(COC)(C)CCCN1C(=O)Cn1cnnc1.C1(C=O)CC2(C1)CC2F.N CC#CCC(C(=O)N(C)OC)NC(=O)CC(O)CN(C)C C1(C)(C(=O)NCC2(F)CC(NC(C(F)=CC)=O)C2)CC(C)=NO1 C1(C(=O)NC2CCC(NC(c3c(C)nn(C)c3)=O)C2)Cc2cncn2C(=O)N1 c1(CC(=O)NC2C(NC(C3CC(=O)NC3)=O)CCOC2)cn2ccsc2n1 c1(C(C)C)cccc(CN2CCC(CCNC(=O)Cc3cncs3)CC2)c1 C(=O)CC(O)CC(C)(C)C.C1CC(=O)N(C2CC2)C1.C1(CC)(C(=O)N)CC1 N1(C(COCCCC)=O)CC2OCCN(C(c3ccc(C(=O)OC)[nH]3)=O)C2C1 C1(NC(c2c(COC)cccc2)=O)CC(C)CN(C(c2cccnc2CO)=O)C1 N1(C(C2=C(C)CCC2)=O)CCN(C(c2ccccc2O)=O)C2CCCC12 CC(C)(C)CCC(=O)N1CCC(NC(C2(c3ccc(F)cn3)CC2)=O)C1 C1(C(=O)NC(C(=O)NCCCc2cn(C)nc2)CC2CCC2)CCCOCC1 C12(C(=O)NC3C(C)CCN(C(CC4CCC(C)CC4)=O)C3)CCC(=O)N1CCS2 C(N=c1cc(C(=O)O)nc(Cl)[nH]1)C1CC(NC(c2ccc(SCC)cc2)=O)C1 c1(C(=O)NC2CC(C(=O)N)C2)c(O)c(Cl)cc(Cl)c1Cl.c1(CCO)ccccn1 C1(C(C#C)C)CCN(C(=O)C=CC2CCCN2C(=O)C(C)CC2CCC2)CC1 Cc1cnoc1C1(C(=O)NCCC(O)CNC(C2CCCN2C)=O)CC1 C(=O)(C1=NOC2(CCOC2)C1)N1CCC(NC(C(COC)N(C)C)=O)(CO)CC1 N1(Cc2cc(C)c(Br)cc2)CC(NC(c2cc(C(C)C)no2)=O)CC(F)(F)C1 c1(CC(=O)NC(C)CCNC(c2cscn2)=O)csc(-c2cnccn2)n1 CN1CCN(C(C2CC(=C3CCC3)C2)=O)C(C(=O)NC2CCN(C)C2)C1 c1(C(N(C(C)C)CCN(C)C(C2CCOC2=O)=O)=O)nnc(O)nc1O CCCC(CC)C(=O)NCCC1CC(NC(=O)C(c2ccc(Cl)cn2)(F)F)C1 CCC(C(=O)NCC=CC(=O)NC1CC1(C)C)C(C)(C)CC c1(C(=O)NCC2CN(C(c3c(C)n[nH]c3)=O)CC2O)cc2sccc2[nH]1 c1(C(N(C2CCCN(C(C3(C)CCOC3)=O)CC2)CC)=O)cc(C)cc(C)c1C C(CC(C(=O)NCCC1CCN(C(=O)CC(C)(C)O)C1)OC)OC c1(OCCC#N)ccc(-c2ccncc2)cn1.C12CC1C2 c1(C(=O)NCC2(C(=O)NC(CCC)C)CC=CC2)cc(F)ccc1F c1(CNC(CP(C)(C)=O)=O)n[nH]c2c1CN(C(=O)Cc1ccc(F)c(F)c1)CC2 N1(C(=O)CNS(N)(=O)=O)CC2CCC(C1)N2N(c1cncc(N)n1)C N1(C(CCC)=O)CCc2c(C(=O)Nc3cc(OC)cc(C)c3)n[nH]c2C1 c1(C(=O)NCC2CC2CF)cc([N+](=O)[O-])sn1 C1(CC(=O)NCC(CCNC(CCCC#C)=O)O)CCCNC(=O)C1 Cc1ccc(I)c(C(N2CCC2(C)C(=O)NC(C)(C)CO)=O)c1 c1(C(N2CCN(C(c3cc(Br)cnc3F)=O)C(CO)C2)=O)cc(Br)ccc1Cl C1(NC(C(n2ccc(C3CC3)n2)C)=O)CC12CCN(C(c1cc(O)cs1)=O)CC2 C(c1c[nH]cn1)=C(C(=O)NCC1CC(NC(C(C2CCOCC2)C)=O)C1)F Cc1ccc2c(CN(C)CCN(C)CCO)csc2c1.c12cc(ncn1)N2 c1(NC2C3N(C(c4cncc(C)c4)=O)CC(CC3)C2)nc(Cl)nc2c1ncn2C Cc1ccc2c(c1)CCC2C(=O)N1CCCC1CCNC(C1CC12CC2)=O c1(C(=O)NC2(CNC(C3CCCC34CCC4)=O)CC2)[nH]nc2ncnc(O)c12 c1(CC)ccc(C(N2CCC2CNC(=O)Cc2ccc(OC)nc2)=O)cc1 N1(C(C(CCC)OCC)=O)CCN(C(c2ccn(C(C)C)n2)=O)CC1C(C)C c1(NS(C)(=O)=O)ccc(C(=O)NC2CN(C(=O)Cc3ccsc3)C2)cc1 Cc1cnc(O)c(NC(=O)CNC(=O)CCC2CC2(C)C)c1 C1(C2(O)CCN(C)CC2)(C(N(CC)CC)=O)CC1.C1(C=O)C=CCCC1.CO C=C(C)CC(=O)N1CC(C)(NC(=O)CCCc2nc(-c3cccs3)no2)C1 N1(C(C2ON=C(CC)C2)=O)CCN(C(=O)CCS(=O)(=O)N(C)C)C(C(F)F)C1 n1(C(C)(C)C)cc(C(=O)C(=O)NCCCO)cn1.C(C1CCCO1)=CC(=O)N N1(C(=O)Nc2ccc3nncn3c2)CCC2(CCCC2C(=O)N=c2cc(Br)[nH][nH]2)C1 Cc1nnc2ccc(C(N3CC4(CCN(C(C5CCC(C)CC5)=O)C4)C3)=O)cn12 c1(C(N2CCCC(O)(CO)C2)C(=O)NCCOC)cc(C2CC2)ccc1F C1(NC(=O)C2=CCC2)CCN(C(C2(C(F)(F)F)CCCCO2)=O)CC1O CCC(CCC(=O)NC1(C(N2CCCCC2C)=O)CCC(C)(C)C1)OC C=C(Cl)CC(C(=O)NCCc1ccncc1F)NC(c1cncn1C)=O Cc1c(C)nnn1C.C1(CC(=O)N(CC(=O)N)C2CCC2)NC(=O)NC1=O N1(C(COCC(=O)OC)=O)CCC2(C1)CN(C(=O)C(CO)c1ccccc1)C2 C1(NC(C(C)N(C)C)=O)CCCC1NC(C1(CC#N)COC1)=O c1(C=O)cccc(-n2ccnn2)c1.C1(OC)(C)CN(C(=O)Cn2cnnc2)C1.N [N-]=[N+]=NCC(C(=O)NCCCc1cccs1)NC(c1ccon1)=O Cc1cc(Cl)c(C(N2CC3(CCC3)C2)=O)cc1C c1(C(=O)NC2CCC(NC(c3c(C)nc(CO)s3)=O)C2)cccc(Cl)c1Cl C1(NC(c2c(C)nsc2)=O)CC2CC1CN2C(=O)C(c1cccc(Cl)c1)O n1(CC(COC)OC)c(N2CCN(C(C)C)CC2)nnc1Cc1ccc(C)o1 Cc1cccc(C2(C(=O)N(CC(C)O)CC)CC2)c1.c1(CC=O)ccnn1C.N N1(C(C(C)N(C)C)=O)CC=C(CC(=O)N2CC(CO)C3(CCC3)C2)CC1 C#CCCCCCC(C(=O)NCC1(OC)CCC1)N(CC(C)C)CCN(C)CC c1(C(=O)NC(CC=C)CNC(=O)C(C)(C)C2CCOC2)nn(C)c2c1CCC2 c1(C(=O)NCC2CCC(NC(C3(Cl)CC3)=O)C2)cc(Cl)nnc1O c1(Cn2cc(C3CCN(C(Cn4c(C)nc(C)n4)=O)C3)nn2)sc(C)c(C)c1C C(=O)(C(O)CCNC(=O)C(N)=O)N(C(c1cccnc1)C)C c1(C(N2CCCC(O)(CN(C(CN(CCC)C)=O)C)C2)=O)cc2ccccn2n1 C(C1CN(C(c2nnc(S)n2C)=O)CC1C(=O)NC1C2CCCCCC12)=CC Cc1cnc(C(=O)NCCCCCNC(C2CC(C)CC(=O)N2)=O)cc1C#N C(C(CO)CO)N(C(C=CCN(C)CC)=O)C.c1(C(C=O)F)ccc(C)cc1.N C=CC1(CC(=O)NC(C)CNC(=O)C(C)Cc2ccco2)CCC1 c1(C(N2CC3CN(Cc4ccc(F)cc4Br)CC3C2)=O)cc([N+](=O)[O-])ccc1Br N1(C(CC(N2CCC(NC(c3c(CC)ocn3)=O)C2)=O)C)CCc2ccccc21 C1(SC)CN(C(=O)CCc2ncccn2)CC1NC(=O)C(C)(C)c1cnn(C)c1 C=CC(C)(CC)C(=O)N1CCCC(CCC)(NC(=O)CCc2ccc(C)cc2)C1 c1(C(N(C(C)CNC(=O)CN2CCC(C)(O)C2)C)=O)cccc2cc(O)ncc12 C1(C2CCCC2)(C(N2CC(N(C)C(C3CC34CCC4)=O)C(O)CC2)=O)CCC1 c1(CC)cc(C)c(C(N2CCC=CC2C(=O)N(CCC(C)C)C)=O)o1 C(=O)(C(F)C(C)CNC(c1ccnn1COC)=O)N1CC(N(CC=C)C)C1 N1(C(C2C(CC)N(C)CC2)=O)CCC(O)(CNC(=O)CC)CC1.C(=O)C.N CC1(C)CC(NC(=O)Cc2cccc(Cl)c2F)CN1C(C1CC(C(F)F)C1)=O N1(C(c2noc(C)c2C)=O)CC2(CC2)CC1C(N1CCC1CO)=O C1(C2(O)CCN(c3cc(O)nc(O)n3)CC2)(NC(=O)C=C2CCC2)CC1 Cc1nn(C)cc1SC1CCCNC1 C(=O)(C(O)C1=CCCCC1)N1CCC(CNC(C(C)N(C(C)=O)C)=O)CC1C N1(C(CCc2ccc(C)c(Cl)c2)=O)CCCC2C1CCN2C(=O)C(C)SC(C)C C1(CC)(CC)CC(C(=O)N(C(C)CC(=O)NCC2(C)CSC2)C)C1 C12(C(=O)NC3(C)CC(O)(CO)C3)CCCC1N(C(=O)C(F)F)CC2 Cc1ccccc1OCC(=O)NC1(CO)CCN(C(C2CC2C)=O)C1 CC1(CC(=O)NC(CNC(C2CC(F)C2)=O)C2CC2)CCOC1 C(=O)(C1CNc2ccccc21)N1C(C)(CNC(C2CN(C)C(=O)C2)=O)CCC1 CC(CC(=O)NCC1CCC1NC(=O)C=C1CCC1)c1ccsc1 c1(OC)cc(F)c(NC(C2CNCC2C2CC2)=O)cc1C(F)(F)F c1(CN(C(C(C)NC(=O)CSC(C)(C)C)=O)C)nccn1C C(C)(C(=O)NCC1(N(C)C)CCC1)N(C(CNC(CC)=O)=O)C N1(C(C2CN(C(C3(CC(C)C)CC3)=O)C(C)(C)CC2)=O)CCC2(CCC2)C(O)C1 C1(C(C)(C)C)CN(C(=O)C(O)CNC(c2sccc2C#N)=O)CCO1 CC1(CC(N2CCC(CCO)C2)=O)CCN1C(C1CCCCO1)=O n1(-c2c(C(=O)NC(CNC(CCN(CCC)C)=O)CO)ccs2)c(C)ccc1C Cc1c(C(=O)NCC2C3CN(C(C4C5CCC4CC5)=O)CC23)nn2c1CCCC2 c1(OC)ccc(N(C)Cc2noc(-c3ccc(Cl)nc3)n2)cc1 C(=O)(C1c2c[nH]nc2CCC1C)NC(CNC(C(=O)NCC)=O)(C)C N1(C(C(=O)NCCCCCC)C2CC2C)CC2CC1C1OC(C)(C)OC21 CC1(C)CN(C(C2CCC(n3cc(CCCN(C)C)nn3)CC2)=O)CC(C)(C)O1 c1(C(N(C)CC2CCN(C(c3cncc(C)c3)=O)CC2)=O)cc(I)c(O)c(I)c1 c1(OC)ccc2c(C(=O)NC3CC3NC(c3ccccc3O)=O)csc2c1 c1(C(=O)NCCN(C(C2CCCC(OC)C2)=O)CC)ccc2ccccc2c1C Cc1nn(C)c(C(=O)NCCN(C)C(C2CCC2Cc2cccnc2)=O)c1Cl C1(CNC(C2CCC(NC(c3ccsn3)=O)C2)=O)CCS(=O)(=O)C1 Cc1cc(C(=O)NCC2CN(C(=O)CCP(C)(C)=O)C2)ccc1S(C)(=O)=O N1(C(C(C(CC)C)O)=O)CCC2(CC1)CN(C(=O)CC1CC(CF)C1)C2 C1(CC(=O)NCC(CC)(C)Cl)CC(C)(C)CN1C(=O)CC(C)(F)F Cc1cc(N2CCC(C)S(=O)CC2)nc(=NCCSCC(F)(F)F)[nH]1 c1(CCC)cc(C(=O)NC2CCN(C(C3COCCN3C)=O)C2C2CC2)n(C)n1 N1(C(COCCOC)=O)CCCC(C)(C)C1.c1(C(=O)N)ccc(C(F)F)nc1 n1(CCc2onc(C)n2)c(C)cc(C)c(Cc2ccccc2)c1=O c1(OC)ccc(C)c(C(=O)NCC2CC2)n1.c1(C=O)cnc(N)c(Br)c1.N C1(NC(c2cc(C)ncc2)=O)CCC12CN(C(=O)CC1CC(C(F)F)C1)C2 c1(C(=O)N)n[nH]c2c1CS(=O)(=O)CC2.c1(C(=O)NCCCC=C)ccc(C)n1C C1(CNC(C(C2CC2)SC)=O)CC12CCN(C(=O)C(C)(C)C(N)=O)CC2 CC1(c2ccc(C(=O)NC3CN(c4ccccc4)C3=O)cc2)NC(=O)NC1=O CC#CCC(C(=O)N1CCC(C)(OC)CC1)NC(C1CCC(O)C1)=O N1(C(c2ccc(C3(C)CC3)cc2)=O)CC2CC3CC2C1C3OCc1ccsc1Cl CCC(C)(CO)C(=O)NC1CCC(CCNC(c2cnc(C(C)(C)C)[nH]2)=O)C1 O=C(C(C(F)(F)F)C(F)(F)F)NC1CN(C(=O)Cn2ccc(O)nc2=O)CC1O c1(Cn2cc(-c3cncc(C(=O)OC)c3)nn2)ccc(F)cc1C c1(CC)nc(C)c(C(=O)NCC(C)(C)CNC(C2CCCC23CC3)=O)o1 CC(=O)CC(C)(C)C(=O)NCC1CCCC1C(=O)NCC1COC(=O)C1 Cc1cc2nc(NCC3CCC(NC(C4CCC(=O)N4)=O)C3)cc(=O)n2o1 c1(C(N2CCC(NC(CCC(=C)Cl)=O)CC2C2CC2)=O)cnc(C)c(C#N)c1 Cc1oc2ncnc(O)c2c1C(=O)NCC(CC(C)C)NC(=O)C(C)C1CCC1 c1(C(=O)NCC2CC2NC(c2ccc(Br)cc2F)=O)cc2cccnc2s1 C(=O)(CCCCCCCCCO)N1CC(N(C(C2(n3cccn3)CC2)=O)CC)C1 C1(C(=O)NC(C2CN(C(CC(=O)OCC)=O)C2)C)CCc2[nH]nc(O)c2C1 N1(C(C2C(OC)CN(C(c3cc(C)c(C)cn3)=O)C2)=O)CC(F)CC(F)C1 C1(OC)CC(C)CN(C(=O)C(C2CCCC2)NC(=O)C(C)n2ccnc2)C1 Cc1cc(C(N2C(C(=O)Nc3cnccc3I)CC3CC23)=O)cc(Cl)c1 C1(O)(CNC(CC2N(C(Cc3ccn(C)n3)=O)CCCC2)=O)CCC(C)(C)C1 N1(C(CNC(=O)NC)=O)CCN(C(=O)COc2ccc(OC)cc2)CC1 N1(CC(N2CC3CN(C(C(C)O)=O)C3C2)=O)C(=O)c2ccccc2C1=O C=CCC(CNC(=O)C1=CC(C)(C)C1)C(=O)NCC(c1ccnn1C)O c1(CCC(C(=O)NCCCC)N2CCC(C)(F)C2)cccc(OC)c1F CCCCCCNC(C1(C)CCCN1C(C)=O)=O.C1(C=O)CCC1.C1CC1.N CC(CC(=O)NC1CCCC12CN(C(=O)CCc1cnn[nH]1)C2)CC(C)(C)C c1(OC)cccc(OC)c1CC(N1CCN(C(c2cscc2Cl)=O)C(C)C1)=O C1(C(N2CCC(F)(c3ccccc3F)C2)=O)(CC)CCN(C(=O)O)C1.C(C)(C)C C(CC(=O)NC)(C(N)=O)NC(C)=O.C12CC1CN(C(=O)CC)C2.CC(C)C C=C(C)CCCC(=O)N1CCCC(N(C(=O)CC=CCC)Cc2ccccc2)C1 Cc1conc1NC(=O)NC(C(C)(C)O)c1ccccc1 c1(C(C)OC(=O)CNC(=O)OC2CC2)ccccn1 CC(O)C(C(=O)N(CCCCCNC(C1CC(F)C(=O)N1)=O)C)N(C)C S(=O)(=O)(c1ccc(F)c(F)c1)N1CCCC(CNC(=O)CC2CCCCC2)C1 Cc1nsc(C(=O)N(CCCNC(=O)Cc2cnn(C)c2)C(C)C)c1N CCCC(C(O)C(=O)N1CCCCC1CC(C)C)NC(=O)C(=O)NC(C)C Cc1cc(C(N)=O)cc(C=O)c1.CC(C)CN(C)C(C1(C(F)F)CCC1)=O.N c1(NCC(C)N(C(=O)NCC)Cc2ccccc2)ncc(C(F)F)cc1F N1(C(CC(C)(C)O)=O)CCC2(CCCC2NC(=O)C2=CCCC2P(C)(C)=O)CC1 CC1(C(=O)NC2CCN(C(c3cncnc3C(C)(C)C)=O)CC2)CC(C#N)C1 C(=O)(C1=CCCC1(C)C)N1CCN(C)C(CNC(c2nc(Cl)cs2)=O)C1 C1(C(N2CC(N(C)C(c3ccsn3)=O)C3(C2)CC3)=O)COc2cc(F)ccc2O1 c1(CNC(=NCCC#C)NCC23CCCC(CO2)C3)oc2ccccc2c1C n1(CC(=O)NC2CCC(NC(CC(C=C)C)=O)C2)nc2c(n1)CCCC2 CCS(=O)(=O)CC(=O)N.c1(C2C(C=O)C2)ccc(C)c(C)c1.CCC1CCC1 C=CC1CN(C(=O)C(CC(N)=O)NC(=O)C(CSC)OC)CCO1 c1(C(N(CCn2cc(-c3cccnc3F)nn2)CC)=O)cc(Br)c(F)cn1 C1CC(C(N)=O)=NO1.Cc1c[nH]nc1C(=O)NCc1cc(C(=O)N)on1.C CC(CC(=O)NCCOCCCN(C(=O)CC1CCSCC1)C)c1ccco1 C1(C)(COC)CN(C(C2C3CN(C(=O)CNC(=O)OC)CC23)=O)CCO1 C1(C)(C(=O)NCc2ccn(CCC)n2)CCN(C(=O)C(C)CC(=O)OC)CC1 C1(CNC(CCOCCOC)=O)CCC(C(=O)NCC(C)C(C)O)CC1 Cc1cncc2cc(C(=O)NCC3CCN(C(=O)CC4CCCCO4)C3)sc12 Cn1ncc2c(NC(C3CCCCC3F)=O)ncnc12 CC(CC(=O)NCC#CCNC(=O)C(C)(C)CC1CC1)C(F)(F)C(F)(F)F C(CC(F)F)(C(=O)NC(CO)CCCO)N(C(C1CC(C)C1)=O)C Cc1cc(C(N2CC(NC(=O)C(C)Cc3cnco3)CC2(C)C)=O)c(C)c(C)c1 c1(CNC(C2C(CCOC)C2)=O)ccnc(C(=O)N)c1.C(C)(CO)CCF c1(C=O)cc(F)cc2nc[nH]c12.C1(C(=O)NCC(C)(C)OCC)CCC1(F)F N1(C(C(C(CC)(F)F)(C)C)=O)CC(S(=O)(=O)C2COC2)C1 C(CC(C)C(C)C)NC(C=C(C)C(C)(C)C)=O.c1(CC=O)cc(F)ccc1C.N CC1=NOC(CNC(=O)C(Cc2ccco2)NC(=O)CC2(C)CCOC2)C1 c1(OC)ccc(C2CCCN2C(C(=O)NCCC#N)c2cc[nH]n2)cc1C c1(OC)cc(C(=O)NC2CC3CN(C(c4ccncc4)=O)CC23)cc(Cl)c1 C1(C(=O)N(C2CCN(c3ccnc(Cl)n3)CC2)c2ccncn2)CC2CCC1CC2 c1(C(N(C(CCNC(C(COC)(C)C)=O)C)C)=O)cccc(OC)c1F c1(-c2nc(NC(COC(CSC=CCC)=O)=O)sc2)cccc(Br)c1 O=C(CCC(F)F)NC1(CF)CCN(C(c2ccccc2OC(F)F)=O)C1 C=CCC(C)(C)C(=O)N1CCC(C)C(CNC(C2SCC=C2C)=O)C1 C(=O)(CC(=O)N(CC(=O)NCCC(O)C1CC1)C)NCC#C c1(C(=O)NC(CNC(C2CCC(C)(C)C2)=O)(C)C)cc(C2CC2)cc(F)c1 C1(CNC(COCCOCC)=O)CCOCC1.C(=O)C=C(C)C.C N1(C(C(CCC)C)=O)CC2CCC1C(NC(C1CC3CC1C1CC31)=O)C2 C1(NC(c2ccc(C=C)cc2)=O)CCCC12CCN(C(C1CCN1CC)=O)CC2 C=Cc1ccc(C(=O)NC2CC(CNC(c3cscc3C(F)F)=O)C2)cc1 c1(CC(=O)NCCC(C)C)cccc(C(N)=O)c1.C(=O)(CCc1cc[nH]n1)N Cn1cc(C(=O)NCCNC2CCC2)c(C(F)(F)F)c1.c1ccn(CCF)n1 C1(CNC(C2C(C(C)C)OCC2)=O)CCN(C(C2C3COCC23)=O)CC1O c1(CC(N2CCC(CNC(CCC#N)=O)C2)=O)ccc2oc(O)nc2c1 c1(N2C(C)CCC(NC(COCCOC)=O)C2)nc2c(cc1C#N)CCOC2 C1(C(=O)NCCC(C(=O)NCC(O)C(C)(C)O)OC)CC2(CCC2)CO1 c1(C(=O)NCCCOCCNC(=O)CC2CCC2(F)F)ccc2ccccc2c1 C(C)(CCC(=O)NCC1CCC(=O)O1)NC(Cc1nc(C)oc1)=O C(=O)(CCCC(=O)N)NCC.c1(C(N(C2CCCCC2)C)=O)cn(C)c(=O)n1C CC1CN(C(=O)CSc2n[nH]c(=N)s2)CC(CC)O1.C(c1ccsc1)=CC=O CCC(CNC1(c2nnnn2C2CCC2)COC1)C(C)C c1(C(N2CCC(NC(c3n(C(C)C)ncn3)=O)C(F)C2)=O)cc(N)c(Cl)c(O)c1 c1(CNC2C(C(=O)NC(c3ccc(Br)s3)CC)C2)cc(C)cs1 c1(OC)cccc(C(N2CC3(CNC(=O)CS(C)(=O)=O)CC2CO3)=O)c1F C1(N(CCC)C(C2CCN2CC)=O)CCN(C(c2ncn(CC)n2)=O)CC1 CC1(C(=O)NOCC(=O)NCCC2COCC2O)COC(=O)N1 c1(CC)ccccc1C(=O)N(S(=O)(=O)CC)CC.C(=O)C(C)C1CCC1.N Cn1ncc(C(N2CCC(C(=O)NCCN3CCC(CO)C3)C2)=O)cc1=O c1(C(N(C(C)CCNC(=O)CC2COCC2O)C)=O)ccc(-c2ncc[nH]2)cc1 c1(C(C(=O)NCC=C)N(C(C)CCO)C)cccc(C(C)(F)F)c1 CC(C)(C)C#CC(=O)N1CCC(C(C)(C)C)(C)C1.C1(C=O)CCC(F)(F)C1.N C1(C(=O)OC)CCC2(CCC2)CN1C(c1ccc(C2CCNC2)cc1)=O Cc1cc[nH]c(=N)c1C(=O)NC1CCC1CNC(C1CC(C2CCC2)C1)=O N1(C(c2c(OC)ncc(Cl)c2)=O)CCC2C(C1)OCCN2C(c1cn(C)cn1)=O C(C)(c1ccccc1Cl)=CC(=O)NC1COCCN(C(C(C)(C2CC2)OC)=O)C1 C1(C(N(CC(C)O)CCNC(c2cnc(SC)n2C)=O)=O)OCC2CCCC12 c1(OC)cnccc1C(=O)NC(C1CCN(C(c2cc(C)cs2)=O)C1)C c1(C(N(CCOC)CCNC(c2ccc(Br)o2)=O)=O)cncc(OC)n1 C(=O)(CC(C)CC(C)(C)C)NC(CNC(c1c(C)nn(C)c1)=O)(C)C C1(C(=O)Nc2cc(CC)c(C)nc2)CC2CC1CN(C(c1cc(CC)sn1)=O)C2 c1(N(C2CNCC2(F)F)C(COC)=O)ncc2ccc(F)cc2n1 C=CC1CCCN(C(C2CN(C(C)=O)C2)=O)C1.C12(C=C)CCN(C1)C2=O c1(C(=O)NCC2CC3CCC2N3C(=O)CCc2nncs2)ccc2scnc2c1 CC(C)(F)CCC(=O)NC1CC2CCC1(NC(=O)Cc1cc[nH]n1)C2 Cc1nc(C)c(C(=O)NCC(C)(O)CNC(=O)CO)[nH]1.c1ccc(F)cc1 C(=O)(CCC(=O)NC(CO)C(=O)NCc1ccnn1CC)NCC c1(CNC(C=CCC)=O)ccc(CC(C)NC(c2cccn2CC)=O)cc1 C#Cc1ccccc1CNC(=O)C(C)N(C(C12COCC1C2)=O)CC c1(C(N2CCC(N(C(CCCCC=C)=O)C)CC2)=O)ccc(S(C)(=O)=O)o1 C1(CC(N2CC(C)C(NC(=O)C=CC3CCOCC3)C2)=O)CCCC(C)(C)O1 N1(CNCc2n(CCCC)nnn2)C(=O)NC(C)C1=O N1(C(c2cnsn2)=O)CC(CNC(C2(O)CC(c3ccccc3)C2)=O)C(O)C1 N1(C(c2ccc(OC)cn2)=O)CCN(C(=O)C(O)Cn2cncn2)CC1C c1(C(N2C(C(=O)NC(c3ccncc3F)C)CCC2)=O)nnc(O)nc1O n1(CC(=O)N(CC(C)NC(COCCCC#C)=O)CC)cnc(Br)n1 N1(C(C2CC(CC)(CC)C2)=O)CC(C=O)C(F)(F)C1.CCC=O.CC(C)C.N N1(C(C(C)n2cccn2)=O)CC2CC1C2C.C12(C(=O)N)CCCC1(C(N)=O)C2 C1(CNC(c2c(OC)c(Cl)ccc2)=O)CCCCN(C(c2ccn(C)c2)=O)CC1 n1(C(C)C(=O)NC(C)(C)CN(C(=O)Cc2cnoc2)C)cc2ccccc2n1 c1(C(=O)NC(CNC(CN2CCN(C)CC2)=O)C2CC2)ccc(CO)c(F)c1 C1(C(C(=O)NCCSC)N(C2CCCC(C)(C)C2)C)CCC(C)=CC1C c1(OC)cccc(C(=O)NC2(C)CCCN(c3cc(O)ncn3)C2)c1C Cc1[nH]nc(C(N2CCC(=CCNC(c3cscn3)=O)CC2)=O)c1[N+](=O)[O-] N1(C(CCOCC)=O)CC2CN(C(=O)CC)CC12.c1(NCC)ccc(C)o1 c1(C(N2CCC(NC(C3CC3F)=O)CC(O)C2)=O)cnn2c1OCC1(CC1)C2 C1(NC(=O)OC(C)(C)C)CN(C(c2c[nH]nc2C2CCOCC2)=O)CC1(C)C NS(=O)(=O)c1ccc(CN)c(F)c1.n1(CCC(=O)O)nc(C(F)(F)F)cc1 Cc1cnc(CCCC(=O)NCC2(F)CN(C(C3CC(C)C3)=O)C2)o1 C=CCCC(F)(F)C(=O)NC1CC(F)(F)CC1NC(c1cc(C)ccc1F)=O c1ccc(C(N2CCCC2C2(O)CN(C(C3(C)CC(C)=NO3)=O)C2)=O)nc1.CN C#Cc1ccc(C(N2CCCOC(CNC(=O)C(C)(O)CCC)C2)=O)cn1 C(=O)C1=NOC(C(C)(C)C)C1.C(C)(C)C(C)C.c1(C(C)C)cc(C=O)no1.N N1(C(Cc2ccn(C)n2)=O)CCOC(C(N2CCC2C(N)=O)=O)C1 c1(C(=O)NC(C2OCCN(C(CC3(OC)CC3)=O)C2)C)sc(C#N)cc1Cl c1(OC)nc(C(c2nnnn2C2CCCC2)NC2CCN(C)C(=O)C2)ccc1C C1(COC)CCN(C(C2C3CCC(C3)N2C(c2ccc(C)s2)=O)=O)C1(C)C c1(OCC)cccc(CC(=O)NCCCCCNC(c2ocnc2CC)=O)c1 C1(C(=O)NC(CCC=C)(C)C)CN(C(C2(C#N)CCCO2)=O)CCC1(C)C C1(COC)(NC(=O)CC2CC(F)C2)CCN(C(c2cc(N)cnc2C)=O)CC1 C=CCC(CC)C(=O)NC(CNC(C1COCCN1C=O)=O)C(C)C Cc1cc(C(N2CCOC(CNC(C3COC3)=O)C2)=O)c2ccc(F)cc2n1 c1(C(=O)NCCCCNC(=O)CC2CC=CCC2)csc2c(F)cccc12 c1(C(N2CC=C(CNC(C3(CC)CCOC3)=O)CC2)=O)cccc2[nH]c(=N)oc12 N1(C(C2(C)CC(C#N)C2)=O)CC(C2(NC(=O)CCC3CCC(O)CC3)CC2)C1 N1(C(CCC=CCC=C)=O)CC(C(=O)N)C(C2CC2)C1.c1(C(C)C)cn(C)nn1 c1(CC)ccc(C)cc1C(=O)NCCN(C(=O)CC(O)CC)CC1CC1 Cc1cc(C=CC(N2CC(c3ocnc3C)C2)=O)c[nH]c1=N.C(=O)CN(C)C CC1CC(C)(C)CN1C(=O)CC1(C)CCN(C(=O)CCc2cnoc2)C1 C1(NC(c2c(C)csc2)=O)CCC2CN(C(=O)C3=CCOCC3)CCC2C1 C1(CNC(C2CCCCC2F)=O)CCC2(CCC2)CN1C(c1ccc(Cl)cc1)=O C1(C)(C(=O)NCCN(C(=O)CCc2cccc(F)c2)C)CCCNC1=O Nc1ncccc1CC(N1CCOC(C2CCCOC2)C1)=O c1(C(=O)NC2CC(NC(c3c(Cl)cc(C)s3)=O)C23CCC3)cc(N)cc(O)c1C CC1CN(C(=O)C(c2ccccc2)NC(=O)C2=C(Cl)CCC2)C(C)CCO1 CCC(CC)C(O)CNC(C1OCCC1NC(C1CCC(CC)O1)=O)=O c1(C(=O)NC(CCOC)CNC(=O)C(C)n2cccn2)occc(=O)c1OC C(=O)(CCC(C)Sc1nocc1C)OCC CC(C)C(=O)C(=O)N1CC2C(NC(=O)CC3CCCCO3)C2C1 C(=O)(C(CC#CC)NC(C1CC(=O)N(CC)C1)=O)N(CC=C)CCO Cn1ccn2ncc(C=O)c2c1=O.N1(C(=O)N)CC(C)OC(C)(C)C1.C(C)(C)C C12(NC(=O)CSC(F)(F)F)CCOC(CNC(=O)Cc3cc[nH]n3)(C1)C2 c1(COC(c2ccc(N3CCN(CC)CC3)cc2)=O)cc(C#N)ccn1 c1(C(N2C3CC(NC(c4nocc4Cl)=O)CC2CC3)=O)cnn2c1C(=O)NCC2 C1(CC(=O)NC2CC(C)N(C(C3COC4COCC34)=O)C2)CCCNC(=O)C1 C(=O)(CC(C(C)C)OCC)NC(CC=C)CNC(=O)CCc1ccccc1O C1(C(=O)NCC2(NC(=O)Cc3cc(Cl)cs3)CCC2)CC(O)C(F)C1 N1(C(CSCCN(CC)CC)=O)CCOCC1.C(=O)(CC1CC1)NC.C C1(CNC(c2ccc(C)c(F)c2)=O)C2CCCC1N(C(=O)C1=COCCO1)C2 N1(C(C2CN(C)C(=O)CC2)=O)CCOCC(F)(CNC(c2coc(O)n2)=O)C1 c1(CN2C3CN(C(Cn4c(C)cc(C)n4)=O)C(C3)C2)cc(F)c(O)cc1F CC1=NC(C)(CN2CCC(c3cnco3)CC2)CS1 C(=O)(C1Cc2ccc(F)cc21)N(C1CCN(C)CC1)Cc1c(OC)nn(C)c1 N1(C(C2CC(CCNC(C3(CO)CCOCC3)=O)C2)=O)CCC(F)(CO)C1 Cc1ccc2c(n1)CN(C(c1ccc(-c3cc[nH]n3)o1)C(=O)NC1CCOC1)C2 C(=O)(CCC(F)(F)F)NC(C(=O)N(CCc1ccccc1)CC)CC1CC1 N1(C(c2ncc(F)cc2F)=O)CC(C2CCCCN(C(C3OCCCO3)=O)C2)C1 Cn1cc(C(F)F)c(C(=O)NC=O)n1.C1CC1.C(C)(C)C.C(=O)(C)N c1(CCC(=O)N(CCCCN(C(C(CCC)C)=O)C)C)ccccc1C#N c1(C=O)ccc(S(N)(=O)=O)nc1.N1(C(c2c(CC)nc[nH]2)=O)CC2CCC1C2.N c12cc(no1)C(=O)N1C(CC1CO)NC(=O)COCC2.C1CCCC1CO C1(NC(C(c2ccc(Cl)cc2)C)=O)CN(C(=O)CCc2cnc[nH]2)CCC1F N(C(=NCCOC)NCC(C)SC)C(C#C)C(C)C c1(C(=O)NC(CNC(C(CC)COC)=O)(C)C2CCC2)ccc(F)c(SC)c1 c1(C(=O)NCC(CNC(COCC(=O)OC)=O)CO)cnc2[nH]ncc2c1 c1(CC)cc(C(=O)N(CC(C)NC(C2(O)CC(C)(C)C2)=O)C)cc(Cl)c1 C1(NC(CC(=O)OCC)=O)CCCC(NC(C2(CCOC)CC2)=O)C1 c1(C(=O)NCCCCNC(c2c(C)nco2)=O)cccc2c1OCCN2C c1(NCCC(C(C)C)N(C)C)ccc(S(=O)(=O)NCC2CC2(Cl)Cl)cc1F C1(O)(C(=O)NC(CSCC)C(=O)NCc2cncc(O)c2)CC2CCC1C2 N1(C(COCC=C)=O)C(CC(=O)NCC2(C)CCC(=O)N2C)C2CCCC12 c1(C(N(C)C)=O)ccnc(NC(=O)N(C2CC3(CCC3)C2)CCO)c1 c1(C(COC(c2c(N)snn2)=O)=O)ccc(N2CCNC(=O)C2)nc1 C1(NC(C2(C(C)(C)OC)CC2)=O)CC(F)(C)C1.C1(C)(C=O)CCCO1 O=C1CCC(CCC(=O)N2CC(C3CCCN(C(C4CSCCS4)=O)C3)C2)=NN1 c1(CC(C)NC(=O)CCC2CCC2)cnccn1.C1(C(=O)N)CCC1.C1CC1 C(C)(CCC(=O)N(C1CCCN(C(c2ccc(CF)cc2)=O)C1)C)OCC Cc1cc(C(N2CCOCC(CNC(C34CC(C)C3C4)=O)C2)=O)c2nccn2c1 c1(C(=O)Nc2cccc(NC(C3CN(C)CC(C)O3)=O)c2)cnc2n1CCOC2 C12(NC(C(C3CC3)OC)=O)CCC(CC1)N(C(=O)C(c1ncccc1F)(F)F)C2 C1(OC)(C)CCN(C(=O)CCC2(C)CC2)C1.C(=O)CS(=O)(=O)N(C)C.N N1(C(CC(C)O)=O)CCC(O)CC1C(=O)NCC1CC(=O)N(C)C1=O Cc1cc(C(=O)NCCCCC2CCCN(C(=O)C(C)c3cccs3)C2)cn1C N1(C(C)C(=O)NCC2(NC(=O)CCn3cnnn3)CCOC2)CCCCC1=O C(=O)(CC(CC)CC(C)C)NCCCN(C(C12CCC(OC)C1C2)=O)C1CC1 N1(C(COCC=C)=O)CCC2CCC(C1)N2C(=O)C(c1cccc(Cl)c1)SC N1(C(C2(C)CC(C)OC(C)C2)=O)CC(NC(=O)CC(C)(C)O)CC2(CCC2)C1 C1(CNC(c2cc(C(C)C)no2)=O)CN(C(=O)C=CC2CCC2)CC1C Cc1ccc(F)c(C(=O)NCCCCC(=O)NC2CCC3CCC2C3)n1 Cc1csc(=O)n1CCC(=O)NC(C)(CNC(=O)C)C1CCC1.C1CCC1 C1(C(N(C2CCN(C(=O)CCCc3cc[nH]n3)C2)CCC)=O)CC(C)(C)CO1 c1(CC(N2CCC2C2CC2)=O)cn2cc(-c3cccc4ccsc34)ccc2n1 c1(CCC)cc(C(=O)NC(C)CCCNC(C2CCCN2C=O)=O)n(C)n1 n1(CC(=O)NCCN(CC(C)O)C(c2cnc(C)[nH]2)=O)ncc(Br)c1C N1(C(C(CC=CC)C)=O)CCC2(CCN(C(c3cnc(Cl)s3)=O)CC2)C1 C(CC(C(C)C)NC(C1CC2CC2C1)=O)NC(C(c1ccc(C)s1)C)=O c1(OC)ccc(CC(=O)NC(C)CC)cc1[N+](=O)[O-].C(c1cnc[nH]1)=CC=O.N CC(N)(Cc1ccc(Br)cc1)C(=O)NCC(O)Cc1ccccc1 N1(C(c2cccc(N3CCCCC3)c2)=O)CCN(C(=O)C(O)CCl)C2(CC2)C1 c1(C(N2CC(NC(C(C(C)(C)F)(C)F)=O)C(O)C2)=O)cc2n(n1)CCCCC2=O C(=O)(C(C#N)CC)NCC1(O)CC(C(N(C2CC(OCC)C2)C)=O)C1 C12CC(CO1)N(C(C1(C)CCC(F)(F)C1)=O)C2.c1(OC)ccnc(C(=O)N)c1 CCCCC(CC)C(=O)N1CC(N(C(=O)CCCCCNC(C)=O)C)CC1CO C(C(=O)N1CCC1CNC(=O)Cc1ccccc1)(C(C)C)SC.C(C)C.C C1(C(=O)NCC(CO)C2CCC2)CC(O)CN1C(=O)C=C1CCOCC1 C=C1CCC(C(=O)NC2CN(C(C3(C)CC=CC3)=O)CC2OC)CC1 CCCC(C(O)C(=O)Nc1ccccc1SC)NC(C1COCC(C)O1)=O C(C(=O)N(CC)OC)N(C(C(CC)C)=O)C CCC(C(=O)N1CC2C(C)C2C1)C(C)(F)F.c1(C2(C=O)CC2)ccc(C)nc1.N c1(-n2c(-c3csc(-c4ccncc4)n3)nc(CSC)n2)ccc2ccccc2c1 c1(-c2c(C(N3Cc4cccc(O)c4C3)=O)cccn2)cnc2c(c1)NCCO2 C(c1cccc(F)c1)=CCC=O.C(C)(C(=O)N)NC(CC)=O.C1(CC)CCC1 Cc1ccc(F)c(C(N2CC(CNC(c3ncn4c3CCC4)=O)C(F)(F)C2)=O)n1 c1(NC(C)=O)cccc(CNC(C2OCCC2)=O)c1Cl.C(C)(C)C.C=O.N N1(C(CC2(C)CC2)=O)CC(NC(=O)CCc2csnn2)CC12CCOC2 N1(C(C(C)C2CC2)=O)CC(CC(=O)NC2(C)CCCC2(F)F)CC1(C)C C1(NC(=O)CN2CCN(C(c3cnn(C4CC4)c3)=O)CC2)CCn2ncnc2C1 N1(C(=O)CC(C2CC2)C2CC2)CCC2CCCC(C1)N2C(=O)Cn1cnnc1O C1(CCCN(CCOC)C)CCN(N2CCC2c2cccc(C(C)C)c2)CC1 N1(C(c2cc(CCC)on2)=O)CCC(CC)(NC(C)=O)CC1.c1ccc(N)cc1.C c1(C=O)cccnc1.C(=O)(CCCC=C(C)C)N1CC(CCO)(COC)C1.C C(=O)(C#CC1(C)CCCO1)NC1C(CNC(CCNC(=O)OC)=O)COC1 C1(O)(CNC(=O)CO)CCN(C(c2cncn2-c2cccc(F)c2)=O)CC1 CCC(C)C(C(=O)NCCCNC(c1cn(C(C)C)cc1C)=O)NC(C)=O C1(O)CCN(C(=O)CC2CC(C)=NO2)C1.CCC(=O)N.C(CO)OCC C(C1=CCCN(C(C2OCCC2(C)C)=O)C1)NC(CC1C(CC)C1)=O C(=O)(C(C)(O)C(F)(F)F)NC1C(C)N(C(c2cc(C(F)(F)F)ns2)=O)CC1 N#CC1CCN(C(C2CN(C(=O)CCc3ccc(C(F)(F)F)cc3)C2)=O)CC1 N1(C(C(=O)NC(CNC(C=C(C)C(C)C)=O)CO)C)CCOCC1 N1(CC)CCCC(NC(C2(CNC(=O)CC3CCC3)CC23CCC3)=O)C1 CC1(C)C(CC(N2CCC(CF)(NC(=O)COC3CCCOC3)C2)=O)C1(C)C C#CCC(CC(F)F)C(=O)NC(C1(C(=O)NCC2CC2CO)CC1)C N1(c2nccc(OC)n2)CCC2CCN(C(=O)C=Cc3nccs3)CC2C1 N1(C(C(C(C)C)CNC(c2cc(C(N)=O)[nH]n2)=O)=O)Cc2ccc(O)cc2C1 C1(NC(C2ON=C(C)C2)=O)COCCC1NC(C1CC(C)(O)C1)=O C(CC)(C(=O)NCCNC(C1CC2CC2C1)=O)=CC C1(CNC(c2cc3nc(C)n(C)c3cc2)=O)CC(N=c2nc(C#N)[nH]cc2C)C1 c1(-c2c(C)nc(C)s2)cccc2[nH]nc(C(=O)Nc3ncc(Br)nc3Br)c12 C1(C(=O)N)CCC(C)=C(C)C1.N1(C(C)=O)CCCC1(C)C(N1CCC(CC)C1)=O N1(C(CSCC)=O)CCC12CN(Cc1ccc(-c3ccccc3)nc1)C2 C(=O)(C1Cc2ccccc21)N1C(C(N2CC(CCC)C2)=O)CN(C)CC1 N1(C(c2ccn(COC)n2)=O)CCOCC(CNC(C2(OC)CC(C)C2)=O)C1 c1(C(N2C(C)CCC(NC(CCCOC(C)=O)=O)C2)=O)c(O)nnc2c1CCC2 C(=O)(C1CC(NS(=O)(=O)c2cnn(-c3ccccc3)n2)c2ccccc21)OCC C1(C)CCN(C(=O)C(S(C)(=O)=O)C2CC2)CC1.C(C(=O)N)NC(=O)NC C=CC(CC)CC(=O)NC(CCNC(=O)CCCc1nc(CC)no1)C(C)C C(c1ccncc1)=CC(=O)NC(Cc1cc[nH]n1)C(=O)NCCCCC1CC1 C1(C(=O)OC)C(F)(F)C12CC(C(N1CCN(C(C3(F)CCC3)=O)CC1)=O)C2 C12(CNC(CCCC(=O)NCC)=O)CCCCC1N(C(c1c[nH]nc1F)=O)CC2 c1(CC)ccccc1C(=O)N(CCNC(C1(c2ccncc2F)CC1)=O)CC Cc1ccc(-n2nnnc2N2CC(O)(CNC(c3sccc3C(C)C)=O)C2)cc1 c1(C(N2CC(NC(C(=CC3CCCC3)C)=O)C(O)C2)=O)cc(F)cc(F)c1N c1(C(=O)NCC2(Cn3cc(-c4cccs4)nn3)CC2)cccc(F)c1Br c1(NC(C2CCCC(NC(C(C)NC(C)=O)=O)C2)=O)ccc(C#N)c(Cl)c1C N1(C(c2n(CC)c(O)nc2)=O)CCN(C(c2coc(C(F)F)n2)=O)C2(CCC2)C1 N1(C(C(CSC)(C)C)=O)CCC(NC(=O)C(C2(O)CCOCC2)(F)F)C(C)C1 C1(OC)(CNC(=O)Cn2cc(CN3CCOCC3=O)nn2)CCCC(C)C1 Cc1cccn2cc(C(N3CC4(CC(NC(C5(C(F)F)CC5)=O)C4)C3)=O)nc12 C(C(=O)N1OC2C=CC1CC2)(C1(O)CCC1)NC(c1cccc(C)n1)=O CC1(C)Cc2cccc(C(N3CCN(C(C45CC(C)(C4)C5)=O)CC3CO)=O)c2O1 C1(NC(C(C)CN2CCOCC2)=O)COCCN(C(=O)C2=CCCO2)C1 N1(C(C(CCCC)(C)F)=O)CCC2(C1)CN(C(=O)COc1ccsn1)CCO2 N1(CCC)CCCC(C(N2CC3CC3(NC(=O)C(CO)N(C)C)C2)=O)C1 CC1CN(C(C)C(=O)NCSc2ccccc2)CCN1C(C1CC=CCC1)=O CCCCC(C(=O)N(CC)CC1(n2ccnn2)CC1)NC(N)=O CN1C2CCC1CC(N1CCCC(c3nnc4ccccn34)C1)C2 c1(C(N2CCCC(C(CNC(COC(C)C)=O)(C)O)C2)=O)ccc2n[nH]cc2c1 c1(C=O)cccc([N+](=O)[O-])c1.C1CCN(C(=O)C)C1.C(C(=O)N)=CC.CC N1(CCOC)CCN(C(c2sccc2Cl)C(=O)NCC2CCOC2)CC1 C(C)(C(O)C(=O)OC1CCOCC1)N(C(C)=O)C(c1ccco1)=O c1(C(=O)NC(CN)CCOC)cc2ccc(O)cc2[nH]1.CCC(C)CC=O C(c1ccc(F)cc1)=CC=O.C1(F)(CNC(CCC2C(C)(C)C2)=O)CCC1 CC(F)(C(=O)NCC1CCN(C(=O)CCC2CC(F)(F)C2)C1)c1ccccc1 c1(C(=O)NCC(C)CNC(C2(C#N)CC2)=O)cc2sccc2cn1 C1(C(C=O)N(C2CCC(C=O)C2)C)CCC(=C2CCC2)CC1.C(C)=O.CC c1(CNC(C2CC=C(C)CC2)=O)nc(CNC(C2COCCO2)=O)cc(O)n1 CC1CCCN(C(c2n[nH]c3c2CCC3)=O)C1CNC(=O)Cn1cccnc1=O C1(C(=O)NC2CC(C(=O)NCC(COC)(C)C)OCC2)CCC2(CCC2)C1 c1(C(=O)NCC2CCC(NC(CCCC(C)C)=O)C2)cc2cc(Cl)ncc2[nH]1 N1(C(C(C=C)(C)C)=O)C2CCC1C(CNC(=O)CC1CCOC(CC)C1)C2 c1(C2C3CCCN32)ccc(Br)c(Cl)c1.c1(C(Cc2n(C)nnn2)=O)ccc(Br)cc1 C1(C(=O)NCc2c(C)nc(C)c(Cl)c2)CC(c2c(F)cccc2F)=NO1 C1(C(=O)NCCNC(C2CCS(=O)(=O)C2)=O)CCCCN1CCO c1(C(=O)NC2C(NC(C(CC)CC)=O)CC2)cc(F)c2nc(O)ccc2c1 c1(OC)cccc(C(=O)NC2CN(Cc3nc(Br)cn3C)CC2(F)F)c1[N+](=O)[O-] Cc1nc(C(=O)NCCN(C(=O)C(c2ccccc2)F)CC(C)O)c(C)o1 c1(C(N2CCCC(NC(C3CC(O)C3)=O)C2)=O)cc(F)c(F)c(Cl)c1F c1(C(=O)NC2(C(=O)NCCn3ncc(C)c3)CCCC2C)ncc2ccccn12 c1(C(N2CCC(C)(NC(=O)C=Cc3ccc(C(F)F)o3)C2)=O)cnccc1C#N C(C(C)(CC(=O)N(C)C)C(F)(F)F)N(C)C.C1CCCN1C(C1COC(=O)N1)=O N1(C(CC2ON=C(C)C2)=O)CC(CNC(C2CCC2)=O)C2(CCC2)C1 C1(C(NOCCCC)=O)C(CC)CCN1C(c1nonc1CC)=O c1(C(=O)NCCC(C)F)c[nH]nc1CNC(c1c[nH]nc1Cl)=O CCC(C)C(C)C(=O)NC(CO)CCCNC(=O)CC#N Cn1cc(C(=O)NCC#CCNC(C2(C3CCCO3)CCC2)=O)cc1Br Cc1cnccc1CCNC(=O)CCN(C)C(C1(CN(C)C)CC1)=O c1(OCC)c(C(N2CCCC2C2CCN(C(=O)CCC(C)(C)O)C2)=O)cccc1F c1(CNC(C(=O)NCCC(C)(C)OC)=O)cc(C)ccc1N1CCCC1 N1(C(CC(n2c(C)cc(C)n2)C)=O)CC2CC(NC(=O)C(F)C(C)C)CC1C2 c1(NC(C(CNC(C=CCN(C)CC)=O)CC2CC2)=O)ccc(O)cc1C C1(CNC(c2ccc(CCC)[nH]2)=O)CCCN(C(=O)CCc2nc(O)n[nH]2)CC1 c1(C(N2CC(CNC(C3CC(=C)C3)=O)C3(C2)CC3)=O)cc(Br)c2nccn2c1 N1(C(C(C)NC(C)=O)=O)CCC(C)(C)C(NC(c2cn(C(C)C)nn2)=O)C1 C=CCCCC(=O)NC(C)CNC(=O)CSCCN(C)C.c1ccccc1 C1(N(C)C(C23CC2CCN3C(=O)C=O)=O)CS(=O)(=O)C1(C)C.C1CC1.N C1(CNC(CC2CC(OC)C2)=O)CCC(F)(C)CC1.c1(C(=O)N)cocn1 CC(C)C(C(=O)N1CCC2CCC12)C(C)NC(=O)CCCC(=O)C1CC1 CC(C)(C)C#CC(=O)N1CCN(C2CN(C(C3(C(F)(F)F)CC=CCO3)=O)C2)CC1 C1(CC(=O)NC2CCC(N(C(C3C(C)CC=CC3)=O)C)CC2)CCC2(CC1)CC2 N1(C(C(C(C)C)c2cnn(C)c2)=O)CCOC(C)(C)C1.C(=O)(CN=S(C)(C)=O)N c1(C(N(C(CCNC(C(N2CC(C)C2)C)=O)C)C)=O)cc(CCO)on1 C1(NC(c2cc(O)no2)=O)CCN(C(c2cc(Cl)c(Cl)[nH]2)=O)CC1F N1(C(C(C2CN(C(C3CCCC3F)=O)C2)OC)=O)CC2(CO)CCC1CC2 N1(C(c2c(C)cncc2)=O)CCOC(C)(CNC(c2cnns2)=O)C1 C1(CC=O)C=NN(C)C1=O.c1(C(C(=O)NC2(C)CC2)OC)ccccc1.N N1(C(c2ccc(I)cc2)=O)CCN(C(=O)C(c2ccc(F)cc2F)O)C2CC12 c1(C(C(=O)NCC2CCOC2)N(CCC)CC)ccc(COC)cc1 N1(C(c2cccc(C#N)c2Cl)=O)CCC2(CCCCC2NC(=O)C(F)(F)F)C1 CC1CN(C(c2cn(C)nc2C(F)(F)F)=O)CCCN1C(c1ccc(F)nc1)=O N1(C(c2cc(OC)no2)=O)CC(OC)C(NC(c2ccnc(S)c2)=O)C1 C(=O)(C1=CCC(C)CC1)NC1CCN(C(C)=O)C1.c12coc(n1)CNC2=O N1(C(CNC(c2ccc(C)cc2)=O)=O)CCCC(C)(C(=O)NCC(=O)O)C1 CCC(C)(C#N)C(=O)N1CCC(NC(c2[nH]c(C)c(C)c2C)=O)C(F)C1 c1(CC(=O)NCC(CO)NC(=O)CC2NC(=O)NC2=O)cc(Cl)cc(Cl)c1 c1(OC)cnc(F)c(C(=O)NCC2CCN(C(C3CCCC3)=O)C2(C)C)c1 N1(CC)CCCC(C(N2CCC(C(C)NC(c3cnc(S)n3C)=O)C2)=O)C1 C1(NC(C(CC)N(C)C)=O)CC2CCC1N(C(C1CC(C#N)(OC)C1)=O)C2 Cc1cnc(NC(C2(C)CCC2)C)c(S(=O)(=O)NC(c2cc(Br)ccc2C)C)c1 C1(CN(C)C(c2c[nH]cc2C(C)(C)C)=O)CCN(C(C2CCCCC2F)=O)CC1 N1(C(c2cc3occc3[nH]2)=O)CC2CCCN(C(C3CCCCC3O)=O)C2C1 C1(C(=O)NC2CCC(C)(O)CC2)CC2(CCC2)CN1C(C1CN(C2CCC2)C1)=O N1(C(CSCCCC)=O)CCC(F)(C(=O)NCC2(C)COCCO2)CC1 C(C)(CS(N)(=O)=O)NC(c1cc(F)ccn1)c1n(CC(=C)C)nnn1 c1(NCC(CC)OC)[nH]c(=NCCCN=c2nccc[nH]2)nc2c1cnn2C CC(C)CC(O)CC(=O)N1C2CCC(C2)C1C(N1CC2CC2C2CC12)=O c1(NCC=C=C)[nH]c(=NC2CCSC2C)nc2ncn(CC)c12 C1(NC(COC)=O)(CNC(=O)C=CCOc2ccccc2)CCOCC1 C(=O)CCCC.C(=O)(CC)N(C(C)C1CC1)C.C1CCCO1.C(=O)C1CC1.S N1(C(c2c(OCC)nccc2)=O)CCCC12CCN(C(=O)CCC(C)OC)CC2 Cc1ccc([N+](=O)[O-])c(Nc2cc(=NCc3cc(Cl)cc(Br)c3)[nH]c(C)n2)c1 c1(C(N2CCN(C(C3CC(F)C3)=O)CC23CC3)=O)cccc2c1CCOC2 C1CCN(C(C2(C)CC(C#N)C2)=O)CC1.c1nocc1C(=O)NC1CC1.CC C1CN(C(=O)C2=NOC(C)(C)C2)C2CCN1C2.Cn1cc(C(=O)NC)n(C)c1=O C1(C)(NC)CCN(C(=O)CC2(C)CCN2C(=O)C(O)CC2CCCC2)C1.CC N1(C(CSC(C)C)=O)CCC(NC(=O)CC(F)(F)C(F)F)C2(CCC2)C1 C1(CN(C)C)CCCCN1C(C1CC(C)(C(=O)OCc2ccccc2)C1)=O C=CCC(CC=C)C(=O)NC(C)(CSC)C(=O)NCCC(C)OC Cc1ccc(C)c(C(N2CCOCC2CNC(C2CCSC2)=O)=O)n1 C1(CC(=O)NC(CC)C(=O)NC)CCN(C(=O)CC(O)COC)CC1 C1(NC(C(N2CCSCC2)C)=O)CC2(C1)CCC2.C1(CC(=O)N)CC(C)(C)C1 N1(C(C)C(=O)ON2CC(C)CC(C)C2)CCN(C2CCc3ccc(Cl)cc32)CC1 C(C(CO)(CO)NC(=O)CC1CCNC1=O)N(C)C(C1C2COCC12)=O Cc1ncc2ccccc2c1C(=O)NCCC(C)N(C)C(c1ccc(F)cn1)=O C1CCN(C(=O)C=CC(C)(C)C)CC(C)(C)C1.CCCCCC(=O)NCC(=O)N N1(C(c2n(CC=C)ccc2)=O)CCN(C(c2ccc(F)o2)=O)CC1CCC N1(C(C(CCC)NC(=O)CCCCOCC)=O)Cc2ccc(C)nc2C1 c1(C(=O)NCC(C)(C)CNC(c2cc(C(F)F)[nH]n2)=O)cc2cccnc2o1 N1(C(c2c(OC)ccs2)=O)CC(C)(C)OCC1C.C(=O)C(C(C)O)N(C)C.N c1(C(N2CCC(C)(CCNC(CC(=C)C)=O)C2)=O)cccc2ccccc12 c1(N(C)C)ccc(Br)cc1NC(=O)C(=O)N(Cc1ccccc1O)C.C1CC1 C12(NC(=O)Cc3cccs3)COCCC1CN(C(=O)Cc1cccs1)C2 c1(CC(=O)N(C(CNC(C(C)Cc2ccnn2C)=O)C)C)ccc(C#N)cc1F c1(C(=O)NCC(C2CCCN2C(=O)C2CC2)(C)C)ccc2cnccc2n1 c1(CCNC(=O)CC23CNC(C2)C3)cc(C(F)(F)F)cc(C(F)(F)F)c1 N1(C(C(CC)C2CCOCC2)=O)CCOC(CN(C)C(C2(OC)CCC2)=O)C1 C1(CCOC)CN(C(=O)CO)CCN1C(C1CCC(F)(F)CC1)=O.C1CCOC1 CC1=C(C(=O)NCC2CCN(C(c3csc(=N)[nH]3)=O)C2)CCCC1 C1(NC(c2ncn(C)n2)=O)CCCCCCC1NC(c1cc(O)cc(C#N)c1)=O c1(CNC(=O)NCC2C3CCN(C(C)=O)C32)cc2c(O)ncnc2cc1F c1(C(=O)NCC(C)OC)ccccc1C.C1(C=O)CCC1(C)C.C(C)(=O)N C1(C)(NC(C(CC=CC)C)=O)CCCN(C(=O)CCc2ncccc2C)C1 c1(OC)cccc(C(=O)NCC(F)CNC(=O)CC2CCC(F)(F)CO2)c1 c1(SCCCCOC)ccccc1C(=O)NCC1(c2ccccc2)CC(S)=NO1 N1(C(c2nc(C)[nH]n2)C(=O)NCC2CCCO2)CC2(C)CN(C)CC2(C)C1 C1(CC(C)O)CCCN1C(=O)CNC(=O)CNC(c1ccsn1)=O c1(C(=O)NCC2CCN(C(COCCCCCC)=O)C2)cc2scnc2[nH]1 CCC(C)(O)C(=O)NCC1CC(O)CN1C(=O)Cc1ccccc1OC C1(C(=O)NC(CN(C(c2cc(C(=O)OC)n(C)c2)=O)C)C)CCC2(CC1)CC2 C1(CNC(C2N(C(c3c(C)noc3N)=O)CCC2)=O)CCCC12CCC2 c1(C(=O)OC)cn2[nH]c(=NC(C)CCN3CCOCC3)ccc2n1 c1(C=O)c(Cl)ccc(Cl)c1O.n1(CC=C)cc(C(=O)NC2CC(F)C2)cn1.C C(=O)(C1=C(Cl)CCCC1)NC(CCC=C)C(=O)NCCCC1(O)CC1 N1(C(c2cncc(SCC)n2)=O)CC2(CCN(C(c3cc[nH]c(=NC)c3)=O)C2)C1 CN1CCC(C)(C(N2CCC(O)(CNC(C3CC34CCSCC4)=O)CC2)=O)C1=O c1(C(N2CCN(CC)CC2)=O)cc(F)c(F)c(F)c1.C12(C(=O)N)CC(F)C1C2 N1(C(CC2(C)CCC2)=O)CCC2(C=C(C(=O)NCCn3ccnc3)C2)C1 N1(C(C2(C)CCCS2)=O)CCOC(CCNC(=O)Cc2ccccc2Cl)C1 C(=O)(CCC(=O)CNC(c1cc(Cl)ccc1NS(C)(=O)=O)=O)OC c1(C(=O)OC)cnc(-c2cn(CCOCCOCC)nn2)nc1.C(=O)C=C N1(C(c2snc(O)c2Cl)=O)CCC(C2(O)CN(C(=O)C(F)CC3CCC3)C2)CC1 c1(C(=O)NCCOCCNC(c2cccc(C)c2F)=O)[nH]c2c(c1C)CCCC2 CC(CC(C)NC(=O)Cc1nnc(O)s1)NC(=O)C(C)(C)N(C)C c1(SC)ccc([N+](=O)[O-])c(C(N2CCC2)=O)c1.C1(C=O)CCS(=O)(=O)C1.C c1(-c2nc(C)on2)cccc(C(N2CCCC(CNC(=O)C)C2)=O)c1.C1CC1.O CCCC(CC)C(=O)NCc1ccccc1CNC(=O)CCC(C)CC C1(N(C)CC=CC(=O)NC2CCCC2)CC(OC(C)(C)C)C12CCC2 CN1CCC2(CC2)C1=O.C1(C=O)C2CC3C(C2)C13.C(=O)C=C.N1CCC1 N1(C(C(C(C)C)C)=O)CCCC(O)(CN(C)C(c2[nH]nnc2C2CC2)=O)C1 CC(CNC(=O)C(CC(N)=O)NC(=O)C(C)n1cccn1)CC(F)(F)F Cc1nc(C(=O)NC2(C(=O)NC(CCO)C3CC3)CCOCC2)ccc1C#N N1(C(C2CN(C(C)=O)C2)=O)CCC(F)CC1.C1(C=O)CCN1S(C)(=O)=O.C C1(C2CCC2)(C(=O)NC2(CNC(C(COC)OC)=O)CCCC2)CC1(F)F c1(CNc2c(C(=O)NCc3cc(Br)ccn3)n[nH]c2)cc(F)c(F)cc1F Cc1cc(-c2cccc(-c3nc(C(N4CCCC(CO)C4)=O)cs3)c2)ccc1F CC1(C)Cc2ccc(Cl)c(NC(=O)NCCOC3CCOCC3)c2O1 C1(C(C)NC(CC2CC(OC)C2)=O)CCCN(C(=O)C(C)(C)N2CCCCC2)C1 N1(C(CC(COC)C)=O)CC=C(CCNC(c2conc2C)=O)CC1 N1(C(c2scc(C)c2)=O)CCC2CC12C(=O)NC1CC(O)C1O CC(CNC(C1OCCC1(C)C)=O)CC(=O)N1CC([N+](=O)[O-])C1 C1(N(C(=O)C)C)C=CCN(C(c2n[nH]c(C(C)(C)C)n2)=O)C1.c1cnn(C)c1 C(=O)(CCCC(C)(C)C)N1CCOC(C)C1C(N1CCCC(CC2CC2)C1)=O c1(C(CN2CC(C(C)Nc3ccc(C)c(F)c3)OCC2)=O)cc(Br)cc(C)c1N N1(C(c2ccc(CC)s2)=O)CCN(C(C2CC(=O)NC(=O)C2)=O)C(C2CC2)C1 c1(CC)ncc(C(=O)NC(C)CC2CN(C(=O)CCC)C2)s1.c1ccccc1.O C1(NC(CCN(c2cc(Cl)cc(Cl)c2)C)=O)C2CCC1N(C(=O)CC1CC1)C2 Cc1cccc(C)c1.C1(CC(=O)N(CCN(C(CO)=O)C)C)CCC(F)(F)CO1 O=C(O)CCCCCCNC(C12CC(CO1)N(C(=O)OCc1ccccc1)C2)=O N1(C(c2cccc(C)c2C)=O)CCN(C(c2cc(Cl)nnc2Cl)=O)CC(C)(F)C1 C(=O)(C1CSc2ccccc21)NC(C1CN(C(c2c(OC)ccc(Cl)c2)=O)C1)C c1(C(N(C(CSC)=O)C)=O)cc2c(cc1[N+](=O)[O-])OCCO2.C(=O)C=O.CC.N c1(C(=O)NC2CC3(CCN(C(CC)=O)C3)OC2)cn(C)c2c(cnn2C)c1=O N1(C(COc2cc(C)on2)=O)CCC(C)(CCNC(=O)C(C2CCOCC2)F)C1 c1(C2(CC(=O)NC3CC3NC(C3CC3F)=O)CC2)ccccc1 CCCCC(CC(=O)N(C)CCc1ccccn1)NC(C1CCCS1)=O CCC(C)CCC(=O)NCC1CCN(C(c2cnc(C3CC3)s2)=O)C12CC2 C#CCC(CC(=O)NCC(CC)C(C)(F)F)NC(C1(OC)CCC(C)C1)=O n1(CC(C)NC(C2(CCNC(c3ccsc3)=O)CC2)=O)ccnc1 C(=O)(C1=NOC2COCC12)NCC(CNC(c1c(C)c(F)ccc1N)=O)CO N1(C(C2(C(C)C)CC2)=O)CCC2CCN(C(C34CC5CC3C4C5)=O)C2C1 N1(C(c2ccc(C(F)(F)F)s2)C(=O)NC)CC(CC(N)=O)OC(C)(C)C1 COn1cnc(C)c1C(=O)NC.C1CC(C(F)(F)F)CN1C(C1CCSCC1)=O CC1=C(C(=O)NC2CCCC(NC(c3nnc(S)n3C)=O)CC2)C(C)(C)CCC1 c1cc(=O)n(C)cc1C(=O)N(C1CCCC1)C.N(S(N)(=O)=O)CC=O.CO c1(OC)noc(C)c1NC(C1CCC1)=O.c1(CCC)cccnc1.C(C=O)O CC1CCN(C(C2CC(CF)C2)=O)CCN1C(C1CC(=C2CCC2)C1)=O C1(CNC(C(C)C)=O)CC(C)N(C(=O)C(C)(C)C2CCOCC2)C1 CC1(CO)CC(c2nnnn2-c2ccccc2)(NC2(CF)CCC2)C1 C#CCCCCC(=O)NCC1(NC(=O)C(n2ccc(C(F)(F)F)n2)C)CCOC1 C12(C(=O)NCCN(C(=O)C(O)Cc3cn(C)cn3)C)CCCCC1CCCC2 Cc1ccc(F)cc1NC(=O)CCNC(C1CC=CC(N)C1)=O c1(N(C)C)ccc(Cl)cc1NC(c1ccc(CCC(=O)O)cc1)=O CC1CC(CC(N2CC(F)(F)CC2C)=O)CC(C)(C)C1.C1(C=O)CCC1(C)C.N Cc1c(Cl)cnc(NC(C)CC(C)NC(C2(c3ccccc3)CC2(C)C)=O)c1C#N N1(C(C(CSC)(C)NC(=O)C(C)SC(C)C)=O)Cc2ccc(O)cc2C1 Cn1nc(Cl)c(C(=O)NC2CC3(C2)CN(C(C2CCC24CCC4)=O)C3)c1Cl CC(C)CC(F)C(=O)N1CCC(CCCCCNC(=O)C(C)SC(C)C)CC1 C1(CNC(C(C)Oc2ccccn2)=O)CCN(C(C2CC2Br)=O)CC1 CON1CCC(C(N2CCOC(C(=O)N(C)CC3CCCO3)C2)=O)CC1 N1(C(C2C(C)(C)OC2(C)C)=O)CCC(C2CC(NC(c3ccns3)=O)C2)C1 C1(C(N2CCC(SC)CC2)=O)CCN(C(c2cnsc2C)=O)C(C)(C)C1 CCC(C)(C)C(=O)NC(C1CCCC1)CNC(=O)Cn1c(C)csc1=O c1(C(N(CCNC(C2CC(C)(CC)C2)=O)CC)=O)c(N)cc(Cl)cc1F N1(C(c2cnc(-c3ccccc3)[nH]2)=O)CCCC(c2ccccc2F)C1 C1(N(C)C(c2n[nH]c3c2CC(C(C)(C)C)CC3)=O)C2CC3CC1CC(O)(C3)C2 CCCCC(=O)C(=O)N1CCCC1(C)C(=O)NC1(C2CCCO2)CC1 C(C(C(=O)N=S(C)(=O)c1ccccc1F)OC)c1c(CC(=O)OC)cccc1 O=C(C1=NN2CCCN=C2N1)NCC1(O)CN(C(C2CC(n3ccnc3)C2)=O)C1 CN1CCC(C(=O)NCCCS(C)=O)(NC(c2cn[nH]c2)=O)C1 C(C(C)C)(C(O)C(=O)N1CCC(CCNC(c2cn3ccsc3n2)=O)CC1)OC c1(CC)c(C(=O)NCC2(NC(=O)C(O)C3CCC3)CC2)cnn1CC N1(C(c2scc(C)c2)=O)CC2(C1)C(NC(=O)C#CC1(C)CCCO1)CCS2(=O)=O CCCCCC(C)(C)C(=O)NCC1CCOC1C(=O)NC(C1CCCCC1)C C(CC(=O)NCc1noc(C)n1)(C(F)F)NC(C1N(CC)CCCC1)=O.O c1(C(=O)NCC2CCN(C(C(CC)OC)=O)C2)ccnc2cc(F)cnc12 C(=O)(C(C(C)(C)C)OC)N(C(CC)CC(=O)N1CCCCC1CN(C)C)C C1(C)(COC)CC(NC(c2ccc(Cl)cc2)=O)CN1C(=O)C=O.CC(F)F CN1CCC(C)(C(N2CC(N(C(=O)C=CBr)C)C(C)(C)C2)=O)C1=O C1(CC(=O)NCC2N(C(C3CCC(C)(C)C3)=O)CC2)CCCCC1(C)C Cc1cc(Br)cc(F)c1C(=O)NC1CC1CNC(=O)Cn1cnnn1 N1(C(c2c(C)nn(C)n2)=O)CCN(C(c2cncn2C2CC2)=O)CC(C)C1 C12CCCCN1C2.c1(C(C)NC(=O)NC)ccc(OCC#N)cc1 N1(C(C)=O)CC2CC1(C(N1CCOC(CNC(=O)CC)C1)=O)C2.C(N)=O.N c1ccc2c(c1)CCC21CC1CNc1cncnc1 C12(CC(=O)OCC)CCCCC1N(C(c1cnc(F)c(C)c1)=O)CCC2 c1(C(=O)NCC(CN(C(=O)CCC2CCCN2C)C)(C)C)ccc([N+](=O)[O-])o1 N#Cc1c(N2CCC(CNC(C3CC34CCSCC4)=O)C23CC3)cccc1F c1(C(N(C(C)C)C)=O)ccc2c(c1)nc(C)n2C.C1(CCOC)(C=O)CCC1.N C1(NC(c2cnc(C(C)C)[nH]2)=O)CCN(C(=O)Cn2cc(C(C)=O)nn2)CC1 C1(NC(Cn2cc(C(=O)NC)nn2)=O)CCC(C)N(C(c2ccoc2)=O)C1 c1(C(=O)NC(CC)CNC(c2cnccn2)=O)c[nH]c(C#N)c1C c1(OC)ncc(F)cc1C(N1CCN(C(=O)C(C)(O)c2ccccc2)C(C)C1)=O C1(NC(C2(OCC)CCC2)=O)CCN(C(c2[nH]c(=N)ccc2C)=O)CC1(C)C C1(NC(C2CCOC2)=O)CC(NC(C2C3CCC2(c2ccco2)C3)=O)CC1O C1(CCOC)(CNC(=O)C(Cc2ccccc2)N(C)C)CCCC1 C(=O)(CCCN(C)C(C)=O)N(CCCC)C.C(=O)(C=CI)NCC(=O)N C(=O)(CC(C(F)(F)F)OC)N1CC(CNC(c2c(C#C)c[nH]n2)=O)C(F)(F)C1 C(CC(C(=O)NCCNC(=O)CCn1ccnc1)N(C)C)N(C)C.C1CC1.C C1(CNC(CCC=C)=O)CN(C(c2cn(C)nc2OCCC)=O)CCO1 c1(CC)cnc(CC(=O)NCC(C)CN(C(=O)CC2COC(=O)C2)C)[nH]1 c1(C(N)=O)cccc(CCC(N2CCC(NC(=O)CC3CC4CC4C3)C2)=O)c1 CC1CC(C(N2CCC(O)C(C)C2)=O)CN(C(=O)CC2CC=CC2)C1 Cc1cc2[nH]c(=O)c(C(=O)NC3CC3NC(=O)C#CC3CCC3)cn2n1 N1(C(c2ccc(SC(C)C)cc2)=O)CCC(C)(C)C1.C1(C)CCC1.C(=O)C.N N1(C(c2ccn(CC)c2C)=O)CC(C)CN(C(c2cn(C(F)F)cn2)=O)CC1C C1(C(=O)NC2(C=C)CCCC2)CN(C(c2cccnc2S)=O)CC1C=CC C1(NC(c2cc(OC)ns2)=O)CCCCC12CCN(C(c1coc(C#N)c1)=O)C2 C(=O)(C(C)(C)CC(=O)N(C1CN(C(=O)C#CC(C)C)CC1(C)C)C)OCC N1(C(c2n(CCC)ncc2)=O)CC2(CC(C)C2)C1.c1(C(C(=O)N)O)ccnn1C Cc1cc(C)c2cc(C(=O)NC3C4CC3N(C(=O)Cc3ccco3)C4)sc2n1 N1(C(C=Cc2ccc(C)s2)=O)CCCC12CCN(C(=O)CN1CCC(C)(O)C1)C2 c1(C(N2CCC(N(C(COC(CC)C)=O)C)C2)=O)cncc(-n2cnnn2)c1 c1(OC)cc(C(=O)NC2(CO)CCN(C(c3ccoc3)=O)CC2)cc(Br)c1Cl C1(O)(CNC(Cc2cc(C)[nH]n2)=O)CCCN(C(C2CN(C)C(=O)N2)=O)CC1 CCC(CNC(=O)C=CC(C)NC(=O)C(c1cnn(C)c1)C)(CC)CO O=C1CCC(C(=O)NCC2(C(=O)NC3(C4CCC4)CC3)CCCO2)CC1 N1(C(c2c(C)cccc2C)=O)CC2(C1)SCCC2NC(C1CC2CCC2C1)=O C1(CCC(=O)N(CCNC(C=C(CCC)C)=O)CC2CC2)CCC(C)O1 C1(C)(CC)C=C(C(=O)N2CC=CC2CNC(=O)CCC2CCN(C)CC2)C1 N1(C(CN(C)CC)=O)CCCC1(C)C(=O)N(C1CCN(C)C1=O)C N1(C(C(CC)Cl)=O)CC2CN(C(C3CCCSC3)=O)CC2C1 c1(C(=O)Nc2cc(C)ns2)cc(-c2ccc(C3COC3)cc2)ccn1 N1(C(CCOCC#C)=O)CCC(C(=O)NCC)C(O)C1 C1(CC(=O)N(C(C)C)CCF)CCCC(NC(=O)Cc2ccnn2C)C1 CC(C)CC(CNC(=O)Cn1cc(C(F)(F)F)nn1)NC(c1cnco1)=O c1(C(N2CCOCC2(C)C)C(=O)NCCCSC)ccc(-n2cccn2)c(F)c1 C1(C(N2CC(C)(CC)C2)=O)N(C(=O)CCOC2CCCC2)CC12CCCC2 C12(C(N(C(CC)C)CCO)=O)CCCC1CN(C(c1cscn1)=O)C2 N1(C(CC2CCC(=O)O2)=O)CCC2(C1)CN(C(C1CC3CCC1C3)=O)C2 C(=O)(C#CC1CCC(=O)CC1)NC1CC(C)N(C(c2cnn3cc[nH]c23)=O)C1 c1(N2CCCCC(NC(=O)Cc3ccoc3)C2)ncnc2sc([N+](=O)[O-])cc12 c1(CC)c(C(=O)NC(C(F)(F)F)C2CCCC2)cnn1-c1ccc(F)cc1 c1(NCC2C(C)COCC2)nc2ccccc2nc1N1CCn2c(O)nnc2C1 N1(CCC)CCCC(C(=O)NCC(C(C)(C)C)NC(C2(CCO)CC2)=O)C1 c1(C(=O)NC(C2CCCN(c3snc(COC)n3)C2)C)ccc(C)c(F)c1 c1(NC(C(C)C)CNC(=O)C2=C(Cl)CC2)cc(S(C)(=O)=O)ncn1 C(C1CN(C(C2(C#N)CC2)=O)CC1C(=O)NCCN(CCC)C)=CC Cc1c(S(N)(=O)=O)sc(C(N2CCC(C)C2C)=O)c1Cl.c1(C(=O)N)cc[nH]n1 c1(C2(C(=O)NCC(CNC(c3c(C)snn3)=O)O)CCCC2)cccc(Cl)c1 C1(C(=O)NCC2CN(C(C3CCC(F)C3)=O)CCO2)COc2ccc(O)cc2O1 C(N=c1[nH]nc(-c2ccccc2)o1)(c1ccccc1)c1ccnnc1 Cc1ccc(Br)cc1C(=O)NC1CCC(NC(C2C(C)C2C)=O)CC1 c1(-c2nc(NC(=O)CNc3ccc(Cl)c(F)c3)[nH]n2)ccc([N+](=O)[O-])cc1 C1(NC(C(CC)F)=O)CN(C(c2cnsn2)=O)CCC12CCOCC2 N1(C(c2cc(C)c(C(N3CCC(O)C(F)C3)=O)o2)=O)CCC2(CC1)CC(O)C2 c1(NC(C(COC)(C)C)c2nnnn2C2CCCC2)cc(F)cc(Cl)c1 c1(CCC(N2CCC(CNC(C(C)=C3CC3)=O)C2)=O)cc(C)nc(C)c1 C1(NC(=O)CCCc2cncs2)COC2(CCN(C(C3CC=CC3)=O)CC2)C1 c1(CC(N2CC(NC(=O)COC3CC=CC3)C3C2C3)=O)ccc(O)c(F)c1 C1(F)(C(=O)NC)CCN(C(C(=O)NCCCS)C2CC(CC(C)(C)C)C2)C1 CC(C#N)CCC(=O)N1CCC(O)C(NC(c2ccco2)=O)C1 Cc1cc(CC(=O)NC2CCN(C(=O)CCC3(C)CCC(=O)N3)C2)ccc1O N1(C(C(C(CC)O)C)=O)CC(C)N(C(=O)CC23CCC(CC2)C3)CC1C c1(CCC)ccc(C(=O)NC(CNC(C2CC2Br)=O)C(C)C)cc1 C(CCCCC(=O)NC1CCCN(C(c2cc3sccc3[nH]2)=O)C1)OCC Cc1cc(S(N)(=O)=O)oc1C(N1CCN(C(=O)CCCCCF)CC1)=O Fc1cccc2[nH]c(=NCC3CCCS3(=O)=O)[nH]c(=NCCn3cncn3)c12 C(=O)(C1=C(C)CCOC1)N1CC(C(=O)NC(CC)COC)C(F)(F)C1 C(=O)(C(C)(C)CNC(c1cncc(C)n1)=O)NC(CCC)CO Cc1cc(C)cc(C=CC(=O)NC2CCCCC2)c1.c1(CC=O)cnn(C)c1.N C1(C(=O)NCC2N(C(CC3CCC(C)(O)CC3)=O)CC2)CCc2nnnn2CC1 c1(C(N2CCN(C(C(C)OCCCC)=O)C(CO)C2)=O)cn(C)c(=O)nc1O CCCC(C)(CC)C(=O)NCC1CC(O)CN1C(=O)CNC(C)=O c1(NC(C2(C)N(C(c3c(C)c(F)ccc3)=O)CC2)=O)ccnc(O)c1[N+](=O)[O-] C12(C=O)CCCCC(=O)N1CCC2.C1(C(N(C)CCOCC)=O)CC1(C)Br.N C=CC1(C(=O)NCCCC(C)NC(c2cnncc2OC)=O)CCOCC1 c1(C(C)C(=O)NCC(F)CNC(C2(Br)CC2)=O)cncnc1 C(CN=c1cc(C)nc(CC2CC2)[nH]1)N(C(C1Cc2ccncc2C1)=O)CC C1(C)(C(=O)NC(CNC(c2cnc(C)nc2)=O)C2CC2)CCNC(=O)C1 S(=O)(=O)(c1[nH]c(=NC2CCN(c3nccs3)C2)ccc1Br)NCC(CO)OC n1(CC(=O)NC2C(C)N(C(C3CC3C(N)=O)=O)CC2)cnc2sccc2c1=O Cc1ccc(F)c(CC(=O)NC(C)C(C)(C)NC(c2ccnnc2C)=O)c1 CCCC(C)(O)C(=O)NCC1CC(NC(c2cnc(-c3ccccc3)[nH]2)=O)C1 c1(C=O)ccc(S(N)(=O)=O)cc1Cl.C(C)(C)(CC)NC(C(C)n1cccc1)=O.N n1(CCNC(=O)NCC2CC(C(C)(C)C)C2)ncc(F)n1 n1(CC(N2CC=CC(NC(CCCC#C)=O)C2)=O)c(C)c(C)sc1=O C(CCCCCC(=O)N1CCCC(SC(F)F)C1)c1nnc(C2C(C#N)CCC2)o1 C1(C2CCN(C(C3CCCC3)=O)CC2)(NC(=O)Cc2ccc(Cl)cc2F)CCC1 N1(C(C2ON=C(C)C2)=O)CC2CCCC1C2CNC(=O)C=CC1CCCC1 c1(NCC(C)CO)cc(=NCC(C)c2ccc(N3CCCC3)nc2)[nH]cn1 N1(C(CSSC)=O)CCC2(CCCN(C(=O)CCc3cccnc3F)C2)C1 C12(NC(Cc3ccc(OC)cc3Cl)=O)CCCN(C(c3cnsn3)=O)CC1C2 c1(CCC(=O)N(C(C)CNC(=O)CCS(N)(=O)=O)CC)c(C)ncnc1O N(C1CCC(NC(=O)C(O)C2CCC2)c2ccccc21)c1ncnc(C)c1C#N c1(CCCC)cc(C(=O)NC(CN(C)C(C2CCCOC2C)=O)CC)c(C)o1 c1(C(=O)NC2CC(Nc3ncc(OCC(F)F)cn3)C2)occ2c1CCC2 C(CC1=CCCCC1)N(CCNc1ccccc1)C.c12nccn1CC2 C(=O)(C1(C)CCc2ccccc21)NCc1ccc2scc(C)c2c1 C1(CN(C(C2C(C=C)C2)=O)C)COCCN1C(c1csc(-c2cn[nH]c2)n1)=O C1(NC(C2CCCN(C)C2)=O)CC(F)(F)CC1NC(c1nonc1N)=O C1(C(N2CC(C(C)(C)C)C2)=O)CC(C)(C)C1.C1(CC(=O)N)(N(C)C)CC1 C(=O)(CC(C)(C)CCC)NC1CN(C(c2cn(CC=C)nc2)=O)C1 c1(NC2(CO)CCCN(C(C3CC(C)(C)C3)=O)C2)ccc([N+](=O)[O-])cc1 Cc1cc(C(=O)N(CC)C2CC2)cc(C)c1F.c1(C(=O)N)cnnn1C1CC1 C=CC1(NCC2CC(C(C)C)=NO2)CCCCC1 C1(C(CC)C)CCCN1C(=O)COC1CCN(C(=O)CCc2ccn(C)c2)C1 N(C1c2ccccc2CC1C)C(C1C(c2ccc(OC)cc2)N(C)C(=O)C1)=O O=C1NCC(OC(C2(O)Cc3ccccc3C2)=O)n2ncc(Cl)c21 Cc1cccn2c(=O)c(C(=O)NCC(O)CCNC(C3(C)CC3)=O)cnc12 N1(C(CCCNC(=O)OCC)=O)CC2CC(C)N(C(=O)CCc3cnn[nH]3)C2C1 CC(C)C(F)(F)F.C1(C#N)(C=O)CC1(C)C.c1(COC)cc(C=O)on1.N N1(C(C2CN(C(c3cnc(CC)s3)=O)C2)=O)CC(C)OCC1C c1(CC(=O)N)cc(C(F)(F)F)cc(Cl)n1.C=C(Cl)CCC(=O)N1CCC(CF)C1 n1(CCOC)cc(C(N2CCC2CCNC(=O)CC)=O)nn1.C(C)(C)C C1(NC(C(CC)(C)C)=O)CCCCN(C(=O)COC2CCOC2)C1 Cc1cc(C(=O)NCCCC2CCN(C(C3CCCCC3C)=O)CC2)c(C)cn1 Cc1cc(C(=O)N(C)CC2CCN(C(C3CC34CC4(F)F)=O)CC2)c(C)cn1 C(=O)(CCCC(C)(C)C)N1C(CNC(C(CC)CC)=O)CC(C(F)(F)F)C1 c1(COC)nc(C)c(C(=O)NCC(O)CCNC(=O)CC2CCCC2)s1 CC(C)C(CCN(C(=O)C(C)OC1COC1)C)NC(=O)Cc1cnoc1 c1(NC(CC2CCN(C(c3n(CCOC)ncc3)=O)C2)=O)cccc(O)c1 N1(C(c2c(CNC(CC(C)C3CCCO3)=O)n[nH]c2)=O)CCS(=N)(=O)CC1 C1(C(=O)N)CC2(CCOCC2)C1.C1(C(C(=O)NCCC2CCCC2)=O)CCCCC1 N1(C(c2n(C)ccn2)=O)CCCC2(NC(=O)CCc3cccnc3)CC2C1 C(=O)(C=CSNC(=O)OC(C)(C)C)NC(c1noc(C)n1)CC CC#CCCCC(=O)NCC1CC2CC2N1C(=O)C(C1CCCCC1)C N1(C(C(CC)N(C)C)=O)CCCC2(CN(C(=O)CC(O)CC3CC3)C2)C1 N1(C(CCCOC)=O)CCCCC2(CCN(C(c3nccc(C)c3N)=O)C2)C1 C1(C(=O)NC(CNC(c2cc(CC)ncc2)=O)(C)C(C)C)CCCCN1N=O CCC(CC)(CCNC(C1CCCC1OC)=O)NC(=O)C(=Cc1cccs1)C c1(C(=O)NCC2(OC)CN(c3nnc(O)s3)C2)cc2c(nc1O)CCC2 CCCC(C#N)C(=O)N1CC(OCC)C(NC(=O)CSc2cccc(C)c2)C1 CCCCCC(O)CC(=O)N1CCC(NC(=O)Cc2nn(C)cc2Cl)C12CC2 C1(CC(N2CC(C)C2)=O)CCCCC1C.c1(CC(C)NC(=O)CO)nncn1C Cc1nc2ccc(C(N3CCC(N(C)C(c4cccc(Br)c4)=O)C3)=O)cn2n1 C(=O)(CC1=CCN(C)CC1)N1C(C)(C(=O)NCCCCCN(C)CC)CCC1 C(=O)(C(CC(C)c1ccccc1)N(C)Cc1n[nH]c(C)n1)NCC=C C1(C(N2C(C)CC(CCNC(=O)C=C3CC3)CC2)=O)CCc2ncncc2C1 Cc1c(C(N2CCC(NC(c3cn(C)c(C(F)F)n3)=O)C2)=O)nc2sccn12 c1(C(=O)NC2C3CN(C(C4OCC(C)(C)OC4)=O)C2C3)cc2c(F)cccc2[nH]1 C(C(F)(F)C(=O)NCC1CC(C(=O)NCCOC(C)=O)CO1)OC N1(C(c2cc(C)sc2C)=O)CC(NC(=O)Cc2ccnc(O)c2)C(C)(C)C1 c1(C(N(c2nnn(C)n2)C(=O)CN2CCNCC2)=O)nc2ncccn2n1 c1(C(N2C(C)CC(NC(c3c(C)[nH]nc3Cl)=O)C2)=O)cc2cnccc2[nH]1 N1(C(CN(C2CC2)CC)=O)CC(CNC(=O)CCc2nncn2C)C1.C C1(CCC)CN(C(c2cc(C)nc(O)n2)=O)CCN1C(=O)C(O)CC(C)C c1(NCc2c(C)cn(C)n2)[nH]c(=NCC(=O)NC2CC2)nc2c1cnn2C(C)C c1(CC(C(=O)N(C2CCCN(C(C3(CCF)CC3)=O)C2)C)O)c(F)cccc1Cl Cc1cnccc1C(=O)NC1CCN(C(C2CCCS2(=O)=O)=O)C1 CC1CC(C)CN1C(=O)Cc1ccccc1Cl.c1(C(=O)N)cc(C2CC2)n(C)n1 N1(C(C2=CC(C)C2)=O)CC2(CC2)CC1CNC(=O)C1=C(Cl)CCC1 C1(C)(C(=O)N)Cc2ccccc2C1.C1(N(C)C)(C(=O)NCC2CC2)CCCC1 N1(C(C(CNC(c2cn(C(C)C)cn2)=O)OC)=O)CCOCC(C)(F)C1 O=C1CC(C(=O)NCCCNC(C2CCN(Cc3cccnc3)CC2)=O)CCN1 C1(C)(C(=O)NCC(C)(C)C)CCN(C(c2ccsc2)=O)C1 C1(=CCOC(C)C=O)CCN(C)CC1.N12CCCC1CC1CCOC1C2=O.N n1(COC)cc(CNc2cnnn2CC)c2ccccc12 c1(C(N(CC(CCC)O)C)=O)ccc(CNC(C2CCC(C)C2)=O)nc1 n1(CC(=O)NCCCn2ccnc2)cc(C2(O)CCCC2)nn1 C1(CNC(c2c(SC)cn(C)n2)=O)CCC12CCN(C(=O)C1=CCOCC1)CC2 N1(C(c2ncn(CC)n2)=O)CC=C(C(C)(C)C(=O)N2CCC2C(=O)OC)C1 C1(NC)CCCCC1.C1(Cn2cc(C(C3CCCC3)OC)nn2)CCC(C)CO1 N1(C(CN(CCC)C(C2CCCN2C)=O)=O)CCC(C)(F)C1 C1(NC(=O)C=CC2CCC2)CCC(Cn2cc(C3CC4C=CC3C4)nn2)CC1 C(C(C)C)(C(O)C(=O)NC(C)(C)C(=O)NCC1COC(C)(C)C1)OC c1(C(N2CCC(C(C)(O)CNC(c3nc(Cl)cs3)=O)CC2)=O)cnn2ccsc12 C(=O)(C1=C(Cl)CCOC1)NC1C(NC(CCCC(N)=O)=O)CS(=O)(=O)C1 C(=O)(CCC(=O)NC(C)C(C)(C)C)N(CC)CC.c1(C=O)cccnn1.N C1(NC(=O)CN2CC3CCC2C3)CCCC2CN(C(=O)C3=NNC(=O)C3)CC12 c1(OC)ccc(C(N2CC(O)CC2C)=O)c(F)n1.c1(C(=O)N)c(O)cccc1Cl N1(C(C2(C#N)CCCCC2)=O)C2CC=C(C(=O)N3CC(F)(C4CC4)C3)C1CC2 c1(C(C=O)=O)cc(F)ccc1F.Cc1ccc(C(=O)NCC2CC2C)cn1.N N1(C(C(CCCC)O)=O)CC2CCCC1(CNC(c1cc[nH]c(=NC)c1)=O)C2 CCC(C)(COC)C(=O)NCC1(C)CCCN1C(=O)C=CC1(C)COC1 c1(OC)ncc(-c2cn(C(C)C(N3CCOC(C(=O)N(C)C)C3)=O)nn2)cc1F c1(CNC(c2snc(O)c2Cl)=O)cccc(NC(C2CCC2F)=O)c1 C#Cc1ccc(C(=O)NCC2(C(=O)N)CCC2)cc1C.C1(C(C)(F)F)CC1 C1(CNC(C2(C#C)CCC2)=O)COCCN(C(=O)Cn2c(C)csc2=O)C1 C#CC1CN(C(C2CC23CCCCC3)=O)CCN1C(C1CSC1)=O c1(C(=O)NCC2(NC(CCCC)=O)CCC2)ccccc1-c1ncn(C)n1 C(=O)(C1=CC(C)(C)C1)NC(C)CC.C(=O)CCN(C)C=O.C(C)(C)C.N C1(C)(NC(C(c2ccccc2)Sc2c(OC)cccc2)=O)C(C)(C)C1(C)C c1(C(=O)NCC(CNC(C(CCC)O)=O)O)cc2cccnc2cc1F C#CCC(C)C(=O)NC1CN(C(C2(O)CC2)=O)CC1SC C(=O)(C(CC#CC)NC(=O)CCOC)NC(CSCC)CO C(C(C)(C)C(=O)N)OCC.C1CN(C(=O)CCC2CCC(C(N)=O)O2)C1 c1(NC(=O)NC(c2ccncc2F)C)ccc(Cl)c(-c2ccccc2)c1 Cc1[nH]c2ccccc2c1NCc1ccc(OCC#N)cc1 N1(C(c2cccnc2F)=O)CC2(CCC(C(N3CCC(F)C3)=O)O2)C1 C(=O)C(C)C=O.c1(CC)ccccc1F.C1(NC(CNC(C)=O)=O)(C)CCC1 c1(NCCSC(C)C)ncccc1S(=O)(=O)NC(C)CCC(C)(C)C Cc1nc(Cl)ccc1CN1CCOC(CC(=O)Nc2cc(Br)cnc2Cl)C1 CCC(CC(F)F)C(=O)NCC(C1CCCN1C(=O)C(C)N1CCC1)(C)C c1(C(=O)NC2(COC)CN(C(=O)CCC(C)C)C2)sc2sccc2c1Cl CC1CC(C(=O)NCCC(C)NC(c2cccc(C3(C)CCO3)c2)=O)CCC1C CC(C)(C#N)CCC(=O)NCC1CN(C(C2CCCC3CC23)=O)C1 c1(CCC(N2CC(CC(C)NC(CCC#C)=O)C2)=O)ccc(C)cc1Br Cc1ccc(C=CC(N2CC(NC(C3CCCC3C(C)C)=O)CC2(C)C)=O)cn1 C(=O)(CC1CN(C)c2ccccc21)NCCNC(C=CC(C)C)=O.C1CC1.C N1(C(C2C(C)C2)=O)CC=C(C(=O)NCC2(C)CCOCC2)C1 CCC(CC)(C(N)=O)NC(=O)CC(C(F)F)NC(=O)COCC(C)C C1(NC(C(CCOCC)NC(=O)CCC2OCCO2)=O)CNC(=O)C1(C)C C12(C=O)CC3CC(CC(C3)C1)C2.c1(CNC(C2CC2)=O)ccccc1.C C(=O)(C#CC1(C)CCCO1)N1C(C(N2C(C)CC3(CCC3)C2)=O)CC(O)C1 c1(C(N(C(CC)C)C)=O)oc(CNC(=O)CC2(SCC)CC2)cc1C.C c1(C(=O)NCC(CC)NC(c2cnc(C)s2)=O)csc(C(F)F)n1.C1CC1 Cc1nnc2n1CC(C(=O)N(C1CCN(C(c3cc(F)cc(F)c3O)=O)C1)C)C2 C1(CC)CCCCC1.C(=O)C(F)CC1CN(C(=O)CN(CC(C)(C)C)C)C1.C c1(CNCC23C(CN(C(Cc4cc(C)n(C)n4)=O)C2)C3)cc(Br)c(F)cc1O C1(NC(C2CC(F)CN2C(c2ccnnc2O)=O)=O)CC(=O)N(C2CC2)C1 C1(NC(C2(C)CCCO2)=O)CCCC(CNC(=O)C(=O)NC2CC2)C1 C(C)(C)(C(=O)NCC#CCNC(=O)CCCSc1ccccc1)OC C1(NC(C2CN(S(CC)(=O)=O)C2)=O)CCN(C(=O)CCS(=O)(=O)N)C12CC2 Cc1cc(C(=O)NCC2CCCCCN2C(C2CCS(=O)(=O)N2)=O)cc(O)n1 C(CCN(C)C)(C(=O)NC)NC(C=CC=CCCCCC)=O.c1cnnn1C.C C=C(C)C1OCCC1CNCCCCc1cccc(C(F)(F)F)c1 C1(NCCN(C(C(C)NC(=O)NC)=O)C)CN(C(C)=O)CC12CC2 C(=O)(C(C)(O)C(F)(F)F)N(CCCCNC(C1C(C)(C)C1(F)F)=O)C c1(C(=O)NC2CC(CC(=O)NCC)C2)ccc(C)cc1 N1(C(c2c(CC)ocn2)=O)CCC(NC(=O)Cc2c(O)ncnc2O)C12CC2 C(=O)(C1=CCN(C(C2(C)CNC(=O)C2)=O)CC1)NCC1C(C)(C)C1(C)C CC1CCCCC1CNC(c1ccc(F)cc1N)=O.C12(C=O)CC(C)(C1)C2.N C1(C(=O)NC(c2nc(CC)on2)C)CCC2(CC2)N1C(=O)C(C)CO N1(C(CCCC)=O)CCCC(C(=O)N(CCNS(=O)(=O)NCC(F)(F)F)C)C1 C1(CC)CN(C(c2csnn2)=O)CCC1N=c1cc(C(N)=O)nc(Cl)[nH]1 S(=O)(=O)(c1ccc(-c2ccc(F)cc2C)s1)NCC(CC)N1CCCC1 c1(CC)ccoc1C(=O)NCC1CCN(C(=O)CCN(CC)CC)C1 C(=O)(C(CO)C(F)(F)F)N1C(C(=O)NCC2(C#C)CCOCC2)C(C)CC1 S(=O)(=O)(c1cc(C(F)(F)F)ccc1N1CCCCC1)N1CCCC(C)(C(=O)O)C1 C1(C(=O)NC2CCCC2CCO)CSCCN1C(=O)CCC1CCOCC1 N1(C(CC2(N(C)C)CCCC2)=O)CCC(O)CC1.C1(F)(C=O)C(C)(C)C1(C)C.N Cc1cc(C(=O)NCCCCNC(C2CC(C)(C)CO2)=O)ncc1Cl C(CCCC(=O)N(C)CC1CCCN(C(C2CCCC2(C)C)=O)C1)N(C)C C1(NC(=O)C(C2CCN(C(c3ccn(CCF)n3)=O)C2)F)CC(O)C(O)C1 C(C)(CCC(=O)N1CC2CC1C2CNC(=O)C(F)(F)C1CC1)SC c1(C(=O)NCCC2CC(NC(c3cc(CC)ncc3)=O)C2)cc(C)ccc1Cl c1(C(N2CC(C)C(NC(C3CCCCC3O)=O)C2)=O)ccc(S(=O)(=O)N(C)C)o1 C1(C(=O)NC2C3CN(C(C(C)CC4CCCC4)=O)C2C3)CNC(=O)CC12CCC2 C1(CCOC)(NC(C2CCCC(=O)N2)=O)CCN(C(c2c(C)cnn2C)=O)CC1 Cc1nc(O)nc(O)c1CCC(=O)NC(C(F)(F)C(=O)O)c1ccccc1 n1(C(CNC(C(C2CCCCC2)OC)=O)C)cc(CC2CCCC2)nn1 c1(C(=O)N)ccc([N+](=O)[O-])n1C.N1(C(C(C)n2cccc2)=O)CC2(CC2)CC1C C1(C(N2CCC(C)(C)C2)=O)CNC(=O)CC1(C)C.CN1CCC(CC(=O)NC)C1 C1(C(=O)NCC(CC)NC(=O)Cc2ccc(C(C)=O)cc2)COCC1(C)C c1(C(=O)NC(CNC(c2c(Cl)ccc(C#C)c2)=O)C)cccc2c1ccn2CC Cc1ccc(C(=O)NC2(C(=O)N(C3CC(C)CC(C)C3)C)CCCCC2)cc1C N1(C(C2(C#N)CC23CCC3)=O)CCOC2(CCN(C(c3ccc(=O)oc3)=O)C2)C1 c1(SC(C(=O)NC2CCN(C(c3cc(OC)no3)=O)C2)C)ccccc1Cl Cn1ncc2ccc(CN3CC(NC(c4ccccc4)=O)C(F)C3)cc12 Cc1cc([N+](=O)[O-])cc(C(N2CCC(CO)(NC(=O)C(O)CC(N)=O)C2)=O)c1Cl C=CCCC(C(=O)NC1COCC1OC)NC(C1CCCCC(=O)N1)=O c1(N2CC(N(C(=O)CCc3ccccc3Cl)C)C2)ncnc2c1CCC2 c1(C(=O)NCCC(CNC(C(CC)SC)=O)O)ccc(S(N)(=O)=O)c(Cl)c1 CS(=O)(=O)c1ccc(NC(C2CC(NCc3ccnc(F)c3Cl)C2)=O)cc1Cl c1(C(C)=O)cccc(N(Cc2ccccn2)Cc2cccnc2Br)c1 N1(C(C(CC)n2nccc2C)=O)CC2CCN(C(C3CCS3(=O)=O)=O)CC12 n1(C(C)(C)C)cnc2c(NOC3CCCCO3)nc(C(F)(F)F)nc12 c1(OC)cccc(SCC(=O)N(C2CC(NC(=O)Cn3cnnc3)C2)C)c1 C1(CNC(C(C2CCC(=O)N2C)C)=O)CCCN(C(C23CSCC2C3)=O)CC1 c1(CC(=O)OCC(c2c(C)nn(C)c2)=O)csc2nc(-c3ccc(F)cc3)cn12 C(=O)(C1=C(C)CCCC1)N1CCCC(NC(CSC)=O)CC1 N1(C(c2cc(C)on2)=O)CCOC2CN(C(c3[nH]c(=N)sc3C(F)(F)F)=O)CC12 C1(CNC(C2CCCN2C(=O)Cc2cnoc2)=O)CC12CCCCC2 CCC(CC)CCCC(=O)NCc1cncc(C(N2CCC(CC(C)C)C2)=O)c1 O=C(C1=CCC(NC(c2csc(F)c2)=O)C1)NCC(F)CO C1(CNC(CCOCC#C)=O)CN(C(=O)Cn2nccn2)CCC1C N1(C(c2c(C)nccn2)=O)CCOC2(CCN(C(c3cc(Br)ccc3F)=O)C2)C1 C1(C)(NC(C2C=CCN(C(C(C(C)(C)C)N(C)C)=O)C2)=O)CCC2(CC1)CC2 N1(C(C2(C(N(C)C)=O)CC2)=O)CC(O)(c2cn(CCCC(=O)O)nn2)C1 c1(NC)cc(C(N2CC(N(C(=O)C(O)C3CCC3)C)C2)=O)cc(Cl)n1 CC(C)C(C(=O)N(CCC(C)NC(=O)Cn1ccnn1)C)n1cccc1 C12(C(=O)NC3C(NC(c4cnc(CC)[nH]4)=O)CCC3)CCC(CC1)C2 c1(C(N2CCOC(CNc3ccnc4ncnn34)C2)=O)cc2cccnn2n1 N1(C(=O)C=Cc2ncc[nH]2)CCC2(CC1)CCN(c1ncc(I)cn1)C2 C1(CNC(CCc2ccn(C)n2)=O)C2CC1N(C(=O)C(C)(C)c1sccc1Cl)C2 C1(CC)CC(OC(C2CCN(C(=O)CN(C)C)CC2)=O)C(=O)O1 c1(C(=O)N)n[nH]c2c1CC(C)CC2.C1(OC)CC(C)N(C(=O)CC)C1.C(C)=O C1(C(N(C2CCSCC2)C)=O)CC(NC(=O)CCC2CC2)CCO1 C1(NC(C=C(CC)CC)=O)CCCC(NC(c2cnn(C)c2-n2cccc2)=O)C1 c1(C(N(CCC(NOCCOC)=O)C)=O)c(C)nc2ncnn2c1C c1(CCC(N2CCN(C(CC)=O)CC2CC(F)F)=O)ccc2c(c1)COCC2 N1(C(C2CCCCN(C(C3CC3C3CCC3)=O)C2)=O)CC2CC(O)CC1C2 C1(C)(CNC(C(C=C)O)=O)CN(C(=O)C(c2ncccc2OC)(F)F)CC1C C(=O)(C(C(C)C)OC)N(C1CCN(C(=O)CC)C1)CC#C.C1(C=O)CCCC1 C1(NC(C2N(C(COCCOCC#C)=O)CCC2C)=O)CCN(C)CC1C C(C1=CCSC1)N(C(C=C(C)CNC(c1cnn(CCF)c1)=O)=O)C c1(C(N(CC(C)NC(c2cc(CC)[nH]n2)=O)CC)=O)cc(O)cc(C)n1 C1(C(N2C(C)(C)C(NC(c3ccsc3)=O)CC2)=O)CC2CC(O)CC(C1)C2 N1(C(C2N(C(C)(C)C)CC2)=O)CCCC(C)C1.C(=O)C(F)(F)F.C(=O)C.C Cc1cc(C(N2CC(CNC(=O)CN3CCN(C)CC3)C2)=O)c(Cl)cn1 CCC(C)N(OC)C(=O)C1=CCN(C(c2snnc2C)=O)C1 C(=O)(N=c1[nH][nH]c2ccccc12)C1C2CN(C(C(C(=O)OC)C)=O)CC1CCC2 Cc1nsc(C(=O)NCC2CCCN(C(C3(CO)CC(C)(C)C3)=O)C2)c1N c1(C(N(CCNC(=O)C(F)C2CC2)CC)=O)ccc2nccn2n1 C1(CNC(C2=C(C)OCC2)=O)Cc2ccccc2CN1C(C1COCCO1)=O c1(C(N(CCC(C)NC(C2(F)CC=CC2)=O)C)=O)ccc(-c2cnn(C)c2)cc1 c1(C(=O)NC2C(C(=O)NCC(C)(C)F)C2)cccc(O)c1O C(=O)(CC1=Cc2ccccc2C1)NC(C)CCNC(=O)COC1CCOC1 c1(CNC2(CC(N3C(c4ccc(C)cc4)CCC3)=O)CCC2)ccc(Cl)c(C)c1 Cc1cc(CCCC(=O)NCC2(CNC(C3CC3(C)Br)=O)CCC2)on1 C(=O)(C(CC(C)CC)NC(c1n[nH]c(O)n1)=O)NC1CCC(CCC)CC1 C1(NC(COCCCOC)=O)CCCCN(C(=O)C=Cc2ccccc2)C1 c1(OC)cc(C(=O)NCC23CC(CN2C(C2C(C)C2C)=O)C3)ccc1F c1(C(N(C2CCCN(C(C3(CF)CCOCC3)=O)C2)CC)=O)cnc2n1CCC2 N1(C(c2cn(CCOCC)nc2)=O)CC(C)(C)CC1C.C1(C=O)C=C1C c1(C(=O)NCC(C)CNC(=O)CCC2CC2(Cl)Cl)ccc(O)c(F)c1 C(CCCCCC(=O)NC1CCC2(CC2)C1)NC(C(C(C)C)NC=O)=O N1(C(C(C)SC)=O)CC(C)CN(C(c2cc3ccccn3n2)=O)C(C)C1 C1(NC(C(C=C)O)=O)CN(C(=O)CCc2cncc(C)c2)CC2CCCC12 C(=O)(CC1=NNC(=O)C1)N1CCCN(CCN(C(=O)Cc2ccno2)C)CC1.C N1(C(C2=CC(C)(CC)C2)=O)CCC(C(=O)NC(C)C=O)CC1(C)C.C(C)C N1(C(CC)=O)CCCC(NC(C2CCC(NC(=O)COCCF)CC2)=O)C1 CC1C(NC(=O)Cn2cncn2)CCN1C(c1csc(C(F)(F)F)c1)=O C(C(C)(C)CNC(c1n[nH]cc1C(F)(F)F)=O)NC(C(C)C1CCC1)=O N1(C(=O)CC2CCCC(O)C2)CCOC2(C1)CN(C(c1ns[nH]c1=O)=O)C2 CCCCCCC(C)CC(=O)N1CCC(NC(=O)C#CC2CCCCO2)C(F)C1 C12(C(=O)N)CC(C1)OC21CCC1.c1(CC)ccc(C(=O)N(CCC)CC)s1 c1(C(=O)NC2CC(CNC(CC3CCCC(OC)C3)=O)C2)cncc(F)c1Cl C1(NC(=O)CCC2CC2)CCCCC1NC(C1CCCCN1c1ccncc1)=O C(C)(C)(C(C)CC(=O)NCCC(O)CO)NC(C(C(C)C)C#N)=O N1(C(c2c(C)nc(C3CCOC3)s2)=O)CCC2(CC1)CN(C(=O)C1=CCOC1)C2 CC(CN=c1[nH]c2c(c(=NC(C)c3cc4cnccc4o3)[nH]1)CCC2)OC(F)F c1(C(N2CC(C)C(CNC(=O)CC(=O)N(C)C)CC2)=O)[nH]nc2c1COC2(C)C c1(C(N2C(CNC(C3(C)CCCO3)=O)CC2)=O)ccc([N+](=O)[O-])nc1 CC(C)CC(O)C(C)C(=O)NC1CCCC(CC(=O)NC2CCN(C3CC3)C2)C1 C1(Cl)(C=O)C2CCC(=O)C12.C1(NC(COCCOC)=O)CCCCC1C Cc1cc(C(=O)NCCCN(CCO)C(c2cnc3n2CCS3)=O)c(C)cn1 N1(C(C2CCOC2c2ccncc2)=O)CCCC1C(O)C(F)(F)F N1(c2n(CCC=C)c(-c3[nH]nc(O)c3Br)nn2)CCCC2(CCSC2)C1 C1(C(=O)NC(C(N2C(C)(CCC)CC2)=O)C2CCCC2)CCC(=O)N(C)C1 c1(C(N2C3CC(C2)C3)=O)cc(=N)[nH]c(=N)[nH]1.c1(N(C)C)cccc(C(=O)N)c1 C(=O)(NN1CCCC1C(=O)NCCC1C=CCC1)c1c(C)nn(C)c1 CC1CN(C(=O)CCCS(C)(=O)=O)CCN(C(c2cn(C)[nH]c2=N)=O)C1 C(C1Cc2ccccc21)NC(CCN(C(C1CC(=C)C1)=O)C)=O C12(C(=O)NCCC3CCCC3O)CCC(n3cc(CCO)nn3)(CC1)C2 C#Cc1ccccc1CC(=O)NCC1(C)CCCN(C(c2conc2C)=O)C1 O=C(CCCC(F)(F)CO)NCC1=NOC2CN(C(=O)CCc3ccco3)CC12 C1(C)(C(N2CC(O)(CNC(c3ccc(C(C)=O)[nH]3)=O)C2)=O)CCCCO1 C1(c2cn(CC(C)NC(C3CC3c3cccc(Br)c3)=O)nn2)CCCC(F)(F)C1 CC(CC1CCC1)C(=O)NC1CC(C)(NC(C2CCN(C3COC3)C2)=O)C1 c1(CNCC2N(C(c3cc(C)on3)=O)CCC2)cc(O)c(Br)cc1O C#CC1CN(C(C2CC=CCN2C(c2cncc(NC)c2)=O)=O)CCO1 N1(C(CC(C)C)=O)CCN(C(C2(O)CCCC2)=O)CC(C)(F)C1 Cc1sc2ccc(F)cc2c1C(=O)NC(CO)C(C)NC(=O)Cc1ccon1 C(=O)(C1=Cc2cccc(Br)c2OC1)N1C(C)C(NC(C2CC23CC3)=O)CC1 N1(C(=O)NCCc2nnc(CO)s2)CCOC2CS(=O)(=O)CC12 C(CN=c1nc2c(c[nH]1)CCCCC2)C1CC(NC(C2CC(C)OC(C)C2)=O)C1 C1(C)(NC(c2c(CC)csc2)=O)CCN(C(c2ccc(C)nc2N)=O)CC1 N1(C(C2(C#C)CCCC2)=O)CCCC(C2CCN(C(=O)C(C)(C)C(=O)NC)C2)C1 C1(C(=O)NCCC(C)NC(c2c(C)onc2)=O)CCC(C)(O)CC1 C1(OC)C(C)(C)CN(N2CCCCCC2CCN2CCCC2)C1(C)C N1(C(c2c(C)csc2)=O)CC(NC(c2cc(C(C)(F)F)on2)=O)CC12CCOC2 CCCC(CO)NC(=O)CCNC(C1CC1(C)CC)=O CC1CNc2c(C(=O)NC(C)CN(C(=O)C3=CCCCO3)C)cnn2C1 c1(C(=O)NCC(CC)(C)NC(=O)Cn2cccn2)ccc(S(C)(=O)=O)[nH]1 C(C(C)(C)CC)NC(C(C)C1CCC1)=O.c1ccccc1C(N)=O.C(=O)(C)N C(=O)(C1=Cc2ccccc2OC1)NCC1N(C(C2OCC(C)C2)=O)CC1 C#CCCCC(C(=O)NCSc1cccc(F)c1)N1CCCC1(C)CC1CCC1 C1(C#N)(C(=O)NC(C2CCN(C(C3COC(=O)N3)=O)CC2)C)CCCC1 c1(C(N2CC=C(CNC(C(=O)NCC)=O)CC2)=O)cc(O)c2ccccc2c1 C1(NC(=O)CCOCC2CCCO2)CCN(C(C2CCCSS2)=O)CCC1CO O(N=C(C)c1cccc(=N)[nH]1)CC(CC)C N1(CC)CCOCC1C(=O)NCc1ccc(C(N2CC(c3nncs3)C2)=O)cc1 C(=O)(CC1=CCCCC1)NC(C)C(C)C(=O)N(C)CC1CCCC1(C)C C1(CCNC(C2CC2c2cccs2)=O)CCCN1C(=O)C=C(Cl)Cl N1(C(CCCCC)=O)CCN(C(c2c(Br)cnn2C)=O)CC1CCOC C1(c2nccc(CN(CC(=O)OCC)C)n2)Cc2ccccc2O1 CCC(C(=O)NCC(C)=CC(N1CC(C)(CO)C1)=O)SC C(=O)(C(C)C(C)NC(c1nocc1Cl)=O)NC(c1n[nH]c(CO)n1)C C(=O)(CCCC(F)(F)F)NC1C(CC)N(C(C2COCCN2C=O)=O)CCC1 n1(CCC=O)nc(C)c([N+](=O)[O-])c1C.N1(C(COCCOC)=O)CCC2CC12 C(=O)(C1=NOC2COCC12)N(C)CCOCCN(C)C(C1(F)CCOC1)=O C1CC2(CCCCN2C(=O)Cc2ccc(F)cc2Cl)C1.CC(C(=O)N)NC(N)=O N1(C(c2c(C)scc2)=O)CCCC(NC(c2cccc(C(F)(F)F)c2Cl)=O)C1C c1(OC)cccc(CC(C)CC(=O)NC2CC3(C2)CC3NC(=O)CCC(C)C)c1 C1(C)(CC)CC(NC(c2sc(O)nc2O)=O)CN1C(=O)C(c1cccnc1)C c1(C(N(CCC(C)NC(c2ccc(O)nn2)=O)C)=O)ccc2c(c1)NCCC2 c1(NC(C(=O)N(C(c2cncn2C)C)CC2CC2)=O)cc(O)nc(O)n1 Cc1cn(-c2ccccc2)[nH]c1=NC(=O)NCC(N)C1CCC1 CCCCCCCCC(=O)N1CC2CC1CCC2NC(=O)CSc1nncn1C c1(C(=O)NCC(CNC(C(C)NC(CC)=O)=O)(C)O)ccc(Cl)c(F)c1N C1(O)(CNC(=O)Cc2nnc(O)s2)CCN(C(=O)CCCn2ccnn2)CC1 N1(C(C2CCC(OC)CC2)=O)CCN(C(=O)CN(CC(C)(C)C)C)C(CO)C1 C1(CNC(c2cc(OC)ncc2)=O)CN(C(C2C3COCC23)=O)CC12CC2 c1(C(Cc2ccccc2)Nc2ccc(SC)cc2)cc2cc(Br)ccc2[nH]1 CC(C)N(O)C(=O)C(=O)N1CCC(O)(CNC(=O)CN2C(=O)CCC2=O)C1 C(=O)(CC(=O)OCCC(C)O)NCCNCC.C(C)(C)C.C(C)(C)C C1(NC(C(C(C)(C)C)OC)=O)CN(C(C2(OC)CCC2)=O)CC(C)(C)C1 N1(C(c2cnc(CC)nc2)=O)CC2(CO)CC1(C(=O)N)C2.C1(C)CCCCO1.C C=C(C)CC(C(=O)NCc1cscn1)NC(=O)CCN(C)CCC CC(C)(C)C(C(F)F)NC(c1cccc(-c2cc[nH]n2)c1)=O Cc1ccc(C(=O)O)c(N2CC(c3cccs3)CC2C)n1 C(=O)(CC(C)C)C1(C(C)C)CC1.C(C(=O)NCC)OCCOCC C1(CNC(C2C(C)(C(C)C)C2)=O)CCCCN1C(=O)CC1CCN(C)C1=O CC1CC(NC(=O)CCC(C)(C)F)CCN1C(=O)C=Cc1cccc(CO)c1 CCCC(O)C(=O)NCC1(O)CN(C(c2cncc(C(C)(C)C)c2)=O)C1 C1(C(=O)NC(CN(CC(N)=O)Cc2cccs2)=O)CCCC1 c1(C(N2CC(C(C)NC(C3OCCN(CC)C3)=O)OCC2)=O)cc(Cl)ccc1C Cc1nn(C)cc1S(=O)(=O)NC1CCN(C(c2ccc(S)cc2)=O)C1 Cc1nc(C(N2CCC(C=CC(N3CCC(CC(F)F)C3)=O)CC2)=O)cc(O)n1 N1(C(C=CC)=O)CCC(CC2CCN(C(C3COC(=O)N3C)=O)CC2)CC1 c1(C(=O)NC2CN(C(C3C(C=C)C3)=O)CC23CC3)cccn2nncc12 C(c1csc2ccccc12)=CC(=O)NCCCNC(C1CC2CCC1C2)=O C1(C(N2CCCC(NC(C34CC(F)(C3)C4)=O)C2)=O)CCC12CCC2 C=C(Br)CC(C)(C)C(=O)NC1CN(C(=O)CCc2ncccn2)CC1F CCS(=O)(=O)CC(=O)N1CC(CNC(c2cc(F)ccc2C(C)C)=O)CC1C N1(c2c(S(=O)(=O)NCC(C)C)cncc2)CCCC(C2CCCC2)C1 c1(C(=O)NC(CC(C)NC(c2ccc(C)s2)=O)C)ccc2nc[nH]c2n1 Cc1cc(C(=O)NC(C(=O)NCc2cc(O)ns2)C(C)C)nnc1O c1(C(=O)NCCNC(C(CCC)=CCC)=O)cc(N)ccc1Br c1(C(=O)NC2C(C)(C)CN(C(=O)C#CC3CC3)C2)ccc([N+](=O)[O-])cn1 C1(O)CCN(C)CC1.Cc1ccc(C(=O)NC2CC(CC(=O)NC)C2(C)C)n1C c1(OC)sc2c(-c3cccc(-c4ncco4)c3)cccc2c1C N1(C(=O)Nc2nc(C3CCC(c4ccccc4)CC3)no2)CCC(O)C12CCC2 c1(C(N2CC(C)(NC(c3cccnc3S)=O)C2)=O)ncc(F)cc1F c1(CC(=O)NC(C2CCN(C(C(C)OC)=O)C2)C)ccc(CO)cc1 c1(OC)cccc(C(=O)NCC23COC(C2)C3)c1.C1(C)(C=O)CC1(Cl)Cl C(=O)(C(C)CS(C)(=O)=O)NCC(C)NC(C1(C#C)CC1)=O C(C(C)(C)C)NC(C1CCC(C=O)C1)=O.c1(C=O)ccon1.C(C)(C)C C12(C(=O)N)CCCC1CCN2C(=O)CN1C(=O)CNC1=O.C1(COC)CC1 C12(C(=O)OC)CN(C(=O)NCCCCn3cc(CC(C)C)nn3)CC1CCO2 N1(c2nnc(C(CC)(C)C)o2)CCC(O)(C(C)NC(C2CC3CCC2O3)=O)CC1 C1(C(=O)NC2CCC(C(N3CCOCC3C3CC3)=O)C2)CC2(CCO1)CC2 C(N=c1nc2sccc2c(NC2CC2F)[nH]1)C1CC(CC)C1 N1(C(C2CC(n3ccnc3)C2)=O)CCC(CNC(C2(CO)CCCO2)=O)CC1 c1(C(=O)NC2C3CN(C(C(C(CC)O)C)=O)CC32)ccc2nc(N(C)C)sc2c1 Cc1cc(NC(c2nnnn2CC(F)F)c2ccns2)cc(CO)n1 C(=O)(CCCS(N)(=O)=O)NCC=CCNC(C(C=C=C)C)=O N1(C(CCC(=C)C)=O)CCC2CN(C(=O)C=Cc3cocn3)CCC2C1 C1CCN(C(=O)C(C)=C(C)C)CCC1(F)F.c1(C(=O)OC)cc(C(=O)N)on1 c1(CN2CCC(C)(C(N(C)Cc3ncon3)=O)C2)c[nH]c2cc(Br)ccc12 CC1OC2(C(=O)NC3CCC(NC(C4CCS(=O)(=O)CC4)=O)CC3)CCC1CC2 Cc1cccc(C2CCCCN2C(=O)CCc2nc(-c3cccs3)no2)c1 C1(C(N2CCC(CNC(c3cc(CCC)[nH]n3)=O)CC2)=O)CCn2nncc2C1 CCC(CNC(C1CN(C(=O)CN(C)C=O)CC1(F)F)=O)(CC)C(N)=O.O C1(CC=C)(NC(=O)C(C)CO)CCN(C(C2(COC)CCCCC2)=O)C1 C1(C2CCCCC2)(C(=O)NC2CCN(C(C(c3ccccc3)C)=O)C(C)C2)CC1 c1(C(C(=O)NCCCC)N(C2CCS(=O)(=O)C2)C)cccc(C(F)(F)F)c1 O=C(C1=CCS(=O)(=O)C1)NCC1CC2CCC1N(C(C1(O)CCCC1)=O)C2 C(=O)(CCS(=O)(=O)C1CCCC1)NCC(C)NC(=O)C=Cc1ccccc1C#N c1(C=O)c[nH]c(=O)c2ccnn12.Cc1cc(CO)oc1C(=O)NCC1CC1.C c1(SC)ncc(C(=O)NCCCC2CC2)s1.C1(C)(CC(=O)N)CC1(F)Cl C1(CC)CCCCN1C(=O)Cc1cc(C)on1.c1(C(=O)N)cncc(N(C)C)n1 C1(C(=O)NCCCNC(C2ON=C(C)C2C)=O)CCc2nnn(C)c2C1 Cc1cc(C(=O)NC2(CC(=O)NCC(C)(C)C3CC3)CCC2)cnn1 c1(COC)cn(C2CCCC2)nn1.CC(C)NCC1CC1F N1(C(C(COC)C)=O)CCCC1(C)CNC(C1CCOC1)=O C12(C(N(CCCCC)CCO)=O)CC3CC1C2C3.C(=O)CCOC.C(C)=O.N C(=O)(C1=C(Cl)CCC1)N1C(C)(CNC(=O)COCCCF)CCC1 N1(C(C2(CCOC)CC2)=O)CCC(O)C(NC(=O)C=CC2CCCC2)C1 Cc1nc(C2CCCN(C(=O)OC(C)(C)C)C2)oc1.c1(C(=O)O)cnc(O)n1C c1(C(=O)NC2CC(C(=O)Nc3ccc(C)c(F)c3)C2)cnc2cc(Cl)ccc2c1 c1(C(N2CC(C(=O)NC3CCC(F)(F)C3)(CC)C2)=O)cccc(=O)n1C c1(C(=O)NC2CCN(C(c3c(C)con3)=O)CC2F)cc2nccn2c(O)n1 c1(C(=O)NC(C)C)ccc(C(=O)NC2CCCC2)cc1.C(=O)C(C)(C)C.C N1(C(C(C)OCCC#C)=O)CC2CCC(C1)N2C(=O)C(C1CC1)SC c1(C(N2C(C)CCC(C(=O)NCCOC)C2)=O)cc2cc(N)ccc2o1 c1(OC)cc(C(=O)NC2CCN(C(C3CC(C)N(C)C3)=O)C2)c(F)c(Cl)c1 Cc1cc(C(=O)NC2CCCC(c3ccc(F)c(F)c3)C2)nc2c(Br)cnn12 c1(CC)cccc(C(N2CC(NC(c3cc(N)ccc3O)=O)C(C)C2)=O)c1F Cc1cc(OC(F)F)c(N)c(NC(=O)CCn2nc(C)nc2C)c1 CN1CCC(NCc2cccc3c2OCC3)C2CCCC12 N1(C(C(Cn2cncn2)NC(c2c(CC)nn(C)c2)=O)=O)CCCCC(C)(F)C1 c1(NC(C2CCN(C(c3c(I)ccnc3Cl)=O)CC2O)=O)cccc(F)c1F C(=O)(C1=C(C)C(C)(C)OC1=O)NCC(CNC(CS(=O)(=O)NC)=O)CO C1(C=O)CC2(CCCC2)C1.c1(C=O)cccc(NS(N)(=O)=O)n1.CCC(C)C.N C1(C(N2CC(OC)C2)=O)CCCCCN1C(=O)Cc1cnsc1 C1(CNC(CCc2c(C)noc2C)=O)CCCN(C(C2(CO)CCCC2)=O)CC1 N1(C(Cc2ccccc2)=O)CCC(O)(C(N)=O)C1.C(C(=O)NCC=O)N(C)C.N c1(C(=O)OC)c(C)oc2[nH]c(=NC3CCCC(C(F)(F)F)C3)ccc12 CCC(CC)CC(=O)N1C(C(=O)Nc2cncc(C(N)=O)c2)CC1C c1(C(N2CCN(C(C(C)C#N)=O)C(CF)C2)=O)c2c(nn1C)CCC2 N1(C(CSc2ccc(C)cc2)=O)CC2CC1CN(C(c1cnc(C)o1)=O)C2 N1(C(C(C)OCC#C)=O)CCCC2(NC(=O)CN(C3CCSC3)C)CC2C1 C1(CC=C)(NC(C2CC2c2cnn(C)c2)=O)CCN(C(c2ccncc2)=O)CC1 C1(CC(=O)N(CCCCCCNC(=O)CCC2CCC2)C)CC(C)(C)CCO1 CC(C)CCC(=O)NC(C(=O)NC1CCC1(C)C)C1CCCC1 C(=O)(C(C)(C)CCC#N)N1C(C)CC(OC)C1.C(=O)(C(C)Cc1ccnn1C)N C=C(C)CC(=O)NCC(CCOC)NC(=O)C(C)C1(O)CCC1 C1(C(=O)NC(C(=O)N(CC=C)CC=C)C2CCC2)CC=CCC1C C(=O)(C1=C(C)OCC1)NCC1CCC(NC(c2ccc(OC)s2)=O)CC1 CC1(C)CC(CO)N(S(=O)(=O)CCCC2CC2)C1 Cc1cc(NC(C2CC2C(=O)Nc2cccc(C(C)O)c2)=O)cnc1Br N1(C(C)(C)C)CCN(C(=O)CCC2(NC(C3CC4CC4C3)=O)CCC2)CC1 c1(C(=O)NC2(c3cn(CC(F)(F)F)nn3)CCC2)cccc(-n2ccnc2O)c1 C(=O)(CC(C)(C)C1CC1)NCCCN(C(=O)C=C1CCSCC1)C(C)C CC1CCC(C(=O)NCC23CC2CN(C(=O)Cc2cccnc2F)C3)CC1 C(c1ccc2c(c1)COCC2)=CC(=O)NC(CC1CCOC1)CO C1(NC(C(C2CCN(C(C3C4CCCCC34)=O)CC2)C)=O)CC2CCCC2C1 c1(C(C(=O)NCC2CCC(NC(C3CSCCS3)=O)C2)=O)cc(F)c(F)cc1F CCCC(C)CC(=O)N1CCC(NC(=O)C(C)c2ccco2)C(CC)C1 c1(C(=O)NC(C)CNC(c2ncn3c2CCCC3)=O)nccc2c(Cl)cccc12 c1(C(=O)NCCC(C)NC(=O)CCc2cnc[nH]2)ccc(C(N)=O)[nH]1 CCC(CN(C)C)CC(=O)N(C(C)C(=O)NCC1=CCN(C)CC1)CC c1(OC)cccc(O)c1C=O.C1(CC=O)CC(C2CC2)C1.C1CC(CC)C1.N N1(C(C2C(CC)OCC2)=O)CC2(CCN(C(C3CCCCN3C(N)=O)=O)CC2)C1 C1(COC)CC(C)N(C(c2csc(O)n2)=O)C1.C1(CC(=O)N)CCOC1=O c1(OC)cccc(C(=O)NCC2(F)CCC2)c1.C1(C=O)ON=C(C)C1C.C C(=O)(C(CC(F)F)c1ccccc1)NC12C(CN(C(CN(C)C3CC3)=O)C1)C2 C1(N(C)C)CCCN1NC(=O)C1N(C(=O)COCC(C)(C)C)CC12CCCC2 c1(C(N(CCCOC(C)C)C)=O)c[nH]nc1C(C)(F)F C(C)(CNC(=O)C(=Cc1cccs1)C)(C)OC.C1(C(=O)N)CNC(=O)C1 C1(C=O)COC(C)(C)CN1C=O.N1(C(COCC)=O)CCCC1.C(C)(C)C CCCCC(O)C(C)C(=O)NC12CC(C(=O)NC3CCc4n[nH]cc4C3)(C1)C2 C1(CNC(Cc2n(C)cnn2)=O)CCCCN1C(=O)CC1CCN(C2COC2)C1 N1(C(C2C(C)=C2)=O)CCC(C2CC2)C1CNC(=O)CC1CC2(CC2)C1 C(=O)(CCC(=O)NCC1(CNC(=O)CC(C)(C)OC)CC1)NCC N1(C(CCc2[nH]c(=N)sc2)=O)CC2CCC1C(NC(C1CCC1C(N)=O)=O)C2 c1(C(=O)NCC(=CC(=O)NCC(CC)N(C)C)C)cc(O)cs1 N1(C(c2coc(CCCCCC3CN(C(C)=O)C3)c2)=O)CCCC1C(=O)OC c1(CC(N2CCC(CNC(C=C(C)C)=O)CC2C)=O)ccc2ccccc2c1 c1(C(=O)NCC(C)(C2CC2)NC(CCC2(C)CC2)=O)ccc(O)c(N)c1 C1(CC)CCN(C(=O)CSC2CC2)C1C.c1(C=O)ccc(C(C)C)[nH]1.N c1(OC)ccc(C=CC(=O)N(C2CN(C(=O)C(O)C(F)F)CC23CC3)C)cc1F c1(C(=O)NC2CCC(NC(c3nc(CC)oc3)=O)C2)ccncc1OC N1(C(COCCCC)=O)CCC(C)C(N(C(=O)Cc2cccc(C)c2F)C)C1 CC(C)C1=CCC(NC(C2(F)CN(C(c3csc(F)c3)=O)C2)=O)CC1 N1(c2cc(NCC3(N(C)C)CCCC3)ncn2)CCC2(CC1)CC(O)CCO2 C1(CNC(=O)CCCc2nccs2)C2CN(C(C3(N4CCCC4)CC3)=O)CC12 c1(C(=O)NC2CC(NC(C3(CC#C)CCCC3)=O)C2)c(C)oc(Br)c1C N1(C(CC(=C)C)=O)CC2CC1(CNC(c1cnn(-c3ccccn3)c1C)=O)C2 C=CC1CN(C(c2n[nH]c3c2COC3)=O)CC1NC(c1nc(C)ccc1C)=O c1(C=O)cn2c(n1)CCCC2.C1(C(N2CC(COC)C2)=O)CC=C(C)CC1.C c1(C(=O)NCC2CN(C(=O)CCCn3cccn3)C2)cc(O)cc(O)n1 C=C1CCN(C(c2cnccc2OC)=O)C(C(=O)NCC(C)(O)C(F)(F)F)C1 C(=O)(CC(C)(C)F)N(C)CC1CCCN1C(=O)C(=O)NCc1cccnc1 C1(C(N(CC(C)C(N2CCC3(CCC3)C2)=O)C)=O)CN2CCN1CC2 C1(OCC)(CNC2(COC)CC2)CCCC1 CON(CC1CC1)C(=O)C(Cn1cncn1)NC(=O)CN1CCCCCC1 C=CC1CN(C(=O)CN(C)C(C)=O)CC1.c1(C=O)cccc(C(C)(F)F)n1.N c1(OC(C(c2ccc(C)o2)C)=O)cccc2c1C(=O)c1ccccc1C2 C(=O)C1=CCC(C)(C)CC1.N1(C(CC(=O)NCC#C)=O)CC2CCC2(C)C1.N c1(C(N2C(CCNC(c3c(C)ccs3)=O)COCC2)=O)cccc(S(N)(=O)=O)c1 n1(C(C)C)nccc1C(=O)NC1CCCC1NC(=O)C=CC=O.C1CC1 C1(C(=O)NC(COC)CNC(=O)C(C2CC2)SC)C(C)C1(F)F C(=O)(CCCC(C)(C)C#N)N(C(C(N1CCC2(CCCCC2)C1)=O)C1CC1)C CS(=O)(=O)c1cnn(CC(O)CNC(c2ccc(Br)cn2)=O)c1 CN1C(=O)CSC1=CC(=O)NC1C=CCN(C(=O)CC2CCCC(=O)N2)C1 C(=O)(C1CCCn2cnnc21)NCC(COC)NC(c1cc(C#N)ccc1F)=O c1(CC(=O)N(CC(C)NC(=O)C)CC)csc2sc(C)cc12.CC(C)C.O C12(C(=O)NC3(C)CCSC3)CC(CN(C(=O)Cc3ccc(F)nc3)C1)C2 C1(CC=O)CC2(C1)CN(C(=O)CN1CC3CCC1C3)C2.n1(CC)cccn1.C Cc1cnc(NCC2COCCN2C(=O)CCc2cccc(Br)c2)nc1 CC1=CCN(CCNC(=O)CC2CC(NC(=O)CCC3CCCOC3)C2)CC1 C(C(C)N=c1[nH]nc(CO)s1)(c1ccccc1)NC(C(CCCC)C)=O O(NC(=O)CCN(C)C(c1cc(C)n(C)c1)=O)C(C(=O)OC)(C)C C1(C(N2CC(N(C(COCCC)=O)C)C(C)(C)C2)=O)CC(C2CCCC2)C1 N1(C(C(=O)Cc2ccsc2)=O)CC2CC(NC(=O)CC(F)(F)F)C2C1 N1(C(CCCCC)=O)CCCC(NC(=O)Cc2cnc(C3CC3)[nH]2)C1C O=C1NCC2C1CCCN2C(=O)CCCn1cc(C2CC3CCC2CC3)nn1 C1(C=O)CC2CCC(C1)C2=O.C1(OC)(C)CCN(C(=O)C(C)=C2CCCC2)C1 C1(NC(CCNC(CC(C)C)=O)=O)CC(NC(c2ccn(C)c2)=O)C12CCC2 c1(C(N2C3CC(CNC(C4(C)CC4(Cl)Cl)=O)C2CC3)=O)ccc2c(c1)CCO2 C1(C(N(CCN(C)Cc2nnc(C3CC3)n2C2CC2)C)=O)CCCC12CC2 c1(NC(C)=O)cccc(C(N2CC3CC(C(=O)O)C3C2)=O)c1C C1CC(F)(CNC(C2(C(=O)OC)CCCO2)=O)C1.C1(=O)CC1.C1CC1 c1(OC)coc(C(=O)NC2CN(C(=O)Cc3nnc(O)s3)CCC2CO)cc1=O C(=O)(CCCCCCn1cc(-c2cnccn2)nn1)NC(C1CCC(=O)C1C)C C(Cn1cncn1)(C(=O)NCc1ncco1)NC(=O)CC1CCCCO1 CCCCCCCCCCC(=O)N1CC(NC(c2cc(F)ncc2Br)=O)C(C)C1 C(=O)(C(C)CNC(=O)CCCN1CCCC1)NC(C1CCOC1)C#C C(=O)(C(C)CC(C)C(C)=O)NCC(CN(C(c1ccc(C)c(F)c1)=O)C)O C(=O)(C1=Cc2ccccc2OC1)NC1CC(C)(C)N(C(c2cnnc(O)c2)=O)C1 C(=O)C(C)(C)S(C)(=O)=O.C1(CC)OCCCC1C(=O)NC(C)(CC)CC.N N1(C(C(C)CC2CC2)=O)CCC(CO)(CNC(=O)C=CC2CCCC2)CC1 C1(CNC(CNC(N)=O)=O)(CNC(c2cnccn2)=O)CC2CCCC2C1 C(=O)(C(F)CC(C)(C)C)NCc1cn(CC(=O)Nc2c(C)ccnc2)nn1 CS(=O)(=O)c1ccc(C(=O)NCC2CC(O)CN2C(=O)Cc2csnn2)[nH]1 S(=O)(=O)(c1nc(N2CCC(F)(CO)C2)ccc1Br)NCCCS(CC)(=O)=O CN1C(=O)CCC12CCN(C(=O)COCc1ccc3c(c1)OCO3)CC2 C1(CC(=O)NCCNC(CC2C(C)C2(F)F)=O)CCCC12CC2 C#CCCCC(C)C(=O)N1CCC2(CC(C(N3CCCC(C(C)C)CC3)=O)C2)C1 C1(NC(=O)CC2C=CCC2)CCCC12CCN(C(c1cnsn1)=O)CC2 c1(C(N2CC(CN(C)C(C3C4CCCC34)=O)C2)=O)ccc2n[nH]cc2c1 N1(C(COCc2n(C)c(S)nn2)=O)CCCN(C(c2ccnn2C2CC2)=O)CC1 c1(NC(C2(O)CCN(c3ncc(CCC)cn3)C2)=O)cccn2nc(C)nc12 c1(C(=O)NC2(C)CCN(C(C3(CCC)CCC3)=O)C2)ccc(F)c2ccoc12 n1(CC(=O)NCc2cc(C)on2)cc(C#CC(C)(C)NC(=O)CCC=O)nn1 CCCCC(CNC(c1cc(Br)sc1C)=O)NC(c1ccncc1)=O C(=O)(C#CC1CCOC1)NC1CCC(Cn2cc(-c3cccc(CC)c3)nn2)C1 C1(CC(=O)NCCCSC)CCN(C(=O)Cc2nc(C)cs2)C1 c1(C(=O)N)ccccc1.C(=O)(CC(=O)N1CCC1C)NCC#C.C(=O)CC C1(NC(c2c(C)c(C3CC3)[nH]n2)=O)CCN(C(C2SCCS2)=O)C(C2CC2)C1 CCCC(CNC(=O)CCC1CC1)C(=O)NCc1cc(Cl)no1 c1(C(=O)NC2CC(F)(CNC(C(CCC)(C)C)=O)C2)ccc(C)cc1[N+](=O)[O-] Cc1cccnc1C(=O)NCC(C1CCOC1)NC(=O)CCc1ccccc1O Cc1c(C(=O)NCC(O)CNC(=O)CC2CC3CC3C2)sc2nnc(S)n12 Cc1cc(C)c(CNC(=O)CC2(O)CCC2)s1.C1(CC=O)CCCCN1C.N C(=O)(C1=CC(O)CCC1)NCCC1(O)CN(C(C(CC)(F)F)=O)C1 C=CCC(COC(c1cncc(COC)c1)=O)CC(C)C CCCCCCCCCC(C)CC(C(=O)NC1CC1)N1CCSC2CCCCC12 N1(C(c2nc(C3CC3)cs2)C(=O)NCCOC)CCC2(CC(=O)NC2=O)C1 N1(C(C(c2c(F)cccc2F)C)=O)CCC(C)C(N(C(=O)CC2OCCO2)C)C1 c1(C(N2CCC(C(C)NC(CCC(C)SC)=O)CC2)=O)c(C)nc(C)nc1C C1(C(N(CCOC)CC)=O)CCC(=O)C(C)C1.c1(CC=O)cccc(C)c1 C1(CN)CCN(C(=O)Cn2ncc3c(N)ncnc23)CC1C1CC1 c1ccc(O)c(=O)cc1.N1(C(C(C)NC(C)=O)=O)CCC(C)(C)C1CC(=O)N Cc1ccc(C(F)C(=O)NCC2CC2C)cc1.n1(CC=O)ccccc1=O.N Cc1ccc(C(=O)NC2CCCC(C(=O)Nc3ncc(C)cc3Cl)C2)c(C)c1 c1(C(=O)NC2CCC(N(C(CCN(C)CC)=O)C)C2)ccc(Cl)cc1O C1(F)(CNC(=O)CC2CCCSC2)CCN(C(=O)CC2(O)CCCOC2)CC1 CCCCC(CNC(=O)C=CC1CCCO1)NC(c1cc(C)sc1C)=O N1(C(c2cc(C)oc2)=O)CCC2CN(C(=O)CCC3(C)CCC(=O)N3)CC12 C(=O)(CCCCSC)NC1(CNC(CCc2onc(CC)n2)=O)CCOC1 CC1CCC(CC(=O)NC(C(=O)Nc2cncnc2O)C2CCC2)OC1 c1(C(=O)NC(C(C(C)C)C)CNC(=O)CCF)cnc2occc2c1 c1(SC(C)C(N2CCC(NC(=O)CN3CC=CC3)C2)=O)nncn1C CCCCC(CN=c1ccnc(C2CCCC2)[nH]1)NC(C1OCCC1CC)=O c1(C(=O)NCc2c(CNC(c3cnn(C)n3)=O)cccc2)csc2c1CCCC2 c1(C(N(CC(C)N(C(C(C)NS(CCC)(=O)=O)=O)C)C)=O)ccccc1C.C C1(NC(COC(CC)C)=O)CC2CCC1N(C(c1nc(OCC)ccc1Cl)=O)C2 C1(NC(CCC2CCN(C)CC2)=O)CCN(C(C2(C)CC2)=O)CC1F CC1CN(C(=O)CCNS(C)(=O)=O)C(C)CN1C(c1cccc(Cl)c1)=O C1(N(C(CNC(CCC)=O)=O)C)CCN(C(=O)CCOCC(F)(F)F)C1 C1(CC(=O)NC(CNC(C2(C#N)CCCC2)=O)CO)CC2(CCC2)CO1 CCC(C)C(=O)NC1(CCC(=O)N(C2CCN(C)C2)C)CCC1 C(=O)(CCCC(F)(F)F)N1C(CNC(c2cc(F)cc(Br)c2)=O)COCC1 CCC(C(=O)N1CC(CNC(=O)CO)C1)Sc1ccccc1.C1CCC1(F)F CC1=NOC(CC(=O)NCCN(C(=O)C(C)Sc2ccccn2)C)C1 C(=O)(CC(O)C(C)C)N1CC(CC)(NC(c2occc2)=O)C1.N1(C)CCOCC1 C#Cc1cnn(C)c1C(=O)NC(C)CN(C(=O)CC1CCOC1=O)C C1(C(=O)NCC2CN(C(C3(CC#C)CCC3)=O)C2)C2CS(=O)(=O)CC12 CC(C)CC(C)OCCC(=O)NCC(c1ccccc1)C.C(=O)(C=C1CC1)N c1(C(=O)NCCC(C)NC(=O)C(F)C(C)(C)O)cc2cc(Cl)ccn2n1 N1(C(c2c(C)ncs2)=O)CCCCC1CCCNC(c1cc(=O)cc[nH]1)=O Cn1nc(C(N2CCC(C(=O)NC3COC(C(F)F)C3)C(O)C2)=O)cc1C#N Cc1nc(NC(C)C(C)C)cc(C(C)C)n1.C(=O)(C1=NNC(C(F)(F)F)C1)N c1(C(=O)NC(C)CCNC(C2CCCN2C=O)=O)c[nH]c2c(F)cccc12 C(=O)(CC(C)(C)C)N(CC(C)C)C.C(CC(=O)N)NC(C)=O.C(C)(C)C c1(C(=O)NC2CN(C(Cn3c(C)nnn3)=O)C3C2C3)ccc([N+](=O)[O-])cc1 c1(CC)ccc(C)c(NC(C2C=CCN(C(c3ccc(CF)cc3)=O)C2)=O)c1 N1(C(c2cn(C)c(C(=O)O)n2)=O)CCC(O)(c2cn(C3CCOCC3)nn2)CC1 C1(C(=O)NCC2CN(CC(C3CCCC3)OC)C2)Oc2ccccc2OC1C N1(C(C(C)Cc2ccnn2C)=O)C2CCC1C(CNC(=O)C1=CCCOC1)C2 N1(C(c2c(O)ncc(CC)c2)=O)C(C)CC2COCC12.c1(C(=O)N)cnn(C)c1 CCC(C(=O)NC(C)CN1CCN(C(=O)CCn2nc(C)cc2C)CC1)C(C)C CC(C)CCCC(=O)N1CCCC1CCNC(=O)Cc1cnccn1 C1(CCC)CN(C(=O)C(COC)COC)CCN1C(=O)CC1(CO)CC1 N1(C(c2c(C)nccc2)=O)CC(NC(=O)Cc2cncs2)CC2(CCOCC2)C1 CN=S(C)(=O)c1ccc(C(=O)NCC2COCC2NC(=O)CCCN=[N+]=[N-])cc1 C1(NC(CCCCNC(c2cnc(C(C)C)o2)=O)=O)CN(C)C(=O)C12CC2 C1(N(C(C(C)OCCCC)=O)C)CCCC1(C)NC(=O)C(CC)OC C(C1CN(C(=O)C(C)C(C)O)Cc2ccccc21)NC(CCCCC)=O c1(C(N(C)CC2CCSC2)=O)coc2c1CN(C(C1(N(C)C)CCCOC1)=O)C2 C(=O)(CCCC(CC)CC)NC(C(=O)NC1(C#C)CCCOC1)(C)CSC CCC(C)(CC)C(=O)NCc1ncoc1CCNC(=O)C(CC(C)C)OC N(C1CCCc2ncccc21)C(C(=O)NCC(c1cccc(Cl)c1)SC)=O N1(C(CN(C(c2nc(C)oc2)=O)C)=O)C2C=CC(C2)C1CO C1(NC(C(C)O)=O)CC2(C1)CC(CNC(c1cn(CCCF)nn1)=O)C2 C(=O)(C(C)CCCC(C)C)NC(CC)CCC(=O)NCC1CCC(C)(C)O1 Cc1sc(C(=O)NC2(C3CN(C(=O)C(C4CCOCC4)F)C3)CC2)c(C)c1C C1(CC(=O)NC2(C)CN(C(C3CC(C)(CC)C3)=O)C2)CCC(F)(F)C1 C=CC(C)(O)CC(=O)NC(C1CCN(C(=O)C(CCC)NC(N)=O)CC1)C c1(NC2C(C)C2)nc2ccccc2c(=NCCc2csc(N(C)C)n2)[nH]1 c1(C(N2CC(NC(C3(CC)CCC3)=O)C3C2C3)=O)cc(Cl)cc(F)c1N Cc1ccc(C(=O)NCCCC(CO)NC(C2CC=CC2)=O)c(F)c1 C12(NC(=O)C(CC(F)F)c3ccc(F)cc3)CC3CC(C1)CC(C(F)(F)F)(C3)C2 n1(CCC=C)cc(C(=O)N(CC(C)N(C)C(c2cscc2C2CC2)=O)C)nn1 N1(C(c2ccc(NCc3ccc(Cl)s3)cn2)=O)CCC(O)(CO)CC1 C1(C(N(CC(CC)(C)OC)C)=O)CCC(C)(C)N(C(=O)Cc2cn[nH]c2)C1 c1(CC(N2CCC(NC(C=C(C)C)=O)C2C)=O)cccc([N+](=O)[O-])c1C C1(C(N(CC(C)N(C(=O)Cc2cccs2)C)C)=O)CCC12CCOCC2 N1(C(COCCC)=O)CCCC(CO)CC1.C(=O)(CS(=O)(=O)Cc1cccs1)N c1(C(=O)NCC2(C)CCC(NC(=O)C#CC3CC3)C2)ccc(F)c(F)c1F c1(C(=O)NCC(COC)NC(c2cnn(C(F)F)c2)=O)cc(CO)[nH]n1 Cn1[nH]nnc1=NC1CCC(NC(c2cc(Cl)ccn2)=O)c2ccccc21 C1(COC)CCCC(c2nnnn2CCCC2CC2)(NCCCC2CC2)C1 CCCCCCC(C)CC(=O)N1CCC(n2cc(-c3cncnc3)nn2)C1 C(=O)C1SCCc2sccc21.c1(OC)cc(C(=O)NCC2(C)CC2)cc(F)n1 Cc1cccc2oc(CNC(c3ccc(Cl)c4c3OCC4)=O)nc12 CCC(C(=O)N)C(C)(F)F.c1(C(n2cc(C3(O)CCCCC3)nn2)=O)cccc(F)c1 c1(CCNC(C(CP(C)(C)=O)N)=O)cc(F)cc2c1OCOC2 Cc1cc(N)c(C(N2CC3CN(C(C4(C)CC(C)C4)=O)CC3C2)=O)cc1F Cc1cc(C)on1.N1(C(C)=O)CCC(N(C)C(c2ccoc2C(F)(F)F)=O)C1.O N1(C(C(CC=C)(F)F)=O)CC(C(=O)N(C)CC2CC(F)(F)C2)CCC1(C)C N1(C(c2cnoc2)=O)CC(S(C)(=N)=O)C1.C=C1CC(C=O)(COC)C1 N1(C(CC2NC(=O)OC2)=O)CCC2(C1)CN(C(c1ncc[nH]1)=O)CCO2 C(=O)(CN=S(C)(C)=O)N1CCN(C(CNC(CC(C)c2cccnc2)=O)=O)CC1 N1(C(CCCC(=C)C)=O)CC2ON=C(CNC(=O)CCC(=O)NC)C2C1 C(=O)(CC(C)(C)CC(=O)N1C2CCC1CC(CNC(C1(F)CC1C)=O)C2)OC C=CCC(CC=C)C(=O)NC12CCC(CC1)N(C(c1cn(CCOC)nn1)=O)C2 c1(CCC)cccc(C(=O)NC2CC23CC(NC(=O)C=C(Cl)Cl)C3)c1 C1(c2nnc(C)o2)CCCN(C(c2ccc(Br)nc2)C(=O)NCC2CC2)C1 C(C1c2ccsc2CCN1C(C1CC1C(F)F)=O)NC(c1c(C)cn(C)c1)=O CC1CN(C(=O)C(F)C2CCOC2)CCN1C(c1ncsc1C1CC1)=O C1(CNC(c2c(NC)nccc2)=O)CC2CCC1N2C(=O)C(C)=C(C)C C(=O)(C(C)(Cc1ccccc1F)NC(=O)C(N)Cc1cc(Br)sc1Br)OC c1(C(=O)NC(CCN(C(=O)CC2CCCOCC2)C)(C)C)cccc2occc12 c1(C(=O)NCC2(NC(=O)C=CCF)CC3CCC2C3)cccc2nccn12 C(CCCCCN(C(=O)CSc1cn[nH]c1)C)NC(C(F)=C(C)C)=O CCCCCC(C)CC(=O)NCc1occc1C(N1CCOC(CO)C1)=O N1(C(COc2c(CC)cccc2)=O)CCC(CC)CC1.C1(C=O)CCS1(=O)=O.N C(=O)(CC(=O)NC(Cc1cnc[nH]1)C(=O)NCCC(C)C)OC C1CCN(C(=O)C(C)(C)C(F)c2ccccc2)CCC1(F)F.CC(C)(C)OC(=O)N C(=O)(CC(C)(C(F)F)N(C)C)NCC(CC)NC(=O)CCC(=O)c1ccncc1 Cn1ccc(C(=O)NCC2CN(C(c3cnc(F)cn3)=O)CCO2)cc1=O c1(OC)ccc(C(N2CCC(C)C(N(C(=O)CCCF)C)C2)=O)c(OC)c1C c1(-c2cn(C3CN(C(c4c(OC)scc4)=O)C3)nn2)ccc(OC(F)(F)F)cn1 N1(C(c2c(C)c[nH]n2)=O)CCCC(CNC(=O)CC2CCNC2=O)CC1 Cc1c(C(N2CCOC(Cc3cn(CCN4CCCC4)nn3)C2)=O)nnn1C C1(NC(c2c(Cl)cn(C)n2)=O)CN(C(=O)CC(=O)NC2CC2)CC1C1CC1 C1(CC(=O)NCCCC(=O)OC)CCCN(C(=O)C(F)C2CCCC2)C1 N1(Cc2c(C)con2)CCCC(CNC(C2CC3(CCC3)C2)=O)C1 N1(C(CC(C)=C(C)C)=O)CCN(C(C2CCCCCN2C)=O)CC1CC(F)F c1(CNc2ccc(OCC)nc2C)oc2ccccc2c1OC Cc1cc(C(=O)NCC2CN(C(=O)C)C2)nc(C)c1.c1ccccc1C(C)C c1(C(=O)NC(CNC(c2ccc(C)n2C)=O)C)ccc(S(C)(=O)=O)cc1N c1c[n+]([O-])ccc1[N+](=O)[O-].CCC(CC)C(=O)NCC(=O)NC(CN)C(C)(C)C C1(C(N2CCC(c3ccccc3)C2C)C(=O)NCC=C)CC2(CCOCC2)C1 c1(C(N2C(CCNC(C(CC)N(C)C)=O)CC(OC)C2)=O)cc(C)ccc1C Cc1nc(NC2CN(C(=O)CCCN3C(=O)CCC3=O)CC2(C)C)c(C)c(O)n1 c1(C(C)O)cn(C2CCN(CC(C)(C)NC(=O)OC(C)(C)C)C2)nn1 C(CC(O)CC(=O)N1CCC(OCCCNC(C2(C)CC=CCO2)=O)CC1)SC Cc1ccc2c(=NCC3C(C)(C)C3(C)C)[nH]c(=NCCCn3cccn3)[nH]c2c1 N1(C(CNC(CC)=O)=O)CCCC2(C1)CN(C(C1CNC(=O)N1)=O)CCO2 N1(C(C2(COC)CC(=C)C2)=O)CCC2CCCC(C1)N2C(C1SCCS1)=O C1(NC(Cc2cnc(C)o2)=O)CCCCC1CNC(=O)CCCc1cccs1 C1CCC12CCC2.c1(OCC)nc(C(=O)N)co1.c1(C=O)cnc(C(C)C)s1 CC1CC(C(N2CCN(CCNC(=O)CC3CC(=O)NC3=O)CC2)=O)C(C)O1 c1(OC)ccc(Cl)c(C(N2CC(CC(=O)NCc3cccc(C)n3)C2)=O)c1F N1(C(C2(CC#C)CCOCC2)=O)CCC(C)N(C(=O)Cc2cccc(C)c2)CC1 C1(C(N(CCCCCO)C(C)C)=O)CC12CCN(C(c1c(F)cccc1I)=O)C2 C(C)(C)(CC(F)C(=O)NCC(C)(C)C1CCCC1)NC(C(n1ccc(C)n1)C)=O C(=O)(CCC(C)(C)[N+](=O)[O-])N1CC(C)N(C(c2cc3cc(Cl)sc3[nH]2)=O)CC1 C(=O)(C1=CCCCC1C)NC(CNC(CCCOCCC)=O)C(C)(C)C CC1CN(C(=O)CCC(F)(F)F)CCC1NC(=O)CN(C)C(c1cccs1)=O C#Cc1ccc(C(N2CCC(C3CCCN3C(=O)CC3(O)CC3)CC2)=O)c(C)c1 C1(NC(C(CCC)(C)O)=O)CCN(C(c2cc(C)nn2C)=O)CCC1CO C1(C(N2CCC(NC(C=C3CCC(C)C3)=O)(C)C2)=O)CCS(=O)(=O)C1(C)C c1(C(N(C(CCNC(c2scc(OC)c2)=O)C)C)=O)cnc(C(=O)O)nc1 C1(C(=O)NCCC2CCCN(C(CCCOCC=C)=O)C2)CCCC(F)(F)C1 c1(C(N2CCN(C(CCCC=C)=O)C3C2C3)=O)cnn2c(C)cc(C)nc12 N1(C(C(C)(C)N(C)C)=O)CCN2CCN(C(=O)Cc3cncn3C3CC3)CC2C1 Cc1ccc(C(=O)NC2CC3CCC(C2)N3C(c2cc(Br)n[nH]2)=O)c2c1CCC2 C1(C)(CC(=O)NCc2onc(CC)n2)CCN(C(=O)Cc2ccsc2C)C1 c1(CC(=O)N)csc2nccn12.CC(C)CCC.C1(C=O)(C(=O)N(C)C)CC1 Nc1cncc(-c2cn(CCCC(N3CCC4CC34CO)=O)nn2)n1 Cc1cn2cc(NC(C3CN(Cc4nc5ccccc5o4)CCS3)=O)ccc2n1 C1(OC)C(c2nc(C3CCC(OC(F)F)CC3)no2)COC12CCC2 c1(OC)ccc(Cl)c(F)c1C(=O)NCCN(C(c1ccncc1)=O)C1CC1 c1(C(N2CCC(CNC(CCCC(C)=O)=O)CC2)=O)cc(F)c(F)c(C#N)c1F c1(C(=O)NC(CCC=C)C(=O)NC2CCN(CC)C2)cccc(C)c1C#N c1(C(N2CCC(NC(C=C(COC)C)=O)C2)=O)ccc(OC)c(Br)c1N Cc1cccc(CC(N2CC(NC(C3CC(F)C3)=O)C(c3nccn3C)C2)=O)c1 C(C(=O)N1CC(c2ccc(Br)cc2)CC1C)(C(C)C)Nc1c(C(C)=O)ccs1 C1(NC(C2CCN(C)C2=O)=O)CC2CCC(C1)N2C(c1cccc2ccsc12)=O c1(C(N2C(CNC(c3nn(C)c(=O)cc3)=O)C=CC2)=O)cnc2c(n1)CCCC2 C1(CNC(C=C(CCC)C)=O)CC(C)CO1.c1(C(=O)N)cnnn1C(C)C c1(C(C)=O)c(Cl)c(Cl)cc(Cl)c1Cl.c12nccn1C1CCN(C1)CC2 c1(C(C)(C)C)[nH]cnc1C(=O)NCC1(F)CC(NC(c2n[nH]cc2Br)=O)C1 C1(CNC(C(CC)(C)O)=O)CCCN(C(c2ncn(C(C)(C)C)n2)=O)CC1 c1(C(=O)NC(CCC(=O)OC)C(C)C)ccc2c(c1)OC(C(=O)O)C(=O)N2 N1(C(C2CC(=O)N2)=O)CC(C(=O)NCc2cc(Br)ncc2F)CC(F)C1 N1(C(C2(OC(C)C)CCC2)=O)CCC2CC2C1.c1(C=O)cc(C(F)(F)F)ns1 N1(C(c2cc(CC)on2)=O)CC(NC(c2csnn2)=O)CC1(C)C c1(C(=O)NC2(CF)CCN(C(c3ccc(O)cc3)=O)C2)ccc([N+](=O)[O-])[nH]1 c1(OC)cc(Cl)c(C(N2CCC(NC(C3CCCN(C)C3)=O)C2)=O)cn1 C1(NC(c2c(C)n(C(C)C)cc2)=O)CC2CCC1CN2C(=O)CC1CC(F)C1 C(=O)(C(C)CN(C)C(C1CCN(C)C1)=O)N(CC#C)CC1CCCO1 c1(C(CNC(=O)CSC)NC(C(C2CCC2)OCC)=O)ccccc1 C1(CC(C)NC(C2CN(C)C2)=O)CC2CCC(C1)N2C(=O)CC1CCSCC1 N1(C(C(CC(N)=O)O)=O)CCC(CCNC(=O)Cn2cncn2)C(F)(F)C1 c1cccc(F)c1F.C1(NC(=O)NCCC2C(C)(C)C2)CCS(=O)(=O)C1.C c1(OC)cc(C(C(=O)NC2CCOC2)N(C)Cc2ccccc2C)c(F)cc1Br c1(NC(C(CC)N(CC)CC2CC2)=O)cccc(OC)c1 C1(NC(C2C=CCN2C(=O)CN2CCC(F)CC2)=O)Cc2ccccc2C1 N(C1CCCc2c(Br)cc(Br)cc21)NCC(c1ccccc1)(C)F N1(C(C2(NC(C)=O)CCC2)=O)CC(C)C(O)C1.C(=O)(C(C)=C(C)C)N Cc1cnc(C)c(C(N2CCC2CC(=O)NOCC2CCC2)=O)n1 c1(CC(=O)N)ccc(F)cc1Cl.c1(SC)ncc(C(=O)NCC2CCCC2)[nH]1 C1(C(=O)NCCCCCNC(C(C=C=C)C)=O)CCC(=O)N(c2cnn(C)c2)C1 c1(C(C)C)ccc(CCC(=O)NCCCCN(C(=O)Cc2cnnn2C)C)cc1 N1(Cc2c(C)nc(C)[nH]2)CC2(C1)OCc1cc(-c3ccncc3)ccc12 N1(C(CCOCC)=O)CCC(O)(CN(C)C(C2(C)CNC(=O)C2)=O)C1 C1(NC(C(C(C)(C)C)SC)=O)CC2(CCCCN2C(=O)C(C)C(C)(F)F)C1 c1(C(C)C)ncc(C(=O)NCC2COCC2NC(=O)CC2CC(F)C2)o1 C(=O)(C1=NNC(=O)CC1)N(C)CC1CN2CCC1CC2 C1CN(C(C23CC(CCO2)C3)=O)CC1C.C(=O)(C=CC(=O)N)OCC.C C(=O)(C1=CC2(CCOCC2)C1)NCC(C)NC(=O)C(c1cccc(Cl)c1)(C)C CCCC(CCNC(=O)C(C1(O)CN(C(C2CC(=O)C2)=O)C1)F)C1CC1 c1(CC)cc(C(N2CCN(C(c3coc(C4CC4)c3)=O)C(C)C2)=O)ccc1C Cc1cc(Br)cc(C(N2CC3CCN(C(C4CC4C)=O)CC23)=O)c1C C(CCC(=O)NC1CCC1CNC(C1CC(C)(F)C1)=O)=CC(C)C c1(C(=O)NCC23CC(CO2)N(C(=O)Cc2cnsc2)C3)cc2ncccn2n1 n1(CC(=O)NCCC2N(C(C3C(=C)C3)=O)CCC2)c(C)cc2ccccc12 O=C(CCC(CF)CF)N1CCC(C(F)C(N2CCC(OC3CC3)C2)=O)C1 N1(C(C(CCC)OC)=O)CCC(C)(C)C1C(N1CCC(N(C)C)C(C)C1)=O CCC(Cc1cccc(C)c1)C(=O)NCCCC(C)NC(C1(CC)CCCC1)=O C(=O)(CC(C)CC(C)(C)C)NCC(CC)(C)C(=O)N1CCN(CC(C)C)CC1 C1(CNC(c2nc(C(=O)OC)sc2)=O)CCCCC1.C(=O)CCc1cnoc1 C1(C(C)C)CC(N2CCCC2)CN1C(=O)Cc1nc(Cl)sc1Cl N1(C(c2cc(C(C)(C)C)no2)=O)CCC(CC)CC1.C1(CC(=O)N)CCC(O)C1 c1(C(=O)NC2CCN(Cc3ncsc3Br)C2)occ2c1CCC2 CCC1=NOC(C(N2CC(O)CC2CC(=O)NCC(C)OCCO)=O)C1 CC1(C)CN(C(=O)CN2CCN(C(C3CC3(C)C)=O)CC2)CC1O c1(OC)ccc(CCNC(=O)NCCc2ccc(F)c(F)c2C)c2ccccc12 CC(C(=O)NC1CCN(C(c2cn(-c3ccn(C)n3)cn2)=O)CC1)C(C)(C)C C(CC(C)CC)(C(=O)N=c1cc2n([nH]1)CCCC2)NC(C(CCCCC)F)=O Cc1ccc(C2CC2)c(C(=O)NCCC(C)NC(C2(C)CC=CCC2)=O)c1 c1(CNC(=O)NCC2CC3(CC3)C2)cc2c(cn1)OCCO2 N1(C(c2n(CC)ccc2)=O)CCC2(CCCC2NC(=O)C(C)CF)CC1 N1(C(c2n(CC)ccc2)=O)CCOC(C(=O)NCC2CCSCC2)CC1 Cc1ccc(C)c(CC(N2CCCC(N(CCO)CC3CCC3)C2)=O)c1 CCCS(=O)(=O)CC(=O)NC1(C)CN(C(c2ccc(-n3nnnc3O)cc2)=O)C1 N1(C(CCC(=O)NCC)=O)CC2(CC(C(=O)N(C)CCC3CCCC3)CO2)C1 N1(C(C2CC(C#N)C2)=O)CC2CCCN(C(C3CC3(Cl)Cl)=O)C2C1 c1(CSC)ccc(C(C(=O)NC2CCCCC2)N(C2CCNC2=O)C)cc1 c1(C(=O)NC2CCN(C(C(c3ccn(C)n3)C)=O)CC2O)nccn2cnnc12 C1(NC(C2C(=C)C2)=O)COCCN(C(C2(O)CCSCC2)=O)C1 C1(NC(Cc2n(C)nnc2)=O)CCCCCC1NC(=O)COc1ccsc1 Cc1cnc(N2CCCC2C2(NC(=O)CN3CCC(C)CC3)CC2)nc1N(C)C C1(NC(C2CC(SC)C2)=O)CCN(C(c2cnc(N(C)C)s2)=O)CC1F CC(C)CC(CNC(C1CCCC(O)C1)=O)C(=O)N(C(C)C)CC1CCCO1 C(C1=CCN(C(c2cc(CC)[nH]n2)=O)CC1)NC(C(CC)=CC)=O N1(C(C(CC)(F)F)=O)CCC(C)C(NC(=O)C(=Cc2cccnc2)C)C1 c1(C(=O)NCC(CCNC(c2cncc(OC)c2)=O)O)cc2cccc(F)c2o1 C1(C(=O)N)CC2CCC(C1)N2C(=O)CN1CC(C)(C)C1.Cc1csc(CC)n1 c1(C(=O)NC(c2cccc(OCC)c2)C)cc(C)c(OC)c(Cl)c1 N1(C(C2C(CC)N(C(=O)CCP(C)(C)=O)CCC2)=O)CCC(C)C(C)(C)C1 C(=O)(CCCC(=O)N1CCN(C)C(CNC(C2CC(CC)C2)=O)C1)NCC C1(CC(=O)NC2CC(n3cc(COC)nn3)C2)CSC2CCCC12 C1(C(=O)NC2CCC(C(=O)NCCc3n(C)cnc3)C2)CC(C2CC2)C1 c1(C(c2n(C)nnn2)NCc2ccc3ncsc3c2)nc2c(s1)CC(C)(C)CC2 C(=O)(C1=CCC2CCC1N2C(=O)CC1CCCOCC1)NC(C=C)(C)C c1(CCN(C(c2ccn(C)n2)C(=O)NC2COC2)C)ccncc1 C1(NC(c2c(C)cc(F)s2)=O)CN(C(C2(C(C)(F)F)CCC2)=O)CC12CCC2 C1(NC(COCCC)=O)CC2CCC1CC2NC(c1c(N)ccc(C)c1F)=O C=C(C)C1OCCC1CNC(=O)CCCCn1cc(CC(C)(O)CC)nn1 C(CCC(=O)NCC1(CNC(c2coc(O)n2)=O)CC1)NC(N)=O c1(CN2CCC(N(C)C(c3cnc(Cl)cc3Cl)=O)C2)cnc2cc[nH]c2c1 C(=O)(C(CC)N(C(c1cc(Cl)ns1)=O)CC)NCCC C12CCC(C1)OC2.C12(C=O)CC(F)(C1)C2.c1(C(=O)N)cc(C(F)F)cs1 C(CC(=O)NC)(C(F)(F)F)NC(C1(C)CC=CC1)=O.c1ccc(C(N)=O)o1 CCC(C)C(C)C(=O)NC(C)(C)CNC(=O)CCC(=O)c1ccncc1 C1(NC(C(COC)COC)=O)CCN(C(=O)C(C)C(C)(F)F)C12CCC2 Cc1cc(N(C)CCOC(F)F)nc(N2CCC(CF)C2)n1 C1(O)(CNC(C2(CCC)CCC2)=O)CCN(C(C2(N(C)C)CCC2)=O)CC1 C1(C(N)=O)CCC(C(=O)NCCCNC(C2CC(OC(F)(F)F)C2)=O)O1 N1(C(c2cncc(C(=O)OC)c2)=O)CCC(C)N(C(=O)C(C)C2CCCC2)CC1 C(=O)(CCCC1CC1)NC(C)(C)CNC(=O)CN(C)C1CC1 C1(C(=O)OC)(C(=O)N(C(=O)CC)C)CCCO1.C1CN1 c1(C(N2C(C(=O)NCC)CCC2)=O)cccc(NCC2CC(F)(F)C2)c1C CC#CCCC(=O)NC(C)(C)C(C)NC(=O)C(c1ccc(C(C)(C)C)cc1)=O c1(C(N(C2CC(NC(c3cnn[nH]3)=O)C2)C)=O)cc(C2CC2)ccn1 C(=O)(C(C)CC(F)(F)F)NCC1CCC(NC(c2cc(C)ncn2)=O)C1 CN1CC(C(=O)NC2(CC(=O)N(C3CCC3)CCO)CC2)CCC1=O C1(N(C)C)CN(Cc2nnnn2-c2ccccc2)CC12CC2 c1(C(=O)NC2(CO)CN(C(c3nn(CC)c(C)c3)=O)C2)csc2nccn12 c1(OC)ccc(CCC(N2CCOCC(NC(C3CC(C)(C)C3)=O)C2)=O)cc1F CCCC(C)(O)CC(=O)N1CC2CC1(CNC(c1c(F)cncc1Cl)=O)C2 Cc1cc(C(=O)NC2CC(C(C)NC(c3cnco3)=O)C2)c(C)cn1 C(=O)(C(CC(F)F)NC(C1CCC(C(N)=O)C1)=O)NCCCOC=C c1(C(=O)N)cc2sccc2[nH]1.N1(CC(N2C(CC)CCC2)=O)CCN(C)C(=O)C1 c1(C(=O)NC(C(CO)NC(C(COC)OC)=O)C)cn(C)cc1C CC1(C)CCC(C(N2CCN(C(=O)CCc3ccco3)CC2CF)=O)CO1 c1(N(C(CNCC(C)CNc2ccccc2)=O)C)cccc(Cl)n1 CC(C)CC(C(=O)NC12CC(NC(C3CC4CC4C3)=O)(C1)C2)N(C)C N1(C(c2ccc(OCCCC)cc2)=O)CCN(C(=O)C=Cc2cscn2)C(C)C1 C1(C#N)(C=O)CC2(CC2)C1.c1(CCC)ccccc1.CCCCSCC(=O)N Cc1c(O)ccc(C(=O)NCC2CCCCC2NC(=O)CC(C)C)c1C C1(C(=O)OC)C2CC2CN1C(c1cccc(Cl)c1)C(=O)NC1CCC1 C(C)(C)(CCNC(=O)CN1CCC(C)C1)NC(CC1(OC)CC1)=O C(=O)(CC(C)CNC(C1(COC)CC1)=O)N1CCC(COC)C1 c1(CC)cccc(C)c1NC(=O)CC1CN(Cc2ccc(F)nc2)CCO1 c1(C(=O)NC2C3CC(NC(C(CC=C)OC)=O)CC32)cc(OCC)ccc1O N1(C(C(c2cnn(C)c2)C)=O)CC2CC(NC(=O)C(C)(C)c3cc[nH]n3)C(C2)C1 c1(CC(N2CCC2)=O)nn(C)cc1Cl.C=C1CC(CC(=O)NC)C1.C(=O)C c1(CC)cc(NC(C2CCN(C(=O)C=CC(=O)O)CC2)=O)cc(F)c1.C Cc1nc2ccc(N(C(=O)C(C(C)C)n3ccc(C4CC4)n3)C3CC3)cc2s1 C1(NC(CSCCC)=O)CN(C(=O)C(C)(O)CCC)CCC12CCC2 c1(C(N2CCCC(F)(CNC(CC(C)F)=O)C2)=O)c(S(N)(=O)=O)cnn1C C1(C(=O)NCCC2CCCN2C(=O)Cc2ccon2)COc2ccc(Cl)cc2O1 C1(C)(CC=O)CCS(=O)(=O)N1.c1(CCC)c(C(=O)N(C(C)C)C)cnn1C N1(C(COCCC#C)=O)CC2CCN(C(C3CN(C)C(=O)CCO3)=O)C(C2)C1 C1(CNC(C=CC)=O)COCCN(C(=O)COCc2nc(C)no2)C1 N1(C(C2C(C)(C)C2(C)C)=O)CC2ON=C(CNC(c3n[nH]c4c3CCC4)=O)C2C1 C1(C=O)CCCO1.C1(OCC)CCC1C(=O)NCC(C)OCCO.C=O c1(C(N2CC3(C(NC(=O)CC(O)C4CC4)CCS3)C2)=O)c(Cl)ccc2ccoc12 C(CCC(C(=O)NCc1ccccc1)NC(=O)C(n1cc(C)cn1)C)OC c1(N2CCC(C)C(NC(=O)C(C)(C)C3CCC3)C2)nc2c(cc1C#N)CCOC2 Cc1ccc(C)n1-c1ccsc1C(=O)NC1CC(NC(c2nsnc2O)=O)C1 C#Cc1ccc(C(N2CCOCC2CC(N2CC=CCC2)=O)=O)cc1C C1(CC(=O)NC)CCC(C)CO1.N1(C(C2CN(C(=O)NC)C2)=O)CC(O)C1 N1(C(c2c(NC)scn2)=O)CCN(C(=O)C(C)SCC)C(c2cn[nH]c2)C1 c1(C(N2CCCC(C)C2CCNC(=O)Cc2ccco2)=O)cncc2ccsc12 c12ccc(cc1)S(=O)(=O)N2C.N1(CC)CCOCC1.CC(C)CN(C(=O)C)C.O CCCC(C)(O)CNC(=O)C(C(C)O)NC(C1CCS(=O)CC1)=O c1(C(=O)NCC(CC)NC(C2CC(c3ccccc3)O2)=O)ccsc1C(F)F C12(C(N3CCCC(CNC(CCCCOC)=O)C3)=O)CC1COC21CCC1 c1(N(C)C)ncccc1C(=O)NCC1(O)CN(C(C2CC23CC3(F)F)=O)C1 Cc1cc(C(=O)NCC2CCC2NC(=O)Cc2ccccc2)n2nccc2n1 C(c1c(C)cc(C)cc1C)=CC(C=O)N(CC(C)C)CC(C)C.C(CC)SC.N c1(CC)nc(C)n(C)c1C(=O)NCC1CCCCC1.C(=O)C1=COCCC1.C C(=O)(C(C)CC#N)N1CC(C(=O)NC(C2CCC2)C2CC2)(CC)C1 c1(N(CCOCCNC(C(CCCC)O)=O)C)cc(=O)n2cc(Cl)ccc2n1 CCC(CC(=O)NCCCCCN(C)C(c1cn(CC)nc1C(C)C)=O)SC C1(NC(c2nc(C)oc2)=O)CCCN(C(=O)CC2CCCS(=O)(=O)C2)CCC1 C(=O)(CC(CC)C(C)(C)C)NC1C2CC(NC(C(CCCC#C)C)=O)CC21 CC(C)C(C(=O)NCC1(F)CCOCC1)NC(=O)COCC1CCC1 c1(CC(N2C(CNC(C(C)Cc3ccccc3)=O)C=CC2)=O)cc(F)ccc1F c1(C(=O)NC(CNC(c2ccc(C)c(F)c2)=O)C(C)C)cnc2sccc2c1 N1(C(c2cn(CCC)nn2)=O)CC(OC)C(C(=O)NCCC2(C)CC2)C1 C(CCCC(=O)NC1(CNC(=O)Cc2cccc(Cl)c2)CC1)N(C(C)=O)C C1(C(N(CCNC(=O)C(C)NC=O)CC)=O)CC(O)(C(=O)OC)C1 c1(C(=O)NCCC(C)NC(c2ccc(C)c(O)c2)=O)cn2ccc(F)c(C)c2n1 Cc1cc(C(F)F)nn1CC(=O)NCCCCCNC(=O)C1=COCC1 CCCCCCCCC(C)C(=O)NC1CC2(C1)CC(NC(C1CC(C)=NO1)=O)C2 N1(c2cc(N(C)Cc3ccnc(N(C)C)c3)ncn2)CCCN(CC(N)=O)CC1 C1(C(N(CC)Cc2ccccc2)=O)CCCN(C(c2nccs2)C)C1 CC1(C)CC(CCNc2cc(C(C)(C)C)sc2C#N)CCO1 N1(C(C=C(CC)CC)=O)CCCN(C(C2(C(=O)OC)CCCC2)=O)CC1 c1(C(=O)NC2(C)CCN(C(C(C(=O)OCC)F)=O)C2)ccc2nc(O)[nH]c2c1 CCCCC(O)C(=O)NC1CCCC(NC(c2cnc(C(C)=O)s2)=O)C1 N1(C(CCCNC(C)=O)=O)CCC(F)C(NC(c2csc(-c3nc[nH]n3)n2)=O)C1 Cc1cc(C(N2CCCC(c3ccc(NC(c4ncco4)=O)cc3)C2)=O)nn1C c1(N(C2C(C(C)C)NCC2)CCN2CCCCC2)cc(Cl)cc(Cl)c1 S(=O)(=O)(C1CCCc2ccccc21)N(CC(C)C)Cc1ccc(C)s1 Cc1ccc(Br)cc1C(C)(C)C(=O)NC1OC(=O)CC1(C)C CC(CC(=O)N1CC(CNC(=O)CC2CSC2)CC1(C)C)C(C)(C)C C(=O)(CC(O)CCSC)NCCN(C(=O)C(c1cccc(Cl)c1)O)CCC C(=O)(C(C)CC(N)=O)NCC1(C(C)(C)O)CN(C(C=C(CC)CC)=O)C1 O=C(C1Cc2ccccc21)N1CC2OCCN(C(c3cc(F)n[nH]3)=O)C2C1 N1(C(c2ccc(C)c(O)c2)=O)CCC=C(C(=O)NC(C)(C)C(O)CO)C1 C1(NC(C2CC(C#C)(O)C2)=O)CN(C(c2ccnc(O)c2)=O)CCC1F C1(NC(c2cc(C)oc2)=O)CCC(O)CN(C(=O)C(c2ccc(O)cc2)(C)C)C1 CN=c1[nH]cc(C(=O)NC2CCC2NC(=O)CCC2CCCN(C)C2)s1 CC(C)(F)C(C)(F)C(=O)NCC(F)C.c1(C(=O)N)ccc(C(F)(F)F)cc1O C1(NC(=O)NC(c2ccccc2)C)CC2(CCN(C(C3CCCC3C)=O)CC2)C1 n1(CCCSC)nnnc1C(C1CC=CC1)(C)NCC1CCOC1 c1(C2(C(N3CCN(C(COC)C(F)F)CC3)=O)CC2)ccc(Br)cc1Cl c1(C(N2CCC(NC(=O)C(C3CCCCC3)O)C2)=O)cccc2c1C(=O)NC2 N1(C(c2ncccc2NCc2cc3cnccc3[nH]2)=O)CCN2CCOCC2C1 c1(CCCC(=O)NC2CCCC(NC(=O)Cc3ccno3)C2)cc(F)ccc1F C1(NC(C(CNC(c2c(CCC)n[nH]c2)=O)CC2CC2)=O)CCOC12CCCC2 n1(CCC)nc(C)c(C(c2nnnn2Cc2ccco2)NCCCCO)c1Cl N1(C(C(c2c(F)cccc2F)C)=O)CCC(N=c2[nH]c(C3CC3)nc(=N)[nH]2)C1 Cc1cccc(C(N2CCCN(C(C34CCOC(C)(C3)C4)=O)CC2)=O)c1Br c1(OC)cc(OC)cc(C(O)CN(C(=O)CC2CN3CCC2CC3)C)c1 C1(CC(=O)NCC(CC)N(C(=O)C=Cc2nccs2)C)CC2CCC1C2 C=CC(CCC)CC(=O)NCC(C)(C1CCC1)NC(c1ccccc1CO)=O c1(C(=O)NCCC2CCCN2C(C2CC(C3CC3)=NO2)=O)cnn2ccncc12 Cc1ccc(F)cc1C1(C(=O)NC2CN(C(C3CC(N(C)C)C3)=O)C2)CC1 c1(OC)ncc(Cl)c(=NC(C)C2CCCCN2C(=O)CN(CCO)CCO)[nH]1 c1(C(=O)NC2(C)CCN(C(c3cc(OC)n(C)n3)=O)C2)c(Cl)cc(Cl)cc1Cl Cc1ccc(C(=O)N(CCCN(C(=O)Cc2ccc(C(N)=O)cc2)C)C)cc1Cl c1(C(=O)NCC(CO)NC(c2occ(C)c2)=O)coc2ccccc12 N1(C(C=CSC)=O)CC2CCC(C1)N2C(c1ccnn1CCc1ccccc1)=O c1(C(N2CC(C)(C(=O)Nc3c(C)n[nH]c3)C2)=O)cc(CC(C)C)nn1C c1(SC(C)C)ncccc1C(=O)NCC1CCN1C(c1cnc(C)cn1)=O C(c1cccc(Br)n1)=C1CN(C(=O)OC(C)(C)C)C1 C1(N(C(C2CC2)=O)C)CC2CCC(C1)N2C(C1CCN(C2CC2)CC1)=O.CC C#CC1CC2(CC2)CN1C(=O)C(CCOCC)NC(=O)C(C)C1CCC1 C1(NC(C(=O)NC(C)C)=O)CCN(C(=O)C=Cc2ccccn2)CC1(C)C C#CC1(C(=O)NC2CCN(C)CC2C#N)CCN(C(c2ccncc2)=O)CC1 CC(C)C(C)CC(=O)NC(C)CC(C)NC(c1cc(O)nc(C2CC2)n1)=O CC1COc2c(C(=O)NC(C)CNC(C3CC4C(C3)C4(F)F)=O)cnn2C1 c1(CC(=O)NC2CCN(C(C3COC(=O)N3)=O)C2)cc(F)ccc1Cl C1(NC(=O)Cn2cnnc2O)CCCN(C(=O)C(F)(F)CC2CC2)C1 c1(OC)cc(C(N2CCOCC(CNC(c3sccc3F)=O)C2)=O)c(N)cc1F C1(O)(C(C)NC(c2c(C)occ2)=O)CCN(C(C2CCC(=O)N2)=O)C1 CC(=Cn1ccnn1)C(=O)NCCCCN(C)C(C1OCCCC1(C)C)=O N1(C(=O)NC(CCC=C(C)C)C)CC(CCC=O)CCC1C(=O)O.C(C)(C)C c1(OC)ccc([N+](=O)[O-])c(N(C(C)CNC(C2COCCN2C)=O)C)n1 N1(C(C2(CCCNC)CCCN2C(=O)C)=O)CCCC(CSC)C1.CC=O.S C1(C(N2CCC(NC(c3cc4cccn4cn3)=O)CC2)=O)CCn2nncc2C1 CCCC(C)(O)CC(=O)NCC(O)CN(C(=O)CCc1ccc(OC)cc1F)C S(=O)(=O)(c1cc2oc(=O)[nH]c2cc1F)N1CCC(N2CC(C)(O)C2)CC1 c1(NCC2(CNC(CCCC#CC)=O)CCC2)cc(C(F)(F)F)ncc1[N+](=O)[O-] CC#CCCC(=O)NCC1CC(O)CN1C(=O)C(C)CSc1ccccc1 C=C1CC(CC(=O)NCCCOCCNC(=O)CCn2ccnc2)C1 CCC(CC(=O)NC1C2CN(C(c3cnc(Cc4ccccc4)s3)=O)CC12)SC CC1=C(C(=O)NCC2C3CCC(C3)N2C(=O)CC2CCOC2(C)C)CCO1 C1(NC(C(CCCOC)C)=O)CC(N=c2[nH]c3ncnc-3c(C(F)(F)F)[nH]2)C1 N1(CCc2cn(CC3N(C(=O)C(O)C4CCCC4)CC3)nn2)CCC(O)CC1 c1(C(=O)NCC(CCNC(C(CC=C)C(C)C)=O)=C)cc2cc(C)ccc2o1 c1(CC)c(Cl)cc(C(N2CC3CC2CN3Cc2cccc3sccc23)=O)cc1Cl C1(NC(=O)NC2CCOC(c3cccnc3)C2)CCc2nccn2C1 C1(C(=O)NC)CC2(C1)CC(C(=O)N(C(CSC)C=O)C)C2.C(C)(C)C.O N1(C(C2(C(C)(F)F)CC2)=O)CCN(CC2CCCN(C(C3CC=CC3)=O)C2)CC1 c1(C(C(=O)NC2CCOCC2)N(C(C)(C)C)CC)ccc(Cl)c2c1CCC2 C1(OC)CN(C(=O)CCOC2CCCCC2)CC1.C(=O)(C(C)(C)c1cc[nH]n1)N N1(C(CC(CC)OC)=O)CC2(CCCN(C(C3CCCN4CCCCC34)=O)C2)C1 C(=O)CCC(C)(F)F.C1CC(F)(F)C1.C(=O)(C=O)NCCNC(C)=O.N C=CCN=C(NCC(Br)=C(C)C)NCC1COCC(C)(C)O1 C1(c2cccs2)(C(=O)NCC2CC(OCC)C2)CCCCC1 c1(C(N2CCCC(Cc3ccc(F)cc3)C2)=O)nc2ccccc2n1C(F)(F)F C1(N(C(c2c(C)onc2)=O)C)CCN(c2cncc(Cl)n2)CC1 CC(CS(C)(=O)=O)C(=O)N1CCCC(C)(C)C1.C1(CC=O)CC(N(C)C)C1.C C(=O)(C(C)(C)CCCNC(=O)Cc1ccc(O)nc1)NC1C(N(C)C)CC1 CC1(C)OC2CC(C(N3CCOCC3CCNC(=O)Cc3ccns3)=O)CC2O1 Cc1oc(S(N)(=O)=O)cc1C(=O)NCCCNC(=O)C(C)O N1(C(c2cc3scc(C)c3[nH]2)=O)CCCC2(C1)CN(C(=O)C=CCF)CCO2 N1(C(C(CC)(C)O)=O)CC(C2CCN(C(=O)CCc3cnc[nH]3)CC2)C1 C(=O)(C1Cc2ccc(Cl)cc21)N1CCOCC(NC(c2cc(Cl)cc(Cl)n2)=O)C1 CCCCC(C)(F)C(=O)NC(C)CCNC(c1cnc(C2CCC2)nc1O)=O c1(C(=O)NCCCCN(C(C2(COC)CCCC2)=O)C)cccc2sncc12 CCC(CC(=O)N1CC2CCC(C1)C2NC(c1cnn(C)c1)=O)C(C)(C)C N1(CC(=O)NCCC)CCN(C)C(=O)C1.C(=O)CC.C1(C=O)CCC1.CC CN=C(NCCC1(O)CCOC1)NC(c1csnn1)C c1(C(N2CC(C)C(NC(C3CC4CCCC34)=O)C2)=O)cc([N+](=O)[O-])cnc1O C(=O)(C1=C(C)OCCS1)NCC(c1ccc(F)cc1F)NC(C(CC)C)=O C1(C(=O)NCCNC(c2c(OC)cccc2Br)=O)CCn2ccnc2C1 C=CCCCC(=O)N1CCSCC1CCNC(=O)Cc1ccns1 C1(C(=O)Nc2ccc(C)cc2C(N)=O)C2CCC1CN(C(c1occc1C)=O)C2 C(c1ccc(Cl)c([N+](=O)[O-])c1)=CC=O.C=C=C(C)CC(=O)N1CCCC1CC.N Cc1c[nH]c(C#N)nc1=NC(CN(C(c1coc(C(F)F)n1)=O)C1CC1)C1CC1 c1(NCC(=O)N(C2(C(=O)O)CC(O)C2)C)ccc2ncccc2c1 c1(OCC)cc(C(C)NC2C=CC(C(=O)NC)C2)sn1 N1(C(C(C)NC(CC)=O)=O)CCC2(CC1)CCN2C(c1cc(Br)cc(C)c1C)=O c1(C(N2CCN(C(COCCC=C)=O)C(C)C2)=O)[nH]c2ccc(Cl)cc2c1Cl C(C)(C(C(=O)N1CC(CC(=O)NCc2ccc(C)s2)C(C)C1)N(C)C)OC C(C1c2ccccc2CCN1C(C1CCCO1)=O)NC(c1cc2ccsc2[nH]1)=O C1CC(=O)N1.C1(CNC(C)=O)CCC1C(=O)N(CC(C)C)C1CC1 c1(SC)ccc(CNC(c2ncnn2C)C(F)F)s1 c1(C(N(CC)CC)=O)ccc(-c2cc(O)ns2)cc1.c1(CC=O)cnc(C)[nH]1 N(C(=NCC(O)c1ccc(Cl)cc1)NC(C)CC)CC(=O)N(CC)CC c1(CNC(=O)CCc2cc3ccccc3o2)ccc2oc(O)nc2c1 C1(CC)CC12CCN(C(c1sc(Br)nc1Cl)C(=O)NC1(C)CC1)CC2 N1(C(CCC2C(C)C2)=O)CC=C(C(C)(C)C(=O)NC(c2ccc(F)cc2)C)C1 C(c1cncc(O)c1)=CC(=O)NCC1CC(O)CN1C(C1CSCCS1)=O C(C(CNC(c1sccc1C)=O)C(F)(F)F)NC(CC1CCC(OC)CC1)=O C1(CNC(c2n(C)ncc2C(N2CCSCC2)=O)=O)CCCC12NC(=O)NC2=O C1(NC(C(CC)OC)=O)CCN(C(c2ccc(O)c(F)c2)=O)C12CC2 c1(CC(=O)N(C)CC2OCCN(C(C(CC=CC)C)=O)C2)ccc(C)c(O)c1 C(C(=O)NCCC(C(=O)N1CCN(C(=O)OC)CC1)OC)(C(C)C)OC C=CC1OCCC1C(=O)NCC1CN(C(=O)C(C)(C)COC(C)C)CC1 C1(N(C)C)CCN(CC(=O)NCC2CCCN(C(=O)Cc3nccn3C)C2)CC1 N1(C(C2(C)COC2)=O)CCN(C(c2cncc(OC(F)F)c2)=O)C(C2CCC2)C1 Cc1c(C(=O)NCCCCNC(C2CCC2F)=O)cnn1C(C)(C)C CCC(C(=O)NC1(C(=O)NC2CCCC2C#N)CCSC1)C(F)(F)F C(=O)CC1=CCOCC1.C1(C(=O)C2CC2)CCC(c2n[nH]c(-c3ccccc3)n2)O1 N1(C(c2cc(C)no2)=O)CCN(C(C2CCOC3(CCCC3)C2)=O)CC(C)(F)C1 c1(C(=O)N)cc2ccc(F)cc2o1.C(=O)(C(O)P(C)(C)=O)NCC(C(C)C)C CC1CN(C(=O)Cc2n[nH]c(=N)s2)CC(C)N1C(=O)C(C)CN1CCOCC1 c1(NC(c2c(C)ncs2)=O)nccc2ccc(-c3ccc4cnn(C)c4c3)cc12 C(CC)(CCC(=O)NCc1cnc(C)[nH]1)NC(CCCOCC)=O N1(C(Cc2cccc(OC)c2)=O)CCC(C)(CNC(=O)C(=O)N(C)C)CC1 c1(OC(C(=O)OC)C)ccccc1CNS(=O)(=O)CC1(C)CCCCC1 n1(C(C)(C)C)cnc(C(=O)NC2CC2)n1.c1(C(=O)N)cocc1.[nH]1cccn1 N1(C(c2c(C)cn(C)n2)=O)CCCC(C)(CNC(c2cc(N)ccc2Cl)=O)C1 C(C)CS(C)(=O)=O.C1(C=O)C(C#N)C1(C)C.C1CCC1.C(=O)(CO)NC c1(OC)ccc(NC(=O)C(c2cccc(I)c2)N(C)CCN2CCOCC2)cc1 C1(NC(c2[nH]cc(CC)c2)=O)CC2CC1N(C(c1ncn(C(C)C)n1)=O)C2 c1(CN(C(C=CCOC)=O)C)ccc(CNC(c2ncncc2F)=O)cc1 C(=O)(CCC(=O)NC(C)CC(N1CC=CC1(C)CO)=O)NCCC c1(C(N2CCC(CCOC)(NC(=O)COC(F)F)C2)=O)cc2sc(C)cc2s1 c1(C(N(C)CCNC(=O)CN2CCCC2C(F)F)=O)cccc(CO)c1 c1(C(N2CCCC(NC(CC(N3CCCCC3=O)C)=O)C2)=O)cnc(N)c(N)c1 c1(NC(C)=O)nc(-c2ncccc2C)nc(Cl)c1NC(C)(C)C C1(C=O)(CC)CS(=O)(=O)C1.CCCC1CC1.C(=O)C=CCN.N C(C)(c1ccccc1)=CC(=O)N(C(C(=O)N(CC(CC)O)C)C)CC Cc1ccc(F)c(C(N2CCC(C(C)C(N3CC(=O)NC(C)C3)=O)CC2)=O)c1Cl C1(C(N2CCC(C)C2)=O)OC(C)(C)OC1(C)C.C(CC(=O)N)OCCOCC N1(C(c2c[nH]c(=NCC=C)s2)=O)CC2(CCCC(C)O2)C1.C(=O)C(C)=C(C)C.N N1(C(c2c(CC)scc2)=O)CCCC2(NC(c3cc(O)nc(Cl)c3)=O)CCCC12 NC1CN(C(c2ccc(N3CCN(C(=O)CSC)CC3)cc2)=O)CC2(CCC2)C1 NS(=O)(=O)c1c[nH]c(C(N2CC3CC2C3NC(c2ccc(CO)cc2)=O)=O)c1 c1(N(C)C(c2sccc2C(=O)OC(C)(C)C)=O)cccc(Br)n1 CCN=c1[nH]c(C(N2CCC(C)C(CNC(c3n[nH]c(C)c3Cl)=O)C2)=O)cs1 c1(C(C(=O)NCCCCCN(C(CC)=O)C)O)ccc(C(C)C)cc1 O=C1COCC2(CCN(C(c3cn(CC4CCOCC4)nn3)=O)CC2)N1 C1(C(=O)NCC2CCCC(NC(CCc3cnc(C)o3)=O)C2)Cc2nncn2C1 c1(C(=O)N)ncn2c1CCC2.C1(CNC(COC(CC)CC)=O)(C)CCCCC1 CN=c1nc(N2CCCC(NC(C)=O)C2)[nH]c(=NCc2ccc(N)c(C)c2)[nH]1 c1(CC(=O)NCC(CC=C)NC(=O)C(CC)=[SH]C)sc(SC)nc1C c1(OC)cccc(-c2nc(C(c3cnn(C)c3)C)n(C3CCCOC3)n2)n1 CCC(C(=O)NCc1ncoc1CCNC(c1coc(Cl)c1)=O)N(C)C N1(C(C2C(=C)C2)=O)CCC(F)(CNC(c2cc(-c3ccco3)cs2)=O)C1 c1(C(=O)NC2COCCC2NC(C2CC(O)C2)=O)c(F)ccc(F)c1F C(=O)(CCCc1ccncc1)NCC(CC)NC(=O)C(CSC)c1ccccc1 N1(C(C(CCC)C)=O)CCC(C2CN(C(=O)CC3CCSCC3)C2)CC1 C(=O)(CCC(F)(F)F)N1CCC(N(C(=O)CCCc2nccs2)CCC)C1 CC1(C)COCC(C(=O)NCCOCC)O1.C1(CC=O)CCCS1(=O)=O.N c1(CC(=O)NCCCC=C)cccc(SC)c1.C1(CC=O)SC(=N)NC1=O N1(C(c2cccc(CC)c2O)=O)CC2COCC(C1)C2NC(=O)COCCCF C#CCCC(O)C(=O)N(C)CC1CCCN(C(=O)C(c2ccc(OC)cc2)=O)C1 N1(C(=O)OC(C)(C)C)CCCCC1.c1(C(=O)N)ncoc1.C1(F)(C=O)CC1 C=CC1OCCCC1C(=O)NC1CCN(C(=O)CC(C)C(F)F)CC1O c1(OCC)ncc(C(N2CCCC2C(C)C)=O)s1.C1(CCC=O)CCCCO1.N n1(C(C)C)nccc1C(=O)NC1C=CC(C(N2CC(C)(c3ccccc3)C2)=O)C1 N1(C(CC2(COC)CC2)=O)C(C)C2CC1C2NC(=O)CCC1CC1(Cl)Cl Cc1ccc(Cl)cc1C(=O)NC12CC(C=O)(C1)C2.c1cccc(N(C)C)c1.N C#Cc1cnn(C)c1C(N1CCC(CCC(N2CCCCC2CF)=O)C1)=O C#CCC(CC(=O)NC(C1CCCC1O)C)NC(c1c[nH]nc1[N+](=O)[O-])=O N1(C(C(CC)(C)OC)=O)CCC2CN(C(c3cscc3C(F)(F)F)=O)CC2C1 N1(C(C(CC2CCC2)NC(Cn2ncc(C)c2)=O)=O)CCCC(C)C1CO N1(C(C2(C(C)C)CC2)=O)CC2(CC(NC(C3CC(=O)NC3(C)C)=O)CO2)C1 n1(CCCOC)cc(C(=O)N)cn1.CCCCCN(C(=O)CN(C1CCC1)C)C c1(C(C)=O)ccc(C(=O)NC(C)CNC(=O)C=CSc2nc[nH]n2)c(F)c1 N1(Cc2c(C#N)cncc2)CC2CCC1CN(C(c1ncccc1Br)=O)C2 C1(C(=O)NC2CN(C(c3c(C)csc3)=O)CC2n2cccn2)CC(C2CC2)=NO1 N1(C(c2c(CC)cco2)=O)CCN(C(c2c(F)ccc(F)c2O)=O)CC(O)C1 N#Cc1ccc(C(N2CCN(C(=O)CC3CC=CCC3)C(CCO)C2)=O)c(F)c1 c1(C(N2CCC(C)(NC(C(C)n3cnnn3)=O)C2)=O)ccnc2ccc(N)cc12 N1(C(c2cnn(CC)n2)=O)CCN(C(c2cn(C)c(C)cc2=O)=O)CC(C)(F)C1 c1(OC)c(C#N)ccnc1NC(C1CNCCN1Cc1ccc([N+](=O)[O-])cc1)=O C1(NC(c2n(C=C)ncc2)=O)CCN(C(=O)C(C)CF)C(C)C1 C12(C(N(CC)CC)=O)CCOC(C)(C1)C2.C1(N(CC(=O)N)C)CCSC1 c1(C(N(CC)C)=O)ccc2c(c1)OCC2.C1CCCN1C(=O)CN(C)CC C1(CCNC(c2n(CC)ncc2)=O)CSCCN1C(=O)C(F)C1CC1 c1(C(N2CCC(N(C(C(c3cnn(C)c3)OC)=O)C)C2)=O)sc2cncn2c1C C(=O)(C(CC(C)C)c1ccccc1)N1CCCC1.C1(C(=O)OC)(CC)CC1C.S CCC(O)CC(=O)N1CC(C(=O)NCCSCCOC)(COC)C1 c1(NC(CC)C(O)C(C)C)ncc(S(=O)(=O)N2CCN(C(C)C)CC2)cc1Cl c1(C(N2CC(CNC(c3cc(Cl)c(Cl)s3)=O)C2)=O)ccccc1OCF C1(CC)CCN(C(c2oc(CNC(C3CC4CCC4C3)=O)cc2C)=O)C1C c1(Cc2nnnn2CCC2(C)CC2)nc(Br)cn1C.C1(COC)(N)CCCC1 C(=O)(C(NC(C1CCCN1)=O)=Cc1ccco1)OCC c1(NC(=O)C(=O)NC2CC3CCC(C2)C3O)cccc2c1COC2=O N1(C(CCc2c(C)cccc2)=O)CCN(C(c2cn(C)cn2)=O)C(C(F)(F)F)C1 N#Cc1ccc(C(N2CC3C(C(C4CC4)=O)C3C2)C(=O)NC2CCC2)cc1 N1(C(C(C2CCCOC2)OCC)=O)CCC(CF)(NC(C2CCSC2)=O)C1 c1(C(C(=O)N)(F)F)ccc(F)cc1C.C=CC1CC1C(=O)NC1CC(CC)C1 n1(CC(C(=O)N2C(CNC(CNC(CCC)=O)=O)CC2)C)nnc2ccccc12 c1(OC)ccc(=NC(=O)C2CCCN2C(c2cccc(C#N)c2Cl)=O)[nH]c1OC c1(SCc2n(CCOC)c(N3CC(F)C(F)C3)nn2)ccc(C#N)c(C)c1 N1(C(C(CCC)OCC)=O)CCCC(C2CCN(C(C3COC3)=O)CC2)C1 N1(C(C(C)CN(C)C(C2CCC(N(C)C)C2)=O)=O)CCCC(CO)C1 c1ccc(F)cc1O.CC1=CCC(C(N2CC(O)CC2CNC(=O)C)=O)CC1.O N1(C(C=C(CC)C)=O)CC(NC(C2CC=CCC2C(F)(F)F)=O)CC(C)(C)C1 C(=O)(C#CC1CCCCO1)N1CCC(C)(CNC(C(C)=CC)=O)C1 c1(C(=O)NC2C(OC)CN(C(c3ccc(CC)[nH]3)=O)C2)ccc2c(c1)CCOC2 C(=O)(C1=NOC(CNC(C2CC=CCC2)=O)C1)NCCCCCN(C)C c1(C(=O)NCCNC(C2CCC(C(=O)OC)C2)=O)ccc(Cl)cc1 C(=O)(CS(=O)(=O)C(C)C)N1CCC(N(C(C2C3CCN2CC3)=O)CC)C1 c1(CC)cc(C(=O)NC(c2ccncc2)C2(C(C)OC)CCC2)ns1 C1(C(=O)NC(c2ccncc2F)C)CCN(C(C2CN(C)C2)=O)CCO1 N1(C(C=CCC(C)(C)NC(CC2C(C)CCC2)=O)=O)CCC(C)(O)C1 C1(NC(c2cc(Br)ccc2Cl)=O)CC2(C1)CN(C(=O)Cc1cccc(Cl)c1F)C2 C1(C(NOCC(=O)NCC2(CC)CC(C)(C)C2)=O)C2CC3C(C2=O)C13 C12(C=O)C(=O)C3CC1C2C3.C1(C(N2CCC(n3ccnn3)C2)=O)CC(O)C1.N C1(NC(c2nccn2C)CC)CCNC(C)(C)C1 c1(N2C(C(N=c3cc(C)o[nH]3)=O)CC3CC32)ncnc2ccc(Br)cc12 C(=O)(C1=CC2CCCC12)NCC(C1CCCCC1)NC(C=C(CC)CC)=O N1(C(CNC(c2n(CCOC)ncc2)=O)=O)CCN(C(C2CC2Cl)=O)CC1 Cc1cc(N2CC(C)OCC(C)(C)C2)ncc1S(=O)(=O)NCc1ccnn1C(C)C CC(=O)CCC(=O)N1CCOC(C(=O)NC2CC(=O)N(CC)C2)C1.C(C)(C)C N1(C(C23CC(C)(OCC2)C3)=O)CCOC2(CCN(c3ccc(C#N)nn3)C2)C1 C1(N(C(C=C(C)CNC(=O)C(F)=CC2CC2)=O)CC2CC2)CCCC1 c1(CC(N2CCC(N(c3nnco3)CCO)C2)=O)cnn2ccccc12 c1(OC)cc(OC)c(C(C)NCC2(CCO)CC2)c(Br)c1 N1(C(CCCCN(C)C)=O)CC2(CC2)CC1CC(=O)N(C)Cc1cscn1 C(CC)(CCCC(=O)NC(C)CN1CCOCC1)NC(C=CCC)=O CC(CCS(C)=O)NC(=O)NC(N1CC(OC(F)F)C1)=O N1(C(=O)CSCc2cccnc2)CCC2CN(C(=O)CCCCCO)CC2CC1 C1(C(=O)N)CC2CC(O)CC(C1)C2.C1(CNC(C2CCC(C)C2)=O)CCOCC1 c1(C2C(C)C2)cc(C(=O)N(CC)CCC)no1.C1(C=O)COCC1C(N)=O C1(C=O)CCCS(=O)(=O)C1.C1CCCCC1.c1(C(=O)N)ccn(C(F)F)n1.C N1(C(CC)=O)CCC2(C1)CN(C(c1ccc(N)c(N)n1)=O)C2.C(C)OCC.O c1(OC)ncc(C(=O)NC(CNC(=O)CC)C(C)C)c(C)n1.C1COC1.O Cc1ccc(CC(=O)NCCC2CC(NC(c3ccccc3C)=O)C2)cc1 O=S(=O)(c1[nH]c(=NCC2CCCCO2)ccc1Br)N1CCC(c2ccncc2)C1 C#CCCC(O)C(=O)NC1CN(C(=O)CNC(=O)C2CC2)CCC1F C1(NC(=O)Nc2nnc(C(=O)OC)s2)CC2CCC(C1)N2C.c1ccccc1 C1(NC(C(C)OCC#C)=O)CCCN(C(=O)CSc2ccccc2O)CC1 C(c1ccccc1Cl)=CC(=O)NC(C1N(C(CCCC#C)=O)CCCC1)C C1(NC(CCCc2nc(C)sc2)=O)CCOC(C2CCN(C(=O)C(N)=O)CC2)C1 CC(CNC(C1CC2CCC2C1)=O)CC(=O)N(c1cccc(Cl)c1)C Cc1cc2ccc(C(N3CCCC3CNC(=O)CCOCC(F)F)=O)cn2c1 N1(C(c2cnc(C(C)C)s2)=O)CC(NC(=O)COC(C)(C)C)C(C)(C)C1 CC1(C)C(C(=O)NCC2CCCOC2)CCN1C(=O)Cn1c(O)nnc1O C1(C(=O)NCC(C)CN(C(=O)CNC=O)C)CC2CCC(C1)O2 C12(C(=O)N)CC3CC(O)(C1)CC(O)(C3)C2.c1ccc(N2CCCS2(=O)=O)cc1 c1(C(N(C2CCN(C(c3cccc(SC)c3)=O)CC2)C)=O)cnc(Cl)cc1N c1(SCc2cc(C)sc2)ccc(-n2cc(C(C)N(C)C)nn2)cn1 c1(CCNC(C=CCNC(C(C)OCC)=O)=O)ccc(F)cc1 n1(CC)cnc(=NC(=O)c2ccc(C(F)F)cc2F)[nH]1 C1(C)(CNC(CC2C(CC)C2)=O)CC(F)(F)CN1C(=O)Cc1ccsn1 Cc1cccc(C(=O)NCC(F)CNC(=O)C(C)Cc2cccc(Cl)c2)c1N N1(C(C2CC(OC)C(OC)C2)=O)CCCN(C(=O)C(=O)N(C)C)C(CO)C1 C1(C(=O)NC(C=C)(C)CC)CCC2(CC2)N1C(c1c(C)cncc1C)=O C1(CNC(c2ccc(C)[nH]2)=O)CCN(C(C2CS(=O)(=O)C2)=O)CC1C N1(C(CCCC=C)=O)CCC(CO)C(NC(c2cc(Cl)cs2)=O)C1 c1(C(=O)NCC2(C3CCCCC3)CC2)cnn(CC)c1.C1(O)COC1.C=O C1(NC(CC(CC)SC)=O)CCN(C(c2cc[nH]c2C(=O)OC)=O)CC1CO Cc1nn(C)c(N)c1C(=O)NC1CCC1NC(c1noc(C2CC2)c1C)=O Cn1nccc1C(=O)NC(C1CCCCC1)CNC(C1(CC(F)F)CC1)=O Cc1ccc(NC(C2(CNC(c3ccccn3)=O)CC2)=O)nc1Cl CC1=NOC(c2ccccc2)(C(=O)NCC(C)(C)CNC(C2CCCN2C)=O)C1 c1(-c2cn(C(COCC)C(=O)NCCn3cncn3)nn2)nn(C)cc1Cl N1(C(CCC(=C)C)=O)CCC2(CNC(C3(CCF)CC3)=O)CCCCC12 C1(NC(CC2N(C(C(COCC)C)=O)CCOC2)=O)C2CCC(F)(F)C12 CC1CC(=O)NC1C(N1CC(NC(c2cccc(-c3ccc(F)cc3)n2)=O)C1)=O C(c1ccc(Cl)cc1)=CC(=O)NCC1C(CNC(CC=C=C)=O)C1 C1(NC(C2(C)CCN(C)C2)=O)CC(F)CN(C(=O)CCc2cccs2)C1 N1(C(C(C)c2cccs2)=O)CC2(CC(NC(c3ncc(Cl)cc3O)=O)C2)C1 N1(C(CCn2ncc(C)c2)=O)CC2C(CN(C(=O)C=Cc3ccccc3)C)C2C1 c1(C(N(C)CC2CCC(NC(CC3CN(C)C3)=O)CC2)=O)cc2ccccc2[nH]1 N1(C(c2c(C)ccs2)=O)CCC2(CCN(C(C3(Br)CC3)=O)CC2)C1 c1(CC)ccc(CC(N2CCCC2CCNC(C2(C=O)CCC2)=O)=O)cc1.O Cn1ccc2cccc(C(=O)NC)c12.C12(C(N3CC=CC3)=O)CCC(C)(C1)OC2 c1(CC)noc(CNC(=O)C(Cn2cccn2)NC(C2CC2(C)C)=O)n1 c1(C(=O)NCC2COCCN2C(c2ncc(Br)cc2Br)=O)cc(F)c(Cl)cc1F c1(OC)ccc(C=CC(N2CC(O)(C)C2)=O)cc1.C(=O)(C(C)CC(F)F)N C12(C(N(CC(C)C)C)=O)CC3CC1C2C3.C(=O)C=CC=O.CC=O.N C1(C(=O)NC(C(=O)N(C)Cc2ncccn2)Cc2cnc[nH]2)COC(=O)N1C C12(NC(CC3(C)CCCCC3)=O)CCN(C(c3cccnn3)=O)CCC1C2 c1(C(N)=O)ccc(Cl)c(C(N2CCC2Cn2cc(CCC3CCC3)nn2)=O)c1 C1(N(C(CS(=O)(=O)NC)=O)C)CCN(C(c2ccc(OC)c(N)n2)=O)CC1C C1(NC(C2CC(NC(CC(C)=C(C)C)=O)C2)=O)(CO)CC2CCCC12 c1(NC(C(c2cccs2)OCC)=O)ccc(C(F)F)nc1 CC(C)CC(CNc1nccc(N2CCC(C)(CC#N)C2)n1)N1CCCCC1 N1(C(C(C2CCC2)OC)=O)CC2(CCCC2NC(c2cc3cscc3s2)=O)C1 c1(C(N2CCN(C(c3ncccn3)=O)C3CC23)=O)cnc2c(c1)CCS(=O)(=O)C2 N1(CCCC(=O)N(CCCNC(C2(C)COCCO2)=O)C)CCc2ccccc21 C1(NC(C=CC)=O)CCCC2CN(C(c3cccc(OC)c3[N+](=O)[O-])=O)CC12 c1(C(=O)OC)nc2ncn(CC)c2c(N2CCC(F)(F)C(O)C2)c1C N(C1COCc2ccccc21)C(Cc1c(NC(C2CC(=O)NC2)=O)cccc1)=O C12(C(N(C3CCN(C(C4N(C)CC(C)(C)C4)=O)CC3)C)=O)CCCCN1CCC2 CCCC(C)C(=O)N1CC2CC1C2NC(c1cnnn1CC)=O c1(C(N2CC(NC(c3ccc(C#N)o3)=O)C3(C2)CC3)=O)ccc2cnnn2c1 C(CCCN=c1[nH]c(=NCCN2CCC(C)(F)C2)c2sccc2[nH]1)OC c1(C(=O)NCC2CCCN2C(c2ccnn2C(F)F)=O)cc2n(n1)CCC2 CC1=C(C(=O)NC2CC(CC(=O)NCc3cccnc3)C2(C)C)CCC1 c1(C(N2CCC(C(C)NC(=O)CC(C)(C)C3CC3)CC2)=O)cn2c(n1)SCC2 C1(CC(=O)NC(C(C)C)C2CC2)CC(F)CN1C(=O)CN1CCNC1=O c1(C(=O)NCc2occ(C(=O)NCCOC)c2)cc(O)ncc1F c1(C(=O)NC(C2CN(C(C3C(C)N(C)CC3)=O)C2)C)ccn2ccnc2c1 c1(C(N2CCC(NC(Cc3ccc(C)s3)=O)C2C)=O)ccnc2c1CCO2 CCC(CC)C(C(=O)NC)N1CCC2(CC1)CC2C(=O)NCc1ccco1 c1(NC(CC)CSC)[nH]c(=NCc2n[nH]c3c2CCCC3)nc2c1ncn2C N1(C(c2c(OC)[nH]c(=N)cc2)=O)CC2CCN(C(=O)CCOC3CCCC3)CC12 C1(NC(COCCOC)=O)CC2CCC1C2.C(=O)(CCN(C)C(C)=O)N C1(NC(Cc2ccc(C)nc2Cl)=O)CCC2(CCCCC2)C1 c1(OC)ccc(Br)c(C)c1C(=O)NC.c1(C(N2CCC2)=O)cc2cccn2cn1 N1(C(c2ccn(CC)n2)=O)CC2CCCC(C1)N(C(=O)CCC(C)(F)F)C2 c1(CC(=O)OC)cc(F)c(N(C2CC3CC2CN3)C(=O)C(S)C(C)C)c(F)c1 C1(NC(c2ccn(C)c2)=O)CC2CCC1N(C(C1CC13CCC3)=O)C2 C1(C(=O)NCC(C)(C2CCC2)NC(C2CC2(Cl)Cl)=O)CC2(C1)CC(O)C2 CCC(C)C(C(=O)N1CCN(C)CC1CCO)NC(=O)CCC1CCCO1 CC1CN(C(=O)COCc2ccncc2)CC(C)CN1C(c1ccc(C#N)[nH]1)=O c1(CC(=O)NCC2C(NC(C3(C=C)CCC3)=O)C2)cccc(F)c1 c1(C(C(=O)NCC(=C)C)N(CCCO)C)ccc2ncccc2n1 C(=O)(C(F)(F)C(F)(F)F)NCCCCC(N)=O CCC(C(=O)N(CCC(N)=O)C)NC(=O)CN(C)C(=O)OC(C)C C1(CNC(=O)C(O)C2CCCC2)CC2CCC1N2C(=O)CN1CCCCCC1 c1(CC)c(C(N2CCCC(N(CCO)C(C3COC(=O)N3)=O)C2)=O)cccc1C CC1(C)CCCC(CC(=O)NCCCNC(c2ccc(SC3CC3)cc2)=O)C1 N1(Cc2c(Cl)cccc2)CCC(O)(CN2CCS(=O)(=O)CC2)CC1 c1(OCC(=O)NCC2CCCC2)cnc2n1CCCC2 c1(CNC(CN(CC(C)C)C(C2CCC(C)C2)=O)=O)c(F)cccc1F N1(C(C(c2ccc(C3CCC3)cc2)C)=O)CCCN(C(=O)CO)C(CO)C1 c1(CCC(N2CC(OCCNC(C3CC34CCC4)=O)C2)=O)c(F)cccc1Cl N#Cc1cc(F)ccc1NC(C12CCC(C(=O)NCC(O)CO)(CC1)CC2)=O n1(CC(C(=O)NCC2CC(NC(CCC=CC)=O)C2)C)nnc2ccccc12 c1(C(=O)Nc2ncc(C)cc2C)ccc2c(c1)CN(C(C1(Br)CC1)=O)CC2 C1(NC(=O)CSc2ccc(O)cc2)CCN(C(C2CC(C3CC3)=NO2)=O)CC1F c1(NC(C(=O)NCC(C)(O)c2ccco2)=O)cc(F)c(N(C)C)c(F)c1 C1(CC(=O)NC2C(CNC(CC=CCC)=O)C2)CCCCC1C(=O)O C(CC(CNC(=O)C=C(C)C)NC(C1(Br)CC1(C)C)=O)OC c1(C(N2CC(NC(c3c(C)cno3)=O)C(F)C2)=O)cc2nc[nH]c2cc1[N+](=O)[O-] c1(-c2cc(C(=O)NC3CCOCC3C(F)(F)F)on2)c(F)cc(F)cc1F c1(C(C(=O)NC(CC2CN(C(C(C)=O)=O)C2)C)C)cccc(C2CC2)c1 N1(C(C2C(C=C(C)C)C2(C)C)=O)CC2=C(C1)CN(C(C1Cc3nccn3C1)=O)C2 Cc1cc(C(=O)NC2(C(N3CCCC(CC(C)C)C3)=O)CC(F)C2)c(C)nn1 Cc1ccc(C(N2CCC(OCC(C(=O)C)=O)C2)=O)o1.c1nncn1C.CC.N c1(C(N2CCC(NC(=O)CC3CCC3)C2)=O)ccc2c(=O)n3c(nc2c1)CCC3 c1(C(=O)NCC2(SC)CC2)cc(CNC(c2cnco2)=O)cs1 C(C(O)(C(=O)N1CCC(NC(C2(F)CC2)=O)C(O)C1)C(F)(F)F)N(C)C N1(C(C2C(=C)C2C(=O)OC)=O)CCC2(CCC2NC(=O)CCC)CC1 CC1CN(C(=O)COCC2CCCCO2)CCN1C(c1c[nH]c(C#N)c1)=O C12(NC(c3cc(C)no3)=O)CCN(C(c3cc(N)nc(Br)c3)=O)CC1C2 C1(C(=O)NCCN2CCC(C)C2)C2CN(C(=O)CCc3nc(O)n[nH]3)CC12 O=C1CCC2C(C(=O)OCCSCCC34CCC(CC3)C4)C12 c1(C(=O)N)cccc(Cl)c1F.C(C(=O)NCC1(C)CC1)OCCN(C)C c1(C(N2CCC(C(C)NC(c3n(CC)ncn3)=O)C2)=O)ccnc(OC(F)F)c1 C=Cc1cc(C(N2CC3CCC(C2)N3C(c2cnn(CCC)c2)=O)=O)cc(F)c1 Cc1cc(CNC(c2c(C)nsc2N)=O)oc1C(=O)N(C)Cc1cc[nH]n1 c1(OC)nc(N2CCN(C(c3cc(F)ccc3Br)=O)C(C#N)C2)ncc1C#N C1(NC(c2ccc(CC)s2)=O)CCCN(C(c2cccc(SC)n2)=O)C1C C1(NC(CC2N(C)CCC2)=O)CN(C(c2cc(Cl)c(Br)[nH]2)=O)CC1O N1(C(=O)CSc2cccc(F)c2)CC(C2CCCCN(C(C34CCC3C4)=O)C2)C1 C1(CC)CN(C)C(=O)CN1C(c1ccnc(Cl)c1Br)C(=O)NC.CCCC1CC1 Cc1scc(C(N2CC(C)CC2C(=O)NC2CNC(=O)OC2)=O)c1C c1(CNc2ccc(C(=O)NC(C3CC3)C3CC3)cn2)cccn2ccnc12 c1(C(=O)NCCCCC2CN(C(c3ccc(C)o3)=O)C2)ccc2n[nH]cc2c1F c1(Nc2cc(C)c(O)c(N)c2)sc(S(C)(=O)=O)cc1[N+](=O)[O-] c1(C(CCO)NC(=O)NC(c2nc(C)on2)c2ccccc2)ccc(Cl)c(Cl)c1 C1(C(=O)NC(CCN(C(CSC)=O)C)C)NC(=O)OC1(C)C C1(NC(=O)C(F)=CC2CC2)CCOC(C2CCN(C(c3cnc(S)[nH]3)=O)CC2)C1 C1(C(N2C(C3CCCN(C(COC)=O)C3)CCCC2)=O)CC2(C1)NC(=O)NC2=O N1(C(c2c(C)ncs2)=O)CCc2sccc2C1CNC(C1(C2CC2)CC1)=O N1(C(c2nccc(C)c2F)=O)CC(C)CN(C(=O)CCc2nc[nH]n2)C(C)C1 N1(C(c2cncc(CNC(CCC#CC)=O)c2)=O)CC(C)CCC1CC C1(CN(C(CCN(CCC)C)=O)C)CN(C(=O)C(C)Cc2ccnn2C)CCO1 N1(C(=O)C(F)=C2CCC2)CC2CCC(C1)N(C(c1ccnc3ccnn13)=O)C2 Cc1ccc(C(=O)NC2CCN(CCCNC(C3CC(F)(F)CS3)=O)C2)nc1 C1(NC(=O)COC2CCOC2)CC2CC1N(C(=O)C1=COCCO1)C2 Cc1ccnn1C(C)C(=O)NCCn1cc(C(C)O)nn1 C(CC(C)(C)C)(C(=O)NCc1ccoc1C(N1CCC(N=[N+]=[N-])CC1)=O)OC N1(C(C(CCC)CNC(=O)C(C2CC2)OCC)=O)CCC2(CCCC2)CC1 N1(C(CCn2cc(C(CC)(C)O)nn2)=O)CCCNC(=O)C(F)(F)C1.CCC=O c1(C(N2CC(C(=O)NCC(CC)OC)(CC)C2)=O)ccc(F)cc1F CCCCC(O)C(C)C(=O)N1CCC(NC(c2c(C)ncn2OC)=O)C(F)C1 C1(C)(CC)CCC(C(=O)NC23CC(C2)C3)O1.C(=O)(CC(C)C1CCCO1)N Cc1nc(C=CC(=O)NCCCCC(C)NC(C2(C3CCCO3)CC2)=O)cs1 C1(C(CC(=O)NCC(C)CN2CCCCC2)C)CCC(N)CC1 CC(=Cn1ccnn1)C(=O)NCC1CC(NC(c2cn(C)ccc2=O)=O)CC1O CC1=C(C)CC(C(=O)NC(CC(=O)NCC2(CO)CC2)C2CC2)CC1 c1(OC)nc(Cl)ccc1C(=O)Nc1ncc(-c2cccs2)cc1O c1(NC)ccc([N+](=O)[O-])cc1C(=O)NCCC(C)NS(C)(=O)=O c1(C(N2CCCC3(C(C(=O)OC)C3)C2)=O)nn(C)c2ncccc12 C=C(CNC(=O)CSCCNC(C1(C)CCCO1)=O)c1ccccc1 CC1CC2(CO1)CN(C(C13CC1CCN3C(=O)CC1=CCCCC1)=O)C2 c1(C(=O)NC2(CO)CCCN(C(C3(C4CC4)CC3)=O)C2)cccc2c1CCCC2 N1(C(c2c(CCC)n(C)nc2)=O)CCC(NC(c2ccc(C#N)s2)=O)C(CC)C1 c1(C(=O)NC2(CC)CCN(C(c3cc(F)c[nH]3)=O)CC2)cc2ccsc2n1C C(CC(C(N)=O)NCc1csc(CC2CC2)n1)OC N1(C(CSC)=O)CCC2(CC1)CCN(C(c1ccc(CS(C)(=O)=O)cc1)=O)C2 Cc1cc(=O)c(C(=O)NCC(C)C(=O)NCC(c2ccccc2)O)c[nH]1 C(=O)(N=c1ccn(CCO)[nH]1)C1C(C)N(Cc2cc3n(n2)CCC3)CC1 N1(C(C2(CC=C)CCOC2)=O)CCC2(C1)CN(C(c1[nH]cnc1C#N)=O)C2 Cc1n[nH]c(C)c1Cn1cc(NC(C2CC(O)C2)=O)nn1.c1ccc(Cl)cc1.C C(=O)(C1=CC2C=CC(C1)C2)NCCC(C)NC(=O)Cc1cc2ccccc2s1 C(CCCC(C)(C)C)(C(=O)Nc1ccccc1Cl)N1CCC(C)OCC1 CC1CC(NC(=O)Nc2cccnc2I)c2ccccc21 N1(C(Cc2ncc(C)s2)=O)CCC2CCC(NC(C3(C)CC3)=O)C12 N1(C(CSC)=O)CCCC(C)C1CNC(c1ccnn1CC1CC1)=O C(=O)(CC1=CCCCC1)N1CC(NC(c2cccc(OCCF)c2)=O)C1 O=C(C(O)C(F)(F)F)NC1C=CC(CC(=O)NCCCC(O)CO)C1 CC(C)(O)C(F)(F)C(=O)N1CC(C(N2CCCC(F)(CO)C2)=O)C2(CCC2)C1 N1(CCn2cc(CCCCOC(C)=O)nn2)CCN(C(=O)CN2CCOC2=O)CC1 N1(C(C(F)=C(C)C)=O)CC2(CC(NC(=O)CC3(C#N)CCC3)C2)C1 NS(=O)(=O)CCC(=O)NCC1CCN(C(c2cnn(CC3CCC3)c2)=O)CC1 CCCC(C(O)C(=O)N1CCC(CN(C)C)C1)NC(=O)C#CC(C)C N1(C(C=O)=O)CC2(C1)CN(C(=O)C=Cc1ccc(F)c(F)c1)CCO2.CCC.N c1(C(=O)NC2CC(C)N(C(c3ccc(Cl)o3)=O)CC2)cnc2c(n1)CCCC2 S(=O)(=O)(c1c(C)ccc2ccccc12)Nc1cc(C)ns1 N1(C(CNC(=O)NCC(N2CCCC2)C)=O)CCC2C(=O)NCC2C1 Cc1onc(CC(=O)NC2CN(C(C3CC(=O)NC(=O)N3)=O)CC2(C)C)c1C#N C1(C=O)COC2(C1)CN(C(=O)CC1CCC(C)(C)O1)C2.n1(CC)ccc(C)n1 C(=O)(C(O)CC(C)(C)C)N1C(C(N(C)Cc2ncc(C)o2)=O)CC=CC1 C1CCN(C)C12CCCN(C(C1(C(N)=O)CC1)=O)C2.c1(CC)nonc1C=O.N c1(C(=O)NC2CC(NC(C3C(CC)C3)=O)C2)ccccc1.[SH](C)(=O)=O C1(C(=O)NCC2N(C(CSC(C)C)=O)CCN(C)C2)CCc2cc(F)ccc2O1 c1(CC(=O)NCC23N(C(C(C)CF)=O)CC(C2)C3)ccc(S(C)=O)cc1 C#CCC(C)(C(=O)N(C)Cc1cocn1)NC(=O)CSCCOC c1(OCC)cccc(CN(CCC#N)C(=O)NCCc2cnccc2C)c1 C(C(COC)CC(=O)N1CCC2C(NC(c3cccc(Br)c3)=O)CC12)OC CCC(C)(C)CC(=O)N1CCC(C)(C)C1CC(N1CCCC(C)(N(C)C)C1)=O N1(C(CCCCC)=O)CC2ON=C(CNC(=O)COc3ccccc3CC)C2C1 C#CC1(O)CC(C(N2CC(CNC(=O)Cc3ccc(O)nc3)(O)C2)=O)C1 CC(CC(=O)NC1(c2nn[nH]n2)CCSCC1)C(C)(C)C Cc1ccc(CC(=O)NCC(C)NC(c2cc3sc(Cl)cc3s2)=O)c(F)c1F N1(C(c2cc(=N)[nH][nH]2)=O)CC(C(N2CC3CC3(CO)C2)=O)C2(CC2)C1 C(=O)(C(C)(C)CF)N1CCC(C(C)NC(c2c(CC)nco2)=O)C1 C(=O)(C(=O)C(C)(C)C)NC(C(=O)NC1(C)C(C)CCC1)CCN(C)C c1(CCF)ccccc1.C(C)(C=O)NC(C1C(OC(C)=O)C1)=O.C1CC1.C CC(CS(C)(=O)=O)C(=O)NC1CCCCC1NC(C1OCCO1)=O CC1(NC(C2CC2c2ccncc2)=O)CCN(C(C23CCC(C2)C3)=O)C1 N1(C(C(C(CC)CC)C)=O)CC(NC(=O)CCCC(C)(C)CC)CC12CCCC2 C1(CNC(C(N2CCOCC2)C)=O)CCN(C(C2CCCC23CC3)=O)CC1C c1(C(C(=O)NC2CCC(NC(c3ccc(CCC)s3)=O)C2)(C)C)cnccc1C C1CN(C(=O)CN(S(C)(=O)=O)C)CC12CCOCC2.C(C)(C=O)(C(C)C)OC c1(C(N(C)C)=O)cncc(CO)c1.c1(OC(C(=O)NCC)=O)ccc(F)cc1 n1(CC(=O)NCCC2CN(C(=O)CNc3ccccc3)CCO2)ccccc1=O C12(CNC(CN3CC(C)(C)C3)=O)CCCC1CCN2C(C1CCN(CCF)CC1)=O C1(C(N2CCN(CCNC(c3c(C)onc3O)=O)CC2)=O)C2(CCC2)C12CCC2 C1(C(=O)NC2CCN(C(c3nnn(C)n3)=O)CC2)C2CCC3C(C2)CC13 C=C1CC(N=c2[nH]c(N3CCS(=O)(=O)C(CO)C3)nc3c2CCCCCC3)C1 Cc1c(C(=O)NCC(C)(CC(C)C)NC(c2cnsn2)=O)cnc2ccnn12 C(=O)(C(O)CCC(F)(F)F)N1CC(C2N(C(=O)CC3CCCOC3)CCC2)(O)C1 C=CCC(C(=O)N(CCCN(C(=O)CSc1ccc(C(C)C)cc1)C)C)C(C)C C(=O)(CCCS(N)(=O)=O)N(C1CCCN(C(=O)C(Cc2ccsc2)NC=O)C1)C C1(NC(c2ccc(C)s2)=O)CC2CCC1(C)C2.n1(CC=O)cc(C2CC2)cn1 C(CC(C)(C)C)(C(=O)NCC1CC(O)CN1C(c1ccc2snnc2c1)=O)OC c1(C=O)ccc2c(=O)n(C)c(O)nc2c1.C1(NC(C2C(=C)C2)=O)(C)CCC1 C1(N(C(C2C(C)CCC2)=O)C)CC2CC1N(C(=O)Cc1cnns1)C2 N1(CCNC(C(C)Cn2cccn2)=O)CCN(C(=O)CC2CC=CC2)CC1 C(C(F)(C(=O)NC)C(C)C)NC(c1c(OC)cncn1)=O.C1CC12CCCCC2 C1(CCNC(CC)=O)CSCCN1C(c1oncc1C)=O C(C)(C)(C(C)CC(=O)NCCOCC(=O)NC)NC(C(CC)N(C)C)=O CC(C(=O)N(CCCN(C)C(c1cnn(C)c1)=O)C)C(F)(F)C(F)F c1(C(C(N2CCC(N(CCC)C(c3ccco3)=O)C2)=O)C)cccc([N+](=O)[O-])c1 C(c1ccccc1C#N)=CC=O.Cc1cc(CO)oc1C(=O)NC12CC(C1)C2 c1(C(N2CC3CCCC3C2)C(=O)NC2CCOC2)cc2cnccc2o1 N1(C(C2(SC)CC2)=O)CC(O)(C(C)(C)CNC(C23CCCC2C3)=O)C1 C1(C(=O)NCCCC(CO)NC(CCC(C)SC)=O)CC2CCC(C1)C2=O C(=O)(C(F)CC(C)C)N1CC(NC(c2c(C)sc(C(F)(F)F)n2)=O)(CO)C1 c1(OC)cncc(C(=O)NC2CCCC2(C)NC(=O)CN2CCCCC2)n1 C1(NC(CN(CCC)C)=O)CC(C)(C(=O)NCC(C)C(C)O)C1 N1(C(Cc2cn(CC)nc2)=O)CCC(C2CN(C(C3CC=CCC3)=O)C2)CC1 N1(C(C(C(C)C)OC)=O)CC2(C1)CN(C(=O)CNC=O)CC2CO C(=O)(C1CCCc2nc[nH]c21)NC(C)CC1CCN(C(c2cc(O)no2)=O)CC1 N1(CCCSc2nnc(CC)n2CCC(N)=O)C(=O)C2C3C=CC(C3)C2C1=O C#CCC(CC(=O)Nc1ccccc1C)NC(=O)CCOCCCOC C1(C(=O)NC2CCN(C(C=CC)=O)C2CC)CC(C)(C)CC(C)(C)C1 N1(C(C=CCCC=C(C)C)=O)CCCC12CCN(C(C1CC3CC3C1)=O)C2 CCCC(C)C(=O)N(C(CNC(C1CN(C)C(=O)N1)=O)Cc1ccccc1)C c1(OC)ccc(C=CC(=O)NC(C)(C)C2CC2)cc1.C(=O)C.CC#N.N CC1(NC(=O)C=Cc2nccs2)CCCCC1C(=O)NC1CCC12CCCC2 CC1CCC(N=c2[nH]c(=N)[nH]c(=NCCc3nc[nH]c3Br)[nH]2)Cc2ccccc21 c1(C2C(C(=O)NCC(CC)NC(=O)C)C2)ccccc1Cl.c1cccc(C)c1.O Cc1cc(CC(=O)NC23CCC(C2)N(C(=O)C(c2cnn(C)c2)C)C3)ccc1Cl Cn1nc(C(=O)NCC2(F)CC(NC(c3cscc3Cl)=O)C2)cc1Cl N1(C(C)=O)Cc2nccn2CC(NC(c2c([N+](=O)[O-])c(C)nn2C)=O)C1 C1(C(N(C2CCCN(C(=O)C=CCO)C2)CC)=O)CC(=O)N(C2CC2)C1 CC(C)(CC1CC1)C(=O)N.C1CCCC1.c1(C=O)ccc(SC(F)(F)F)s1.C c1(OC)ccc2nc(N(CC(O)CN(C(=O)CC3CC3C)C)C)sc2n1 C12(C(N(C3CCCN(C(=O)C4=CSCS4)C3)C)=O)CCCCC1C2Br c1(C(=O)NCC2(CNC(=O)C(F)OC(F)(F)F)CCC2)sccc1Cl C(=O)(C1CC(=O)Nc2ccc(Br)cc21)N1C(C)(C)CC(O)C1 CCC(CC(=O)N(CCCNC(C1CC(F)C1)=O)C1CC1)SC Cn1nnnc1N1CC(C(=O)OC2CCN(C(=O)Nc3ccncn3)C2)C1 CC(CNC(C1CC(C)CC(=O)N1)=O)CC(=O)NOCCCCC1CC1 Cc1ccc(NC(C2CC(F)CN2C(c2csc(=N)[nH]2)=O)=O)cn1 c1(C(N2CCC(NC(C(c3cccc(Cl)c3)CC)=O)CC2)=O)cc(N)ccc1F C1(C(N(CC)Cc2ncc[nH]2)=O)C2CN(C(=O)C(C)SC)CC12 C1(C(=O)NC(C#C)C2CCC2)CCC(C2CC2)N1C(c1ncccc1F)=O c1(C(N(CC(C)NC(c2ccc(F)c(C)c2Cl)=O)C)=O)cnc2cccnc2c1 N1(C(C#C)C2CC2)CCN(C(=O)NOCc2ccccc2Cl)CC1 CC1(C(=O)NCC(O)C)CC1C(F)(F)F.C1(C=O)CCN1C1CCCC1.N c1(C(NNC(C2CCCC(C)C2)=O)=O)ccnn2ccnc12 C=CCCCC(=O)N1CC(NC(C2CCCN(CC(C)C)C2)=O)C(SC)C1 C1(C2CCN(C(C3(C)CCNC(=O)C3)=O)C2)(NC(C(C=C)O)=O)CC1 c1(C(c2nnnn2CC2CCC2)NCCSC)ccc(C)cc1Br C(=O)(CC(C)C(C)(C)C)NC(CC=C)CC(=O)Nc1ccc(C(C)C)nc1 N1(C(Cc2ccc(OCC=C)cc2)=O)CC2CC(NC(=O)CS(=O)CC)C1C2 CCC(C(=O)N1CCC(N(CC(N2CCCC2CN(C)CC)=O)C)C1)OC c1(-n2ncc(C=O)c2)ccccc1F.C=CCCCNC(C1(C(N)=O)CC1)=O.N C(C(C)C(C)C(=O)NCCC1(CNC(c2[nH]cnc2C)=O)CC1)OC c1(C(N2CCC(N(C(=O)CC3(C(F)F)CC3)C)C2)=O)cc2n(n1)CCCC2=O C=C(F)C1(CC(N2CCCCC2CCNC(C2CC2F)=O)=O)CCOCC1 N1(C(c2c(CNC(C(CCCOC)C)=O)c[nH]n2)=O)CCC2(CCSC2)C1 CCC(CC(=O)NC(CC(C)C)C(=O)NCCC(C)(C)N(C)C)C(C)C CC1OCCC1(C)C(N1CCCC1c1nc(NC(c2ncc(Cl)cn2)=O)no1)=O C1(C(N(CCCNC(C(C)C2=CCCC2)=O)C)=O)CCOCC12CCCC2 N1(C(=O)CC2CCCC(O)C2)CC2(CO)CC1(C(=O)NC)C2.c1ccc(F)cn1 CC(C)CCC(F)C(=O)NCCOC(C)(C)CNC(=O)C(C)n1ccnc1 C1(C)(NC(=O)Nc2c(C)c(C(F)(F)F)ccn2)CCC(=O)N(C)C1 c1(OC)cc(F)cc(C(N2CC(NC(=O)CC3(O)CCCN(C)C3)C2)=O)c1N C#CC1CCC(C(N2CCOCC(C(=O)NCC3CC3)C2)=O)CC1 C1(NC(C(n2ccc(C)n2)(C)C)=O)CCOCC1NC(C1(O)CCOCC1)=O C#CC1(OCCOC(C2CCC(=O)N2C(c2ccccc2)=O)=O)CCCC1 N(C(=NCCCC1CC1)NCC1(OC(F)F)CCS(=O)(=O)C1)C(C)C c1(C(=O)NCCC2CC(NC(C3CC(C)C3)=O)C2)nc2ccccn2c1F c1(C(C)NC(N2C(COC(=O)NC)CCCC2)=O)c(F)cccc1I N1(c2snc(SC)n2)CCCCC(CNC(C2CCC3CC3C2)=O)C1 C1(Nc2cc(NCc3cnc(C(F)F)s3)nc(C)n2)CCc2nnnn2CC1 c1(C(=O)NC2CC(NC(c3cnn4ccccc34)=O)C2)c[nH]c2cccnc12 Cc1cc(C(=O)NC(CNC(=O)C(O)CCN(C)C)CO)cc(F)c1 C1(c2nnnn2C(C)(C)C)(NC2CC(SC)C2)CN(Cc2ccccc2)CC1C CC(CN=c1[nH]c(=NCCc2ccccc2F)[nH]c2c1CCCC2)S(N)(=O)=O CC1CCCC(C(=O)NCCCC(=O)NC2(C(F)(F)F)CC2)C1 CCC(O)(CC)C(=O)N1CCN(C)C(c2cn(Cc3ccco3)nn2)C1 Cn1cc(C(=O)NCCOCCOCCN2CCOCC2)c2ccccc12 N1(C(CCOCC)=O)CCC(NC(=O)CCCc2cccs2)C(C)C1 Cc1cc(CCC(=O)NC(C)CN(C(=O)CC(C)C2CCCO2)C)c(C)s1 CC1CCC(NC(C2CN(CC3OCCC3C(F)(F)F)C2)=O)CC1 N1(C(c2cc(CCC)oc2C)=O)CC(NC(c2scnc2CC)=O)CC1(C)C N1(C(C(C(C)O)(F)F)=O)CC2CCCC(C1)N2C(C12CCOC1CCOC2)=O Cc1cc(C#N)ccc1C(N1CC=C(C(=O)NCC23CCCC2CCC3)C1)=O Nc1cccc(C(=O)NC2CCC(NC(=O)CN3CC4C=CC3C4)CC2)c1F CCC(C)(C)CC(=O)NC12CCC1CN(C(C1CCC1Cc1ccccc1)=O)C2 c1(C(N2C(CNC(C3(OCC)CCC3)=O)C=CC2)=O)cc(F)ccc1.N CCCCC(F)C(=O)NC(COC(C)C)C(=O)NCCC1CC=CCC1 c1(C(=O)NC2CC3CN(C(c4cc(CC)[nH]n4)=O)C2C3)c(C)nn2cccnc12 Cn1oc(C(=O)NC(C2CCCN2C(c2cc(Br)n[nH]2)=O)(C)C)cc1=O CC(CC(=O)N1CC(NC(c2cscc2C(N)=O)=O)CC(C)C1)C(F)(F)F N1(C(CCCC)=O)CCOCC1CN(C)C(C1CC(O)CN1C)=O C(C(=O)N1CC(CNC(c2cnc(S)n2C)=O)C(F)(F)C1)(C(C)(C)C)OC C12CCN(CC1)CC2.C1(C(C(=O)N(C2CCNC2)C)N(C)C)CC(C)(C)C1.C N(C1CCCc2[nH]ccc21)C(=O)NCC1(C#N)CCCO1 C#Cc1cc(C(=O)N(CC)CC2CCN2C(=O)C=CC2CCCO2)ccc1C C1(C(=O)NC2CC2C(=O)NCc2cn[nH]c2)CCCS1 C(CCC(=O)NCc1coc(CO)c1)N(C(=O)C(Cl)Cl)C C1(NC(C2C(CNC(c3c(C)ocn3)=O)CCCC2)=O)C2CCC(C2)C1C C(=O)(C1=Cc2c(ccc3ccccc23)CC1)N1CCC(N(C)CC)C1 C1CN(C(=O)CC(F)(F)F)CC(F)(F)C1.Cc1ccc(OC(C)C(=O)N)c(C)c1 CCCC(C(=O)OC)C(=O)N1CC(COC)(NC(=O)C(CCO)N(C)C)C1 c1(C(=O)NC2CN(C(c3cnc(C)[nH]3)=O)C(C)(C)C2)cc2c(s1)COCC2 CC1(C)CCCC(C(=O)NCC2(F)CN(C(=O)CCCc3cc[nH]n3)C2)CC1 CCS(=O)(=O)C1(Cc2ccc(NC(C3CCC(=O)N3C)=O)cc2)CC1 C1(CNC(CSC)=O)CN(C(=O)CC(=O)N(C)C)CC(C)(C)C1 CCC(CC)C(C)C(=O)NCC1CN(C(c2cc(O)ncc2F)=O)CC1N(C)C C(=O)(CC1=CCOCC1)N1CCCC(CC(=O)NCCC(O)C2CCC2)C1 C#CC1COCCN1C(=O)CC(CC1CC1)NC(c1cnc(C)nc1)=O C1CN(C(=O)C(C)Cc2ccco2)CC1F.C(=O)(CC1(CC(=O)N)CC1)OC N1(C(CC(CC)OC)=O)CC(CNC(c2c(OC)cccc2Cl)=O)C(C)(C)C1 N1(C(c2ccc[n+]([O-])c2)=O)CCC2CN(C(C3CCc4c[nH]nc4C3)=O)C2C1 O=C1Cc2ccc(NC(c3sccc3NC(c3ccc(Cl)c(O)c3)=O)=O)cc2N1 c1(OC)ccc(C(=O)NC2(CCCNC(C3CC4CCC4C3)=O)CC2)cc1N N1(C(C2OCCN(C(=O)C=Cc3ccncc3)C2)=O)CCCC12CCCOC2 c1(NC)nc(C)ccc1C(=O)N(CC)C(C)C.c1(C(=O)N)ncc(C)cc1 C1(C(=O)NC2C(OC)CN(C(c3cc(C#N)c[nH]3)=O)C2)CCOC(C)(C)C1 C#CCCCCCCC(=O)N1CC(C)(NC(c2cnnc(C)c2C)=O)C1 C(=O)(C(F)(F)c1cnccn1)N1CC(NC(c2coc(Cl)c2)=O)C1 C(=O)(CCC(F)(F)F)NC(C1CCCN1C(c1ccon1)=O)C N1(CCC=CCC)CCC2(CN(C(c3cn(CCC)nn3)=O)CC(C)O2)C1 N1(C(C2CC(C#N)(OC)C2)=O)CCCC(C)(NC(=O)CCc2cncs2)C1 C1(C(=O)NCC(CN(C(Cn2nc(C)c(Cl)c2)=O)C)C)CN(S(N)(=O)=O)C1 O=C1NCCC2(CN(C(=O)Nc3ccc(C(F)(F)F)cc3)C2)O1 C1(C(=O)NC2CN(C(C3SC4C=CC3CC4)=O)CC2O)CS(=O)(=O)CC12CC2 c1(C(NC(C)C)=O)ccc2nc(C)[nH]c2c1.C1(C=O)CC1C(F)(F)F.CC N1(C(=O)C=Cc2ccc([N+](=O)[O-])o2)CC2CCC1CN(C(=O)C1CC1)C2 n1(CC(N2C(CNC(CC(CC)(F)F)=O)CC(F)(F)C2)=O)nnc2ccccc12 N1(C(C2C(C)C2)=O)CC2CC(C1)CN(C(c1nocc1C(C)(C)C)=O)C2 C12(NC(c3ccc(CCCCC)o3)=O)CCC(C1)N(C(c1cncnc1)=O)C2 C12(NC(c3ccc(C)[nH]3)=O)CCCCCC1N(C(C13CCCN1CCC3)=O)CC2 CC1CN(C(=O)Cn2nc(Cl)ccc2=O)CCN(C(C2CC(=C3CCC3)C2)=O)C1 C#CCC(CC#C)C(=O)NC1CS(=O)(=O)CC1NC(=O)CC(C)(C)C(F)F CCC(C)CCCCC(=O)N1CCN(C(C2CCCC(C)(C)C2)=O)CC1 C12(NC(COC3CC(NC(=O)CC4COC(=O)C4)C3)=O)CCCCC1OCC2 Cc1c(C(=O)NC(C2CCCN2C(C2CN(C(N)=O)C2)=O)C)nn(C)c1Br S(=O)(=O)(c1ccc(NCC2CCC(F)C2)c(Br)c1)N(CCCCO)C N1(C(c2cn(C)nc2)=O)CCC2(CCOC2)C(CNC(C2OCC2(C)C)=O)C1 c1(C(N(CC(=O)N(C2CCC(F)(F)C2)C)CC#C)=O)cnn2cccc2c1 c1(OC)nc(N(C(C2CCCNC2)C)Cc2ccc3ncoc3c2)ncc1C#N C(=O)(N=S(C)(=O)c1cnn2c1CN(C(C1(Br)CC1)=O)CC2)c1c(C)sc(O)n1 C(CC(F)F)(C(=O)NC1CN2CCC1C2)NC(c1c(C)sc(O)n1)=O C12(C(=O)NC3C(C)C3)CC(NC(=O)C(O)C3CC3)(C1)C2 c1(NC(C)=O)ccc(C(=O)N)cc1.C(C)(C)C(C)C.c1(C=O)cc[n+]([O-])cc1 N1(C(C=CCN(C)CC)=O)CCC2CN(C(c3cnc(C(=O)NC)s3)=O)CC12 c1(N2CCC(C(=O)NCC)CC2)nc(=NCC2CNC(=O)C2)[nH]c2c1ncn2C C1(NC(c2c(C)nc(CO)s2)=O)COC2(CCN(C(c3ccnnc3)=O)C2)C1 Cc1ccccc1C1CN(C(c2cc(C(F)(F)F)n(-c3ccccc3)n2)=O)C1 N1(C(C2C(C=O)C=C2)=O)CCC(O)C1.c1(C=O)csc(C(F)(F)F)c1.CO C1(NC(=O)Cc2cccnc2)C2CC3CN(C(C4(C5CCCO5)CC4)=O)C1C3C2 CC(C)C(CCC(=O)NC1CC(N2CCC2)C1)NC(=O)C(CO)C(C)(C)C C1(CNC(C(C)(C)F)=O)CCCCCN1C(=O)CC(=O)Nc1nccs1 c1(CC(=O)NCC(C2C3CCC2CC3)=O)cccc(SC(F)F)c1.c1ccccc1 C#Cc1cncc(C(=O)NC2CCCCN(Cc3cnn(C)n3)C2)c1 C12(C(N(CCC)CCNC(=O)C(c3cnccn3)C)=O)COC(C)(C1)C2 C1(C)(CNC(C)=O)COCCN(C(c2cccc(C(F)(F)F)c2O)=O)C1 CCC1=NOC(CN2C(c3ccccc3)(C(=O)NCc3ccccc3)CCC2)C1 c1(C(=O)N)cc(C2CC2)ncn1.C(C(C)CO)NC(c1coc(C(F)F)n1)=O CC1(C)C(C(=O)NCC2CCC2NC(c2cnccc2Cl)=O)CC1(F)F CC1CC(C(=O)NC2CC(n3ccnn3)C2)CN(C(c2cnnc(O)c2)=O)C1 c1(C(=O)NC(CC)(C)CNC(=O)C(F)n2ccnc2)cc(F)cc2nc(S)[nH]c12 c1(C(=O)NCC2CC(OC)CN2C(=O)C)n[nH]c2c1COC2.c1cnn(C)c1 c1(OC)ccc(Br)c(C(=O)NC2CCCC(NC(c3cccn3C)=O)C2)c1 C12(NC(c3[nH]c4c(F)cc(Br)cc4c3CC(=O)O)=O)CC3CC(CC(C3)C1)C2 N(C)(C(=NCCOC)NC1CC1c1ccc(Br)cc1)CCCC(=O)NC CCCC(CC)CCC(=O)NC(CC(=O)NC1CCCC1F)C(C)CC C1(C(=O)NC(C(=O)NCC(F)Br)c2ccco2)CCCCCCC1 N1(C(CCc2n(CC)ccn2)=O)CC2CN(C(C3(O)CCSC3)=O)CCC12 C1(C(=O)NCC2(C)CCC2)CC(NC(c2ccco2)=O)C12CCC2 c1(CCCCC)nc(Cc2ncccc2F)n(-c2ccn(C3CCOCC3)n2)n1 C(=O)(C(C)(C)CS(N)(=O)=O)NC1C(NC(c2n(C)ccc2)=O)CCCC1 c1(C(=O)NCCC2CC(NC(C3(C)CCNC3=O)=O)C2)nc2ccccn2c1F CCCCC(CNC(=O)CC12COC(C)(C1)C2)NC(=O)COC(C)C Cc1nn(-c2ccccc2)c(C)c1CNCCC1CNC(=O)N1C N1(C(=O)Cn2ccnn2)CC2(CCCN2C(=O)C(F)(F)C(F)F)C1 c1(OC)cc(C(N2CCC(O)(CC)C2)=O)cc(Cl)c1.C(=O)(CC1(C)CC1)N C1(NC(C2(C)N(C(C(SC)SC)=O)CCC2)=O)CC2CC(O)C1C2 C1(C(N2C(CN(C(=O)CC3CCC3)C)CCCC2)=O)CC2(CCCC2)C1 C1(CNC(c2scc(C)c2Cl)=O)CC(F)(F)CN1C(C12CCCC1C2(F)F)=O c1(C(=O)NCCOC2CN(C(=O)C(F)F)C2)ccnn1-c1ccccc1 C1(n2cccn2)(C(=O)NC2CC(C(C)C)C2)CCN(C(=O)C(O)C(C)(C)C)CC1 c1(C(=O)NC2CSC2)cc(C(F)(F)F)ccc1F N1(C(C2C(=C)C2)=O)CC2(CC(NC(C3CCc4ccnn4C3)=O)CO2)C1 c1(OC)ccc(C(=O)NC2CC2CNC(=O)CO)nc1Cl.C1CCCO1 C(C)(C)(CC(=O)NC1CC(CCNC(C2(C)CC2)=O)C1)OC C1(N(C(C(CC=CC)C)=O)C)CC2CCC(C1)N2C(=O)Cc1c(C)cnn1C c1(CC(=O)N)cscn1.c1ccccc1.C(C(=O)NC1CC1)N(C1CCC1)C C1(O)(C(C(=O)N(CC=C)CC)F)CN(C(=O)C(O)c2ccsc2)C1 c1(C(N(CC(C)NC(C2CC(C)(C)CN2C)=O)C)=O)c(N)ccc(F)c1F C1(C2CCN(C(=O)C=CCCC=C(C)C)CC2)CC1.C(C(C)(O)CC=O)OC C1(C(C)C)CN(C(C2CNC(=O)N2)=O)CC1C(=O)NC1(C(C)(F)F)CCC1 c1(C(=O)NC2CC3(C2)CN(Cc2cc(Cl)ccc2Br)C3)cccc(Br)c1[N+](=O)[O-] Cc1cn(C)cc1C(=O)NC1CN(C(c2cnco2)=O)CC1C C1(C(N(C(CC(=O)OC)C)C)=O)CC(F)CCN1C(c1cc(C)cc(C)n1)=O C(=O)(CCCCS(=O)(=O)N1CCC(CC(=O)NCC2CCOC2)C1)OC C=CC(C)(CC)C(=O)NC1CCC(N(C)C(c2coc(SC)c2)=O)CC1 N1(C(CC)=O)CC2CC(NC(=O)CCN3CCC3)CC(C2)C1 N1(C(C(=O)Nc2ccccc2)c2cscn2)CCOc2cc(F)ccc2C1 CCCCCCn1nnnc1C(CC1CCCO1)NCCOC(C)C C1(C(N(C2CC2)Cc2cccc(OC)c2)=O)CCCC2CC(O)CCC12 c1(OC)ccc2c(C(=O)NCCCCCCC3CC3)cc(O)nc2c1 CC(C)C(C(=O)N1CCCC1)OCC(F)F.C(C(=O)NO)OC1CCCC1 Cc1ncc2n1CCC(C(=O)NC)C2.C1CN(C(=O)CC2CC(=O)C2)CC12CC2 c1(C(=O)NC(=O)NC(C(=O)NCCN(CC)CC)C)cc(C)cs1 C(=O)(C(C)(C)CCF)NC1C(C(=O)NC(c2cncs2)C)CC1 C(=O)(C(C)(C)CC(F)F)NCC(C)(C)OCC(=O)NC(CC)CO CC#CCC(C(=O)NC1CCCC2(C1)N=N2)NC(c1ccccc1O)=O c1(C(N(C)CC2CCN(C(c3[nH]cc(C)c3C)=O)C2)=O)cccn2c(O)nnc12 C1(C(=O)NC)(NC(C(CCOC)C)=O)CCC(C)(C)C1.C1(C#N)CCOCC1 Cc1cnc(C(C(=O)NCC2CCN(S(C)(=O)=O)C2)N(C)C)cn1 c1(C(N(C2CC(NC(Cc3c(C)nn(C)c3)=O)C2)C)=O)cc2cccnc2s1 N1(C(C2CCN(C(=O)NC)C2)=O)CCC(NC(C2CC2C(N)=O)=O)CC1 C1(OC)CN(C(=O)C(=O)N)CC1C(=O)NOC1COC(C2CC2)C1.CC(F)F Cc1ccc(C(=O)N(CCCCCNC(=O)C=CS(C)=O)C)c(C)c1 C1(C(=O)NCC(CCCC)NC(c2c[nH]cc(Cl)c2=O)=O)CC12CC(C)(C)C2 C1(NC(c2ccc3[nH]ccc3c2)=O)CN(C(=O)CC=C(Cl)Cl)CC1C1CC1 C1(C)(CC(=O)NC(CC)CCOC)CCN(C(=O)C(C)(CO)OC)C1 C(CC(C(=O)N(C)CCN(C)C)NC(c1ccc(C(N)=O)[nH]1)=O)SC N1(C(c2c(C)ncn2C)=O)CCC2CN(C(c3ncccc3C(F)F)=O)CC2C1 C(=O)(C(F)CCC(C)C)NCCCN1CCC(NC(C2N(C(C)=O)CCC2)=O)C1 N1(C(=O)OC(C)(C)C)CCCCC(CNC(=O)NC2CC3C(O)CC3O2)C1 N1(C(CCCOC(C)C)=O)CC(C)C(F)(F)C1.c1(C(=O)N)cc(C2CC2)cs1 c1(OC)c(C(N2CCCN(C(c3sc(F)cc3C)=O)CC2)=O)cccc1F c1(C(=O)OC(C)C(Cl)(Cl)Cl)ccc2c(c1)NCCS2 CC1Cc2c(Cl)cccc2C1Nc1nccc(=NCCc2ccn(C)n2)[nH]1 Cc1cc(C(=O)NC2CCCCC2NC(=O)CCC(=O)Nc2nccs2)c(C)s1 C1(C(N2CC3C(CNC(C4OCCN(C)C4)=O)C3C2)=O)CCCCC12CC2 N1(C(Cc2cc(C)oc2C)=O)CC2CC1CN2C(c1ccsc1-n1cnnn1)=O c1cc(C)c(C)cc1Cl.c1(NC(COCCOC)=O)cccc(F)c1C(=O)N C(C)(C1Cc2ccccc21)NCC1N(C(=O)OCC)CC1 S(=O)(=O)(c1ccncc1)N1CC(C(=O)Nc2cccc(O)n2)C1 N1(C(CC(C(C)OC)NC(C2CCCCCCC2)=O)=O)CCn2c(O)nnc2C1 N1(CC2C(CS(C)(=O)=O)C2)CCC2(NC(=O)CCCc3cccs3)CCCC12 Cc1csc2nc(CC(N3CCC4(C3)CN(C(C3CC(O)C3)=O)C4)=O)cn12 c1(NC(CCC2CC(NC(C(CC#C)O)=O)C2)=O)c(C)cc(C)nc1C C1(CC)(NC(=O)C(C)O)CCN(C(c2cc(F)ccc2Br)=O)CC1 Cc1ccncc1C=CC(N1CCC(NC(=O)COC2(C)CCCC2)CC1C)=O c1(C(N(CC(C)NC(CC(C)C2CCCO2)=O)C)=O)cc([N+](=O)[O-])cnc1N c1(CC(N2CCCC(N(CC(CC)OC)C)C2)=O)c(C)nc2ccccn12 N1(C(c2cc(CC)ncc2)=O)CCC2(CCCN2C(=O)C=Cc2csc(C)n2)C1 CCC(CNC(C1CC=CCC1NC(c1ncccc1O)=O)=O)CC(C)C N1(C(c2n(C)c(Cl)nc2)=O)CC(C2CN(C(=O)CN3CCc4sccc4C3)C2)C1 c1(C(N2CCCC(CCNC(c3ccnc(Br)c3)=O)C2)=O)cc(F)c(Cl)c(Cl)c1 c1(NC(CCSCC)=O)cccc(CN(C(=O)CCCOCCOC)C)c1 CC1CCC(NC(=O)Cn2cc(-c3cccc(C(C)N(C)C)c3)nn2)CS1(=O)=O C1(N(C(C2C(C#C)C2)=O)C)CCCN(C(C2(C(C)(C)C)CCC2)=O)C1 N1(C(COCCOCC#C)=O)CCC(C(C)NC(c2cc(C)on2)=O)C1 C1(CC)(NC(=O)C(O)C2CC2)CCN(C(=O)C(CCCO)c2ccccc2)CC1 N1(C(CCC=C)=O)CCC(C(=O)NC(CCF)C(=O)OC)CC1CC N1(CC(=O)N(C(C)CCNC(c2ccnn2C2CC2)=O)C)CCCCCCC1=O C1(C(=O)NCc2cc(OC)cc(C(F)(F)F)c2)CCOCC12CCC2 Cc1ccc(C(C)C(=O)N(C2CCCCC2)CCNC(c2ccn(C)c2)=O)s1 n1(CCC(=O)NC2C(NC(c3c(CC)n[nH]c3)=O)CCC2)ccc(O)nc1=O C=C(C)CC(C)C(=O)NCC1CC1NC(c1ccc(OCC)c(C)c1)=O C1(NC(c2nccc(C)n2)=O)CC2CC(NC(=O)CCc3ncc(C)[nH]3)CC12 C(=O)(C(CC(C)C)ONC(=O)COCCO)N1CC(C(=O)NCC)C1.C c1(OC)ccccc1C(F)(F)C(=O)N.C(=O)(C1=NOCC1)N(CCC)C(C)C C1(NC2(c3n(CCSC)nnn3)CC(C)(CO)C2)CC(C2CCC2)C1 c1(C(N(CC(C)C)C)=O)cc(F)c(F)c(F)c1N.C(=O)C(F)(F)c1cncs1.N C1(NC(C(COC)COC)=O)C2COCC1CN(C(=O)C#CC1CCCOC1)C2 C(=O)(C(CC(C)(C)C)OC)N(CC(=O)N(C(CCC)C)C)CCC c1(OC)c(NC(C2(O)CCN(C(=O)Cc3cc(Br)cs3)C2)=O)cc(Br)cc1F CS(=O)(=O)c1ccc(C(=O)N)[nH]1.C1(C=O)(C2CC2)CCCO1.CCC1CC1 C1(C2CC2)(CNC(CC2(C)CC2)=O)CCN(C(C2CCCCC2(F)F)=O)C1 C1(CCCC)CCC(NC(=O)C(=O)NC2CCOC2C2CC2)C1 C1(O)(CC)CCCN(C(C2(NC(c3ncc[nH]3)=O)CSC2)=O)C1 C1(c2n(C)ncc2)CN(C(=NCCc2cnccn2)NCC2CCCO2)CCO1 c1(C(N2CCC(NC(C3C(OC)CCC3)=O)C2C)=O)cc(C)cc(Cl)c1N C1(CNC(Cn2c(=N)scc2)=O)CC2CCC1N2C(C1COC2COCC12)=O n1(CC(N2C(CNC(C3CC34CC(O)C4)=O)CC2)=O)ccc(O)nc1=O C1(NC(CC2CCC(C(C)C)CC2)=O)COCCN(C(C2(C(N)=O)CC2)=O)C1 c1(CC(=O)NCC(CC)NC(=O)C(c2ccc(Cl)nc2)(F)F)cnccc1Cl N1(C(c2nnc(C)s2)=O)CCCOC(CNC(c2occ3c2CCC3)=O)C1 Cc1c(Cl)c(C(=O)NCCN(CC(C)O)C(c2ccc(Cl)[nH]2)=O)nn1C C=CC1(CC(N2CCCOC(CNC(c3cnnc(Cl)c3)=O)C2)=O)CCOCC1 c1(OC)ccc(C)c(C(N2CCN(C(=O)C(c3c(C)n[nH]c3C)C)CC2C)=O)n1 c1(C(=O)NC2CCC(NC(Cc3ncc(C)[nH]3)=O)C2)ccc2c(c1)nc(O)n2C Cn1cnc2cc(-c3cccc(C(CC(=O)O)Nc4ncccn4)c3)ccc12 c1(OC)ccc(Br)cc1C(N1CC(OC)CC1C(N1CCOC2CC12)=O)=O N1(CC)CCC(NC2=NCCc3cnc(OC)cc3N2)CC1C.CCCOC c1(SCc2ncc(C(F)F)cc2Br)nc2c(s1)COCC2 CN1CC2(CN(C(C3CN(C(=O)Cc4ccc(Cl)cc4)CCC3O)=O)C2)C1 C1(CC=C)(NC(c2ccccc2Cl)=O)CCN(C(=O)C(C)(C)O)C1 c1(C(=O)NCC(CN(C(Cn2c(C)nc(C)n2)=O)C)O)ccc(C2CC2)nc1O Cc1cccc(C(=O)NC(CC2CC2)C(=O)NCC23CCC(CC2)C3)c1 n1(CC)nc(C)c(C(=O)NC)c1C.C1CN(C(=O)CCCn2cncn2)C2CC12 C[Si](C)(C)c1cc(C(=O)NC23CCC(CC2)C3)co1.C1(C#N)(C(=O)N)CC1 c1(N(C)CC2CCN(C(c3cc(Br)c[nH]3)=O)C2)ccnc(C(F)(F)F)n1 c1(C(=O)NC2(CC=C)CCN(C(C3(N(C)C)CCC3)=O)C2)cc2cccnc2s1 c1(C(N2CC=CC(NC(C3CCC(OC)CC3)=O)C2)=O)c(C)cncc1F CN1C(=O)CSC1=CC(=O)N1CCOCC(CNC(C2CC2C(F)F)=O)C1 c1(C(COC(C2(Br)C(C)C2C)=O)=O)cnc(O)n(C)c1=O N1(C(C(CCC)OC)=O)CC(CO)C2(C1)CN(C(C13CCC(C)(CC1)CO3)=O)C2 C(=O)(C1Cc2ccc(Cl)cc21)NCC1C(NC(c2cccc3c2OCO3)=O)C1 O=C1NCCc2c(NC(C34CC(C(N5CCCC5CO)=O)(C3)C4)=O)cccc21 CC1CCN(C(C2CCCCCC2(F)F)=O)CC12CCC2 c1(NCCC2CC(C)OCC2)ccc(S(=O)(=O)NCC(C)(C)CCO)c(Br)c1 C1(NC(C(n2ccc(C)n2)C)=O)CCOC(C(=O)NC2(CC(N)=O)CCC2)C1 C(=O)(CC=C(Cl)Cl)N1CC(C(N)=O)(CNC(C2(C)CC2)=O)C1 CC1(C)CC(C#N)(CNC(C2C3CC2N(C(=O)Cc2ccc[nH]2)C3)=O)C1 C(=O)(CCCC(C)(C)C#N)N1C(C(N2C(C)CC2(C)C)=O)CC(O)CC1 C1(CNC(=O)C2=CCCS2)CC2(CCC2)CN1C(c1n[nH]c2ccccc12)=O c1(NC(c2cc(C)ncc2)=O)ccc(=NCc2ccc(Cl)cc2Br)[nH]c1 c1(C(=O)NCC(CSC)OC)ccc(C(N2CCCCC2)=O)cc1 C1(C(=O)NC(C(=O)NCC)CC)C(C)CCN1C(C1COC(=O)N1)=O O=C(NNS(=O)(=O)N1CC2CCC1C2)c1cc(Br)ccn1 c1(C(=O)NC2(C)CCC2)ccc(O)c(Br)c1.c1(C2(C=O)CC2)cccs1.N C1(C)CCCCC1C(N1CCC(O)(C(N)=O)CC1)=O.c1(CC)cc(C=O)n[nH]1.N c1(C(=O)N)cnc([N+](=O)[O-])n1C.CC1CN(C(=O)CC2(O)CCC2)CC(CC)O1 CC1(C)CN(C(=O)CCCn2cccn2)CC1NC(c1ccc(C#N)s1)=O N1(C(=O)C=CCO)CCCC2C1CCCN2C(=O)Cn1cnc(C(F)(F)F)n1 CC1(C)CN(C(C23COC(CCO2)C3)=O)CC1NC(=O)Cn1ccc(=N)[nH]1 c1(OC)ccc(S(=O)(=O)NCCC2CC=CCC2)cc1[N+](=O)[O-] N1(C(C2(O)CC(C)(C)C2)=O)CCC2(CO)CN(C(=O)C=CC=C(Cl)Cl)CC2C1 N1(C(C(C)C2CC2)=O)CCN(C(c2c(O)cncc2F)=O)CC1c1cn[nH]c1 c1(CNC(N2CCCC(NS(CC)(=O)=O)C2)=O)ccc2[nH]c(C)cc(=O)c2c1 C1(NC(c2ccncc2-c2ccccc2)=O)CCCCNC1=O c1(C(=O)NC(C)CN(C)C(C2CC(N3CC(O)C3)C2)=O)c(Cl)cnn1C Cc1cnccc1C(C)C(=O)NCC1CCN(C(c2cn(C)cn2)=O)C1 CN1CCC2CCN(C(=O)C(Cc3cn[nH]c3)NC(=O)CCc3ccsc3)C2C1 Cc1cc(=NCc2ccn(C(F)F)n2)[nH]cc1S(=O)(=O)N1CCCC1CC(C)O N(C1CCOc2c(Cl)cccc21)c1cc(NC2CC(O)C2)ncn1 c1(CCN(C(=O)C(C)C2CC2)C)cnn(C)c1.C(c1ccsc1)=CC(=O)N C1(NC(Cc2c(C)nc(-c3cc[nH]n3)s2)=O)CCN(C(=O)CNC=O)C12CCC2 N1(C(Cc2c(C)scc2)=O)CCC2CCC(C1)N2C(=O)C=Cc1nnn(C)n1 c1(C(=O)NCCC(C)N(C(=O)CC2CC2)C)cnc(S)nc1 n1(C(C(C)C)C)nc(COc2ccccc2)nc1-c1cc(O)nn1C C(=O)(CCCCC#N)NC(C1CCCN(C(C2(CCCC)CC2)=O)C1)C Cc1ccc(S(C)(=O)=O)cc1C(=O)NCC1CCCN1C(C1CC1C)=O C=C(C)CCC(=O)N1CC(n2cc(-c3ccnc(C)c3)nn2)C(SC)C1 Cc1cccc(C)c1NC(=O)C(N1CCCC(C)CC1)c1ccccc1 CCCC(C(N)=O)NC(=O)C(C1CN(C(c2cc(C)sc2C)=O)C1)OC N1(C(CCSC)=O)CCOC(C(=O)NC(C)CCN(C)C)C1 C#CCCCCCCC(=O)NC1(CN2CCN(C(c3ccsc3)=O)CC2)CC1 Cc1cccc(OCCC(=O)NCC(O)CNC(c2ccns2)=O)c1 c1(CC(C)C)ccc(CCCC(=O)NCC2CC2)cc1.C(=O)C(C)=C1CCC1 N1(C(CN(C(=O)CC(F)(F)F)CC#C)=O)CCn2cncc2C1 c1(C(N2C(CN(C(=O)C3=CCCSC3)C)CC(F)C2)=O)cccc2c1OCCC2 c1(C(N(C2CC(NC(c3c(SC)cn(C)n3)=O)C2)C)=O)c[nH]cc(C)c1=O C(Cc1ccsc1)(C(=O)NC1CCOC1)N(C)Cc1c[nH]nn1.C1COCCO1.C N1(C(CCCOC)=O)CCN(C(C2CCS(=O)(=O)N2)=O)CC(C)(F)C1 C1(NC(=O)CCC2CCCCC2)CCN(C(c2ccc(CO)c(F)c2)=O)CC1O CN=c1[nH]ccc(C(=O)NCC(F)CNC(C2(F)CC2)=O)c1[N+](=O)[O-] C12(C(=O)OC)CCCC1C2.C(=O)CCCSCCO.CC.CC.C(N)=O N1(C(C(C=CC)O)=O)CC2CCCC(N(C(=O)C(F)OC)C)C2C1 N1(C(CC(C)(C)O)=O)CCCCCC1CNC(=O)Cc1c(O)ncnc1O Cc1cc(Br)c2oc(C(N3CC(CNC(=O)COC(F)F)C3)=O)cc2c1 C1(C(N2CCC3(CN(C(=O)C4CC4)C3)C2)=O)CC2(CCCCC2)S1(=O)=O C(=O)(CS(=O)(=O)Cc1ccccn1)N1CCC(CC(=O)NCC2CCOC2)CC1 N1(CC)CCC(NC(=O)CN(CC(C)C)C(c2cnn(C)c2C)=O)C1=O c1(NC(=O)CC2CCCN2Cc2cccc(OC(F)(F)F)c2)cc(I)ccc1F c1(C(N2CCC(O)(C(=O)NCC3CCCCO3)C2)=O)cnc(O)c(Cl)c1 c1(C=O)cc(C#N)ccc1C.C1(F)(CNC(C(C)SCCCC)=O)CCC1.C C1(NC(c2c(CC)nns2)=O)CC2(C1)CC(C)C2.C1(C(=O)N)CCCOC1 [N-]=[N+]=NC1CCC2(C(N3CCCC(NC(=O)C4=CCCOCC4)C3)=O)CC12 C1(CC(=O)NC(CN(C)C)CO)CN(C(=O)CSCC(F)F)C(C)(C)C1 N1(C(CCC(=O)NCC)=O)CCOC2CN(C(=O)CC3(O)CCCCC3)CC12 C1(C(=O)NCC(=C)CC)COCCN(C(C2(C)CCNC2=O)=O)C1 CC(C)CC(O)CC(=O)NCC1CC(C)(C)CN1C(c1ncoc1C1CC1)=O C(=O)(C(C)(C)C(=O)NC1CCC(N(C(=O)C)C)C1)NC.c1ccc(F)cc1F C1(C(N(C(CC)COC)C)=O)COCCN(C(C2CSCC(=O)N2)=O)C1 CC(C)CCC(C(=O)NCC1OCCCC1(C)C)NC(c1cnccn1)=O Cc1cc(C)c(C(N2CC3CSCC3(C)C2)C(=O)NCc2ccccc2)c(C)c1 N(C(=NCC1CCN(CC2CCCC2)C1)NC1CCOCC1)C(C)C N1(CCC)CCCCC1C(N1CCCC(NC(C)=O)C1)=O.c12cn(nn1)CCC2 N1(C(=O)CC(F)(F)F)CCCC2(CCN(Cc3coc(-c4ccccc4)n3)C2)C1 N1(C(CCc2nc(=N)[nH][nH]2)=O)CCC(CNC(c2ccc(F)cc2Cl)=O)C12CC2 C(=O)(C1=CCCCC1C)NC(C(C)C)CC(=O)NC1CN(C(C)C)C1 c1(C(=O)N)cc2c([nH]1)CCCC2=O.N1(C(CSCCOC)=O)CC(C)CCC1C C1COC2(C1)CN(C(=O)C(C)=C(C)C)C2.c1(OC)ccc(F)c(CC(=O)N)c1 c1(CC)cc(C(=O)NCCC2CCCN2C(=O)CCc2nncnc2O)n(C)n1 CCC(C(=O)N(C(C)C(=O)NC1CCC1C)CC)N(C)C Cc1ccc(Cl)c(OC(C)C(=O)NC(CO)CC)c1.C(=O)(CCc1cscn1)N CC1(C)CC(NC(=O)C(N)C[Si](C)(C)C)c2ccccc21 C1(CNC(C(C)CC2CC2)=O)C2CN(C(=O)CN(C)CCO)CC12 C(=O)(CS(N)(=O)=O)NCC(CC)(C)NC(c1cccc(CS(C)=O)c1)=O C1(C(=O)NC2CC2C)(CC)CCCC1.C1(C=O)CC(C(F)(F)F)C1.N CCC(C)(C)CC(=O)N(C1CN(C(=O)CN2CSCC2=O)CC1(C)C)C c1(C(N2C3CC(CNC(C45CC(C)(C4)C5)=O)C2CC3)=O)ccn2ccnc2c1 C(=O)(C1=CCCOCC1)N1C(CNC(c2ncccc2F)=O)C(O)C(O)C1 C=CCCCC(C(=O)NCC1(F)CC(O)C1)NC(c1ccc(C=C)cc1)=O CC1(C)C(CNC(c2ccc(F)s2)=O)CCN1C(=O)C=O.CC(F)(F)F.N C1(NC(CC(C=C)(C)C)=O)CCN(C(c2cnc(C)c(N)c2)=O)CCC1CO C1(C(N2CC(n3cc(CCSC)nn3)C(C)C2)=O)CC2CC1CC2(F)F C1(CNC(CCCCC=C)=O)CN(C(c2ccc(CO)nc2)=O)CC(C)(C)C1 N1(C(C)=O)CCCCC1CC(=O)NCC(C)N(C(=O)CCc1cccs1)C CC#CCC(C(=O)N1CCCCC1CF)NC(=O)C(C(C)OC)N(C)C C(=O)(CS(=O)(=O)C1CC1)NCC12C(CN(C(Cc3cn(CC)nn3)=O)C1)C2 N1(C(CC(=C)Br)=O)CCCCC(CNC(=O)CCCOCC)C1 C1(C(=O)NCCSCC(=O)NC(C=C)C2CC2)CC(O)C1 N1(C(C(F)=C(C)C)=O)CC(NC(=O)C(C)(C)CO)C(C2CC2)C1 N1(C(C(C)NC(CC)=O)=O)CCN(C)C(C(=O)N(CC(C2CCCC2)O)C)C1 C1(OC)CCN(C(c2c(C)coc2C)=O)C1.C1(C=O)(C(F)F)CC(F)(F)C1.C CC(C(=O)NOCC1(C)CC1)N(C)C(C1CC=CCC1C)=O c1(C(=O)NCC(CC)NC(=O)Cc2cc(OC)ccc2Cl)cccc2ccoc12 Cc1cc(C#N)c(O)nc1C(=O)Nc1cc(C2CCCCC2)ccc1O C1(C(N(C)CCNC(c2ccc(N(C)C)cc2)=O)=O)CCCCC(F)(F)C1 C1(NC(c2ccc(C)n2C)=O)CC2(C1)CC(NC(C1CC1C1(C)COC1)=O)C2 C1(CNC(C2CC2F)=O)CN(C(C2(c3cccc(F)c3)CCC2)=O)CC12CC2 C12(NC(C=Cc3c(C)ncs3)=O)CCCC1N(C(C1(C)CCOCC1)=O)CC2 CCC(C)C(C(=O)NCCCc1ccnn1C)NC(=O)C(C)c1ccsc1 C=CCC(CNC(=O)CC1CCSC1)C(=O)N(C)Cc1nc(=O)o[nH]1 N1(C(CN(C)C)=O)C(C(=O)NCc2cn(C)nn2)CCC12CC2 C=CC(CC)CC(=O)NC1(CC2CCN(C(C)C(=O)N)CC2)CC1.c1ccccc1 c1(CC(=O)Nc2c(C(=O)OC)n[nH]c2)csc(S(N)(=O)=O)c1 C12(C(=O)NCC3N(C(C=CCCC)=O)CC3)COC(CF)(C1)C2 c1(C(=O)NCCN(C(=O)C(C)SC)CCC)ccc2nc(S)[nH]c2c1 c1(OC)ncc(Cl)cc1NC(C1(F)CCN(C(C2(O)CC2)=O)C1)=O N1(C(c2cccc(SC)c2)C(=O)NCCCC(=O)OCC)CCCC(O)C1C CC1CC(=O)Nc2ccc(C(N3CCCCC3C(F)F)=O)cc2N1 CC1(NC(=O)CSc2ncccn2)CCCN(C(=O)CC2CCNC2=O)C1 C(=O)(CCCCCF)NCC(C)(C)NC(C1N(C(=O)OCC)CSC1)=O C=C=C(C)CC(=O)NCC1CCOC1C(N1CCC(C(C)(C)C)C1)=O CCCC(CCC)C(C)Nc1ccc(N=[N+]=[N-])cc1 C=CCC(C(=O)N1CCCC(NC(c2cccc3nccn23)=O)CC1)C(C)C C(=O)(C1c2c[nH]nc2CN1C(c1cc(N)cc(F)c1)=O)NCC(CC(C)C)O N1(C(CC2C(C)CCO2)=O)CC(F)(F)CC1C.c1(C=O)cn(CC(N)=O)nn1.N N1(C(C(C)n2ccnc2)=O)CCCCC(CCC(=O)NC2(CCO)CCCC2)C1 Cn1cc(I)cc1C(N1CCCCC1c1ccccc1)C(=O)NC1CCCCC1 C12(NC(c3ccoc3Cl)=O)CCCCCC1N(C(=O)CN1CCC(F)CC1)CC2 N1(C(c2ccc(C)[nH]2)=O)CCCC(C2(NC(c3ccc(Cl)cc3)=O)CC2)C1 Cc1cc(C2(C(=O)NC(C)C(O)C(F)(F)F)CC2)cc(C)c1 N1(C(C2CCCCC2(F)F)=O)CCC2CN(Cc3ccc(C(F)(F)F)nc3)CC12 C(=O)(CCC(C)(C)[N+](=O)[O-])N1CC(CC)C(C(=O)NC2(C(F)F)CCCC2)C1 CCCCC(CC)CC(=O)N1CCn2c(CNC(=O)C3=CCOC3)nnc2C1 C1(NC(C(CC)NC(N)=O)=O)CCN(C(c2cccc(C(=O)OC)n2)=O)CC1O C1(C)(CC)CN(C(=O)CN(C(C2CC2(F)Cl)=O)C2CC2)CCO1 N1(C(C(=O)NCC(C)C)c2cnsc2)CC=CCC12CCCC2 C1(O)(C(N2CC(CN(C)C)OCC2)=O)CCN(C(c2cnco2)=O)CC1 c1(C(=O)NCC2(OC)CCN(C(C=CC)=O)C2)c(Cl)ccc(C)c1O n1(C(C)C)ncc(C(=O)NCCCN(C(=O)CSc2ccncc2)C)c1Cl CC(C)C(C)(O)C(=O)NC1C2CN(C(C3(C(F)F)CCCC3)=O)CC12 C1(CNC(c2cnc(C(C)O)s2)=O)CCCN(C(C2(F)CCCC2)=O)CC1 C(CNC(C1(C)CC(F)C1)=O)(CC(=O)NC1CC(F)(F)C1)OC c1cccc(C)c1Cl.N1(C)CCC(N2CC(C3CC(NC(=O)NCC)C3)C2)CC1 c1(C(=O)NC2CN(C(CC(=C=C)C)=O)CC2(C)C)cc2c(C)ccc(C)c2[nH]1 CC1(NC(=O)C(O)CN2CCCC2)CCN(C(c2nnn(C(C)(C)C)n2)=O)C1 Cc1ccc(C2CC2)c(C(N2CCC(NC(C34CCC3C4)=O)C2)=O)c1 CCCCCC(CC)C(=O)N1CCN(C(c2c(Cl)c(CC)nn2C)=O)CC1C1CC1 C(=O)(CCCCCCSC)NCC(CC)NC(=O)CC(N1CCCCC1=O)C CC(C)(C)CC(O)C(=O)NC.C1(F)(C(N2CCC(C)C2)=O)CCS(=O)(=O)C1 c1(C(N2C(CNC(C(C)C)=O)CCCC2)=O)ccc2c(c1)NCCC2=O C1(CNC(c2cn(CCC)nn2)=O)C2CC1N(C(=O)Cc1nocc1C)C2 N1(S(CC)(=O)=O)CCN(C(=O)N(C2(C)CC3CC3C2)C)C(C)C1 N1(C(c2c(CC)cncc2)=O)CC2(C)CC1(C(=O)N(C(C)C(F)F)C)C2 c1(C(=O)NC(C)CCCCNC(C2CCC(O)CN2C)=O)cnn2c1OCCC2 C1(CNC(c2c(C)con2)=O)CN(C(=O)Cc2n[nH]cc2Br)CC(C)(C)O1 C1(C(N2C3CN(C(c4ccc(C#N)o4)=O)C(C3)C2)=O)CCc2nncn2CC1 N1(Cc2ccc(C)o2)CCN(C(c2nccnc2Cl)=O)C2CC12 N1(c2ccc(C(=O)OC)c(C)n2)C2CCC1C(C)C(NC(=O)CC(C)C(F)F)C2 C(=O)(CC(C)CC(C)C)NC1C2(CN(C(c3ncc(NC)nc3)=O)C2)CC1 c1(-c2c(OC)c(C)ccc2)cccc2nc(C(=O)Nc3cnc(C)c(Br)c3)cn12 C(=O)(NNc1cccnn1)C1C(OC)CCC1.c12ccc(C(F)(F)F)cc1C2 N1(C(c2c(C)nco2)=O)CCN(C(=O)Cc2csnn2)CC1C(C)C C(C(CNC(c1ccc(Cl)o1)=O)CO)NC(c1ccsc1)=O CC1OC2(CO)CC1(C(=O)NC1CCN(C(C3CC3(F)F)=O)CC1F)C2 c1(OC)cccc(C2CCCN(C(=O)NCc3cc(C(N)=O)ccc3F)C2)c1F C1(C(=O)N)CCC2CC2CC1.O=C1CCCC(C(=O)NCc2ccccc2C)O1 C(C(CC(F)(F)F)NC(=O)COCc1ncnn1C)NC(CCCC)=O c1(C(=O)N)cnc(O)n(C)c1=O.CCS(=O)(=O)CC(=O)NCCCN1CCCC1 c1(C(=O)NCC2(C)CCCN2C(=O)CCS(C)(=O)=O)cncc([N+](=O)[O-])c1 Cc1c(Cl)ccnc1C(=O)NCCC1(O)CCCN(C(=O)CC(C)(C)C)C1 NS(=O)(=O)c1ccc(C(=O)N(CC)CC)s1.C1(C=O)CC(n2cnnc2)C1 C(C)(CCCC(=O)N1CC(c2ncccn2)C1)NC(CSC)=O NS(=O)(=O)c1scnc1C(=O)NCC1CCN1C(c1cnc2[nH]nnc2c1)=O CCCC(C(=O)N1CC(c2ccccc2)(NC(C2CCOC(C)C2)=O)C1)OCC C1(N)(C(=O)NC2CCN(c3cc(C)[nH]n3)CC2)CCC(C)(C)C1 N1(C(C2C(C(=O)OCC)C2)=O)CCCC1CCNC(=O)CC1CC1 C1(NC(C(C(=O)NC)(C)C)=O)CC2CCC1C(NC(=O)C)C2.c1cccnc1 c1(CNC(CCN(C(CCN(CC)CC)=O)C)=O)cc(C)ncn1 C(CC(=O)N(C(C)CN(C(=O)C=Cc1c(C)noc1C)C)C)C(F)(F)F.CO c1(C(N(CCNC(c2c[nH]nc2Br)=O)CC)=O)cc2ncn(C)c2cn1 c1(CCC)nc(C)c(C(=O)NCc2ccc(C)cc2)o1.C1(C=O)CCCO1.N C(C(=O)N1CC(C(N)=O)(CNC(c2ccccc2O)=O)C1)(C(C)(C)C)OC N1(C(CCOC(C)=O)=O)CCC2CC(NC(c3cnc(C)n3C)=O)CCC2C1 C1(CCC)CN(C(C2CCC(C)O2)=O)CC1NC(C12CC(F)(C1)C2)=O N1(C(c2cc(CC)on2)=O)CC(C)N(C(=O)COCC(=O)OC)CC1C N1(C(C(C2(O)CN(C(C3C(C=O)C3)=O)C2)F)=O)CCC2(CCC2)C1.CC.O C1(NC(=O)CC(O)C2CCCC2)CCCC(NC(=O)C(F)(F)c2ncccn2)C1 CC1Oc2ccccc2N(CC(=O)N(C(C)CNC(=O)Cc2ccns2)C)C1=O N1(C(C(C=C)(C)CC)=O)CC2(C1)CN(C(C1CC(C)CC(C)C1)=O)CCO2 C1(C2(C)CC2)CCS(=O)(=O)C1.n1(C)nnnc1Cc1nc[nH]n1.C1CCOCC1 C1(O)(c2cn(C(C)CNC(=O)CC3COC(=O)N3)nn2)COC(C)(C)OC1 C(CC)(CCC(=O)NC1C=CC(C(=O)OC)C1)NC(c1c(CC)n(C)nc1)=O CC1CN(C(c2cnc(O)n2C)=O)CC2(CCN(C(=O)C(O)C3CCC3)CC2)O1 C=CC1(CC(=O)NC2CCN(C(c3c(C)cccc3Cl)=O)CC2O)CCCCC1 c1(C(=O)NCc2nnc(CC(=O)O)s2)cc(C(F)(F)F)c(Br)s1 c1(NC(C2CCN(C(Cc3c(OC)cccc3)=O)C2)=O)ccc(Br)cc1Br Cn1ncc(S(N)(=O)=O)c1CNCc1ccc(C(C)(C)O)cc1 N1(C(C=NOC)=O)CCCCC1C1CCCN(C(=O)C(C2CCCC2)OC)C1 C=C1c2ccccc2C(=O)N1CC(N1CCN(C(=O)CCC=CC)C2CC12)=O Cc1ccc(C(=O)O)cc1CN1CCOC(C(=O)Nc2onc(C)c2Cl)C1 c1(CC(N2CC(C)(NC(CNC(=O)OC)=O)C2)=O)cc(OC)ccc1.O C(C)(CC(=O)NC(C)CC1CN(C(c2cc(CC3CC3)on2)=O)C1)SC C1(C(=O)N)CC2CCC(C1)C2O.CC(C)(C)C(C(=O)NC(C)(C)C)C1CCC1 C(C(F)(F)C(F)F)N1CC(n2ccnn2)C1.C1(CCOC)(C(=O)NC)CC1 c1(C(=O)NCC2CCCN2C(C23CCCN(CC2)C3)=O)coc2ccccc12 C1(CN(C(=O)Cn2ncnn2)C)CC(F)CN1C(c1cncn1C)=O C1(C(=O)NC2CCC2C)(NC(Cc2ccn(CC)n2)=O)CC(F)(F)C1 C1(CCC(=O)N(C)CC2(NC(C(C)NC(C)=O)=O)CC2)CCCOC1 C1(O)(C(CNC(CC(=O)OC)=O)C)CCN(C(c2ccccn2)=O)C1.C(CF)O Cc1ccc(Cl)c(CC(=O)NCCC2(C)CCCO2)c1 c1(CN(C2CN(C3COC3)C2)C(c2[nH]nnc2C2CC2)=O)ccccc1Br N1(C(C(C=C)C)=O)CCC(C)(C)C(NC(=O)CCc2cccc(O)n2)C1 CC#CCC(C(=O)NCC(O)CC(=O)OCC)NC(c1ccc(CC#N)cc1)=O S(=O)(=O)(c1cccc(NC(=O)C(N2CCCC(F)(CO)C2)=O)c1C)NC N=c1[nH]cc2c(c1C(=O)NCC1CCCN(C(=O)C(F)(F)C3CC3)C1)CCC2 c1(C(N2CC(CN=[N+]=[N-])C2)=O)cnc(CNC(=O)C(F)C2CCOC2)nc1 c1(NC(C(c2n(CC)nc(C)c2)N2CCCOCC2)=O)ccc2c(c1)OCCO2 Cc1cc(O)nc(C)c1C(=O)NCC1CCN(C(c2c[nH]c(=S)cn2)=O)C1 Cn1nc(C(=O)NCCOCCOCC)c2c1CCOC2.C1(C=O)CCCS1 C1(CNC(C(C#C)(C)C)=O)CCC2(CN(C(c3c(C)oc(C)c3Br)=O)C2)O1 c1(NC(CC(n2c(C)cc(C)n2)C)=O)ccc(Cl)cc1-n1cccn1 C1(C2N(Cc3cnc(C)s3)CCC2)CCCN(C(=O)CSc2ccc(O)nc2)C1 Cc1ccc(C)c(C(N2CC(NC(C34CC3CCC4(F)F)=O)C2)=O)c1N C(CCC(C)(C)NC(c1ccc(-c2cn[nH]c2)cn1)=O)NC(CSCC=C)=O N1(C(C(CC)CC)=O)CCC2CCCN(C(=O)C=CCOCCOC)C2C1 C1(NC(C(N(C(CC(C)CN(C)C)=O)C)C2CC2)=O)CCCC1N=[N+]=[N-] N1(C(c2nccc(C)n2)=O)CC2CC1CCN2C(c1nn(C)c(Br)c1C)=O C(CN=c1nc2scnc2c[nH]1)(C1CC(C)(C)C1)OC CC1(C)CN(C(=O)C2=NNC(=O)C2)CCC1NC(c1ccn(C2CCC2)n1)=O c1(CC)cccnc1C(=O)NC1C2CC1N(C(c1ccnc(C)n1)=O)C2 Cc1c(C(=O)NCC(C(C)(C)C)NC(c2cccnc2OC(F)F)=O)nnn1C C(=O)(C(C)CC1CC1)NCC(C)OCC#C.c1(C=O)cc(C)c(C)[nH]1 O=C(C1=CS(=O)CCC1)NCC1=CCN(C(c2ccc(C3CC3)o2)=O)CC1 N#Cc1ccc(C(=O)NC(Cc2cn[nH]c2)C(=O)NCC2CCC=CCCC2)cc1 C1(CNC(C(CC#C)O)=O)CCN(C(=O)C(C)(C)CC)CC1C1CC1 c1(N(C)C)cc(C(=O)NCC(C2CCN(C(C3(O)CCC3)=O)CC2)(C)C)ccn1 C1(C(=O)NC(C)C(=O)N(CCCN2CCCC2)C)CC2(CC(=O)C2)C1 c1(C(CNC(CN(C(COCCCC#C)=O)CC(C)C)=O)O)cnn(C)c1 c1(CC(=O)NCC2CC(NC(c3cccnn3)=O)C2)csc2cccc(F)c12 [N-]=[N+]=NC1CCC(C(N2CCCCC2CCNC(=O)CCc2ccc(Cl)s2)=O)C1 C(=O)(CC(C(F)(F)F)NC(=O)C=CCN1CCC1)N1CCC(CC)CC1 CC1(NC(=O)CSCC(N)=O)CCN(C(=O)C(c2ccc(Cl)cc2)=O)C1 N1(C(c2c(=N)[nH][nH]c2)=O)CCCCCCC1C(=O)NCC12CC(CO)(CO1)C2 c1(C(=O)NC(C2(O)CN(C(C3COCCO3)=O)C2)C)cc(C2CCC2)nn1C C1(C(=O)NC(CC)CCC)(NC(C(C)=CCC)=O)CCOCC1 c1(CC=C)ccc(C(=O)N(C(C)C)C(C)C)c(N)c1 Cc1cccc(CNC(=O)CC2CCN(C(C3(C)CCCN3)=O)C2)c1 CCC(C#N)(CC)C(=O)N1CC(C2CN(C(=O)C#CC3CCOC3)C2)C1 c1(N(C23CC(N)(C2)C3)C(c2c(C(C)C)cccc2)=O)ccn2ncc(Br)c2n1 C1(OC)CN(C)C(C)(C(=O)NC2CCC(C)N(C(C3CC(F)(F)C3)=O)C2)C1 c1(C(N2CCC(N(C(=O)C(F)CC3CC3)CCC)C2)=O)ccc2nccn2c1 Cc1cc(C)c(C(=O)NC2CCN(C(C3CCC3(F)F)=O)CC2)c(O)n1 C=C(CNC(C1(C)CCOC1)=O)CCNC(c1ccc(OCC)s1)=O c1(C(C)=O)cccc(OC(C)C(=O)NCCC)c1.c1(CC(=O)N)cnccc1C c1(C(N2CCC(O)(CN(C(C(CC=C)C)=O)C)C2)=O)ccc(C#N)cc1O CCCCCCCCNC(=O)C(C)(C)C(C)NC(=O)CC1(N(C)C)CCC1 CC(O)CCCCCC(=O)NCC1CN(C(c2cc(CF)on2)=O)CC(C)(C)O1 Cc1cc(C(=O)N(CCC(=O)NC(C)(C)C(O)C(F)F)C)cnc1C Cc1ccc2[nH]cc(CC(N3CCC(S(=O)(=O)NCC4CC4)C3)=O)c2c1 N1(C(C=C(C)C(F)F)=O)CC2(CCCN(C(c3scc(C)c3Cl)=O)C2)C1 c1(C(=O)NC2CCC2NC(C2CC2c2ccco2)=O)cc(Cl)c(F)cc1O C1(NC(=O)CSC2CC2)C2CC1CN(C(=O)COC1CCOC1)C2 C(CCCC(=O)N1CCC(N(C(=O)Cc2c(Cl)cnn2C)C)C(C)C1)(OC)OC N1(C(C(C)=CC2CC2)=O)CCN(C(c2ncc(F)cn2)=O)C(C)C1C c1(NC2C(NC)COC2)ccc(OCCCN(C)C)cc1 c1(C(N2CCC(NC(C(CC)OCC)=O)(COC)C2)=O)noc2c1COCC2 c1(C(CN(C)Cc2cccc(OC(F)F)c2)=O)ccc2ccccc2n1 c1(C(=O)NC2CC(CNC(c3c(CC)n[nH]c3)=O)C2)cc(N)cc(F)c1 c1(CNC(C2CC(O)CN2C(c2sc(Cl)nc2Cl)=O)=O)c(F)cc(O)cc1F N1(C(CN(C(C)=O)C)=O)CC(C)OC(C)(C)C1.c1(C(C=O)O)cccc(Cl)c1.N C1(C(C)C)(NC(c2ccc(C)cn2)=O)CCCCC1.C(=O)C(C)CCN(C)C.N N1(CC)CCCC1C(=O)N(CC(C)CNC(c1coc(C(F)(F)F)n1)=O)C C(=O)(C(C)(O)CC(C)C)NCC1C=CC(NC(c2ccc(C)c(C)c2)=O)C1 N1(C(C2C(OC)C2)=O)CCC2(CCN(C(c3c4c(c[nH]c3=N)CCC4)=O)C2)C1 C1(NC(c2c(C)nc(CO)s2)=O)COC2(C1)CN(C(=O)CCO)C2.C(N)(=O)N C1(C(N2C(C)(CC(N3CC(C(C)C)C3)=O)CC2)=O)CC(C)(C)CO1 c1(CC(C)(C)C)ccccc1C(=O)N(CCNC(c1cnc[nH]1)=O)C1CC1 C(C(CNC(=O)C)S(C)(=O)=O)NC(CC1OCC(C)(C)C1)=O.c1cn[nH]c1 C1(C(=O)NCC(CC)(C)C)CCCCCCN1C(=O)CCc1ccc(C)o1 N1(C(Cc2cc(CC)no2)=O)CCC2(CC1)CC(NC(=O)CC1CC(C)C1)CO2 Cc1c(Cl)ccnc1C(=O)NCCC1CN(C(C23CCC(F)(CC2)C3)=O)C1 C1(C)(CC(=O)NCC=CCNC(c2scc(C)c2Cl)=O)CCCCCC1 CCC(CC(=O)N(C)CCOCCN(C)C(c1coc(C)c1)=O)OC C1(F)CCC1.C(=O)(C(=O)NC)NCC.c1ncc[nH]1.C(=O)C.CC(C)C Nc1ccc(Cl)nc1C(=O)NCc1cccc(NC(c2cncs2)=O)c1 CC1(C)CC(C(N2CCCC2CCCO)=O)CN1C(c1cccnc1O)=O C1(CNC(c2cn(C)c(=O)n2C)=O)CCCCN(C(=O)C(=O)C(C)(C)C)CC1 Cc1cc(Br)c(Cl)cc1C(=O)NCCC1(O)CCN(C(=O)C(C)O)C1 Cc1nc(C2CC2)ccc1C(=O)NCC(C)C.c1(C(C(=O)N)C)cn(C)nc1C c1c(S(C)(=O)=O)cnn1C.C(CCCNC(=NC)NC)OC.C(C)(C)C.C=O c1(CC(N2CCC(N(CCC)C(C3CC3(C)C)=O)C2)=O)ccccc1.C(C)C Cc1c(C(=O)NC(CCC(C)C)C(C)(C)C)nc2sccn12 Cc1cc(Cl)c(C(N2CC3CC(NC(=O)C4=CCCCC4)C3C2)=O)cc1C C(=O)(C#CC(C)(C)C)N1CC2CC2C1.Cc1[nH]nc(C(F)(F)Cl)c1C(=O)N.C C(=O)(C1Cc2ccc(F)cc21)N1CC2C(NC(CN3C(=O)CNC3=O)=O)C2C1 N1(C(c2c(CNC(C(n3ccc(C)n3)C)=O)c[nH]n2)=O)CC(C)c2ncccc21 CC(C)(C)[Si](C)(C)OC1CCN(C(=O)NCCSC2CCCCC2)CC1 C1(C(C)C)CN(C(c2cnc[nH]2)=O)CCC1NC(=O)Cn1cc(C#N)cn1 c1(C(N2CC(O)(C(C)NC(=O)CCn3cncn3)C2)=O)ccn2nnnc2c1 N1(C(COC(C)=O)=O)CCC2CCN(C(c3c(Cl)n[nH]c3C)=O)CC2C1 c1(CCC(N2C(C)CC(NC(c3c(C)n(C)cc3)=O)C2)=O)ccc(F)c(F)c1 O=C(C1=CC2CCCCC12)NCC(CO)NC(c1cc(C2CCC2)no1)=O S(=O)(=O)(c1ccc(CCNC(c2cscc2OC)=O)s1)N(CC)CC c1(C(=O)NCCN(C(C2CC(C)OC2=O)=O)C)cc(Cl)c(F)cc1Br CCC(CC)C(C(=O)Nc1ccc(F)cc1)N1CCN(CCO)C(=O)C1 C1(C(N2C(CN(C(=O)CCCCCO)C)CCC2)=O)CCc2nnc(O)cc2C1 c1(C(=O)NCC2C(NC(C(CC)(C)F)=O)COC2)cccc(C2CC2)c1.O C1N(C(c2ccn(C(C)C)c(=O)c2)=O)CCC1(C)C.CC(C(F)F)=CC(=O)N C1(CC(N2CC(CN(CCN(C(C3C(C)C3)=O)C)C)C2)=O)CCCCC1.C N1(CC(=O)NC)CCC(CNC(=O)C(c2ccccc2C)(F)F)C(C)C1 c1(CC)cc(C)c(C(N2CC(C(C)NC(C3CCC(C)(C)C3)=O)C2)=O)o1 c1(C(N2CCCC(C)(NC(c3nncs3)=O)C2)=O)cc2sccc2cn1 c1(OC)ccccc1C=CC(N1CC2CC2C1)=O.C(=O)C(C)(C)CN(C)C.C c1(C(=O)NC2C3CN(C(C4CC45CC5)=O)CC23)ccc(Br)c(C(F)(F)F)c1 c1(C(=O)NCC2(OC)CN(C(=O)O)C2)cc(O)cc(=O)o1.C(C)(C)C N1(C(=O)Cc2cncc(F)c2)CC(NC(C2(c3ccc(F)cc3)CC2)=O)C2CC12 c1(C(N2C(C)(Cc3cccc(F)c3Cl)CCC2)=O)cccc(F)c1CN C1(NC(CCCC(C)=O)=O)C(C)(C)C(NC(=O)CCC=O)C1(C)C.C(C)(C)C c1(C(=O)NC(CC=C)CNC(c2ccc(CO)nc2)=O)coc2cc(C)ccc12 Cc1ccc(C(N2CCN(C(=O)C(C)NC(c3ccccc3)=O)CC2)=O)c(F)c1 C1(C(=O)OCC2CCC3(C2)CC3(F)F)Cc2ccc(Br)cc2C1 CCC(CC(C)C)C(=O)N1CC2CCC1C(NC(c1ccc(N(C)C)cn1)=O)C2 N1(C(C(CC)C)=O)CC(NC(c2[nH]ccc2-c2cccs2)=O)C(C)C1 C1(Cn2cc(C(C)NC(c3nc(Cl)cs3)=O)nn2)CC(C2CC2)C1 c1(N(C(c2cc(I)n(C)n2)C(=O)NCCC2CC2)C)ccc(Cl)cc1 Cc1ccc2c(=NC3CCC4(CCCCC4)C3)[nH]c(=NCc3ccco3)[nH]c2c1 CC1(C)C(=O)CC1C(=O)NCC1CCN(C(=O)COCCO)C1 C1(c2ccc(CC)cc2)CN(C(=O)CC(=O)OC)CCN1C(=O)C(F)CC1CC1 O=C(C#CC1CCCCO1)N1CC2CN(C(=O)Cc3ccns3)CC2C1 c1(SC)cc(C(=O)NC(C)(C)CNC(=O)C(C2CC2)N(C)C)co1 C(CC1CC1)CC=O.C(C)(C=O)(C1(C)CC1)OC.C(C(F)F)N(CC)C.N c1(C(=O)NC2C(CNC(CCC(CC)O)=O)CC2)cn(C2CC2)c(C)cc1=O c1(C(=O)NC23CC(NCc4cnc(Br)s4)(C2)C3)c(F)ccc(F)c1F C12(NC(=O)Cn3cnnn3)CCCN(C(=O)CCC[N+](=O)[O-])CC1C2 N1(c2nnc(-c3c(OCC)cc(Cl)c(Br)c3)n2CC)C2CCCC1CC(=O)NC2 c1(CC(=O)NC2C(NC(C(CC)O)=O)CCC2)cccc(OC)c1Cl Cc1cc(F)c(C(=O)Nc2ccc(NC(C3(O)COC3)=O)c(C)c2)c(Cl)c1 N1(C(C2C(C(C)C)C2)=O)C2CCC1CN(C(c1cc(C)c(O)c(C)c1)=O)C2.C CCCCC(CC)C(C(=O)NCCCC1CC1)N1CCCC2(CC(O)C2)C1 c1(N(CCOCCN(C)C(C2CCCC2c2ccccc2)=O)C)nnc(CO)s1 N1(C(CCC(C)OCC)=O)CC2CC(NC(=O)Cc3cccc(C)c3F)C(C2)C1 C1(NC(c2cccnc2O)=O)CN(C(=O)COCCc2cccs2)CCC1CO C(=O)(C1=C(F)CN(C(=O)C(C)n2ccnc2)CC1)N1CC(OC)C(OC)C1 c1(CC=O)ccccc1C(F)(F)F.CC(CNC(=O)C=O)C.CC(F)F.N Cc1nc(N2CC3(CNC(c4c(C)nn(C)c4C)=O)CC2CO3)ccc1[N+](=O)[O-] N1(C(Cc2c(CC)con2)=O)CC(C)CCC1C.N1(CC(=O)N)CC(=O)NC1=O C1(C(N(CCCCN(C(C(C)CC2CCC2)=O)C)C)=O)CC2CCC1C2 C1(C2CC2)(CNC(C(C)C(C)(C)C)=O)CCN(C(c2cc(Cl)ncc2N)=O)C1 C1(NC(CCC=CCC=C)=O)CC2CC(NC(c3cncc(CO)c3)=O)CC12 N1(C(CC2C(CC)C2)=O)C(C)CN(C(c2cnnc(C3CC3)c2)=O)CC1C N1(CCC=CC)CCC(CNC(c2nocc2COC)=O)(CC)CC1 N1(C(C2C(CCOC)C2)=O)CCC(NC(c2ccc(C)nn2)=O)CC1 C(CCCC(=O)N(CCCNC(=O)C(C)Cc1ccc(C)cc1)C)OC O=C1CN(C(=O)C=Cc2ccccc2)CCN1C1CCCN(C(=O)C2CC2)C1 CC1CCCCC1(CNC(C1CCCCC1C)=O)NC(=O)CC1CC1(Cl)Cl N1(C(C(C)(O)C2CCC2)=O)CC2(CCC2NC(c2nc(Cl)sc2Cl)=O)C1 c1(C(N2CC(NC(c3c(C)cc(Br)cn3)=O)C(F)C2)=O)ccc2c(c1)CC(=O)N2 CC1(C)CC(C(=O)NCC2(CCCO)CC2)CCN1C(C1CCCCO1)=O N1(C(c2nccc3ccccc23)C(=O)NC2COC2)CC(O)CC2CCCCC12 C1(N(C(=O)C(F)C2CCC2)CC(C)C)CCN(C(C2CCCN2CC)=O)CC1 C(=O)(C(CC)(CC)CC)N1CCC(CC=C)(NC(=O)C=Cc2cnccn2)CC1 n1(C(C)C)ncc(C(=O)N)n1.C1CCC1.C1(C=O)CC(C=O)C1.C(C)(C)C Cc1cccc(Cl)c1C(=O)NCCNC(c1ncn(C)n1)=O N1(C(C(C)=O)=O)CCC2(CCCN2C(c2cc(Cl)cc([N+](=O)[O-])c2C)=O)CC1 C1(NC(c2ccnc(C)n2)=O)C2CCC(C2)C1C(=O)NCC1CC12CCC2 c1(SC)nc(Cl)cc(=NC2CN(C(=O)CCc3cncn3C)CC2C)[nH]1 C1(CNC(=O)CSc2ccsc2)CCN(C(=O)CC2CCCC23CC3)C12CC2 C1(C(=O)Nc2cnn(CCN3CCOCC3)c2)CC2(C1)CC(CF)C2 N1(C(CC(COC)C)=O)CC2CCN(C(=O)Cn3cc([N+](=O)[O-])nc3C)C2C1 c1(CCN=C(NCC(=C)CC)NCC2CC2)ccc2c(c1)CCO2 CN=c1[nH]ccc(=NCC2CCC(C(N)=O)O2)[nH]1 c1(C(=O)NCCC2CCC2)ccc2nncn2c1.C1(C=O)C(Cl)(Cl)C12CC2.N c1(CCC(=O)N(CCCNC(c2cnc(O)o2)=O)CC)ccc(O)c(F)c1 C#CCCCC(C)C(=O)NCCCCCC(=O)NC(c1ccccc1)CF C(CC(C)(C)CNC(=O)C(=O)NC(c1ccccc1OC)C1CC1)OC CCC(CC)C(C)C(=O)N1CC(OCCC(N2CCC3CCC(C3)C2)=O)C1 C(C(CC(F)(F)F)NC(c1ccncn1)=O)NC(CC1C(C)(C)C1)=O.C1CC1 C(=O)(C(C)(O)C1CCC1)N(CCC)CC.c1(C=O)ccccc1.C(=O)CC.N C1(CNC(C(CC)N(C)C)=O)CC(C)(C)CN1C(C12CCC(CC1)C2)=O.O N1(C(c2nncn2C2CC2)=O)CCN(C(=O)CCC2CC2)C(CC(F)(F)F)C1 C1(C(=O)Nc2ccc(Cl)cn2)CCCC12CCN(Cc1cocn1)C2 C1(CCC(=O)NCCC2C(C)C2)CCCN1C(c1nc[nH]n1)=O Cc1cc(C(=O)NCC2CN(C(=O)Cc3[nH]cnc3C)CC2C)c2nccn2c1 c1(CN2CCN(C(c3sccc3Cl)=O)C3C2C3)ccn2ccnc2c1 c1(C(=O)NCC(CNC(C2(Cl)CC3CCC2O3)=O)OC)cc(C)ccc1C C1(C(N2CC(C(=O)N(C)CCF)(COC)C2)=O)CCNC(=O)C1 c1(CCC)ccc(CC(N2CCC(C)(CNC(=O)CCn3cccn3)C2)=O)cc1 N1(CC)CC(C(=O)N(C)C)CC1=O.c1(C(N2CCCC2)=O)cncc(N(C)C)c1 C1(CCNC(=O)NCCCOc2ccc(C)cc2)CC(C)OC(C)C1 N1(C(c2c(C)cc(C)o2)=O)CC2(C1)SCCC2NC(c1cccc(CO)c1)=O c1(OC(C(=O)Nc2c(C)cc(Cl)cc2)C)ccc2cccc([N+](=O)[O-])c2c1 N1(C(c2ccc(SCC)nc2)=O)CC2CCC2(CC)C1.c1(C=O)cnc(C)[nH]1.N C1(CC)CCN(C(c2cnsn2)=O)C1CNC(C1CCC(OC)CC1)=O C(CC(C)C)(C(=O)NC1(C(=O)NCCSC(C)(C)C)CC1(C)C)OC c1(C(=O)NC(c2cccnc2)C(=O)N(C)CC2(C)CC2)ccc(NC)cn1 C(CSC)(C(=O)N(CCCNC(C1OCCC1C)=O)C(C)C)OC C(=O)(C(C)(C)CCCNC(c1cncc(CC)c1)=O)N1CC(CCC#C)C1 C(=O)(C1=CC2CCC(C1)C2)NCC1CC(C)(C)CN(C(C2CNC(=O)C2)=O)C1 CC(C)CC(CNC(c1snnc1C1CCC1)=O)NC(C1CCCSC1)=O N1(C(C(C)NC(N)=O)=O)CCC(NC(=O)CCc2ccn(C)c2)C12CC2 c1(NC(C#CCNC(C2ON=C(C)C2)=O)=O)ccc(C(C)C)cc1 Cc1ccc(SC(C)C(=O)NC)cc1.c1(C=O)ccc(F)cn1.C1(CC)CC1 CC1(C2CC2)CN(C(c2cc(OCC3CC3)ccn2)C(=O)NCCC#N)CCO1 CC1(C)CC(CC(N2CC(NC(=O)CCC(F)(F)F)C3(CC3)C2)=O)C(=O)O1 c1(C(N(CC(=O)N=c2cc[nH]cc2)C)=O)ncnc2c1ccn2CC(=O)O n1(CC)nc(C)cc1C(=O)NCC1C(C=O)C1(C)C.C(CO)C1CC1.N C(=O)(C(F)CCC(C)C)N1CCC(C(CNC(c2c(CC)nccn2)=O)O)CC1 C1(C(N2CC(CCNC(C3CC4CC4C3)=O)(OC)C2)=O)SC2C=CC1CC2 C1(CC(=O)N(CCC)CCNC(=O)CCN2CCC2)CCCCCC1 C=CC(C)(O)CC(=O)NCC1(C)CCCN(C(C2(C(C)C)CCC2)=O)C1 N1(C(CN2C(=O)CCC2)=O)CC2C3CCC(C2C1)N(C(c1n[nH]cc1[N+](=O)[O-])=O)C3 C(=O)(C1=CCCOCC1)N(C1CC(NC(=O)Cc2ccno2)C1)C Cc1ncc(C(=O)NC2(C)CCC2)c(C)n1.C(=O)C(C)C(=O)N1CCOCC1.N C1(C(=O)N)CC(=O)N(C)C1c1ccc(Cl)c(F)c1.Cc1cnc(C2(C)CC2)o1 [SH](=O)(=O)c1cccs1.C(c1cc[nH]c1)=CC=O.C(CC)N(C)C(C1CC1)=O C1(CNC(C=C(CNC(c2ccc(CC)o2)=O)C)=O)CCCNC1=O c1(N2CCC(O)C(F)(F)CC2)ccnc2cc(Br)c(F)cc12 C12(COC)CCC(C(=O)N(CCCCC)C)(CO1)C2.C1(C(=O)N)CCCN1C=O C(CN=C(NCC12CCC(CC1)C2(C)C)NC1CCC1)(C1CCC1)OCC C1(N(C)C)CCN(CC(=O)NC2CCCC2NC(=O)Cc2cccc(Cl)c2)CC1 c1(CC)ccc(C(N2CCCCC2CCN(C(=O)CCSC)C)=O)nc1 N1(C(CCCSC)=O)CCC(F)(CNC(=O)CC2(C)CC2F)CC1 C1(CN(C(=O)CNC(=O)CC(F)(F)F)C)CCCN(C(=O)CC(Cl)Cl)C1 c1(C(=O)NC(CCNC(C(C)OC)=O)C(C)C)cc2cccnc2[nH]1 C1(C(=O)OC)CCC(C(=O)N(CC(C)NC(=O)C(C2CCOCC2)C)C)CC1 [nH]1nc(C2CC2)cc1C(=O)N(C(C)CN(C(=O)Cc1cncnc1)C)C.CC c1(C(N(C(CCNC(CCSCC(C)C)=O)C)C)=O)cccc(CF)c1 N1(C(C2(C)C=CCC2)=O)CC(NC(=O)CN2CCCCC2=O)CC2(CC2)C1 N1(C(C2C(C(=O)OC)C2)=O)CC(OC)C(C(=O)N(C)Cc2ccoc2)C1 C1CS(=O)(=O)C2CN(C(c3coc(C)n3)=O)CC12.C1(C=O)(C=O)CCC1.C C(=O)(CCC(C)(C)C)NC1C(NC(COc2c(CC)cccc2)=O)C1 C=C(C)CC(C(=O)N1CC(C(C)(C)O)C1)NC(=O)CC(C)(C)CC N1(C(CC(CNC(CCSCC)=O)OC)=O)CCOCC(C2CC2)C1 N1(CC(=O)NCCCOCCC(=O)NC(C2CCCC2)C)CCSCC1 N1(C(CCOCCC)=O)CCC(CF)(NC(c2cn(C3CCOC3)nn2)=O)C1 N1(C(C(C)=C2CC2)=O)CC(NC(c2nc(Cl)sc2C)=O)CC1C c1(N2CCN(CCCNC(CC(CC)CC)=O)CC2)ncn(C)c(=O)c1Br N1(C(C2CCN(C(c3c[nH]c(=O)cn3)=O)CC2)=O)CCC(O)(CO)CC1 C(=O)(CCP(C)(C)=O)NC1(C(=O)NCC(F)C2CCC2)C(C)CCC1 c1(CC(N2CCC(O)(C(C)NC(C3CC(O)C3)=O)C2)=O)ccc2cccnc2c1 Cc1nc(CO)sc1C(=O)NC1CCCC(NC(=O)C(c2ccnn2C)O)C1 C(C(O)CC(=O)NC1(CC(N2CC=CC2CF)=O)CC1)N(C)C C(=O)(C1=CCCCCC1)NC1CCCC(NC(=O)CCCN2CCCC2)C1 c1(C(=O)NC2CCN(C(C3CCC(C)CC3)=O)C(C)C2)cc2ncccc2[nH]1 N12CCN(CC1)CCC(=O)NCC2.c1(C(N2C(NC)CCC2)=O)ccnc(S)c1 C1(NC(c2cn(CC(F)(F)F)nc2C2CC2)=O)CCCCCC1O c1(OC)ccc(Cl)c(C(=O)Nc2ccsc2C(=O)NCc2cc[nH]n2)c1Cl Cc1ccc(Br)cc1S(=O)(=O)N1CC(NC(=O)C(C)Cn2cccn2)C(C#N)C1 c1(OC)ccccc1NC(=O)C(O)CCNC(c1ccnn1C1CC1)=O Cn1cnc(C(=O)NCCCC(C)(C)NC(C2CCC3CCC23)=O)cc1=O C1(CNC(c2cnc(C)n2C)=O)CN(C)CCN1C(=O)CCCCC1CC1 C(C(CC(C)C)C(=O)NCC1(F)CN(C)C1)NC(C1(C=C)CCCC1)=O CC1CCCCC1OCC(=O)N(C1CCN(C2CC2)C1)C.c1c[nH]nc1C1CC1 N1(S(CCC)(=O)=O)CCCCC1C(=O)NC1(CNC(=O)COC)CCOC1 c1(C(N2CC3C(CN(C(C(C)=CC)=O)C)C3C2)=O)cc2cc(O)ccc2n1C N1(C(C2(CC)CCCC2)=O)C2CCC1C(C)C(NC(=O)C(O)C1CCCC1)C2 Cc1ccnc(C(=O)NCC2CCCN2C(c2nc(-c3cccs3)oc2C)=O)c1 CCC(C)(C(=O)NCC1(C)CN(C(c2cc3ccccc3[nH]2)=O)CCO1)C(F)F C=Cc1cnn(C)c1C(=O)NCC(C)(C)CN(C(=O)C=O)CC.C1CC1 c1(C(N2C(CC)C(NC(=O)Cn3cncn3)CCC2)=O)ccc([N+](=O)[O-])cc1 Cc1cc(C(N2CC3CC2(CNC(C2CC(N(C)C)C2)=O)C3)=O)ncn1 N1(C(c2onc(CC)n2)=O)CCCC2(CNC(=O)Cn3ccnc3C)CCCC12 c1(C(=O)NC(CNC(C2C(=C)C2)=O)C2CC2)cc2ccc(F)cc2nc1C C(CO)(CC)NC(C(c1ccccc1)N(CC)CC)=O.C1(C)(C=O)CC=CC1 c1(C(N2C(C(=O)NC)CCC2)=O)c(C)c(C)nc2ccccc12 N1(C(c2c(CC)cco2)=O)CCC(C(=O)NCC2CC=CC2)C(O)C1 c1(N(CCCCN(C(Cc2cnc(C)s2)=O)C)C)cc(C#N)c(F)cc1[N+](=O)[O-] N1(CC=O)CCCCC1.[SH](=O)(=O)CC.CC(F)(F)F.N(C=O)(CC)CC c1(C(=O)OC)cnc(N)c(C(N2CCCC(C(c3ccccc3)O)C2)=O)c1 c1(C(=O)NCCN(C(CCc2nc(C)sc2)=O)C2CC2)ccc2nnc(C)n2c1 N1(C(CCC)=O)CC(NC(C2CCCN2C)=O)C(C)C1 Cc1cnnc(O)c1C(N1CC(O)(CNC(=O)CS(N)(=O)=O)C1)=O N1(C(COCCC=C)=O)CCCCC1C1CCN(C(c2c(C)csc2Cl)=O)C1 c1(NCc2n(CC)cnc2)cccc(C(N2CCC(O)(C(F)(F)F)C2)=O)c1 N#CC1CN(S(=O)(=O)NCC(C)CC(F)(F)F)C1 CC(C)CC(O)C(C)C(=O)NCCCN(C(C1(CO)CC1)=O)C1CC1 C1(CNC(CCC(=C)Cl)=O)(NC(c2sc(C)cc2C)=O)CCCCC1C C1(NC(c2ccc(OC3CCC3)cc2)=O)COCCN(C(=O)Cn2nccn2)C1 c1(NC(C2CC(O)CN2C(c2ccoc2)=O)=O)c(O)cccc1[N+](=O)[O-] C(=O)(C1=C(Cl)CCC1)NC1(C)CC(NC(C2CCC(CCC)CC2)=O)C1 CC1CCc2nc(C(C)NC(c3cc(OCc4ccccc4)ccn3)=O)sc2C1 Cc1nc(NC(c2ncncc2-c2ccn(C(C)C)n2)=O)nc(Cl)c1Br CC1CCN(C(=O)CCc2ccn(C)c2)CCN1C(=O)CC1CCCC1C N1(C(c2n(CC)nc(C)c2)=O)CCC(NC(C23CCC(CC2O)C3)=O)CC1C C1(F)(CNC(CNC(C(CC)C)=O)=O)CCN(C(=O)C(C)(C)SC)C1 C1(NC(C(CN(C)C)N(C)C)=O)C2CC(NC(=O)CCC3CC3(F)F)CC12 NS(=O)(=O)C1CN(C(C2CCCC2CNC(=O)CSC(F)F)=O)C1 c1(N2CCCC(C(=O)NCC(COC)O)C2)ccnc2[nH]ncc12 N1(C(c2ncc(C)c(Cl)c2)=O)CCN(C(C2(C)CCCS2(=O)=O)=O)C2(CCC2)C1 c1(C(N2CC(NC(C(CC)(C)F)=O)C(OC)C2)=O)cc([N+](=O)[O-])oc1C C=CC1COCCN1C(C1CCCC1NC(C1CCN1CC)=O)=O c1(C(N2C(C(C)NC(CC(CC)CC)=O)CCCC2)=O)ccnc2ccnn12 C(C(=O)N1NC(=O)CC12CCN(Cc1ccccc1)C2)c1c(C)nc(C)s1 N1(C(CS(CC)=O)=O)CCN(C(=O)CSc2n[nH]c(=N)s2)C(CC(F)F)C1 CCCCS(=O)(=O)CC(=O)NCCCCC1CCN(C(C2(F)CCCC2)=O)CC1 C1(NC(c2cn(C)nc2)=O)CC2C1CCN2C(=O)C=CC1COC(C)(C)O1.C C1(C(N(C2C(C)CCN(C(C3(C)CC3)=O)C2)C)=O)CC2(CCC(F)(F)CC2)CO1 c1(OC)cc(CC(=O)NCC2CN(C(=O)CC3CC3(C)C)CC2C)ccc1Cl c1(C(=O)NC2C3CCN(C(c4ncn(C(C)C)n4)=O)CC32)cc2n(n1)CCCC2 c1(NCC2CN(C)C2)ccc(S(=O)(=O)N2CCCCC2Cc2nccs2)cc1Br NC(=O)C(CC(F)C(N)=O)NC(=O)NCC1CCN(C2CCCCC2)CC1 C(=O)(C1Cc2ccc(Cl)cc21)N1CCCCC1.c1(NCC)scnc1C(=O)NC C(CC(C(=O)NCCCCCN(C(=O)C(C1CCC1)OC)C)OC)OC c1(C(=O)NCC2(CCNC(CC3C(C)OCC3)=O)CC2)ncc2n1CCCC2 C1(C(N2C(CNC(c3c(C)n(C)cn3)=O)CC(F)C2)=O)CCc2cncn2C1 C1(NC(=O)Cn2cnnc2O)CC2CCC(C1F)N2C(=O)CC1CCNC1=O C#CCC(C)C(=O)N1CCOCC1CNC(=O)C=Cc1ccc(SC)s1 N1(C(C2(NC(c3cccc(C)c3)=O)CCC2)=O)CCC12CCC(O)CC2 c1(C(N(CC(C)C)C)=O)ccc(S(=O)(=O)N(C)C)o1.C(=O)(C1=NOCC1)N CC1(C#N)CC(NC(C2CC2c2ccc(CN)cc2)=O)C1 C1(C)CCN(C(=O)C(F)C=O)CC1.C1(C)(CC)CCC(C=O)O1.C(C)(C)C.N C=C(C)C(CC(=O)NC(C)(Cc1ccccn1)C(=O)OC)OCC C(=O)(C(C#N)C(C)(C)C)NC1CC(N(C(CCC(C)N(C)C)=O)C)C1 N1(C(C(C)C2CC2)=O)CC(C2(NC(=O)CS)CC2)C1.c1ccccc1.CC=O N1(C(c2ccc(C(C)C)cn2)=O)CC2CCC1CC2NC(=O)Cc1ccno1 C1(CNC(c2[nH]cc(C#N)c2)=O)CCCCC12CC2(F)F Cc1ccc2cc(C(N3CC4C(C(N5CCCC(CO)C5)=O)C4C3)=O)n(C)c2c1 CC1CN(C(c2ccns2)=O)CC(CCNC(=O)Cc2nn(C)cc2Cl)O1 C12(CC(F)(F)C1)C(=O)N2.C1(CNC(CSCC)=O)CCC(C)N1C C1(O)(C(C)NC(=O)CCF)CCN(C(=O)CC2(C)CC2(Cl)Cl)C1 C1(CCC(=O)NCCN(C(CCC=C(C)C)=O)C2CC2)CCCCN1C c1(C(N2CCN(CCN(C(C(CC)(C)CO)=O)C)CC2)=O)cc2sccc2cn1 C(O)(C(F)(F)F)(C(F)(F)F)c1ccccc1.C1(C[SH](=O)=O)CCCC2(CCC2)O1 C(=O)(C1=Cc2ccc(Cl)cc2OC1)N1CC(CNC(c2cc(C)no2)=O)C2C1C2 Cn1nccc1C(C(=O)NC1CCN(CCF)C1)NC(=O)C=CC(C)(C)C Cc1cc(Cl)ccc1OC(C)C(=O)N(CC(O)CNC(=O)CCC(N)=O)C Cc1[nH]nc2c(CNC3CC(n4ncc5ccccc45)C3)cccc12 c1(SC)ccc(Cl)c(C(=O)N(CCCn2cc(C(O)CC(C)C)nn2)C)c1 N1(C(=O)NC(c2ccccc2Cl)COC)CC(=O)NC2CCCC2(C)C1 c1(C(=O)NC(COC)C(=O)N2CCC2CO)cccc2cc[nH]c12 CC1(C)CC(C(=O)N2CCN(C(=O)C=Cc3cocn3)CC2c2cn[nH]c2)=NO1 Cc1ccc(=N)[nH]c1C(N1CC(c2ocnc2C)C1)=O.C1(C(=O)N)CC1(F)Cl N1(C(CC(CN(C)C)O)=O)CCC2(C1)c1ncn(C)c1CCN2C(C1CSC1)=O C(=O)(C1=C(c2ccccc2)SCCO1)NCC1C(NC(C2C(C)C2)=O)CCC1 C(=O)(C1c2ccccc2C(=O)N1C)N1CC(NC(c2c(CC)nco2)=O)C1 c1(C(=O)NCC2(CO)CCN(C(C(C)Cc3cnc[nH]3)=O)C2)cc(F)ccc1Cl c1(C(=O)NC2CN(C(c3n(C)ccn3)=O)CC2F)ccc(O)c(O)c1Cl C(=O)(C1=CC2(CCN(C(C3CCCCNC3=O)=O)C2)C1)N1CC(N(C)CCO)C1 c1(C(=O)NCCCN(C(c2cnc(CC)s2)=O)CC)cc2ccncc2[nH]1 C1(CNC(c2ccc(CC)s2)=O)CCN(C(c2cscc2F)=O)C12CC2 C(CC(C)(C)C)(C(=O)NC(N)=O)N(c1cccc(Br)c1)C Cc1ccc(F)c(C(N2CC(CNC(c3oc(C)cc3C)=O)CC2C)=O)n1 CCCS(=O)(=O)C(C)C(=O)NCC(C)NC(c1ccn(C(C)(C)C)c1)=O.C C1(NC(CCOCC)=O)CCCCN(C(=O)CCc2cccs2)CC1.C(C)(=O)N C(C(=O)NCC1CCCCC1)(C(C)(C)C)OC.C(c1ccccc1)=CC=O.C c1(C(=O)NC2C(CC(N3C(C#C)CC3)=O)CCC2)c(F)cncc1F Cc1cccc(C(C)C)c1NC(=O)C(=O)NC(C)Cc1ccco1 N1(C(C=CC=CCC)=O)CCCC12CCN(C(C1CCc3n[nH]c(C)c3C1)=O)C2 C1(NC(c2ccc(C(N)=O)s2)=O)CCCC12CN(C(=O)Cn1cnnc1O)C2 c1(C(C(=O)NC2CCOC2)N(C2CCC2)CC2CCC2)cccc(OCF)c1 CCCCC(C)C(=O)N1CC(CNC(=O)CN(CCO)CCO)C1 C(=O)(CN1C(=O)CCCc2sccc21)NC1C(NC(=O)Cn2ncnn2)CC1 C1(NC(C2CC(CF)C2)=O)CCCCCC1C(N1CCCCCCC1)=O N(C1CCCc2c(F)cccc21)C(c1c(C)occ1)c1nnnn1C(C)C c1(CC(N2CC(=C(CNC(=O)CC3C=CCC3)F)C2)=O)cc(F)ccc1F Cc1cc(NC2(c3nnnn3CC(F)F)CCSCC2)cc(C)c1F C1(C(=O)NC(COC)(C)C(N)=O)CCN(C(=O)CSCCOC)O1 N1(C(=O)Nc2c(SC(C)C)ccc(Cl)c2)CCC2C(O)C(C)(C)C12 C#Cc1cncc(C(=O)NC2(CCC(=O)NC(C)CCSC)CCCC2)c1 CC(C)(CO)C(N1CCN(c2ccc(OC(F)(F)F)cc2)CC1)c1ccccc1 C(=O)(C(F)(CNC(=O)C=CC1CCC1)C(C)C)NCc1c(C)ocn1 C1(NC(c2nc(C)n(C)n2)=O)CCN(C(c2cc(C#N)cs2)=O)C12CC2 C(CC(C(=O)NC)NC(=O)Cc1cnccc1C)=CC.C1CC(CN=[N+]=[N-])C1 C12(NC(c3n(C)cnc3)=O)CCCN(C(=O)Cn3nnc(C(C)(C)C)n3)CC1C2 Cc1cc(O)cc(=O)n1CCC(=O)N(C1CCCN(C(=O)C2CC2)C1)C C12(CNC(C3CCC3n3ccnc3)=O)CCCC1CN(C(c1ccncn1)=O)C2 Cc1ccc(=O)n(CC(N2CCC(O)(CN(C)C(C3(Cl)CC3)=O)C2)=O)c1 C=CCCCCC(=O)N1CCC(CNC(c2nnc(Cl)cc2N)=O)C(CC)C1 CC(CC(=O)N1CC2OCC(CNC(=O)CSc3nc[nH]n3)C2C1)CC(C)(C)C c1c(F)c(F)cc(F)c1F.NC1C2CCCCC12 Cc1ncc(CN(Cc2ccoc2)CC2CCCO2)o1 C(=O)(CCCCCCCCC)NCC1(O)CCCN(C(C2C(OCC)C2)=O)CC1 C#Cc1ccc(C(=O)NC2CC23CC(NC(C2CC2C)=O)C3)c(F)c1 c1(C(=O)Nc2nc(C)nc(O)c2)ccc2[nH]c(C(N3CCC(C)C3)=O)cc2c1 Cc1nc(NC(c2cn3cccc(C)c3n2)=O)c2c(ncn2C)n1 c1(C(C(=O)N(C)CC2(O)CN(C(CCSCC)=O)C2)=O)ccc(F)c(F)c1 N1(C(=O)OC(C)(C)C)CCOCC1CCNC(=O)NC1C=CCC1 N#Cc1cccc(C=CC(N2CC3CC3(CN)C2)=O)c1.c1cnc(Cl)c(Cl)c1.C c1(COCC(N2CCCC(NC(C(C)OCC)=O)C2)=O)cc(C)ccc1 Cc1ccc(Br)c(C(=O)NCC2CCN(C(=O)CCCF)CC2C)n1 N1(C(C(C2CC2)SC)=O)CCC2(CC(C(=O)NC3CCN(C4CC4)CC3)C2)C1 c1(NC(C2N(C(C(CC)C)=O)CC(O)C2)=O)ccc(F)c(Cl)c1Cl C1(NC(=O)CC2CCCC2O)CCN(C(C23CCCN(CCC2)C3)=O)C12CCC2 CC(CC(=O)N1CCC1CNC(c1c[nH]nc1-c1ccn(C)n1)=O)CC(F)(F)F c1(OC)ncc(Cl)c(=NC2CCCN(C(C3CCCN(C(N)=O)C3)=O)CC2)[nH]1 C12CC(C1)C(C)(C)O2.C(C(=O)N)(C(C)(C)C)SC.C1CCOC1.C(=O)C C1(C(N(CC(=O)N)C)=O)CC2(CC2)CN1C(c1nc(=N)cc[nH]1)=O.CCC CC1CCC=C1C(=O)N(C1CN(C(c2ccc(C(N)=O)cc2)=O)CC1(C)C)C C(=O)(CCC(C)(C)[N+](=O)[O-])NC1C(NC(C(c2cn(C)c3ccccc23)C)=O)C1 CC(F)(F)CC(=O)N1CC(CC(F)C(=O)NCCN2CCNC2=O)C1 N1(C(C2CCN(C(CCOCC)=O)CC2)=O)CC2(CCOC(=O)N2)C1 Cc1cc(CNc2cccnc2C(=O)NCC2CCO2)c(C)cc1Br C(=O)(CS(=O)(=O)C(C)C)NC1(CO)CCN(C(C(CC#C)C)=O)CC1 N1(C(C(C=C)CC)=O)CCC2(C1)CN(C(=O)CC1CCC(C)O1)C2 c1(CCC(=O)NCC(CC=C)NC(=O)C(C)(C)OC)ccc2[nH]ccc2c1 c1(CC(N2CCC(N3CCN(C(C4CC4F)=O)CC3)CC2)=O)ccc(Br)cc1 C#CCC(C(=O)Nc1cnn(CC#C)c1)NC(=O)CC1C=CCCC1 c1(C(N2CCC(NC(C=C(C)C(F)F)=O)(CF)C2)=O)cc(N)c2ncccc2c1 C1(NC(CSCCN(C)C)=O)CN(C(=O)Cc2nn(C)cc2Cl)CCC12CCC2 C1(CNC(Cc2ccc(C)cc2)=O)CCCCN(C(=O)CCC(C)(C)C)CC1 N1(C(c2n(C)ccn2)=O)CCC(NC(=O)CCC2(C)CC2(F)F)C(F)C1 c1(C(N2C(CNC(C(c3cccc(F)c3)C)=O)CCC2)=O)nnc(O)cc1O C(C(=O)NC1CCN(C(c2ccc(-n3nnnc3C)cc2)=O)C1)(C(C)(C)C)OC c1(C(=O)NC(CN(C(=O)Cn2nnc(C)n2)CC)C)c(C)nn(C)c1C c1(OC)ccc(Cl)c(C(N2CC(C)C(O)C2)=O)n1.C1(=CC(=O)N)CCCC1 Cc1cc(C)c(NC(=S)NC(C)C)c(C)c1 C(CO)(CCCCNC(=O)CN1CCC(C)CC1)NC(C=CCOC)=O Cc1cc(C(=O)N)nn1C(F)F.C1C2CN(C(=O)CC3CCNC(=O)C3)CC12 Cc1c(C(=O)NCC(C)CNC(=O)CC2CCCCO2)cnn1C N1(C(C)=O)CCN(C(=O)CN2CCSCC2)C2CCCCC2C1 c1(C(=O)NCCN(CC(C)O)C(=O)CC2CCCCN2C)cnc(Cl)cc1N C(=O)(C(C)P(C)(C)=O)N1CCC(NC(c2c(C)cn(C)c2)=O)(CO)C1 C1(C(=O)OC)CCC(C(=O)NC2CN(C(C3CCN(C)C3C)=O)C2)CC1 C1(CCC(=O)NCC(Cn2cc(C3CC(F)(F)C3)nn2)OC)CCC(=O)N1 c1(C(N(CCCNC(C(CC)OCC)=O)C)=O)cc(C)nc2c1c(O)nn2C O=C(C(F)C1=CCCCC1)NC12CCCN(C(C3CCCSS3)=O)CC1C2 C(=O)(C(F)C(F)(F)F)N1CC(CC(C)NC(c2ccc(C(C)C)s2)=O)C1 CC(C)(CN=c1[nH]c(N2CCC(F)(F)C2)nc2cccnc12)c1cccs1 C1(NC(COCC)=O)CCC(NC(=O)C(C)(C)c2cnco2)CC1 N1(C(CCC#C)=O)CCC2CCC12CNC(=O)CCc1ccc(C)cc1 N1(C(COCCOCCOC)=O)CC(C)C2(CCC2)C1.C(=O)C=NOC.N c1(C(=O)NC2CC(NC(C3CC4CCC3C4)=O)C2)n[nH]c2c(F)cccc12 c1(NC(c2ncc(-c3cncc(OC(C)C)c3)cn2)=O)cnnc(O)c1Cl C1(C(=O)NCc2ncn(C)c2)CCCCN(C(=O)CCc2cnn[nH]2)C1 N1(C(C2(CNC(CC(C)C)=O)CC23CCC3)=O)CCC2(CCSC2)C1 c1(C(N2CCC(Cc3ccccn3)C2)=O)noc2ncccc12 C1(C(N2CCC(NC(=O)OC)CC2)=O)CCN(C)CC1c1cnn(C)c1 Cc1cc(C(N2CCC(CNC(=O)C(F)C(C)(F)F)C23CC3)=O)c(F)cc1N c1(C(N2CCC(F)(CNC(c3c(C)c[nH]n3)=O)C2)=O)cc(C)c(O)c(N)c1 c1(C(=O)NC(C(=O)NCC)C2CCOC2)c[nH]c(=O)cn1.CCC1CC1.O c1(N2C3CN(C(=O)CC4CC5(CC5)CO4)C(CC3)C2)ncnc2cccnc12 C1(C(=O)Nc2ccc(OC)c(C(F)F)c2)CC12CCOc1ccc(F)cc12 CC1CC(C(N2CC(N(C)CCO)C2)=O)CN(C(=O)CSC(F)(F)F)C1 c1(OCCNC(c2ccc(F)c(F)c2F)C)ccc2ccccc2c1 C(=O)(C1CCc2cccc(O)c21)N1CCC2(C(CNC(C3CCCC3)=O)C2)CC1 N1(C(C(c2cccnc2)N(C)C)=O)CCC(C(C)(C)NC(c2sccc2F)=O)C1 C12(NC(CNS(NC)(=O)=O)=O)CCN(C(c3cc(C)c(C)s3)=O)CCC1C2 c1(C(=O)NCc2cc(C(N3CC(c4ncc[nH]4)C3)=O)n[nH]2)cnn2c1OCC2 N1(C(C(CC)COC)=O)CCC2(CCC(NC(C3(CC(C)C)CCC3)=O)C2)CC1 C1(NC(C(n2cc(Cl)cn2)C)=O)CC(O)(CNC(C2CCCC2F)=O)C1 N1(C(C2(CCCC)CC2)=O)CCC2(CC1)CN(C(=O)C(O)CCCC)CC2CO CCC(CNC(c1cn(CCO)nn1)=O)(CC)NC(=O)C(C1(O)CCCC1)F Cc1cc(F)cc2c1CN(C(=NCC1CCN(C)C1=O)NCC(=O)N(C)C)CC2 c1(NC(C2COCCN(C(Cn3ccc(C)n3)=O)C2)=O)cccc2c1OCCO2 C(=O)(C1=CC2(CCOC2)C1)N(C(C(=O)N(CC(=C)C)C)C)CC c1(COC)cnc(C(=O)NC(CCN(C(=O)C=CBr)C)C(C)C)nc1 c1(C(N(CC(C)Nc2ncnc(Cl)c2C2CC2)C)=O)ccc(C2CC2)c(F)c1 C#CC1(NC(C2CCOCCN2C(=O)C(O)C=CC)=O)CC(F)(F)C1 c1(C(=O)N)cnn2c(C)ccnc12.Cc1ccc(CC(=O)NC2CC2C)c(F)c1 N1(C(C2(CC#C)CCC2)=O)CC2(CCCC2NC(=O)CCC2CCOC2)C1 N1(C(C=C(C)C(F)F)=O)CCCC2(CCCN2C(c2nn(C)cc2C)=O)C1 c1(NC(=O)CN(C)C)ccccc1.c1(C(CC(=O)OC)NC)ccccc1.C Cc1ccccc1S(=O)(=O)NC(c1ccc(-c2ccccc2Cl)cc1)=O C1(CC(=O)NC)Cc2ccccc2NC1=O.C1CC(O)CN1C(=O)C=C1CCC1 C1(NC(COCCC)=O)CC12CCCCC2.c1(C=O)cc(S(C)(=O)=O)cs1.N CC1(C(=O)NC2C3CN(C(C4(c5ccno5)CC4)=O)CC23)CCCC1(F)F n1(CC(=O)NC2C3CC(NC(=O)Cc4ccsn4)CC32)nc(O)ccc1=O c1[nH]nc(SCC(=O)N(c2cnn(C3COC3)c2)C2CC2)c1.c1ccccc1.C c1(NCc2cc(C)no2)[nH]c(=NCC2CCCN(CC(F)F)C2)nc2sccc12 c1(CNC(C(C=C)O)=O)ncccc1CNC(c1c[nH]nc1-c1ccsc1)=O C1(NC(c2c(CC)occ2)=O)CCN(C(c2cn(CC)nc2C)=O)C1C1CC1 c1(C(=O)NCC(CC)NC(=O)C#CC2(C)CC2)cc(C)n(C)c(=O)c1 C1(CCCCNC(=O)C=Cc2ccsc2)CCCN(C(c2cc(O)cs2)=O)C1 C1(NC(C2(CC(F)F)CCC2)=O)CCCC1.C1(n2cccn2)(C(=O)N)CCC1 c1(NC(N=c2c(C)cn(CCS(CC)(=O)=O)[nH]2)=O)cc(Br)c(C)c([N+](=O)[O-])c1 C(C(CC(C)C)NC(c1nsnc1O)=O)NC(C1(CC#C)CCCC1)=O C(=O)(C(F)C(C)C)NC1CC(C(=O)NCC(C)(C2CC2)OC)C1 CS(C)(=O)=NCC(=O)NC1CC(CO)N(C(=O)CSc2nc[nH]n2)C1 c1(C(C)=O)cc(Cl)ccc1NC(C1CN(C(c2ccnnc2O)=O)CCC1O)=O CCC(C)C(CC(=O)NCP(C)(C)=O)NC(=O)Cc1cccn1C C(CC(C)(C)C)(C(=O)N1CCC(c2cnco2)C1)NC(c1nccc(CC)c1)=O c1(C(N2C(C3(NC(c4nsnc4O)=O)CC3)CCC2)=O)nc2c(s1)CCCC2 C1(CNC(C2C(C)(C)CC2)=O)COCCN(C(c2cccc(C(N)=O)n2)=O)C1 N1(C(C(C)OCC#C)=O)CCC(N(CC#C)C(c2cc(C(F)F)no2)=O)C1 c1(C(N2CCC(C(C)(C)NC(C(C)C(C)(F)F)=O)CC2)=O)cc2ccsc2n1C C(=O)(C1=CCCOC1)NC(c1ccccc1F)CNC(C1(C(C)(F)F)CCC1)=O C=CC(CCC)CC(=O)NC(C)C=CC(=O)NCCC(C)C(C)C N1(C(C2CCC(C)O2)=O)CC(NC(c2noc3c2CCCC3)=O)C2(CCC2)C1 N1(CC(=C)C)CCCC(NC(=O)CC2CCN(C(C)C(N3CCCC3)=O)C2)C1 C1(C=O)CN(C(=O)CC2CC23CC3)CC1.C1CCC1.C(C)(C)C.C=O.C N1(C(CCC)=O)CCC(F)(CNC(=O)C(c2ccccc2OC)OC)C1 C(=O)(C(O)CC(F)(F)F)NC(CC)CC(=O)NCC(c1ccsc1)O Fc1ccc(CN2CCCC(c3noc(C4CC4)n3)C2)c(F)c1Cl N1(CC(=O)OCC(=O)CCC2CC2(F)F)C(=O)c2ccc(O)cc2C1=O N1(C(CCc2ccn(C)n2)=O)C2CCC(C2)C1CNC(=O)CCc1ccsc1 Cc1cc(C(=O)NC2CC3(C2)CC3C(=O)NCCOCC(C)C)ccn1 CC1CCN(C(=O)CCSCc2ccccc2)CC1NC(C1(C)CSC1)=O NS(=O)(=O)N1CC(C(N2CCC(O)(C)C2)=O)C1.c1(C=O)cn[nH]c1.C1CC1 CC1(C(=O)O)CCN(CC(c2ccc(F)cc2Cl)O)CC1 CC1(C)CN(C(c2cnn3c2CCCC3)=O)Cc2c(Br)cccc21 C(=O)(C(C(C)(C)C)NC(=O)CCCC1CC1)N(C)CCC1CC1 c1(C(N(C)CC2CCCN(C(c3nc(C)sc3)=O)C2)=O)ccc2c(ccn2C)c1 CCCCCCC(CC)(CC)C(=O)NC1CC(C)C1.C1(C(=O)N)CC1C(F)(F)F CS(=O)(=O)CCCCN1CCCC1(c1ccccc1)CO c1(C(=O)NC2CC3CCC2CC3)c(Cn2cc(CCCO)nn2)nn2c1CCC2 C1(C(=O)NC2C(O)C3CCCC23)C2CCCC2CN1C(C1CN(C2CCC2)C1)=O c1(C(N2C3CN(c4cc(CC)ncn4)C(C3)C2)=O)c(Br)ccc(OC)c1F CC(CN(C)C(c1ccoc1Cl)=O)C(=O)NCCC(C)(C)N(C)C C1(CCN(C(C=C2CCN(C)C2)=O)C)CCCCN1C(C1CC1c1ccoc1)=O c1(NC(C(C)OC(c2[nH]cc(C)n2)=O)=O)ccc2c(c1)OCCO2 C1(CNC(C(C2CCCC2)OC)=O)CC(C(N2CC(C#N)C2)=O)CO1 Cc1cc(N2CCOC(C)CC2)nc(N2CCN(CC(C)O)CC2)n1 C1(NC(C2CCOC2)=O)CCCN(C(C2(CO)CC2(F)F)=O)C1 Cc1cc(C(N2CCN(C)C(CNC(C3(C)CSC3)=O)C2)=O)nc2[nH]nc(O)c12 n1(CC(=O)NCC(F)CNC(C2CCCO2)=O)cc(Br)cn1 C1(Oc2cccc(NC(C)=O)c2)CC2CC(CO)CC12 N1(C(C2C(OCC)C2)=O)CC2(C1)CN(C(C1CCCC1CC)=O)C2 C(=O)(C(C(C)C)C(C)C)NC1CCN(C(c2cc(C)cc(Br)c2)=O)CC1O C1CN(C(=O)C(C)n2cnnn2)CC(C)(C)O1.c1(COC)ccc(C(=O)N)s1 n1(CC(=O)N(C2CCCC2)C)c(C2CC2)nnc1S.C(=O)(C(C#N)C1CC1)N CC(C)(F)CCC(=O)NC1CCC(CCNC(=O)C(c2ccc(Cl)cc2)=O)C1 C1(N=[N+]=[N-])(C(N(CC(C)O)C)=O)CCN(C(c2ccncc2F)=O)C1 Cn1ccnc1C1OCCC1C(=O)NC(c1cn(CC2C3CCCC23)nn1)(C)C N1(C2CCN(C(C3(C)CC(=C)C3)=O)CC2)C2CCC1CN(C(c1csnn1)=O)C2 C1(C)(C(N2CCC(C)C2)=O)CCC(=O)N(C)C1.CC(O)C(C(=O)N)NC(N)=O Cc1ccc(C(N2CCCC(CCNC(=O)CC(=O)N(C)C)C2)=O)cc1Br c1(C(N2CC(CC)C(NC(c3ncoc3C)=O)CC2)=O)cccc(S(C)(=O)=O)c1 N1(C(c2ccc(C(N)=O)nc2)=O)CCN(C(=O)CC2COCCO2)CC1CCO C1(C(=O)NC2CC3(C2)CC3)(CC)CCCC1O.C(C(C)(C)C)=CC=O.N N1(C(C(C(C)C)OC)=O)CC2(CCC2)C1.c1(C=O)c[nH]nc1-c1ccc(Cl)s1.N C1(C(=O)Nc2ccc(F)cc2)CCC2(CCN(C(=O)C(O)c3ccco3)CC2)O1 C1(C(C)C)C(=O)N1.c1(C(N2CC(C(C)OC)C2)=O)oc(C(=O)OC)cc1C N1(C(c2nn(C)c(C(N)=O)c2)=O)CCC(F)C(NC(=O)C2=C(Cl)CCC2)C1 C(CCC(C)C(=O)NC1CCC(N(C(=O)CCC(C)N(C)C)C)CC1)OC c1cc(C2(C(=O)N(C)CCN(C)C(C3(C)C=CCCC3)=O)CC2)ccc1F.CO Cc1ccc(NC(C2(C)CN(C(=O)CCC3CCCC3)C2)=O)c(Cl)n1 N1(C(C(N(C(c2n(C=C)nnc2)=O)C)C2CC2)=O)CCN2CCCCC2C1 C1(CC)COC(C)CN1C(C12CCC(NC(=O)CCC(=O)C3CC3)(CC1)C2)=O c1(SC)nc(=NC(=O)N2CCCC(OCc3ccccc3)C2)[nH]s1 C(=O)(C(C)(C)CCCNC(c1ccncn1)=O)NC1CC(C)(CC)OCC1 N1(C(c2n(C)nc(Cl)c2)=O)CCC2(C1)CN(C(=O)Cn1cnnn1)CCO2 c1(C(=O)NCc2ccnc(OC)n2)ccc(S(=O)(=O)N(C)C)o1 C(=O)(CCC(C)(C)F)N1CC(C(=O)NC2C=C(C)CCC2)(SC)C1 CCCCCC(O)CC(=O)N1CC2CCN(C(=O)CC3(C)CCOC3)CC12 N1(C(c2c(CC)cccc2)=O)CCC(NC(=O)CCn2cnnn2)C(F)(F)CC1 C(CC(C)(C)C(=O)NCC1CC(SC)C1)NC(CNC(C(CC)C)=O)=O CC(C)(CS(C)(=O)=O)C(=O)N1CC2CC1C2NC(c1cc(Cl)ns1)=O C1(CC(=O)NC(CC)(C)C2CC2)CCN(C(=O)C(C)OCCO)C1(C)C Cc1cccc(CC(=O)NC(C2CCN(C(c3cc(O)ccc3O)=O)C2)C)c1Cl CC(C)CCCCC(=O)N1CCCC1C(C)(C)NC(=O)C(CO)NC(N)=O Cc1nc(CC(C)C)oc1C(=O)N(CC(C)O)CC.c1(C=O)nc(O)c(C)s1 Cc1ccc(CC(=O)NC2CC(C(=O)NOCCOC(C)C)C2(C)C)cc1 C1(COC)CCCN(C(c2cc(Cl)ccc2Cl)C)CC1 C12(C=O)CC1COC2(C)C.c1(SCC)ccccc1C(=O)N.C1(CC)CCC1 c1(CNC(C2CC(=C)CN2c2cc(COC)ncn2)=O)cccc2[nH]ccc12 c1(C(N2CCCC(NC(C(C)=C3CCC3)=O)C2C)=O)nc2ccccc2s1 C(=O)(C1CCc2ccccc21)N1C2CC(NC(C(C3CC3)OCC)=O)C(CC2)C1 CCCC(CC(=O)N(CC(F)F)C1CCC1)NC(=O)C(n1cc(C)cn1)C c1(C(N2CCC(CNC(c3ccc(CO)cc3)=O)C2)=O)cccnc1CO N1(C(C(C(CCC)NC(=O)C(F)(F)C(C)(C)O)O)=O)CC23CCC2(COC3)C1 CC1(CNC(=O)C(CCC2CC2)NC(c2nc(=N)cc[nH]2)=O)COCCO1 N1(C(C(C2CCCN(C(C(C(C)OC)N(C)C)=O)C2)(C)C)=O)CC2CC(C)C2C1 c1(C(=O)NCC=C)ccc(NC(c2ccc(Br)cn2)=O)cn1 Cc1cc(Cl)c(Cl)cc1C(=O)NC1CCC(C(=O)Nc2cccc(F)c2O)C1 N1(C(C(n2cc(Cl)cn2)C)=O)CCC(C)C1CNC(=O)C=CC1CC1 CC1CCC(C)(C(N2CC(CCNC(c3ccc(Cl)s3)=O)C2)=O)CC1 c1(C(N(C2CCCN(C(c3c(C)nn[nH]3)=O)C2)CCF)=O)ccc2ccsc2c1 c1ccc(Cl)c(Cl)c1.C1(NC(C2(OC)CC2)=O)CC(CC)C1.C(=O)(C)N CCC(C)CC(=O)N1CCC=CC1C(=O)NCCCC1CCOC1=O N1(C(C(C2CN(C(c3c(CC)ncnc3)=O)C2)O)=O)CCCC(C)(C#N)C1 C(CC(C)C(=O)NCC(C)(O)CNC(=O)CSCC(F)F)OC CCC(CCC(=O)N1CCC2(CSC2)C1)NC(=O)COCCCN(C)C C1(N(C(C2CC(=C)C2)=O)C)C2CN(C(c3ccc(C4CC4(F)F)cc3)=O)CC12 C(=O)(C#CC1(C)CCCO1)N1CC(C2CN(C(C3C(C)(C)CC3)=O)C2)C1 c1(NC(C2(c3nn[nH]n3)CCOC2)=O)ccc(C(F)C(F)(F)F)cc1 Cc1occ(C(F)(F)F)c1C(N1CCCC1CCCNC(=O)C(C)(F)F)=O S(=O)(=O)(c1ccccc1)N(CCCN1C(CCC)CCCC1)C(C)=O N1(CCN(C)C(C2CC(NC(C3CCCC3)=O)C2)=O)CCCC1 N1(C(c2c(C)cc(C)cc2Br)=O)CC(CO)C2(C1)CN(C(=O)C1=CCC1)C2 Cc1scnc1C(=O)NCCC(C)NC(=O)CN(C)C(N)=O c1(C(=O)N)ccc(N(C)C)c(C)c1.n1(C2(C=O)CC2)cc(C#CC)nn1.CC CC(C)(F)CC(=O)N(CCOC1CCCCC1)Cc1ccccc1.C(=O)(C)N C(=O)(C1CCCc2nnn(C)c21)N1CCC(NC(c2ccn(C)n2)=O)C12CCC2 N1(C(c2cc(C)ns2)=O)CC(C)(C)CC1CNC(c1ccc(F)cn1)=O C(CC(CNC(=O)CCSCC(C)C)NC(C1CCC(=O)O1)=O)OC N1(C(COCCOC)=O)C(C)CC2CCCC12.C1(=CC=O)CCC(C)C1.N C(C(CNC(c1scnc1C)=O)S(C)(=O)=O)NC(c1c[nH]c(=NC)s1)=O CC1CC(NC(=O)CC2(C)CCCC2)CN(C(c2ccnn2CC(F)(F)F)=O)C1 CC1(C)CN(C(c2sccc2C(F)F)=O)CCN(C(=O)C(C)(C)CC#N)C1 C(=O)(CCCCN(C)C)NC(C1(CNC(C2(C#C)CCC2)=O)CC1)C CCCC(O)CC(=O)NCC12CC(CO1)N(C(=O)Cc1ccc(Cl)nc1)C2 N1(C(c2cc(OCC)ns2)=O)CCCC2(CCN(C(=O)C=O)CC2)C1.C1CC1.N c1(OC)cc(F)c(C2CC2)cc1-c1ccc(CNC(c2ccccc2C)=O)nc1 CC1CN(C(=O)C(CNC(c2ccn(C(F)F)n2)=O)CC2CC2)Cc2c[nH]nc21 C1(CCCC)CCN(C(C2CC(NC(=O)C(C)SC)C2)=O)C1 c1(C(N(C2CCCSC2)C)=O)sccc1CNC(=O)COC1CCOC1 N1(C(c2c(C)ccs2)=O)CC2CC(CNC(C3CCC(C(C)C)CC3)=O)C2C1 c1(CNC(C2OCC(C)(C)C2)=O)cc(Cl)ccc1OC(F)F N1(C(=O)COC(F)(F)F)CCCC(O)(CCNC(C2(CCF)CCC2)=O)C1 C=CCCCCCNC(=O)CC(C)(C)NC(c1n[nH]c(C)c1C)=O N1(C(CCC2C(C)=NOC2=O)=O)CCCCCC(NC(=O)CCCCC(N)=O)C1 c1(CC(N2CC(C(=O)NCC(C)(C)O)SCC2)=O)cccc(Cl)c1F Cc1c(C(=O)NCC2CC(CNC(c3n[nH]c4c3CCC4)=O)CO2)cccc1N Cc1ncc(NC(=O)C(C)CCN(C)C(c2ccccc2)=O)cc1Cl C1(NC(CS(CCC)(=O)=O)=O)CCC2CN(C(c3[nH]ccc3C)=O)CC2C1 N1(C(C2(C(C)C)CC2)=O)CCC(C)(NC(c2ccc(C3CC3)cc2)=O)CC1 c1(C(N2CCC(n3cc(-c4c(C)ccs4)nn3)C2)=O)nc(Br)sc1C N1(C(CC2(C)CCN(C(C3(C(N)=O)CC3)=O)C2)=O)CCc2ncsc2C1 C1(CC)CN(C(c2ccc(F)c(CN(C)C)c2)=O)CCN1C(=O)CCCF C1(F)(CNC(c2nc(Cl)sc2Cl)=O)CCCN(Cc2cnco2)C1 C1(CC=O)CCC(F)(F)CO1.c1(C(=O)NC(C)CC)cnn(CCN(C)C)c1 C(CCC(=O)NC1(CC)CC1)NC(=O)OC.C1(C=O)CCCC1C(N)=O CCC(C)C(C(=O)NC1CCCN(C(C2NC(=O)CC2C)=O)CC1)N(C)C c1(CN2CCC(C(N3CCCC(F)CC3)=O)CC2)cc(F)ccc1Cl CC(C)(C)CCC(F)C(=O)N1CCC(C)(NC(=O)CC2COCCOC2)CC1 CCC(CCOC)C(=O)NC1C2CCN(C(c3cccn3CC)=O)C12 N1(C(C(CC)N2CCCC2=O)=O)CCC2(CC1)CN(C(C1(C(N)=O)CC1)=O)C2 N1(C(c2c(SC)cnn2C)=O)CCC(NC(C2(O)COC2)=O)C(CO)C1 c1(C(N(CCOC)CCOC)=O)sccc1CNC(C1CC1F)=O N1(C(C2CC2C2CCC2)=O)CC2(C(N3CCCC34CC4)=O)CC1CCO2 c1(C(=O)NC2CC(NC(C=CCCC)=O)C2)cn(C)nc1C(C)C n1(CCCC)nnnc1C(C1C2COCC12)(C)Nc1cnoc1 N1(C(C(CCC2CCC2)NC(c2c(C)n[nH]c2)=O)=O)C2CCCC1CC2 CCC(C)CCCCC(=O)N(C)CC1CCCCN1C(=O)C1=COCCC1 C1(C(N2CC(OC)C(C)C2)=O)CN(C(=O)COCCCF)CC(C)(C)C1 Cc1oc(CO)cc1C(=O)NCC1CCC1NC(=O)CCc1nncn1C C1(C=O)CC2(C1)CC(F)(F)C2.C1CCCC1.CC(C(=O)N)OCCN(C)C c1(C(N(C)CCOCC)=O)cnc2[nH]ccnc1-2.C1(N(CC=O)C)CCCC1 C#CC1CCN(C(=O)C=CC(C)(C)NC(c2ccnnc2C)=O)CC1 c1(CC(=O)NCC2CN(C(CC(=C)Br)=O)CC2C)cc(Cl)ccc1O c1(C(N(C2CCN(CC(=O)NCCc3cccs3)CC2)C)=O)cn(C)ccc1=O c1(CNC(C2CCC(OC)C2)=O)cnn(C)c1C(=O)N(C1CN(C)C1)C c1(CCC(N2CC(NC(C3N(C)C(=O)CCC3)=O)C2)=O)nc2cccc(F)c2[nH]1 c1(N2CCC(NC(C3CCN(C4CCCC4)CC3)=O)C2)ncc2sccc2n1 c1(C(=O)NCCC(C)(C)NC(C(C(C)SC)O)=O)cnn2ccn(C)c12 Cc1cc(CC(=O)NCC2CCCCC2NC(c2ccnc(S)c2)=O)n(C)n1 C1CC2(CN1C(=O)C=Cc1ccc(F)cc1)CC2(F)F.C(C(=O)N)N(C)CC C(CCCCC(=O)N1CCC(C(C)(C)NC(=O)C(C)COCC)C1)=CC C(=O)(C1=NOC(C)C1)N1CCC(C(C)C(=O)NCCc2nccc(O)n2)CC1 C(=O)(CCCC(=O)N1CC=C(C(=O)N2CC(O)C(F)C2)C1)N(C)C c1(C(=O)NCCNC(COCc2ccc(OC)cc2)=O)ccc(=N)[nH]c1Cl CC1CC(C(=O)NCC2COCC(C)O2)CN(C(=O)CC2CC3(CC3)C2)C1 C(CN=c1[nH]c(=NC(C)CSCC(C)C)[nH]c2cccnc12)NC(CC)=O C1(C(N2C(CNC(c3cnc(SC)nc3)=O)CC(OC)C2)=O)CC12CCSCC2 C(=O)(CN=c1[nH]c(=NCC(C(C)C)C(C)C)[nH]c2c1CSC2)N(CC)CC C(=O)(C(C)(C)CC(=O)NCCCOCCN(C)C(c1cnoc1)=O)OC CCC(C(=O)NC1CCCC1NC(=O)Cc1cncs1)C(C)(C)CC CCCCCC(O)C(=O)NCC(C)CNC(c1cccc(SC)c1Cl)=O Cc1noc(N)c1C(N1CC(C(=O)NCC2(O)CCOCC2)C(F)C1)=O N1(C(c2cc(OC)no2)=O)C2CCC1CN(C(c1cc(C)ccn1)=O)C2 C1(NC(c2cc(C)n(C(C)C3CC3)n2)=O)CN(Cc2nccs2)CCC1C C(=O)(CCCCC(N)=O)NC(C)C(CO)NC(=O)Cc1ccc(C(N)=O)cc1 c1(OC)ncnc(C)c1C(=O)NC1CCN(C(=O)C(=Cc2ccco2)C)CC1C C(=O)(CC(CC)C1CC1)N1C(C(=O)NCC(C#C)OC)CSC1 c1(C(N(CCC(=O)NC2CC(=O)NC2)C2CC2)=O)coc2ccccc12 N#Cc1ccccc1CNC(C12CC1CCN2C(c1cn(C2CC2)nn1)=O)=O c1(C(=O)NCCCNC(=O)Cc2ccc(O)nc2)cc([N+](=O)[O-])cc(Cl)c1Cl S(=O)(=O)(c1cccnc1N)NCc1cnn2ccn(C)c21.C1CC2(CC2)CO1.C CC(C)CC(C)(C)C(=O)N1CC(C(N2CCC(C#N)C2)=O)C(F)C1 N1(C(CC(=O)OCC)=O)CCC2(CC1)COCC2.C1(C=O)CC1CC(C)C.C C(=O)(C(O)C(C(C)C)OC)N(CC(=O)NC12CCCC1C2)CC N1(C(C(CCC)NC(C)=O)=O)CCC2(CCCN(S(=O)(=O)CCCCCl)C2)CC1 C(=O)(CCCCCSC)NC(C(N1CCC(C)(COC)C1)=O)CCC1CCC1 c1(C=O)ccc(O)c(Cl)n1.c1(C(=O)NCC(=O)NC(C)CC)cccnc1.N N1(C(CCC#CC)=O)CCC2CCCC12C(=O)NC1C(C)CCCC1C C1(C)(C(=O)N)CN(C(C2CCSC2)=O)C(C)(C)C1.C1(CCOC)(C)CC1 C(CCNC(=O)C(=O)NC(c1ccc(F)cc1)CF)(C(C)C)OC N1(C(c2c(CC)noc2)=O)CCN(C(=O)C(Cl)=CCl)C(CC(C)(C)C)C1 c1(-c2ccn(CC)n2)nc(CSc2ccccc2)nn1CC1CCCO1.C1CC1C C(C#CC(=O)NCC(F)CNC(c1cc(C)nn1C1CC1)=O)OCC.O Cn1cnc2c(NCCC3(F)CCCC3)nc(Cl)nc12.C12CC(C1)CCNC2=O CC(C)CN=C(NC1CC1)N1CCC(CC2(CN3CCC3)CC2)CC1 c1(C(N2CCC(NC(CN(CCC#C)C)=O)C(C)C2)=O)ccc2c[nH]nc2n1 S(=O)(=O)(CCC(=O)NCC(O)CNC(=O)Cc1nc(=N)[nH][nH]1)NC N1(C(Cc2ccc(SC)cc2)=O)CCC2(CCCN2C(=O)C(C)NC(N)=O)C1 CC(C)(C(=O)N1CC(O)C(O)C1)C1=CCN(C(=O)Cn2ccnc2)C1 C(=O)(C(C(=O)NCCN(C(=O)C(C1CCOCC1)F)C(C)C)OC)OC c12cccnc1C1CCN(CC1)C2.C1(NC(=O)OF)CCN(Cc2ccccc2)C1 N1(C(c2c(OC)nccc2)=O)C2CC1CN(C(c1cc(C)cc(Cl)n1)=O)C2 C1(NC(COCCOCC#C)=O)CN(C(C2CC2(C)C)=O)CC1CO N1(C(CC#C)=O)Cc2ccccc2C1C(=O)NCc1cccc(F)n1 Cc1c(C(N2CCC3CCN(C(C4CC=CC4)=O)C3C2)=O)[nH]c2cc(F)ccc12 Cc1cc(CNC(=O)NNC(=O)C2CCC(=O)N2)c(C)n1-c1ccnn1C c1(C(=O)OC)c[nH]c2cc(NC(C3CCCC(=O)C3)=O)ccc12 c1(Cn2cc(CCSCC)nn2)cccc2nonc12 c1(C(=O)NCC2C(NC(c3ccc(C)cc3)=O)C2)cc(C#N)cc2ccccc12 C1(F)(C(=O)NC2C(C)CCN(C(C3(C#C)CCC3)=O)C2)CCC(F)(F)CC1 c1(C(=O)NC2CN(C(CCCCC#C)=O)CC23CC3)ccc2ccccc2c1Br C1(NC(c2conc2C(F)(F)F)=O)CCN(C(=O)C(F)C(F)(F)F)CC1C N1(C(=O)OCc2ccccc2)CCC2CN(N3CC3c3ncco3)CCC12 c1(CNC(CNC(CC)=O)=O)ccc(C(=O)N(C)CC2CCN(C)C2)cn1 CC1CCC(CC(=O)NC2CCCCC2NC(C2CCCN2C)=O)CC1C N1(C(CC(CC)OC)=O)C2CCC1C(C(=O)NCCCc1ncc[nH]1)C2 CN(C)S(=O)(=O)N(C)CC(=O)NC.C1CC2CC2N1C(=O)CC.C1CCCC1 C1(C)(C=O)CCC(C)C1(C)C.C=C(Cl)C(C)(C)C(=O)NC(C)C(C)(C)C.N c1(NC(C2CCC(NCc3n(C)ncc3)C2)=O)ccc(I)cc1C#N C1(CNC(CCN(C)CC)=O)CCCC(NC(=O)C(C2CCOCC2)C)C1 Cc1noc(C2OCCC2NCCc2ccsc2Cl)n1 CC1CN(C(=O)CCC(C)(C)F)CCC1N(C)C(c1cc(C(F)F)no1)=O C1(C(=O)NCCC(C)N(C(C(C)OCCC(C)C)=O)C)CC1C1CCCCC1 c1(C(=O)NCC2(CNC(COCC)=O)CC23CCC3)ncc(Br)cc1C CN1CCN(CC(N2CC(F)CC2C(N2CCCCC2CCCO)=O)=O)CC1 C1(C)(C(=O)NC2C(CNC(C3(C)CC(F)C3)=O)CCCC2)CCNC(=O)C1 c1(CCC(=O)NC2C(CC=C)CCCC2)ccc(F)c(OCCCN(C)C)c1 N1(C(Cc2nc(C)oc2)=O)CCC2(CCCN2C(=O)Cn2cc([N+](=O)[O-])cn2)C1 N1(Cc2ccc(OCC)c(-c3ccc(C)o3)c2)CCC2(O)CCCCC2(O)C1 N(C1CCCc2cccnc21)(C(C1(OC)CCCCC1)=O)CC C1(OC)CCN(C(=O)CNC)C1.C1(C(F)(F)F)(C=O)CCC1.C1CC1.C N1(C(CC2CC(OCC)C2)=O)CCC(CCC(=O)NCc2cnc(C)cn2)CC1 CC1C(NC(c2cccc(C(F)(F)F)c2)=O)CCCN1C(=O)C=C1CCSCC1 C#CCCCC(=O)NC1(CCNC(=O)C=Cc2cocn2)CCC1 N1(C(C(C)Cc2ccco2)=O)CC(O)C(O)C1C.n1(CC(=O)N)cccnc1=O c1(CC)c(C(=O)NCCNC(=O)CCC2CC3CCC2C3)nnn1C O=C1CCc2ccc(C(N3CCCN(C(=O)Cc4ccccc4)CC3)=O)nc2N1 c1(Oc2cccc(C(N3CCC(CN4CCCCC4)C3)=O)c2)cccc(Cl)c1Cl C(=O)C(CC)(CC)CC.C(=O)(C(F)C(=O)NCC1(C)CCOCC1)OCC c1(N(CCCNC(c2c(C)noc2)=O)C)nc(C(C)(C)C)ccc1C#N N1(c2nnc(C)s2)CC2CC(NC(c3c[nH]c4nccc-4c3)=O)CC2C1 C(=O)C=CS(F)(F)(F)(F)F.C(C)(C(=O)NC1(CCC)CC1)OCCCC.N C(=O)(C(O)CC(F)F)N1CCC(CCNC(C2C3(CC3)C23CC3)=O)C1 C(=O)(C(C)(COC)COC)NCC(CO)NC(COCCC)=O c1(NC(c2c(CCO)cn(-c3ccc(C)cc3)n2)=O)c(O)cccc1Cl N1(C(C2(NC(c3cscn3)=O)C(C)C2)=O)CCCC(O)(CO)C1 c1(C(C(C)OC(c2ncn(CC)n2)=O)=O)ccc(C)cc1 c1(N2C(c3ccc(F)cc3)CC2)cc(C2CC2)nc(C2CC2)n1 c1(C(N2CCC(CCCNC(CC(C)F)=O)CC2)=O)cc(F)cc2nccnc12 C(=O)(C(C(Cc1ccccc1)OC)N1CC(C)=CC(C)C1)NCCCC Cc1cc(C(N2CC(NC(=O)C(F)C(C)(C)O)C(n3ccnn3)C2)=O)nc(O)n1 N(C1CC2(CCOCC2)Oc2ccccc21)C(=O)NC(CC)CSC C(=O)(CCNC(=O)C(C)N(C(c1cc[nH]n1)=O)CC)NC(CC)C CCCCCC(O)C(=O)N1CC2CCC(C(=O)N(C)Cc3ccc(O)cc3)(C2)C1 C1(C(=O)NCC2(O)CCN(C(c3cc4sccc4s3)=O)C2)CC2(CCCC2)CO1 C1CCN(C(=O)CC2CCC(O)C2)C1(C)C.c1(C(=O)OC)ccnc(C=O)c1.N C=CCC(CNC(=O)Cn1cnnc1O)C(=O)NCc1ccoc1C c1(C(=O)NC2C(NC(C(c3ccc(F)cc3)OC)=O)CCC2)ccc(=N)[nH]c1Cl N1(C(c2cc(C)c(C)o2)=O)CCC(N=[N+]=[N-])(C(=O)NC2(CO)CC(O)C2)C1 N1(C(Cn2cc(CN(C)C)nn2)=O)CC2CC2(NC(=O)CC2CCSCC2)C1 C=CCC(F)(F)C(=O)N1CC(C)C(C)(CNC(=O)CCCCCOC)C1 C1(N(C(C2C(C)CN2C(c2cnc(O)nc2)=O)=O)C2CC2)CCC(=O)N(C)C1 c1(C(=O)NC(C)CCNC(=O)C(F)(F)c2ccccn2)ccc2nnnn2c1 C(=O)(CCCCNC(C)=O)N(CCC(=O)NC(C1CCOC1)C#C)CC#C C1(NC(C(CC=C)C)=O)CCN(C(=O)CCCCC(=O)OC(C)(C)C)CC(O)C1 C(=O)(C(C)C(O)C(C)C)NCc1c(C(N(C(CC#C)C)C)=O)[nH]cc1 CC(C)(C(=O)NCC1CC1)c1cnsc1.C(=O)C(Cc1ccccc1)C1CC1 C1(OC(C(c2cccc(C)n2)(F)F)=O)C(=O)NCC12CCOCC2 C1(C(N2C(C(C)C)CCC2C(=O)NCc2cn(CC)nn2)=O)CC2CCCC2C1 C1(NC(C(C#N)C2CC2)=O)CCCC12CN(C(c1c[nH]nc1Br)=O)C2 CS(=O)CCC(=O)NC1(CNC(=O)CCC(=O)c2ccncc2)CCC1 O=C(O)CC1CN(Cc2nc(C3CCCCC3)cs2)c2ccccc21 C(=O)(CCCCCF)N1CC2C(CNC(C(c3ccc(C)s3)C)=O)C2C1 c1(C(=O)NCC2C(C)CCN(C(c3cc(Cl)no3)=O)C2)ccnc2ccncc12 Cc1nc(N2CCC(C(=O)NC3CCSC3)CC2)nc(O)c1C C#Cc1ccc(F)c(CNCc2cnn3c2NCC(C)C3)c1F N1(C(C(C)CC(N)=O)=O)CC(NC(=O)Cc2ccc(C(F)F)cc2)C(N=[N+]=[N-])C1 c1(C(=O)NC2CC(CO)C23CCC3)ccc2c(c1)nc(O)n2Cc1ccccc1 c1(NC(C(CC)(C)C#N)=O)ccc2c(c1)C(=O)OC2 Cc1cc(F)c(C(=O)NC(CO)C(C)NC(c2cnn(C)c2Br)=O)c(F)c1 C1(NC(C(C(COC)C)C)=O)CC2CCC1CN(C(C1CC(OC)(OC)C1)=O)C2 C(C(C)(C(=O)NC1CNC(=O)OC1)NC(C1CCCC(=O)N1)=O)SC N1(C(CCCNC(=O)OC)=O)CC2CC1C2NC(=O)CCC1CCCC1 Cc1cc(Cl)ccc1C(N1CC(NC(c2nc(Cl)ccc2F)=O)CCC1C)=O C(=O)(C(F)(F)C(F)(F)F)NCCCCCNC(c1cnnn1-c1ccccc1)=O Cc1cc(Cl)ncc1NC(=O)CC1CCN(C(=O)Cc2csnc2C)C1 C1(C(C)NC(=O)CC2CCN(C)C2)CCN(C(=O)CS(C)(=O)=O)CC1 c1(CNC2CC(NC(c3ccc(CO)cn3)=O)C2)ccnc(-c2ccccc2)c1 C1(C(=O)NCCC(=C)CNC(=O)C=CCN2CCOCC2)C2CCCOC12 CC1(C)CCOC1CCNC(c1coc(CNC(=O)Cc2ccon2)c1)=O C1(NC(CC(C)c2ccncc2)=O)CN(C(c2cccnc2Cl)=O)CC1(C)C N1(C(C(CC=C)OC)=O)CCC(CNC(=O)CCCC2CCC2)C1(C)C C1(C(=O)NC(CNC(CN2CCC(C)C2)=O)(C)C)CCc2cn(C)nc2C1 C1(NC(c2ccccc2-n2ccnn2)=O)CC2(C1)CC2.C1(C=O)CC1(F)F.N c1(CNC(C2(CNC(=O)Cc3csnn3)CC(=C)C2)=O)cccc(O)n1 c1(C(N2CCC(SC(F)F)C2)C(=O)NCCC)cccc(OC)c1 c1(C(=O)OC)cc(NCC2CC3C(C2)C3(F)F)cc2c1OCCO2 C(C(CC(F)(F)F)NC(c1ccsc1Cl)=O)NC(C1CCN(C)C1=O)=O CC(F)(C(=O)NCC1(O)CCN(C(c2cc(Cl)ccc2Cl)=O)C1)C(F)(F)F c1(C(=O)NC(c2ccc(Br)cc2)CC(=O)OC)cncc(S(N)(=O)=O)c1 c1(CC)cc(Cl)ccc1NC(c1nc(Br)ccc1OC)c1nnnn1CCOC c1(C(C(=O)NC2CN(C(=O)CC3(OC)CC3)C2)OC)ccc(F)cc1 C1(C(N(CCCC=C)CC)=O)CCN(C(c2ccncc2N)=O)CC1C Cc1ccc2nc(Cn3cc(COC4(C(=O)O)COC4)nn3)cn2c1 c1(SCC(=O)NCCC2CCCN(C(C(CC#C)O)=O)C2)cc(C)ccc1C c1(CC(=O)NC)ccc(C(=O)N)cc1.C(c1cccnc1)=CC=O.C1CCC1 C1(NC(c2cccc(F)c2Cl)=O)CCC2(CC1)CCN(C(C1CCCCS1)=O)C2 Cc1nc(C)c(C(=O)N(C2CCC2)C)s1.c1(-n2ccnn2)cccc(C(=O)O)c1 CC1C(NC(c2cncn(C)c2=O)=O)CC2CCC1N2C(=O)Cn1ncnn1 C(=O)(N=c1nn[nH]n1Cc1ccccc1)N1CCCC(C(C)(C)O)C1 C(CCS(N)(=O)=O)C=O.C1(C(=O)OC(C)(C)C)CCN(Cc2ccncc2)CC1 C#CC1CN(C(C2CC23CCCC3)=O)CCN1C(=O)CSC(C)C C1(NC(C(C(CC)C)O)=O)CC2CCC1CN(C(=O)CCCc1ccccn1)C2 c1(OC)cc(C)c(C(N2CC(NC(c3ccc(F)cc3N)=O)C2)=O)cc1Cl C1(CC=C)(C(=O)NCC#CC2CC2)CCCN1C(=O)CC(C)N(C)C c1(C(N2CCCC(CN(C(=O)CC(C)(F)F)C)C2)=O)cnn2ccn(C)c12 c1(OC)ccccc1C=CC(=O)NCC(C)(CO)NC(C1CCCN1N=O)=O N1(C(c2ccc(OCC)cn2)=O)CC2(CCCN(C(C3CC3(C)CC)=O)C2)C1 Cc1cc(C(CO)NC(=O)NCCC(=O)NCc2ncc(Br)s2)cc(F)c1 N1(C(CN(CCC)C)=O)CCN(C(=O)C(C)n2ccnc2)C(c2nccn2C)C1 CCCCCCCCCCCNCC1(C)CCCCC1 CN1CCN(C)C(CN=C(NC2CC2)NC2CCC2(C)C)C1 Cc1ccc(NC(C2CCOCC2NC(C2(CO)CC(C)(C)C2)=O)=O)cc1O C1(CC(=O)NC(c2ccccc2Br)C)CCN(C(=O)CCc2ncc[nH]2)CC1 CCCCCCCCNC(N1CCC(C(=O)Nc2ccc(CO)c(OC)c2)C1)=O C1(NC(c2cc(C(=O)OCC)n[nH]2)=O)CC(C)CN(C(c2cncs2)=O)C1 Cc1cccc(Br)c1C(N1CCOCC(NC(c2nnccc2C)=O)C1)=O C(=O)(CCCCC(=O)NCc1nnn(C)c1C=O)NC.C(C)(C)CN(C)C N1(CC(=O)N)CC(C)N(C)C(C)C1.c1(CC(=O)N(CC)CC)ccccc1 C=CCCC(C)(C)C(=O)N1CCC(OC2CN(C(=O)C(O)C(C)OC)C2)CC1 C(COC(C)C)(C(=O)N1CC1)NC(COC)=O.CCN(C)CC.O Cc1nc(C(=O)NC2CCCC(CNC(=O)CS)C2)nn1C.c1cccs1.C Fc1ccc2cc(Cl)nc(NC(C(F)(F)F)C3CCCNC3)c2c1 C1CN(C(C2CC2(C)C)=O)CCN1C(=O)Cc1ccc(C(C)=O)cc1F.CO.C N1(CC)CCCC2C1CCCN2C(=O)NCCC1CC12CCOCC2 c1(C(N(CC=C)Cc2cscn2)=O)cccc(SC)c1[N+](=O)[O-] C1(C(N(C)CCNC(=O)CCc2ccsc2)=O)CC(=O)OC1(C)C Cn1nnc(CNC(=O)C(O)C2CN(C(=O)CCN3CCOC3=O)C2)n1 N1(C(C(C)CC2CC2)=O)CC2CCC(C1CO)N2C(c1snc(Cl)c1Cl)=O c1(NC(C2CCCC2)CC)cc(N2CC(CSC)CC2C)ncn1 N1(C(C)=O)CCCCC1CC(N1CCC(CN(C(=O)CN(C)C2CC2)C)C1)=O N1(C(C2(C(C)(C)C)CCC2)=O)CC(NC(c2c[nH]c(=N)o2)=O)CC2(CCC2)C1 Nc1cc(Cl)ncc1C(=O)NCC1CC2CN(C(C3(CF)CCOCC3)=O)CC12 C1(NC(c2cscn2)=O)CC2C1CCN2C(=O)Cn1cnc([N+](=O)[O-])c1 CCC(C)C(O)CC(=O)N1CC(CCn2cc(C(C)(C)CCCOCC)nn2)C1 c1(C(N2CCN(C(c3ccc(O)nc3)=O)CC2CO)=O)cnc2ccccc2c1 n1(CC)ncc(C(=O)NCc2cnc(C(C)(F)F)s2)c1Br C1(C(=O)NCC2(C(N)=O)CN(C(c3cc(C)sc3)=O)C2)CCCCC1O N1(C(=O)C=CCn2cncn2)CC(C2CCCCN(C(=O)C3=COCCC3)C2)C1 c1(C(=O)NCC2CN(C(C(C)=C3CC3)=O)C2)cnc2cc(C)ccc2c1 CC1(C)CCCN(C(C2CC23CCN(C(C2CC4CC(=O)C2O4)=O)C3)=O)CC1 N1(C(c2cnc(C)s2)=O)CCC(NC(=O)C(C)(C)c2ccno2)C(CO)CC1 N1(C(C23CC(CN(C(=O)CCCn4cccc4)C2)C3)=O)CCC2CCC(O)C1C2 C1CC2CCC(C1)N2C(=O)Cn1cc(S(C)(=O)=O)cn1.C(C=O)N(C)CCO N1(C(C(=O)NC(CC)CC)C)CCCC1(C)CCCO C1(C(=O)NCCC(C)N(CCC)C)CCN(C(c2snnc2C)=O)C12CCC2 C(=O)(C1=NOC2COCC12)N(CCCNC(C1CC2(C1)CC2F)=O)C C1(CC)CCC(C(N2CC3CC2(COc2cn(C)nc2Cl)C3)=O)CC1 C1(NC(c2c(F)cccc2Br)c2n(C(CC)(C)C)nnn2)CC(C)(C)OC1=O C1(CNC(=O)NCC(C)Cc2cccs2)COC(=O)O1 C(CC(CNC(C1CSCCS1)=O)NC(c1ccc(C(C)=O)[nH]1)=O)OC c1(C(=O)NC(C2CCN(C(c3c(C)nc[nH]3)=O)C2)C)cc(O)cc(Cl)c1 c1(SCC(=O)N(C2CCN(C(=O)CC3CC3)C2)C)ccccc1Cl C=C(Cl)CCC(=O)NCC1CCCN(C(c2ccn(-c3cccc(Cl)c3)n2)=O)C1 N1(C(C2CC3(CC(=O)C3)C2)=O)CCC2(CC1)CN(C(=O)C1=CCCOCC1)C2 C1(CC)(C)CCOCC1.C1(C(=O)N)CCC(O)C1.c1(C=O)ccc(C(F)F)o1 C1(OC)CCOCC1NC(C1CCC(n2cc(-c3ccccc3F)nn2)C1)=O C(C(CNC(=O)C(CC(F)F)C1CCC1)C(F)(F)F)NC(c1n(C)nnc1)=O N1(C(C#CC(=O)O)=O)CCC2C1CCCN2C(c1ccc2nncn2c1)=O C1(NC(c2cnc(OC)nc2C)=O)CC2CCC(C1C)N2C(=O)CCCCF N1(C(c2cc(OC)nc(Cl)c2)=O)CCC2C(C1)CN2C(=O)COCCSC c1(C(=O)NC2C=CC(CNC(C(C(C)C)F)=O)C2)cc(Br)c(O)cc1F N1(C(C(CC)=CC)=O)CC2CCCC(C)(C2)C1.C1(C(=O)N)CCCN1C=O N1(C(C2(CO)CCOC2)=O)CCC2(CC2C(=O)Nc2cccc(O)c2)C1 N1(C=O)CC2C3COCC3C2C1.c12cccc(c1)C(=O)N(C)C2=O.C(C)(C)C.O C1(C(=O)N(CC(=O)OC)C)(COC)C=CCN1C(=O)CCCC1CC1C CCCCC(O)CC(=O)N1CCN(CCCNC(=O)CCC(C)(C)C)CC1 C1(C(=O)NC2CN(C(c3cnc(C(C)O)s3)=O)CC2C)CCC(=O)C(C)C1 N=c1[nH]c(CCC(=O)NC2(C)CC(NC(C3CNC(=O)N3)=O)C2)cs1 N1(C(c2nc(C(CC(C)C)N)sc2)=O)CCCCC1C(F)(F)F c1(C(N2C(CC)CCC2)=O)cccc2c1NCC2.C1(C(=O)N)(OC)CC(C)(C)C1 CCC(CC)C(C)C(=O)N1CC(CNC(c2cc(Br)cc(C)c2N)=O)C1 c1(C(=O)NC(C(=O)NC(CC#C)CC(F)F)(C)CO)cnn2cccc2c1 N1(C(C2C(C)OCC2)=O)CCC2(CC1)CCN(C(c1scnc1C1CC1)=O)CC2 c1(C(=O)NC(CNC(CC(C=C)CCC)=O)C)cnc2cc(C)ccn12 c1(C(N2CCCC(NC(CC(CC)C3CC3)=O)CC2)=O)cccc([N+](=O)[O-])c1 N1(C(C(CSC)C)=O)CCN(C(=O)CSc2nnnn2C)C(c2ncc[nH]2)C1 N1(NC(C(c2ccn(C)n2)C)=O)CCN(CCc2nnnn2C2CC2)CC1 n1(CC)nc(C)cc1C(=O)N(CCC(C)NC(=O)CCOCC1CC1)C N1(C(C(C)OCCC#C)=O)CCCCCC(NC(=O)Cc2ccc(Cl)cc2F)C1 N1(CCOC)CC(NC(C2(CNC(c3ccsc3C)=O)CC2)=O)CC1=O C1(C=O)CCS(=O)(=O)N1.CC(C=O)NC(=O)C1CC1.C1(CCC)CC1.N c1(OC)ncc(Br)cc1CNC1CCC(N(C)C)C1 C1(OC)CCCC(C(=O)NC(C)CCN(C)CCC)C1.c1ccc(C(=O)N)cn1 CC1CC(C(=O)N(C)CC2(C)CC2)CC(C)O1.N1(CCC=O)CCOC1=O.N c1(CCC(N2C(c3onc(C)n3)CC(O)C2)=O)cc(Br)cc2c1OCC2 c1(C(=O)NC(C2(O)CN(C(c3ccc(F)s3)=O)C2)C)csc(C(F)F)n1 Cc1nc(N2CCC(CCNC(=O)C(C)Cc3cnc[nH]3)CC2)cc(O)n1 C1(NC(C(COC)O)=O)CN(C(c2[nH]ccc2C2CC2)=O)CC1OC C1(NC(=O)C=Cc2cscn2)CC(=O)NC1.C1CN(C(=O)C=CCF)C1.C C1(C2CC2)CCN(C(=O)C(CO)C(C)(C)C)C1.Cn1nc(C(F)F)cc1C(=O)N c1(C(=O)NCC23OCC(NC(CC)=O)(C2)C3)c(N)sc(C)c1C C=CC(C)(CC)C(=O)NC(C)C(CO)NC(=O)C(c1ccccc1)N(C)C C1(C(=O)NCCCC(C)(C)NC(=O)CSc2ccccc2)Cc2ccccc2S1 N1(C(C(C2CN(C(C3(F)CC=CCC3)=O)C2)OC)=O)CCN(C)CC1C c1(C(N2CCN(Cc3ccco3)CC2)C(=O)NCC2CC2)ccc(Br)c(F)c1 CC1C(NC(c2ccc(Cl)cc2Cl)=O)CCCN1C(=O)CCc1ccc(=N)[nH]c1 C1(CC)CCN(C(=O)C(C)(C)NC(c2c[nH]nc2C)=O)C1C Cc1oc(C)c(C(=O)NC2CCCN(C(=O)CCCc3nncn3C)CC2)c1C c1(CNC(C(C(C)O)NC(C(CC)SC)=O)=O)cnnc(C)c1C C1(C(C)C)CN(C(=O)C(O)CNC(=O)CC2CCC(=O)N2C)CCO1 c1(C(=O)NCC=C2CCN(C(C(C)C(F)(F)F)=O)CC2)cnn2ncccc12 C1(CC(C)C)C(=O)N1.c1(NC(c2cc(COC)no2)=O)cc(C)cc(Cl)c1 N1(C(C(C(CC)O)C)=O)CCC2CCC(C1)N2C(c1nc(OC)ncc1Cl)=O C(=O)(C1CCCn2cnnc21)N1CC(CNc2c(C#N)cccn2)OCC1 c1(C(=O)NCC(C)(O)C2(C)CC2)sccc1C.C(=O)C(C)(O)C1CCC1 C(=O)(CC1C(=O)Nc2ccc(Cl)cc21)NC(C)CNC(=O)Cc1ccnnc1O C(=O)C#CC1(C)CCCO1.N1(C(c2c(CN(C)C)ccs2)=O)CC2CC2(C)C1.N c1(C(=O)NCC2C(C)CCN2C(=O)C=Cc2nccs2)cnc2nccnc2c1 c1(NC(C(c2cccnc2S)N(CCOC(C)=O)C)=O)cccc([N+](=O)[O-])c1 C1(CNC(c2cnc(OCC)s2)=O)CCCCN(C(=O)C(F)(F)CO)C1 Cc1c(C(=O)NCC(F)C)[nH]c2c(C)cccc12.C1(CC=O)CC2(CC2)CO1.N C1(NC(CS(N2CCN(C)CC2)(=O)=O)=O)CC2CN(C(C3(C)CC3)=O)CC2C1 N1(C(CCC(C)(C)F)=O)CCC2(CC1)CC2NC(=O)C(C)(C)C1CCCO1 Cc1ccc2c(CC(=O)NC3CN(CC(F)F)C3)cc(=O)oc2c1 Cc1cccc(NC(=O)CC2COCCN2C(=O)CCc2ccccc2Cl)n1 C(CCCCCN(C(=O)C=Cc1ccccc1)C)NC(CCOCCC)=O S(=O)(=O)(c1cccnc1N1CCC2CC2C1)NC(CC)Cc1ccc(C)cc1 Cc1cnc(O)c(CNC(=O)CCCCNC(=O)CCn2ccnc2)c1 c1(C=O)cccnc1C.CC(F)(F)F.C(=O)(C(=O)N(C)C)N(CCC)CC.N N1(C(CC2C(C)CCC2)=O)CC(NC(=O)CC2CCOC2)CC2(CCC2)C1 C(CC(C)(C)C(=O)NCC(C)=CC(=O)NCc1ccnn1C)OC C#CCCC(O)CCNC(=O)CC1CSCCO1 C1(C(=O)NCCCC(=C)Cl)CC12CCN(C(=O)CN1C(=O)CNC1=O)CC2 c1(OCCC)cccc(-c2nc(C3CCCC3)nn2Cc2ccc(F)cc2)c1 CC(C)CC(C(=O)N1CCC(N(C(=O)Cn2cccc2)C)C1)C(N)=O N1(C(=O)CN2CC3CC3C2)C2CCC1CN(C(=O)C=Cc1ccccc1F)CC2 C1(CC(=O)NC(C2CN(C(C3CC4(CC4)CO3)=O)C2)C)COCCN1C C(=O)(C1CC(O)c2ccccc21)N(C1CN(C(C2N(C(C)=O)CCOC2)=O)C1)C C=C=C(C)CC(=O)NCC(O)C(N1CCC(CC)C1C)=O C1(CC)CN(C(=O)CCCOC)CCN1C(=O)C=Cc1ccccc1.C1(S)CC1 C1(C(=O)NCCCCN(C(CCCN(C)C)=O)C)CC12CCCCCC2 C1(CNC(C2(CCC)CCC2)=O)CCC(C(=O)NC(c2ccccn2)C)C1 N1(C(Cc2cn(CC)nc2)=O)CCCC(F)(CNC(C2CCC(C)C2)=O)C1.O c1(C(N2CCCC23CC3)=O)ccc2c(c1)CCN2.C(C(=O)N)N(C1CC1)CC C1(CCC)CN(C(=O)CCOCC(C)C)CCN1C(=O)CC1CC1(Cl)Cl Cc1[nH]nc(C(N2CCC(OCc3ccnn3C)C2)=O)c1O.C12CCN(CC1)C2 C(CCC=C(C)C)(C(=O)NC(C)C)N(Cc1cccc(CC)c1)CC NC(=O)CCCC(=O)NC12CC1CN(C(C1(c3ncco3)CCC1)=O)C2 Cc1c[nH]c2cc(C(=O)NCC3(C)CCCCO3)ccc12 C12(NC(C3CCC(=O)N3)=O)CCCC1(F)CN(C(c1[nH]nc3ncccc13)=O)C2 N1(C(C2CC=CC(NC(C3(C)CCC4CC4C3)=O)C2)=O)CCc2ncsc2C1 N1(C(c2c(C)c(O)ccc2)=O)CCN(C(=O)CN(CC(C)(C)C)C)CC(C)(F)C1 c1(COC)cccc(C(N2C(C)CC3CC23)=O)c1.C(=O)(CCc1cncs1)N c1(C(=O)NCCCN2CCN(C(CCNC(C)=O)=O)CC2)cc2c([nH]1)CCC2 c1(C(=O)NC2C(NC(c3ccc4c(c3)CCN4)=O)C2)nc2ccccn2c1F CC(C(=O)NCC(C)NC(c1c[nH]cc1C1CC1)=O)C(F)F CCCC(C(O)C(=O)N1CC=CC1)NC(c1nccn1C(C)C)=O C1(COC)N(C(=O)C(C)(C2CCC2)NC(=O)CCCCSC)CC1(C)C c1(C(N2CCC(N(C(C(C)O)=O)C)C2)=O)cc2c(c(S(N)(=O)=O)c1)CCC2.CS n1(CCC)ncc(C(=O)NC2(C)CCN(C(c3cnn(CCOC)n3)=O)C2)c1C c1(C(CSCCC)(C)N)nnnn1CCOCCOCC=CCl c1(C(C(N2CCCC(n3cc(C4C5COCC45)nn3)C2)=O)O)ccc(F)cc1 c1(CCN2C(=O)CN(CCc3n(CC)c(S)nn3)C2=O)c[nH]c2cc(Cl)ccc12 c1(C(=O)NC(CC=C)CNC(C2(N(C)C)CCC2)=O)ccc(SC)cc1O CC(CC(=O)N1CC=CC1C(=O)NCc1cncn1C)C(F)F N1(C(c2c(CC)n(CC)nc2)=O)CC2(C1)CN(C(C1CC(OC)C1)=O)CCO2 CC1(C)CCCC(C(N2CCC(C3CCCN3c3ccc(C#N)cn3)C2)=O)C1 COC1CN(C(=O)C(=O)NCC2CC(C)(C)CCO2)CCc2ccccc21 C(C)(C(=O)NCC(C1CCC1)O)NCC.C1(C=O)CC(=C2CC2)C1 Cc1ccc(S(=O)(=O)N2CCCC(CN(C)C(C)C)C2)c2ccccc12 O=C1COc2ccc(C(=O)NCC3C4CCCC34)cc2N1 N1(C(CN(C(=O)C(C2CC2)C2CC2)CCOC)=O)CCC1.C(N)=O.N c1(NC(c2c(-c3cncc(C)c3)c[nH]n2)=O)cccc2c1CCN2C C1(CC(=O)NCC23CC2CN(C(C2CCCCO2)=O)C3)(OC)CCCCC1 c1(C(=O)NCC(=O)OCC2(C)CC2Br)c(F)cccc1Cl c1(C(=O)NCCN(C(=O)CC2CC2(C)C)C)ccc(-c2cccs2)s1 c1(C(N2CCCN(C(CSCC)=O)CC2CO)=O)cc2c(n1C)CCOC2 Cc1ccc(C#N)cc1S(=O)(=O)N1CC(F)CC1C(=O)NCc1cc[nH]n1 C1(CNC(C(CC)(C)OC)=O)(NC(C2CC23CCOCC3)=O)CCCCC1C N1(C(c2cc(CC)cc(F)c2)C(=O)NC(C)C(=O)OC)CCCCc2sccc21 C1(NC(c2c(COC)cco2)=O)CN(C(=O)CC2CC2)C2(CCC2)C1.O Cc1nc(C(C)NC(=O)C(C2CCOC2)NC(=O)C(C)c2cc[nH]n2)cs1 c1(C(=O)OCC2CC3CC2CC3NC(=O)Cc2ccccc2)cc(I)ccc1Br CC(C)C(N=[N+]=[N-])C(=O)NC(CC(F)F)C(=O)NC1(C)CCCC1C Cc1ccc(S(=O)(=O)Cc2nc(C3CC34CC4)nn2Cc2ccccc2Cl)cc1 Cc1csc(C)c1C(N1CCCC1CNC(=O)C(c1ccn(C)n1)C)=O N1(C2CN(C=O)C2)CCN(CCCC2CCC(=O)N2)CC1.CC(C)(C)NC=O C1(NC(=O)C=Cc2ccc(Cl)s2)CCCN(C(c2cc3ccsc3s2)=O)CC1 C1CCC2(COC2)O1.C1(CN(C)C=O)CN(C(=O)OC(C)(C)C)CCO1.N C(c1ccc(F)c(C)c1)=CC(=O)N(C1CN(C(C(C)OC)=O)C1)C C(=O)(C(C)S(C)(=O)=O)N(C1CCN(C(C2(C)CC=CCC2)=O)CC1)CC Cn1cnnc1CCC(=O)NC1CC(C(=O)NCC(O)(C2CC2)C2CC2)C1 c1(N2CC(NC(c3ccc(O)c(F)c3F)=O)C(F)C2)ncnc2cccnc12 C=CCC(C)C(=O)NC(C)(CNC(=O)C(C1CCCCC1)O)Cn1cccn1 N1(C(CC)=O)CCC2(CCCCN(C(c3cc4n(n3)CC(C)(C)CO4)=O)C2)C1 C1CS(=O)(=O)CC(=O)O1.C1(c2c(C(=O)OCC)cn(C)n2)Cc2ccccc2O1 Cc1cnc(C(=O)NC2CC23CCC3)cc1Cl.c1(C(=O)N)c(Cl)n[nH]c1C1CC1 CC1(C(=O)Nc2ccc(CS(C)(=O)=O)nc2)CCCN1C(c1ccc[n+]([O-])c1)=O Cc1coc2c(CNC(=O)CC(C)CC(C)C)cccc12 C1(CCNC(C2CC(SC)C2)=O)(NC(=O)Cc2cncn2C)CCCC1 CN1CCC(c2cn(CC3CCCN(C(c4c(Cl)cnn4C)=O)C3)nn2)CC1 C1(CC)CCCC(NC(=O)C(C)(C)NC2CCN(C3CCCC3O)CC2)C1 c1(C(=O)NC2(CC(=O)NC(C(CC)C)CO)CCC2)cnc2ccc(Cl)cn12 C1(C(=O)NCCn2ccnn2)CC2(CCC2)CN1C(C1CN2CCN1CC2)=O CC(CCCCNC(C1(C)COC(=O)C1)=O)NC(=O)CCCCn1ccnn1 c1(OC)cc(C)cc(-c2nc(CCn3ccnc3)nn2C23CC(C2)C3)c1C CC1CCN(C(c2cnc(CNC(=O)CCC3CC3)nc2)=O)C1C c1(C(=O)NCC=CCNC(c2cc(Cl)ns2)=O)ccc([N+](=O)[O-])cn1 C1(C)(C(=O)Nc2cccc(C)c2F)CN(C(C2CCCSC2)=O)C(C)(C)C1 S(=O)(=O)(c1ccc(F)c(Br)c1)N1CC(F)CC(C(=O)NCC2CCSCC2)C1 c1(OC)cc(C(=O)N)ccc1C.C1CC2CCC1N2C(C1CC(N(C)C)C1)=O.C c1(C(N2C(C)CN(C(c3sccc3OC(F)F)=O)CC2)=O)cnc(O)n(C)c1=O C1(N(C(Cc2c(C(C)C)con2)=O)C)C2CN(C(=O)C=C(Cl)Cl)CC12 c1(CC(=O)NC2(C)CN(C(CC(C(C)C)C)=O)C2)cc(Br)ccc1C#N C#CCC(C)(CC)C(=O)NCc1nc(C)cc(O)n1.c1(CC=O)occc1C.N c1(CNC(=O)C2CC2)ccc(S(=O)(=O)NC(CCCO)c2cccnc2)cc1 C1(C(=O)NC2(CO)CN(C(c3cc(C(C)(C)C)no3)=O)C2)CC(=O)N(O)C1 c1(OC)cccc(SCCC(=O)NC2CCC2NC(c2ccc(Cl)s2)=O)c1 CCN(C(C)CO)N1CCC(C(C)=O)CC1 Cc1cnc(C)c(NC(C2CCN(C(=O)CN3CCCC3)CC2C)=O)c1 c1(OC)ccc(C(=O)NC2(C)CCCCC2C(=O)NC2CNC(=O)C2)cc1O C1(C)(C=O)CCC(=O)CC1.c1(OCC)cc(C(=O)NC2CCCC2)ccn1.C N1(C(CCCC(CC)C)=O)CCC(C2(NC(C3CCCOC3C)=O)CCC2)CC1 c1(C(=O)NC2C(NC(=O)CC3CCSC3)CS(=O)(=O)C2)ccn2cccc2c1 CC1(C)CCC(C(=O)NC2CN3CCC2C3)(NC(=O)CN=[N+]=[N-])C1 C#Cc1ccc(F)cc1C(=O)NCC(C)CC.C(=O)(C(O)Cc1cnn(C)c1)N C1(C(N2C(CCC=C)CCC2)=O)CC(NC(C2CC(C)N(C)C2)=O)C(O)C1 C(CC(C)C=O)=CC.c1(CC)ccccc1.C1(CS(C)(=O)=O)(C=O)COC1.N C(=O)(C1=NN(C)C(=O)CC1)N1C(C2CC2)CCC1.CC(C)CC=O.C(N)(=O)N c1(NCC(C)N(C(CCn2c(C)csc2=O)=O)C)c(Cl)cccc1[N+](=O)[O-] C1(C(N(CC(N2CC(CCC)CC2)=O)C2CCC2)=O)CC2(C1)CC2(F)F.C CN1CCN(C(C2CC3(CSC3)C2)=O)CC1CNC(c1cnn(C)c(=O)c1)=O Cn1cnc(C(=O)NC2CCN(CC(N3CCCCC3)=O)C2)c1 CC(CN(C)N1CCOCC1Cc1cccc(Cl)c1)C(F)(F)F Cc1ccc2scc(CC(=O)NCC3(O)CCCN(C(C4CCO4)=O)C3)c2c1 N1(C(CC(C=C)(C)O)=O)CC2CCC(CNC(C3(F)CC=CC3)=O)(C2)C1 CC(CCNC(C1CC(O)CN1C(=O)Cc1csnn1)=O)C(F)F c1(C(c2cnc(C3CC3)o2)NC(COCC)(C)C)nnnn1C N1(C(c2ccc(CCC)[nH]2)=O)CC(C)(C)CC1CNC(C1(O)CCSC1)=O N1(C(C2CCCN(CC)C2)=O)CCC(Cc2cc(CN)on2)(CC)CC1 c1(CC)ccc(NC(=O)C(=O)Nc2nc(C(C)C)cs2)c(Cl)c1 c1(N(C)Cc2nnc(O)o2)nc(=N)[nH]c(=NCCc2nc(=N)[nH][nH]2)[nH]1 C1(C(=O)NC2CCCN(C(=O)C(c3cnn(C)c3)C)C2)(CC)CNC(=O)C1 CCCC(CNC(c1csc(C)n1)=O)NC(C1(C2CCCO2)CCC1)=O c1(C(=O)NC2CCC(CNC(c3c(C)ncnc3)=O)CC2)csc2ccncc12 C#Cc1cnc(NC(N2CCC(CC3CC3)C2)=O)c(C)c1 C1(C(N(C(CC)CNC(C2CC(=O)N(C)C2)=O)C)=O)CCC(C)(C)OC1 C(C(CNC(C1(C2CCCCO2)CC1)=O)CO)NC(c1cncs1)=O c1(C(N2CCCC(N(C(=O)C=CC3CCOCC3)C)C2)=O)cn(C)c(=O)nc1O C12(NC(c3cc(C(N)=O)no3)=O)CCCC1CN(C(=O)C=CC(F)(F)F)C2 C1(NC(COCCC)=O)CN(C(c2c(Cl)cncc2Br)=O)CC(C)(C)C1 C12(CCNC(C(CC=C)C)=O)CCC(CC1)N(C(=O)CC1CC(C)(C)CO1)C2 C1(C)(CC)CCC(C(=O)N)O1.C1CC(F)C1.C1(C=O)CC(=C2CCC2)C1 N1(c2cc(N(CC(=O)NC(C)C)C)ncn2)CCC(C2CCCOC2)CC1 N1(C(c2ccn(C)n2)C(=O)NCC)CCN(C(C)COC)CC1 c1(OCCNC(C(=O)OC)CCCl)ccc2c(c1)CN(C)C2=O c1(C(=O)NCC(CC=C)NC(C2(F)CCC(C)CC2)=O)c(F)cc(Cl)cc1Cl C(=O)(C1=C(C)OCCS1)NCC1(C)N(C(=O)Cc2cnoc2)CC(OC)C1 C(C(O)CN=c1[nH]cnc2[nH]ccc12)NC(C1CNC(=O)N1)=O c1(C(=O)NC(C(CO)NC(C(c2ccc(Cl)s2)C)=O)C)cc2c(s1)COCC2 Nc1c(C(N2CC3(C2)CN(C(c2ccc(Cl)cn2)=O)C3)=O)ccc(F)c1F N1(C(c2nn(C)c(CO)c2)=O)CCC2(C1)CN(C(=O)C=Cc1ccco1)CCO2 C1(NC(c2cccc(OC)c2)=O)COC2(CCN(C(=O)Cc3cnsc3)CC2)C1 c1(C(N2CC3CN(C(CCCOCC=C)=O)C3CC2)=O)coc2ccc(Cl)cc12 c1(C(=O)NC(C)C(C)NC(c2cc(P(C)(C)=O)cs2)=O)csc2c1CCCC2 c1(C(=O)NC(CCC=C)C(=O)NCC2(C)CCC(=O)N2C)coc2ccccc12 C(C(=O)N=S(C)(=O)CCO)(C1CCC(F)(F)CC1)OC N1(C(c2n(C)cnn2)=O)CC2CCN(C(C3CCCC3(F)F)=O)CCC2C1 C=CC(C)C(=O)N1CC(CC(N2CCCC2C(N)=O)=O)(OC)C1 c1(C(=O)N)cc(C)nc2ncnn12.N1(C(C(C)SC)=O)CCN(CC2CC2)CC1 N(C(=NCCF)N1CCC(OCC(F)(F)F)CC1)CC(c1cn(CC)nc1)O c1(C(=O)NC2(CNC(C3(C)CC3)=O)CCOC2)c(Cl)nc2ccccn12 Cc1cn2c(n1)CC(C(=O)NCC1CCCN1C(=O)C(c1c(C)n[nH]c1C)C)C2 c1(SCC)nc(C)c(CC(=O)NC2CCC(C)C2)s1.C(=O)C(C)(C)CC.C C(=O)(CCC(F)(F)F)NCC12C(CN(C(C(Cc3ncn(C)c3)O)=O)C1)C2 C(=O)(C(C)C(F)(F)F)NC(CCN(C(c1c(CCC)onc1C)=O)C)C C1(CNC(c2cnn3c2CCCC3)=O)CN2CCCCC2CN1C(=O)CC1CC1 C(C)(CCCCNC(c1ccc(C2(F)COC2)cc1)=O)NC(C1C(=C)C1)=O C1(C(N2CCC(C)(NC(=O)Cn3cnnc3O)CC2)=O)CCn2cnnc2C1 C1(C(=O)NCC(CC(=O)NCCC(C)(C)N(C)C)OC)(CC)CCCC1O C#Cc1cccc(C(=O)NC2CC(CC(=O)NC(C)CC(=O)NC)C2(C)C)c1 c1(CC(=O)NC(C2CN(C(c3cc(CC)c(C)s3)=O)C2)C)cc(F)ccc1C C(=O)(CCCC(=O)N(C1CCCCC1N(C(=O)CC(C)(C)OC)C)C)OC C(CCCCCNC(c1cc(Cl)n[nH]1)=O)NC(C1CC(=O)NC1)=O N1(S(CC2(C)CCCOC2)(=O)=O)CCOC2(CC2)C1 N1(C(COc2cc(C)on2)=O)CCOCC(NC(=O)C2CC2)C1 c1(OC)cc(Br)cc(CN2CC(NC(=O)Cc3ncccn3)C2)c1O c1(COC(C2CC2(c2ccccc2Br)F)=O)ncc(Br)cc1Cl c1(OCCOC)cccc(NC(=O)C(N2CCC(C(O)C(F)(F)F)C2)=O)c1 c1(NC(C2CC(NCc3c(OC)ccc(C)c3)C2)=O)cnc2c(F)cccc2c1 C(=O)(CCCCC(F)F)N1CC(O)CC(NC(CSCCC)=O)C1 N1(C(CCc2ccc(=N)[nH]c2)=O)CC2CC(NC(c3cc(C(F)F)cs3)=O)C1C2 c1(C(N2C(CNC(C(CC)(C)C)=O)CCC2)=O)ccc2occc2c1 C#CCC(CC(=O)N1CCC(n2ccnc2)C1)NC(C1CN(C)C1)=O CCCCC(CC)C(=O)NCC1(C(C)(C)O)CN(C(=O)CC2(CO)CC2)C1 c1(C(N2CC(NC(c3c(CC)cco3)=O)(C)C2)=O)cccc2c1C(=O)NC2=O N#Cc1cc(F)c(C(=O)NCC2CCN(C(c3cnn4c3OCC4)=O)C2)c(F)c1 C(=O)(C1=CS(=O)CCC1)N1CC(CC=C)C1.c1(C(=O)N)cncc(C(N)=O)c1 N1(C(c2cc(C)no2)=O)CCN(C2CCC(NC(=O)CC3CC(C)(C)C3)C2)CC1 CC(N=c1[nH]c2c(c(=NC(CN(C)C)CC(C)(C)C)[nH]1)CSC2)c1cnsc1 CON1CCC(CC(=O)NC2CCC(CNC(c3cc(Cl)ncc3O)=O)C2)CC1 N1(C(C=Cc2ccc(C)cn2)=O)CCC2CN(C(C3(Br)CC3(C)C)=O)CC12 c1(C=O)c(F)c(F)cc(F)c1F.C(c1nc[nH]n1)=CC(=O)NCC.C1CC1 c1(-c2ccc(C)cc2O)cc2c(s1)CCN(Cc1cnccc1C#N)C2 N1(C(C(CCC)C)=O)CC(CC(=O)NC2CC(CO)C3CC23)C2(CC2)C1 CCC(C)CCC(=O)N1CC(F)(CNC(C2CC(OC)C2)=O)C1 n1(CC(N2CCCCC2)=O)cc([N+](=O)[O-])nc1C.C(=O)C=CC(N)=O.C=CC C1(CC)CC(O)CN1C(C1(CC)CN(C(=O)C(=O)NCC(F)F)C1)=O CC(CC1CCCCN1C)N=c1[nH]c(=N)[nH]c(=NCCCCN2CCCCC2)[nH]1 c1cc(C(=O)Oc2c(Br)cc(Cl)cc2C#N)cc2c1OC(C)C2.CCN N1(Cc2cc(OC(CC)C)c(OC)cc2)CCCCC2(CCNC2)C1 Cc1[nH]c(C(=O)NC2(CF)CCC2)c(C)c1C(=O)NC(C1CCOC1)C C(=O)(C1CCc2c[nH]nc21)NCC(C12CCC(CC1)C2)NC(=O)CCC1CC1 Cc1sccc1CC(=O)NC(C1CCOC1)CNC(=O)CCOc1ccccc1 C1(F)CCN(C(c2cc(C(F)F)cs2)=O)CC1.CC1(C(=O)NC)CCC(=O)N1 c1(C(=O)OC)ccc(C(O)CNC(c2cn(C)nc2OC(C)C)=O)cc1 C1CCCCCC1F.C1(C(C)CCC=C)CCN(C(=O)C(C)CC=Cc2ccccc2)CC1 C(N=c1[nH]c(=NCC2CCOC2C)c2ccccc2[nH]1)c1cc(C)c(Br)c(C)c1 C1(S(C)(=O)=O)(C(=O)N)CCC1.C(C)(C)(CO)NC(CSC(C)(C)C)=O c1ccc([N+](=O)[O-])cc1[N+](=O)[O-].c1(CCCC(=O)OCC)cc(F)ccc1F CC1Cc2cc(CC(N3CCC4C(NC(=O)CCc5cscn5)C34)=O)ccc2O1 C(C(=O)NN1CCCC1C(N1CC(O)CC(O)C1)=O)n1cnc(=N)[nH]1 N1(C(Cc2cn(CC)nc2C)=O)CCC2CN(C(C3CCN(C)C3)=O)CC12 c1(-c2nc(C(CC)CC)nn2C(C)C(C)(C)C)cccc(=O)n1C N1(C(c2scc(COC)c2)=O)C2CCC1CC(N(C)C(c1cccc(=O)o1)=O)C2 c1(OC)ccc(CN(C(c2ccc(Br)s2)C(=O)NC2CCCC2)C)cc1 N1(C(C(CCC)OC)=O)CCC2CC1CN(C(c1ccc(C(C)C)s1)=O)C2 c1(C(=O)NC(c2ccccc2)C(C)NC(=O)CCc2c[nH]nn2)csc(C#N)c1 C12(C(=O)NC3CCN(C(c4n(CC)ncn4)=O)C3)CC(C)(C1)OC21CCC1 N(C(=NCC1CCCO1)NC1CCC(C(=O)OC)C1)CCc1ncc(CC)s1 CC(C)C(CC(=O)NCC1CCN1C(=O)CN1CCCOC1=O)C(C)C c1(C(=O)NCCN(C(C2CCNC(=O)C2)=O)CC)c(F)ccc(F)c1N Cc1ccc(CCC(N2CCCC(CN(C)C(C3(Br)CC3)=O)C2)=O)cc1 C1(NC(C2CCCCNC2=O)=O)COCCN(C(c2cncc(C3CC3)c2)=O)C1 C1(NC(C)=O)CCC(C(=O)NC2CCCC2C)CC1.c1(CC=O)scnc1C c1(C(=O)N)csc(N=S(C)(=O)N(C)C)n1.CC1CCCN(C(C2CC(O)C2)=O)C1 Cc1cncc(C(=O)NC(C2CCCCC2)CNC(c2ncccc2O)=O)c1 Cc1nc(C(C)C)ccc1CSCc1nc(C)c(C)o1 c1(C(=O)NCC(CNC(COCC=C)=O)C)sc(Br)cc1C S(=O)(=O)(c1cccc([N+](=O)[O-])c1)NCCC(NNC(=O)NC(CCCC)CCC)=O C(=O)(CCCC(C)CC)NC(CC=C)CNC(C1(c2ccc(Cl)cc2)CCC1)=O c1(CNC(CC=CC=C)=O)ccc(C)nc1.C1CCCC2(CC2)C(=O)N1 Cc1cc(O)ccc1C(=O)NCCNC(=O)Cc1ccon1 c1(C(C(=O)NC(C(C)NC(C=C(C)Cl)=O)C)(F)F)ccc(Cl)cn1 C=CCCC(F)(F)C(=O)N1CCC(CNC(=O)CC2CCC(C)O2)C(O)C1 Cc1ccsc1C=CC(=O)NC1(CO)CCCCC1.C12CCCN1C(=O)C21CC1 c1(C(N2CCC(N(c3cc(OC)nc(C)n3)C)C2)=O)cccc2ccc(Br)cc12 CC1(C)CC=CCN(c2ccnc(N3CCN(c4nccs4)CC3)n2)C1 N1(C(CCCCCCCC)=O)CCCC2(CCN(C(=O)CC3CSC3)CC2)C1 C(=O)C(C)(C)n1cc(Cl)cn1.N1(C(CCCN(C)CCN(C)C)=O)CCCC1 C1(C(=O)NC2CC(NC(c3ccnnc3)=O)C2)CCOC2(CCCCC2)C1 N1(C(=O)NCC2C(c3ccc(F)c(F)c3)(C)C2)CC2(CCC2)C1c1ccsc1 C1(C(=O)NCC=CC(N2CC(O)(CCC)C2)=O)CCC(C2CC2)C1 C(C(C)N=c1[nH]c(=NCC2(C)CCCO2)[nH]c2c1SCC2)N(CC)CC CCC(C)CCC(=O)NC1CC1NCCC1CC=CCC1.C(C)(C)C.C=O.N C(C(C)(CO)CO)NC(C(C)NC(C(n1ccc(C)n1)C)=O)=O C1(CNC(C2(OC)CCSCC2)=O)CCCCCN1C(=O)Cc1ccc(Cl)cc1 CC1CCC(CO)(NC(c2ccncc2Cl)=O)c2ccccc21 c1(C(N2CC(O)CCC2)=O)ccc2cnn(C)c2c1.C1(C(=O)OC)CC1C=O.N C1(C(N(CCCCCC)CCNC(C2C(=C)C2)=O)=O)CCCS(=O)(=O)C1 C1(Br)(C(=O)NCC#CCNC(CN(CCC)C)=O)CC1(F)F N(C1CCc2c(Cl)cccc21)C(C(=O)NC1C(C)(C)NC1)=O O=C(C1=CCS(=O)(=O)C1)N1CCCC(N2CCN(c3ncc(O)cn3)CC2=O)C1 N#Cc1cc([N+](=O)[O-])c[nH]c1=NCCC1CCN(C(c2cccc(Cl)n2)=O)C1 c1(-c2c(C)c(C#N)ccc2)n[nH]c2cc(C(=O)Nc3scnc3C(N)=O)ccc12 C1(NC(Cc2n(C)nc(C3CC3)n2)=O)CC2(CCN(c3cc(F)ncn3)C2)C1 C1(CC=C)(NC(c2cn(C)nc2Br)=O)CCN(C(c2nn(C)cc2C)=O)C1 C1(CCC)CCCN(C(=O)C(COC(C)C)NC(c2cc(OC)ns2)=O)CC1 N1(C(c2c(CC)noc2C)=O)CCCC(F)C1.c1(C=O)cc(C(N)=O)cn1C.N c1(NC(C2C(CNC(CCC(=C)Cl)=O)OCC2)=O)cc(Cl)ccc1C Cc1ccc(=NCCC(=O)N2CCCC2(C)CNC(c2cc(Cl)c(Cl)[nH]2)=O)[nH]c1 N1(C(C(=O)NCC(C)C)CC2CC2(Cl)Cl)CCOCC12CCC2 C#Cc1ccc(C(=O)NC2CC(NC(=O)Cc3scnc3C)C2)cc1C c1(CCC)cc(C(=O)NC(CNC(C2(n3ccnn3)CC2)=O)CC)n[nH]1 c1(-c2ccc(OCC(C)C)cc2)cnc2[nH]c(C(=O)NCc3ccoc3)cc2c1 c1(COC)cc(C(c2nnnn2Cc2cccs2)NC2CSC2)no1 C(CNC(=O)C(SC)SC)(C(C)C)NC(C1(CSC)CCC1)=O O=C(NOCC(F)(F)F)C(CNC(C1(O)CCC1)=O)CC1CCCC1 C1(C(=O)NC)(OCC)CCOCC1.N1(CC(N2CC(O)C2)=O)CCNCC1 Cc1cccn2cc(C(N3CCCCC3CNC(c3cccnc3S)=O)=O)nc12 Cc1cnsc1C(=O)NCCN(C(=O)Cc1cnc(C(C)C)[nH]1)C1CC1 C1(C(=O)NCC(COC)O)CCN(C(C2(NC)CC2)=O)CC1(C)C.C(C)C C1(C(=O)NC2(CC)CCOC2)(C)CCCCC1.C(=O)C(CN(C)C)N(C)C C=CCCCCC(=O)NCCN(CC(C)O)C(c1cc(NC)nc(Cl)c1)=O c1(N(C)C)ccccc1CN1CCC(C(=O)N(CCCO)C)CC1 S(=O)(=O)(c1cc(C)cnc1NC1CCCn2ncnc21)NC(CCC)C1CCC1 N1(C(C(C(C)(F)F)(C)C)=O)CC2CCCC(O)C2C1 c1(OC)cccc2c1OCCN(C(c1cncc(=O)[nH]1)=O)C2 C1(C(N2C3CCC(NC(CC(C(C)C)C)=O)(CC3)C2)=O)CCc2nccn2CC1 c1(C(=O)NCC(c2ccccc2)N(C(C(CC#C)C)=O)C)nn(C)cc1C#C C1(NC(C2CCCN(CC)C2)=O)CCCCN(C(=O)CC2(O)CCC2)CC1 c1(CNCC23C(CN(C(C(N)=O)=O)C2)C3)c(Cl)ccnc1Br C(CC(F)F)(C(=O)NC1CCCN(O)C1=O)N(C(=O)C=CCF)C c1(C(N2CCCN(C(C34C(C(N)=O)(CCC3)C4)=O)CC2)=O)cccc2nn[nH]c12 N1(c2cccc(OC)c2)CCN(C(c2cc(OC)cc(Br)c2O)=O)CC1C#N CC1(C(=O)NCCc2ccco2)CCN(C(=O)CC2CC=CC2)C1 C1(COC)CN(C(=O)Cc2cncnc2)CCN1C(=O)C(C)C.C1CCCC1.S CCCC(C#N)C(=O)NC(C)(C)C(C)NC(=O)Cc1cccc(Cl)c1 C1(NC(c2c(C)ccnc2C)c2n(C(CC)C)nnn2)CC2CCCCCCC12 C=Cc1ccc(C(N2CC=CC(C(=O)NC3(C(O)COC)CC3)C2)=O)cc1 c1(C(N(C(CCNC(C(C(C)C)C)=O)C)C)=O)cc(S(C)(=O)=O)ccc1O CCC(C)(CNC(c1cc(C)cc(C)n1)=O)C(=O)NC(C)CCC(C)C C#Cc1ccc(C(=O)NC2CCN(C(=O)C(N)=O)CC2c2ccccc2)cc1Cl C1(CCNC(=O)C=Cc2cncs2)CN(C(C2CCCS(=O)(=O)C2)=O)CCCO1 C1(NC(CS(CC)=O)=O)CCCCCN(C(=O)COc2ccc(F)c(Cl)c2)C1 C1(OC)CN(C)C(C)(C(N2CCC(C)C2)=O)C1.c1(C=O)ccc(C)c(N)c1.C O=S(=O)(NC(C1CCC(F)(F)CC1)C(F)(F)F)N1CCC(F)(F)CC1 N1(C(CC)=O)CCC(C2CCCN(C(c3c[nH]c4nccc(Cl)c34)=O)C2)C1 N1(C(c2c(CC)cc(Cl)cc2)=O)CC2CC1CN(C(=O)C(O)C1CC1)C2 N1(C(C2CSCC(=O)N2)=O)CCN(C(=O)CCc2ccc[nH]2)C(CCO)C1 c1(OCC(=C)C)ccc(C(=O)NCCO)cc1.C(=O)C.CC.C(C)=O N#Cc1ccsc1S(=O)(=O)NC1CC2CC3C(C2)C13 C1(NC(C(C)SCC)=O)CCN(C(c2cnc3c[nH]nc3c2)=O)CC1(C)C c1(OC)ccc2c(c1)CCC2C(=O)NCCC(C)NC(=O)CN1CCCC1 C=C(Cl)CC(C(=O)NCC)NC(=O)CC(=O)NCCc1ccnc(C)n1 C1(CC(=O)N)CCC(=O)NC1.C1(OC)CCC1CC(=O)NC1CC1C=O CC(C)(O)C(F)C(=O)NCC.c1(C(=O)N)ccc(C(F)(F)F)cc1C(F)F C1(CNC(CCN(C(CC)CC)C)=O)CCN(C(=O)Cc2csc(C)n2)CC1O N1(C(CCc2scc(C)c2)=O)CC2(CC(C(=O)NCC3CCCCC3)CO2)C1 C1(CC(N2CC3C(NC(c4c(C)nc(O)[nH]4)=O)(C3)C2)=O)CC2(CCCC2)CO1 C(CCCC(F)(F)F)NC(C1C2(CC(NC(=O)CC3CC=CCC3)C2)C1)=O N1(C(c2nc(C)oc2)=O)CCc2nc(CNC(=O)C(C)(C)c3cnco3)sc2C1 n1(CCC(=O)NC2C(NC(C(C)O)=O)CCC2)c(=O)oc2cc(Cl)ccc12 C(CC(C)(C)CC(=O)NCC=CCC(=O)NC(c1csnn1)C)OC C(=O)C(F)(F)C(C)O.c1(OC)ccccc1CCC(N1CCC(CCOC)CC1)=O C1(C(=O)NCc2cn(C(C)C)nn2)CCCCN(C(=O)C=C2CCC2)C1 c1(C(N2CC(O)(NC=O)C2)=O)cc(SC2(CCC)CCOC2)nn1C.OC c1(OC)ccc(C(=O)NC2CC(NC(=O)C(C)C(F)(F)F)C(O)C2)c(C)n1 c1(OC)cc(N)c(F)cc1C(N1CC(OC)CC(NC(=O)CC(C)F)C1)=O c1(C(N2CCC(CC(N)=O)(NC(c3cccs3)=O)CC2)=O)cnc2[nH]nnc2c1 n1(CCCOC)c(N2CCCC(COC)C2)nnc1Cc1cc(C)on1 c1(CC(=O)NC2CC(O)C2)cccc(CN2CC3C(Cn4cccn4)C3C2)c1 C1(C(=O)NCC(CCOC)NC(C2(C)CCCCC2)=O)CCc2ccnn2C1 O=C(C1CCCc2nccn21)NC1CN(C(=O)CCc2ccsc2Cl)CC1O C1(C(=O)NCc2c(COC)noc2)CN(C(=O)C(C)CO)CCN1C C1(c2ccccc2)(CNC(=O)NC(c2nnc(C)o2)C)CCOCC1 n1(CCCC)nnnc1C(c1cc(C)co1)NCC(CC)OC N1(S(CC(C)C)(=O)=O)CC2(CC2)CC1C(=O)Nc1ccc(OC(F)F)cc1 c1(CNC(CC(CN(C)C)O)=O)cnn2c1CN(Cc1sccc1Cl)CC2 Cc1ncc(C(=O)NC2(CC)CC2)c(C)n1.c1(CC=O)cc(F)cc(Cl)c1.N C(C)(C)(C(=O)NCCOCCNC(=O)Cc1cnccn1)OC C1CCN(C(c2scnc2C(F)(F)F)=O)CC1.C12(C(NCC)=O)CCCC1C2 c1(N(C)C)ccc(C(N2CCCC(Sc3ccc(CN)cc3)C2)=O)cn1.C=O N1(C(CC(=C)I)=O)CCC(NC(C2CC(C)(CC)C2)=O)C(O)C1 C1(NC(CCCc2ncc(C)o2)=O)CN(C(=O)C(C)(C)CF)CCC1C Cc1cc(O)ccc1CC(=O)NCCOCCNC(c1cn(CCO)nn1)=O c1(C(N(C)CCOCCNC(C23CC(CO2)C3)=O)=O)nnc(O)nc1O c1(C(N2CC3C(CNC(CC=C=C)=O)C3C2)=O)cc(N)cnc1Br C1(OC)(CO)CCN(C(C2(CC)CC2)=O)C1.N1(CC(=O)N)CCC(=O)CC1 c1(NC(CC2CCN(C(c3n[nH]c(CC)c3F)=O)C2)=O)cnc2ccc(Br)cn12 c1(C(N2CCC(OC)C2)=O)sc(Cl)nc1C(F)(F)F N1(C(c2cccc(OC)c2)=O)CC2C=CC1C(C(=O)NC(C)CSC)C2 CC(CCCNC(C1(O)CC1)=O)NC(c1n[nH]c(C2CC2)n1)=O Cc1ccncc1C(N1CCCOCC1)C(=O)NCc1cccs1 C1(NC(c2cnn(C3CCC3)c2)=O)CCCC(C)C1.C1(F)(C(=O)N)CCOC1 C1(NC(c2c(CCC)cccc2)=O)CC2CN(C(c3cnoc3C3CC3)=O)CC12 C(=O)(C(F)(CNC(=O)Cc1nonc1C)C(C)C)NC(CC=C)C1CC1 CCC(C)C(C(=O)NCC1(O)CN(C(=O)CCOC2CC2)C1)OC C1(CCNC(C(C)(C)C2CCCCO2)=O)CCCCN1C(=O)CC1CCC(O)C1 N1(C(C=C(CC)C)=O)CCC2(CCCN(C(=O)C3=CC(C)CC3)C2)C1 c1(C(C(=O)NC2(C(=O)NCCOC(C)C)CCC2)O)cnn(C)c1 c1(-c2cc(C(NOC)=O)c(C)cc2)cc2c(s1)CCN(C(c1ccccc1)=O)C2 Cc1ccc(N)c(C)c1C(N1CCC12CN(C(=O)C(O)C(C)C)C2)=O c1(CC(=O)NCC(CC)NC(=O)C(F)(F)CC2CC2)ccc(F)cc1Cl C1(NC(C(CNC(C)=O)(C)C)=O)CCN(C(c2ocnc2C)=O)CC1O C1(C(=O)NC(CC=C)CNC(=O)Cn2cncn2)Cc2cc(Br)ccc2O1 Cc1ccc(C2CC2)c(C(N2CCOC(CNC(C3CCC(=O)N3C)=O)C2)=O)c1 N1(C(COC2(C)CN(C(C3(CC#C)CCOC3)=O)C2)=O)Cc2cccc(O)c2C1 c1(OCCC=C)ccccc1C1CCOC1 c1(SCC(=O)NC(CNC(C=COCC)=O)CCOC)cc(F)ccc1F c1(C(C)C)nnnn1CC1C2COCC12.c12cn(nn1)C1CN(C1)C(=O)C2 C(C(CC(C)C)C(=O)N(C)CC1CN(C(=O)Cc2c(C)cnn2C)CCO1)OC CC1(C)COCC(CC(=O)N(CCNC(C2CC=CCO2)=O)CC)O1.CCO.O c1(N2CCCC(C#N)C2)ccc(S(=O)(=O)NCCC2CCCS2(=O)=O)cn1 C1(OC)(CNC(=O)Cn2cc(NC(=O)N)nn2)CCOC1.C1CC1.C N1(C(=O)Cc2cc3ccccc3o2)CCCC2(C1)CN(C(c1occc1F)=O)C2 CN1CCC2(CCCN(C(=O)C3=C(Cl)CCCC3)CC2)CC1 CC1(C(=O)NCCCC2(NC(=O)Cn3cnc(Br)c3)CC2)CC=CCO1 c1(C(N2C(CCN(C(c3c(C)cno3)=O)C)CCCC2)=O)cc(F)c(F)cc1F CC1(C)CCC(C(=O)NCCC2CCC2)O1.c1(C=O)ccc(C(F)(F)F)nn1 C(C)(C(C)(C)C(=O)N1CC(C)(OCC(N2CCC2CF)=O)C1)OC C1(C(C)NC(c2cnn(CCF)c2)=O)CCN(C(=O)CC2CCCCC2C)CC1 n1(C(CC(=O)N(C(C)CNC(=O)C(C)(C)C)CC)C)nc(C)cc1C c1(C(N(CC(=O)NCCCO)CC#C)=O)c[nH][nH]c1=N Cc1c(-n2nc(CCn3cncn3)nc2CC2(C(F)(F)F)CC2)cccc1Cl C1(NC(c2c(Cl)cnc(C)n2)=O)CCSC12CN(C(=O)C=Cc1ccccc1)C2 N1(C(COCC(C)(C)C)=O)CC(C(=O)NC2CCC(O)CC2)C2(CC2)C1 C(C(CC(C)C)NC(=O)C(C)(C)n1ccnn1)n1cc(CCSC)nn1 CCC(C(=O)NC(C)CC(C)NC(c1nc(C(F)(F)F)cs1)=O)OC c1(C(=O)OC2CCN(C)C2)cnn2c(C(F)(F)F)cc(C3CC3)nc12 c1(C(=O)NCCCCCNC(COC(C)(C)C)=O)csc(C#N)c1 N1(C(C2C(=C)C2C(=O)OC)=O)CCOCC1C=O.C1(CC2CCC2)CCC1 C=CCC(C)(CNC(C1CCCCCC1)=O)CO.C1(C(=O)N)(CCC)CC(=O)C1 C1(CC)CC(CC(N2CCC2CNC(=O)CC2CCCCO2)=O)CCO1 c1(C2C(C=O)C2)cnn(C)c1C(C)C.c1(CCC)nnsc1C(N1CCC1)=O C(CC(C(C)C)NC(C1CCC(C)(C(=O)O)O1)=O)NC(C1(SC)CC1)=O S(=O)(=O)(c1ccc(NS(C)(=O)=O)cc1Br)NCc1cnn2ccn(C)c21 c1(C(NC)=O)cccc(Cl)c1C.C1(CNC(CC(=O)NCC)=O)CCCCC1 C1(C(N(CCOCC)C)=O)CCC(n2cc(CCN)nn2)C1.[SH](C)(=O)=O C(CC1=CCCCCC1)NC(C1CCN(C(=O)c2c(C)n[nH]c2)O1)=O c1(CC)cnc(F)cc1C(=O)NC1(CNC(c2cnn(C)c2Cl)=O)CC1 c1(C(=O)NCC(CNC(C2ON=C(C)C2)=O)O)cnc2ccccn2c1=O c1(C(C)C)nocc1C(=O)NC(CNC(=O)CCC1CCCN1C)C1CC1 N1(C(c2cn(CCC)nc2)=O)CC2CC(NC(=O)CCN(CC)CC)CC1C2 N1(C(CN2CC(CC)C2)=O)CCC(C)C1.c1(C=O)cn(C(F)F)nc1C(F)F Cc1nc(=N)[nH]c(C)c1C=O.c1(C(N(C2CCC2)C)=O)noc(C2CC2)c1C.N CC(C)C(C(=O)NC(C)C(C)(C)C)n1cnnc1.C1(C=O)CC1(C)C(C)C.N N1(C(COCC)=O)CC(C)N(C(c2cn(CC(F)F)cn2)=O)C(C)C1 N1(C(CCCCN(C(c2c(CC)c[nH]n2)=O)C)=O)CC(C)C(C)C1C C12=c3c(scn3)=NC(=NCC3(CC3)N1)N2.C1(CC2(C)CC2)CCOC1 Cc1[nH]c(=N)ccc1C=CC(=O)NCC1CC1.c1(C=O)cc(=O)cc[nH]1.C C1(C(=O)NC2CCCN(C3CC3)C2)(NC(=O)Cc2cncnc2)CC(F)(F)C1 C(C(CNC(=O)CCN1CCCC1)S(C)(=O)=O)NC(c1cc(C)nn1C)=O c1(C(=O)NCC=CC(=O)NCCCCSC)coc(C(F)F)c1 C(CCC(=O)NCC1CC1NC(c1cc(CO)on1)=O)NC(=O)OC C1(N(C(C2CCC(=O)C2)=O)CC)CCCN(C(C2CCCC2)=O)C1.N(C)C.C c1(C(=O)NCCCCCNC(C(CC=C)CC)=O)cc(F)c(N)c(F)c1F N1(C(CCc2c(C)[nH]n(-c3ccccc3)c2=O)=O)CCC2OCC(=O)NC2C1 Cc1ccc(C2(C)CCN(C(=O)CC3CC(N)C34CCC4)C2)cc1 CC1(C)CCN(C(c2cncnc2)=O)C(C(=O)NC2COCC2CO)C1 c1(C(=O)NC2CC(C)(C)SC2)c(O)cnc2ccc(Br)cc12 C(=O)(C(C)(C(C)C)O)NC1(c2cccc(F)c2)CCN(C(C2CC(=C)C2)=O)C1 N1(CC(c2c(C)coc2C)=O)CCc2cc(O)ccc2C1C1CC(=O)CC1 c1(CC#N)ccc(C(=O)Nc2cc(C(F)(F)F)ccn2)cc1 C(N=c1cc[nH]cc1)C1(C(=O)OC(C)(C)C)CC1(C)C Cc1cc(C(=O)NCC(C2CCC2)NC(C2CC=CCC2)=O)nc2[nH]nc(O)c12 CC(C)(CO)C(=O)NCCC1CCN(C(c2cccnc2OCCO)=O)C1 N1(C(c2c(C)scc2)=O)CCCC(CCNC(=O)CC2(N(C)C)CC2)C1 c1(C(C(=O)NC(C)C)N(CCOC)CC#N)cc(Cl)c(OC)cc1OC C1(C(=O)NC(C(=O)N(CCF)CC)Cc2cnn(C)c2O)CC(C)(C)CCO1 c1(CN(C2CCCC(c3ccccc3)C2)C)ccccc1OC(F)(F)F C1(C2CCOCC2)(C(=O)NCC2CCN(C(=O)C3=CCCSC3)C23CC3)CC1 C(=O)(CCC(CC)OC)N1CCC(C(C(N2CC(CCC)OCC2)=O)C)CC1 c1(C(=O)NCC#CCNC(C(N2CCN(C)CC2)C)=O)ccc2cccnc2c1 C(=O)(C(CCC(C)(C)C)N1CCC(F)(CO)C1)NCCCOC N1(C(C(=O)NC(C(C)NC(C=C(C)C)=O)CO)C)CCc2ccccc2C1 C(=O)(CC(C)(C)c1cccs1)NCCC(=C)C.C(=O)(C(C)N(C)C(C)=O)N C#CCCC(C(=O)N1CCC1CO)NC(c1cc(C)c(N)cn1)=O C(=O)(C1=CS(=O)CCC1)NCCCCN(C(c1ncnc(OC)c1F)=O)C c1(C(=O)NC2CC(CNC(C(C(CC)C)C)=O)C2)ccc2c(c1)CCC(=O)N2 c1(C(N2CC(NC(C(N3CC(C)C3)C)=O)C(O)C2)=O)cnc2c[nH]nc2c1 C1(N(C)C)CCC2C(C1)OCCN2C(=O)CSc1ccc(F)c(F)c1 c1(C(=O)NCCNC(c2ncsc2Cc2ccccc2)=O)[nH]nc2ncccc12 CCC(CNC(C1(c2ncco2)CCC1)=O)NC(=O)COC1CCOC1 C1(NC(CCC2(C)CN(C(C(CC)OCC)=O)C2)=O)CN(C)C2(CCC2)C1 Cc1n[nH]c(C)c1C(C)CC(=O)N(CC)C1CC1.c1(C=O)cncn1C(C)C c1(C(N2CCN(C(Cc3ccc(C)c(Cl)c3)=O)CC2)=O)cnc2[nH]cc(C)c2c1 C(=O)(CC(C)P(C)(C)=O)N(CCCN(C(c1c(C)snc1)=O)C)C N1(C(C2(OC)CCCSC2)=O)CC2(CCCCN(C(C3CCN(C)C3)=O)C2)C1 C=CC(CC(=O)N(CC(C)NC(C1C2(CC2)C12CC2)=O)C)c1ccccc1 N(C(=NCC(C)N1CCCC1)NCC1CCCCC1)Cc1c(C)cccc1C c1(C(N2C(CNC(C3CCSC3)=O)CC(OC)C2)=O)ccc2sc(O)nc2c1 CCCCCC(C)(C)C(=O)N1C2CCC1C(CNC(=O)CC1CC(OC)C1)C2 N1(C(CSCCC)=O)CCC(C)C(CNC(C2(c3n[nH]cc3C)CC2)=O)C1 c1(NC(C2(O)CCN(Cc3c(Br)ccc(Cl)c3Cl)C2)=O)cc([N+](=O)[O-])ccc1Cl C12(C(=O)Nc3cc(C)cc(Cl)c3)CCC(CN(C(c3cnc(O)c(C)c3)=O)C1)C2 O=C(C(F)C(F)(F)F)NCC1COCCN(C(c2nc(Cl)ccc2Cl)=O)C1 Cc1coc(C=CC(=O)N(C)CC2(O)CCN(C(=O)C#CC3CC3)C2)n1 c1(COC)nc2n(n1)CC(NC1CCNC13CCC3)CC2 N1(c2nc(C(C)OCC)nc(Cl)c2)CCCC2(CCN(C(C3CC3CC)=O)C2)C1 C1(C(=O)NC2C(NC(C=CCOC)=O)CCOC2)CC2(CCC2)CO1 C=CCC(C(=O)NCCN1CCCOCC1)NC(=O)C(n1nccc1C)C C1(C(=O)NCC(N2CCCC2)=O)CC12CCN(C(=O)C(F)(F)Cl)C2 N1(C(Cc2c(C(C)C)con2)=O)CC(NC(C2CCCCO2)=O)CC(F)C1 C(=O)C1=CCc2ccccc21.CC(O)(C(=O)NCC1CC(C)CO1)C1CCC1.N C1(C(=O)NC(CCCC)C(=O)NC(C)C(=O)OC)Cc2ccccc2C1 C1(CN(C)C)CCCCO1.C1C(C)(C)NC(=O)COCCCN1C C1(C)(CN(C(c2cn(CCCC)nn2)=O)C)CCCC1.c1(C=O)ccc(F)o1.N N1(C(C2C(CC)CCO2)=O)CCCC(CNC(=O)CN2CCCCC2=O)C1 C1CCCC1.c1(C(=O)N)ccnn1CC(F)(F)F.C(=O)C(C1CC1)C1CC1 C(C1CCCc2sc(C)nc21)N(C(=NCC(=C)C)NC(c1nncs1)C)C C(=O)(C(F)CC1CN(C(=O)CC2CC2(C)C)C1)N(C)CC1CCCO1 c1(CN(C(=O)COc2cccnc2)C)cc(-c2ccc(CO)nc2)ccn1 C1(F)(C(=O)NC(CCCC)CNC(c2cccc(=O)o2)=O)CCC(F)(F)CC1 C12(OC)CCC(C(=O)N)(CC1)C2.C1(O)CCN(C(=O)Cc2nc(C)sc2C)C1 CC(CCCNC(c1nc(C(F)(F)F)cs1)=O)NC(=O)CCCn1ccnc1 c1(NCC(CC(C)C)NC(C2CC3(C2)CC(F)C3)=O)nccnc1C#N C1(C)(C(=O)NCCSC(C)C)CC12CCN(C(c1ccc(O)cc1)=O)CC2 N1(C(C(C=CC)O)=O)CCN(C(c2ccnc(Cl)c2N)=O)CC1CO c1(Cc2c(C)sc(-c3cnn(CCCNC(C)(C)C)c3)n2)cccc(C#N)c1 C12(CNC(c3ccc(C)n3C)=O)CC(CO1)N(C(=O)CCC)C2.[SH](C)(=O)=O c1(CN2CCC(NC(c3c(C)cnnc3)=O)C(O)C2)cccc([N+](=O)[O-])c1 Cc1cc(C(=O)OC(c2ccccc2)C)c(C)n1-c1cccc(F)c1 c1(C(=O)NC(CCC)C(=O)NCCCN(C)C(C)C)cc(C#N)ccc1N c1(C(N(CC(C)CNC(C2OCC2(C)C)=O)C)=O)ccc2snnc2c1 N1(C(C(Cc2ccsc2)OC)=O)CCN(C(=O)C=C2CCC2)C(C)C1 C(=O)(C1CCOc2ccccc21)N1CC(C)N(C(C23CC(C2)C3)=O)CCC1 c1(C(N(CCC)CCNC(=O)CC(C)F)=O)ccnc(OCC(F)F)c1 C#Cc1ccc(C(=O)NC(CNC(=O)C(C)c2cncs2)C(C)(C)C)o1 N1(C(C2C(C=C)C2)=O)CCC2(CCN(C(c3cc(C)c(C)[nH]3)=O)C2)C1 N1(C(c2ccc(C(C)=O)[nH]2)=O)CC=CC(NC(=O)Cc2cnsc2)C1 CON(CCC(=O)NC1CC=CC1)C(=O)CC1CCCC2CC12 CC(N=c1cc[nH]cc1S(=O)(=O)NCC1(CSC)CC1)c1ccccc1N(C)C Cn1cnnc1C1CCC1C(=O)N.CCC(O)C.C1(C=O)(CCN(C)C)CC1 c1(OC)ccc(CC(=O)N(C2CCN(C(=O)C)CC2)C)cc1[N+](=O)[O-].C(N)(=O)N c1(CC)ncsc1C(=O)N(CCC(C)(C)NC(=O)CC1CCC(C)C1)C CC1(C)C(S(=O)(=O)NCCN2CCc3sccc3C2)C1(C)C Cc1onc(Br)c1C(=O)NCC1COCC1.c1(C(=O)N)cccc(C2CC2)n1 c1(C(C)C(N2CCN(CC3CCOC3)CC2)=O)ccc(S(N)(=O)=O)cc1 c1(C(N(C(C)CC)C)=O)coc(S(N)(=O)=O)c1.c1(C=O)cc(C(F)F)[nH]n1.N C=CCC(C)(C)C(=O)N1CCCC1CCC(=O)NC(C)C(N)=O C1(C(N(C2CC(=C)C2)C)=O)CC(O)(CNC(C2CC(F)(F)C2)=O)C1 Cc1cc(CNC(c2ccns2)=O)oc1C(N1CCCC1(C)C1CCC1)=O N1(C(c2cnc(OC)s2)=O)CCCC(NC(C2COCC2(C)C)=O)C1.C1CC1.C Cc1cc(O)ccc1CN1CCCCC(NC(c2cc(Cl)ccc2Cl)=O)C1 C(=O)(C1=NN(C)C(=O)CC1)N.N1(C(C2(CC#C)CCC2)=O)CC2CCC(C2)C1 c1(C(C(=O)NCCC)N(C2CC(=O)NC2=O)CCOC)nccnc1C CCC(CCCC(=O)NC(C)(CC(C)C)C(N)=O)NC(=O)C1=CCN(C)C1 C(=O)(C1=CCCC1P(C)(C)=O)N1CC(NC(CCC2CCC(C)O2)=O)C1 N1(C(c2cn(CCOCC)nc2)=O)CC(C)N(C(c2ccn(C)n2)=O)CC1C CC(CNC(c1sccc1CNC(C1CCCOCC1)=O)=O)CC(F)(F)F CC(COC(=O)CC1CCCC(C(F)(F)F)C1)C(C)(F)F N1(C(C(C)O)=O)CCC2(CCC(C(F)(F)F)N2C(=O)CN(C)C)CC1 c1(CN(C)CC2CN(S(=O)(=O)c3cn[nH]c3)C2)cc2ccc(Br)cc2s1 c1(OC)ccc2[nH]cc(C(N3CCC(C)(NC(=O)C(C)N(C)C)C3)=O)c2c1 N1(C(C2CCCC(C)(C)C2)=O)CCCCCC(NC(C23CSCC2C3)=O)C1 C1(OC)CCCN(C(C2(c3ccncc3)CC2)=O)C1.c1(CC(=O)N)ncc(C)[nH]1 Cc1c(-c2ccccc2)nn(C)c1NC(C1CN(C(=O)C(C)O)CCC1O)=O C1(CC#C)(C(=O)NCC(C)(O)CNC(=O)CCc2cccn2C)CCOC1 C1(C(=O)NC)CCCN(C(C2COCC2NC(c2nc[nH]n2)=O)=O)C1 C1(CC)CCC(C)N1C(=O)C(O)C1CN(C(=O)C=C2CCOCC2)C1 c1(CNC(C2CCCC2NCC(O)Cc2ccccc2)=O)ccnc(Br)c1 c1(NC)cnc(C(=O)N(C2(C(=O)NC3COC(C(F)F)C3)CC2)C)cn1 N1(C(c2cnc(CC(F)(F)F)s2)C(=O)NCC(C)C)CCCc2ccc(F)cc21 Cc1ncc(Br)c(C(=O)NC2(CN(C(=O)C#CC3(C)CC3)C)CC2)n1 C(CCCNC(c1cc(C(N)=O)cs1)=O)OC.c1(CCC=O)cnc(O)[nH]1.N c1(C(=O)N)cc2c(s1)COCC2.Cc1nn(C)cc1C(=O)NCC(C)C1CCC1 n1(C(C)C)cccc1C(=O)N(C(C)CCNC(c1csc(C2CCCO2)n1)=O)C c1(C(=O)Nc2ccc(C(C(=O)O)(F)F)cc2)cc(Cl)cc2cc[nH]c12 C1(NC(c2cc(C)nn2C)=O)CN(C(C2(c3cccs3)CC2)=O)CC1C#N c1(C(=O)NC2C3(CC(NC(C(C)CN(C)C)=O)C3)C2)cnc2sccn2c1=O C(=O)(C(O)C(C)CC)NCCN(C(C=C(CCC)C)=O)CCC c1(OC)ccncc1C=O.C1(CC=O)CCCS1(=O)=O.C(C)(C)C1CCC1.N C=C(Cl)CC(C(=O)NOC(COC)COC)NC(c1cc(COC)on1)=O Cc1cccc2ccc(C(N3CCC(C)(NC(=O)C4=NOC(C)C4C)C3)=O)nc12 C(=O)(C(F)(F)CCC(=O)O)NC1(CC(=O)OCC)CCNCC1 C(=O)(CC(C)CC(C)(C)C)N1CCC(CC)CC1.O(C(F)(F)F)CC=O.CO.N C#Cc1ccc(C(N2CCCCC2CNC(C2CCCCNC2=O)=O)=O)c(F)c1 C1(C(=O)NCC(C)N(C(Cc2cccc(OC)c2)=O)C)Cc2cc(C)ccc2O1 N(S(=O)(=O)N1C(C(=O)O)CCC1(C)C(=O)O)c1cc(C)nnc1C N=c1[nH]cnc2cc(C(=O)NC(C)C3CC3)ccc12.CC(F)(F)F.C(=O)(C)N c1(C(N2CC3(CCN(C(C(C(CC)C)O)=O)C3)C2)=O)sc2cc(Cl)ccc2c1Cl C1(NC(CNC(N)=O)=O)CS(=O)(=O)C12CCN(C(C1CC3CC3C1)=O)CC2 N1(C(C=CC(C)(C)C)=O)CC=CC1C(N1CC(OCCO)C1)=O C1(C=O)CC2(CC(C)=NO2)C1.C(=O)(C(F)=C1CCCC1)N(C(C)C)CC c1(NCCC(c2ccccc2)Oc2ccc(F)cc2)ccc2c(Cl)cccc2n1 c1(C(=O)NC(c2c(C(C)C)cccc2)(C)C)cc(I)ccc1N c1(NC2(CC)CCCCC2)nc2ccccc2nc1N1CC(C)OCC(C)(C)C1 Cc1ccc(C)n1CC(=O)NCc1cc(C(N2CCC3CC23C)=O)ccn1 N1(C(c2c(C)cccc2)C(=O)NC(C)C)CCCCC1P(C)(C)=O c1(COC(C2CN(C(C)C3CC3)C(=O)C2)=O)cc(F)cc(C#N)c1 C1(NC(=O)CSCC(F)F)CCCN(C(=O)C=Cc2cc[nH]c2)CC1 c1(OCC(=O)NC2CCCN(C(CCC)=O)CC2F)ccc(S(N)(=O)=O)cc1F C1(C(=O)NC2C(CNC(C(c3cn(C)nc3)(C)C)=O)C2)CCC(F)(F)C1 C=CC(CC)CC(=O)N1CCCC1CCNC(c1conc1C1CC1)=O N1(C(CCCCOCC)=O)CCC(C)(C)CC1C(N1CCCC(C)(CC)CC1)=O c1(C(N2C(C(C)(C)NC(C3CCCOC3)=O)CCC2)=O)noc2c(F)cccc12 C(=O)(C1CCCc2ncnn21)N1C(C)CN(C(c2cc(C(N)=O)co2)=O)CCC1 C1(COC)CC2CCC1N2C(c1csc(-c2cnc[nH]2)n1)=O C(=O)(CCCCC(c1nnnn1CC1CCOCC1)NCC1(C)CC(C)C1)OC C1(O)(C(=O)NC(CNC(C(COC)OC)=O)CO)CCCCCC1 c1(COC(C2(c3ccc(C#N)cc3)CC2)=O)cc(Br)ccc1[N+](=O)[O-] c1(CC(=O)N(CCCNC(c2c[nH]c(-c3ccncc3)n2)=O)C)ccncc1Cl C=CCC(C)(C)NC(c1coc(C(C)NC(=O)CN(C)C(=O)OC)n1)=O N1(C(C2(C=O)CC2C)=O)CCCCC(C(N2CC(C(=O)N(C)C)C2)=O)C1.CO C(=O)(CCC1CC1)N(CC)CC1CC1.C(=O)CC1(N(C)C)CC1.N Cc1noc(C(=O)NC2(CNC(=O)Cc3ccnn3C)CCC2)c1C n1(CCC)nc(-c2cc(Cl)ccn2)nc1-c1coc(-c2ccccc2)n1 c1(C(N2C(CC(=O)NC)CN(C(=O)C(C)(F)F)CC2)=O)cc2ccncc2s1 Cc1cc(C(C)NC(c2n[nH]cc2C)c2nnnn2CC2CC2)cc(C)c1 C1(CC(N)=O)CCCCN1C(c1cccc(C(F)(F)F)c1)C(=O)NC1CCCC1 c1(C(N2CC(C(=O)Nc3nccc(C)c3Br)SCC2)=O)cnc2ccccn12 C=C=CC(C)C(=O)NC1CCN(c2cc(C(=O)OC)ncn2)C1 c1(C(=O)NCCC(C)C)cc(S(C)(=O)=O)cs1.C1(CC=O)CCC(=O)NC1 Cc1cc(NC(=O)CNC(c2cnn(C3CCN(C)CC3)c2C)=O)ccc1Br N1(C(C2(COC)CC2)=O)CCC(CNC(=O)CCC2CC2(C)C)C1.O N1(c2nnn(C)n2)CCCC2(NC(c3cc4c(nc3O)CCC4)=O)CCCC12 c1(C(N2CC(NC(c3cnc(O)c(F)c3)=O)C(O)CC2)=O)onc2c1CCCC2 c1(SC2(C)CC(C(=O)OC)C2)nc2ncccc2o1 C1(C#N)(C(N2CCN(C)C(CNC(=O)C(C)(C)CO)C2)=O)CC2C=CC1C2 c1(CSC(C)C(c2ccccc2)=O)c(Cl)cc(Br)cc1Cl N1(C(C)=O)CC2CC(NC(=O)C(c3ccc(F)c(Cl)c3)(C)C)CC1C2 c1(CCC=C)ccc(C(=O)NCC2COCC2NC(C2CCO2)=O)cc1 N1(C(C2CCCN(C(=O)CCc3cncs3)C2)=O)CC2CCOC2C1 c1(C(N(CCNC(=O)CCc2cn[nH]c2)CC)=O)cc[nH]c(=N)n1 C1(NC(CCN(C)CCO)=O)CCCCCN(C(c2ncc(C(F)F)s2)=O)C1 C1(C=O)CC(C2CCCC2)C1.c1(CCC(=O)NC2CC(O)(C)C2)ncc(F)cn1 CC1C2CCCCC2CN1C(=O)NCC1CCCCC1(F)F C(=O)(C1Cc2ccc(Cl)cc21)NCC(C)NC(=O)CC1OCCC1C C1(C(=O)NC2(CN(C(C3=NOC(C)C3)=O)C)CC2)CC(=O)N(C)C(=O)N1 CCS(=O)(=O)Cc1ccccc1.Cn1cc(CC2CC(N3CCOCC3)C2)cn1 C1(C(=O)NC2CN(CC)CC2(C)C)CCCN1NC(=O)CC(COC)COC C1(NC(CC=CC)=O)CN(C(c2cc(C(=O)OC)c[nH]2)=O)CC1C(F)F c1(CNC(C2(C)CCC2)=O)nocc1C(=O)NOCC(O)CO c1(OCC)cc(N2CCC(C)C(NC(=O)C(C)(C)C)C2)nc(C)n1.C(C)=O CCCCCN(CCC(=O)N1CC(CNC(=O)CCN(CC(F)(F)F)C)C1)C c1(NC(C2CCCC2NCc2cc(CO)ccc2O)=O)c(Cl)cc(Br)c(Cl)c1Br Cc1nc2ccc(O)cc2cc1C(N1CC(NC(=O)C)CC1(C)C)=O.C(N)(=O)N C1(NC(c2cc(C)ncn2)=O)CCN(C(=O)CCC(C)(F)F)C1(C)C c1(C(NOCCCCC)=O)ccc2c(n1)CN(C(c1ccc(C)n1C)=O)CC2 c1(CC)cc(C(N2CC(CO)C(O)C2)C(=O)NC2CCOC2)sc1C c1(C(=O)NC)cc2cc(NC(N3CC4(F)CCC3(CO)C4)=O)ccc2[nH]1 c1(C(N(C2CCN(CC=CCl)C2)CC)=O)cc(C(N)=O)[nH]n1 CC(C)C(C(=O)N1CC2(CC2)CC1CO)C(C)NC(=O)C=CC1CCCC1 c1(CC)nn(C)c(CC)c1S(=O)(=O)NC(C)C(=O)NC(C)C c1(C(N(CC(=O)NCC(Cl)C(C)(F)F)C)=O)cncc(C#N)c1 N1(C(C(C)CO)=O)CCN(C(=O)COc2cccnc2)CC(CO)C1 c1(C(N2CC3C(C(=O)N)(C3)C2)=O)cc(Br)cc(F)c1F.c1(OC)cccc(C)n1 C1(C(N2CC3CN(C(C4(C)COC4)=O)CC3C2)=O)COc2ccccc2O1 C1(C(=O)NCC2CCCOCC2)C2CC(O)C(C2)N1C(C1CCOCC1)=O C12(C(N(CCC(C)NC(C3CC34CC4)=O)C)=O)C3C4C1C1C2C3C41C CC(C)CC(CNC(=O)Cc1cccn1C)C(=O)NC1CC=CCC1 N1(C(c2nccc(C)c2)=O)CC2CCC(NC(c3cc4sccc4[nH]3)=O)CC2C1 N1(C(c2ncnc(OC)c2F)=O)CC2CCC1CN2C(c1nnc(O)nc1O)=O Cc1cc(C(N2CCC(C(=O)NCc3cnsc3)C2C(C)C)=O)[nH]c1C c1(N2C(=O)CCn3cc(cn3)C2=O)cc(C)c(S(N)(=O)=O)cn1.CC#CCO N1(C(c2ccc(N)cc2Cl)=O)CCC2CC(NC(c3cnoc3)=O)CCC2C1 C1(C(C(=O)NCCSC)N2CCC2c2ccc(Cl)cc2)CC(C)CC(C)C1 c1(C(N2CC3(CN(C(=O)CC45CCC(CC4)OC5)C3)C2)=O)n[nH]c2c1CCCC2 C(=O)(C(F)CC(CC)CC)NC1CN(C(c2c(CC)nn[nH]2)=O)CC(F)C1 c1(C(=O)NC(C)CCCCNC(=O)C(C)C(F)F)ccc2ccnc(Cl)c2n1 S(=O)(=O)(c1ccc(C(F)F)cc1F)N(C1CCCCCC1O)C C(=O)(C1=NOC2(CCOC2)C1)NC(CN(C(C1=CC(C)(CC)C1)=O)C)(C)C C(=O)(C(CC)CC(C)C)N1CC(CCC)C(C(=O)NC23CCCC2CCC3)C1 c1(NC(c2c(CC)cc[nH]2)=O)ccc(CN2CCNCC2)cn1 C1(C(=O)NCC(C)NC(c2cc[nH]n2)=O)CCN(c2ccc(Br)cn2)CC1 Cc1nnnn1CC(=O)NC1CCCC1NC(c1cc(-c2ccn(C)n2)on1)=O N(C1COc2c1ccc(Cl)c2Cl)C(CCCCCn1cc(COC)nn1)=O Cc1c(Cl)nc(CC(C)C)[nH]c1=NC(C)CC(C)NC(C1CC(C(C)C)=NO1)=O C1(C(=O)NC(CNC(C=CCC)=O)C)CC(=O)N(C2CCCC2)C1 CCCCC(CC(=O)NCc1c[nH]nc1OC)NC(C1CC12CC2)=O N1(C(c2c(C)nc(CC3CC3)o2)=O)CCCC2(C1)CN(C(C1CC=CCO1)=O)C2 C1(C(N2C(C(N3CC(O)(c4cnn[nH]4)C3)=O)CCC2)=O)CCC(F)CC1 C(=O)(C1CCc2cc(C)ccc21)NC1CC(NC(CNC(COC)=O)=O)C1 CC1CCN(C(c2ccc(S(C)(=O)=O)s2)=O)CCN1C(=O)CCc1ncco1 C(C(C)(O)C(=O)NCCC(C)Nc1nccc(-c2ccccc2F)n1)OC c1(C(=O)NCC2CCC(NC(CC3N(C)CCCC3)=O)C2)ccc2[nH]ccc2n1 N1(C(C(C(C)C)N(C)C)=O)C2CCCC1CN(C(c1cc(F)cc(Cl)c1)=O)C2 CC(=O)C(C)CC(C)C(=O)NC1(CNC(=O)C(C)(O)C2CCC2)CCC1 CC(C)CCC(C(=O)NCCC(=O)NC(N)=O)NC(c1ccc(N)c(F)n1)=O c1(C(C)C(N2CC3C(N(C(=O)CSC(F)(F)F)C)C3C2)=O)ccc(F)cc1F c1(NC(C2(O)CCN(C(Cc3ccc(C)nc3)=O)C2)=O)cc(I)ccc1C CC1(C)CN(C2CCCNC2=O)CC1NC(c1ccccc1C1(C)CC1)=O c1(OC)cc(CC(=O)NC(C)CC(C)NC(c2cscc2C)=O)c(F)cc1O c1(OC)cccc(O)c1C=O.c1(C(N2CCC2)=O)nc(C)[nH]c1C(F)(F)F.N C1(C)COCCN(C(=O)CCC2CC(F)(F)C2)C1.C(CC(=O)N)SCCOC CCC(CC(=O)NC1CCCCC1C(=O)N(C)CC1CCC1)C(F)F C(=O)(C1=NOC2(CCC2)C1)NC1(CNC(C(CC)C(C)O)=O)CCOCC1 C1(CC)CC(O)CCN1C(C1CC(OC)CN1C(c1cnns1)=O)=O N(C(=NCCCC(C)(F)F)NC1CCN(c2ccn(C)n2)C1)C(C)C C1(NC(c2n(CCCSC)nnn2)CCSC)CCC2(CCCC2)C1 c1(CN2CCC(N(C(c3c(C)nns3)=O)C)C2)cccc(I)c1F C1(C(=O)NCC(=O)NC)CC2(CC2)CN1C(c1cnnc(O)c1)=O c1(C(=O)NC(c2cn(Cc3ccccc3)nn2)C)c(F)c(F)cc(Br)c1F CCCCCS(=O)(=O)CC(=O)NCC1CC1C.c1(C(=O)N)cccc(C#N)c1 N1(C(C(COC)(C)OC)=O)CC2(CCC(CNC(C3(C)CC3)=O)O2)C1 N1(C(=O)OC(C)(C)C)CCC(N(C(C2CCCCC2O)=O)C2CC2)CC1 c1(NCc2ccc(C)c(C#N)c2)nccc(=NC(C)c2ccns2)[nH]1 c1(C(=O)NC(CNC(CC)=O)(C)CO)ccc(OC)c(C(C)C)c1 C1(CN(C)C(C2(O)CCOC2)=O)CCC(NC(C2CS(=O)(=O)C2)=O)CC1 C12(NC(=O)CC3CC4CC4C3)CCCC1N(C(C13CC=CC(C1)OC3)=O)CCC2 c1(C(N2CCC2)=O)ccc(F)c2c1OCC2.C(C(=O)NC)(C(C)O)NC(C)=O Cc1cc(=NC(=O)C(C)SCC(=O)NCC(C)NC(c2sccc2C)=O)[nH]o1 N1(C(c2c(C)nccc2Cl)=O)CC(C)CC(C)(C)C1.C1(C=O)C2(CC2)C12CC2 c1(CCC)occc1C(=O)NC(CNC(=O)CC1(N2CCCC2)CC1)CC c1(C(N2CC(C)(NC(c3n(C)cc(C(N)=O)c3)=O)C2)=O)cc2ccccc2nn1 C(CC(C(=O)N1CCC(C(C)O)CC1)NC(=O)C(C)C(F)F)=CC C12(NC(C3C(CC)CCC3)=O)CCCC1N(C(=O)C#CC1CCOCC1)CCC2 C1(CNC(c2c(CCC)nco2)=O)CCC2(CN(C(C3CC3(C)C)=O)C2)O1 CN(C)NC(=O)CCC(=O)N1CC2CCC1C(C(N1CNC(=O)C1)=O)C2 c1(C(N(C2CCN(C(=O)C(C)NC(C)=O)CC2)CC)=O)ccnc2ncccc12 CC1CC=C(C(=O)N2CC(O)(C3CCCN3C(=O)CN3CCCOC3=O)C2)CC1 c1(C=O)nnn(C)c1C.C1(C(=O)NCC2(C(=O)OC)CCC2)CCCO1.C c1(C(N(C(C2CC(C)OC2)=O)C)C)ccccc1Cl N1(C(CCCC(=O)OCC)=O)CCC2(CC1)OCCCC2NC(C1CCC1)=O CC1CC(CCNC(=O)C(c2cccs2)NC(=O)CC2C=CCC2)C1 c1(C(=O)NC(C)CNC(c2cnc(-c3cccs3)o2)=O)cc2c(Cl)cncc2o1 c1(C(N2CC(COC)(C)C2)=O)cnc(C)nc1.C(=O)(CCCn1ccnc1)N c1(N(CCN(CCC2CCC2)C)C)csc(C=O)n1.C(C)(C)C.C(=O)N c12cc(Cl)cc(Br)c1NCC(=O)N2.n1(CC(=O)O)cccc(C(F)(F)F)c1=O N1(C(c2ccnc(C(C)C)n2)=O)CCN(C(C2CCCO2)=O)CC(C)C1 Cc1nnc(NC2CC(CNC(c3cc(C)n(C(C)C)n3)=O)C2)c(C#N)c1C N1(C(C2CC(CC)C2)=O)CCC(NC(c2ccc(CCO)cc2)=O)C(F)C1 Cc1nc(C(=O)NC2CCC2)ccc1[N+](=O)[O-].C1(CC(=O)N)CC(O)C12CCC2 c1(OC)cccc(C=CC(N2CCC(NC(C3CC(F)CN3C)=O)C2)=O)c1 c1(C(C)(C)C)ccc(C(=O)NCC2CC2)cc1.c1(C=O)ccn(C2CC2)n1 C1(CC(N2C(CNC(C(SC)SC)=O)CC2)=O)CN2CCN1CC2 N1(C(C2(C)CC2)=O)CCN(C2CCN(C(C3CCCS(=O)(=O)C3)=O)CC2)C(=O)C1 N1(C(C(n2cc(CN(C)C3CC3)nn2)C)=O)CCN(C)C2CC12 C(=O)(C#CC(C)(C)C)NC1(C(=O)NC(C(=O)OC)CCF)CC(O)C1 C(=O)(C1=CCC(NC(c2cnn[nH]2)=O)C1)NCC1(C(N)=O)CCCC1 c1(C(=O)NCC(CN(C)C(C2(C)CSC2)=O)O)cc(N)c(F)cn1 CCC(CCCC(=O)NCCC(C)C(C)C)NC(=O)CC(C)(C)OC c1(C(=O)NCC2C(C(N(CC(Cl)Cl)C)=O)OCC2)sccc1C#N C(=O)(CCCC(N)=O)N(C(C)(C)CN1CCCC1)CC.C1CC2CCC(C1)S2.N C1(C(=O)NCCOc2ccccn2)C2CCC1CN(C(c1csnn1)=O)C2 C1(CCC)(NC(=O)Cn2cncn2)CCCN(C(C2(C)CC2(F)F)=O)C1 N1(C(c2c(CC)nccn2)=O)CC2CCC1C2NC(c1ccc(CSC)cc1)=O C1(C(C)(C)N(C)C(=O)NC2CC(OC(C)(C)C)C2)CCCO1 C=C(C)CCCC(=O)N1CCC(CCNC(c2coc(COC)n2)=O)C1 n1(CC(C)NC(=O)CCc2csnn2)cc(C(c2cccnc2)O)nn1 OC1CCC2(CCN(Cc3nc(-c4ccccc4Br)n[nH]3)C2)C1 C1(CCNC(CC(C2CC2)NC(C2(CC)CC2)=O)=O)CC2C=CC1C2 C1(NC(c2nc(C)oc2)=O)(CNC(=O)CS)CCOCC1.c1cccnc1.C c1(C=O)ccc2c(c1)ncn2C(C)C.C(C)C(C)C.C1CC1C=O.COC Cc1nn(C)c(I)c1C(=O)NCC(c1ccon1)C1CC1 C(=O)(C1=CC2(CCN(C(=O)C(C(C)C)C3CCC3)C2)C1)N1CCCC1.CC(=O)O N1(C(C(CC(=O)OC)C)=O)CCC2(CC1)CC(NC(c1c[nH]c(=O)cn1)=O)C2 c1(Sc2cc(C(F)(F)F)cc(C(C)=O)n2)ccc2oc(O)nc2c1 C1(NC(C2(C)CCOCC2)=O)CC=C(C(=O)N2CC3CC2CC3CF)C1 C1(=CCNC(CCN(CCCCC)C)=O)CCN(C(C2CC2Cl)=O)CC1 c1(CC=O)ccc(C)cc1.c1(OC)cc(C(N2CC(C(N)=O)(C)C2)=O)on1 C(CC(=O)Nn1ccccc1=O)(C(F)F)NC(c1c(N)non1)=O Cc1nnnn1CC(=O)NC(c1cccnc1)CNC(=O)CC1CCCCO1 C(C1CCCCCC1)=CC(=O)N(CCCNC(C(C)OCC=C)=O)C N1(C(C(C(C)C)F)=O)CC2CCN(C(C3(C)CCNC3=O)=O)CCC2C1 CCC(O)C(F)(F)C(=O)NC(C)CN(C)C(c1cnncc1C)=O C12(CN(CCS(=O)(=O)N(CC)CC)C=O)CCCCC1C2 C(CCNC(c1ccnn1CCF)=O)(C(=O)NCCC1(C)CCCC1)OC c1(C(=O)NCCC2(NC(C3SCCS3)=O)CCC2)scnc1C(F)(F)F N1(C(c2c(C)cc(N)cc2)=O)CC(C)CN(C(=O)Cn2cncc2C)CC1C C(c1cccnc1)=CC(=O)NC1C2CC1N(C(=O)C(F)CC1CCCCC1)C2 c1(C(N2C(C)CCN(C(C(COC)(C)OC)=O)CC2)=O)sc2cccnc2c1Cl c1(CC)ccc(C(N2CCC(C)C2CNC(=O)CC2CCCC2)=O)cc1F C1(OC)CC2(CCC(C(=O)NCCCCNC(=O)CCF)CC2)C1 N#CC1(C(N2CCCC(NC(c3cc(-n4cccn4)ccn3)=O)C2)=O)CCOC1 N#Cc1csc(C(=O)NCC2CC2)c1.c1(C2(C=O)CC2)ccc(Cl)cc1.C N1(C(c2cnc(CC)o2)=O)CCCC(N(C(=O)CC2CCCN(C)C2)CC)CC1 CCCC(CC)C(=O)NCC1COCCN1C(c1cc(O)ccc1OC)=O CC1(NC(c2ccc(-c3cnco3)cc2)=O)CCCN(C(=O)C(F)(F)C(F)F)C1 N1(C(C2CCC(CO)CC2)=O)CC2CC1CC2N1CCN(CC2CC2)CC1 C12(CC=O)CC3CC(CC(C3)C1)C2.Cc1nsc(NC(C2CC2)=O)c1C#N.C N1(C(C(CC)CC)=O)CCN(C(c2cccc(Cl)c2)=O)C(C2CC2)C1 c1(CC)nc(Cl)c(C)c(=NCC(C)(C2CC2)NC(=O)CCc2ccncc2)[nH]1 Cn1nc(C(=O)NC2CC3(C2)CC3)cc1C(F)(F)F.C1(C=O)CC=CC1.N CCC(CC(C)C)C(=O)NC(CCCOC)C(=O)NC1CCCC1(C)N(C)C N1(C(COC(CC)C)=O)C2CCC1CC(CC(C)NC(=O)C(C)C(C)(F)F)C2 C1(NC(=O)C=Cc2cnc[nH]2)CC(F)CN(C(=O)CCn2ccnc2C(F)F)C1 C1(CC=C)(NC(=O)CC(F)(F)Cl)CCN(C(c2cc(C)oc2C)=O)C1 Cc1c(F)ccc2[nH]c(C(N3C4CCC3CC(NC(=O)CC(F)(F)F)C4)=O)cc12 N1(C(CN(C(Cn2ncc(C#C)c2)=O)CC(C)C)=O)CCCCCCCC1 C1(NC(c2ccc(Cl)s2)=O)CN(C(C2CC23CCC3)=O)CC(F)(F)C1 c1(N2CCC(C(C)NC(C3CN(CC(C)C)C(=O)C3)=O)C2)ncc2c(n1)COC2 c1(C(=O)NC2CC3CN(C(=O)CCc4ncccn4)CC23)ccc2sncc2c1 Cn1c(C(N2CC=C(Br)CC2)=O)cc2cc(Cl)ccc12 N1(C(CC(=C)C)=O)CC2CC(F)(F)CCC2(NC(c2cccc3sccc23)=O)C1 N(C(=NCCOC)NCc1cc(C(F)(F)F)co1)C1CN(CC)C(=O)C1 CC(C)C(C#N)C(=O)N1CCCC(CN(C(=O)Cc2ccccc2)C)C1 C1(C(=O)NCC(N(C(CCc2onc(C)n2)=O)C)C2CC2)COC2(CCC2)C1 c1(C(C)C)nnc(CNC(=O)C(n2cc(CCN3CCCC3CO)nn2)C)n1C C#Cc1cccc(OCC(N2CCCC(NC(c3ocnc3CCC)=O)C2)=O)c1 CC(CC(=O)NC)P(C)(C)=O.C1CN(C(=O)C(c2cnn(C)c2)=O)CCC1(C)C C12(C(=O)NC(C3CCCN(C(Cc4c(C)cc(C)s4)=O)C3)C)CCCC1C2(F)F C1(CNC(CN(C(C)C)C)=O)CC(NC(c2ccc(CO)cn2)=O)C1(C)C C1(C=O)CN2CCCN1CC2.C1(C(=O)NC2CC(F)(C)C2)CCS(=O)(=O)N1 C1(C(C)C)CCC(C(=O)NCCC2(C)CC2)CC1.C1(C=O)CCCC2CC12.N C1(O)CCC(F)(F)CC1.c1(N(CCOC(C)=O)CCO)ccccc1.C1CC1 c1(CNC(C2CCC(C)O2)=O)ccc(CN(C(=O)Cn2ccnn2)C)cc1 CCC(F)(C(=O)OC)C(=O)NCC(N1CCN(C(=O)C=C2CC2)CC1)C CC1(C)CCc2c(sc(NC(c3ccc(C(N)=O)c(Cl)c3)=O)c2C(N)=O)C1 C1(N(C(Cc2c(C)non2)=O)C)CCN(C(C2CCCC(F)(F)C2)=O)CC12CC2 C12(NC(C(CC)SC)=O)CC(C1)N(C(=O)CCCC1CCOCC1)C2 CC1CCC(C)(C(=O)NC2CCC2C)C1.c1(C=O)cnc(-c2ncccn2)s1.N c1(NC(C)=O)ccc(C(=O)NC(C)CC)c(Cl)c1.C(=O)CCc1cncs1.N Cc1cccc(C(=O)NCCOCC(=O)NCC2CC2(Cl)Cl)c1C N1(C(NNC(=O)c2ccncc2)=O)CC2(CCC2)OC2(CCC2)C1 CC1(C)CCC(CC(=O)NCC(O)CNC(=O)CC2(C)CCOCC2)C1 c1(C(N(C(C)C2CC2)C)=O)cnc(F)c(F)c1.C(=O)(C(F)OC(F)(F)F)N N1(C(CCC)=O)CCCC1C(=O)NCCCCNC(C1CCC1)=O.C(C)(C)C c1(C(=O)NC2CC(C)N(C(c3ccc4oncc4c3)=O)C2)c(F)cc(F)cc1Cl C1(C(N(C2CCN(C(CC(CC)SC)=O)C2)CC2CC2)=O)CN(C)CCN1C C(CC(C(=O)NC(C1CCCOC1)=O)NC(c1cccs1)=O)=CC c1(C(=O)NCC(C2CCCC2)NC(C=CS(C)=O)=O)cc[nH]c(=N)c1[N+](=O)[O-] C(=O)(C1=CC2CCC(C1)N2C(=O)OC(C)(C)C)N1CC(C)OC(CC(=O)O)C1 C(=O)(CC1=CCCC1)N1CC(OC)C(CNC(C2CCN(C(C)=O)CC2)=O)C1 C12(CC(N3CC(N(CC(C)C)C)C3)=O)CCC1CN(C(=O)C1=CCCOC1)C2 C1(C(N(CC(C)NC(c2ccnc(OC)c2)=O)CC)=O)CCc2ncsc2C1 c1(NC(C2CC2NCc2cc(Br)ccc2Cl)=O)cc([N+](=O)[O-])ccc1Br Cc1ccc(C(=O)NCC2CCCCN(C(C3(F)CCOC3)=O)C2)c([N+](=O)[O-])c1 C(=O)(C(CC)CC(C)C)NC1(C)CCN(C(CCCN(C(=O)OCC)C)=O)CC1 c1(CC)ccccc1CC(N1CCOCC1CNC(C1CNC(=O)N1)=O)=O C1(C(C)C)(CNC(=O)CC2CSC2)CCN(C(=O)C(N2CCOCC2)C)C1 c1(C(=O)OC)ccc(C(N2CC3CC(F)(C2)C3)=O)c(F)c1.C(=O)C(C)O.C Cc1ccc([N+](=O)[O-])cc1C(N1CCC(N(C)C(c2ccn(C3CC3)n2)=O)C1)=O c1(C(=O)N)cccnc1SC(F)F.c1(CCC(=O)N(CC(C)C)C)cn(C)nn1 CC1Cn2nccc2CN1C(=O)C(Cn1cccn1)NC(c1ccsc1Cl)=O N1(C(c2cccc(O)c2)=O)CC2CCN(C(=O)CC(F)(F)F)C2C1 CC(C(=O)NCC(C)(C)CCNC(c1cnnc(O)c1)=O)C(C)(C)C C1(C(N2CCCCC(N(C)C(c3cc(F)c[nH]3)=O)C2)=O)C(C)(C)CCCC1(C)C Cc1cccc(C)c1CNC(C1CCC1)=O.C(=O)(CC)N.C1(C=O)CC1C C1(NC(C2C(C)(C)C2)=O)CC12CCN(C(c1cc(O)cc(Br)c1)=O)CC2 CC1(CONC(C2CCC(CNC(c3cnn(CCF)c3)=O)O2)=O)CC(O)C1 C12(CC)CCC(CC1)N(C(=O)C(F)=CCCF)C2.CCC=O.C(CO)OCC Cc1cccc(C(N2CC(NC(=O)Cc3ccc(Cl)c(Cl)c3)C(F)C2)=O)c1O C(CCOC)(C(=O)NOCCCCC1CC1)NC(c1cc(CC)ncn1)=O c1(CCNC(=O)NCCc2ccccn2)nnc(S)n1C1CC1 C(=O)(CCCCc1ccccc1)N.n1(CC)ccc(CC(=O)NC23CC(C2)C3)n1 C(=O)(C#CC1(CC)COC1)NCCCC(C(=O)NC(C1CCCCC1)CC)O CC1=NOC2(C1)CC(C(=O)N(C)CC1CCCCN1C(C1CCCN1N=O)=O)C2 C(=O)(CCCC(C)NC(c1cc(F)c[nH]1)=O)NC(CCC)(C)CC C(=O)(C(F)C(CC)CC)N1CCC(N(C(C2ON=C(CC)C2)=O)CC)CC1 N1(C(CC2CCC(C)O2)=O)CCC(OCC(C)(C)CC2CN(C(=O)CO)C2)CC1 C1(NC(=O)C=C(Cl)Cl)CN(C(=O)CONC(=O)OC(C)(C)C)CC12CCC2 C1(CC(=O)NCCC(C)N(C(=O)CCc2cc(C)no2)C)(CC=C)CCCC1 C1(CNC(C2CN(C(Cn3ccc(C)c3)=O)CC2F)=O)CC2(CCO1)CC2 O=S(=O)(c1ccc2[nH]c(=NCc3ccoc3)sc2c1)N1CC(F)C(F)C1 Cc1cc(C(N2CCCC2CCC(=O)Nc2ncco2)=O)c(C)n1C c1(C(N2C(C(=O)NC3CCCCC3)CC(=C)C2)=O)c(OC)ccc(Br)c1C C1(N(c2nnc(CC)s2)C)(CO)CCCN(C(C2C(F)(F)C23CCC3)=O)C1 CCC(C)(C)C(C)CC(=O)N(CC(C)NC(=O)CC1(C)OCCO1)C c1(NC(N2CCC(OC(F)(F)F)CC2)=O)cc(F)cnc1OC1CCCC1 c1(C(N2CCC(CC)CC2)=O)ccc2c(c1)[nH]c(=N)n2C.C1(CC)CC1C=O.N c1(C(=O)NC(CC2CN(C(C(CC)O)=O)C2)C)nn(C)c(=O)cc1C C#CCC(C)(CC)C(=O)N1CCN(C(=O)C=Cc2cccc(O)c2)C(C)C1 C1(OC)CCN(C(c2cccc(Br)n2)C(=O)NCc2ccccc2)CC1F C1(C(=O)OC)CCC(CN2C(C(=O)NC3CC3)CC3CC23)CC1 N1(C(Cc2c(C)nn(C)c2)=O)CCCC(NC(c2cocn2)=O)C1C C(=O)(C(C)C(F)(F)F)NCC1CCN(C(CSc2nc(C)[nH]n2)=O)C1 Cc1nc2nccc(N3CC4CC(O)CC(C4)C3)n2n1 C1(C2CN(C(C3CC4CC4C3)=O)C2)(NC(COCC(=O)OC)=O)CC1 N1(C(c2onc(CC)n2)=O)CCC(NC(=O)CC(C)c2cnn(C)c2)C(C)C1 Cc1ccc(C(C)N(C)CCN(C(c2cn(CC(N)=O)nn2)=O)C2CC2)cc1Cl C(=O)(C(C)(C)C(F)(F)F)N1CC(C=C)(CC(N2CCOCC(O)C2)=O)C1 c1(CNC(C2(CC=C)CC2)=O)ncc(C(=O)N)cn1.CCCCCCC1CC1 Cc1cn2cc(-c3nc(-c4ccc5c(c4)CCC(=O)N5C)no3)nc2c(C)n1 CC(C)CCC(O)C(=O)NCc1occc1C(=O)NC1CCCC1C1CC1 c1(C(=O)N)cc2cccc(C)n2n1.CCC(C(=O)NC(C)(C)CC)NC(N)=O O=S1(=O)CCC(n2nc(-c3ccc(Cl)cc3)nc2C2CC(=C3CC3)C2)C1 Cc1cnc(CNC(C2CN(C(=O)CCc3ccccc3Br)CCS2)=O)cn1 N1(C(CC2(CS(C)(=O)=O)CC2)=O)CCCC12CC2.c1(C=O)csc2nccn12.N N1(C(C2(C)CC2(Cl)Cl)=O)CCOC2(CCN(C(=O)C3=CCOCC3)CC2)C1 C(C)(C)(S(C)(=O)=O)c1cn(C(C)C(N2CCCC(C(=O)N)C2)=O)nn1.C1CC1 C1(C(F)(F)F)(OC(CNC(C(=O)OC)CCSC(C)=O)=O)CCCCCC1 C(=O)(CC(Cc1ccc(Cl)cc1)n1cc(CO)nn1)OC.CC N1(C(CCC(=O)OC)=O)CC2(COC(CNC(C3CCCCN3C)=O)C2)C1 c1(C(N2CC(OCCNC(CN(CCOC)C)=O)C2)=O)oncc1C C12(C(N3CCC(CC=C)C3)=O)CC(CN1C(=O)CCC1CCCO1)C2 c1(C(N(C)C)=O)ccc(C(N2CCCCC2CF)C(=O)NCC(F)F)cc1 C1(C(N2CC(F)CC(NC(c3ccc(C)o3)=O)C2)=O)OCCOC12CCC2 C(=O)(C1=CNC2=NCCC2=C1)N1CC2(OCCN(C(C(CCOC)OC)=O)C2)C1 c1(C(N2C(CNC(CC3CC(=C)C3)=O)(C)CCC2)=O)ccc2c(c1)SCCN2 CC1C2C(CCN2C(=O)C2=CCCCCC2)CN1C(C1CC(OC2CC2)C1)=O C(CC1=CCN(C(=O)CCc2cscn2)CC1)NC(C1CCC2C(C1)C2(F)F)=O N1(C(CC(=C)C)=O)CC(F)(F)CC1(C)CNC(c1ccc(C)c(CO)c1)=O N1(C(c2c(CC)cco2)=O)CCN(C)CC1C(=O)NC(c1cnccn1)C C1(C(C)(C)C)(CNC(C2(c3cn(C)nc3)CCCO2)=O)CCN(C(=O)CO)C1 c1(C(N)=O)cc(C(=O)NC2CN(C(C3CCC(C(F)(F)F)C3)=O)C2)co1.C C1(NC(C(C)N(C(CCCCOCC)=O)CC)=O)CC2CC3C(C2)C13 C#CC1(C(=O)NCC2(O)CC2)CN(C(=O)C=CCOC)C1 Cc1cc2c(CC(N3CC(CNC(=O)C4=COCCC4)C4CC34)=O)csc2s1 C1(C(N2CC(NC(c3ccc(C)cc3)=O)C(F)CC2)=O)CC2(C1)CC1(CCC1)C2 N1(c2ncc(CC)cn2)CC2(CCC(NCc3cccc(C(=O)O)c3)C2)C1 C12(NC(CC3C(C)CCC3)=O)CCOC(C)(C1)C2.c1(C(=O)N)c(N)cccc1Cl N12CCCC(C1)NCc1cc(cs1)C2=O.N1(CC)CCOC(C2(C)CC2)C1 C(=O)(C(F)(CNC(c1nc(C)oc1C)=O)C(C)C)N1CCC=C(C)C1 C1(C#N)(C=O)CC2C=CC1C2.C(C)(CC)OC.C(=O)CC(C1CC1)C1CC1 Cc1cc2c(CC(=O)NCCN(C(=O)CC(C)(C)F)CC(C)O)csc2s1 c1(C(C)C)nccc(C(=O)NC2(C)CN(C(=O)CCSc3nccn3C)C2)n1 N1(Cc2cc(C(CC)CC)no2)CCCC2(CCCCC2O)C1 CC(C)(O)C(F)C(=O)N1CCC(CCNC(=O)CC2(n3cncn3)CC2)C1 N1(C(c2n(C)cnn2)=O)CCn2ncc(CNC(=O)C3=CC4CCCC34)c2C1 c1(C(C(=O)NCC(CC=C)NC(=O)C(C2CCC2)O)(C)C)cccc(C)c1 c1(N(C2CCNCC2F)C(=O)Cc2ccc(Br)cc2F)nc(Cl)c2c(n1)COC2 C1(O)(C(=O)CC23CC(C(=O)NCC4CCN(C)C4=O)(C2)C3)CCCCCC1 C1(CC(=O)NC2CC(C)N(C(=O)CCOCC(F)F)C2)CCC2(CC2)CO1 CC1C(C(=O)N2CC3C=CC2C(C(N2CCN(C)C(CO)C2)=O)C3)=NOC1C c1(NC(c2nc(C(N3CCC(N(C)C)CC3)=O)cs2)C)n[nH]c2cc(I)ccc12 Cc1ccc(C2OCCCC2CNCc2ccc(SC(F)F)cc2)cc1 CC1=C(C(=O)N2CCC23CN(C(C2CCC(=O)O2)=O)C3)Cn2nnnc2N1C c1(-c2nc(-c3ccc(N(C)CC)cc3)nn2C(C)C2CC2)ncc(OC)cc1F N1(C(C(C)OCCCC)=O)CCN2CCOCC2(CNC(=O)CSCCCC)C1 c1(NC(C(N2CCN(C(C(=O)NCCCC)=O)CC2)C)=O)cc(Cl)ccc1OC CC(C)(C)C#CC(=O)NC1CCCN(C(c2cc(C3CCC3)[nH]n2)=O)CC1 N1(C(CC2N(C)CCCC2)=O)CC(N(C)C(C2OCCCC2(C)C)=O)C(C)(C)C1 C(=O)(CC=C(Cl)Cl)NCCN(C(c1c(C)cco1)=O)Cc1cccc(Cl)c1 c1(C(=O)NCCCC)scc(OC)c1OC.c1ccccc1.C(=O)(C)N.C=O c1(C=O)cc(S(=O)(=O)N(C)C)c[nH]1.Cc1cc(C(=O)NC(C)CO)n(C)n1 Cc1nc(Cl)ncc1NC(C1CC(NCc2ccc(Cl)cc2O)C1)=O C1(C(=O)NC(c2ccns2)C)C=CCN1C(C1CCC1C#N)=O N1(C(c2ccc(Cl)cc2F)C(N2CCC(C#C)C2)=O)CCC2CCCCC2CC1 C=C(F)C1(CC(=O)N(C)CCC2CCN(C(c3cc(CC)[nH]n3)=O)CC2)CCC1 N1(C(c2c(OC)ccnc2)=O)CC2CC1CN2C(c1c(OC)ccnc1OC)=O CC1Cc2cnccc2N1C(C1CCON1)=O Cc1cccc2oc(=NCC(C)N(C)C(C34CC5CC(C3)CC(O)(C5)C4)=O)[nH]c12 C1(C(C)C)CCC(C)CC1C(=O)OCC1=NOC2CC12 Cc1ccc(C(N2CC3CN(C(=O)CCOCC(C)(C)C)CCC23)=O)c(=O)n1C C1(C(=O)NCC(CNC(c2c(F)ccc(C)c2)=O)(C)O)CCc2ccnn2C1 Cn1cc(NC(C2C=CCCN2C(=O)Cn2ncn(C)c2=O)=O)c(C#N)n1 N1(C(C(C)OCCC=C)=O)CCCC1C(C)(C)NC(=O)Cc1cnn(C)c1 C(C1CS(=O)(=O)c2ccccc21)NC(=O)NCC1(OC)CCOC1 N1(C(c2cc(OCC)no2)=O)CCC2C(C1)CN2C(=O)CCC(C)OC c1(C(=O)NCCCCNC(C(C)(O)c2ccccc2)=O)cc(N)ccc1F C1(C#N)(C(=O)NCC2C(NC(c3nc(C)oc3C)=O)CCCC2)CCCCCC1 c1(C(N2CC(C(=O)Nc3cnccc3I)SCC2)=O)cccc2nc[nH]c12 C1(CNC(C2CC(=C)C2)=O)CC2(C1)CN(C(c1cc([N+](=O)[O-])c[nH]1)=O)C2 C1(CCC)(NC(=O)Cc2ccc(Cl)cc2F)CCN(C(c2cc(F)n[nH]2)=O)CC1 c1(C(=O)NC2(CO)CCN(C(CCC(N)=O)=O)C2)ccc2nccnc2c1 c1(C(N(C(C)C)CC)=O)ccc([N+](=O)[O-])cn1.C1(C=O)CC1C(F)F.N N1(C(c2c(C)noc2)=O)CCN(C(c2cncc(N)c2C)=O)C(CCO)C1 C(CCCCCN=C(NCCC1COCCO1)N1CCC(C)C2(CCC2)C1)SC C1(C(N2CC(C(=O)NCc3cnnn3C)(SC)C2)=O)CC2CCCC2C1 N1(C(C(C(=C)C)(C)C)=O)CC2CCN(C(c3cc4occc4[nH]3)=O)CCC2C1 N1(C(=O)C=C2CCC2)CCC2(CCCN2C(c2cc3cnccc3[nH]2)=O)C1 CN1CC(C)(C(=O)N(C2CCN(C(C3(CO)CCCO3)=O)CC2)C)CC1=O CC1(C)OCC2CC12C(N1CCCOC(CCNC(c2cnn[nH]2)=O)C1)=O c1(C(N2CCCC(CN(C(C(CCCC)C)=O)C)C2)=O)cnc2sc(C)cn12 c1(OC)ccc(C(=O)NC(c2ccc(C)cn2)C)cc1S(=O)(=O)NC1CC1 c1(CCCC(=O)NC2CCC(NC(COCC(N)=O)=O)C2)ccc(Br)cn1 CC(C)CC(CN(C)C)NC(=O)C(O)CCNC(=O)Cc1cn(C)cn1 S(=O)(=O)(C1CC2C(C1)C2(F)F)NCC1(C)C=CCCN1 C(=O)(N=c1ccn(CCF)[nH]1)C1CCN(C(C)=O)C1.N1(C=O)CCSC(C)CC1 N1(C(c2c(CC)ncs2)=O)CCC(C(=O)N(C2CC3(CCC3)C2)C)CC1 CONC(=O)C(=O)NCCOC1CCN(C(=O)C(C)(C)CN(C)C)C1 CC1(C(=O)Nc2cccc(CCO)c2)C=CCN1C(=O)CCc1ncccn1 C12(C(=O)NCC3(CF)CCNC3)CC3CC(O)(C1)CC(O)(C3)C2 N1(C(C(C=C)C)=O)CC(NC(c2ccc(C(F)F)cn2)=O)CCC1C C1(F)(C(=O)NC(C2CCOC2)CO)CCCN(C(C23CCC(CC2)CO3)=O)C1 c1(C(N2CC(C)(C)C(CNc3nc4cccnc4s3)C2)=O)ccn2cncc2c1 C(C(=O)NC(c1cnn(C2CCC2)c1)C)(C(C)C)SC [N-]=[N+]=Nc1cccc(C(=O)NC2CN(C(=O)C3=COCCO3)C2)c1 C(CCC(C)C)(C(=O)NCCC(O)CO)NC(C(C(=O)OCC)OC)=O C(CNC(c1ccc(F)s1)=O)(C(C)C(C)C)NC(Cc1c(C)n(C)nc1)=O CCC(C)C(C(=O)NCC(O)Cn1cccn1)OC Cc1cc(C=CC(=O)NC2CC(CNC(=O)C(C)CF)C2)ccc1Br CC1CCN(C(=O)OC(C)(C)C)CC1CC(=O)Nc1cnn(C)c1.CCF.C c1(CC)c(CNC(c2ccccc2)C(C)O)cccc1C c1(N2CCC(CNC(CC3(OC)CCC3)=O)C(F)(F)C2)ncnc2c(Br)csc12 C(=O)(CC(F)(F)C(F)(F)F)NC1CN(C(Cc2c(CO)nc(C)c(C)c2C)=O)C1 C1(NC(=O)CNc2ncccn2)CCCC2CN(C(=O)Cn3cnnn3)CC12 Cc1cc(NC(CC(C)C)C(=O)NCC2CCCn3ccnc32)c(Br)c(C)c1Br c1(C(N2CCCC(N(C(C3CC3F)=O)CC)C2)=O)ccc2nnc(O)n2c1 c1ccc(NC)c(OC(F)F)c1.C(CC(O)C(C)C)NCC1C(OC)CCC1 c1(C(N2CC(O)(CNC(CC(C=C)(C)C)=O)C2)=O)cc(C)cc(C)c1O C1(NC(C2(C)CCN(C(C3CCC3(F)F)=O)C2)=O)CCCCC1N=[N+]=[N-] C1(CNC(C2(CCC)CC2)=O)CN(C(=O)CCO)CC1(F)F.c1cccnc1 CN1CCOC(C(=O)NCc2ccc(CNC(c3ccnc(O)c3)=O)cc2)C1 c1(CC(=O)NCCCNC(c2ccnc(OCC(F)F)c2)=O)cccc(F)c1F C(=O)(CC(CC)C(C)(C)C)N1CCC(C#C)(C(=O)NCC(=O)N2CCCO2)C1 c1(NC(C2N(C(c3[nH]cc(CC)c3)=O)CCC2)=O)ccc(C(F)(F)F)cc1C#N C1(NC(c2n(C=C)nnc2)=O)CC(NC(c2c(F)cccc2Cl)=O)C12CCC2 c1(C(N2C(C(N3CCC(OC)C3)=O)CC3CC32)=O)cc(Cl)c(Cl)cc1F C(CCC)(C(=O)NC(C1(O)CN(C(c2cncc(F)c2)=O)C1)C)=CCC c1(C(=O)NC2(C)CCN(C(C3C(OCC)C3)=O)C2)cccc(F)c1N N1(C(C(CC)Oc2cccc(Cl)c2Cl)=O)CCN(C(=O)CC2(C)CC2)CC(O)C1 N1(C(c2nc(C)n(C)n2)=O)CCOCC(CNC(=O)C(C)n2cncn2)C1 c1(NC2CN(C(CCCCC)=O)C(C)C2)ncnc2cnccc12 c1(C(N2CCCC(N(C(CN(CCC)C)=O)CC)C2)=O)cc(N)cc(O)c1F C1(c2nnnn2CCOC)(NC2(COC)CCCCC2)CC2CCN(C2)C1 C1(OC)(CNC(=O)NC(c2cccc(Nc3ccccc3Cl)c2)C)CCOCC1 CC1CN(C(=O)CC2CCCS2(=O)=O)CC1CNC(=O)C.C1CCOCC1.O N(C1CCCn2cnnc21)C(CCCC(CC)NC(=O)C(c1ccn(C)n1)C)=O NC(=O)CC(C(=O)N1CCN(C2CC2)CC1)NC(=O)CC1(O)CCOCC1 C1(CN(C(c2cc(Br)no2)C(=O)NC)C)CCSC1(C)C c1(OC)cc(C#N)ccc1F.c12cc(nc(C)c1)CN1CC3CN(CC13)C2=O C=CC1(CC(=O)NC2CN(C(=O)Cn3cc(CC)cn3)CCC2O)CCCCC1 c1(C=O)n[nH]c(C)c1[N+](=O)[O-].CC(C)(C)C.C1(C=O)CC1C=O.C#CC.N C1(Nc2cccc(C(=O)OC)c2O)CCC2(CCO2)CC1 c1(C(N2CCN(CC)CC2)=O)cc(F)cc(S(N)(=O)=O)c1.CC(F)(F)CC(=O)N C1(NC(c2cc(CC)nn2C)=O)CN(C(c2ccnc(C)c2)=O)C2(CCOC2)C1 CC1(C)NC(=O)CC1C(N1CC(O)(CNC(C2CC=CCC2)=O)C1)=O C1(NC(C2C(OC)CCC2)=O)CCCCC12CCCN(C(=O)C(F)(F)C(F)F)C2 N1(CCC=O)CCSC(C)(C)C1.CC(C)(C)CC(=O)NCC1COC(C)C1.N C1(NC(CN2CCN(C)CC2)=O)CC2CC(NC(C3CSC3)=O)C1C2 C1(C(N2C(C(CCC)C)CCC2)=O)CCC2(CC1)CCC2N N1(CC(=O)NC(C)=O)CC(C)(C)CCC1C.c1(C=O)ccnc(C2CC2)c1 C1(CCCNC(CC2(OC)CC2)=O)CN(C(=O)CCOC2CC2)CCO1 C1(C(=O)NC(COCCOC)C)C=CCN(C(=O)COCCCC(C)C)C1 C(c1ccncc1)=CC(=O)NCCOCCN(C(c1c(C)ocn1)=O)C C(=O)(CC(O)CC(C)(C)C)N1CC(C(C(=O)NCC2(C(C)C)CC2)O)C1 C1(C(=O)NCC2C(NC(C3(SC)CC3)=O)CCC2)CCOC(C)(C)C1 C1(NC(C2(C)CC(C)C2)=O)CN(C(=O)C(F)(F)c2cncs2)CC2(CCC2)C1 CC1CCCCC1C(=O)NOCC(=O)NCCC1CCCN1C1CC1 C1(C(=O)NC2CN(C(C3CC(C(C)C)C3)=O)C(C)CC2)CCC2(CCC2)CO1 c1(C=O)c(S(C)(=O)=O)cnn1C.Cc1nn(C)c(C)c1C(=O)N.C1CC1.C CN1CC(C(=O)NC2CCN(C(=O)CSCc3csc(=N)[nH]3)CC2)CC1=O C1(NC(C2(OC)CCSC2)=O)CCN(C(c2c(C)ccnc2O)=O)CC(C)(C)C1 Cc1csc(C(N2CCC(O)(C(C)NC(=O)CC3(C)CC3)C2)=O)c1C CCC(CC(=O)N1CC2CC2(C(N2CC=CCC2C(=O)OC)=O)C1)CC(C)C C12(NC(CSCCC#N)=O)CCC(CC1)C2.C1(C=O)CCC(C(N)=O)C1.N C(=O)(C1=CCCCCC1)NC1C(C(F)(F)F)CCN(C(c2c(C)noc2)=O)C1 C(CCN(C(=O)CSc1nc[nH]n1)C)(C(C)C)NC(C(c1ccc(C)s1)C)=O N1(C(c2cc(I)n(C)n2)C(=O)NCCC)CCCC(C(F)(F)F)CC1 N1(C(C(COC)NC(C)=O)=O)CC(C)CN(C(=O)CC2CC2)C(C)C1 C(C(C)(O)CC(=O)N1CCOCC1CNC(c1cc(C)c(C)s1)=O)OC C1(CN(C(c2n(C)nnn2)CCc2ccccc2)Cc2ccsc2)COC(C)(C)C1 N1(C(C(C2(C)CC2)NC(c2cc(C(C)C)[nH]n2)=O)=O)CCc2nocc2C1 C1(C(=O)NC2CC(OCC)C2OC)CCCC2(CCOC2)O1 C1(C(=O)NCC(C#C)CC)CCN(C(C2CCN(OC)CC2)=O)CC1C c1(C(=O)OC)cc(NS(=O)(=O)c2ccc(C(F)(F)F)o2)c(F)cc1C C(=O)(CS(=O)(=O)CCC)N(CC(C)O)CCNC(C(CCC)CC)=O N1(C(C(CC)C)C(=O)NCC2CC(F)(F)C2)CC2CCC(N(C)C)C2C1 c1(C(N(CCCNC(=O)CC2(C)CCC2)CC)=O)n[nH]c(C)c1Cl C(C(O)C(=O)NCCN(C(=O)Cc1c[nH]nc1O)C1CC1)OC C(=O)(CC(O)CC(C)C)NCC(C)NC(c1cc(C)c(N)cn1)=O c1(C(=O)NC2(C)CCN(C(C(n3ncc(C)c3)C)=O)C2)nc2ccccn2c1F c1(CC)cccc(CC)c1C(=O)NC1CC1C.c1(CC=O)cncnc1O.N CP(C)(=O)CC(=O)NC(C1C=CCN1C(=O)Cc1cccc(C(N)=O)c1)=O CCC(C(=O)NCC(N1CC(CCOC)C1)=O)NC(C)=O c1(CC(N2CC=CC2)=O)ccc(C2CCCC2)cc1.C1(C(=O)NC)CC1(Cl)Cl C1(C)(C(=O)NC(CC)CN(C)C(C2CN(C)C2)=O)CCC(=O)C1 C1(NC(C2(C(=O)OCC)CCO2)=O)CCCCCN(C(C2CC(O)C2)=O)C1 C1(CC(=O)NCC2CN(C(c3ccc(CC)s3)=O)C2)(CC=C)CCCC1 c1(-c2c(SC)cccc2)cnc(C(=O)NCc2cccc(F)c2)cc1C C1(CNC(CCCCC=C)=O)CC2(CC(NC(=O)CCCOC)CCS2(=O)=O)C1 N1(C(CCc2ncn(C)c2)=O)CC2(C1)CN(C(c1cnnc(Cl)c1)=O)CCO2 C1(C)(CNC(C(c2ccc(C)s2)C)=O)CCN(C(=O)C=CC2CCC2)C1 N1(C(CCN(CCC)C)=O)CC(O)CC1(C)C(=O)NC(C)Cc1cn[nH]c1 C1(NC(Cc2cc(C)nn2C)=O)CCN(C(c2cc(Cl)cs2)=O)C(C2CC2)C1 N1(C(C2CC2F)=O)CC2CC(NC(C34CCC(CC3)CC4)=O)CC1C2 C1(CNC(CN(C)CC)=O)C2CCCC1N(C(=O)CS)C2.c1cccc(C)c1 N1(C(Cc2cccc(C)c2)=O)CCOC2(CCCN(C(c3n[nH]cc3C)=O)C2)C1 C1(NC(C(CO)OC)=O)CN(C(=O)CCc2ccc(F)cc2)CC12CC2 C1(CC(C)C)CCN(CC2CCCCC2CC(F)(F)F)CC1 C1(C(N(C2CN(C(=O)C=Cc3cc[nH]c3)CC23CC3)C)=O)OCCOC12CCC2 CCC(CC)N=c1ccc2cc(S(=O)(=O)NCC(c3ccco3)O)ccc2[nH]1 c1(CC(=O)NC)ccc(O)c([N+](=O)[O-])c1.C1C2CN(C(=O)CC(C)(C)O)CC12 c1(C(=O)NCC2(O)CC(NC(CCC#C)=O)C2)c(Cl)ccc(Br)c1F c1(C(=O)NC(c2ccccc2)CNC(c2nc(Cl)cs2)=O)ccc2ncnn2n1 C=CC1(C(=O)NCc2cccnc2O)CCN(C(C2CC23CCC3)=O)C1 C1(C(CNC(c2n(C)cnc2)=O)(C)O)CCCN(C(=O)CSc2cn[nH]c2)C1 c1(NC(c2cn(CC(CC)C)nn2)C)cc2cc(F)c(OC)cc2[nH]1 c1(OC(C(N2CC(CCNC(CC(CC)C)=O)C2)=O)C)cc(Cl)cc(Cl)c1 c1(C(=O)NC(CNC(C2CC(SC)C2)=O)C(C)C)snc2ccccc12 c1(C(=O)Nc2ccc(Oc3ccc(F)cc3)cc2)cc(F)ncc1Br C(=O)(CCCCCF)NC1(C)CN(C(C(c2cccc(OC)c2)OC)=O)C1 Cc1nc(C(=O)NCC2CCC(C)N(C(c3cnc(C)c(C)c3)=O)C2)cc(O)n1 C(=O)(CC(C)(O)CCC)NCC1N(C(CC(=C)C)=O)CC1 c1(CCC=O)cnccn1.C(C)(C)C.C(C)(C)(C)OC1(N(C)C=O)CC1 C(CCC)(C(=O)NC(c1ccccc1)CNC(=O)C)=CCC.c1ccccn1.O c1(NC(Cn2cc(CC(C(=O)OCC)(C)C)nn2)=O)ccc(F)c(F)c1F C(=O)(C(CC(C)C)NC(=O)CC1CC1C)NC.c1(C=O)cc(=O)cc[nH]1 c1(C(=O)NC2CC(C)(NC(CC3C(C)CCO3)=O)C2)n[nH]c2c1CC(C)(C)CC2 C(=O)(C1=CN=C2N=CNN2C1)N.N1(C(C2N(C(C)=O)CCC2)=O)CC2CC(C1)C2 C(C)(N=c1[nH]c2c(c(=NC(CF)c3ccco3)[nH]1)CCC2)c1ccc(C)c(N)c1 C1(C(=O)NC2CCN(C(Cc3cc(C)[nH]n3)=O)C(C)C2)CC2CCCC(C1)C2=O C(C)(CO)(C(=O)NC(CCNC(=O)C=C(C)C)c1cccs1)OC CS(C)(=O)=NC(=O)C(=O)N1CC(NC(=O)CC(C(F)F)c2ccccc2)C(O)C1 CCCCCC(O)C(=O)N1CC(OC)C(NC(=O)C(c2ccccc2Cl)(F)F)C1 c1(C(=O)NC2C(NC(=O)CN3CCC(O)CC3)COC2)ncc(Br)cc1F c1(C(N(C2CN(C(C(CC=CCC)C)=O)C2)C)=O)cn2c(Br)cccc2n1 c1(C(=O)NC(CNC(c2cnc(C(C)C)[nH]2)=O)C)n[nH]c2ccc(O)cc12 C(=O)(N1OC2CCC1C2)C1CCN(C(C(N2CCNC2=O)C)=O)C1 Cc1cnc(C(N2CC(NC(=O)Cc3cn(C)nc3C)CC(C)C2)=O)cc1C C1(CNC(CN2C(C)CCC2)=O)CN(C(c2cnnc(C3CC3)c2)=O)CCCO1 c1(C=O)ccccc1.C(=O)(C(F)(F)F)N(C)CC.CCC.C1(C=O)CC1F.O N1(C(C2N(C(CCC#N)=O)C3CC(F)C2C3)=O)CCc2sccc2C1 c1(C(=O)NC(CC(C)NC(c2c(C)scn2)=O)C)ccc([N+](=O)[O-])cc1N CC1=C(C(=O)N2CCCCC(N(C(=O)C(F)C3CCCC3)C)C2)COCC1 Cc1cc(CCC(=O)N2CCC2CNC(=O)C(C)(C)C2CCOCC2)cc(C)c1 C(N=c1[nH]c(=NCCC2=CCOCC2)c2[nH]ccc2[nH]1)C1(CO)CC(C)C1 C1(C(N2CCC(CNC(C(C)=C(C)C)=O)C2)=O)CC(=O)CCO1 O=C1CCc2ccc(C(=O)NCC34CCC(CC3)N4C(=O)CCCF)cc2N1 C1(C(=O)NC(C2CN(C(c3ccc(F)c(Br)c3)=O)C2)C)C2C3CCC(C3)C12 c1(OC)ccc(OC)cc1.c1(N(C(C=CC=O)=O)CC#N)ccc(C)cc1.N c1(C(=O)NCC(CN(C(c2n[nH]cc2)=O)CC)(C)C)ccc(O)c(F)c1 C(C(=O)N1CCN(CC(=O)NCC(CC)N2CCCC2)CC1)(C(C)C)SCC c1(C=O)nc(O)c(C#N)cc1C.N1(C(c2n(CC)cnn2)=O)CC(C)C(O)C1.N c1(OCCC(N2CCN(C(=O)C(O)CC3CC3)CC2)=O)ccc(Cl)cc1Cl N1(C(CC2CC(=C)C2)=O)CCCC(C(C)NC(c2ccccc2SC(F)F)=O)C1 N1(CC(=O)N(CCC)CCC)CCN(C(=O)CC(CC)C2CCC2)CC12CCC2 CC(C)CCC(F)C(=O)NN1CCCC1C(N1CCC12CCCC2)=O N1(C(=O)N(C(C)(C)C)CCO)CCN(C(=O)CC2CCC3CC23)C(C)(C)C1 C1(NC(CNC(C)=O)=O)CN(C(c2cc(C)nnc2O)=O)CCC12CCOCC2 c1(OC)ccccc1S(=O)(=O)N1CCC(O)(C(=O)Nc2nc(C)c(C)nc2Cl)C1 N1(C(CCC=CC)=O)CC2(CCOCC2)CC1C.c1(C(=O)N)cnc(C(C)O)s1 c1(CCC(=O)NC(CNC(c2cn(C)nn2)=O)(C)CO)cccc(O)c1 CC(C)(Cc1ccccc1Br)C(=O)N1CC(CCNC(C2(CF)CC2)=O)C1 N1(CC)CC(C(=O)NCC2CCN(C(c3nonc3N)=O)C2)NC1=O C(=O)(CC(C)CCCCC)N1CCC(C=C)(C(=O)NCc2cccc(C)c2O)C1 CCCC(CCO)CN=C(NCC1C(F)(F)C12CCOCC2)NC1CCOCC1 N1(C(C(C#C)(C)C)=O)CC2(C1)CN(C(=O)CC1CC3(CCC3)CO1)C2 CC1(NC(=O)CC(c2ccc(Cl)cc2)O)CCCN(C(c2ccns2)=O)C1 C(=O)(CCC(=O)NC(C)(C)CN(C(=O)C(c1ccc(Br)cc1)C)C)OC c1(C(=O)NC2C(C(=O)Nc3ncc(C(=O)OC)s3)C2)c(I)ccnc1F C(=O)(CC(C)C(C)(C)NC(C1CCC2(CCC2)O1)=O)NC(c1scc(C)n1)C C1(CC)CN(C(C2CCCC2OC)=O)CCC1NC(=O)C(C)(C)CC1CCC1 c1(C(=O)NCCN(C(C2C3(CC(OCC)C3)C2)=O)C)cc[nH]c(=O)c1 Cc1nccc(C(=O)NCC2(C)CCCCC2)c1N.C1(CC(=O)N)CC1(C)C C1(C(=O)Nc2c(OC)cc(Br)cc2)CCC2(CN(c3ncc(F)c(C)n3)C2)O1 n1(CC(=O)N(C2C(NC(Cc3c(C)ncs3)=O)CCCC2)C)nc(C)n(C)c1=O C1(C(=O)NCC(C2CC2)NC(C(N)=O)=O)CCCC1CF CCC(C(=O)NCc1ncnn1CC)NC(C1CC1[N+](=O)[O-])=O C1(NC(Cc2ccc(OCC)cc2)=O)CCCN(Cc2cnc(Cl)s2)C1C C1(C(N2CCC(C(=O)NCCC(O)C(C)C)(CC)C2)=O)CCC(C)(O)CC1 Cc1ccc(NC(=O)CC2(C)CCN2C(=O)C(C)N2CC(C)C2)cc1C#N C(C)(C(=O)N1CC2COCC2O1)N(C(=O)Cc1nonc1C)CCC c1(-c2c(C(=O)NC(C)CNC(=O)C(O)C3CC3)c[nH]n2)ccc2c(c1)OCO2 C1(C(=O)NCC(C2N(C(CCC(C)=O)=O)CCC2)(C)C)CNC(=O)CC1(C)C N1(C(c2[nH]cc(CC)n2)=O)CC(C2CCN(C(C3CCN(C)C3=O)=O)CC2)C1 c1(C(=O)NCC2CN(C(c3n(C=C)ncc3)=O)C(C)C2)cnn2cc(C)cnc12 Cc1[nH]c(C#N)cc1C(=O)NCC(C)(C)CC(=O)NCCC1CCCC1O c1(C(N(CCCC)C)=O)ccc2c(c1)CCO2.C1(C(=O)N)CC(CC(F)(F)F)C1 c1(C(N2CC(O)(C(C)NC(c3cccn3C)=O)C2)=O)cc2c(F)cccc2s1 c1(C(=O)NC(C2(C(=O)NCC3(CSC)CC3)CC2)C)csnn1 c1(CN(C)CC2CN(C(c3ccc(CC(C)C)o3)=O)C2)ccc(C(C)C)cc1 C1(C(N2CCNC(C)C2)=O)CC=CCC1C(N1CCCC1c1nc(OC)no1)=O c1(C(N2CC(CC(=O)NCCC3CC4CCC3O4)(OC)C2)=O)cc(Cl)cn1C N1(C(Cc2scc(C)c2)=O)CCCC(C)(C)C1C(=O)N(CCC1=CCCCC1)C C(=O)(C(C(=O)N(CC(C)CNC(=O)C(n1cc(Cl)cn1)C)C)OC)OC C(=O)(CC1CCc2cc(Br)ccc21)N(CCNC(CC(C=C)C)=O)CC N1(C(=O)NCC(c2cc(C)cc(C)c2)C)CCc2c(Br)ccc(Cl)c2C1C C1(C(N2CC(C(=O)OC)(CC)C2)=O)CC(C)CN1C(c1cccc(O)n1)=O C1(C(N(C2CCN(C(=O)CCc3ccn(C)c3)C2)CC)=O)CC2CCC(C1)N2C C1(C(=O)NCCN(CCC)C(c2cc(F)cnc2Cl)=O)Cc2cccc(C)c2O1 C(=O)(C1=C2CCN=C2NC=C1)N1C(C)CN(C(c2cnc(Cl)s2)=O)C(C)C1 C(=O)(C(CC1CCOCC1)NC(=O)Cc1ccoc1)NC(C1CCC1)C C(c1ccnn1C)=CC=O.C1(CN(C)C)COCC1NC(=O)CC1CC1.N c1(C(=O)NC(C2OCCN(C(CN(C)CC)=O)C2)C)ccccc1F.C(C)=O.N N1(C(c2ccc(CC)nc2)=O)CC=C(CCNC(=O)C(O)C(C)CC)CC1 C(=O)(CCC(F)(F)C(F)F)N1CCC(NC(c2cc3nc[nH]c3cn2)=O)C1 C(CC(C)C(=O)NCC(C(N1CC2C(N(C)C)C2C1)=O)N(C)C)=CCC C1(C)(CNC(CC(c2ccc(C)cc2)C)=O)CCN(C(=O)Cn2cnnn2)CC1 C1(CC=C)(NC(c2coc(O)n2)=O)CCCN(C(C2(n3cncn3)CC2)=O)C1 CCCC(CNC(=O)C(C)(C)C(C)C)C(=O)N1CCC(CC)(CC)C1 c1(C(=O)NC2CC(CNC(CC(C(C)C)O)=O)C2)cnn2ccccc12 c1(C(N2CCCC(N3CCCS3(=O)=O)CC2)=O)ccnc2c1OCO2 C(=O)(C(C)(C)CCCNC(C1CC2CC(=O)C1C2)=O)NCC(CCC)(C)O c1(CC(COCC)C)nc(C2CCN(C(C)=O)CC2)nn1-c1ccn(C)n1 c1(C(=O)NC(CNC(c2cnn[nH]2)=O)C2CCC2)ccc(F)cn1 c1(CC(C)C(=O)NC2CC2NC(=O)C(=Cc2c[nH]cn2)F)ccc(C#N)cc1 c1(C(=O)NCC2CCCCN(C(C(C(C)C)N(C)C)=O)C2)cc2cc(Cl)sc2[nH]1 c1(CN2C(C(=O)Nc3cc(Cl)ccc3F)CC3CC32)cnc2c(Br)cc(Cl)cn12 N1(C(C(=O)NC(CC)(C)C)C2CC2(C)Br)CCCC2(C1)CC2(F)F c1(OCC)ccsc1C(=O)NCC1CC1CNC(c1csnn1)=O C1(NC(CN(CCC)C)=O)CCSC12CN(C(C1CCC(=O)CC1C)=O)C2 N1(Cc2cnc(SC)nc2Cl)CC2CCN(Cc3ccccc3OC(C)=O)C2C1 C(=O)(CCCS(N)(=O)=O)N1C2CC(CNC(C3(C#N)CC4CC4C3)=O)C1CC2 C(=O)(C1CCCc2nncn21)NC(COC)(C)C1CC1 N1(C(c2c(-c3ccc(C)cc3)ocn2)=O)CC(N)CCC1(C)C c1(OC)cccc(CCC(=O)NCCCOCCCNC(=O)C(O)C(F)F)c1 N1(C(C(ON=C(C)C)C)=O)CC2CC1CN(C(C1CCc3ccoc3C1)=O)C2 Cc1ccc2occ(CC(N3CC4CC(NC(=O)CC5CC5)C4C3)=O)c2c1 Cn1ccc2c(C(=O)NCCCNC(=O)CP(C)(C)=O)ccnc12 C12CCC(C1)CCC(=O)N2.C(CCC(=O)OC)NC(CC1CC(CC#C)C1)=O O=C1CC(C(=O)NC2(C(=O)O)CCOC2)N(C(=O)CC23CCCC2C3)C1 N1(Cc2ccc(OC)c(Br)c2)CCC2(CCCN2S(=O)(=O)c2cccs2)CC1 C1(NC(CC2(C)CCC2)=O)CN(C(c2cc(Br)no2)=O)C2(CCCOC2)C1 Cc1ccc(C(N2CCC(NC(=O)C(F)C(F)(F)F)C(F)C2)=O)c(C)c1 CC1(C)CC(C(N2CCC(NC(c3ccc(Cl)cc3O)=O)CC2)=O)CNC1=O C=C=CCC(=O)NCCSCC(=O)NC1(CCC=C)CCC1 Cc1c(C(N2CCC(O)(C(=O)NCCS(C)(=O)=O)C2)=O)cc(F)cc1Cl S(=O)(=O)(c1ccc(Br)cc1NC1CCCCCC1F)NCc1n(C)cnc1 c1(CCC(=O)NC(C2CN(C(C(C)=C(CC)C)=O)C2)C)ccn(C)c1 O=C1CC(C(N2CC3CC(NC(=O)CCc4ncc(F)cn4)C2C3)=O)CC(=O)N1 N1(CC(=O)NCCN(C(=O)Cc2ccnn2C)C)CCCOC1=O Cc1nc2cncc(C(=O)NCC(CO)NC(C3CC4CCC3C4)=O)c2[nH]1 C(CN=c1nc(N2CCCC(F)C2)c2c([nH]1)COC2)OCCC Cc1nc[nH]c1CC(=O)NC(C)CCCNC(C1OCC1(C)C)=O C1Cc2ccccc2C1.n1(CCCSCC)nnnc1C(C1(n2ccnn2)CC1)N c1(C(C)C)cnc(Cl)nc1N1CCCC(C)(CNC(C2(C(F)F)CCCC2)=O)C1 c1(C(c2nnnn2CC(F)F)Nc2ncn(CCC)c2)ccc(Br)cc1OC CC1CN(C(c2cnc(Cl)c(F)c2)=O)CCN1c1ncc(F)cn1 C12(NC(c3ccc(=O)oc3)=O)CCCC1N(C(=O)Cc1ccco1)CCC2 C12(C=O)CC(C1)C(C)(C)O2.c1(OC)ccc(CC)cc1.c1(C=O)ccco1.N C1(C(N2CC(CNC(C3CCCCO3)=O)C(F)(CO)C2)=O)CCC(C2CC2)CC1 N1(C(=O)OC(C)(C)C)CC2OCC(C(=O)NC(C3CCC3)C3CC3)OC2C1 Cc1cc(C(=O)NC2CC(NC(c3cccc(C(N)=O)c3)=O)C2)cn1C C(=O)(C1COc2ccccc21)NCCC(C)NC(c1ccsn1)=O CCCCC(O)C(=O)N1CCOCC1CCNC(C1C2COCC12)=O c1(-n2cc(C3N(C(CC4(C)CC4(Cl)Cl)=O)CC3)nn2)ccc(F)cc1 N1(C(c2ccc(C(=O)OC)cc2)C(=O)NCC(F)F)CCN(CCO)C(C)C1 C1(=O)N2OCCC2N1.c1(C(COC)(C)O)cn(CCC(=O)OC(C)(C)C)nn1 c1(C(=O)NCCOC)cccc(S(=O)(=O)NC2COCC2C)c1 C1(C(N(CCC#C)CC)=O)CCCCN(C(c2cc(C3CC3)ncn2)=O)C1 C12(CNC(CCC=C(C)C)=O)CCCC1CN(C(c1nccc(C)n1)=O)C2 Cc1c(F)ccc(OC(F)F)c1Cl.C(CCC(=O)OC(C)(C)C)(C(=O)O)O c1(SC)c(C(=O)NC2CCC(NC(C3COC(=O)C3)=O)CC2)cccc1F C(C(CNC(=O)Cc1ncccc1C)C(F)(F)F)NC(COC(C)=O)=O O=C(CCC1CCc2ccccc21)NC1CC(CNC(C2(Cl)CC2)=O)C1 N1(C(c2cc(C)oc2C)=O)CCC(NC(c2c[nH]c(C(F)(F)F)c2)=O)C12CC2 c1(C(=O)NCC2CC(NC(C3(C=C)CCC3)=O)C2)csc2c1CCC(C)C2 N1(C(C(C)C#N)=O)CCC2(CC1)CC(CNC(=O)CCc1cccc(Cl)c1)C2 Cc1cn2c(n1)C(C)N(C(=O)COC(c1cccc3ccnn13)=O)CC2 c1(C(N2C(CNC(c3ccc(Cl)cc3F)=O)CC2)=O)ccc2c(=O)cc[nH]c2c1 Cn1cc(Br)cc1C(=O)NC1CCN(C(c2cc(C(F)F)n(C)n2)=O)CC1 CC(C)(C)C(C#N)C(=O)NC12CC(C1)N(C(=O)C(CO)NC(N)=O)C2 C(CC)(C(=O)N1CC(CCO)C1)=CC.n1(CC(=O)N)cc(-c2ccccc2)cn1 CC1CCOCC1C(=O)NCc1ccc(CNC(=O)CCCc2ccsc2)cc1 C1(NC(Cc2cnc(C)s2)=O)(CF)CCN(C(C2(N3CCCC3)CCC2)=O)C1 S(=O)(=O)(c1cccc(NCc2ccc(C(F)(F)F)s2)c1)N1CC(C)OC(C)C1 C(=O)(C1=C(F)CNCC1)Nc1cncc(OC)c1C N1(C(CC(CNC(CCSCC)=O)O)=O)CN2CCC(O)C2C1 Cc1ocnc1CC(=O)N(C1CC(NC(C2CCC2c2nc[nH]n2)=O)C1)C C1(NC(C(CC)NC(N)=O)=O)CCCC12CN(C(c1cnc3cccnn13)=O)C2 c1(NC(c2nc(-c3cc(OC(C)(C)C)c(O)cc3)sc2)=O)cc(F)c(Cl)cc1F C=CC1(CC(N2CCC(NC(C3CCCN3C(N)=O)=O)C(O)C2)=O)CCOCC1 c1(C(C(=O)NC(C)C)N(C2COC(C)(C)C2)C)cnc(Br)n1C N1(C(=O)Nc2c(C)nn(-c3ccccc3)c2)CC(c2cc[nH]n2)C(C)(C)C1 C1(n2c(-c3cnc(C4CCOC4)s3)nc(-c3scc(C)n3)n2)CCOC(C)(C)C1 c1(CCC(=O)N(CCCN(C(C2C(C)OCCC2)=O)C)C)n[nH]c2c1CCCC2 c1(NCc2ccc(S(C)=O)cc2)ccc(S(=O)(=O)NC2(CO)CCC2)cc1Cl c1(C(N2CCC(C)(CCNC(c3nncs3)=O)C2)=O)cccc(N)c1F c1(C2N(Cc3c(O)ccc(Br)c3)CCCC2)c[nH]c2ccccc12 C(c1ccccc1)=CC=O.C1(C)(OC)CN(CC(=O)NC2(C)CC2)C1.N Cc1cc(C)n(CCC(=O)N(C2CCCN(C(C3CNC(=O)C3)=O)C2)CCF)n1 Cc1csc2ccc(CC(=O)NCC(C)CNC(C3C(C#N)C3(C)C)=O)cc12 C1(C(C)C)Oc2ccc(C(N3CCC(Cc4ccncc4)C3)=O)cc2NC1=O C1(CC)CN(C(C23CC(C2)C(C)(C)O3)=O)CCN1C(=O)Cc1ccccc1.O c1(C(=O)NCC23N(C(Cc4n(C)ncc4)=O)CCC2CC3)cc2cnccc2o1 C(CCC)(C(=O)NC(CCOCCO)C(=O)NC1CCN(CCC)C1)=CCC c1(N2CCCC(C(N(C)C)=O)C2)nc(=NCc2cccc(Cl)n2)[nH]c2c1SCC2 C1(C2CC2)(C(=O)NC(c2cc(C)on2)C)CN(C(=O)CC(C)F)C1 C1(O)(C(N2CC(C)C2)=O)CC2CCC1C2.c1(COC)nc(C)c(C(=O)N)s1 C1(NC(C(CNC(=O)CC2(C)CC2)OC)=O)CCCCNC1=O C(=O)(CN=c1cc[nH]cc1)NCC1(C(=O)OC)CC1(F)F C1(C(=O)NC(CCCC)CO)C2CCC(C2)C1NC(=O)Cc1cccnc1 C1(OC)CC(NC(c2ccccn2)=O)C12CCN(C(C1CC(=O)N(C)C1)=O)CC2 N1(C(C2C(C)C2)=O)CCC2(CC1)CC(NC(c1ccc(F)cc1F)=O)C2 N1(C(c2cc(C)oc2)=O)C2CCC1CC(NC(c1csc(-c3cnc[nH]3)n1)=O)C2 C1(CNC(=O)Cc2ccsc2)CN2CCCCC2CN1C(=O)COCCF C#Cc1ccc(C(=O)N(C(C)C(=O)N(CC(F)(F)COC)C)C2CC2)o1 C(=O)(C1CCCc2ccccc21)NC1CCC(NC(C(C(C)(C)O)F)=O)C1 C1(CNC(c2nc(CC)sc2)=O)CC(O)CN1C(=O)C=Cc1cccn1C C1(C(NNC(=O)OC(CC)C)=O)Cc2ccc(F)cc2C(=O)O1 N1(C(C#CC)=O)CCC(O)C(NC(=O)CCc2ccncc2)C1 CCC(O)C(C)C(=O)NC(C)CC1CN(C(C2COCCN2CC)=O)C1 c1(N2CCC(OC)(CO)C2)nc2c(c(=NCC3CC(C)(C)CCO3)[nH]1)CSC2 N1(C(c2cnc(C)o2)=O)CC(S(=O)(=O)N2CCN(C(=O)CC3CC3C)CC2)C1 C1(CNC(C(CCC)OC)=O)CN(C(C2CC3(CCC3)CO2)=O)CC(C)(C)O1 c1(C(=O)NCCC2CCCCN2C(C2CC2C(F)(F)F)=O)cccc(Cl)c1O Cc1cc(Br)c(CNC2CC3(C2)CC32CC2)cc1O c1(C(N2C(c3cc(C)cc(C)c3)CC2)=O)cc(=NCc2cc(C)cc(F)c2N)[nH]cn1 C(C)(C)(CC(F)C(=O)NCC1NC(=O)CC1(C)C)NC(C(CC(C)C)=O)=O c1(N(C)C)ncc(Br)nc1NC(C1CCCN(C(=O)NC2CCC(C)CC2)C1)=O CS(=O)(=O)CCC(=O)NCCC1(C)CC1.c1(C=O)cc(C2CCC2)no1.N c1(NC(C2CCC(CNCc3c(Cl)cccc3Br)CC2)=O)ccc2[nH]ccc2c1 CCCC(C(=O)NC(C1CCN(C(c2cc(C)c(C#N)cn2)=O)C1)C)S(N)(=O)=O c1(C(=O)NC2(C)CC(NC(c3sccc3F)=O)C2)cc(F)cc2ccoc12 C(=O)(N=c1[nH]nc(Cl)cc1Br)c1c(NC(c2c(CN(C)C)cccc2)=O)c[nH]n1 c1(C(=O)NCC2CN(C(c3cc(C)oc3)=O)C(C)CC2)ccn2c(C)ncc2c1 C1(CC=O)CC(=O)NC1=O.CC1(C)CN(CC(=O)NC(C2CCCC2)C)C1.N C(N=c1ccnc(Cl)[nH]1)C1(NC(c2cc(O)cc(O)n2)=O)CCOCC1 C1(CNC(=O)NCC(N2CCCS2(=O)=O)C)CCC2CC(C)CN2C1 CCC(C(=O)NCc1nc(C(N2CCCN(C)CC2)=O)co1)C(C)C C(C(=O)NC(C)C)(C(C)(C)C)SC.c1(C(N2CC(CO)C2)=O)ccccc1C C1(OC)CCC(C(N2CC(F)CC2)=O)CC1.c1(CC(=O)N(C)C)c(C)noc1C c1(C(C2CC(N(C)CC)C2)NC(CCO)c2cccs2)nnn[nH]1.C1CCCO1.C C(CCCC(N)=O)NC(C1(C(C)NC(C(C)OCC#C)=O)CC1)=O C1(C(N2CCC(NC(c3nc(C4CC4)oc3C)=O)C2)=O)CC(C)CC(=O)N1.C CC1(SC)CCOCC1.C1(C=O)CN(C=O)C(=O)O1.c1ccon1.C(C)(C)C C1(OC)CN(CCc2cccs2)CCC1Cc1ccccc1 c1(OC)cccc(CC(=O)NC2(CNC(=O)CC3CC34CC4)CCOC2)c1 C1(C(=O)NC(C)CCCO)CN(C(=O)CCCCNC(N)=O)CC1(C)C [SH](=O)(=O)c1ccc(Cl)s1.C1CCN(C(=O)C=CC2CC2)C12CC2.O=CCN N1(C(c2nn(C)c(O)c2)=O)CCc2ccc(C(N3CCOC(CO)C3)=O)cc2C1 CCC(C)C(O)CC(=O)N(C(C)(C)CC(=O)NCC(C)(C)CC1CC1)C c1(C(=O)NCc2cc(C)c(Br)c(Cl)n2)c(C)nc2ncnn2c1N C(=O)(N1CCC(C(=O)NCC2CCC2C)O1)c1c(OC)nccc1 C(=O)(CCCC(C)(C)C)NC(C(=O)NCc1onc(C)n1)CO C(=O)(NNC(=O)CCO)NC(c1ccc(C(C(C)C)C(=O)O)s1)=O CC1CCC=C1C(=O)N1CCOCC1CC(=O)NCCC1COC(C)(C)C1 C1(CCC(=O)N(C(C)CN(C(=O)CC2CSC2)C)C)CCN(C)CC1 C1(F)(C(=O)NCCCP(C)(C)=O)CCCN(C(=O)CCCCC#N)C1 C(c1scnc1C)=CC(=O)NCC(CNC(CC1ON=C(C)C1)=O)(C)O C(CC(C)(O)C(=O)NC1COCC1C(=O)NCC1(CCO)CCC1)N(C)C c1(C(=O)NC2CC3CN(C(CN4CC(C)(OC)C4)=O)C2C3)ccc2ncsc2c1 C1(C(=O)NC(C)CCF)CCCCC1CNC(c1c[nH]nc1Cl)=O C1(CNC(CCOCC)=O)CCC(NC(c2ccncc2N)=O)CC1 C1(NC(Cc2c(C)nc(C)s2)=O)CN(C(C2CCCC(=O)N2C)=O)CCC1(C)C c1(C(=O)NCC(COC)NC(=O)C(CCS)N(C)C)c(C)ccc(C)c1O N1(CCCCCNC(C2(C(=O)OCC)CCCO2)=O)CCN(C(=O)CCF)CC1 c1(C(N(C2CCN(C(C3SCC=C3C)=O)C2)CC#C)=O)cn(C)nc1C Cc1cccc(CN)c1C(=O)N(C1CCN(C(C)C)CC1)C Cc1c(C(=O)NCCC(C)NC(=O)C(CC(F)F)C2CCC2)cc(C2CC2)n1C C1(NC(C2CC(=O)NC2)=O)CCCCC1NC(=O)CC1CC12CC2 N1(C(CCc2n(CC)ccn2)=O)CCC2C1CCCN2C(c1nc(O)c(C)s1)=O CCC(C)(CNC(=O)C=CBr)NC(C1CC(C(F)(F)F)CO1)=O c1(C(N2CCCC(NC(C3CC(C4CC4)=NO3)=O)C2)=O)cc2c[nH]nc2s1 C(=O)(C#CC1CCCOC1)NC(C)CC1CN(C(C2CCC3(C2)N=N3)=O)C1 O=C(C1CCCn2cncc21)NCC12CCC1(C(F)(F)F)CNC2 C(=O)(C(C)C(C)C(C)(C)C)NCCN1CCN(C(C(C=C)(C)C)=O)CC1 Cc1c(C(=O)NC2CCN(C(=O)C(c3ccc(Cl)cc3)O)C2)cccc1[N+](=O)[O-] c1(C(C)NC(=O)NCc2nc(CS(C)(=O)=O)no2)cc(F)cc(F)c1 c1(N(C)C)nnc(-c2cc(-c3cccnc3)on2)n1CC1CCCCO1 n1(C(C)C)nnnc1C(C1CC1)NCCOc1cccnc1 C1(C(N2CCC(O)(C(C)NC(C(C3CCC(=O)N3)C)=O)C2)=O)CCCCC1(F)F N1(C(CSc2cccc(OC)c2)=O)CC(C)N(C(C23CC(CO2)C3)=O)CC1C N1(C(CCC)=O)CC(CNC(=O)C(C2CCCCC2)SC)C(c2cncn2C)C1 C1(C(=O)NC2C(C)N(C(c3ccncc3O)=O)CCC2)CC(C)(C)SC(C)(C)C1 CCCC(C(=O)NCC1(F)CCC1)N(C)C.c1(C=O)c[nH]nc1C1CCOC1.N CCCC(C(=O)OC)C(=O)NC1CN(C(c2coc3ccccc23)=O)C1 C12(CC(=O)NC3(CCF)CCC3)CCC1CN(C(=O)CC=Cc1ccccc1)C2 c1(OC)cc(C)cc(C(=O)NC2CCCC2NC(C2C=CCC2)=O)c1C N1(C(C(=O)NCCOC)c2ccns2)CC2(CCC2)CC1CO Cc1ccc(NC(C2CCN(C(c3ccnc(OC4CCC4)c3)=O)C2C)=O)cc1 Cc1c(C(=O)NC2CC3(C2)CN(C(C2CC(F)(F)C2(C)C)=O)C3)cccc1C#N N1(C(C(CC)SC)=O)CC(CN(C(=O)CCc2ccccc2F)C)C2(CC2)C1 C(=O)C(C)CSC(F)(F)F.C1(C(NCC)=O)CN(C(=O)N(C)C)C1.C n1(CC)cc(C(=O)NCC(C)(CC)NC(c2cc(CCOC)on2)=O)cn1 C(=O)(CS(=O)(=O)N(C)C)N(C1CCN(C(C2CC23CCC3)=O)CC1)CC C1(C(N2C(C(=O)OC)C=CC2)=O)CCCCCC1.N1(CC=O)CC(C)(C)C1.N C1(C(N2CCC(NC(CCCOCC)=O)C2C2CC2)=O)CCC(C2CC2)CC1 N#Cc1cc([N+](=O)[O-])ccc1C(=O)OCC(=O)CC1CCCOC1 N1(C(C2N(CC)CCC2)=O)CC(=O)NCC1C(=O)NC1CC(CC(=O)O)C1 c1(CN(C(N(CCSC)CC)=O)Cc2cn(C)cn2)ccccc1OC N1(C(c2ccc(-c3cnc[nH]3)cc2)=O)CC2CCCN(C(C3CC3(Cl)Cl)=O)C2C1 N1(C(c2ccc(CC)[nH]2)=O)CCCC(N(C)C(c2ccc[n+]([O-])c2)=O)C1 C(=O)(CCCCCc1cn(CCCCNC(=O)C(F)CC2CCOC2)nn1)OC c1(C(N2CC(CNC(c3ccc(OC)cn3)=O)C3C2C3)=O)ccc2ccsc2c1 N1(C(C=C(C)Cl)=O)CCC2(CC1)CC2CNC(c1ccon1)=O.N(C)C.C C(C(C)(O)CC(C)C)NC(C1(CCNC(C(CC)CN(C)C)=O)CCCC1)=O C(=O)(CCC(=O)NCC1CC1)N(CC)CC.C12(C=O)CCCC1C2.C C1(CC(=O)NC(C)CN(C(=O)CCn2cnnn2)C)CCC2CC12 CC1(C)CC(C(=O)N2CC=CC2C(=O)NC2(c3nc[nH]n3)CC2)=NO1 c1(C2(C(=O)NCC(C)N(C(C(C(C)C)C)=O)C)CC2)cc(Cl)cc(Br)c1 C(=O)(C(C)(CC)C(N)=O)N1CCC(NC(c2c(N)ccc(CC)c2)=O)C(C)C1 Cc1cc2cc(C(=O)NC(C)C(C)NC(=O)Cc3ccc(O)nc3)oc2cc1C c1(C(=O)NC2CN(C(c3c(CCC)n[nH]c3)=O)C2)csc2cnccc12 CC1(C)CCCCC1NC(C1C=CCN1C(c1cnc[nH]c1=N)=O)=O C1(C(=O)NCC2CSCCO2)CCCCN(C(C2(c3cc[nH]n3)CC2)=O)C1 Cc1ccc(NNC(=O)NC2CCCCC2N2CCOCC2)c(Cl)c1 C(C(=O)N(C(C)C(C)SC)C)(C(C)CC)N(C(C1N(CC)CC1)=O)C c1(C(=O)NCC(CNC(COC(CC)C)=O)F)cc2cn[nH]c2cn1 c1(N(CCCNC(C2CCNC2=O)=O)CC)nc(Cl)ncc1Br C1(C=O)C2CCC(CC2)C1C(F)(F)F.C1(CC(=O)N)CCC12CCC2.CC#CC CCC(C(=O)NCC1CN(C(c2ccc(Cl)c(F)c2)=O)CCO1)C(C)O Cc1oc(C2CC2)nc1C(N1CCCC1(C)C)=O.c1(C=O)cscc1C(F)F.N CCC(CCO)C(C)NC(c1ccc(C2COCCN2)n1C)=O C#CCC(CC(F)F)C(=O)NC1C(CNC(C2CCCC2O)=O)CCC12CCC2 C(C(=O)N=S1(=O)CC(O)(C(=O)O)C1)c1nc(NS(C)(=O)=O)sc1 C1(CC(=O)N(C(c2ccc(C(F)(F)F)cc2)CC)C)CC(c2ccccc2)=NO1 c1(COCC)ccccc1CNC(c1cccs1)=O.C1(C(=O)N)CC1 C(CC1=CCN(C(=O)CCC2CCC(C)O2)CC1)NC(c1ccc(C)cc1C)=O c1(CC)[nH]nc(C(N2CCC(C)(C(=O)Nc3cnn(C(C)(C)C)c3)C2)=O)c1C CC1(NC(=O)Cn2cc(C3CCOC3)nn2)CC(C(F)(F)F)C1 C(CC(C(C)(C)C)NC(C1CCCS1(=O)=O)=O)N(C)C(c1ccc[n+]([O-])c1)=O Cc1cnc(CCNC(=O)NCc2oc(=O)oc2C)c(C)c1 c1(C=O)ccc(=O)n(C)c1.C(CC(C(=O)NCCCCCC)NC(N)=O)SC.N c1(NC(C(c2oc(C)nc2C)N(CC(=O)NC)CCC)=O)ccc(F)cc1C CCC(C)CCC(=O)NCc1ccsc1C(N1CCC12CC(O)C2)=O C=CC1(CC(=O)NCC(CCCC)NC(=O)CCC(C)N(C)C)CCOCC1 CC1(C)CN(C(=O)C=Cc2cocn2)CC(CNC(c2cncnc2)=O)O1 C1(C)(CNC(CCCCCC)=O)COCCN(C(C2(F)CCOCC2)=O)C1 C1(S(C)(=O)=O)(C(N2CCCC(C)(NC(C3CCC(C)O3)=O)C2)=O)CCOCC1 N1(C(C(=O)NCCOC)=O)CCC(C2CCN(C(=O)CCC=CC(C)C)C2)C1 N1(C(C(C(C)C)N(C)C)=O)CC2(C1)CN(C(c1[nH]cnc1C#N)=O)CCO2 N1(C(Cn2nc(C)oc2=O)=O)C2CCCC1CN(C(=O)C(O)C1CC1)CC2 c1(CS(=O)(=O)NC(C(=O)OCC)CCC2CC2)cnc(C)c(OC)c1 N1(C(CS(C)(=O)=O)=O)CCCCC1C1CC1.c1(C=O)cncc(C(F)(F)F)c1.N c1(C(C)C)ccc(C(=O)NC2C=CCN(C(c3ncc(F)cc3N)=O)C2)c(F)c1 C(=O)(CCCNC(=O)Cn1cc(COCCCCO)nn1)OC c1(C(N(CCC(C)NC(=O)CCc2cccnc2)C)=O)cnn2ccncc12 CCCCN=C(NCC1CCc2ccccc2C1)N1CCC(CCOC)C1 C(=O)(C(O)C(F)(F)F)NCC(CNC(c1cc(C#N)n(C)n1)=O)OC Cc1ccc(CNC(C2CCN(C(C34CC(F)(C3)C4)=O)C23CC3)=O)c(C)c1 Cc1cc(CC(=O)NC2C3CN(C(=O)CCCSC(C)(C)C)CC23)nn1C C1(NC(c2cncc(Cl)c2)=O)CN(C(C2COC3CCCCC23)=O)CC12CCC2 n1(CC#C)cccc1C(=O)NC1(C(=O)NCCC(O)CC)CC(CO)C1 C1(C(=O)NC2CN(C(CSC)=O)CC2O)CCc2nnc(O)cc2C1 C1(CC)CCC(C)N(C(c2oc(CNC(=O)C#CC(C)C)nc2C)=O)C1 C1(O)(C(C)NC(=O)C=Cc2cnc[nH]2)CCN(C(c2cc[nH]c2)=O)CC1 C(CCCCCN=c1cccc(S(=O)(=O)NCCN(C)CC2CC2)[nH]1)NC(C)=O C=CCCCCCCC(=O)N1CC2CC1CN(C(c1cocc1Br)=O)C2 c1(C(N2C(CNC(C3(C)CC3)=O)CC2)=O)ccc(Br)cc1C#N C(=O)(C(F)(F)C(C)(C)O)N(C(C)CN(C(=O)CN(C)C)C)C c1(CC(=O)NC(CCN(C(c2c(COC)[nH]cc2)=O)C)C)ccnc(OC)c1 c1(CC)ccc(NC(C2C=CCCN2C(=O)C(O)CC)=O)cn1 N1(C(CCC=C=C)=O)CCC(CNC(=O)C(C)OCC)C(F)(F)CC1 c1(N(CC(C)NC(c2ccn(CC(C)C)n2)=O)C)nc2cc(Br)cnc2s1 C1(C)(NC(COC(CC)C)=O)CCCN(C(c2cn(CC(F)(F)F)cn2)=O)C1 CCCCC(C(=O)NC1(CNC(c2cc3ccsc3s2)=O)CCOCC1)C(C)C Cc1nc(CNC(=O)CSCCNC(=O)C(C)C2(O)CCC2)co1 N1(C(C2CC(CCC)C2)=O)CCC(C(C)(C)C(=O)NCCc2cncn2C)C1 C(C)(CC1CCC1)(C(=O)NCC(F)C)OC.c1ccc(F)cc1.C(=O)CC.N C1(CC(=O)NCCCN(C(C)C)C(c2cc(CF)on2)=O)Cc2ccccc2O1 CCC(CC(=O)N(CC(C)N(C(=O)CCc1cc(Cl)cs1)C)C)OC C1(C(=O)NCCC=CCCC)CCCN1NC(=O)Cn1ccnc1 Fc1cncc(-c2nc(-c3cc(C4CC4)[nH]n3)n(C3CSC3)n2)c1 c1(C(N(CCNC(=O)Cc2cc[nH]c2)CC2CC2)=O)ccc(Br)cc1 CC(C)(C)CCCCC(=O)N1CC(C)(NC(c2cc(C3CC3)[nH]n2)=O)C1 N1(C(c2c(C)cn(C)c2)=O)CC(CNC(c2cncs2)=O)C(C)(C)C1 CC(C)=C=CC(=O)NCC1(CNC(=O)CCCCN(C)C)CCC1 N1(C(C(C)NC(=O)NC)=O)CCC2CN(C(=O)C=Cc3cc(C)no3)C2C1 Cc1[nH]c(C)c(C(=O)OC2CCOC2)c1C.C1CCCC1.C1(NC(=O)N)CC1 C=C=C(C)CC(=O)NC(C)(CNC(=O)C(=O)NCC)CO.C(C)=O.N CCN=c1cc[nH]c(C#N)n1.c1(OC)nc(C(=O)NC2CCN(C(=O)C)C2)co1.O C1(CCC(=O)NC)CCN(C(=O)C(=O)NC)CC1.C1CC1C=O.C1CC1 N1(C(C(CC)(C)OC)=O)CC2CC(C)N(C(c3ccc(C)c(Br)c3)=O)C2C1 C(C(C)NC(c1cc(-c2ccc(F)cc2)n(C)n1)=O)(C(C)C)NC(CCCC)=O c1(C(N2C(CCNC(c3c(C#C)c[nH]n3)=O)COCC2)=O)nnn2c1CCC2 N1(C(c2c(CC)cno2)=O)CC23CCCC2(C1)CN(C(=O)CC(C)C(C)(C)C)C3 N1(C(c2c(C)nc(CC(C)C)o2)=O)CC(C)(C)CC1CNC(=O)C(Cl)=CCl C(=O)(C1CCc2c(Cl)cccc21)NC1C(C)(C)CCN(C(CCOCC)=O)C1 c1(CSC)ccc(C(=O)NC(C)C(C)NC(c2sccc2F)=O)o1 CN1CCc2nc(C(N3CCCC(NC(C4CC5C=CC4C5)=O)CC3)=O)sc2C1 N1(C(c2n(CCC)ncc2)=O)CC2CN(C(C3(CO)COC3)=O)CCC2(CO)C1 C12(CN=C(NCC3(O)CCC3)NCCN3CCOCC3)CCC(CC1)OC2 C1(O)(CCNC(CN2C(C)CC2)=O)CCN(C(=O)C(C)(C)N2CCOCC2)C1 C1(NC(Cc2c(C)nn(C)c2Cl)=O)CCN(C(=O)CC2CC3CC3C2)C12CCC2 N1(C(C(C=C)(C)O)=O)CCC2(C1)CN(C(c1c(CC)nc(C)n1C)=O)C2 CCS(=O)(=O)c1ccc(Cc2noc(-c3nc(C)c(C)nc3O)n2)cc1 C(=O)(C(O)CCC)NCC1(OCC)CC1.c1(C=O)cc(C(C)C)on1.N C1(C(N2C(C)CCC(NC(c3nc(OC)oc3)=O)C2)=O)CCC2(CC1)CC2(F)F c1(CC)ccc(C)c(NC(C2CN(C(=O)C=C=C(C)C)CC23CC3)=O)c1 C(C)(CC(=O)NCCCOCCC(=O)NC(C1CC(F)(F)C1)C)SC Cc1ccc(C(=O)NCCCC2CCCN2C(=O)COCP(C)(C)=O)c(F)c1F Cc1csc(C(C)(C)NC2(C3CCCN3C(=O)C(=O)NCC(F)F)CC2)n1 C1CN(C(=O)CC2(O)CCOC2)CCC1C(F)(F)F.Cc1ncn(C)c1C=O.N S(=O)(=O)(c1cccnc1)N1CCN(C(c2cc(C(C)C)ncc2)=O)C2C1C2 CC1(O)CCC(CC(N2CCN(C(=O)CNS(=O)(=O)C3CC3)CC2)=O)CC1.C N1(C(Cc2c(C)noc2Cl)=O)CC2CC(NC(C3(CC4CC4)CCC3)=O)C2C1 C(CN=[N+]=[N-])(C(=O)N(C1CCN(C(C)C)C1)C)NC(CCOC)=O c1(C(=O)NCC2CCN(C(c3cc(CCC)c(C)s3)=O)C2)ccc(N)c(F)c1 c1(N2CC3C(CNC(CN4CCC(C)(C)C4)=O)C3C2)ncc(Br)c(O)n1 C=CC(C(=O)NC(CNC(=O)CC1CCCC1)CCOC)c1ccccc1 c1(CC(N2CCC(CC=C)(NC(=O)CC(C)CC)CC2)=O)ncn2c1CCCC2 c1(C(=O)NCC2(c3c(C)cccc3)CC2)cc(Br)cc2cccnc12 N1(C(C(=O)Nc2ccc(Cc3nnc4n3CCC4)cc2)=O)CCCC12COC2 CCCC(CC)CCC(=O)NC1(CNC(C2CCN3CCCCC23)=O)CC1 CN1CCCC(C(=O)NC2CCCC2(C)CNC(c2ncoc2C2CCC2)=O)C1 c1(C(N(C2CCN(C(C3CC(=O)C3C)=O)C2)CC)=O)ccc(C(=O)OC)o1 C1(C(=O)NC(c2ccc(C)cc2)CO)COCCN(CC2CC3(CCC3)C2)C1 CC(CS(C)(=O)=O)C(=O)NC(C1CCN(C(c2ccc3oncc3c2)=O)CC1)C C1(C(C)C)CCC(C(N2CCC(NC(C3(F)CC3)=O)C2)=O)CC1 c1(C=O)ocnc1-c1ccccc1.C(C)(C(=O)N1CC(CC)C1)NC(=O)NC C(C1=NOC2CN(C(c3cc(F)ccc3N)=O)CC12)NC(C=C(C)Cl)=O C(=O)(CC(O)C1CCCC1)N(CC(C)N(C)C(c1coc(Br)c1)=O)C c1(CC(N2CC3(CNC(=O)OCC(F)F)CC2C3)=O)ccc2nsnc2c1 Cc1cc(C(N2CC3(NC(=O)CN4CCC(C)(C)C4)CCC2C3)=O)ccc1Cl c1(CNC(CN(C(=O)C(CC)NC(C)=O)CCC)=O)cc(C)co1 CCC(CCOC)C(=O)N1CCC(C)C(CNC(=O)CSCCC(F)(F)F)C1 C1(C)(NC(C(CN(C)C)NC(C2C(=C)C2)=O)=O)CC(O)(CO)C1 c1(CC)c(N2CCC(F)(CNC(C3CC(O)C3)=O)CC2)nc(C)nc1Cl N1(C(c2cccc(N=[N+]=[N-])c2)=O)CC2C3CCC(C2C1)N(c1cnc(F)cn1)C3 C1(CNC(c2c(C(C)C)n(C)nc2)=O)C(C)CCCN1C(C1CC12CCOC2)=O c1(C=O)c[nH]c2ccc(F)cc12.C1(CNC(COC(C)(C)C)=O)CCC1(C)C CON(CCC(=O)NC(c1cncc(F)c1)C)C(=O)C(C)OCC(C)C c1(NC(=O)CC2CCCN2C(c2ccoc2)=O)cc(Cl)ccc1F N1(C(CCNC(=O)NC)=O)CCC2(C)CCCCC12.C1(C(=O)N)CCOC(C)C1 CCCCC(CC(=O)NC1CCC2CCC12)NC(c1sccc1CO)=O CCC(F)(F)C(=O)N1CCC(C(F)C(=O)NCCc2cccnc2)C1 N1(C(C(C(C)OC)NC(=O)CC2C=CCC2)=O)CCCC2(CC(O)C2)C1 N1(C(C(C=CC)O)=O)CC2(CCC2)CC1CNC(c1cc(O)ncc1Br)=O C(CC(=O)NCC1(C2(O)CCC2)CC1)(C(C)(C)C)NC(C(C=C=C)C)=O N1(C(C(C)Cc2ccc(O)cc2)=O)Cc2cc(F)c(F)c(F)c2C1 c1(CN2CCC(NCC(CC)NC(C)=O)C2)ccn(C=O)c1.C(C)(C)C.O N1(Cc2c(C#N)cncc2)CC2CN(C(C3CCCO3)=O)CC2C1 c1(C(=O)NCCC2CN(C(C(CCC)NC(C)=O)=O)C2)csc2cnccc12 N1(C(c2cc(NC(=O)OC)c(F)cc2)=O)CCC(NC(=O)C=CSC)C12CCC2 C(=O)(C1=NOC(C)C1)NCC1CN(C(c2cc(CC)c(C)s2)=O)CC1O CCC(CC)CCCC(=O)NC1CC(C)(CNC(C2(C)CC(F)(F)C2)=O)C1 C1CN(C(c2ccc(C#N)c(C)c2)=O)CC(C)(C)C1.C(CC(O)C(=O)NC)SC C1(NC(CCc2cccc(OC)c2F)=O)CN(C(C2CC2(Cl)Cl)=O)CC12CCC2 C(=O)(CC(C)CC(C)C)N1CCC(N(CCC)C(C2CN3CCN2CC3)=O)CC1 CC(c1cnn(C)c1)=CC(=O)NCCC1CCCCN1C(C1CCC(=O)N1C)=O C1(C(N2C(C)C(NC(c3cnc(C(C)(C)C)[nH]3)=O)CC2)=O)CCc2cncn2C1 C#CCC(C)C(=O)NCC1CCCCN1C(c1cccc(Oc2nccs2)c1)=O S(=O)(=O)(c1ccc(NC(CC(N)=O)c2cccs2)cc1Br)N1CCC(CSC)C1 C12(C(N(CC(=O)Nc3cnn(C4CC4)c3)CC3CC3)=O)CCCC1CCC2 N1(C(CC=CC(C)(C)C)=O)CC2CN(C(c3cc4[nH]ccc4s3)=O)CCC12 N1(C(CC=C(C)C)=O)CC(N(C(=O)CCc2cc(Br)cs2)C)C(C)(C)C1 N1(C(C2=CCN(C(c3ccc4[nH]ccc4c3)=O)C2)=O)CCC12CCCOCC2 C(=O)(C(O)C1=CCCCC1)N(C(C(=O)NCC(CC=C)(C)C)C1CC1)C CCCCC(CN=c1cc(COC)nc[nH]1)NC(=O)CN1CCCCC1=O C1(C)(COC)CCCN1C(=O)CCCCC1CC1.C1(C(=O)N)(CCF)CCC1 c1(CCC(=O)OC)ccc(C(N2CC(CC(=O)N)C2)=O)cc1.c1cc(F)c[nH]1 N1(C(C2(C)COC2)=O)CCN(C(c2ccc(-c3ccc(F)cc3)s2)=O)C2CC12 N1(C(C(CC=C)C)=O)CCc2ccccc2C(N(C)C(C23CCN(CC2)C3)=O)C1 N#Cc1ccc(C(N2CC(CNC(=O)CC3CC3)C3(CC3)C2)=O)c(O)c1 N1(C(c2c(C)cccc2)=O)CCC2CCCC12C(=O)NOCCN(C)C c1(OC)cc(C(=O)NCCCNC(C2(F)CC=CCC2)=O)ccc1C(F)F c1(N2C(C)CC(CNC(CCCc3onc(CC)n3)=O)C2)nc(OC)cc(C)n1 C1(NC(c2cccc(C(=O)NC)c2)=O)CN(c2ncc(C)c(C)n2)CCC1C c1(CC(=O)NC(C)CCNC(=O)Cn2cccc2)cccc2ncccc12 c1(OC)ccc(CN(C(CCC)=O)C)cc1.C1(C)CCCN1C(=O)CCCSC.N C1(NC(C2(OC)CCCCC2)=O)CCC2(CC1)CN(C(C1CC(F)C1)=O)CCO2 N1(C(c2c(CC)n(CC)nc2)=O)C2CC1CN(C(c1ccncc1F)=O)C2 c1(CC(=O)NCC(C)(CO)NC(c2cccc(OC)c2)=O)csc2nccn12 c1(C(N2CCC(C(N(C)CCO)=O)C2)=O)cccnc1O Cc1ccc(C(=O)NCC(O)CN(C)C(c2c[nH]c(C(N)=O)c2)=O)c(C)c1 C#Cc1cc(C(=O)NC(C2CN(C(=O)CCSC)C2)C)cc(F)c1 C1(CNC(C(CC)(C)O)=O)CN(C(=O)CCSc2nccn2C)CCCO1 C1(CC)CCCC1(C)C(=O)NCCC(=O)NC1(CCF)CC(O)C1 C1(CNC(c2c(C)nncc2)=O)C2CCC(C2)N1C(=O)C#CC(C)(C)C C1(C(=O)NCCCn2cccn2)CC(F)CN(C(C2CCC(F)(F)C2)=O)C1 c1(CCC(=O)NC2CCC(NC(c3ccn(C4CC4)n3)=O)C2)ccc(Cl)cc1 N1(C(c2cc(C)oc2)=O)CCOC2CCN(C(c3ccn(C4CC4)n3)=O)CC12 c1(C(N2CCC(OCCNC(c3c(C)nsc3N)=O)C2)=O)cccc(F)c1.C c1(C(N2CC(CNC(C3=NNC(=O)C3)=O)OCC2)=O)cnc2n1CCOC2 N1(C(CCC(=C)C)=O)CC2CCC2(NC(c2ccc(-c3ccccn3)s2)=O)C1 c1(C(=O)NC(C)C(C)NC(C2(F)CC2C)=O)ccsc1C#N CCC(CCCC(F)(F)F)Nc1ncnc(N2CCC(CC(=O)NC)CC2)c1C N1(C(CC2CC(N(C)C)C2)=O)CC(C)(C)OCC1C.c1(C(=O)N)cncc(F)c1 C1(NC(CCCN(C(C)C)C)=O)CCN(C(C2(C(F)F)CCC2)=O)CC1C c1(C(N2CCC(NC(C(C=C=C)C)=O)C2C)=O)cc(OC)cc(F)c1 N1(C(CNC(CC)=O)=O)CCN(C(c2ccc(C#N)cc2)=O)C(C)C1C C(=O)(C1CCCc2ncccc21)NC(C(C)NC(c1cc(OC)nn1C)=O)CO Cc1ccc(C(=O)NC2(CO)CCN(C(=O)C(C)P(C)(C)=O)CC2)nc1C c1(C=O)oc2ccccc2c1Cl.c1(C(=O)NCCC2CC2)csc(C(F)F)c1.N CC(C)C(CNC(=O)C1=NOC(C)C1)C(=O)NCCCC(N)=O Cc1ncc(C(=O)NCCCCCCN(C)C(C2(O)CC2)=O)c(=N)[nH]1 C1(C)(NC(CC2(N(C(CC(C)O)=O)C)CC2)=O)CCC2(CC1)CC2 C(=O)(C(C)CS(C)(=O)=O)NCC#CCNC(C1C(C=C)CC1)=O O=C(C1=CCOCC1)NC1CN(C(C2C(F)(F)C23CCC3)=O)CCC1O CC1CN(C(C2(F)CCCN(C)C2)=O)CCN1CCO C1(C)(C(=O)NCC=CCSC)CCCN1C(C1CC1(F)Cl)=O CCCCC(C(=O)N1CC(C(C)(C)C#N)C1)NC(C1CC(=O)OC1(C)C)=O c1(C(C)OCC)nc(C)c(C(=O)NCC(C)CO)s1.C(=O)(C#CC1CC1)N O=C(NN1CCN(c2ccc(Cl)cc2)CC1)c1c[nH]nc1[N+](=O)[O-] C1(NC(c2ccc(CCC=C)cc2)=O)CCSC12CN(C(=O)CC(C)(O)C=C)C2 O=C1OC(c2cnn(-c3cc(C4CCC4)[nH]n3)n2)c2cc(Br)ccc21 C(=O)CCC(C)(F)F.C12(CNC(C3(CC(C)C)CC3)=O)CC(CO1)C2.N c1(CCC)nc(C(N2CC(O)(CCNC(=O)CC)C2)=O)cs1.c1ccccn1.S c1(OC)ccc(C(=O)NC(C)CCN(C(=O)C)C)o1.c1(CC)ccccc1.O C(=O)(C(CC1(C)CC1)N(C(C)(C)C)CCOC)NC(CC)C CCCC(C)CCNC(c1cc(CNC(c2cc(O)cs2)=O)[nH]n1)=O N1(C(c2c(CC)onc2C)=O)CC2(C)CN(C(=O)C(CC)C(=O)OC)CC2(C)C1 S(=O)(=O)(c1cccc(Br)c1)N1CCOCC(NC(CC=C)=O)C1 CC(C)(O)CC(=O)NCC#CCNC(=O)C(CC1(C)CC1)c1ccccc1 Cc1cc(C(=O)NC2C=CC(CNC(c3ncoc3C)=O)C2)cc(O)c1 C1(NC(CCC=CC)=O)CN(C(c2ccnn2CCF)=O)C2(CCCC2)C1 N1(C(c2cc(CCOC)on2)=O)CC(NC(=O)C)CC1C.c1(C=O)ccoc1 c1(NC(c2cc(C)no2)c2nnnn2CCSC)cnn(C(F)F)c1C c1(CC=O)ccc(Cl)cc1Cl.C=C1CC(C(F)(F)F)(C(=O)NCCC(C)C)C1 C1(O)(CNC(c2cccc(CO)c2)=O)CCCN(C(C2CCCCC2(F)F)=O)C1 Cc1cc(C(N2CCC(C(=O)NC3CCCCC3)C2)=O)cnn1 c1(C(=O)OCc2ccccc2)ccc(NCc2c[nH]nc2C2CC2)cn1 c1(CC)cccc(CC)c1C(=O)NC(C)CC(C)NC(C1C(C)C1C)=O c1(OC)c(C(=O)NC2CCCN(C(=O)CC3(CO)CC3)C2)cccc1Br C(=O)(C1(C)CCc2ccccc21)NCC1(C)CCCN(C(c2c(C)c[nH]c2)=O)C1 c1(C(=O)NC2C(CC(=O)Nc3c(CC)csc3)CCC2)cc(C)n(C)c1 c1(C2CCCC2)cccc(NC(C(C(C)OC(COCC)=O)C)=O)c1 c1(C(=O)NCC(C(C)C)NC(C2=CC(C)(CC)C2)=O)ccc2occc2n1 C1(C(=O)NC(C)CCNC(C2CC23CCC3)=O)CCCC2C1C2(F)F C(=O)(C#CC1CCCC1)NC(CNC(C(C)OCC=C)=O)(C)C(C)C c1(C(=O)NC2(C)CC(NC(COCC(=O)OC)=O)C2)ncncc1Cl CC1(C2CCCN(C(C3CCN(C(=O)CC4COC(=O)C4)CC3O)=O)C2)CC1 CCCCCC(O)C(=O)NCC1CN(C(c2cnoc2-c2ccco2)=O)CC1C C1(CC)COC(C)C1.C(CCC=CC)=CC(=O)N.C(=O)C.C(=O)CO C1CC(C)CC(C)C1.CCC(C(=O)N1CCCC1Cn1cc(CNC)nn1)SC C1(=O)CCCCCCNC(=O)CC(C)C(=O)C(C#C)CCN1.OC C(CCN=c1nc(C(=O)O)cc(COCC)[nH]1)=CC=C C1(NC(c2cncc(Cl)c2)=O)COCCC1NC(c1coc(Cl)n1)=O Cc1c(CN=C(NCC(F)F)NC2CCOC3(CCC3)C2)cccc1[N+](=O)[O-] Cc1ccc(C)c(C(=O)NCC2CN(C(=O)C=C3CCN(C)CC3)CC2O)c1 C1(C(=O)NC(C(=O)OCC)C)CNC(=O)CN1C(=O)CC(=O)N(C)C O=C(C1=C(Cl)CCCC1)N1CCC(OC2CN(C(C34CC(F)C3C4)=O)C2)CC1 Cc1ccc(S(=O)(=O)N2CCCCC2C(=O)NCC(=O)NCC(F)(F)F)s1 Cc1cc(=O)oc(C)c1C(=O)NC1CCCC1NC(c1ccccc1O)=O C=CC1(c2cn(C3CCC(C)(C)CC3)nn2)COCCN1C(=O)C(C)OC CC(C)(C)CCCC(=O)NC(C1CCOC1)CNC(=O)CSS(C)(=O)=O c1(C(N2CCN(C(=O)C=CC3CCC3)C(CO)C2)=O)cccc(O)c1Br C1(C)(C(=O)NCC2(F)CCN(C(C(C)CO)=O)CC2)CC(C2CC2)=NO1 Cc1ccc(NC(=O)CC(C)CNC(=O)C(C)(C)CC(F)F)cc1C#N C=C(CNC(=O)C(F)(CNC(=O)C1=CCC(C)CC1)C(C)C)c1ccccc1 C1(C)(C(=O)NCc2[nH]nc(COC)n2)CCCN1C(c1cscc1C)=O C1(NC(c2cc(Cl)nc(Cl)c2F)=O)CCC2(C1)CN(C(c1nccnc1Br)=O)C2 Cc1cc(NC(C2CCCN2C(=O)CC2CCC(=O)NC2)=O)c(=O)n(C)c1 C(N=c1[nH]c(C)cc(=NC2CSCc3ccccc32)[nH]1)c1nccc(C)c1 CN1CC(NC(C2(C3CCCN3C(c3cc(F)n(C)n3)=O)CC2)=O)CC12CCC2 n1(CC)ncc(NC(=O)NCC2CCC2O)c1C(=O)OC c1(C(N2CC(N(C(C3NCC3)=O)C)C(C)(C)C2)=O)oc(S(N)(=O)=O)cc1C.C c1(C(N(C(CNC(C=COCC)=O)C2CC2)C)=O)cccc(C2CC2)c1 N1(C(C2(CC=C)CCOC2)=O)CC(N(C)C(c2ccnc(C)c2O)=O)C(C)(C)C1 N1(C(C2(SCC)CC2)=O)CC2CN(C(C34CC3COC4(C)C)=O)CC2C1 C=C=CC(C)C(=O)N1CCN(C(c2ccncc2N2CCCC2)=O)CC1 N1(C(c2[nH]ccc2)=O)CCC2(C1)CN(C(C13CC(C(C)C)(CO1)C3)=O)C2.CC C(C(CC)(CC)C(=O)NCCC(CO)C(C)C)NC(C(CCCC)=O)=O c1(C(N2CCCC2C)C=O)ccc2c(c1)CCC2.C(=O)(CCC(C)(F)F)NC.N CC(CC(N)=O)C(=O)NCC(C1CC1)NC(=O)CCF CC1CCN(C(=O)CCc2ccc(Cl)cc2)CCN1C(C1CCOC1)=O c1(C(=O)NCCCCC(C)NC(c2cc(C)nc(C)n2)=O)c(O)nnc(C)c1C CCC(O)C(C)C(=O)NCC1CCN(C(C2CC3(C2)CC(O)C3)=O)CC1 C12(C(=O)NCCCN(C(c3ccsc3Cl)=O)CCO)COCC(C1)OC2 CC(CC(=O)N1CCOC(C2CN(C(=O)C(C)Cn3cccn3)C2)C1)C(F)F N1(C(C2(C(C)C)CCCO2)=O)CCc2cccc3c2C(CCC3)C1 C1(CN(C(CC2(OCC)CC2)=O)C)CCCN(C(=O)C2=CCCC2)C1 c1(C(N(C(CNC(c2c(C#C)c[nH]n2)=O)C)C)=O)cc2cc(OC)ccc2cn1 C1(C(N(CCCCNC(c2c(C)con2)=O)C)=O)CC2CCCC2C1 Cc1cc(CNC(c2csc(CNC(c3csc(O)n3)=O)c2)=O)n[nH]1 c1(C(=O)NC(C)C(C)NC(c2nc(Cl)c(=O)[nH]c2N)=O)cccc([N+](=O)[O-])c1Cl c1(C(=O)NC(CNC(C2C(CC)OCC2)=O)(C)C)cc2c(cc1N)CCCC2 Cc1cc(C(N2C3C=CCC2CC3)=O)nc2nc(O)nc(O)c12 C(=O)(C(O)C1CCCC1)NCC(=O)NCC(=O)NC1CC(CO)C1 S(=O)(=O)(c1cc(C(=O)NC(C)C(C)C)c(C)o1)NC.C(=O)(CC(C)F)N c1(C(=O)NCCCC(C)NC(C=CC(CC)C)=O)cc2c(OC)cccc2s1 N1(C(c2ncc(C(C)(C)C)s2)C=O)CCCC(C(F)(F)C(F)(F)F)C1.C=CC C(C(C)(C)C(=O)NC(C)CCSC)NC(C1N(CC)CCC1)=O c1(C=O)cc(C(C)=O)c[nH]1.C1(C=O)CC(F)CN1S(=O)(=O)CC1CC1 c1(C(=O)NCC(C2CCN(C(CCCC#C)=O)CC2)(C)O)cc(OC)nc(C)c1 C1(C(=O)NCC(CCNC(CC2(C=C)CCC2)=O)O)CCN(C)S1(=O)=O c1(C(N2CCN(C(CCC(=O)c3ccc(C)s3)=O)CC2)=O)c([N+](=O)[O-])cnn1C C(C(=O)N(C)CCNC(c1cnc(O)o1)=O)(C(C)(C)C)OC c1(C(N(C2CCCC(N(C(=O)C3=CCOC3)C)C2)C)=O)ccncc1Br c1(C(C)=O)ccc(C(=O)NCC2CC2(F)F)o1.C(C(C)(C)C)=CC=O CC(C(=O)N(CCCOCCN(C)C(c1cccnc1S)=O)C)C(F)(F)F N1(C(c2cnn(CC)c2Br)=O)CCCCC(NC(C2CCC(=O)O2)=O)C1 Cc1cnc[nH]c1=NCc1cc(O)nc(CNC(c2cnncc2O)=O)n1 N(C(=NCCCC(C)(F)F)NCc1cccc2c1OC(F)(F)O2)C(C=C)C C1(CNC(=O)CC2CCOC2)CC(F)CN1C(=O)CNc1cnccn1 CCC(C)C(CC(=O)N(CCN=[N+]=[N-])C)NC(c1cncnc1)=O C1(OCC)CC2(C1)CC2C(N1CC(N(C)C(c2cnco2)=O)C1)=O Cc1ccc(C(C)C(=O)NCCC(C)(C)NC(=O)C(C2CC(F)(F)C2)O)s1 N1(C(c2c(C)c(O)ccc2)=O)CCC2(C1)CN(C(C13CC(CO)(C1)C3)=O)CCO2 c1(C(=O)NC(CNC(C2(CC=C)CC2)=O)C)cnc(OC)c(Cl)c1 C1(C(N2CCC(C)(CN(C)C)C2)=O)COC2(C1)CN(C(=O)Cc1cnns1)C2 C1(C(=O)NC2C(CNC(c3c[nH]c(Br)c3)=O)C2)C2CC3C(C2)C13 c1(C(N(CCCCNC(c2cc(OC)no2)=O)C)=O)ccc(-c2csnn2)cc1 c1(C(=O)NCC(CCCC)NC(c2sccc2C)=O)cc(Cl)c(OC)cc1OC C1(C(=O)NC2CCC(NC(C(C)C#N)=O)CC2)CCC2(CCCCC2)CC1 C1(CNCCC2S(=O)(=O)CCC2)C2CCCCCC12 N1(C(COCC)=O)C2CCC1CC(CNC(=O)CC1Cn3ccnc3NC1=O)C2 N1(C(CCC2CCN(C)CC2)=O)CCC2CN(C(=O)C3=CCSC3)CC2C1 N1(C(c2cccc(C)c2I)=O)CC2(CCC(C(=O)Nc3cc(Cl)cnc3O)O2)C1 C1(NC(Cc2nc(C)nn2C)=O)CCCN(C(=O)C=CC(C)C)CC1F c1(-c2cccc(C)n2)cccc2nc(C(=O)CC(N3CC4CC4C3C#N)=O)cn12 Cc1ccc(CNC(=O)C(C2CCCCCC2)(C)C)cc1[N+](=O)[O-] O=C(C(CNC(C1(CO)CCC1)=O)CC1CC1)NCC(O)CCC1CC1 CN=c1cc(C)[nH]c(-c2ccc(CNC(CC3CCCO3)C(=O)OC)cc2)n1 N1(C(C2C(CC)C2)=O)CC(NC(c2cncc(CO)c2)=O)CC(C)C1 c1(C(N2CCC(OCCNC(C(C)C)=O)CC2)=O)ncc(C(F)(F)F)cc1N Cn1ncc(Cl)c1C(N1CCCCC1CCNC(C1(CC(F)F)CC1)=O)=O Cc1ccc(NC(=O)CC(C)N(C)C(C2C3CC4C(C3)C24)=O)c(C)n1 C(C(C(=O)NC1CC(NC(=O)C(C)(F)c2ccccc2)C1)N(C)C)OC C=C(CCNC(c1cncn1C(F)(F)F)=O)C(=O)OCC C=CCC(CC=C)C(=O)NC1CCCN(C(=O)C=Cc2cc[nH]n2)CC1 C(CN=C(NCCOc1c(C)cccc1C)NCc1cc(C)cs1)OC C1(OCC=C)CCN(C(=O)C(CCF)NC(C2CC(C)=NO2)=O)CC1 C1(C(C(=O)NCC=CCNC(C2(C#N)CCC2)=O)O)CCCCCCC1 S(=O)(=O)(c1cnc(NCCN2CC=CCC2)c(Cl)c1)NC1(CO)CCC(C)C1 C(=O)(CC(C)C(F)(F)F)N1CCC(CN(C(c2c(C(C)C)con2)=O)C)CC1 C#Cc1ccccc1CNC(=O)C(C1CC=CCC1)NC(=O)C(C)(C)O C1CCN(C(c2cc(C)c(C)o2)=O)CC1C1CC1.C1(CCOC)(C(=O)N)CC1 C1(NC(C(C(C)C)O)=O)CC(F)CN(C(=O)CCCSc2ccccc2)C1 N1(C(c2ccoc2Cl)=O)CCN(C(C2(Nc3ccccc3)CC2)=O)CC1C1CC1 n1(CCC)nccc1C(=O)NC1C=CC(C(=O)N(CC(C2CCC2)O)C)C1 CCC(C(=O)N(C)CC1CCCC1)N(C)C.C1CC(C)(C)C1.c1(C=O)cnn[nH]1 C(=O)(C1COc2ccc(F)cc21)N1CCN(C(=O)CNC(N)=O)CC(C)(C)C1 N1(C(C(C(C(C)C)O)C)=O)CCN2CCN(C(=O)C(O)C3=CCCCC3)CC2C1 C1(C(=O)NCC)CCCN1C(=O)C(n1cc(C2(C)COC2)nn1)C c1(-n2c(-c3cc(C)ncc3)nc(CCC3CC3)n2)cc(Cl)ccc1Oc1ccccc1 c1(C(=O)NCC2CCN(C(Cc3c(C)ncs3)=O)C2(C)C)cnc2[nH]ccc2n1 c1(C(C)C)ccc2cc(C(=O)NC)[nH]c2c1.C1CCN(C(C2CC(C)(O)C2)=O)C1 CCN=c1ccc(C(=O)NC2CN(C(C)C)CC2C)c[nH]1 c1(C(=O)NCC2(C)CCN(C(C3CCCNC3=O)=O)C2)cc(F)cc(Cl)c1 c1(C(=O)NC2CN(C(c3c(Br)cn(C(C)C)n3)=O)C2)cc2ccccc2nn1 c1(OCC)ccc(NC(=O)CN(C(c2coc(C#N)c2)=O)C2CC2)cn1 C1(c2cn(C)nc2)CC(COC(=O)C(F)F)CCO1 N1(C(c2ccc(-n3cc(COCC(C)O)nn3)cc2)=O)C2CCC1CC(=O)NC2 C(=O)(C1=CCCCC1C)N(C(CCNC(Cn1nc(C)c(Cl)c1C)=O)C)C CCC(C(C)(C)C)NC(=O)C(N1CCC(CF)C1)=O Cc1cc(C(=O)NC(C)C(C)(C)NC(C2CCC3CC23)=O)nnc1O c1(OC)ccc2c(C(=O)N(CCCNC(c3cc(N)c(F)cn3)=O)C)csc2c1 c1(C(=O)NC2CCN(C(c3ccncc3F)=O)CC2CO)ccc2snnc2c1 Cc1ocnc1CNC(=O)C(C1CCCCC1)O N1(C(c2c(OC)n[nH]c2)=O)CC2=C(C1)CN(C(c1cc(O)n(C)n1)=O)C2 N12CCCC(C1)CNC2=O.c1(C(=O)OC)scnc1C(F)F c1(C(=O)NCCC2CCCN(C(C(CC)C)=O)C2)ncc(C(F)(F)F)cc1F Cc1cccc(S(C)=O)c1NC(=O)NC1CCCC(CC(N)=O)C1 N1(C(C2CCCC2)=O)CC2OCC(NC(C3(c4ccccc4)CCOC3)=O)C2C1 C(=O)(C1=CCCN(C(c2ccccc2Cl)=O)C1)NCc1ccc(OC)c(I)c1 c1(C(N2C(C(=O)NCCOCCN=[N+]=[N-])C=CC2)=O)cc(N)cc(F)c1 C(=O)(CC(C(C)O)NC(C1CC2CC2C1)=O)NC(C(=O)OC)C1CCC1 Cn1c(NC(NC2CCn3nncc32)=O)cc2ccccc12 C1(C(N2C(C)CCC2C)C)CCCN(C(=O)C=CC(N)=O)CC1 Cc1ccc2c(C(N3CCOCC(NC(C4CCCC4)=O)C3)=O)cnn2c1C N#CC1CCC(OC(C23CC(CO2)C3)=O)CC1 N1(C(C(Cc2cn[nH]c2)NC(C=CCOC)=O)=O)CC2CC1C2C(=O)O C1(C2CC2)(NC(C2CCN2C(=O)CC2COCCO2)=O)CCOCC1 c1(C=O)cc(C)c(Cl)c(N)c1.C1(CNC(COCCC)=O)CC(F)C1.C CCCCCC(C)(CC)C(=O)NC1C2CC1CN(C(=O)C(C)(C)OC(C)=O)C2 N1(CC(=O)NCCOCCC(C)C)CCc2c(C#N)cccc21 c1(C(C)(C)NC(C)C)cn(C2CN(C(c3cc(-c4cnn(C)c4)on3)=O)C2)nn1 N1(C(c2ncn(C(C)C)n2)=O)CC(NC(C2CC2(C)C)=O)C(C2CC2)C1 C(c1cc(F)cc(F)c1)=CC(=O)N.C1CCCCC1.C1(C=O)CC(=C2CC2)C1 C(CC(C)C)(C(=O)NC1COCC1CN(C)C)NC(CCC(C)OC)=O c1(C2(C(N3CC(N(C(=O)CC4CC(=O)C4)C)C3)=O)CC2)cc(F)ccc1F C(CCCCNC(c1ccc(CC2CC2)s1)=O)NC(=O)Cc1ccsc1Cl c1(C(=O)Nc2cccc(NC(c3c(CC)ocn3)=O)c2)cc2nccnc2[nH]1 CN1CC(C(=O)N(CCN(C(=O)C)CN)C2CC2)NC1=O.c1ccccc1F C1(O)(C(C)NC(Cc2c(C)con2)=O)CCN(c2cncc(C#N)n2)CC1 C(C1=CCCN(C(C2CC2(F)F)=O)C1)NC(C(C(C)C)C)=O c1(C(N(CC)C(C)C)=O)ccn2ncc(C)c2n1.CC1=NOC(C)(C(=O)N)C1 C1(C2CCC2)(CNC(C(c2ccnn2C)NC(CCSCC)=O)=O)CC1 C1(NCC(=O)N(C)CC2N(C(COC)=O)CCC2)CCc2n[nH]cc2C1C C=CCC(C)(CC)C(=O)N1CC(C(=O)NC(c2c(C)noc2C)C)C(C)C1 C1(NC(CCC(=O)N(C)C)=O)CC=C(C(=O)N(C)CC2CCCS2)C1 c1(C(=O)NC2(CO)CCN(C(CC=C)=O)C2)cnn2c1NCCC2 C1(CNC(c2occ(C)c2)=O)CCC(CN(C)C(C2(CO)COC2)=O)CC1 CC(CC(F)(F)F)C(=O)NCC1(C)CCN(C(=O)C=C2CCN(C)C2)C1 n1(CCCC)nc(Cc2ccccc2Br)nc1-c1n[nH]c(O)n1 C(=O)(CC(C(F)F)NC(=O)C(C)OC)N(CC)Cc1ccoc1 CC1CC(NC(C2CSCN2C)=O)CCN1C(c1ccc(F)o1)=O N1(C(C)=O)CCc2ccccc2C1CC(=O)NCC1C=CC(NC(=O)CO)C1 CN1CCCC(C(N2CCCC2(C)CNC(C2(C)CC3CC3C2)=O)=O)C1 N1(CC)CCOCC1CC(=O)NC1(CNC(=O)CCCC2CC2)CCCC1 c1(OC)ccc(CNC(C2(C)CN(C(=O)Cc3cccc(F)c3)C2)=O)cn1 C1(C=O)CCCCN1CC(F)F.C(C)(C)(C(=O)NC(C)CCC)OC(C)=O.N C(C)(C)C(C)C.C1(C=O)CCCN(S(C)(=O)=O)C1.c1(CC)occc1C=O CCCCCN(C(=O)C=C1CCSCC1)C.C1(COC)(CO)CC1C=O C1(N(C(=O)Cc2csnn2)C)CCC(NC(c2cc[nH]c2C2CC2)=O)CC1 N1(C(Cc2c(C)non2)=O)CC(CNC(=O)COCCC(C)C)C(C)(C)C1 C1(C(N2CC(CCC)N(C(c3onc(C)c3C)=O)CC2)=O)CCc2cnnn2C1 c1(C(=O)NCCC(C)(C)NC(CS(CC)(=O)=O)=O)cccc2nn(C)cc12 Cc1cc(F)c(C(N2CC(CN(C(=O)CCCC(C)(C)C)C)C2)=O)cc1F N1(C(CCCSC)=O)CCC2(CCN(C)CC2)C(CNC(=O)OC(C)(C)C)C1 c1(NC(C2(F)CCCN(C(c3n[nH]c(C)c3C)=O)C2)=O)cnc2[nH]cnc2c1 CCCCC(CC)CCCN(C(c1nccc(Cl)c1Cl)C(=O)NC(C)(C)CC)C CC1CC(C(=O)NCCC(C)(C)C)CC(=O)N1.C1(C(=O)N)C(C)(C)C1(C)C Cc1nc(C(=O)N(C2CC(NC(c3c[nH]nc3C(C)C)=O)C2)C)c2ccccn12 C(=O)(C(F)C(F)(F)F)NCCC(C)N(C(=O)CCc1nncn1C)C c1(C(=O)NCC2(C)CCCN2C(C2CC3CCC3C2)=O)nc2ccccn2c1F C1(NC(=O)NCC(CO)C2CCC2)CCCN(c2ccc(Br)cc2)C1=O C1(NC(C(c2cnn(C)c2)C)=O)CC2CCC1N(C(c1ccc(N)c(Cl)n1)=O)C2 c1(C(C)NC(=O)C(O)CN2CCCC2)cccc(OC(F)F)c1Br c1(C(=O)OCC)noc(CSCC(F)(F)CC2CC2)n1 N1(C(Cc2cn(C)nc2)=O)CCC2CCN(C(=O)CC3(O)CCCCC3)CC12 O=C(C1CCCc2nncn21)NC1C=CCN(C(c2cnn3cccnc23)=O)C1 c1(C(NCCNC(c2cc(CC)oc2C)=O)=O)ccc(C2CC2)c(C)c1 c1(C(=O)NCC(C)NC(c2cccc(=S)n2O)=O)cnc(C2CC2)nc1O C1(C(=O)NC2(CC=C)CN(C(=O)CCCF)C2)CC(O)CN1Cc1ccccc1 c1(C(N2CC(NC(c3c(C)cnn3C)=O)C(C)C2)=O)ccc([N+](=O)[O-])cn1 C1(=CC(=O)NCC(C2CC2)NC(c2ccc(C)cc2)=O)CCCCC1(C)C N1(C(CC(CC#C)NC(C2(OC)CCC(C)C2)=O)=O)CCn2c(C)cnc2C1 N1(C(C2CC(OC)C2)=O)CCC(C(N2CC(C3CCCO3)C2)=O)CC1(C)C n1(CC=O)ncc(C#N)c1N.c1(COC)ccc(C(=O)NC)o1.C1CCC1 n1(CC)nc(C(N2CCSCC2C(=O)NCc2nc(=O)o[nH]2)=O)cc1C N1(C(CNC(C=C)=O)=O)CCC(NC(=O)CS(=O)(=O)CC)C(F)C1 Cc1ccc(C(=O)NCC(C)(C)CN(C)C(C2CCCC(N(C)C)C2)=O)cn1 C=CC(C)(O)C(=O)NCC(C1CCCCC1)NC(c1cnc(CC)cn1)=O c1(C(N(CCCCCC)CCNC(c2ccsc2C)=O)=O)cc2n(n1)CCO2 CC(CNC(c1cocn1)=O)C(=O)NC(c1cnsc1)C c1(C(N2CC(O)(CCNC(C=CC3(C)COC3)=O)C2)=O)c(Cl)nsc1Cl CCC(CC)(C(=O)N1CCC1Cn1cc(CCC2CCOC2)nn1)OC N1(C(CSCCOC)=O)CCC(CC(=O)NCC2COCC(C)O2)C1(C)C c1(C(N(CC)C2CC2)=O)ccc2sc(C)nc2c1.C(C)(CO)C=O.CC(=O)N C=Cc1cnn(C)c1C(=O)NC1CCN(C(=O)CCC2CC2)CC1 CCC(C)CCC(O)CC(=O)N1CC(NC(C2(C)CCC3CC3C2)=O)C(CO)C1 C1(CNC(C2(COC)CCCC2)=O)CCCCN1C(C1OCCC1(C)C)=O C1(NC(C2(CC=C)CC2)=O)CCN(C(=O)CCc2nccs2)CC1CO N1(C(C2(C#C)CC2)=O)C2CCCC1CN(C(c1nn(C)c3c1CSCC3)=O)C2 N1(C(C2(CC=C)CC2)=O)CCCN(C(=O)Cc2ccc(C(N)=O)cc2)C(C)C1 C(=O)(C(CC)C(C)C)NC(CCC)C(=O)NC(c1cnn(C)c1)CC c1(C(=O)NCC2CCN(Cc3ccncc3)C2)cc(Br)cnc1Br c1(C(N(C2CN(C(c3ccc(C(O)CF)cc3)=O)C2)C)=O)ccn(C)c(=O)c1 c1(NCC)ccc(C(=O)NC(C)C(C)NC(c2ccc(Cl)o2)=O)c(Cl)c1 C(C(C)(C)CCNC(=O)CCn1cc(Br)cn1)NC(c1n(CC)ccc1)=O C1(CNC(c2n(C=C)ncc2)=O)N(C(=O)CC2CCC(=O)C2C)CCCC1(C)C C12(CCC)CC(C(N3CC(NC(=O)CCC4CNC(=O)N4)C3)=O)(C1)C2 C(CC(C)C(=O)N1CC2C(C(=O)NCCN3CCC(O)CC3)C2C1)=CCC CCCC(C)(O)CC(=O)NCC(C(=O)NCCc1ncoc1C)C(C)(C)C C(=O)(CN1C(=O)COc2ccccc21)N1CCN(C(CCC=CC)=O)CC1C C12(CNC(c3ccc(SC)o3)=O)CC1CN(C(=O)Cc1csnn1)C2 c1(C(=O)NC2CC(CNC(Cn3ccc(C)n3)=O)C2)ccc(Cl)c(O)c1N CN1CCCC1C=CC(=O)NCCNC(=O)C(c1cscc1Br)=O c1(C(=O)OC)c[nH]c(C(=O)NC(C)CNC(=O)CCC2CCC2)c1 C1(C)(C(=O)NCCCC2(NC(c3ccc(C(C)C)s3)=O)CC2)CCCCO1 C(=O)(C1CCc2cccc(O)c21)NCC1CCN(C)CC1 c1ccccc1.C1(C(=O)NCC2(COCC)CC2)CN(C(=O)CCF)C1 N1(C(Cn2c(=O)ccc(C)n2)=O)CCC2CN(C(C3CCCOC3)=O)CC2C1 N1(C(C2CCN(c3n(C)ccn3)C2)=O)CCC(CN(C(C2CCC2)=O)CC)CC1 C1(CNC(C2CC(C#C)(O)C2)=O)CN(C(c2ccn(CCCC)n2)=O)CCC1C Cn1ncc2ncc(C(N3CCC(O)(CNC(=O)C)C3)=O)cc12.C(C)(C)C.O C(CCCCNC(c1cnn(C2CC2(F)F)c1)=O)N(C)C(C1CCC2CC12)=O C12(C(N3CCC(OCC(N4CCN(CC=C)CC4)=O)C3)=O)CCCC1CCC2 C(=O)(C1=CCCN(C(C2(c3ccnn3C)CC2)=O)C1)NC(C1CCC1)C Cc1cccc(=O)n1CCCCNC(=O)NC1CCN(CC(C)O)C1 C1(CC=O)COc2ccccc2O1.C1(COCC(=O)NCC(F)C)CCOC1.N Cc1nc(C(=O)NC(C2CCN(C(=O)Cn3ccsc3=N)C2)C)c(C)o1 C1(NC(C2CCC(COC)C2)=O)CC(OC)CN(C(c2cnc[nH]2)=O)C1 C(C(F)(F)C(C)(C)O)NC(C1(CCNC(CCCN(C)C)=O)CC1)=O n1(CC)ncc2c(C(N3CC4C(C)C4C3)=O)cc(C)nc12.C(=O)C(C)(C)CO.N S(=O)(=O)(CC(C)CC(C)C)N(CC)Cc1cnn(C)c1 CC(C)C(O)CC(=O)N1CC2(CC(CC(=O)NCC3CC(CF)C3)C2)C1 C1(C(C(=O)N(C(C(=O)NCC=CCCC)C2CC2)C)O)CCCCC1 CC1CC(CNC(c2cccnc2F)=O)CN1C(=O)Cn1ccccc1=O c1(C(=O)NC2(CC=C)CN(C(=O)C(CC(C)C)OC)C2)cnc2sc(C)nc2c1 CC(C)CC(F)C(=O)NCC12CCC(NC(=O)CC3(C)OCCO3)(CO1)C2 N1(C(C2CC(C)(C)O2)=O)CCC(NC(c2cccn2C)=O)C(O)C1.c1cccs1 CN(CCCc1nc(-c2cccc(Br)n2)nn1CC(C)(C)C)N=O C1CN(C(C2CCSCC2)=O)CCC1C(F)(F)F.c1(COC)ccoc1C=O.N C1(OC)CC(CNC(=O)CC2CC23CC3)N(C(c2ccc(Cl)o2)=O)C1 c1(CC(N2CCCC(NC(C3CC4CC3CC4O)=O)C2)=O)cc(O)ccc1Br C(=O)(C1=CCCSC1)NCC(CCCC)NC(C1CC(C(C)C)C1)=O C(=O)(C(CC(C)C)CC(C)C)NCCN(CCC)C(C1C2CCCCCCC12)=O CCC(C(=O)OC)C(=O)N1CCCC(N(C(=O)C=Cc2ccc(CC)o2)CC)C1 c1(C(N(CCn2cc(CC(C)O)nn2)C)=O)c(F)cc(Cl)cc1F Cc1ccc(F)c(C(N2CC(CCO)(NC(=O)CC)C2)=O)c1Cl.CCN(C)C.O N1(C(C(CSC)(C)C)=O)CCN(C(=O)CC2CCCCC(=O)N2)CC(CO)C1 C1(NC(CC(C)O)=O)CC2CC(C1)CN(C(=O)CCCn1ccnn1)C2 c1(OC)cnc(C(=O)NCC2(OC)CN(c3nnc(CC(F)(F)F)s3)C2)nc1 c1(C(=O)NCC2(F)CN(C(c3nc(CCC)oc3)=O)C2)ccc(OC)cc1 C(=O)(CCC(F)(F)C(F)(F)F)NC(CNC(C(C)OC)=O)C1CCC1 C(=O)(C1=C(C)OCCS1)NC1CCC(N2CCN(C(C3(C#C)CC3)=O)CC2)CC1 C(=O)(CCCC(=O)c1ccccc1N)NC1CCCC(NC(C=CCCC)=O)C1 N1(C(CS(=O)(=O)NC)=O)CCC2(CC1)CC(NC(c1nnccc1C)=O)CCO2 CCCC(CC)C(=O)N1C(C)C2CC1C2NC(c1cc(C(C)C)on1)=O N1(C(C(CCC)CC)=O)CCC2(CCCN2C(=O)Cn2nnc(=O)[nH]2)CC1 c1(CC(=O)NC2CC(N(C(C(CC)SC)=O)C)C2)ccc(F)c(C(F)(F)F)c1 C1(CC)CN(C(C2(N=[N+]=[N-])CC2)=O)CCO1.n1(C(C)C)cnnc1SCC=O.N c1(NC(C2CN(Cc3c(C#C)cccc3)CC(F)C2)=O)c(C)ccnc1C#N Cc1ccnn1C(C)C(=O)NCC(O)CNC(C1(C(=O)N(C)C)CC1)=O C(=O)(C(C)(C)CC(C)(C)C)N.CC1CC(C(=O)NCC2(CC)CC2)CCO1 CCC(CC)(CC(=O)OC)C(=O)NC.C1(O)CN(C(=O)C(n2cc(Cl)cn2)C)C1 C1(NC(COCCC=C)=O)(CNC(C2CCC2C=O)=O)CCOCC1.O Cc1ncoc1C(=O)NCC(C)CNC(=O)C(O)CC1CCCC1 N1(C(CCC(C)N(C)C)=O)CCCC(CCNC(=O)CCC(N)=O)CC1 C(=O)(CCCC(C)(C)CC)NCC1(C)N(C(CCCC#C)=O)CCC1 N1(C(CCc2nc(C)c(C)[nH]2)=O)CCC(CNC(=O)CCc2ccc[nH]2)C(O)C1 C#CCC(C(=O)NCCc1cccc(F)n1)NC(c1cc(C#N)cs1)=O N1(C(C2(CC=C)CCOCC2)=O)CC2CCCC(C1)N2C(=O)C(CC(C)C)OC N1(CC(CC(=C)C)NC(=O)OC(C)(C)C)C(=O)CCCC1=O C=CC(C)(C)NC(=O)CCNC(=O)CCSCC c1(C(N2CCC(c3ccc(Br)cn3)C2)=O)cccc([N+](=O)[O-])c1Br c1(NC(C2CC(NC(c3ccc(Br)c(Cl)c3Cl)=O)C2)=O)cc2[nH]ccc2cc1Cl C1(C(N2CCC(NC(Cc3ncc(C)s3)=O)C2)=O)C2CCCCCC12 C(=O)(CC1=CCCCC1)NC(CC)C(=O)NC(CC)C1CCC1 c1(C(=O)NCCC2OCCN(C(CC(=C)C)=O)C2)cc(S(N)(=O)=O)cnc1C CC1(C)CC(NC(=O)CC2CCCCCO2)CN1C(=O)C.c1(C=O)ccoc1.N O=C1CCCCC(C(N2CCCC(NC(=O)CC3CN4CCN3CC4)CC2)=O)N1 c1(OC)ccc(C(C)C(=O)NCC(C)(C)C(F)(F)F)cc1OCC(=O)O c1(C(=O)NC(CNC(CCCC=C)=O)(C)C(C)C)ccc(=O)n(C(C)C)c1 Cc1cccc(-c2ncccc2C(=O)N(c2cc(=O)cco2)C(C)C)c1 C1CC2CCC(C1)N2C(=O)Cc1cnns1.C1(COC)CCC1C(=O)N.C C1(CC#C)(C(=O)NCCC(O)C2CCCC2)CCN(C(C2CCC(=O)O2)=O)C1 c1(OC)nccc(-c2cc(Cl)ccc2CO)c1CN1CCN(C)C(C(C)(C)C)C1 c1(OC)cccc2c(NC(C3CCN(C(C4(F)CCC4)=O)C3)C)ncnc12 C1(CC)CCN(C(=O)CC2CCCO2)C(C(=O)NC2CCC2C(=O)NC)C1 c1(CNC(C2CCC(C)C2)=O)cc(O)nc(CNC(c2sncc2Br)=O)n1 Cc1nn(CC(=O)NCC(CNC(c2ccc(C(F)(F)F)[nH]2)=O)CO)cc1Cl n1(CCOC)cccc(C(=O)NCCC)c1=O.c1(C=O)ccc(C(F)(F)F)o1 C1(C(=O)NCCCNC(C(C(C)O)N(C)C)=O)COc2ccccc2C1 C12(NC(c3c(=O)ccn(C)c3)=O)CCCC1CN(C(C1(O)CCSCC1)=O)C2 C(=O)(C(C)(CO)NC(C1CCC1)=O)NC(C)Cc1nn[nH]n1 C=CCC(C)(C)CC(=O)N1Cc2[nH]nc(C(N3CC(C4CC4(F)F)C3)=O)c2C1 CSC1=C(C(=O)NC2CC2CNC(=O)Cc2csc(C)n2)CCCC1 C1CCN(C(C2CC(C(F)(F)F)C2)=O)CC1.C1(C(C)(C)C)CCCC1.CNC C(=O)(C#CC1CCCC1)N1C(C)C(C(=O)NCC2(C(C)(F)F)CC2)CC1 N1(C(C(CC)(C)OC)=O)CCCC(C2CN(C(c3oc(SC)cc3C)=O)C2)C1 C1(CC(=O)NCC2CCCC2C(F)(F)F)CNC2(CC2)CO1 c1(CC(N2CCCCC(NC(c3c[nH]c(Br)c3)=O)C2)=O)cc(F)c(N)cc1F C1(O)(CN(C)C(C2COC(CNC(C3CC(O)C3)=O)C2)=O)CCCC1 C(c1ccnn1C)=CC(=O)NCC(CC=C)NC(C1(C(C)C)CCCO1)=O C#Cc1cn(C)nc1C(=O)NC1(Cc2ccccc2)CCOC1 Cc1ccccc1C(=O)CN1CCCCC1CCn1ccnn1 CC(C)C1=NOC(C(=O)NCC2CCCN(C(=O)C(N3CCOCC3)C)CC2)C1 C(=O)(C(C#N)C(C)(C)C)NC(CCC=C)C(=O)N(C)C[Si](C)(C)C C#Cc1ccc(Br)c(C(N2CCCN(C(=O)NC(C3CCC3)NC)CC2)=O)c1 Cn1cccc(C(=O)NC(C(=O)NC2CC3CCC2(CO)C3)C2CC2)c1=O C1(CNC(COCC#C)=O)N(C(=O)CC(C)C)CCCC1(C)C C1(C(CNC(c2cc(C(F)F)no2)=O)F)CCN(C(c2cncnc2)=O)CC1 c1(CC)cccc(C(=O)NCCC(O)C(=O)N2CC3CC2CS3)c1 Cc1ccc2c(c1)CN(C(=O)C(N1CCN(c3nc(C)cs3)CC1)=O)C2 C1(NC(c2ccc(CC)o2)=O)CC2CCCC12.C1(C(=O)N)C2(CC2)C12CC2 CCCC(C(=O)OC)C(=O)N1CCC(CCNC(=O)Cn2ccccc2=O)C1 c1(C(=O)NC(C(C)NC(=O)CC=CC(C)(C)C)C)nnc(O)nc1O Cn1ncc(CNC(c2cncc(Cl)c2)=O)c1C(N1CC(n2ccnc2)C1)=O C1(c2c[nH]nn2)CN(C(=O)C=CC(F)F)CC1NC(c1cscn1)=O.CC c1(NC(C2CN(Cc3ccc4nccn4c3)C2)=O)cc(Br)cc([N+](=O)[O-])c1 c1(C(=O)NC2CN(C(c3c(OC)ccs3)=O)CC2C)cnc(O)c(F)c1 N1(C(c2ccc(C=C)cc2)=O)CCC2CCN(C(=O)CCc3cccn3C)CC12 C1(NC(C2CCC3CC3C2)=O)CN(c2ncnc(O)c2Br)C2CCCCC12 C1(C#CC(=O)NC(CCN(C)C(c2nn(C)nc2C)=O)C(C)C)(CC)COC1 c1(C(N2CC(C)(NC(C(C)=Cn3ccnn3)=O)C2)=O)cc(C)c2c(c1)CCCN2 N1(C(C(CC)O)=O)CCCCC1CCCNC(c1cccc(C(N)=O)c1)=O N1(C(c2cc(CC)c(C)s2)=O)CCN(C(C2CC23CCOCC3)=O)CC1COC C1N(C(C2CSCN2C(C)=O)=O)CCC1(C)C.n1(CC=C)cccc1C(=O)N c1(C(N(C)C)=O)nccc(C#N)c1F.c1(OCC)n[nH]cc1C(N1CCCC1)=O c1(N2C3(CC3)C2=O)ccccc1Br.C(C(C)(C)CO)C1C(C)C1 C(CNC(=O)C(O)C(C)C)(CC(=O)NCC1CCCSC1)OC N1(C(CCC2N(C(c3c(OC)csc3)=O)CCC2)=O)CCC(N(C)C)C(C)C1 CC1(C)CCCCC(C(N2CCC(NC(=O)CCCS(C)(=O)=O)C(CO)C2)=O)C1 Nc1ncccc1C(=O)NC1CCN(C(c2ncoc2-c2cccc(F)c2)=O)C1 C(=O)(C1=CCN(C(C2CCC3(CCC3)O2)=O)CC1)N(C)CCc1ccccn1 C(CC(F)(F)F)OC(C(C)N(C(CC1N(C(COCCC)=O)CC1)=O)C)=O C1(C)(CC)C=C(C(=O)NC2(C)CCN(C(c3cn(C4CCC4)nn3)=O)C2)C1 CCCCCCC(=O)NC(C1CN(C(=O)Cc2nc(CC)cs2)CCO1)C c1(C(N(CC(=O)N(C(=O)C2CC2)CC)C2CC2)=O)cc(C)co1 c1(C(N(C)CC2CCCN2C(c2coc3c2CSC3)=O)=O)cnn2c1CCCC2 C1CN2CCC1(F)CC2.n1(CC)nncc1C(=O)NCc1cc[nH]c1C(=O)N n1(CC(=O)O)cc(CC(C2CC2)NC(=O)C(F)F)nn1 C1(N(C)C(c2cscn2)=O)CC2CCC(C1)N2C(C1CCCSS1)=O C1(C(C)=O)CCN(c2ccc(-c3ccc(F)cc3)cn2)CC1 N1(C(c2c(C)n(C)nc2)=O)CCC(C)C(N(C(=O)CN(C(=O)C(C)C)C)C)C1 N1(C(Cc2cc(C)nn2C)=O)CCN(C(c2c[nH]c(=N)cc2C)=O)C(C(F)F)C1 CC1CC2CN(C(=O)C=Cc3nnn(C)n3)CC2N1C(C1CN(C)C1)=O C1(NC(c2ccc(C)nc2N)=O)CC2CC(C1)N(C(C1(C)CCCCCC1)=O)C2 c1(C(N(CCCCCC)C)=O)ccc(S(C)(=O)=O)s1.C1(C=O)(COC)COC1 N1(C(CC(n2ccc(C)n2)C)=O)CCC(CNC(=O)C(C)C)C12CC2 N1(C(C(CC)CC(F)F)=O)CCCC(C2CC2NC(c2cnn(CC)n2)=O)C1 Cc1cc(C(=O)N(c2cccc(-c3cccc(OC(C)(C)C)n3)c2)C)cc(O)c1 C1(CCNC(C(C2CCN(C(C(C)CO)=O)C2)(C)C)=O)CCN(C)CC1 C=CC(C)CC(=O)N1CCCC(C(=O)NCC)C1.N1(CC(=O)N)CCC(O)CC1 C(=O)(CCCC(C)CC)N(C1CCCCN(C(CNC(CC)=O)=O)C1)C C(C(=O)N1CCC(C)(NC(c2coc(C3CCCC3)n2)=O)C1)(C(C)(C)C)N(C)C c1(C(=O)OCC)cnc2c(Br)cncc2c1NCc1sccc1C C=CC(CCC)CC(=O)N1CCC(O)CC1C(=O)NCC1CC(O)C1 C(c1ccc([N+](=O)[O-])cc1)=CCN(CC(CN1C(=O)CCC1)O)Cn1cccn1 Cn1c(C(=O)NC2(C)CCCN(C(=O)CC3CCNC(=O)C3)C2)cc2ccsc12 CC1CCN(C(=O)CC(C)P(C)(C)=O)CCN1C(c1cc(=O)c(O)c[nH]1)=O Cn1c(CCC(N2CCC(N(C(=O)CS(C)(=O)=O)CCO)C2)=O)nnc1S Cc1cc(C(N2CCC(NC(c3cnc(C)c(N)c3)=O)C2)=O)ccc1Cl C1(NC(=O)COC2CCCC2)CCCC(CNC(c2cncc(Cl)c2)=O)C1 C1(C(=O)NC(C=C)CO)CC(OC)CN1C(=O)CC(C)n1ccnc1 CC1c2nncn2CCN1C(=O)N(C1CCCC1)CCN1CCCCCC1 CC(C)CC(C)(O)C(=O)NCC1CC(O)(CNC(c2cnc(Cl)s2)=O)C1 N1(C(c2c(C)ncn(C)c2=O)=O)CC(C2CCCN(C(c3ncn(C)n3)=O)C2)C1 CC1(C)C(NC(c2cnn(C3CC3)c2)=O)CCN1C(C12CC(C1)C2)=O c1(C(N(C)CC2CN(C(C3CC3(C)C(F)F)=O)C2)=O)cccn2nncc12 Cc1cc(CNC(C2COCCO2)c2nnnn2CC2CC2)on1 C1(CNC(c2c(CC)non2)=O)CN(C(C2COCCN2C)=O)CC(C)(C)O1 N1(C(c2c(C)ccc(F)c2)=O)CCN(C(c2scnc2C)=O)CC1C#N CCCCS(=O)(=O)N1CCCCC1C(=O)NCCCNC(=O)CCC(N)=O C1(C(=O)NC(CCC)C2CC2)CC(NC(=O)COC2CCCC2)C1(C)C N1(C(C2(COC)CCCO2)=O)CC(NC(=O)COC(F)(F)F)C(C)C1 Cn1cnn(CCC(=O)NC(C2CCOC2)CNC(=O)CCc2ccoc2)c1=O N1(C(=O)NC2CC3(CC(C#C)C3)C2)CCc2nc(C(C)C)ncc2C1 c1(CN2C(CC(=O)NCC(C)(F)F)COCC2)cnc2cc[nH]c2c1 C(=O)(C1=C(C#N)CCC1)N(C(C)CNC(c1cccc(F)c1Br)=O)C c1(C(=O)NCC2CC(C)N(C(=O)C=Cc3cncnc3O)C2)cccc(F)c1Cl Cc1cccc(CC(=O)NCC2CCC(C(=O)NCCC3CCC3)CC2)c1 CN=C(NCC(CO)C(C)C)N1CCC(CC#N)CC1 CCC(CCCC(=O)NC1(C(N)=O)CCCOC1)NC(=O)CC1CCCCCC1 C12(NC(=O)Cc3ccc(Cl)cn3)CCCC1CN(C(=O)CC1(O)CCCC1)C2 N1(C(c2ncc(C)nc2)=O)CCC(C)(C)C(C(N2CC3CC3C3CC23)=O)C1 c1(C(C=O)(C)C)ccc([N+](=O)[O-])cc1F.CCC.C1(C=O)CC1C(F)(F)F.N C1(OC(C(C)c2cc[nH]n2)=O)CCC=CCCC1 Cc1nc(N(C)C)nc(N2CCC(CC(N3CCCC(C(C)C)C3)=O)C2)c1C C#CC1(C(=O)NC2(C)CCOC2C)CN(C(c2ccn(C)c2)=O)C1 N1(C(c2ccc(C(C)=O)[nH]2)=O)CCCC2(NC(C3CCCOC3C)=O)CCCC12 C1(C2CCCN(C(=O)Cc3cnsc3)C2)(NC(C2CN(C(N)=O)C2)=O)CC1 N1(C(C2C(C)C3CCC2C3)=O)CCC2(CCN(C(C3CN4CCC3CC4)=O)C2)C1 n1(C(C)(C)C)cnc(C(=O)N)n1.C1CCCC1.c1(C=O)cnc(C(N)=O)s1.C N1(C(C(CCC)C)=O)CC(C)CCC1CNC(c1cnn(CCF)c1)=O C(=O)(C(CC)CC)NCC1CC(COC)CN1C(C1CCS(=O)CC1)=O.O c1(C(=O)NCC(=C)CCNC(=O)C(C)CCCOC)ccc(F)c(C)c1Cl c1(C(=O)NC(CNC(=O)CCOC2CCCOC2)CO)ccc(O)cc1Cl c1(CCC(=O)NCC2CN(C(C3(Cl)C(C(C)=O)C3)=O)C2)cn(C)cn1 C(=O)(C1=C(CCOC)N(C2CC2C)C(=S)NC1c1c(F)cccc1F)OCC C(c1ccc(F)c(F)c1)=C(C=O)C.C(C)(CC(=O)NCC1CCC1)OC.C c1(C(C)=O)ccc(C(=O)NCC(C)(C)CN(C(=O)Cc2nncn2C)C)nc1 c1ccc(F)cc1.C(C)(C(=O)NCCNC(=O)CC1(O)CC1)=C(CC)C CCC(C(=O)NC)NC(C1CC(n2cc(C(C)(C)CO)nn2)C1)=O Cc1nc2c(s1)CC(CNC(=O)C(=O)NCC(c1ccccc1)N(C)C)CC2 C1(NC(=O)CC2COCCO2)CCC2CN(c3ncnc4c3CCO4)CCC2C1 C(c1ccc(F)nc1)=CC(=O)NCC1(C)CCN(C(C2(C)CC2(F)F)=O)C1 CCC(CCc1ccccc1)C(=O)NCC(O)CNC(c1n[nH]c(C)n1)=O Cc1cc(=NC(=O)C(=O)N2CCC2CNC(c2ccc(Cl)nc2)=O)[nH]o1 CCCC(C)(C)C(=O)N1CCCC(C2CCCN2C(=O)CCN(S(C)(=O)=O)C)C1 CCCCC(CC)CC(=O)N1CC2(CCC2NC(=O)Cc2cn[nH]c2)C1 c1(C(=O)NC2CCC(CCNC(C(CCCC)C)=O)C2)cc2sccc2cn1 C1(CCOC)(NC(c2c(CC)n[nH]c2)=O)CCN(C(c2cnc(O)s2)=O)CC1 Cc1cccc(C(N2CCC(C)C2CNC(=O)CCc2ncc(F)cn2)=O)c1O C(=O)(CCCC(=O)NCC1CN(C(=O)Cc2nc(CC)cs2)C1)NCC N1(C(C=CC(C)(C)SC)=O)CCN(C)C(C(N2CC3CC2C3)=O)C1 c1(SC)cc(C(=O)NCCCC2CCCCN2C(=O)C=CC2CCCC2)oc1C c1(NC(CC2CN(Cc3n(C)cnc3)C2)=O)ccc2c(c1)ncn2C C1(C(N2CC(C)N(C(=O)CCCF)CCC2)=O)CCC2(CCCCC2)C1 c1(C(=O)NCCN(C(C(C)N2CCCC2)=O)C2CC2)ccn2ccccc12 c1(CN(C2CCN(C(CC(=O)OC)=O)C2)C)cccc(-c2ccncc2)c1 c1(C(=O)NCC2CCN(C(CCOC(C)C)=O)C2)cc[nH]c(=N)c1 N#CC1COCCN1C(c1cc(CC2CCCO2)on1)C(=O)NCC1CCOC1 C1(C)(C(=O)NCCN(C(=O)Cc2ncc(C)s2)CCOC)COCCO1 CC1OC(C)(C)OC1(C)C(N1CCN(C(c2cnc(C3CC3)nc2)=O)CC1)=O Cc1c([N+](=O)[O-])c(C(=O)NC2CCC(N(C)C(c3nsnc3O)=O)C2)nn1C C(=O)C(C)(C)C(=O)N(C)C.c1(C(NCCCC)=O)ccc(C2CC2)cc1.CC N1(C(C(C)(Cl)Cl)=O)CC2CCN(C(=O)CC3CCSCC3)CC(C2)C1 C1(NC(CCC(C)(C)C)=O)C2COCC1CC(NC(C1COCCC1(F)F)=O)C2 CCC(C(N)=O)NC(c1ccoc1C(F)(F)F)c1nnnn1CC1CC1 FCCCN=C(NCCN1CCCC1)NC1CCC(OC(F)(F)F)CC1 Cc1nc(O)c(Br)cc1C(=O)NC1CCC12CN(C(=O)C1=CCCC1)C2 C1(C(N2CC(c3cn(CC(CC)O)nn3)(C)C2)=O)CC(S(N)(=O)=O)C1 C(=O)(C(CC)C(=O)N1CCC(NC(c2sc(C)cc2C)=O)C(O)C1)OCC c1(C(N2C3C(NC(c4n(C)ncc4Br)=O)C(C3)C2)=O)ccc(N)cc1F C#Cc1cc(C(=O)NC2CCN(C(c3ccc(Cl)c(F)c3F)=O)C2)cc(Cl)c1 c1(C(N2C(C)CC(CC(=O)NC(CSCC)CO)C2)=O)ccc(=O)n(C)n1 C1(C)(CC(=O)NCCN(C(=O)CC2CCC2C2CC2)CCC)CCCCCC1 C12(NC(c3c(C)nn(C(C)C)c3)=O)CCCN(C(C3CCCO3)=O)CC1C2 c1(-c2cc(CNC(C3(O)CCC3)C)[nH]n2)ccc(C(=O)N)cc1.C(C)(C)C Cc1nn(C)cc1C(C)C(=O)NCC1(C)CCN(C(=O)CC2CC=CC2)C1 C(C)(C)(CC(C)NC(C1CCN(C(c2ccccc2C(=O)O)=O)CC1)=O)OC c1(C(N(CC(C)NC(c2cccnc2C(F)F)=O)C)=O)c(F)cc(Cl)cc1F n1(CC(N2CC(c3nc(C(C)C)on3)OCC2)=O)nc2ccccn2c1=O C1(C(=O)NC(C(C)C)CCNC(C2CNC(=O)N2)=O)CC1C1CCOCC1 CCCCC(C)C(=O)NCC1CC(CNC(c2cscc2C(C)C)=O)C1 Cn1cc(C#CCNC(=O)CN(C(c2cccc3ccoc23)=O)C2CC2)cn1 CC(C)CC(CNC(C1CCCC(F)C1)=O)C(=O)NC1CC(F)C1 C#CC1(C(=O)N(C)CC2CCCN(C(=O)COc3cccc(O)c3)C2)CCCC1 N1(C(C(C)C)=O)CC(C)OC(C)C1.c1(C=O)ccc(C2(C(F)(F)F)CC2)nc1O c1(C(=O)NC(C2(O)CCN(c3ccnc(C4CC4)n3)C2)C)cc(Cl)ncn1 C(CS(=O)(=O)c1ccc(F)cc1)NC(C(C)SCc1ccc(OC(F)F)cc1)=O C1(N(C)C)CCC2CN(C(=O)Nc3n[nH]c(C(C)(C)C)c3C#N)CC12 c1(CC(=O)N(CCCN(c2cc(C)nc(C)n2)C)C)ccc2c(c1)CCO2 N1(C(CCCC)=O)CC2(CCN(C(=O)Cn3nc4n(c3=O)CCCC4)CC2)C1 c1(C(=O)NC(CCOC)CNC(C2(C)CC3CC3C2)=O)nnc2ccccc2n1 c1(CC)cc(C(=O)N)cn(C)c1=O.C1(O)CCCN(C(=O)Cn2cccc2)C1.C N1(C(C)(C)C)CC(n2cc(-c3[nH]nc4c3COC4)nn2)CC12CCCC2 C#CC1CCCN(C(C2CC(C)(NC(=O)C(O)C3CCC3)C2)=O)CC1 C1(C(=O)NC(CCC=C)C(=O)OC)CCN(C(=O)C(C)COC)C12CCC2 C(=O)(C1=CCCOCC1)N1CCC(C(=O)NC2C(C)(C)C(F)(F)C2)C12CC2 C1(NC(C(CC)Br)=O)CC2CCC(C1)N2C(c1ccc(O)nc1)=O Cc1cccc2[nH]c(C(N3C(C(=O)Nc4ccc(I)c(F)c4)CC4CC34)=O)nc12 N1(C(c2ccc(Cl)cc2Cl)C(=O)NCC(=C)C)CC2(C)COCC2(C)C1 N1(C(c2c(NC)nccc2)=O)CCC(F)(C(=O)Nc2cnc(Cl)c(C)c2)CC1 C(=O)(C(F)(F)C(F)(F)F)NCC1C(C)CN(C(=O)CN2CSCC2=O)CC1 c1(C(N2C(CNC(CC(CC)C)=O)(COC)CCC2)=O)ccc(C)c(C)c1N c1(C2C(NCC(COCc3cccc(OC)c3)O)C2)ccc(Br)c(Cl)c1 c1(C(N2CCC(n3ccnn3)C2)C(=O)NCCC)cccc(CO)n1 c1(C(=O)NCC2(C(=O)NCCC(C)OC)CCCCC2)ccc(C#N)n1C C12(CNC(CC(CC)O)=O)CN(C(c3cc(Cl)no3)=O)CC1CCO2 C(CC(C)(C)C(=O)NC(C)C(C)NC(c1cc(OC)ncc1Cl)=O)OC C(C(O)CC(=O)NC1CCN(C(c2cn(-c3ccccc3Cl)nn2)=O)C1)N(C)C C1(C(N(CC(=O)OC)C)=O)COCCN1C(=O)CC1CCC(=O)NC1 c1(SC)nc(NCC2(NC(=O)CCC(C)N(C)C)CCCCC2C)ncc1C c1(C(=O)NC23CCN(C(c4cc(Cl)c(Cl)s4)=O)CC2C3)ncc2ccccn12 n1(CCOCCCOC)cc(C#CCNC(c2nn(C)c(C)c2Br)=O)nn1 N1(C(C(C)CF)=O)CCCC(CNC(C2(S(N)(=O)=O)CC2)=O)C1 c1(C(=O)NCC(CNC(C(C=C)O)=O)(C)C)cc([N+](=O)[O-])c[nH]1 c1(C(=O)NCC2CN(C(CCC(C)C)=O)C(C)C2)ccc2c(c1)n(C)c(=O)n2C c1(C(N2CCC(N(C(C3C(C(=O)OC)CC3)=O)C)C2)=O)cc(F)cc(Cl)c1 C12(C(N3CCC(CCC(=O)NC(CC)(C)C4CC4)C3)=O)CC(C)(CCO1)C2 C1(N(C(=O)CC2NC(=O)NC2=O)C)CCN(C(=O)Cc2cccs2)CC12CC2 Cc1ccc(C(C(=O)N)NC(=O)OC(C)(C)C)cc1.C1CC1.C(C)C.C c1(-n2ncc(C)c2)ccc(C(C)NC2(C(F)(F)F)CC=CC2)cc1F C1(NC(c2c(C)noc2N)=O)CC(F)(F)CC1NC(c1cncc(Cl)c1)=O c1(CCC)c(C(=O)NC(CNC(=O)C=CBr)CC)cnn1CCO N1(C(c2cn(CCC(C)C)nn2)=O)Cc2ccccc2C(NC(=O)CNC=O)C1 c1(C(N2CCC(NC(c3n(C(C)C)ccc3)=O)C2)=O)cc(F)c2[nH]nnc2c1 c1(OCC(=O)NCCCNC(C(COC)N(C)C)=O)cccc(F)c1 C1(NC(CC(n2c(CC)ncc2)C)=O)C=CCN(C(C2(C)CCC(=O)C2)=O)C1 C1(C(N2CCC(OC)C2C)=O)(CC)CCN(C(=O)C(C(C)C)OC)CC1 N1(C(C(CC)(C)O)=O)CC(NC(=O)Cc2ccc3nsnc3c2)C2(CCC2)C1 C(=O)(CC(CC)CC(C)C)Nc1cccc(NC(C(C)OCCCC)=O)c1 C1(NC(C(C)OCC)=O)CCC(O)CN(C(=O)CN2CCCCC2=O)C1 N1(c2n(CC(CC)(C)OC)nnn2)CC2(CCCCC2)CC1C C(=O)(C(F)CC(CC)CC)NC(C1CCN(C(C=C(CCC)C)=O)CC1)CO Cc1ccc(Br)c(F)c1C(=O)NCC.c1(C(N(CC=O)C)=O)ccccc1.N CC1CCC(CNC(=O)CCc2cnn(C)c2)CN1C(c1ccccc1F)=O c1(C(N2C(C)CC(NC(=O)C3=NOCC3)C2)=O)ccc(F)c(O)c1F N1(C(c2c(C)ccc(Cl)c2)=O)CC2CC(C1)N(C(c1cc3cccnn3n1)=O)C2 N1(C(C2(C=C)CCC2)=O)CCCC2(CCC(NC(c3cc(C(N)=O)[nH]n3)=O)C2)C1 c1(C(N2CCC(C(=O)OC)(C(C)C)C2)C(=O)NC(CC)C)cccc(CO)c1 S(=O)(=O)(c1ccc(Br)cc1N1CC2CCCC2C1)N1C2CC(=C)CC1CCC2 c1(C(C(=O)NCC2CCCO2)N(CCCC)C(C)CC)cnc2ncccn12 c1(CC(=O)N(CCCOCCNC(C(C)c2cc[nH]n2)=O)C)cncnc1O c1(C(N(C(C#C)C2CCC2)C)=O)n[nH]cc1C.C1(C=O)CC1C(C)(C)C c1(OC(=O)CC(C2CC2)C2CC2)nc(C2CC2)nc2scc(-c3ccccc3)c12 N(C(=NCCc1cnn(C)c1)N(C)Cc1ccc(Cl)cc1)C(C=C)C CC(C)C(C(=O)NC(C)CCCNC(C1(c2ccno2)CC1)=O)n1cnnn1 c1(SC)ccc(C(=O)NC(C)C(C)C)o1.c1(C=O)nc(C(C)(F)F)cs1.N c1(C(=O)NC2(CNC(C3(C)CC3(F)F)=O)CCOC2)ccnc2ncsc12 C(CC(O)CC(=O)NCC1CN(C(=O)C=CC=C(Cl)Cl)CCO1)SC CC1CCN(C(C2(CF)CCOCC2)=O)CC1CNC(C1(F)CC1)=O c1(NC(CCN(C(=O)CCC=CC)CC#C)=O)ncc(CC)cc1C N1(C(C=C(CCC)CCC)=O)CC(C)CCC1C(=O)NCCOCCCF Cc1nn[nH]c1C(=O)NCCCN(CCCCNC(=O)CCCc1ccsc1)C S(=O)(=O)(c1ccc(Cl)c(Cl)c1)NC(CC#CC)C(=O)O c1(C(=O)NCC(C2CC2)NC(C(C)n2cncn2)=O)ccc2cccnn12 CC1(C(=O)NCC(N)=O)CC12CCN(c1ccc(CC#N)cn1)CC2 c1ccccc1C#N.C1(C(N2CC(CN(C)C(C3(C)CC3)=O)C2)=O)CCCC1O C(=O)(C(F)(F)C(F)F)NCC1N(C(c2cc(C(=O)OC)[nH]c2)=O)CCCC1 C(=O)(C1CCc2snnc21)N1CCC(O)(CNC(CC(C)n2ccnc2)=O)CC1 n1(C(CC)C)nnnc1C(C1(CSC2CCCC2)CC1)NCCOC N#CC1(C(=O)NCCC2CN(C(=O)COCCc3cccs3)C2)CC=CC1 C1(OCC(CN2CCN(c3nc(C)c(C)s3)CC2)O)CCOC2(CCC2)C1 c1(CC(=O)NCC(C2CC2)NC(c2cc(C(C)C)[nH]n2)=O)cccc(Br)c1 N1(C(c2cccc(Br)c2Cl)=O)CC2CN(Cc3n[nH]c4ccccc34)CC2C1 C#CCCCC(=O)N1CCC(N2CCC(NC(=O)Cc3cccs3)CC2)C1 C1(OC(C)C(=O)NC23CC2CN(C(C2(C(C)C)CC2)=O)C3)CCCCCC1 C1(NC(CC=CCNC(CCC(C)=O)=O)=O)CCC(=O)NC1=O c1(CC)cc(C#N)ccc1NC(C1(C)CCN1S(=O)(=O)C(Cl)(Cl)Cl)=O CCC(C)C(C(=O)N1CC(Cc2c(C)cccc2C)C1)OC.n12cc(nn1)CC2 CS(=O)C1CN(C(=O)C(O)C2CN(C(c3ccc(F)cc3)=O)C2)C1 C(=O)CC1=NNC(=O)C1.c1(COC)ccc(C(=O)NC2CCCC(C)C2)cc1 Cc1ccc(C(N2CCN(c3ccc(Cl)c(Cl)c3)CC2)=O)c(Cl)c1Cl c1(C=O)ccc2nnc(C(F)F)n2c1.N1(C(C=CCOC)=O)CCCCC1C.N Cc1cc(C(N2CC(CC(C)NC(C3CNC(=O)N3)=O)C2)=O)cc2c[nH]nc12 CCCCC(O)CC(=O)N1CCCC1C1(NC(C2CC(SC)C2)=O)CC1 C1(C(=O)NC2CCC(NC(CC3(C)CCC3)=O)CC2)CS(=O)(=O)CC12CCC2 Cc1cc([N+](=O)[O-])cnc1N1CC2(CN(C(C3CC3(C)C(C)C)=O)C2)C1 CC1(C)CN(C(C2(CO)CC2)=O)CC(C)(C)C1.C1(C(=O)N)CC1(C)C(F)F C(C)(CNC(=O)CCSC1CCCC1)(C)OC.C1(C=O)CC(=O)C1C.N Cc1cc(C#N)cc(Cl)c1NC(C1CCCN(Cc2cc(Br)co2)CC1)=O C#Cc1ccc(C(=O)N(C2CCCN(C(=O)CCC3CCC3)C2)CC)cc1C N1(CC)CCCN(C(c2nccc(Cl)c2F)=O)CC1.C(C=CC(=O)N)(CC)=CC C(=O)(CCCCC(C)C)N(CC(CC)NC(c1ccc(-c2ccsc2)cc1)=O)C C(F)(c1ccccc1)=CC(=O)NCCCCN(C(C1(C)C(C)C1)=O)C C=CC1(C(=O)NCCCCC(CO)NC(C2CS(=O)(=O)C2)=O)CCOCC1 C=CCCCC(C(=O)NC(c1ccnn1C)CC)NC(c1coc(C2CC2)n1)=O N1(C(=O)NCc2cnccc2C2OCCO2)CCC(CC2CC2)CC1 c1(C(N2CCC(O)(CNC(C(=O)NC)=O)C2)=O)cc(F)cc(I)c1 n1(CC(C2CN(C(C3C(C)(C)C3)=O)C2)F)cc(C2(O)CCOC2)nn1 N1(C(COc2c(C)ccc(C)c2)=O)CCC(C2CC2)(C)C1.C(=O)CC1CC1.N CC(C)CC(CO)CN=c1[nH]c(=NCc2cc(Cl)ccc2F)[nH]c2c1CCCC2 C1CN(C(c2ccc(CC(N)=O)cc2)=O)C(C)(C)C1.Cc1cc(C)c(C(=O)N)o1 c1(CSC)ccc(C(=O)N(C(CNC(C2(F)CCOC2)=O)C2CC2)C)o1 N1(C(C(C=C)OC)=O)CCCC(NC(c2ccc(C(=O)NC)o2)=O)C1 C=C=CC(C)C(=O)NC1CC(NC(c2nccc(-n3ccc(C)n3)n2)=O)C1 CCCCC(CC(=O)N(C)CCOC(F)F)NC(C1(C#N)CCOC1)=O C1(NC(c2c(C)cc(C)nc2Cl)=O)CCC2CN(c3ncns3)CCC2C1 c1(C(C)C)ncc(CNC(C2CC2C)=O)[nH]1.C1(CC=O)CC(F)(F)C1 CC1CCc2[nH]c(=NCCC3CCSC3)nc(N3CCC4(C3)CC(F)(F)C4)c2C1 c1(-c2c(C)nc(CC)s2)cnc2c(C(=O)NCCCCN(C)C)c[nH]c2c1 N1(C(c2n(C)c(S)nc2)=O)CC2CC(O)C1C2NC(C1CCC2(CC2)C1)=O N1(C(CCNC(C(C)=C2CCCC2)=O)=O)CC(C)C(N=[N+]=[N-])C1 c1(C(N2CCC(N(CCC)C(C3CCC3C=O)=O)C2)=O)ccc2occc2n1.O c1(C(=O)NCC2N(C(c3c(CC)cncc3)=O)CC2)ccc2nonc2c1 C12(OC)CCCC(C(=O)NC(C)CNC(=O)C=Cc3ccco3)(CC1)C2 C#Cc1cccc(C(N2CCC(O)(CN(C)C(C3(C)CCCC3O)=O)CC2)=O)c1 N1(C(c2cc(C(C)C)[nH]n2)=O)CC(N(C)C(c2cc(CCO)on2)=O)C(F)C1 Cc1ccc(O)c(C(=O)NCC(C)(C)OCC(=O)N)c1.C1CCNC(=O)C1.C Cn1ccc(S(=O)(=O)N2CCC(CN=c3cc[nH]c(=N)[nH]3)C2)n1 N1(C(C(COCC)C)=O)CC(C=O)C2(CCC2)C1.c1(C2CC2)cnn(C)c1.N c1(C(=O)NC2CCC(C)N(C(C3COC(=O)N3)=O)C2)c[nH]c2ccccc12 Cc1coc(C)c1C=CC(=O)N.C(c1ccc(F)cc1)=CC(N1CCC(C)C1)=O N1(C(CC2N(CC)CCC2)=O)CCC(F)C(NC(=O)CCN2CCN(C)CC2)C1 c1(C(N2C(CCCNC(c3cc(OC)ns3)=O)CCC2)=O)ccc2cc[nH]c2n1 c1(C(N2CCCC2)=O)cccc(C(C)(C)C)c1.c1(NC)nnc(C(C)(C)C)o1.C C12(NC(c3cc(C)c(C)nc3)=O)CCC(CN(C(=O)C3=CCCC3C)C1)C2 C1(C(=O)NCC#CC(=O)NCC(C(C)(C)C)(C)O)Cc2ccccc2C1 N1(C(C(C)=C(CC)C)=O)CCCCC(C2CN(C(c3cn(CCO)nn3)=O)C2)C1 c1(C(=O)NCC(CNC(c2c(N)c(F)ccc2)=O)F)cnn2ccc(O)nc12 N1(C(C(COCC)C)=O)CCC(O)(C(C)NC(c2ccc(O)nn2)=O)CC1 C1(C)(C=O)CCS(=O)(=O)CC1.CC1(C)CC(O)(C(N2CCC(F)C2)=O)C1.C C1(C(=O)NC(CC)(C)CNC(=O)Cc2ccc(OC)nc2)CCc2nc[nH]c2C1 Cc1ccc(C(C)C(=O)N(CC(=O)O)Cc2cn(CCCCCO)nn2)s1 C1(NC(C2(C)CC2)=O)CN(C(=O)CCSC2CCCC2)C2CC12 c1(SC)nc(Cl)cc(=NCC2CC(CNC(c3nc[nH]c4nccc3-4)=O)CO2)[nH]1 C(C)(C)(CC(=O)N1CCC(CN(C(=O)C(C)OCC(F)(F)F)C)C1)OC c1(C(N2C(C(=O)OC)CCC2)=O)ccc(CN2CC(C)C2)cn1.N1CCCC1.C C(CNC(c1n[nH]cc1C)=O)(C(=O)NC1CCC1)OC.c1(C=O)ccccc1 CC(C)(CCCNC(c1cc(Cl)c[nH]1)=O)C(=O)N1CC2(CC(CO)CO2)C1 c1(C=O)cncc(F)c1.c1(CCC(=O)N(CCC)CC)ccc(C(F)F)cc1.N CCC(CC(F)(F)F)C(=O)N1CCC(C)C(NC(C23CCC(CC2)C3)=O)C1 N1(C(C(C)OC)=O)CC(C)CN(C(=O)CCSc2n[nH]c(C)n2)CC1C CCC(CC)CC(=O)NCC1(CNC(=O)COC)CCC1.C1CCCOC1 N1(CC)CCOC(C(=O)OCC(c2ncn(C)n2)=O)C1 c1(OC)cnc(F)cc1NCc1ncccc1C(=O)NCc1ncccc1.O c1(C(N2CCCC(C)C2CNC(=O)OC(C)(C)C)=O)coc2c1CCCC2 c1(C(=O)NC2CC(C)N(C(=O)C(c3ccccc3)F)C2)cnc(Cl)c(Cl)c1 c1(C(=O)NC(C)CC(C)NC(C2CCCC(=O)CC2)=O)c(F)cc(F)c(F)c1F N1(C(C2(CC=C)CCCN2C(=O)CCc2cscn2)=O)C2CCC1CC1(C2)N=N1 C1(CCC)(NC(c2cc3occc3s2)=O)CCCN(C(=O)Cc2nnc(C)o2)C1 c1(NC(c2ccc(C)c(Br)c2C)c2nnnn2C2CC2)ccc2ncc(C)n2c1 N1(C(c2ccc(CC)s2)=O)CC(C(N2CCOC(C3CC3)CC2)=O)CC(C)(C)C1 C1(C)(Cn2cc(-c3cn(CCN(C)C)nc3)nn2)CCNC1=O c1(C(N2C(C)(CNC(CCC(=C)C)=O)CCC2)=O)c(F)c(F)cc(F)c1F c1(N2CC(CC(C)NC(CCCCOC)=O)C2)cc(C(=O)OC)nc(Cl)n1 c1(NC(C2CC(NC(C3CCCC3(F)F)=O)C2)=O)ccccc1CCO c1(C(N(CC)CC)=O)ccc(=O)n(CC(C)O)c1.C(=O)(CC)N.C(N)=O c1(C(=O)NCC(CCNC(c2nccc(C)n2)=O)O)cc(F)cc2nccnc12 C1(C(=O)NCC#CC(=O)Nc2cc(F)ccc2O)CC12CCOCC2 C(=O)(C(C)CC(=O)OC)NCC(=CC(=O)N(CC(C)(C)C)CC)C C1(C(N2CC(O)(CCNC(CCOC(C)=O)=O)C2)=O)CCCOC1C C(c1ccsc1)=CC(=O)NC1CC(C(=O)NC(C2CCCO2)CO)C1 C1(OC)CN(C(C2CCN2C(C)(C)C)=O)C(C)(C(=O)O)C1.c1ccccc1.C CCC(C)(C)CC(=O)NC1(C(=O)Nc2cnn(C)c2C)CCC(C)(C)C1 c1(C(=O)NCC(=C2CN(C(CCN(CCCCC)C)=O)C2)F)noc(CC)c1C Cc1sc2ncc(C(N3CC(CNC(C4CCCC4(C)C)=O)C(C)C3)=O)n2c1C C(=O)(Nn1cnc2ccccc12)C1(CC)CN(C(c2c(CC)n(C)nn2)=O)C1 Cc1ccn2cnc(C(=O)NC(C)C(C)C)c2c1.C1(C(=O)N)CCS(=O)(=O)C1 c1(C(N2C(CNC(=O)CCc3ccccc3F)C=CC2)=O)ncc(Br)cc1F c1(C(=O)NC(c2ccc(OC)c(F)c2)C(F)F)cc(Cl)c(N)cc1F c1(C(N2CC3C(NCc4c(Cl)ccnc4Br)C3C2)=O)cccc2cccc(Br)c12 N1(C(C(c2c(C)ccnc2)(C)C)=O)CCCC(NC(=O)C(C)OC2COC2)CC1 Cc1oc2cc(C(=O)OCC(CO)n3cccn3)[nH]c2c1C CC1COc2c(C(=O)NCC3CCN3C(c3[nH]nnc3C3CC3)=O)cnn2C1 N1(C(c2ccc(SC)s2)=O)CC2CCCC(C1)N2C(c1cncc(C(C)C)c1)=O C1(OC)CC(NC(c2csc(C)n2)=O)CN(C(c2cncc(C(C)=O)c2)=O)C1 C1(CC)CN(C(=O)COCC2CCCCO2)CCN1C(=O)Cn1cc(C)cn1 C1(CNC(C(C(=C)Cl)(C)C)=O)N(C(=O)C=CSC)CCCC1(C)C N1(C(C(C=C)(C)C)=O)CC2(CC(C(=O)NCCN(C3CCCC3)C)CO2)C1 c1(CCC(=O)NCC=CCNC(C(C)OC)=O)ccc(Cl)c(Cl)c1 c1(C(N2CCC(OCCNC(c3c(CC)cno3)=O)C2)=O)cc(S)ccc1F c1(C(N(CC(C)NC(C2(n3ccnc3)CCCC2)=O)C)=O)cc([N+](=O)[O-])n[nH]1 c1(C(N(CCCNC(c2cccn3cnnc23)=O)C)=O)ccn2[nH]c(=N)nc2c1 c1(N(CC(=O)NC)Cc2ccc(C(=O)N)cc2)ccc(C(=O)OC)cc1 CC(O)C(C)C(=O)NCC1CCN(C(=O)CSCc2cccnc2)CC1 Cc1csc(C)c1C(=O)NC1CCC(CNC(c2nn(C)cc2Cl)=O)C1 c1(CC(=O)NCC(CC=C)NC(C2CC23CCCC3)=O)cc(C)ccc1O N1(C(c2cn(C)nc2)=O)CCCC2(NC(=O)C3=COCCC3)CC2C1 C12(NC(c3c(CC)cno3)=O)CCC(NC(=O)C(C)(C)C)(CC1)C2 n1(CC(=O)NC2(COC)CCCN(C(C(CCC)O)=O)C2)ccc(=O)n(C)c1=O CC(C)CC(C)CNC(C1CC2C=CC1C2)=O.c1(C(=O)N)cocn1.C(C)C c1(C(N2C(C)CN(C(=O)CS(C)(=O)=O)CC(C)C2)=O)cc([N+](=O)[O-])c(O)cc1N N1(CCN(CC(O)CN(C)C(C2(F)CCOC2)=O)C)C(=O)NC(C)(C)C1=O C1(N(C(C2(NC(CC3(CSC)CC3)=O)CSC2)=O)C)CCCC(C)C1 n1(CC(=O)NC2CCSC2)cc(CNC(C2(F)CCC2)=O)nn1 Cc1ccsc1CC(=O)NC(CO)C(=O)N(C)CCC1CCC1 c1(-c2c(C(=O)NCc3cnc(-c4ccccc4)s3)csc2)ccc(OC(F)F)cc1 N1(C(C2C(=C)C2)=O)CCC2(CC1)CN(C(c1c(O)cccc1Cl)=O)C2.C1CC1.C CCC(C)(F)C(=O)NC(C)CCCNC(c1ccc(C(=O)OC)cc1)=O c1(C(N2CCC(O)(CC)C2)=O)cccc2c1SCCC2.C(C(F)(F)F)=CC=O.N CC(O)C(F)(F)C(=O)NC1CCC(NC(C2CCC(n3cccc3)CC2)=O)C1 c1(CNC(C2(C)CCN(CC(=O)NC3CC3)C2)=O)cc(Cl)ncc1Cl CCC(CC(=O)NC(C)(C)CN(C)C(c1cn(C)cn1)=O)C(F)F c1(C(=O)NCCCCC2CN(C(CC(CC)SC)=O)C2)cc2sccc2cn1 CC1CN(C(=O)CCN(c2ccccc2)C)CC1NC(C1CCN(C)C1)=O N1(C(c2c(C)nns2)=O)CCN(C(c2cnccc2Cl)=O)C(CCO)C1 C1(F)(CNC(c2c(CC)cns2)=O)CCN(C(C2CCCS2)=O)CC1 Cc1cc(C(=O)NCCCCC2CN(C(=O)C(C)N(C)C)C2)c(C)n1C(C)C C(=O)(C(C)(C)CC(=O)Nc1ccc(C(=O)NC(C)C)cc1F)OC C(CC(C(=O)N1CCC(OC(C)=O)C1)NC(=O)C(CO)OC)OCC N1(C(C2(CSC)CCOCC2)=O)CCN(C(C2CCC(=O)N2C)=O)C(CCO)C1 CC(C)(O)CCN(C(=O)CC1(N)CCOC1)C1CC1 CC(CCCC(=O)N(C)CC1(O)CCOC1)NC(=O)CC1(CO)CCC1 CC1CCc2nc(C(=O)NC3CCCC3NC(C3CC4C=CC3C4)=O)cn2C1 Cc1csc(=O)n1CCC(=O)NC1CCC(NC(C2CCCSC2)=O)C1 C1(N(C(c2c(CC)c(C)sc2)=O)C)CN(C(=O)CC2CCCCC2O)CC12CC2 Nc1c(Cl)cc(NC(=O)C(=O)NCc2ccc(F)c(F)c2F)cc1Cl C(CCOC)(C(=O)NCCC1CCC(=O)N1)NC(CC)=O Cc1ccnc(C)c1C(N1CCCCC1C(N1CCOC(C)C1C)=O)=O C1(N(C)C(c2ccc(Cl)cc2Cl)=O)CCCN(C(c2coc(C(F)F)c2)=O)CC1 C(CC(C(=O)NCC(=O)NC(c1cn(C)nc1C)C)OC)OC C#Cc1ccc(F)c(C(=O)NCCCN(C)C(C2CCCC(=O)O2)=O)c1 Cc1cc(C=CC(N2CCCC2CNC(=O)Cc2occc2C)=O)ccc1F CCCCCC(CC)C(=O)N1CC(C(=O)NCC(c2cn(C)cn2)O)C(CC)C1 c1(OC)cc(CN2CCCCC2C(=O)NCc2cc(Br)cs2)ccc1[N+](=O)[O-] c1(C(=O)NC(CNC(CC2CCN(C)C2=O)=O)(C)C)ncnc(O)c1F Cc1c(C(C)(C)C)o[nH]c1=NC(=O)N1CCCC(C(=O)C(C)(C)C)C1 N1(C(c2ccc(OC)o2)=O)CCCCC(NC(c2cc3c[nH]cnc-3n2)=O)CC1 n1(CCC)ncc(C(=O)NCC(C)(C)CN(C(=O)C(C)NC=O)C)c1Cl C1(O)(CNC(c2cc(C(C)C)no2)=O)CCCN(C(=O)C(O)CC(N)=O)CC1 C#CCCN=C(NCC1C(C)C1C)N1CCC(c2ccc([N+](=O)[O-])cc2)CC1 CCCC(C)(O)C(=O)NC1CN(C(=O)CC(c2cccc(F)c2)O)CCC1C n1(CC(=O)NC2CCCC(NC(c3n(CC)ncc3)=O)C2)ncc(O)nc1=O C1(C2CCCN(C(=O)CN3CCCC3)C2)(NC(c2n[nH]c3cccnc23)=O)CC1 N1(C(CSCC#C)=O)CC2CC1CCC2NC(c1cc2nc[nH]c2cn1)=O C(=O)(CCC(=O)N(C1CN(C(=O)C(CC)CC)CC1O)CC)NCCC C#CC(CO)(CO)NC(C1CC(O)CN1C(=O)CC1CCCOCC1)=O c1(C(N(C(CNC(C=C)=O)C2CC2)C)=O)[nH]c(C)nc1C S(=O)(=O)(c1c[nH]ccc1=NCc1ccsc1)N(c1c([N+](=O)[O-])cccc1)C1CCC1 C1(NC(CC2(C)CCCC2)=O)CCCCC1CNc1ncnc(C(C)(C)C)n1 C(=O)(C1Cc2ccc(F)cc21)N1CC2C(NC(CCC(=O)NC)=O)(CCCC2)C1 N1(C(=O)CC2CCOCC2)CCOCC(C(N2CC(N3CCOCC3)C2)=O)C1 C1(NC(Cn2c(C)ncc2)=O)C2CC3CN(C(=O)COCCCC(C)C)C1C3C2 C(=O)(CC(O)CN(C)C)N1CC(C(C(=O)NC(C(=O)OC)(C)C)O)C1 c1(C(N2CC3(CC3C(N3CCCC3CO)=O)C2)=O)cccc2c1OCC2 C#Cc1cn(C)nc1C(=O)NC1CCN(C(c2[nH]ccc(=O)c2C)=O)C(C)C1 CC(C)C(F)(F)CC(=O)N1CCCC(NC(=O)Cc2ccc3sccc3c2)C1C C1(F)(CNC(c2cc(C)nn2C)=O)CCCN(Cc2ncccc2C)C1 Cc1c(OCC(N2CC(C)(NC(C3CCC(C)(C)O3)=O)C2)=O)cccc1Cl C1(C(N2CCN(c3cccc(C)c3)CC2)=O)CC1C1CC(N=[N+]=[N-])C1 C=C(C)CC(=O)N(CCNC(=O)C(C)(C)C1CCCCC1)CCc1ccccc1 C(C)(N=c1nc(NCc2ccc(C#N)cc2)c2[nH]ccc2[nH]1)c1nc(CC)[nH]n1 Cc1c(C(=O)NC(C)(CNC(c2cc(Cl)c[nH]2)=O)CC(C)C)sc2cncn12 c1(NC(N(CCCC)CCCO)=O)ccc2c(c1)CCC(=O)N2COC N1(C(C=Cc2cn(C)nc2)=O)CC2CCC(NC(C3CCC3(C)C)=O)(C2)C1 c1(C(=O)NCCN(C)C(c2sc(F)cc2Cl)=O)cc(F)c(F)cc1Cl C(CC)(CC(=O)N(C(C)CCCC)C)NC(c1n(CC#C)ccc1)=O Cc1ccc(Br)c(C)c1C(N1CCC(NC(c2ccc(Cl)cc2)=O)C(O)C1)=O C1(CCOC)CN(C(=O)CC(C)F)CCN1C(=O)C(F)CC1CCOCC1 N1(C(c2ccnc(C)c2C)=O)CCC2CC2(C(=O)NOC2CCC2)CC1 C(=O)(C(C)(C)C#N)N(CC(C)(C)NC(=O)Cc1ccn(-c2ccccc2)n1)C c1(CC(=O)NC2CC(CCNC(Cc3ccc(C)s3)=O)C2)cccc(F)c1O Cc1ccc(CC(N2CCC(CO)(CNC(C3(C)C=CCC3)=O)C2)=O)cn1 C1(CC=C)(C(=O)NCC2CCN2C(=O)C(C)Cn2ccnc2)CCOCC1 c1(C(N(C2CCCCN(C(C3(SC)CCC3)=O)C2)C)=O)c[nH]c2cc(F)ccc12 c1(N2CC(C(=O)Nc3c(C(=O)OC)ccs3)SCC2)ncc2c(Cl)cccc2n1 c1(CC)cc(C(N2CCC(CC)CC2C)=O)cc(Cl)c1.C(=O)CN(C)C(C)C.N N1(C(CCN(C)CC)=O)CCC(NC(C23CCOC2CCOC3)=O)C(CO)CC1 c1(CNC(C(=O)Nc2ccc(CC)cc2)=O)ccc(OC(C)C)c(Cl)c1 N1(C(CC(=O)OC)=O)C2CCC1CC(O)(CNC(=O)C)C2.c1ccccc1Cl.S N1(C(=O)NC2(CCC)CCOC2)CC(C#N)C2(CCC2)C1 c1(N(CCCNC(c2n[nH]cc2Cl)=O)CC)ncnc2sc3c(c12)CCC(C)C3 Cc1scnc1C(N1CCCC1C(C)NC(=O)CCN1CCC1)=O c1(C(c2nnnn2C2(C)CC2)NCC(=O)OCCCC)ccnc(F)c1F C1(CCCC)CCN(C(=NCC2CCC3(CCC3)O2)NC(CC)CC)C1.CSC N1(C(C(C)(C)SC)=O)CCN(C)C(C(=O)NCC2CC(O)C2(C)C)C1 Cn1cc(C(N2CC3CC(NC(C4(C)CCCCO4)=O)C3C2)=O)ccc1=O C1(CCC)CN(C(=O)CC(CC)SC)CC1C(=O)NC(c1ncc(C)o1)C c1(C(=O)NCC2CCCN(C(CC3C(C)C3(F)F)=O)C2)csc(=NC2CC2)[nH]1 C(C(C)C(F)C(=O)N(C1CCCCC1)C)NC(C1C(C(C)=O)C1(C)C)=O c1(CC(CC)Sc2ccc(Br)cc2)ccc(C)cc1.C12(CC1)C(=O)N2 c1(C(N2CCCC(CC#C)CC2)C(=O)NCCCC)cc(Cl)c2c(c1)OCO2 c1(CNC(C2CCCN(C(C3(OC)CCOCC3)=O)C2)=O)cccc(C)c1O N1(C(C2C(C)CCC2)=O)CCCC1(C)CNC(=O)CC1CC(C)OC1C CCC(C)C(CC(=O)NC1CCC(=O)N(C)C1=O)NC(C1(C)SCCCS1)=O c1(CCC)cc(C(=O)NC2(CCNC(=O)C(C)(C)OC)CC2)n(C)n1 C(=O)(C(C)C(F)(F)C(F)F)NC(CC)CNC(C1CCC(C(N)=O)CC1)=O CC(C)C1=NOC(C(=O)NCC2CC(NC(C3CCCCCC3)=O)C(O)C2)C1 CC1(C)C(NC(c2cc(Cl)c[nH]2)=O)CC1CC(=O)NOCC(O)CO C(=O)(C(C)CC(=O)OC)NC(CCC)C(=O)NCC(C)CC(=O)OC C1(C=O)CCN(C(=O)C2CC2)CC1.C(C(=O)N(CCC)C)N(CCOC)C.N c1(C(=O)NCC2(NC(=O)CC3C=CCC3)CCCCC2)cn2cccc(Cl)c2n1 C1(NC(C2(C)C(C)(C)C2)=O)C=CCN(C(=O)Cc2cnn(C(F)F)c2)C1 N=C1c2ccccc2NC(=O)C(=O)NC2C1=CC=CC=C(F)C2CCCC C1(NC(c2ccc(CO)cc2)=O)CCN(C(=O)Cn2ccnn2)CC1C(=O)O N1(C(c2c(CC)non2)=O)CCN(C(=O)C(c2ccccc2)SC)C2(CC2)C1 C1(CCC)CN(C(C2C=CC=CC=C2)=O)CC1C(=O)NC(c1ccns1)C Cc1coc(C)c1C(N1CC(=C(F)CNC(C23CC(C2)C3)=O)C1)=O Cc1ccc(CCNC(=O)Cc2csc(NC=O)n2)cc1C#N.C(C)(C)C.O CCC1=NOC(CC(N2CC=CC2C(=O)NCC2CCSC2)=O)C1 C=C(C)CC(C=O)NC(=O)CC1C(C)(C)C1(C)C.n1(CCC)cc(C)cn1.N c1(C(=O)NC2C(NC(Cc3cnc(C)s3)=O)C2)cn(CC(F)F)nc1C C(=O)(C1CCCc2nccn21)NC1CC(NC(=O)CC2COC(=O)C2)C1 c1(C(N2CCN(C(CCC(=O)OC)=O)C(C3CC3)C2)=O)ccc2oc(=O)oc2c1 N1(C(c2cccc(SC)n2)=O)CCC2(CCCN2C(C2CC3CCC(C2)C3)=O)C1 C#Cc1cn(C)nc1C(=O)N(CC(=O)NCC(c1ccncc1)C)C CC1CC(NC(=O)CC2CCC(F)(F)C2)CCN1C(c1ccc(CO)c(F)c1)=O N1(C(CC(C)OC)=O)CC(NC(c2cc(OC)cc(C)c2)=O)CC(O)C1 N1(C(CCN(C)CC)=O)C(CNC(C2(C(F)F)CCCCC2)=O)CC2CC12 N1(C(C(C)Cc2ccc(Br)cc2F)=O)CCC(=O)C2(CCOCC2)C1 C(CC(C)C(=O)NCc1nc(C(N2CC(c3ccccn3)C2)=O)c(C)o1)OC C(=O)(CCC(C)(C)[N+](=O)[O-])NC1C(CNC(c2ccnc(C)c2C)=O)C1 C1(CNC(Cc2c(CC)cccc2)=O)CCCCN(C(c2cc(C)[nH]n2)=O)C1 c1(C(N(C)CC2CCN(C(CC3(C=C)CC3)=O)C2)=O)c(C)cccc1N C1(CNC(c2c(C)oc(Cl)n2)=O)CCCCCN1C(=O)C(C)c1ccco1 C1(NC(c2c(C)nn(C)c2)=O)COC2(CCN(C(C3CCOC3)=O)CC2)C1 Cc1ncccc1CC(=O)N(CCCCC(=O)NC(c1ccn(C)n1)C)C c1(C(N2CC(N(C(=O)CCc3cc(Cl)cs3)C)C2)=O)cnc2nccn2c1 c1(C(=O)NC23CC(CNC(CC)=O)(C2)C3)cnc2cnc(Cl)cc2c1 C(C(C(=O)N1CCC(C(=O)NC(=O)C(C2CCCCC2)=O)O1)C1CC1)OC c1(SC)cccc(C(N2CCCC2C2CCN(C(=O)C(C)N(C)C)CC2)=O)c1F c1(C(N2C(C)CCC(CO)C2)=O)ccc(Cl)c2ccccc12 c1(OC)ccnc(C(=O)NC(C2CCOC2)CNC(c2cscn2)=O)c1O C(=O)(CCC(=O)Nc1ccccc1)NCC(C)NC(c1ccc(C)s1)=O N1(C(CCCN(C)C)=O)CCC2(CC1)C(NC(C1(C)CCOC1)=O)CS2(=O)=O CCC(C)(C)C(O)C(=O)NC(c1ccnn1C)C(=O)NCC1C=CCCC1 C1(C)(C(=O)NCCCC(C)NC(C(CC)(F)F)=O)CC(C(C)C)=NO1 N1(C(c2c(C)nc(Cl)cc2)=O)CC2(C1)SCCC2NC(C1CCCOC1)=O N1(C(c2c(C)cc(CC)o2)=O)CCC(C)C12CC2.c1(C(=O)N)ccnc(Cl)c1Cl N1(C(CCc2cc(OC)no2)=O)CC(NC(=O)CC2(O)CCCCC2)C(C)C1 c1(C(=O)N)ccc(C)cn1.C1(C(N(CC)CC2CCCO2)=O)(CC)CCC1 c1(CNC(Cc2cc(C)on2)=O)ccc(N2CCN(CC3CCC3)CC2)cc1 Cc1oc2cc(C(=O)NC3(CO)CN(C(C4CCCC(C)C4)=O)C3)[nH]c2c1C c1(CCC)ccc(C(=O)NC(C)(C)C(C)NC(=O)CC2(C)CCCO2)cc1 C(=O)(C(F)CC(C)C)NCC(C(=O)OCC)C.C(=O)C(O)CCN(C)C n1(CC(=O)N(CC(C2C(C)(C)C2)=O)C2CC2)ncc(O)nc1=O c1(OC)ccc2cc1NC(=O)N1CCN(CC1)C2=O.C12(CO)CCCNC1C2 C(C1=CCN(C(=O)CC2CCCC(=O)C2)CC1)NC(C1(C)CCCOC1)=O O=C1CCc2ccc(NC(C3CN(Cc4cc[nH]n4)CCC3O)=O)cc2N1 c1(CN2C(C(N3CCC(F)C3)=O)CC3CC32)cc(Br)c(O)cc1O Cc1cc(N2CC(NC(c3cc(O)n(C)n3)=O)CC2C)nc(C2CC2)n1 Cc1cc(F)ccc1C(=O)N(CCCN(C(=O)CCOCC1CCCO1)C)C c1(C=O)cn2c(n1)CC(C)CC2.Cc1cccnc1C(=O)NC1C=CC(C)C1.N c1(OCCC(=O)NCCOCC)cccc(F)c1.C1(CC=O)CCC2CC12 c1(OC)cc(C(N2CCN(C(c3ccc(OC)nc3)=O)C(C)C2)=O)ccc1O c1(C(N2CCC(C(C)(C)NC(c3cnc(Cl)s3)=O)C2)=O)nccc2ccccc12 C(C1CCCN1C(=O)Cc1ccns1)=CC(=O)NC(C)CC1CCOC1 C#Cc1ccc(C(N2CCC(C(=O)Nc3ccc(N(C)C)nc3)CC2C)=O)nc1 S(=O)(=O)(c1ccc(N2CCC(Cc3nccn3C)C2)c(C#N)c1)NCCCC=C C1(CC(N2CC(=C(CNC(=O)C(c3ccccn3)O)F)C2)=O)CCCCO1 N1(C(c2c(C)n[nH]c2)=O)CCC(F)(C(=O)NC2CCN(C3CC3)C2=O)C1 CCC(C(=O)N1CC2(CCN(C(=O)CCc3cccnc3C)C2)C1)C(C)(F)F N1(C(c2c(CC)c[nH]n2)=O)CCC2C(CCCN2C(C2(C#N)CCCC2)=O)C1 Cc1ccc2oc(C(N3CC4CC(N(C(=O)C=CS(C)=O)C)C3C4)=O)cc2n1 c1(C(=O)NCC(C)NC(c2ccncc2)=O)ccc(O)c(Br)c1 C12(C(=O)NC(C)CCN(C)C)C(NC(c3n[nH]c(O)n3)=O)C3CC1C2C3 c1(CC(=O)NCC2(O)CCCN(C(C(CC)(C)F)=O)C2)ncn2c1CCCC2 c1(NC(C2COCCN2Cc2cccnc2Cl)=O)ccc(C(F)(F)F)c(F)c1 C(C(CNC(=O)CNC(c1ccsc1)=O)CO)NC(=O)CCC1OCCO1 C=CCCC(F)(F)C(=O)NCC(CC1CCCC1)C(=O)Nc1cnsc1 Cc1ccccc1-c1nnc(N(C)CC2(O)CCCC2)n1CC(C)(C)O Cc1cccc(C(N2CC(O)CC2CNC(C2CC(F)(CO)C2)=O)=O)c1C C1(C(=O)NCCNC(C(N2CCCC(C)C2)=O)=O)CC12CCC1(CC1)CC2 C(=O)(CCC(=O)NC1(CO)CCN(C(C2CC3(CCC3)C2)=O)C1)OCC CC1=NS(=O)(=O)NC=C1C(=O)N(C1CCN(C(=O)C=Cc2cncs2)C1)C C=CCC(C(=O)NCC1CN(C(c2ccc(Cl)nc2N)=O)CCO1)C(C)C C1(CC=C)(NC(c2cc(Cl)ccn2)=O)CCCN(C(C2(OC)CCCCC2)=O)C1 CN(C)NC(=O)CCC(=O)NCCC1(C)CC1.c1(C=O)sccc1S(N)(=O)=O C(=O)(C1=CC2(CCOCC2)C1)NC1C2CN(C(c3nn(C)c(O)c3)=O)C(C2)C1 C(=O)CC(C)(C(F)F)N(C)C.CCCC(C)CC(=O)NCC1(F)CC(C)C1.N C1(C(N2CCC2)=O)CCCC2(CC2)C1.N1(CC)CC(NC(=O)CO)C(C)C1 C1(NC(C(N2CCN(C(CC)C)CC2)=O)=O)CCC(=O)N(C)C1 N1(C(=O)OC(C)(C)C)CCC(C(=O)N)C1.C1CN(C(C2CC(O)C2)=O)C1 C1(CC)(CC)NC(=O)N(CC(=O)NCCNC(=O)C2=CCOC2)C1=O C(=O)(CC(O)C(Cl)(Cl)Cl)N1CCC(N(C(c2[nH]nc(OC)c2Cl)=O)C)C1 N1(C2CCN(Cc3c(C)nns3)C2)CCN(C(c2cc(Br)c(C)o2)=O)C(=O)C1 n1(CC)nc(C(C)NCCc2nn(C)cc2C)c(C)n1 N1(C(=O)NCC(N2CCCCC2)=O)CCCc2c1ccc(F)c2F C1(CCC)CCN(C(=O)C(C)(C)N(C)C)CC1.C(C)(C)C1(C=O)CC1.CO CC1CCC(O)CN1C(c1ccc(CNC(=O)CC2(O)CCC2)s1)=O C(CN=c1ccc(S(=O)(=O)N2CCCC2C2OCCO2)c[nH]1)n1c(C)ncc1 C1(c2cn(C)nc2)CC2CCC(C1)N2C(=O)NCC1CCC2CCCCN12 c1(C(N2CC(O)(C(C)NC(C3(O)COC3)=O)C2)=O)cc2cc(Cl)ccc2[nH]1 c1(OC)ccc(CC(N2CCCC2CNC(c2ccnc(C)n2)=O)=O)cc1OC C1(NC(C=CC(c2ccc(C)cc2)=O)=O)(C)CCCN(C(=O)C(C)C(C)C)C1 Cc1[nH]nc(CO)c1C(=O)NC1CCC(C(=O)NCC2CCC2)CC1 c1(-c2cn(CCCN(C(C(CC)OC)=O)C)nn2)ccc(F)cn1 C(C)(CC(C)C)(C(N)=O)NC(C1C(NC(CC(CC)(F)F)=O)CCC1)=O CC(CCCCNC(=O)C(CO)c1ccccc1)NC(=O)CC1COC(=O)C1 c1(CCC)cc(C(=O)N(CCCCNC(c2ccc(OC)nn2)=O)C)sc1C C(=O)(C(C)CCCC(C)C)NC(CCOC)C(=O)NCC1CC(CF)C1 CCC(C(=O)N1CC(CO)(NC(C2CC(CF)C2)=O)C1)Sc1ccccc1 c1(C(=O)NC2C(C)CCN(C(c3cc(C)ncc3)=O)C2)ccc2c(C)[nH]nc2c1 N1(C(CCCCCC)=O)CCC2C1CCCN2C(c1[nH]cc2c1CCS2(=O)=O)=O N1(C(C(c2ccccc2)C)=O)CCN(C(c2cc(C#N)on2)=O)C2(CC2)C1 N1(C(C(CC=C)OC)=O)CC2CCC(CNC(C3(C)C=CCCC3)=O)C2C1 CC(Cl)(Cl)C(=O)NCCCC1(NC(c2ccnn2CC(F)F)=O)CC1 c1(C(=O)NC2CCN(C(C3C(=C)CC3)=O)C(C)C2)ccnc2c1CC(=O)N2 CC(C)CC(C(=O)NC(C1CCCN1C(c1ccncn1)=O)C)C(C)C C(=O)(C1CCCc2nc[nH]c21)N1CC(N(C(C=Cc2c(C)ccnc2)=O)C)C1 C1(CNC(COCC(=O)NC)=O)CCCN(C(c2[nH]ncc2C#N)=O)C1.C N1(C(C(F)=CCC)=O)CCC(OCC)C1.C1(N(CCC(=O)N)C)CCCCC1 N1(C(c2n(CC)ccc2)=O)CCOC(CC(=O)NCC(C(F)(F)F)OC)C1 CCC(C(=O)NCC(C)(C)CNC(=O)CO)C(F)(F)F.c1c(C)cccc1C Cc1cccc(C(=O)NCC2CCCC2NC(=O)CC2CC3CCC2O3)c1C c1ccc(F)cc1Cl.C1(CC(=O)NCC2(O)CN(C(=O)CC)C2)C=CCCC1.S N1(C(C2(CNC(C(CCCC)O)=O)CCCC2)=O)CCn2ncnc2C1 C1(C(=O)NC2(c3nnnn3C3CCCC3)CC=CC2)C2CN(CC(F)(F)F)CC12 c1(CC)nc(C(=O)NC(C(=O)NCCCCOC)C2(O)CCC2)c(C)o1 CCC(C)CC(C(=O)NCC(C)(C)C#N)NC(=O)CCn1cnc(=N)[nH]1 c1(CNC(c2c(C)c[nH]n2)=O)ccc(CNC(=O)C(CO)N(C)C)c(F)c1 C1(C(=O)OC)CSCN1C(=O)Cn1cc(CC2CCOC2=O)nn1 c1(SC)cncc(NC(C2C(C)CN2C(=O)Cc2csc(C)n2)=O)c1 C1(C(=O)NCC(C(=O)NCC2(CSC)CC2)OC)COCC(C)O1 c1(CCC)ccc(C(=O)NCC2CCC2)cc1.C(c1scnc1C)=CC(=O)N N1(CCC)CC(C(=O)NCC23CC(NC(c4cnsn4)=O)(C2)C3)CC1=O C1(C(N2CCN(CC3CN(C(CCCC=C)=O)C3)CC2)=O)CC2C(C1)C2(C)C c1(NCCN(C(C2CCN(CC=C)C2=O)=O)CC)cc(O)nc(C)n1 c1(C(=O)NC2(CF)CN(C(C3CC34CCCC4)=O)C2)cnc2ccoc2c1 c1(N2CCC(N(C(C3C(OCC)C3C)=O)C)C2)nc(Cl)nc2c1CCC2 C(N=c1[nH]cnc(NCCCS(C)=O)c1C)c1c(OC)c(=O)cco1 Cc1ccc(Cl)c(C(=O)NC(C)(CNC(C2CSCCS2)=O)C2CC2)c1 C(=O)(C1=CC2(CN(C(=O)CCC(C)=O)C2)OC1)NC(c1noc(C)n1)CC C#Cc1cc(C(=O)NCC2CN(C(=O)CC3CC3)CC2C)cc(Br)c1 C12(CNC(C3CC(=O)OC3)=O)CCC(CC1)CO2.c1(C=O)ccc(F)cc1F.N c1(C(N(C(C)CNC(=O)CCCN=[N+]=[N-])CC)=O)c(C)ncc2ccccc12 N1(c2nnc(C)n2CC#CC2CC2)CC2(CCCC2)C1c1ccccc1 N1(C(=O)N(C(c2cccc3cc[nH]c23)C)C2CC2)CCC2OCC(=O)NC2C1 c1(C(=O)NCCC(CNC(CCC(C)OCC)=O)O)c[nH]c2cccnc12 c1(NC(C)=O)ccc(CN2CC(F)CC2C=O)cc1.c1cccc(C(C)C)c1.N CC1CCC(=CC(N2CCC(CC(C)NC(c3ccnc(O)c3)=O)CC2)=O)CC1 c1(N2CCC(C3N(C(C(COCC)C)=O)CCCC3)C2)cncc(C#N)n1 C#Cc1cc(C(N2CC(NC(=O)CC3(O)CCOCC3)C(C=C)C2)=O)ccc1C C1(F)(CNC(C(=C(C)C2CC2)F)=O)CCN(C(c2cc(Cl)ccn2)=O)C1 c1(C=O)cn(CC)cn1.C1(C#N)CC1C(F)(F)F.C(=O)C=O.C1CC1.N C1(C(N2CC3CN(C(C=CCC)=O)CC3(C)C2)=O)Cc2ccccc2C(=O)O1 c1(C=O)cc2sc(Cl)cc2[nH]1.C1(C(N)=O)(C(=O)NCCC2(C)CC2)CC1 C1(CNC(c2c(CC)ncs2)=O)CC2CCC1N2C(=O)C(C)S(N)(=O)=O c1(C(C)C)cc(C(=O)NCCCOCC)ccc1F.c1(C(=O)N)cc(Cl)cn1C Cc1cc(NCC2CC(NC(=O)C(F)OC(F)(F)F)C2)c(F)cc1[N+](=O)[O-] C1(C(=O)NCCN(CCC)C(c2c(C)nn(C)c2N)=O)SC2C=CC1CC2 N1(C(c2cc(C)nc(C)n2)=O)CCC2(C(=O)NCCN=S(C)(C)=O)CCCC12 N1(C(C(COCC)C)=O)CC(C(N2CC(C)CCC23CC3)=O)C2(CCC2)C1 N1(C(C(CC=C)(F)F)=O)CCCC2(CCCN2C(c2ccc(C)s2)=O)C1 C1(NC(C=CC(C)(C)NC(C2C(C)(C)C2(C)C)=O)=O)CC1C1CCCC1 C(CCCCC(=O)NC(C)C(C)SC)NC(C(C)(C)SC)=O N1(C(c2cc(OC)no2)=O)CC2CC2(NC(c2cccc(C(C)C)n2)=O)C1 Cc1ccc(C(=O)NC(C)CNC(=O)Cc2cccc(Cl)c2)c2ncccc12 N1(C(c2cc(C)nn2C)=O)CC(C)(C)CC1CNC(=O)C.[SH](C)(=O)=O C1(N(C)C)CCC(N=c2[nH]c(=N)[nH]c(=NCC3(CC4CCCCO4)CC3)[nH]2)CC1 C(=O)(C(C)C(F)(F)F)N(C(C)CNC(C1(CC(C)C)CC1)=O)CC C(C)(CCCC(=O)N1CCC1(CC)CC)NC(CC1ON=C(CC)C1)=O C1(CC(=O)NC(c2nc(C)[nH]n2)C)CN(C(c2nn(C)cc2Cl)=O)CCO1 Cc1cc(C(=O)NCC(C(=O)NCc2ccsc2C)N(C)C)on1 c1(CNC(C2CCN(C(=O)CC3CCSC3)C2)=O)cnc2[nH]cnc2c1 CC1CCC(C(=O)N(CCCNC(=O)CSCc2ccncc2)C)O1 C#CCCCC(C)C(=O)NCC=CC(=O)NCC(O)CC c1(N2CCCN(CC(=O)NC(C(F)F)C3CCCO3)CC2)nc2ccccc2s1 C1(NC(c2nncc(C)c2)=O)C(C)CCN(C(=O)Cc2ccccc2C)C1C N1(C(CC(CC)C)=O)CCC(NC(c2ccc(C(C)C)cc2N)=O)C(F)(F)CC1 C12(CCOCC1)CC(=O)NCCO2.C(C(=O)NCC=C)(OCC)OC N1(C(C(C)NC(C)=O)=O)CCN(C(=O)Cc2cc(C)on2)C(CO)C1 C1(CCCNC(c2cn[nH]c2)=O)CN(C(c2cc(C3CCC3)no2)=O)CCO1 c1(C(N(C(c2cc(OC)ncc2)C)CC2CCCC2)=O)ccc([N+](=O)[O-])cc1C Cc1cc2c(C(=O)N)ccc(C)c2[nH]1.c1(C(N(CCC)C)=O)ccc([N+](=O)[O-])o1 Cc1cc(C(=O)NCC2CC(C)CN(C(=O)CCn3cnnn3)C2)cn(C)c1=O C1CCN(C(C2CC(N3CCOCC3)C2)=O)C1C.C1(CC(=O)N)(C(=O)OC)CC1 C(=O)(C(C)(CC)CCC(C)C)NC1C(CNC(C(C)=CC)=O)CCC1 C1(NC(CC(=C)C)=O)CN(C(c2ccc(C(=O)OC)cc2Cl)=O)CC(C)(C)C1 c1(C(N(CC(C)NC(c2ccc(C)c(Cl)c2)=O)C)=O)cnc2cccnc2c1 N1(C(C(C)OCC#C)=O)CCCOC(CNC(C2(CC)CCNC2=O)=O)C1 C1(NC(C(n2c(C)ccn2)C)=O)CCCCC1NC(c1ccc(O)cn1)=O N1(C(C(CC)OCC)=O)CCCC(N(CCF)C(c2ccc(F)s2)=O)C1 c1(C(=O)NC(C)CCNC(=O)C(C)C2CC2)cccc([N+](=O)[O-])c1 C(C)(CO)(CC(C)C)NC(C(C1CN(C(c2cc(CC)[nH]n2)=O)C1)OC)=O c1(OC)cc(Cl)ccc1CNC(C1CCC1)=O.c1(C(=O)N)cc(C#N)c[nH]1 N1(C(c2c(F)cccc2Cl)=O)CCC2CCN(C(=O)C3=CCCSC3)C2C1 O=C(C1=CCCN(C(c2cc(Br)cnc2F)=O)C1)NCC1(O)CC1 C=CCC(CC(C)C)C(=O)N1CCN(C(=O)C2=CCSC2)C(C)C1 c1(CC)cc(F)cc(Cl)c1.C(C=O)(C(C)C)NC(C)=O.C(=O)CC(C)(F)F.N C(CN=c1[nH]c(Cl)ncc1Cl)C1CCCN(C(c2cccc3nnn(C)c32)=O)C1 c1(C(=O)NCC(N(C(c2c(OC)ccs2)=O)C)C2CC2)cc(Cl)ccn1 c1(NCc2c(OC)ccs2)cnc(Cl)cc1C(=O)Nc1[nH]cnc1C(N)=O c1(NCC(C(C)O)(C)C)[nH]c(=NC2CC2)nc2sccc12 CC1CCC(NC(=O)CCC(=O)OC(C)(C)C)CN1C(C1CCCOC1C)=O CC1(C)CCN(C(c2ccncc2F)=O)C1CC(=O)NCCc1ccccc1O CN1CCC(NC(=O)CC2CCN2C(C2CCCC2O)=O)C1(C)C N1(C(C2CCC(CC)CC2)=O)CC(NC(=O)Cc2ccccc2O)CC2(CC2)C1 C1(NC(c2c(CC)onc2C)=O)CCC(C)N(C(c2cc(F)n(C)n2)=O)C1 CC(C)C(CCNC(c1snc(Cl)c1Cl)=O)NC(C1OC(C)CC1C)=O c1(OC)ccc(F)c(C(=O)NCC2CCCN2C(=O)CC2CCCC2)c1Cl.O c1(C(c2n(C(C)C)nnn2)NC2CC=CC2)ccccc1C(F)(F)F c1(C(=O)NCC(C2CC2)NC(CN(C(COC)=O)C)=O)cc(O)cnc1N CC(CCc1ccc(F)cc1)C(=O)N1CCCC1C(C)C.C1(CC(=O)N)CCOC1 CC(C)C(CO)C(=O)NC1CC(C)N(C(c2cccc(CN(C)C)c2)=O)C1 c1(C(C)=O)cc(C(=O)NCCc2nc[nH]c2Br)c(C)o1 N1(C(c2ncc(CC)cn2)=O)CCC(O)(C(C)NC(=O)Cc2cscn2)CC1 c1(C(NC2CCN(C(C3(CCN(C)C)CC3)=O)CC2)=O)cc(Cl)cnn1.CC N1(C(CC(CC2CC2)NC(c2c(C)ccs2)=O)=O)CCC(C)(F)CC1 C1(CC)(NC(c2cncc(N)c2)=O)CCN(C(C2(F)CCCOC2)=O)CC1 c1(C(=O)NCCCCC2CN(C(C=C(C)Cl)=O)C2)cc(C)cc2ccncc12 C=C1CC2CCCC(C1)N2C(C12CCC(CC1)N(C(c1nnc(S)n1C)=O)C2)=O C(C)(CCCCC#N)N1CCC(c2nc(C)c(C)s2)CC1 C(=O)(NNC(=O)CNn1nc(C)c(Br)c1C)c1ccc(OC)cc1 C(CCC)(C(=O)N(C(C)CCNC(c1nocc1C(C)(C)C)=O)C)=CCC C1(C(=O)N)Cc2ccccc2C1.C12(C(N(CCC)CC)=O)CCC(CC1)C2(C)C c1(-n2c(CNC(CCCC)C)nnn2)cnn(C(F)(F)F)c1OC CC(F)CCN=C(NC1CCC1N1CCOCC1)N1CCC2(CCC2)C1 N1(C(c2ccnc(C)n2)=O)CCC(NC(=O)C=Cc2ccnn2C)CC1C Cc1cc(-n2ccnc2)ccc1C(=O)NCC1CC1NC(=O)C.C(N)=O CCC(CC)CCC(=O)NCC(O)CNC(C1(C)C=CCC1)=O c1(NC(c2cn(CCC(C)C)nn2)=O)cccc(C)c1.C(=O)C(C)C1CCC1.N C1(CNC(CC(C)OC)=O)CN(C(C2CCC(F)C2)=O)CCO1 C1(CC)(NC(=O)CS(=O)(=O)N(C)C)CCCN(C(=O)CC2CCCN2C)C1 C1(NCCC(=O)OC)CC(C)(C)CC1C c1(C(C)C(=O)NCCN(C(=O)C2=COCCC2)CC2CC2)cc2ccccc2o1 C(C)(CO)(C(C)(C)O)NC(c1cncc(CNC(CC(CC)C2CC2)=O)c1)=O N1(C(CSCC=C)=O)CCC(c2ccccc2CNC(=O)C(C)C(C)O)CC1 N1(C(COc2cc(C)on2)=O)C2CCC1CN(C(=O)CCC1CCC1)CC2 N1(C(CCCc2[nH]c(=N)sc2)=O)CCC2CN(C(=O)CC(O)C3CCCC3)CC12 c1(C(N(C2CCC(NC(CCSC)=O)CC2)C)=O)cc2c(Cl)cccn2n1 C(C1c2ccccc2CN1C(C1CC2CC2C1)=O)NC(C(C1CCOCC1)C)=O c1(OC)ccc(CC(=O)NCC2(F)CN(C(=O)CN(C)CCO)C2)cc1Br c1(C(N2CC(C)N(C(=O)Cn3nccn3)CC2)=O)cc(S(N)(=O)=O)ccc1O N1(C(c2c(C)ccnc2)=O)CCC(CNC(C2(C)CC2)=O)C(C)C1 N1(C(c2sc(CC)c(Br)c2)C(=O)NC2CC2)CC(CCOC)c2ccccc21 CC1(C)C(NC(=O)CN2CCCC2=O)C2CCCN(Cc3ccc(F)c(F)c3)C12 c1(C(=O)NCC2C(NC(c3cc(Br)c[nH]3)=O)C2)ncccc1Cl CC1CN(C(c2snc(Cl)c2Cl)=O)CC1NC(c1ccc(OC(F)F)cn1)=O N1(C(C(C)(C)Cl)=O)CC2CCC2(CC(=O)NCCC(C)(C)C2CC2)C1 Cc1nnc(CC(=O)NCCOC2CN(C(c3nocc3Br)=O)C2)o1 N1(C(c2n(CCC)ncc2)=O)CCC2(CC1)CC2NC(=O)C(C)OC N1(CC(N(C)CCNC(C2CCCC(C)(C)O2)=O)=O)CCn2ccnc2C1 N1(C(C(C)c2cccs2)=O)Cc2[nH]nc(NC(=O)C=Cc3ccccc3Br)c2C1 C(=O)(C(C)(O)C(F)(F)F)N1CCC(C(N2C(COC)COCC2)=O)C1 C(=O)(C(C1=NOC2CC12)N1CCC(c2n[nH]c(C)n2)CC1)NCC N1(C(c2c(C)nc(CC)o2)=O)CCN(C(C2CCN2CC)=O)C(CCO)C1 c1(C(N2CC3C(NC(CCCOC)=O)C(C3)C2)=O)cccc2ccoc12 N1(C(c2n[nH]c(C)c2Br)=O)CC2CC(NC(C3(CF)CCC3)=O)CC2C1 c1(C(=O)NCC2COCCN2C(=O)C)cc2c(Cl)cc(F)cc2[nH]1.C1CC1.O C12(c3onc(C)n3)CCCC1CN(C(=O)C(C)S(C)(=N)=O)C2.n12nccc1C2 c1(C(N2CC=CC2C(N2CCC2CO)=O)=O)cccnc1OC(F)F C1(NC(C(CC)(C)CNC(=O)C(C#N)C(C)C)=O)CCCCCC1(C)C c1(C(N(CC(CC)NC(=O)Cn2nnnc2C)C)=O)cnc(C)cc1C C1(CNC(CN(C(COC)=O)C)=O)CN(C(C2(C)CSC2)=O)CCC1(F)F CC(CC(=O)NCCNC(c1cn(CC2CCOC2)nn1)=O)C(C)(C)C C1(C(N2CCC(CNC(c3c(C)nsc3)=O)C(O)C2)=O)CCCCC1N=[N+]=[N-] Cc1nc(-c2ccccc2)c(NC(=O)NCC(C2CC=CCC2)(C)O)n1C Cc1c(C(N2CC(CC(N3CC=CC3CN(C)C)=O)CC2C)=O)ccn1C CCC(CC)(CCCn1cc(-c2cc(F)ncc2C)nn1)C(=O)OC C1(C(=O)NC(CNC(C2C(C(=O)OC)C2)=O)(C)C)CCCN1N=O C1(NC(C(C)OCC)=O)CCC2(CC1)CCN(C(=O)C(F)CC)CC2 N1(C(c2nc(OC)oc2)=O)CC(NC(=O)Cc2nnc(C)o2)C(C2CC2)C1 CC(C)CC(O)C(=O)NCC(C)(CC(C)C)NC(=O)C=Cc1nccs1 C1(CN(C)C(c2ncoc2C)=O)CCC(C)CC1.C1(C(=O)N)(OC)CCOCC1 N1(C(CNC=O)=O)CCN(C(C2CC(CC(F)F)C2)=O)CC2(CC2)C1 C1(C(=O)NCC(O)C2CC2)C2CCC(C2)N1C(c1cncc(Cl)c1)=O N1(C(C(CCC(C)C)F)=O)CCC2(CCC2NC(=O)CC2CCC(C)(C)O2)CC1 C(=O)(CC(C)(C)CCOC)NCC1CN(C(C2(COC)CCCCC2)=O)C1 C(=O)(C1=NN(C)C(=O)CC1)NC1C2(CCN(C(C(=O)N(C)C)=O)CC2)C1 N1(C(CN2CC(CC)C2)=O)CC(C)C2(C1)CN(C(c1ccc([N+](=O)[O-])[nH]1)=O)C2 N1(C(c2c(N)cc(OC)c(F)c2)=O)CCC2(CNC(=O)C(C)CO)CCCCC12 C1(C=O)CN(C(C2CC2Cl)=O)CC1C(F)(F)F.n1(C(C)C)cc(CF)nn1 C(=O)(C1=CCS(=O)(=O)C1)N1CC(O)(CN(C(=O)CCCF)C)C1 C12(CNC(CCC=C(C)C)=O)CCCCC1CN(C(c1cc(C)ccc1Cl)=O)C2 c1(C(=O)NCCNC(c2cnc(C#N)s2)=O)cnn2cccc(Br)c12 N1(S(CC)(=O)=O)CCCC(C(C)NC(C2C3CC2(c2ccccc2)CO3)=O)C1 N#Cc1ccc(NC(C2CC(F)CN2C(=O)CCc2cc(Cl)ccc2Cl)=O)cc1 N1(C(CC2CC(NC(c3cc(C)sc3N)=O)C2)=O)CC2(CCC(=O)N2)C1 c1(C(=O)NC(CN(C(C2CSCCS2)=O)CC)C)c(F)ccc2nc[nH]c12 C1(C(=O)NC2CC(O)(Cn3cc(-c4cnccc4Cl)nn3)C2)CCOC(=O)CC1 C1(NC(C(C(C)C)n2cccc2)=O)CCN(C(c2ccc(CO)s2)=O)CC1(C)C C(CCCCC(=O)NC(C1CSC1)C)NC(C(CC=CC)C)=O c1(-n2ccc(C(=O)NC(CC)CNC(c3csc(C)c3)=O)n2)ccccc1Cl N1(C(CCn2cc(C(C)(C)CC3CCC3)nn2)=O)CCCC(CC(F)(F)F)C1 N1(C(C2C3N(C(C(CCC)OC)=O)C(CC3)C2)=O)CCCC2OCCC12 N1(C(c2c(C)cns2)=O)CCCC(C2CCN(C(=O)C3=CC4(CCOC4)C3)C2)C1 CC1CC(NC(C2CCC(C(N)=O)C2)=O)CN(C(c2coc(O)n2)=O)C1 c1(C(N2CC=CC2)=O)ccccc1CS(C)(=O)=O.Cn1cc(CC(=O)N)cn1.C c1(-c2nc(C(C)C)nn2C2CCCS(=O)(=O)C2)ccc2c(c1)OCCO2 C1(C2N(C(C3(CN(C(C4CCOC4)=O)C4CC4)CC3)=O)CC2)CCOCC1 C(=O)(CCCc1cccs1)N(CCCNC(C(C)NC(C)=O)=O)CCO N1(C(c2scc(C(N)=O)c2)=O)CCN(C(=O)CCC2CCCOC2)C(CCO)C1 c1(C(c2nnnn2CC2CCOCC2)NCC(CC)C)ccc(F)c(F)c1Br C1(C(N(CC(C)(C)O)C)=O)CCN(C(C2CC3(CCC3O)C2)=O)CCO1 n1(C(C)C)ncc(C(N2CCN(CCNC(=O)CCCOC(C)C)CC2)=O)c1N CCCCC(CNC(=O)CC1CC(C)C1)NC(C1(C2CCCCO2)CCC1)=O c1(C(C)C)cccc(C(N2CCC(C)C2C)=O)n1.c1(C=O)ncoc1C1CC1.N C1(NC(C2C(C)(C)C2)=O)CN(C(=O)Cc2ccncc2Cl)Cc2ccnn2C1 C1(NC(c2coc(CO)c2)=O)CC2CCC(C1)N2C(C1(CO)CCOC1)=O C(c1ncco1)=CC(=O)N(CCC(c1cccs1)NC(=O)Cc1ccsn1)C Cc1csc(C(C)C(N2CC(O)(CN(C(=O)Cc3nncn3C)C)C2)=O)n1 CCC(CC(=O)N(CCC(=O)NC1CC1CC(C)C)OC)SC n1(CC)nncc1C(=O)N(C1CC(C(=O)NCC(C)(C)O)C1)C C1(NC(c2ncn(CC)c2)=O)CN(C(c2csc(-c3ncc[nH]3)n2)=O)CC1O CCCC(C)(O)CC(=O)NC(CC1CC1)C(=O)NCCc1nc(C)no1 c1(SCC)cncc(C(=O)NCC(O)CC)n1.C(c1cccnc1)=CC(=O)N N1(C(C=CC(C)C)=O)CCCC1CCCNC(c1ccncn1)=O c1(C=O)cc(F)c(F)c(F)c1.N1(C(=O)CNc2ccccn2)CCCC(F)(C)C1 C(=O)(CCCCCSC)NC1C=CCN(C(c2c(OC)nn(C)c2)=O)C1 C1(NC(c2cc(CC)c(C)cc2)=O)CC2CN(C(=O)CC(C)C)CC2C1 c1(C(N2CC(C)C(NC(c3cnncc3O)=O)C2)=O)c(C(F)(F)F)cccc1F Cc1c(C=O)cnn1CCO.C12(CC=O)COC(C)(C1)C2.C12CC(C1)C2.N CCC(C)(C(=O)NCC1(NC(c2csc3cncn23)=O)CCC1)C(F)F c1(C(N2CC(CCNC(=O)COC(F)F)C2)=O)scc2c1CCCC2 CN1CCC(C(N2CCCC(C)(CNC(c3nnc(O)nc3O)=O)C2)=O)S1(=O)=O C(=O)(C1=C(Cl)CCC1)NCC(C)(C)NC(=O)COc1ccccc1C#N N1(C(c2cc(C)cc(OC)c2N)=O)CCCC2(C1)CN(C(c1ccc(C)o1)=O)C2 C(CCCCCNC(=O)C(C)OCCC(C)C)NC(c1c(CC)onc1)=O c1(NC(N2CCOCC2C2CCOC2)=O)ccnc(C2CCC2)c1 C(=O)(C(CO)C(F)(F)F)N1CC(O)(CN(C(=O)CSC2CC2)C)C1 O=C1NC(C(N2CCC(NC(c3cnns3)=O)C2)=O)CO1 c1(NC(C2CN(c3cccc(CC)c3)C(=O)C2)=O)ccc2sccc2c1 Cc1cc(C(=O)NCCCOCCN(C)C(C2CCCCC2C)=O)cc(N)c1 N1(C(COC(CC)C)=O)CCOCC1CCNC(=O)CCC1CC1 c1(C(=O)NC2CC(NC(Cn3c(=O)ccc(C)c3)=O)C2)c(F)ccc(C#N)c1F C1(CNC(C(C(C)C)SCC)=O)CN(C(=O)C(C)S(C)(=O)=O)CCN1C n1(CCC)cc(C(=O)NC2(CCNC(c3c(C)n[nH]c3C)=O)CC2)c(C)n1 C#CCC(CC(=O)N(C1CCC1)C)NC(c1cnn(C)c1C#N)=O C(=O)(C(C)C(C)(F)F)NCCN(CC(C)O)C(c1cnsn1)=O C1(F)CCN(C(=O)CCC2C(=O)ON=C2C)CC1.C(C(=O)N)(C1CC1)OC.C n1(C(C)C)cc(C(=O)NC2CCCC2NC(=O)C)c(O)nc1=O.C1CCC1.O CCCC(C(=O)NC(C)(C)CC=CC(=O)NCC(C1CCC1)OC)N(C)C c1(C(=O)NC(CCNC(C=CC(C)C)=O)C)sccc1I c1(CNC(=O)C(=O)NC2CCN(C3CCOC3)CC2)ccccc1I N1(C(c2c(C)coc2C)=O)CCN(C(C2OCC3CCCC2C3)=O)CC(CO)C1 C1(C(=O)NCC(C2CC2)NC(Cc2ccc(C)s2)=O)Cc2ccccc2N1 C1(C(=O)NCCC2(NC(C(=O)N(C)C)=O)CC2)Cc2c(F)cccc2O1 c1(C(c2n(C(C)C)nnn2)NCC2CC23CCCCC3)noc2c1CCCCC2 CC1(C)CC(NCC2CCCCC2)C1OCc1ccccc1 O=C1NCCCC1n1cc(C2CCN(C(=O)CC3CC4(CC4)CO3)CC2)nn1 c1(OC)c(C(N2CCCC2CC)=O)occc1=O.C1(CC=O)CC(C)(C)CO1.N N1(C(C(c2ccn(C)n2)(C)C)=O)CCC(O)(CNC(=O)CC)C1.C1COC1.O c1(C(=O)NCC(CC)NC(c2ccc(C)nc2OC)=O)cnc2n1CCC(C)C2 N1(C(C=C(C)C(C)C)=O)CCOCC1C(=O)NC(C(N)=O)C1CCCC1 CC1CCCC=C1C(=O)N1CC(C(=O)NC(C)C(C)(C)C)OC(C)C1 c1(OC)ccc(CC(=O)NC(CO)CC)cc1.c1(C=O)cnc(C(C)(C)C)[nH]1.N c1(C(C(=O)NCCCNC(=O)C(O)C2CCCC2)O)cccc(Br)c1 C=CC(CC)C(=O)N(C)CC1CCCC1NC(c1c(C2CC2)noc1C)=O C(CC(=O)NC(C)CO)(C(C)(C)C)NC(C=Cc1ccc(C)cc1)=O C1(NC(c2ccc(CO)cn2)=O)CCN(C(c2nnc(O)cc2O)=O)CC1CO c1(C(=O)NCCC2CN(C(C(COC)OC)=O)CC2C)cccc(OC)c1F C(c1cnccc1C)=CC=O.C1(OC)CCC(CC(=O)N(CC)C2CC2)CC1.N c1(C(=O)NCC2CN(C(C(CC)=CC)=O)CC2O)ncn2c1CCCCC2 C(=O)(C(F)C(C)C)N(C(C(=O)OC)C)C1CC1.C(=O)CCC1OCCO1.N Cc1nc(NC(C2(C)CCCN(Cc3ccnn3C)C2)=O)cnc1C#N c1(CC)nc(C(=O)NC(C2CN(C(=O)Cc3ccccc3)C2)C)c(C)o1 C(CCN=c1nc(S(C)(=O)=O)cc[nH]1)N(C(C(C(=C)C)(C)C)=O)C CCCC(C)(O)CC(=O)NCC=CCC(=O)NCC1CCC(=O)O1 c1(C(=O)NC(CN(C(c2nc(C)c(C)s2)=O)CC)C)cc(N)ccc1Cl CC1(C(N2CC(O)(CCNC(=O)CCCC3CCC3)C2)=O)CCCC1(F)F N1(C(c2n(CC)c(O)nc2)=O)CCN(C(C2CCC2(C)C)=O)C(C2CCC2)C1 c1(C(N2C3C(NC(C(COC)O)=O)CC(C3)C2)=O)c(C)cc(OC)cc1C C1(N(C)C(C2CC=CC2)=O)CCC(NC(c2cc[nH]c2)=O)C1 c1(NC(C2(O)CCN(C(c3ccccc3)=O)C2)=O)cc2c(F)cc(F)cc2[nH]1 N1(C(CC2(CC)CCOCC2)=O)CC(NC(c2csc(CO)n2)=O)CC(C)(C)C1 c1(C(N(CCN(C(=O)C=Cc2ccc(Cl)nc2)C)C)=O)cnc2cccnn12 C(=O)(C1CCc2nccn21)NC(C(=O)NC1CC(CC)(CC)C1)(C)C C1(CCC)CN(C(=O)C(c2ccccc2)OC(C)(C)C(F)F)CC1C(=O)N C(=O)(C1=CCN(C(=O)C#CC2CC2)CC1)NC(C1CCCCC1)C#C O=C(N=c1[nH][nH]c2cccnc12)C1CN(Cc2n[nH]cc2Cl)CCS1 c1(N(CCN(C(C2C(CC)OCC2)=O)C(C)C)C)nn2cc(C)nc2s1 N1(C(CC(C)n2ccnc2)=O)CCC(NC(=O)CCOC2CCCCC2)C(O)C1 C1(C(=O)N)CCOC(C(F)(F)F)C1.C1(CC(=O)N(CCC)C)(CSC)CC1 C1(C2CCCN(c3cc(C4CC4)ncn3)C2)(NC(c2cccnc2O)=O)CC1 C1(CC(=O)NC(COCC)C(=O)N2CC(C(F)(F)F)C2)CCCC(=O)C1 C=CC(C)(O)C(=O)N(C)CCN(C(=O)CCC(C)NC(C)=O)C(C)C c1(NC(C2(C)CCN2Cc2ncccc2F)=O)ccc(O)cc1-c1ccccc1 N1(C(C2CCC(CC)O2)=O)CCCC(C)(C(=O)N(C2CC(C(N)=O)C2)C)C1 c1(C(N2C(CNC(CN(C)CC)=O)C(C)CC2)=O)ccc(O)c(C)c1C c1(OC)ccnc(C(=O)NC)c1.C1(C=O)C2CC3C(C2)C13.C1(O)CCC1 C(=O)(C(CC(F)F)N(C(=O)CSC(F)F)C)N(C)Cc1cccs1 CCC(COC)C(=O)N(CCCCC(=O)NC(C1CCOC1)CO)C C(=O)(C1=Cc2ccccc2C1)NCCCN(C)C(c1[nH]ccc1-c1cccs1)=O C(=O)(CC(O)Cc1ccccc1)N1CC(CNC(c2ccc(CCC)s2)=O)C1 c1(OC)nc(C)c(C(=O)Nc2ccccc2)s1.c1(C(=O)N)nocc1C(C)C Cc1cnn2ccc(C(=O)N(C3CCCN(C(c4ccn(C)c4)=O)C3)C)nc12 C(=O)(CC(C(F)F)C(C)(C)C)N1CCN(C(CC)=O)CC1C(C)C.C(=O)(OC)N C1(C(N2CCC(NC(C3(C)CC(=C)C3)=O)C2)=O)(CC)CCCCO1 Cc1ccc2occ(C(N3CC=CC(NC(C4CCC=CCC4)=O)C3)=O)c2c1 c1(NCc2n(CC)ncn2)[nH]c(=NC2COCCOC2)nc2c1cnn2C c1(C(=O)NC(CC)(C)CNC(c2[nH]c(C)nc2C)=O)cccc(F)c1Br c1(SCC)cccc(CC(=O)N)c1.C1C2CCN(C(C3CCC3)=O)C12.C1CC1 CC1N(C(C2CCN(C(=O)C34CCC(CO)(CC3)C4)O2)=O)CCCC1(C)C c1ccc2c(c1)CN(C(=NCCCOCC1CCC1)NC1CCCC1)CCO2 C1(C(N(C)CC2CN(C(=O)Cc3ccsn3)CCO2)=O)CCCCC1(C)C N#Cc1ccc(Br)c(NNC(=O)NCCS(=O)(=O)NCC2CCC2)c1 CC(C)CCC(c1nnnn1CC1CCOC1)NCc1ncnn1C c1ccccc1.C1(C(NC)=O)CC1C1CC1.C(C)(C(=O)N)OCCOCC N1(Cc2ccc(C(=O)O)c(Cl)c2)CCC=C(C(=O)NCc2cccnc2Cl)C1 C=C=CC(C)C(=O)N(C)CC1CCCN(C(=O)COc2ccc(Br)cc2)C1 C(=O)C1SCCc2sccc21.c1(CNC(C2C=CCC2)=O)nc(C)cc(O)n1.N Cc1nn(C)c2c1CC(NC(=O)C(=O)NC(C)CCc1cccn1C)CC2 S(=O)(=O)(c1cccc(C(=O)NCCCCC)c1)NCC.C1(C(=O)N)CCC1 C(=O)(CCCCC(C)C)NC1CC(N(C(c2n[nH]c(C)c2C)=O)C)C1 N1(CCOCC)CCN(C(=O)Nc2cc(CC)ccc2CC)CC1C c1(C=O)ccnc(F)c1N.Cc1noc(C)c1CSCC(=O)N.C(C)C1CC1 c1(C(=O)NC23CC(CNC(=O)CCc4cn[nH]c4)(C2)C3)cccc(Cl)c1O C=CC1CCCCN1C(C(=O)Nc1ccccc1C)C(C)C1CC1 c1(C(N2CCCC(C(C)NC(C3C4CCC3CC4)=O)C2)=O)c(F)ccc(F)c1N c1(OC)nsc(OC)c1C(=O)NCC1CC1C.C1(O)(C=O)CCC1.N N1(C(c2nc(C)oc2C)=O)CCC(C)(C)C(C(N2CC3CC3(CO)C2)=O)C1 N1(C(C2(C)OCC(C)OC2)=O)CC2CC(C1)CN(C(C1CC(=O)C1C)=O)C2 c1(N2C(CN(C(CC)=O)C)CCC2)[nH]cnc2nc(Cl)cc1-2 N1(C(=O)CCc2cc[nH]n2)CCCC(CN2CCN(C(C3(O)CCC3)=O)CC2)C1 CC(C)=C=CC(=O)N(C1CN(C(=O)Cn2cc(C3CC3)cn2)CC1O)C CCCC(CCCNC(c1n[nH]cc1Cl)=O)NC(c1[nH]ncc1C#N)=O c1(C(N2CCCC(NC(Cc3c(C)ocn3)=O)(CO)C2)=O)cc2scc(C)c2[nH]1 C1(C(N2C(CNC(C3C(OC)CC3)=O)CCCC2)=O)Cc2cc(C)ccc2O1 CC1CN(C)CC1C.C1(CC=O)CCCC2CC12.C1(CC=CC=O)CCC1 C(C)(C(=O)N)(c1ccccc1)OC.C1(C)(CC(=O)N(CC)C)CCCO1.CC N1(C(CC2C(C)CCN(C(Cc3c(C)con3)=O)C2)=O)CCC(F)(F)C(O)C1 c1(CNC(C=CCC)=O)ccc(C(=O)NCc2cnco2)cc1 N1(C(=O)C2CC2)CCN(C(=O)CNC(=O)NC2CC2)CC2(CC2)C1 N1(C(C2CC(=C)C2)=O)CCN(C(=O)C(C)OCC(F)(F)F)C(c2cccnc2)C1 C1(CC(N2C(CCNC(CCCSC)=O)CCC2)=O)NC(=O)CN(C)C1=O c1(NCC(C(C)(C)F)(C)F)[nH]c(=NCCc2ccccc2CO)nc2scnc12 N1(C(CCCSC)C(=O)NCCCC2CC2)CC2CCCCCCC12 Cc1c(C=CC(=O)NC2CC(C)(NC(=O)C3=NOC(C)C3)C2)cnn1C N1(S(C(C)C#N)(=O)=O)CCC2(CC1)CC(C(=O)NCCN1CCOCC1)CO2 N1(C(c2cc(C)[nH]c2)=O)CCCC1(C)C(=O)Nc1ccc(O)cn1 c1(C(=O)NC2CCN(C(C(CC)SC)=O)C2C)cc(F)c(OC)cc1Br Cc1cc(-c2nc(CC(N)=O)nn2-c2ccc(C(C)C)cc2)ccc1O N1(C2CCN(CC)CC2)CCOCC(C(=O)NCC(C)(C)CN(C)C)C1 C1CC2CCC(C1)N2C(=O)CC1CCC1.C1(CC)CC(C(=O)N)C1.N(C)C C(C(C(=O)NC(C)Cn1ccnc1)NC(=O)C(=O)C1CCCC1)SCC C1(N(C(=O)CSc2ccccn2)CCO)CCC2(CC1)CNC2 c1(C=O)ccc(O)c(C)c1C.C1(C(=O)NCCC2CCC2)(OC)CCOCC1.N Cc1c(C(N2CCN(CCC(C)C)CC2)=O)ccc2c1CCNC2 N1(C(C(C(C)C)NC(N)=O)=O)CCCC(CCNC(=O)C(F)C(C)C)CC1 C(C(C)NC(c1snnc1C)=O)(C(C)C)NC(CC(=O)NCC#C)=O C(=O)(C1=C(C)OCC1)N1CC2C(C(N3C(C(=O)OCC)COCC3)=O)(C2)C1 CC(C1COc2ccccc21)NC(=O)CCOC1CCNCC1 c1(NC2CCN(C)C2)cc(S(=O)(=O)NCC2CC(F)C2)ccc1C#N C1(OC)(C)CCN(C(=O)C)C1.C1(C(=O)N)CC1C1CC1.c1(C=O)cscn1 C1(O)(CNC(C2(CC(C)C)CCC2)=O)CCN(C(C2CCC2F)=O)CC1 N1(C(C(C)Cc2ccc(C#N)cc2)=O)CCCC(C)(NC(=O)C(O)C(C)(C)C)C1 C(=O)(C(CN=[N+]=[N-])NC(=O)C=C1CCOCC1)NC(C(=O)OC)CCF Cc1noc2ncnc(N3CCC(CNC(c4c(Cl)ccnc4F)=O)CC3)c12 N1(C(C(=O)NC(C2CN(C(C(CC)N(C)C)=O)C2)C)=O)CCCC(C)C1 c1(C2(NC(c3ccc(C(F)F)c(Cl)c3)c3n(C)nnn3)CC2)ccc(F)cc1Br CCCCC(C)C(=O)N1CCC(CCNC(=O)C(N2C(C)CCC2C)C)CC1 C1(CC)CCN(C(=O)CCc2ccc[nH]2)C1.n1(CC(=O)N)cnc(C(F)(F)F)n1 N1(C(CSC(C)(C)C)=O)CC2CC(NC(=O)CCCC(O)c3ccccc3)C1C2 N1(CC)CC(C(=O)NC)CCC1C(=O)O.c1ccc(C(=O)O)n1C C(=O)(CC(CC)N(C(=O)CSCCNC(c1cccnc1)=O)C)OCC C12(C(N(C(C=C)C3CC3)C)=O)COC(C1)C(NC(=O)C#CC(C)(C)O)C2 CC1CC(N(C)C(C2CC(F)(F)CN2C(=O)CCC2CCCN2C)=O)CC(C)C1 N1(C(CCN(S(C)(=O)=O)C)=O)C2CCC1CN(C(=O)CCC(C)(C)F)C2 C1(CS(C)(=O)=O)CN(C=O)CCN1C(=O)CCn1ccnc1.C1CCC(=O)O1 C1(O)(CNc2nccc(OCC)n2)CCCN(C(=O)CCc2cnc(C)s2)C1 c1(C(N(C(C)C)CC)=O)csc([N+](=O)[O-])c1.c1(C(=O)N)ccc(C2CC2)o1 N1(C(c2cccc(C)c2Cl)=O)CC2CCCC(C1)N2CCOCC1CC1 C(CN=c1[nH]c(=NC2CCS(=O)CC2)[nH]c2c(F)cc(F)cc12)SCS(C)(=O)=O N1(C(CN2CC(C)(C)C2)=O)CCC(C(F)C)CC1.c1(C=O)cc(C(N)=O)cs1.N C1(C)(C(N(C(C)C2CC2)C)=O)CCCO1.C1(C(N(C)C)=O)(C(=O)N)CC1 c1(C(C)NC(C(CCCC)C)=O)cc2cccc(F)c2o1 C(O)(CCNC(=O)NC1COCC1C(N)=O)(C(F)(F)F)c1n(C)ccn1 C#CC1CN(C(c2cccnc2SC)=O)CCN1C(c1cncc(C(C)C)c1)=O C=CC1(O)CCN(C(C2CCC(C(C)C)N2C(C2CCCOC2)=O)=O)C1 c1(C(=O)NC(c2cn(CC3CCOC3)nn2)C)cc2cncn2c(O)n1 N1(C(c2n[nH]c3c2CCCC3)=O)CCC2C(CCCN2C(=O)Cn2nccn2)C1 n1(CCOCC)nnnc1C(C)(CSC(C)(C)C)NCCCC1CC1C N1(C(C2CC(C)N(C)C2)=O)CCN(C(=O)C(C)(C)S(C)(=O)=O)C2(CCC2)C1 C(C)(CO)(C(F)(F)F)N(C(C1CCN(C(CSCCCC)=O)C1)=O)C(C)C Cc1cccc(CC(N2CCC(CCCNC(=O)COC3CC3)CC2)=O)c1Cl C1(C(=O)NC(CNC(C2(CSCCOC)CC2)=O)C)CCCN1C C(=O)(C1=CCCCO1)NCC1C(NC(C=CC(C)(C)C)=O)C1 CCC(C)CC(C(=O)NCC(C(F)(F)F)OC)NC(=O)C1=CCSC1 N1(C(c2ccc(C(C)=O)cc2)=O)CCCC(NC(=O)C(O)C2CC2)C1C N1(C(C(=O)N(CC(F)(F)CC)CC#C)=O)CC2(CCC2)C1C1CCOCC1 C(C(C)(C(=O)N1CCC(CN=[N+]=[N-])C1)NC(C12CSCC1C2)=O)SC C1(NC(c2cncnc2)=O)CCCCN(C(=O)C=Cc2ccc(Br)o2)C1 C(=O)(CC(C)C)NCC(=O)N(CCCNC(C=C(C)C(C)C)=O)CCO N1(C(C2C(=C)C2)=O)CC(C2CCN(C(c3nn(C)c4c3CSCC4)=O)CC2)C1 C(=O)(C1=C(Cl)CCOC1)N(C)CCN(C)C(c1cnoc1-c1ccc(Cl)cc1)=O c1(N(C2CC3(CNC3)C2)C(C2(C)C(C)C2)=O)ccc(S(F)(F)(F)(F)F)cc1 c1ncc(N)c(C(=O)N(C2CN(C(=O)Cn3cc(C4CCC4)nn3)C2)C)n1.CS C(C(=O)NC(C)(CO)C(=O)NC(c1cncs1)C)(C(C)C)OC N1(C(C(F)=CCC)=O)CCC2(CC(NC(c3ccc(F)c(CC)c3)=O)CO2)C1 n1(C(C(=O)N(CC(C)OC)C)C)cc(C(C)(C)C(N)=O)nn1 C(C)(C(C)(C)C(=O)N1CCC(CC(C)(C)C)C1)NC(c1cncc(C)c1)=O N1(C(CC2(CSC)CC2)=O)CCC(O)(CNC(=O)CN2CCCC2C)C1 Cc1cccc(C(=O)NCC(CC2CCCC2)C(N2CCC3(CCC3)C2)=O)c1O c1(C(=O)NC2C(C(N(CCNC(C)=O)C)=O)CCC2)cc2ccccc2[nH]1 C1(CNC(c2c(CC)ncs2)=O)CC(C)CN(C(C2CCCCC(=O)N2)=O)C1 O=C(CN1CCN(C2CC2)C1=O)N=S(=O)(c1ccc(F)cc1Cl)C1CC1 c1(C(N(C(C)CNC(c2ccc(Br)cc2)=O)CC)=O)cncnc1C1CC1 C(=O)(C(OC)OCC)NCCNCCC.C12(COC1)C(=O)NC2 c1(C(N(CC(Cc2ccccc2)NC(CCC)=O)C)=O)ccnnc1C(F)(F)F Cn1nccc1C=CC(=O)NCC(C)(O)C.CC(F)(F)C(F)F.C(=O)(CC)N C1(C(C)C)(C(N2CCC3CCC23)=O)CCN(C(c2sccc2Cl)=O)C1 C1(C(=O)NCCc2c(C)ncs2)C2CCC(C2)N1C(c1cccc(O)c1)=O c1(C(=O)OC)cc(Br)c(CNc2ccc(F)nc2)[nH]1 CC(CC(=O)NCC1(NC(c2cc3n(c2)CCCC3)=O)CCOC1)CC(C)(C)C n1(CC(CNC(C(=Cc2ccncc2)C)=O)O)ccc2ccccc2c1=O C(=O)(C(CC1CC1)OC)NC(C1CN(C(C=CC(CC)=CC)=O)C1)C c1(C(N2CCC(C(C)NC(CC(=C)C)=O)CC2)=O)cc(OC(F)F)cc(F)c1 n1(C(CC)C)nccc1C(=O)N(CCC(C)NC(=O)CCNC(N)=O)C C1CC(C)CN(C(=O)C=Cc2ccnn2C)C1.C1(C(=O)N)(COC)C=CCC1 c1(C(=O)NCC(C(C)C)(C)NC(C2CN(C)C2)=O)cc(Cl)c2n[nH]cc2c1 C(=O)(C(C)(O)C(F)(F)F)N(CCCCN(C(C(c1cncnc1)C)=O)C)C c1(C(=O)NCC2C(C)CCCN2C(C2CCC=CO2)=O)cc(F)c(F)cc1Cl N1(C(COC)=O)CCOC(C(N2Cc3ncsc3C2)=O)CC1 c1(N2CCC(NC(N(c3cn(C)nc3Cl)C)=O)C2)cccc(Cl)c1 C1(C(N2CCCC(CCC(N3CC(C(C)(C)O)C3)=O)C2)=O)CCC2(CCC2)C1 C1(CNC(COCCCC#C)=O)CCCC(NC(C2CCC2OC)=O)C1 C=C(C)CC(C(=O)N(C1CN(C(c2cccc(=O)o2)=O)CCC1O)C)OC N1(c2nccc(C(=O)OC)n2)CC2COCC2(C(=O)N(C)CC2CCCCC2)C1 N1(C(c2cc(C)on2)=O)CCC(CNC(c2cnn3cc[nH]c23)=O)C12CC2 c1(OC)ccc(C(=O)NC2COCC2C(=O)N(C)CC2CN(C)C2)cc1 c1(NC(C2C(C(=O)NC(CCCC)CO)C2)=O)c(C)cc([N+](=O)[O-])cc1Cl c1(OC)ccc(C(=O)NCc2nnc(C3CCN(C(N)=O)CC3)s2)c2[nH]ncc12 Cc1cc(C)c2c(c1)C(NC(=O)C(=O)NCC1CCOCC1(C)C)CCO2 C1(NC(N2CC(c3ncnn3C)(OCC)C2)=O)CCC(C#N)C1 C=CC1CCCCN1C(=O)CCOCCCNC(=O)Cn1cccn1 c1(C(=O)NC2CCCCN(C(CC)=O)CC2)cc(S(C)(=O)=O)ccc1C c1(C(=O)NCC(C)CNC(=O)COCCCF)sccc1S(C)(=O)=O O=S(=O)(c1cccnc1N1CCn2c(Br)cnc2C1)NC1CC=CC1 Cc1cc(C(=O)N(C)CCOCCNC(C2CC23CCOCC3)=O)c(F)cc1Cl c1(C(=O)NCC2CC(NC(C(C(C)(C)C)SC)=O)C2)cccc2c1NCCC2 c1(C(N2CCN(C)C(CNC(c3ccc(Cl)cc3)=O)C2)=O)nnn2c1CSCC2 c1(C(C(=O)NCCCc2cncc(F)c2)O)ccc(F)c(Br)c1 N1(C(=O)NC(c2scc(C)n2)C(F)(F)F)CC2(COC(=O)C2)C1 Cc1c(C(N2CCN(C(C3CC4C=CC3C4)=O)CC2)=O)ccc(Cl)c1Cl c1(NC2C(N)CC2)nccc2c1CCO2 C1CN(C(C2C3CCC(=O)C23)=O)CCC1(C)C.c1(OC)ccccc1C(=O)N.C c1(C(N2CCN(C(C3CC=C(C)CC3)=O)CC2)=O)cc2cc(Cl)cc(Cl)c2[nH]1 C(=O)(C(CCC)C(C)C)N1CCN(c2ncc(C#C)cn2)C(CCO)C1 C(=O)(CCC(C)C#N)N(CC(C)O)CCNC(=O)CS.c1cccc(Cl)c1 C1(COC)CCCCN1C(c1scnc1C)C(=O)Nc1ccccc1C C12(NC(CCNC(=O)OCC)=O)CC(C1)C2.C(=O)(C)N.CC(F)F C=CCCC(C1CC1)NC(C1CC(F)(CNC(=O)C(C)OC)C1)=O c1(C(c2nnnn2C2(C)CC2)NCCn2c(C)ncc2)cnc(C(C)C)n1C N1(C(C2C(CC)C2)=O)CCCC2CN(C(=O)CC(C)(C)C)CCC12 O=C(CCC1CC1)NCCCN(c1nnco1)C1CC1 C=CCC(C)C(=O)N(C)CC1CN(C(C2(OC)CCSC2)=O)CCO1 N1(C(c2n(C)c(S)nn2)=O)CC2CN(C(=O)Cn3cnnc3)CCC2(CO)C1 c1(C(N2C(C)CCC(CNC(c3c[nH]c(=N)o3)=O)C2)=O)ccc2nc(S)[nH]c2c1 N1(C(C2(CC=C)CCC2)=O)CC(NC(c2cc(Cl)sc2Cl)=O)CC(O)C1 c1(CC(=O)NC2(C)CCN(C(=O)Cn3cnc(C#N)n3)C2)cc(F)cc(Cl)c1 c1(CC(=O)NC(c2cn(Cc3ccncn3)nn2)CCC)nocc1C C1(C(N2CC(C)(CF)C2)=O)CC12CCN(C(=O)CC1CC3C=CC1C3)CC2 O=C(C1=CC2CCCC12)N1CCCC1C1(C(=O)NCc2ncccc2F)CC1 C1(C(=O)NC(C)CCN(C)C(C2(C)CSC2)=O)CCc2ccccc2O1 C#CCC(CC#C)C(=O)N1CC2=C(C1)CN(C(c1cccnc1S)=O)C2 Cc1ncncc1C(=O)NCCn1cc(C(=O)NC(c2cc[nH]n2)C)nn1 c1(C(=O)NC(C(C)C)CNC(c2cc(F)c[nH]2)=O)ccc2ccc(Br)cc2n1 c1(CCC(=O)NC(CNC(CCCC=C)=O)CO)cc(OC)cc(OC)c1 N(C(=NCC(C)c1cccc(C(F)(F)F)c1)N(C)Cc1ccon1)CCOC C1(O)(CCC(=O)N(CCCNC(C2CCN(C=O)C2)=O)CC)CCCOC1 C1(CC)CCCN(C(=O)CN(C)C(=O)C2CC2)C1.c1cccnc1.C(=O)C.N Cc1cc(CNC(=O)CC2C=CC(NC(=O)COCC=O)C2)no1.O C(=O)(C1CCCc2ncnn21)N1CC2OCC(NC(CN=S(C)(C)=O)=O)C2C1 c1(C(=O)NC(CCCNC(C2C(C)CCCC2)=O)(C)C)ccc(C#N)c(F)c1 C(=O)(C1CCCc2ncccc21)NC(C1(O)CN(c2ncncc2Br)C1)C C(=O)(C1c2ccoc2CCN1C(=O)OC(C)(C)C)N1CCc2n(C)nnc2CC1 C=CCCC(CC(C)C)C(=O)N(CCC(C)NC(=O)CN1CC(=O)N(C)C1=O)C Cc1cc(C(=O)NCC2(C)CC(NC(C3(C#N)CC3)=O)C2)c(C)nc1C N1(C(C(COC)O)=O)CC2(CCN(C(=O)C3=CC(C)(C)C3)C2)C1 C(=O)(CC(C)(O)COC)N(C1CCCN(C(c2cc(C)c(CC)o2)=O)C1)CC c1(CC(=O)NC2CC(CCNC(CCn3ncc(C)c3)=O)C2)c(C)noc1Cl C1(CC)CC(C(=O)NC2(CC3CC3)CC2)CCN1C(=O)C(=O)N(C)C Cc1cc(CN2CC3C(C(N4CCCCC4C#N)=O)C3C2)cc(C)n1 C1(NC(c2nccc(=NCC3(N(C)C)CCOCC3)[nH]2)C)CCCCCC1(F)F N1(C(CN=[N+]=[N-])=O)CC(O)CC1(C)C(=O)NCC(=O)NC1CC1 C(c1ccoc1)=CC(=O)NCCC1CCCN1C(=O)CC1CC1 C12(NC(C3CCC(C)N3C(=O)CN3CCCCCC3)=O)CCC(C1)OC2C C(=O)(C(C)(C)C(C1CC1)NCc1ncoc1C)OC Cc1cc(Cl)nc(Cl)c1-n1cc(C)nn1.C1(C(=O)N)(C(=O)O)COC(C)(C)C1 O=C1CC(C(=O)NCC2CN(CC3CCC4(CC3)CC4)C2)C2CCCCC2N1 CS(=O)(=O)CCC(=O)NC12COC(C1)C(NC(=O)C)C2.CCN(C)C.O N1(C(C2N(C)C(=O)OC2)=O)CCC(C)C(F)(F)CC1.C(=O)C(F)=C1CCC1.N c1(C(=O)NCCCN(C(c2nc[nH]c2C(F)(F)F)=O)CC)csc(C)c1 CC1(C)OCC2CC12C(=O)NC1(C2CCCN2C(c2cc(F)ccc2Cl)=O)CC1 CCC(C)(CNC(C1CCN(OC)CC1)=O)C(=O)NCC1=CCCC1 c1(CC(=O)NC2(CC)CCC2)ccnc(F)c1F.C(c1cccs1)=C(C(=O)N)F C1(C(C)NC(C2CCCC2)=O)CN(C(=O)C=Cc2ccsc2)CCO1 c1(C(N2CCN(C(C(C)Cn3ccnc3)=O)CC2)=O)ccc(Br)c(O)c1 C1(NC(c2n(C)ncc2C(F)F)=O)C2CCCC1CC(NC(c1ccco1)=O)C2 c1(N2CCC(CC(=O)N(C(C)C(N)=O)CC)C2)ncc(Cl)cc1F C#CCC(C(=O)N(C)Cc1ccncc1F)NC(C1CC1C(C)C)=O Cc1ccc(O)cc1CNC(C1CC(O)CCN1C(=O)C(F)CC1CCOC1)=O C1(NC(c2n(CC)nnc2)=O)CN(C(=O)CC2CCC3(CC3)CO2)CCC1C c1(C(N2CCC(NC(C(SC)SC)=O)C(C)C2)=O)nccc2ncccc12 c1(OC)ccc(CC(=O)NCCCCCN(C(=O)Cc2nnc(C)o2)C)c(F)c1 c1(C(C)C)[nH]nc(C(=O)N(CCCCCNC(c2ncccn2)=O)C)c1Br CCCC(CCCNC(c1ccc(C(C)(C)CC)cc1)=O)NC(=O)C(C)C(C)C CCC(C(=O)N1CC2C(CNC(=O)C=CC3CCCC3)C2C1)C(C)(F)F C(N=c1nc2scnc2c(NCC2CCCC2C)[nH]1)c1c(C)nccn1 C1(OC)CN(C(=O)CCCF)CCC1NC(c1sc(C2CC2)nc1C)=O C1(O)(C(=O)NC2C(C)N(C(=O)Cn3cnnc3)CCC2)CCCC(C)(C)CC1 C1(C(C)C)CCC(C)CC1C(=O)NCC1CCN(C(c2cccc(F)c2N)=O)C1 c1(OC)ccc(NC(=O)CC(C)CNC(c2ccc(C)o2)=O)c(C)c1 CC1CN(C(C2CC(n3ccnn3)C2)=O)CC1NC(c1cscn1)=O c12ccc(c(Cl)c1)CCNC2=O.N1(CC)CCC(N)(c2cccc(OC)c2)C1 N1(C(CC2(C=C)CC2)=O)CCN(C(=O)C(C)(C)n2cnnn2)CC1CS(C)(=O)=O C(CN=C(NCCc1csc(Cl)c1)NCc1ccc(F)cc1)c1c(C)cncc1 Cc1nc(N(C)CC2CCCN2C(c2cocn2)=O)c(C)c(O)n1 C#CC1CCCC(NC(C2COCCN2C(=O)C(O)C=CC)=O)C1 N1(C(C(C)CC(C)(C)C)=O)CCCC2(CCN(CCO)C2)C1 N1(C(C2C(C3(C)COC3)C2)=O)CCC2(CC(C=O)C2)C1.C1CC2CC1CC21CC1.N CCC(C(=O)NC(C1(O)CCN(C(=O)CS(=O)(=O)N(C)C)C1)C)C(C)(F)F Cc1nnccc1C(=O)NC(C1CCCCN1C(=O)CN(C)C1CC1)C C(=O)(C1CCCc2ccnn21)N(C1CN(C(c2ccccc2S(C)=O)=O)C1)C c1(CC(N2CCCC(C(C)NC(c3cc(C)nnc3)=O)C2)=O)ccc(O)c(Cl)c1 C1(C(=O)NCCN(CCC)C(C2CCC2)=O)C2CC1(c1cccnc1)CO2 c1(C(N2CCC(N(C(=O)CCSC(F)(F)F)CC)C2)=O)nc(C)sc1C C1(OC)CN(C(=O)CC2CC=CCC2)CC1NC(c1[nH]c(C)nc1C)=O C#CCC(C(=O)NCC12CC1CN(C(=O)C(c1ccc(O)cc1)=O)C2)C1CC1 C12(NC(c3nc(CC)sc3)=O)CCC1CN(C(=O)CC1(OC)CCOCC1)C2 C1(C(C)NC(c2nc(CC)sc2)=O)CCCN(C(=O)Cc2[nH]cnc2C)C1 N1(C(C(C)(C)OC)=O)CC2CCN(C(=O)CCc3cc(C)cc(C)c3)C2C1 c1(C(N2CCC(O)(C(C)NC(COCC)=O)C2)=O)cccc2ccnn12 c1(CNC(C2(NC(C3N(CC)CCOC3)=O)CC2)=O)ccc(C)nc1O c1ccc(C#N)cc1.c1(-c2n(CC)c(N3CCCCC3)nn2)cc(OC)nc(=N)[nH]1 C#CC(C)(C)C(=O)NC1CC(NC(C2C3COCC23)=O)C(O)C1 c1(C(=O)NC2CCN(C(c3c(CC)oc(C)c3)=O)CC2C)ccn2nncc2c1 C(N=c1ccn(CC(N2CCC(CO)CC2)=O)c(O)n1)c1cc(C)ncc1 c1(C(C)NCC#CC2CC2)cncc(F)c1 C1(COC)(NC(C2COCCO2)=O)CCN(C(=O)C(c2ccc(F)cc2)C)CC1 N1(C(c2cccc(C(=O)NC)c2)=O)CCC(NC(c2nncs2)=O)C2(CCC2)C1 c1(C(=O)O)ccc2[nH]cc(CN3CC4CCCCCC4C3)c2c1 N1(C(C(C=CC)O)=O)CCC(NC(C2(C)CCC(=O)NC2)=O)C(C)C1 CC(C)(C)CCCCCC(=O)NC1C=CC(CNC(C2CC23CCC3)=O)C1 C(=O)(C1=CCCCCC1)N1C(C(C)(C)NC(CN(S(N(C)C)(=O)=O)C)=O)CCC1 O=S(=O)(c1n[nH]c2ncccc12)N1CC2CC2C1 C1(C(=O)NC(c2ccccc2F)CC)C2CC1N(CC)C2C C1(CCCNC(c2c(C(C)C)nns2)=O)CN(C(=O)CCc2nccs2)CCO1 CCCC(C)CCCC(=O)NC1CN(C(=O)C(C)(C)NC(=O)C(F)(F)F)CC1C C(=O)(C1CCc2ccccc21)N1CC(NC(C(C2CC2)OC)=O)C2C1CCCC2 C(=O)(CC(F)(F)F)NC(C(=O)NC(c1ccccc1)C(=O)OCC)C Nc1c(C(=O)NC2CCCC(NC(c3cscc3F)=O)C2)cc(F)cc1Cl CC1CC(NC(=O)C(C)(C)C2CCC2)CCN1C(=O)C(c1ccccn1)O c1(OC)cc(C(=O)N(CC(C)N(C)C(c2[nH]nnc2C)=O)C)c(F)c(Cl)c1 C12(CNC(c3cc(Cl)n[nH]3)=O)CCC(CN(C(c3ccnc4c3CCO4)=O)C1)C2 C1(CCN(C)C(c2ncccn2)=O)CCN(C(=O)CC2CCCO2)CC1 Cc1cn2ccc(C(=O)NC3CCCC(NC(c4cncc(O)c4)=O)C3)cc2n1 N1(C(c2c(C)scn2)=O)CC2CC(NC(C3(C(C)(C)O)CC3)=O)C(C2)C1 c1(NCCN(CCOC)C)ccc([SH](=O)=O)cc1Cl.C1CCCC1C(N)=O.N c1(OC)cccc(C(C)CC(=O)N(CC(C)(C)O)C2CC2)c1 c1(NC)ccc(C(N2CCC(NC(=O)C=Cc3sccc3C)C2C)=O)cc1F c1(C(N2CC(OCCNC(C=C(C)C)=O)C2)=O)c(N)cc(Cl)nc1Cl C1(C(N(CCCCCC)CCN)=O)CCCN(C(=O)COCC(C)C)C1 C1(C(=O)NCC2(C(=O)NCC(O)COC)CC(=C)C2)CCCOC1C Cc1ccc(-n2cc(C(C)N(C)C(c3csc(-c4cnc[nH]4)n3)=O)nn2)cc1N c1(C(=O)NC(CC)CNC(c2cnn(C)c2F)=O)sc2cc(C)ccc2c1Cl c1(C(=O)NC2C(NC(c3cc(C)[nH]c3C)=O)C2)ncsc1S(N)(=O)=O C(=O)(C1CCc2ccccc21)N1CCCCC(C(=O)NC2C(CCOC)C2)C1 c1(C(=O)NCCN(C2CCN(C)CC2)CC)c(Cl)ccc(CO)c1Cl Cc1ncnc(O)c1CCC(N1CCCCC(NC(=O)C=C(Cl)Cl)C1)=O C1(C)(CC)C=C(C(=O)N(C2CCCCC2N(C)C(C2CCC2(F)F)=O)C)C1 CC(C)(C)CC(O)C(=O)N1CCN(C(c2ccc(O)nc2)=O)CC1CF C(=O)(C1=CCCCCC1)NC1CC(CNC(c2cnn(CC)c2Cl)=O)C1 Cc1cc(Cl)c(C(=O)NCC2COCCN(C(c3ccc(Cl)o3)=O)C2)cc1C C(=O)(CC(C(F)F)NC(c1nnn(C)c1C)=O)NC(C(=O)OCC)CC CCCCC(CNC(=O)CC1OCCC1(C)C)NC(=O)COC1CCCCC1C c1(C(N2C(C(=O)Nc3cc(SC)n[nH]3)CC(F)(F)C2)=O)cc(Br)c2cn[nH]c2c1 C1(CCNC(c2n(CC)ncc2)=O)CN(C(=O)C(C2CC2)SC)CCO1 C1(CC#C)(C(=O)OC)CCN(c2nccc(C3CCCCN3)n2)C1 C1(C(=O)NC23CC(F)(C2)C3)CC2(CCN1C(=O)CSC(F)(F)F)CC2 C(CC(C(=O)N(C)OCc1ccccc1)NC(=O)Cn1nnc(C)n1)=CC CCC(O)C(C)C(=O)N(C1CCN(C(c2cc(C)ncc2C)=O)CC1)CCOC CC1(C)CN(C(C2(F)CC=CC2)=O)CC1CNC(=O)C(Cl)=CCl C1(NC(C(=Cc2cccs2)C)=O)CCC(C(=O)NCc2cccs2)CC1 C(=O)(CCC(=O)N1C(C(=O)NC(CO)C(C)C)CC2CC12)NCCC CC1C(=O)CCC1CC(=O)N(O)Cc1cn(CCc2ccccc2)nn1 Cc1noc(C)c1C(C)(C)C(=O)NCC(O)CNC(=O)CC1CCC1 C(=O)(C1=CN=C2N=CNN2C1)N1C(CN(C(=O)CCc2ncc[nH]2)C)CCC1 c1(OCCCC(=O)NCC2CCN(C(C3C(C#C)C3)=O)C2)ccccc1Cl C1(NC(CC2C(C)(C)C2)=O)(CNC(=O)Cc2csc(Br)n2)CCCCC1 CCC(C(=O)NC1CN(C(c2cccc3nncn23)=O)C1)C(C)(F)F c1(C=O)cc(F)c(O)c(Br)c1.C1(OCC)CC1C(=O)N(CCC)CC.N N1(C(C(C)OC2CCCC2)=O)CC(CC(=O)NC)C2(CC2)C1.c1ccc(O)nc1 Cc1cc(=NC(=O)C2CCN(C(=O)CC(C)(C)C)CC2)[nH]o1 c1(N2CCN(CC)CC2)ccc(CO)cc1[N+](=O)[O-].c12ccc(nc1)NC(=O)N2 c1(C(=O)NCC(C)NC(c2c[nH]nc2C(C)(C)C)=O)ccccc1Br CC(=O)C(C)CC(C)C(=O)N1CC=CC1(C)C(=O)NC1(C)CCCCC1(C)C c1(C(=O)NCC(CN(C(C2ON=C(C)C2)=O)C)(C)C)cccc(CS(C)=O)c1 CC1OCCN(C(C2SCCS2)=O)C1C(=O)NCC1(CO)CC=CC1 S(=O)(=O)(C1CC2(CNC2)C1)Nc1cc(Br)cc(C)c1F N1(C(C(C)N(C(=O)CNC(=O)OC)CC)=O)CC2(C)CCC2(C)C1 c1(C(N2CC3(CCN(C(C4C5CC6C(C5)C46)=O)C3)C2)=O)ccn2c1CCCC2 C1(C(N2CC(CNC(C3C(C)(C)CCCC3)=O)C2)=O)CCCN2CCCC12 N1(C(C2CC=CCC2)=O)CCC12CN(C(=O)Cc1cc(O)cc(F)c1)C2.COC C(=O)(CC(F)(F)C(C)C)N1CCCC(CCNC(c2ccn(COC)n2)=O)C1 C1(C(=O)NC(CN(C(C(CC=C)NC(C)=O)=O)C)C)CC2C=CCC(C1)C2 c1(C(N2CCC(CCNC(C(CCCCC)O)=O)C2)=O)ncc([N+](=O)[O-])cc1C N1(c2cc(NCc3scc(COC)c3)ncn2)CCCCC(c2ccccc2)C1 CC(C)C(CN(C)C)C(=O)NC(C(=O)NC1CCC(O)CC1)C1CCC1 C1(NCCC2CCCC(C)(C)O2)(CO)CCS(=O)(=O)CC1 CN1C(=O)CSC1=CC(=O)NC12CCCN(C(C3(C#N)CC3)=O)CC1C2 N1(C(CCc2cnn(C)n2)=O)Cc2ccnn2CC(NC(c2ccc(Cl)s2)=O)C1 C1(NC(c2cn(CCC=C)nn2)=O)CCCN(C(=O)C=CCN(C)C)CC1 c1(CCC(=O)OC)ccc(NC(=O)NCCC(C)(C)F)cc1 N1(C(C=C(CCC)CCC)=O)CCN(C(=O)Cc2cc(C)nn2C)C2CCC12 c1(C(=O)NCC(CO)NC(C(CC=CC)C)=O)c(CO)nc2ccccn12 C1(NC(c2c(CC)con2)=O)CC2CCC(C1)N2C(c1cnoc1C(C)C)=O C(CC1CC1)(C(=O)NC(Cn1ccnn1)C(=O)N(C)Cc1cccs1)OC C(=O)(C1=CCCOCC1)NC1C(C(C)(C)C)N(C(=O)CCc2cnc(O)[nH]2)CC1 C(=O)(CC(C(F)(F)F)NC(=O)C(C1CCCCC1)=O)NC1(CCC)CCOC1 N1(C(c2ccc(C#C)s2)=O)CC2(CC2)CC1C(=O)NCCCS(N)(=O)=O C1(C(N(C2CC(NC(=O)Cn3ccc(Br)n3)C2)C)=O)C2CCC(=O)C12 CONC(=O)C(=O)NCC1(C(=O)NCC(C)(C)N(C)C)CC12CCC2 Cc1cccc(N)c1C(=O)NCC(C1CC1)NC(c1cc2n(n1)CCO2)=O N1(c2c3occ(C)c3ccc2)CCCC12CCN(Cc1ccccc1)C2 C1(C(N2CC(NC(=O)CCc3ccc(O)nn3)(CO)C2)=O)CCc2nncn2C1 c1(C(N2CCC(NC(C3C=CC(=O)N=N3)=O)C(F)C2)=O)ccc(O)c(O)c1O CC1(C)CC1CCC(=O)NC1(C2CCCO2)CC1 c1(C(C)N(C)C(c2cnn(CC3CC3)c2-c2ccccc2)=O)ccc(F)cc1 C1(NC(c2cc(OCC)n[nH]2)=O)C(C)CN(C(=O)C2=CCOC2)CC1C c1(OCc2c(C)ccc(F)c2)ccc(C#N)c(I)c1C N1(C(c2ccc(CC)s2)=O)CC(C)CC1C(N1CC(c2ccncc2)C1)=O C(CCC1CCC1)(C(=O)NCCC(O)C1CC1)NC(c1cn(C)nc1)=O C(c1ccc(C(F)(F)F)cc1)=C(C(=O)N)F.C=C1CCC1C(=O)NCCCC N1(C(C2COCCN(Cc3cnc(CC)nc3)C2)=O)CCC(=O)NCC1C C1(O)(C(N2CCN(CC#N)CC2)=O)CCN(C(=O)Cn2cnc(Br)n2)CC1 CC(C)(C)C(CNC(c1nc(Cl)cs1)=O)NC(=O)CCCCN1CCCC1 C(CCCC(=O)NC1CN(C(c2cnc(C3CC3)nc2)=O)CC1C(F)(F)F)OC C12(NC(c3ccnc(CO)c3)=O)CCCC1CN(C(C1(F)CCCC1)=O)C2 CC(O)C(C(=O)NCCN(C(=O)C(C)(C)C1CCCC1)C)N(C)C c1(C(N(C)CCNC(c2ccc(C(C)(C)C)[nH]2)=O)=O)c[nH]c(C#N)c1 C1(NC(C2(CC=C)CN(C(C3CC(F)C(=O)N3)=O)C2)=O)CCC(O)CC1 C#CCC(C)(CC)C(=O)NC(C1CC(NC(=O)CSC(F)F)C1)C N1(C(CC(C)CF)=O)CC(C)C2(CCC2)C1.C(=O)(CS(=O)(=O)Cc1cccs1)N c1(C=O)cc(C)ccn1.C(C(C)(C)C)N(C(C1(C(=O)OCC)CC1)=O)C N1(C(CC(CNC(Cc2n(C)ccc2)=O)O)=O)CC2CC1C(F)(F)C2 O=C(C(Cl)=CCl)NCC(c1ccccc1)NC(c1ccc(-c2cccs2)[nH]1)=O C(=O)(CC(C)(F)F)NC(CCN(C(C1N(CC)CC1)=O)C)C c1(OC)nc(N2CCCC(NC(=O)CCCCN3CCCC3)CC2)nc(C)c1F CC1CC(=O)NCC1C(N1CCCC(NC(=O)Cc2ccc(Cl)cn2)CC1)=O c1(NC(c2cccc(C(=O)OC)c2)c2n(CC=C)nnn2)ccc2nonc2c1 C(CC(N=c1cccc(S(=O)(=O)N(C)Cc2ccoc2)[nH]1)C(C)C)OC c1(C(N2CCCC2)=O)cc(F)ccc1C1CC1.c1(CC(C)C)cc(C(=O)N)no1 Cc1cnc2c(C(=O)N(C3CC3)CC3COCCO3)cccc2n1 CCCCCC(=O)NCC(=O)N(C)CC1CCN(c2nc(COC)ns2)C1 c1(CC(=O)NCC(C)NC(C23CCCN2CCC3)=O)coc2c(F)c(F)ccc12 C1(CCCC)CN(C(c2cc(SC)ccc2O)=O)CCN1C(=O)CCSCC C1(NC(C(Cc2ccc(C)cc2)C)=O)CCC2CN(Cc3cncs3)CC2C1 C1(C(=O)NCC(C)NC(=O)C(C)C)(C(C)C)CNC(=O)C1.c1ccccc1 c1(SCC)ccnc(NC(=O)CONC(C2CCC(C)(CC3CC3)C2)=O)c1 Cc1nc(CO)oc1C(N1CCC(O)(CCNC(C2(Cl)CC2(F)F)=O)C1)=O C1(OC)CC(CCNC(=O)CCCF)N(C(=O)Cc2ccnc(O)c2)C1 c1(NC(N(CC(C)(O)CN)C)=O)cc(C(F)(F)F)cc2c1OCC(=O)N2 c1(C(=O)NC2(C)CN(C(C#CC3(CC)COC3)=O)C2)ccc(Cl)c2occc12 C1(C(=O)NCC(CC=C)NC(c2occc2C(C)C)=O)COCCN1CC CC1CCN(S(=O)(=O)CC(=O)NCCC)CC1.C1(C=O)CC1(C)C(F)(F)F.N C=C1CN2C(=O)CCC2(C=O)C1.C1(C(N(CC)CCC)=O)CC1C(C)C.N c1(COC)cc(C(=O)N(CCC(C)NC(=O)CCC2CCCOC2)C)n(C)c1 C1(NC(c2c(CC)onc2)=O)CC1C1CCCN(C(=O)CCc2cn[nH]c2)C1 c1(C(=O)NCCCCCN(C(C2C(=C)C2)=O)C)ccc(C(F)F)c(OC)c1 C1(NC(C2N(C(c3cc(C(N)=O)ncc3)=O)C3C(C2)C3)=O)CCC=CCCC1 N1(C(CC(=C)C)=O)CCCC(N(C(=O)CC2SC(=N)NC2=O)CCO)C1 c1(OC)cc(C=O)ccn1.C1(O)(CC)CN(C(=O)C)C1.c1(C=O)ccco1.N C1(C)(C(=O)N)COC(=O)C1.C1(C(N(CCC)CC)=O)CCC(C(N)=O)C1 CCCC(C(O)C(=O)N1CC(C(C)(C)C#N)C1)NC(C1CC(=O)N(CC)C1)=O c1(C(=O)NC2CN(C(Cc3c(C)scc3)=O)CC2C)cc2c(Cl)cncc2s1 C(=O)(C1=NNC(=O)CC1)N1CC(NC(=O)C(=O)N)CC(OC)C1.C1CC1.C N1(C(CCc2n(C)cnn2)=O)CC(=O)NCC1C(=O)NC1CC2(CCC2)C1O Cc1cc(=NC(=O)C2CC3(CCN(C(C4(CO)CCCC4)=O)C3)C2)[nH]n1C1CC1 C#CCCCC(C)C(=O)NC(CCCC)C(=O)N1CC2(CC2)CC1C c1(NC(C2C(O)CCN(C(CCC(=O)OC)=O)C2)=O)cc(F)c(Br)cc1[N+](=O)[O-] c1(C(=O)NCC(CN(C(C(C)SCC)=O)C)O)cn(C(C)(C)C)cn1 N1(C(CC(CC)O)=O)CC(NC(c2ccn(C3CC3)c2C)=O)C2(CCOCC2)C1 C#Cc1cccc(C(=O)NC2CC(NC(=O)C=CC3CCC3)C2)c1Cl Cc1cc(C)nc(N2CCC2)n1.C(=O)CCSC(F)(F)F.CC.C(=O)C1CC1.O CC(CC(=O)NC(CNC(C12CCC(CC1)OC2)=O)CC(F)(F)F)C(F)(F)F CCCCCCCCOCC(=O)NC1COCCN1C(=O)C1=NOC(C)C1 c1(N2CCC(CF)C2)nc(=NCCC2CC3CCC2O3)[nH]c2c1CCCCCC2 N1(C(CS(CCC)(=O)=O)=O)CC2(C)CN(C(=O)Cc3sc(C)nc3C)CC2(C)C1 c1(CC)ncnc(CC)c1C(=O)NCCC(C)(C)NC(=O)CCCC.C(N)=O CC1(C)C(CO)CN1C(=O)CCN(C(=O)C(N)=O)CC1CC1 CN1C2CCC1CC(NC(C13CC(CO)(CN1C(C1(CO)CC1)=O)C3)=O)C2 c1(C(=O)NCCCN(C(C2CCC2)=O)C2CC2)c[nH]nc1-n1cnnn1.C C=CCC(C(=O)N1CCC1C)NC(C)=O.C(=O)C(C(C)C)c1cnc(C)s1.N C(c1nc(C)co1)=CC(=O)N(CC(C)NC(=O)CCN(C)CCO)CC c1(C(=O)NC(CC)CNC(c2oc(C(F)F)cc2C)=O)ccc(Br)cc1NC C(=O)(CCCC(=O)N1CCN(C(c2ncoc2C2CCCCC2)=O)CC1)OC C(=O)(C(C#N)C(C)(C)C)N(CC)C1CC1.c1(C(C)(F)F)n[nH]cc1C=O.N c1(C(N2CCC(N(C(CC(C)N(C)C)=O)CCO)C2)=O)ccn2c(O)nnc2c1 Cc1csc(=NCC(=O)N2CCCC(NC(c3cccc4ccccc34)=O)C2)[nH]1 CC1CN(C(c2cnn(C)c(=O)c2)=O)CCN1C(=O)C(F)n1ccnc1 Cc1cc(NC2CC2)ncc1S(=O)(=O)N1CCCN(C(C)CO)CC1 CC(C)CC(F)C(=O)NC(CNC(C1(O)CCSCC1)=O)C(C)(C)C CS(=N)(=O)c1cnc(N2CCN(C(N)=O)CC2)nc1 c1(C(=O)NCC(c2ccc(C)cc2)NC(C2(C#N)CCC2)=O)ccc(C)nc1C C1(C(=O)NCCN(C)CC)COCCN(C(=O)C(c2cccc(Br)c2)(C)C)C1 [SH](=O)(=O)c1c(F)cccc1F.C1(C(=O)N)(OC)CCC1.C1CCN1C(=O)C CC(C)CC(C)CC(=O)N1CC(NC(c2cccn2C(C)C)=O)CC(F)(F)C1 CC1(C)CC(CO)(CNC(C2CCC(=O)C2)=O)C1 c1(C(N2CCN(CCC)CC2)=O)sc(=NCc2c(F)cccc2I)[nH]c1C N1(C(CC(C)(C)CNC(C2CCC2(F)F)=O)=O)CCC(C#N)CC12CC2 c1(C(=O)OCC)c[nH]c(=NCC2(C)CCN(C(C3CC3CO)=O)C2)cn1 C(C(C)(C)CC(=O)NCC1C=CCN1C(C1CCS(=O)(=O)CC1)=O)N(C)C CC(C)C(C(c1nnnn1CC1CC1)NC1COCC1n1ccnc1)C(C)C S(=O)(=O)(c1cnccc1N(C)CCO)NC(c1ccc2c(c1)CCO2)C C1(CCCC)CN(C(C2CCCC(CF)C2)=O)CCN1C(=O)C1=CCCCO1 C1(C(=O)NCC2(OC)CCN(C(c3[nH]cnc3C)=O)C2)CCN(C)S1(=O)=O c1(-n2ccc(C(=O)N)n2)c(F)cccc1F.O=C(CCC1CC1(Cl)Cl)NC1CC1 C#CCC(C)(C(=O)N1CCOC(CF)C1)NC(=O)CCC1CCOC1 N1(c2nc(C)c(F)cn2)CCC2(CCN(c3ncnc4c(Br)c[nH]c34)C2)C1 CCC(C)C(C)C(=O)NC1CN(C(c2ccoc2C)=O)CC1C CC(C(C(=O)NCCC1CC1)N(C1CCCCC1C)C)C1CCCOC1 C1(CNC(N2CC(CCCOCC)C2)=O)CC2CCC1CC2 C(CS(=O)c1ccc(CC(=O)NC)cc1)OC.C1C=CCN1C(=O)CCC1CC1 c1(C(N2CCCC(C)C2CNC(c2cncs2)=O)=O)ccc2nc(O)n(C)c2c1 C(C)(C(=O)N(CC(CC)NC(=O)Cn1cnnn1)CC)=CC C1(NC(=O)C=C2CCC2)C2CCN(C(C3CCN(CC(F)(F)F)CC3)=O)C12 c1(C(=O)NC(CN(C)C(c2ccn(CC(F)(F)F)n2)=O)(C)C)ccc[n+]([O-])c1 C1(C(C)(C)C)(C(=O)OC)CN(N2CCCC(C)(C(=O)OC(C)(C)C)C2)C1 N1(C(CC2=NNC(=O)C2)=O)CC2CCCC(C1)N2C(=O)CC1CCCCC1O N1(C(CC2CC(C)C2)=O)CCOC(CNC(=O)CCc2cccnc2F)C1 CC(C)(C#CC(=O)NCc1ccc(Cl)cn1)CNC(=O)CN1CCC(F)CC1 C12(C(=O)N)CCN(CC1)CC2.C1(NC(=O)CCC2CCC2)(C)CC(F)(F)C1 c1(C(N(CCCNC(C2CCC2(F)F)=O)C)=O)cc2c(cnn2C)nc1O Cc1ccc2c(=NCc3nc(C)ccc3C)[nH]c(=NC3C=CCCCC3)[nH]c2c1 N1(C(C(CC)C)=O)CC2(CC2)CC1CNC(=O)CO.C1CN(C(C)=O)C1 c1ccc(F)nc1.O=C(CCc1cn[nH]c1)NCC1(CCNC(=O)C)CC1 c1(CNC2CC(CC(=O)Nc3c(C)cccc3Br)C2)cc(F)cc(C)c1O C(CC(C)(C)CNC(=O)Cc1ccccc1C)NC(c1cc(CC)no1)=O CC(C)C(C(=O)NCC1(CC(=O)N(CC(F)F)CC(C)O)CC1)C1CCC1 C(N=c1[nH]nc(C2CC2)o1)c1c(C)c(C2CC2)on1 Cc1cc(O)ccc1CN(C(=O)COC1(C)CCCC1)C N1(C(c2n(CCC)ncc2)=O)CCC(CC(C)NC(c2oc(C)cc2C)=O)CC1 C1(C(N(C(C(=O)NCC=CCCC)C)CC)=O)CC2CCC1C2 C1CCC2(CC2)C(CN=C(NCC2CCCCC2)NC2CN(C3CC3)C2)C1 c1(CSC)ccc(C(=O)NC2CN(C(C3(n4cccn4)CC3)=O)CC2O)cc1 C(=O)(C(C)(O)c1ccccc1)N(CCCCNC(=O)CCc1cscn1)C Cc1cnc(C(=O)NCC2(O)CCCCC2)c(Cl)c1 N1(C(=O)OC(C)(C)C)CCC(C2CCN(C(c3ccc4c(c3)OCC4)=O)C2)CC1 c1(C(N2C(CNC(c3c(Cl)cn(C)n3)=O)CC2)=O)cc(CN)cc2ccccc12 c1(OC)ccc(S(=O)(=O)N2CC(NC(c3ccsc3)=O)C3(CC3)C2)cc1F C(CCCC(=O)NCCCCC1CN(C(C23CCC2C3)=O)C1)OC c1(C(N(C2CCCN(C(=O)C(O)CC3CCCC3)C2)C)=O)cc2c(s1)CCC2 C1(C(N(C)CC2COC(=O)N2)=O)CN(C(=O)Cc2cnsc2)CC12CCC2 n1(CCC)nccc1C(=O)NCC(CNC(c1ccc(C(C)=O)[nH]1)=O)CO Cc1cc(Cl)cc(C)c1C(=O)N.C1CC(C)CCN1C(C1CCC(C)(C)O1)=O.C c1(C(=O)NCC2N(C(c3ncn(C)n3)=O)CCOC2)ccc(S(N)(=O)=O)o1 c1(CN2CCC(O)(C(=O)Nc3ccc(SC(F)(F)F)cc3)C2)cnc2cc[nH]c2c1 C12(C(=O)NCC(CN(C(=O)CCc3cn[nH]c3)C)O)CCCN(CCC1)C2 C(=O)(C(CO)C(C)(C)C)N.C1(CC=C)CCN(C(c2cc(CCC)n(C)n2)=O)C1 C1(OCC)CCC(OCC(C(=O)N2CCOCC2)n2cc(CO)nn2)CC1 N1(C(CCCOC(C)C)=O)CCCC2(CCN(C(C3COCCN3C)=O)CC2)C1 CCC(C)C(C)C(=O)N1CCN(CCCNC(=O)Cc2ccccc2Cl)CC1 C1(NC(CCNC(=O)Cn2ncccc2=O)=O)CCC2(CCCC2)C1 c1(C(=O)N)cc(C(F)(F)F)cnc1N.c1(OCC)sccc1C(N1CCC1)=O C(=O)(C1=CS(=O)(=O)CCC1)N1CCCC(C)(CNC(C2CCOC2)=O)C1 c1(CC)oc(C(=O)NC2(C(=O)NC3CC3C(F)(F)F)CC2C)cc1C C1(C(F)(F)F)(C(=O)OC)CCCN(Cc2cc(-c3nn[nH]n3)c(C)o2)C1 C1(C(N(CC(=O)NCC(C(CC)C)C)C)=O)C2CCCC(=O)C12.C1CC1 C1(CC(N2C(C)(CC(=O)N(C3C(C)CC3)C)CC2)=O)CCOC1(C)C c1(CN(CC(C2CC2(F)F)OC)CCOC)ccccc1 c1(C(N2CCC(NC(C3COCCO3)=O)C2)=O)cc(F)cc2ccccc12 C(=O)(C1=CCC(NC(c2ccco2)=O)C1)NC1CCN(C(N)=O)C1 C1(F)(CNC(CCC2CCCN(C)C2)=O)CCN(C(C23CC(F)(C2)C3)=O)CC1 c1(CC)cnc(C(N2CCCC2CCNC(=O)C)=O)nc1.c1cccc(Cl)c1.O N1(C(C(CCF)NC(CC(C)n2cccc2)=O)=O)CC2C3CCC(C3)C12 C(=O)(C(C(C)(C)C)NC(C1CCCC(OC)C1)=O)NC(c1nn[nH]n1)CC c1(C(N2CCN(C(C(F)=C(C)C)=O)C3C2C3)=O)cc(C)c(C#N)c(C)c1 CCCC(C)(O)CC(=O)N1CC(CCCCNC(=O)CCCC(=O)NC(C)C)C1 C(CN=c1cc(C)nc[nH]1)OCCN(C(C(C(C)C)OCC)=O)C CCCCC(C)C(=O)N1CCOC(CNC(C2CC3(CCC3O)C2)=O)C1 N1(C(CSCCCC)=O)CCC(C2CC2)(NC(C2CC(C)(C)OC2(C)C)=O)C1 c1(OC)cc(C(c2nnnn2CCC2CC2)NCC2C=CCC2)cc(Cl)c1 N1(C(C(CSC)OC)=O)CCC2CCN(C(c3c(C)nsc3Cl)=O)CC12 N1(C(CSSC)=O)CCCC(C2CCCCN2C(=O)C(=Cc2cccnc2)C)C1 C1(C(C)NC(C2CC(=C)C2)=O)CCCN(C(c2cc(-c3ccccc3)ns2)=O)C1 CC1(C)CC(CC(N2CCC(C(C)(C)NC(C3CC(CCO)C3)=O)C2)=O)NC1=O C1(C(N(CC(C)NC(c2cc(-c3cccnc3)on2)=O)C)=O)COC(=O)N1 C1(C(N2CCC(C(N3CCCC3)=O)(C(C)C)C2)=O)CN2CCCC1C2.CC(C)N CCC(CC)CC(=O)NCC1CC1NC(c1ccccc1)=O.[nH]1cc(Cl)cn1.C c1(NC(C)=O)cccc(Cl)c1C1CCN(C2CCN(C3CCCCC3C)CC2)C1 c1(C(C)=O)cc(C(N2CC3CC3(NC(=O)C=C(Cl)Cl)C2)=O)ccc1C C(=O)(CCNC(=O)CSC(C)(C)C)N(C(C)CO)C1CC1 N1(C(C2CC(C)CC(C)C2)=O)CCC(C2(NC(C3CCC(C)(O)CC3)=O)CC2)C1 CCCCCC(C)(C)C(=O)OC1CCC(C)CC1 c1(CC)cncc(C(C(=O)NCC(F)F)N(CC(=O)N(CC)CC)C)c1 C(=O)(C1=C(C#N)CCC1)NCCCNC(c1c(C)cnnc1)=O C(=O)(C1c2ccccc2OCC1C)N1CCC(CCNC(CCCOC)=O)CC1 Cc1cc(C)c2c(C)c(C(=O)N(C3COCC3O)C)[nH]c2c1 C1(C(N(CCCC)C2CC2)=O)CCCCN(C(c2cnc(NC)s2)=O)C1 N1(C(C2CCC(=O)C2)=O)CCC(CF)(NC(=O)CCCc2cccc(Cl)c2)C1 N1(C(C2C(C=C)CC2)=O)CC2(CCCC2NC(=O)CSc2ccc(F)cc2)C1 C(=O)(C1=NNC(=O)CC1)N1CC2CC2C1.c1(CCOCC)nc(C=O)co1.N C(=O)(CCC(=O)NCC(c1ccc(F)cc1)NC(C1CCCC1C)=O)NC c1(N2Cc3c(cc(Br)s3)C2)nc(=NCC2COCCO2)[nH]c2c1CCCC2 C(=O)(C#CC1(C)CN(C(=O)OC(C)(C)C)C1)NCCSC(CCC)(C)C C(CCCCC(=O)N(C1CCC(O)CC1)C)NC(C(C1CCOCC1)C)=O N1(C(c2cc(CC)[nH]n2)=O)CCC(F)(CNC(c2ccsc2OC)=O)C1 N1(c2n(CCCN=c3[nH]ccc(Br)c3)nnn2)CCC2(Cc3ccccc3C2)C1 N1(c2n(C)nnn2)CCC(NC(=O)Cn2nccn2)C(CO)CC1 C1(C)(CNc2ccnc(N(C)Cc3ccc(CO)cc3)n2)CCOC2(CCC2)C1 C(CC)(CC)(CCO)NC(c1cccc(F)n1)c1n(CCCC)nnn1 N1(C(c2cn(CCC)nn2)=O)CCCC2C1CCCN2C(=O)C=CC1CCCC1 Cc1cnc(CC(=O)N(C2CCCC2)CCNC(C2(F)CC2C)=O)s1 CC1C(=O)N(C)C(C)C(C)N1C(=O)Cc1cn2ccsc2n1 N1(C(C2C(C(N)=O)C2)=O)CCC2(CC2)CC1C(=O)N(C1CC2CCC1CC2)N C(CN=c1nc2c(ncn2C)c(NCC2CC(F)C2)[nH]1)NC(=O)NC C(C(=O)NC1CCCC(CC(=O)NCC2CC(CF)C2)C1)(C(C)C)OC c1(C)cc2n(n1)CCCC2O.C1(CC(=O)N(C(C)C)CC)C=CS(=O)(=O)C1 c1(C(N2CCN(C(C=C3CCC(C)C3)=O)C(C)C2)=O)cn2ccc(F)cc2n1 CC1(C)CCC1CC(=O)NCC(O)CNC(=O)CCCc1cccs1 C1(NC(CC(C)(C)O)=O)CCN(C(c2c[nH]ccc2=N)=O)CC(O)C1 C(CC)(CCC(=O)N1CCC(O)C1(C)C)NC(COCCCC)=O C1(NC(CC(c2cccc(F)c2)C)=O)CC2CCC(C1F)N2C(C1(F)CCC1)=O Cc1nccnc1C(C)NC(C1(C(C)NC(=O)C(C)CC2CC2)CC1)=O C1(C(N2C(CC(C)O)CCC2)=O)(CNC(=O)CCc2nccn2C)CCCCC1 C(=O)(CCCCC(C)CC)N(CCC)CCNC(C12CCCCN1CCC2)=O C1(CCC)CN(C(C2CC(O)(CNC(c3cc[nH]c3CC)=O)C2)=O)CCO1 N1(C(c2nnn(CC)c2C)=O)CC(CO)C2(C1)CN(C(=O)CCCC(C)=O)C2 C12(C3CC4CC(C3)CC1C4)c1c(C#N)c(ccn1)N2.C(C(F)(F)F)OCCO c1(N2CC3CN(Cc4ccc(C)nc4Br)C3C2)ncnc2occc12 c1(OC)cc(-c2cn(CC3COCCN3C(=O)COC3CC3)nn2)cc(Cl)c1 CCCCC(C)(F)C(=O)NC1CC2(C1)CN(C(C1(C)CCC3CC3C1)=O)C2 C1(CNC(CC2C(CC)C2)=O)CCN(C(c2cnnn2C2CC2)=O)CC1.C c1(CC(CC)Nc2ccc(CC(C)N(C)C)cc2)ccc(Cl)cc1 C(=O)(C(C#N)C(C)C)N(C1CCCN(C(=O)Cc2cc(Cl)cs2)C1)CC N1(C(c2c(N)cc(Cl)cc2)=O)CCCC2CN(C(=O)CCCCC(F)F)CCC12 CC(c1ccccc1)=CC(N1CC(C)(NC(C2CC(C)(C)CO2)=O)C1)=O c1(CC)nccnc1C(N1CCCC(CCNC(C2CC2c2cncs2)=O)C1)=O c1(C(=O)NCCC(C)NC(CCNC(C)=O)=O)ccc2scnc2c1 c1(C(N2C(CNC(C3C=CCC3)=O)CC2)=O)cc(O)nc(C2CCOCC2)n1 c1(N2CCN(CCSC)CC2)[nH]c(=NC2CCCN(CCCO)C2)nc2scnc12 C#CCCCCCCC(=O)NCC1CN(C(c2ncncc2Cl)=O)CC1C Cc1cc(F)c2cc(C(=O)NC3CC(N(C)C(C4CCC(C)O4)=O)C3)[nH]c2c1 Cc1cc(C(=O)N(CC(C)NC(=O)C(C)(C)n2cc(Br)cn2)C)cs1 c1(CCC)nc(C(=O)NC(C)CC2CCCCC2)cs1.c1(C=O)cnc(S)[nH]1.N C1(n2cc(C(C)(C)C(N)=O)nn2)CCCN(C(=O)C(C)(O)C2CCCCC2)CC1 CCC(CC(C)C)C(=O)N1CCN(C(=O)Cc2cncn2C2CC2)CC1CC C1(C(N2CC(NC(=O)Cn3cnnc3O)CC(C)C2)=O)CCCCC1C1CC1 N1(C(=O)Nc2sc(C(=O)OC)c(-c3ccccc3)n2)CC(CO)CC1(C)C c1(C(C(=O)N(CC(=O)N(C(C#C)(C)C2CCC2)C(C)=O)C)F)ccccc1 CN1c2ccc(C(=O)OCC(=O)CCCS(C)(=O)=O)cc2C(C)(C)S1(=O)=O C12(NC(C(C)NC(N)=O)=O)CCCCC1CN(C(c1cnc3ncccn13)=O)C2 c1(C(=O)OCc2cccc(-c3ccncc3)c2)cc2c(O)cccc2[nH]1 CC(C)C(Cc1ccccc1)C(=O)N1CC(C(C)NC(=O)CC2CCCC2C)C1 c1(C(=O)NC(C)CN(C)C(c2scnc2Cl)=O)ccc(P(C)(C)=O)nc1 c1(C(=O)NCC(CC=C)NC(C2(OC)CC2)=O)ccc(C)nn1 c1(CC(N2CC(C)(CCC(N3CC4CC4(CO)C3)=O)C2)=O)ccc(O)cn1 c1(C(N(C)CC2(O)CN(C(C(=O)NCCOC)=O)C2)=O)scnc1Cl.O C1(C(N(CCCO)C)=O)CCN(C(C2CC(C)(C)CCO2)=O)CC1(C)C C1(C#N)(C(=O)NCCCCC(C)NC(=O)CO)CCCC(=O)C1.C1CCCO1 c1(OC)ccc(C(O)C(=O)N(CC(C)(C)NC(=O)CC(C)F)C)cc1 c1(C(=O)NC(CCC)CNC(c2ccccc2)=O)nnn2ccccc12 C1(C(=O)NCCNC(c2[nH]cc(C)c2)=O)Cc2cc(C)c(C)cc2O1 CC(C)C(CC1CCCCC1)C(=O)NC(CO)C(C)NC(=O)CO.c1cn[nH]c1 C(C1COc2ccccc21)NC(=O)CCn1cc(C2CC23CC3)nn1 C1(C(=O)NC(c2ccncc2)CC)CCN(C(=O)Cc2nccs2)C1C C(CC(C)CCNC(c1cnc(CCCC)s1)=O)NC(CCC=CC)=O Cc1cc(C=CC(N2CCN(C(=O)C(C)OC3COC3)CC(O)C2)=O)ccc1F c1(CC)cccc(C(N2CCN(C(=O)CC3CCC(C(F)(F)F)O3)CC2C)=O)c1N N1(C(C(CC)=CCCC)=O)CC2CCC(CNC(C3CC3C3CCCC3)=O)C2C1 C(C(N=[N+]=[N-])C(=O)NCCC(=O)N(CCCCO)C(C)C)OCC CC(C)C(CCNC(=O)CC1CSCCS1)NC(C1C(c2ccccc2)C1C)=O O=S(=O)(c1ccc(NC2CCCn3nccc32)cc1Cl)NC1CC2C(C1)C2(F)F c1(C(=O)NCC(N(C(C(C)OCCC=C)=O)C)C2CC2)cn2ccsc2n1 c1(C(N2CCC(CC)C2)=O)cc(F)c(N)c(F)c1.C(=O)C(C(C)(C)C)N(C)C N1(C(CC(=C)C)=O)C2CCC1CC(NC(c1ccc(OC(F)(F)Cl)cc1)=O)C2 C1(O)(CN(C(c2c(C)[nH]c(=N)s2)=O)C)CCCN(C(C2CC2[N+](=O)[O-])=O)C1 c1(C(N2CC(C(C)NC(C3(C)COCCO3)=O)C2)=O)cc(O)nc(N(C)C)n1 c1(OC)cc(C(=O)N(C)Cc2ncnn2C)cc(N)c1O C(=O)(C#CC(C)(C)CNC(=O)Cn1cnnc1O)Nc1c(CC)onc1C c1(C=O)ccc2c(c1)CC(=O)NC2.C=C=C(C)CC(=O)NCC1COC(C)C1 C12(C(=O)NCC3(C)CCN(C(C4(C)CC4)=O)C3)CCCC1CCC2.C1CCC1 N1(C(C2C(C=C)C2)=O)CCC2(CC1)CC2.C1(CC=O)CCCCC1.C(=O)(C)N N1(C(C=CCCC(C)C)=O)CCC(CN(C(=O)CCCc2ccncc2)C)CC1 Cc1cc(-c2nc(-c3ccc(SC(F)F)nc3)n(CC3CCCOC3)n2)c(C)o1 C1(CNC(C(N2CCCCC2)C)=O)CCOC1C(=O)NCC1(C#N)CCC1 c1(NC(C2OCCN(C(C3CN(C)C3)=O)C2)=O)cc(Cl)cnc1O CCCC(CC)C(=O)NC(CCN(C)C)C(=O)N(C1CSC1)C c1cc(C)c([N+](=O)[O-])cc1C#N.N1(C(C2CC(OC)C2)=O)CCCC(C)C1CN C(=O)(C(CC(C)C)NS(=O)(=O)c1cccs1)NCCCCNC(C(CC)CC)=O c1(N(CC(CNC(C(CC)N(C)C)=O)C)C)nc(O)c2c(ncn2C)n1 c1(OC)ccc(CC(O)C(=O)NCCCN(C)C(c2sccc2SC)=O)cc1 C1(CNC(C(C)N(C)C)=O)CC(F)(F)CN1C(=O)CCc1cccnc1 C(CN=C(NCC1CN2CCCC2CO1)N1CCC(CC(F)(F)F)CC1)OC N1(C(C=CC=CC)=O)CC2CC(NC(C3(C)CCOC3)=O)CC(C2)C1.O c1(CCCC=O)ccc(F)cc1.c1(C(=O)NC)conc1C.c1ccccc1.N N1(C(C(C)NC(CC)(C)C)=O)CCC(C(N2CCC=C(Cl)C2)=O)CC1(C)C C1(O)(CC=O)CCCCC1.n1(CC)ccnn1.C1(C(C)(F)F)(C=O)CC1.C C1(C(=O)NC(C)CN2CCCC2=O)CN(C(=O)CSCC(F)F)CC12CC2 C1(C(=O)NC2(CCCC(=O)NCC(CC)CC)CCC2)CC(=O)NC(C)C1 S(=O)(=O)(c1ccc(C)c(NC2CCOCC2OCCCC)c1)N C1(C(=O)OC)CC(F)(CNC(=O)NCC(C)C(C)O)C1 C1(N(C(Cc2c(C)n[nH]c2)=O)C)CN(C(c2nn(C)cc2Cl)=O)CC1(C)C c1(C(N2CCCC(C3(C)OCCO3)C2)=O)ccc2c(c1)C(=O)CCN2 CCC(C)(CNC(=O)CCc1ccsc1)NC(c1coc(C2CCCCC2)n1)=O c1(CN2CC3N(C(Cc4cc(C)on4)=O)C(C3)C2)cc(F)c(F)cc1O c1(CN2CCC(C)(C(N3CCCC(C(=O)OC)C3)=O)CC2)cc(F)cc(F)c1O CCCCCCNC(=O)C(C)OCC(N)=O.c1(C(=O)N)ccc(OC(F)F)cc1 N1(C(Cc2nc(C)sc2)=O)CCCCCCC1C(=O)NCCCS(N)(=O)=O C1(c2onc(C)n2)CC(O)CN1C(C1CNCCC1c1ccc(F)cc1)=O C=C=CCCC(=O)NC1CCC1NC(c1cc(-c2ccccc2OC)on1)=O c1(C(=O)NCC2(NC(=O)Cc3nnc(O)s3)CCC2)cnc2[nH]cncc1-2 O=C1CCC(NC(=O)N(C2CC2)Cc2cccc(Br)c2)C(=O)N1 N1(CC(N2CC(OC)C(F)C2)=O)CCN(C(c2ncccn2)=O)CC1=O N1(C(CCN(C(C)C)C(c2c[nH]c(=O)cn2)=O)=O)CCC2CN(C)CC12 N1(C(C(C(C)C)CNC(=O)CN2CCCCC2C)=O)CC(O)C(N=[N+]=[N-])C1 CCC(F)(F)CC(=O)N1CC(F)CC1CNC(c1cc(C)n(C2CC2)n1)=O c1(C(=O)NCC2CC(OC)CN2C(c2snnc2C)=O)cnn(C)c1C#N CC(C)(C)C(C(=O)N)NC(C1CCCN1C(N)=O)=O.C12CC(CCO1)C2.C CC(C)CS(=O)(=O)CC(=O)NCC1CCN1C(=O)CC1CCCC1O N1(C(c2cccc(C(F)(F)F)c2)=O)CCc2sc(-c3c(O)cccc3F)nc2C1 c1(-c2cc(C(N(CC(O)CNC(C3COC3)=O)C)=O)on2)ccccc1Cl Cc1nc(NCC2CCC2)c2c3c(sc2n1)CCC3.N1(CC=O)CCN(C)CC1.N c1(C(C)C)ncc(C(N2CC(NC(=O)C(C)(C)c3cccs3)C(C)C2)=O)n1C C1(C(N2CC(C(C(=O)N(C3(C)CCCC3)C)OC)C2)=O)(CC)CNC(=O)C1 C1(CC(N2CC(CNC(C=CSC)=O)C3(C2)CC3)=O)CCn2cncc2C1 CC(C)(C)CCCCC(=O)NCCCCCCC(=O)N1CCC1C1CCC1 Cc1noc2ncc(C(=O)NCC(O)CNC(C3CCCCC3CO)=O)cc12 n1(CC)cc(Cl)c(C(N2CCC(C)C2CNC(C2(CCF)CC2)=O)=O)n1 C(C(C)(C)CC(=O)N1CC(C(=O)Nc2ccccc2C(C)C)C(C)C1)OC C1(C(N2CC(CCC)N(C)CC2)=O)CC12CCN(CCC(=O)OCC)CC2 C=CCCCCCCC(=O)NCCCCN(C(=O)CCC(CC)OC)C N1(C(Cc2n(C)c(S)nn2)=O)CC2COCCC2(NC(c2ncc(F)cn2)=O)C1 c1(C(=O)NC(C2CCCN2C(C2(Sc3ccccc3)CC2)=O)C)cccnc1S Cn1cc([N+](=O)[O-])cc1C(N1CCC2(NC(=O)C(F)CC3CCOC3)CC2C1)=O C1(NC(CC(C(F)F)NC(C(C(C)C)C)=O)=O)CC2CC1OC(=O)N2 N1(C(c2cc(CC)n(C)n2)=O)CC(C2CCN(C(C3CCOC3=O)=O)CC2)C1 c1(C(N(C2CCN(C(C3CC(OC)C3)=O)C2)CCO)=O)c[nH]c2nc(F)ccc12 CC1CN(C(=O)COc2cccnc2)CCC1C.C1(CC=O)(N(C)C)CCC1 Cc1ccc(CC(N2CCCCC2CNC(C2CCCCNC2=O)=O)=O)c(Cl)c1 CCCCC(=O)C(=O)N1CCCC1C(C)(C)C(=O)NCC(C)Cn1cccn1 c1(-c2cn(CCCC(=O)NC(c3ncoc3CN)C)nn2)ccc2n[nH]cc2c1 N1(C(CSC(C)C)=O)Cc2[nH]nc(C(=O)NCc3nc(N(C)C)no3)c2C1 n1(CCC)nnnc1C(c1nscc1Br)NCc1ccc(C(N)=O)o1 c1(OC)ncc(C=O)c(C(F)F)n1.C1CN(C(c2cnsn2)=O)CC1C(F)F.N c1(C(=O)NCC(C(=O)NCC(C)F)O)csc(C#N)c1 CC1CCCCC1n1nc(-c2ccncc2)nc1-c1ccc(CO)o1 c1(C(=O)N)ccc(C)c(C)c1Cl.C1(CC)CN(C(=O)CC2(OC)CCC2)CCC1 c1(C(=O)NCCCNC(=O)CC2CCCS(=O)(=O)C2)ccnc2c1CCO2 C(CCCCC(=O)N1CCC(CCCO)C1)N(C(CC(=O)N(C)C)=O)C c1(C(=O)NCCN(C(=O)CC)CCC)cc2ccc(C)cn2c1.CC(F)(F)F N1(C(C)=O)CCCCC1C1CC1.N1(C(C)=O)CCC1.C(=O)CN(C)C1CC1.O c1(C(N2C(CNC(c3cc(-c4cn(C)nn4)on3)=O)CC2)=O)n[nH]c2c1CSCC2 c1(NC(=O)C(=O)N2CC(N)C2)ccc(Cl)cc1.c1cc(C(=O)C(F)(F)F)c[nH]1 C12(CCNC(c3cc(C)ncc3)=O)CCC1CN(C(c1cccc(C)c1F)=O)C2 Cc1c(C(N2CC(NC(=O)C(N3CCCCC3=O)C)C(O)C2)=O)sc2cncn12 c1(C(N2CCCC2)=O)cc(=O)cc(Cl)[nH]1.C1(OCC)CC(CC(=O)NC)C1.C C1(C(=O)NC(CC=C)CO)CCC(C2CC2)N1C(c1cncc(F)c1)=O c1(C(N2C(C(=O)NC(CC#CC)CO)CC=CC2)=O)cc(C)c(C)cn1 c1(C(N2C3CC(NC(C(CSC)C)=O)CC2CC3)=O)ccc2c(c1)NCCC2=O c1cccc(C)c1.c1(CCC)ccc(C(=O)N(C)CC2CC2)s1.C(=O)(CC)N c1(CC)ccc(C(=O)NCC=CC(N2CCCC2CC(C)(C)C)=O)cc1 CCCCC(O)CC(=O)NC(C)(CNC(c1cccc(CC(F)(F)F)c1)=O)CO c1nc2c(NCCC34CC(CO3)C4)[nH]c(=NCC3CC34CCOCC4)nc2s1 C(=O)(CCCC#N)NCC12CC(NC(c3nc(C(C)OC)sc3)=O)(C1)C2 S(=O)(=O)(c1cc(Br)ccc1C)N1CC(F)CC(C(N2C(COC)CCCC2)=O)C1 c1(C(c2nnnn2CC2CC2)NCCC(CC)O)ccc2c(c1)CCC2(C)C CC1CCN(C(c2cnc[nH]c2=N)=O)CC1CNC(C1(CO)CCC1)=O N1(C(C=CCOC)=O)Cc2ccccc2C(NC(c2nn(C)c(C)c2Cl)=O)C1 C1(C(=O)NCC2C(C)CN(C(=O)C(C)(C)C3CCCC3)C2)CC2CCC(C1)S2 c1(-c2c(CNC(c3cncs3)=O)n[nH]c2)ccc(O)c([N+](=O)[O-])c1 n1(CC(=O)N(CCC)CCO)nc(C)c(Cl)c1C.N1(CC)CCOC(C=O)C1.N c1(C(N2CCCC2)=O)ccccc1.C1(CC)CCC(C(=O)NC)O1.C(C)(C)C CCC(C(=O)N1CCN(C(=O)Cc2cocn2)C(COC)C1)C(C)C CCC(CNC(=O)CCCN(C)C(C1CNC(=O)N1)=O)(CC)CC N1(C(c2nc(C#C)sc2)=O)CCN(C(=O)C(C)CCCC)CC1CC(=O)NC c1(CCNC(=O)OC)cn(C)nn1.C1CCN(C(=O)C=C(C)C(F)F)C1 N1(C(C(C)CC(N)=O)=O)CCC2(CC1)CC2C(=O)N(C1CCCC1(C)O)C C(C(C(=O)NC1CC2CC1CC2CO)C(C)(C)C)NC(COC(C)=O)=O S(=O)(=O)(c1cccc2c1COC2)NC1CN(Cc2cnc(C)o2)C1 C(=O)(C(O)CCSC)N1C(CN(C(=O)Cc2occc2C)CC)CCC1 c1(CC)nc(C(N2CC(NC(=O)C=Cc3sccc3C)CC2CO)=O)c(C)o1 C1(NC(CNC(c2c(C)occ2)=O)=O)CC(C)CN(C(C2CCCC23CC3)=O)C1 N1(C(CSc2nc(C)[nH]n2)=O)CCCC(C2CCN(C(=O)CC(C)C)C2)C1 CCCCCCCC(=O)NCC(C)(CO)NC(c1nc(OC)ccc1Cl)=O CCC(CCCC(=O)NCC1(CSC)CC1)NC(C1CC2CC2C1)=O c1cc(S(=O)(=O)N(C2C(CC(C)(C)C)C2)CCO)ccc1C#N.c1ccc(Cl)o1 C1(C(=O)NCC(C#C)CC)CCCC(NC(C2(C=C)CCC2)=O)CC1 N1(C(CC(C(=O)OC)C)=O)CC(NC(C2(CO)CCOCC2)=O)C2CCCCC12 CN1CCOC(NCCc2ccccc2CN2CCCC2)C1 N1(C(C23C(CCN(C(c4cn(CC)nn4)=O)CC2)C3)=O)Cc2ccc(O)cc2C1 C(=O)(C1=CC(C)(C)C1)N.c1(CNC(C(N2CCCC(O)C2)C)=O)ccccn1 C1(CNC(C2CCCS2(=O)=O)=O)CC2CCC1N2C(c1occc1Br)=O C(c1cccc(Cl)c1)=CC(=O)NCCC1CCN(C(=O)CN2CCCCC2=O)C1 N1(C(CN(C)CC)=O)CC(OC)C(OC)C1CNC(c1nccn1CC)=O N1(C(c2c(C)ncn2O)=O)CC2CC(NC(=O)CC#N)C(C2)C1 C(=O)(CC(C)(C)C)N1CCC(O)(CC)C1.C1(C=O)(SC)CCC1.C(C)=O.N CC1CCc2cc(NC(=O)C(=O)NC3CCCC3c3ccccc3Cl)ccc2N1 c1(C(N2C(C(C)(C)NC(C3C(C)C3)=O)CCC2)=O)ccc2cc(F)c(F)cc2n1 N1(C(C(C=CC)O)=O)CC(C(=O)NCCNS(N)(=O)=O)C(C(C)C)C1 c1(NC(CC2N(C(C(C(=O)OC)C)=O)CC(O)C2)=O)ccc(O)c(Cl)c1 n1(CC)c(C)nn(CC(N2CC=CC(NC(C3(C)CCNC3=O)=O)C2)=O)c1=O C1(OC)CCN(C(CC(C)SC)C(=O)NCC2CC2)C1(C)C C1(C(N2C(C(N(CC(=O)NCC)C)=O)CCC2)=O)CCCCC(=O)C1 C1CCN(C(=O)CC)CCC1(F)F.C(C)(C(=O)N)NC(=O)NC.CC(F)F.C c1(C(=O)NC(C)CCNC(C2COCC2(C)C)=O)ccc2cccc(O)c2c1 Cn1cc(C(F)(F)F)cc1C(=O)NCCCCC.C1(C(=O)N)(C(N)=O)CC1 N1(C(c2c(C)nncc2)=O)CCC2CN(C(=O)CNC(=O)CN(C)C)C2C1 C1(CNC(C(CC)(C)C)=O)C(C2CC2)CCN1C(C1SCCCS1)=O c1(C(N2CC(NC(C(N3C(=O)CCC3=O)CC)=O)C2)=O)cnc2sc(C)nc2c1 c1(NC2C3(CCN(C(C4CC(=O)N4)=O)CC3)C2)ncnc2ccc(I)cc12 C1(NC(CCCC#C)=O)CCN(C(=O)Cc2ccc(C(F)(F)F)cc2C)CC1O c1(C(N2C(COC)(C)CCC2)=O)nccc(Cl)c1Cl.C1(C=O)(CCO)CC1.N Cn1cnc(C(N2CC3C(C(=O)N)C3C2)=O)c1C(F)(F)F.C1CCC(=O)NC1 N1(C(C(C=C)O)=O)CCCC(C2CCCN(C(C3CCCC(F)(F)CC3)=O)C2)C1 N1(C(C2(C(=O)OC)C(=C)CC2)=O)CCC(O)(CC)C1.c1(C=O)cc(Cl)cnn1 C1(C(N2CCC(NC(C3CC(C)(C)C3)=O)(CO)CC2)=O)CCc2nc(O)[nH]c2C1 Cc1c(C(N2CCC(C)(NC(c3cnco3)=O)C2)=O)[nH]c2c(F)cc(F)cc12 c1(C(N2C(CN(C(=O)C(C#N)C(C)(C)C)C)CCC2)=O)cc2nc(Cl)ccc2o1 CCC(C)(C)CC(=O)NCC1CCN(C(c2ccc(Cl)nc2OC)=O)C1 c1(C(N2C(C(=O)OC)CCC2)C(=O)NCCCSC)ccc(S(C)=O)cc1 CC1(C(=O)NCC2CCN(C(c3[nH][nH]c(=N)c3Cl)=O)CC2)CCCCC1 N1(C(C(C)(CO)NC(C2CN(C)C2)=O)=O)CCC2(C=CCO2)CC1 C1(C(=O)NCCC(C)NC(=O)Cc2nccs2)CCOC(C)(C)C1 C1(C(N2C(C(C)C)C(C(=O)N(CC(C)(C)CO)C)CC2)=O)CC(=O)OC1(C)C n1(C(C(=O)NCCCCC(CO)NC(C=CC)=O)C)c(C)cc(O)cc1=O c1(C(N2CC(N(C)C)C(C=O)C2)C(=O)NCC(=C)C)cc2ccccc2s1.O C=Cc1cc(C(N2CCCC(NC(=O)CSc3nncs3)C2)=O)cc(F)c1 Cc1ccc(Br)c(F)c1C(N1CC(c2ocnc2C)C1)=O.C(=O)C=CCO.N Cc1cc(C(=O)NCC2(F)COCCN(C(=O)C(C)(C)CS)C2)cc(=O)n1C n1(CC(=O)NC2CN(C(c3c(C)c(F)ccc3)=O)CC2C)cc([N+](=O)[O-])nc1C c1(NCC(C)N(C)C(C2CCCC(=O)N2C)=O)cc(=O)n2cc(Cl)ccc2n1 c1(C(N2CCN(C(COCCOC)=O)C(C)C2)=O)ccn2nccc2c1 C1(CC)COC(C)CN1C(c1ccnc(C)c1)=O.C1(C=O)C(C)(C)C1(C)C.N CC1CCC(CNC(=O)CC2C=CCC2)CN1C(c1ccc(C2CC2)o1)=O c1(C2C(C(=O)OC(C)C=CCOc3ccccc3)C2)ccc(Br)cc1 CC1CC(C(N2CCC(C)C2(C)C)=O)CC(C)C1.C1(CC(=O)N)CCC(=O)NC1 C1(CC(=O)N2CCC2)COCC1NC(C1CCS1(=O)=O)=O c1(C(=O)NC2C(NC(C3ON=C(CC)C3)=O)C2)cccc2oc(C)cc12 CCCCC(C)C(=O)NC1CCN(C(c2[nH]nnc2-c2ccccc2)=O)CC1O n1(CC)ncc(C(N2CCC=CC2C)=O)c1C1CC1.C12(C=O)COCC1C2.N C(=O)(C1COc2ccccc21)N1CC(C)C(CNC(=O)CO)C1 C1CN(C(C2CC(C(F)(F)F)C2)=O)CC1(F)F.c1(CC)cnn(CC(=O)N)c1 N1(C(C(C(=O)OC)C)=O)C2CCC1CC(C(N1CCC(O)CC(C)C1)=O)C2 c1(C(C=O)NC(C=CC)=O)cccc(C(F)(F)F)c1.c1(CC)ccccc1F.N c1(C(C(=O)NC(C)C)N(c2c(C)scc2)C)ncc(Cl)cc1F c1(CC)oc(C)cc1C(=O)N(C1(CC(=O)N(C(CC)CC)C)CC1)C CCC(C)C(C)C(=O)NCC(C(=O)NCC1CCC(=O)NC1C)N(C)C Cn1cc2cc(-c3cnc(C4CCCN4C(=O)CO)[nH]3)ccc2n1 c1(OC)ccc(CC(N2CCCC(NC(C3CC3(C)C(F)F)=O)C2)=O)c(C)c1 c1(OCOC)ccc(C(N2CCC(NC(C3CC3(F)F)=O)C2)=O)cc1F c1(N2CCC3(C(C(=O)OC(C)(C)C)C3)CC2)nc2ccc(Br)cc2o1 C1(NC(C2Cc3cncn3C(=O)N2)=O)CN(C(=O)C=CCF)CCC12CCC2 N1(C(C(c2ccccc2)OC)=O)CCC(NC(c2cn[nH]c2)=O)C(CO)CC1 C#CCCCCCCC(=O)N1CCC(CN(C)C(c2ccc(F)s2)=O)C1 c1(C(N2CCCC(NC(CCc3onc(C)n3)=O)C2)=O)cc2c(s1)CCC(C)C2 C=C(C)c1cn(CC(c2ccc(F)cn2)C)nn1 CC(C)CCC(=O)N(C)CC1CCN(C(=O)C(F)(F)CN2CCCC2)C1 CCC(CC)(CCNC(=O)CC1CCOC1(C)C)NC(=O)CSC(C)C C1(NC(c2cc(OC)n[nH]2)=O)COCCC1NC(=O)C=C1CCSCC1 c1(C(=O)NC(C)CN(C)C(C2(C3CC3)CC2)=O)c(O)nc(=O)n2c1CCC2 C#Cc1ccc(Br)c(C(N2CCC(CO)(NC(=O)C=Cc3cc[nH]n3)C2)=O)c1 c1(CNC(=O)CCc2nncs2)ncoc1CCNC(c1cnccn1)=O c1(C(N(C)CC2CCCN2C(=O)C(O)C2CCCC2)=O)cc(Cl)c(O)c(Cl)c1 c1(OC(C(=O)NC2C(NC(CSC)=O)CCC2)C)ccc(C)cc1C N1(C(C2C(C(=O)O)C2)=O)CCCC(N(C(=O)Cc2ccc(Br)s2)CCO)C1 c1(C(=O)NC2CCCC(NC(Cc3c(C)ocn3)=O)CC2)cc(F)c(F)cc1Cl C(=O)(C1CC(=O)Nc2ccccc21)N1C(CNC(Cc2c(C)nsc2)=O)CCC1 c1(OCC(N2CC(NC(CC=CC)=O)(CO)C2)=O)ccc(C#N)c(Br)c1 c1(C(=O)NCCC2N(C(CS(CC)(=O)=O)=O)CCCC2)ccc2oc(S)nc2c1 N1(C(CC(C(C)OC)NC(=O)C=Cc2cc[nH]n2)=O)CCCC12CCOC2=O N1(C(C(C(C)(C)C)O)=O)CCCC(F)(CNC(C2(CO)CCOC2)=O)CC1 N1(C(CCC=CCC=C)=O)CC(NC(C2CC(N3CCOCC3)C2)=O)C(C)C1 C(=O)(C1CCCc2ncnn21)N1CCC(C2N(C(c3ccc(SC)o3)=O)CCC2)C1 c1(N2CC(CS(=O)(=O)NC)OCC2)nccc2ccc(F)cc12 Cc1cn2cccc(C(=O)NC(C3CN(C(c4ccncn4)=O)CCO3)C)c2n1 C=CCC(C(=O)OC)NC(c1ccccc1OCCCOC)=O CC1(C)COCCC1C(=O)NC1CCCC1NC(C1CCCC2(CC2)C1)=O c1(C(=O)NCC(CC)NC(=O)CC2CC3(CC3)CO2)cnc2sccn12 C1(C=O)C(C)CCN1C(=O)Cc1cnn(C)c1C.C(=O)(CC)N(CC)CC c1(C(N2C(C(N3CCC(COC)CC3)=O)CC2)=O)ccc(I)cc1OC C(=O)(C(CO)C(C)(C)C)NCCC1CCCN(C(c2c(C)nc(C)n2O)=O)CC1 CC1CN(C(=O)CSc2nc[nH]n2)CCN1C(=O)CCc1ccccn1 C1(C(N(C(CCSC)C)C)=O)CCCN(C(=O)CNC(C)=O)C1C S(=O)(=O)(c1nc(N(C)CC2CCC(F)(F)C2)ccc1Br)NC(CC)CN(C)C C(C(C)CC(=O)NC(C)CN(C)C(c1ccc(C(F)F)nc1)=O)OC N1(C(c2cc(C)no2)=O)CCC(C)(CNC(C2CCCC(C)C2)=O)C1 N1(C(c2cnc(CC)[nH]2)=O)CCCCC(NC(c2ccccn2)=O)C1.C(C)(=O)N c1(C(N2C(C)C(NC(c3ccncc3)=O)CC2)=O)cc(F)c(F)cc1O CC1CC(C)(C)CN1C(C1CCCC1CNC(=O)C(F)C1CCCC1)=O N1(C(CCCCOCCC=C)=O)CCN(C(=O)Cc2c(Cl)cnn2C)CC(C)C1 C(=O)(C(O)CC(C)(C)C)NCc1c(C(N(C(CC)CO)CC)=O)n(C)nc1 N1(CC(=O)NCCN(C(=O)CS)CC)CCCCC1=O.c1ccc(F)cc1 S(=O)(=O)(c1cccc(=NCC(O)C2(Cl)CC2)[nH]1)NCCS(CC)(=O)=O C=C(Cl)C(C)(C)C(=O)NCC(CC)NC(c1cc(-c2cccn2C)[nH]n1)=O CCC(C)(C)C(C)CC(=O)N1CCC(NC(=O)C(C)=C(C)C)C1(C)C c1(CNC2(C(=O)NCCCNC(c3c(C)nns3)=O)CC2)ccccc1Cl N1(C(c2ncc(SCC)cn2)=O)CCCCC(CNC(=O)CC(C)(C)C)C1.S C1(C(C)C)CCC(CN(C)C(=O)NCC2(c3ccc(Cl)cc3)CCCCC2)CC1 N1(C(C(C)(F)F)=O)CC2ON=C(CNC(=O)COCCCF)C2C1 C1(CCNC(CC=CC=C)=O)CC(OC)CN1C(=O)C(C)CC=CCC CCC(C(=O)NCC(C)(C)C)Sc1nc(=N)[nH][nH]1.C12(C=O)CCC(C1)C2.N Cc1cn2nnc(C(=O)NCCOCCNC(c3ocnc3C)=O)c2c(O)n1 CCCCC(F)C(=O)NC1CC2CC(NC(=O)CC3OCCCO3)C1C2 c1(C(N2CC(CC(F)C(=O)NC3CCOC3)C2)=O)[nH]ccc1C1CC1 N1(C(COCCC)=O)CCC(F)(F)C(CNC(C2CCC(C)=C(C)C2)=O)C1 c1(N(C2CCNCC23CC3)C(C(C)(F)F)=O)ccc2nccnc2c1 c1(OC)cncc(C=CC(=O)NCCc2ccccc2F)c1.C1(C=O)CCC1.N CC(C(O)C(F)F)NC(=O)C(CCF)NC(C1CCS(=O)CC1)=O N1(CCOCC)CCC(C)(NC(C2CCC(C)C2)=O)C1 C#Cc1ccc(F)cc1C(=O)NCC#CC.C1(C(=O)N)CCC(C(F)(F)F)CC1 N1(C(CCC(C)OCC)=O)CCCC2(C1)CN(C(C1SCCS1)=O)C2 C(C#Cc1ccc(F)cc1)CN1CC(C(C)NC(c2cc(C3CC3)on2)=O)C1 C=CC(O)C(=O)NC(C)CCNC(c1ccc(OC)o1)=O N1(C(C(CC=C)NC(=O)C(OCC)OCC)=O)CC2CCN(C)C2C1 C1(C#N)(OC)CC(C(N2CCC(CNC(=O)C(F)=CCCF)C2)=O)C1 c1(OC)cc(C(N2CC(CNC(=O)C=CSC)C2)=O)cc2c1OCC2 N1(C(CC=CC)=O)CCC2CCN(C(C3CCN(c4ccccc4)CC3)=O)CC12 S(=O)(=O)(C1CC2(CCNCC2)C1)N(C)Cc1cc(C(C)C)no1 c1(C(N(C2CCN(C(c3cc(C#N)cs3)=O)C2)C)=O)nnc(O)nc1O C1(CCC)CN(C(C2CC23CCC3)=O)CC1NC(=O)C(C)=C(C)CC N1(C(Cc2c(C)cco2)=O)CCC(C)N(C(c2n[nH]c3c2CSCC3)=O)CC1 CC1CCN(C(=O)C(=O)Nc2cccc(NC(=O)C(C)C(C)C)c2)CC1 C(CC(C)C)(C(=O)NC(C)CCCNC(C1CCC=CCCC1)=O)NC(C)=O C(=O)(C(C(=O)OCC)C(C)(C)C)NC(CCNC(CC=C)=O)C CCC(C)(C(=O)NCc1ccc(C)c(F)c1)C(N)=O.C(=O)C(C)c1ccsn1 N1(C(C(C)n2cccn2)=O)CCC(C(=O)NC2CC(C)(O)C2)C1(C)C N1(C(C2CC2(Cl)Cl)CC)CCc2c(c(-c3ccccc3)nn2CC)C1 c1(NC2CN(C(C(CCCC)O)=O)CC(C)(C)C2)ccc([N+](=O)[O-])c(OC)c1 Cc1n[nH]c(C)c1CCC(=O)NCc1cccc(CN(C)C(c2cccs2)=O)c1 CC1(C)C(C)(C(N2CCCC(CCC(N3CC4CCC=CC34)=O)C2)=O)C1(C)C c1(C(=O)NCCCCNC(c2ccn(CC)n2)=O)ccnc(C(=O)OC)c1 CCC1=C(C(=O)N2CCC3CN(C(=O)CC4CC=CCN4C)CC23)CCCO1 CC1CN(C(c2[nH]cnc2C#N)=O)CC2(CCN(C(=O)CSCC(F)(F)F)C2)O1 c1(OCC(=O)NCC(F)CNC(=O)CC=C(Cl)Cl)ccc(F)c(Cl)c1 N1(C(c2c(NC(C(CC)NC)=O)ccs2)=O)CCn2c(C)nnc2C1 N1(C(CC(CCC)C)=O)CCC(C2(NC(c3cn(C4CC4)cn3)=O)CC2)C1 N1(C(C=CC)=O)CCC(CNC(=O)Cc2ccn(C(C)C)n2)C12CCC2 CC1(C)CN(C(c2cc(F)n[nH]2)=O)C(C)CO1.C1(C(=O)N)CCCN1C(N)=O c1(-c2cn(CCC(=O)NCCC3CC(OC)(OC)C3)nn2)c(C)nn(C)c1C Cc1nccc(CCNC(C2(C3CCCN3C(C3CCCCS3)=O)CC2)=O)n1 Cc1c(C(=O)NCC2C=CCN2C(c2cc3c(o2)CCCC3)=O)nc2sccn12 Cc1cccc(C(N2CC(COC(=O)Nc3cc(C(F)(F)F)ns3)C2)=O)c1 Cn1nc(C(N2CC3C(CNC(c4cc(Br)c[nH]4)=O)C3C2)=O)c2c1CCCC2 N1(CCCC)CCCCC1CNC(=O)NCC1CCC(=O)N1C c1(OC)ccc2c(c1)CC(C)N2S(=O)(=O)Cc1noc2c1CCCCC2 c1(CC)conc1C(=O)NCc1cc(C(=O)NC2(CC)CC2)cs1 C(=O)(C(CC(C)(C)C)NC(=O)CCN=[N+]=[N-])N(CCC(C)N(C)C)C C1(C)CN(C(C2CCCN2C)=O)C(C)(C)C1.c1(OC)ccccc1CC(=O)NC CN1CC=C(CC(=O)NC(C)(CO)C2CCCC2)CC1 c1(N2CC3CCC(=O)N3CC2)nc2c(c(=NCCCc3cnccn3)[nH]1)CCC2 c1(C(N2CCC(C)(C(=O)Nc3c(Cl)ccnc3Cl)C2)=O)ccc2cc[nH]c2c1 C(C(C)(C)CO)OC.C(=O)(C(C)(C1CC1)N(C(=O)C=Cc1ccsc1)C)N C(=O)C(C)S(N)(=O)=O.C1(CC(=O)NCCN(CC=C)C)CCCCC1.C C1(COC)CCCCN1C(c1cc2c(s1)CCC2)C(=O)NCCCSCC Nc1cc(F)cnc1C(=O)NC12CCN(C(=O)CC3CC3)CC1C2 CC1CC(NC(c2ccc(N3CCC(O)C3)cc2)=O)CN(C(=O)C=C2CC2)C1 CC1CC(CNC(c2cc(CNC(c3cocn3)=O)no2)=O)=NO1 Cc1cc(CS(=O)(=O)CCC#N)ccc1F c1(C(N2CCCC(CNC(C3C(C4C(C)C4)C3)=O)CC2)=O)cccc2nsnc12 C1(C(=O)N)CN(C(=O)C(C#N)C(C)(C)C)C2(CCC2)C1.C1(CCC)CC1C CC(C)CC(C)CNC(=O)C(C1CC1)C1CC1.c1(C(=O)N)cc(Cl)cnn1 c1(C(N2CCN(Cc3c(C)nn(C)c3)C(C(C)C)C2)=O)ccc2sccc2c1O C1(NC2(c3nnnn3C3CC(F)(F)C3)CC(C)C2)CCc2ccccc2OC1 CC(CC(N)=O)C(=O)NC1CN(C(c2ccncc2-c2ccccc2)=O)CC1F CCC(C)(O)CCNC(C1(CNC(c2ccc(Cl)s2)=O)CC(C)(C)C1)=O c1(CC)onc(C(=O)NC(C)(CNC(=O)Cc2ccc(Cl)nc2)CC)c1C N1(C(CCCC=C)=O)CCCC(CO)(NC(c2ccc(-c3cn[nH]c3)cn2)=O)C1 Cc1cn(-c2ccc(F)cc2)[nH]c1=NC(=O)C(=O)N1CCCC(C)(c2nn[nH]n2)C1 N1(C(c2cnc(CC(C)C)[nH]2)=O)CCCN(C(=O)C(C)CC2CCCCC2)CC1 C(=O)(CCCCC(C)C)NC(CC)CNC(c1c[nH][nH]c1=N)=O c1(SCCOC(C(C(C)SC)O)=O)c[nH]c2ccccc12 C1(C(=O)N)OCCN(C)C1=O.C1(C2CCC2)CC1.C(=O)(C=O)N1C(CC)CC1 Cc1ccc(F)c(N)c1C(=O)NCC1CCCN1C(c1ccc(F)c(Cl)c1F)=O C1(NC(c2n(COC)ncc2)=O)CCCC2CN(C(c3ccc(O)cn3)=O)CC12 N1(C(C2CC(C)(CC)C2)=O)CC(C)OC(C)(C)C1.c1(C=O)cnn(CCO)c1 C(=O)(C(F)C(C)CNC(=O)CNC=O)NCCC=CC c1(CNC2C=CC(C(=O)NCc3cn(CCC)nc3)C2)cccc(C)c1Br c1(C(N(C(CCNC(C(C)Cc2ccncc2)=O)C)C)=O)c[nH]c2cnccc12 N1(CCC2N(C)CCCC2)CCCC(C)(C(N2CCOCC(CO)C2)=O)C1 C1(NCc2c(N)c[nH]n2)CC=CCC1C(F)(F)F CCC(O)CC(=O)NCCCCC1CN(C(C2CCCN2C(C)C)=O)C1 C(C(=O)N1CC(O)CCO1)SCCNC(C1COCC(C)O1)=O c1(C(=O)NCCN(C(=O)CC(F)(F)C(F)F)CC)ccc2ccccc2c1 N1(CC)CCCC(C(N2CCCCC2CCNC(c2cc(C)no2)=O)=O)C1 N1(C(CCCOCC)=O)CCN(C(C2CCCNC2=O)=O)C2CCC12 c1(C(N2CC(CNC(Cc3c(C)ccs3)=O)OCC2)=O)ccc(C(F)F)c(C)c1 c12ncc(cn1)C(C(=O)NC)N1CCOC(C1)N2C.C1(C(=O)OC)CC(OC)C1 C(CCCCNC(=O)C(F)Cc1ccccc1)NC(C(C)n1ccnn1)=O c1(C(=O)Nc2nc(C(=O)OCC)c(Br)s2)cccc(C#N)c1Cl.C1CC(O)C1 CC(C)C(C)(O)CNC(=O)C(C)CN(C)C(C1CC(=O)C1)=O N1(C(c2nn(C)c(O)c2)=O)CCC2CCCN(C(c3ccoc3Cl)=O)C2C1 O=C(CS(=O)(=O)CCO)NC1CCC(CNC(C2CC3(C2)CC32CC2)=O)C1 c1(CC(=O)NC(CC)CN(C(=O)CCCSC)CC)c(C)nc2ncnn2c1C C1(NC(=O)NC(CC=C)C)CCN(S(=O)(=O)CCC)C1 N1(C(C(C)NCc2ccccn2)=O)CCC2OCCCC2(NC(C2(F)CC2)=O)C1 C1(NC(=O)CC23CCC(CC2)C3)CC2(C1)CC(C=O)C2.CCC.C1CCC1.N c1(C(=O)NCCC2N(C(C(C)c3ccsc3)=O)CCSC2)ncc2[nH]ncc2n1 C1(C(=O)OCC)CC(F)(C=O)C1.C1(CC)CN(C(=O)CC2CCCC2)C1 CC1C(C(=O)NCC(C2CCN(C(=O)COc3cccnc3)CC2)O)CCN1C c1(CC)ccc(C(=O)NC(CO)C(=O)NCCOCC2CCC2)[nH]1 N1(C(CCNC(=O)CO)=O)CC(NC(=O)C=Cc2cncs2)C(O)C1 C1(NC(C=C(CC)C)=O)CC2CCC1(NC(=O)CCc1cccc(Cl)c1Cl)C2 C1(C(=O)NCCc2cc(C(=O)NCCc3nc(C)[nH]n3)no2)CN(C)CCO1 N1(C(C(=O)NC2COC2)CCc2ccc(Cl)cc2)CCc2cc(Br)ccc21 C1(CCC)(NC(=O)CC2CC(C)C2)CCCN(C(C2(CC)CC2)=O)C1 Cc1cc(=NC(CNC(c2ccnn2C(C)C)=O)C2CC2)[nH]c(Cl)n1 c1(CC)nc(C)c(C(=O)NC(C)(C)Cn2cccn2)s1.C(=O)C=CCF C(N1CCC(C2(C(F)(F)F)CCC2)CC1)N1C(=O)C(=O)N(CC(C)(C)C)C1=O C1(C(N2C(SCC)CCC2)=O)(NC(C2CCN(C)CC2)=O)CCCCC1 N1(C(CC(CNC(CN2CCC(C)C2)=O)O)=O)CC(C)(C)OC(C)(C)C1 C1(CC)C(C(=O)N(C2CCN(C(=O)C=Cc3cn(C)cn3)C2)CC)CCN1C C1(C(N(CCCC=C)CC)=O)CCC(C2CC2)N1C(=O)CC1COCCO1 CCCCC(CNC(=O)C(C1CCCC1)OC)NC(c1ccc(C)n1C)=O Cc1nc2cc(C(N3CCOC(CN(C(=O)CC(C)(F)F)C)C3)=O)[nH]c2s1 C(=O)(CS(=O)(=O)CCO)N1CCC(NC(C(C(=O)OCC)C2CC2)=O)CC1 C(=O)(C(O)CC(F)(F)F)N1CC(C)(C)C(C(=O)NCC2CCC=CCC2)C1 c1(N(CC=O)C)ccccc1[N+](=O)[O-].Cc1cc(CC(=O)NC2CC2)c(C)s1.N Cc1ncsc1C=CC(=O)NC.C1C2CC1N(C(c1sc(C3CC3)nc1C)=O)C2 C1(NC(C2=NOC(C)(C)C2)=O)CCN(C(=O)CCC2CC2(C)C)CC12CCC2 C(=O)(C1=NNC(=O)C1)N(CCC(=O)NCCc1nncn1C)CC Cc1csc(C(N2CC(C(O)C(=O)NCC(CO)N(C)C)C2)=O)c1 Cc1c(C)c(CC(C)N(C2COC2)CC2CC2)c(C)c(C)c1Br C1(C(=O)OC)CCC2CN(C(c3c[nH]c(=N)cc3C)=O)CC2C1 C(CCN(C)C(c1coc(C2CC2)n1)=O)(C(C)C)NC(CC=CC=C)=O C1(NC(c2occc2)=O)CCC(CO)C1.C1(C=O)(C(=O)C2CC2)CC1.C N1(CC)CCOCC1C(=O)NC1CC2(C1)CC2NC(=O)C1=CSCS1 O=C(CC1=CCCC1)NCCC1CC(F)(F)CN1C(c1cc(C(F)F)no1)=O C(c1ccc([N+](=O)[O-])s1)=CC(N1CCC(O)(CC)C1)=O.C(=O)C=O.CC.N CCC(C)(CC(=O)O)NC(=O)CSCc1cn(-c2ccc(OC)cn2)nn1 c1(C(=O)NCCN(C)C(C2CS(=O)C2)=O)occ2c1CCOC2 c1(OC(C)C)cncc(C(N2CC(NC(=O)CC3(O)CCCOC3)CC2C)=O)c1 Cc1ccnc(C(F)(F)C(=O)NC2CCC2NC(c2cocc2C)=O)c1 N1(C(Cn2nnc(C)n2)=O)CC(=O)NCC1C(=O)NCC1CCC(=O)N1 c1(C(C)NC(C(=O)NC2(C#C)CC2)=O)ccccc1-n1cccn1 C#Cc1cc(C(=O)NCC(C2CCOC2)NC(=O)C(C)(C)C2CCC2)ccc1C N1(C(c2cncc(CC)c2)=O)CCC(CNC(=O)Cc2n[nH]c(=N)s2)CC1C c1(NC(=O)NCCCC(c2ccccc2)OC)ncnc2c1COCC2 C1(O)(CNC(CC(CNC(Cn2ccc(C)c2)=O)C2CCC2)=O)CC2C=CC1C2 C1(CC)CCN(C(=O)Cc2nc(=N)[nH][nH]2)C(C(=O)NCCC2CC(C)C2)C1 CCS(=O)(=O)CC(=O)NC1CCCN(CCOCC(F)F)CC1 CC1(C)OCC(C=CC(=O)NCCC2(O)CN(C(C3(C)CCC3)=O)C2)O1 c1(C(N(CC(C)NC(=O)CCc2n[nH]c(C)n2)CC)=O)cccc2nsnc12 CC1(C)CCCN1C(C12CC(CN1C1CC1)C2)=O.c1(C(=O)N)cncc(Br)c1 N1(C(C(C)Oc2ccc(Cl)cc2)=O)CCn2c(cnc2C2CCC2)C1 c1(CC)cc(C(=O)NC(C)(CNC(c2ncn[nH]2)=O)CC(C)C)ccc1F.C C(=O)(C1=CC2CCC(C1)C2)N1C2C(NC(C(CC)CN(C)C)=O)CC(C2)C1 C(CC1=CCOCC1)NC(CN(CCC)C(C1CCC(N=[N+]=[N-])C1)=O)=O C1(C(=O)NCCC2COCCO2)(CC)CCN(C(=O)C(C)SC)C1 c1(C(=O)NC2CN(C(c3noc(CC)c3C)=O)C(C)C2)cc(C)ccc1N Cc1nc(-n2cc(CCOCC(N3CC(C(=O)O)CC3C)=O)nn2)sc1C N1(C(C(C(C)C)F)=O)CC2CCN(C(=O)CC(C)F)CCC2C1 N#Cc1cccc2c1CCCN2C(=O)C=Cc1ccc(S(N)(=O)=O)cc1 Cc1ccc(C=CC(N2CCC(C)(NC(=O)CCC3CC(C)(C)CO3)C2)=O)s1 C1(CNC(c2cnc(C)[nH]2)=O)N(C(=O)C(O)Cc2cn(C)cn2)CCC1(C)C Cc1cc(C)c(C(=O)NC2CC2CNC(C2CC3C=CC2CCC3)=O)cc1Br N1(c2nnc(C(N)=O)s2)CC2CC1CN2C(C1CC1C)=O c1(C(=O)NCCCCCNC(c2nc(C(C)OCC)sc2)=O)oc(C)cc1C C(=O)(C#CC1(C)CCCO1)N(CC(C)(C)NC(Cc1c(C)n[nH]c1)=O)C Cc1cccc(OC(C)C(N2CC3CC3C2)=O)c1.C1(C=O)(C(N)=O)CCC1.C c1(OC)ccc(S(N)(=O)=O)cc1C(N1CCC(O)C(C(=O)N(C)C)C1)=O c1(C(N2C(CNC(c3nc(C)nn3C)=O)CCCC2)=O)ccn(C)c(=O)c1O c1(-c2nc(-c3cccc(CC)c3)n(CCN(C)C)n2)ccc(N(C)C)cc1F C1(CC(N2CC(CC)C2)=O)CC2(CC2)CO1.Cc1csc(C(F)(F)C(=O)N)n1 C1(COC(C(C)OCC)=O)CCCCC1(C)C C1(C(NOCC(CC)C)=O)(CNC(c2ccc(Cl)s2)=O)CCCO1 CC1CN(C(=O)CC2CC2(Cl)Cl)CCN1C(c1c(Cl)n[nH]c1C1CC1)=O c1(CN2CC(CN(C(C(COC)OC)=O)C)OCC2)cc2ccccc2o1 C(=O)(C#CC1CC1)NC1CCC(CCC(=O)N(c2cnn(C)c2)C)C1 Cc1cnc(N2CCCC2C(C)(C)NC(=O)C(C)O)nc1SC(C)C CCCCCCC(C)(C(=O)O)NC(c1ccc2c(c1)CCN2)=O C(=O)(C1=CS(=O)(=O)CCC1)NCC.c1(C(N2CCCC2)=O)cncc(Cl)c1.C C1(COC)CCCCN(C(C2CCN(C(C3C4CCC(C4)C3C)=O)CCO2)=O)C1 c1(NC(C(=O)NC(c2cccnc2)CCNC(C)=O)=O)cncc(F)c1 N1(C(CCC(N)=O)=O)CC(O)C(O)C1CNC(c1cc(Cl)no1)=O N1(C(CCOCCOC)=O)CCC(OCCNC(c2csnc2Cl)=O)C1 c1(C=O)cccc(C)c1.c1(C=O)c(C)noc1C1CC1.C1(OCC)CC1.C Cc1nc2cc(NC(C3CCCN(C(C4(C)COC4)=O)CC3)=O)cnc2[nH]1 C1(COC)CCCC12CCC2.c1(C(=O)NOC)ccc(OCC(F)(F)F)cc1 CCC(C(=O)NCC12CC(CO1)C2)C(C)C.c1(CCC=O)ccc(F)cc1Cl.N C1(O)(CNC(CC2C(C)CC2)=O)CCCN(C(c2cccc(Cl)c2F)=O)CC1 C1(NC(CC(CC)C2CC2)=O)COC2(C1)CN(C(=O)C(C1COC(C)(C)O1)O)C2 C1(C)(OC)CC(NC(=NC)NCc2cnnn2C)C1(C)C c1(C(N2C(CNC(CC=C=C)=O)CCC2)=O)cc(C)c2sccc2c1 c1(CC(N2CCN(C3CN(C(COC)C)C3)CC2)=O)nc2ccc(C)cc2[nH]1 C1(CNC(C(CC#C)O)=O)CCN(C(c2cc3scnc3[nH]2)=O)CC1C1CC1 Cc1cn2nc(C(N3CCN(Cc4ccc(Br)cc4C)CC3)=O)cc2c(=O)[nH]1 C1(C(N(CC(CC)O)C)=O)CC12CC(NC(c1ocnc1C)=O)C2 c1(OC)cc(F)ccc1C(=O)NCC1CCC1.C1(C=O)CN(CC(C)C)C1 N(C(=NCCc1cccs1)NC(C)COC(F)F)CC1CC(SC)C1 C1(NC(C(CC)Oc2cccc(C)c2)=O)CC2CC1N(C(C1CC(C)(O)C1)=O)C2 C1(C(=O)NCC(CN(C)C(c2cc[nH]n2)=O)(C)C)CC2(CO1)CC(F)(F)C2 c1(OC(C)C)ccc([N+](=O)[O-])cc1C(=O)NCC.C(c1cn[nH]c1)=CC=O Clc1nn(CC(F)F)cc1CNCCCNCc1ccccc1 C1(NC(C2CC(=C)C2)=O)CC(NC(c2ccc(O)cc2Cl)=O)C12CCOCC2 C(C)(C)(CS(N)(=O)=O)NC(=O)NCc1cc(OCCN(C)C)ncc1 C(C)(Cc1ccnc(N2CCC2)n1)(C(=O)O)NC(=O)OCC.C(C)(C)C Cn1ccc2c(N(CCC3CCCNC3)Cc3cc(I)c[nH]3)ncnc12 N1(C(C(C)OCC#C)=O)CCC(c2ccccc2C)CC1.C1(C(=O)N)SCCS1 C(=O)(CC1OCc2ccccc21)N1CC(C)(F)CN(C(c2csc(=N)[nH]2)=O)CC1 C(=O)(C1=C(Cl)CCOC1)NCCCCC1CN(C(C(c2c(C)cccc2)C)=O)C1 CCCS(=O)(=O)C(C)C(=O)NC(CNC(c1nnn(C)n1)=O)C1CCC1 c1(C(=O)NCCC)ccccc1S(=O)(=O)C(F)(F)F.C1(C)(C=O)CC2CC2C1 C1(NC(c2cnc(C(C)C)s2)=O)CCC(NC(c2cccc(N)c2)=O)CC1 Cc1cccc(Br)c1C(=O)N(c1ncncc1C#N)C1(C#N)CCNC1 Cc1nn(C)c(C)c1C(C)C(=O)N.C(=O)C(C)C.C1(CC)CC1.C(N)=O c1(CCC(N2CC(NC(c3nc(C)c(C)s3)=O)C(C)C2)=O)ccc(N)c(F)c1 N1(C(C(=O)NCC(C)C)CCc2ccc(F)cc2)Cc2c(F)ccc(Br)c2C1 c1(NCCCc2ccc(Cl)s2)nc2ccccc2nc1NCC1CC(=C2CC2)C1 C(=O)(C1=NNC(=O)CC1)NC1CCC(CCNC(CCc2cc(C)no2)=O)C1 c1(OC)nc2sc(NCc3noc4ccc(F)cc34)nc2cc1Br C1(C(=O)NC2C(C)(C(F)F)C2)C2CC1N(C(=O)CCCn1cccc1)C2 CC1CC(NC(C2CCC3CCC23)=O)CCN1C(C1CCC1)=O.[SH](C)(=O)=O.N N1(C(C(C)C(C)n2cccn2)=O)CC2(CCN(C(=O)CCCn3cncn3)C2)C1 C(CC(C)C(=O)NCC1CCC1C(=O)NCCc1[nH]cnc1C)=CCC N1(C(C(C)OCC=C)=O)CCC(C)C12CCC2.c1(C=O)ccc2c(n1)CCO2.N C1(CNC(C2(C=C)CCC2)=O)CCCCC1NC(c1c[nH]c(C=O)c1)=O.O C1(CC)(NC(=O)C(F)OC(F)(F)F)CCN(C(=O)CC2CCN(OC)CC2)CC1 O=C1CCN(CC2CC(=O)NC2)C(=O)N1CCc1cccc(F)c1.C1(S)CCC1 C1(C(=O)NCC2(C)CCN(C(CNS(NC)(=O)=O)=O)CC2)CCn2nncc2C1 C12CCN(CCC1(F)F)C2=O.[SH](=O)(=O)C(F)F.n1(C2(C(=O)N)CC2)cncn1 c1(C(N2CCOC(C(C)C)C2)C(=O)NC)ccc(F)c2ncccc12 C(C)(C)(CC(=O)NC)n1ccnn1.C(COC)(CO)(c1ccccc1)N(C)CC Cc1sc(O)nc1C(N1CCC1CC(=O)NCC1CCC(F)C1)=O Cc1cc(CNC(=O)Cc2cnn(C)c2)ccc1F.C1(C=O)CCS1(=O)=O.N c1(C(N2CC3N(C(C4CC(=O)N4)=O)C3C2)=O)c(Br)cc(F)c(Cl)c1F CC(C)C(CN(C)C)C(=O)NC1CCN(C(C2(O)CCOC2)=O)CC1 C(=O)(C1=CCCC1C)N1CC(NC(C(CC)CC)=O)(COC)C1 C(C(=O)NCCC1CC1)(C(C)CC(C)C)N1CCCC(OCC#C)C1 C12(C(N3CCN(CC4CN(C(C(N)=O)=O)C4)CC3)=O)CCCN(CCC1)C2 c1(C(C(=O)NCC(=C)C)N(C2(CC(C)(C)C)CC2)C)sccc1C c1(C(=O)NC(C(C)NC(C2(CC=C)CCCCC2)=O)C)c(C)nc(=N)[nH]c1C Cc1cc(C(N2CC(CNC(=O)CC(C)N(C)C)C(C)C2)=O)ccc1Cl c1(C(=O)NCc2ncc(C(=O)NC(c3ncc[nH]3)C)cn2)cc2ccccn2n1 N1(C(C)C)CCCC(NC(=O)C(=O)NC2CC(c3ccon3)C2)C1 c1(Nc2cc(C)[nH]n2)ncnc2c1cnn2CC(=O)OC(=O)N(C)C Cc1nc(C)n(CC(=O)NCCC2CN(C(=O)C(C)Cc3ccco3)C2)n1 CC(C)C(N)C(C)(C)C(=O)NC(c1cc(Cl)ccc1OCC1CCCCO1)=O C1(C(N(C2CCCC2)CCNC(c2nsnc2O)=O)=O)CC2CCCC2C1 C1(NC(C(C)=C2CC2)=O)C(C)(C)CC1(C)C.c1(C=O)cc(O)nc(Br)c1.N C1(OC)CN(C(c2ccc(C(F)F)cn2)=O)CC1NC(=O)CCC(=O)N(C)C N1(C(C2CN(C)CC2C(F)(F)F)=O)CCN(C(=O)CCC(=O)N(C)C)CC(O)C1 c1(OC)ccc(C(=O)NC2C3CC2(C)CN3C(c2ncccc2F)=O)c(Cl)c1 C1(NC(CN(C)C)=O)CCC2CN(C(C3(C)CC(F)C3)=O)CCC2C1 C1(NC(C(C)CNC(C2CC(=O)C23CCC3)=O)=O)CCC2CCCC1O2 Cc1nc(NC(C)(C)Cn2cccn2)c(F)c(C)n1.c1(C(=O)N)nc(C)sc1C C1(NC(c2cc(C)n(CCO)n2)=O)CCC(C)N(C(=O)C2=CCCCO2)C1 CC(C)(C)C#CC(=O)N1CCC(C)(NC(c2c[nH]nc2OCC(F)F)=O)C1 CCC1=C(C(=O)N2CC(F)(F)CC2(C)CNC(C2(CO)CC2)=O)SCCO1 c1(-c2c(CC)con2)nc(CS(C)(=O)=O)nn1CC1CCCO1 c1(-c2c(C)cncc2)cc(C(=O)Nc2noc3cnccc23)cc2[nH]ncc12 c1(C(=O)NC(C(CC2CN(C(C(C)C#N)=O)C2)F)=O)cccc2ccncc12 c1(C(=O)NCCC2N(C(C=C(COC)C)=O)CCOC2)ccc(Cl)c(Cl)c1 c1(CC(=O)NC2C(CNC(CCCCC#N)=O)C2)coc2cc(F)ccc12 C1(NC(c2cc(C)nnc2)=O)CCC2(CC1)CC(NC(c1cc(Cl)ns1)=O)C2 C(C(=O)NC1CCC(CC(N2CC3CC2CC3CF)=O)CC1)(C(C)(C)C)N(C)C CC1c2ccccc2CC1C(=O)N(C1CCN(C(=O)CN(C)C)CC1)C.C1CC1 Cc1sccc1CC(=O)NC(C(=O)NCCNC(=O)C(C)C)C1CCCO1 c1(NC(c2cn(C)nn2)C)ccc(S(=O)(=O)NCC(C2CCCC2)O)cc1F Cc1sc2cncn2c1C(=O)NC1COCC1n1cc(CN(C)CCO)nn1 CCC(CCC(=O)N(C1CCCC1C#N)C)NC(c1coc(COC)n1)=O C=CCCCCCCC(=O)N1CCC2CN(C(=O)C=C3CCN(C)CC3)CC2C1 CC1CN(C(C2CN(CP(C)(C)=O)C2)=O)C(C)CN1C(=O)CN1CCS(=O)CC1 C(c1c(C)noc1C)=CCNC(Cc1cc(C)no1)=O c1(C(N2CC(CNC(CCCOC)=O)N3CCC2C3)=O)ccc(F)c2c1OCC2 CC1(C)Oc2ccc(Nc3nc4ccccc4nc3NC3C4CCCC34)cc2O1 C#CC1(O)CCCN(C(=O)CCC2CCCCN2C(=O)COC(C)(C)CC)C1 N1(C(CC(C)C(F)F)=O)CC2(CCCC2)C1C(=O)NCC(=O)NC1CCC1 C#Cc1cccc(C(=O)NC(CO)C(C)NC(c2sccc2C2CC2)=O)c1Cl CC(CC1=CCCCC1)(C(=O)O)NCC1COC(=O)O1 C(CCCCCN=c1cc[nH]cc1[N+](=O)[O-])N(C)C(c1ccns1)=O C1(C(=O)NC(C(=O)OC)CCF)N(C(c2nccn2C)=O)CCCC1(C)C CC(F)CC(=O)OCC1(Sc2nncs2)CC1 c1(C(N2CCC(O)(C(=O)NCc3ccc(F)nc3)C2)=O)cc(Br)cnc1F C1(C)(CNC(Cc2ccn(C)n2)=O)CCN(C(C2CCCN2C2CCCC2)=O)C1 C12(CCNC(CNC(N)=O)=O)CCC1CN(C(=O)CCc1ccncn1)C2 C1(CNC(CC)(COC)c2nnnn2Cc2ccco2)(CC)CCOCC1 C1(C(N2CC(C(C(=O)N)OC)C2)=O)CC(=O)CC12CCC2.C12CCC(CC1)CC2 C1(NC(CCc2ccc(SC)cc2)=O)CC(C)CN(C(c2cnn(C)c2)=O)C1 C1(CC)CC(F)(F)CN1C(C1CC(C(C)C)=NO1)=O.C(C=O)=CCOC.N S(=O)(=O)(c1cccnc1NCCC(C)CCO)NC(CN(CCCC)C)C c1(C(C)=O)cc(CCC(N2CC(F)(C(N3CC4CC4C3)=O)C2)=O)oc1C N1(C(C2=C(C)CC2)=O)CCC2(C(=O)NC(CCO)C(F)(F)F)CCCC12 N1(C(CSCC=C)=O)CCCC1C1CC1.C1(C(=O)N)CCN(c2ncccn2)C1 C1(NC(c2cnco2)=O)CN(C(c2c[nH]c(=O)cn2)=O)CC(F)(F)C1 C=CC(C)CC(=O)N1CCC(OCCNC(C23CC(CC)(CO2)C3)=O)CC1 c1(NC(c2cc(C)n(-c3cccc(F)c3)n2)=O)ccc2c(c1)C(=O)CCCC2 N1(C(c2nc(C)n(C)n2)=O)CC(C)(C)OC2(C1)CN(C(=O)CCS(N)(=O)=O)C2 c1(C(=O)NC(C(=O)NCCn2ncc(C)c2)CC2CCCC2)cc(Cl)n(C)n1 c1(C(N2CCOCC(CC)C2)C(=O)NC2COC2)oc2ccccc2c1Br CCCCCCCc1ccc(C(=O)NCC(C)N(C(=O)C(C)C2CCC2)C)cc1 N1(Cc2cccc(C#C)c2)CCC2(CC1)CC(C(=O)NCCn1cccc1)C2 N1(C(=O)CCCCCBr)CCc2cc(-c3ccc(F)c4[nH]ccc34)ccc2C1 C(=O)(C(O)CNC(C1CCCOC1)=O)N1CC(OC(=O)NC)C1 C(=O)(C1=CCC(C)(C)CC1)NC(CNC(CCCC(CC)C)=O)CC(C)C C1(O)(CC(N2CC(CC)(OC)C2)=O)CCCCCC1.C1(C)(C=O)C=CCCC1.N C1(NC(c2scc(C)c2Cl)=O)CCC2CCN(C(C3CC3F)=O)C12 c1(N(CCC)CC)ccc(C(=O)N)cc1.C1CCC1.C(=O)CC.C(C)=O.C N1(C(c2c(C)oc(C)c2C)=O)CCC2(CC(NC(=O)C(C)CC(C)C)C2)C1 N#CC1CN(C(=O)NC(c2ccccc2)C2CC2)CC1.C1(C(=O)N)CCSCC1 N1(C(C=CC(C)C)=O)CCC(C)CC1C(N1CCCC(N(C)C)C1)=O N1(C(C(CCC)OC)=O)CCC2C(CCN2C(c2cn(CCF)nn2)=O)C1 C(=O)(CCCC1CCC1)NC(C(=O)OCCC)C.C1(C=O)CCC(=O)O1.N CCCC(C(O)C(=O)NCC(c1nccs1)C)NC(C12CC1CNC2=O)=O C=CCC(C(=O)N1CCC(CNC(=O)CC23CC(C2)C3)C1)C(C)C c1(NCCOCCOc2c(OC)cccc2)nc2sc(-c3ccccc3)cc2s1 c1(C(N2CC(CNC(C3C(OC)C3)=O)N(C)CC2)=O)ccc2ccncc2c1 S(=O)(=O)(c1cc(Br)ccc1Br)N1CC(NC(C#CC)=O)C(F)(F)C1 c1(C(=O)NC(C#C)(C)C)c(CNC(C2(CCCC)CCC2)=O)nnn1C c1(C(N2CCCC(C)(NC(C3=CC(C)(C)C3)=O)C2)=O)cccc2ccoc12 C1(NC(c2cc(N)c(Cl)nc2)=O)CC2CC1CN(C(=O)C(O)Cc1cnc[nH]1)C2 Cc1ccc(O)nc1CNC(=O)CCCCN(C(=O)C(O)C(F)(F)F)C N1(C(c2cc(C(F)F)cs2)=O)CCC2CN(CC34CC(CC(F)F)(C3)C4)CC12 c1(NC(C2CN(C(C3=CC(C)(CC)C3)=O)C2)=O)cc2c(cc1F)NCCC2 c1(CC)cccc(CNC(C2CC=CCN2C(=O)C(SC)SC)=O)c1 N1(C(C2C(NC(CNC(=O)OC)=O)C3CCC2C3)=O)CCn2nccc2C1 C(=O)(C(C#N)=COC)N1CC(C(C)NC(c2cccc(SCCC)c2)=O)C1 c1(C(=O)NC2CCC2NC(C2(O)CCC2)=O)cc([N+](=O)[O-])cc2c1OCCO2 c1(N(C)CC2CCN(C(c3cn(C)nc3C(F)F)=O)C2)ncc(Br)c(O)n1 N1(C(Cc2cccc(C)c2)=O)CCN(C(=O)C(c2ccnn2C)C)CC(C)(C)C1 C1(CCC)CN(C(c2cc(C)c(C)[nH]2)=O)CCN1C(=O)CCCc1cnccn1 C1(C(C)C)(C(=O)NCC2CCCN(C)C2)CCN(C(=O)Cc2ccon2)C1 N1(C(C2(CC=C)CCCCC2)=O)CC2(NC(=O)C(C)NC(C)=O)CCC1CC2 N1(C(CCC)=O)CCCC(N(C)C(C2CC(C)(C=O)C2)=O)C1.C(C)OCC.O O=[N+]([O-])c1cc2c(cc1CN1CCC(c3nccs3)CC1)OCCO2 n1(CC(=O)N(CC(C)(C)NC(=O)C=CS(C)=O)C)ncc2ccccc2c1=O N1(C(CCC(C)C)=O)CCC2(CC1)CC2(C)C(N1CCN(C(C)C)CC1)=O c1(CNC(=O)NC(c2nc(=N)[nH][nH]2)C)ccc2c(c1F)OCCO2 C1(F)(C(=O)NCCCCC)CCCN(C(c2ccc(=NC)[nH]c2)=O)C1 c1(OC)ncc(NC2CCC(n3nnnc3O)CC2)cc1C(N)=O CCCCCC(O)C(=O)NCC1N(C(c2ccnnc2)=O)CCCC1(C)C C12(NC(=O)C3=CCCCO3)CCN(C(C3(n4cccn4)CCC3)=O)CCC1C2 C1(C(N(CCCC(N2C(COC)C=CC2)=O)C)=O)C2CCC(F)C12 N1(C(C2C(CC(C)C)C2)=O)C2CCC1C(CNC(c1c[nH]nc1F)=O)C2 N1(C(c2cn(CC)nc2C)=O)CC2CCN(C(c3cn(C)nc3SC)=O)CC2C1 Cc1nc(NCc2cc3n(n2)CCN(C)C3)c(C#N)c(C)c1C C1CCN(C(C23CC(C)(C2)C3)=O)CC1.c1(C(N(CCC)C)=O)nccn1C Cc1cc(=NC(=O)C2CCCCCC2NC(=O)CC(O)C(C)C)[nH]n1C(C)C c1(OC)ccc(C(N2CCCC2(C)C(=O)NCCc2c(O)n[nH]c2C)=O)c(C)c1 Cc1cnccc1C(N1CCCCC1C1CCCN(C(=O)C(F)(F)CO)C1)=O c1(C(=O)NCC2CN(C(C=COCC)=O)CC2C)c(C)ccc(F)c1N C1(C(N2CCN(C(c3cnnc(O)c3)=O)C(CF)C2)=O)CC12CCCCC2 Cc1cccc(C(N2CCC(C#N)(NC(c3ccc(Br)c(CO)c3)=O)C2)=O)c1I C=CCCCC(C(=O)NC1CCNC(=O)CC1)NC(=O)C1=NOC(C)C1C N1(C(C(CCC)(C)C)=O)CC(CNC(=O)CCC(C)(F)F)CC(C)(C)C1 N1(C(Cc2cn(CC)nc2)=O)CC=CC(NC(c2nsnc2O)=O)C1 C1(CNC(CCC#CC)=O)CC(C)(C)CN1C(c1n[nH]c(C)c1C)=O C1(C(N2CC3C(NC(C4CCOC4)=O)(C3)C2)=O)CC2OC1C1CC21 C(=O)(C(CC(C)C)NC(C1(CC(C)C)CC1)=O)NCC(CC=C)(F)F C(=O)(C1CCCn2nccc21)NCCN(C(C1C(c2onc(C)n2)C1(C)C)=O)C c1(CC(=O)NC(C)CC2CN(C(C34CCCN3CCC4)=O)C2)ncc(F)cc1F N1(Cc2cccc(N(C)C)n2)CCC2(CC2C(=O)Nc2cncc(O)c2)C1 c1(C(=O)NCC(CNC(c2c(CC)ncnc2)=O)OC)cnc(C)cc1Cl Cc1ncn(O)c1C(=O)NCCN1CCCOCC1 N1(C(CCN(CC)CC)=O)CC2CC1(C(=O)NC(CC)(CC)CC)C2 C1(CNC(N(c2nc(C)sc2Br)CC)=O)CC2(CCC2)C1.C(C)(C)C.O C(C)(C)(C(=O)NCC=O)ONC(=O)OC(C)(C)C.C1(n2cncn2)CCC1 C(CC1=CCN(C(=O)Cc2ccsn2)CC1)NC(=O)CCCn1cccn1 c1(OC)cccc(CN2CC=CC2C(N2CCCC(CO)C2)=O)c1Br c1(C(=O)OCC(C)CC(F)(F)F)cc(Cl)c2c(c1)OCCCO2 C12(CNC(C(C)CC3CCCO3)=O)COC(C)(C1)C2.C1(C=O)CCCO1.N N1(C(CSC)=O)CCCCC2(CCN(C(c3c(Br)c(C)nn3C)=O)C2)C1 C1(CC)CN(C(c2occc2F)=O)CCN1C(=O)C(O)COCc1ccccc1 C(=O)(CC(F)(F)C(F)(F)F)NCC(CNC(Cc1c(C)cc(Cl)cc1)=O)C c1(C(N2CCCC(F)(CNC(C3(CC=C)CC3)=O)C2)=O)cc2ncccc2[nH]1 c1(N2CCN(Cc3cccc(OC)c3)CC2)ncc(C(C)(C)C)cc1C#N C#Cc1ccccc1CNC(=O)CC1(CNC(=O)C(O)C=C)CC1 CC(C)CCCCc1nc(-c2ccc(N(C)C)nc2)nn1C1CC1 c1(C(N2C(C(=O)Nc3ccc(C)cn3)CC(C)C2)=O)cc(F)ccc1C CC(C)(CF)C(=O)NCC1C=CCN1C(c1cnn(CCO)c1)=O c1(CC(=O)NCC2(O)CN(Cc3ncccn3)C2)cccnc1Cl CCS(=O)(=O)C=CC(=O)N1CC2C(C)C2C1.c1(C=O)ccnn1C(C)(C)C.N N1(C(c2c(C)cc(O)cc2)=O)CCC(NC(=O)C(F)OC(F)(F)F)C(C)(C)C1 N1(C(C(COC)(C)O)=O)CCC2(COC(CNC(C3(F)CCOC3C)=O)C2)C1 c1(OCCC(=O)NC2C(NC(C(C)(C)SC)=O)CC2)cccc(Br)c1 c1(OC(C)C(=O)N(CCCNC(=O)Cc2cnoc2)C)ccc(F)cc1 c1(C(C=O)C)ccc2c(c1)OCO2.n1(CCCOC)cc(C(=O)NCC)cn1.N C#Cc1cc(C(=O)NC2CCC3(CC3)N2C(=O)C(=O)CC(C)CC)ccc1C Oc1cc(CNC(=NCCOCC2CC2)NCC(F)F)cc(Cl)c1 c1(C(=O)NCCC2(NC(C3CC(C)OC3)=O)CCC2)cc([N+](=O)[O-])n[nH]1 N1(C(CCCCOCC)=O)CCN(C(c2cc(OC)ncc2F)=O)C(CF)C1 N1(C(C(C)n2cncn2)=O)CCOC(C)(CNC(C2(F)CCCCC2)=O)C1 c1(CC)c(OC)cccc1C(=O)N.C(C)(CC)CC.C(=O)CN(C1CCC1)C C1(CNC(c2nc(C)sc2)=O)CC2CCC(C1)N2C(C12CC(F)(C1)C2)=O C(=O)(C1SCCc2sccc21)NCC(C)(CO)NC(c1nc(OC)c(C)s1)=O c1(C(=O)N)ccc(C(F)(F)F)c(F)n1.c1(C(C)(C)C)ccc(C(F)(F)F)cc1F C#Cc1cc(F)c(C(=O)NCCC(C)NC(=O)C(c2ccccc2)F)cc1F N1(C(C(C)n2cnnn2)=O)CCSCC1C(N1CCOC2CC12)=O c1(NC(C#C)CC2CCCC2)cncc(CC(=O)OC)n1 CCC(CC(=O)N(CC(O)CC)C)N(C)C(c1cnn(C)n1)=O N1(C(CCOCCCOC)=O)C(C(=O)N(C(C)CC(C)CC)C)CC2CC12 c1(CCCNC(=O)NC(c2nccn2CC)CC)c[nH]nc1C O=C(CC(C(F)(F)F)NC(c1cc(O)ccc1F)=O)NCc1cocn1 c1(C(=O)OC)cccc2c1CCCN2C(=O)Cn1nnnc1-c1ccccc1 C1(C(=O)NCCSCC(N2CCC(OCC)CC2)=O)C2CCCCCC12 Cc1c(Cl)ccc(C(=O)N(C)CCN(C(=O)C2=COCCO2)C)c1O C1(NC(C2(C)C(C)C2)=O)CN(C(c2cn(C3CC3)nn2)=O)CC1C(F)(F)F C1(O)(CC=O)CCN(C)CC1.c1(COC)ccc(C(=O)NC(C)C)cc1.N c1cc(C)c(F)c(C)c1.c1(OC)ccc(C(=O)NC(C2(C=O)CC2)C)o1.N C=CC(C)(O)C(=O)N1CCN(CCNC(c2nccn2C(C)C)=O)CC1 c1(CNC(C2CCC(NCc3ccc[nH]3)CO2)=O)ccncc1Cl C1(CC(=O)NCc2cc(C)sc2)CCC(NC(=O)CCc2ccnn2C)CC1 c1(C(N2CCC(NC(CC3CC(CC)C3)=O)C2)=O)c(C)n(C)c2ccccc12 C(=O)(C1=CCN(C(=O)CC(=O)NCC2CC2)C1)N(C1CC1Cl)C CC(CC1CC1)C(=O)N1CCCC1CC(=O)N(C)C(C1CCOCC1)C N1(C(=O)C2=CCCS2)CCN(C(c2cc(C3CCOC3)[nH]n2)=O)C(CCO)C1 c1(C(c2nnnn2CCCC2CC2)NCCOCCCC)ccc2c(c1)CC2 C1(C(=O)N)CCOCC1(C)C.C1(OCCNC(C(C)(C)O)=O)(C)CCOCC1 C1(CNC(c2cc(F)ccc2Br)=O)CCCC2(CCNC2)O1 c1(OC)ncccc1CNC(=O)NCC(C)Oc1ccccc1F N1(C(c2c(CC)con2)=O)CC2OCCN(C(=O)COc3cc(C)on3)C2C1 C1(CC=C)(NC(=O)CCC2CC(F)(F)C2)CN(C(=O)CC2COCCO2)C1 Nc1ccc(O)c(C(=O)NCC(F)CNC(=O)C(c2ccc(Cl)nc2)(F)F)c1 c1(C(=O)NCC(N(C(C(c2ccncc2)C)=O)C)C2CC2)c(F)ccc(Cl)c1F C1(CNC(CC2N(C)CCC2)=O)CCN(C(=O)CCn2cccn2)C1(C)C CCS(=O)(=O)CC(=O)NC1CC(C(=O)NC23CCC(C2)OC3C)C1 N1(C(CCC(=O)N(C)C)=O)CCCCC2C(NC(=O)CC34COC(C)(C3)C4)C12 c1(CC)ccc2c(c1)CCN2C(c1cc(Cl)c(Cl)s1)C(=O)NC1(C)CC1 N1(CC(=O)N(C(C(=O)NCCCSC)(C)C2CC2)C)CCNC(=O)C1 C#Cc1ccc(C(=O)NC(C2CN(C(=O)COC)CCO2)C)cc1F c1(C(=O)NC(CC=C)CNC(c2ncn(C(C)(C)C)n2)=O)cccc2sccc12 c1(C(=O)NC2C(O)CCN(C(c3ncn(C(C)C)c3)=O)C2)cc([N+](=O)[O-])cn1C C1(C(=O)NCC2CN(C(c3cn(C)nn3)=O)C2)CCC(C)(C)OC1 N1(C(C2CCOCC2)C(=O)NCC=C)CCC(=CC(=O)OC)CC1 N1(C(CC(C)F)=O)CCC(C)(CCNC(c2[nH]nnc2C(F)F)=O)C1 c1(CN)ccccc1.c1(CCN2C(CS(=O)(=O)N)CCC2)cccc(C2CC2)c1 C1(CCC)C(=O)NCCN1C(c1cc(C(F)(F)F)ccc1C)C(=O)NCCC#N C(O)(C(=O)NOCCCO)C1CN(C(CC2CCC(=O)C2)=O)C1 N1(CC(=O)NCc2c(C)cccc2)CC2CC1CN2C(=O)Cc1cnn(C)c1C S(=O)(=O)(c1ccccc1Br)N1CCN(Cc2cc(C(=O)O)cc(Br)c2)CC1 Cc1cc(F)cc(C)c1C(N1CC2CN(C(c3cc(Cl)cnc3Cl)=O)CC2C1)=O Cc1ccc(C=CC(=O)NCC(C)(O)C)c(C)c1.C1(C(=O)N)CC1C1CCC1 Cc1cc2cc(-c3ncccc3C(=O)Nc3cc4cc[nH]c4cc3F)ccc2[nH]1 C1(Nc2nccc(C)n2)CC(NC(=O)CCc2cscn2)C12CCOCC2 Cc1nnc(CN2CCCCC2C(=O)N(C)Cc2ccccc2Br)n1C CC(C)CCC(O)C(=O)N1CCCC1CN(C(=O)C(F)=C1CCC1)C c1(C(N2CCC(C(C)NC(c3ccc(CCC)s3)=O)C2)=O)c(Cl)cnn1C C1(C=O)CC=C(C(C)C)CC1.C(C(=O)NC1CC1C)OCCOCC N1(C(CC(C)(C)O)=O)CC2CC(C(=O)NC3(C4CCC4)CC3)C(C2)C1 C(=O)(CC(C)CC(=O)NC1CC(CNC(C2Cc3cccnc3C2)=O)C1)OC C(=O)(CC(CN(C)C)C(F)F)NCCN1CCN(C(CCC(CC)OC)=O)CC1 c1(CNC(CSCCCC)=O)cc(C(=O)NCc2cc[nH]n2)on1 N1(C(C2(N(C)C)CC2)=O)CCCC2(C1)CN(C(c1cc(C3CCCC3)[nH]n1)=O)C2 CCC(C(C)CNC(C)=O)NC(=O)CN(C(=O)CCCC1CCCO1)C N1(C(C(CC)CC2CCCC2)=O)CCC2(CC1)CCN(C(C1CC(SC)C1)=O)CC2 N1(C(CCCC=C)=O)CCC(C2CCN(C(=O)C(=C3CCCCC3)F)CC2)C1 C(c1ccc2c(c1)COCC2)=CC=O.C(C)(CCC(=O)NC(C)(C)CC)OC.N C=CC1(NC(=O)CC2(CC(=O)OC)CC2)CC1 Cc1cc(CC(=O)OC(C)(C)C)ccc1CNC1CC2(C1)CC2(F)F N1(C(CSCC)=O)CC(C)(C)OC2(C1)CN(C(C1CCC3CC13)=O)C2 c1(C(=O)NCC(CC)NC(C2CC2C(F)(F)F)=O)cc([N+](=O)[O-])cnc1C c1(C(N2CC(C)(NC(c3cnc(CCCC)s3)=O)C2)=O)cnn2cc[nH]c(=O)c12 N1(C(=O)Cc2cc(F)cc(F)c2)CCN(C(c2ccnnc2Cl)=O)CC(O)C1 c1(C(=O)NCC2CCN(Cc3cccc(OC(C)C)c3)C2)ccc2ncnn2c1 C1(C(N2CC3C(NC(c4cnc(=N)[nH]c4)=O)C3C2)=O)CCC2CC2CC1 c1(C(=O)NC(CC)CNC(=O)C(F)OC)ccc(OC(C)C)c(N)c1 c1(OC)cc(CCNC(=O)C(=O)NC2CC2(c2ccccc2Cl)C)cc(C)n1 N1(C(CC2CC(=C)C2)=O)CCC(F)(C(=O)N(C)OC)C1.C C1(C(=O)NC2C(C(=O)O)COC2)(CO)CCCCO1 C(=O)(C1=CCC(C)CC1)N1CCN(C(c2nc(CC)sc2N)=O)C(C)C1.C1CC1 C1(CC(=O)NC(C(CC)CC)C)CCN(C(=O)Cc2cccnc2C)C1(C)C c1(CC)c[nH]nc1C(=O)NC1CC(C(=O)N(C(C)CS(C)=O)C)C1 C1(CC)CCCCCN1C(c1ncc(C(=O)OC)s1)C(=O)NC1CCOC1 c1(CN(C(=O)CCc2ccc(F)nc2)C)ccc(C)cc1F.C(=O)(C1CC1)N C(=O)(C(F)C(F)(F)F)NCCNC(C(C)C=Cc1ccccc1)=O.C1CC1 C1(NC(c2ccc3nccn3n2)=O)CN(C(C23CCC2C3)=O)CC2(CCC2)C1 N1(C(C(c2ccc(CC)cc2)C)=O)CCOC(C)(CNC(c2ccnn2C)=O)C1 n1(CCC)c(=O)n(CCNC2CC(C)CN(C(=O)CC3CC3)C2)c2ccccc12 C1(N=[N+]=[N-])(C(N2CC(C)C(NC(=O)CC(F)(F)C(F)F)CC2)=O)CCOCC1 C1(C2CCCN(C(=O)C(C)(C)c3cnn(C)c3)C2)(NC(CCC(CC)C)=O)CC1 C#Cc1cc(NC(=O)C(c2ccco2)NC(c2cc(OC)no2)=O)ccc1C c1(C(N(CC(C)NC(C2(COC)CCOC2)=O)C)=O)ccc(C)nc1O CC(C)C(C(=O)NCCCn1cccn1)C(C)NC(c1n[nH]c(=N)[nH]1)=O C1(C2CCN(C(c3ccc4n[nH]cc4n3)=O)CC2)(NC(CS(CC)=O)=O)CCC1 C1(C#N)(SC(C)C(=O)Nc2c(C(=O)NC(C)(C)C)scc2)CNC1 C(=O)(C(CC1CCCO1)C(F)(F)F)N(C)CC.C1(=O)CO1 c1(CCC(=O)NCCC)c(C)nn(C)c1C.C12(C=O)CCC(C)(C1)OC2.CC c1(CC)cscc1NC(C1CCN(C(=O)C(CSC)OC)C1)=O N1(C(C2C(NC(c3cnn4ccccc34)=O)COC2)=O)Cc2cc(O)nnc2C1 N1(C(c2c(CC)non2)=O)CCC(C)C1CNC(c1ccc(CCF)cc1)=O CS(=O)C=CC(=O)N(CCCNC(C1(C)C=CCCC1)=O)Cc1cccnc1 C1(C(N2CC3CC2C3)=O)(OC)CCC(C(F)F)CC1.C(C(C)(C)C)=CC=O CCC(CNC(c1nnn(C)c1N)=O)(CC)C(=O)NC1CCC(=O)NC1=O c1(OC(C)C)cc(F)cc(F)c1.C1(N2c3c(nccc3)C2=O)CCNCCC1C c1(NC(C(CCSC)NC(=O)CCCn2cccn2)=O)ccc(C)cc1CO Cc1nc2ncccc2cc1C(=O)NCC1CN(C(=O)C(C)O)CC12CCC2 C=CC(C)(O)CC(=O)NCC1CCN(C(=O)C(CCC)OC)CC1 c1(CC)c[nH]nc1CNC(=O)C(F)C1CC(NC(=O)C(C)N2CCCC2)C1 c1(NC(C2C3CN(c4ncccn4)CC23)=O)ccc(Cc2ccccc2)c(O)c1 c1(C(C(=O)N)C)ccc(F)c(Cl)c1.c1(C(=O)NCCC)cc(-c2ccco2)no1 C(CC(=O)NC(C1CCCC1)CNC(c1cnn[nH]1)=O)OCC(C)C c1(CC)cccc(C(N2CCCC(c3cn(CC4C5CCCC45)nn3)C2)=O)n1 N1(C(C(CCC#C)O)=O)CCCC2(CCN(C(=O)C(C)(CC)CCC)C2)C1 c1(C(=O)NC2CCC(NC(C(C=C)(C)O)=O)CC2)ccc2nc(C3CC3)oc2c1 c1(CC(=O)NC2CCn3nccc3C2)cn2cc(Cl)ccc2n1 C1(C(C(=O)Nc2ccccc2)N(CCCC)Cc2snnc2C)CCN(C)CC1 CN=C(NCc1c(-c2ccccc2)coc1C)N1CCC(S(C)(=O)=O)CC1 N1(CC)CC(C(=O)NC)CCC1=O.C1CCCC1.c1(C=O)cnc(C(C)=O)s1 N1(C(C(CC)CCOC)=O)CC2CC1CN(C(C1(C3CC3)CCCO1)=O)C2 C1(C(=O)NCC(COC)C)CCN(C(c2nocc2C)=O)C1 c1(C(N2CCCCC(NC(CN(CCC#C)C)=O)C2)=O)c([N+](=O)[O-])cnn1CC c1(OC)ncncc1CN(CC(F)(F)CO)C CCCCC(C(=O)NCCCF)N1CCC(c2ccc(Cl)cc2)C1(C)C C1(CCC)CN(C(c2c(C)noc2C(F)F)=O)CCO1.C=CCCOCC(=O)N c1(C(=O)NCC2CCN2C(=O)Cc2cnc(C3CC3)[nH]2)cn2ccccc2n1 C(Cc1ccco1)(C(=O)N(C1(CCO)CC1)C)NC(CC=C(C)C)=O c1(CC(=O)N(C2CCN(c3ncns3)C2)CC)nonc1C c1(C(=O)N)cnc2c(ccn2C)c1.c1(NC(C)=O)ccc(C(=O)NCCC)cc1 c1(C(N2CCN(C(C(C)OCC=C)=O)C(C(C)C)C2)=O)cc2ncccc2[nH]1 c1(C(=O)NCCOC2CN(C(=O)CC3COCCO3)C2)c(Cl)ccc(Cl)c1O c1(CC(=O)NC2CC(CNC(=O)C(F)C(F)(F)F)C2)ccc(Cl)cc1F c1(CC(=O)OCCSC)ccc(C)c(F)c1F Cc1cc(C(=O)NC2CCC3CCC2C3)c(C)n1C1CC1 C1(OCC)CC(CC(=O)NC2CCCO2)C1.C12CC(C1)CCO2.C(=O)C c1(C(N2CCC(C)(NC(c3c(C)nc[nH]3)=O)CC2)=O)cc(N=S(C)(C)=O)ccn1 c1noc(C)c1C(=O)NC.C1(C(N2CCCC2)=O)C(C=C(C)C)C1(C)C N1(C(CCCC2C(C)C2)=O)CCC2C(CCCN2C(c2cnoc2C2CC2)=O)C1 c1(C(N(CCC)CCNC(C2CC(C)(C)C2)=O)=O)cnc2ccccn12.O Cn1cnc2cc(C(=O)NC3(C)CCN(C(C4CCCCC4F)=O)CC3)ncc12 C(CCO)(C(C)(C)C)NC(C=CC(C)(C)NC(Cc1n(C)ccn1)=O)=O c1(C(N2CCC(NC(Cc3cc(C)on3)=O)C2)=O)cc(F)c(F)cc1.C(N)=O.N Cc1ccnc(C(=O)NCCC2CCC(NC(=O)CSS(C)(=O)=O)C2)c1 C1(N(C(c2ccc(C3CC3C)o2)C=O)C)CCOCC1.C(=O)CC.C1CC1.CC CC1CN2CCN1CC2C(=O)NC1CCC(CNC(C2(C)C=CCCC2)=O)C1 N1(C(c2cc(CCC)[nH]n2)=O)CCC(C)C(NC(c2cnc(C(C)C)o2)=O)C1 C(c1ccnn1C)=CC(=O)NC1(C(N(CCC)CCC)=O)CC1(C)C CCC(C)(C)C(C)CC(=O)N(C)CC1COCCN1C(c1[nH]c(C)nc1C)=O C(C)(C(C)(C)C(=O)NCCC1COCCO1)NC(C(CC)CN(C)C)=O C12(CC(=O)NCc3c(C)nn[nH]3)CCC1CN(C(c1cc(C(C)C)no1)=O)C2 C1(CNC(c2c(NC)cccc2)=O)CCC2(CCC2)C1.C1(C(=O)N)CCC1 N1(C(CC2(C)CC2)=O)CCC(O)(Cn2cc(CC3CCCOC3)nn2)C1 c1(C(=O)OCC(=O)NCC2CCN(CC(F)(F)F)C2)cn2c(Br)cnc2s1 N1(C(CNC(=O)OC)=O)CCCC1.C1(C(NC)=O)OCCC1.C1CC=CC1.C Cc1cc(O)ncc1C(=O)NCC1CCCCC1.C1(C=O)CCS(=O)(=O)C1.C c1(C=O)cc(O)nc2[nH]c(=N)ccc12.C1(C(N(CC)CC)=O)CC12CCOC2.N c1(C(=O)NC2CCC(CCNC(c3c[nH]nc3Cl)=O)C2)cnc2ccncc2c1 N(C1CCc2c(F)cc(F)cc21)C1(c2n(CC)nnn2)CCC(=O)N(C)C1 c1(OC)cc(C)c(CNC(=O)C(c2ccccc2F)C)cc1OC C(CC(C)(O)CNC(=O)CC1CC(F)CN1C(c1cnncc1C)=O)OC C1(NC(c2c(C)cnnc2)=O)CCC(O)CN(C(c2cc(CN)ccc2C)=O)C1 CC(C)(C)C#CC(=O)N1CCC(C)(NC(=O)CC(F)(F)F)C1 c1(CC(N2CC(NC(c3c(C)nsc3)=O)C(F)C2)=O)coc2ccccc12 C1(NC(C2C(C)OCCC2)=O)CCSC12CN(C(c1ncc(F)cc1F)=O)C2 CON(C(=O)C1C2CC3C(C2NC(C2CCC(OC)CC2)=O)C13)C(C)C c1(C(=O)N)cnc2c(c1)nnn2C.Cc1ccccc1C=CC(=O)NC1(C)CC1 C1(CCCNC(C(C)n2cccn2)=O)CCCN1C(=O)CCOc1cccnc1 c1(C(=O)NC2(C3CCCO3)CC2)cn(CC)nn1.C(=O)(C(F)n1ccnc1)N CCC(C)(C)CCCC(=O)N1CCC(C(C)NC(=O)CC2(O)CCN(C)CC2)C1 O(NC(=O)C(C)(CO)OC)CC(N1CCCC(CCC)C1)=O N1(CC2CN(C(C(C)C3CCC3)=O)C2)CCN(C(c2cnc(C(F)F)s2)=O)CC1 Cc1cnccc1C(N1CCN(C(=O)C(c2ccccc2)N(C)C)CC1)=O O=C1CCC(C(=O)N(C2CCCC2)CCCNC(C2C=CCC2)=O)C1 CC(C)CC(CNC(c1nccnc1N)=O)C(=O)N1CC2C(C1)C2(F)F C1CCN(C=O)CC1.C(C(C)C(=O)NCC(=O)NCC(=O)N)OC.C(C)C N1(C(c2c(N)ccc(OC)c2)=O)CC2CC1CCC2NC(=O)C(C)(C)CF c1(C(N2C3CN(C(C(CCCC)=O)=O)CC2CC3)=O)cc(F)c2c(c1)CCC2 N1(C(C2(C)C=CCC2)=O)CCC(O)(CCNC(c2sc(C#N)cc2Cl)=O)CC1 c1(C(=O)NCCC2(O)CN(C(c3cc(CCC)[nH]n3)=O)C2)cnc(OC)cn1 c1(C(N2C(C(=O)NCCS(C)(=O)=O)CC3CC32)=O)cc(O)cc([N+](=O)[O-])c1 N1(C(C2C(CC)CCO2)=O)CCC(N=[N+]=[N-])(C(=O)N(CCCN=[N+]=[N-])C)C1 C(=O)(C(F)CC(C)(C)C)N1CCC2(NC(c3ccc(C)c(F)c3)=O)C(C1)C2 C1(CNC(CC(CC)OC)=O)CC(C(=O)NCC(C(F)(F)F)OC)=NO1 N1(C(c2c(CC)ocn2)=O)CC(CNC(=O)C(c2ccccc2)S)C(C)C1 C12(OC)CCC1CN(C(=O)C(F)C1CCC1)C2.c1(CC=O)c(C)nn(C)c1C.N c1(C(C)NCC(c2ccoc2)N(C)C)cc(-c2ccccc2)ccc1Cl c1(CC)cccc(C(=O)NCC2CCCC2NC(=O)C(F)(F)C(C)O)c1O C(=O)(N=c1ccn(CCO)[nH]1)C1(CC)CCN(C(c2nc(O)sc2C)=O)C1 C1(C(N2C(CCNC(C(C)=CC3CC3)=O)CSCC2)=O)CC2CCCCCCC12 c1(C(=O)OC)csc2c1CCN(C(C1C=CCN1C(=O)CS)=O)C2.c1nc[nH]n1 Cc1cc(Br)cc(F)c1C(=O)NCC1CCN(C(c2ccnc(Cl)c2C)=O)C1 C12(NC(c3c(Cl)cn(CCC)n3)=O)CCCCC1CN(C(C1CC1(C)C)=O)C2 C1(CC(=O)NC(CC)CNC(=O)CCc2ncc(C)[nH]2)COc2ccccc2O1 Cc1c(C(N2CCC(C)(CC)C2)=O)nnn1C(C)C.n1(CC(=O)N)nccc1C N1(C(c2cc(C)n(C)n2)=O)CC2CCCCC2(CN=c2[nH]c(Cl)ncc2F)C1 N1(C(CC=CC)=O)CCC(O)(CN(C(=O)CC2CC(O)C23CCC3)C)CC1 C(CCCCC(=O)NCc1occc1C(N1C(C)CCC1(C)C)=O)=CC C(=O)(C(C)CC(=O)N=c1ccn(-c2ccnc(C(F)F)c2)[nH]1)OC C1(CNC(CN(CCC#C)C)=O)CCCC1NC(=O)CC1CCN(C)C1 C=CC1(CC(=O)N(C)CC2CCCC(NC(=O)Cc3cscn3)C2)CCOCC1 C1(NC(C(C)=C2CCCC2)=O)CCCC(NC(C2CC(C)(O)C2)=O)C1 C1(NC(C(C)(c2ccccc2)OC)=O)CCC(NC(=O)Cc2ccsc2)CC1 CC1(C2CCC2)CN(C(C2(F)CCN(C(=O)COC3CCCOC3)C2)=O)C1 c1(CCCCC)ccc(C(=O)NCC#CCNC(=O)Cc2cc(C)nn2C)cc1 Cc1ccc(C)n1S(=O)(=O)NCc1cn(C2COCC2O)nn1 c1(CC(=O)NCCN(C(c2c(CC)cccn2)=O)CC)ccc(F)c(F)c1 CC1CN(C(C)C(=O)N(C)C(CC(c2cccc(Cl)c2)O)=O)CCN1CC(F)F C(N=c1[nH]c(=NC2CCSC2C)[nH]c2ccsc12)c1c(C)n[nH]c1C Cc1cc2ncn(CC(O)CN3CCCCC34CCCNC4)c2cc1C c1(C(=O)NC2(CNC(CC(COC)C)=O)CC2)cnn2c1CC(C)CC2 N1(C2(c3ncon3)CC2)CCN(CCC)CC1 c1(OC)c[nH]c(C(=O)NC2CN(C(=O)CC3CC4CC4C3)CC2O)cc1=O c1(NCCC2CCN(C(C(C)(C)N(C)C)=O)CC2)snc(Cl)c1C#N C(CCCCCN(C(=O)C(c1ccc(F)cc1)C)C)NC(C(C)=C1CC1)=O C=CC(C)(C)CC(=O)NC1CCOCC1NC(c1cc(-c2ccccn2)c[nH]1)=O C(=O)(C1=CCCN(Cc2ncn(-c3ccccc3)n2)C1)Nc1c(C)ccc(OC)c1 N1(C(CC(C=C)C)=O)CC(NC(=O)COCCOCCO)CC12CCCCC2 N1(C(Cc2c(C)n[nH]c2C)=O)CCCC(C)(CNC(C2CC23CCCC3)=O)C1 c1(C(N2CC(C)N(C(C34CCC(C3)C4)=O)CCC2)=O)cc2ccc(Cl)cc2[nH]1 c1(CC)cccc2c(CC(=O)NC3CN(C(=O)C(F)C(C)(C)O)C3)c[nH]c12 N1(C(C(C)(C)C2CCC2)=O)CCC2(CC1)CN(C(=O)CO)CC2CO CCC(CN(C)C)CC(=O)N1CCCN(C(=O)CC2OCCCO2)CC1 c1(C(N2C(C(N3CCC(C(F)F)C3)=O)CC(OC)C2)=O)cccn(C)c1=O c1(OC)cccc(C(=O)N(C(C)CC)C)c1N.C1(CC(=O)N)CCCC(C)(C)O1 CC1CN(C(c2csc([N+](=O)[O-])c2)=O)CCC1NC(=O)CC1CCCNC1=O c1(C(N2CC(C=C)(CC(=O)NCC3(C=C)CCC3)C2)=O)cc(C)n(C)c1C C1(CNC(c2ccc(C(C)C)o2)=O)CN(C(=O)CCN(C)C)CC(C)(C)O1 Cc1[nH]nc(C(N2CCCCC2C(=O)NCCN(C)CCF)=O)c1C C1(CC)CC(O)CN1C(c1csc(C(C)C)n1)C(=O)NCSc1ccc(F)cc1 c1(C(N(C2C(C)CC2)C)=O)occc1CNC(=O)CN1CSCC1=O CCCCC(C(=O)N(CCCCN(C)C(C1CCCC1C)=O)C)NC(N)=O CN1CCC2CCC(C1)N2C(=O)CC1(NC(=O)CS)CCCCC1.C(C)(C)C C(=O)(CCCC)NC(C)CNC(c1cnn(-c2ccccc2)c1)=O.C(C)(C)C.S c1(C(N2CC(NC(=O)C(c3cccc(Br)c3)O)C(F)C2)=O)cc2ccccc2s1 C1(NC(c2cc(CCC)on2)=O)CC(CNC(=O)CO)CC1O.CC(F)F c1(CNC2CN(C(C(C)Cc3ccco3)=O)CC(C)C2)ccc2ncccc2c1 C(C(=O)NCC=C)(C(C)NCC(C)C)NC(C=CC=CC)=O.O N1(C(C(CC#C)(C)NC(=O)CCC2CCOC2)=O)CC2(COC(=O)N2C)C1 N1(C(C(C)NC(C2CCC2)=O)=O)CC2(C1)SCCC2.c1(CC=O)ccsc1Cl.N N1(CCC)CCCC(C(=O)N(C)CCNC(=O)C(c2cccnc2)O)C1 C1(C(N2CC(CNC(CC=CC)=O)C(OCC)C2)=O)CCCCCS1(=O)=O c1(C(c2n(C)nnn2)NCCc2cncs2)ccc(F)cc1C(F)(F)F O=C1CN(Cc2cn(Cc3cccc(NC(=O)CCCF)c3)nn2)CCN1 Cc1cc(N2CC3(CC3)CC2CNC(c2cc(Cl)ccc2F)=O)nc(CO)n1 c1(C(C(=O)N(C2CN(C(=O)CCc3cnoc3)C2)C)O)ccc(F)c(Cl)c1F c1(C(C(=O)NCCNC(C2C(C(=O)OC)C2)=O)C)ccccc1 Cc1oc(C#N)cc1C(=O)NCC(F)CNC(=O)C(C)CC(C)C Cc1nnc(N2CCC(C3CC3)(CNC(=O)CCC3CCCO3)C2)c(C#N)c1C N1(C(c2ccccn2)=O)CC(C)(C(N2CCC(C3(C)N=N3)C2)=O)CC1(C)C.CO CC(C)CS(=O)(=O)CCC(=O)NCC(C)(C)CN(C)C(C1CCC(=O)N1)=O c1cncc(C(=O)N(C2COCC2O)C2CC2)c1.C1(C(=O)NC)CC1C1CC1 Cc1cc(C(=O)NC2CCC(NC(=O)CN3CCCCC3=O)C2)n(C(F)F)n1 c1(CC)oc(C(=O)NCC2(NC(=O)CC=O)CCCC2)cc1C(=O)O CCC(CC(=O)NC1(CC(N2CCC(OC(C)=O)C2)=O)CCC1)C(C)(C)C N1(C(c2c(C)scn2)=O)CC2CC(C1)N(Cc1cccc(OCCO)c1)C2 c1(OC)nn(C)cc1N.c1(C(=O)C2CC2)ccn(CCNC(=O)C=O)c1 c1(C(=O)NCc2nc(C)nn2C)ccc(N2CCNCC2)c(F)c1 C1(NC(CCC(C)OCC)=O)CCN(C(C2CN3CCN2CC3)=O)CC(O)C1 C12(CNC(Cc3ccc(C)s3)=O)CN(C(c3cnsc3)=O)CC1CCO2 C1(C)(C(=O)NCCCN(C(c2nnsc2-c2ccccc2)=O)CC)CCOC1 c1(C(N2CC(CNC(CSC(C)(C)C)=O)C2)=O)cccc2c1CCCN2 C(=O)(C(C)C(O)CC)NCc1oc(C(=O)NCC(=O)OCC)c(C)c1 C1(n2cc(CN(C)C(c3ccc(Cl)nc3)=O)nn2)CCC(C(C)(C)C)CC1 c1(COC)ncc(C(=O)NC2CC2)s1.c1(C=O)cnn(-c2nccs2)c1.C C#Cc1ccc(CC(N2CC(CNC(=O)CSc3cccs3)C(C)C2)=O)cc1 c1(C(=O)NCC(CO)NC(C(CC)F)=O)ccc(C(=O)O)cc1.C(C)(C)C Cn1cc2c(n1)CCN(C(=O)CC1CN(Cc3c(Cl)cccc3Cl)CCO1)C2 c1(C(=O)NC2CCN(C(COCCSC)=O)C2)ccc(OC(F)F)cc1F c1(C(N2CC(C)(NC(C3C(C(C)O)C3)=O)C2)=O)ccc(C(F)F)c(F)c1 N1(C(c2c(C)nc(C)[nH]2)=O)CC(NC(=O)C(O)Cc2ccccn2)C2(CCC2)C1 C1(=C(C=O)F)CCCCC1.C(=O)(CC1CC1)N(CC#C)CC1CC1.C CCCCC(C)CCC(=O)N1CCN(CCN(C(=O)CS(=O)CC)C)CC1 C12(CNC(N3CC(OCCOC)C3)=O)CC1CN(Cc1ccccc1)C2 C#Cc1cc(F)c(C(=O)NCCCCCCNC(=O)C(C)(C)CF)c(F)c1 N1(Cc2cc(OC(CC)C)c(OC)cc2)CCCC(B(O)O)C1 CCC(C(=O)NC(CC(=O)NCC1CCC(=O)NC1C)C(F)(F)F)C(F)(F)F N1(C(C(C)CO)=O)CC2(CCC(CNC(C3CCCC4CC34)=O)O2)C1 C1(NC(C2(C(N)=O)CCC2)=O)CCC2CCN(C(c3ccnc(F)c3Cl)=O)C1C2 N1(C(C(C)C(F)F)=O)CCOCCC1C(N1CCN(C2CCC2)CC1)=O c1(C(=O)N)cccc2scnc12.CC1(CNC(=O)C=Cc2ccoc2)CCCC1 Cc1cc(OCC(=O)NCC2CN(C(=O)CC3CC3(Cl)Cl)C2)cc(C)c1Cl CCS(=O)(=O)c1ccccc1CC(=O)NC1CC1NC(=O)CC(C)n1cccc1 CC1=C(C(=O)N2CC3CC(NC(c4cc(Cl)ccc4Cl)=O)C2C3)C(=O)OC1(C)C c1(C(=O)NCCOC2CCN(C(C3CC3F)=O)CC2)cc(O)ccc1O O=C(C1Cc2ccc(F)cc21)NCCOC1CN(C(C2CCCOC2)=O)C1 c1(C(N2CCC(C3N(C(C4C(OC(C)=O)C4)=O)CCC3)C2)=O)cc(C)nn1C N1(C(C=Cc2ccc(CC)o2)=O)CC2CC1CN(C(C1CCC13CCC3)=O)C2 c1(C(=O)NC2CCC(NC(c3cncs3)=O)C2)cccc2c1COC2 C1(C(=O)NCCOC(CNC(C(CC)=CC)=O)(C)C)CCCN1C=O C1(O)(CCNC(C(CCC)N(C)C)=O)CCN(C(=O)C2=CCCCC2)CC1 c1(CNC(C(COCC)NC(=O)C(C)n2cccn2)=O)ccc(F)cc1O C12(C(=O)NCC(CO)NC(CCC3(C)CC3(F)F)=O)CCC(CC1)C2 N1(C(CCC)=O)CCOCC1CN(C(=O)CC(O)Cc1ccccc1)C C(C(=O)NC(C)CC)(C(C)C)(C(C)C)NC(C)=O.c1(C=O)cccc(C)c1C C1(NC(CCCSC)=O)CCC(CN(C)C(c2c[nH]cc2C)=O)CC1 c1(OC)cccc(C(=O)NCC2CCN(C(C3C(C)C3(F)F)=O)C23CC3)c1 C1(C)COCCN(C(=O)C(CC)C2CCC(=O)N2)C1.C1(OC)CC(C(=O)N)C1.C C1(C(N(CC(C)NC(C2(C)CC(F)(F)C2)=O)C)=O)CN2CCCN1CC2 CC(N=[N+]=[N-])C(=O)NC1CCCCC1NC(=O)CCc1nccn1C C1(C(N(CCCN(C)C(c2c[nH]c(C#N)c2)=O)C)=O)CN2CCN1CC2 c1(-c2cc(C(=O)N=c3cc[nH][nH]3)c(F)nc2)ccc2scnc2c1 c1(NC(=O)NC(C2(O)CCCC2)CC)ccc(C2CC2)cc1C C(C(=O)NCC1CC2(CC2)C1)(C(C)CC)N(C(c1c(CC)c[nH]n1)=O)C S(=O)(=O)(c1cc(C(=O)OCC)c(Br)cc1Br)NC(C(=C)Cc1ccccc1)=O c1(OC)ccc(C(=O)NCC(C)(C)C)c(C)c1.c1(C(=O)N)sc(C#N)cc1Cl N1(C(C(C2(O)CN(C(c3cc(C)[nH]c3C)=O)C2)F)=O)CCC(F)C(F)C1 c1(C(=O)NCC2CN(C(CSC)=O)CC2C)cncc2cc(Cl)ccc12 C1(C(N2CCC(C)(NC(C3CC3F)=O)CC2)=O)CSC(c2ccccc2O)=N1 C1(NC(C2(C=C)CCC2)=O)CC2COCC(C1)N2C(C1CCCO1)=O C1(C(N(C(C)C)CCO)=O)CCN(C(=O)C(C)(C)C2CC2)O1 Cc1cc(C(=O)NC2CCCN(C(=O)COc3ccc(Cl)cc3)C2)ncc1C#N n1(CC=O)ncc2ncccc12.c1(C(N(CCC)CC)=O)csc(C(C)C)n1.N CN1CCCC(CC(=O)NC2(C(=O)N)CC2(C)C)C1.c1cc(C(N)=O)co1.C CCCC(C(=O)NCC(c1ccncc1)C)NC(=O)CCNC(N)=O N1(C(C2(CC)CCCN(C(=O)Cc3cc(C)no3)C2)=O)C2CCCC1CN(C)C2 C1(NC(c2cc(C3CCC3)no2)=O)CCC(Cn2ccnn2)C1.n1(C)cccc1 n1(CC)ncc(C(=O)NCCCC(C)NC(=O)CC2CC3(CC3)C2)c1Br c1(C(=O)NCCCN(C(COCC)=O)C(C)C)ccc(F)c(Cl)c1 C1(C(=O)NCC2(C=C)CCC2)(CNC(=O)CC(C)O)CC2(CC2)C1 CC1(C)C(CO)CN1C(C1CCN(CC2CCNC2)CC1)=O C(c1ccccc1)=CC(=O)NC1C(CNC(C(C)C)=O)CCC1.C(C#N)O c1(C(N(C)CC2CCN(C(=O)C(F)(F)CO)C2)=O)cc(F)c(N)c(F)c1 c1(COC)nc(CC(=O)N)cs1.C(=O)(C(CN(C)C)N(C)C)N(C(C)C)C C1(C(=O)NC2(COC)CC=CC2)(CC)CCCN1C(C1CCC(=O)C1)=O c1(C(=O)NCC(CC)NC(c2cnc(N)cn2)=O)nnc(O)c(Br)c1O C=CCC(C(=O)N1CCC2(CCN(C(c3ccc(NC)cn3)=O)C2)C1)C(C)(C)C N1(C(c2scnc2Br)C(=O)NCC)CCC(C(N2CCCC2)=O)CC1 c1(C(C)(C)C)ccc(CNCC#CCNC(=O)O)c(O)n1.c1ccccc1.C CCC(C)(C#N)C(=O)NCCC(O)C(=O)N(CCS(N)(=O)=O)C c1(CCC(=O)NC(CCNC(C(F)OC)=O)C)cnc(C)o1 c1(C(N2C(C)C(NC(=O)CCc3cccs3)CCC2)=O)ccc2c(c1)ncn2C C1(O)(CNC(C2C(CC)OCC2)=O)CCCN(C(c2sccc2F)=O)C1 c1(NC(c2c(OCC)cccc2)C)ccc2c(c1)CCCC2O Cc1oc(CO)cc1C(=O)NC.C1(C(C)(C)C)CCN(C(c2cnn[nH]2)=O)C1 C(C1C(C)C1(Cl)Cl)=CC(=O)N.C(=O)CC(c1ccccc1)N(C)C.CCCC c1(CCC)sc(C(=O)NC(C)(C)CNC(C2CCN(CC)CC2)=O)cc1.C Cc1csc(CNC(c2csc(CNC(C3CCCCO3)=O)c2)=O)c1 C1(CC#C)(C(=O)NCC2C=CCCC2)CCCNC1 C1(C(=O)NCCCCCNC(CN(C(C)=O)C)=O)(CO)CCOCC1 C1(CC(N2CC(CC)C2)=O)N(C(=O)CNC(C2CC2C)=O)CCC1(C)C N1(C(CC2(C)CCCC2)=O)CCC(C)(CCNC(C2CC(N3CCCC3)C2)=O)C1 c1(C(=O)NC2CS(=O)(=O)C2)nnc2ccc(-c3ccc4sccc4c3)cn12 N1(C(c2c(OC)cccc2)=O)CC(CNC(=O)CCCF)CCC1C N1(C(c2nnc(C)s2)=O)CCCCC1CN(C)C(C1CC1(C)C(F)(F)F)=O c1(C(=O)NCC(CNC(C2(C#C)CC2)=O)CO)c(C(F)(F)F)coc1C c1(NC(C2CCC(NCc3scnc3Cl)C2)=O)cc(CO)ccc1Cl c1(C(N2CCCN(Cc3cccc(Cl)c3)CC2)=O)c(Cl)ccc(F)c1F CC1CN(C(c2cccnn2)=O)CC1CNC(c1sc(Br)cc1Cl)=O c1(C(N2CC(NC(C=CCC)=O)C2)=O)cc(Cl)on1 c1(CN)nc(N2CCOCC2C2CCCC2=O)cc(Cl)n1 C(CC(C)C(=O)NCC(N1CCN(C(=O)C(CCN(C)C)N(C)C)CC1)=O)OC c1(C(N2CC(CC)NC(=O)C2)C(=O)NCCOC)cc(Cl)cc(C#N)c1 O=C(C1=CCCO1)NCC1CCCC(NC(c2csc(C3CC3)n2)=O)C1 c1(C(N2CC(CN(C(c3nccc(C)n3)=O)C)OCC2)=O)c(C)cc(F)cc1C CC1(C)CC(C(=O)N2CCCC2C(C)(C)CNC(c2ccoc2)=O)=NO1 Cc1ccc2cc(C(=O)NC(C3CCN(C(=O)C4=CCCC4)C3)(C)C)cn2c1 c1(C(=O)NC2CC(C(=O)Nc3ncn(C)n3)C2)ccc2c(c1)n(C)c(=O)n2C C1(CNC(CCN(C)CCO)=O)CN(C(=O)CCCCc2cnn[nH]2)C(C)(C)C1 C(=O)(CN=c1cc[nH]cc1)N1CCC(c2c(CNC(C(CC)SC)=O)c[nH]n2)C1 c1(NC(C2CC(=C)CN2C(=O)CCOC)=O)ccc(C(N)=O)nc1Cl C(CC(C(C)(C)C)NC(c1csc(O)n1)=O)N(C(C(C=C)(C)C)=O)C c1(OC(C)C)cnc(C(=O)NC2CCCN(C(C3CC3(C)C)=O)C2)cn1 C1(CC#C)(C(=O)O)CN(N(C)C(C)C2CCCCC2)CCO1 c1(CN(CCCNC(=O)C(C)C)C(c2c(C)onc2)=O)ccc(F)c(F)c1 c1(C(=O)NCC(CCNC(c2c(C)[nH]nc2Cl)=O)O)ccc2ccsc2c1 C(=O)(C1=CCCOC1)N1C(CC(=O)NC2CCC(C(N)=O)CC2)COCC1 C1(O)(CNC(C(c2cnn(C)c2)C)=O)CCCN(C(C2CCC2)=O)CC1 N1(C(c2cc(OC)no2)=O)CCCN(C(=O)Cc2ccccc2C(C)C)C(C)C1 C=C(C)CC(C(=O)NOCC(O)C(C)C)NC(C12CCC(C1)C2)=O N1(C(C=C(CCC)C)=O)CC(C)(C)OCC1CNC(C1CC1C#N)=O c1(C(=O)NC(CC(C)NC(C(CC)CC(F)F)=O)C)cc(C)cc([N+](=O)[O-])c1N N1(CC(=O)NC2COCC2n2cc(CC(CO)C3CC3)nn2)C(=O)CCC1CF c1(-c2ccc(COC)c(C)c2)ccc(C(N2CCc3ccsc3C2)=O)c(C)c1F C1(C(=O)NC2CCCC(NC(c3c(C)onc3)=O)C2)Cc2ccc(F)cc2O1 C1(C(=O)NC2CC2c2nc(Cc3nn[nH]n3)no2)(CC)CC1(F)F C1(C)(CNC(CCC=CC)=O)CN(C(=O)C(C)Cc2c(C)noc2C)CCO1 C1(C(C(=O)NC(C)(C)C)N(CCCOCC)C)CCCC1C C(=O)(CCC(CC)NC(c1ccn(C2CC2)n1)=O)NC(CC)C(N)=O c1(CC(=O)NC2CC2C(=O)Nc2cncc(Br)c2)cc2ccccc2s1 C(C(O)CC(=O)NCC1(O)CC(NC(=O)CSC2CC2)C1)N(C)C c1(C(N(c2nc(C#N)cc(C)n2)C2CCC(N)C2)=O)cc2cc(F)ccc2s1 CC1SCCCC1NC1CCN(c2ccccc2OCc2ccccc2)C1=O C1(C(=O)NCC(CCOC)NC(=O)CN2CCCCCC2=O)COC2(CCC2)C1 c1(C=O)ccc2c(c1)C=CCC2.Cc1cc(C(=O)NCC(F)C)n(C(F)F)n1.N N(C1CC2(CN(C(=O)CC(C)C)C2)n2ccnc21)C(c1cc(CCC)on1)=O Cc1ccc(C(C)C(=O)N2CC(NC(=O)CSc3nccn3C)C2)cc1 Cc1cc(C(N2CC(NC(C3COC(=O)C3)=O)C(C)(C)C2)=O)nnc1O O=C(C1=CC2CCC=CCCC12)NC1CCCN(C(=O)CCn2cnnn2)CC1 c1(OC)coc(C(=O)NCC(C)N(c2cc(C(C)(C)C)nc(Cl)n2)C)cc1=O N1(C(C=CCCC=C(C)C)=O)CC(C2(NC(=O)CC3OCCCO3)CC2)C1 Cc1cncc(C(=O)NC2CCC(NC(=O)C(C)(C)C3CCCO3)CC2)n1 N1(C(C(F)=CC)=O)CCC(NC(c2cc(C)ccc2OC)=O)C(F)C1 N1(C(c2cnn(C(C)C)c2Cl)=O)CCCC12CCN(C(c1nnc(S)n1C)=O)C2 c1(C=O)ccc(=O)n(C)n1.C(C(C)(O)CNC(C1(C)CC1)=O)N(C)C.N Cc1cc(C(N2CC(N(C(=O)CSC3CC3)C)C(C)(C)C2)=O)nc(C)c1 N1(C(C23CC(OC)C2C3)=O)CCCC1(C)C.C1(C=O)CCC(C(N)=O)CC1.N c1(C(=O)NCC(CC)NC(=O)C(c2cnn(C)c2)C)scnc1C(C)C c1(OC)ncc(C(=O)NCCC2CCN(C(=O)Cn3[nH]cnc3=N)CC2)cc1C c1(OC)cc(C2(C(=O)NC(C)CCCC)CC2)ccc1Cl.C(=O)CC1CCC1.N CC1CCN(C(C23CCC(F)(CC2)CC3)=O)CCN1C(=O)C(N)=O Cc1cc2c(cc1Br)N(C(c1ccc(F)c(Cl)c1F)C(=O)NCCC#N)CCC2 c1(SCC(=O)NC2C(NC(c3cnc(N(C)C)o3)=O)CCC2)ccccc1Cl c1(C(N(C2CCN(C(=O)C(C)(CC)CCC)C2)CCC)=O)ccc2nncn2c1 c1(C(N)=O)n[nH]c(=NC23CCC(CON)(C2)OC3)s1 C1(CCNC(c2n(CCC)nnn2)C(C)CC)COC(C)(C)C1 C1(NC(C(CC)c2ccccc2)=O)CC2CCC(C1)N2C(=O)COC1CCOC1 C(c1cnn(C)c1)=CC(=O)NC(CNC(C=C(COC)C)=O)CO C=CC(C)(C)CC(=O)N1C(C(=O)NCc2nc(C)c(C)s2)CCC1C(C)C C(=O)(C(O)CCC(C)C)NCCNC(c1c(CC)ccs1)=O CC1(C)CC(C)CN(C(=O)CNC=O)C1.C1(C(=O)N)CC1.C(=O)C1CC1 c1(N2CCC(CNC(C3CCCC(C)C3)=O)CC2)ncc(C#N)cc1Cl CCC1=C(C(=O)NCC(C)NC(=O)CC(=O)NC2CC2)CCCO1 C1(CC(=O)NCC2C(C(N(C)Cc3nncs3)=O)C2)COC(=O)C1 c1(CC)nc(CNC(=O)CC2CCN2C(c2c[nH]nc2CC)=O)co1 C12(CNC(C(N3CCN(C)CC3)C)=O)CC1CN(C(=O)Cc1cnn(C)c1)C2 Cc1nc(NC(C2(N)CC23CC3)=O)cs1 c1(C(N2CC3N(C(Cn4c(C)ccn4)=O)C(CC3)C2)=O)ccnc2ncccc12 C1(NC(c2csc(C(F)(F)F)c2)=O)CCN(C(c2ccncn2)=O)CCC1CO N1(C(C2N(Cc3c(C)cccc3C)C3C(C2)C3)=O)CCN(C)C(=O)C1C CC1=C(C(=O)NC2CCN(C(=O)CCC3CC3)C(C)C2)CCO1 N1(C(c2c(C)ncs2)=O)CCCC(C)(NC(=O)CCn2ccc(O)nc2=O)C1 N1(C(C(CN(C)C)O)=O)CC(C2CCCN(C(C3(S(C)(=O)=O)CC3)=O)C2)C1 O=C(CC(F)(F)c1ccccc1)NCC(O)CCNC(C1CCC1(F)F)=O C1(C(=O)NCC(CC)NC(c2cc(Cl)ccc2N)=O)CCc2nnc(O)cc2C1 c1(C(C)C)cc(C(=O)NC2CC2NC(C2CC(C#N)C2)=O)n(C)n1 Cc1cc(C(N2CCCC(N(C)C(C3CCCN3C)=O)C2)=O)c2scnc2c1C C(C(C)(C(=O)NC1(CCCCO)CC1)NC(C1CCNC(=O)C1)=O)SC C(CC)(CCC(=O)NC1(C(=O)OC)CC(C)C1)NC(c1ccc(CC)cc1)=O C#CCCCCC(=O)N(C)C(c1cn(Cc2cccc(C)c2)nn1)C c1(-c2cn(Cc3c(CC)nco3)nn2)cccc2cnccc12 C(CCC(O)C(=O)N1CC2C(CO)C2C1)NC(c1ccc(CO)s1)=O N1(C(C(C2CCOCC2)OCC)=O)CC(C)(C)CC1C.C(=O)C(C)(C)C.N O=C1NC2(C(=O)NCC3CCN(CCCC4CCC4)C3)CC3CC1C2C3 c1(C(=O)NC2CCN(C(COCC(C)(C)C)=O)CC2)cnc2occc2c1 CCCC(C#N)C(=O)NCC1(F)CC(NC(=O)CSc2cccc(C)c2)C1 O(N1CCC(CC(=O)NCC2CCCC2NC(C2C3COCC23)=O)CC1)CC C(CCC1CC1)(C(=O)NCC(=O)N(C)OC)NC(CCCNC(=O)OC)=O N1(C(C(CCC)C#N)=O)CCCN(C(c2cn(C)c(=O)nc2O)=O)C(C)C1 c1(C(=O)NCC(CNC(C(C)OCC(C)C)=O)C)nc(F)ccc1Cl C1(NC(=O)C(Cl)Cl)CCC(C(=O)NCC2(F)CC(O)C2)CC1 C12(NC(CCN3CCC(C)CC3)=O)COC(C1)C(NC(C1CN(C)C1)=O)C2 Cc1cc(C(N2CC3CN(C(C4CC45CC5)=O)CCC23)=O)ccc1[N+](=O)[O-] c1(C(N2CCC(C(C)(C)NC(C34COCC3C4)=O)C2)=O)ccc2cc[nH]c2n1 C1(NC(CCc2n(C)ncn2)=O)CCC(F)(C)C1.c1(C=O)coc(C(F)F)n1.N C1(CC)C(=O)N1CCOCCO.CCC(CC)NCC=O.N(C)C c1nc2ccccc2o1.c1(C(=O)NO)cccc(C(F)(F)F)c1 C1(NC(c2cnc(O)c(Br)c2)=O)CCCN(C(c2cc(Cl)cc(Br)c2)=O)CC1 Cc1[nH]c2cc(Br)ccc2c1C(=O)NC1CCOCC1NC(C1CC1F)=O N1(C(C(CC)=CCCC)=O)CC(C)CCC1C(=O)NCC1CCSC1 CC(C(O)C(F)F)NC(=O)C(C)(C1CCC1)NC(c1coc(C(N)=O)c1)=O c1(OC)ccccc1C(C)NC1CCN(C(=O)CSc2cccs2)C1 CC1CCc2cc(C(=O)NCCNC(=O)CC3CCCN3C)ccc2N1 c1(NC(C(CCC2CCC2)NC(c2cc(CC)no2)=O)=O)cnc(Cl)c(C)c1 Cc1ccc(NC(=O)C)cc1.C1CC(C2(C(F)(F)F)CC2)C1.C(=O)(C)N N(C1CCc2cccnc21)C(C1CC2(CC2)CN1C(c1ccc(Br)c(Br)c1)=O)=O c1(C(C)NCC(c2cc(OC)c(Cl)cc2)F)nc2c(s1)COCC2 c1(OC)ccn2ncc(C(=O)NCC#CC)c2c1.C(=O)(CC1=NN(C)C(=O)C1)N Cc1nnnn1CC(=O)NC(C1(C(=O)NC2CC3CC3C2)CC1)C c1(NC(=O)NCCc2nc(C)oc2)ccc(Cn2cncn2)cc1 N1(C(c2cc(OC)ncc2)=O)CCCC(CNC(C2CCCC(F)(F)C2)=O)CC1 CCCCCC(F)C(=O)N1CC2CCC1CN2C(C1COCCN1C)=O C1(C(N(C2CCCOC2)C)=O)(CNC(c2cnc(O)o2)=O)CCCO1 C(=O)(C(CC1CCCCO1)N1CCC(c2ncccn2)C1)NCCC C(c1ccccc1F)=CCC(N1CCC(C)(CNC(C(CC=C)C)=O)C1)=O n1(CC)cc(C(=O)NC2CCOCC2C(=O)NC)c(C)n1.c1c(C)noc1C.C Cc1csc(CC(=O)N(CCCOCCN(C(=O)C(C)C2CCC2)C)C)c1 C(=O)(C1=CCCCC1C)NCCC(C)NC(=O)CN1CC=CC1 N1(C(COCCOCC)=O)CC2(NC(=O)CCc3cc(Cl)no3)CCC1C2 C1(C(=O)N(C)OCC(F)(F)F)(COC)C=CCN1C(=O)CSC1CC1 c1(CCCC)ccc(C(=O)NNCN2CCC(O)CC2)cc1[N+](=O)[O-] Cc1cc(CC(=O)NC2(C(=O)NCC(N3CCCCC3)=O)CC(O)C2)n[nH]1 C(=O)(CCCCC(C)=O)N1CC(CCC=C)(C(=O)NC(C2CCOC2)CC)C1 C1(NC(CSCC=C)=O)CCN(C(C23CCCCC2C3Br)=O)C1(C)C c1(C(=O)N)ccc(F)c(Cl)c1F.C1(NC(CC2(OC)CC2)=O)CCC(CC)C1 N1(C(c2ccc(OCC3CCCC3)s2)=O)CCC2(CCCN(C(=O)CO)C2)CC1 Cc1c(Cl)ccc(C(=O)NC(C2CCN(C(c3nn(C)cc3Cl)=O)C2)C)c1O c1(OC)ccc2c(N3CCC(O)(C(C)NC(=O)C(C)C)C3)c([N+](=O)[O-])cnc2c1 c1(C(N2CCC(C(=O)NCCCC)(C(C)C)C2)=O)cccc(C)c1C c1(C(C(F)F)NC(CCCc2onc(CCC)n2)=O)cccc(Cl)c1 c1(-n2cc(C(C=C)(C)O)nn2)ccccc1CCC(=O)NCCN1CCOCC1 C1(C)(CC)CCCN(C(=O)C(C2CCCC2)NC(c2cn[nH]c2)=O)CC1 c1(C(=O)NCCC(C)C)ccc(C(F)F)cc1F.c1(C(=O)N)cc(O)nc(O)n1 C(c1ccccc1F)=CCC(=O)NC(CC(C)C)CNC(C1CSCCS1)=O C(C)(C)(CC(=O)N(C1CCC(NC(=O)CCn2ccnn2)CC1)C)OC CC(C)CC(C)C(=O)NC1(C)CCN(C(=O)COc2cc(Cl)ccc2Cl)C1 C1CC(C)(C)OC1(C)C.C(C)(C=O)(N(C(=O)CCc1ccn(C)c1)C)C1CC1 c1(C(=O)NC2CCC(N(C)C(C3CN4CCN3CC4)=O)C2)ccc2c(c1)CCC2 c1(C(=O)NC2C(NC(c3cn(CC)nc3)=O)CCCC2)c(C)ncnc1O CC1CNc2c(C(=O)NC3CC34CC(NC(=O)CN(C)C3CC3)C4)cnn2C1 Cc1cc(NCCc2cc(C(F)(F)F)ccn2)c([N+](=O)[O-])cc1C(=O)O C12(C(N(C3CCN(C(COC(C)=O)=O)CC3)C)=O)CCN(CC1)S(=O)(=O)C2 C1(NC(C(COC)NC(c2cc(O)ncn2)=O)=O)CCCCC1(C)C CN=c1ccc(C(N2CCC(OCCNC(C3C4CCCC34)=O)C2)=O)c[nH]1 C1(CC(=O)NCC(C)(CO)NC(c2c(C)ncs2)=O)COCC(C)(C)O1 C1(NC(c2ccc(CNC(C)=O)s2)=O)CCCCC1.C1(Cl)(C=O)CC1.C N1(C(c2cc(C)[nH]c2)=O)CCC2(NC(=O)C(CO)c3ccccc3)CCCC12 c1(C(N)=O)nccnc1C(=O)NC1CC(C)C1.N1(C=O)CCCC1.C(=O)C CN1CCN(C)C(C(N2CCOCC2CC(=O)NCCC(C2CC2)C2CC2)=O)C1 c1(CC)cc(NC(C2CCC(O)CN2C(=O)C(CC(C)C)N(C)C)=O)cc(C)c1 N1(C(CC=CC(C)(C)C)=O)CCC(O)C1C(=O)NC1CC1(C)C C1(C(=O)NC(C)C(=O)O)CCN(C(C23CC(F)(C2)C3)=O)C1.C(C)(C)C C1(CC(=O)OCc2c(OC)cc(OC)c(C(=O)O)c2)COc2ccccc2C1 C1(C(NC)=O)CC2C=CC1C21CC1.N1(C(C2(SCC)CC2)=O)CCCCC1.C C1(CC(=O)NCC2(NC(CC(CC)OC)=O)CCCCC2)C(=O)N(C)N=C1C C1(COCC)CCCCN1C(=O)CC1CCCN1C(=O)Cc1cc(C)[nH]n1 N1(C(C(CC)=CC)=O)CC2CC(N(C)C(c3cn(CCC)nc3C)=O)C1C2 N1(C(C(C(C)(C)O)F)=O)CCC2(CC1)CC2CNC(C12CCCC1CCC2)=O C(=O)(CC(=O)N(C)C)NCC=CC(=O)NC(C)Cn1cccn1 C1(CCC)CN(C(=O)C(C)O)CCN1C(=O)CC(C)(C)c1ccc(F)cc1 C1(C(=O)NCCSCC(=O)N(C(CC#C)C)C)CC2(CCC2)C1 c1(C(N2CCC(N(C(CC3CC(=C)C3)=O)C)C(C)C2)=O)csc2ccc(C)cc12 C(=O)(C(O)CCC(F)(F)F)NC(c1ccccc1)CNC(CC(C)C(C)(C)C)=O CC(C)C(c1ccccc1O)NC(C1(O)CC(O)C(O)C(O)C1)=O C1(CC)CCCC1N=c1[nH]c(N2CCN(C3CCN(C)C3=O)CC2)nc2ccsc12 Cn1cnnc1SCC(=O)NCC(C)(CO)NC(=O)C(F)OC(F)(F)F C1(CC(=O)NCC=CC)CCN(C(c2ccc(C)cc2C)=O)C1(C)C C1CC2(C1)CN(C(C1CCC1)=O)C2.C1(CC#C)(C(=O)N)CCOC1.N(C)C C1(CNC(COC(C)C)=O)CC2(CC(NC(c3cc(Cl)ns3)=O)C2)C1 c1(C(N2CC(NC(C3(c4ccc(C)cc4)CC3)=O)C2)=O)ccc(O)c(C)c1 Cc1csc2c(C(=O)NCC(C)N(C)C(C3COCCC3(F)F)=O)cccc12 C1(CNC(c2[nH]cc(CC)c2)=O)CC2COCC2N1C(=O)CN1CC2CC2C1 Cc1cc([N+](=O)[O-])cnc1NCCNC(=O)C(C)CCCc1ccccc1 c1(-c2cc(C(=O)N)n[nH]2)ccccc1F.C12(C(N3CC(CC)C3)=O)CC(C)C1C2 C(C(C)C(C)C(=O)NC1(C)CCCCC1)OC.c1(C(=O)N)cc(=O)n(C)cn1 c1(C(N2CC(CC=C)C2)=O)cccn2nnnc12.C1(CC(=O)N)COC(C)(C)C1 c1(C(C)(C)C)cc(Br)ccc1NC(C1CC2CC2N1c1ccncn1)=O C(CNC(C1CC2CCC1O2)=O)(CCCC)NC(C1(CC#C)CC1)=O c1(OCC)cc(C(=O)NCC(c2ccccc2)(O)C2CC2)sn1 c1(C(N2CC3CN(Cc4cnc(C5CC5)s4)CC3C2)=O)cc(Cl)cc(Cl)c1O C(C)(CCCC(=O)NC1CCCCC1OC)NC(c1ccnc(OC)n1)=O CC1CCN(C(c2coc(O)n2)=O)CCN1C(c1cn(C)ccc1=O)=O CC1CCCCC1(CNC(C1(S(N)(=O)=O)CC1)=O)NC(c1ccoc1)=O N1(C(C2N(CC)CCCC2)=O)CC(NC(=O)CCc2ncccn2)CC2(CC2)C1 c1(CC(C)(C)O)cccc(N=c2ncc3cc(Br)cc(F)c3[nH]2)c1 C1C(C2CC2)CCN1C(c1cocc1C)=O.C(C(=O)N)(C(C)(C)C)NC(C)=O N1(Cc2ccc(N3CCN(CC)CC3)cc2)CCN(C(=O)C(C)N(C)C)CC1 N1(Cc2c(O)ncc(C)c2)CCc2sc(-c3ccc(F)s3)nc2C1 c1(C(=O)NCCCN(CCCNC(=O)CCF)C)cc(Cl)nn1C C1(CNC(C(C)OC(CC2(OCC)CCC2)=O)=O)CSc2ccccc2O1 CC1CCC(N(C)C(=O)NC2CN(C(c3cnc(=N)[nH]c3)=O)CC2O)CC1 c1(C(N2C(C3(C(=O)NC(C=C)(C)CC)CC3)CCC2)=O)ccc(C)nc1O Cc1cc(=O)c2cc(C(=O)NC3CCCN(c4ccccn4)C3)ccc2[nH]1 c1(C(=O)NCC(CC)NC(C2(CCC=C)CC2)=O)ccc2nc(O)[nH]c2c1 CC(C)C(O)CC(=O)NC(C(=O)NCCN1CCC1)C(C)(C)C N1(C(C(C)=CC2CC2)=O)CC2(C)CN(C(=O)CC3(O)CCC3)CC2(C)C1 C(c1cc(C)c(C)cc1C)=CC(c1nnnn1C)NC(C(=O)NCC)C C#CC1(C(=O)NC2CCC(=O)NC2C)CCN(C(=O)C(N2CCCCC2)C)CC1 N(C(=NCCOC1CCOCC1)NCc1cc(C(C)(C)C)on1)CC(C)(C)C c1(N2CCC(N(C)C(c3cccc(F)c3F)=O)C2)nccn2nnnc12 C1(CNC(COCC(=C)C)=O)CN(C(=O)CSCC(C)C)CC1(C)C CC(CC(=O)N=c1cc2n([nH]1)CCCC2)NOCCC(F)(F)F N1(C(c2cn(CCC)nn2)=O)CCCC1(C)C(=O)Nc1ccc(C2CC2)nc1 N1(C(C2N(C(CCC)=O)CC(O)C2)=O)CCC2(CC1)OCCO2 Cc1nc(CNCc2cccc(F)c2)n(C)c1C c1(C(N2CCC(O)(CCNC(C(C(C)C)OC)=O)C2)=O)ccc2cncn2c1 C1(C(=O)NC(C(=O)OC)CCF)CC(O)C(O)CC1.C(=O)C(C)=C1CC1.C N1(Cc2c(NC)cc(Cl)cc2)CCC2CN(c3nc(Cl)c4c(n3)COC4)CC2C1 C#Cc1ccc(C)cc1.C(=O)(C(F)CC1CN(C(c2ocnc2C2CC2)=O)C1)N C1(CNC(=O)CC(F)(F)F)CC(F)(F)CN1c1cc(C(F)(F)F)ncn1 N1(C(c2c(C)nco2)=O)CCN(C(=O)Cn2nc(C3CC3)n(C)c2=O)CC1CF CC1=C2CC(NC(=O)N(CC(C)C)C)CN=C2NN1.c1cn(C)nc1C(C)C Cc1cnc(C(=O)NC(c2ccnn2C)C(=O)N(C(C)C(C)(C)O)C)c(C)c1 c1(C(N2CCC(F)(C(N3C(C)CCC3CO)=O)C2)=O)c(Br)cc(F)c(F)c1F c1(CNC(C2(C)CCN2C(c2cc(C#N)c[nH]2)=O)=O)ccc(I)cc1Br c1(C2N(C(=O)C(F)(F)C3(O)CCCC3)CCC2)cc(F)cc(F)c1 c1(C(N2C(C(CNC(C3(C)ON=C(C)C3)=O)(C)C)CCC2)=O)nccc(Cl)c1F C1(CCC(=O)N(CC(C)N(C(CC)=O)C)C)(C=O)CCCC1.C#CCCO C1(C(=O)NCC(CC(C)C)NC(=O)CCc2ccc(Cl)nc2)CN2CCC1CC2 c1(C(=O)NCC2(C(=O)NCc3conc3)CC(=C)C2)ncncc1OC C(Cc1cn[nH]c1)(C(=O)Nn1cnn(C)c1=S)NC(CN(C)CC)=O C1(N(C(=O)COCCCF)C)CCC(NC(c2cc(C3CC3)no2)=O)CC1 C1(CNC(C2N(C)CCC2)=O)CC2CCC1N2C(c1ccnc(Cl)c1F)=O C1(NC(C2=C(C)OCC2)=O)CC2CCCC(C1)N2C(c1ccc(F)cn1)=O N1(C(C2=CCCC2(C)C)=O)CCC(C2CCN(C(C34CCCC3C4)=O)CC2)C1 n1(CCOC)cc(C)c(=NC(=O)N(CCC2CC2)CC2CC2)[nH]1 c1(C(N(C2CN(C(C3(C4CCCCC4)CC3)=O)C2)C)=O)ccc([N+](=O)[O-])cc1N c1(OC)ccc(CCC(=O)NCCC2CCCN2C(=O)Cc2ccsc2)cn1 c1(C(=O)NCC(O)CCNC(C2CC3CC3C2)=O)cc2n(c1)CCCC2 C1(CNC(c2ccnnc2)=O)CCCC2(CCN(C(C34CCC3C4)=O)CC2)O1 C(CN=c1[nH]c(=NCc2cnns2)[nH]c2ccsc12)(C1CCOC1)OC c1(C(=O)NCC2(O)CN(C(C3(COC)CCOC3)=O)C2)cncc(O)c1 C(=O)(C1CCCn2cnnc21)N1CC2C(N(C(c3cc(C)cc(C)c3)=O)C)C2C1 Cc1ccc(Cl)c(F)c1C(=O)NCC1CCN1C(C1CN(C(C)C)C1)=O C(=O)(C(CC(C)C)OC1CN(C(=O)CCC2CC(C)C2)C1)OCC c1(OC)cccnc1C(=O)NCC1CCCCC1.c1n[nH]c(=N)s1.C(=O)C.N CC(C)C(C)(CNC(=O)C(O)CN(C)C)NC(=O)CC1CCC(=O)NC1 C1(NC(c2c(C)onc2Cl)=O)CCN(C(c2ccoc2C(C)C)=O)CC1O CON1CC(C(=O)NCC2CN(C(=O)Cc3ccc(C)cc3Cl)C2)CC1=O C(CC(O)CC(=O)NCC(C)(C(C)C)NC(=O)CCC=CC(C)C)SC N1(C(c2cc(OCC)no2)=O)CCC(C(=O)NC2C(O)CC2O)(CO)C1 c1(C(=O)OC)ccc2c(n1)CN(C(=O)COc1cc(OC)ccc1Cl)C2 N1(C(C(CSCC)NC(c2nnc(O)nc2O)=O)=O)CC2CCC(O)C2C1 C1(NC(c2c(CC)nccn2)=O)CCC2CC1CN2C(c1cnc(C)[nH]1)=O Cc1cnnc(O)c1C(=O)NCC1C(C)CCN1C(C1OCCO1)=O C(N=c1[nH]c(C)cc(=NCc2cc(Cl)sc2Cl)[nH]1)C1N(C(C)=O)CCC1 N1(C(Cc2c(C)noc2C)=O)CC2(C1)SCCC2NC(C1CSCC(=O)N1)=O N1(C(c2c(C(C)(C)C)[nH]cn2)=O)CCCC(C)(NC(=O)CCCC2CCCC2)C1 Cc1nc(C)c(C(=O)NC2CCN(C(=O)CCCC(C)(F)F)CC2CO)nc1C n1(CC(=O)N)ccc(C)cc1=O.C1(C)(C=O)CCC(F)(F)C1.C(C)(C)OC N1(C(C(F)OC)=O)CC(CO)C2(C1)CN(C(=O)Cc1ccn(C(F)F)n1)C2 C(=O)(C1CCCc2c(O)cccc21)N1CC2CN(C(C3CC(C)(C)C3)=O)CC2C1 Cc1nn(C)c(=O)c(C(=O)NC)c1C.C12CC(C1)C(C)O2.C(=O)C.CCF N1(C(=O)Nc2ccc(OC(C)C)nc2)CCc2c(C(=O)O)ccc(F)c2C1 CCC(CC)C(C)C(=O)NCC(CNC(C1CC2CCC(C1)C2=O)=O)CO N1(C(C(C)O)=O)CCN(CC(=O)Nc2ccccc2)CC1 C(CCN=C(NCC1(O)CC2CCC1CC2)N1CCCC(C2(C)OCCO2)C1)OC n1(CCC=O)c(C)cc(O)cc1=O.C1(CNC(CCOCC)=O)CCCC1.N c1(C(=O)OC(CCSC)C(C)C)cc(C)ccc1C C1(C(N2C(C=O)CSC2C)=O)CCC(=O)N(C(C)C)C1.C(=O)(CC)O.CC O(S(=O)(=O)c1cnn2c1OCC(C)(C)C2)c1c(C(=O)OC)cc(OC)cc1 Cc1cc(O)c(C(=O)NC(C)CN(C)C(C2CC=CCO2)=O)nn1 CC1CCc2c(C(N3CC(NC(c4ccnc(Cl)n4)=O)C(F)(F)C3)=O)n[nH]c21 C(=O)(C1=COCC1)N(C1CCN(C(CCc2cnc(C)o2)=O)C1)CCO N1(C(C(C)Oc2c(OC)cccc2)=O)CCN(C(=O)CCC(=O)NC)C(CF)C1 N1(C(C(C)OCC)=O)CC(C2CN(C(=O)Cc3ncc(C)s3)C2)C1 C(CCCC(CO)NC(=O)Cc1cc(C)on1)NC(c1cc(CCC)nn1C)=O C1(CC=C)CCCCC1NC(c1nn(-c2ccccc2)cc1O)=O Cc1cccc2c(SC3CCOCC3N)ncnc12 N1(C(C(CC)NC(N)=O)=O)CCC2CC(C)CCC2C1.C(=O)(CS(=O)(=O)CC)N C(=O)(CC1=CCCCC1)NC(CN(C(c1cnc(C(C)OC)s1)=O)C)(C)C c1(C(=O)N)cc(F)cnc1.c1(C(N2CC(COC)(C)C2)=O)cccc(O)n1 C=CC1CCCN1C(=O)COC1CC(NC(=O)C(c2cnn(C)c2)C)C1 C1(NC(C2CCC(C)N2C(=O)C=Cc2ccc[nH]2)=O)CC(C2CCCC2)C1 CC1(C)CCCC(C(=O)NCCCN(C(=O)CN2CCCCC2=O)CCO)C1 n1(C(C)C)nccc1CC(=O)NCCN(C(C12CC(O)C1C2)=O)C1CC1 NS(=O)(=O)c1ccc(F)c(C2(C(=O)Nc3ccc4nncn4c3)CC2)c1 N1(C(C(C=C)OC)=O)C2CCC1CN(C(c1nccc(N)c1Cl)=O)CC2 O(NS(=O)(=O)c1ccc(F)cc1)CC(=O)NCCC(C)N(C(=O)C(N)=O)C CC1C(NC(=O)C=CI)CCCN1C(=O)CN1CCN(C)CC1 Nc1c(C(=O)NC2(CCNC(c3cccn4nnnc34)=O)CC2)ccc(F)c1F c1(CC)cc(=NC(C)CC(C)NC(=O)C2=CCCS2)[nH]c(CC)n1 C1(CNC(=O)CN2CCCC2CO)CCCN(C(c2ccc(F)cn2)=O)CC1 c1(C(N(CC(C)NC(C(C)OC)=O)C)C)ccccc1Br.C1C(=O)N1 C(CC(F)(F)Cn1cc(-c2nc(C3CC3)cs2)nn1)NC(c1cnc(CC)o1)=O c1(C=O)ccc(Cl)c2occc12.N1(C(CC(=O)OCC)=O)CCC(F)(C)CC1.N C(=O)(C(F)(F)CC)N1CCC(n2ccnn2)C1.N1(CCC)CCCC1C(=O)NC c1(OCC=C)ccc(C(C=O)N(CCCN(CC=C)CCC)C)cc1.C(C)=O CC1C(NC(C2(C)CCC(F)(F)C2)=O)CC2CCC1N2C(C1CCN(C)C1=O)=O C1(CNC(c2c(CC)cc[nH]2)=O)CC(C(=O)N2CCCCC2)=NO1.C1CC1.C c1(OC)ccc2c(c1)C(NC(c1nnc3ccccc3c1N)=O)C(=O)N2 CC1(C)CC(C(=O)NC2CC=CCC2)CCN1C(=O)Cn1cccnc1=O CC(C(=O)N1CCCC(NC(=O)CCc2cnc[nH]2)CC1)C(F)(F)C(F)F C#CC1(C(=O)NOCC2(F)CCC2)CCN(C(=O)C(C)=C2CC2)C1 N1(C(C=Cc2ccc(OC)cc2)=O)Cc2ccccc2C1.C12CC(C=O)(C1)C2.N Cc1ccc(C=CC(=O)NC(C(=O)NOC2CC2)C2CCOC2)o1 C(=O)(CCCCN1CCOCC1)NCC(C)CNC(C1C2(CC2)C12CC2)=O c1(C(=O)NCCN(C(=O)CSC(F)(F)F)C)cn(C)nc1C1CCCCC1 C(CCCCNC(=O)CC(=O)NCC1CC1)N(C(C=C(C)Cl)=O)C Cc1cc(C(=O)NC2COCCN(Cc3cn(C)nc3C)C2)cc(Br)c1 Cc1cc(C(N2CC3CC2CCC3(F)F)=O)c2c(O)nn(C)c2n1 Cc1cn2ccnc(C(=O)NC3CC(CCNC(=O)CO)C3)c2n1.C1CCC1 c1cnc(N)c(N)c1.Cc1nnccc1C(=O)NCCOCCO.CC.CC N1(C(c2cc(OC)c(Cl)cc2)=O)CCC(C2(NC(=O)C3=CCCSC3)CC2)CC1 N1(C(CN2CCN(C)CC2)=O)C2CCC1CN(C(c1ccc(C(F)F)cc1)=O)C2 C1(OC)C(OC)CN(C(c2onc(C)c2C)=O)C1CNC(c1ncsc1C)=O C#Cc1ccccc1CC(N1CCCC1CNC(=O)C=C(C)c1ccccc1)=O C1(C(CC)(C)C)CCCC(NC(=O)NC(COC)CC2CCOCC2)C1 c1(OC)cccc(CC(C)CC(=O)NC23CC(C2)C3)c1.C(=O)(C)N.C1CC1 CCCCC(C)CCC(=O)N(C)CCOCCCNC(C1C2CC(=O)CC12)=O CCC(CC)C(C)C(=O)NCC(C)(C)NC(c1cccc2ncsc12)=O C(C1CCC(C)CC1)=C(C)C(=O)NC1CN(C(=O)Cc2cccc(F)c2)CC1C Cc1cc(C(=O)NC2CCC2C)c(C)[nH]1.c1(C(=O)N)cnsn1.c1ccco1 CN=c1[nH]cc(C(=O)NCC2(CC(=O)NCCC3(O)CCC3)CC2)o1 N1(C(C2(COC)C=CCN2C(=O)C(C)CC(F)F)=O)CCc2nc[nH]c2C1 c1(C(N(CCCN(C(=O)Cc2cnc[nH]2)C)C)=O)c[nH]cc1-c1cnn(C)c1 c1(NC(C)=O)cccnc1NC=O.C1(O)CN(C(=O)C(C)c2cccs2)C1.N c1(OC)ncc(Cl)c(C)c1C(=O)NC1CC1C.n1(CC(=O)N)ncnn1 c1(CC(C=C)O)cn(CC2CN(C(C3(N(C)C)CCCC3)=O)C2)nn1 CC1(F)CC(C(=O)NCCCC(=O)N2CCC(CC(F)F)C2)C1 CCC(COC)C(=O)NCc1nocc1C(=O)NC1(c2cccnc2)CC1 N(C(=NCC1CC1)NCc1ncccn1)Cc1nnc(COC)s1 n1(CC)nccc1C(=O)NC(Cn1ccnn1)C=O.C(C)CC=O.C(C)C.N c1(C(N2C(CCC3N(C(CCC)=O)CCOC3)CCC2)=O)cc(=O)n(C)cn1 C=CC(COC)N=c1nc2sccc2c(NCC(c2cnc[nH]2)C)[nH]1 N1(C(CN(C(c2c(C#C)cnn2C)=O)C)=O)CCC(F)(F)C(F)C1 c1(C(N2CC(CNC(C(C=C)(F)F)=O)C(O)C2)=O)c(F)cccc1[N+](=O)[O-] C(=O)(CCCCCNC(=O)Nc1ccccc1)N(c1oc(C2CC2)nc1C#N)C CC(CN(C)C)CCC(=O)NC1CCCCC1C.c1(CCC(=O)N)cnn(C)c1 N1(C(CN2CC(C)(OC)C2)=O)CCC(C)(C)C1.C(=O)(CC(C)c1ccccc1)N c1(C(N2CC3C(NC(c4cccn5nnnc45)=O)C3C2)=O)c(Cl)ccc(Cl)c1Cl C1(C(=O)NCCN(CCO)C(C2CC(C)(O)C2)=O)(CC)CC1(F)F N1(C(c2cc(CCC)nn2C)=O)CCN(C(=O)CC=C)CCC1C C1(CC)C(C(=O)NCCc2ccccc2)CCN1C(=O)CCc1ccccn1 N1(C(CC(C=C)CC)=O)CC2OCC(NC(c3cscn3)=O)C2C1 c1(CCNC(c2c[nH]c3ccccc23)=O)c[nH]c2ccc(Br)cc12 C(C)(CNC(=O)C(N)=O)(CO)NC(C(c1ccccc1)SC)=O CCC(C)C(=O)C(=O)NC1COCCC1C(=O)NOCc1nc[nH]n1 c1(C(N2CC(O)(CC)C2)=O)ccc(F)c2c1CCC2.c1(SC)ncc(C(=O)N)s1 C1(N(C)C(c2cc(Cl)n[nH]2)=O)CN(C(=O)CN2CC3CC3C2)CC1F C(=O)(C1=CS(=O)CCC1)NCCNC(C1(C)CCCCCC1)=O N1(C(C(C(C)C)F)=O)CC2(C1)CN(C(=O)CCC(C)(C)N1CCOCC1)C2 c1(OC)cc(S(=O)(=O)NCc2cccc(OCC(F)F)c2)sn1 CC(C)C(C(=O)NC1CN(C(C2CC(=O)N(C(C)(C)C)C2)=O)CC1C)C(C)C C#CCCCCC(=O)N1CCC(C(CO)NC(=O)CN(CCCCCC)C)CC1 Cc1cc(S(C)(=O)=O)ccc1NC(N1CC2CCC1CN(C(C1CCC1)=O)C2)=O c1(C(N2CC(NC(=O)CO)C(C3CC3)C2)=O)ccc2c(c1)S(=O)(=O)N(CC)C2=O C#CCC(C)(C)C(=O)N1CCC(C=CC(=O)NCc2cc(C)[nH]n2)CC1 C1(C=O)NC(=O)CC1c1ccccc1.CC(C)CC.C12(C=O)CC(F)(C1)C2.N C1(n2cc(-c3ccc(C)nc3)nn2)CCCN(C(=O)CCC2CCCO2)CC1 C=CCC(CC(C)C)C(=O)NCC(C)CO.C(C(F)(F)F)N(CC=CC=O)C N1(C(CCc2n(C)cnc2)=O)CCCC(CNC(C2(C)CC=CCC2)=O)C1 Cc1c(C(=O)NCC2(NC(C3CCCC3C)=O)CCC2)sc(Cl)c1Cl C1(OC)CN(C(=O)Cc2cc(C3CC3)on2)CC1.c1(C=O)ccc(C2CC2)s1 C(=O)(CCC(F)(F)C(F)F)NC(C)CCN(C(=O)CCCCN1CCCC1)C CC(CC=Cc1ccccc1)C(=O)NC(Cc1cccc(Cl)c1)CO C1(NC(C(CC)C2CCOCC2)=O)CCC12CN(C(=O)CN1CCN(C)CC1)C2 C1(C(=O)NCC2CCN2C(=O)CN2CCNC2=O)CC2(CCCC2)C1 C1(CNC(c2cc(CC)ncc2)=O)CC2(CCN(C(=O)CCCSC)CC2)C1 Cc1c(C(=O)NC2(C3CN(C(=O)C(C)OCC(F)(F)F)C3)CC2)cncc1F N1(C(COCC(C)C)=O)CCOCC(F)(C)C1.C1(=CC(=O)N)CCN(C)C1 c1ccc(C(F)(F)F)cc1Cl.C1(CC(=O)N)CSCN1C=O.C(C)(C)C.C N1(C(CCc2cc(OC)ncc2)=O)CCC2(C1)CN(C(c1cc(=O)cco1)=O)C2 C1(NC(C(c2ccccc2Cl)OC)=O)CC(F)CN(C(C2CC2)=O)C1.N(C)C.C C1(NC(C(C)CCN(C)C)=O)CC2CN(C(C3(O)CC4CCC3C4)=O)CC2C1 CC(C)(C)C(=O)C(=O)NC1CCCN(C(C2CC(S(N)(=O)=O)C2)=O)C1 Cc1cc(NC(=O)C)ccc1.c1ccccn1.C(=O)CC1CC1C(F)(F)F.S N1(C(CNC(=O)NC)=O)CCC2C(NC(=O)C(c3ccc(Cl)cc3F)O)CC12 C(=O)(C(C1=CCC(C(C)(C)C)CC1)N1CCOCC1c1cc[nH]n1)NCCC#N N1(C(CC2(C)CC2(Cl)Cl)=O)CC2(CC(NC(C3CC=CCC3)=O)CO2)C1 N1(C(C(CCC)N(C)C)=O)CCOCC(NC(c2ccc(C)nc2NC)=O)C1 c1(OC)ccc(CN2CCC(C(N3CCC(O)C3)=O)CC2)c(C)c1 N1(C(c2c(OC)ccc(C)n2)=O)CCN(C(=O)C2=CC3CCCC23)CC12CC2 Cc1c[nH]c(C(=O)NC2CN(C(c3csc(Br)n3)=O)CC2O)cc1=O CC1OC2(CO)CC1(C(N1CCCC(N(C)C(c3cccs3)=O)C1)=O)C2 C1(C)(C(N2CCCCC2)=O)CCC(=O)N(C)C1.CC(C)CCC=CC(=O)N(C)C C1(CNC(C(CC)C2CCOCC2)=O)CCC(NC(c2snc(C)c2N)=O)CC1 C(C)(c1ccccc1)=CC=O.C(C)(CCNC(=O)Cn1nnnc1C)OC.N C#Cc1ccc(NC(=O)C(=O)NCc2ccnn2CC)nc1C C1(NC(CCc2onc(C(C)(C)C)n2)=O)CCCCC1.C1(C(=O)N)CCS1(=O)=O C1(NC(C2CC2)=O)CC2CN(c3cc(Cl)nc(C(F)(F)F)n3)CC2C1.C1CC1 c1(C(N2CCC(CN(C)C)C2)C(=O)NC(C)(C)C)csc2ccccc2c1=O c1(C(N2CCCC(NC(CC)=O)C2C)=O)sc2ccc(OC)cc2c1C Cc1cnc(N(C)Cc2ccno2)c(S(=O)(=O)N2CCC3C(C2)C3(F)F)c1 C1(C(=O)NCC(CO)OC)C(C2CC2)CCN1C(c1cc(C)nnc1O)=O CCC(C)CC(=O)N1CCC(C(=O)NC(C)Cn2cnnc2)(CO)C1 c1(C(=O)NC2CN(C(c3c(C)ccnn3)=O)CC2C(F)F)ccnn2ccnc12 c1(C(=O)NCC2(O)CC(CNC(C(COC)O)=O)C2)c[nH]cc(C)c1=O CN1CCC(C2(C(=O)NC3C4CN(C(C5COC(C)(C)CO5)=O)CC34)CC2)CC1 c1(C(CC)C)nc(C)cc(=NCC2CN(C(=O)Cc3cc(C)no3)CCC2C)[nH]1 c1(N2CCCC(NC(C)=O)C2)nc(=NCC2CCN(C)C2)[nH]c2ccc(Cl)cc12 CC(C)CC(C)CC(=O)NC12CC(NC(C3CC4(C3)CC(F)C4)=O)(C1)C2 C(=O)(CCC(=O)c1cccnc1)NC1CC(NC(=O)CN2CC3CC3C2)C1 C12(NC(C)=O)CCC(CC1NC(c1cc(-c3cc(C)ccc3C)on1)=O)C2 C(=O)(C1Cc2ccccc21)N(CC(=O)NCCC1CCCCO1)C1CC1 c1(C(N2CCC(=CCNC(c3c(C)cn(C)n3)=O)CC2)=O)c(O)ccc(Cl)c1F C=C1CC2CC1CN2C(C1C=CCCN1C(=O)C(CC1CCC1)OC)=O c1(CSCCC(=O)NCCNC(c2cocn2)=O)ccccc1 c1(C(=O)NC2CCN(C(Cn3ncn(C)c3=O)=O)C2)cccc2c(C#N)c[nH]c12 C=CCC(CNC(C1(COCC)CCC1)=O)C(=O)N1CCCC(OCC)C1 CP(C)(=O)CC(=O)NCCC1(CNC(c2cncs2)=O)CC1 N1(C(c2cn(C)c(O)n2)=O)CCCC12CCN(C(c1cc3c(o1)CCCC3)=O)C2 C12(C(NC3CC3)=O)CCCCC1CCC2.C(=O)(C#CC(=O)N1CCCC1)N(C)C.C N1(C(c2c(OC)scc2)=O)CCC2(CC2)C1.C(=O)C(C)Cc1cnn(C)c1.C c1(NC(C2(C)C(C)CN(C(C(CC)C)=O)C2)=O)c(C)cc(C)cc1C C(CCC(C(=O)NCCCF)N(C)CC1CN(C)CCO1)SC C(CC1=CCN(Cc2ccccc2)CC1)NC(c1c(C)n(C)c(C2CC2)c1)=O N(C1CC(C)(C)c2ccccc21)C1(c2n(CC=C)nnn2)CC2(CCOCC2)C1 C1(C(N(CC(C)O)CCOC)=O)CCN(C(=O)c2cc(C)n(C)c2C)O1 C1(CC(=O)NC2CC(C(C)NC(=O)CCC3CCCCC3)C2)CCCC(C)C1 c1(C(N2CCCC(COC)C2)=O)[nH]c(C)c([N+](=O)[O-])c1C.C(=O)C1=CCCC1.N N#Cc1cc2c(nc1NCC1CC(NC(=O)C3CCCc4ccnn43)C1)CCC2 Cc1cc(=O)n(C)cc1C(=O)NCC1CC1.C1(C)CCOCC1.C(=O)C.C C1(OC)(C)CCN(C(=O)C(C)(C)F)C1.c1(C=O)ccc(C=O)cc1.C(C)C C1(NC(c2c(CC)n[nH]c2)=O)CC2CC(C1)N(C(C1CC13CCCC3)=O)C2 CC(O)CCCNC(C1CC(CNC(C2CCCCO2)=O)C1)=O c1(OC)ccc2c(c1C(=O)N(C)CC1CC1)CCC2.c1(C=O)ccccc1F.N N1(CC)CCCC(C(N2CCCC2CN(C)C(C2(C#N)CCCO2)=O)=O)C1 c1(C(=O)NC2CC(C)CN(C(=O)C(C3CC3)C3CC3)C2)nccc2ccncc12 N1(C(C(CC)N(CC)CC)=O)CC(C)(C)CC1CC(=O)NC1(CCF)CCC1 O=C(O)C(C1CC1)NC(=O)C(c1cscn1)NC1CC1 CC#CCCC(=O)NC1(CNC(=O)C(Cc2ccccc2)OC)CCCCC1 [nH]1nc(C)c(C=O)c1C.C1(C)(CC)CCN(C(C2CC2C(C)(C)C)=O)C1.C N1(C(CN(C)CCO)=O)CC(O)CC1CNC(=O)CSCC(N)=O c1(N2CC(CC)OC(C)C2)nc(=NCCc2cnn(CC)c2)[nH]c2c1CSC2 c1(-c2cccc(C#N)c2F)cnn2cc(C(=O)NCc3cscn3)cnc12 O=S(=O)(c1ccc(Cl)nc1)N1CCC(c2nc(O)n[nH]2)CC1 C12(C(=O)NC)COC(C1)C(NC(C1(C#N)CCOC1)=O)C2 C1(C(=O)Nc2ccc(C#C)cc2)CCN(C(C2(O)CCSCC2)=O)CC1(C)C C1(C)(C(=O)NCC2N(C(C(CC)=CC)=O)CCOC2)CCCC(F)(F)C1 N1(C(CC(C(=O)OC)C)=O)CC(NC(c2ncnc3c2CCC3)=O)C2(CCC2)C1 C1(CC(=O)NC(CCNC(C(c2scc(C)n2)C)=O)C)CC2CCC1CC2 CCCC(C)(O)CNC(C1CCCN(C(c2cc(C(C)C)on2)=O)C1)=O C1(C)(C(=O)NCCC(=C)C)CC(NC(c2ccc(NC)s2)=O)C1 N1(CC=O)C(C)CCC1C.c1(C(N(CCC)CC)=O)cccc(CC(C)C)c1.N c1(C(N2CCC(C)C(CNC(C3CCSCC3)=O)C2)=O)ccc2c(c1)nnn2C C=CCC(CNC(C1CCCS1)=O)C(=O)N(C1CCC1)CC1CC1 c1(OC)cc(C(=O)NCCCN(C(C2COCCO2)=O)C2CC2)cc(Cl)n1 C1(NC(CCC=CC(C)C)=O)CCC(C)(CNC(=O)CCCn2cccc2)C1 c1(C(N2CCC(O)(CN(C(CCC=CC)=O)C)C2)=O)nnc(O)cc1O C12(NC(c3ccc(C)nc3N)=O)COCCC1CN(C(C1(C)CCCCC1)=O)C2 C1(CCC)CN(C(=O)Cc2cnc(C)s2)CC1C(=O)NC(C)CO.C1CCC1 CC1CCC(C)(C(=O)NCCOCC(=O)NOCC2CCCO2)C1 C(=O)(C1CCc2ccccc21)NCC(CC)NC(=O)CN(C1CCC1)C Nc1cc(C(=O)NCCC2CN(C(c3c(F)cccc3Br)=O)C2)nc(O)c1 Cc1c(C(=O)NC2CN(C(c3nncs3)=O)CC3(CC3)C2)c2ccccc2n1C c1(C(N2CCC(F)CC2)=O)ccc2[nH]nc(-c3cnn(C4CCCCC4)c3)c2c1 C12(NC(Cc3c(C)scc3)=O)CC1CN(C(=O)CC(C)n1cccc1)C2 C(=O)(CCC(O)C(C)(C)C)N(CCN(C(c1cc(CC)on1)=O)C)C Cc1cc(C(N2CC3(CCC3)C23CCC3)=O)c2cccc(C)c2n1 C12(C(N)=O)CC(CN1C(c1nc(Br)sc1Br)=O)C2 C1(NC(c2cnc(SC)s2)=O)CCN(C(=O)Cn2c(C)csc2=O)CC1 c1(OC)c(C(=O)NC2CN(C(c3ncc(Cl)cc3Cl)=O)CC2O)cccc1C C(=O)(C1=CCS(=O)(=O)C1)NC(C)CCCCNC(=O)C(C)n1ccnc1 C=C1CCN(C(c2ccn(C3CC3)n2)=O)C(C(N2CC(c3cccnc3)C2)=O)C1 Cc1nc(CNC(=O)C(c2cccnc2)NC(C2CCCC2)=O)[nH]c1C C1(C=O)COC2(CCOCC2)C1.C1C2CCC(C2)C1.CC(C)(C)OC(=O)N.C C1(CC)CN(C(=O)C(F)(F)C2CC2)CC1.C1(C=O)CC(=O)N(C2CC2)C1.N C1(CNC(c2c[nH]c(=O)cn2)=O)CC12C(=O)Nc1ccccc12 C(=O)(C(O)COC)N(CC(C)N(C)C(c1cc(Cl)no1)=O)C.c1ccccc1 C(C)(CNC(=O)CCn1ccnn1)(C(C)C)NC(c1cc(C)[nH]n1)=O N1(C(Cc2ccn(C(C)C)n2)=O)CCC2CC1CN(C(=O)C(C)c1ccco1)C2 c1(CC(=O)NC2(CO)CN(C(Cn3cc[n+](C)c3)=O)C2)cc(F)ccc1Cl CCC(C(=O)N1CCC(C)C(NC(=O)C(c2ccc(F)cc2)O)C1)C(C)C N1(C(C(CCC)C)=O)CCC(CO)C(NC(C23CC(C)(C2)OC3C)=O)C1 C(=O)(C1=NN(C)C(=O)CC1)N1CCCC(C(C)NC(CCc2ncc(C)[nH]2)=O)C1 Cc1ccc(C(=O)C(N2CCCC2C(C)NC(C23CC(CO2)C3)=O)=O)cc1.C CCC(CC)CCC(=O)NCC(O)CNC(=O)C(CC)(CC)CO c1(C(=O)N)cc(Cl)cc([N+](=O)[O-])c1.C1(N(C(C(C)CC2CC2)=O)C)CCCCC1 c1(N(C=O)C2CC2)cc2ncccc2[nH]1.n1(C2CCC2)cc(C(F)(F)F)cn1.N Cc1nc(S(=O)(=O)N2CC3(CN(C(=O)C(F)(F)F)C3)C2)ccc1C(=O)O N1(C(C(CC2CC2)OC)=O)CCOC2CN(C(=O)Cc3n[nH]c(=N)s3)CC12 Cn1cnc(C=CC(=O)NCCn2cc(C(=O)N)nn2)c1.CCCSC(F)F N1(C(C2CC(CF)C2)=O)CC2(CCCCN2C(C23COCC2C3)=O)C1 C1(C2CCCCO2)(C(N2CCC(F)(c3cn(CCCC)nn3)CC2)=O)CCCO1 N(C)(S(=O)(=O)N(C)C)CC(N1CCC(C)C1)=O.Cc1ncc(CCC(=O)N)o1.C N1(C(C2(C=C)CCC2)=O)CC2CCN(C(=O)CCC(=O)OC(C)(C)C)C(C2)C1 N1(C(CCC=CCC=C)=O)CCC(C(=O)NC2C=CC(COC)C2)(CO)C1 C12(NC(CCOC)=O)CCCCC1CN(C(c1cn(C)nc1SC)=O)C2 n1(C2CN(C(C3N(CC)CC3)=O)C2)cc(CNC(C2CC3CC2C3)=O)nn1 C(=O)(C1CCc2cccc(=O)n21)N1CCCC(CCNC(CSC(C)(C)C)=O)C1 c1(C(=O)NC2C(C)CN(C(c3cnc(Br)s3)=O)C2)cc(O)ccc1Cl C1(O)(C(C)NC(C2CC2c2cncn2C)=O)CCN(C(c2ncccn2)=O)C1 C(CNC(=O)NC1CC(F)C1)(CCNC(=O)OC(C)(C)C)OC C1(NC(CC=CC)=O)CCN(C(c2cc3c(s2)CCC3)=O)CC1C(C)C C1(C(N2CCCC(C)(CNC(CC(=C)C)=O)C2)=O)Cc2nccnc2C1 c1(NC(C2CCC(NC(=O)CN3CCCC3=O)C2)=O)c(F)cc(Cl)cc1I c1(NC(=O)OC(C)(C)C)cccc(C#CC)c1.C12(C(=O)O)CC1CCC2(F)F c1(CN2CC(NC(c3cccc(Br)c3Br)=O)C2)cnc2cc[nH]c2c1 C1(NC(CC2(C)N(C(c3cc(C)cc(C)c3)=O)CC2)=O)CCc2n[nH]cc2C1 CCC1=C(C(=O)NCCCCC(C)(C)NC(=O)C(C)=CC2CC2)CCCO1 C#CC1(O)CCN(C(C23COC(C2)C(NC(c2cn(CC)cn2)=O)C3)=O)C1 N1(C(=O)CC2(NS(=O)(=O)CCBr)CCC2)CCS(=O)(=O)CC1 c1(C(=O)NC2CC(n3cc(-c4cnc(C)o4)nn3)C2)ccc2[nH]cc(C#N)c2c1 c1(C(N(CCC(C(C)C)NC(CCCN(C(C)C)C)=O)C)=O)csc2nnsc12 c1(C=O)onc2c1CCCC2.c1(C(C)=O)nc(C(=O)NCC2(C)CCC2)cs1 N1(C(N(C)Cc2cc(C)c(Br)cc2)=O)CCN(C)Cc2cccnc21 N1(C(c2c(C)nn(CCC)c2C)=O)CC(C)CN(C(=O)C(C)=C2CCC2)CC1C C1(CNC(C(C2CCCN(C(C3(C)CCC(=O)N3)=O)C2)C)=O)CCCCCCC1 C1(C#CC(=O)N2CCC(NC(=O)C(c3ncccc3C)(F)F)C2)(CC)CC1 CC(C)CC(C(=O)N1CCC(N(C(=O)CC)C)C1)NC=O.C1CC1.C1CC1.N n1(CC)cnc2c(N(C)CCN(C)CC)[nH]c(=NCC3CNC(=O)C3(F)F)nc12 c1(CC(=O)NC2CCN(C(C(C(CC)C)C)=O)C2(C)C)csc2ccccc12 N1(C(CC(CC)SC)=O)CCC(NC(c2nc(N(C)C)nc(=N)[nH]2)=O)C(O)C1 CCC(C)(C(=O)NCC(O)CNC(=O)Cn1ccc(=O)cc1C)C(F)F c1(CC=O)ccc(S(N)(=O)=O)s1.CC1(C)CCN(C(C2CNC(=O)N2)=O)C1 CC1(C)CCCC(CNC(C2(CNC(=O)CN=[N+]=[N-])CC(C)(C)C2)=O)C1 C(C(CO)(CO)NC(=O)N(C)C)N(C(c1c(C(C)C)ncs1)=O)C Cc1ccc(C)c(CNC2(c3nnnn3C3CCC3)CCCC(N(C)C)C2)c1 c1(C(N(C2CCCN(C(C3(C)CC(=C)C3)=O)C2)CCO)=O)cc([N+](=O)[O-])oc1C C1(O)(C(C)NC(C(C)C2CC2)=O)CCN(C(=O)CC(O)c2ccccc2)CC1 c1(CC)cc(C(=O)NC2(C(=O)NCCC(O)COC)CC2(C)C)n(C)n1 C(=O)(C(C)CCC)N(CC(=C)C)Cc1ccccc1.C(=O)(C(=O)N(C)C)N C1(CC(C)CO)CCN(C(=O)NC2CCS(=O)(=O)C2)CC1 CCCCCC(O)CC(=O)NC(C)(C)CCCC(=O)NC(c1ccns1)C Cc1ccc(C=CC(=O)NCCC2CCN(C(c3cscc3Cl)=O)C2)o1 Nc1c(C(=O)NC2C3CN(C(c4n[nH]c5c4CSCC5)=O)CC23)cc(F)cc1F N1(C(Cc2n(C)ccn2)=O)CCC(NC(C2CC3CCC2O3)=O)C1C1CC1 CC(C)C(F)C(=O)NCCc1cc(C(=O)NC2(C3CCCO3)CCC2)no1 C(=O)(C1COc2ccccc21)NC1C(NC(=O)COc2ccc(Br)nc2)C1 c1(C(=O)NC(CC)(CNC(C2CC2C)=O)CC)ccc(N)cc1C(F)(F)F C=CCCC(C(=O)N(C1(CCO)CC1)C)NC(c1n[nH]cc1C)=O C1(CNC(c2ccc(N(C)C)cc2)=O)CCCCC1N=c1[nH]nc(C(N)=O)s1 C1(C(=O)NC2CCC2)(CC)CCN(C(c2cnn(C)c2OC)=O)C1 c1(OC)ccc(OC)c(C(=O)N(C2CCCC(NC(c3csnc3C)=O)C2)C)n1 c1(CC)n[nH]cc1C(=O)NCC1CCN1C(=O)CN1CCC(C)C1 C1(C(=O)N(C)CC)(CC)CCCN1C(=O)CNC1CC1.C(=O)C(C)C c1(OC)cc(N)c(C(=O)NCC(O)CNC(C2CCOC2)=O)c(F)c1 n1(CC(C)NC(=O)O)cc(NC(=O)C(=O)N(C)CCO)nn1.C(C)(C)C C1(CNC(c2cnn[nH]2)=O)COCC1n1cc(COCCCO)nn1 c1(-c2cn(C(C)C)nc2)cnc2n[nH]c(C(=O)Nc3onc4ccccc34)c2c1 c1(C(N2CC(O)(Cc3ncccn3)C2)=O)cn(CC(F)(F)F)cn1 C1(COC)(C)CCCN1C(C1CC12CC2)=O.c1(CC=O)cn(C)nc1C.N c1(C(N2CC(C)C(NC(C3(C)CC=CCO3)=O)C2)=O)cc2n(n1)CCCCC2=O C1(NC(C2(CC=C)CN(C(=O)CP(C)(C)=O)C2)=O)CNC(=O)C12CC2 C#Cc1ccc(NC(c2ccc(CNC(C3(C)CCC(C)C3)=O)o2)=O)cc1 C(=O)C(F)(F)c1nccs1.C(C)C(=O)NCCCC.C(C)O.CCSCC Cc1c(C(=O)NCC2(O)CCN(C(c3nnn(C)c3N)=O)C2)ccn1CCO c1(C(=O)NC2CCN(C(C(COC)(C)O)=O)C2)c(C)nn(CC(F)F)c1C Cc1cc(C(=O)N)nn1C(C)(C)C.C1(C(N(CC)C)=O)CC2CCC1O2.CC c1(OCC2(NC(C(=O)O)CN3CCCCC3)CCSCC2)ccc(F)cc1 CC1CN(C(C2(C)CCOCC2)=O)CCN1c1nccc(-c2cnccn2)n1 C1(NC(C(F)=CC)=O)CC2(C1)CC2NC(=O)C(C)Oc1ccccc1 c1(C(=O)NC2CC(C)(C)N(Cc3ccccc3)C2)cc(Br)cc([N+](=O)[O-])c1 C1(c2cn(CCOC)nn2)CCCN(C(=O)C(n2cnc(C#N)n2)C)C1 C(=O)C1=NOC(C)C1.C(CC(C)C)=CC=O.C1(CC(=O)OC)CCC1.C N1(CCNC(c2n(C(C)C)nnc2)=O)CCCCC1CCC(=O)OC C(C=O)(C1=CCCCCCC1)N1C(C(=O)OCC)CCC1C(=O)OC.C1CC1.N c1(C(=O)N)nc2c(s1)COCC2.c1(CC)ncncc1C(=O)N(CC(C)(C)C)C c1(N2CCCC(CCCO)C2)nc(=NCCC2CCOC2)[nH]c2c1CCC2 N1(C(c2cncc(OCC)c2)=O)CC(NC(=O)C#CC2(C)CC2)CC12CCCC2 C(=O)(C1=CC2CCCC12)N.c1(CCC(=O)NCC2CC(C)C2)ccc(O)cc1 Cc1[nH]cc([N+](=O)[O-])c(=O)c1C(N1CCOC(C)C1)=O.c1(CC=O)ccns1.N Cc1cc(C)cc(C)c1.N1(C(c2cc(C(=O)O)c(C)o2)C=O)CCOC(C)C1C.N CC(N=c1[nH]c(N2CC=CCC(C)(C)C2)nc(=N)[nH]1)c1ccns1 N1(Cc2nnc(C)s2)CCOC(COCCn2c(C)csc2=O)C1 Cc1cn(C(C)C)cc1C(N1CCC(NC(C2CCCCC2)=O)C1C(C)C)=O C(=O)(C(CC)CC(F)F)NCC(CCCC)NC(c1onc2ccccc12)=O c1(C(N2CCCC(C(C)NC(CCOCC(C)C)=O)C2)=O)cc(C#N)ccc1F c1(C(=O)NC2CCN(C3CCCCC3O)CC2)ccc2c(c1)C(CC(=O)O)CCC2 Cn1cnn(CC(N2CCCC2CNC(=O)CSCc2ccccn2)=O)c1=O c1(SCC(=O)NCCC)ccc(Cl)cc1Cl.C(=O)C(C)Cc1cnn(C)c1.N Cc1cc(C(N2CC(CNC(=O)C=CCO)CC2C)=O)nn1-c1ccccn1 N1(C(C2CCC2)=O)CC(C2CC2)C1C1CC1.c1(C(=O)N)occc1C1CC1 c1(OC)cc(NCC2CN(C(=O)C(C)CC3CCC3)CC2C)ncn1 N1(C(CN2C(C)CC2)=O)CCN(C(=O)Cc2scnc2-c2ccccc2)CC1C c1(NC(=O)OCC(N2CCC(O)(CC(C)C)C2)=O)ccc(Cl)c(F)c1O c1(CNC(C2CCN(c3nc(OC)nc(C)c3)C2)=O)ccnc2ccccc12 CC(C)C(N=[N+]=[N-])C(=O)NC1(CNC(c2nc(Cl)cs2)=O)CCC1 Cn1cc(Cl)cc1C(N1CCCC1C(C)(C)C(=O)NCC(O)CC1CCC1)=O C1(NC(c2cc(C)c(F)cn2)=O)CC2CC1CN(C(c1n[nH]c(C)c1Cl)=O)C2 c1(C(N2C(C3CCCN(C(C(C=C)O)=O)C3)CCC2)=O)cc(C)c(=O)n(C)c1 Cc1nn(C)c(C(=O)NCCC2CC2)c1[N+](=O)[O-].C1(C#N)(C=O)CCOC1.N N1(C(c2c(OC)oc(C)n2)=O)CCN(C(C2CN(C)C2)=O)C(C)C1 c1(C(=O)NC2CN(C(C(c3n(C)cnc3)O)=O)C2)cc(N)cc(O)c1F N1(Cc2cccc(C#C)c2)CC(NC(c2ccc(OC)cc2F)=O)CC(F)(F)C1 Cc1ccc2c(c1)CC(C(N1CCC(N(C(=O)CCc3cccnc3)C)C1)=O)O2 N1(C(c2c(SC)cnn2C)=O)CCC(C)CC1.C1(F)(C=O)CC2(CCC2)C1.C C(c1ccc(Cl)cc1F)=CC(N1CCN(C(C2CC(C)(O)C2)=O)CC1)=O.CO.C n1(CC)nc(C)c(CN2CC3CC2CN3C(c2cnn(C(C)(C)C)c2Cl)=O)c1C CC(F)(F)C(C)(C)C(=O)N.C12CC1CN(C(c1ccc(C(F)(F)F)cn1)=O)C2 C1CC2(CC2)CN1C(C1CCCC(C(N)=O)C1)=O.c1(CC)cnoc1C(=O)N CC(CNC(c1ncoc1C(C)(C)C)=O)N=c1[nH]nc(-c2ccccc2)s1 CC(C)CC(Cn1cc(CCc2ncccn2)nn1)NC(C1CC(F)C1)=O CC1(C)C2CCC(NCCS(=O)(=O)CC3CC3)C1C2 N1(CC(N2CCC(CNC(CC=C=C)=O)C(F)(F)C2)=O)Cc2ccccc2C1=O C=CC(C)(CC)C(=O)NCC(O)CC(=O)NC(c1noc(CC)n1)C C1(C)(CC)CCN(C(=O)C2=CCN(C(C3CSCC(=O)N3)=O)C2)CC1 C(=O)(CCCC(C)(F)F)N1CC(CNC(C2CC(C)=C(C)CC2)=O)C(C)(C)C1 N1(C(C(OCC)OCC)=O)CCCC(F)C1.C(=O)(C(O)CC1CCCCC1)N C#CCCCCCCC(=O)N1CCCC(NC(c2nnsc2C)=O)C1C C(=O)(C(C(C)O)NC(c1nnnn1C)C1CC(n2ccnn2)C1)OCC c1(C(C(=O)NCC(=C)C)N(C(C)C2CC2)CC)cccc2sccc12 Cc1cc(C(=O)N(CC(=O)NCC2(C)CCCCCC2)C)nc(O)n1.C1CC1 c1(OC)ccc(C(c2nnnn2-c2ccccc2)NCCCF)c(F)c1Br N1(C(C(C=C)CC)=O)CCC(C(N2CCCN(CCC)CC2)=O)C1(C)C C1(CC)CN(C)CCCN1C(=O)C(Cn1cncn1)NC(=O)C=CCF N1(C(CN(C)C(N)=O)=O)CC(c2cn(C3CCCC3O)nn2)(N(C)C)C1 c1(C(=O)NCC2CCC(CNC(C3(C)CC3)=O)CC2)cnc2cccnn12 c1(OC)c(C(=O)N(CC(C)NC(=O)CCCN=[N+]=[N-])C)ccnc1F C(=O)(C(C)(O)C(C)(C)C)N1CC(C)C(NC(c2cnn(C(F)F)c2)=O)C1 c1ccc(C#N)cc1.C=CC(C)(C)C(=O)NCC1(NC(=O)CC)CCOC1.O C12(C(=O)NC(CCNC(CNC(C)=O)=O)(C)C)CCCC1CC2 c1(CN(C(c2[nH]nnc2C)C(=O)Nc2c(OC)cccc2)C)ccc(F)cc1F C1(NC(c2c(C)n(C)nc2)=O)CC2CC1N(C(c1c(Cl)cncc1Cl)=O)C2 C=CCC(CC)C(=O)NCCC1CCCN1C(=O)C(=Cc1ccccn1)C N1(C(C=NOC)=O)CCCC2CN(C(c3cc(Cl)cc(C)c3O)=O)CCC12 N1(C(c2cn(C(C)C)nn2)=O)CCN(C(c2cc(S(N)(=O)=O)cs2)=O)CCC1C C1(C(=O)NCCCC)CCCN1S(=O)(=O)CC.c1(C=O)cnn(CC(C)C)c1 CC(CC(=O)NC1CN(C(=O)COc2cccnc2)CCC1(C)C)C(F)(F)F c1(OCCC)cc(OC)ccc1NC(=O)NC1CC(C(C)C)C1 N1(C(c2occ(C)c2)=O)CCCC(C(N2CC(F)(CF)C2)=O)C1 C#Cc1cc(C(=O)NC)ccc1C.c1(C(N2CCC2)=O)ccc(C(C)=O)c(C)c1 N(C(=NCCc1ncc(Br)s1)N1CCCC(O)CC1)C(CC)CC C1(NC(c2c(C)nccn2)=O)CCC12CN(C(c1cnc(C(C)(C)C)o1)=O)C2 c1(C(=O)NCC2N(C(c3occ(C)c3)=O)CCOC2)cc(Cl)cc(Cl)c1Cl Cc1ccc(CCNC(=O)NC2C=CC(C)(C)CC2)c(Cl)c1 C1(NC(C(CC)=CC)=O)CCN(C(C2(C3CC3)CC(=O)C2)=O)CC1C CC(C)CC(CC(=O)NCc1nc[nH]n1)NC(C1CC1c1ccccc1)=O N#Cc1cc2c(nc1N1CCCC3C(NC(=O)C=CBr)C(C)(C)C13)CCOC2 n1(CC)nnc2cc(C(=O)NCCCCNC(c3cc(F)ccc3Cl)=O)ccc12 Cc1cc(C)c(C=CC(=O)N)c(C)c1.C1(CC)CCN(C(=O)C)C1.CC(C)C CN1CC=C(CCNC(C2CCCCN2C(c2cc(N)cc(F)c2)=O)=O)CC1 N1(C(Cc2nc(C)[nH]n2)=O)CC(CC(=O)N(CC(N)=O)C)C2(CC2)C1 c1(C(=O)NCCC(C)C)ccc(N(C)C)c(F)c1.C1(CC(=O)N)CCCCCO1 C1(C(=O)NCCCOC2CCCC2)(CCl)CCCCCC1 C(=O)(CCC(CC)NC(=O)CC1COCC1O)NCC(=O)NCCC C1(C(N(C2CC(CO)C2)C)=O)CN(C(C2CCC3(CCC3)O2)=O)CCN1C c1(C=O)cc(N)c(Cl)c(O)n1.C(=O)(C(C)(C)C(=O)NC1CCCC1)N(C)C.N C1(C(N(CC(C)CNC(c2sccc2CO)=O)C)=O)CCCN1N=O C1CC2CCC1N2C(c1cn(C)c(=O)cn1)=O.n1(CC(C)C)cc(C(=O)N)cn1 C1(NC(c2cnnc(Cl)c2)=O)CCOC2(CCN(c3ncns3)CC2)C1 C1(C(N(CCNC(c2n(C(C)C)ncc2)=O)C2CC2)=O)CCC(C)NC1=O C1(NC(C(C(C)(C)F)(C)F)=O)CC1C1CCCN(C(=O)CCN2CCOC2=O)C1 CCCCCCC(=O)N1CCN(C(c2cccnc2S)=O)CC1CCO CC1(C)CCCOC1CC(=O)NC1CN(C(=O)CC2CCC2)CC1F c1(NC2C(C)(C)C(NC(c3cc(Cl)ncc3Cl)=O)C2)ncc([N+](=O)[O-])cn1 Cc1ccnc(O)c1C(N1CC(CC(F)C(=O)N(C(CO)C2CC2)C)C1)=O CC1CCN(C(c2n[nH]c(=N)s2)=O)C(C)C1.c1(C(=O)N)cnn(C2CC2(F)F)c1 C#CC1CC2CCC1N(C(C1CC13CCN(C(=O)C(C)(F)C(C)(C)F)CC3)=O)C2 Nc1cccc(-c2nc(-c3ccnc(C(F)(F)F)c3)n(CC3CC3)n2)n1 N1(C(C2C(C)(C)COC2)=O)CCC2(CCN(C(c3cnc(C#N)s3)=O)C2)C1 C1(C(=O)O)CCCCC1NS(=O)(=O)CCCOc1ccccc1 Cc1cc(O)cc(O)c1CNC1C=CC(C(=O)Nc2cc(Br)c(F)cc2I)C1 c1(C(C)C)cc(C(N2CCC(C(C)NC(=O)CCC3CCC(C)O3)C2)=O)no1 C1(C(N2CCCN(C(c3c(O)nnc(C)c3C)=O)CC2)=O)CC2CCC(C1)C2=O C1(NC(C=CC=CC)=O)CC2CCC(C1F)N2C(=O)CCc1cc(C)on1 Cc1cc(C(=O)NCC2CC(O)(CNC(C3CC3(Cl)Cl)=O)C2)ncc1N C1(C(N2CC(N(C)C(c3cc4n(n3)CCCC4)=O)C2)=O)CC12CCC(F)(F)CC2 Cc1nn(C(C)C)cc1C(=O)NC1CCCCC1NC(c1cc(O)n(C)n1)=O CC(C)(C)C(=O)CCCC(=O)N1CCCOC(CNC(=O)C#CC2CC2)C1 CC(C)(CCCCNC(c1cc(Cl)ccn1)=O)C(=O)NNC(=O)c1ccc(F)s1 C(C(=O)N1CC(F)CC1C(C)(C)O)(C(C)C)c1cnc(C)s1 Cn1nc(C(N2CCC(C)(NC(c3cccc(=O)o3)=O)CC2)=O)c2ccccc12 Cc1ccc2ncc(CNC3(CNCc4ccnc(Cl)c4)CC3)n2c1 C#CCC(CC#C)NC(=O)C(c1cccs1)NC(=O)C(C)C#N c1(C(N2C(C(=O)NCCN(C(CC)C)C)CSC2)=O)nc(C)sc1C CC(F)(F)CN=C(NC1CCC1)NC1C2Cc3ccccc3C12 c1(CN2CC3C(C(=O)Nc4cccc(CC)n4)(C3)C2)ccc(C2CC2)c(F)c1 c1(N(CCC(C)O)C)ccc(S(=O)(=O)NCC(O)C2CC2)c(Cl)c1 C1(C=O)CC=C(C)CC1.C(=O)(C(CCN(C)C)N(C)C)N1CC(OC)(C)C1 c1(C(N2CC(N(C(C(COCC)C)=O)C)C2)=O)ccc2occ(C)c2c1 C1(NC(=O)CC2CC2)CC2(CCCN(C(c3ccc(C(F)F)o3)=O)C2)C1 CC1(C)CCC(CC(=O)NC2(C3CCCN3C(=O)CCCC(F)F)CC2)CC1 c1(C(=O)NC(C)CN(CCCO)C)cccc2c1ncn2C c1(C(=O)NC2COCCC2C(N2CCC(O)(CO)CC2)=O)cc2ncccc2[nH]1 C1CC2CN(S(=O)(=O)CC3CCC4(C3)CC4(F)F)CC2C1.CC(C)C.C(=O)O C1(OC)CCCC(C(=O)NCCN(C)C(C2CCSCC2)=O)C1 Cn1nc(C(F)(F)F)nc1-n1nc(-c2ccsc2)nc1C(O)P(C)(C)=O C1(C(=O)NC2CCC(NC(CCC(C)N(C)C)=O)CC2)CCc2nncn2CC1 CCC(COC)(CC)C(=O)N1CCC(C)(CNC(=O)C(=Cc2ccco2)C)C1 C(CCCCC(=O)NC(C)(C)CCNC(=O)C(c1ccc(F)cc1)=O)=CCCC CCC(C)(C)C(C)CC(=O)N1CCC2(CC1)CN(C(=O)Cc1ccsc1C)C2 Cc1cc(Cl)c(C(=O)NCc2cccc(C)c2)cn1.C1(C(=O)N)CC(F)C1 C1(NC(c2cc(CC)on2)=O)CCCC1(C)CN(C)C(c1ccc(C)nc1)=O C1CCN(C(C23CC4CC2C3C4)=O)C(C2CC2)C1.c1(C(=O)OC)ncncc1N c1(CCC)c(C(=O)NC2CCCN(C(C3(C)SCCCS3)=O)C2)cnn1C c1(-c2cn(CC3CCN(C(c4scc(C)n4)=O)C3)nn2)ccnc(Cl)c1Cl C(CCCCCNC(c1c(C)nsc1N)=O)N(C(C(C1CC1)OCC)=O)C N1(C(C2(C)CCN(C)C2=O)=O)CC2(NC(=O)CCC3CCCO3)CCC1CC2 Cc1nc(=N)[nH]cc1C(N1CCC(C(C)(C)CNC(c2nsnc2O)=O)CC1)=O c1(OCC)cccc(C(=O)NC(C)(C)CO)c1N.C(c1ccccn1)=CC=O C1(CC)CC(CC(N2CCC(CNC(=O)Cn3cnnc3O)C2)=O)CCO1 N1(C(CC2C(C)(C)CCN2C(=O)Cc2ccsc2)=O)CCC(C2(C)CC2)C1 c1(C(C)C)cc(F)cc(F)c1.c1(C(=O)NCC)cn(C(COC)C(=O)N)nn1 C1(C(N2CCC(C(C)NC(=O)Cc3cc[nH]n3)CC2)=O)OCCOC1(C)C C(C1=CCCN(C(c2cc(C#N)n(C)n2)=O)C1)NC(C1C(C)OCC1)=O c1(CNC(C(N(OC)C)=O)C)cc2cc(Cl)ccc2[nH]1 C=C(C)C(C)(C)C(=O)NC1CC2(C1)CC2C(=O)NC(CC)C1CCC1 c1(NC(N2CC(C(=O)OC)C(F)(F)C2)=O)ccc(S(=O)(=O)C(F)F)cc1 C1CC2(CCN(C(=O)CN3CCCC3=O)CC2)CO1.C1(C(=O)N)(CC)CCC1.C C1(C(c2n(CCC(=O)OCC)nnn2)NC2(C3CC3)CC2)CCOCC1.C c1(C(=O)NCC(C)N(C(C(COC)CC(C)C)=O)C)ccc2c(c1)N(C)CCO2 C1(CC(N2CCC(OCC(C)(C)C)C2)=O)COc2ccccc2O1 c1(OC)ccc(O)cc1C(=O)NC1CCCC1C.c1(C(C=O)O)ccccc1.N C(=O)(C1=CCC2CCC1N2)N1C(C(=O)O)C2CC2C1 c1(C(=O)NC2CCN(C(CCCN(C(C)=O)C)=O)C2)ccnc(C2CC2)c1 c1(C(=O)N)cccc2ccn(C)c12.CC1SCCCC1C(=O)NCC1CC1C CC(C)CC(C)(CNC(C1CC1C(F)(F)F)=O)NC(=O)C.c1ccsn1 CC(C)(CCC(=O)N1CCN(C2CN(C(=O)CCCC(N)=O)C2)CC1)[N+](=O)[O-] NS(=O)(=O)CCCC(=O)NC1(CF)CCN(C(c2cc(O)cc(O)n2)=O)C1 N1(C(c2c(C)nc[nH]2)=O)CCC2CN(C(=O)Cc3ccnnc3O)CC2CC1 C(C)(C)(CCCNC(C1CCCOC1c1cc[nH]n1)=O)NC(c1nc(C)sc1)=O c1(C(N2C(C(=O)NCc3ccc(Cl)cc3)CC(F)C2)=O)cnc(O)nc1O CN1CC(CNC(C2C3CC3CN2C(c2ccccc2Cl)=O)=O)CC1=O C1CCC2(CCN(C(C3(C(=O)N(C)C)CC3)=O)C2)C1.c1ccc(C=O)s1.CO c1(C(=O)NCCN(C(C2(C)CC(F)C2)=O)CC)ccc(C)s1 c1c(Cl)cccc1Cl.C1(COC)OCCC1C(=O)N.C1(CC)CN(C(=O)C)C1 Cc1cc(C#N)ccc1C(=O)NC1CCCC1NC(C1CC(F)(F)C1)=O C1(C(=O)NCC2C(NC(C(C)N3CCCC3)=O)COC2)CCCC2(CC2)C1 C1(C(N2CC(CC=C)(NC(=O)COC(F)(F)F)C2)=O)CC2C=CC1C2 C1(SCc2cnc(C3CN(C(=O)OC(C)(C)C)C3)s2)CCC(=O)NC1 Cc1c(CC(N2CC3CC3(CNC(=O)C(F)F)C2)=O)c(O)nc2ccccc12 C#CCC(C(=O)NC1CCN(C(=O)CC2CC3(CCC3)C2)C1C)C1CC1 N1(C(c2cc(C)c(C)cn2)=O)CCN(C(c2cc3cccnc3s2)=O)CC12CC2 c1(C(N(C)CC2CCN(C(=O)Cn3ncnn3)C2)=O)cc2ccc(Cl)c(F)c2[nH]1 N1(C(C(CC)C#N)=O)Cc2[nH]nc(C(N3CCOCC3C)=O)c2C1 CC1CN(C(C2CC(C)CN(C(C3CCC(C)(O)CC3)=O)C2)=O)CCN1C C1(C)(NC(C2N(C(c3cc(C)c(C)nn3)=O)CCC2C)=O)CCCC(C)(C)C1 N1(C(C(C)CCO)=O)CCCC(C2(NC(=O)C=C(Cl)Cl)CC2)C1 N1(CCNC(c2c(CCC)nco2)=O)CCCN(C(=O)OC(C)(C)C)CC1 C1(NC(=O)NCc2nc(CC(=O)OCC)[nH]n2)CCC(F)(F)C1 c1(C(=O)N)ncc(C(F)F)s1.C1(O)(CC)CN(C(C2(N(C)C)CC2)=O)C1 Cc1cc(C)c(CNC(N2CCCC(Nc3ccccc3[N+](=O)[O-])C2)=O)cc1C c1(C(=O)NCC(C)C(F)C(=O)N2CCC3CCCC23)nccc2cc[nH]c12 C1(C)(C(=O)NCCC2CCN(C(C3(O)CC(C)(C)C3)=O)CC2)CC2CCC1O2 C1(C(=O)OC(C(C)=O)C)CC2CC1(c1ccc(Cl)cc1)C2 C1(CC)C(NC(=O)C(N2CCCCC2=O)C)CCN1C(C1CCC(OC)CC1)=O c1(CN2C(C(N(C3CC3)Cc3ccc(CC)o3)=O)CSCC2)cccc(O)c1 c1(C(=O)NC23CC(C(=O)Nc4cn(C)nc4)(C2)C3)cc(Br)ccc1C#N C1(C(N(CC(C)(C)C)CCO)=O)CCCCN1C(C1CCCOC1)=O C1(CCC)(NC(=O)CC(C)C(=O)O)CCN(C(=O)C)CC1.C(=O)C(C)(C)C C(=O)(C1=C(C)S(=O)(=O)CC1)NCC(C)(CC(C)C)NC(C(CC#C)C)=O C(C(F)(C(=O)NOCCC1CC1)C(C)C)NC(C=C(CCC)C)=O C(=O)(C(O)CNC(=O)C(C)N1CCCC1)N(CCN=[N+]=[N-])CC c1(C(N2CCC(F)(C(N(CCOC)C)=O)CC2)=O)cc(Br)c(C)cc1O c1(C(N2CCC(N(C)Cc3sccc3Cl)C2)=O)cc2c(s1)CCC2 N1(C(Cc2cccc(C)c2)=O)CC2CCC1C2NC(c1ccc(C)cc1Cl)=O c1(C(N2C(C)CCC(NC(=O)C=CCF)C2)=O)cccc2c1nnn2C C12(C(=O)NC3(C4CCCN4C(c4cncc(Cl)n4)=O)CC3)COCC1C2(F)F Nc1cc(Cl)cc(F)c1C(N1CC2CC1CC2NC(c1cc2n(n1)CCC2)=O)=O c12ccc(cc1)c(=O)[nH]2.C(C(C)N(C(=O)CNC=O)C)N(CC)CC c1ccc(Cl)cc1.C(CCC(=O)N(CCCNC(=O)CO)C)N(C(=O)OC)C C(=O)(C1=CCCCCC1)N1CCC(CC=C)(NC(C)=O)C1 C(=O)(C1=C(Cl)CCCC1)N1CC(O)(CCNC(c2ccc(CO)nc2)=O)C1 C1(CNC(C2CC(C)(C)C2)=O)CN(C(C2CCCC(=O)CC2)=O)CCC1(F)F c1(CNC(c2ccc(C3(C(=O)O)CCC3)cc2)c2n(C)nnn2)cccnc1Br C1(NC(=O)CC2CCC2)(CNC(=O)CCc2cn[nH]c2)CCCC1 C(=O)(C1=NOC(CNC(=O)CCCN(C)C)C1)N1C(CC(C)C)CCC1 CC1CCC(C(=O)N(CC(O)CF)C)CN1C(=O)CSC(F)F C1(NC(C(=O)N(C)C)=O)C(C)(C)CN(C(c2ccc(C3CC3)[nH]2)=O)CC1(C)C c1(N2CCN(C(=O)NCC3CCN(CC)CC3)CC2)cnc(C)c(C)n1 CCCC(O)CC(=O)N1CCCC1C1(O)CN(C(c2nc(C(C)C)cn2C)=O)C1 Cc1cc(C(=O)NC2(CC)CC2)nc(C)n1.C1(C=O)CCN(C2CC2)C1=O.N c1(C(CNC(=O)C2CC2)NC(C(c2ccn(C)c2)C)=O)cccc(Cl)c1 C(=O)(C(C)CC(=O)N1CC(O)(CCNC(=O)C(CO)N(C)C)C1)OC Cc1ccc2oc(NC(=O)NC(COC(C)(C)C)C(F)(F)F)cc2c1 CCCCC(O)C(C)C(=O)N(CC(=O)NC(COC)CCO)C(C)C CC1CC(NC(=O)C=C(Cl)Cl)CN1C(=O)CCc1ccccc1Br C1(NC(c2n(C)cnc2Br)=O)CCN(C(c2ccc(F)cn2)=O)CC1F O=C1CC(NC(=O)COC2(C(F)(F)F)COC2)CN1 C12(C(=O)NCCCC(=O)NCCCN=[N+]=[N-])C(=O)C3CC1C2C3 N1(C(C(CC)n2cccn2)=O)CC=C(CNC(c2cc(C(C)(C)C)n[nH]2)=O)CC1 C(C(O)(CO)CO)NC(C(c1cccnc1)NC(C1CCC(=O)C1)=O)=O C1(C(N2CCN(C(c3cc4n(n3)CCC4)=O)CC2CO)=O)CC2CCC(C1)C2O c1(C(C)NC(=O)NC(C)CCC(F)(F)F)c(F)cc(Br)cc1F N1(C(C2CC(N=[N+]=[N-])C2)=O)CCOCC(C(=O)N(C2CCOC2)CCF)C1 c1(OC(C)C(=O)Oc2ccc(Br)c(Cl)c2)ccc(F)cc1Cl C(=O)(CCCN(C)N=O)NCC(Cn1cc(C(CC)(C)O)nn1)(F)F C(=O)(C(C)(C)CC)N1CC2C(CNC(C3(OCC)CCCC3)=O)(C2)C1.S N1(CCO)CCOC(c2cccc(OC(F)(F)F)c2)C1.N1(C(C2CC2)C)CCCC1 c1(C(=O)NCC(C)(C)NC(CCC)=O)ccnc2[nH]c(CC3CC3)nc12 CC1(C)CCN(C(c2ncncc2Cl)=O)CC1NC(=O)Cn1ncccc1=O N1(C(C2=NOC(C)C2C)=O)CCc2sc(CNC(=O)CSC(F)(F)F)nc2C1 c1(C(=O)NC(C)CCNC(c2cc(C3CC3)nn2C)=O)cc2ccncc2[nH]1 C12(NC(c3ccc(Br)s3)=O)CCC1CN(C(=O)C(c1cccnc1)O)C2 c1(C(C(=O)NCCN(C(=O)C(F)C2CC2)CC)O)ccc(OC)c(Br)c1 Cc1ccc(C(=O)Nc2cccc(NS(=O)(=O)C3CC3)c2)c(N)n1 c1(C(=O)NCc2c(C(N(C)Cc3c(C)ccs3)=O)cco2)cccn2ccnc12 c1(COC)ccc(C(=O)NCC)o1.C1(C=O)CN(C(C2CCO2)=O)C1.N C(=O)(C(C)(C)CCNC(=O)CC1CC=CCC1)NC(C)CC1(O)CCC1 N1(C(C(N(C(c2cc(OC)n[nH]2)=O)C)C2CC2)=O)CCC(C2(C)CC2)C1 C(C(C)(C)C(=O)N(C1CCCCCC1)C)N(C(C(C1CCC1)OC)=O)C Cc1cc(N2CC3CC(NC(=O)Cc4ccc(F)cc4)C3C2)n2ncnc2n1 C#CC1CCCN(C(=O)CC(C)NC(c2c(C)ccn2C)=O)C1 C1(C=O)CN2CCN1CC2.C1(CC=C)CN(C(C2CC2c2cnn(C)c2)=O)C1.N N1(C(C(C)NC(C)=O)=O)CCCC1C1(O)CN(C(c2csc(C)n2)=O)C1 c1(CC)ccc(C=CC(=O)N)cc1.C(=O)CS(=O)(=O)N(C)C.C1CC1.C C(C)(CCCN=c1[nH]c2ccc([N+](=O)[O-])cc2s1)NC(Cn1nnc(C)n1)=O C1(CC(=O)NCCNC(C)=O)CN(C(C2(C3CC3)CCCO2)=O)CC1C N1(C(c2cnc(C)[nH]2)=O)CCCC(CO)(NC(c2cn(CC3CC3)nn2)=O)C1 c1(C(c2cn(CC(O)CC3CCN(C(=O)CC(Cl)Cl)C3)nn2)N(C)C)ccccc1 C1(C(=O)NC(C2(O)CCCCC2)C)CCCN(CCc2ccccc2)C1 c1(OC)c(C)cc(CNC2CC(C(=O)Nc3cnccc3C)C2)cc1C CC1(C2CC2C(=O)NC(CC2CCC2)C(=O)NCC2CC2(Cl)Cl)COC1 C1(NC(CCC2CCN(C(C3(C)CCCS3)=O)CC2)=O)CC2CC1CC21CC1 C12(NC(C(C)OC3CCOC3)=O)CC(C1)C2.c1(C=O)cc(C2CC2)no1.N CC(F)(F)C(C)(C)C(=O)N1CCCC2(NC(C3(C4CCCO4)CC3)=O)CC2C1 C1(OC)CCCC(c2nnnn2CC(F)F)(NCCCCCCSC)CC1 c1(C(=O)N)ccc2c(c1)CCO2.c1(OC)cnccc1C(=O)NCCC(C)(C)C C(Cn1ccnn1)(C(=O)N1CC(C)(O)CO1)NC(c1c(CC)cccc1)=O C1(NC(Cc2cccc(OC)c2C)=O)CCC2CN(Cc3nn[nH]n3)CC2C1 c1(NC(c2c(NC(c3nc(C)[nH]n3)=O)cnc(F)c2)=O)ccc2c(c1)CNC2=O N1(C(c2c(SC)scc2)=O)CC(C)N(C(c2cccc3c2CCN3)=O)CC1C C1(C(N2CCC(F)C2)=O)CCC2CC1C2(C)C.c1(CC)conc1CC(=O)NC C1(O)(C(=O)NCc2nc(Br)n[nH]2)CCN(C2CCOCC2)CC1 CCCCCC(O)CC(=O)N1CC2CCC(NC(c3cc(Br)co3)=O)CC2C1 CC1CCC=C1C(=O)NCC1CC(C)(C)CN1C(=O)C(O)C1CC1 CCCC(C(O)C(=O)NCCC1NC(=O)NC1=O)NC(=O)CCCC(C)=O N1(C(=O)N(C(C)(C)C)C2CC2)CCC(C2CC(c3nc(CCCCO)no3)C2)C1 c1(CC)cc(F)ccc1CC(=O)NC1CCN(C(C2CCCCC2)=O)CC1F C1(C(C)NC(c2c(C)csc2)=O)CCN(C(c2cc(Cl)cs2)=O)CC1 CC(C)CC(C)(O)c1cn(CC(F)(F)CNC(C2CN(C)CCO2)=O)nn1 Cc1c(C(=O)N(CCC(C)NC(=O)C(=O)NCC(F)F)C)cccc1O CCCC(C)(CC)C(=O)N1CC(CNC(C2(C)CC(C)=NO2)=O)(OCC)C1 Cc1cc(C(=O)NC2(C)CCN(C(c3c(C)cc(O)nc3C)=O)C2)ccc1C#N C1(OC)CC(C(=O)NCC2(O)CSC2)N(C(C2CC2)=O)C1.C(C)=O.O c1(C(=O)NC(CCC)CCCNC(c2cnc(O)s2)=O)cc(C#N)c(C)cn1 CCCCC(C)C(=O)NC(C)C(CO)NC(c1cnc(C2OCCO2)s1)=O C(=O)(C1=Cc2ccccc2C1)NC1C(C)N(C(=O)CN2CCc3ccccc32)CC1 Cc1c(NCC23CCCC2C3)nc[nH]c1=NCC1CCCCC1NS(C)(=O)=O C1(C(N2C(CCCNC(CCC=CCC=C)=O)CCCC2)=O)CCCOC1C=C N1(C(CC)=O)CCN(C(c2n[nH]c(C)c2C(F)(F)F)=O)CC1C1CC1.CC=O C12(C(=O)N)CC3CC(CC(C3)O1)C2.N1(C(c2cc[nH]c2)=O)CCCC2(CCC2)C1 C(=O)(C(C1CCC1)NC(=O)CC1CCSC1)NC(C=C)C CCCC(C(=O)N(C(c1ccccc1)C(C)O)Cc1ccccc1)NC(=O)C C1(C(=O)Nc2cc(OCC)nn2C)CCN(c2ccnc(C3CC3)n2)CC1O N1(C(CC2CN(C)CC2O)=O)CCC(C)C1(C)C.C1(O)(C(=O)N)CC(C)(C)C1 c1(-c2n(C)ncn2)ccccc1NC(=O)NC(c1ccccc1)C1(CO)CCCC1 N1(C(c2cnc(OC)c(Cl)c2)=O)CC(C)CN(C(C2(C)CC(C)(C)C2)=O)CC1C n1(CC(=O)NC(CC(C)NC(=O)CN2CCC(N(C)C)CC2)C)ccccc1=O Cc1c(NCCc2ncoc2C)ncnc1NC1CCN(CC(F)(F)F)CC1C c1(CC(=O)NCC2(F)CCN(C(C34CC(C3)C4)=O)C2)ccc(F)c(F)c1 C1(NC(CCCN(C(c2c(CC)csc2)=O)C)=O)CC12CCCCCC2 C1(CC(=O)NC(CCNC(C2CCC(OC)C2)=O)C)CC2CCC1CC2 C1(C(N(CC(C)(C)Nc2ccnc(SC)n2)C)=O)CCc2nccn2C1 C(CCF)(C(=O)N1CCC1(C)C(=O)NC)NC(C1C(OC)CCC1)=O Cn1ncc(Cl)c1NC(C1CC12CN(C(=O)C=Cc1cnccn1)C2)=O c1(C(=O)N)cc2ccc(Br)nc2[nH]1.C(C)(C(=O)NC(C)(C)C1CCC1)=CC Cc1cc(C(=O)N(C)CC2(O)CCCN(C(=O)CC(C)CF)C2)cc(N)c1O c1(C(=O)NCCN(c2cc(Cl)ncn2)CC)nc2cnccc2s1 C1(NC(C(C#N)C2CC2)=O)CCC(O)C(O)CC1 CS(=O)(=O)c1sccc1CNC(c1ccccc1)c1ccco1 C1(C(N(CC(C)O)CC)=O)(CNC(=O)CC2(C)CC2)CC12CCC2 N1(c2nc3cccc(C)c3s2)CCC(C2CCCN(C(C3CCCN3C)=O)C2)C1 c1(C(=O)NC(C2CCN(C(c3ccsn3)=O)C2)C)cc(N)cc2ccccc12 CN1CCc2cc(C(=O)NC3CN(C(C4C=CCCC4)=O)C(C)(C)C3)sc2C1 C1(CN(C(C(C)c2ccsc2)=O)Cc2ccc(Cl)s2)COCCN(C(C)=O)C1 C(CCC(N)=O)(C(=O)N(CCNC(=O)Cc1ccsc1)C1CC1)N(C)C C1(CNC(C(C)OC)=O)(OC)CCN(C(c2c(C(F)(F)F)ncn2O)=O)C1 c1(OC)ccc(C(=O)NCC(CNC(=O)C(CO)N(C)C)CO)c(C)n1 C1(NC(CC2(C=C)CC2)=O)COCCN(C(C2CCN(CC(F)(F)F)CC2)=O)C1 c1(CC(=O)NCC2C(C(N3CCC(CC)C3)=O)CC2)cccc(C)c1F c1(C(=O)NC(C)CCNC(c2n[nH]c3c2CCC3)=O)cc(=O)c2ccncc2o1 C1(C(N(CCCNC(c2c(C)c[nH]n2)=O)C(C)C)=O)CC2CSCC(C1)C2 C1(C(=O)NC(C2CCN(C(=O)CCc3ccon3)C2)C)CC(C)(C)C1 CC1CC(CNC(=O)CCN2CCCC2=O)CCN1C(C1CCCN1N=O)=O C1(NC(C(C)OCC#C)=O)CCCC(CC(=O)NC(C)C)C1 N1(C(C2(CC)CCCC2)=O)CCC2(CCN(C(C3(C)CCCO3)=O)C2)C1 C(=O)(C1=CC2C=CC1C2)N1CCC(C(c2ccccn2)=O)C1 C12(CN(CCNC(=O)CC(C)(C)COC)CC)CCCN(CCC1)C2 C(=O)(C(CO)C(F)(F)F)N1CC(O)CC(NC(C(CC)n2cncn2)=O)C1 c1(CCCC)ccc(C(C)C(C)OC)cc1.C12CCCC(C1)CCN2 N1(C(c2c(C)cc(Cl)cc2)=O)CC2(CCN(C(=O)C(F)=C3CCCC3)CC2)C1 c1(NC(C)CO)ccc(S(=O)(=O)NCC2(CO)CCOC2)cc1Br CCC(C)CCCC(=O)N(C)CC=CC(=O)NC1CCN(CC)C1 c1(OC(C)C)cncc(C(=O)NCC2CCCC2)c1.C1(C=O)CC2CC2C1.N N1(C(c2nc(C)sc2)=O)CC(C(N2CCCCC2CCO)=O)CC(F)C1 C1(NC(COc2cn(C)nc2)=O)CCCC2CN(C(C3CN(CCF)C3)=O)CC12 CC(C)(C)CCCC(=O)NC1CC12CC(NC(=O)CCNC(=O)C=CCl)C2 c1(CC)cc(C(=O)NC2CC(C)(NC(c3cnnn3C)=O)C2)ccc1OC c1(SC)cccc(N2CC(C(=O)NCC(C)Oc3ccccc3Br)CC2=O)c1 c1(C(NC)=O)c2c(nn1C)CCS(=O)(=O)C2.C(C)(C)C(=O)N1CC(O)C1.C c1(OC)ccc(CC(=O)NCCC2CC(NC(=O)CC3CCCCC3O)C2)cc1 C1(C(=O)NC2(C)CCCN(C(C(C)(C)C3CCCC3)=O)C2)CC2CCC1C21CC1 c1(C(C)(C(=O)O)NC(Cc2n(C)ncn2)=O)ccc(Br)cc1 C(=O)(CC1CCc2ccc(O)cc21)N(C)CCNC(=O)CCC(F)F C1(C(N2C(CCC)CN(C(c3[nH]nnc3C)=O)CC2)=O)Cc2c(C)cccc2O1 C(CC(C)(C)C(=O)N1CCC(C)(CC(=O)NCCC(O)CCO)C1)SC C1(C)(CNC(C(C)NC(CC)=O)=O)COCCN(C(=O)Cc2cnoc2)C1 C1(c2cn(C)nc2)CCCN1Cn1nc(C2CC2)n(-c2ccccc2)c1=S N1(C(C2N(C(C(C=C)(C)O)=O)CSC2)=O)CCCC[Si](C)(C)C1 Cc1cccc(C)c1C(=O)N(C)CC1CCN(C(=O)CCCCn2ccnn2)C1 c1(CCN(C2CC3CNC2C3)C(c2ccc(C)s2)=O)ccc(Cl)c(Cl)c1 N1(C(=O)CN2CCCNC2=O)CCCC(C2CN(C(C3CCCSS3)=O)C2)C1 CC(O)CCCCCC(=O)NCC1CCC1NC(c1ccsc1Br)=O C1(N(C(Cc2c(C)ccnc2)=O)C)CN(C(=O)CN2C(=O)CCC2=O)CCC1O c1(C(N2CCC(C(C)C(N3CCCC3C(C)O)=O)CC2)=O)cccc2ccnn12 CN1CCCCC1C(=O)NCc1n[nH]cc1C(N1CCCC1C(O)CO)=O C12(NC(CN3CCCC(CC)C3)=O)CC(C)(C1)OC2C.C1(O)(C=O)CCOC1 c1(C(C(=O)NC(c2cc(NC(CC)C)sc2)C)C)c(C)noc1C C(=O)(C#CC(C)(C)CNC(=O)CC1CCCCC1C)N(CCCC)CCOC Cc1ccc(C(=O)N(C2CCCC(NC(C3CC4(CCC4)C3)=O)C2)C)nc1C N1(CC2CC(=O)N(C3CC3)C2)CCC(c2ccccc2)(CO)CC1 C1(NC(CCOCCN(C(CCc2cnc(C)o2)=O)C)=O)CCN(C)C1(C)C N1(C(C=C(C)c2cccs2)=O)CCC(C2CCCN(C(c3cocn3)=O)C2)CC1 CC(C)C(CNC(C1(c2ccnn2C)CC1)=O)NC(=O)C(F)=CC1CC1 c1(CNC(=O)NCC2(CC)CCCCO2)cc2ccc(Cl)cc2[nH]1 CCCC(C(=O)NCc1cnn(CC)c1)NC(c1cn(C)nc1CC)=O C1(NC(c2ccc(C)c(-c3cnn(C)c3)c2)=O)CCN(C(=O)C(N)=O)CC(O)C1 N1(C(c2c(C#N)scc2)=O)CCN(C(=O)CCc2ccccc2F)C2CC12 c1(C(=O)N)cn(C)c(=O)cn1.c1(SC)cccnc1C(N1CCC(C)(C)C1)=O n1(C(CC)C)cc(C(C(=O)NC(C)C)N(C)CC2CC2)cn1 CC1CN(C(C2C(C)(C)C2(C)C)=O)CC(C)N(C(=O)C=Cc2cscn2)C1 Nc1cc(Br)ccc1C(N1CCN(C(=O)Cn2cccn2)CC1C(F)F)=O C#CCCCCCCC(=O)NC1CC(NC(=O)C2=CCOCC2)C12CCOCC2 C(C1CCN(C(=O)CCn2cncn2)CC1)=CC(=O)NC(CC#C)CC c1(C(=O)NCc2cn(C3C(CN)COC3)nn2)c[nH]c(=O)c2ccnn12 Cc1ccc([N+](=O)[O-])c(C(N2CC(CC)C2)=O)c1.C(=O)(C(F)CC1CCCC1)N C(=O)(C(F)C(F)(F)F)NCC1N(C(c2cc(C(C)=O)[nH]n2)=O)CCC1 C1(NC(c2c(C)nn(C3CCC3)c2)=O)CCSC12CN(C(=O)C(C)C(F)(F)F)C2 c1(CCC(=O)NC2(C)CCN(Cc3ccc(Cl)s3)C2)cccc(C#N)c1 CCC(C)CCCCC(=O)NC1CN(C(c2ccc3occc3n2)=O)CC1(C)C N1(C(C2N(CC)CC2)=O)CCCCC(NC(=O)C(C2CCOCC2)OC)C1 C(C(C(=O)NCCCC(C)O)N(C)C)NC(C=CC=CC)=O Cc1ccc2oc(C(N3CC4CC4(NC(C4CCC5CC45)=O)C3)=O)cc2c1 C(=O)(C1CCc2c(Cl)cccc21)N.C(C)(C(=O)NCCOCC)OCCCC C1(C(=O)N)(CC)CCC(F)(F)CC1.C1(O)CN(C(c2sccc2CC#N)=O)C1 N1(c2ccc(C(=O)OCC)cn2)CCN(C(=O)CCC2CC2(Cl)Cl)CC1C N1(C(C=C(C)Cl)=O)CC2CC2(NC(=O)C(O)Cc2ccccn2)C1 C(=O)(C(F)(F)C(C)O)NC(C1(CNC(c2c[nH]c(=N)s2)=O)CC1)C C(=O)(C(C)C(F)(F)F)NC1CN(C(CC(=C=C)C)=O)CC1C c1(CNC(C2(NC(=O)CCc3nncs3)CC2)=O)ccc(F)c(F)c1 c1(C(N2CC(CCNC(CCC(C)(C)F)=O)OCC2)=O)cc(O)cc([N+](=O)[O-])c1 c1(C(=O)NCC#CCNC(C(C)C2(O)CCC2)=O)ccnc(N2CCOCC2)c1 c1(OC)cc(CO)ccc1C(=O)NCCC(C(C)C)NC(C1CCCC1(C)C)=O CC(C)(CC(F)F)C(=O)N1CCN(C(C2CCn3ncnc3C2)=O)C(CF)C1 N1(C(Cn2ncc(C#C)c2)=O)CC(CNC(=O)CCc2ccn(C)c2)CC(C)C1 CCC1CNC1=O.c1(CC(Cc2cn(C3CCOCC3)nn2)OC)ccccc1 c1(C(N2C(CC(=O)N(CCCCN(C)C)C)CC2)=O)ccc(CO)nc1 N1(C(C(c2c(C)cncc2)C)=O)CC(NC(=O)CN2CCNC(=O)C2)CC(F)C1 c1(-c2c(C)nn(C)c2)cnc(Cl)c(C(=O)N(CCCCCO)C(C)C)c1 c1(N(CCN(C)C(c2nn(C)nc2Br)=O)C)ccc(Cl)c(Cl)c1 O(N=C1CCCCCC1)CC(=O)N(C1CCN(C(c2csc(C)c2N)=O)CC1)C C1(C(N(C)CC)=O)C2CC3C(C2NC(c2ccc(=N)[nH]c2)=O)C13 N1(C(CNC(CCC(C)C)=O)=O)CC(NC(C2CC3CC2C3)=O)CC(O)C1 C1CCN(C(=O)C(C)(C)c2ccsc2)CC1.C1(CCOC)(C(=O)N)CC1.CC C=C(CNC(=O)CCCOC)CCNC(C1CC1(C)C)=O c1(SC)cccc(F)c1CNC(C1(CC2CC23CNC3)CCOC1)=O c1(C(c2nnnn2CC2CCOC2)NC(C)C2CC2)cc2occc2s1 C1CCCN(C)C1.c1ccsc1C(=O)NC.C1(C(=O)OCC)CC1C=O.N C1(=CC(=O)NCC(C)NC(=O)CC2CN(C)C2)CCCCC1(C)C C1(NC(c2coc(Cl)c2)=O)CCSC12CN(C(=O)CN1CC3CC3C1)C2 c1(CC=C)cc(F)c(NC(=O)C(C)(C)Oc2nc(C)cs2)cc1OC c1(C(N2C(C)(CC=O)CCC2)=O)cc2ncccc2[nH]1.C1(C(=O)NC)C=CCC1 Cc1nn(C)c(C)c1-c1cc(C(=O)N(C)CCNC(C2CC3CC3C2)=O)n[nH]1 c1(C(N(CC(CO)(CO)NC(=O)CCCC(N)=O)C)=O)ncc2cc(Cl)ccn12 C(=O)(C1=CCCCC1)NCc1c(C(N2CCC(C)(C(=O)OC)C2)=O)nco1 N1(C(CSC)=O)CCCC(C2CN(C(C3C4Cc5ccccc5C34)=O)C2)C1 N1(CS(c2n(C)ncc2C2OCCO2)(=O)=O)CCN(S(=O)(=O)N2CCCC2)CC1 c1(C(N2CC(O)(C3CCCN3C(C3CC3C3CC3)=O)C2)=O)onc2c1CCCC2 c1(C(N2CCC(=CCNC(=O)C(C3CCCCC3)O)CC2)=O)cc(Cl)ccc1F C(=O)(C(O)C(C)(C)CC)N(CC(CC)NC(=O)C=CC1(C)COC1)C C=C(C)CCCC(=O)NC1CC2(C1)CC2C(=O)NC1(C(N)=O)CCC1 C1(C(=O)NCC(CCC)(C)O)CCN(C(=O)c2cnncc2OC)O1 CC(C)(CCC#N)C(=O)N1CC=CC(NC(=O)Cc2cnn3c2CCCC3)C1 C(=O)(C(CC=CC)NC(C1CCC2(CC2)C1)=O)N(C(C#C)C1CCC1)C c1(CC=O)c[nH]c2cc(F)ccc12.C(CCC(=O)NC1CC1C)NC(C)=O.N c1(OC)ccc(C(N2CCC(CN(CC(=O)NC(C)C)C)CC2)=O)nc1 N1(C(c2c(OCC)cccn2)=O)CC(C)OC2(CCN(C(C3(O)CC3)=O)C2)C1 CC1CN(C(=O)CC(C)(C)N(C)C)CC1C.n1(CC=O)cc(C2CC2)nn1.N CC1CC(NC(C2CC(C)(F)C2)=O)CN1C(c1cccc(OC(F)F)c1)=O CC1CCN(C(C23C(=O)C4CC2C3C4)=O)C(C(=O)NCCC(F)(F)F)C1 c1(C(=O)N(c2cc(F)cc(Cl)c2)C2CC3CNC2C3)n[nH]c2c(F)cccc12 c1(C(=O)NCCCNC(=O)CC2CCC(C3CC3)O2)ccncc1.C1CC1.O c1(OC)cc(Nc2nnnn2C)ccc1NC(=O)NNC(=O)c1cccc(Cl)c1 CC1(C)CC(CNC(c2ncccc2Cl)=O)N(C(C2CCCN2N=O)=O)C1 N1(CC(C)O)CCN(C(C2(CO)CCN(C(=O)COC3CC3)C2)=O)CC1 N1(C(CCC=CC)=O)CC(NC(=O)C(=O)C(C)CC)CC12CCOC2 C(C(CN=c1[nH]cnc2c1SCCC2)C(F)(F)F)NC(c1c(C)sc(Cl)n1)=O N1(C(CC2CC(C)(C)OC2)=O)CC(CNC(c2nonc2N)=O)C2(CC2)C1 c1(OC)cccc(C(=O)N(C2CC2)Cc2ccc(-c3nn[nH]n3)cc2)c1 Cc1cc(Cl)cc(NC(C2CCCN2Cc2ccc(F)nc2)=O)c1Cl C(N=c1c(C#N)c[nH]c2c(F)c(F)c(F)cc12)C1CC(NC(C(C=C)(C)O)=O)C1 CCCCCCC(=O)N1CCC(C2CCCN2c2cc(Cl)nc(C(F)(F)F)n2)C1 C(C)(C)(CC(F)C(=O)NCCCC1CCOC1)NC(CCCC#C)=O C(=O)(C=C=C(C)C)NC(C(N1CC(C#C)C1)=O)C1CC1 CC(C)C(N=[N+]=[N-])C(=O)N1CCCC(C(=O)NC(C)C)CC1 C(c1cc(F)c(O)c(F)c1)=CC(N1CCCC1)=O.C1(C=O)C(F)(F)C12CC2 N1(C(C2CCN(S(=O)(=O)c3cccnc3)C2)=O)C2COCC1CC(F)C2 Cc1cc([N+](=O)[O-])c(S(=O)(=O)N2CC(c3cccc(F)c3)C2)cc1F c1(CCn2nnc(C)n2)nc(CN(C)C)nn1-c1ccnc(Br)c1 C1(N(C(COCCOC)=O)C)CCN(C(=O)C(C)(C)C)CC1C.C(C)(=O)N Cc1csc(C)c1C(=O)NCc1ccsc1C=O.c1cn(C)nc1C(N)=O C1CN(C(c2coc(C)n2)=O)C(C)(C)C1.n1(CC)nc(C=O)cc1C1CC1.N C1(C(N(C)CC2(F)CCOC2)=O)CC2(CCN(C(=O)O)CC2)C1.C(C)(C)C c1(C=O)c(C)oc(C)c1Br.c1(OCCOC)ccc(C(=O)NC2CC2)cc1 C(=O)(C1=CC(C)(C)C1)NCC1C(C)CCN1C(c1cc(O)ncn1)=O c1(-c2ncc(-c3n(C(C(=O)NCC)C)ccn3)s2)ccc(O)cc1OC c1(C(N2CCCC(O)(CCNC(C(C)NC(C)=O)=O)C2)=O)ccn2nncc2c1 c1(OC)cc(N(CCCCN(C)C(C2CC2C)=O)C)c(Cl)cc1[N+](=O)[O-] C(=O)(CCC1CCCC1)NC1CN(C(=O)OC)C1.N1(CC=O)CC(C)C1 c1(C(N2CCCC(CC(=O)NCCCn3cnnc3)C2)=O)c(O)cccc1F CCCC(C(=O)N1CCCC(CN(C)C(C2CCC(C(C)(C)O)CC2)=O)C1)OC C(=O)(C1CCCc2n[nH]cc21)N1C2CC(CC(NC(C(CC)OCC)=O)C2)C1 c1(C=O)cccc(=O)o1.C12(CCNC(Cc3ccc(C)s3)=O)CCC(CC1)C2.N c1(CC)cc(F)c(C(N2CC(F)(C)C2)=O)cc1F.C1(C)(CC=O)CC1(F)F C1(CC(=O)NCCCCCNC(C(C)(C)OC)=O)CC(C)(C)CCO1 CC1=CCC(C(N2CCC(CN(C)C(c3occc3C(C)C)=O)CC2)=O)CC1 C1(NC(CCn2ccc(C)n2)=O)CC2(CCN(C(=O)C(=O)N)CC2)C1.C1CC1.C CSC=CC(=O)NCC1CC1NC(c1c[nH]nc1-c1ccn(C)n1)=O CCC(C)CCC(=O)N(CC(C)(C)CNC(C1(C)CCNC1=O)=O)CC c1(C(=O)NCC23CC(C2)C3)cnn2cccnc12.C1(C=O)OC2CCC1C2.N c1c(C)cc([N+](=O)[O-])cc1[N+](=O)[O-].C(C(C)C(=O)NC(C)(C)CN)OCC CC(C)(CCCC(=O)NCC(N)=O)NC(=O)C(C1(O)CCCC1)F N1(C(CC2CCC(OC)CC2)=O)CCCC12CCN(C(=O)CC1(C)CC1)CC2 C#Cc1ccc(C(=O)NCC(C2(O)CCN(C(=O)CC(C)(C)O)C2)C)c(F)c1Cl CC1(C)OCCN(Cc2ccc(N3CCC(O)C3)cc2)C1CO N1(C(C2(C)CCC(F)(F)C2)=O)CCC2(CCN(C(=O)C3=CCCSC3)CC2)C1 C#CC1CCN(C(=O)CCC(CC)NC(C2CCCCC2(C)C)=O)CC1 CS(=O)(=O)c1ccc(NC(C2CN(C(c3ccc(S)cc3)=O)C2)=O)c(Cl)c1 c1(OC)ncnc(OC)c1C(=O)NCC(C)N(C)C(C1CCC1(C)C)=O CC1CC(CNC(=O)CSCCC#N)CCN1C(c1cnc(O)c(Cl)c1)=O c1(C(=O)NC2CCC(N(C(c3ncn(CC)n3)=O)C)C2)cccc2oc(C)cc12 C(=O)(CCN=c1cc[nH]cc1S(=O)(=O)N1CCS(=O)(=O)CC1CO)N(C)C c1(CN(CC(=O)OC)C(c2cnc(Cl)[nH]2)=O)cn(CC2CCCO2)nn1 C(=O)(CC(C(F)F)n1cccn1)NC1C2CN(C(CCc3nc(=N)[nH][nH]3)=O)C1C2 C1(NC(CC(C=C)CC)=O)CN(C(C2C3CCC(C3)C2(C)C)=O)CCC12CCC2 c1(C(N2CCC(O)(c3ccccc3F)C2)C(=O)NCC)nn(C)cc1Br Cc1c([N+](=O)[O-])cc(C(=O)NC(C)(C)CO)cc1[N+](=O)[O-].C1(C(=O)N)CC1 c1(CC(=O)NC(C(C)NC(=O)C=C2CCSCC2)CO)cc(F)ccc1O c1(C(=O)NCC=CCNC(C(c2cn(C)nc2)O)=O)cccc2c1COC2 c1(C(N2CC(NC(C3(C=C)CCCCC3)=O)C(OC)C2)=O)cc2ccccn2c1 N1(C(CC2(N(C(C(COC)C)=O)C)CC2)=O)CC2(CCC2)CC1C Cc1ccn2c(C(N3CCCN(C(=O)CCN4CCCC4=O)CC3)=O)cnc2c1 C12(C)CN(CCC1(C)C(=O)OC)C(=O)N2.c1(CC)ccc(CC)cc1 C(c1ccccc1)=C(CC)C(N1CC2C(CNC(=O)Cc3nc[nH]n3)C2C1)=O C(=O)(CCC(CF)CF)N1C(C(=O)NC2CC3CCCCC23)C2CC2C1 C1(NC(C(CCCC)C)=O)CCS(=O)(=O)C12CN(C(=O)CS)C2.c1cnn(C)c1 C1(NC(C2N(C(C)=O)CCOC2)=O)CCN(C(=O)CC2(O)CCC2)CC1F CCC(C)(CO)C(=O)N(C)CC1CN(C(c2csc([N+](=O)[O-])c2)=O)CCO1 Cn1cc(S(N)(=O)=O)cc1C(=O)N.C(=O)CCS(C)(=O)=O.C1(CC)CC1 Cc1cnc(CNC(=O)CNC(=O)CNC(c2cccnc2)=O)[nH]1 C1(NC(c2c(C)cncc2)=O)C(C)CN(C(=O)CC23CCC(CC2)OC3)CC1C c1(C(=O)NCCC2CCCN(C(C3CN(C(C)C)C3)=O)C2)cccc2ncnn12 C1(C(=O)NCC2OCCN(C(CC(C)(C)OC)=O)C2)Cc2ccncc2C1 c1(OC)c(C(N2CCCC(N(C(=O)CC3C=CCC3)C)CC2)=O)ccc(Cl)c1Cl c1(CNc2cc(N(C)CC3CCN(C)C3)ncn2)ccc2ccn(C)c2c1 C1(CC(=O)N(CCC)CC)C(=O)NN=C1C.C1(C=O)CC(C(F)F)C1.N C(C)(CCCCC#N)(c1nnnn1C1CCCC1)NCC(CCC)OCC N1(C(c2ccc(CSC)o2)=O)CCC2C(C1)CN2C(=O)C=Cc1scnc1C C1(NC(CCn2ncc(C)c2)=O)CC2CC(NC(c3cc(C(F)F)cs3)=O)CC12 c1(C(N2C(C)C(C)N(C(c3ns[nH]c3=O)=O)CC2)=O)cnc2ccncc2c1 C1(F)(c2cn(C(CC)CC)nn2)CCN(C(C2CN(CC(F)(F)F)C2)=O)CC1 C1(Cn2cc(C(C)OC)nn2)CCN(C(=O)CCc2nncnc2O)C12CC2 Cn1cc(F)c(C2CC2CNC(N2CC(n3ncnc3Br)C2)=O)n1 C1(C(=O)NCCCOCCNC(C2CC(C)C2)=O)CCCCN1C1CCCC1 C1(CNC(c2n(C)nnc2)=O)CCC(NC(=O)C(C)(O)C2CCOC2)CC1 C(CC(CC)C(=O)NC(CNC(c1cn(CCO)nn1)=O)CC)=CC N1(C(c2ccc(C)cc2)=O)CCC(C(N2CCN(CC(N)=O)CC2)=O)C12CCC2 c1(C(=O)NCC(C)NC(C2(C)CCC(=O)N2)=O)cccc2[nH]nc(O)c12 N1(C(CCCC)=O)CC(C)(C)C1C1CCN(C(c2oc(C3CC3)nc2C)=O)CC1 c1cc(=O)n(C(C)C)c(O)n1.C(C)(C(C)(C)C)NC(CCc1cc(C)[nH]n1)=O.N N1(C(C=CCOC)=O)CCCC(O)(CNC(C2(C)CC(C#N)C2)=O)C1 C1(C)(CC)CC(NC(=O)C2=COCC2)CN1C(c1ccc(C)cc1SC)=O C1(C(N2C(CNC(C3C(C)=C3)=O)CCC2)=O)CC(C)CC(C)C1 c1(CC(=O)NCCOC2CCN(C(c3c[nH]c(Br)c3)=O)CC2)c(O)ncnc1O c1(C(=O)NC2C(C)CN(C(c3ccc(Cl)cc3)=O)C2)ccc(F)c2ccncc12 Cc1cc(C)c(C)c(S(=O)(=O)NCc2noc(-c3ccc(F)cc3F)n2)c1C c1(C(=O)NCC2OCC(CNC(=O)Cn3cccn3)C2)cc2n(n1)CCO2 N1(C(C2C(OC)C2)=O)CCC2CCCC(C1)N2C(=O)CS(=O)(=O)C1CC1 C=C(C)CC(C(=O)NCC1(SC)CCC1)NC(=O)CC1CCCCN1C CN1C(=O)CSC1=CC(=O)NCC1C=CCC1.C12(C=O)CC(C#N)(C1)C2.N C1(CNC(c2n(C)ncc2)=O)CC2(CC2)CN1C(=O)CCc1cn[nH]c1 C1(O)(C(=O)NCCNC(c2cc(C)cc(C)n2)=O)CCc2ccccc2C1 Cc1cc(OC(F)F)c(C(=O)N(CC(C)NC(=O)CCCF)C)s1 CN1CC(NC(=O)CCC2CC(NC(=O)CCc3ccccc3)C2)CC12CCC2 n1(CC(C)C)ccc(C(=O)NCCN(C(C2CCCO2)=O)C2CC2)n1 C(=O)(CCC(CC)OC)N1CC(C=C)(CC(=O)NC2CC3C=CC2C3)C1 c1(C(N(CCCC(N2CCC(N(C)CC)C2)=O)C)=O)n[nH]c(C)c1O C(=O)C1=CC2(CN(C(=O)CC3CNC(=O)O3)C2)OC1.CC1NC(=O)NC1=O.C C=CCC(CC)C(=O)NCC(C)(C)CC1CN(C(C2CC2F)=O)C1 c1(C(N(C2CN(C(c3cnc(CCC)s3)=O)C2)C)=O)cc2c(nc1O)CCSC2 C=CCCC(O)CNC(C1(C(C)C)CCN(C(c2conc2CC)=O)C1)=O CON(CCC(=O)NCC1CC2CCC1CC2)C(=O)CCCCC1CC1 N1(C(CC)C(=O)NCCNC(=O)COCC(C)(C)C)CCN(C(C)C)CC1 Cc1nc(O)c(C(=O)NCC(C)NC(c2cccc(C#N)c2C)=O)nc1C Cc1snnc1C(=O)NCC1C=CC(NC(c2cc(C(N)=O)cs2)=O)C1 C=C(C)C1OCCC1CNC(C1CCCCCC1)c1nnnn1CCCOC c1(C(=O)NC(c2ccc(-c3cccc(CCC)c3)cc2)C)ccc2c(c1)OCO2 c1(C(N2CCCC2)=O)[nH]nc([N+](=O)[O-])c1Cl.Cc1nc(C2CC2)oc1C(=O)N.C c1(C(=O)NC(CNC(C2C(=C)CC2)=O)CC(F)(F)F)ccc2ccncc2n1 c1(OC)ccc(C(=O)C(C)OC(C2(C#N)CC(=O)C2)=O)cc1Cl N1(C(c2c(C)n(C)c(C3CC3)c2)=O)CCC2(CCC(NC(c3cnns3)=O)C2)C1 N1(C(C(C)=C(C)C)=O)CC(NC(C2COCCN2C=O)=O)C2(CC2)C1 c1(C(=O)OC)cn(CCNC(c2nnnn2C2COC2)C2CC2(Br)Br)cn1 Cc1c(NCCCC2CCC2)nc[nH]c1=NCCN(c1ccccc1)C C1(CC)CN(C(=O)CC2(NC(=O)CC3CC(C4CC4)C3)CCC2)CCO1 c1(C(=O)NC2CC(CNC(=O)CC3CC4CCC3C4)C2)cnc2cccnn12 CC(C#N)CN=c1[nH]c(=NCCC2CCCCC23CC3)c2cccc(F)c2[nH]1 C1(C(=O)NC2CC(c3ccc(F)c(Cl)c3)C2)CC(c2ccccn2)=NO1 c1(CCC)cccc(C(N2CC(C(C)NC(c3cncc(C4CC4)c3)=O)C2)=O)c1 C1(C(N2CC(CCC=C)(C(=O)Nc3ccc(Cl)cc3)C2)=O)CC(=O)CC12CCC2 c1(NC(=O)NCc2c(OCC#C)noc2C2CC2)cnc(O)cc1C c1(C(N2CCCCC(C)(C)C2)C(=O)NCC)cc(Br)cc([N+](=O)[O-])c1.C(C)(=O)O c1(OC)ncc(C)c(C(=O)NCCCCC(C)NC(C2CCCN2C=O)=O)c1Cl CCC(C)C(CC(=O)NCCc1cnnn1C)NC(=O)Cn1[nH]cnc1=N C(=O)(C(C)CC(=O)N1CC2CC2(NC(c2nc(C)n(C)n2)=O)C1)OC c1(C(N2CCC(NC(C=CC)=O)C(C)(C)C2)=O)cnn2c1CCCC2C N1(C2CCN(CCC)CC2)CCC2CC(C(=O)NCc3ccon3)C2C1 Cc1nccc(C(=O)NCc2cc(C(N3CC4CCC4(C)C3)=O)ccn2)c1N CC(C(C)C)NC(=O)CC.c1ccccc1.C(=O)C=CCO.C(C)(C)C N1(C(C(C)OCCC=C)=O)C2CCC1CC(NC(c1cccc3c1CCO3)=O)C2 N1(c2ncc(SC)cn2)CCCC(C2CN(C(c3cscn3)=O)C2)C1 Cc1ccsc1CNC(=O)CNC(C1(C)CCCS1)=O c1(C(=O)NC2CCC(C(=O)Nc3c(C)cc(Cl)nc3)OC2)cc(C)c(C)cc1I c1(C(=O)NCC2(NC(CC=C)=O)CCC2)nccc(OC)c1OC c1(N(C(CSCC)C)C)cncc(C)c1 C#Cc1cnc(C(=O)NC2(CC)CCN(C(=O)C(O)CC)CC2)c(C)c1 C1(CNC(C(C2CCC(=O)N2)C)=O)CCC(Nc2cc(Cl)ncn2)CC1 C1(C(=O)NC2CC(NC(=O)C(C)n3cnnn3)C2)(CC)CC1(F)F Cc1cccnc1CCC(=O)NCCCNC(C1CC1c1ccoc1C)=O C(=O)(C(C(C)O)NC(=O)C1CC1)NC1CN(C(CC(C)C)=O)C1 C1(C(NCP(C)(C)=O)=O)CN(C(=O)Cc2cc[nH]n2)C2(CCC2)C1 c1(C(N2CCCC(C(C)NC(C(C)(C)OC)=O)C2)=O)c(Cl)ccc(F)c1F c1(C(=O)NCC(CN(C(c2c(OCC)ccs2)=O)C)C)cc(C)c(O)nn1 N1(C(c2c(C)ncs2)=O)CCCC(O)(CNC(=O)C(=Cc2cccnc2)F)C1 c1(C(=O)NCCN(C(C2CN(S(CC)(=O)=O)C2)=O)C)cn2cccc(Cl)c2n1 Cc1cc(C(=O)NCCOCC(=O)NC2(CO)CC2)ncc1N N1(C(c2c(Cl)nc(OC)s2)=O)CC(NC(=O)Cc2cccc(C)c2)CC(C)C1 C1(C(C)C)CCC(C)CC1NCc1ccc(Br)c(C(F)(F)F)c1 c1(C(N(CC(C)NC(=O)C#CC2CCOC2)CC)=O)cc2c(F)c(F)ccc2s1 C(=O)(CS(=O)(=O)CCC(F)(F)F)N1C(CN(C(C(CC#C)C2CC2)=O)C)CCC1 N1(C(C(C(C)C)N(C)C)=O)C2CCC(C2)C1C(=O)NCCc1cc[nH]n1 c1(CCC)nc(=NCC2(C)CCCN(C(C3CCS(=O)(=O)N3)=O)C2)s[nH]1 N1(C(C2(CCCC)CC2)=O)CC2COCCC2(NC(=O)C(C)c2cccs2)C1 N1(C(C2C(O)CCN(Cc3c(C)nccc3)C2)=O)CC(O)C(O)C(O)C1CO C(=O)(C(F)(F)C(C)(C)O)N1CC(c2cn(CC(CC)O)nn2)N(C)CC1 N1(C(C2(COCC)CNC(=O)C2)=O)CC2COCC2(C(=O)NOCC=O)C1 CC(C1=NOC2COCC12)NCCCCCCCCO c1(C(N(CC(C)(C)CNC(C2CCNC2=O)=O)C)=O)nnn2ccccc12 S(=O)(=O)(c1ccc(N(CCC#N)C)cc1Br)N1C(CC)CCCC1 Cn1ncc2c(N3CC4CCC3C(NC(C3CCS(=O)(=O)CC3)=O)C4)ncnc12 N1(C(C(=O)NC2CC(CCNC(c3cnc(C)[nH]3)=O)C2)C)CCN(C)CC1 N1(C(c2cn(C)c3c2cccc3)=O)CC2(C1)CCCS2(=O)=O.C(=O)(C=CCO)N N1(C(COC2C(CC)CCCC2)=O)CC2CCC1CN2C(C1CC(N(C)C)C1)=O C1(C(N(CC)CC2CCC2)=O)CCCC1C.n1(CCC(=O)N)cnc(=N)[nH]1 c1(N2CC3CCN(C(C(c4n(C)ccc4)=O)=O)C3C2)ncnc2c(Br)cccc12 C1(NC(C=CC)=O)C(C)CCC12CCC2.C1(C=O)CC2(COC(=O)N2)C1.N C(=O)(C(C)CC(N)=O)NC(C(C)C)CNC(=O)CCc1cccs1 C1(C(N2C(C)(C)CCC2)=O)CC2(C1)CC(F)(F)C2.C1(C=O)CC2(CCC2O)C1 N1(C(c2cc(C)nn2C)C(=O)NC(C)C)CC2CCC(C1)C2(F)F N1(C(c2ccc(C#C)cc2)=O)CC2CC(C1)CN(c1ncc(CC)cn1)C2 Cc1cc(=NC2C=CCC2)[nH]c(N(C)Cc2cc(Br)cn2C)n1 C1(CNC(C=CCOC)=O)CCN(c2nc(C(=O)OCC)ns2)C12CC2 c1(N(c2cc(OC(C)C)ncn2)C2CCCN2)nc(Br)ccc1Br C1(NC(CCC=CC)=O)CN(C(c2cc3c[nH]cnc-3n2)=O)CC12CCOCC2 C1(NC(CNS(CC)(=O)=O)=O)CCC(C)CC1.N1(CC=O)CC2CCC1C2.N C(C(CC(F)(F)F)NC(c1cncn(C)c1=O)=O)NC(C(C(C)C)OC)=O c1(OC)cc(N)ccc1C(=O)NCC1CC(O)CN1C(C1CC1Br)=O c1(OC)cc(C(=O)NC(CC(N2CCOCC2C2(C)CC2)=O)C2CC2)nn1C c1(C(=O)NCCCN(C)C(C2CCC2F)=O)cc(C(F)(F)F)ccc1Br N1(C(c2n(C(C)C)ccc2)=O)CC2CCCC(NC(C3CCCCC3)=O)C2C1 c1(C(=O)NC2CC(NCc3cnc4ncccn34)C2)cc2cc(Br)ccn2n1 C=CC(CC)CC(=O)N(C1CCCN(C(=O)CCNC(N)=O)C1)CCCC n1(CC)ccc(=NC(=O)C2CN(C(C3CC3C(C)C)=O)CCC2(C)C)[nH]1 Cc1ccccc1C(C)C(=O)NCC(O)CCNC(c1ccccc1Cl)=O CC(C)CC(F)(F)C(=O)NC1CCCN(C(=O)Cn2cnc(C(F)(F)F)n2)C1C n1(CC)cncc1C(N1CCC(SC)C1)C(=O)NC(C)C N1(C(C2N(C)CCC2)=O)CC(C(=O)NCC(O)CC2CCCC2)C(C2CC2)C1 C(=O)(C(C1=NOC2CC12)N1CCN(CCS(N)(=O)=O)CC1)NCCOC N1(C(CC(C)n2cccc2)=O)CC2(CC(NC(c3cc4sccc4s3)=O)CO2)C1 c1(CNc2c(OC(C)C)cc(Br)cc2)cc(F)c(F)c(F)c1 c1cc(C)cc(C)c1.Cc1ccc(COC=O)cc1.N1(CC=O)CCC(=C)C1.N C1(NC(CC2CCN(C)CC2)=O)CN(C(=O)C(O)C(F)(F)F)CC12CCC2 C1(NC(=O)CCN2CCCC2=O)CCN(C(c2ccc(OCF)cn2)=O)CC1F C#Cc1cnn(C)c1C(N1CCC(O)C(NC(C2CCOC2)=O)C1)=O C1(NC(CSCc2[nH]c(=N)sc2)=O)CN(C(=O)CCC2CC2)CCC1CO C(=O)(C(C)CS(C)=O)N(CCN(C(C=C(C)I)=O)C)C c1(CCCCCC)nc(-c2csnc2Cl)n(C(C)C(C)(C)C)n1 Cc1ccn2cc(C(=O)NCC3(C)CCCN3C(=O)Cc3cccnc3)nc2c1 c1(CC)cc(C(=O)NC2CN(C(c3cn(CCO)nn3)=O)C2)c2c(c1)CCO2 C1(F)(C(=O)NC(C(=O)OC)CCF)CCN(C(=O)CC2CC(F)C2)CC1 C1(CNC(C=CCCC)=O)CN(C(c2cn(C)nc2C)=O)C2CCCCC12 C1(C2CCN(C(=O)C=CI)C2)CCCCN1C(C1CCS(=O)(=O)C1)=O c1(CC(N2CC(NC(C=CCN(C)CC)=O)C(O)C2)=O)cc2ccccc2o1 c1(C(N2CCC(c3nc(=N)[nH][nH]3)CC2)=O)cnc(Cl)c(Br)c1 C=C(C)C1OCCC1C(=O)NC1CC(C(N2CCCC(C)(C)C2)=O)C1 Cc1cc(C(N2CC(O)CCC2C(=O)NCc2ncc[nH]2)=O)nc(C)c1 C=CC(C)(O)C(=O)NC(C)CC.C1(CC=O)CCN1C=O.C(C)(C)C.N C1(C)(C=O)CN(C(C2COCCC2C)=O)C(C)(C)C1.CCS(=O)(=O)NCC.N c1(N2CC(CNC(c3c(C)nn(C)c3C)=O)N(C)CC2)nc(Cl)[nH]c2ncnc1-2 N1(C(C=C(C)C(C)(C)C)=O)CCN(C(=O)C(C(C)C)n2cc(C)cn2)C(C)C1 C1CN(C(c2ccc(O)c(C)c2)=O)CC12CC2.c1(CC)c(C(=O)NC)cnn1C c1(C(C(=O)NCCC#N)N(C2CCC(F)(F)CC2)C)ccc2nonc2c1 Cc1[nH]nc(C(=O)NC(C2CCN(C(=O)C3=COCC3)C2)C)c1C(F)(F)F C1(CNC(C(C2N(C(CCOCC)=O)CCC2)(C)C)=O)NC(=O)CC1(C)C C(=O)(C1=CCC(F)(F)CC1)N1CC(NC(c2cnn3ccsc23)=O)C(F)C1 N1(C(C2CC(C)(C)N(C(=O)C3=CCCCC3)C2)=O)CCC12CCCCC2 C1(NC(Cc2cc(OC)ncc2)=O)CN(C(c2ncccc2F)=O)CC12COC2 NS(=O)(=O)CCC(=O)NCCCC1CCCN1C(c1cocc1Br)=O Cc1nc(N2CC3(CN(C(=O)CC4CCCC(C)C4)C3)C2)c2c[nH]nc2n1 C1(C(N2CCN(C(C)CNC(=O)CN)CC2)=O)(COC)CCCCC1.C C1(C#N)(C(N2CCC(C)C2)=O)CCS(=O)(=O)CC1.C(CC=O)OCCCOC.N C=CCC(C(=O)N1CCOC(CNC(C)=O)C1)NC(=O)COC(CC)CC c1(C(=O)Nc2c(C)cccn2)cccc(S(=O)(=O)N2CCCC2CN(C)C)c1 c1(C(=O)N)cccc(C2CC2)c1Cl.C1(O)(C(C(=O)N(CC)CC)F)CCCC1 CCC(CO)CN=c1nc(N(C)CCc2ccc(F)cc2F)c2c([nH]1)CCS2 N1(C(C2(CCCF)CC2)=O)CCC(O)(c2cn(CC3CCCO3)nn2)CC1 C1(NC(C=COCC)=O)CN(C(c2nc(C)c(N)cc2C)=O)C2CCCCC12 CCCCC(C(=O)NCCCCNC(=O)C(C)CO)C(C)C c1(OC)ncc(NC(C2CC2C(=O)Nc2nc(OC)ccc2Br)=O)cc1F c1(C(CNC(C2CC23CC3)=O)NC(c2c(CC)nc[nH]2)=O)cccc(C)c1 N1(C(C)C)C(=O)COCC1C(N1CCC(F)C(NC(c2c[nH]c(=N)s2)=O)C1)=O c1(C(=O)OC)ncccc1C(=O)NCCC1CCCOCC1 C1(CNC(=O)CSCC(F)F)CCC2CN(C(c3cnc4c[nH]nc4c3)=O)CC12 c1(CNC(C(n2cc(CC3(O)CCSC3)nn2)C)=O)cc2ccc(Cl)cc2[nH]1 C12(CN(C3CCN(CC(=O)Nc4ccccc4Cl)CC3)C)CC1COC21CCC1 Cc1cc(S(N)(=O)=O)sc1C(=O)NC.C1CCOC1.C(=O)C(C)n1cccn1 c1(CCC(N2CC(CN(C(=O)C=Cc3cccs3)C)C2)=O)ccncn1 Cc1ccc(F)cc1CNC(C1C(C)CN1C(c1snnc1C)=O)=O c1(C(N(CC(CNC(C(C)CC(F)F)=O)C)C)=O)cc(O)c2sccc2c1 N1(C(C(C)SCCCC)=O)CC(NC(=O)CC2CCCOCC2)C(C)C1 C1(NC(C(CC)C)=O)C2CC3C(C2)C13C(=O)Nc1ccc(N(C)C)cc1 C(=O)(C(O)CC(C)(C)C)N1CC2C(CC(N3C(CC)C(O)CC3)=O)C2C1 C1(NC(C(CCC)N(C)C)=O)CC2(CCN(C(c3ccc(C)c(C#N)c3)=O)C2)C1 C1(NC(C(C)CSc2ccccc2)=O)CN(C(c2ccccc2O)=O)CCC1F N1(C(C=CC2N(C)CCC2)=O)CCC2CN(C(c3cc(=O)n(C)o3)=O)CC12 C(=O)(C1Cc2ccccc21)OCC1ON=C(C(N2CCC(OC)C2(C)C)=O)C1 C12CCC(CC1)C2.c1(CCC=O)nnc(C2CC2)o1.C1CC1C=O.CCO CC1CCC(C)(C)CN1C(=O)C(CNC(C1CC(=C2CC2)C1)=O)N(C)C N1(C(c2cc(CNC(=O)C=CC3CC3)on2)=O)CCCC2(CCCO2)C1 C(=O)(CCCCC)N1CC(OC)(C)C1.C(=O)(C(C)(C)C1CCOC1)N.C(N)=O CCCC(CNC(C1(C(C)(C)O)CC1)=O)C(=O)N1CC(C2CCCO2)C1 N1(CC)CCn2nncc2C1.c12sc(nc1O)COC2=O c1(C(=O)Nc2ccc(C(c3cccnc3)=O)cc2)ccc2ncccn12 c1ccc2c(c1)n(C)c(=O)n2C.C1(C(N(CCNC(C)C)C)=O)CC1(C)C.C Cc1ncc(C)c(=NCCCCNC(=O)C2CCCc3sccc32)[nH]1 Cc1cc2nc(NC(=O)CC(O)C(C)C)sc2cc1C CCCCC(CC(=O)Nc1cnc2ccnn2c1)NC(C1CCC(C)(O)CC1)=O Cc1cnncc1C(=O)NC1CC(NC(C2CCCOC2c2ccnn2C)=O)C1 C1(NC(CC2(CC=C)CCCC2)=O)CN(C(c2cnc(OC)s2)=O)CC1C N1(C(c2cc(CC)no2)=O)CCOCC1C(=O)NCCc1ccc(F)cc1 C(CC(C)(CC)NC(=O)CC1CCC=CCC1)NC(C(C)OCC)=O c1(CC(=O)NCCOCCCNC(C2(C)CC2F)=O)cccc2cnccc12 CCCCCCCC(=O)NC1CCC(CNC(c2cc(O)ccc2OC)=O)C1 Cc1cc(C(N2CC(NC(=O)CCCCCCBr)C(F)C2)=O)c(F)cc1F CC1(C)CC(C)(C)CN1C(c1cc2nc[nH]c2cn1)=O.C1(=CC=O)CCCC1.N Cc1cc(=NCC(C)OC(C)C)[nH]c(N2CCCC(C(N)=O)(N(C)C)C2)n1 C1CC2CC2N1C(=O)CCCN1CCCCC1.c1(COC)csc(C(=O)N)c1.C c1(C(=O)NCC2CN(C(C3(C)CC3)=O)C2)cncc(S(N)(=O)=O)c1 C(=O)(C(C(C)(C)C)NC(=O)NCc1cncc(C#N)c1)NC n1(COCC2CN(C(C(=C)CN3CCOCC3)=O)CC(C)O2)cnc([N+](=O)[O-])n1 Cc1ccc(C(=O)NCCCCCN(C(=O)CCc2ccn(C)n2)C(C)C)o1 C1(C(=O)NCCCNC(C2C(C)C2C)=O)CCCCN1CC(F)F N1(C(c2ccccc2)C)CCC(N=c2ccnc(N3CCCN(C=O)CC3)[nH]2)C1 c1(OC)ccsc1C(=O)NCCCC.C1(C=O)CC=CC1.C(C)(C)C.C=O C(=O)(C1=CCOCC1)NCC(C)CN(C)C(C1(C(F)F)CCOCC1)=O Cc1cccc([N+](=O)[O-])c1C(=O)NC(C)CC(C)NC(=O)C(O)C(C)(C)C c1(NC(C)=O)cc(C(F)(F)F)ncc1NC(=O)NC1CCCC1C1CC1 Cc1cccnc1CCNC(=O)CCN(C)C(C1C2CCC(=O)C12)=O N1(C(C(CCC)O)=O)CC2CCN(C(c3cnc4onc(C)c4c3)=O)CCC2C1 N1(C(c2c(C)noc2C(F)(F)F)=O)CCN(c2nccc(C#N)n2)CC(C)(F)C1 N1(C(c2n(C=C)ncc2)=O)CCC(C(=O)NCCCS(C)=O)C(C)C1 Cn1ncc(Br)c1-c1noc(-c2ccc(CSc3ncccn3)o2)n1 c1(C(N2C3CN(C(Cc4cnc(C)s4)=O)C(C3)C2)=O)cn2[nH]cnc(=O)c2c1C C(=O)(C(C)(C)CC(F)(F)F)NC1OCCCN(c2ncc(C(=O)OCC)nc2)C1 C1(CC(=O)N(CC(C)N(C(CCc2ncc(C)[nH]2)=O)C)C)CCCC(=O)N1 CC1(C)C(C#N)C1(C#N)C(N1CCCC1(C)c1cn(CCC=CCO)nn1)=O C1(CNC(c2cncn(C)c2=O)=O)CC2COCC2N1C(=O)CCCC(F)(F)F C#Cc1ccc(C(N2CCOC(CC(N3CCC(COC)C3)=O)C2)=O)nc1 C1CC(C)CN(C(C2CC(S(C)(=O)=O)C2)=O)C1.c1(C(C)C)ncc(C(=O)N)o1 C(=O)(C(C)(Cc1ccc(F)cc1)NC(=O)CNC(C1CC1C)=O)OC C1(CC(N2CCCCC(N(C)C(C3CC(F)(F)C3)=O)C2)=O)CC2(CCCC2)CO1 N1(C(c2c(CC)ccs2)=O)CC2(CC2)CC1C(=O)NC(c1cc(C)on1)C C(C(N)=O)(C(C)(C)C)NC(CC1CCN(C(C2N(C(C)C)CCC2)=O)C1)=O C1(CC(N2CCC(C3CCCN3C(C3CCOC3)=O)CC2)=O)CC(O)C12CCC2 c1(C(=O)NCC(C)CN(C)C(C2CCOCC2)=O)ccc2c(c1)CC(=O)N2.C C1(C=O)CC2(C1)CC21CC1.C1(C(=O)OC)CCC(C=O)O1.C1(C)CCC1.N C1(CNC(c2n(CC)ccc2)c2nnnn2C2CCC2)CCCCC1(C)C CC1(C)CC(C(N2CCC(n3ccnn3)CC2)C(=O)NCC2CCOC2)CCO1 CSC1=C(C(=O)NCC2(C)CCC(NC(c3cccc(F)c3)=O)C2)CCCC1 N1(C(C(C)OC2CCCC2)=O)CCC(C(N2CCCC(C)CC2)=O)C(C)(C)C1 Cc1nnc2n1CC(C(=O)NCCCNC(C1CCC(=C3CCC3)CC1)=O)CC2 c1(OC)cc(C)sc1C(=O)NCC1(F)CCC1.c1(C=O)nc(C)n(C)n1 C(=O)(C(O)C(C(C)C)O)NCC(CN(C(c1c(CCC)n(C)nc1)=O)C)(C)C Cc1cccc(C(=O)NC2CC(CC(=O)NC)C2(C)C)c1.c1nn(C)c(=O)o1 c1(C(=O)N(C2CC3CNC2C3)Cc2ccc(F)c(F)c2)c(Cl)ccc(Br)c1Cl C1(C(=O)NCCC)(COCC=C)C=CCN1C(=O)C(c1ccccc1)C.S C(=O)(C(C)(C)CCCO)N(CCNC(=O)CC)CC.c1ccc(F)c(F)c1.O C1(CNC(C(C)O)=O)CC(C)(C)CN1C(c1ccnc(C(C)(C)C)n1)=O c1(C(=O)NC2CCN(C(c3cc4c(s3)COCC4)=O)C2)nc2cc(F)ccc2s1 C12(C=O)CC3CC(C)(C1)CC(F)(C3)C2.N1(C(C=CC)=O)CC(F)CC1C N1(C(C(Br)=C(C)C)=O)CCC2(CCCC2C)CC1.C1(C=O)CC(N(C)C)C1.N C(=O)(CCCC(=O)N)NCC.C1CC(C)N(C(C2CCCC(C(N)=O)C2)=O)C1 C1(NCc2ccc(C)nc2)CN(C(c2cccc(O)n2)=O)CCC1(F)F N1(C(c2cnc(C)[nH]2)=O)CCC2(CCCN(C(c3cc(C)c(Br)s3)=O)C2)C1 N1(C(C(CC)NCC)=O)CC(CCNC(=O)C(C)(C)C2CCCC2)C(C)C1.C c1(CN(C)C)ccc(NC(c2cccc(NCc3ccccn3)c2)=O)cc1O c1(C(C=O)C)cc(F)cc(F)c1.c1(C(N2CC(OC)C2)=O)cn(C)c(O)n1.C c1(C(C)NC(COCC(C)C)=O)nc(C=O)co1.c1(CC)nc(=O)o[nH]1.N Cc1cn2c(n1)CCC(CN(C(=O)CCN1CCCCC1)C)C2 CCCC(C(=O)NCC12CC(C1)C2)C(C)C.c1(C=O)ccc[nH]1.C1CCC1.N S(=O)(=O)(c1ccc(N2CC(C)C(C)C2)nc1)N(CCC(C)C)CCC(C)C c1(C(N(C(CNC(c2ccc(C#C)cc2)=O)C)CC)=O)cc2c(s1)CCC2=O c1(C(N2C(C)(CNC(CC(COC)(C)O)=O)CCC2)=O)ccc2cccnc2c1 c1(C(N(C2C(C)CCC2)C)=O)ccc2c(n1)CN(C(C1CCCCO1)=O)CC2 Cc1cc2ccc(C(N3CCC(NC(c4cnc(Cl)cc4N)=O)CC3)=O)cc2o1 N1(CCNC(CC2(C)CC2(F)Cl)=O)CCC(NC(C2CC2(Cl)Cl)=O)CC1 C#Cc1ccc(C)cc1.C1(C(N(CC(=O)N)CC(C)C)=O)C2CCC(=O)C12 Cc1cc(C(=O)NCC2CCC2NC(=O)CC2CN3CCC2CC3)nc(O)n1 c1(C(=O)NC2CC(NC(c3ccnc(OC)n3)=O)C2)ccc(Cl)cc1N c1(C=O)ccc(C#N)c(C)c1.C1(C(=O)NCCNC(CC)=O)CC1(C)C.N Cc1c[nH]c(=NCCCNC(=O)COc2cccc(CC3CC3)c2)nc1O C(=O)(C1=C(Cl)CCCC1)N(CCC(=O)NCCCCCCCO)CC=C C(=O)C1=CS(=O)CCC1.c1(C(=O)OC)cccc(NC2CCCCC2C=O)c1.N CCC(C)C(C)CNC(C1CCCN1C(c1c[nH]nc1C1CC1)=O)=O n1(CC)cnc2c(NCC3CCCC3)nc(N3CCCC(C)(C(F)(F)F)C3)nc12 N1(CC)CCOCC1CC(=O)NC1(C)CC(NC(=O)C=Cc2cc[nH]n2)C1 Cc1cncc(NC(=O)C(Cc2cn[nH]c2)NC(c2[nH]cc(C)c2C)=O)c1 N1(C(C(C=C)O)=O)CCC(C2CCCN(C(c3nc(=O)n(C)[nH]3)=O)CC2)CC1 N#CC1(CC(=O)NCC(CO)NC(C2CCCCO2)=O)CCS(=O)(=O)CC1 C1(C(=O)NC(CCC=C)C)CCCCN1C(c1n[nH]c(C)c1Cl)=O C1(CCCC)CCC(C(N2CCSC(C(=O)Nc3cc(CO)ccn3)C2)=O)CC1 C1CS(=O)(=O)CC1.c1(C=O)cc(N)ccc1C.c1(COC)cc(C=O)no1.N C1(CC(=O)OC)Cc2ccccc2CN1C(c1nc(O)c([N+](=O)[O-])c(O)n1)=O N1(C(C)C)CCN(C(=O)C=CC(=O)N(C)C)CC1.c1(CC)c[nH]nc1C=O.N C1(CC=C)CC(O)CC(CNC(Cc2ccc(OC)cc2)C(C)C)O1 C(=O)(C(C)OC(=O)C=C(CC)C#N)NCCC N1(S(Cc2cccc(C)c2)(=O)=O)CC2CN(C(c3ccc(Cl)c(Cl)c3)=O)CC2C1 C(=O)(C1CCCc2ccccc21)N(CCn1cc(-c2cc(Cl)ccc2C)nn1)CC C1(C(C)(C)C)CCN(Cc2cn(-c3cccc(Cl)c3Cl)nn2)C(C(N)=O)C1 CC(C)(C)C#CC(=O)N1CC(O)CC1(C)C(=O)Nc1cnn(C(C)(C)C)c1 N1(C(c2cnc(Br)s2)C(=O)Nc2ccc(F)cc2)CCc2ccc(Cl)c(Cl)c2C1 C#Cc1ccc(C(=O)NCC23CC(C2)C(C)O3)cc1Cl.C(=O)C1=CCCCO1.N Cn1cncc1C(=O)C(N1CCC(C(=O)NC2(c3ncc[nH]3)CC2)C1)=O C1(C(N2CCC(CCNC(CCCOCC)=O)C2)=O)CCC(=C(F)F)CC1 Cc1ncc(C(c2nnnn2CCCF)NCCCCO)cn1 N1(C(C=O)C)CC2CCCN(C(=O)Cc3ccc(O)nc3)C2C1.C(=O)NCC.N C1(NC(CCCc2c(C)ccs2)=O)(CO)CCN(C(=O)CCC2CCCOC2)C1 N1(C(C)C)CCCCC1C(=O)NCCN1CCN(C(=O)CCC2CC2)CC1 N1(C(CN(S(C)(=O)=O)C)=O)CC(NC(=O)C)CC12CCC2.c1cccs1.C C(=O)(CCCCN(C)C(c1csnn1)=O)NC(COCC)C C(=O)(C(CCC)O)NCC1(F)CC(CNC(CC2(C=C)CCC2)=O)C1.C C(=O)(CC(C)CC(C)(C)C)N1C2CC(CN(C(c3c(OC)noc3C)=O)C2)C1 C(C)(C)(C(C)CC(=O)N(C)CC1(C#N)CC1)NC(C1CC(SC)C1)=O C(C(CC1CC1)CO)NC(=O)CN(C(=O)Cn1cccn1)C1CCC1 c1(C(=O)N)cc(Cl)c(Cl)c([N+](=O)[O-])c1.C1(C(N(C(C)C)C)=O)CNC(=O)N1C C1(NC(=O)NC(C2CCCOC2)C)CN(C(=O)OC(C)(C)C)CC1(C)C c1(C(N(CCCN(C(C(=Cc2ccccn2)C)=O)C)C)=O)coc2c1CSC2 Cn1ccc2cc(CN3CCSC(C(N4CCC5(CC4)OCCO5)=O)C3)ccc12 C1(CCC)CCCN(C(=O)Cc2nnc(C)s2)C1.C1(C(=O)N)CCC(C)=C(C)C1 N1(C(C2(N(C)C)CCCOC2)=O)CC2(C1)SCCC2NC(=O)CCn1ccnn1 Cc1cc(NC(c2ccc(Cl)c(N(C(C)C)CC3CCOC3)c2)=O)ccc1C#N Cc1c(CCC(=O)NC2C=CCN(C(C3CCC3C)=O)C2)cnn1C Cc1ccc(C(=O)NCC2(C)CCC(NC(=O)CC(C)C)C2)c(Cl)c1C n1(C2CN(C(C(C3CCC3)OCC)=O)C2)ccnn1.c1(CC=O)ccsc1.C C(=O)(C(CC(C)C)NC(c1cccc(F)c1O)=O)NC1C(CC)CCCC1 N1(C(C2C3CCC2CC3)=O)CCCC(C(C)C=O)C1.C1(C=O)(COC)CC1.N C1(CNC(Cc2c(C)con2)=O)C(C)CCN1C(c1onc(Br)c1C)=O N1(C(c2n(CC)ccn2)=O)CC(O)CC1C(=O)NCC1CCOC1 N1(C(C2CC(CNC(C3(CC)CCCO3)=O)C2)=O)CC2COCC2(C)C1 N1(C(CC2C(COC)C2)=O)CCCCCC1C(=O)NCC(C)C(=O)OC C(=O)(CCS(=O)(=O)C(F)(F)F)N(CCn1ccnn1)CC.C(C)C(=O)O.C S(=O)(=O)(c1ccc(NCC2CCCN(C)C2)c(Cl)c1)N1CCn2c(C)cnc2C1 c1(OC)cc(-c2nc(C3CC3)nn2CC2CC2C)c2cnccc2c1 C(=O)(C(C)C(C)(C)C)NCC(CC)NC(c1ccc(F)c(C(C)C)c1)=O C1(NC(c2cn(CCC)nn2)=O)CCCCC1C(=O)NCC(F)(F)C(F)F c1(C(=O)NCC(C)(C2CC2)NC(=O)C2=CCSC2)cccc(Cl)c1O C(=O)(CC1=CCN(C)CC1)N1C(CC(N2CCC(C(=O)OCC)C2)=O)CC1 CCC(C)(O)C(=O)N1CC(N2CC(NC(=O)CCc3ccncc3)CC2=O)C1 N1(C(C(CCOC)OC)=O)Cc2[nH]nc(C(N3CCN(C)C(C)C3C)=O)c2C1 c1cc(F)c(C)cn1.c1(C(=O)OCC)ccc(CN2CCC(C)(C=O)C2)nc1 c1(C(=O)NC2CC3CN(c4ncnc5c4CCO5)CC23)noc2ccc(F)cc12 S(=O)(=O)(c1cc(Cl)c(F)cc1F)N1CCCN(C(Cn2ccc(C)n2)=O)CC1 c1(-n2c(C(C(CN(C)C)(C)C)NCCS(C)=O)nnn2)ccc2c(c1)CCC2 N1(Cc2ccc(OCC)s2)CCN(Cc2c[nH]ccc2=N)CC1 C1(C(=O)NCC(c2nncn2C)C)(SC)CN(C(c2cn(C3CC3)nn2)=O)C1 N1(C(c2ccc(C)o2)=O)CCC(C(C)CNC(C2(n3cnnn3)CC2)=O)CC1 N1(C(CNS(CC)(=O)=O)=O)CCC2CN(C(c3ccc(OC)cc3F)=O)C2C1 N1(C(C(C#C)(C)C)=O)CC(OC)CC(NC(=O)Cc2coc(C)n2)C1 CCC(CC)CCC(=O)N1CCC(C)(CC(=O)NCC2CC(O)CN2C)C1 c1(C(=O)N)scc(Cl)c1Cl.O=C(CC(O)C1CCCC1)NCC1(O)CC(C)C1 CC(CC(=O)NC(CC(=O)NCC1CN2CCC1CC2)C(C)(C)C)C(F)(F)F N1(C(c2c(NCC)scn2)=O)CCC(C)(C)C1.c1(C=O)oc(C(F)F)cc1C C(=O)(C1CCCc2scnc21)N(CC(CNC(Cn1cc(C(C)=O)nn1)=O)O)C C1(CNC(CC2CC(=C)C2)=O)(CO)CCN(C(=O)C(O)CN2CCCC2)CC1 N1(c2ccc(C(=O)OC)cn2)CCC(NC(=O)CC2CCCCC2C)CC1C c1(-n2ncc(C3C(CN4CC(O)C(c5ccccc5)C4)C3)c2)ccc(Cl)c(Cl)c1 C1(NC(C=COCC)=O)CCCCC12CCCN(C(c1ncccc1F)=O)C2 Cc1cnc(C#N)c(-c2cc(N3CCC(CCCO)CC3)n[nH]2)c1 C1(C(=O)NC2(C)CCN(C(C(C)CF)=O)C2)CC12CCC(F)(F)CC2 c1(C(=O)NCC(C)(O)CNC(c2nncs2)=O)cnc(O)n(C2CC2)c1=O c1(C(=O)NC2CC(C(N3CC(OC)C(O)C3)=O)C2)cc(F)cc(F)c1Cl C(=O)(CCC1=NNC(=O)CC1)NC1C2(CN(C(C(CCOC)C)=O)C2)CCC1 c1(NC(CC)C(c2cccc(Br)c2)C)nc(C)cc(=NCC2COC(C)(C)CO2)[nH]1 C(=O)(CC(C)(C)C(=O)O)N1CCC(C)(CC(N2CCCC(OCC)CC2)=O)C1 c1(C(N2CCC(N(C(=O)C(F)F)CC3CCCC3)CC2)=O)ccc([N+](=O)[O-])o1 N1(C(CSCCC)=O)CCCCC1CN(C)C(C12CC(F)C1C2)=O Cc1cc(C(=O)NCC23CC2CN(C(C2CC24CCC4)=O)C3)c2nccn2c1 C1(CC)CN(C(=O)Cc2n[nH]c(=N)s2)CCN1C(=O)CC1C=CCCC1 C=CCC(CC)C(=O)NCCC(O)CNC(c1cc(CC2CCC2)c[nH]1)=O c1(NCC2CCC(SCC)CC2)nccc(=NCC2(C)CCN(C)CC2)[nH]1 C(C(C)(C)CCCO)NC(C1N(C(c2c(C)coc2)=O)CC1)=O C(C(CNC(C1CC1c1ccccc1)=O)CO)NC(c1ccsc1Cl)=O C(=O)(C1CCCn2cncc21)N1CCCC(NC(C2COC2)=O)C1 N1(C(C2CC(C)OC2)=O)CCCC2(CCN(CC3CCC(F)(F)C3)C2)C1 c1ccccc1F.c1(C(CNC(C2(C)C(C)C2)=O)NC(=O)C)cccc(Cl)c1.O c1(C(=O)NCCCN(C)C(C2(C)CCC(=O)C2)=O)c(F)ccc2[nH]ccc12 c1(C(N(C)CC2CCN(C(=O)COC3CCC3)C2)=O)ccc2[nH]ccc2c1 C1(CC(C)NCCc2cc(-c3ccncc3)n[nH]2)CCCS1(=O)=O c12ccc(c(Cl)n1)NC(=O)C1CC(C1)O2.C1(CC)CC(O)(c2cccnc2)C1 C(=O)(C(CCCCNC(=O)C1CCc2ccccc21)CC(F)(F)F)OC C1(NC2CCC(NC(N(C)Cc3onc(C(C)C)n3)=O)C2)COC(C)(C)O1 C1(NC(CC(OCC)O)=O)COCCC1NC(=O)C=Cc1ccncc1.C C(=O)(C(C)(C)CCC(=O)N(CCCCNC(=O)C(Br)=C(C)C)C)OC Cc1ccc(C)c(C(=O)NCC(C)(C)NC(=O)CO)c1.c1(CC)ccccc1 N1(C(C(=O)NCCc2cc(OC)ncc2)=O)CC2CCCC(=O)NC2C1 Cc1cc2ncc(CNC(=O)NCC(C)(C)CC(C)C)cn2n1 c1(SC)cc(C)ccc1C(=O)N(CCCNC(C1CC2(CSC2)C1)=O)C CCCCC(CCCC)NC(C1CN(C(c2n[nH]c(C)c2C)=O)CCC1(C)C)=O N1(O)CCOCC(F)C1.C(=O)C(C)(CC)C(N)=O.CCC(C)Cc1ccco1.C=O c1(C(=O)OC)cc(F)cc(C)c1NC(=O)NCCC1CCCCC1C C(c1ccc(Br)cc1)=CC(=O)N(C1CCN(C(C2CCC2)=O)C1)C.N(C)C.C C1(C)(C=O)CCCNC1=O.C1(NC(c2c(NCC)scn2)=O)CCCC(C)C1 c1(SCC(=O)NC2(CCNC(C3C=CCCC3)=O)CCC2)cccc[n+]1[O-] Cc1ccc([N+](=O)[O-])c(C)c1C(=O)NCC1CCN(c2cc(C3CC3)ncn2)C1 CCC(CO)C(=O)N1CCCC1CNC(C1CCC(C)(C)C1)=O c1(C(N2C(C)CC(NC(=O)C=CC3CCCCC3)CC2)=O)cncc2ccsc12 C1(CN(C(=O)CC2CCN(C(=O)Cc3ccc[nH]3)CC2)C)CCCC2CC12 N1(C(CSCCOC)=O)CCN(C(=O)CCC2CCOCC2)CC1C1CCCC1 N1(C(C(C2CC2)SC)=O)CCCCC1CNC(=O)CCc1cn(C)cn1 n1(CCC(N2CCC(CN(N3CCCC3)CC3CCNC3)C2)=O)ccc2cccnc12 CC1CCC(C)C1NC(C1(NC(=O)C=C2CCCCC2)CSC1)=O CCC(C)C(O)C(=O)NC(CN(C)C(c1cnn(C)c1C1CC1)=O)CC c1(OC)ccc2cc(C(=O)NC(CO)C(C)NC(=O)C(F)C(C)C)nnc2c1 c1(C(=O)NCC2CC2C2CC(F)(F)C2)cc2cccnc2nc1C1CC1 c1(OC)noc(C)c1C(N1CCC(C(=O)NOCC(N)=O)C1)=O N1(C(C2(CC#C)CCCC2)=O)CCC(CNC(C2CCC(OC)C2)=O)(O)C1 C12(CNC(N3C(c4ccc(C)cc4C)CCC3)=O)COCC(COC1)O2 N(C1CCc2c(Br)cccc21)C(C1CC(O)CN1C(c1ccc(I)c(Cl)c1)=O)=O Cc1nonc1CC(=O)NCC12CC(NC(=O)C(c3ccccc3)F)(C1)C2 c1(C(=O)NCC(C)NC(CN(C(C)C)C)=O)cnn(CC2CCOC2)c1 N1(CC2(OC)CC(C)CC(C)C2)CCCC2(CCOC2)C1 S(=O)(=O)(c1cnccc1N(CC(C)C(C)C)C)NC(COC)CO c1(C(=O)NC2C(NC(C3(C)CCOCC3)=O)CC2)cc2occ(Br)c2[nH]1 Cc1cc(C)c(C(N2CC3C(CNC(=O)C(C)C(C)O)C3C2)=O)c(O)n1 c1(CNC)ccc([N+](=O)[O-])c(F)c1.c1cc(O)ccc1NC(C1CC1)=O c1(C(N2CC(N(C(CS(CC)(=O)=O)=O)C)C2)=O)cc(S(=O)(=O)O)ccc1O c1(CC)cccc(C(=O)NCC2COCC2NC(=O)C(F)C(C)C)c1 N1(C(C(C2CC2)OC)=O)CC(OC)C(C(=O)NCC2(F)CC(O)C2)C1 c1(OC)cc(C(=O)NCCC(C)N(C)C(C2CCCC(N(C)C)C2)=O)cc(C)c1 N1(C(c2c(C)cc[nH]c2=N)=O)CCC2C(C1)CN2C(c1cc(C(C)(C)C)on1)=O C(CCCC(=O)NC1CCCC1NC(=O)CNC(=O)C1CC1)N(C)C N1(C(CCC=C)=O)CCC2CN(C(=O)CC(C)(C)CCC)CC2CC1 c1(C(=O)NC(C2N(C(C(COC)C)=O)CCC2)C)ccc2c(c1)CNC2=O c1(C(N2C(CNC(CSC(C)C)=O)CCCC2)=O)cc2ccc(F)c(F)c2o1 C1(CC(=O)NC(CN(C(C(C)C2CCCC2)=O)C)(C)C)CCC=CCC1 N1(C(C2(SC)CC2)=O)CC(NC(c2cn(CC(F)(F)F)cn2)=O)C(SC)C1 C(C(C)(C)CC(=O)NCc1ccsc1C=O)N(C)C.C1CC(=O)N(C)C1=O.N N1(C(c2ccc(CC)cc2)=O)C2CCC(C(N3CCn4ccnc4C3)=O)C1CC2 N1(C(C(C(C)C)F)=O)CC23CCCC2(C1)CN(C(c1cc(CCCO)on1)=O)C3 C(CN=c1ncc(Cl)c[nH]1)C1CCN(C(CC(=C)C)=O)CC1 C1(NC(c2ccc(C)nn2)=O)CCCCCN(C(=O)C(C2CCCCC2)C)C1 N1(C(CC(C)CF)=O)CCC(F)C(NC(=O)CCOCc2ccccc2)C1 C1(COC)CC(C)N(C(c2ccon2)=O)C1.c1(C=O)ccc(C(N)=O)o1.N C=C(C)C(CC(=O)N1CC2(CC2)CC1CNC(C1CCSC1)=O)OCC CN1N=C(CC(=O)N2CCCC3(NC(C4CC5CCC4O5)=O)CCCC23)CC1=O c1(OC)cccc(Cl)c1C(N1CCOCC(NC(=O)C(C)NC(N)=O)C1)=O c1(C(=O)NC2CC23CC(NC(C2CC24CCSCC4)=O)C3)ccc2c(c1)CCC2 c1(CC#N)ccc(C(=O)NC(c2ccc(C(F)(F)F)cc2)CF)cc1 C1(C(=O)NC2CC(NC(CCc3cc(OC)no3)=O)C2)CCCCC1C C(=O)(C1CCc2cc(F)ccc21)N1CC(COC)N(C(=O)CN=S(C)(C)=O)CC1 C(=O)(CCCS(N)(=O)=O)N1CC2(C(NC(C3C(C)OCCC3)=O)CC2)C1 Cc1c(C(=O)NC2CCCC(NC(C34CC(C3)C4)=O)CC2)cccc1F N1(C(CC(=O)NCC)=O)CCC(NC(=O)Cn2cc(O)c(=O)cc2C)CC1C C(=O)(C(CNC(=O)C1=NOC(C)C1C)C(C)(C)C)Nc1c(C)cc(F)nc1 C=C1CC2(C1)CC(C(=O)N(C)CC1CN(C(C3CCCCC3(F)F)=O)CCO1)C2 CC1(c2cn(Cc3csc(Br)n3)nn2)CCN(C(c2occc2C2CC2)=O)C1 N1(C(c2csc(C(F)(F)F)n2)C(=O)NCCC)CCOC2(CC2)C1 N1(C(C(C)NS(C)(=O)=O)=O)CCCC(C2CCN(C(c3nscc3N)=O)CC2)C1 C1(N(C)C(C2CC3C=CC2C3)=O)CCCCN(C(=O)C2=C(Cl)CC2)C1 c1(NC(Cc2nc(-c3c(OC)ccc(Br)c3)sc2)=O)cc(Cl)c(F)cc1[N+](=O)[O-] N1(C(C(C)(C)C2CCN(C(=O)CN3CC4CC4C3)C2)=O)CC(O)C(C2CC2)C1 C1(O)(Cc2occ(C)n2)CCN(C(=O)CCCn2cc(C3CC3CO)nn2)CC1 c1(OC)ccc(C(N2CCC(N(C)C(C3OCCOC3(C)C)=O)C2)=O)c(OC)c1 C1(NC(COCC#C)=O)CCC12CN(C(c1ccc(C(C)=O)c(O)c1)=O)C2 Cc1cc(C(N2CCCC2CN(C(=O)C(C)C(C)C)C)=O)cnc1C(F)F N1(C(Cc2c(C)nc[nH]2)=O)CC2(NC(c3coc4c3CCCC4)=O)CCC1CC2 C(=O)(C(C)(F)C(C)(C)F)N1CCC(O)(C(C)NC(=O)CCCN(C)C)C1 c1(N(CC)CC)ccc(C(=O)NCC(C)C)cc1.c1(C=O)nn(C)cc1N.N C(=O)(CCCCC(F)(F)F)N1CC(CC)N(C(=O)C(C(C)C)n2cnnc2)CC1 CC1C(C(F)(F)F)N(Cc2ccccc2)CN1CC(c1ccccc1)O c1(CC(N2CCC(C)C2c2cn(C3(C)CCOCC3)nn2)=O)cc(F)cc(F)c1 c1(C(N2OCC(n3cc(CCCC)nn3)C2)=O)ncn2ccc(C)cc12 C1(C(=O)Nc2ccc(I)cc2)C2CCCC1CN(C(c1cc(F)ccc1O)=O)C2 Cc1c[nH]cc(C(=O)NCC2CCCN2C(C2CC2C)=O)c1=O c1(C(C)C(=O)NCCC2(C)CC2)nc(F)ccc1Cl.C1(C=O)CCCC1(F)F.N C(=O)(NN1CCCC1C(=O)NC(C)Cc1ccnn1C)c1n(OC)cnc1C CC1(C)CC(NC(=O)C(F)=CCCF)CCN(C(c2cc(C#N)ccc2Cl)=O)C1 C1(NC(c2cc(C)sn2)=O)CCOC12CCN(C(C1CN(C(N)=O)C1)=O)CC2 N1(C(c2cc(C)ncc2)=O)CCC(O)(CCNC(c2cc(CO)n(C)n2)=O)CC1 c1(NC(c2n(CC)nnn2)CCc2ccsc2)ccc(-c2cn[nH]c2)cc1OC N1(C(c2cnccc2)=O)CC2(CCC(O)CC2)C1.C(=O)(COCC(=O)N)NC Cn1ccnc1C(=O)NCC1CCN1C(c1ccc(-c2cccnc2)s1)=O N(C1c2ccccc2CC1NC(=O)CC1COC2CC1C2)C(C1N(CC)CC1)=O c1(CN2CCC(CC#C)C2)cc2ccnc(F)c2o1 c1(CC)c(C(=O)NC(C2CCOC2)CNC(=O)C)nnn1C.c1ncc[nH]1.S Cc1oc([N+](=O)[O-])cc1C(=O)NC1CN(C(=O)CC2CC(=O)NC2=O)CC1C CC1CN(C(=O)CC2CCC3CC3C2)CCN1C(=O)CCCCF C(CC(C(F)(F)F)N1CCOCC1)OC(=O)C(c1ccc(Cl)s1)=O c1(C(C(=O)NCCOC)N(C(C2CCC2)C)CC)cnn(CC)c1 c1(CN(C2CN(C(C3CC4CC4C3)=O)CC2)CC(=O)OC)cccc(C)c1 CC(C)CCN=C(NCCCC1CCCCO1)NCC1CS(=O)(=O)CCO1 C(=O)(CCCCCC#N)N1CC=CC(NC(c2nn(C)c(Cl)c2Br)=O)C1 c1(C(N2C(C)CCC(NC(CC(=C)C)=O)C2)=O)ccc2c(n1)CCC(C)C2 c1(C(=O)NCC2CCN(C(C(C)CC(N)=O)=O)C2)cc2c(nn1)CCC2 C1(NC(CN(C)OC)=O)CC(C(=O)NC(C)COCC2CC2)C1.C c1(CC(=O)NC2(CNC(C3CCC4CCC34)=O)CCCC2)cnn2ccccc12 c1(C(=O)NC(C2CCCN(C(c3c(C)coc3)=O)C2)C)cccc2ccnn12 C1(CCO)(CNC(=O)Nc2c(C(C)C)c[nH]n2)CCCCC1 C1(NC(C(CC)OCC)=O)CC12CCN(C(=O)C(C#N)(CC)CC)CC2 N1(CCNC(c2ccnc(O)c2)=O)CCN(C(=O)CN2CC=CC2)CC1 C(C)(CC(F)(F)F)NC(c1cc(C)oc1C)=O.C(=O)(CC)N.[SH](C)(=O)=O C1(C(=O)NC(c2ccc(C)cc2)C)CCN(C(C2(CF)CC2)=O)CC1(C)C Cc1c(C(N2CC3(CCN(C(=O)C(O)CC[S+](C)C)C3)C2)=O)nn2c1CCCC2 Cc1nc(C)n(-c2ccc(-c3noc(C(CC(C)C)c4nc[nH]n4)n3)cc2)n1 c1(CC(N2CCC(OCCNC(C(C)C)=O)C2)=O)cccc(C(F)(F)F)n1 c1(OC)ccc(C(N2CCCC2(C)CNC(C2CC23CC3)=O)=O)c(O)c1 C1(C)(C(=O)NCC2(O)CN(C(C3C(CCOC)C3)=O)C2)CC=CCC1 CCCC(CC(C)C)C(=O)N1CCN(C(c2nnc(C)s2)=O)C(C)C1 c1(OC)cccc(OC)c1CC(=O)N(CCC)C.c1(C(=O)N)[nH]ccc1C1CC1 c1(OC)cc(C)cc(C(N2CCC(CNC(C3CCCS3)=O)CC2C)=O)c1C S(=O)(=O)(c1cccc(S(=O)(=O)N2CCC(C)(F)C2)c1)N(C1CCCN(C)C1)C N1(C(=O)CCF)CCN(C(C2CC23CCOCC3)=O)C(c2ccccc2)C1 C(CNC(C1CCC1(F)F)=O)(C(=O)N1CC(O)(c2nn[nH]n2)C1)N(C)C C1(NC(c2ccc(CC)cc2)=O)CCN(C(=O)C(CO)C(C)C)CC1CC C(C(=O)NCCc1cn(CC(N)=O)nn1)(C(C)C)N(CC)C.c1ccccc1 C1CC12CCN(C(=O)C)CC2.[SH](=O)(=O)c1cccs1.C(C(=O)NC)OCC Cc1cn2c(n1)CC(C(=O)NCC1CC13CCN(C(=O)CC(C)C1CC1)CC3)C2 N1(C(C=COCC)=O)CCC(F)C(NC(c2ncc(F)c(OC)n2)=O)C1 c1(C(=O)NCc2ccc([N+](=O)[O-])cc2Cl)ccc2c(c1)C(=O)CCS2 c1(CC)ccc(C(C)=CC(N2CC(C)C(C)(C)C2)=O)cc1.C(=O)C.C1CC1 C1(C)(CNC(CCN(C(CC)CC)C)=O)COCCN(C(=O)C(C)(C)C#N)C1 c1(C(N(CCNC(C2C(c3ccc(C)s3)C2)=O)C)=O)cccc2c1NCC2 N1(C(C2CNC(=O)N2)=O)CCC(NC(C2(c3ccccc3)CCOCC2)=O)CC1 C1(C(=O)NCC(CNC(c2coc(CO)c2)=O)O)CC2C(C1)C2(F)F C#CCC(C(=O)N1CCC(C(N)=O)C1)NC(=O)CCOC(C)=O C(=O)(N=c1ccn(C2CC2)[nH]1)C1N(C(CN2C(C)CCC2)=O)CC(=O)C1 N1(C(c2n[nH]c(CC)c2[N+](=O)[O-])=O)CCC2(COC(CNC(=O)CF)C2)C1.O c1(C(=O)OC)nsc(N2CC(CCNC(C3C4COCC34)=O)(OC)C2)n1 CC(C)(C)C(C(=O)N1CCC(CCNC(c2ccc(=N)[nH]c2)=O)C1)C1CCC1 C1(C(=O)OC)C2CCC1(C1CCCN(C(=O)CC(C)n3cccc3)C1)C2 N1(C(CC2C(C)CCCC2)=O)CCCC(NC(C2CCCN2N=O)=O)C1C N1(C(CCCC(=C)C)=O)CC(C(=O)NCC2CC23CCOCC3)CC(C)(C)C1 C1(C(=O)NCC2(OC)CCOC2)CN(C(C2CCSCC2)=O)CC1(F)F C1(NC(C2C(C(C)O)C2)=O)CCC(N2CCN(c3nnc(O)s3)CC2)CC1 C1(NC(Cc2ccn(CC)n2)=O)CN(C(c2nn(C(F)F)cc2Cl)=O)CC1(C)C C(=O)(C1=CCCCCC1)N1CCCC1(C)C.N1(C(C)=O)CC(O)CC1C(=O)N.C C1(C(C(=O)NC(C(=O)OCC)Cc2cccc(OC)c2)C)CCC(C)(O)CC1 C1(C(N2C3C(NC(CC(C)C4CC4)=O)C(C3)C2)=O)Cc2ccccc2C1 S(=O)(=O)(CC(=O)N(CC(C)NC(=O)CCNC(N)=O)C)NCC c1(CCNC(=O)C(N2CCOC(Cn3cncn3)C2)=O)ccncc1Br C1(CN(C(=O)CC(O)C2CCCC2)C)COCCN1C(=O)COC1CCOC1 C(=O)(C(C(C)C)NC(c1csc(C)c1C)=O)NC(c1cnn(C)c1)CC C=Cc1ccc(NC(C2(F)CN(Cc3ccc(C)[nH]3)C2)=O)cc1 N1(C(C(=O)OC)=O)CCc2nc(-c3ccnc(C(F)(F)F)c3F)sc2C1.C1C(=O)N1 CC(C)CS(=O)(=O)N1CCOCC1c1ccc(C(=O)N2CCCO2)n1C C(=O)(CC(C=C)CCC)NC(CC#C)C(=O)NCCN1CCC(C)C1 C12(C=O)CCCC1C2.C1(C=O)CC(C)C1.C(CCOC)OC.C(=O)CC.N N1(C(CCc2nnc(C(C)C)o2)=O)CC2CC2(CNC(C2CC(O)CN2)=O)C1 c1cc(Cl)ccc1[N+](=O)[O-].c1(OC)ccc(Cl)c(C(=O)NC2CC(NC)C2)c1F N1(C(C2CN(C(C(C)C)=O)CC2(C)C)=O)CCC(C2CCCC2)C1 c1(CN2CC3C(C(=O)NCCc4ccncn4)(C3)C2)cc(O)ccc1[N+](=O)[O-] c1(OC)ccc(C(=O)NCC2(CCNC(C3CCC3)=O)CC2)c(Br)c1 c1(C2(N(C(C(CC)O)=O)CCCNC(C3CCCC3)=O)CC2)ccc(C)nc1 C(C(C)C)(C(O)C(=O)N1CC(=O)NCC1C(=O)Nc1ccc(Cl)cc1O)OC c1(C(N2C(CC(=O)NCCc3ccnc(O)c3)COCC2)=O)cc(Cl)cnc1F C1(CC)(NC(c2nccc(C)n2)=O)CCN(C(c2cn(C)ccc2=O)=O)CC1 Cc1cc(C(=O)NC2CCC2NC(=O)C(O)CCc2ccccc2)c(C)cc1Cl N1(C(Cc2ccc(C(=O)OC)cc2)=O)CC(NC(c2ccc(F)s2)=O)CC(O)C1 NC1Cc2ccccc2N(C(c2ccc(-c3ccccn3)s2)=O)C1 CC(C)(C)CN(C(=O)CC1CCC(C)C1)C.C(C=O)OCCOCC.N C1(N(C)Cc2ccccc2)CCN(N2CCN(C)CC2C2CC2)C1 n1(CC(=O)NCC(C)N(C(C2C(=C)C2)=O)C)c(CS)nc2ccccc12 c1(C(=O)NC(C)CN(C)C(C2CNC(=O)C2)=O)cc2ccc(Br)cn2c1 Cc1cc(Cl)nc(Cl)c1NC(C1CC(F)CN1C(=O)CCc1ccc(O)cc1)=O c1(C(CNC(C(F)=CC)=O)NC(=O)C(c2ccccc2)S)ccccc1 c1(CN(C(C2(NC(=O)CCOC(C)=O)CC2C)=O)CC)ccccn1 CC1CCC(N(C)C(c2coc(CNC(=O)CCc3cnco3)c2)=O)C1 c1(C(=O)NC2C(O)CCN(C(c3cc(C)sc3)=O)C2)cn2c(n1)CCCC2C N1(c2cc(N(C)CC3CCCOC3)nc(C)n2)CCC2(CCN(C)C2=O)C1 N1(C(C2N(C(C)=O)CSC2)=O)CCCC(C(=O)NC(C)(C)C)C1 Cc1cc(CCC(=O)NCC2C(C)CCCN2C(c2sncc2C)=O)cc(C)n1 CCCCN=C(NCC1(C)CCCC(=O)N1)NC1CCN(C2CCCC2)C1 N1(C(c2cc(CCC)on2)=O)Cc2[nH]nc(C(N3CC4(CC(C)CO4)C3)=O)c2C1 CC1CC(C(=O)OCC2CC(c3ccccc3)C2C)OC1C(=O)O.C(C)(C)C O=C(C1=CC2C=CC(C1)C2)NC1(C)CC2CCC1CC2.c1(C=O)cnc(S)[nH]1.N C1(C(=O)NC2CCN(C(c3c(OCC)nccc3)=O)C2)CCC2CC2CC1 C#Cc1cc(C(N2CCC2C(=O)NCc2cnco2)=O)ccc1C C1(NC(c2ccc(CNC(C)=O)o2)=O)COCCN(C(=O)Cc2ccco2)C1 C1(C(N(C(C)CCNC(=O)C=Cc2ccco2)C)=O)CCCCCC1 CC(CN=c1nc2sccc2c(N2CCN(CC(C)O)CC2)[nH]1)c1ncc[nH]1 c1(OC)cc(C(F)(F)F)[nH]c(=NCC2(C)CCN(C(=O)C(C)CC(F)(F)F)C2)n1 c1(CCC(c2n(C(CC)C)nnn2)NCCCO)c(Cl)cccc1Cl C(=O)(C1=C2CCN=C2NC=C1)N1C(CNC(=O)C2=CCOCC2)COCC1 c1(CCC(N2C(C(C)NC(CCCC=C)=O)CCC2)=O)cccc(F)c1F C1(CC=O)CC2(CCCC2)CO1.C1(CC=C)CCN(C(c2c(C)cnn2C)=O)C1.N C1(CNC(C(CC)SC)=O)CCN(C(c2scnc2C(C)C)=O)CC1C1CC1 C(=O)(C1=CC2CC(C1)CC2O)N1CCCC(N(C(=O)C2=CCSC2)C)C1 C(CCCC(=O)N1CCCC(NC(C2CCCCC(=O)N2)=O)CC1)(OC)OC Cc1c(C(=O)NC2CCN(C(=O)CCF)C2c2ccccc2)cnn1CC(F)F C(C1CCOC1)=CC(=O)N(C(C)C1CC1)C.C(C=O)N(C)C(=O)C1CC1 CCCC(CNC(=O)C=CC1CCC1)C(=O)NC(C)(CO)C1CC1 N1(C(CNC(CCC)=O)=O)CCN(C(=O)C#CC(C)(C)C)C(C)C1C c1(C(=O)NCCC2(NC(C3CCN(CC)C3)=O)CCCC2)oc(C)nc1C C1(NC(CN(CC)CC)=O)CCN(C(=O)C(c2cccc(Cl)c2)(C)C)CC1C c1(C(=O)NC2CN(C(C3(C(=O)O)CCCC3)=O)C2)cccc(-n2cncn2)c1 C=C(Cl)CC(C(=O)NC1CC2C(C1)C2(F)F)NC(=O)Cc1c[nH]nc1C C1(NC(CC(=O)NCC)=O)CC(C)CN(C(=O)C(c2ccc(F)cn2)(F)F)C1 c1(C(=O)NC2CC(NC(CCC(=C)Br)=O)C2)cccc2nc(O)[nH]c12 N(C1CCc2ccccc21)C(c1cc(-c2c(C)ccc(OC)c2)c(C)cc1F)=O C12(C(N3C(COC)CC3)=O)CCCC1CCN2C(c1coc(C)c1)=O C1(C(NCCNC(c2cnc(-c3cnccn3)s2)=O)=O)CCOC(=O)N1.CC c1(C(=O)NC2CN(C(CCC3C(C)=NNC3=O)=O)C2)c(F)cccc1F C(CC(C(=O)NCC(COC)C(C)C)NC(c1cnsn1)=O)=CC C(=O)(C1=CCOCC1)NCC1(CC(=O)NC(COC)(C)C2CC2)CC1 N1(C(C2(CC)CC2)=O)CCC2(CC1)CC(NC(=O)C=Cc1ncccc1C)CO2 c1(OC)cc(C)c(C(=O)NC2CN(C(C3CC4CC4C3)=O)CC2O)cn1 c1(C(=O)OC)cccc(C2CN(Cc3cccc(-c4cnn(C)c4)c3)C2)c1 c1(C(=O)NCC(CNC(c2ccc(OC)cc2OC)=O)O)scc2c1OCCO2 N1(C(C(C)N(C)C)=O)CCCC2CN(C(=O)C=Cc3nc[nH]n3)CC12 c1(N2CCCC(C=C)C2)nc(=NCc2nn(C)cc2OC)[nH]c2cccnc12 Cc1ccc(C#N)cc1NC(c1cc(CCNC(c2c[nH][nH]c2=N)=O)on1)=O C1C2CCC1CN(C(=O)CS(N)(=O)=O)C2.C1(CCOC)(C(=O)N)CCCC1.C N1(C(C2(CC)CC2)=O)C2CCC1C(F)CC2.C1(C)(CC=O)CC(F)(F)C1.N C1(NC(c2c(C(C)C)ccc(C)c2)=O)CC2CCC1CC2NC(=O)C.C1CC1 C(=O)(C1=CCS(=O)(=O)C1)N1CC2(CN(C(C(c3cccc(O)c3)(C)C)=O)C2)C1 N1(C(CCN(CCOC)C)=O)CCC(OCC)C1.C(c1nccs1)=CC=O.N Cc1cc(C(N2CCCCCC2CNC(=O)C(F)C2CC2)=O)c(N)c(Cl)c1 c1(C(=O)NC2C(NC(CC3C(C)=NOC3=O)=O)CC2)ccc2nccnc2n1 N#Cc1ccc(OC2CCN(C3CCN(c4ccccc4F)C3=O)CC2)cc1 C1(OC)CN(C(=O)Cc2nc(-c3ccccc3C(=O)O)cs2)C(C)(C)C1 N1(C(c2c(C)c[nH]c2)=O)CCc2[nH]nc(-c3cnn(-c4ccccn4)c3)c2C1 Cc1cc(CC(=O)NC(C2CC=CCC2)C(=O)NCCSc2nnnn2C)n[nH]1 c1(OCC)ccc(Cl)c(C(=O)N(C)CCN(C(=O)CC)C)n1.CC(N)=O.S c1(C(=O)NCCN(C(CCCC=C)=O)C2CC2)nc(C(C)CC)ncc1Br Cc1cccc(C(C)NC(=O)C(Cc2ccoc2)NC(=O)CNC=O)c1 Cc1ccc(CC(=O)N(CCCCN(C)C(c2cc3n(n2)CCO3)=O)C)cc1Cl C(=O)(C(CNC(c1cncnc1C)=O)CC(C)C)NCC(CC)(C)CC N1(C(C=CC=CC)=O)CCCC(CCCCNC(=O)C(=O)NC2CC2)C1 C(=O)(C1=CCN(C(=O)CCCN2CCCC2)C1)NCc1c(C)n(C)nn1 n1(C(C)C)ncc2c(N(C)CC3CC3(F)F)[nH]c(=NCc3cccc(Cl)n3)nc12 C1(NC(c2ccc(OC)cc2)=O)CC(C)CN(C(c2ccc(C(C)=O)cn2)=O)C1 c1(C(=O)N)cc(F)cc(F)c1.C(C)(C)(C(=O)N1CC(O)(CC)C1)OC(C)C Cc1ccc(Cl)c(C(=O)NCCN(CC(C)O)C(C2CC2[N+](=O)[O-])=O)c1 C(=O)(C(CC)CCOC)N1CCC(N(C(COCCC=C)=O)C)C1 C1(OC)CCCC(c2nc(CCCCCCC3(c4ccc(=N)[nH]c4)CC3)no2)C1 CC1ON=C(C(=O)NC2CN(C(c3ccccc3SCC(F)(F)F)=O)C2)C1C Cc1ccc(C(N2CCN(C3CCCC3NC(=O)C(=O)NC(C)C)CC2)=O)cc1 C(N=c1[nH]cncc1Cl)C1CC(NC(C2(N(C)C)CCCC2)=O)C1 c1(CCC(=O)N(CCC(C)NC(=O)CCN2CCC(F)C2)C)csc(=N)[nH]1 C(=O)(CC(CC)c1ccccc1)N1C(CN(C(c2c(CC)onc2)=O)C)CCC1 c1(NC(c2ccccc2N)COC)ncnc(NCc2cccc(Cl)c2F)c1C N1(C(c2cnc(C)s2)=O)CC(C)(C)CC1CNC(C1CCC(O)CC1)=O c1(C(C)=O)ccc(OC(F)C(=O)N2CC(CC(C)NC(=O)C(C)C)C2)cc1 C1(C=O)CC2(CCCCC2)C1.C1(NC(C2(C)CCN(C)C2)=O)CC2(C1)CCC2.N C1(CC)CN(C)CCN1C(C1(C)CC(C=O)C1)=O.C1(C=O)CC1NCC C#CCC(C=O)NC(=O)CC=CCNC(=O)C(CSC)OC.O(C)CC C(=O)(CC1=CCCC1)NC1CC(NC(c2cccc(-c3nc(C)sc3)c2)=O)C1 CC1(C)CCC1CC(=O)NCC1CCCN1C(c1ncnn1C1CCOCC1)=O c1(C(C)C)ccc(CCC(=O)NC2CCC2CNC(C2CCCN2N=O)=O)cc1 N1(C(CCCC)=O)CCC(C)C(NC(C2CCCN2CCC)=O)C1C c1(C(C)C)n[nH]cc1C(=O)NC(c1nocc1C(=O)NCCCS(C)=O)C CC(C)(CCC#N)C(=O)NC1CCCC1NC(C1(C)CC(C2CC2)=NO1)=O C1(NC(=O)CCCCNC(C2CS(=O)(=O)C2)=O)CC2CCC(C1)O2 FC(F)(F)C(CC)C(F)(F)F.c1(Cc2nnnn2C2CC2)cc(Cl)c(F)c(Cl)c1 CCC(C)C(C(=O)N1CCC(C)C1)NC(=O)OC.N1(CC=O)CCN(C)CC1.N C(=O)(CC(C)C(F)F)N(C(CC)C(=O)NCCc1csc(C)n1)C n1(CCCC)cc(C(=O)NCC2CCN2C(c2cc(CC)on2)=O)nn1 C(C)(CCC(=O)NCC(C(=O)N(CCC(O)CO)C)N(C)C)SC C=CC1CCCC(c2nnnn2CCCF)(NCCC(F)(F)Cl)C1 C1(O)(CCNC(C(C)OCCCC)=O)CCN(C(=O)C(C)(C)CF)C1 N1(C(C2(CC)CCCC2)=O)CCOC2(CCN(C(c3nccc(C)c3F)=O)C2)C1 C1(CCNC(c2n[nH]cc2F)=O)CN(C(=O)C(O)Cn2cncn2)CCS1(=O)=O Cc1oc(S(=O)(=O)N(C)C)cc1C(N1CCC1C)=O.C(=O)CC.C1CCC1 c1(CN2CC(NC(c3c(C)cc(C)c(Br)c3)=O)C(F)C2)c[nH]c2ncc(Cl)cc12 Cc1ccc(F)c(C(=O)N(C2CN(C(C3CN(C)CC(C)O3)=O)C2)C)n1 c1(NC(C2CCN2C(c2ccncc2Br)=O)=O)cccc(OC(F)(F)F)c1 N1(C(C2CCCN(C(c3cc(C)c(O)nc3)=O)CC2)=O)CCCC2(C=CCO2)C1 c1(CC(N2CC(O)C2)=O)c(Cl)cccc1Cl.C(C(F)C(=O)NC)N(CC)CC N1(C(C2(COC)CN(C(c3cnccc3C#N)=O)C2)=O)CC2(CCOCC2)C1 CC1CC(NC(=O)CC2(N(C)C(C3(C)CCC(=O)CC3)=O)CC2)CCN1C C(=O)(CC(C)CC(C)C)N1C(C(N2CCC(C)(CC)C2)=O)CCC12CC2 C1(C)(C(=O)NCC(C2N(C(CC)=O)CCC2)(C)C)CCC(F)(F)C1 N1(C(c2cnc(C)s2)=O)CC2OCC(NC(C3(C4CCCO4)CCC3)=O)C2C1 C1(C(=O)NCc2n(CC)nnn2)CN(C(C2(F)CCCCC2)=O)CC1(C)C C(C(CCO)NC(C1CCC(CNC(c2cnnn2C)=O)C1)=O)N(C)C N1(C(C(=O)NCC(F)F)=O)CCCC2C1CCCCN2C(=O)C1=COCC1 Cc1ccc(C(=O)N(C)C)cc1NC(=O)C(N1CC(F)CC1c1ccccc1)=O N1(C(CC2N(C(C(CCC)OC)=O)CCC2(C)C)=O)Cc2c[nH]nc2C(C)C1 N1(C(c2ccc(CC)[nH]2)=O)CC2CCC(NC(C3(CO)C=CCC3)=O)CC2C1 N1(C(C(N2CCOC2=O)C)=O)CCN(C(C2CC=CCO2)=O)C(C(C)(C)C)C1 C1(OC)(CNC(=O)C(O)C(C)C)CCN(C(c2cc(C)sc2C)=O)C1 CCN=c1[nH]cnc2cc(C(=O)N(C(C)CNC(c3cnccn3)=O)C)ccc12 c1(C(C)=O)cnc2sc(C(N3CCC(C)(NC(=O)C)C3)=O)c(C)c2c1.C(C)C C(=O)(C1CCS(=O)(=O)c2ccccc21)N(CC(C)NC(=O)CC(F)(F)C(F)F)C c1(CNC(CN(C(C)C)C(c2ccoc2Cl)=O)=O)cccc(CSC)c1 CCCC(CNC(C1(F)CCCCCC1)=O)C(=O)NC1CCC(=O)NC1=O CC1CCCC(n2nc(COC(C)(C)C)nc2-c2ccccc2)C1.C1(C=O)CC1 C1(C(=O)NCC2C(CNC(CCCc3nc(C)sc3)=O)C2)Cc2ccccc2C1 C1(NC(C(CO)NC(c2cnc(CC)nc2)=O)=O)CCCCC1(F)F c1(CC)cccc(C(=O)NC(C)Cn2cc(C3(CCO)CC3)nn2)c1 C=CC1(C(=O)NCCC(C)(C)CC=C)CCN(C(c2cccn(C)c2=O)=O)CC1 N1(C(C(CC)C)=O)CCCCCCC1C(=O)NCCC(O)CO C1(CN(C=O)Cc2csc(C3CC3)n2)C(F)(F)C12CCOCC2 C#Cc1ccc(C(N2CCC3(CC2)CC3NC(=O)C(CO)C(C)(C)C)=O)cc1Cl C1(C(N2CCC(C(C)(C)C)C2)=O)CCCN1NC(=O)COC1CCCC1 C1(NC(=O)C(N2CCOCC2CC2CCOCC2)=O)CCc2ncc(Br)n2C1 C1(C(=O)NC(COC)C(C)C)C2CCN(C(=O)Cc3cc(C)on3)CC12 C(=O)(N=c1cc[nH]c(C)c1C)C1CN(C(c2c(C)cc(Br)cc2)=O)CC(F)(F)C1 N1(C(CC(C=C)(C)O)=O)CCC(C)(C)CC1C(N1CC2(CSC2)C1)=O C(=O)(CC(F)(F)Cl)N(C)CCN(C(=O)CCN(C(=O)C=CCl)C1CC1)C CC(C)(CN=c1ccnc(Nc2cnn3c2C(=O)NCC3)[nH]1)OCCO CC(C)(C(=O)NCC1CC1)c1csc(-c2cccs2)n1.C1(C(=O)N)CCC1 C(=O)(C(F)(F)C(F)(F)F)N1CC(Nc2nccc(OCC)n2)C(F)CC1 NS(=O)(=O)CCC(=O)N1CCC(NC(c2c(Cl)nsc2Cl)=O)C(F)C1 c1(C(=O)NC2(C)CC(NC(=O)C#CC3CC3)C2)cc2n(n1)CCNS2(=O)=O c1(C(=O)NCC(CCNC(C(COCC)C)=O)O)c(F)ccc(Br)c1OC C=CCCCCC(=O)N1CCCCC(N(C(=O)CCCc2cncs2)C)C1 C1(OC)C=CCN(CC(=O)NCc2nc(-c3ccc(C)cc3)cs2)C1 C1(NC(CN(C(c2ccn(COC)n2)=O)C2CC2)=O)CCn2nccc2C1 Cc1ccccc1C=CC(=O)NCC1CC2CN(C(c3[nH]nnc3C)=O)CC12 Cn1ccc(C=CC(N2CC(NC(C3CC3C(C)(F)F)=O)C(O)C2)=O)c1 CN1C(=O)CCCC1=O.C1(C=O)C2CC(O)C(C2)N1C(C12C=CC(CC1)C2)=O Nc1ccc(C(N2CC(F)CC2CNC(=O)CCn2cncn2)=O)nc1 C1(CN(C(CCC=C)=O)C)CN(C(=O)C(C)Cc2ccco2)CC12CC2 C12(C(=O)NCCCN(c3cc(O)nc(O)n3)C)CCCCN1CCC2 N12CCCC(O)(C1)C2.c1(NCCCC=O)ccc(F)cc1.C(C[SH](=O)=O)OC.C c1(CN2C(C(=O)Nc3ccc(OC)nc3C)CC(F)C2)cn(C)c2ccccc12 N1(C(CC(=O)N(CC#C)CC=C)=O)CCC(C=C)C1.C(C1CCC1)=CC=O C(=O)(C1=C(Cl)CCC1)NCC(C)(CC)NC(c1c(CC)cc[nH]1)=O C(=O)(CC(C(F)F)NC(=O)CC=C(Cl)Cl)N1CC(C)C1(C)C c1(CCC(=O)NC(C2(CNC(C)=O)CC2)C)ccc(=N)[nH]c1 Cc1cc(N2CCC(NC(c3ccnnc3Cl)=O)CC2)n2nc(C)cc2n1 N1(c2c(C)cnc(C)n2)C2CCCC1CN(C(C1CN3CCN1CC3)=O)C2 C1(C)(CNC(C(C)(C)C)=O)CCCN(C(C2CC2c2cccc(C#N)c2)=O)C1 C=CCC(CC=C)C(=O)NCC1CC(CNC(=O)CC(C)(C)F)CO1 Cc1ccc(C(=O)NC2CCC2NC(=O)COC(C)(C)C)nc1O N1(C(CC2N(C)CCOC2)=O)Cc2ccccc2C(NC(=O)C=CC=C(Cl)Cl)C1 N1(C(C2(C(=O)OC)CC2)=O)CCC(F)(C(=O)NCc2c[nH]nc2C)C1 N1(Cc2nnc(C)n2C)CC(NC(C2CCN(C)CC2)=O)C(C)(C)C1 C#Cc1cnc(NC(C23CC2CN(Cc2cc(Cl)cc(Cl)c2)C3)=O)cn1 CC(CC(=O)NC(C)(C)CCCNC(C1OCC2COCCC12)=O)C(C)(C)C N#Cc1ccccc1-c1cn(C2CCN(C(=O)CCc3cccnc3Cl)C2)nn1 Cn1cnc(N2CCCCC(NC(=O)C=C3CCSCC3)C2)c(Br)c1=O CN1CC2CN(C(=O)C(C3CCN(C(=O)CC4(C)OCCO4)C3)F)CC2C1 c1(OCC(=O)NC2CC23CCC3)c(F)c(F)cc(F)c1F.C1(C=O)C=CCC1 C(=O)(C1=C(Cl)CCC(C)C1)NC1CCN(C(C=Cc2ncc(C)[nH]2)=O)CC1F C(=O)(CCN(OC)C(=O)COC1CC1)NCC(C)(OC)OC c1(OC)c(NC(c2[nH]ccc2CNC(=O)C(O)CSC)=O)cccc1Cl c1(NC(C)=O)cccc(C(=O)NCC2CCC2)n1.C1(C(=O)N)CCCOC1C c1(C(C(N2C(C(C)(C)NC(CCC)=O)CCC2)=O)F)ccc(C)cc1 C=C(C)CC(C(=O)NCC(c1ccccn1)O)NC(=O)Cc1cccs1 Cc1cccc2c1CC(C(=O)NC(c1ccccc1)c1cnn(C)c1)N2 C(=O)(C1=CC(O)CCC1)N(C1CCN(C(c2ccc(-c3ncc[nH]3)cc2)=O)C1)C CN1C(=O)CSC1=CC(=O)N1CC(NC(c2csc(C3CC3)n2)=O)C(F)C1 Cc1nonc1CC(=O)NCC1COC(CNC(=O)Cc2cc(Cl)cs2)C1 N1(C(c2c(C)nccn2)=O)CCN(C(c2cc(F)ccc2Cl)=O)CC(O)C1 C1(NC(C2C(C)CC(C)O2)=O)CC(N=c2[nH]cnc3cnn(C)c23)C1 c1(C(N(c2c(CC)cccc2C)C2CCNCC23CC3)=O)cc(C)c(F)cc1N CC1(C(=O)NCCc2n[nH]cc2C(=O)NC23CCCC2C3)CC(F)C1 CCC(C(=O)N(C(CNC(=O)CSCC(C)C)C1CC1)C)c1cccnc1 N1(C(C2N(S(C)(=O)=O)CCC2)=O)CCC2(CCCN(c3cnc(F)cn3)C2)C1 C12(C(=O)NC(C(C)NC(c3cn(CCC)nn3)=O)C)CC1Cc1c[nH]nc12 C1(CC(=O)N(CCC#C)CCO)CCCN(C(=O)CC(CC)OC)C1 CCC(F)(F)C(=O)N1CCN(CCNC(c2ccnnc2O)=O)CC1 C(=O)(C1=CNC2=NCCC2=C1)NC1C2CCN(C(c3c(C)nc4sccn43)=O)C21 C1(NC(c2cn(C)nc2C(F)(F)F)=O)CN(C(=O)Cc2ccsc2)CCC1C CCC(CC)C(C)C(=O)N1CCCCC1CCN(C)C(C1(n2cncn2)CC1)=O N1(C(c2cc(CC)oc2C)=O)CCC(NC(=O)C(CC(C)C)OC)CC1C c1(C(N2CCC(N3CCCC3)C2)C(=O)NC(CC)C)ccc(Cl)c(F)c1 Nc1ccc(F)cc1C(N1CCC(F)C(NC(=O)Cn2ccc(C3CC3)n2)C1)=O N1(C(C=CC)=O)C2CCC1CC(N(C(=O)CC(C)Cc1cccc(OC)c1)C)C2 CC(C)C(C)(C)C(=O)N1CCC1CC(N1CC(OCC(=O)N(C)C)C1)=O c1(CC(=O)N)ccccn1.C(C)(C(=O)NCCC)OCCOCCOC c1(OC)ccc(NC(C2(C(C)C)CCN(C(c3cnnn3C)=O)C2)=O)c(C)c1 N1(C(c2ccc(OCCCC)cc2)=O)CCC(NC(=O)CCC2CC2)CC1C N#Cc1ncc(NC(c2nc(-c3ccc(OC4CCCCO4)cc3)cs2)=O)cn1 CC1(C)CCN(C(=O)C(c2cccc(F)c2)(C)O)CC1NC(=O)CN=S(C)(C)=O c1(CC)ccc(C(=O)N)cc1[N+](=O)[O-].C1(O)CN(C(C2(C#N)CC2C)=O)C1.C N1(C(c2ccccc2)C)CC2CC(NC(=O)Nc3nc(C#N)c(Cl)s3)CC1C2 CCCC(C)CC(=O)NCC1CCCN(C(=O)C(F)Cc2ccccc2)C1 c1(N2CC(C(CC)CC)OCC2)nc(N(CC(=O)NC)C)cc(C)n1 Cc1cnc(NCc2ccc(N)cn2)c(S(=O)(=O)NC(c2ccsc2)C)c1 C(C(CC(C)C)N)NC(C)=O.C(=O)(C(C)(C)c1ccno1)N1CC(CC=O)C1 c1(C(N2C3CN(C(=O)OC)C(C3)C2)=O)cc(F)c(F)cc1Nc1ccncc1 C#CC1(C(=O)NC(C=C)C2CCC2)CN(C(C2CCCC(C)O2)=O)C1 C#CC1(C(N2CCN(C)C(C(C)C)C2)=O)CCN(C(=O)C(C(C)C)C2CCC2)C1 N1(C(CC(CC)C)=O)CCC(C(=O)N(C(C)CN(C)C(C)=O)C)CC1(C)C Cc1ccc(C#N)cc1S(=O)(=O)NC12CC(NC)(C1)C2.c1cc(Br)ccc1C#N C1(CC(N2CCC(NC(c3ncn(C)c3)=O)C2)=O)Cc2cccc(Cl)c2O1 C1(CC)CCOCCN1C(C1(NC(c2cccs2)=O)CCCCC1)=O N1(C(c2cc(CC)sn2)=O)CCC2(CC(C(=O)N)C2)C1.C1CCN(C(C)=O)C1 C1(NC(c2c(C)nc(CCC)o2)=O)CC2CCC1N(C(c1cc(C)c[nH]1)=O)C2 C1(C(=O)NCCCCCCNC(C(c2n(C)cnc2)O)=O)COCCC1(F)F CC1CC(C)OC1C(=O)NC1CCCC1CNC(c1ccccc1)=O.CC#N Cc1cc(=NC(=O)C2CC3(CC(NC(c4c(F)cccc4F)=O)C3)C2)[nH]n1C C#Cc1ccc(NC(=O)C(CC)N(C)C(C2CCN(C)C2=O)=O)c(C)c1 c1(C(N2C3CC(NC(C(C)CO)=O)C3CC2)=O)ccc2c(ccn2C)c1 N1(C(c2c(CC)nc[nH]2)=O)CCN(C(c2coc(Br)c2)=O)CC1c1cn[nH]c1 Cc1cnc(C)c(NC(C2CC2NC(c2nc(Cl)ccc2F)=O)=O)c1 Cc1cc(C(N2CC(F)(C(=O)NC(C(C)C)C3CCC3)C2)=O)ccc1O CCC(C)(CCC(C)C)C(=O)N1CC(C(=O)NCCCn2ccnc2)CC(F)C1 c1(CC(=O)NCC(C)(C(C)C)NC(Cc2scc(C)c2)=O)c[nH]c2ncccc12 C(=O)(CC(C)(C)C(F)(F)F)N1CCC(NC(C2N(CCC)CCCC2)=O)C1(C)C c1(SCCC(N2CCC(C(N(C)C)=O)C2)=O)nc2ccccc2s1 Cc1cc(C(=O)NC(C)CCCNC(=O)C(C)N)cc(C)c1F.[SH](C)(=O)=O N1(C(Cc2c(C)noc2C)=O)CC(C)(C)CC1C.c1(CC(=O)N)nnc(O)s1 C(=O)(CCC(C)(F)F)NC(CC)CN(C)C(C1CCN(C)CC1)=O CCC(C)C(CC(=O)N(CC(C)OC)CC)NC(c1nc(C)c(C)s1)=O C1(C(=O)NCC)CN(C(c2ccc(C)o2)=O)CCN1 CC(C)CCCCCC(=O)N1CCC2(CC2C(=O)NCCCC(O)CO)C1 N1(c2n(CCOC)c(-c3ccco3)nn2)CC(OC)CC1(C)COC C(=O)(C1=CC2(CN(C(C3(C)CC3C)=O)C2)OC1)NC1C(C)NC(=O)CC1 C1(CNC(c2cccc(CC=C)c2)=O)CC(C(=O)N)=NO1.C1CCCC12CC2 c1(-n2c(-c3[nH]ccc3C)nc(CCOC)n2)ccc2c(C)cc(C)c(O)c2n1 C1(C(N2CCCC(c3cc(CC)c(F)cc3)C2)=O)CC(C(C)(C)C)=NO1 C1CN(C(C2(C)CC(C)=NO2)=O)CCC12CCC2.C(C)(C(=O)N)OCCOC N1(C(C2COCC(C)O2)=O)CC2(C)CC1(C(=O)NCc1cncn1C)C2 c1(CC)cnc(CNC(C2CCCC2NC(=O)C=Cc2ccsc2)=O)s1 N1(C(CCCCC=CCCC)=O)CC2COCC(CNC(=O)NC)(C1)C2(F)F c1(NC(c2cc(F)ncc2NCc2ccc(Cl)o2)=O)cccc2c1OCO2 C1(C(=O)NC2CCCC2NC(=O)CCc2ccccc2)(OCC)CCCSC1 N1(Cc2cc(Br)c(O)c(Br)c2)CC2(CCC(N=c3nc[nH]n4cc(Br)cc34)C2)C1 c1(N(CCC(=O)N2CCCC2)C(C)C)nc(Cl)ccc1CS(N)(=O)=O N1(C(CC2C(C)(C)CCO2)=O)C2CCCC1CN(C(=O)CC1CCOC1)C2 c1(OC)cc(CN(C(=O)CC2COC(C)(C)CO2)C)c2ccccc2n1 c1ncc(S(C)(=O)=O)cc1Cl.C1(NC(c2c(CC)cno2)=O)CC2(C1)CC2.N C(CC(C(=O)NCCNC(=O)COC(C)(C)C)NC(N)=O)SC C1(CC(=O)NCCC2CN(C(c3ccc(Cl)cn3)=O)CCO2)CN2CCN1CC2 C1(NC(CCS(N)(=O)=O)=O)C2CCN(C(=O)CSc3ccccn3)CCC12 CCCC(O)CC(=O)NC(C1(O)CN(C(c2cn(C)[nH]c2=N)=O)C1)C c1(C(=O)NC(C)CCNC(=O)C(C)c2cccs2)ccc2cnnc(O)c2c1 N1(c2c(C)cccc2)CCCC(NC(=O)NCc2cn(C3CC3)cn2)C1=O S(=O)(=O)(c1c(Cl)cc(Br)cc1Cl)N1CCOCC(C(=O)NC(CC)C(=O)NO)C1 CC1CCN(CC(=O)NC2(C)CC(NC(c3scnc3C3CCCC3)=O)C2)CC1 CCCC(C(=O)OC)C(=O)N1CCC2(CC1)CC2C(=O)NOCC1(C)CC1 N1(C(C(C)(C)OCC)=O)CCC2(C1)CN(C(C1NC(=O)CC1C)=O)CCO2 O=C(C1c2ccccc2CN1Cc1cccc(Br)n1)Nc1cc(F)ccn1 c1(C(=O)NCCN(C(=O)CC2CCCCC2)CCC)cc(C)c(C)c(C)c1 c1(C(=O)NCC2CCCN2C(=O)CS)cc2n(c1)CCSC2.c1cccnc1 Cc1ccc(C(=O)N(C)CC2CCCN(C(=O)COC3CCCOC3)C2)nc1O C1(C(N2CCC(CO)C2)=O)(CC)CCCN1C(=O)CCCC1CCCC1 C(=O)(C#CC(C)(C)C)NC1CC(CC(=O)NCCC(C)C)C1 CCCC(O)C(=O)N(CC(C)N(C(=O)CNc1ccccn1)C)C C1(CNC(C(Cn2ccc(C)n2)C)=O)CC2(C1)CN(C(=O)CC1CCCC1)C2 C1(CC)CN(C)C(=O)CN1C(=O)CC=CCNC(c1cc[nH]c1C)=O c1(C(C)N(CCNC(=O)CCC(N)=O)C2CC2)cccc([N+](=O)[O-])c1 N1(C(C2(c3ccccc3)CCOC2)=O)CCOCC(C2CCC2)C1 c1(C=O)ccc(S(N)(=O)=O)s1.N1(C(C2(CC)COC2)=O)CCCC(CO)C1.N C(=O)(C(C)(Cn1ccc(C)n1)N(CC(=O)OC(C)(C)C)CC(C)C)OC C1(C(N2CCC2)=O)CC2(CCC2)CN1C(C1CC12CCCC2)=O.C(=O)(NC)N CC1(N=c2[nH]c(Cl)nc3c2COCC3)CC(NC(=O)C(C)(C)CC(F)F)C1 c1(N(C)C)ccc(-c2nc(-c3cc(F)n[nH]3)n(Cc3cccnc3)n2)cc1 C12(C(=O)NCC(C)(CO)NC(CCCCC)=O)CCC(CC1)C(C)O2 C1(C(=O)NC2(CNC(c3ccnc(O)c3)=O)CCCCC2)COC2COCC2O1 C(CC(F)(F)C(F)(F)F)NC(c1nc(C)c(C)[nH]1)c1nnnn1C1CCOC1 C(=O)(C1=C(Cl)CCCC1)N1C(C)CN(C(=O)C(O)C2CC2)CC1 n1(CCC(CC)O)cnc2c(N3CCN(CC4CCOC4)CC3)ncnc12 C=CC1(c2cn(CCC(=O)OC)nn2)COCCN1C(c1c(Cl)c(C)nn1C)=O N1(C(c2c(C)ocn2)=O)CC2C3CCC(C(NC(=O)C(O)CCC(C)C)C3)C2C1 c1(CC(N2CC3C(C3)C2)=O)ccc2c(c1)OC(F)(F)O2.CCCC=CC(=O)N CC(C)(CC(=O)NCC1CC2CC2N1C(=O)C=Cc1ccccc1F)C(F)F C1(C(CC)NC(=O)Nc2cnoc2C2CCOCC2)CCOCC1 c1(C(=O)NCCC2(NC(=O)C=CC3CCC3)CCC2)cc2cc(Cl)cnc2o1 N1(C(CCC(=C)Cl)=O)CCC(NC(=O)C(C)CCCc2ccccc2)C1(C)C C(=O)(CCCCc1ccc(F)cc1)N(CC(C)N(C(C(C)O)=O)C)C.C1CC1.C C1(NC(=O)Cc2ccc(F)c(F)c2)C2CCc3ccccc3C12 N1(C(=O)C(F)=CC2CC2)CC2(C(=O)NC34CC5CC(CC3C5)C4)CC1CCO2 C1(CCCC)CN(C(=O)C(C)OC)CCN1C(=O)CC1CC2CCC1O2 N1(C(Cc2c(C)n[nH]c2)=O)CC2CC2C1CNC(=O)CCc1ccccc1 C1(NC(C2(SC)CC2)=O)CC2CCC(C1)N2C(=O)C(C)Cc1ccnn1C CCN=C(NCC1(OC)CCCOC1)NC(c1cn(C)nn1)COCC c1(C(C)(C)C)ccc(CCC(=O)NC(CNC(=O)C(F)n2cccn2)CO)cc1 C(=O)(C(CNC(=O)CCc1cnc(C)o1)OC)N(CCOC)CCO C1(O)(C(=O)NCC2C(CC)(CC)C2)CCN(C(c2c(Br)cnn2C)=O)CC1 c1(COC)ccc(C(=O)NCCC(C)NC(=O)C(C)n2cncn2)cc1F C12(NC(CC3(CS(C)(=O)=O)CC3)=O)CCCC1N(C(=O)C(Cl)=CCl)CC2 c1(CC(=O)N(CC(C)(C)C)CC)cccc(F)c1.C(=O)(CC)N.CC(F)F N1(C(C2(COC)C=CCC2)=O)CCC2(CC1)CC(NC(c1ncc[nH]1)=O)C2 CCC(C(=O)N(C)CC1CCN(C(=O)Cn2ccnc2C(C)C)CC1)C(C)O C#Cc1ccc(C(N2CCCCCC2C(=O)NCC(CC)C(C)(F)F)=O)cc1 c1(COc2c(C(=O)NCC=C)ccnn2)nc2ccccc2o1 Cc1ccn(C(C)CC(=O)NCCC2CC(NC(=O)C(c3cnccn3)C)C2)n1 N1(CC)CCCC(C(=O)NCC(CCOC)NC(=O)C(C)(O)COC)C1 Cc1ccc(C=CC(=O)NCC2OCCC2C=O)o1.C1(CC)CCCC2CC12 C1(NC(C(C)Sc2nnnn2C2CC2)=O)COCCN(C(C2(C#N)CCC2)=O)C1 c1(C(=O)NCCC(CC)(C)NC(=O)CCC(C)(C)OC)cc[nH]c2nccc1-2 C(=O)(CCCC1CC1)NCc1c(C(C)C)n[nH]c1.C1(CC=O)COCC(C)O1 CC(CCC#N)NCc1nc(-c2ccccn2)no1 c1(C(=O)NC2CCCN(C(c3c(OCC)n[nH]c3)=O)C2)cc(=O)n(C)cn1 C1(NC(C2(CCOC)CCC2)=O)CCCN(C(c2sc(C(C)C)nc2C)=O)C1 C=CCC(C(=O)N(CCC(=O)NCCOCC1CCC1)CCCO)OC n1(CC#C)c(C)cc(C(N2CC3(CCC3)C2)=O)c1C.C(=O)(CCS(N)(=O)=O)N C1(NC(C(C)NC(N)=O)=O)C=CCN(C(=O)C(O)C(C)c2ccccc2F)C1 C(c1nc2ccccc2o1)=CC(=O)NC1(C2CCN(C(CS(CC)=O)=O)C2)CC1 C1(C)(N(C(C(c2cc(C)sc2)(F)F)=O)C)CC2CC2C1 C1(C(N2CC=CC2)=O)CC2(C1)C(F)(F)C21CCC1.Cn1cc(C(=O)N)cn1.C CC(C)CC(O)C(C)C(=O)N1CC(F)(C)C1.c1(CC=O)ccccc1.C(C)C.N Cc1cccc(O)c1C(=O)NC1CC(CNC(C2CCCC2(C)C)=O)C1 N1(C(CC(C)(F)F)=O)CCC(NC(c2cccc(C(=O)N(C)C)c2)=O)C12CCC2 C(=O)(C(CC1CC1)CC1CC1)NCC(C)NC(C(CC)C1CCOCC1)=O N1(C(C2(F)CCN(C(=O)CC3CCCO3)CC2)=O)CC2(CCC2)CC1CO C1(CNC(C2ON=C(C)C2)=O)C2CC2CN1C(=O)CCc1ncc[nH]1 C(CCC(=O)NCC1CCC1)NC(=O)NCC#C.C1(CC=O)CCC1 c1(C(N2CC3(CC(NC(C4(CC)CC4)=O)C3)C2)=O)csc2c(Br)cccc12 CN1CCN(C(=O)CC2CCCC(=O)N2)CC1C(N1CCOCC1)=O C1(CC)CN(C(=O)CC(CC2CC2)NC(=O)CN2C(=O)CNC2=O)CC1F C(N=c1[nH]c(=NCc2nc(C(F)F)n[nH]2)[nH]c2c1CC(C)CC2)c1c(C)nn[nH]1 C1(NC(c2c(C(C)C)onc2)=O)CCCN(C(C2CC2C(C)(C)C)=O)C1 N1(C(=O)C(O)C2CCCC2)CCN(C(C2(CCO)CC2)=O)CC1C1CCCC1 CC1(NC(c2sccc2C#N)=O)CCCCC1C(=O)NC1CC(n2ccnn2)C1 CN1C(=O)CSC1=CC(=O)NCC1CCCCN1C(=O)Cc1ccoc1 N1(C(c2cc(C)[nH]c2C)=O)CCC(C2(NC(c3nccc(F)c3Cl)=O)CC2)C1 CC(C)(C)C(C(=O)NC1CCOCC1)NC(C1CCCCC1(C)C)=O C12(C(=O)NCC3(NC(CC(C)c4cccnc4)=O)CCOC3)CCC(CC1)C2 c1(C(=O)NCCN(C(C2(F)C(C)OCC2)=O)C)ccc([N+](=O)[O-])c(N)n1 C1(NC(c2c(C)snn2)=O)CC2(C1)CC(C#N)C2 C(C(O)CC(=O)NCC1COCCN1C(=O)CS)N(C)C.c1ccc(F)cc1.C n1(CC=O)ccc(=O)c([N+](=O)[O-])c1.c1(OC)cc(C(=O)NCC(F)C)[nH]n1 C1(C(=O)NC(C)CCCO)C=CCCN1C(=O)Cc1cnns1 c1(NC(C)CC(C)NC(c2cnc(C(F)(F)F)s2)=O)ncnc(Cl)c1F O=C1CC(N2CCC(NC(C3(c4cnccn4)CC3)=O)C2)C(=O)N1 C1(Nc2cc(NC3CC3)nc(C)n2)CCc2ncc(C)n2C1 CCC(CCC(=O)NCCNC(=O)C(=O)NC1CC2CCC12)OC CCCC(CCC)=CC(=O)NC(C1CCCN1C(=O)CSCC(N)=O)C c1(SC)cncc(C(N2CCC(C)C2C)=O)c1.c1(C=O)ccc(C2CC2)cc1.N CCC(CNC(=O)Cn1nccc1C)(CC)NC(c1cccc(CO)n1)=O N1(C(Cn2c(C)cc(C)n2)=O)C2CCC1CC(CNC(C1CCCN1N=O)=O)C2 c1(CCC)cnnc(C(N2CCC(NC(C3(CC)CCCCC3)=O)C2)=O)c1 N1(C(C2(N)CC[Si](C)(C)C2)=O)CCC2(CCCCCO2)C1 N1(C(C(CC)(CC)CC)=O)CCC2(C=C(C(=O)NCCCC3C=NNC3=O)C2)C1 C1(NC(C2CC(C)(C)C2)=O)CCN(C(c2cnc(S(C)(=O)=O)s2)=O)CCC1.C c1(CC=O)cc(C(F)(F)F)cc(Cl)n1.C(C(C)(C)C)NC(C=C(CC)C)=O c1(C(=O)NC2CC(C)N(C(C3CC(N4CCCC4)C3)=O)C2)cccc(=O)n1C Cc1ccc(O)c(C(N2CC(C)C(C)C2)=O)c1.c1(C(=O)N)ccc(C(C)C)cn1 C(=O)(CCCCCc1cccs1)NCC(CNC(C=Cc1nnn(C)n1)=O)(C)C n1(CCCC)nnnc1C(c1cn(C2CCOC2)nn1)NCCC(N)=O C1(C(=O)NC(c2nc(C)[nH]n2)(C)C)CC2CC1CN(C(c1nccnc1C)=O)C2 C(C(=O)NNc1cc(F)cc(Br)c1)c1cc(C#N)on1 c1(N(C)C(c2ccc(-c3nn[nH]n3)nc2)=O)ccc2cc(Br)ccc2c1 Cc1cccc(C(N2CCCC2(C)C(N2CC(CO)C(CO)C2)=O)=O)c1F N1(C(Cc2cc(C)ns2)=O)CCC(C2CCOCC2)(CNC(=O)C=C(Cl)Cl)C1 C1CN(C(=O)CC2CCC(C)(C)CO2)C(C)(C)C1.c1(CC)cnoc1C(=O)N c1(C(=O)NCC2CCN(C(C3C(C)COCC3)=O)CC2)cc2n(c1)CCC2 [SH](=O)(=O)c1ccc(Cl)cn1.CC1(C(=O)N)CCN(C(C2CC3(CCC3)C2)=O)CC1 C(C)(C)(CN=c1cc(C)nc(NC2CC2)[nH]1)NC(C1(C=C)CCC1)=O c1ccc(O)c(Cl)c1.c1(C(N2CCC(C=O)C2)=O)cc(F)ccc1C(F)(F)F.N O(P(C)(=O)CNC(C1(NC(C2(N3CCCC3)CC2)=O)CC(C)C1)=O)CC N1(C(C(COC)N(C)C)=O)CC2CC(NC(c3ccc(C)cc3OC)=O)C1C2 c1(CN(C(C)C)CC)ccnc(C(C)(C)C)c1.c1(C=O)cocc1C(N)=O c1(C(=O)NCCCCNC(C2(CC)CCNC2=O)=O)ccc2c(C)nn(C)c2n1 CCS(=O)(=O)c1ccc(F)c(C(=O)NCC2COCCN(C(=O)C=NOC)C2)c1 Cc1nc2cc(C(=O)NCC3C4CC3N(C(=O)CP(C)(C)=O)C4)ccc2o1 c1(NCC(CC)(CC)CO)[nH]c(=NCCC=CBr)nc2ncn(CC)c12 C(CC(=O)NCc1ccccc1)(C(F)(F)F)OC.C(=O)C1=CC2C=CC1C2.C C(CC(C)(C)CC(=O)N(CCC(=O)NCCCOCCCO)CC1CC1)OC O=S(=O)(c1cnn(-c2ccc(Cl)c(F)c2)c1)NCc1cnn(C2CCC(O)C2)c1 C1(C(=O)N)(COC)CCC(=O)N1.C1(CC)CN(C(=O)C)CCO1.C1CCC1 N1(C(Cc2c(C)cco2)=O)CC(NC(=O)C(F)OC(F)(F)F)C(S(C)(=O)=O)C1 c1(C2(C=O)CC2)ccc(F)cc1.C1(CC(=O)NCC(C)OC)CCNC1=O c1(C(=O)NC(CC=C)CNC(C2CC2F)=O)ccc(N2CCCCC2=O)cc1 c1(OC)c(C(=O)Nc2cn(C)nc2OC)cccc1Br Cc1occc1CNC(=O)C(F)C1CC(NC(=O)CCc2cnoc2)C1 C1(C(=O)NCC(CNC(CCn2ccc(C)n2)=O)(C)O)COc2ccccc2C1 C=CCC(CNC(c1ccc(O)nn1)=O)C(=O)NC(CO)C1CCC1 C(=O)(C(C)S(N)(=O)=O)NCc1cc(C(=O)NCCC(C(C)C)C)sc1 C(c1ccc(F)cc1)=CC(=O)N(CC(C)(C)C)C.C1(C)(C=O)CC1(C)C.N c1(CC(=O)NCC2(COCC)CC2)ccc(C2CCCCC2)cc1 CCCCCC(CC)C(=O)N1CCCC(O)C1C N1(C(CCC=C=C)=O)CC2(CCC2NC(=O)C(CC(C)C)NC(N)=O)C1 C(=O)(C(CC)C(C)(F)F)N(CCC)CC.c1(C=O)n[nH]c(C)c1C(F)(F)F N1(C(C2C(C(C)O)C2)=O)CCC2(CCCN(C(c3cc(C(F)F)no3)=O)C2)C1 C(C(C)C(C)C(=O)NC12CC(C)(C1)C2)OC.c1(C(=O)N)ccc(F)cc1N Cc1cc(C(N2CC3CC2C3NC(c2ccns2)=O)=O)nn1-c1ccc(F)cc1 c1(C(N2CC(C(C)NC(C3CCC4(CC3)CC4)=O)C2)=O)cc(F)cc2cc[nH]c12 c1(C2C(NC(=O)NCC3CCCS3)C2)cccc(Br)c1 CC1(C)C(C(=O)NC2(C)CCCC2(C)C)CCN1C(=O)CCC(=O)C1CC1 C(=O)(CC(C)CC(C)(C)C)N1CCC(N(C(=O)C(C(CC)CC)OC)CC#C)C1 C1(CC(C)NCc2ccc(C(F)C(F)(F)F)cn2)CC2CCC(C1)N2 C(CN=C(NCC1COCCOC1)N1CCC(Cc2ccccc2F)C1)OCC c1(C(=O)Nc2cccc(OC)c2Cl)cnc2cc(Cl)ccn12 C(C(=O)N1CCOC(C(=O)NC(C)CCCO)C1)(C(C)(C)C)OC c1(C(=O)NC(CC=C)CNC(=O)CCC)cc2ccc(Cl)cc2nc1C N1(C(C(C)OC(C)=O)=O)CC(F)(CNC(=O)C(C)(O)C2CCC2)C1 c1(C=O)cc([N+](=O)[O-])ccc1.CCC(F)C(=O)NC(C)C(C)C.[SH](C)(=O)=O c1(Oc2c(C#N)ccc(C)c2)ncc(B2OC(C)(C)C(C)(C)O2)cn1 c1(CC(=O)NC(C(C)NC(c2cnc(CC)[nH]2)=O)C)cc(C)sc1C N1(C(Cc2nc(COC)sc2)=O)CCN(C(C2C(C)(C)C2(F)F)=O)CC1 c1(OC)sccc1C(=O)NCC1CC1NC(=O)Cc1ccoc1 C1(C(=O)NCC2(OC)CCCC2)CC2(CCC2)C1.C1(C(=O)N)CCCCO1 N1(C(CC(C)c2ccncc2)=O)CC(C2CN(C(c3cc4ccsc4s3)=O)C2)C1 Cc1csc(C(N2CCC(C(C)(C)NC(=O)CCCn3ccnc3)C2)=O)c1 c1(-c2cc(OC)ncc2Cl)ccc2[nH]c(C(=O)N=c3nn[nH][nH]3)cc2c1 c1(C(N2C3CC(NC(CC(C)(C)C)=O)(C3)C2)=O)cc(F)c(Cl)cc1F c1(NCC(=O)NCCc2c(C)ccs2)cccc(OC(F)F)c1 CCC(C)C(C(=O)N1CCOCC1CCNC(c1csc(C(C)C)n1)=O)N(C)C C1CCC2(CN(C(=O)CCC3OCCO3)C2)O1.c1(C(=O)NC)c[nH]cc(Cl)c1=O N1(C(c2ccc(C(F)(F)F)nn2)=O)CCc2ccc([N+](=O)[O-])cc2C1 Cc1cc(C(=O)NC(C)CCNC(=O)CC2CC(C)OC2C)c2c(C)n[nH]c2n1 c1(CC=O)ccc2[nH]ccc2c1.C1CCC12CCC2.C(C)(C)(C=CC=O)SC.N Cn1cc(C(=O)NC2C3CN(C(c4ccc(CO)s4)=O)CC23)c(C2CCC2)n1 N#CC1(C(N2CC=CC(C(N3CCC3CO)=O)C2)=O)CCCO1 C=CC1(CC(=O)NCC(CC)NC(c2sccc2-n2cnnn2)=O)CCOCC1 C(=O)(CCCC(C)(C)C)N1CC(NC(C=C(CC)C)=O)C(n2ccnn2)C1 C=CC(CCC)CC(=O)NCCC(=C)CNC(C1(O)CCCCCC1)=O C1(NC(=O)CCC2CCOCC2)CC2CC1N(C(=O)CCCCCF)C2 c1(CCC(=O)NC(C)CN(C(=O)CN2CCC(O)CC2)C)nc2cccnc2[nH]1 N1(C(CC2N(C(C(CCC)F)=O)CCOC2)=O)CCC(C)(C)CC1 C=CCCCCC(c1nnnn1C1(C)CC1)NCc1c(C2CC2)cccc1F CCC(C(=O)N1CC(CNC(c2cccc(C)c2)=O)C1)C(C)(F)F c1(N(CCNC(=O)CC2CCCOC2)C2CC2)ncnc2[nH]c3ccccc3c12 C1(NC(=O)COC2CC2)C2CC3CN(C(=O)CC4CC4(Cl)Cl)C1C3C2 C1(CCNC(c2cncnc2)=O)COCCN1C(c1ccc(Cl)s1)=O C(=O)(CCC(F)(F)C(F)(F)F)NC1CCN(C(C2(CC=C)COC2)=O)C(C)C1 N1(C(c2cnc(CC)nc2)=O)CCN(C)C(C(=O)NCCCC2CCOC2)C1 C1(NC(C2(CC=C)CC2)=O)CC(F)CN(C(=O)CCOCC(F)(F)F)C1 N1(C(C(CC=C)CC=C)=O)CC(NC(C2CCC(=O)N2C)=O)CC12CCCCC2 C1(C(=O)NCc2ncc(C)o2)(CC)CCCN(C(C2CCCN2C=O)=O)C1 C1(CNC(C(C)CN(C)C)=O)CCCN(C(c2cc(C3CCOCC3)[nH]n2)=O)C1 N1(C(c2cnn3ccc(C)nc32)=O)CCCC1C1CCCCN1C(=O)C=C(Cl)Cl c1(C(N2CC(NC)C(C)(C)C2)=O)cc(S(=O)(=O)CC2CC2)ccc1F N1(C(c2c(CC)nccn2)=O)CCOC2CCN(C(=O)C(C)CO)CC12 C=C(Cl)CC(C(=O)NCc1nc[nH]n1)NC(=O)C(C1CCCC1)OCC c1cnc(C(=O)N(C(C)C)C)c(F)c1.c1(C=O)c(C)noc1C(F)(F)F.C C1(CC(=O)N(C(C)C2CC2)CC)CCC(NC(=O)CCC2CCCC2)C1 c1(CC)cccc(C(=O)NC)n1.C1CCCCC1.N(C)(S(N)(=O)=O)CC=O N1(C(C(C(=O)OCC)F)=O)CCCCCC1.c1(C=O)ccc(N(C)C)c(F)c1.N C1(CNC(C2CCCC2O)=O)CN(C(c2ccc(-c3cc[nH]n3)s2)=O)CCO1 Cc1cnc(NCC2CN(C(C)C)C2)c(S(=O)(=O)N2CCC(C3CCCC3)C2)c1 C1(C(N(C2CCCN(C(=O)COC3CCC3)C2)CC)=O)CC12CCCCCC2 C1(CC(=O)N(C(CN(C(CN(C(C)=O)C)=O)C)C)C)CCCC(C2CC2)O1.C C(=O)(C1=CCc2ccccc21)NC(C(C)(C)C)CNC(=O)CC1CCCCC1O CC1CN(CC2CC3CC4C(C3)C24)CC2(CCC2)O1 C#Cc1ccc(F)cc1C(=O)NC1CC(CC)C1.N1(CCC(=O)N)CCCC1=O C1(NC(C2(CC#C)CCC2)=O)CN(C(c2ccc(Cl)cc2)=O)CC2CC12 O=C(CCCC1CC1)NCCC1CCCN1C(=O)CC1CCCCO1 C(=O)(CC1=C(C)NS(=O)(=O)N=C1C)N.C1(CC)CN(C(c2[nH]cnc2C)=O)CC1 c1(OCC)cccnc1C(=O)NCCCN(CCO)C(c1ccc(C)o1)=O C(=O)(CCCC(CC)NC(c1ccnn1COC)=O)N1CC(C#C)(N(C)C)C1 CCC(C)(C)CC(=O)N1CCCC1C1(NC(c2cccc(CS(C)=O)c2)=O)CC1 c1(C(N2CCCCC2)=O)cc(S(N)(=O)=O)ccc1N.C1(O)(C(N(C)C)=O)CC1 c1(-c2cn(CC3(C(=O)O)CCCO3)nn2)ccc2ncccc2c1 CCCC(C(O)C(=O)NCC1(CCO)CCC1)NC(=O)C(C)=CC1CC1 C(=O)(C1=NN(C)C(=O)CC1)NCCCN(C)C(c1ccn2nncc2c1)=O C12(CNC(CC3ON=C(C)C3)=O)CC1CN(C(C1CN(C(N)=O)C1)=O)C2 C1(NC(c2ccnc(OC)n2)=O)CCN(C(c2ccn(C)c2)=O)C12CCC2 NC(=O)C(C(N)=O)NC(c1ccc(C(F)F)cn1)=O N1(C(C(C)C#N)=O)CCCC2(CCCCC2NC(c2ccc(CO)o2)=O)C1 N1(C(c2cc(C)cc(C)c2)=O)CC2CC(C(N3CCC(O)C3)=O)C(C2)C1 C1(NC(c2cc(C)c(Br)s2)=O)CCCCN(Cc2ccc(O)cn2)C1 C1(C)(C(=O)NCC(C)(C2CC2)OC)CCCN1C(=O)CC1CSCCO1 Cc1cc(C(=O)NC2CCC(C(=O)NC3CC3)C2)cc(O)n1.c1ccccc1.C C(CC(=O)NOC1CC1)(C(F)(F)F)NC(COCC(C)C)=O c1(C(N)=O)ccc(C=CC(=O)NC(C)(C)C)cc1.C1(C=O)CCOC(=O)N1 C#CCCCC(C)C(=O)NC1CCCC1(C)CNC(=O)CCc1ncccn1 C1(C(=O)NCC(C#C)OC)CC2(CCC2)CN1C(C1CC(F)CN1C)=O C1(C(N(CCOC)CC2CCCS(=O)(=O)C2)=O)COc2ccc(OC)cc2C1 c1(-c2cnc(CC)s2)nc(C2CCCO2)nn1C1CCCCC1 C(=O)CCS(=O)(=O)C(F)(F)F.c1(CC(=O)N(C)CC)ccc(C(N)=O)nc1 C1(CNC(C2(C)CCOC2)=O)CCC(F)CC1.c1(C=O)cc(C(N)=O)cs1.C C=CC(CC)CC(=O)N(CC(=O)NCC(C)N(C1CCCC1)C)CC1CC1 C(=O)(CCCCC=O)NC.C1CC(=O)N(C2CN(C(=O)CC3CN(C)C3)C2)C1.N N(C(=NCCCF)NCc1ccc2c(c1)COC2)CCCN(c1ccccc1)C Cc1cnc(CC(N2CCC(n3cc(CNC(c4cnsn4)=O)nn3)C2)=O)s1 c1(C(N2CCC(C(C)(C)NC(c3ccc(Cl)cn3)=O)C2)=O)ccc(=N)[nH]n1 C1(C(=O)NCC2CC23CCC3)CCCCCCN1C(=O)CN1CCNC1=O c1(C(=O)NCC2C3N(C(C(CC=CC)C)=O)C(CC3)C2)cc2c(F)cccc2s1 Cc1cc(=NC(=O)C(C)SCC(=O)NCCCCCN(C(=O)C(C)(C)O)C)[nH]o1 C(CC(C)N=c1[nH]c(=NC2CCC(C#N)CC2)c2c(F)cccc2[nH]1)SCC c1(C(=O)NCC2CN(C(C(CSC)O)=O)C3(C2)CCC3)ccc2c(n1)OCCO2 C1(C(=O)NC(C2CCN(C(=O)C=Cc3cncs3)C2)(C)C)CCc2c[nH]nc2C1 N1(C(=O)Cc2csc(Cl)c2)CCC2C(CCN2C(C2CCOC2)=O)C1 C1(C)(C(N2C(C(=O)NCC(C=C)O)CC(C)C2)=O)CC(=O)N(C)C1 c1(CN2CC(F)(C(=O)NCC3COC3)C2)cnc(Cl)cc1Br CCCCCC1CN(C(C2CC(CCNC(C3(CSC)CCC3)=O)C2)=O)C1 c1(CC(N2CCC(CC(=O)Nc3ccc(Br)cc3Cl)C2)=O)cccc(Br)c1F c1(CN(C)C(=O)NC2CC3CCC2C3)nc2ccccc2o1.C(C)(C)C.C=O N1(C(CCC(=O)OC)=O)CC2ON=C(CNC(=O)CC3(O)CCC3)C2C1 Cc1ccc(CC(N2CCC=C(CNC(=O)Cc3csnn3)C2)=O)cc1Cl C#CC1CCCCN1C(=O)CN(C(c1cc(C)nc(O)n1)=O)C(C)C N1(C(CC(C=C)(C)O)=O)CCC2(CC1)CCN(C(C1CCC3CCC1O3)=O)CC2 C(C)(C)(CCCNC(c1ccccc1C(=O)OC)=O)NC(C=CCC)=O c1(C(=O)NCC2CCCC3(CCOC3)O2)cc2c(Cl)cccn2n1 c1(C(=O)NC(CCNC(c2c(CC)ncs2)=O)C)ccnc(N2CCCC2)c1 c1(C=O)cccn(C(F)F)c1=O.CC1CC(C(=O)NCCOCCC)CCS1.N N1(C(C(=O)NCCOC)=O)CCC(C2CC2)C1.N1(CC=O)CCC(C)C1.C CC1CCCCC1C(=O)NCCCC1CCN(C(=O)COC2CCCC2)CC1 N1(C(C(CC#C)C2CC2)=O)CC2=C(C1)CN(C(=O)C(C)COC(C)=O)C2 C1(C(=O)N)CCc2nn[nH]c2C1.c1(CN(C(=O)C=CCF)C)ccccc1C Cc1ccc(NC(=O)CSCCNC(=O)ON2CCCC2)c(C)c1 c1(OC(C)C(=O)NCCC(C)CCNC(C2(C)CCNC2=O)=O)ccccc1Cl c1(C(=O)NCCC2CCCCN2C(C2CC2(F)F)=O)cc2cc(F)ccc2cn1 c1(NC(C2OCCN(C(C3C(CC)C3)=O)C2)C)cc(OC)c(OC)cc1[N+](=O)[O-] c1(C(N(C)CCN(C)C(C2(C)CC2F)=O)=O)cc2ccccc2nc1O C(C(C(C)(C)C)NC(c1cnn(C)c1F)=O)NC(c1cc(C(C)C)[nH]n1)=O C(=O)(C#CC1(C)COC1)N.C(=O)(CC1CCCO1)N(CC(=O)NC(C)C)C Cc1ccc2n[nH]cc2c1C(=O)N(C)CC1CN(C(C2(C)CCCC2)=O)CCO1 N1(C(CCCOCC)=O)CC2CCCC1C2CNC(=O)C(C1CCOCC1)F CC1=C(C)CC(C(=O)NC2(C)CCOC2)CC1.c1(C(=O)N)nn(C)c(C)c1Cl c1(C(=O)NCC=CC(=O)NC(c2cn(C)nn2)C)ncoc1C1CC1 C1(NC(Cn2ncc(C)c2)=O)CCSC12CN(C(c1sccc1CN(C)C)=O)C2 CN1CCCC(C(=O)NCCNC(C2CC3(F)CC2C3)=O)C1.c1ccccc1.C C(=O)(C(CC(C)C)N1CCCCCC1)NCCOCCNC(C(CCC)O)=O N1(C(c2c(C)n(C)cc2)=O)CCCC(C(N2CC(O)C(O)C2)=O)CC1 Cc1nc(C(=O)NC2C=CC(CNC(=O)CCOC3CCOC3)C2)nn1C Cn1ccc2cccc(C(N3CCC(C(=O)N=c4nc[nH]n4C)(C)C3)=O)c12 c1(C(N(CCOC)CC)=O)ncnc2c1ccn2C.C1(C=O)CC2(CC2)CO1.N C(=O)(C(CC)C(C)(F)F)NCC(CC)NC(c1cc(C)c(Cl)cn1)=O C(=O)(C(C(C)C)OC(c1nc(-c2ccccc2)oc1C)=O)OCC n1(CCN(C)C)cc(NC(c2ccc(O)nc2)=O)ccc1=O S(=O)(=O)(c1ccc(C)c(N(C)C)c1)NC(c1ccccc1F)C=C c1(C(N(CC(C)NC(=O)CN2CC(C)(C)C2)C)=O)sccc1C(C)(C)C C1CC12CCN(C(=O)C(F)(F)c1cscn1)CC2.C1(C(=O)N)CC2(CCC2)C1.C Cn1nccc1CN1CCC(NC(=O)NCCCCc2ccccc2)C1 c1(NC(C(C)Oc2cccc(C(C)C)c2)=O)cc(F)c(I)c(F)c1 N1(C(c2cnc(C(C)(C)C)[nH]2)C(=O)N)CC2(CCC1)CC2.C(CC)SCC c1(C(=O)NC2(C3CCN(C(=O)CO)C3)CC2)[nH]nc2ncnc(O)c12 CC1=NNC(=O)C1CC(=O)NCc1ccc(C(=O)NOC(C)(C)CO)cn1 C1(N(C)C)(CC)CCN(C(C2CCOC(c3cccc(F)c3)C2)=O)C1 CN1CCCC(C(=O)N(CC(C)(C)NC(=O)CCC2OCCO2)C)C1 c1(-c2nc(CCCOC)nn2CC2CCOC2)ccc(OC)c(OC)c1 C1CN(C(=O)Cn2cnc(=N)[nH]2)CC(C)(C)C1.C1(C(=O)N)(SCC)CC1 C(CCF)(C(=O)NCC(=O)NC1CCCC1)NC(C1CC(=O)OC1)=O c1(C(N2CCN(C(C(CN(C)C)O)=O)CC2)=O)ccc2oc(=O)oc2c1 N1(C(CCOCC#C)=O)CC(NC(=O)Cc2ccc(Br)s2)C(O)C1 n1(C2CN(C(C(F)=C(C)C)=O)C2)cc(C)nn1.C(=O)C(C1CC1)N(C)C C1(CCC(=O)NCCCCNC(C2(CO)CC2(F)F)=O)CCCC(=O)N1 c1(CNC(=O)C=CC=Cc2ccccc2)ccc(Br)nc1Cl Cn1ncc(C(N2CCC(CNC(=O)CCC3CCOC3)C2)=O)c1N N1(C(=O)C=C2CCOCC2)CC(C2CN(C(=O)CSCCN(C)C)C2)C1 CC1(NC(=O)CC23CCCC2C3)CCN(C(c2cnccc2C(F)(F)F)=O)C1 C(CCCCF)NC(C=CC(C)NC(C1CC2(CC2)C1)=O)=O c1(CNc2cc(N3C(CC)CN(C)CC3)nc(C)n2)c[nH]c2ncc(Br)nc12 N1(C(C(C)OC(C)(C)C)=O)CC(O)(C2CCN(C(C3CC(F)C3)=O)CC2)C1.C CCCCCCC(F)C(=O)N1CCCC1C(C)(C)CNC(=O)C=Cc1cccs1 c1(CN2CC3C(C(=O)Nc4cc(C)nn4C)(C3)C2)cnc2cc[nH]c2c1 C1(CC)CC(C(=O)NOCC(N)=O)CCN1C(=O)CCn1cccc1 CC1(NC(c2ccccc2)=O)CN(C(C2CC(C(F)(F)F)CO2)=O)C1 c1(C(N2CC(NC(c3cccc(F)c3Cl)=O)C3C2C3)=O)cc2ccc(F)cc2[nH]1 C(CNC(c1sccc1CO)=O)(C(=O)NCCCC(=O)NC1CC1)OC C1(CNC(c2c(C)csc2)=O)CN(C(=O)C2=CCCOC2)CC2(CCC2)O1 C1(C(C(=O)N(CC(C)C)C(C)C)C)CCCN(C(=O)CCn2cnnn2)C1 c1(CSCC(=O)NCCN(C(=O)CC(C)CF)CC)ccc(Br)cc1 C1(OC)CN(C(=O)C=Cc2cc[nH]c2)CC1.c1(C(=O)N)c[nH]nc1C1CCCO1 c1(C(=O)NCC(c2ccccc2)NC(C(C(C)C)(C)O)=O)noc2c1CCCC2 C(=O)(C(O)C(F)(F)F)NCC1C(C(=O)NC2(CC)CCCCC2)CCO1 C#CCC(C)(C(=O)NCCC1CCCOC1)NC(C12COCC1C2)=O C(=O)(C(C)S(N)(=O)=O)N1C(CCNC(C(CC)(F)F)=O)CCC1 C1(CNC(C2(CC=C)CCCC2)=O)CCCCC1NC(=O)C(C)C(F)F N1(C(c2ccc(CCC)s2)=O)CC(NC(C2(SC)CCC2)=O)C2CC12 C(=O)(C1=Cc2c(ccc3ccccc23)OC1)N1C(C)(C)C(=O)CC1 Cn1c(C=CC(=O)NC2COCC2NC(=O)CCCCCF)cc2ccccc12 C1(NC(CN(CCC#C)C)=O)CC12CCN(C(c1ccsc1C#N)=O)CC2 N1(C(C2CC(=C)C2)=O)CCC(O)C(N(C(=O)C(C)CSC)C)C1 C1(CNC(C(CC#C)C2CC2)=O)CCC2(CN(C(c3cccc(N)c3)=O)C2)O1 C(CN=c1[nH]cc([N+](=O)[O-])cc1CO)N(C(c1csnc1C)=O)CC c1(C(N2CC(C)(NC3CN(C(c4c[nH]c(=O)cn4)=O)C3)C2)=O)c(F)cccc1Cl C1(CNC(CSCCNC(CC2(N(C)C)CCC2)=O)=O)CC(C)(O)C1 N1(C(c2c(C)nc(CNC(C3=C(C)OCCS3)=O)o2)=O)CCc2cc(F)ccc21 N1(C(C(CC)CCCO)=O)CCC(O)(Cn2cc(C3CCN(C)C3)nn2)CC1 C1CC2CC(C1)N(C(C1CC1c1ccccc1)=O)C2.CC1OC(=O)NC1C(=O)N C1(CNC(C2CC(SC)C2)=O)CC2CCC1N(C(c1c(Cl)cncc1Cl)=O)C2 N1(C(CC(C)F)=O)CCN(C(c2ns[nH]c2=O)=O)CC1c1cn[nH]c1 c1ccccc1Cl.c1(C(=O)NCC2CCCN2C(=O)C)nccc(C(F)F)n1.N C1CCCC2CC12.C(C(C(=O)N1CCC1)n1cc(CC2CCOCC2)nn1)OCC.C N1(C(C(C)(N(C(c2nc(OCC)oc2)=O)C)C2CC2)=O)CC2(CCCO2)C1 N1(C(c2ccc(NC(CC(C)C)=O)c(F)c2)=O)CCC2(CCCN2)C1 N1(C(c2cnc(CCCC)s2)=O)CC(NC(C2(SC)CCC2)=O)C(C(F)F)C1 c1(OC)cc(Cl)ncc1CN1CCC1C(N1CCN(C(=O)C(F)(F)F)CC1)=O C1(Cn2cc(CN3CC(c4nc(C(C)C)[nH]n4)OCC3)nn2)CCCNS1(=O)=O C(CCCC(C)C)(C(=O)NC1CC(F)(F)C1)N1C(CCCC)CCC1 Cc1cc(N)cnc1C(N1CCN(CC(=O)NCC(O)C(N)=O)CC1)=O C1(C)(CNC(C2(C=C)CCC2)=O)COCCN(C(c2cccc(F)c2OC)=O)C1 CCC(CCC(=O)NCCN(C(c1nc(C2CC2)ncc1Cl)=O)C1CC1)OC C1(C(C)(C)C)CC2(C1)CC2c1nc(C2CC2(C)C)nn1-c1cccnc1 c1(CNCC(C=C)(C)O)csc2ccc(C)cc12 CCCCC(CCCC)C(=O)NCC1CC1NC(=O)CCc1ccc(OC)cc1 C1(NC(c2cnn(C)n2)=O)CCCN(C(=O)CCc2nc[nH]n2)C1 N1(C(c2cc(C(C)C)no2)=O)CCC=C(C(=O)NC2C(C)CCCC2C)C1 c1(C(N(CCC)CCNC(C2CCOC2)=O)=O)cn2cccc(C)c2n1 Cn1cc(Cl)c(C(N2CC3CC3(CNC(=O)C=Cc3ccccn3)C2)=O)n1 C(=O)(C(CN=[N+]=[N-])NC(c1ccc(Cl)cn1)=O)N1CC(C)SCC1 C1(NC(CN(CC#C)C(C2CCN(C)C2)=O)=O)CCSCC1 C1(C)(C(N(C)CCn2cnnc2)=O)CCCN(CCC(C)(C)O)C1 N1(C(C=Cc2n(CC)ccn2)=O)CCCN(C(=O)CCC=CC(C)C)C(C)C1 c1(OC)ccc(CC(=O)N(CC(C)CNC(c2coc(Br)c2)=O)C)c(C)c1 C(=O)(C(F)CC(C)C)NCC1CC(NC(C(C=C)(C)O)=O)C1 c1(C2(C(=O)NC3CN(C(COCC=C)=O)C3)CCCC2)cccc(Cl)c1F CCC(C)CCCCC(=O)N1CCC=C(C(=O)NCC(Cl)C(C)(F)F)C1 c1(C=O)cscc1S(C)(=O)=O.C1(C)(COC)CCCN1C(C1CC(O)C1)=O C(C)(C(=O)NNC(=O)c1cccc(Cl)c1)n1cc(C2C(C(=O)OC)C2)nn1 N1(C(CN(CCCC)C)=O)CC2CCN(C(=O)CSCc3ccccc3)CC2C1 C=C=CCCC(=O)NCC1CCCCN1C(c1cc(C)ns1)=O C1(CNC(C2(OCC)CCC2)=O)CN(C(=O)Cc2ccno2)CC1O.C CCCCCC(C)(CC)C(=O)NC1CN(C(c2ccn3cncc3c2)=O)CC1C Cc1cccc2oc(=NCC(O)CNC(C3(C)CC3(F)F)=O)[nH]c12 Cc1ccnc(-c2cn(C(C)(C)CC(=O)N3CCC(C)(C(=O)O)C3)nn2)c1 Cc1ccc2oc(N3CCCC(NC(C4(c5cccs5)CC4)=O)C3C)nc2c1 CCC(C)(C#N)C(=O)NC(C)CNC(C1CCC(C)=C(C)C1)=O C1(SC)CCCC1n1cc(CCCNC(C2(C3CCCO3)CCCC2)=O)nn1 c1(C(N2CC(C(C(=O)NCc3[nH]c(C)nc3C)OC)C2)=O)c[nH]c2ncccc12 c1(C(=O)NC(CCC)CCCNC(C2(C)CC2)=O)ccc2c(c1)CCCCS2 C(=O)(CS(C)(=O)=O)NCC(C(C)C)NC(C1(C)CC1(C)C)=O C(=O)(C(C)(C)C(=O)NCC(C)(C)Cn1cc(C)nn1)NC.c1ccccc1.N C(=O)(CCC(C)(C)[N+](=O)[O-])N1CC(C(N(CC(C)CO)C)=O)CC12CCC2 C1(NC(C2(C)CC2(F)F)=O)C2CN(C(c3ccc(-n4cccn4)nc3)=O)CC12 C1(NC(=O)CCC(F)(F)F)CN(C(c2ccnnc2)=O)C2(CCOC2)C1 C(=O)(C(F)(F)C(F)(F)F)N(CCCC(C)(C)C)C.CN1CCC(CC(=O)N)CC1 c1(NC(C(C2CCCC2)NC(CS(C)(=O)=O)=O)=O)cnc2ccnn2c1 c1(C(N(C(C)CCNC(C2(N=[N+]=[N-])CC2)=O)C)=O)ccc2c(c1)CCC(=O)N2 c1(C(=O)OC)cnc(C)nc1N(CCCC)C.c1(CC(=O)N)ccc(Cl)c(F)c1 c1(C(N2CCC(O)(C(=O)NCC3CC3)CC2)=O)ccc2nc[nH]c2n1.C1CC1 c1(C(=O)NC2CCN(C(c3nnn(C)n3)=O)CC2)cc2cc(Cl)cnc2[nH]1 c1(NC(=O)N)ncccn1.C12CC(C1)C2.c1(CCCC)ccc(C(F)(F)F)o1 C1(CC)(NC(C2CC(F)CN(C(c3cnco3)=O)C2)=O)Cc2ccccc2C1 C1(CNC(C(c2ccccn2)C)=O)CCN(C(c2cnc(S)nc2)=O)C1(C)C C(=O)(CCCCCNC(C1CC(C)(C)CN1C)=O)NC1(C(=O)OC)CCC1 CC1CCn2ncc(C(N3CC4CC(NC(=O)CCCCC(N)=O)C3C4)=O)c2C1 c1(CN)cn2cccc(C(N3CCN(Cc4ccno4)CC3)=O)c2n1 CCC(CC)(CO)C(=O)NC1CCC(NC(c2[nH]c(C3CC3)nc2C)=O)C1 N1(C(=O)OC(C)(C)C)CCC2(CC(C(=O)N3CCC3)=NO2)C1.C12CC(C1)N2 CCC(CC)CC(F)C(=O)NC(C1CCCN(C(c2cnsc2)=O)C1)C C1(NC(C(c2cccc(F)c2)C)=O)CCCN(Cc2nc(Cl)cs2)C1 CC1(C)CC1(C#N)C(=O)NC1CCN(CCNC(=O)CCc2cncnc2)CC1 C1(C(=O)NCC(CC)CC)CCC(C2CC2)N1C(c1cccc(CO)n1)=O n1(CC(=O)OCC=C(C)Cl)ccc2cc(C)ccc12 O=C1CC(C(=O)Nc2ccc3c(n2)NCCC3)c2cc(Br)ccc2N1 c1(C(N2CC(C(C)NC(c3ccc(C)c(F)n3)=O)C2)=O)ncc([N+](=O)[O-])n1C N1(C(C(CCOC)C)=O)CC2C3CCC(C2C1)N(Cc1cc(F)ccc1Br)C3 CC1CCN(C(c2cc(F)cnc2O)=O)CC1NC(=O)Cc1ccnc(F)c1 C(=O)(C(C)(F)CCCC)NC(CC=C)CNC(c1ccn(C(C)C)n1)=O c1(C2(C)CCO2)cccc(C(N2CCC(C)(NC(=O)CC3CCCC3)C2)=O)c1 c1(C(=O)NCC=CC(=O)NC(c2nc(C)on2)C)ccc(F)cc1F C#CCCCC(=O)N1CCCC1(C)C(=O)N(C)Cc1cc(C)cs1 CCC(CC(F)(F)F)C(=O)NC1(CC)CCCC1.C1(CC=O)CCC(C)(C)C1.N C1(C(N2CCC(C(=O)OCC)C2)=O)CCN(C(=O)c2cnn(C)c2Cl)O1 C(=O)(CC(CNC(C1CCC1CO)=O)C1CCC1)NC(n1cnnn1)(C)C c1(C(N2C(CCNC(C)=O)CSCC2)=O)ccc(Cl)c(C)c1N N1(C(c2ccn(C(C)C)c2)C(=O)NCC2CCCO2)CC(CCO)OCC1(C)C N1(C(C(CC(C)C)N(C)C)=O)CC2OCC(NC(=O)CC(C)C3CCCC3)C2C1 c1(C(=O)NC(C(=O)O)Cc2ccc(F)c(Cl)c2F)ccc2c(c1)COC2 C1(C(=O)N)CCC(C)(C)N(C(c2c[nH]c(=O)cn2)=O)C1.C1(OC)(C)CCOC1 c1(OC)cc(C(N2CC(C(C)NC(=O)C(N3CCNC3=O)C)C2)=O)cc(F)c1 N1(C(c2c(C(=O)OC)cccc2)=O)CCC2CN(C(=O)C(F)(F)C(F)(F)F)CC12 c1(C(=O)NCCCN(C(=O)C(C)(O)CC)CC)ccnc2nc(C)nn12 N1(C(Cc2c(C)noc2Cl)=O)CCC(NC(c2nncs2)=O)C(F)(F)CC1 c1(N(C(c2cnc(NC(N)=O)s2)C(=O)NC2CC2)C)ccc(F)cc1.CC C1(CNC(C(NC(CSCCOC)=O)SC2CC2)=O)CCOC1=O C(=O)(CCC(C)(C)[N+](=O)[O-])NCCC1CC(NC(C#CC(C)(C)C)=O)C1 C1(NC(C(c2csnc2OC)N(CCC#N)CCC)=O)CCCCC1 c1(OC)cccc(Cl)c1CC(=O)N(C)C.C1(O)CN(C(=O)CCc2cnco2)C1 C(=O)C(C)N(C1CC1)C=O.C(C)(C)(CC)NC1CCCC1.C1CC1.C C(CN=c1ccnc(N)[nH]1)C1CN(C(=O)Cc2ccccc2)C1.c1nncs1 CN=c1ccc(C(=O)NC2CCCC(C(=O)NC3CCNC3=O)C2)c[nH]1 C1CC2(CN1C(=O)C=C1CCC1)CC2(F)F.c1(C=O)cc(C2CC2)[nH]n1.N c1(NC(C)=O)c(C(=O)NC2CCCN(C(C3(CO)CCCO3)=O)C2)cccc1C C(C(C)(C)C#CC(=O)NC1CCC2CC1CO2)NC(C(C)OCCC(C)C)=O C1(CC)CN(C(=O)C2=CCCCC2)CCC1NC(c1ccc(C)c(CO)c1)=O CCCCC(C)C(=O)N1CCC(N(C(=O)Cc2cnnn2C)C)C1 CN1CCC2CCN(C(C3(CO)CCC3)=O)CC12 C1(C(N(C2CCC(CO)CC2)C)=O)CN(C(C2(C)CCSCC2)=O)CC1(C)C CC1(CNC(C2(NC(=O)C=Cc3ccccc3)CSC2)=O)CCCCO1 C1(C(=O)Nc2c(C#N)nc[nH]2)CCN(C(c2cc(O)ccc2Br)=O)CC1O CC(O)(C(=O)N1CCCC(C(N2CCOC(c3ccccc3)C2)=O)C1)C(F)(F)F Cc1ccc(C(=O)N(CCCNC(=O)Cn2ncnn2)C(C)C)c(=O)n1C C12(C(=O)NCCCNC(C(c3cc(C)sc3)(C)C)=O)CCC(CC1(F)F)C2 c1(OC)cc(N)c(F)cc1C(=O)N.c1(C=O)cc(S(N)(=O)=O)co1.CCCO c1(C(c2n(CC)nnn2)NC2CC(=C3CC3)C2)cc(Cl)cc(Cl)c1F C1(CN(C(=O)CCn2ccnn2)CC)CCCN(C(=O)CCO)C1.C(N)=O.N c1(C(N2CC(CCCC)N(C(C3CCCCS3)=O)CC2)=O)nnn2c1CCCC2 C(C(O)(CO)CO)NC(C(c1n(C)ncc1)NC(=O)CC1CCCO1)=O C1(CNC(CCSCCCC)=O)CN(C(=O)CNC=O)CCC12CCOC2 c1(N2CCC(NC(CC3C(OC)COCC3)=O)C2)snc(C)c1C#N N1(c2nnc(C)s2)CCC(C2CCCN(C(=O)COCC3CCOC3)C2)C1 C1(C)(COC)CN(C(=O)C(n2cc(-c3ccnc(C)n3)nn2)C)CC1C N1(C(c2ccc(OC)c(C)c2)=O)CC(NC(c2nnc(S)n2C)=O)C2CCCC12 CC(CC(N)=O)C(=O)NCC1CN(C(=O)COC2CCOC2)CCO1 c1(OC)cc(Cn2cc(CNCS(=O)(=O)C3CC3)nn2)c(F)cc1C N1(C(C(CCCC)NC(=O)C2=NOC(C)(C)C2)=O)Cc2cccc(O)c2C1 c1(C(N2CCC(NC(C3(CC)CCCC3O)=O)CC2)=O)ccnc(Cl)c1O c1(C(=O)NCCOC2CCN(C(C(C(CC)C)O)=O)C2)c(C)ccc2n[nH]cc12 Cc1ccnc(C(=O)NC(c2ccnn2C)C(N2CCCC(N(C)C)CC2)=O)c1F CC1(C)COc2c(C(N3CCC(C)(CCNC(C4CC45CC5)=O)C3)=O)cccc21 C1(NC(c2nc(CC)sc2)=O)CCC(C)(C)CC1.C(c1ncc[nH]1)=CC=O.C C(=O)(C#CC1CCOCC1)N(C)CC1N(C(C(C(C)C)n2cnnc2)=O)CCC1 Cc1cc(Cl)c(C(N2CCC(CCNC(=O)CCSCC(N)=O)CC2C)=O)cn1 C1(CN(C(=O)CSC(F)F)C)CCCN(C(C2CCCCC2C(F)(F)F)=O)C1 C(=O)(C1=C(C)CCC1)N1CCC(O)(CCNC(C(C)NC(C)=O)=O)C1 C(CC(C)(C)CO)NC(c1c(C)ocn1)c1nnnn1CCN1CCOCC1 CC1(C)CCC(C(N2CCCCC2CCNC(=O)COCCO)=O)CO1 C1(NC(C(C)OCC#C)=O)CN(C(=O)CSC2CC2)CC(C)(C)C1 Cc1nc(C(N2CC(CNC(C3CCOC3)=O)C(O)C2)=O)c2n1CCCC2 c1(OC)cc(C)c(Cl)cc1C(=O)NC1CCN(C(=O)CC2CCN(C)C2=O)C1 CC(C1CC1)=CC(=O)NC(C1(CNC(C2(N(C)C)CC2)=O)CC1)C c1(OC)nscc1C(N1CCCC1CNC(=O)CNC(=O)C1CC1)=O CC(CC(=O)NCCOCCNC(c1ccc(=N)[nH]c1)=O)P(C)(C)=O C1(C(=O)Nc2n(CC)nc(C)c2Cl)COCCC12CN(C(=O)C(Cl)CC)C2 c1(C(N2CCCCC2)=O)cn(C)c(=O)n(C)c1=O.C(C)(C(=O)NC)NC(C)=O N1(C(C)=O)CCC(C(=O)NCC(O)CC)C1.c1(C=O)nnn(C(C)(C)C)n1.N C=CCCC(CC(C)C)C(=O)N1CC=C(CNC(c2ccnc(CC)c2)=O)CC1 N1(C(CCc2cncc(OC)c2)=O)CCOCC(NC(=O)Cc2cccn2C)C1 C1(C(=O)NCC(CN(C(COCC)=O)C)O)CCCC2(CCC2)C1 c1(C(N2CC(C(C)NC(C3C(C)=CCS3)=O)C2)=O)cnn(C)c1Cl CC(C)(CCCCNC(=O)Cc1cncnc1O)NC(=O)Cc1ccc(O)cc1 c1(C(=O)NC(C)CCCCNC(C2CCN(C)C2)=O)ccc(=O)n2c1COCC2 CC(CNC(C1(CCNC(C2CCCN2C)=O)CCCC1)=O)C(F)F c1(C(=O)NC2CN(C(C(CC)(CC)CC)=O)CC2(C)C)c(C)nn2cccnc12 c1(C(N2CCC(NC(CC(=O)NCC#C)=O)C(C)C2)=O)cnc2cccc(C)n12 N1(C(CN(CC)CC)=O)CCCCC1C(C)NC(C1CCS(=O)CC1)=O n1(CC(N2C(CN(C(C(CCC)(C)C)=O)C)CCC2)=O)cc([N+](=O)[O-])nc1C N1(C(c2c(CC)nccc2)=O)CCC2CN(C(=O)C(n3ccc(C)n3)C)CCC12 C1(C)(C=O)CCCCO1.c1(CC(=O)N(CC)CC)nc(C2CC2)nn1C.CO C(CC(C)C)(C(=O)N1CCC(C)C1)NC(C)=O.c1(C=O)cc(C2CC2)on1.C c1(CCC)ccc(CN2CCC(C(=O)Nc3ccnc(OCCOC)c3)C2)cc1 c1(C(N2C(CNC(C3C(C=C)CC3)=O)CCC2)=O)ccccc1-c1cnn(C)c1 Cc1ocnc1CC(=O)NCCOC1CN(C(=O)C=CC2CCCO2)C1 N1(c2cc(OC)ncn2)CCC(NC(c2nc(F)ccc2Cl)=O)C(O)C1 c1(C(=O)NCC(N2CC3C(NC(CC(C)(C)C)=O)(C3)C2)=O)ccc(F)cc1F CC(CS(C)(=O)=O)NC(c1ccc(C)o1)=O.C1(CC=O)CCC(=O)NC1.N O=C1CC2(CCC(C(=O)NC3CC(C)(NC(C4CC(F)C4)=O)C3)CC2)CN1 N1(C(C(C)CSCc2ccccc2)=O)CCC(N(C)C(C2CCN2C)=O)C(F)C1 c1(CC)nnsc1C(N1CSCC1C(=O)NCCOCCF)=O c1(CN(C(=O)NCCN(CC(O)C(F)(F)F)C)C)ccc(Br)cn1 c1(C(N(C2CCCOC2)CC)=O)cc(CNC(c2ccc(C)o2)=O)cs1 c1(N2CCN(c3cccc(OC)c3)CC2)nc(C)cc(=NCCSCC(C)C)[nH]1 n1(CC(=O)NC2CCC(CNC(C(CC)(C)O)=O)CC2)ccc(=O)c(O)c1C C(=O)(C(C)(C)CNC(c1cnc(N)cn1)=O)NCCCCCOC c1(C(N(CCCCCNC(c2cccc(NC)n2)=O)C)=O)c(Cl)c(CC)nn1C CC(C)C(N=[N+]=[N-])C(=O)NCc1nocc1C(N1CCC2C(C1)C2(F)F)=O c1(C2(CCNC(=O)NCCN(C(CC)C)CCO)CC2)ccc(F)cc1 CCS(=O)c1ccccc1C(=O)NC1CCCC(NC(c2nc(C)nn2C)=O)C1 Cc1csc(=O)n1CC(=O)NC(C1CN(C(=O)CCNC(=O)CO)CCO1)C C1(c2nc(C3(C4CCN(CC#N)CC4)CC3)on2)CCC(C2CCCO2)O1 C1CCCC(=O)N1.C1(C(N)=O)COCC1C(=O)NCc1nocc1C(=O)N c1(CC)nc2ccccn2c1C(=O)Nc1cc(C(F)(F)F)nc(Cl)n1 c1(CC)cc(C)c(C(=O)NC(CC)C(C)C)o1.c1(CC=O)sc(S)nc1C.N N1(C(CC2(OC)CCC2)=O)CCC(NC(c2ccc(OC(F)F)cc2)=O)C1(C)C CCCCCCC(C)C(=O)NC1CC1C1CCCN(C(c2ccc(CO)o2)=O)C1 C1(COC(CCCc2n(C)cnc2)=O)CCCCC1(F)F C1(C)(C(N2CC(CC)NCC2)=O)CCCN(CC2CN(C)C2)C1 CC(C)CC(C(=O)NC1C=CC(CNC(=O)CCCC2CCOCC2)C1)C(C)C C=C=C(C)CC(=O)N1CCC(N(CCOC)C(c2nsc(OCC)n2)=O)CC1 c1(C(=O)NC2C(C)C3N(C(C)=O)C(CC3)C2)[nH]c2c(Cl)cccc2c1C C(c1ccc(Cl)cc1F)=CC=O.Cc1cc(C(=O)N(C)CCOCC)ncn1.N Cn1nc2c(c1C(N1CCC(F)(F)C(CNC(c3ccsc3Cl)=O)C1)=O)CCC2 C(=O)C=O.CC(C)CC=O.CCC.C1(C(=O)O)CC1CC.C(C)(C)C C1(C(=O)NC2(C)CCCN(C(c3c(CC)cno3)=O)C2)CCC2(CCCCC2)C1 Cc1nc2ncc(C(=O)NC3COCCC3NC(=O)CC3CCSCC3)cc2o1 c1(OCC)ccnc(NC(CNC(=O)CC2CSCCS2)C2CCC2)n1 Cn1ccc2c(NC(c3scnc3-c3c(F)ccc4[nH]ccc34)=O)ccnc12 c1(OC)ncc(C(=O)NC2(CC)CCC2)c(C)n1.C(=O)C(C(C)C)C1CCC1 C(C)(C)(C(C)CC(=O)NC)NC(C(=O)NCC)=O.C1(C)CSC(C)=N1 CC1CN(C(c2c(N)cncc2Br)=O)CCCN1C(=O)CC1C=CCC1 CCCCCCC(CC)C(=O)NC(CNC(C1CCCCS1)=O)C(C)(C)C CC1(CC(=O)NCC(C2CCOC2)NC(=O)CCCn2cccc2)CCCCC1 C#Cc1cc(F)c(C(=O)N(CCC)CC)cc1F.c1(C(=O)N)cncn1C(C)C C1(C(N2CCCC(CCC(=O)N)C2)=O)CCCC12CCC2.C1(SCC)(C)CC1 c1(C(C)Nc2cc(N3CCC(NC(CC)=O)CC3)ncn2)ccc(C)c(C)c1 c1(CNC(CNS(N)(=O)=O)=O)ncccc1.C1(CC=O)CC2CCC1O2.C c1(OC)ccc(N(C(=O)CCCCCO)CCC(=O)N2CC(N)C2)cc1OC N1(C(C(C)CO)=O)CCN(C(c2cnn(C3CCCC3)c2)=O)CC1CC(F)(F)F c1(OCC=C)cccnc1C(=O)N(CC(C)N(C)C(c1ccns1)=O)C N1(C(c2cncc(C)c2)=O)CCC(F)(C(=O)NCc2cccc(O)c2F)CC1 C1(C)(CC)CCC(NC(=O)CC(C)(C)N(C(=O)CC(C)C(F)F)C)CC1 c1(C(N2C(CNC(C3CC4C=CC3C4)=O)CC(OC)C2)=O)cnc2c[nH]nc2c1 C1(NC(c2n(CC)ccn2)=O)CCCCC1NC(=O)C(C)(C)OC C1(CNC(C2CC(CCOC)C2)=O)CN(C)CCN1Oc1ccccc1 Cc1nc2cccc(C(N3CCOCC3c3cn(CC(C)(C)O)nn3)=O)c2[nH]1 O=C1CC(CC(=O)NC(CC2CCOCC2)C(=O)NCCCCCF)C(=O)N1 c1(CCC)cc(C(=O)N(C(C)C(=O)NCC2CC(O)C2)C2CC2)n[nH]1 CCC(CC(=O)NC1CCC1C(=O)NCC1CCC(F)(F)C1)CC(C)C N1(C(Cc2c(C)non2)=O)CCCC(C(C)C(=O)N(CC(O)CO)C(C)C)C1 C(=O)(C1Cc2c(Cl)cccc21)NC(C1CN(C(C(C(C)C)SCC)=O)C1)C c1(NC(C(Cc2c(C)nc[nH]2)O)=O)cccc(NC(C23CCC(C2)C3)=O)c1 c1(NC(C2(CCCOC)CC2)=O)cc(O)ncn1.C1(N(CC)C)CCC1 CC1(C)C(CNC(c2cnc(C3CCC3)o2)=O)CCN1C(=O)C=CBr N1(C(c2c(CC)nc(C)o2)=O)CCC2(CCCC2)C1.C(=O)C(C)S(C)(=O)=O.N N1(C(CC2CC2)=O)CCC2(CC2)CC1C=O.CC(C)(O)C(F)(F)F.CC=O.N c1(C(N(C2CCN(C(=O)CCCNC(=O)O)C2)CC#C)=O)cn(C)nc1C C(CCN=C(NCc1cc2c(s1)CCC2)N1CCC2CCCCC2C1)OC C1CCN(C(=O)CC2CCC3CC3C2)C12CCC2.c1(COC)cc(C(=O)N)on1 C(=O)(C(CCC(C)C)NC(C1COCC(C)O1)=O)NCCC(C=C)(C)C C1(C(=O)NCC(C)(C)C)CC(O)CN1C(=O)C(F)n1ccnc1 c1(OC)cccc(C=CC(N2CCC(O)(C(=O)NCC)CC2)=O)c1.C(C)=O N1(C(CCCCC#C)=O)CCC2(CCC2)C(NC(c2ccc(Cl)nn2)=O)C1 Cc1cc(C(=O)NCCNC(c2ccccc2C2CCCC2)=O)c(O)c(C)c1 C1(C)C(=O)N1CC.C(C(C)(C)OCC(=O)N(C)C)NC(CC)=O C1(C(=O)NCCCCC2CN(C(C3C(=C)C3)=O)C2)CC2CCCN(C1)C2 Cc1cc(C(=O)NCC2CCN(CCC3CCS(=O)(=O)C3)C2)nn1C N1(C(CC2C(C)OCC2)=O)CCN2CCN(C(c3cc(C#N)c[nH]3)=O)CC2C1 c1(C(=O)NCCCN(C(c2cc(C)ccc2C)=O)CC)cnc2n[nH]c(C)c2c1 c1(C(C(=O)NCC2CC2C)N(C(C)C)Cc2cccnn2)noc2c1CCCC2 N1(c2n(CCCCCCO)ccn2)CCCCC1C1CCCO1 C1(CC(=O)N)CC2C=CC1C2.c1(C(N(C)CC)=O)cc(-c2ccn(C)n2)on1 C(CO)(C(O)CCC)NC(C1(CCC=C)CN(C(c2cn(C)c(=O)cn2)=O)C1)=O N1(C(C=C(C)C)=O)CC(NC(C2CCCC2(C)C)=O)C2(CCS(=O)(=O)CC2)C1 C1(CNC(CC(=O)N(C)C)=O)CC2(CCC2)C1.C(c1cocn1)=CC=O.N C1(C(N2C(CCC)CN(C(=O)Cn3nnc(C)n3)CC2)=O)CCn2cnnc2C1 N1(C(CCc2c(C)n(C)nc2)=O)CCN(C(C2CC(F)C2)=O)CC1CCO C(CCC(N)=O)(C(=O)NCC1CCCN1C(=O)C=Cc1ccco1)N(C)C N1(C(C2C(CC)CCC2)=O)CCCC(NC(=O)CC2CCCC(C#N)C2)CC1 C1(CC(=O)NCCCOCCNC(Cc2ccc(C)nc2)=O)OCCOC1(C)C C1(C)(CNC(C(N2CC(C)C2)C)=O)CN(C(=O)C(C)(C)C(N)=O)CCO1 c1(OCC)ccc(C(N2CCCC(NC(C3(C(C)C)CCCO3)=O)C2)=O)cc1Cl C1(N(C)C(=O)C2CC2)CCN(C(c2ccc(C3CC3)o2)=O)CC1 c1(C(C)C)cc(C(=O)NC(C(=O)NCCCCC2CCCC2)c2cccs2)no1 N1(C(C(C)N(C(CC=CC=C)=O)CC)=O)CCCC(F)(F)CC1 Cn1ncc2cc(CC(=O)NC3(C)CC3)ccc12.C(=O)(C(CC(F)F)N(C)C)N O=C1CCC(C(=O)N2CCC(NC(=O)Cc3c(F)cncc3Cl)C23CCC3)=NN1 CCC(C)C(C(=O)NC1CC(C)C1)c1ccccc1.C1(C)(C=O)CNC(=O)C1.N c1(C(=O)Nc2ccc(-c3ccc(C(=O)O)o3)cc2)ccnc2cc(Cl)ccc12 c1(C(=O)N)ccc2c(C)noc2n1.N1(C(C2(CC=C)COC2)=O)CCC2(CC2)C1 c1(CC)occ(C)c1C(N1CCCC(C2CCCN2C(=O)CC(=O)N(C)C)C1)=O C1(NC(CCc2ncc(C)[nH]2)=O)CCN(C(C23COCC(C2)C3)=O)CC1(C)C c1(C(N2CC(C(C)NC(=O)C=CS(C)(=O)=O)C2)=O)ccc2nc(CO)[nH]c2c1 C12(C(=O)NCc3ccc(CC)cc3)CC3CC1C2C3.C(=O)C(O)C(C)(C)C Cc1ccc(C(N2CC(CNC(=O)CN3CCOCC3=O)CC(C)C2)=O)c(N)n1 N1(C(C(C2CC2)OC)=O)CCC2(CCCN(C(=O)Cc3coc(C(F)F)n3)C2)C1 O=C(CCCC(F)(F)F)NCC(C1CCC1)NC(=O)CCCc1ccc(Cl)cc1 C(N=c1nc(N2CCN(C)C(=O)C2)c2c([nH]1)CCCC2)c1ccc(SC)c(C)c1 C1(C)(CCNC(C(C(C)C)n2cnnc2)=O)CCN(C(=O)C(F)(F)C2CC2)CC1 c1(CC(=O)N(C2CCN(C(c3[nH]ccc3C)=O)C2)CCC)c[nH]c2ccccc12 Cc1cc(C(N2CC3CC2C3CNC(=O)C(C)O)=O)nc(C)n1.C1CC1.C Cc1oc(CO)cc1C(=O)NC12CC(NC(C3CCC4CCC34)=O)(C1)C2 C(CC(C)(C)C)(C(=O)NC1CCCCC1NC(=O)CCCN1CCOCC1)OC C1(C(=O)NC(C2CCN(C(C(C=C)(F)F)=O)CC2)C)CC12CCCCC2 c1(CC)cc(C)[nH]c(=NCC(F)(F)C2CCN(C(C3C4C5CCC(C5)C34)=O)CC2)n1 c1(C(C)(C)C(=O)NCCC2CC(NC(=O)C)C2)c(F)cccc1F.C(N)=O C=CC(C)C(C)C(=O)N(CCCNC(c1cc(C)sc1SC)=O)CCO C(=O)(C1=CCC(C)(C)CC1)N1C(C(=O)N)CCC(C)C1.C(=O)(OC)NCC N1(C(CC(=O)NCC#C)=O)CC(O)CC1CC(=O)NC(c1nccn1C)C n1(C(C)C(=O)NC2CC2NC(=O)CCn2cnnn2)cc(Br)cn1 C(CC(C)C(=O)NCC12CC1CN(C(C1(OCC)CCCCC1)=O)C2)=CC N1(C(CNC(C)=O)=O)CCN(C(C2CN(C(C)C)C2)=O)CC1C1CCC1 C1(CC)CCCN1C(c1cc(C2CCC2)on1)=O.C1(OCC)C(C=O)C1C.N c1(CNCc2ccc(OCC)cc2)cccc(F)c1N C1(O)(CC)CCCN(C(c2csc(Br)c2)C(=O)NCCOCC2CC2)C1 CCCC(C(=O)NCC(C)(C)NC(C1(c2cc[nH]n2)CCC1)=O)NC(N)=O C(c1cccc(F)c1)=C(C(=O)N)F.C(=O)(C(C)C(=O)NC1(C)CCC1)OC O=C(CCc1ccccc1)C(=O)NCC(C1CC1)NC(=O)CCC1CCOC1 N1(c2cc(CC)nc(C)n2)CC2(CN(C(C3CSCC(=O)N3)=O)CC2CO)C1 C12(NC(=O)CC3CCCC3)CCN(C(c3cc(C4CC4)[nH]n3)=O)CCC1C2 C1(NC(c2c(OC)noc2C)=O)CN(C(c2cccc(CF)c2)=O)CCC1O c1(C(=O)NC2CC(C)(CNC(C(C)SC)=O)C2)ccc([N+](=O)[O-])cc1O C1(CNC(C(CC)(C)O)=O)CC2(CC2)CN1C(=O)Cc1ccc(O)cc1C c1(N2CCN(CC)CC2)nc(=NC(C)c2ccc[nH]2)[nH]c2ncn(CC)c12 N1(C(C2C(OC)CC2)=O)CCC2(CC1)CC(NC(c1cn3ccncc3n1)=O)C2 C1(O)(CC)CCN(C(=O)C(C)(C)CC)CC1.C1(C=O)(COCC)CC1.N Cc1cnc2n1CC(C(=O)NC1CN(C(c3ccc(F)c4occc34)=O)C1)CC2 c1(CC(=O)NC(C)CC2CN(C(C3CC34CC4)=O)C2)cnc2ncccn12 C1(O)(CCNC(C2C(C3C(C)C3)C2)=O)CCN(C(c2cnc(F)c(Cl)c2)=O)CC1 Cc1nc(C(C)(C)C)c(C(=O)NCCC2CCC2)s1.C1(C(=O)N)COCCO1 C1(C(N2C(C=C)CC2)=O)CCN(C(c2cc(C)c(N)cn2)=O)C(C)(C)C1 N1(C(c2ccc(=O)oc2)=O)CC2CN(C(C3CSC3)=O)CC2C1 n1(CCC)cc(Cl)c(C(=O)NC2CC(C)N(C(c3nccnc3N)=O)C2)n1 c1(C(=O)NC(C)CC2CN(C(=O)CCc3ncc[nH]3)C2)ccc2c(c1)N(C)CC2 C1(NC(C2CC(C(F)F)(OC)C2)=O)C=CCN(C(=O)Cn2ccnn2)C1.C c1(C(N2CC(C)C(NC(C3C(F)(F)C34CC4)=O)C2)=O)cc(Br)cnc1O c1(CC=O)ccc(F)c(F)c1.N1(C(c2cc(OC)ns2)=O)CCC(F)(C)C1.N CN1CCC(C(=O)NCC2(CCNC(c3cnc(Cl)s3)=O)CC2)CC1 N1(C(C=CCC2(NC(C(C3CCOC3)OC)=O)CCC2)=O)CCCC(C#N)C1 c1(OC)cc(C(=O)NCCNC(c2ccc(C(F)F)o2)=O)ccc1O C1(C)(OCC)CCN(C(=O)C(CC)NC(=O)C(C)(O)C2CCC2)CC1 Cc1nnc(O)c(C(N2CC3(C2)CN(C(c2c(N)cc(Cl)cc2Cl)=O)C3)=O)c1C S(=O)(=O)(c1c(C)nn(C)c1C)N1CCN(C(C2CN(CC)C(=O)C2)=O)CC1 Cc1cnn(C)c1C(=O)NC.C1C(C)CCN1C(=O)C(C1COC(C)(C)O1)O C1(CN(c2snc(CCOC)n2)C)CCN(C(c2ccc(C(N)=O)nc2)=O)CC1 c1(CN(CCCNC(CCC)=O)C(c2cnc(CC)s2)=O)cccnc1 N1(C(c2ccn(C(C)C)n2)=O)CCCC1C=CC(=O)N(C)CCc1cccnc1 C(=O)(C(C)(CC)C(=O)N1CCC(O)(CC)C1)OCC.c1(C(=O)N)cc[nH]n1 C(=O)(C(F)(CNC(c1csc(O)n1)=O)C(C)C)NC1CC(OCC)C1 C(=O)(CC(O)C(C)C)N(C(c1ccc(-c2ncc[nH]2)nc1)=O)C.C1(CCC)CC1 c1(C(=O)NC2(C)CCN(C(C(CC=C)(C)C)=O)C2)nc2ccccc2cc1Cl c1(C(N2C(C3CCN(C(CNS(N)(=O)=O)=O)C3)CCC2)=O)cccnc1O C(=O)(C1CCCc2n[nH]cc21)N1CCC(N(CCC)C(C2COC(=O)O2)=O)C1 N1(C(CSC(C)C)=O)CCC(NC(C2CC3CC3C2)=O)C(F)C1 C(CC(C)C(=O)NCC(CNC(c1ccc(=N)[nH]c1)=O)CO)=CC Cc1cccc(C(=O)N(CCN(C)C(c2n[nH]c(O)n2)=O)C(C)C)c1 C(=O)(C1=CCC(NC(C2CC=CC2)=O)C1)N1CC(n2ncc(C)c2)C1 CN1CC2CN(C(C3CCCC(NC(c4coc(C(N)=O)c4)=O)C3)=O)CC2C1 c1(C(N(C2CCN(C(=O)CC3CCCO3)CC2)CC)=O)cccc(F)c1C c1(COC)cccc(C(c2nnnn2-c2ccc(F)cc2)NC2CSC2)c1F C1(NC(c2ccc(SC)o2)=O)CCCN(C(c2cn(CCO)nn2)=O)CC1 CC1C(NC(C2CCC(=O)N2)=O)CCCN1C(c1cccc(C(F)F)c1)=O C1(N(c2ncn(C)n2)C(C(C)C)=O)CN(C(=O)Cc2sc(O)nc2O)CCC1F N(S(=O)(=O)N(C)C)CC=O.C1(CC=C)CN(C(=O)C)C1.CC(F)(F)F.C N1(C(C2C=CC(NC(c3c(OC)cc(I)cc3)=O)C2)=O)CCc2sccc2C1 N1(C(CC(=O)OCC)=O)CC2OCC(NC(=O)C(c3cncnc3)C)C2C1 N1(C(Cc2nc(C)sc2)=O)CC(C2CCCN(C(=O)Cn3ncn(C)c3=O)C2)C1 C1(C)(NC(C=C(COC)C)=O)CCN(C(c2cc(C)n(C3CC3)c2C)=O)CC1 c1(C(=O)N)cc(Cl)c(F)c(Cl)c1.C(C(=O)NCC#CC)(C1CCC1)OCC n1(CC)nc(C)c(C(N2CC(Cc3ccc(CO)cc3)C2)=O)c1C(=O)OC c1(C(=O)NC2CN(C(c3ccc(C)o3)=O)C(C)C2)cc(Cl)c(Br)cn1 CCC(C)(CC)C(=O)NCC1COCC1NC(c1ccnc(C)c1C)=O C1CN(C(c2c(C3CC3)cnn2C)=O)CC2CC12.CC(C)CCOC(C)C(=O)N C=CC1(O)CCN(C(C2CCN(C(=O)c3cccc(NC)c3)O2)=O)C1 N#Cc1cc(C(=O)NC2CC3(C2)CC(NC(=O)CN2CCCC2=O)C3)ccc1Br c1(C(=O)NC(CNC(c2ccnn2C2CCC2)=O)C2CCC2)ccccc1F C1(NC(C(CC=CC)CC)=O)CC2CCC(C1)N2C(c1cccnn1)=O CCC(C)C(C(=O)NCCCC(C)(C)CO)N(C)C(c1ccnnc1)=O N1(C(C2(C)CCN(C)C2)=O)CCC2(CC1)CC2C(=O)NC1(C)CCCC1 C=Cc1ccc(C(=O)NC(C2CCN(C(=O)CCS(N)(=O)=O)CC2)CO)cc1 N1(C(c2cn(C(C)C)nc2)=O)CC(C)N(C(=O)C=Cc2ccncc2)C(C)C1 c1(C(N(CCNC(C2C(COC)C2)=O)C)=O)ccc2c(c1)C(=O)CCN2 c1(C(=O)NC(CNC(C2N(C(=O)OC)CCC2)=O)CO)cc2ncccc2s1 CN1CCN(C(C2CCN(c3ccccc3Cl)C2)=O)CC12CC2 C1(C(N(C)CC2(C)CC2)=O)CSc2ccccc2O1.C1(CC=O)CCCOC1.N CCCC(C(=O)N(CC(C)(C)NC(c1ccc(C(C)C)nc1)=O)C)NC(N)=O N1(C(C(C)(CO)NC(c2n(COC)ncc2)=O)=O)CCC(F)(CF)CC1 N1(C(C(N)=O)=O)CCCC2C(CCCN2C(=O)CC2CC2)C1 CCC(C)CC(=O)NC1CCC(CNC(=O)CC2CN(C)CC2O)CC1 c1(CN2CC(COCCC)OCC2)cc(Br)cc(F)c1O C1(C=O)CC12CC(F)(F)C2.CC(C)CC.c1(CCC=CC(=O)N)ccccc1 C12(NC(c3ccc(Cl)s3)=O)CCCC1CN(C(c1ccc(F)c(CO)c1)=O)C2 C(=O)(CCC(CC)CCC)N1C(C(N2CC(C(=C)C)OCC2)=O)CCCC1 N1(C(c2c(C)cc(C)s2)=O)CCC(C(N2CC(C)C(C)C2C)=O)C1(C)C c1(OC)ccc(OCCC(=O)C2CC2)cc1.C1CCN(C(=O)C)C1.C(C)=O.N c1(N(CC(=O)NC2CC2)C(C2CC3(N)CC2C3)=O)nc2ccccc2s1 C(=O)(C1=C(Cl)CCC(C)C1)NCC1(O)CCN(C(C2CCN(OC)CC2)=O)C1 c1(C(=O)NCC2CCN(C(Cc3c(C)ocn3)=O)C2)cn(C)nc1C1CCC1 c1(C(N2CC=CC(NC(C3C(CCC)C3)=O)C2)=O)ccnc(F)c1OC C1(O)(CC(=O)N(C(C)C)CC)CCCCC1.C(=O)C(O)Cc1cn(C)cn1.N C(=O)(C(C)CC(C)(C)C)N1CC(F)CC(NC(c2c(OCC)cccc2)=O)C1 C1(NC(c2c(Br)cc(CCC)s2)=O)CCN(C(=O)CSC)CC1O CC1CN(C(c2cnn(C)n2)=O)CCN1C(c1c(N)cnn1C)=O N1(C(C(CC)SC)=O)CC2C3CCC(C2C1)N(C(c1c(C)cc(O)nc1C)=O)C3 Cc1ccsc1C1CCCN1C(=O)NCc1cnsn1 C=CC(C)(O)CC(=O)N1CCN(CC(=O)NC(C2(O)CCC2)C)CC1 C(=O)(C(C(C)(C)C)NC(=O)CC1CCN(C(c2c(O)cccc2Cl)=O)C1)NC CCC(C)(CNC(c1cc2occc2[nH]1)=O)C(=O)N(CC(C)(C)OC)C c1(OC)c(C(=O)NC2CC(F)CN(C(=O)C)C2)ccnc1Cl.c1cccc(Cl)c1.O CCC(CN(C)C)C(=O)N(C1CCC(NC(c2ccc(C)o2)=O)CC1)CC c1(OC)cccc(C=CC(=O)NC2CC(NC(c3ccc[n+]([O-])c3)=O)C2)c1 C1(C=O)C2CCC1CN(C(=O)CS(=O)(=O)N(C)C)C2.c1(OC)ccc(O)cc1.N c1(C(N(CCC)CCNC(=O)C(C)c2cccs2)=O)cc(C)c(C#N)[nH]1 N1(C(C23CC(NCc4ccc(F)cc4I)(C2)C3)=O)CCc2ccccc2C1 N1(C(C)=O)CCCC12CCN(C(=O)C(C)CCN)C2.C#CCOCCOCCO N1(C(C(CC)CC(C)C)C(=O)NCCCC2CC2)CCC2(C)C(F)(F)C2(C)C1 CC1CCN(C(C2(C)COCCO2)=O)CC1CC(=O)N(C)Cc1ccccn1 C1(C(=O)NCCC(C)N(C(=O)CS)C)CCc2cn(C)nc2C1.CCC(F)(F)F C12COC(C1)CC2.C(C=O)(C1CC1)OC.C(=O)CC.C(=O)C.C(C)=O.N CCC(F)C(=O)NC(C)CCCNC(=O)C(C1CCCOC1)OC c1(C(=O)OC)cc(C)c(NC(=O)C(C)Oc2cccc(C(C)C)c2)cn1 C(=O)(C(Cc1cn(CCCCF)nn1)NC(c1ccc(CN(C)C)s1)=O)OC C(=O)(CC(C)N(C)C)NC(C1CC(NC(C2CCOC2)=O)C1)C C1(C(N(CCC(C)NC(=O)C(C)C2(O)CCC2)C)=O)CCCC1F CCCCCC(C(=O)N(C1CCC(NC(c2cc(CO)on2)=O)CC1)C)C(C)C CCCCC(C)(F)C(=O)NCC(C)(C)CN(C(=O)CCn1cnc([N+](=O)[O-])c1)C c1(CC(=O)NC(CN(C(CC2CC(OCC)C2)=O)C)C)cnn(CC)c1 c1(C(N2CCC(N(CC(C)C)C(C3CCS3(=O)=O)=O)CC2)=O)nnc(O)cc1O CC(O)(CC(F)(F)F)C(=O)N1C2CCCC1CN(C(C1(F)CCCCC1)=O)C2 C1(NC(CC2CCC(C)(C)O2)=O)CC2CC1CC2C(=O)NC1(CCF)CC1 CC1CC(NC(c2coc(C(F)F)c2)=O)CCN1C(c1ccc(CCO)cc1)=O N1(Cc2c(C)c(-c3ccc(Cl)cc3)on2)CCC2(CC1)N=N2 CCC(O)C(C)(C)C(=O)NC1C2CC3C1C3C2C(=O)NC1(C)CCCC1C c1ccc(C)cc1F.C(C)(C(C(C)C)NC(=O)CO)NC(CCSCCC)=O C(=O)(C1=C(Cl)CCC1)NC(CC)(CNC(=O)C(C(C)C)OCC(C)C)CC c1(C(=O)NC2C=CC(C(=O)NCC#N)C2)ccc(Cl)cc1 C=C1CCN(C(=O)CC(=O)OCC)C(C(=O)NCC2(CCO)CC2)C1 Cc1ccc(Br)c(OCC(N2CCC2Cn2cc(-c3ccsc3)nn2)=O)c1 c1(C(N2CCC(NC(C3CC(CC)C3)=O)(CF)C2)=O)cc(F)c(C)cc1O N1(C(CN(C(=O)OC)C)=O)C(C(=O)NCC#CC2CC2)CC1C CCCCC(O)C(C)C(=O)NC(C1CC(NC(c2c(C)coc2CC)=O)C1)C CC1COCCC1NC(C1(CNC(c2cc[nH]c2C2CC2)=O)CCC1)=O CCC(CC(=O)NC1C2CC1N(C(c1nccc(C(F)(F)F)n1)=O)C2)C1CC1 C(=O)(C(C)(COC)COC)N1C(CNC(c2nc(CC)oc2)=O)CC1 C1(C(N2C(C3(NC(C4C(C(C)C)CCO4)=O)CC3)CCC2)=O)CC2(CCC2)C1 N1(C(c2ccn(CC)n2)=O)CCC(CNC(c2ccc(=N)[nH]n2)=O)CC1C CC12CCCC(C(=O)NCC3C4CCCC3N(C(=O)Cc3nccs3)C4)(CO1)C2 c1(CSCC)ocnc1C(N1CCC1C1CCCCC1)=O.C1(SC)C(=O)N1 c1(NC(N)=O)ccc(C(N2CCC(NC(=O)CC3CCCC3)C2)=O)cc1 N1(C(c2c(C)noc2)=O)CCOC(CNC(C2(c3ccno3)CCOCC2)=O)C1 C1(CC=O)CS(=O)(=O)CCN1C.C=C(C)CCNC(C1(SC)CCC1)=O.N Cc1cc(CC(=O)NC(C2CCCN2C(c2[nH]ccc2C)=O)C)c(C)s1 CC1CC(NC(=O)CC2OCCC2(C)C)CCN1C(=O)CSC.c1ccccc1 C1(NC(c2c(C(N)=O)nccn2)=O)CN(C(=O)C(Cl)=CCl)CC2(CCOCC2)C1 C(=O)(C1CCc2ccccc21)N1C2C(NC(C(C)N(C)C)=O)CC(CC2)C1 CC1(NC(C2(O)CCOCC2)=O)CCC2CC2C1.C1C(C)(C)Cn2cc(nn2)C1 C1(C(=O)NCCN(C(C(C)c2ccco2)=O)C2CCCC2)COC(=O)N1 C(CCCC(CO)NC(=O)C(C)C(F)(F)F)NC(c1cnc(C(=O)OC)s1)=O C(=O)(C(CC)C(=O)NC(C1(C(=O)NC)CC1)C)OCC.c1cccnc1 c1(C(=O)OCC)cnc(CC)[nH]c1=NC1CC(F)C1.C(=O)C=CC(N)=O.C CC(C)(C#CC(=O)NCC1CNC(=O)CO1)CNC(=O)C=Cc1ccsc1 CC(C)CC(C)(CO)NC(c1cc(CNC(C2CCC(=O)O2)=O)[nH]n1)=O C(=O)(CCCC(C)(C)C#N)N1CC2(CC(CC(N3C4CC(C)CC3CC4)=O)C2)C1 c1(C(=O)NCC(=C)CCNC(C2COCCC2(F)F)=O)c(C)nn2ccccc12 C1(NC(C(COC)C)=O)CC(NC2CC3CCC2C3)C12CCC2 c1(C(=O)NC2CC(CCNC(CCCC(N)=O)=O)C2)ccc2c(c1)CCCCS2 CC1CCN(C(c2ccc(O)cn2)=O)CC1NC(=O)C(O)C1CCC1 N1(C(C(CC)(CC)OC)=O)CC2CC(C(=O)N(C)CCc3ccncc3)C(C2)C1 CC(CCCNC(c1coc(C2CC2)n1)=O)NC(=O)CN(CC(C)(C)C)C c1(C(=O)N)ccc2c(c1)SCCN2.c1(C(=O)NCC2COCC2)cccc(F)c1 C(C(CCCC)NC(C1COCCN1C)=O)NC(C1(C)CC(=C)C1)=O CC(C)C(CNC(=O)Cc1cn[nH]c1)C(=O)NCC1CCC(C)CC1 c1(NC(C2C=CCN(C(=O)C3=CCOCC3)C2)=O)cccc2c1OCO2 C1(C)(CNC(C2(C(C)C)CC2)=O)CCCC1.c1cccc(F)n1.C(=O)C.N c1(C(=O)NC(CC#C)C(=O)NC(CO)CC#CC)ccn(C)c(=O)c1 CC(C)(C(=O)NC1CCCC1C(N1CC(N2CCNC2=O)C1)=O)n1cc(Cl)cn1 CN1CCCC(C(=O)NCC2CCCN2C(=O)COC(F)(F)F)C1 N1(C(C(C)(C)F)=O)CCN(C(c2ncccc2Cl)=O)C2(CC2)C1 Cc1noc(C)c1C(=O)NC1(C)CCCCC1.C(=O)C(F)(F)c1csc(=N)[nH]1 C1(NC(=O)CSc2n[nH]c(O)n2)CCCN(C(=O)CC2NC(=O)NC2=O)CC1 c1(OCC)cccc2c(=O)c(C(=O)N(CC(C)N(C(=O)C=CSC)C)C)c[nH]c12 c1(C(=O)NC2C(C)CN(C(C3CCCCO3)=O)C2)c(F)c(F)c(F)c(F)c1F c1(OC)ccc(C(=O)NC2CN(C(c3csc(C)n3)=O)CC2C(F)F)c(O)c1 C1(CC(=O)N(CC(C(=O)N(CC(C)(C)O)CC)C)C)CCCCC1O C12(NC(c3cc(C)no3)=O)CCCN(C(c3cccc4nncn34)=O)CC1C2 Cc1cc(C)c(C(=O)NC2CN(C(=O)C(O)C3CC3)CC2C2CC2)c(C)c1 C1N(C(=O)CCCC2CC2)CCC1(C)C.CC(C)(C(=O)NC)Oc1ccccc1 C(=O)(C#CC1CCCO1)NC1(C)CC(NC(=O)CCCCCn2cnnn2)C1 N1(C(c2cnn(C)c2Cl)=O)CCC2(CC(NC(C3CCN4CCOCC34)=O)C2)C1 C(=O)(N1CC(O)C(O)CO1)C1C(CC)CCN1C(=O)C(C)C(F)F C(C1c2ccsc2CCN1C(=O)C=CC1CCOCC1)NC(C(=O)NC1CC1)=O CCCC(N=c1[nH]c(=NCCn2ncnn2)c2ncccc2[nH]1)C1CCC1 Cc1cc(C(=O)NCC(=O)Nc2cccc(Cl)c2Cl)c(C)cc1Br N1(C(C(CCC)OC)=O)CC(CNC(c2cnc(O)c(Br)c2)=O)CC1(C)C c1(SC(C)C(=O)NNC(=O)c2cccc(Cl)c2)nnc2ccc(Br)cn12 N1(C(C=CCN(C)C(c2coc(CO)c2)=O)=O)CCC1(C)CCO C(=O)(CCCCC(F)(F)F)NCCC(C(C)C)NC(C1C(C)OC(C)C1C)=O NS(=O)(=O)CCCC(=O)N1CCCC(O)(CCNC(C2CCCC23CCC3)=O)C1 c1(C(=O)NCCC2CCCN(C(C)=O)CC2)ccc2ccccc2c1[N+](=O)[O-] C12(NC(c3c(C)nc(O)[nH]3)=O)CCC1CN(C(=O)C(C)n1cccn1)C2 c1(C(N(CC(NOC(C(=O)OC)(C)C)=O)C2CCC2)=O)nnn(C)c1CC c1(C(=O)NCC2C(NC(c3ncc(NC)nc3)=O)COC2)ccc2nccn2c1 N1(C(c2ccc(SC)s2)=O)CCC2CN(C(c3cc(C)ns3)=O)CCC2C1 C(=O)(C1CCCc2sc(=N)[nH]c21)NC1(C(=O)OC)COCC12CCC2 Cc1noc(C)c1C=CC(=O)NCC1CCN(C(C2CC(O)C2)=O)C1 C1(C(=O)NC)CCCCN1C(c1cc(C(C)(C)C)oc1C)C(=O)NCC(C)C c1(C(N2CC(OCCNC(C(COC)C)=O)C2)=O)nn(C)cc1N Cc1cccn2cc(C(N3CCC4C(C3)CN4C(=O)C=CC3CCCO3)=O)cc12 C=C1CCN(C(=O)NC2CC(C(=O)Nc3ccccc3)C2)C1 c1(CC)ccc(N(C)CCOCCN(C)C(=O)N(C)C)nc1CC C(CSC)(C(=O)NC(C(N1CC(O)(CO)C1)=O)C1(O)CCC1)OC N#Cc1cc(C(=O)NCC2CC(F)C2)c[nH]1.C(c1cccnc1)=C(C=O)F.C N1(C(C(CC)C(C)C)=O)CC2(C1)CN(C(=O)CN1CCCS1(=O)=O)CC2CO C1(c2nc(C3(CC)CC3)no2)(OCC)CCOC1 c1(-c2cn(C3CC(NC(CC=CCC)=O)C3)nn2)ccc(N)c(C)c1 Cn1cncc(C(=O)NCC2CN(C(c3ccc(F)cc3F)=O)CC23CC3)c1=O O=C1CCC(NC(N2CC(C(N3CCC(C(=O)N)CC3)=O)C2)=O)CN1.C1CC1 c1(NC(=O)NCc2c(C(=O)OC)c(C)on2)nc2c(C)cc(Br)cc2s1 C1(C(N2CCC(CC=C)(NC(=O)CCC=C(C)C)CC2)=O)CCc2c[nH]nc2C1 Cc1ccc2cc(C(N3CCC(C)C(NC(=O)C(F)C(C)(C)O)C3C)=O)[nH]c2c1 c1(OC)ccc(CC(N2CCC3(CC2)CN(C)C3)C)c([N+](=O)[O-])c1 c1(C(=O)Nc2cc(OC)nc(OC)c2)nnn2c1CN(C(=O)C(C)(F)F)CC2 C12(CC(F)(F)C1)C(=O)N2.Cc1snnc1C(=O)NCCSCC(C)C Cc1cc(F)cc(C)c1C(=O)NC(C)C(C)(C)C.c1(CC=O)csc(=N)[nH]1 c1(OC)ccc2cc(C(=O)NC(c3cn(CCC(F)(F)Cl)nn3)C)ccc2c1 C1(C=O)CCS(=O)(=O)C(C)C1.c1(CC(=O)N(CCOC)CC)ccon1 Cn1oc(C(=O)NCC)cc1=O.c1(C=O)cnc(S)n1C1CC1.C(C)(C)C C(=O)(C(F)(F)C(O)C1CC1)N(C)CC1CCCCN1C(C1CCC2CC2C1)=O N1(C(C(C)OCCCCCC)=O)CCCC(NC(C2(C)CCSCC2)=O)C1C CCC(C)CC(=O)C(=O)NC1CC(C(=O)NCc2cnccc2Cl)C1(C)C c1(CNC(CCCC)=O)ccc(CNC(=O)C(F)(F)C2(OC)CCCC2)cc1F C#CC1(C(=O)NOC(C)C(=O)OC)CCN(C(c2nc(Cl)cs2)=O)C1 C1(NC(C2C(C=C)C2)=O)CN(C(=O)C(=Cc2c[nH]cn2)F)C(CC)(CC)C1 CCC(CC)(C(=O)N1CC2CC(NC(c3ccncc3OC(C)C)=O)C1C2)OC C1(CS(=O)(=O)NC2C(C)(C)COC2)CC2COCC2O1 C1(CNC(c2nc(CCC)sc2)=O)(CO)CCCN(C(=O)CCCSC)C1 c1(C(c2nnnn2Cc2ccccc2)NC2CCC(O)CC2)cc(O)ncc1F N1(C(C(C)C2CC2)=O)CCOC(CNC(C2C3CCC2(c2ccccc2)C3)=O)C1 N1(C(CC(C)N(C)C)=O)CC(n2cc(C(C3CCCOC3)C)nn2)CCC1(C)C N1(C(CCCOC(C)C)=O)CCC2CC2(C(=O)N2CC(O)CCO2)CC1 C(=O)(C1=C(c2cscn2)N(C)C(=S)NC1c1nn(CC)nc1Br)OCC C1(NC(C(F)=CCC)=O)CN(C(c2snnc2C(C)C)=O)CC1C C1(C(=O)NC2CN(CC)CC2C)CCN(C(c2cc(Cl)cn2C)=O)C12CCC2 c1(N2CC=C(C)CC2)nc(NC2CCCc3c[nH]nc32)nc2c1CC(C)CC2 c1(C(=O)NC2CCOC2C2CC2)coc2c1CN(C(c1ncc(F)cn1)=O)C2 N1(C(c2n(CCC)ccc2)=O)CC(CC(=O)NC2CC=CCC2C)C2(CC2)C1 C(=O)(CCCCC(C)=O)NC(CSC)(C)C(=O)NC(c1nncn1C)C c1(C(=O)NCC(CC)C)cc(C)c(F)c(C)c1.C(c1cncnc1O)=CC=O.N N1(C(CCC=C=C)=O)CC2(CC(NC(=O)C(C)NC(=O)NC)CO2)C1 c1(CC)ccc(C(=O)NC(C)C(C)NC(c2cc(O)cc(O)n2)=O)cc1F N1(C(CCc2cccc(OC)c2)=O)CC(C)CCC1CNC(c1ccnn1C)=O N1(C(C(F)OC)=O)CCCC(C2CN(C(c3cc[nH]c3)=O)C2)C1 CC1CN(C(=O)Cn2cnnc2O)CCC1N(C)C(C1CCN1C1CCCC1)=O c1(SCC(=O)NCC2N(C(C(OC)OC)=O)CCOC2)ccc(F)c(F)c1 C(=O)(CC(C)(C)C1CC1)N.C(=O)(CCc1ccoc1)NCCN(C(CC)C)C C=CCC(CC=C)C(=O)NC1CN(C(c2c[nH]c3ccncc23)=O)CC1N=[N+]=[N-] C1(O)(CC)CCN(C(=O)C=CC(C)(C)NC(=O)CCc2ccc(C)o2)C1 c1(C(=O)NCCOCCNC(c2ccc(OC)cc2)=O)cccc2cncn12 C(C)(C1CCCCC1)=CC(=O)NCC(C)(C)NC(CCC(=O)OC)=O c1(C(=O)NC(C)CN(C)C(c2nncs2)=O)ccc(N)c(F)c1Br C#Cc1c[nH]nc1C(N1CC(NC(=O)CC2CC3CC3C2)CC1CO)=O c1(C(N2CC(CNC(c3c(CC)n[nH]c3)=O)C3C2C3)=O)nc2sccn2c1C CC(C)CC(O)C(=O)NCC(C1CC1)NC(=O)CO.c1ccc(F)c(F)c1 N1(C(C23N(C(CCc4n(C)ncc4)=O)CCC2C3)=O)CCNC(=O)CC1 N1(C(CCC=CC)=O)C2CCC(C2)C1CNC(C1C(C#N)C1(C)C)=O c1(C(N(C(CN(C(c2c(SC)cn(C)n2)=O)C)C)C)=O)n[nH]c2cc(C)ccc12 C=C(C)CC(C(=O)NC1CCCCN1C)NC(=O)C=CCN1CCC1 C(=O)(C1CCc2ccccc21)NCC(C(C)C)NC(c1cnc(N(C)C)s1)=O Cc1nc(C)c(CNC(=O)CCOCCCNC(C2(F)CCOCC2)=O)o1 CC(N=c1nc2ncn(C)c2c(NCC2(CC3CC3)CC2)[nH]1)c1n[nH]c(=N)s1 C(=O)(CCCCC(C)(C)C)NC1C(CNC(C2C(C(=C)C)OCC2)=O)CC1 C=CC1(C(=O)NC2C(C)(C)C2(C)C)CCN(C(=O)CC2COCC2O)C1 C1(CN=C(NC(C=C)C)NC2CC(c3ccccc3)C2)CCS(=O)(=O)C1(C)C CC(C)(C)CCCCN=c1[nH]c(N2Cc3ncsc3C2)nc2cccc(F)c12 C1(C(CO)NC(C(CO)OC)=O)CCN(C(=O)CC2CNC(=O)O2)CC1 C1(CCC)CN(C(=O)Cc2cnc(C)o2)CCN1C(c1coc(Cl)n1)=O c1(C(=O)NC2CCN(C(=O)Cc3nc(C4CC4)cs3)CC2)cc2c(o1)CCCC2 N1(C(CC2CC(SC)C2)=O)CCCC1C1CCN(C(c2n[nH]c(C)n2)=O)C1 N1(C(c2cnc(C)n2C)=O)C(C)C2CC1C2NC(c1sccc1C1CC1)=O CCC(C(=O)NC1CCCC1N(C)C)NC(=O)CSCC(F)F C1CC2CC1CN2C(c1cnc(S)n1C1CC1)=O.C1(OCC(=O)N)CCCCC1 C1(CC(=O)O)CC2(CCN(C(=O)NCC3C4CCC(F)(F)C34)C2)C1 C1(CNC(CC(CC)O)=O)CN(C(=O)CCC2CC2(Cl)Cl)CCC12CCOC2 C12(C(N(C3CCCC3)CC)=O)COCC(C1)C2.c1(CSCC=O)cccs1 N1(Cc2n(CC#C)ccc2)CCC2CC(C(=O)NC3CCS(=O)(=O)C3)C2C1 C1(C(=O)NC(C=C)CO)CCC(NS(=O)(=O)CC2CCC2)C1 c1(CC)ncsc1C(=O)N(CC(C)NC(C1(COC)C=CCC1)=O)C c1(C(=O)NCCC(=C)CNC(=O)CCOC)ccc(OC)cc1N N1(c2c(C)c(NCc3nc(C)c(C)[nH]3)ncn2)CC2OCCN(C)C2C1 c1(C(N(C)CC2N(C(C(C=CC)O)=O)CCCC2)=O)ccc(C)c2ncccc12 C1(NC(CCC2(C)CN(C(CNC(CN(C)C)=O)=O)C2)=O)CCC2(CCCC2)C1 N1(C(C=Cc2n(C)ncc2)=O)CCN(C(=O)CC2CCCOC2)CC1CCO C1(C(=O)NCCOCCF)CCOCCN1C(=O)Cc1cnsc1 c1(CNC(C2(NC(C(C3CCOCC3)C)=O)CSC2)=O)cc(F)ccc1F C1(c2nnnn2C2COC2)(NCC2(C)CSC2)CCC2(CCOCC2)C1 c1(CCC(=O)NCC(C)C2CCC2)ccc(CO)cc1.c1(C=O)cc(Cl)no1.N c1(CNC(CCC(C)(C)F)=O)nnc2n1CCN(C(C1NC(=O)CC1C)=O)C2 CCC(C)(C)C(=O)N1CC(O)CC1C(N1CCC(Cc2ccc(Br)cc2)C1)=O C1(NC(c2cc(C)[nH]c2)=O)COCCN(C(C2CCC(N=[N+]=[N-])C2)=O)C1 N1(C(C(CC)=CCCC)=O)CCCC12CCN(C(=O)C(C)Cn1cccn1)C2 c1(CC(N2C(CNC(c3cc(CC)no3)=O)CCC2)=O)ccc(Br)nc1 c1(SC)cc(C)ccc1C(N1CCC(C(C)C)CC1)=O.c1(CC(=O)N)cocn1 CC(C)(CC(F)F)C(=O)N1CCC(CCC(=O)NCC2CC(C(N)=O)=NO2)C1 N1(C(c2scc(C)c2)C(=O)NCC2CCOC2)CCC(N(C)C(C)C)CC1 CC#CCCC(=O)NCC1COC(CNC(c2ccc(-c3cnco3)cc2)=O)C1 N1(C(=O)NC2CCC(C)(C(C)=O)C2(C)C)CCN(S(C)(=N)=O)CC1 C1(NC(CCC(=O)NCCC)=O)(C)CCCCC1C.C1(O)(C(=O)N)CCCCC1 O(NC(=O)C=Cc1cc[nH]n1)CC(=O)NC(C1CCCCO1)CC C(c1ccccc1)=CC(C)C(=O)NCCC(C)NC(=O)CCCc1nncn1C N1(C(CCOC)=O)CCN(C(C2CC3(CCC3)CO2)=O)C2CS(=O)(=O)CC12 c1(C(=O)NC(C)(C)CCNC(=O)CCOC2COC2)ccc2ccoc2c1 c1(OC)cc(C)cc(C(=O)NC(CO)C(C)NC(=O)C(C)(C)C)c1C c1(C(N(CCCCN(C(Cn2c(C)cc(C)n2)=O)C)C)=O)ncncc1C#N c1(C(N(CC(C)NC(=O)C(C)(C)CCOC)CC)=O)cnn2ccccc12.O N1(C(C2C(C)(C)COCC2)=O)CC2CC(NC(=O)C(F)=CC3CC3)C(C2)C1 N1(C(CC(CCOC(=O)NC(C)(C)C)O)=O)CCCC(COC)C1 C(=O)(C(C)CC(F)(F)F)N1CCC(C)(C)C1.Cc1cc(C(F)(F)F)sc1C(=O)N C1(NC(C2(OCC)CCCOC2)=O)CN(C(C2(SCC)CC2)=O)CCC1F N1(C(CCSC)=O)CCC12CN(C(=O)CC(c1ccccc1)NC(N)=O)C2 c1(C(=O)NC2(CN(C)C(c3cn(CCCF)nn3)=O)CC2)cccc2cnsc12 N1(C(C(NOC)=O)=O)CCCC12CCN(C(=O)CCC(=O)N(C)C)CC2 CS(=O)(=O)c1ccc(NCC(=O)Nc2ccccc2O)c(S(C)(=O)=O)c1 c1(C2CCCN(C(c3cc(Br)ccc3Cl)=O)C2)c[nH]c2ncccc12 c1(C2CCN(C(C(N3CCC(NC(C)=O)C3)=O)=O)C2)cccc(C(C)C)c1 CC(C)CC(CNC(=O)C(=O)NC1CC1)NC(c1sccc1C(C)C)=O C1(C2CCC2)(C(=O)NCCCN(C(=O)CN2CC3CC3C2)C)CCOCC1 C1(C(=O)NC2CC(NC(c3n4c(nn3)SC(=C)C4)=O)C2)Cc2cccc(C)c2O1 N1(C(C(CC=C)C)=O)CCN(C(C2CCN(OC)CC2)=O)C2CCCC12 C(=O)CCCCS(C)(=O)=O.c1(C(=O)OCC)ccc(C)c(O)n1.C(C)(C)C N1(C(CCc2cnc(C)o2)=O)CCCN(C(c2cc3cc[nH]c3cn2)=O)C(C)C1 N1(C(C(C)Oc2ccc(F)cc2)=O)CC2CC1CN2C(=O)C(F)(F)F n1(C(C)C)ccc(C(=O)NC2(C)CN(C(C3CCCN3c3ncccn3)=O)C2)c1 CCC(CC(=O)NCC(=O)OCCC(C)(C)C(=O)OC(C)(C)C)C(C)C C1(C)CC2(CCC2)C1.c1(CNC(C=CC=CC)=O)cc(C=O)on1.N c1(C(N2CCC(NC(CCNC(=O)C=CCl)=O)CC2)=O)ccc([N+](=O)[O-])o1 c1(C(=O)NC(CNC(C(CC)C(C)O)=O)C)cncc2ccccc12 c1(C(=O)NCc2ccc(O)cc2)ccc2nc[nH]c2n1 N1(C(=O)Cc2cccc(F)c2)CCCC2(CCN(C(c3cc(Cl)no3)=O)C2)C1 N1(C(CC(C(=C)C)OCC)=O)CCCCC2(CCN(CC3CCC3)C2)C1 C12(CC(=O)Nc3ccc(OC(F)F)c(C(F)(F)F)c3)CC3CC(CC(C3)C1)C2 c1(CC)nc(C)c(CC(=O)NC(C)C(C)(C)NC(=O)C(F)F)c(C)n1 CC1CN(C(c2ccnnc2)=O)CCN(C(=O)C(C2CCCCCC2)F)C1 C1(CC=O)CN2CCN1CC2.Cc1nc(CC(=O)NCC2(C)CCC2)oc1C.N Nc1cc(F)cnc1C(N1CCOC(CC)C1)=O.C1(C=O)CN(S(N)(=O)=O)C1.N C#CCC(C)(C)C(=O)NC(C1CC=CCC1)C(=O)NCC1(O)CCCCC1 N1(C(C23C(C)(C)OCC2C3)=O)CC(NC(=O)Cn2cnnn2)C2(CCOCC2)C1 N1(C(C2CC(SC)C2)=O)C(C(=O)NC2CN3CCC2C3)CCC1C(C)C c1(NC(c2c(CC)cccn2)c2nnnn2C(C)C)ccc2nccnc2c1Br CC1CN(C(C2(C)CC(C3CC3)=NO2)=O)CC2(CCN(C(c3cscn3)=O)C2)O1 c1(CNC(C(C)n2cncn2)=O)ccc2c(c1)CN(C(c1cc(C#N)no1)=O)C2 Cc1cc2ccccc2cc1C(=O)NCC1CC1.C1(C=O)NC(=O)OC1(C)C.N O=C1CCC(CC(=O)NC(CC2CC2)C(=O)NCc2cncc(O)c2)CN1 N1(C(C2(CC)CCC2)=O)CCCC(O)(CN(C(=O)C)C)C1.c1ccc(O)cc1 C(C(=O)NNc1ccc(F)cc1Sc1ccccc1-n1ncc(C#N)c1N)OC C1(NC(C(C(C)C)C)=O)CC2(C1)CCC2.c1(C=O)cccc(CS(N)(=O)=O)c1 C1(C(N2C(C)CC(NC(CCc3c(C)noc3C)=O)C2)=O)CCCC12CCC2 N1(C(C(=O)NCC(C(=O)OC)OC)=O)CCOC(C)(CCSC)C1 c1(C(N2CC(NC(C34OC(C)C(C3)C4)=O)C(C)CC2)=O)coc(S(C)(=O)=O)c1 CC1=C(C(=O)NCCC(O)CNC(C2CCN(C)C(=O)C2)=O)CCCC1 N1(C(c2c(C)ncnc2)=O)CC(O)(C2(C)CC2)C1.C1(=CC(=O)N)CCSCC1 c1(OC)cccc2c(CC(=O)NCC(=O)Cc3ccc([N+](=O)[O-])cc3)coc12 N1(C(C2CC(=C)C2)=O)CCC(CNC(c2nc(Br)c[nH]2)=O)C(C)C1 c1(OC)ccc(C(C)C(=O)NCCCC(C)NC(=O)C(C)C#N)cc1 CC(C)(C)CCNC(=O)COCCO.n1(CC(=O)N)cc(C2CC2)nn1 C(C(C)(C)C(=O)NC(C)Cc1cn[nH]c1)N(C(CCC1CC(C)C1)=O)C N1(C(CC(C=C)C)=O)CC(C2CCN(C(=O)Cc3ccc(C(C)=O)cc3)C2)C1 C12(NC(c3cc(OC)cc(C)c3)=O)CCCN(C(=O)CCO)CC1C2.C1CC1 C1(NC(c2cc(CCC)[nH]n2)=O)CC(C)CN(C(C2(C#N)CC=CC2)=O)C1 N1(C(c2cc(Cl)c[nH]2)=O)CCC2CCCC12C(=O)NC1CCSCC1 N1(C(C2C(C(N)=O)COC2)=O)CCCC(CNC(=O)CCn2ccnc2)C1 c1(C(=O)OC)cc(NC(=O)N(C2COCC2O)C)cc(C2CC2)c1 C1(C(N2C(CNC(C3CCCC(=O)O3)=O)CCC2)=O)CSc2ccccc2O1 Cc1ccncc1C=CC(=O)NC1CCN(C(c2cc[nH]c2C(C)C)=O)CC1F C(CNC(=O)Cc1cncs1)(C(=O)N1CC(n2ccnc2)C1)N(C)C C1(NC(C2CCCO2)=O)C2CC(O)C1N(C(=O)CCc1cnco1)C2 C1(C(=O)NC2CC3(C(NC(CCc4c(C)cccc4)=O)C3)C2)CC12CC(F)(F)C2 N1(C(C2CC2)=O)CCCC2(CCN(C(=O)CC3C(=O)ON=C3C)C2)C1.COC c1(OC)cc(C)ccc1C(=O)NCC1CCC1.C1(C=O)C2CC2C2CC12.N c1(C(=O)NC(CC(=C)C)C(=O)NCC(O)COCC)ccc(C#N)c(C)n1 C=CCCCCCC(=O)N1CCC(C(C)C(=O)NC2COCC2N=[N+]=[N-])CC1 C1(NC(C=C(CCC)CCC)=O)CN(C(=O)C(C2CCCCC2)O)CCC1C C1(OC)CCN(C(C2CC2(Br)C(=O)O)=O)CC1.c12ccccc1O2 C1(NC(=O)C(C2CC2)C2CC2)COCCN(C(c2ccc(C(F)(F)F)o2)=O)C1 C1(NC(c2cn[nH]c2)=O)CCN(C(=O)C(c2ccccc2)=O)C1c1ccccc1 C(=O)(C(O)C(F)(F)F)N1CCN(C2CCCN(C(c3c(C)ccn3C)=O)C2)CC1 C1(N(C)C(C2CCOC2)=O)CCC(NC(c2cnc(C3CCC3)o2)=O)CC1 N1(C(Cc2cc(C(C)C)no2)=O)CC2(CC(NC(=O)Cc3cnn(C)c3)CO2)C1 CC1CC(CC(=O)NCCn2ccnn2)CN1C(=O)Cn1ccc(CN)n1 c1(C(=O)N)ccc(Cl)cc1-c1ccsc1.C=CC(O)C(=O)NC(C)(C)C1CC1 CCCCCCCCC(C)C(=O)NCCN(C(=O)C(C)C)CCOC c1(C(=O)OC)ccc2c(c1)C(C(=O)Nc1nc(C(N)=O)cs1)CO2 Cn1ccc2cc(C(N3CCN(C(c4nnn(C(C)(C)C)n4)=O)CC3)=O)ccc12 c1(C(=O)NC(CNC(CCC=CC)=O)(C)C)nn(C2CC2)cc1OC(F)F N1(C(C(c2ccc(CC)s2)=O)=O)CCOCC(CNC(=O)C(C)C(C)(F)F)C1 C12(CNC(c3c(C)cn(C)n3)=O)CCCC1N(C(=O)Cc1c[nH]nc1O)CCC2 c1(CNC(C2C(O)CCN2C(c2ncccn2)=O)=O)cc(F)cc(F)c1 n1(CC)nc(C(=O)NCc2ccsc2C(=O)N(C)CCF)cc1C CCC(Cc1cn(C(C)CN(CCCN(C)C)C)nn1)C(=O)O.c1ccccc1 N1(C(C(C)OCC2CC2)=O)CCCC(C)(C)C1C(=O)NCCCC(N)=O C(=O)(C1=CCC(C)CC1)N1CC(CC)C(NC(=O)C(C)CC(F)(F)F)CC1 Cc1cc(NC(C2CCCN(S(=O)(=O)C(F)(F)F)CC2)=O)cnc1Br CC(C(=O)N1CC(C)(C)CC1C)S(C)(=O)=O.N1(CCC=O)C(=O)CCC1=O Cc1nc(C(N2CC(O)(C(F)C(=O)NC(C)(C)C(O)CO)C2)=O)sc1C C1(NC(N2CCN(C(C3(O)CCCCC3)=O)CC2)=O)CCCC2(CCC2)C1 N1(C(C(=CC2CCCO2)C)=O)CC2(C1)CN(C(=O)CCCc1ccc(N)cc1)C2 Nc1c(C(N2CCC(NC(C3CC(O)C3)=O)CC2C2CC2)=O)cc(Cl)cc1F N1(C(C2CN(C(C)=O)C2)=O)CC(C(=O)NCc2ncccc2Cl)OC(C)C1 c1(C(N2CCC(N(C(C(C)c3cccs3)=O)C)CC2)=O)ccc(N)cc1Cl CC1CC2(CC(C(=O)NCc3ccc(CC)cc3)C2)C1.c1(C(=O)N)cnsn1 CN=c1[nH]cc(C(=O)NCCCN(C(=O)C(c2ccc(Cl)s2)C)C)o1 c1(C(=O)NC(CCOCC)C(=O)N(C2CN(C)CC2O)C)ccc2c(c1)CC2 C(=O)(C1=CCCC(C)(C)C1)N1CC(O)(CNC(C(CC=C)CC)=O)C1 CC1CN(c2ccc(CNC(=O)C(F)(F)CC3CCNCC3)cn2)CCO1 Cc1ccnc(C(=O)NCC(C)NC(C2CSCN2C(C2CCC2)=O)=O)c1 c1(C(N2C(CC)CCC2)=O)cnc(C(F)(F)F)cn1.C(C)(C=O)NC(C)=O.N CCC(C)(CO)C(=O)N1CCOCC(NC(c2ccc(OC)c(F)c2)=O)C1 c1(CNC2CCC(CC(=O)NCC(C)OC)CC2)ccc2cc[nH]c2c1 C(=O)(CC(C)C(F)F)N1C(C(=O)N(CCN=[N+]=[N-])C)(COC)C=CC1 C12(C(N3CCC(C(C)O)CC3)=O)COCC1CN(C(C1CCC(C)O1)=O)C2 C1(NC(c2cc(C)c(C)o2)=O)CCCN(C(c2ccc(C3CC3)cc2)=O)C1C c1(C(N2CC(NC(C3CNC(=O)N3)=O)CC(C)C2)=O)c(F)ccc(F)c1Br c1(SCCC(CC)C)ccc(-c2cccc(C(=O)N(C)C)c2)cc1C C#CC1(C(N2CC=CCC(C)(C)C2)=O)CCN(C(=O)C(C)C(O)CC)CC1 C(C)(C)(C(=O)NC(C)C(c1ccccc1)NC(=O)CN1CCNC1=O)SC C1(C(N2CC(CNC(C)=O)C(C)C2)=O)CC2(CC2)C1.C(C)(C)C.C=O.N c1(CCC(=O)NCCN(C(=O)CC2(C)CCOC2)CC)n[nH]c(=N)s1 CC(CNC(=O)CC(C1CC1)NC(=O)CC1=CCCC1)CC(F)(F)F c1(C(N(CCCCCCNC(=O)CC2CCCCO2)C)=O)ncc([N+](=O)[O-])n1C N(C1CCCn2cnnc21)C(C1N(C(CN(C(C(C)C)=O)C)=O)CC(O)C1)=O N1(C(C(C)OCC=C)=O)CC2(CC(NC(=O)CN(C)CCOC)CO2)C1 C1(C(=O)NC(C)Cn2cccn2)CN(C(=O)C(N)=O)CC(C)(C)C1 CCCCC(C(=O)NC(C)CC(C)NC(=O)C(C)OC)N(C)C C(=O)(C1CCc2c(Cl)cccc21)N1CCC(CNC(=O)OC(C)(C)C)C1(C)C CCCCC(C)(F)C(=O)NC1CCCCC1NC(c1cnnn1CC)=O C(=O)(C1=CCC(C)CC1)NCc1cc(C(N2C(CCC)C(C)CCC2)=O)n(C)n1 C#CCCCCCC(=O)NC(C)(C)C1CC1.n1(CC=O)cc([N+](=O)[O-])c(C)n1.N c1(C2(C(N3CCC(c4cccs4)CC3)=O)CC2)ccc(-c2csc(CO)c2)cc1 CC1(C)CC(NC(=O)C(F)CC2CCOC2)CCN(C(=O)C=CCF)C1 CC(C)CCCC(=O)NC1CCC(F)(CNC(c2conc2C(C)C)=O)C1 c1(C(=O)NC2C(C)CCN(C(c3c(C)ocn3)=O)C2)cnc(O)n(C)c1=O Cc1ncccc1CNC(=O)CCOCCNC(C1CCC1(F)F)=O c1(C(N2CC(CNC(C(C(C)C)OCC)=O)C(O)C2)=O)cc(F)c(F)cc1N N1(C(C2C(CCC)C2)=O)CCC2CN(C(=O)CC(C)(C)C(F)F)CC12 C1(NC(c2ncc(Cl)cn2)=O)CCN(C(c2c(F)cccc2I)=O)CC1F N1(C(=O)OC(C)(C)C)CCC(N(C(=O)C(O)CCO)CCO)CC1C1CC1 C1(C)(CNC(=O)OC(C)(C)C)CCCC1.C1CN(C(N)=O)C1.C=O.N Cc1cccc(C(N2CC(NC(=O)C(c3c(C)nn(C)c3C)=O)CC2C)=O)c1Cl c1(-n2cc(C(=O)NC(CC)CNC(=O)Cc3cc[nH]c3)nn2)ccccc1Cl c1(C(=O)NCCCNC(CC(C=C)C)=O)cc2ccccc2cc1NC(C)=O N1(C(CC2CC(=C)C2)=O)CC2CCN(C(c3cnc(C)nc3C)=O)CC12 c1(C(=O)N)cccnc1C(F)F.CC1(C)CN(CC(=O)NC2(C)CCCC2)C1 c1(C(N2CCC(OC)(CNC(c3ocnc3C)=O)C2)=O)cc(C#N)c(C)cn1 C(=O)(CCCCNC(N)=O)N(C)CC1CCCN1C(=O)Cc1cnn(C)c1 C1(C(=O)NC2(C#C)CC2)(C)CN(C(=O)C(F)=C(C)C)C1.C(C)(=O)O C1(OCC(=O)NC2CCCC2CNC(C2COC2)=O)CC(F)(F)C1.C N1(C(COC(CNC(CCCOCC)=O)(C)C)=O)CC2(CCC(=O)NC2)C1 C(=O)(CCCCC(C)C)N.N1(C(C=CCN(CC)CC)=O)CCC(O)(C)C1 c1(C(N2CCC3(C2)CC3)=O)ccc(S(C)(=O)=O)s1.CC1(C)C(C=O)C1(F)F.N c1(OC)cc(C)nn1-c1nnc(Sc2c(C)noc2C2CC2)o1 c1(C(N(CCC)CCNC(C2CCCN2C(C)=O)=O)=O)c(C)cccc1C C(=O)(C(C)(C)C1CCN(C(=O)CC2CCCC2)C1)NC1(CSC)CC1 c1(C(=O)NCC2N(C(CCC(CC)C)=O)CC2)cc2c(nc1O)CCSC2 c1(SCC)cc(C(C)C)nc2ncnn12.c12cn(nn1)CC(=O)NC2C O=S1(=O)CCCC2(CCN2c2ncnc3ccc(I)cc23)C1 Cc1cccc(OCC(=O)NCCC(C)(C)CNC(C2CCN(C)C2=O)=O)c1 c1(C(=O)NC2C(C(=O)NC3C(CCC)CCCC3)OCC2)ccc(C)c(C)c1 c1(CN2CCN(C(c3cccc(Br)c3)C)CC2)ncc(Br)cc1Cl CN1CCS(=O)(=O)CC1CC(N1CCCCCC1CNC(=O)Cc1cnns1)=O c1(C(C=O)C)ccncc1C.C(C)(C(=O)N(C)CCOCCC)N(C(C)=O)C.N c1(N2Cc3c(nn(C)c3N)C2)nc2c(c(=NCCCS(C)(=O)=O)[nH]1)CCCC2 N1(C(C(C)(C)C2CC2)=O)CC2(C)CN(C(c3ccn(CC#N)n3)=O)CC2(C)C1 N1(C(=O)Nc2ccc(OCF)cn2)CCS(=O)(=O)c2ncc(Br)cc21 c1(C(=O)NC2CC(C)N(C(=O)CCCCC#N)CC2)ccnc2c1CCO2 c1(C(N2C(CC(=O)NC(C(C)F)C)CC2)=O)ncn2c1CCC2 Cc1cc(F)sc1C(=O)N(C1CCCCC1NC(c1ccon1)=O)C.N(C)C.C Cn1cncc1CCNC(=O)C(C1CCOC1)N(C(=O)CCC)C.C1CC1 C(=O)(C1CCCn2nccc21)NCC(CCNC(C=Cc1cn(C)nn1)=O)O N1(C(c2c(OC)ccs2)=O)CCCC1(C)C(=O)NCC(O)CC1CCCC1 c1(CCC(=O)N(CCF)CC)ccc(C)cc1-n1cc(CC(O)C(C)C)nn1 CCC(C)(CC(=O)N1CCOCC1CCNC(c1nc(C)sc1C)=O)C(=O)OC N1(C(C(=Cc2ccco2)C)=O)CCC2(CC2)CC1C(=O)N.C1CCC(F)(F)C1.C N1(C(=O)CCc2ccncc2)CC2CCN(C(c3ccc4nn[nH]c4n3)=O)C2C1 C1(N(C)C(c2cc(Cl)cc(Cl)c2)=O)CCCN(C(c2cccc(CO)c2)=O)CC1 C1(C(C(=O)NC(CC)CNC(=O)CCc2ccsc2)O)CCCCC1 C(=O)(C#CC1(C)CCCO1)N(C(CC(=O)O)C(=O)O)Cc1cccc(C)c1 CC(F)(F)CCC(=O)NC1CCN(C(=O)C(O)Cn2cncn2)C1C1CC1 C1(C2(O)CCC2)(C(=O)NCC(CC(=O)N(C)C)OC)CC1.c1cn(C)cn1 C(C(CO)(CO)NC(c1ccc(N2CCOC2=O)cc1)=O)N(C(CC)=O)C CC1CN(C(=O)C=CC2CC2)CC1CNC(=O)CCc1c(N)cnn1C C1(OCC)COCCC1NC(=O)N(C)CC1(c2ccccc2)CC1 N1(C(c2n[nH]c(=N)[nH]2)=O)CC2CC(NC(c3ccc4cnsc4c3)=O)CC1C2 C(=O)(C(CC(C)C)OC)NCC1(O)CCN(C(C2CC(=C)C2)=O)C1 CS(=O)(=O)C1CN(C(=O)COc2ccc(-c3nn[nH]n3)cc2)C1 C(=O)(CCCC(N)=O)N1CCC(NC(CCC2C(C)(C)C2)=O)C1C1CC1 Cc1nocc1NC(c1nnnn1CC1CC1)c1ccsn1 C(N=c1[nH]nc(C2CC2)o1)C1C2CN(C(C(C)Cc3ccccc3F)=O)CC21 O=C(CCCOc1c(F)cccc1Cl)N=c1nc(C(F)F)[nH]s1 c1(C(=O)NCC2CC(NC(c3c(C)cc(F)s3)=O)C2)cnc2ccccc2n1 C1(CC)CN(C(c2cnoc2)=O)CCC1NC(=O)CCOCC(F)F C1(C=O)CC2(C1)C(F)(F)C21CC1.C1(O)CN(C)C1.C1(C(F)(F)F)CCC1 C1(NC(c2c(CC)noc2C)=O)CC2CC1CN2C(=O)CC1CC(=O)C1 CCC(C)C=CC(=O)NC(C)C=CC(=O)NCC.C(=O)N.C(C)C C1(C(=O)NC2CC(CCNC(c3cc(C)oc3)=O)C2)CCN2CCOCC12 C1(COC(CC#N)=O)CCCN(C(C2CCCN2C(=O)C2CC2)=O)C1 N1(C(c2c(C)nc(CC)s2)=O)CCC(NC(=O)C(C)(C)c2cnsc2)C(C)C1 c1(OC)ccc(C(N2CCCCC(CNC(C3CCC3)=O)C2)=O)c(F)n1 CC1CCN(CC(=O)N(C)CCC2CCCCN2C(C2CC2C)=O)CC1 c1(C(=O)NC2CCCN(C(C3C(C#C)C3)=O)CC2)csc2cc(Cl)cnc12 C1(CC=C)(NC(=O)C(N2CCOCC2)C)CN(C(c2ccc(CCCC)o2)=O)C1 c1(C(C(=O)NCC2CCN2C(=O)CCSC(F)(F)F)O)cccnc1 Cc1cncc(-c2cn(CC34CC(CN3C(C3(C(N)=O)CCC3)=O)C4)nn2)c1 Cc1nc2ccccn2c1C(=O)NCC(C)CNC(=O)C(O)Cc1[nH]cnc1C Cc1cc(O)ncc1C(N1C(C(=O)NCCCCC(C)(F)F)CC1C)=O CCCC(C(O)C(=O)N1CC(CC)(CO)C1)NC(=O)Cc1ccc(C)o1 Cc1c(C(=O)N(CCCNC(C2CC(C)OC2=O)=O)C)cnn1CCC(C)C CC1CN(C(=O)CC2CCS(=O)(=O)C2)CCN1C(=O)CS(C)(=O)=O c1(C(N(C)CC2CCCN2C(C23CC(F)(C2)C3)=O)=O)cnc2cccnn12 c1(OC)ccc(NC(=O)CCOCC)cc1.C(C1(C)COC1)=CC(=O)N C1(CC#C)(C(=O)O)CCCN1C(=O)C(C)OCC(C)C N1(C(C2C(C(C)(F)F)C2)=O)CC2(C1)CN(C(=O)C(O)CCc1ccccc1)C2 c1(C(=O)OC2CC2)cncc(-c2cnn(C3CC3)c2)c1 n1(CC(=O)N(C)CC2CCCN2C(=O)Cc2cn[nH]c2)nc2ccccn2c1=O Cc1cc(C)c(-c2nnnn2C)c(C)c1.C12(c3nnnn3C)CCOC(C1)N2 C(C(F)(C(=O)NC1CCN2CCC1C2)C(C)C)NC(c1n[nH]c(CC)c1C)=O Cc1cc(CN(C)C(=O)NCCC(O)c2cccs2)c(C)s1 C1(CNC(CCCC#CC)=O)(NC(c2ccccn2)=O)CC2CCC1CC2 CC(C)C(C(=O)N1CCN(C(c2nc(O)nc(O)c2N)=O)C(C2CC2)C1)C(C)C CCCC(CCC)=CC(=O)NCC(C)N(C)C(c1n[nH]c(CC)c1Br)=O N#Cc1cccc(C(=O)NCCCCCC(=O)NCC23CCCCC2C3)c1 N1(C(C2C(C)C2C)=O)CC2(CC(NC(=O)Cn3cc(F)ccc3=O)CO2)C1 C1COC2(C1)CN(CC(=O)N(C(C)C)C(C)C)C2.CC(C=O)S(C)(=O)=O.N C1CN(C(c2cccc(C)c2F)=O)C(C)(C)C1.C(F)(F)(C=O)C1(OC)CCC1.N C(=O)(C1=CC2CCCC12)N(C)CCNC(=O)CSCc1cscn1 C(=O)(CCC(C)(C)C(=O)N1CC=C(CNC(=O)CCC)CC1)OC.C(C)=O.N C1(C(=O)NC(C2CCCCC2)CC)CCN(C(=O)C(=O)NCC(F)F)CC1 Cc1ccc(N)cc1OC1CCC(C)(C)N1CCOc1ccc(F)cc1 CCC(C)(C)CC(=O)NC1CCCCCC1NC(=O)C(C)(C1CC1)OC C1(NC(CCN(CCCCC)CC)=O)CN(C(=O)C=Cc2nccs2)CC1(C)C N1(C(C(CC=CC)NC(=O)CN(C(=O)C(C)C)C)=O)CCN(C)C2CC12 Cc1ccc(CC(=O)N(C2CCN(Cc3ccc(Cl)c(Br)c3)C2)C)cc1[N+](=O)[O-] c1(N2CCN(C(=O)OC)CC2)ccc(F)c(CNC(c2cccc(Cl)c2F)=O)c1 c1(OC)cncc(C(N2CC(NC(=O)CN3CCC(OC)C3)C(O)C2)=O)c1 c1(CNC2CCCC(C(=O)Nc3ccc(OC)nc3)C2)c[nH]c2cc(F)ccc12 c1(N2CCCC(c3ccc(N4N=C(C)CC4=O)cc3)C2)cc(C)nc(C2CC2)n1 c1(C(=O)NCCCC2N(C(C3C(OC)C3)=O)CCCC2)cc(Cl)c(O)c(Cl)c1 N1(C(Cc2ccn(C)n2)=O)CCC(C(F)(F)F)C(NC(c2cncc(F)c2)=O)C1 O=C(C1OCCn2ccnc21)NCC1CN(C2CC2)C1 c1(NC(C(N2CC3CC3(CO)C2)c2cc(C(C)C)no2)=O)ccc(F)cc1 C1(NC(C(CC)CC)C)CC(c2ccc(OC)cc2)C1C1CC1 C12(C(=O)N)CC3CC(C(=O)N1)C2C3.C(C(C)(C)CC(=O)NCCCCCC)OC C=C=C(C)CC(=O)NCC1(F)CCC1.c1(C=O)ccc(C)cc1.C(=O)C.C N1(C(c2ncn(C)c2)=O)CC2(CNC(=O)C)CCC1C2.c1(C=O)cccs1.N C(C(N=c1cc[nH]cc1[N+](=O)[O-])C1CC1)NC(c1ccnc2ccsc12)=O C1(CC)CN(C(c2ccncc2C(F)(F)F)=O)CCN1C(=O)CCC.C(N)=O.N CCCCCC(C)NC(C1C2CN(C(=O)C(CC)CC)CC12)=O C(=O)(C(C(C)(C)C)OC)NC1CCCC(CC(=O)NC2(CC#C)CC2)C1 N1(C(C(CC)OCC)=O)CCCC(CNC(c2ccc(COC)[nH]2)=O)CC1 C1(N(C(=O)C)C)CCCN(C(c2ccc(C(N)=O)cn2)=O)C1.[SH](C)(=O)=O.N C(CCC(=O)NCCOCCN(C)C(C1(C#N)CC1C)=O)N(C(C)=O)C c1(C(=O)NCCN(C(C)C)C(C23CC(CO)(C2)C3)=O)cc(O)ncn1 N1(C(C(CCN(C)C)NC(CC(C)C)=O)=O)CC2CCC(C1)N2C c1(C(=O)OCC2CC(=O)C3CC23)cc(O)c2ccsc2c1 n1(CC)ncc(C(=O)NC2CC(CNC(c3cccs3)=O)C2(C)C)c1C.C c1(C(N(C2CCN(C(=O)C3=CCCS3)C2)CCC)=O)cc(C)nc(O)c1[N+](=O)[O-] c1(C(N(C(CC)C(=O)O)Cc2cccnc2)=O)cc(S(N)(=O)=O)c(C)cc1C C(C(CCC)C(=O)NCc1cnn(CC)c1C)NC(CC(C=C)C)=O c1(C(N2CC(NC(C3C(C)(C)COCC3)=O)C(F)C2)=O)ccc(Cl)c(N)c1Cl C(=O)C(C)S(N)(=O)=O.c1snc(O)c1Cl.C1(N(CC)C)CCCCC1.CC=O CC(C)(C)C(CO)C(=O)NC1CCC(NC(=O)CCCc2cccnc2)C1 N1(c2snc(CC)n2)CC=C(CNC(C23CCCN(CC2)C3)=O)CC1 N1(C(Cc2nc(C)[nH]n2)=O)CCOCC(C(=O)NCCc2nc(C3CC3)no2)C1 C1(NC(c2n(C)nc(O)c2)=O)C2CC1CN(C(c1cc3sccc3[nH]1)=O)C2 c1(N2CCOCC(NC(C(=Cc3ccco3)C)=O)C2)nc2cccc(C)c2o1 C1(NCc2scc(C)c2)CCN(C(c2cnc(C(C)C)s2)=O)CC1C C1(C(=O)NC(C2CCN(C(C3(C(N)=O)CCCCC3)=O)C2)C)CCC(C)CC1 C1(CN(c2ccc(C#N)cc2)C)CCN(C(c2ccccc2)=O)CC1(F)F CCCCC(C(=O)NC)NC(C1CC(C)CN1C(c1ccc(=O)n(C)c1)=O)=O C#CCC(CC(=O)OC)NC(C1CC(F)CN1C(C1CC1C(F)F)=O)=O c1(NCC2(CO)C(C=C)C2)cc(N2CC(C)C(C)(CO)C2)nc(CC)n1 c1(C(=O)NC2CCN(C(C(CC)C)=O)C23CCC3)cccc2nc(N(C)C)oc12 c1(C(N2CCCC(C(=O)NC3(C(CC)=O)CC3)C2)=O)ccc(Cl)cc1CSC C1(OC)(C)CCCCC1.C1(C(N(CCC=O)C2CC2)=O)CCC2(CC2)C1.N C(c1ccc(F)cc1[N+](=O)[O-])=CC(=O)NC1CCN(C(=O)CCC(F)(F)F)CC1 C#CC(C)(C)C(=O)NCC1CCCC1.c1(C(=O)N)ccncc1.CC(F)(F)F Cc1ccccc1C=CC(N1CC(NC(=O)C(O)CC(C)C)C(C)(C)C1)=O C1(NC(CC(CC)CC)=O)CN(C(=O)C(CC)CC)CC12CCC2 C(=O)(C(C)CCC(C)(C)C)NC1CC(C(C)NC(C(C2CCOCC2)C)=O)C1 c1(C(N2CC(NC(C3(CC=C)CC3)=O)C(C)C2)=O)cc2cc(F)ccc2o1 C1(O)(CNC(Cn2c(CCC)nnc2S)=O)CCCN(C(=O)CCCCCF)C1 N1(C(C(C)C)=O)CC(NC(=O)CCCNS(C)(=O)=O)C(C)(C)C1 c1(C(N2CC3C(C2)N3S(=O)(=O)c2cn[nH]c2)=O)ccc([N+](=O)[O-])c(F)c1F C(=O)(CCC(C)(F)F)N.N1(C(COCC(c2ccccc2)C)=O)CC2CC2(C)C1 C(=O)(CC(O)C(C)CC)NC(CCOCC)C(N1CCN(CC)C(=O)C1)=O N1(C(C(CC)(F)F)=O)CC(C(=O)NCC2CC[Si](C)(C)C2)C(C2CC2)C1 c1(SCc2onc(C(CC)NC(C)=O)n2)cncc(C)c1 C1(CNC(CCC=CC)=O)CCCN(C(=O)COCCSC)CC1 N1(C(CCN(C(CSCC=C)=O)C)=O)CCC(CO)C(C)(C)C1 C12CCC(CO1)C2.CN1CCC(C(=O)NC)CC1.C(c1ccn(C)c1)=CC=O Cc1cc(C(N2CCN(C(C3CC4CCC3CC4)=O)C(C)C2C)=O)c(F)cc1F c1(-n2cc(CN(C(C3CC(C(C)=O)C3(C)C)=O)C)nn2)c(F)cncc1Cl c1(C(c2nnnn2C2CCC2)NCC2C(C)(C)OCC2)ccc2c(c1)CCC2 C1(C(=O)NC(CC)C)OCCC1NC(=O)C(C)(C1CC1)OC c1(C=O)nc(C(C)C)n2ccccc12.Cc1cnsc1C(=O)NC1CC(C)C1.N C1(C(C)NC(c2cc(SC)oc2)=O)CN(C(c2cnoc2CC(C)C)=O)CCO1 CCC(C)C(C(=O)NCC1CC(C)(C)C1)NC(=O)COCCCOC C1(NC(CC2(N(C(CCC)=O)C)CC2)=O)CCN(C)C(=O)C1 N1(C(Cc2cccc(C)c2)=O)CCOCC(NC(C2CCCC(C(N)=O)C2)=O)C1 C1(CNC(=O)Cc2cccnc2Cl)CN(C(C2CN3CCN2CC3)=O)CC12CC2 Cc1cncc(C(N2CCC(C)C2CNC(c2ccnc(S)c2)=O)=O)n1 CC1COc2ccc(C(=O)NC3CCCN(C(=O)CS(=O)(=O)CCO)CC3)cc21 S(=O)(=O)(c1ccc(C(N2CC(N(C)C(C3CCC(C)NC3=O)=O)C2)=O)o1)NC C(=O)(N1CCCc2ccnn21)C1CC(C)N1C(=O)C(C)(C)C(N)=O c1(C(=O)NC(C(=O)NC(C2CCOCC2)C)C2CCCC2)c[nH]c(=N)o1 Cn1nc(C(=O)NCCNC(C2CC(O)(c3ccccn3)C2)=O)c2ccccc12 N1(C(C2(CC)CC2)=O)CC2CC1C2.c1(C(=O)N)nn(-c2cccc(Cl)c2)nc1C Cn1cc2cc(NC(c3cccn(C4CCSC4)c3=O)=O)ccc2n1 c1(C(=O)NCC2CCN(C(C(CC)SC)=O)C2)cccnc1C1CC1 C1(NC(CCCn2c(C)cc(C)n2)=O)CC2(C1)CC(NC(C1(C)COC1)=O)C2 CC(=O)C(C)CC(C)C(=O)N1CCOCC(CNC(=O)Cn2ncnn2)C1 N1(C(C2CC(SC)C2)=O)CC(NC(c2cc(C)oc2C)=O)C2CCCC12 C12(CNC(CCCOCC)=O)CCCC1N(C(C1CNC(=O)N1)=O)CCC2 C=CCC(CC=C)C(=O)NC(C(=O)NC(c1c(C)n[nH]c1C)C)C(C)C c1(C(C)C)cccc(C(N2CCCC(N(CCO)C(C3CC(C)(C)O3)=O)C2)=O)c1 C12(C(=O)NC3CC(OC)CN(C(CC(CCC)C)=O)C3)CCC(CC)(CC1)OC2 CC(C)(C)C(O)C(=O)NC(C)(C)C1CC1.c1(CC=O)cccc(C(F)F)c1 Cc1nc2ccc(C(=O)N(C)CC3CCN(C(C4CCC(=O)NC4)=O)C3)cc2s1 c1(CC)cccc(C(N2CC(N(C)C)C(CNC(C3CCOC3C)=O)C2)=O)c1F C1(C(=O)NC(CCNC(=O)C2=CCC2)Cc2ccccc2)CC12CCOC2 c1(C(C)C(=O)OCc2cnc(Cl)c(Br)c2)cnc2c(cnn2C)c1 N1(C(C(CCC)C(C)C)=O)CC2(CCN(C(=O)C(CC)N(C)C)CC2)C1 C(=O)(C1=CC(O)CC1)N.C(=O)CCCn1ccnn1.C(=O)(C)NCCOC Cc1cc(-c2nc(CC(C)C)nn2CCC(=O)OC(C)(C)C)cc(Cl)c1Br c1(C(=O)OCC)cc(OC(F)F)ccc1SC.c1csc(CS(C)(=O)=O)n1 C1CC(F)CN1C(=O)Cc1ccccc1C.c1(COC)ccsc1C(=O)NC.C c1(OCC)ccc(CC(=O)NC)cc1.C(=O)C(F)(F)c1cccnc1.C1CC1 C(=O)(C1=CC(C)(C)C1)NCC1CC(C)N(C(C23CCC(F)(CC2)C3)=O)C1 C(=O)(CCC(C)(C)C(=O)N1CCC(C)(C)C(CNC(C2CCCO2)=O)C1)OC Cc1cc(C)n2nc(C(=O)NCCN(C)C(c3ccc(C)n3C)=O)cc2n1 C1(C=O)CCCCN1C(C)C.C=C(C)CCNC(=O)CC(C)c1cnn(C)c1.N CCCC(C)(C)C(=O)N1CCC2(NC(=O)C=C3CCCC3)CC2C1 N1(C(c2ccc(OC)o2)=O)CC(OC)CC1CNC(=O)C(O)CN(C)C C=C(C)C1CC=C(C(C(=O)NC(C)(C)C)N2CCc3sc(C)nc3C2)CC1 Cc1ccnc(CNC(C2CC(C)N2C(=O)Cn2cccc2)=O)c1F N1(S(CC)(=O)=O)CCCC1(CNC(=O)NCC1CC(C)CO1)COC c1(OC)c(F)cc(C(N2CCN(C(=O)C=Cc3cocn3)CC2C)=O)cc1Cl c1(C=O)ccc(O)c(Br)c1.CC1(C(F)(F)F)CC1C(=O)NC1CCC1C c1(C(=O)OCC)cnc2nc(=NC(=O)Nc3ccc(C)nc3C)[nH]n2c1 C1(C(N2C(C(=O)NC)CC2)=O)CC12CC(NC(c1csc(F)c1)=O)C2 N1(C(CCCNC(C)=O)=O)CC(NC(=O)CCCC(N)=O)CC12CCCCC2 c1(N(CCNCc2ccc(C)cc2)C)cc(=NCC(C)(C)N(C)C)[nH]c(C)n1 N1(C(CC2CC(=C)C2)=O)CCCN(C(=O)C2=NOCC2)CC1C C(C1=CCN(C(C2CC=CCC2)=O)CC1)NC(c1scnc1Br)=O c1(C(OC)OC)ccccc1CN.N1CCN(C=O)CC1.C12CC3CC1C2C3 N1(C(C(C(COC)C)C)=O)CC2OCCN(C(c3ccc(Cl)o3)=O)C2C1 c1(CC)cc(C(=O)NC2CC3CN(C(c4cnc(O)n4C)=O)CC23)c(C)nn1 N1(C(c2c(C)cn(C)n2)=O)C2CCC1CC(N(C)C(c1cc(=O)cc(Cl)[nH]1)=O)C2 CC(C)(C)C#CC(=O)NC1CN(C(=O)CC2CCCCC2)CC1c1ccccc1 N1(C(c2c(N)ccc(C)c2)=O)CC2COCC(C1)C2NC(=O)CC(C)F N1(C(CC(=O)N(C)C)=O)CC(CNC(=O)Cc2c[nH]nc2O)CC1(C)C N1(C(C(C(C)(C)O)F)=O)CCOCC(F)(CNC(c2ccc3ncnn3c2)=O)C1 C(=O)(C1=CCC(NC(c2ccnc(CO)c2)=O)C1)N(CCC#C)C C#CCC(C)(C(=O)NC(CCC)c1ccco1)NC(c1cc[n+]([O-])cc1)=O C=CC1(C(N2CCC(F)(CF)C2)=O)CCN(C(C2CC(O)C2)=O)C1 C1CC(O)CN(C(=O)Cn2nnc(=O)[nH]2)C1.c1(SCC)ccccc1CC=O.N Cc1ncc(S(N)(=O)=O)cc1C(=O)NC1(C)CCCCC1.C1(C=O)CC1C.N c1(C=O)nnn2c1COCC2.C1(CNC(CSCC(N)=O)=O)CC(O)C1.C c1(CN2CCC(CC(=O)Nc3cnc(Br)c(Cl)c3)C2)cc2c(cn1)OCCC2 C=C(Br)CC(=O)NC1(CNC(c2cc(CC(C)C)c[nH]2)=O)CC1 C1(NC(C2CCN(C)C2)=O)CN(C(c2c(O)cccc2F)=O)CCC1(F)F Cc1cc(NCC(N2CCN(c3cc(C#N)ccn3)CC2)=O)cc(C)c1F C1(NC(C2C(C)OC(C)C2)=O)CCC(C)N(C(c2ccc(O)cn2)=O)C1 C1(CN=[N+]=[N-])C2CN(C(=O)NC(C3CCOCC3)c3ccsc3)CC12 C1(NC(CCCN(C)C)=O)CN(C(=O)Cc2ccc(S(C)=O)cc2)CCC1(C)C C(=O)(C(Cc1ccoc1)NC(C1CCCN1C)=O)N(CCN(C)C)C Cn1nc(C(=O)NC2C=CCN(C(=O)C(c3ccccc3F)O)C2)cc1C(F)F C1(O)(CC)CCN(C(=O)CC2(C)CCN2C(=O)CC2C(C)(C)C2(C)C)C1 c1(CC=O)c(F)cccc1F.C1(CC)(OC)CN(C(=O)C(F)(F)C2CC2)C1.N C1(C)(C(=O)NC(c2cccc(O)c2)C)CC12CCN(Cc1ccc(O)nc1)CC2 CC(CNC(=O)C)(C1CC1)N(C(=O)C=O)C.C1(C2CC2)CC1.C1CC1 c1(N(C)C)cccc(-c2cn(CC3CCN(C(c4cccnn4)=O)CC3)nn2)c1 C=CC(O)(C(=O)NCC(C)C)C(F)(F)F.C1(n2cnnn2)(C(=O)N)CCCCC1 c1(C(N(C(C)C)CC)=O)cc2c(C)cccc2[nH]1.N1(CC=O)CC2CC2C1.N C1(C(N2CCCC(CNC(Cc3c(C)cco3)=O)C2)=O)CCCCC(F)(F)C1 CC1(CC(=O)OCC(=O)NCCC2=CCCCC2)CCS(=O)(=O)N1 Cc1ccc(C(=O)NCCCCNC(C2(c3ccccc3)CC2(C)C)=O)c(Cl)c1 c1(C(N(CCCNC(=O)CCc2nccs2)C)=O)ccc(C2CCCCC2)cc1 N1(C(C(c2cccs2)SC)=O)CCCCC(Cn2cc(-c3ccncc3)nn2)C1 N1(C(C2(CC)CCC2)=O)CC2CC1C2NC(=O)C(C)Oc1ccccc1 C1(NC(=O)Cc2cccnc2Br)CC2CC1CN2C(=O)CCOC1CC1 CC1(C)CC(NC(c2cnn3c2CCC3)=O)CN1C(=O)COCC1CCCO1 CC1OCCC1CC(=O)NCCC1(C(=O)NCCOC(=N)O)CCC1 CC(C)C(C#N)C(=O)NC1CC(F)(F)CC1.c1(C(=O)N)coc(C2CCCC2)n1 c1(OC)nccc(C(N2CC3(CC3)CC2C(N2CCC(O)C(C)C2)=O)=O)c1F c1(C=O)cnc(-c2ncccn2)nc1.CC1(C)CC1C(=O)NCCC1CCC1.N C(=O)(C(CC)C(C)C)N(CC(C)(C)NC(c1ncn(CC)c1)=O)C c1(C(=O)NC2C(CNC(c3coc(C4CC4)n3)=O)C2)cc2cccnc2[nH]1 c1(C(=O)NCC2C3CN(C(c4c(C)ocn4)=O)CC32)cc(Br)c2occc2c1 C(=O)(C1=NOC(C)C1)NCC(CN(C(CC1(OC)COC1)=O)C)C C1(C(=O)NCCOCCCC)CCCN(C(C2CC(O)C(F)C2)=O)C1 C(=O)(C(O)CCC(F)(F)F)N(CCCNC(C1CCC(C)O1)=O)C C1(CCNC(c2cnc(C)s2)=O)CN(C(c2occc2F)=O)CCCO1 CCC(CCCC(=O)N(C1CCOC1)CCF)NC(C1C2CN(C)CC12)=O C=C(C)CC(=O)NC(CNC(=O)C(O)COCc1ccccc1)C1CC1 CN=c1cc(C(=O)NC2(C(=O)Nc3ccc(C)nc3)CC2C)cc[nH]1 C(=O)(CN=S(C)(C)=O)NCCN(CC(C)O)C(C1Cc2nncn2C1)=O CC1(C)C(NC(C2CCC(F)CC2)=O)C2CCCN(C(=O)CC3CCC(=O)N3)C12 N1(C(C(C2CCOCC2)OCC)=O)CCN(C(=O)CCn2ccnc2)C(CF)C1 c1(C(N(CC)CC2CCCN(C(=O)CO)C2)=O)cc(Br)cc2[nH]ncc12 Cc1ncc2c(n1)CCC(C(=O)NCCNC(c1cccc(S(C)=O)c1)=O)C2 C(=O)(CCC1=CCCCC1)N1CCC(CC(=O)N(CC(CN(C)C)O)C)CC1 C1(NC(C2(C(=O)NC)CCC2)=O)CC2(C1)CC(C)C2.C(=O)C(C)C=O c1(NC(=O)CC)ccccc1F.N1(C=O)CCOCC1.O=C1COCCCN1.C N1(C(c2c(C)sc(Cl)n2)=O)CCC(C)C(CNC(=O)CN2CCCNC2=O)C1 C1(CNC(c2ccc(NCC)cc2)=O)(C)CCCN(C(c2ncsc2C)=O)C1 C(CCC(N)=O)(C(=O)NC(c1n[nH]c(CC)n1)C)n1cc(CCCCC)nn1 C(=O)(CCCC(C)(F)F)NCC(C)N(C(=O)CCOc1cccnc1)C C1(NC(CCc2nc(C)sc2)=O)CN(C(=O)CCCC2CCCC2)CCC1C C=CCCCCC(=O)NC1(CCOC)CCN(C(=O)CCCOC(C)(C)C)CC1 C1(NC(=O)COCCCF)CCCCC12CCN(C(c1ccc[nH]1)=O)C2 CC1CCC(C(=O)NC2CC(CCNC(c3cc(C(N)=O)ccn3)=O)C2)CC1 N1(CC)CC2CC1CN2C(=O)CC(C)CNC(=O)CC1(C)CCOC1 N1(C(C(C(C)C)C)=O)CC(C2CN(C(c3cnn(CC4CCC4)c3)=O)C2)C1 CC(CO)CCc1nc(CC(C)CO)no1 C1CN(C(c2csc([N+](=O)[O-])c2)=O)CCCO1.C(C(C(=O)N)NC(C)=O)OC CC1CN(C(=O)CC2(n3ccnc3)CC2)CCC1COc1ccc(F)cc1F c1(C(N2CCOC(c3cn(CCCF)nn3)C2)=O)ccc(C2CCC2)cn1 C(=O)(CCC(F)(F)Cn1cc(CNS(N)(=O)=O)nn1)NC1CCC(C)(C)C1 N1(C(C2(C)CCC2)=O)C2CCC1CC(O)(CNC(=O)CN1CC3CC3C1)C2 CCCC(CC)CC(=O)N1CCOC(C(C)NC(C23CC(C)(CO2)C3)=O)C1 C1(C(N(C)CC2CCCN(c3cc(O)ncn3)C2)=O)Cc2ccccc2C(=O)O1 N1(C(CC2(C)CC2)=O)CCCC(C)(C)C1CNC(=O)C(c1ccccc1F)(F)F Cc1ccc(NC(=O)NC2CCN(c3cc(C(C)(C)C)ncn3)CC2)cc1Cl N1(C(C(C2CCOCC2)OC)=O)CCC2CN(C(c3ccoc3)=O)CCC12 c1(Cc2nnnn2CCF)cc2n(n1)CCCC2.CC1(CN)CC(C(F)(F)F)C1 C(=O)(C1(C)CCCc2ccccc21)NC1C2(CN(C(C)=O)C2)S(=O)(=O)CC1 c1(OC)noc(C2CC2)c1C(=O)NCCCCC(C)NC(=O)Cn1nccc1C S(=O)(=O)(c1cccc2c1COC2=O)N1C(c2ccc(OC)cc2)CCCCC1 c1(C(=O)NCC2(COC)CCN(C(CC(C=C)C)=O)C2)ccc2ncnn2n1 c1(N2CCC(C)C(CO)C2)nc(N2CCc3[nH]ccc3C2)nc2scnc12 C1(CC(=O)N(C2CN(C(CC3(CC=C)CCCC3)=O)C2)C)SC2=NCCN2C1=O C(=O)(CCS(C)(=O)=O)N1CC(CC(C)NC(c2ccc(OC(F)F)cc2)=O)C1 C1(C(N(C)OC2CCCC2)=O)C2CCC(C2)C1NC(C1CC1Cl)=O c1(CC)ccccc1CC(=O)N(C1CCCCC1)CC(F)(F)F Cc1cc(C(=O)N(CC(C)NC(=O)C(F)(F)C(F)F)C)c(F)cc1N C(C1=CCCOC1)N(C(c1n[nH]cc1Br)C(=O)NCCC1CC1)C N1(C(=O)C2CC2)CC2CCN(Cc3c(F)cc(Cl)cc3F)C2C1 C1(NC(CN(CCC)C)=O)CC(O)CN(C(=O)CN2CCC(C)CC2)C1 C(C1CCOC1)=CC(=O)NCc1cc[nH]c1C(=O)NCCC1CC(F)C1 N1(C(CC2(C)CC2(Cl)Cl)=O)CCN(C(=O)COC(F)(F)F)CC1c1cn[nH]c1 Cc1cnn(CCN(C)C(c2cc(C)[nH]n2)=O)c1.c1(C(C=O)C)ccn(C)c1.N N1(C(C(CCOCCO)NC(=O)Cc2ccsc2)=O)CC2(CCC2)C12CCC2 C1(CNC(=O)CN(C(c2cnco2)=O)C2CC2)CCCC(O)C1 CC1(C)CCCOC1CC(=O)NCC1CC(O)CN1C(C1CC2CCC1O2)=O C#CCC(C)C(=O)N1CCC(CF)(NC(c2oc(-c3cnn(C)c3)nc2C)=O)C1 C1(C(=O)NCC(C)(C2CC2)NC(c2c(Cl)cn(C)n2)=O)CC12CCOCC2 C(CC1=CCN(C(C2CC2F)=O)CC1)NC(c1nc(CCC)oc1)=O C1(F)(CNC(CC=C)=O)CCC(NC(=O)Cc2ccsc2)C1 c1(Cc2nnnn2CCCC2CC2)cccc(Br)n1.C1(CO)(CO)CN(CC)C1 C#CCCCCC(=O)N(CCC(=O)Nc1c(C)ncnc1C)OC CCCC(CC)C(=O)NCC#CCNC(=O)C=Cc1ccc(O)cc1 Cc1ccc(F)c(C(N2CCC(C)(C(=O)NC3(CO)CCC(C)(C)C3)C2)=O)c1 O=C(CC(F)(F)C(F)F)NCCC1CCN(C(c2c(Cl)csc2Cl)=O)CC1 C=CCC(CC(=O)Oc1ccc(C)c(Cl)c1)c1ccccc1 C(=O)(CCCC(C)(c1nnnn1C1CC1)Nc1cc(F)c(Cl)cc1Cl)OC C1(CC)CCN(C(c2cnccc2C)=O)C1C(=O)Nc1ccccc1CCO C(=O)(C1CCNc2ccccc21)NCCC1CCN(C(CCC(=O)N(C)C)=O)C1 C1(O)(C(C)NC(c2n(CC)ccn2)=O)CCN(C(c2cccc(OC)n2)=O)CC1 Cc1cc(C(=O)OCC(c2cc(C)n(-c3ccccc3Br)c2C)=O)nc(C)n1 c1(C(=O)NC2C3CN(C(c4cc(Br)cnc4O)=O)CC23)cc([N+](=O)[O-])ccc1Cl N1(CC)CC(C(N2CCCC2CNC(=O)CN2CCOC2=O)=O)NC1=O Cc1cccc(F)c1C(=O)NC(C1CC1C(=O)NCCn1cnnc1C)C N1(C(c2cnc(C3CC3)s2)=O)CCC(N(C(c2cn[nH]c2)=O)CC2CC2)C1 C1(N2C(C(N3CC4(CC4)C3)=O)CCC2)CCN(C(c2ccc(CO)nc2)=O)CC1 C12CCC(CC1)CO2.C1(CC(C)C)(C(=O)NC)CCC1.C1(C=O)CC12CC2 Cc1ccc(N)c(C)c1C(=O)NC1CCCCN(C(=O)C(C)(C)C2CCC2)C1 C1(n2cccn2)(C(=O)NC(CN(C(=O)CC2CC2)CC)C)CCOCC1.O N1(C(C)C(=O)N(C)C)CC2C(CNC(=O)CCC3CCCCC3)C2C1 C1(CNC(C2(CC)CC2(F)F)=O)CC(O)CN1C(c1ccc(OC)s1)=O CC1NC(=O)OC12CCN(C(c1cnn(C(F)F)c1)=O)C2 N1(C(c2n(C)cnc2)=O)CC2CC1CN(C(=O)C=CCOCC(F)(F)F)C2 c1(C(N(CCNC(CC2(CC)CCCC2)=O)C(C)C)=O)ccc(C)s1.C c1(C(N(C)CC2(NC(C3C(C#C)C3)=O)CC2)=O)cc([N+](=O)[O-])cnc1O C=CC1(C(=O)NCCOC2CCOCC2)CCN(C(=O)CC2CCCC23CC3)C1 C1CC2CCCC2C1.N(S(N)(=O)=O)CC=O.C(C(=O)N)NC(=O)OC.C c1(C(=O)NC(C)CCNC(C2(C)CC2Br)=O)ccn2c(O)nnc2c1 C1(NC(C2CCCCN2C(C2CC=CC(O)C2)=O)=O)CCCN2CCCC12 c1(CNC(CNC(=O)CNC(=O)C(O)C2CC2)=O)ccccc1 Cc1cc(NC(=O)N(C)Cc2ccc(Cl)o2)ncn1 c1(OCC=C)cc(Cl)ccc1C(=O)NCCNC(c1c(C)noc1)=O.C c1(CC)ccc2c(CC(=O)NCC=CC)coc2c1.c1(C=O)scc(C)c1.N CN1C(=O)NC2(CCN(C(=O)Nc3cc(Cl)ccn3)CC2)C1=O c1(CC(=O)NCCCc2cn(Cc3ccncc3)nn2)ccc(Br)c(Cl)c1 C(CN=c1nc(N2CC(F)CC(F)C2)c2c([nH]1)CSC2)Oc1c(OC)cccc1 C1(C(N2CCC(NC(C(C(=O)NC)(C)C)=O)C(O)C2)=O)CC2CCC(C1)N2C c1(C(=O)NCCCC=C)cn(CCC)nc1C.c1(CC(=O)N)nncn1C(C)C CC1(C)COCC(NC(=O)C(C)(C)C2CCCN2C(C2CC23CCCCC3)=O)C1 c1(NCC(C(C)(C)C)NC(C(CC)SC)=O)ccc([N+](=O)[O-])cc1C#N N1(CCN2CC3C(C(N(CCCCN)C(C)C)=O)C3C2)CCCCCC1.CC(N)=O c1(NC(C2C(NC(c3cc(Cl)ncc3Cl)=O)CCC2)=O)nc(Cl)ccc1O N1(C(CC2C(C)(C)OCC2)=O)CCC2OCCN(C(=O)Cn3cncn3)C2C1 C12CN(C(C3(O)CC(F)(F)C3)=O)C(C1)C2.n1(CCC=O)cc(C)cn1.CC N1(C(CCOCCOC)=O)CCC(CNC(=O)CC2CCC2)C12CC2.O c1(C(N2CC(C)(C)OCC2)=O)cc(S(N)(=O)=O)co1.C1(C=O)OC2CCC1C2.N CC(=Cn1ccnn1)C(=O)N1CC2C(N(C(=O)CC(C)(C)N(C)C)C)C2C1 C1(C(=O)NC)CCCN(c2nnc(C(c3c(C)n[nH]c3C)C)n2CC2CC2)C1 N1(C(COC(C)C)=O)CC2(CC2)CC1C.c1(C=O)ccc(C(N)=O)c(Cl)c1 c1(OCOC)ccc(CN2CCC(C#N)(NS(=O)(=O)C3CC3)C2)c(OC)c1 CC1=CCC(C(=O)NCC2CCN2C(=O)CCc2nnc(-c3ccsc3)o2)CC1 C1(C(=O)NCC(CC)(C)NC(=O)C(=O)N=S(C)(C)=O)CCn2nncc2C1 Cc1cc(F)cc(C)c1C(=O)NCC1CCC(C)N(C(=O)CCc2csnn2)C1 C1(C(=O)NC2CC(NC(COCCOCC)=O)C2)CCCC2CCCN12 C1(NC(C(=O)NCC)=O)CC2(C1)CC2NC(=O)COCC(C)C N1(C(C(C2CCC2)OC)=O)CCC2(CC1)COC(C)C2.C1(C(=O)N)CC12CCC2 c1(N(CCN(C(C2N(C(CCOCC)=O)CCC2)=O)C)C)ncccc1[N+](=O)[O-] N1(CC)CC(C(=O)NCC(CNC(c2cc3n(c2)CCC3)=O)CO)CCC1=O C#CC1(O)CCN(C(=O)C(C2CC2)N(C(=O)CC(C)C(F)F)C)C1 CC1(C)CC(NC(=O)C2=CCSC2)CN1C(C1CCCC1n1cccc1)=O N1(C(=O)OC(C)(C)C)CC(NCC2(c3ccccc3)CC2)CC1(C)C.CCO Cc1cccc(O)c1CN1CC(F)CC1C(N1CCCC(CO)C1)=O N1(C(C(C)(C)N2CCCCC2)=O)CCCCC(C2CN(c3ncccn3)C2)C1 Cc1cc2cc(NC(C3CCN3Cc3cccnc3C)=O)ccc2[nH]1 c1(C(C(=O)NC2CCCCC2)N(CC)CC2CC2)cnn2c1CCC2 c1(NC(C2C(CCOC)C2)=O)cccc(C)c1.c1(C(C=O)C)ccc(Cl)cc1 CCCCC(CNC(c1ccsc1OC)=O)NC(c1csc(C(F)F)n1)=O N1(C(CSc2n(C)nnn2)=O)CCC(C2CC2)(C)C1.C(=O)C(O)P(C)(C)=O.N c1(OC)ccc2[nH]cc(CCNC(c3cc([N+](=O)[O-])cnc3C)=O)c2c1 C(=O)C(F)(F)C(F)(F)F.C12CCCN1C2=O.C1(CC)CC1.C(C)(C)C.C Cc1ncccc1CCC(N1CC(N(C)C(c2cccc(CO)c2)=O)C(O)C1)=O Cc1cc(C)c(C(=O)N(C(c2ccccc2)C)C)s1.C1(C(=O)N)CC1.C1CC1 C1(C(N2CCC(C)C2)=O)C2CC3C(C2=O)C13.c1(COC(C)C=O)ccccc1 C1(OC(C)C)CCC(C)N(S(=O)(=O)CC23CC(C(F)(F)F)(CO2)C3)C1 c1(C(c2n(CCC)nnn2)NCCCC(=O)NC)ccc(OCC)nc1 C1(CNC(C2C(C)SCCC2)=O)CN(C(=O)C(C)Cc2cccnc2)C(C)(C)C1 c1(NCCN(CCO)CC)[nH]c(=NCCC(C)C(F)F)nc2ncn(CC)c12 N1(C(CN(CCC#C)C)=O)CCC2(CC1)CC2C(N1CC(F)(CF)C1)=O c1(C(=O)NC2CCN(C(C(CC)COC)=O)CC2CO)nn(C)c(=O)cc1C C1(=CC(=O)NC2CC(OCCCC)C2(C)C)CCC(C)(C)CC1 c1(OC)cccn2c(=O)cc(Nc3cnn(CCN4CCCC4=O)c3)nc12 CCCCC(CC(=O)NC(c1ncccn1)(C)C)NC(c1cc2n(n1)CCC2)=O c1(C(=O)NC(CCCC)CNC(=O)COCP(C)(C)=O)ccc2c(n1)OCCO2 N1(C(c2cc(C)no2)=O)CCCC2(CCCN2C(=O)C(C)Cc2ccco2)C1 C1(NC(c2nc(C)n(C)c2)=O)CC(C(=O)NCCc2ncc[nH]2)=CC1O N1(C(=O)NCCNS(N)(=O)=O)CCC(NC(=O)CC)C1.c1ccccc1.O Cc1cccc(CC(=O)NCC(O)COc2ccc(F)cc2)c1Br c1(C(N(CCNC(=O)C2=CCCC2C)CC)=O)n[nH]c2ccc(OC)cc12 C(=O)(C(CC)C(C)C)NC(C1C(C(=O)OC)C1)C.c1(C=O)cnncc1.N C1(CNC(=O)C2=CCOC2)(CO)CCN(C(=O)C(=O)Nc2ccccc2)CC1 C=C(C)CCC(=O)NCCCC(C)(C)NC(c1cc(OC)ccn1)=O N1(C(c2ccnc(OC)n2)=O)CC(CNC(C2CC3CC3C2)=O)C2(CC2)C1 CC(F)(F)CCCCNC(C1CCN1C(=O)Cc1ccccc1F)=O C(=O)(C(F)(F)C(F)(F)C(F)(F)F)NC(CNC(c1cc(C)cc(O)c1)=O)C CCC(C(=O)NCC1(NC(C2CC(=O)N(CC)C2)=O)CCCC1)C(F)(F)F N1(CC)CCOCC1CC(=O)NCC1CC(NC(C2CCCCS2)=O)C1 C=C(C)CC(C(=O)NC1(CNC(=O)C(F)C(C)(F)F)CCCCC1C)OC c1(-c2c(C)c(F)ccc2)cnc2cc(C(=O)NCCc3ccc(O)cc3)ccn12 c1(CNC(C2N(C(c3ccc(C)cc3)=O)CCOC2)=O)ccc(F)c(C)c1 C1(CNC(C(C)OCc2ccccc2)=O)CC12CCN(C(c1cccs1)=O)CC2 N1(C(C=CC=CCC)=O)CC2(C1)CN(C(C1CC(C)(O)C1)=O)C2 CCCCC(CC)(C1CC1)NC(c1ccc(C(F)F)c(F)c1)c1ccc(F)cc1 O=C1CN(CC2CC3CCC2O3)C(=O)N1CC1CCCC1(F)F CN1CCCC1C=CC(=O)NC(CC(=O)NCC=C1CCSCC1)C1CC1 C#CCCCCCC(=O)NCC1CCCC1C(=O)N(CC(F)F)CCO c1(OC)ccc(C(N2CCCCC2CNC(c2cc(O)ccc2C)=O)=O)c(Br)c1 c1(CC2CC3CC(NC(=O)OC(C)(C)C)C3C2)c(O)ccc2ccccc12 C(c1cc2ccccc2o1)=CC(N1CCC(F)(C(=O)Nc2c[nH]nc2Cl)C1)=O CC1(C)CC=CCN(C(c2cccc(CNC(c3ccco3)=O)c2)=O)C1 c1(C(=O)NCC2CN(C(c3ccc(C)cc3F)=O)C2)cc2cnccc2nc1C C(C(CC(F)(F)F)NC(c1cn(C2CCCC2)nn1)=O)NC(c1n(C)cnc1)=O c1(OC)ccnc(C(=O)NCC(F)CNC(c2cncc(C(F)F)c2)=O)c1 c1(N2CCC(N(C(=O)C(C)CCCOC)CC)C2)c([N+](=O)[O-])cccc1[N+](=O)[O-] C1(NC(c2cc(C(F)F)on2)=O)CC2CC(C1)N(C(=O)C(C1CCOCC1)F)C2 c1(C(=O)NC2C(C)(C)CN(C(=O)C3=NNC(=O)C3)CC2)cccc(Br)c1[N+](=O)[O-] N1(C(c2scc(C)c2Cl)=O)CCOC2CCN(C(C3CCCS3(=O)=O)=O)CC12 C1(CC)CCN(C(=O)Cn2ccnc2C)C1C(=O)NCCC1(C)N=N1 N1(C(C(C2CCOCC2)C)=O)CCC(F)(C(=O)NCC2C(CO)C2(F)F)CC1 N1(C(c2cccn(C)c2=O)C(=O)NCC2CCOCC2)CCCC2(CCC2)C1 C1(NC(Cc2c(C)cccc2Cl)=O)CCC2CCN(C(=O)Cc3ccoc3)C12 N1(C(C)=O)CCN(C(=NCCC2CCOC2)NCC(C)(C)C)CC1 c1(C(N(CCOC)CCNC(C2CCC(=O)N2)=O)=O)cc(N)c(F)cn1 N1(C(c2n(CC)nc(C)c2)=O)CCC(F)C(NC(c2nsnc2O)=O)C1 c1(C(=O)NCC(CNC(CCC2N(C)CCC2)=O)O)ncc(C(F)(F)F)cc1Cl C=CCC(C)C(=O)N1CCCC(CCCCNC(c2nccc(C(F)F)n2)=O)C1 n1(CC(=O)N(CC(C)NC(C(C(C)C)F)=O)C)ccc(=O)n(C)c1=O N1(C(C2CCCC(O)C2)=O)CC2CCCN(C(c3cc(Cl)ns3)=O)C2C1 C1(C(N2CCC(N(C(c3cc(C(C)C)no3)=O)C)CC2)=O)CCC2CCC(=O)N12 C1(N(C(=O)C(CO)N(C)C)CC)CCN(C(C23CSCC2C3)=O)CC1 N1(C(C(C)Cc2ccco2)=O)C2CCCC1CC(C(N1CC(C)(O)C1)=O)C2 N1(C(C(C)OC)=O)CCCCC1CN(C(=O)CO)C.C(c1ccccc1)=CC c1(C(=O)NCC(n2cc(C3(F)COC3)nn2)C)cc2nccc(Cl)c2s1 CC1CN(C(C2COC(=O)N2)=O)CC1(C)C(=O)N(CCC1CC1)C.C1CC1 O=S(=O)(c1ccccc1S(=O)(=O)N1CC2CC1C1CC21)NCC(F)(F)F Cc1ccc(CCCCC(=O)N2CCC(F)(CNC(c3ccn(C)n3)=O)C2)cc1 CC(C)S(=O)(=O)C(C)C(=O)NC.C(=O)(C(C)(C)C(=O)N(C)C)N1CCOCC1 c1(C(=O)NC)c(C)cc(NC(Cc2cccc(F)c2)CC(=O)OC)cc1F C(C(=O)NCC[Si](C)(C)C)(C(C)CC)N(C(CC1CC(=C)C1)=O)C CC1CCOCC1C(=O)NCCOCCN(C(=O)C=Cc1cocn1)C C=CC(C)N=c1nc(N2CCC(N(CCCN(C)C)CC)CC2)c2c([nH]1)CCC2 C#CCC(O)C(=O)N1CC(CC(=O)NC2CC2c2nc[nH]n2)(OCC)C1 CCC1=C(C(=O)NC(CN=[N+]=[N-])C(=O)NCc2nccc(C)c2F)CCCO1 CC1CCCCC1(CNC(c1cccn1C)=O)NC(C12CSC(C1)C2)=O N1(CC(N2CC(OCCNC(=O)CC3CCC4CC34)C2)=O)CCC(C)CC1 C=CCC(CC(C)C)C(=O)N1CC(F)(F)CC1C(=O)N(CCC(N)=O)CC N1(C(C=Cc2ccn(C)c2)=O)CC2CCN(C(=O)CC(F)(F)F)C2C1 O=C(C#CC1CCOC1)NCC1C=CCN1C(c1ccc(Br)cc1)=O C1(C(=O)NC(C)Cc2cnc[nH]2)CC2CCC(C1)N2C(=O)C(F)C(C)(F)F c1(C(=O)NC2CCC(CCNC(CN(C)CC)=O)C2)n[nH]c(C2CC2)c1Br N1(C(c2ccnc(CC)n2)=O)CC(F)(F)CC1C(N1CC(C2CCCO2)C1)=O CCCC(CCCNC(C1CC=CC1)=O)NC(c1cncc(C(=O)N(C)C)c1)=O CC1C2CC(C2NC(=O)Cn2cncn2)N1C(=O)CCN1C(=O)CCC1=O C1(C(=O)NC(C)C(=O)N(C)C)CC2(CC2)CN1C(=O)CN1CC2CC2C1 C1(C(N2CC(C(=O)NCC)C2)=O)CCCCN1C(=O)Cc1csnc1C N1(C(CCCCOC)=O)CCCC12CCN(C(C1C3CC4C(C3)C14)=O)C2 N1(C(c2c(COC)noc2)=O)CCN(C(C2(OC)CCCOC2)=O)CC1C C1(NC(C2CC(CC)(CC)C2)=O)COC2CN(C(=O)CC(C)(C)C=O)CC12.O N1(C(C2CCC(=C)CC2)=O)CCC(COC)(NC(C2CCCC(OC)C2)=O)CC1 CCC(CC)CCC(=O)N1CCCN(C(=O)CCOC2CCCC2)CC1C c1(C(=O)NCC(CC(F)(F)F)NC(C#CC(C)C)=O)cc2ccccc2cn1 Cc1ccc(CCC(=O)NCC#CCNC(C2CC(C)(F)C2)=O)c(C)c1 CC1(C)CCCN(C(C2(F)CCS(=O)(=O)C2)=O)C1.c1(C=O)cn2c(n1)CCC2 C1(C(=O)NCC)C2C3CC4C1C2C34C(=O)NC(c1ccc(F)cc1)CC C(N=c1[nH]c(=NC2CCC(C)(C)C(C)C2)c2sccc2[nH]1)c1cc(CC)[nH]n1 C1(COCC(=O)NC)CCN(C(=O)CC)C12CC2.C(C=O)O.C1COC1 N1(C(C2(SC)CC2)=O)CCC(O)(CNC(=O)CCC[N+](=O)[O-])CC1 Cc1oc(-c2cccs2)nc1CC(=O)NCC1C2CC2CN1C(=O)C(C)O c1(C(N(C)CC2(O)CN(C(=O)OC(C)(C)C)C2)=O)ccc2c(n1)NCC2 c1(OCC)ncnc(OC)c1C(N1CC(C2CC2)C1)=O.C(=O)C#CC1CCC1.N CCC(C(=O)O)N(C)C(C1CC1Br)=O C1(CNC(C(C(C)C)F)=O)CCN(C(c2ccc(F)c(F)c2)=O)C12CC2 CCC1=NOC(C(=O)NCC2(CN)CCC2)C1 C12(NC(C(CCC)O)=O)CCCCC1CN(C(c1cc(C)no1)=O)C2 Cc1nc2cc(C(=O)NC34CCN(C(=O)CC#N)CCC3C4)ccc2n1C N1(C(C(C)OCC=C)=O)CC(CC=C)(C(=O)NC2CC2c2c[nH]nc2C)C1 C(=O)(C1=CCCC1C)N(C)CC1N(C(c2cncc(CC)c2)=O)CC(F)C1 C(=O)(C1Cc2ccccc21)N1C(CC(=O)NCCc2csnn2)CCC1 N1(C(c2c(C)cc(C)[nH]2)=O)CCC2C(CCCN2C(c2ccnnc2S)=O)C1 c1(C(C)C)ccccc1C(=O)NC1CC(C(=O)NCC2CCO2)C1 Cc1cccc(C(C)NC(c2coc(CNC(c3c(C)csc3C)=O)n2)=O)n1 C(CCC(C)(C)C(=O)NC1C2CCCCC12)NC(C(C(C)C)OC)=O C1(NC(CC(C)NC(=O)Cn2cc(C#N)cn2)=O)CC2CCCCCC12 C(=O)(CCCCCN(C)C(c1ccc(=O)n(C)n1)=O)NCc1cc(C)ns1 c1(C(=O)NCC(c2cn(CC)nc2)=O)ccc2cc(F)c(F)cc2n1 C1(NC(C2CCN(CC#C)CC2)=O)CCCCC12CCN(C(C1CC1F)=O)CC2 c1(N(C)Cc2ccsc2)ccncc1S(=O)(=O)NC(C)(CO)C1CCCC1 C(=O)(CC(C(C)C)C(C)C)N1CC(CNC(c2c(C)ncnc2)=O)C(C)(C)CC1 c1(CCNC(NCC(CC)n2cccn2)=NC)ccccc1C C#CCC(C)(CC)C(=O)N1CC=CC(C(=O)NC(C)(C)C#CCCCC)C1 c1(OCC(C)N(CCOC)C(C2(OC)CCSC2)=O)ccc(F)c(Cl)c1 C1(C(=O)Nc2ccc(CC)nc2)C2CCC(C2)C1NC(c1scnc1C)=O Cc1ccc(OCC(=O)OCC2CCCCN(C(C3(C#N)CC3)=O)C2)c(C)c1 C(C(=O)NCC1CCCO1)(C(C)C(C)(C)C)N(C1CCOC1)CCOC C1(CC=O)CCCC(=O)N1.C(CO)(C(=O)NCc1nccs1)NC(N)=O.C N1(CCCC)CCN(C(C2(SC)CN(C(C)=O)C2)=O)CC1 C(=O)(CS(=O)C(F)(F)F)NC(C1CCN(C(c2cc(C)ns2)=O)CC1)(C)C c1(SC)ccnc(F)c1-c1cnc(Nc2ncnc(C)c2Br)c(O)c1 Cc1ccc(CC(=O)NC23COC(C2)C(NC(=O)C(O)C(C)C)C3)c(Br)c1 CC1CN(Cc2nc(C3CC3)no2)CCN1C(c1cc(-c2ccco2)[nH]n1)=O c1(OC)cncc(CCC(=O)NC2C3CCN(C(=O)CN(C)C4CC4)C23)c1 CC(C)CC(C)C(=O)N(CC(CO)(CO)NC(=O)CCC1(C)CCC(=O)N1)C c1(NC(C2CN(Cc3cncc(OC)c3)C2)=O)cc(F)cc(F)c1C#N C(=O)(CCCCCOC)NC1(C(=O)NCC(C#C)OC)CCSC1 C1(NC(c2n(CC)ncn2)=O)CC(=O)NC1.CCC.C(=O)(CC1CC1)N c1(C(=O)NCc2n(CC)cnc2)cnc(C)nc1.c1(CC(=O)N)ccoc1 c1(-c2c(C)n[nH]c2)cc(CNC(c2cc[nH]c2)=O)ccn1 CC(C)(C)CC(C)(C)C(=O)NC1CCOC(C(=O)NC2CCCCCC2(C)C)C1 c1(C(=O)NCC2C(C)CCN(C(=O)C3=COCCO3)C2)ccnc2c1CCC2 c1(C(=O)NCC(C)CN(C(=O)CN2CCCCC2)C)cc2nc[nH]c2cn1 C(C)(N=c1ccnc(NCc2cccnc2N)[nH]1)c1c(OC)cccc1 CC(C(CO)NC(C1(F)CC1)=O)NC(c1cc(-c2cccn2C)[nH]n1)=O N1(C(c2cncc(OC)n2)=O)CCCC(C)C1CCNC(c1nc(C)oc1C)=O c1(OC)cc(C(=O)OCc2cc(C(=O)O)ccc2C)cc(Br)c1O C(=O)(C1=CCS(=O)(=O)C1)NCCC(C)N(C(=O)Cn1cnnc1)C c1(CC(=O)NC(C2N(C(CCC#C)=O)CCCC2)C)c(C)cc(OC)cc1C C=CCC(CNC(C1(C)CCCCC1C)=O)C(=O)NCCOCCCC N1(C(c2c(COC)nn(C)c2)=O)CCC2CCN(C(=O)Cc3sccc3C)C2C1 C1(C(=O)NCC#CC)N(C(=O)C(C)C(O)C(C)C)CC12CCCC2 N1(C(CN2C(=O)CCC2)=O)CCN(C(c2cc(-c3ccco3)cs2)=O)C2CCC12 C1(NC(c2c(C)csc2)=O)CN(C(=O)C2=CCC(C)(C)CC2)C2(CCCOC2)C1 C=C(C)C1CC=C(CNC(=O)NCC(C)F)CC1 c1(C(=O)NC2C(C)CCN(C(c3cc(C4CC4)on3)=O)C2)cc2ccccc2[nH]1 N1(Cc2cccc(C(N)=O)c2)CC2CCC(C1)C2NC(c1ccno1)=O c1(CNC(CN(C2CCC2)C)=O)cccnc1CNC(c1scnc1Cl)=O C1(O)(C(C)NC(C2CCCCCCC2)=O)CCN(C(C2(C)C=CCC2)=O)CC1 c1(C(C)NC(C(C)N(CCC)C(C23CCCC2C3)=O)=O)ncccc1C C12(C(N3CCC(N(C)C(C45CCCC4CCC5)=O)CC3)=O)CCOC(C)(C1)C2 O=C(C1=CCCNCC1)NCC(c1ccc(C2CC2)cc1)F N1(C(C(c2ccn(C)n2)(C)C)=O)CC2CN(c3ncccc3C#N)CC2C1 N1(C(c2c(-c3ccc(C)cc3)nn(-c3ccccc3)c2)=O)CCC(C)C(C)(O)C1 C(=O)(CCCC1CCC1)N1CCCC1.C(CCC(C)C)=CC=O.CC(=O)OC C1(C(N2CCC(c3ccc(OC)c(Cl)c3)(O)CC2)=O)CC(c2cnn(C)c2)=NO1 CC1CCN(C(=O)CC2CCC(=O)NC2)CC1CC=O.C(CC1CC1)C1CC1.N C=CCC(C(=O)NC(CC=CC)C(N1CCC2(CC1)CC2)=O)C(C)C c1(C(C(=O)NC2CCC2)N(C(C)(C)C)CCOC)ccc(Cl)o1 C1(CNC(C2N(C)CCN(C)C2)=O)CCC2CN(C(C3(O)CCCC3)=O)CC12 C(=O)(C(CC=C(C)C)c1ccccc1)N(CC(=O)OC(C)(C)C)C.CC=O N(C(=NCCCC(F)F)NC1CC1)C1CCCC(CC)C1 CC(=O)C(C)CC(C)C(=O)N1CCOCCC1C(=O)NC(c1cnn[nH]1)C Cc1nn2cc(C(=O)N(CCCNC(=O)CN3CCCCCC3)CCO)nc2s1 C1(C(=O)NC(C)CCCNC(=O)CC2(OC)CCC2)(CC)CCCO1 C=CCCCC(C)(C)C(=O)N1CC(OC)C(NC(=O)CC2CCCC(OC)C2)C1 N1(C(Cc2c(C)cco2)=O)CCCCC1CN(C(=O)C(n1cnc(C#N)n1)C)C CCC(C)CCCC(=O)NCC1CC(F)CN1C(=O)Cn1nnc2ccccc12 C1(NC(C)Cc2ccc(Cl)cc2Cl)N(C(=O)OC(C)(C)C)CC12CCCC2 c1(C(=O)NCCCNC(C)=O)cc2cc(C)ccc2[nH]1.c12cc(cc(F)n1)N2 c1(C(N2CC(N(C(C(CCC)CC)=O)C)C(C)(C)C2)=O)c(C)ccc(F)c1N N1(C(C2CCN(C(CC)=O)C2)=O)CCCCC1CN(C(c1c[nH]nc1Cl)=O)CC C12(CCC=O)CCC(CC1)C2.C(C(C)C(=O)NC(c1cnn(C)c1)C)SC.N C12(NC(C(CC)N(C)C)=O)CC(C1)N(C(=O)C(C)SC(F)(F)F)C2 c1(C(N(C)CC2C(NC(C(C)(C)SC)=O)CCC2)=O)cc(F)cc(F)c1F N1(C(=O)CCCn2cccn2)CCOCC(F)(CNC(C2(C3CC3)CC2)=O)C1 c1(C(N2CCC3CCCCC23)C(=O)NCCCF)ccc2c(n1)CCC2 C1CCOC(C=O)C1.C(CC)C(C)(F)F.C1(C(=O)OCC)(C(=O)N)CCC1 N1(C(C2(COC)CCC2)=O)CC2OCCC2C1.c1(C(=O)N)ccoc1C1CC1 c1(C(N2CCC3(CCN(C(C4CCCO4)=O)C3)C2)=O)cc2ccc(Cl)cc2nn1 S(=O)(=O)(c1ccc(NC(C)CS(C)=O)c(Br)c1)NC1CCN(CCOC)CC1 N1(C(C)=O)CCCC2C(CCCN2C(c2c(C(C)=O)sc3ccccc23)=O)C1 C1(c2n(CC(=C)C)nnn2)(Nc2cccc3[nH]ccc23)CCN2CCC1C2 Cc1[nH]c(C#N)cc1C(N1CCC(O)C1)=O.c1(CCC(=O)N)nc(C2CC2)no1 c1(C(N(CCOC)C)=O)cc2cc(C(=O)OC)sc2s1 c1(CC(=O)N(CCCCN(C)C(C2(O)COC2)=O)C)ccc(F)c(Cl)c1 CC(CC1CCC1)C(=O)N1CCCC1CN(C(=O)CCc1nncs1)C c1(C(=O)NCCCC(C)(C)NC(CNC(C)=O)=O)cccc2nc(O)ccc12 CC1(C)CC(CNC(=O)C(F)(F)CCn2cccn2)CN1C(=O)C=CCF N1(C(C(N2CC(C)C2)C)=O)CCN(C)CC1C.c1(C(=O)N)cnc(C2CC2)nc1 c1(C(=O)NC(CC)CN(C(c2cn(C)nc2Cl)=O)CC)cc(C)c(F)cc1Cl C=CCC(CC(C)C)C(=O)N1CCN(C(c2ccc[nH]2)=O)CC1C(F)F C(CCC(C(=O)NCC1CCS(=O)(=O)C1)N(C)CC1CCOC1)=C(C)C C1(N(C(C(=O)Nc2ccccc2)C2CC2(Br)Br)CC)CCN(C)CC1 N1(C(CC2CC(C)C2)=O)CCN(C(c2cn(CCO)c(=O)nc2O)=O)CCC1C C(=O)(C(CC)C(C)(C)CC)N(C(C)C(=O)NC1CC2(CC(O)C2)C1)CCC CCC(CCC(=O)NCC1CCN(C(c2cnc(O)c(F)c2)=O)C1(C)C)OC CCCC(C)(CC)C(=O)N1CCC(C)(NC(=O)Cc2cncc(C#N)c2)C1 c1(C(=O)NCC2CC(NC(c3c(OC)c(Cl)ncc3)=O)C2)[nH]cc2c1CCCC2 c1(CNCc2ccc(F)c(C(=O)OC)c2F)c(N)oc2ccc(F)cc2c1=O C1(C(=O)NCCCC2CCCN2C(c2ccco2)=O)(COC)CC=CCC1.C C(=O)(C(F)(F)C(O)C(C)C)N(CC(C)NC(c1c(C)cc(F)nc1)=O)C C1(C(=O)NCCC(Cn2cc(CC(COC)O)nn2)F)(CO)CCCCO1 c1(-c2ccc(C(=O)NC(C(C)NC(=O)Cc3csnn3)C)o2)cccc(Cl)c1F C(CCC(C(=O)NC1(CC(C)(C)C)CC1)NC(c1ccc(C#N)[nH]1)=O)OC Cc1cc(N(C)C)ccc1C(=O)N(C)CCNC(=O)C(O)CN(C)C CCC(Cc1nc(C2CS(=O)(=O)CC2OCc2ccccc2)no1)CC(F)(F)F c1(NC(C2C(NC(c3cc(C)sc3C)=O)CC2)=O)cnc(C)c(C#N)c1 C1CCC(O)CN(C(C2CCCN2S(C)(=O)=O)=O)C1.C(C(C)(C)C(=O)N)OC c1(C(=O)N)cc2cccc(Cl)c2s1.CC1(C(=O)NCCC2CC2)COC(=O)C1 c1(C(COC(C(CC#C)O)=O)=O)ccc(Cl)c(Cl)c1 CS(=O)c1ccccc1C(=O)NCC(O)CNC(c1cnc(N)c(Br)c1)=O c1(C(=O)NC2C=CCN(C(CC3C(C)=NN(C)C3=O)=O)C2)cnn2c1CCCC2 C1(C2CCC2)(CNC(c2cc3c(Cl)c(F)ccc3[nH]2)=O)CCN(C(=O)CO)CC1 N1(C(CC2(N(C(C)=O)C3CC3)CC2)=O)CCC2CN(C)CC12 Cc1cc(CNC(C2CCN(C(c3cc(C)c(C)s3)=O)C2C)=O)nnc1C c1(CC(=O)N)ccc(O)nc1.n1(CC=C)cccc1C(=O)NC(C)C1CC1 N1(C(c2cccc(SCC#C)c2)=O)CCC(NC(c2cc(C)on2)=O)C(O)C1 C1(NC(c2ccn(C(CC)CC)n2)=O)CCCCC1.N(S(=O)(=O)NC)CC=O.C C1(NC(C=Cc2ccc(C)o2)=O)Cc2ccccc2N(C(c2cscc2C)=O)C1 C1(C(=O)NCC2CCCN2C(=O)Cc2ccccc2)(CC)CCC(O)CC1 C(=O)(CC(C(C)(C)C)NC(=O)CN)NC1C(c2cn(C)nc2)C1 c1(C(N2CC(NC(C3CC4(CSC4)C3)=O)C(F)C2)=O)ccc2c(=O)cc[nH]c2c1 N1(C(C(CCCC)=O)=O)Cc2occ(C(=O)N(c3ccccc3)C)c2C1 CCC(CO)CN=c1[nH]c(=NCc2sccc2Cl)[nH]c2cc[nH]c12 CC1=C(C(=O)NC2CC2C)Cc2ccccc2O1.c1(C=O)cc(C(F)F)no1.N C1(NC(C(CCSC)OC)=O)CC2CCC(C1)N2C(=O)C=C(Cl)Cl N1(Cc2ccc(C)c(C(F)(F)F)c2)CC(=O)N(C)CC1C(=O)O c1(C(=O)NC(COC)C(=O)NCC2CCC2)ncnc(O)c1F.C(C)(C)O c1(CC)ccc(C(=O)N(CC(C)NC(c2cnn(C3CCOC3)n2)=O)C)[nH]1 c1(CN2CCN(C(C(=O)NC(CC)C)C)CC2)c[nH]c2cccc(C)c12 C1(C)(CC)CCN(C(C(=O)NCCCF)C2CC2C)CC1 C1(C(N2CC3(C(NC(C)=O)CC3)C2)=O)CCC2(CC1)COCCO2 c1(NC(c2n(CC)nnn2)C2(C#N)CC2)cc(F)cc(F)c1 C1(CNC(C2(OC)CCCOC2)=O)CCC(F)CC1.c1(CC=O)cn[nH]c1.C C(=O)(CC(C(F)F)NC(=O)CN1CCCNC1=O)NC(C)(C)C C=CC(CC)CC(=O)NCCCN(C)C(C1CCCC1(F)F)=O C(=O)(C(CCF)NC(c1nsnc1O)=O)NCC1(C(=O)OCC)CC1 O=C1NC2(C(=O)NCC3(F)CC4CCC(C3)N4C(=O)CCF)CC3CC1C2C3 CCCC(C)(CCC)C(=O)N1CCCN(C(c2ccc(C#N)cc2O)=O)C(C)C1 CCC(O)(CC(=O)OCc1cc(Oc2ccccc2Cl)ccn1)c1ccccc1 c1(C(N2CCCCC2C(C)(C)C(F)(F)F)C(=O)NCC=C)cccc2c1OCO2 C1(c2onc(C3C(O)CCC(C)(C)C3)n2)CC2(CCCCC2)S1(=O)=O c1(C(N)=O)cnc(Cl)[nH]c1=NCC1CCCCN1C(c1cnn[nH]1)=O O=C1OCC2=C1CCN(C(=NCC=Cc1ccc(F)cc1)NCC1CCCO1)C2 Cc1c(C(=O)NCC2CCC2)[nH]c2c1CCCC2.c1(C=O)cnnn1C(C)C.N N1(Cc2ccc(C)cn2)CCC(O)C(C(=O)NCc2noc(C)n2)C1 C1(C(N2CCCC(CC=C)(NC(=O)C(CC)CC)C2)=O)CCOC2(CCCC2)C1 C=CCC(CC(C)C)C(=O)N1CC(CNC(=O)CC(F)(F)Cl)(OC)C1 CCC(CC)(C(=O)NC(C1CN(C(c2n[nH]c3c2COC3)=O)CCO1)C)OC c1(C(=O)NCC2CCC(NC(c3sccc3F)=O)C2)cc2ccc(F)cc2o1 CC1C(CO)CCCN1C(C1(CNC(=O)CC2CCCC2O)CC(C)(C)C1)=O C1(C(=O)NC(C)CCN(C(=O)CCOC2CCC2)C)COCCO1 C1(N(C(C)C)C)CCN(c2nnc(C3CCCCC3)n2CC2(O)CCSC2)CC1 c1(CC(C(=O)NC(CC=C)CNC(=O)CC2CC=CC2)O)cccc(Cl)c1 N(C1CCOc2c(OC)cc(C)cc21)C(Cc1ccc(C(=O)OC)s1)=O C1(CNC(C2CCC(N(C)C)C2)=O)CN(c2nccc(-c3cccnc3)n2)CCO1 N1(C(c2ncsn2)=O)CC2(C)CN(C(=O)C=C(CC)CC)CC2(C)C1.CCO C1(C(N2CC3C(CNC(CCc4scc(C)n4)=O)(C3)C2)=O)CCCCC1(C)C c1(C(=O)NC(c2cn(Cc3ccncc3)nn2)C)ccc(C2CCOC2)cc1 CP(C)(=O)CN1CC(C(=O)NC2CC2CNC(c2ccc(Cl)cc2Cl)=O)C1 N1(C(Cc2scc(CC)n2)=O)CCCC(CCNC(C2CC(=O)CO2)=O)C1 Cc1noc(C)c1CN1C(C(=O)NCCCCCO)CC2CC12 C(CCCC(C)(C)NC(=O)C1=CCCC1C)NC(C(CCSC)O)=O O=S(=O)(c1ccc(NCC2(C(F)(F)F)CCC2)c(F)c1)N1CCSCC1 C1(C(=O)NCC(=O)OCC=C)CC12CCN(C(C1COCOC1)=O)C2 n1(CCNC(C2(CNC(C(C)=CC=C)=O)CCCO2)=O)ccccc1=O Cc1nn(C)c2c(NCCC(C)CO)nc(=NCCC(C)N(C)C)[nH]c12 Cc1nscc1NC(c1csc(-c2cccs2)n1)c1nnnn1C1CC1 C1(C(N2CCC(O)(C(C)NC(=O)CC3CCCCCC3)C2)=O)CCC(F)(F)C1O Cc1cc(N)c(Br)cc1C(=O)NC1CC(C)(NC(=O)C2=CC(C)(C)C2)C1 C1(C)(C(=O)N)COC(C)CO1.Cc1cccc(C2CC2C(N2CCCC2C)=O)c1 c1(OC)cc(OC)c(CN2CC3CCC2CN3C(c2cncs2)=O)c(Cl)c1 C(=O)(C1=CCN(C(=O)Cc2ccccc2O)CC1)N1C(C(=O)OC)CC1 C1(C(N2CC(F)(CNC(C3(n4cccn4)CC3)=O)C2)=O)(CC)CCOC1 C1(CC(=O)NCC(CC)NC(C2CCC=CCC2)=O)COc2ccccc2O1 n1(CC)nccc1C=CC(=O)NC(C1CCCN1C(=O)CNC(N)=O)C N1(C(C(C(=O)OC)OC)=O)CCC2(CCCC2NC(=O)C(C)C2CCOC2)CC1 C#Cc1cccc(C(N2CCC(NC(=O)Cc3nc4ncccn4n3)C2)=O)c1Cl c1(CC)nn(C)cc1C(=O)NCc1occc1C(N1C2CCC1CC2)=O C(=O)(C(F)(F)C(C)O)N(CCC)CCNC(C1(c2ncccc2F)CCC1)=O C(=O)(C1=C(C2CCC2)N(CCF)C(=O)NC1c1c(C(F)(F)F)cnn1C)OCC C#CC1(O)CCN(C(C2(F)CCCN(C(c3sncc3CC)=O)C2)=O)C1 c1(N(C2CCC2)C(C)C)nnc(-c2cnccn2)n1CCCCc1ccccc1 C(=O)(C(C(=O)N1CCC1CC(=O)NC(CO)CC(C)C)OC)OC N1(C(c2c(C)ccnn2)=O)CCC(NC(=O)CC2CCOCC2)C(C(N)=O)C1 Cc1ncc(CN(C(=O)C(C2CCCO2)NC(C2CC3(CC3)C2)=O)C)s1 C(=O)(CCCC#N)NC(C=CC(=O)N(CC(C(=O)NC)C)C)C CC1CCC(C(=O)NC2CCCCCC2O)CN1C(=O)COc1ccccc1 N1(C(c2cc(OC)ncn2)=O)CCC(N(C(=O)CSc2ccncc2)C)C(C)C1 N1(C(c2c(C)nn[nH]2)=O)CCC(C)C(CNC(c2ccoc2C(F)(F)F)=O)C1 CCCCCC(F)C(=O)NN1CCCC1C(=O)NC1Cc2ccccc2C1 C1(NC(c2c(CC)con2)=O)CCN(C(c2cc(OC)cc(F)c2)=O)CC1F C#Cc1cc(C(=O)NC2CCCC2CNC(c2cc(CC)oc2C)=O)ccc1C c1(C(=O)NC2CCCC(CNC(=O)C=C3CC3)C2)nc2cc(F)ccc2s1 C1(C(N2CC3CC3C2)=O)CCCN(S(N)(=O)=O)C1.C(=O)(C=O)N.C(C)OC C1(C2CCN(C(C34COCC3C4(F)F)=O)CC2)(NC(=O)C2=CCCC2)CCC1 C#Cc1ccc(C(N2CC(C#C)(C(=O)N(c3ccn(C(C)C)n3)C)C2)=O)o1 CC(C(C)C(=O)O)NCc1csc(-c2ccccn2)n1 c1(C(=O)NCC2(F)CC(NC(C3C(C=C)C3)=O)C2)cn(C)nc1SC c1(C(N2CC(NC(COCCCOC)=O)C(OC)C2)=O)ccn2c1CCCC2 CC(C)CS(=O)(=O)CCC(=O)NCCN(C(=O)C(c1ccnn1C)C)CC(C)O n1(CC(=O)NC)[nH]c(=NC(=O)c2cccc(C3(S(C)(=O)=O)CC3)c2)cc1C c1(CNC(C2N(C)CCC2)=O)nc2c(s1)CN(C(c1cc(=O)n(C)o1)=O)CC2 C#CCCCCC(=O)NCC1CCC(F)(CNC(=O)C=CC2CC2)CC1 CCS(=O)(=O)c1ccc(Cl)cc1C(=O)O.c1(C=O)ccc(C2CC2)o1.C(C)C N1(C(=O)OCC)CCN(C(=O)C)CC1.C1(C=O)CC2(CSC2)C1.C(=O)C CC(CNC(=O)Cc1ccco1)CC(F)(F)F.C(C1(C)COC1)=CC=O.N C1(CC(N2C(C(N(C)Cc3ccccn3)=O)CC3CC32)=O)CCC(C)(C)CC1 C1(O)(c2cn(CCNC(C(C)C)=O)nn2)CCN(C(C2CC3(CC3)CO2)=O)CC1 N(C(=NCC(O)c1ccc(OC)cc1)NCc1ccccc1)C(C=C)C N1(CC(C)NC(=O)CSC(F)F)CCN(C(=O)CN2CCCCC2C)CC1 c1(C(N(CC)CCC)=O)ccc(-n2cncn2)nc1.N1(C(C)=O)CCCC1C=O N1(C(c2cn(CCC)nn2)=O)C2CCCC1CN(C(C1CC1C(=O)OC)=O)C2 N1(C(c2cccc(Cl)c2)C(=O)NC2CC(C(=O)OC)C2)CCOCC1C#N C(c1ccccc1F)=CCC(=O)NCCC1(NC(=O)C(C2CCOCC2)O)CC1 C12(NC(CSCC(=O)N(CC)CC)=O)CC3CC(C1)CC(F)(C3)C2 N1(C(=O)NC2CCCN(C3CCCCC3)C2)CCC(=O)C2(CCOCC2)C1 c1(NC)ccc(F)cc1C(=O)NC.C1(C)(C(N2CCCCC2)=O)CC(O)CN1C N1(C(CNC(c2n(CCC)ccc2)=O)C)CCN(C(=O)CC2CCOCC2)CC1 C12(NC(CN3CCC(N(CCCCC)C)C3)=O)CC3CC(CC(C3)C1)C2 c1(C(=O)NCCC(C)NC(=O)C(C)CCO)ccc(O)c2ncccc12 N1(C(c2nn(C)c(OC(F)F)c2)=O)CCN(C(C2CCCC(=O)N2)=O)C2CCC12 Cc1ccc(C(N2CCC(C(C(C)C)NC(=O)COC(C)C)CC2)=O)nc1F N1(C(C2(NC(N)=O)CC2)=O)CCC(NC(=O)C=CCO)CC(O)C1 C12(CNC(c3c(C)ncs3)=O)CCCCC1N(C(=O)CCc1ccncc1)CC2 C1(C(C)NC(c2c(C)nn[nH]2)=O)CN(C(=O)Cc2ccn(C)c2)CCO1 CC(CO)C(C)NC(=O)C#CCNC(=O)Cc1ccnn1C C(=O)(CC1CCN(C(=O)OC(C)(C)C)c2ccccc21)NCCCC(C)=O C1(OC)CC(NC(=O)CCC2CC2)CN(C(C2CC=CCO2)=O)C1 C=CCC(CC)C(=O)NC(C)C(C)NC(=O)COc1ccc(F)cc1 C#CC(C(C)(C)C)NC(C1C2CC2CN1C(=O)CCC(=O)OC)=O CCCC(C)C(c1nnnn1C1CCCCC1)NCc1nc(C(C)C)ns1 C(=O)(C(CC(F)F)NC(=O)C(=O)C(C)C)NC(c1nc(CC)[nH]n1)C c1(OC)cccc(C(=O)NCC23CC2CN(C(C2CC2(Cl)Cl)=O)C3)c1N C(=O)(C(CC(F)F)C1CCC1)NCC(C(C)C)NC(c1coc(Br)n1)=O N1(C(C2C(OCC)C2)=O)CCC(C2CC2)C1.c1(CCC(=O)N)cn(C)nn1 Cc1ccc(NC(=O)CC2(C)CN(Cc3ccsc3)C2)c(Br)c1 c1(CCNC(C(C)OC(=O)CC2CCC(C)(C)CC2)=O)cccc2ccccc12 c1(C(=O)OC)ccc(F)c2c1CN(C(C1CCC3(C1)OCCO3)=O)C2 CC1(C(=O)NCC2(F)CCCN(C(=O)CCc3ccoc3)C2)CCC(O)CC1 C(=O)(C1=NN2CCC(C)N=C2N1)NCC=CC=O.C1(CC=O)CC1.CC c1(OCC(N2CC(NC(CN(C)Cc3ccccc3)=O)C2)=O)ccccc1O C12(CC3CCCN(C(C4(OCC)CC4)=O)C3)CC3CC(CC(C3)C1)C2 C=CCC(CC=C)C(=O)NCC1(Cn2cc(CC(O)C3CC3)nn2)CC1 N1(C(C(C)OCC)=O)CC2CN(C(=O)CCc3nc4ccccc4[nH]3)CC2C1 C1(C(N2CCN(CC(C(C)(C)C)O)CC2)=O)CC2(CCC2)CS1 c1(OC)c(F)ccc(CCNC(=O)C(=O)N(C)CCC2CCCO2)c1F c1(COC)nc(C(=O)NC2CCCC2)n[nH]1.C(=O)(C(C)Cc1ccncc1)N c1(C(N(C(C)C)C)=O)cc(C(N)=O)no1.C(=O)(C=CC(=O)N)OCC c1(CC)[nH]nc(C(=O)NCCC2CCN(C(c3cn[nH]c3)=O)C2)c1C c1(C(N2CCN(C(CCCCSC)=O)C(CO)C2)=O)[nH]nc2ncccc12 Cn1cncc1CCC(N1CCC(NC(C2CC(C)(O)C2)=O)C1)=O C1(=CC(=O)N(CCNC(c2ccc(CSC)cc2)=O)C)CN2CCC1CC2 N1(C(C(CCCC)O)=O)CCC2(CC1)CC(CNC(=O)C1=C(C)CCC1)C2 C1(NC(C(CCC2CCC2)NC(C2C(OC)CCC2)=O)=O)CCn2cnnc2C1 N1(C(CCOCCOCC)=O)CCN(C(c2nocc2Cl)=O)CC1CC(F)(F)F C1(CCOC)CN(C(C2CCCN(c3nc(C(C)(C)C)ns3)C2)=O)CCO1 CC(C)(C)C(C)(O)C(=O)NC1CCN(C(c2nccc3ccsc23)=O)C1 Cc1c(C(N2CCC(C)(NC(c3ncn(C)n3)=O)C2)=O)ccc2c1NC(=O)C2=O C12(NC(CC(C)OC)=O)CCCC1(F)CN(C(=O)CCC(C)(F)F)C2 O=C1NC2CCC1CN(C(=O)C(Cn1cncn1)NC(C1CCSCC1)=O)C2 C(=O)(C#CC1CCOCC1)NCC1CN(C(C2(OC)CCCOC2)=O)CC(C)C1 C=C(C)CC(C(=O)N(CCC(=O)NCC(O)(COC)CO)OC)OC C(=O)(C(C)(CCC)CCC)N(CC(=O)NC(CCC)C(N)=O)C1CC1 C1(NC(=O)CO)CCC(CNC(c2ccoc2Cl)=O)CC1 C1(O)(CNC(CC2C(=O)NC(=N)S2)=O)CCCN(C(=O)C(C2CCCCC2)O)C1 c1(C(=O)Nc2nccn3cc(Cl)cc23)ncc(C2=CCC(C(F)(F)F)CC2)cn1 c1(OC)c(C(=O)N(CCCCCNC(C2(C)CC2F)=O)C)cc(Cl)cc1Cl N1(C(C2C(C)C2)=O)CCOCC(NC(c2cc(-c3ccco3)c[nH]2)=O)C1 C(=O)(C1=Cc2ccccc2C1O)N(C)CC1CN(C(c2cnccn2)=O)CCO1 Cc1cccc(C)c1C(C)NC(=O)C(=O)NCC1CCOC(C)C1 C1(NC(=O)Cc2ccoc2)CCCN(C(=O)CCC2CCCCO2)CC1 c1(CC)[nH]c(Cl)nc(=NCC2CN(C(c3cnn(CC)c3)=O)CC2(C)C)c1C#N c1(OC)coc(C(=O)NCC2CCCC(NC(=O)C=CBr)C2)cc1=O N1(c2cc(OCC)ncn2)C2CCC1CN(C(=O)C(C)C(C)C)C2 c1(CC(=O)Nc2ccc(CCN3CCC(O)CC3)cc2)cc([N+](=O)[O-])ccc1F C(=O)CC(C)CC(F)(F)F.Cc1c(C(=O)NCCC2CC2)ccn1C1CC1.N c1(C=O)ccc(Cl)c(Cl)c1.C1(N(C(=O)C)C)CCCCC1.C1(C(=O)N)CCC1 C1(C(NOCCC(=C)C)=O)CN(C(C2(n3cnnn3)CC2)=O)CC12CCC2 N1(CC)CCCN(C(=O)CCC2CCN(C(=O)CC3CCCOCC3)C2)CC1 N1(C(C)=O)CCC(CN=c2ccn(-c3nnc4cccnn34)[nH]2)C(C2CC2)C1 O=C(CC(F)F)NCC1COCC1NC(c1nn[nH]c1Cl)=O c1(CC)nc(C(=O)N(C2CCCCC2)C)c(N)s1.c1(CC(=O)N)cnn(C)c1C CCC(C)C(C(=O)NCC1CN(C(c2cc[nH]c(=N)c2)=O)CCO1)NC(N)=O C(=O)(C(C(=O)NCC(CCNC(=O)CCc1cnc[nH]1)OC)C(C)C)OC C1(CNC(CCCN(C(c2nc(CC)oc2)=O)C)=O)CC12CCOCC2 C(CC(=O)NC(c1ccncn1)C)(CC(C)C)NC(C1(OC)CCSC1)=O c1(C(N2CCN(C(C3C(C)CC=CC3)=O)C3C2C3)=O)ccn2cncc2c1 CCC(C)CCCCC(=O)NC1CN(C(c2cc(Cl)ccn2)=O)C2CCCC12 c1(C(N(C)CC2(NC(C(C(CC)(C)C)O)=O)CC2)=O)cccc2c1CC(=O)N2 C1(C(N(CCC)CC)=O)CS(=O)(=O)CC12CCC2.c1(C=O)cccc(C)c1.N N1(C(C2CC(=C)C2)=O)CCC(C2(O)CCN(C(C3C4CC5C(C4)C35)=O)CC2)CC1 c1(C(C)NC(=O)C(=O)NC2CC(N)C2)ccc([N+](=O)[O-])cc1 c1(CC(=O)NC2CN(C(CCCCCC)=O)CC(O)C2)c[nH]c2c(C)cccc12 C#Cc1ccccc1CC(=O)NC1CC2CC(NC(=O)CCc3cncs3)C2C1 CC1C(C(N2CC(C)C2(C)C)=O)CCN1C(=O)CCc1ccccn1 C(=O)(C1=CCC(F)(F)CC1)NC1CCCC(CNC(c2c(N)cncc2)=O)C1 N1(C(=O)NC)CCC(C(N2CCCC2)=O)CC1.C1(CC=O)CC(N(C)C)C1.C c1(CNC(=O)CC2CCN(CC(F)(F)F)C2)ccc2c(c1F)CCC2 N1(C(c2ccc(C)c(O)n2)=O)CCC(C)(C)C(C(=O)NCc2cocn2)C1 c1(C(=O)NC(C)CCNC(=O)C(N2C(C)CCC2C)C)cc(O)c2ccsc2c1 c1(SC)cscc1C(=O)NCC(C)(C)NC(=O)CCC1CNC(=O)N1 C(C)(CO)(C(=O)N1CC(C=O)(SC)C1)NC(C)=O.C1(CC)CCCC1(C)C.N C12(NC(c3c(C)c(=O)cc[nH]3)=O)CCC(CC1)N(C(=O)CCC1CCOC1)C2 c1(C(C)C(=O)NC(C2CCN(C(=O)C=CCF)C2)C)cccc(F)c1 N1(C(C2(SC)CCC2)=O)CCC2(CCCN(C(=O)CC3CNC(=O)C3)C2)C1 O=C(O)CCC(CC1CCCCC1)NC(c1cc(Cl)c(Br)cn1)=O N1(C(Cc2c(C)con2)=O)CCN(C(=O)CC2COC(C)(C)C2)C2(CCC2)C1 N1(C(C(C2CCOCC2)C)=O)CC2CC2(C(=O)NCCC2(C)CC2(F)F)C1 c1(C(N2CC3CC(NC(CC(C)C(F)F)=O)C3C2)=O)cc(F)c(F)cc1F n1(CC)cnc2[nH]c(=NC3CCC4CCC3C4)nc(N3CCn4ncnc4C3)c12 C1(NC(C=CCC)=O)CCCN(C(c2cn(C3CCCC3)nn2)=O)C1 c1(N2CCC(C)(N(C)C)CC2)[nH]c(=NCC2CCC3CC23)nc2scnc12 C(CCCC(=O)N1CC2CC2(NC(C2CC2(C)C(F)F)=O)C1)NC(C)=O C1(C(N2CC(N(C)C(C3CCSC3)=O)C2)=O)C2CCN1CC2 O=C1NC(=O)C2(CCCN(C(=O)NC3CC(NCC4CC4)C3)C2)O1 c1(C(N2CCCC(c3ncc(C)s3)C2)C(=O)NCC)cc(C)c(Br)s1 C1(C(N(CC(=O)NC2CC(C(C)O)C2)C2CCC2)=O)CC2(C1)CC21CC1 CCC(C)(COC)C(=O)NCCC(O)C(=O)NCC1CC1(F)F CC(C)C1=NOC(C(N2CCCC(C(=O)N(C)Cc3ccco3)C2)=O)C1 C1(C(N(C(C(=O)N2CC(C(=O)NCC)C2)(C)C2CC2)C)=O)CCCCC1C c1(C(N(CCOCCCN(C(c2c(CC)nco2)=O)C)C)=O)cccnn1.O C(=O)C(C)(C)C(C)(C)C.N1(C(C(C(C)C)NC(N)=O)=O)CC2(CCC2)C1.N C1(OC)CN(C(C2(C(F)F)CCCO2)=O)CC1.c1(C=O)ccc(C(F)(F)F)o1 C1(NC(CN2CCC(C)C2)=O)CN(C(=O)CCc2ccon2)CCC1(C)C C1(O)(CN(C(C2N(C(C(C)C)=O)CCC2)=O)C)CCN(C(c2cnsc2)=O)CC1 CC(CC(F)F)C(=O)N1CC2CC(NC(=O)C=Cc3ccsc3)C1C2 CC1CCCCC1CNC(=O)NC1CCCCC1c1ccc(F)cc1 c1(C(=O)NC2(C)CC(NC(C(CCC)O)=O)C2)cc(C)cc(C)n1 O=C1CCC2(CCCN(C(=O)NCCCC3CCCC3O)C2)CN1 N1(C(c2[nH]c3ncc(C)cc3c2)=O)CC(NC(=O)C(Cl)=CCl)CC12CCOCC2 C1(CC)CCCCCCN1C(C1COCC1NC(=O)Cn1ncccc1=O)=O C1(CC(=O)NCC2CCCCN2C(C2CC(O)C2)=O)NC(=O)NC1=O C#CCC(CC(=O)NCC(C)(C)CO)NC(c1c(CO)n[nH]c1C)=O Cc1nc(NCCCCC(N)=O)cc(=NCc2cc3c(nc2O)CCC3)[nH]1 C(CN(C(=O)CCc1ccon1)C)(CO)(CO)NC(c1c(CC)n[nH]c1)=O C1(NC(=O)C(c2ccccc2)O)CC2CCC1N2C(c1cnc(C(F)(F)F)s1)=O c1(C(=O)NCC2(NC(C3CCCC(C)(C)C3)=O)CC2)cncc2c1CCC2 N1(C(c2c(C)noc2C)=O)CCN(C(=O)C(C)C#N)C(CCO)C1 Cc1cc(Br)ccc1C(N1CCC(C)(CNC(C2CCN(C)C2C)=O)CC1)=O C1(CN(CC(F)CNC(=O)OC(C)(C)C)C)CCCN1c1cccnn1 C1(NC(C=CCCC)=O)(CO)CCCN(C(c2c(C(F)(F)Cl)n[nH]c2C)=O)C1 N1(C(CC(C)CN(C)C)=O)CC(CNC(c2c[nH]c(=N)o2)=O)CC12CCC2 C1(COC)CCCCC1C(=O)NCC1CC1.c1(C=O)conc1C1CC1 C1(CNC(Cc2c(C)ocn2)=O)CN(C(=O)C(C)(C)CC2CC2)CCC12CCC2 C(=O)(C1=CCCOC1)NC1(C2N(C(CCc3n(C)ncc3)=O)CCCC2)CC1 CC1CCN(C(=O)CC2C=CCCC2)CCN1C(=O)COCc1cccnc1 N1(C(=O)CC2CC3CCC2CC3)CCc2ccccc2C1c1cccnc1 C(=O)(C(CCNC(=O)CC1CC=CCN1C)OC)NCc1ccc(CC)s1 C1(NC(C2CC2)=O)CCCCCCC1O.C12(COC)CN(C1)C2=O.C1CC1.C N1(C(C2C(COC)CC2)=O)CCN(C(c2ncnc(O)c2F)=O)C2(CC2)C1 N1(C(CC(C)(C)OC)=O)CCC(C)C(CC(=O)NC2CC(O)C(O)C2)C1 CC1(C)CN(C(C2Cc3nncn3C2)=O)C(CNC(c2cnccn2)=O)CO1 Cc1nc(=N)[nH]cc1C(=O)NC1(CO)CCN(C(=O)C(C)c2ccco2)C1 C1(C(CC)NC(C2(F)CNC2)=O)CCCOC1 c1(CCOC)nc(=NC(CNC(=O)CC(C)OC)c2ccccc2OC)s[nH]1 c1(CC)ncsc1C(=O)NCCC(C)NC(=O)C(=O)NCC(F)(F)F N1(C(C(Cc2c(C)nn(C)c2C)C)=O)CCN(C(=O)CS(C)(=O)=O)CC(CO)C1 C1(C(=O)NC(C)CC2CN(C=O)C2)(COC)C=CCC1.C(C)(C)C.O c1(C=O)cc(F)c(Br)cc1F.c1(C(C)(C)N(C)C)cn(CC2(O)CCC2)nn1.N c1(C(N2CCCC(N(C(=O)C(O)CF)C)C2)=O)cnn2ccn(C)c12 N1(C(c2c(NC)scn2)=O)CCN(C(C2CSCCS2)=O)C(C(C)C)C1 C(CCC1CCCC1)(C(=O)NC(=O)NCCC#N)N(CC(F)(F)F)CCC c1(C(N(C2CCN(C(C3C(CC)CCO3)=O)C2)C)=O)ccc2ccncc2c1 C=C1COc2c(C(N3CCOCC(NC(=O)Cc4csc(C)n4)C3)=O)cnn2C1 c1(C(N2CCN(C(COC)=O)C(C3CCC3)C2)=O)ccc2ccccc2c1C c1(C(C)=O)cccc(OCC(=O)NCCCC)c1.c1(C=O)cnoc1C(C)C.N c1(CC)cccc(C(=O)NC(C)(CO)C(=O)NCC2(C)CCCO2)c1 c1(C=O)ccc(CC(N)=O)cc1.c1(CC)sccc1C(=O)NC1(C)CCC1.N n1(CC)cc(CC(=O)NCC(F)(F)CN2CCCC2)c(C)n1 CCCCC(C)CCC(=O)N(C1CC(C(=O)Nc2cnn3c2OCCC3)C1)C CCC(C)(C(=O)NC1CC(F)(C)C1)OC.c1(C(C)=O)ccccc1.C(=O)C.N Cc1cc(C(N2CC(NC(C3CC3F)=O)C3(CC3)C2)=O)n2ncnc2n1 CCC(CC(=O)NC(C)(C)C(=O)NO)NC(C1OCCC1CC)=O c1(C(=O)NCc2scc(C(=O)NCCC(CC)CO)c2)cc(F)cc(F)c1 C(=O)C(O)P(C)(C)=O.c1(OC)ccccc1OC.C(=O)(CC)N(CC)CC Cc1ccc(SCCNC(C2CCCN2C(c2cnco2)=O)=O)cc1 c1(C(N2C(C)C(NC(C34CC5CC3C4C5O)=O)CC2)=O)cnn2c1N(C)CC2 c1(N(C)C)cccc(-c2ccc(C(F)(F)C(F)(F)F)cc2)c1 N1(C(c2ncc(Cl)s2)C(=O)NC)CC(OC(C)(C)C)CC(O)C1 N1(CCC)CCN(C(=O)CN(C2CCC2)C)CC1.C1(C(C)C)(C(=O)N)COC1 c1(OC)ccc(F)c(C(=O)NC2CCN(C(=O)CCF)CCC2CO)c1OC N1(C(C2OCCN(C(c3c(C#C)cn(C)n3)=O)C2)=O)CC(C)(C)OCC1CC C1(C2CCOCC2)(C(=O)NC2CCCC(NC(Cc3cn(CC)nc3)=O)C2)CC1 c1(OCC)cccc(-c2noc(C(C3CCCC3)CC)n2)c1 C1(C2(O)CN(C(c3nsc(OCC)n3)=O)C2)(CNC(C(CCCC)C)=O)CC1 CC1(C)CN(C(c2ccnn2C2CC2)=O)CC1C(=O)NC(CO)C1(C)CC1 Cc1cc(Br)ccc1C(=O)NC1CN(C(=O)CC(O)C(C)C)CC1(C)C C1(C)(SCc2cn(C(CCSC)C(N3C4CCC3COC4)=O)nn2)CCC2CC2C1 C1(C(=O)NCCCC)CCC(C(F)F)CC1.C1(O)(C(C(=O)N)(F)F)CCCCC1 N1(C(C(C)N(C(=O)C(F)=CC2CC2)C2CC2)=O)CCN(C(C)(C)C)CC1 c1(C(N2C(C)C(NC(=O)CCc3cccc(F)c3)CC2)=O)nc[nH]c2nccc1-2 n1(CC(C)O)cc(C(=O)NCC2CCCN2C(C2CC2(C)Br)=O)ccc1=O CC(C)C(CN(C)C)C(=O)NCC(F)CNC(c1[nH]ccc1C1CC1)=O CC(CC(=O)N1CCC1CNC(=O)CC1CCS(=O)(=O)CC1)CC(F)(F)F c1(C2CC2)ccccc1.CC(C=O)O.CCCN(C(=O)CC1(C(F)F)CC1)C [N-]=[N+]=NCCCC(=O)N(C1CCCC1)CCCNC(c1cnc2n1CCC2)=O C1(NC(C2CCCC(OC)C2)=O)CN(C(=O)C2=CCCC2)C2CCCCC12 c1(C(C(=O)NCCOC)N(C)CC2(C)CCCO2)nc(F)ccc1Br c1(C(=O)NC2CC(CNC(c3ccc(C)nc3)=O)CC2O)c(C)nn(C)c1Cl C#CC1(O)CC(C(N2CCC(O)(C(C)NC(=O)CC3CCCC3)C2)=O)C1.C c1(OC)ccc(CN2CCN(c3cccc(C(N4CCC(O)C4)=O)c3)CC2)cc1 C1(C(N(CCC(=O)NC(C)CC2(O)CCC2)CC=C)=O)CCC(C#N)CC1 N1(C(c2n(C)ccc2)=O)CC(F)(F)CC1(C)CNC(C1(O)CCOC1)=O C#CCCC(C(=O)N1CCC(O)(C=C)C1)NC(C1COCCC1C)=O C1(C(=O)Nc2c(O)cccc2F)C2CCC1CN(C(=O)CCN1CCCCC1)C2 N#Cc1ccc(C(=O)NC2(CCNC(=O)CC3CCCC(O)C3)CC2)[nH]1 N1(C(CCCN(C(=O)OC)C)=O)CCCC(C2CC2)C1.C(=O)(C(F)C(C)(C)O)N N1(C(c2cncc(NCc3ncc(C)cc3F)c2)=O)CCc2ccc(F)cc2C1 c1(CCCOC)nc(-c2ccc(CF)cc2)nn1-c1ccc(OCC(F)F)cc1 N1(C(c2ccc(C#C)nc2)=O)CCC2CCN(C(=O)C(O)CC(F)(F)F)C2C1 N1(C(C(CC)C2CC2)=O)CCC2(CC1)CC(NC(C1(n3cncn3)CC1)=O)C2 Cn1cc(S(N)(=O)=O)c(C(N2CCCC(NC(=O)Cn3ccnn3)CCC2)=O)n1 c1ccsc1[N+](=O)[O-].Cc1nc(C(=O)N(CC(O)CNC(=O)CS)C)c(C)s1 Cc1ccc2ncc(NC(c3ccccc3S(=O)(=O)N3CCCC3)=O)cc2c1 C1(CN(C)Cc2c(C)nn3cccnc32)CCC(N=c2[nH]nc(C#N)s2)CC1 CC1(C)CN(C(c2cccc(=S)n2O)=O)CCC1NC(=O)CC1COCC1O Cc1cccc(C(=O)NCCC(C)NC(=O)C(C(C)C)c2cccnc2)c1F c1(C(=O)NCCCCC2CN(C(COC(C)(C)C)=O)C2)cnc2[nH]nnc2c1 N1(C(C2CC2)=O)CCC2(CC1)C(N(C(=O)C(C)=C1CC1)C)CS2(=O)=O.C CC1(C)CN(C(=O)CC2CC=CC2)CCN(C(c2csc(Br)n2)=O)C1 C1(NC(CCC(C)CN(C)C)=O)CN(C(c2ccccc2O)=O)CC2(CCC2)C1 C#CC1CCC(C(N2CCN(C(=O)COC(C)C)C(c3cccnc3)C2)=O)CC1 O=C1CCCCn2nc(C(N3CCC34CN(C(C3CS(=O)(=O)C3)=O)C4)=O)cc21 c1(C2C(C(=O)N)C2)ccccc1F.CN1CCCC1CCC(=O)NC12CC(C1)C2 C(CN=c1nc(NCCc2ccnn2C)[nH]c(N2CCOCC2)n1)=CC C1(C(=O)NCC2CCN(C(C(CCC)(C)O)=O)C2)CC(C)(C)CC(C)(C)C1.O S(=O)(=O)(C1(Cl)CC12CCNCC2)N1CCC(OCC(N)=O)C1 N1(C(C(C(C)C)SC)=O)Cc2occ(C(=O)NCC(C)(C)C(F)(F)F)c2C1 N1(C(C2C(CC(C)(C)C)C2)=O)CCC(C)(C)CC1.CC(C)(C)C.C(=O)C.C S(=O)(=O)(c1cccc(C#N)c1)NCc1c(C)ncs1.C1CC2(C1)CC21CCC1.N CC(C)=C=CC(=O)NCC1CCCCC1C(=O)NC(c1cnsc1)C c1(C(=O)NC2(C)CCN(C(C3CCC4(CC3)CC4)=O)C2)cncc2nc[nH]c12 c1(OC)ccccc1C(N1CCCC1)CNC(c1ccsc1)C C=CC(CCC)CC(=O)N1CCCC(C(=O)NCCNC(c2cc(F)cs2)=O)C1 CC(C)(C)C#CC(=O)NC1CCN(C(c2cccnc2SC(F)F)=O)CC1CO CN1CCN(C2CCN(C(=O)CSc3nn[nH]n3)C2)CC1 c1(OC)ccc(C(=O)NCc2cn(C(C)C(=O)NCC(F)Br)nn2)cc1 c1(NCCCN(C(C)=O)C)nc(Oc2ccccc2)c2ncn(C)c2n1 C1(CNC(C2CC3(CC3)CO2)=O)CN(C(=O)CCc2ccncc2)CCC1(F)F C1(CC)CN(C(=O)C=CS(C)=O)CCN1C(=O)Cc1ccc(C)s1 c1(NCC(CO)N(CCC)C)ccc(C(F)(F)F)c(C)c1 c1(CC(=O)NCC2C(NC(C=CCC)=O)C2)cccc(Br)c1C C(=O)(CCC(=O)N(C(C)(C(=O)N1CCC(c2cnn[nH]2)C1)C1CC1)C)N(C)C c1(OCC)cc(O)ccc1C(=O)NCCc1ccccc1.C1(C=O)CC1.N C1(NC(CCc2n(C)cnc2)=O)C2CC1CN(C(c1cc(C(F)F)n(C)n1)=O)C2 C1(C=O)CS(=O)(=O)CC(=O)N1.N1(C(c2n(C)c(S)nn2)=O)CC2(CC2)CC1.C C(=O)(C1=CC2(CCN(C(c3cc(F)ccc3O)=O)C2)C1)NC1CC(C=C)C1 c1(SCC(N2CC(CCCNC(C(C)C(F)F)=O)OCC2)=O)cccc(C#N)c1 CC1CC2(CC(C(N3CCCC3C(=O)NCCOC(F)F)=O)C2)C1 C1(N2CCC(NC(=O)CC3CSC3)C2)CCN(C(=O)Cc2cnns2)CC1 C(CCCC(=O)NCc1cnccc1C)NC(C1(CC=C)CCCC1)=O c1ccc(C)nc1O.C1(C)(CC)CC(C(=O)NCC2(C(=O)N)CCCO2)C1 CC1CCC(CNC(C2CC(=O)C23CCC3)=O)N(C(c2cc(Cl)no2)=O)C1 N1(C(c2c[nH]c(=NC)o2)=O)C(C(=O)N(C)Cc2ocnc2C)CC2CCCC12 C1(NC(C2(C#C)CC2)=O)CCCCN(C(c2cnn(C(C)(C)C)c2CC)=O)C1 c1(C(=O)NCCC2CN(C(c3cn(C)nc3)=O)C2)c(F)ccc(Cl)c1N c1(C=O)cc(C(C)(C)C)n[nH]1.C1(O)(CC)CN(C(=O)CC2CCC(O)C2)C1 CCC(C)C(CNC(=O)C(CN(C)C)NC(C1CC12CCCCC2)=O)CO [SH](=O)(=O)c1ccc(Cl)s1.C(C(C)(C(=O)NCC(C)NC(=O)C)OC)OC Cc1cc(C)c(C(=O)NC(CC(N2CC(O)CC2(C)C)=O)C2CC2)cn1 c1(C(=O)NC(C(C(C)C)NC(Cn2ccc(C)n2)=O)C)n[nH]c2c1CCC2 c1(C=O)nc[nH]c2ncnc1-2.C1(O)(CC)CN(C(=O)C=CCN(C)C)C1.N C1(NC(=O)CSC(F)F)CC=C(C(=O)NC(c2nc[nH]n2)C2CC2)C1 C1(NC(c2ncoc2C2CC2)=O)CCCC(NC(c2ccc(Br)s2)=O)C1 N1(C(C2CC(C)C2)=O)CCCC(C2(NC(=O)CSc3ccccc3)CC2)C1 c1(C(=O)NCC(C(C)(C)C)NC(C(CCC)(C)O)=O)c(C)cc(C)nc1Cl N1(C(CSCC#C)=O)CCCC(C)(C)C1C(=O)N(CCOC)CC C1(N(C(Cc2c(SC)cccc2)=O)C)CN(C(C2(O)CCC2)=O)CC12CC2 c1(C(CNC(c2scnc2Cl)=O)NC(=O)C(O)C2CC2)ccc(F)cc1 c1(C(C)C(=O)NC2CC(CNC(=O)C(C)(C)N3CCCC3)C2)ccc(Cl)cc1 C(=O)(C(F)(F)C(O)C(C)C)NCC1(O)CN(C(C(CC)O)=O)C1 CCC(C)(CO)C(=O)NCCCCCCN(C)C(C1CN(C(C)=O)CCO1)=O CCC(C(=O)NCc1cn(CCNC(=O)Cc2cncnc2)nn1)C(C)O Cn1[nH]c(=NC(=O)c2ccc(C(F)(F)F)c(Cl)c2Cl)c2ccccc12 O=C(C1=CCCS1)NC(C1CCOC1)CNC(c1cnc[nH]1)=O c1(CN(C(CC2(OC)CN(C(C3(C)CSC3)=O)C2)=O)C)ccc(C)cc1 CC1C(NC(c2ccc(=O)oc2)=O)CC2CCC1N2C(=O)C(c1ccccc1)=O C1(C(=O)NCC(C)N(C(CC2(OC)CCCC2)=O)C)CCC(F)(F)CC1(C)C c1(C(N2C(CNC(c3ccnc(F)c3)=O)CC2)=O)cnc2[nH]c(O)nc2c1 C(C(CC(C)C)C(=O)NCC(CC)C(C)C)NC(C1CCN(CC)C1)=O c1(C(N2C(C)CCC2)=O)cn2c(n1)CCC2.CC(C)CC1(C(=O)NC)CC1 N1(C(CCOC(C)=O)=O)CCC(C)C(NC(C2(C)CC(F)(F)C2)=O)C1C Cc1cc(NC(c2ccc(COCCO)cc2)=O)ccc1Sc1cccc(Cl)c1 C1(C(=O)NCCC(=C)C)Cc2ccccc2C1(C)C.c1(CC(=O)N)nnc(C)o1 c1(SC)cc(C(F)(F)F)ccc1O.c12nnnn1C1CC(C1)NC2C1CC1 N1(C(c2cc(C(N)=O)no2)=O)CCCN(C(=O)C(O)C2CC2)CCC1 Cc1[nH]c2cc(Br)ccc2c1C(=O)NCC(C)N(C)C(C1CC1F)=O Cc1cc(Cl)ccc1OCC(=O)NCC(C)NC(C1(C)CC2CC2C1)=O CN1CCc2cc(C(=O)NC3CC(CCNC(=O)CC4CCOC4)C3)ccc2C1 c1(C(=O)NC2(C)CC(NC(C(C)C(C)O)=O)C2)cc2cccc(Cl)c2cn1 C1C(C)(C)C(O)C1(C)C.C(CNC(=O)CCc1cc(C)[nH]n1)(C=O)OC.N Cc1cc(F)cc(C(N2CCC(CF)(NC(=O)C(C)CCO)C2)=O)c1N C(=O)(C(C1CCCC1)NC(=O)Cn1cccn1)NC1(C(C)O)CC1 C(CCC(CO)NC(c1n[nH]c(C)c1C)=O)NC(C1(CC=C)CCCC1)=O c1(C(=O)NCCC(C)(C)NC(=O)CNC=O)cc(Cl)c(F)cc1F C1(NC(C(C2CC2)NC(c2ccc(COC)o2)=O)=O)CCCCC1C#N c1(C(N2CC(NC(c3cc(OCC)ncc3)=O)C3C2C3)=O)ccc(OC)cc1C C1(C(=O)NC)CCN(C(=O)C(C)(C)C2CCN(C(c3nc(CN)co3)=O)C2)CC1 c1(OC)ccc(C(N2CCOC(CCNC(c3sccc3OC)=O)C2)=O)cc1 Cc1cc(C(=O)Nc2ccc(-c3ccc(CO)o3)s2)c(C)cc1Br C(=O)(CCOC1CCC1)NCCN(C(C1CC1Cl)=O)CC n1(CC)cc(C(c2ccccc2)N(C)CCc2cnn(C)c2)nn1 C1(N(C(=O)CCC2CC2)C)CCCN(C(=O)C(C)(C)c2ccns2)CC1 c1(C(=O)NCC2CC(NC(C(CCC)C)=O)C2)ccc2c(c1)NC(=O)CO2 C=C1CN2C(=O)CCC2(C(=O)NC(C)C)C1.c1(C=O)ccc(C(C)=O)[nH]1.N C=CC(C)(O)CC(=O)NCc1ccc(C(=O)NCC2CC23CC3)cc1 CS(=O)(=O)C1CCCN(c2ncnc3c2ncn3CCC2(CO)CCC2)CC1 c1(CN(C(C(C2CC2)OC)C(=O)NCC(F)F)C)cc(Cl)c(F)cc1F n1(CC)nc(C(N2CCC(N(C(=O)CCS(C)=O)CCO)C2)=O)cc1C1CC1 c1(C(N2CCN(C(C(F)=CC)=O)C(CO)C2)=O)cc2c(=O)[nH]ccn2c1 c1(NC(c2cc(C#N)cs2)c2n(C(CC)C)nnn2)ccc(OCCO)c(C)c1 O=C1CCCc2cc(C(N3CCC(Oc4ccc(Cl)cc4)C3)=O)ccc21 C(CCS(=O)(=O)C(F)(F)F)NC(C(C)(C(F)F)c1ccccc1)=O N1(C(CNC(CNC(C)=O)=O)=O)CCCC(C)C1.c1(C=O)cc(=N)[nH]n1C.C C1(COC)CN(C(C2(Cl)CC2)=O)CCN1C(c1cc(CO)ccn1)=O Cc1ccc(CN2CCC(N(C)C(c3ncc(C)s3)=O)C2)c([N+](=O)[O-])c1 c1(N2CCN(C(C3CC3C3CC3c3ccccc3)=O)CC2)ccc(F)c(F)c1 CC(C)CC(C(=O)NCc1cc(F)ccc1O)NC(c1cnn(C(C)C)c1)=O CCC(O)C(C)C(=O)NCc1occc1C(=O)N(CC(=O)OC)CC c1(C(=O)NC2CN(Cc3cn(CC)nc3)CC2C#N)cc2cccc(Br)c2[nH]1 c1cccnc1.c1(N(CCC(=O)N(C)CC2CC2)C)ncccn1.C(=O)(C)N C1(C(N(CCNC(C(C)C2CC2)=O)CC)=O)CCN(C)C(=O)C1.CCO.O C(=O)(CC1=CCOCC1)NC1CC(C(=O)NC(C)(C)CC(F)(F)F)C1 C=CC(CCC)CC(=O)N1CC(N(C(=O)C2=NOC(CC3(O)COC3)C2)C)C1 C(=O)(C(O)CCCNC(c1cccc(C)c1C)=O)NCC(CC)C#N C1(NC(Cn2ccc(C)n2)=O)CN(C(c2ccc(N)c(F)c2)=O)CCC1(C)C N1(C(=O)CSC2(O)COC2)CC2(C(=O)Nc3ncccn3)CC1CO2 C(C=O)(C(C)C)OCC.C1CN(C(=O)C)CC1C(F)(F)F.[SH](C)(=O)=O [N-]=[N+]=NCCCC(=O)NCC(C1CCOC1)NC(c1cc(O)ncc1Br)=O C1(C)(C(NCCC(N2CCC(C(=O)NC)C2)=O)=O)CNC(=O)N1.C1CC1 C(=O)(C1CCc2nccn21)N1CC(NC(=O)Cn2ccccc2=O)(CO)C1 N1(C(CC2(COC)CCOCC2)=O)CCC(N(C)C(=O)C2CC2)C(COC)C1 C(=O)(C#CC1CCOC1)N1CC(CCNC(C2(CC(C)C)CC2)=O)C(C)C1 C1(NC)CCCN(c2ccnc(N(C)CC3CCCS3(=O)=O)n2)CC1 c1(CC)ccc(F)c(C(N2CCCC(O)(CCNC(=O)CCCC(C)=O)C2)=O)c1 C1(NC(C=CCCC)=O)CN(C(=O)CC(C)(C)C)CC(F)(F)C1.C(C)(=O)O n1(CCC(C)C)cc(C2(O)CN(C(C3CCC(=O)C3)=O)C2)nn1 Cn1nc2c(c1NC(=O)CC1CCCN1Cc1sccc1Br)CCCC2 Cc1ccccc1CC(C)C=O.C1(C(F)(F)F)(C(N(CC)C2CC2)=O)CCC1 CC1=NN(C)C(=O)C1CC(N1CCCCC1c1cn(CC2CCC2)nn1)=O FCCCN=C(NCC12CCCC(C1)OC2)NCC1CC1 N1(C(c2ccnc(C)n2)=O)CC2CCC(C(=O)NCCC(F)(F)F)(C2)C1 N1(C(c2c(C)nn[nH]2)=O)CC2CCC1CC2NC(=O)C(C1CC(F)(F)C1)O C1(CC(=O)NC(C2N(C(CCC)=O)CCC2)C)CCCN(C(C)C)C1 c1(CC)cc(NCc2cccc(Br)c2)n2nc(C(=O)O)nc2n1 C(=O)C1=CC2C=CC(C1)C2.C1(NC(=O)C(C)CC2CC2)CCCCCC1CO.N C1(C(=O)NCc2c(C)cn(C)n2)CCN(C(=O)CCC2CCCN2C)O1 c1(CNC(=O)C(F)CC2CC2)cccc(C(F)(F)F)c1 CCC(CC(=O)N1CCOC(COC(C)C)C1)NC(=O)C(C(C)C)NC=O c1(C(=O)NCC(CNC(CCN(CCCCOC)C)=O)O)nccn2ccnc12 C1(CNC(C(N2CCOCC2=O)C)=O)CN(C(=O)Cc2sc(O)nc2O)CC1O c1(C(=O)NC(C(C)NC(c2cn(CC=C)nn2)=O)C)nc2ncc(Br)cc2[nH]1 C1(C(=O)NCC23C(CN(C(C=C(CC)C)=O)C2)C3)CCCC2(CC2)C1 Cc1cc(Br)cc2c(=O)c(C(N3CC(CNC(=O)C(C)(C)C)C3)=O)c[nH]c12 c1(C=O)ccnc(Cl)n1.c1(CC)noc(COCC(=O)N)n1.C1(CC)CC1 C#CCC(CC#C)C(=O)N1CCC(N(C(=O)C=CC(=O)OCC)C)C1 CC(=O)n1cc(-c2cnc(C(=O)N(c3cccc(N(C)C)c3)C)nc2)cn1 N1(C(C2C(C)OCCC2)=O)CCOC2(CCN(C(=O)CCOCC(F)F)CC2)C1 Cc1c(-c2cn(C3CCCC3NC(C3CCC(C(=O)O)O3)=O)nn2)cccc1Cl Cc1nn(C2CC2)c(Cl)c1C(=O)N(CCCF)C N1(c2c(S(=O)(=O)NCC(C(CC)C)C)cncc2)CC=C(c2ccccc2)CC1 c1(C(N2C3CC(NC(C(CC)F)=O)C3CC2)=O)ccc2c(c1)CCC2 C(=O)(C(CCOC)NC(=O)Cc1cnn(CC)c1)NCC(=O)OCC C(CC(C)(C)C)(C(=O)NC1CC2CC1CN(C(C1(OC)CCOCC1)=O)C2)OC N1(C(C23CCC(CN(C(Cn4c(C)nnn4)=O)C2)C3)=O)CCCC(C2(C)CC2)C1 Cc1cc(-c2ccnc(C#N)c2)cnc1C(=O)OCC1CCC(C)O1 C(=O)(C(C)(C)S(C)(=O)=O)N1CCCC(N(c2ncc(C(C)=O)cc2C)C)C1 c1(OCCC(N)=O)ccccc1C(=O)N.C1CCCCC1.C(=O)C=C1CCC1 c1(C(N2CC(C)N(C(=O)C(O)Cc3cnn(C)c3)CC2)=O)cnn2c1CCCC2 C(=O)(C(C)CC(C)(C)C)NC1C(SC)CN(C(=O)CCCC(=O)N(C)C)C1 C1(C(=O)NCC(CC)(C)NC(=O)C(C)C)CC(S(N)(=O)=O)C1 CC1(C)C(CC(N2CCCCC2C2(NC(C3CC4CC4C3)=O)CC2)=O)C1(C)C N1(Cc2ncc(CC)s2)CCCC2(C1)NC(=O)C(C)(C)O2 c1(C(N2C3CC(NC(C=CC(C)C)=O)C2CC3)=O)cc2ccc(Br)nc2[nH]1 c1(CC)ccc(C(=O)NC2(C)CC(NC(=O)CCO)C2)cc1.c1ccccc1 C1(CCOC)CN(N2CCN(c3ncns3)CC2)CCO1 Cc1c(Cl)c(C(N2CC(CC(C)NC(=O)Cc3cnccn3)C2)=O)nn1C CC(C)(C#N)CC(=O)NCC1CC(NC(c2cn(CC(F)(F)F)nn2)=O)C1 CCC(CC)(CO)C(=O)NCC1CN(C(=O)C(C(C)O)N(C)C)CCC1C CCC(CC)C(=O)NC1CC(NC(=O)C=C(C)I)C1 Cc1cccn(CC(=O)NCC2CCC(NC(C3CCCC(=O)O3)=O)C2)c1=O C1(NC(c2c(C)nc(N(C)C)s2)=O)CCSC12CN(C(=O)Cn1ncnn1)C2 c1(C=O)cc(Br)ccc1C1CC1.C1(C(=O)NCCC)CC(=C2CCC2)C1.N N1(C(c2cnc(C)o2)=O)CCC(C(=O)NC2CCN(CCF)C2)C(C)C1 C(=O)(C(C)C(C)NC(=O)CNC(=O)Cc1cc(C)no1)OC C1(C(N(CCC(=O)NCCC(C)c2cn[nH]c2)CCO)=O)CCC(N(C)C)C1 c1(CC)c(C(N2CC(F)CC2CNC(C2CCN(CC)C2)=O)=O)cccc1F c1(C(N2CCCC(N(C(=O)COC)CC)C2)=O)cn2c(n1)CCCC2C C1(NC(CNC(C)=O)=O)C2CC3CN(C(=O)Cc4cnc5cccnn45)C1C3C2 C(=O)(C1=C(C(C)=O)N(CCOCC)C(=O)NC1c1ccncc1)OCC.C N1(C(c2cn(CC)nc2C)=O)C2CCC1C(C(=O)N(C1CCSC1)C)C2 N1(C(c2cccc(C)c2)C(=O)NCC(=C)C)CC(C)(C)CCC1C c1(C(N2CCC(C)(NC(C=C(C)Cl)=O)C2)=O)c(F)ccc(OC(F)F)c1F Cc1ccc(NC(=O)C(=O)NC(c2nccn2CCN(C)C)C)cc1C#N CC(CCC(C)(C)C)NC(=NC)NCc1ncccc1Br S(=O)(=O)(c1cccc(NC2CCCC2CCO)c1)N1CCN(C)C(C)(C)C1 N(C(=NCCN1CCNC1=O)NCC1CCC1)Cc1n(C(C)C)ncc1 c1(C(=O)NC2CC(CCNC(C(CC)CC(C)C)=O)C2)nccn2nc(C)cc12 C1(C(N2CCC(=CCNC(CC(C=C)C)=O)CC2)=O)CCCCN1N=O C1(CN(C)Cc2ccc[nH]2)CCN(C(=O)C(c2cccn2C)=O)CC1 c1(COC)cc(C)[nH]n1.c1(C=O)ccnn1COC.C(=O)C(F)C1CCC1.N C(CC)(C(F)(F)F)NC(C1CCC(CNC(C2(C=C)CCC2)=O)O1)=O Cn1cc(S(=O)(=O)N2CC(NC(c3cc(Br)nc(Br)c3)=O)CC(F)(F)C2)cn1 Cc1c(NCc2ccc(F)cc2Br)ncnc1NC1CCNC(=O)CC1 N1(C(C(C)(C)OC)=O)CC(NC(=O)CC2CCCCO2)C(CC2CC2)C1 C#Cc1cnc(C(=O)NCC#CCNC(c2ccc(N)c(O)c2)=O)c(C)c1.C C1(C=O)CC(C)N(C)C1.C1(C(=O)OC)C=CC(C(=O)NC)C1.C1CCC1 Cc1cc(C)c(C(N2CC(CNC(=O)CC(C)F)C(C)(C)C2)=O)cc1Br C(=O)(CC(Cc1ccc(C)cc1)NC(C1CCC(n2cc(CN)nn2)C1)=O)OC CCCC(CC)C(=O)N(C)CCOCCCN(C)C(c1cc(OC)cc(O)c1)=O C1(C2CN(C(c3ccc(C(C)(C)C)s3)=O)C2)(NC(CSC)=O)CC1 Cc1ccc(=NCCC(=O)NC2CC2NC(c2cccc(C(F)F)c2F)=O)[nH]c1 C(=O)(C1Cc2ccc(F)cc21)NC1CCN(c2snc(CC)n2)CC1F Cc1c(C(N2CCC(N(C)C(C3CC3(C)Br)=O)CC2)=O)cccc1F N=c1[nH]c(=NCC2CCCCC2NC(C2CC3(C2)CC3F)=O)[nH]cc1[N+](=O)[O-] C1(O)(C=O)CN2CCC1CC2.c1(OC)ccnc(C(=O)NC2(C)CCCC2)c1.N Cc1c(C(N2CCC(C(C)NC(c3cc[nH]n3)=O)C2)=O)[nH]c2cc(F)cc(F)c12 C(=O)(C(O)CCCNC(=O)C(C)(C)C(C)O)NCC(C)CN1CCCC1 N1(CC2CCC(C)O2)CC2CCC(NC(=O)Cc3ccc(C4CC4)cc3)CC2C1 Cc1cccnc1CC(N1CCOCC1CC(=O)NCc1[nH]nnc1C)=O c1(COC)nc(C(=O)NCC(C)(O)CNC(=O)CCCC2OCCO2)co1 C1(F)(C(=O)NC2CC(C)(NC(C3CCCCO3)=O)C2)CCCOC1 C1(NC(Cn2c(C)ccc2C)=O)CC=C(C(=O)N2CCC(OC(C)C)C2)C1 C1(N(C(CC2N(C)CCCC2)=O)C)CN(C(=O)C#CC2(C)CC2)CC1(C)C c1(C(C)C)cc(CC(=O)NCCCCC2CN(C(C3CC(CO)CO3)=O)C2)on1 N1(C(CCC(C)SC)=O)C(CNC(=O)CS(=O)(=O)C2CC2)CC2COCC12 CCCC(C)CC(=O)NC(C)CN(C)C(c1c(Br)ccnc1OC)=O N1(C(C2C(c3c(C)ccs3)C2)=O)CCC2CN(C(C3CCN(C)C3)=O)C2C1 C=CC(C)(CC)C(=O)NCC(O)CCNC(c1ccccc1C(C)(C)C)=O c1(N2C(C(C)(C)CNC(c3csnn3)=O)CCC2)ccccc1[N+](=O)[O-] C1(CNC(CC(=C)C)=O)COC(C)(C)CN1C(C1CN2CCN1CC2)=O c1(CC)ccc(C(C)C(=O)N(C(C)C(=O)O)S(=O)(=O)CC)cc1.C(C)=O C1(C)(C(=O)NC(C=CC(=O)NCCC(C(C)C)OC)C)CCC2CC2C1 C(=O)(CCCC(=O)NCC1CCN(C(c2nn(C(F)F)cc2Cl)=O)C1(C)C)OC N1(C(c2n(C)c(S)nc2)=O)CCC2CCCC12CNC(=O)Cc1cccc(Cl)c1 c1(N(C)C)ccc(C(=O)NC2CC(NC(C3(F)CC=CCC3)=O)C2)cc1F N1(CCC#C)CCC(C(=O)N(CCC(C(C)C)NC(C2CC2O)=O)C)CC1.C N1(C(c2n[nH]c(C)c2N)=O)CCC2(CNC(C3(C)CCC(=O)N3)=O)CCCCC12 N1(C(CC(=C)C)=O)CCC2(CCCCC2NC(=O)Cn2ncccc2=O)C1 CC1=C(C(=O)NC2CCOC2C2CCN(C(=O)Cc3csc(C)n3)CC2)CCO1 C1(C(N2CCC(C(=O)NCC(C)(COC)CC)(CC)C2)=O)CCCCCN1C N1(C(CNC(CCC)=O)=O)CC(CC(=O)N(CC(=O)NC2CC2)C)(OC)C1 C1(C(=O)N)CCN2CCOCC12.c1(CC(C)C)ccc(C(=O)NC2CC2C)s1 C1(C)(C(N2CC(N(C)C)C(F)C2)=O)CC(O)CN1C(=O)CSCCC#N C(CNC(=O)Cc1cn(C)cn1)(CC(=O)N)OC.C1(CC(C)C)CCC1.C C(N=c1cc(C(F)(F)F)nc(Cl)[nH]1)C1OCCCN(C(=O)CC2=CCCCC2)C1 c1(C(N2CCC(CNC(C3(CC)CCCC3)=O)C(C)C2)=O)cc2c(s1)CCOC2 N1(C(C(c2ccnn2C)NC(C=CC(CC)C)=O)=O)CCSCC1 c1(NCc2c(CC)cncc2)cc(=NC2CN(C(C)C)C2)[nH]c(C(C)C)n1 C1(CC)CC(C(N2CC(C(C)(C)C)C2)=O)CCN1C(c1cnn(C)c1C#N)=O C1(NC(c2cc(Cl)no2)=O)CC2CC1CN2C(c1cnn(-c2nccs2)c1)=O N1(C(C2N(CC)CCC2)=O)CC2CC1(C(=O)NCc1cccc(O)n1)C2 C(C)(CCCC(=O)N(C)CC1(CO)CCC1)NC(c1ccc(CC)cc1)=O C(CCC(O)C(=O)N1CCCC1CC(=O)OC(C)C)NC(COC)=O N1(C(C(C2(C)CC2)NC(c2c(C)cc(F)cn2)=O)=O)CCCN(C)CCC1 c1(C(N2CC(NC(CC(C)P(C)(C)=O)=O)C(F)CC2)=O)cc2ccc(Cl)cc2[nH]1 C1(NC(c2csc(CO)n2)=O)CCS(=O)(=O)C12CN(C(c1cscn1)=O)C2 c1(C(C(=O)NCC(CC=C)NC(C2CN(C)C2)=O)CC)ccc(F)cc1 C(=O)(CCC[SH](=O)=O)N.C(=O)(C(C)C)N(CC)CC.c1cc[nH]n1.C(C)C N1(CC(=O)NCC2(OC)CN(C(c3ccc(CC)o3)=O)C2)CCN(C)CC1 CCC1=NOC(C(=O)NC(c2nocc2C(=O)NOCCCCCC2CC2)C)C1 CCP1(=O)CCN(C(c2cccc(C(F)(F)C(F)(F)F)c2)=O)CC1 C1(C(C)C)CN(C)CCN1C(=O)CC1CCN(C(C2CC(=O)C2)=O)C1 N1(C(C2N(CC)CCC2)=O)CC(NC(c2nnn(C)c2C(F)F)=O)CCC1C C1(CNC(c2cncs2)=O)CN(C(=O)Cc2c[nH]nc2O)CCO1 n1(C(C2CCCCC2)CC)nc(C)nc1-c1cc(OC)c(Br)[nH]1 c1(C=O)ccccn1.C(C)CO.C(C(=O)NCC)NC(=O)NC.C(=O)C C1(N(C(c2cc(C(F)F)[nH]n2)=O)CC)CCCN(C(=O)CN2CCCC2)C1.C c1(C(=O)NCCOCCCNC(CC(C=C)CC)=O)ccc2ccccc2c1F c1(-c2cncc(CN(CC)CC)c2)ccc(C=O)c2[nH]ccc12.CC=C(C)C c1(NC(CC)=O)nc(C)c(S(=O)(=O)N(c2ccccc2)C)s1.c1cccc(F)c1 c1(C(=O)NC2CCCC(CNC(c3ncn(CC)c3)=O)C2)cnn2ccncc12 c1(OC)ncc(Cl)cc1C(N1CC(NC(c2ccc(Br)o2)=O)C(C)C1)=O c1(C(=O)NCCCCNC(c2c(C)cno2)=O)ccc(=N)[nH]c1 C(C(C)(C)CNC(=O)CCCOC(C)C)N(C(c1cccnc1)=O)CC N1(C(Cn2ncc(CC)c2)=O)CC(NC(=O)Cc2cccnc2)CC1(CC)CC CC1CCCCN1CC(=O)NCCCCN(C(=O)CC1C=CCCC1)C C=CC1(C(=O)NCC(c2ccccc2)NC(c2coc(C3CC3)n2)=O)CCC1 C(CC(=O)N1CC(c2n[nH]c(C)n2)C1)(C(F)(F)F)NC(CC(CC)OC)=O S(=O)(=O)(c1ccc(Cl)s1)N1C(COC)CN(C(c2cccc(Br)c2O)=O)CC1 c1(C(N2CC3C(CNC(C4CNC(=O)N4)=O)C3C2)=O)c(F)ccc(F)c1F c1(C(=O)N)ccc(Cl)cc1[N+](=O)[O-].N1(C(C)=O)CC(O)CC1C(=O)N(CCC)C C1(NC(CC2C(C)(C)CCO2)=O)CCCC(C(=O)NC2CC3(CC3)C2)CC1 N1(C(C(COC)C)=O)CCC(NC(C2(C(=O)OC)CC=CC2)=O)C1C C1(N2CCN(C(=O)Nc3ccccc3F)CC2)CCC23OCCC2CC13 CCC(CNC(C1(NC(=O)C=CCN2CCC2)CCC1)=O)N1CCCC1 NS(=O)(=O)c1cccc(C(=O)NC2COCCN(C(=O)CCc3cnn[nH]3)C2)c1 C(CCCCCC(=O)N(C1CN(C)C1)C)NC(C1(C(=O)NC)CCC1)=O Cc1c(-c2ccccc2F)o[nH]c1=NC(=O)C(=O)N1CC=CC1C(=O)O C(=O)(C(C)(C)C(N)=O)NCC1(NC(C(CC)NC(N)=O)=O)CCCCC1 c1(C(=O)OC)cc(C)nn1CC(=O)NCC(O)C.C(=O)CCCC1CCC1.N Cc1cc(=O)ccn1CC(=O)NC(C1CCCN(C(c2ccncc2)=O)C1)C C#Cc1ccc(OC)c(C(=O)NC2(CCCNC(C3CCOC3)=O)CC2)c1.O CC(CO)(C(=O)NCc1nn[nH]n1)NC(c1ccncn1)=O c1(OC)cc(C)c2c(c1)NC(C(=O)NCc1cc(Br)ccc1C#N)C2 C1(NC(CCC(=O)NCC)=O)CCCN(C(c2cc(C)cc(C)c2)=O)CC1 CONC(=O)C(=O)NCCC1CCN(C(=O)CC2CCC(=O)NC2)C1 C1(N(C)C(C2CC3(CCC3)C2)=O)CCCCN(C(=O)CN2CCCCC2=O)C1 C1(CN(C)C(c2ccccc2C2CC2)=O)COCCN1C(=O)C=C1CCC1 C(=O)(C1COc2ccccc21)NCCCC(C)(C)NC(C=CS(C)=O)=O c1(C(N2C(C)CC(NC(=O)C(F)(F)c3cncs3)C2)=O)nn(C)c2c1COCC2 CC1(C)CN(C(c2cnn3ncccc23)=O)CCC1NC(c1c[nH]c(=O)cn1)=O c1(C(=O)NCCOCC(=O)NCC(CC)(C)O)cncc(C#N)c1 C(=O)(CCCCCCN=[N+]=[N-])N1CC(C)N(C(=O)C(F)(F)C(F)(F)F)CC1 CCC1=NOC(CNC(c2ncc(Br)s2)=O)C1 C(c1ccc2c(c1)CC(=O)N2)=CN=c1[nH]c(C(=O)O)cc(OC)n1 C1(NC(CCC(=C)Cl)=O)CC2(C(=O)NCc3ccccn3)COC1C2 c1(C(=O)NC(CC)C(F)(F)F)cc2n(n1)CCCN(Cc1cnccc1Cl)C2 c1(C(=O)NCC(=O)NCCCC=C)ccc2c(c1)CCC2.C(=O)CS(=O)CC N1(C(C(C2CCCC2)OCC)=O)CCC(C)C(CN=c2[nH]nc(C3CC3)o2)C1 N1(C(C(C)SC(C)C)=O)CC2(CNC(C3CC(C)CC(=O)N3)=O)CC1CO2 N1(C(C(CC)(C)OC)=O)CCC2(COC(C)C2)C1.c1(C(=O)N)ncnn1C(C)C C(=O)(C(C)CO)N1CC(C(C)NC(=O)COCC2CCCC2)C1 Cn1c(C(=O)NC2CCC2)cc2cc([N+](=O)[O-])ccc12.C1(C(=O)N)CCC2CC12 Cc1cc(=NCC(C)(C(C)C)NC(=O)C(=Cc2c[nH]cn2)F)[nH]c(C(F)(F)F)n1 C1(CN(C)C(C2CCC(CNC(=O)C(C)(Cl)Cl)O2)=O)CCCCCC1 N1(Cc2cccc(OC)c2Cl)CCC2(CC1)CC2NC(=O)C=C(C)C(=O)O c1(C(=O)NC(C(C)NC(C2ON=C(CC)C2)=O)C)cc(S(N)(=O)=O)cnc1C C1(CC(=O)NCCCOC(C)C)CC(C)N(C(=O)CNC=O)C1 Cc1cc(OCC(N2CC3CCC3(CNC(=O)C3=CCCC3C)C2)=O)cc(C)c1 Cc1cc(=NC(=O)C(=O)NCc2nc3c(o2)CCSC3)[nH]nc1C C1(CC)CN(C(C23CCN(CC2)C3)=O)CCN1C(=O)CN1CCC1C N1(C(C(C(CC)C)O)=O)CC2C3CCC(C2C1)N(C(=O)CCc1cnoc1)C3 N1(C(c2ccc(Br)cc2)=O)CCC2CN(Cc3cc(Cl)ccc3Br)CC12 c1(C(=O)NC2C(OC)CN(C(=O)CCc3cccs3)C2)ccc(C#N)cn1 C(C(CC=C)C(=O)NCCC1CC(F)C1)NC(c1c(C#C)c[nH]n1)=O CC(c1ccccc1)=CC(N1CC(C(N)=O)(CNC(C2CC2(C)C)=O)C1)=O C1(OC)CN(Cc2cc(Br)ccn2)CCC1NC(C1(C)CCCCC1)=O c1(C(=O)NC2CCCC(CNC(=O)CCc3ccco3)C2)nc2cnccc2s1 N1(C(CC(C)(C)n2cc(CCC(C)O)nn2)=O)C2CCCC1C(=O)NC2 N1(C(CCN(C(C)=O)C)=O)CCCC(C)C1CCNC(c1cnn2c1CCC2)=O C(=O)C(O)CCC(F)(F)F.C(=O)(C(CCF)N(C(=O)CCC(=O)O)CC)OC.N C#Cc1ccc(C(N2CCC2C(=O)N=c2ccn(C(C)CC)[nH]2)=O)cc1C c1(CCNc2onc(C)n2)ccc(S(=O)(=O)NCCCc2c(C)noc2C)cc1 N1(C(CCC#CC)=O)CC2(CCCN(C(=O)C(C)OCCN(C)C)C2)C1 C1(NC(COC2CCN(C(C(CCCOC)C)=O)C2)=O)CCC2CC1C2(C)C N1(C(C2CC3(CC3)C2)=O)CCC(F)(c2cn(CCCOC)nn2)C1.C1CCC1 CC1(C)CCCC(CC(=O)NCCC2COCCN2C(=O)CNC=O)O1 C1(C(=O)NCCOCCC=C)CCCN(C(c2cc(CCO)on2)=O)C1 C=CCCCCCCC(=O)NC12CC(CNC(=O)C=CCCC)(C1)OC2C C(=O)(C#CC1(C)CCCO1)NC1C(O)C=C(C(=O)N(C)Cc2ncccn2)C1 C(CN=c1[nH]c(=NCC(C)(C)CN(C)C)[nH]c2c1CSC2)C1CC(C)OCC1 N1(C(CCC(=C)Cl)=O)CCCC(C)(C)C1CNC(C1CCCN1C(C)=O)=O C(=O)(C(F)(F)C(O)C1CC1)N1CCC(N(C(C=CC)=O)C)C1 C(=O)(CCC(=O)NCC)OCC.c1(CC(C(=O)N(CC)C)C)ccccc1Cl c1(C=O)c(Cl)n[nH]c1C1CC1.C1CCCN1C(=O)Cn1ccc(C2CC2)n1.N C1(C(N(CC(=O)OC)CC#C)=O)C2CC3C(C2)C13.c1(C=O)cnn(C)n1 c1(CC(N2CC(C)N(C(=O)CN(C)C(N)=O)CCC2)=O)cccc2cccnc12 CN1C2CCC1CC(=CC(N1CCCC1CNC(c1c(F)cccc1F)=O)=O)C2 Cn1nc(CNC(=O)Cc2cscc2Br)c2c1CCN(C(C1CC1F)=O)C2 C(N=c1nc(NCC2CCc3ccccc32)c2c([nH]1)CCOC2)c1cc(C)oc1 C(=O)CC(F)(F)F.C(c1c[nH]cn1)=C(C(=O)NCC(O)CNC(=O)C)F.N N1(C(c2cnn(CCOC)c2C)=O)CC2CCC1CN(C(=O)CCC(F)F)C2 c1(C(C)(C)OC)ccc(C(=O)NCCC(C)C)cc1.C1(C(=O)N)CC(F)C1 c1(NC2CCC(NC(c3nc[nH]c3C(F)(F)F)=O)CC2)ncnc(Cl)c1CO [SH](=O)(=O)c1ccc(C)cc1.C1CC(C)CN(C(=O)CC)C1.C(F)(C=O)=CC.N c1(CC(=O)NCC2(CNC(C(C)O)=O)CCCC2)cnn2c1OCCC2 N1(C(C2CCN(CC)C2)=O)CCN(C(=O)C2=CC(C)(C)C2)C(CF)C1 Cc1nc(CCCC(=O)N2CC(O)(CNC(=O)CC3CCCN3C)C2)cs1 N1(C(c2cn(CCC=C)nn2)=O)CCCC12CCN(C(=O)CC1CCSC1)CC2 c1(C(C)C)cc(C(N2CC(NC(C3(F)CC3)=O)C2)=O)n[nH]1 C=CC1COCC1NC(=O)CCOCCCNC(C1(CC)CC1)=O c1(CC)cc(C(=O)NC2CCCCC2CNC(C2CCCS2)=O)ccc1F C(c1ccc2[nH]ccc2c1)=CC(=O)NC1C2CCN(C(=O)C=CSc3nc[nH]n3)C12 C(CC(C(=O)NCC1(CO)CCCC1)NC(C1CCC(O)C1)=O)=CC c1(Oc2ccccc2)ccc(Cl)cc1Cl.c1(CC)cccc(NC(=O)CCN)c1 N1(C(CCCOCCC)=O)CCC2(COC(CNC(=O)C3=CCOC3)C2)C1 c1(CC)ccc(O)c(C(=O)NCC(C2CC2)N(C)C(C2CC23CCC3)=O)c1 C1(C2CCOCC2)(CNC(c2ncnc(C)c2C)=O)CCN(C(C2CC2F)=O)C1 c1(C(NC2CCCN(C(=O)CNS(C)(=O)=O)CC2)=O)ccc(F)c(Cl)c1 C(=O)(C(C)C(O)CC(C)C)N1CCCC(NC(c2c(C)nc[nH]2)=O)C1 C#Cc1ccnc(C(=O)NC(C(C)NC(C2(CCOC)CC2)=O)C(C)C)c1 CC(C)C#CC(=O)NC(C1CCN(C(=O)C=CC(c2cnn(C)c2)=O)C1)C c1(CCC(=O)NCC(C)CNC(c2nnc(O)nc2O)=O)ccc(O)c(F)c1 N1(C(c2c(C)nc(CCC)o2)=O)CCC(NCc2ccsc2)C(C)C1 C(=O)(CCS(C)=O)N(C1CCN(C(C2(C)CC2(C)C)=O)CC1)CC#C N1(C(c2cc(C)c(Br)cc2)=O)CCC2CN(C(=O)C(C)n3cccn3)CC2C1 c1(C(N2CC(NC(=O)Cc3ccc(F)nc3)C2)=O)cc(Cl)c(Cl)c(Cl)c1 C(=O)(C1=CCCN(C(C2CNC(=O)N2)=O)C1)N1CC(F)(C(=O)OC)C1 C(=O)(CC(C)C(C)(C)NC(=O)C1=CCCC1)N1C(COC)CCC1 C1(NC(C2C(C=C)C2)=O)CN(C(c2nccc(C)c2N)=O)C(C)(C)C1 N1(C(C2CCCC2)=O)CCCC(C(N2CCC(N3CC(O)C3)C2)=O)C1 N#Cc1sccc1C(=O)N(CCNC(c1cnn(C2CCC2)c1)=O)C1CC1 Cc1nc2c(F)c(F)ccc2c(C)c1CNc1ccc(C(C)(C)C)cn1 c1(CC)c(C(=O)NCC(C(C)C)NC(=O)Cc2nc[nH]n2)nnn1C C1(C)(COC)CCCN(C(=O)CC(C)(C)CNC(=O)CCc2cn[nH]c2)C1 C1(NC(C2CCC(C)(C)CO2)=O)CC2CN(C(=O)CSC3CCOC3=O)CC2C1 c1(C2CN2)ccc(F)cc1C.C1(CCC)CCCN(C(C2(C3(C)CC3)CC2)=O)C1 N1(C(Cc2c(C)nc(S)s2)=O)CC2CCC1CN2C(=O)CCc1ccsc1 Cc1ccc(C(N2CCC(NC(c3ccc(=O)n(C(C)C)c3)=O)CC2)=O)c(Cl)c1 c1(C(=O)OC)cc(C)nn1CC(=O)NC(C)(C)CC.c1(C=O)ccoc1C.N C1CC2CC1CN2C(c1ccncc1C(F)(F)F)=O.c1(OC)ccsc1C(=O)N N1(C(C(n2ncc(C)c2)C)=O)CCCC2(CCCN2C(c2conc2C)=O)CC1 C(CCC(C)C(=O)NCC1(F)CC(NC(=O)CO)C1)OC.C1CCCOC1 CC1CC(NC(=O)C(C2CCCCCC2)F)CN1C(C1CCCC1F)=O N1(CC)CCCN(C(c2cccc(-n3cc(COCCO)nn3)c2)=O)CC1 C(=O)(C1=CC2CCCC12)N1CCC(OCCNC(c2c(SC)ccs2)=O)C1 c1(C(N2C(CNC(CC3N(CC)CCC3)=O)CCC2)=O)cc(Br)cnc1O C(=O)(C1=CC2CCC1C2)NCC(C)NC(=O)Cn1cnc(C#N)n1 CC(C(=O)N(C1CCCN(C(=O)CCCCCN(C)C)CC1)C)S(C)(=O)=O c1(C(=O)NCC2CCN(C)C2)n[nH]c2c1CN(C(c1cnc(O)o1)=O)C2 c1(N(S(=O)(=O)c2ccsc2)C)cc2c(cn1)CCCC2 N1(C(c2cc(C)nn2C)=O)CC2CCC(C1)N(C(c1nc[nH]c3nccc1-3)=O)C2 c1(CC)ncoc1C(=O)NCC(C1CCC1)NC(=O)CN1CCOC1=O C(=O)(C1=COCCC1)N1CCCC(CN(C)C(C2CC3(CC3)CO2)=O)C1 C1(CCN(C)C(c2cc(Cl)no2)=O)CCN(C(c2cc(Cl)ns2)=O)CC1 c1(CC)nc(Cl)nc(N2CC(NC(=O)CCN(C)CCO)CC(C)(C)C2)c1C#N C1(NC(CC(C=C)C)=O)CN(C(c2ccc3scnc3c2)=O)CC2(CC2)C1 C1(F)(C(=O)NC(COC)CNC(=O)CCSC(F)(F)F)CCOCC1 N1(C(C2CCN(C(c3c(C#N)ccs3)=O)C2)=O)CCN2CC(O)CC2C1 C=CCCCCCC(=O)NC12CC1CN(C(c1c(N)cc(C)cc1F)=O)C2 CCC(C)CC(=O)N1CCCCC1CN(C)C(c1scc(OC)c1OC)=O CC1CCC(C)C1NC(C1CC(C)(NC(C23CCCCC2C3)=O)C1)=O N1(C(C23CCC(N=[N+]=[N-])(CC2)C3)=O)CC2CS(=O)(=O)CC2C1.C(=O)C1CC1.N C(C(N=[N+]=[N-])C(=O)NC1(CF)CCN(C(=O)Cc2cnn(C)c2)C1)OCC C12(C(=O)NCCN(C(C3COCCN3C)=O)CC)CCCCN1CCC2 C1(C(=O)NCCC(=C)CNC(=O)C(C)=CC2CC2)CC(=O)N(OC)C1 C(C(O)C(F)(F)F)NC(C1(F)CN(C(CNC(CN(C)C)=O)=O)C1)=O c1(C(=O)NC(CC)(C)CNC(C2COCCO2)=O)cccc2nc[nH]c12 CC1CC(NC(=O)C(C)(C)O)CN(C(=O)Cn2cc(C3CCC3)nn2)C1 C=CC(C)C(C)C(=O)NCC.c1(C=O)cnn(CCC)c1C1CC1.C1CC1.N C1(OCC)CCN(C(=O)C(Cn2cncn2)NC(=O)CCC=C(C)C)C1 C1(C(N2CC(CC)N(C(=O)CCc3ccnn3C)CC2)=O)OCCOC12CCC2 c1(C(=O)OCC)cc2cc(C(=O)N(C)Cc3ccoc3)ccc2o1 C(=O)(CC(CNC(=O)CC1CN(C(C)=O)C1)OC)N1C(CC)CC1 CC1(C)CC(C)N(C(c2cc(C(N)=O)c[nH]2)=O)C1.c1(C=O)cc(O)nc(Cl)c1 CC1=CCC(C)(C(=O)NCC(C)NC(c2n[nH]c(C(C)(C)C)n2)=O)CC1 CCC(C(=O)N1CCCC1C1CC1)n1ccnc1.C(=O)(C=CC(=O)N(C)C)N CCC(C)(CC)C(=O)N1CCCC(CCCCNC(c2csc3nnsc23)=O)C1 N1(C(=O)CN2CCCC2CO)CCCCC(Cc2cn(CC(F)(F)F)nn2)C1 C1(CC)C(NC(=O)C(Cc2ccsc2)NC=O)CCN1C(=O)CCc1ccon1 N1(CCC(=O)NCCCC(C)NC(=O)CCC(N)=O)CCCc2ccccc21 C1(C(N(C2CCCN(C(c3sc(C)c(O)n3)=O)CC2)C)=O)CCCC12OCCO2 CN=c1[nH]c(=NCc2ccncc2Br)[nH]c(=NCCCN2CCNC(=O)C2)[nH]1 C1(CN(C(C(F)OC)=O)C)CN(C(=O)CNc2ccccn2)CCO1 c1(OCC)cc2c(cc1C=CC(=O)NC)OC(C)C2.C1CN(C(C)=O)C1 C1(NC(c2cc(CCC)on2)=O)CCCN(C(c2cnccc2OC)=O)C1C N(C)(S(=O)(=O)N1CCCC(C(F)F)C1)C(CC)C c1(C(N2CCN(C(=O)NCC3(C)CC4(CC4)C3)CC2)=O)cnc(Cl)nc1OC C1(C(=O)Nc2c(C)cccc2)CCN(C(=O)C#CC(C)C)C12CCC2 Cc1oc(Cl)nc1C(=O)N(C1CCCC(NC(=O)CCN2C(=O)CCC2=O)C1)C c1(CC)cnn(C)c1C(N1CCCC12CC2)C(=O)NC1CCOC1 CCCCC(O)CCC(=O)NC1CCN(C(=O)C2=CCSC2)C1(C)C N1(C(C(c2ccc(OC)cc2)CC)=O)CCCCC1CNC(C1CC1(C)Br)=O Cc1nc(C#N)ccc1C(=O)NC.c1(CCC=O)cc(Cl)cs1.C1(CC)CC1 C1(NC(C(C(C)C)F)=O)CN(C(c2cnn(C)c(=O)c2)=O)CC1(C)C C1(C(C)C(=O)NC2COCC2CNC(c2coc(C(F)F)n2)=O)CCCCCC1 c1(CNC(C2(NC(C)=O)CCCC2)=O)ccccc1.C1(C=O)CC(C#N)C1 c1(C(C)(C)C)ccc(CNC(C2(C(=O)Nc3nccs3)CC2)=O)s1 C(=O)(C(O)C(C)(C)C)NC(C(=O)N(C)CC1CCCCC1)Cn1ccnn1 c1(C2C(C=O)C2)cccc(C)c1.C1(COC)CN(C(=O)COC(F)F)C1.N C#CC1(O)CN(C(=O)C(CCC2CC2)NC(=O)Cn2nc(C)nc2C)C1 N1(C(C2(CC3CC3)CC2)=O)CCOC(CN(C)Cc2nnc(C)s2)C1 CCC(C)C(C)CNC(c1n[nH]cc1CNC(C1CCC1C=O)=O)=O.O C1(NC(c2cc(C)[nH]n2)=O)CC2CCC1CC2NC(c1snnc1C)=O C12(NC(=O)CC3CCC3)CCCCCC1N(C(=O)Cn1ccc(C(F)F)n1)CC2 N#CC1(CNC(=O)CC2CC2CNC(=O)C(c2ccccc2)F)CCC1 N1(C(c2cccc(OC)n2)=O)CC(C)N(C(=O)CCn2cnnn2)CC1C c1(C(=O)NC(C2CCN(C(Cc3c(CC)con3)=O)C2)C)ccc(O)cn1 c1(C(=O)NC2C(NC(=O)OC(C)(C)C)COC2)csc2ccncc12 C1(CC=C)(C(=O)NCC(C)N(C)C)CCCN1C(c1cc(C2CC2)[nH]n1)=O C(CCCCOC1CCCCC1)NC(C)Cc1ccno1 c1(SCC)cccc(C(=O)NCCCO)c1.C1(C2(C(=O)N)CCC2)CCCCO1 CC1CC(NC(c2cncc(N)n2)=O)CN1C(=O)Cc1cnn(C)c1 N1(C(c2nn(CC)c(C3CC3)c2)=O)CC(NC(C2CCCC2)=O)CC(C)C1.O C(C(C)(CC(C)C)NC(c1cccc(CO)c1)=O)NC(c1[nH]cc(C)c1C)=O CCC1=C(C(=O)N2CC3CN(C(=O)CC(=O)NC4CC4)CC3(C)C2)CCCO1 C(=O)(C(CC)CCOC)N1CCC(CC=C)(NC(C2Cc3nccn3C2)=O)C1 c1(CC)c(C)nc2ncnn2c1NC(=O)C(N1CCC(C(=O)OC)CC1)=O C1(NC(C=CSC)=O)CN(C(=O)CCc2ccc3ncsc3c2)CC1C1CC1 c1(C(N2C(C)CC2C(=O)NCC2CCC(F)(F)C2)=O)cnc2n1CCC2 CC(C)(C(=O)NCC1(NC(c2cnsn2)=O)CCOC1)C1CCCCC1 C1(C(=O)NCCC2OCCN(C(c3c(N)cncc3)=O)C2)CCCC2(CC2)C1 N1(C(C=CC(=O)OCC)=O)CCC(C)(C(=O)NCc2cnccc2)C1 CS(C)(=O)=NC(=O)C(=O)N1CC2(CC(C)C2)C1.C1(CC=O)CC2CCC1CC2 c1(C(=O)NC2CC(NC(C(n3cnc(C#N)n3)CC)=O)C2)cn2cc(C)sc2n1 n1(CCOC)cc(C(=O)NC2CCCN(C(c3n[nH]cc3Br)=O)C2)c(C)n1 c1(NCCc2cc(C)[nH]n2)[nH]c(=NCC(C)c2ccccn2)nc2c1cnn2C C(=O)(C(C)CC(C)C)NCCC(C(=O)OC)C.c1(CC(=O)N)csc(C)c1 C(=O)(CCCC(=O)NCCN(C(=O)C(C)(C)n1cncn1)C1CC1)OC C1(C(=O)NC2CCC(NC(c3c(CC)nc[nH]3)=O)C2)CCc2ccccc2O1 c1(OC)cccc2c(-c3nc(COC(C)(C)C)nn3CC3CCCOC3)cnn12 C(=O)(C1OCCn2ccnc21)NCC(C)(C(C)C)NC(c1c(C)nn[nH]1)=O CC1(C)C(=O)NC2CCC(C(N3CCC(O)(CO)CC3)=O)CC12 C(=O)(N=c1ccn(-c2nccs2)[nH]1)N(C(c1ccc(C#N)cc1)CF)C C1(=CCNC(C(c2ccc(N)cn2)C)=O)CCN(C(C2(F)CCOC2C)=O)CC1 CC(CC(N)=O)C(=O)N1CC(C(C)(C)C)CC(CNC(=O)C2=CCCCC2)C1 C(=O)(CCCC(=O)N1CCC(CNC(=O)CC(C)CC)C1(C)C)N(CC)CC c1(C(N2C3CCC(C3)C2)=O)onc2cc(C)ccc12.C(C(=O)N)=CCN(C)CC C1(CC=C)(NC(c2cccnc2CO)=O)CCN(C(=O)C=Cc2cc[nH]n2)C1 C(=O)(CC1=CCOCC1)N1CCC(CNC(CSCCCC)=O)C(CC)C1 Cc1nn(-c2ccc(Cl)cc2)cc1C=O.C1CC1.C1(C(F)(F)F)(C=O)CC1.N Cn1c(C(=O)NCC2COC(CNC(=O)CCCCC3CC3)C2)cccc1=O c1(SC)ncc(C(N2CCN(C(=O)CCO)C(C)C2)=O)c(O)n1.C(=O)(C(C)C)N CCN=c1ccc(C(=O)NCC(C2CCCCC2)NC(=O)Cc2cccs2)c[nH]1 C(=O)(NN1CCCC1C(=O)NCCC(O)C1CCC1)c1cc(CC)oc1C N1(C(C(C)CF)=O)CCCCC(NC(c2ccc(OC(F)(F)F)cn2)=O)C1 N1(Cc2ccc(C(=O)OCC)cc2)CCN(C(=O)CC2(C)CCCN2)C(C)C1 c1(C=O)csc(=NC2CCCCC2)[nH]1.C(C#CC)NC(CN(C1CC1)CC)=O.N C(C1CCCCC1)=CC(=O)NC(c1ncccn1)C(N)=O Cc1cc(C)c(CCNCC2(CN)CC2)c(C)c1O c1(C(=O)NCC23CC(NC(C(C)SC)=O)(C2)C3)ccc2n[nH]cc2c1 C=CCC(C)(CC)C(=O)NC1CC(NC(=O)C(=Cc2cccnc2)F)C(O)C1 C1(NC(C(CC)=CC)=O)CC(NC(=O)CCc2nnc(C)n2C)C(O)C1 CCCC(CC)CCC(=O)N(C1CC(NC(=O)C(c2ccc(C)cc2)(F)F)C1)C CC1(C)CCC(CCNC(C2(CNC(c3ccoc3Cl)=O)CC=CC2)=O)C1 CCCCC(CCCC)C(=O)NCC1(F)CCC(NC(=O)CCn2cnnn2)C1 N1(C(C(C)Cn2cccn2)=O)CCOCC(F)(CNC(c2ccnnc2O)=O)C1 N1(C(CCSCC(C)C)=O)CCCC(O)(CNC(=O)CCc2nncs2)C1 N1(C(CCC(CC)C)=O)CC2(CCCC2NC(=O)Cc2ccc3n[nH]cc3c2)C1 c1(-c2nc(C3(c4ccc(C)cc4C)CC3)on2)cccc2cc(Br)cnc12 C(CN=c1[nH]c(Cl)nc2c1SCC2)(C(C)(C)C)SC O=C(C1=CCCOC1)N1CCSCC1C(N1C(CO)CC1CO)=O Cc1cccc(CCNC(C2(CCNC(c3ccoc3)=O)CCCC2)=O)n1 C1(C(=O)N)CCC(C)(C)CC1.c1(C(=O)OCC)cnc(NC2CCCC2)nc1 CCC(CCCC(=O)NC(c1cccc(O)c1)C)NC(=O)C1=C(C)CCC1 CC(C)CC(O)CC(=O)N1CCCC1CS(=O)(=O)NCC(=O)OC(C)(C)C N1(C(C)=O)CC(O)CC1C(=O)N.c1(C=O)cccn1C1CC1.C1(CC)CC1 C#CC1(NC(=O)CCCSC)CCC(C)(C)C1.C(=O)(C(C)C)N(CC=O)C N(C(=NCc1ccc(F)cc1)NCc1csc(C2CC2)n1)CC1COC(=O)O1 CC(C)(C)C(C=O)NC(N)=O.C(=O)(C(O)C(F)F)N(C1CCCC1)CC.N c1(C(N(C2CCN(C(c3ccn(C)n3)=O)CC2)C)=O)cnc2c(F)cccn12 c1cccc(O)c1.C1(CNC(C2(N(C)C)CCC2)=O)CCCC1NC(=O)C Cc1cc[nH]c1C(=O)NCC1(F)CC(NC(C2CCC(F)C2)=O)C1 c1(CCC)sc(C(=O)NCC(C)N(C(=O)Cn2cc(CO)nn2)C)cc1Br c1(N2C(C(=O)Nc3nc(C)c(Br)c(Cl)n3)CSCC2)ncnc2c1CCCC2 c1(OC)ccc2cc(C(=O)Nc3ncccc3C(N3CCC3)=O)sc2c1 C1(C(=O)NC(CCNC(CC(C(=C)C)OCC)=O)(C)C)CCCOC1C(=C)C N1(C(C(C)(C)C2CC2)=O)CCC(NC(=O)CCc2cccnc2F)C(C)(C)C1 c1(CN2CCN(C(c3cnc(OC)nc3OC)=O)C3C2C3)cc(Cl)c(Cl)cc1F c1(OC)ccc(OC)c(CCC(=O)NC2CCC2)c1.C1(C(=O)N)CCC(=O)NC1 c1(C(N(CC(C)N(C)C(C2CCN(C)CC2)=O)C)=O)ccnc(OC(F)F)c1 CC(C)C(O)CC(=O)NC1CCCCC1NC(=O)C(c1c(F)cccc1F)(C)C c1(OC)cc(CCNCC(Cc2ccccc2C)CO)c(OC)c(Br)c1 C1(CC(C)C)CN(C(C2CCCCN2C(=O)CCC(C)N(C)C)=O)CCO1 S(=O)(=O)(c1cccc(=NCc2cncc(Br)c2C)[nH]1)NCC(CC)CO c1(C(N2CCN(C)CC2)=O)cc(F)c(N)c(F)c1.C(C(C)(C)CC(=O)N)OC.C C1(C(N(CCC(N2CC(O)(c3nn[nH]n3)C2)=O)C)=O)C2CC3C(C2=O)C13 C1(O)(C(C)NC(=O)COC(=O)CO)CN(C(=O)CC(O)C2CCCC2)C1 C1(C(=O)NCC2(C(C(C)C)O)CC2)CCCN1NC(=O)C1SCCS1 CCCCCC(O)CC(=O)NC(C)(C)CN1CCN(C(=O)CCOC2CC2)CC1 N1(C(=O)OC(C)(C)C)CC2(CNC(c3ccnc(CO)c3)=O)CC2(C)C1 N1(C(C(c2ccccc2O)OC)=O)CCC(CF)(NC(=O)CCCF)C1 N1(C(C2CCN(CC)CC2)=O)CC2CCC2(C(=O)NC)C1.c1cc(Cl)cc(Cl)c1 c1(NC)cnc(Cl)cc1C(=O)NCC1CCCCC1C.n1(CC=O)cncn1.N n1(CC)c(Sn2cc(CCCc3ccccc3)nn2)nnc1C1(CN)CCCC1 C12(C(=O)NC3CC(=O)NCC3)COC(C1)C(NC(=O)CN1CC3CC3C1)C2 C1(C=O)CCCC(=O)CC1.C(CNC(=O)C=CCC)(C1CCC1)OCC N1(C(C(c2cccs2)SC)=O)CC2CCN(C(c3cnnc(C4CC4)c3)=O)C2C1 CCC(CC)CCC(=O)NCC(C1CCCN1C(=O)C(c1cnn(C)c1)C)(C)C N1(C(C2(C(C)C)CC2)=O)CC2CCOCC2(NC(c2cc3ccsc3n2C)=O)C1 c1(C(N(CCCCNC(=O)C=Cc2ccccn2)C)=O)cnc2ccc(F)cn12 c1(C=O)ccc2c(n1)CCC2=O.C1(NC(c2ccc(Cl)[nH]2)=O)CCCC(C)C1.N c1(OC)ccn2ncc(C(=O)NC(C)C3CC3)c2c1.C(=O)(C(CO)N(C)C)N N#Cc1cc(C(N2CCOCC2C(=O)N=c2cc(Br)[nH][nH]2)=O)ccc1F N1(C(=O)NC)CCC(C(=O)N(C)CCN(C(=O)C=CC2CC2)C)C1 C1(CC=O)SC(=N)NC1=O.Cn1ccnc1C(=O)NCC1(F)CC(C)C1 Cc1cc(=NCCN2CC=CC2)[nH]c(N2CCN(Cc3cncs3)CC2)n1 Cc1ccc(C#CC(=O)NCC(c2ccsc2)N2CCCC2)cc1 C=C(Br)CC(C)(C)C(=O)NCC(C)CNC(c1cc(C)nn1C1CC1)=O Cc1cc(C)c(C(=O)N(C2CCN(C(c3coc(CO)c3)=O)C2)C)s1 c1(C(=O)NC2CCN(C(CC(C)F)=O)C2)cc(Br)cc(S(C)(=O)=O)c1 C12(C(=O)NC(CCC)C(=O)NC(C3CCCC3)C)CCCC1OCC2 N1(C(CNC(=O)OCC=C)=O)CCN(C2CCN(C(C3OCCCO3)=O)C2)CC1 c1(C(C)C)nc(NCCC2CCCCC2(C)C)cc(=NCC2(C)CC=CCC2)[nH]1 c1(C(=O)NCCCN(C(C2N(C)CC(C)(C)C2)=O)CCO)cnn2c1OCCC2 Cc1csc(=O)n1CCC(=O)NCC1C(C)CCN1C(=O)C=C(Cl)Cl N1(C(c2ccc(CO)cn2)=O)CCC2(CCCN2C(=O)C=CCN2CCC2)C1 C1(CCNC(c2c(CC)cno2)=O)CN(C(=O)CC=C(Cl)Cl)CC(C)O1 C(=O)(CCC(F)(F)C(F)(F)F)NCC(CC)NC(C1Cc2ccncc2C1)=O Cc1ccc(C)c(C(=O)NC2CN(C(c3ccnc(C(C)(C)C)c3)=O)CC2F)c1 C1(CC(N2C(CNC(c3c(CC)nco3)=O)C=CC2)=O)CCCC(C)(C)O1 C(C1SCCc2ccccc21)NC(c1cc(Cl)c(Br)cc1)c1nnnn1C1CC1 CC1(C)CC2(CN(C(=O)CC3CCCCC3)C2)C1.C1(C(C)(C)O)(C=O)CCC1 CC(C)C(CC(=O)NC1CCCC12CN(C(=O)C(C#N)C(C)(C)C)C2)C(C)C C#CCC(CC(=O)NC(CSC)CC)NC(c1conc1C)=O C1(C(N(CC(CC)NC(=O)CCc2nc(C)cs2)CC)=O)(CO)CCCO1 CCCCCC(F)C(=O)NCC1CN(C(C2CC2C(C)(F)F)=O)CC1(C)C C=Cc1ccc(C(=O)NCC(C)N(C(=O)C(C)OCC(F)(F)F)C)cc1 Cc1cc(CC(=O)NC(C)C(C)C)cc(F)c1.C(C1COC(C)(C)O1)=CC=O Cc1[nH]c(C(=O)NCC2CCCN(CC)C2)cc1C(=O)O.C(C)C C1(C(=O)NCCC(CNC(c2c(C)nns2)=O)O)CC(=O)N(C2CCCC2)C1 C#Cc1ccc(Cl)c(C(=O)NC(CNC(C2CC23CCCCCC3)=O)CO)c1 C1(NC(CS(CC)=O)=O)CC2CCC1CC2NC(C1CCCCS1)=O C=CC(O)C(=O)N1CC(C)(NC(=O)C(C)Cc2cnn(C)c2)C1 Cc1cc(C(N2CC3CCC3(NC(c3coc(C(C)C)n3)=O)C2)=O)c(N)c(F)c1 C(CC(C)(CC)NC(=O)Cc1sccc1Cl)NC(C1C(=C)C1)=O C1(C=O)CCCC2(CCOC2)O1.C1CN(C(=O)CN(C(=O)C)C)C1.CC=O.N C(=O)(C(F)(F)C(F)(F)C(F)F)N1CCC(CNC(C(CC(C)C)C)=O)C1 CCC(CC(C)C)C(=O)N(CC(C)NC(=O)Cn1cc2ccccc2n1)C CC(O)(C(=O)NC1CC(C)(NC(=O)Cc2ccc(F)cc2)C1)C(F)(F)F c1(OCC)ccc2c(c1)CC(C(=O)NC1C3CC1N(C(=O)COC)C3C)CO2 C1(CNC(C2(CCC)CCC2)=O)CCCC(C)C1.C(=O)(C)N.C(=O)CO C(=O)(CN=S(C)(C)=O)NCCCCC(C)NC(=O)CC1CCCC(=O)N1 c1(COC)nc(NCc2nccn2C)cc(=NC2CCc3cccnc32)[nH]1 C1(NC(C(c2cccnc2)OC)=O)CN(C(c2cncc(CO)c2)=O)CC1(C)C Cc1c(C(=O)NCC(C)(CC(C)C)NC(=O)C(F)C(F)(F)F)cncc1Cl Cc1cc[nH]c(=N)c1C(N1CCC(CNC(=O)CCN2CCCCC2)C(C)C1)=O c1(CC(=O)NC(C(CO)NC(c2c(OC)csc2)=O)C)cncc(Br)c1 c1(CC2CC2)nc(C2CC(=O)NC2)n(-c2ccccc2C(F)(F)F)n1.CC.O c1(CN2CCC(C(C)NC3COCC3n3ccnn3)CC2)cscc1S(C)(=O)=O C1(C(=O)NC(C)C(F)(F)F)CCC2(CC2)N1C(=O)C(C)C1(O)CCC1 N1(C(C2C(=C)CC2)=O)CCC(C(F)(F)F)C(NC(=O)C(C)=C(C)C)C1 c1(C(=O)NC2CN(C(CCN(C)CC)=O)C(C)CC2)cc2c(nn1)CCC2 Cc1cc(C)c(CC(N2CCCC(NC(C3C=CC=CC=C3)=O)C2)=O)s1 c1(C(N2C3CN(C(c4cncc(Br)c4)=O)CC32)=O)c(C)cc(F)cc1C.CC.O C#Cc1ccc(C(=O)NC2CC(NC(C3(C)CCC4CC4C3)=O)C(O)C2)cc1F c1(C(=O)NCC(C)=CC(=O)NCC2CCC(F)C2)ccc2nccn2c1 C(=O)(CCCCF)NCC(C)N(C(C(C1CCOCC1)OCC)=O)C C12(C(=O)NC(C3CCCCC3)C(C)NC(C=C(CC)C)=O)CCC(CC1)CO2 C(=O)(CCCC(F)(F)F)N1CC(CCNC(C(CCSC)O)=O)OCCC1 O=C(C#CC1CCOC1)NCCC1CN(C(C2CC(F)(F)C2)=O)CCO1 CC#CCCC(=O)N1CC(CNC(=O)CCN2CCCCCC2)C(C)C1 C1(C(=O)OC)CCCN(CC(N2CCCC2C)=O)C1.c1(CC(=O)N)ccnn1C c1(OC)ccc2c(C(N3CC4(CCC(NS(=O)(=O)C5CC5)CC4)C3)=O)c[nH]c2c1 C1(CCC)(NC(C(C)=CC)=O)CCCN(C(=O)CC(n2nc(C)cc2C)C)C1 N1(C(c2c(C)noc2)=O)CC(C(=O)Nc2cnc(O)nc2O)CC(F)(F)C1 c1(COC)cncc(C(N2CC(CF)C2)=O)c1.C(=O)(CCCN1CCOC1=O)N N1(C(c2sccc2CNC(C2(F)CCCCC2)=O)=O)CCCC2(CC1)CC2 c1(OC)cc2c(CNC(c3ccc(F)cc3)C3CCCC3)c[nH]c2cc1Cl c1(C(N2CC(NC(c3c(C)ncn3O)=O)C(F)C2)=O)csc2nccn12 c1(C(=O)NCCC2CC(NC(c3c(C)cc(C)o3)=O)C2)ccn2cnnc2c1 C=CCCC(F)(F)C(=O)NC1CCCC1NC(c1ccsc1OC)=O c1(C(N2C(C)CCC(NC(=O)CN(C)CCO)C2)=O)n[nH]c2c1CC(C)CC2 CN1CCOC(CN(C(=O)CCC2(NC(c3ccsc3Cl)=O)CCC2)C)C1 CC1CC(NC(c2cccc(-n3cncn3)n2)=O)CN1C(c1ncccc1N)=O C12(C(N(CC(=O)NCCN3CCC(CO)C3)C)=O)CCCN1CCC2 N1(C(C(CC(C)C)C(C)C)=O)CCCC2CN(C(C3CC4CCC3C4)=O)CCC12 C(=O)(C(C)(C)C(=O)C(C)OC(C1CCCCC12OCCO2)=O)OC C1(CC=C)(NC(=O)Cc2ccsn2)CCCN(C(=O)Cc2ncccn2)C1 c1(CN(c2n(CCCOCC)c(-c3nccs3)nn2)C)cc(F)cc(F)c1 N1(C(C2C(CC)C2)=O)CC2C(CC(=O)NCCn3cccn3)C2C1 CC1CC2CN(C(=O)CCCC(N)=O)CC2N1C(=O)CSc1cccc(Cl)c1 CC1CN(N2CCCN(C(N)=O)CC2)CC2(CCCOC2)O1 Cc1nn2cc(C(=O)NCCCCC3CN(C(C4CN(C(N)=O)C4)=O)C3)nc2s1 c1(CNC(C(C2CN(C(=O)CCNC(=O)NC)C2)OC)=O)ccnn1C C#Cc1ccc(C(=O)N(CCC)CC)nc1.c1(C(=O)N)cncc(C(C)(C)C)c1 Nc1nc(Cl)ccc1C(N1CCC(CNC(=O)Cc2ccsc2)CC1)=O c1(C=O)ccc2nnn(C(C)(C)C)c2c1.C1(NC(C2(C(C)C)CC2)=O)CCC1 C1(C(=O)NC2C(NC(c3csc(-c4cccs4)n3)=O)CC2)C2CCOCC12 C(CCCCCN(C(=O)CC1CCCCC1)C)NC(C(C)CC1CCCO1)=O O=C1C2CC3C1C3C2C(N1CC2(C1)CN(C(c1cc(F)cnc1O)=O)C2)=O c1ccc(C#N)cc1.Cc1ccnn1CC(=O)NCC1(CC)CC1.C(=O)C.N N1(C(C2(CCCC)CCC2)=O)CCC2(CC1)CC2NC(C1CC1C)=O Cc1cc(F)cc(C)c1C(=O)N(C)CCN(C(=O)Cc1cn(C)cn1)C Cc1cc(C(C)C(=O)NC2CCN(c3cnccn3)C2)cc(F)c1 c1(C(N2CCCC(CC=C)(NC(C)=O)C2)=O)c(C)nc2cccnn12 N1(C(C(C)SCCCC)=O)CC2(CO)CC1(C(=O)NC1(CCCF)CC1)C2 c1(OC)ccc(C(C)C(=O)NC(CCN(C)C(c2cnccn2)=O)C(C)C)cc1 c1(OCC)nc(C)ccc1C(=O)NC1CCC(C)(CC)CC1 c1(OC)cc(C)c(C(=O)N)c(C)c1.C(=O)C(F)(F)CC1CCCO1.CC(O)C c1(C(=O)NC23CCN(C(c4cccc(CF)c4)=O)CC2C3)ccc2c(c1)NCC2 C(CCC(=O)N1CC2CCC(C1)O2)(C(C)C)NC(c1ccc(C)[nH]1)=O Cc1ccc(S(=O)(=O)N2CCCC2C(=O)NCc2ccnn2C2CCC2)cc1 c1(C(N2CCN(C(C(CC)=CC)=O)CC2C(F)F)=O)cc2nc(C)sc2[nH]1 N1(C(c2n(CC)ccn2)=O)CCCC(C)C1CNC(=O)C=CC1CCCN1C C1(CNC(=O)CN2CC=CC2)CC2CCCCC2N1C(c1ccsn1)=O C#CCC(CC(=O)N1CCCC(OC)C1)NC(C12CCC(OC)C1C2)=O N1(C(CSC)=O)CC2CCC1C(NC(c1cc(OC(F)F)cc(C3CC3)c1)=O)C2 c1(CC(=O)N)coc2cc(F)ccc12.C1CC2(CC2)CN1C(C1CC(O)C1)=O.C c1(C(=O)NC2C(NC(=O)CCCN3CCCCC3)COC2)ncn2c1CCC2 Cc1ccc(C(=O)N(C(C)CCNC(=O)CCCCc2cnc[nH]2)C)c(N)c1Cl C1(CNC(CCc2nc(C)sc2)=O)CN(C(C2(C)CCCCC2)=O)CC1C c1(C(N(C2CC3CN(C(C4C(C)OCC4)=O)C2C3)C)=O)cn(C)c(=O)n(C)c1=O n1(CC)c(NC(=O)CC(C)n2ccnc2)nc2ccc(Br)cc12 c1(CNC(CCC2CCN(C(CC=CCC)=O)C2)=O)ccnc(C#N)c1 N1(C(C(C2CC2)OC)=O)C(CC(=O)NCC(CO)CC(C)C)C2CCCC12 C(=O)(C1=CCC(C)(C)CC1)NC(C)C(C)NC(c1nc2cnccc2s1)=O c1(CC)[nH]nc(Cl)c1C(=O)NCCCOCC.C(=O)CCC.C1CCCC1.N CC1CC(C(=O)NCC2CCC(NC(=O)CSc3nncs3)CC2)=NO1 Cc1cc(CCC(=O)NCCCOCCC(=O)N(C2CCOC2)CCF)n[nH]1 c1(-c2cc(C(=O)N)no2)ccccc1Br.C(=O)(C1=C(Cl)CC1)N(C)CC1CC1 C(CO)(C(=O)N(C)Cc1cn(C)cn1)NC(C(C)OCC1CC1)=O c1(SC)cc(C(=O)NC2CN(C(C3(CO)CC3(F)F)=O)CC2F)c(C)o1 c1(N(C(=O)Cc2csc3sc(C)cc23)CC)ccc2c(c1)OCO2 N1(CC(COC)O)CC2CCN(C(c3cccc(-n4cnnn4)c3)C)CCC2C1 C(c1ccncc1)=CC(=O)N(C1CCCN(C(=O)C(F)(F)C2CCCCC2)C1)C C=CCN=c1[nH]cc(C(N2CCCC(N3CCCC3=O)C2)=O)s1 N1(C(CCN(C(CCC)C)C)=O)CCOC2(CCN(C(=O)CC3CCC3)CC2)C1 C1(C(N(CCC(N2C(C(C)C)CCCC2)=O)CCO)=O)CC2CCCC2C1 C(N=c1ccc([N+](=O)[O-])c[nH]1)C1CCN(C(C2N(N=O)CCCC2)=O)C1 C12(C(=O)N)CCC(C(F)F)(CC1)CC2.C=CCCCC(=O)NCC1(O)CCC1 N1(C(C(C)SC)=O)CCN(C(=O)CC(F)(F)Br)C(C2CCC2)C1 c1(NC(CCOC)=O)ccc(C)cc1NC(C1CCN(C)C1C)=O c1(C(=O)NC(C(C)NC(CCN(C(C)=O)C)=O)C)cn(C)nn1.C1CCOC1 C1(C)(C=O)CC(C)(C)C1.c1(C(C)(C(=O)N)N(C)C)ccc(F)cc1.C1CCC1 C(C(C)(C)CNC(C1(C)COC1)C)NC(=O)NCC.C(C)(C)C.O N1(C(c2sccc2OC(F)F)=O)CCN(C(=O)CCC2CCCC2)C2(CCC2)C1 Cc1cc(C(=O)NCC(O)C(=O)NCC2CCC(C)(C)O2)ccc1C#N c1(C=O)cc(O)nc(O)n1.C=CCCCNC(=O)C.c1(CC=O)nc[nH]n1.N n1(CC)nc(C(=O)OC2CC(OCC3CC3)C2)cc1C(F)(F)F Cc1ccc(Cl)cc1-n1nc(CC(N)=O)nc1C1CCCOC1CC(C)C C(=O)(C1=C(Cl)CCC(C)C1)N1CCCCCC(NC(c2cnc(COC)s2)=O)C1 N1(C(C2OCC(C)C2)=O)CCCC2(C1)CN(C(c1cc(F)cc(Cl)c1)=O)C2 CCC(C)(C)C(C(=O)N1CCN(CCNC(=O)CN2CCCCC2=O)CC1)OC c1(-c2cn(C(COCC)C(=O)NC3(C(=O)O)CC3C)nn2)cccc(F)c1.O c1(C(N(CC(CN(C(c2cn(CC)nc2)=O)C)O)C)=O)cc(C)c(C)nc1C C1(NC(C(N2CCOC2=O)C)=O)(CO)CCN(C(C2(C)CCOCC2)=O)C1 C1(CNCc2n(C)ncc2C(F)(F)F)COc2ccccc2C1 CC(C)C(C(O)c1ccccc1)NCC1(c2ccccc2Cl)CCC1 c1(C(=O)NC2C(NC(CN(C(C)C)C)=O)CC2)cc(C2(O)COC2)on1 CCC1=C(C(=O)N2CC(N(C(=O)C=Cc3ncc(C)[nH]3)C)C(F)C2)SCCO1 C1(C(=O)N)CC=C(C(C)C)CC1.N1(C(c2c(C)nn(C)c2)=O)CCCC(O)(C)C1 C1(C(=O)NC2(CC(=O)OC)CCS(=O)(=O)C2)Cc2ccc(Cl)cc2C(=O)O1 c1(C=O)cnc2c(c1)CCC(=O)N2.C1(C=O)(OCC)CCC1.C(C)C1CC1 c1(C(=O)NCCCCC(=O)N2CCC(n3cncn3)C2)ccc(O)c(F)c1 c1(C(N2CCN(C(C(C)C#N)=O)CC2C2CCC2)=O)[nH]c2ccc(F)cc2c1Cl c1(C(=O)N)ccnc2cc[nH]c12.C1(C(=O)NCC(C(C)C)OC)CC2CC1CC2 c1(C(N2C(CC)C(NC(c3sc(O)nc3C)=O)CC2)=O)cc(C)nc(O)n1.C c1(C(C(=O)NCC2C3CN(C(C4(C=C)CCC4)=O)CC32)O)ccc(Cl)c(F)c1 C(=O)(CC(O)COCc1ccccc1)N(CCN(C(CC)=O)C1CC1)C C1(NC(CN2C(C)CC2)=O)CCCCC1NC(c1ncoc1C1CC1)=O CCCCCCC(=O)NC(C)CC(=O)Nc1ccc(C)cc1O N(C(=NCCC(C)C)N1CCNC(=O)C1)C1CC(OCC)C12CCC2 C1(C(C)C)CN(C(C2CS(=O)(=O)C2)=O)CCC1NC(=O)C=Cc1ccoc1 N1(CC(=O)NC(C)C)CCCC1C1CCCCN1C(c1ccc([N+](=O)[O-])[nH]1)=O C1(C#CC(=O)N2CC(NC(C3CCC(C)(F)CC3)=O)CC2CO)(CC)COC1 CCC(=O)CCC(=O)N(CC(=O)NC1(CC)CC1)CC C1(C(=O)N)CN(C(C2CCCC(=O)CC2)=O)CC(C)O1.C(CC)NC(=O)NC N1(C(COC(=O)CO)=O)CC2CC1CN(C(=O)Cc1n[nH]c3ccccc13)C2 c1(OC)cc(F)cc(Br)c1NC(C1CC2(CC2)CN1C(c1ccccc1F)=O)=O C1(C#N)(C(=O)NCC2CCC(NC(CC3C(C)(C)CCO3)=O)CC2)CCCOC1 C(C)(C)(CCCC(=O)NCCC(C)C(C)C)NC(CC1(NC(C)=O)CC1)=O C1(CC(N2CCC(C(C)CNC(=O)C(C)(C)CF)CC2)=O)CN2CCN1CC2 N1(C(c2cn(CC)nc2)=O)CCCC2(CCC2)C1.C(=O)C(C1CC1)C1CC1.N N1(C(C)=O)CC2(CCCCC2)C1.C1(F)(C=O)CCS(=O)(=O)C1.CC[SH](=O)=O.N N#Cc1cnc(=NNC(=O)NC2CCc3cc(F)ccc32)[nH]c1 Cc1c(Cl)cccc1S(=O)(=O)NC1CC1C(=O)Nc1c[nH]c2ncc(Br)cc12 CN1CC=C(C(=O)NC(C)(C)Cn2cccn2)C1.C1(C(=O)N)CSCC(=O)N1 c1(C(=O)NCC2CN(C(c3cnc(CCCC)s3)=O)C2)cc(Cl)nnc1O C1CCN(C)CC1C#N.c1(C(C)=O)c[nH]c(C(=O)NCc2n[nH]cc2C=O)c1.N Cc1cc(OC(F)(F)F)ccc1S(=O)(=O)N1CCN(C)CC12CCC2 c1(CN2C(C(N3CC(CC)OCC3)=O)CCCC2)cnn2c1CCCC2 c1(C(=O)OC)cc(=NCC2CCCCN(C(=O)CC(F)(F)F)C2)[nH]c(C)n1 N1(C(CC(C)=C(C)C)=O)C(CC(N2CC(=O)NCC2C(C)C)=O)C2CCCC12 Cc1nc2cc(C(N3CCC(O)(CC)C3)=O)[nH]c2s1.C(=O)(C(C)(C)C(F)(F)F)N N(C(=NCCN1CCNC1=O)NC1CC(=O)N(c2ccccc2)C1)C(CC)C CN=c1cc(-c2ccc(N)c(Cc3ccccc3)c2)cc[nH]1 N1(C(C(C)O)=O)CC(O)CC1C(=O)N(CCC(N)=O)C N1(CCC(C)C)CCN(C(c2cccc(OC(C3CCCC3)=O)c2)=O)CC1 C12(C(N3CC(C)C(CC(=O)NCC4(C)CSC4)C3)=O)CCC(C1)OC2C NS(=O)(=O)c1n[nH]cc1C(N1CCCOC(CNC(C2(F)CCC2)=O)C1)=O C(=O)C(O)C(F)(F)F.N1(C(CNC(C(C)OCC=C)=O)=O)CCCCC1.C C1C2CN(C=O)CC12.C1CCCN1CC(F)(F)F.CC(C)(C)OC(=O)N.C c1(COC)cccc(C(N2CCC(NC(c3oc(SC)cc3C)=O)C2)=O)c1 c1(C(C)C)cc(C(=O)NCC2CC2NC(c2c[nH]c(Br)c2)=O)n(C)n1 c1(C(N2CC(NC(C3CC(C)C3)=O)C(F)C2)=O)cc(Br)c(F)cc1F c1(C(=O)NC2(CNC(C3CCC(=O)O3)=O)CC2)ccc2nn[nH]c2n1 N1(C(C(CC2CCC2)NC(c2csc(C)c2C)=O)=O)CCC(=O)N(C)CC1 C(C(=O)NOCCc1ccccc1)(C1CN(C(C2CCOC2(C)C)=O)C1)OC c1(OC)ccnc(O)c1C=O.C(=O)C(O)(C1CC1)C1CC1.C(C)C1CC1.N C1CC(O)C(O)C1.c1(C(C)C)ncoc1C(N1CC(O)(C(F)C(=O)N)C1)=O.C c1(C(=O)NCCOC2CN(C(C=C(C)C(=O)O)=O)C2)ccc(Cl)s1 O=C(N1OC2C=CC1CC2)C1CCC2(CC2)N1C(C1CCC(O)C1)=O C1(C(N2CC=CC2)=O)C(C(F)(F)F)C1[N+](=O)[O-].c1(C=O)coc(C(F)F)c1 c1(C(=O)NCCOCCN(C(C(C)SCC)=O)C)cnn(C)c1C#N C1(C(N(CC(=O)OC)CC#C)=O)CCC(NC(=O)C(CC)n2cccn2)C1 N1(C(C2(CC)CC2)=O)CCOC2(CCN(C(C3(C)CCC(=O)N3)=O)C2)C1 c1(C(C(=O)N(C(CC=C)c2ccco2)CC)(C)C)ccc(C)cc1C C1(C(N(C)CC2N(C(c3c(C)nc(O)[nH]3)=O)CCC2)=O)CN2CCCN1CC2 c1(NC2CCN(C(C(=O)OC)=O)CC2C)cccc2cn(C)nc12 C1(CNC(C2(F)C(C)C2)=O)COCCN1C(=O)C(c1ccc(Cl)s1)C C1CN(C(C2(C3CCC3)CCC2)=O)CCC1C(F)(F)F.C(CC(=O)N)=CC=C c1ccccc1.c1(C2(C(C)NC(=O)NC(COC)CO)CC2C)ccccc1 Cc1cccc(C(=O)NC2C(NC(=O)NCc3cc(C#N)cs3)C2)c1 C=C(C)CC(C(=O)N(C)CCc1ncon1)NC(=O)C(O)CCSC Cc1ccc2c(c1)CC(C(=O)NCC1CCN1C(c1cccc(CF)c1)=O)S2 N1(C(C(CC)(C)F)=O)CC(NC(c2cc(C)n(C(C)(C)C)n2)=O)CC(C)C1 c1(C(N2CCC(CCCNC(C(C)CO)=O)CC2)=O)ccc2c(c1)NC(=O)CS2 c1(C(C(N2CC(C(C)NC(C3CCC3(C)C)=O)C2)=O)O)ccccc1 N1(C(c2cnn(C(C)C)c2N)=O)CCC2(CCN(C(=O)CC(C)N(C)C)C2)C1 N1(C(C(C(C)C)OC)=O)CCN(C(C23CCC(CC2O)C3)=O)C2(CCC2)C1 C1(C(C)NC(C2CCC2C(F)(F)F)=O)CCN(C(=O)Cc2cnns2)C1 c1(C(=O)NCC(CCOC)NC(=O)CC2CC(=O)C2)ccc(C)c(C)c1F C1(NC(c2c(C)con2)=O)CCC(NC(C2CCS(=O)(=O)C2)=O)CC1 CC(C)N(O)C(=O)C(=O)N1CCC(NC(c2cccc(F)c2)=O)C(CO)C1 CCC(CC)C(C(=O)N1CCC(C(=O)NCC2CCN(C)C2)C12CC2)OC C12(NC(C3C=CC=CC=C3)=O)CN(C(c3ncccn3)=O)CC1CS(=O)(=O)C2 C(=O)(CN=c1ccc(C#N)c[nH]1)N1CC(CNC(C(c2c(C)noc2C)C)=O)C1 c1(C(C)C)ccc2c(c1)CN(C(=O)CCCCCCn1cc(C3CC3)nn1)CC2 c1(NCCN2CCN(C(CNC(CC3C(C)C3)=O)=O)CC2)cnc2[nH]cnc2c1 N1(C(C(C=C)O)=O)CC(C(=O)NOCc2ccc(F)cc2)CC12CCC2 C1(NC(C(CCC)OC)=O)CN(C(c2ncc(F)cc2N)=O)CC12CC2 C=CC(O)C(=O)NCCN(C1CCCC1)C(c1ccnn1C)=O Cc1noc(-c2ccccc2)c1.C1[N+](C)(CCCOC)CC1 C1(NC(c2nc(CC)oc2)=O)(CC)CCN(C(=O)C(C#N)C(C)C)CC1 c1(CC(N2CCC(O)(CNC(c3c(C)cco3)=O)C2)=O)c(F)cccc1F N1(C(C(CC)SC)=O)CCC(NC(=O)C=Cc2ccccc2F)CC1C c1(C(=O)NCC(CNC(c2ccc(C)n2C)=O)F)cc2c(Cl)cc(Cl)cc2[nH]1 c1(C(=O)NCCC2(O)CN(C(c3c(N)nccn3)=O)C2)cc2c(Cl)cncc2s1 N1(C(C2C(C)(C)C2)=O)Cc2ccc(CNC(C3C4CCCCCC34)=O)cc2C1 C1(NC(C23CCC(OC)C2C3)=O)CCN(C(=O)CC2(O)CCC2)C(C)C1 N1(C(CSc2n(C)nnn2)=O)CCC2CCN(C(=O)CC3CC4CCC3O4)C2C1 N1(C(c2c(C)nncc2)=O)CC2(CCNC(=O)CC3CCC(O)C3)CCC1CC2 c1(C(CC)(C)C)ccc2[nH]ccc(=NCc3ccc4c(c3)CCOC4(C)C)c2c1 Cc1c(C(N2CCC(C(C)(C)C(=O)N(C)C)CC2)=O)oc2c(F)cccc12 c1(CC)nocc1C(=O)NC(CO)C(=O)NC(C)Cc1nncn1C CN1CCOC(c2nc(-c3cccs3)nn2Cc2cccnc2)C1 C1(CN(C(CN2CCC(OC)C2)=O)C)CC(F)CN1C(=O)C(C)n1ccnc1 C1(CC)CN(C(=O)Cc2ccc(O)nc2)CCC1NC(c1cc2c([nH]1)CCC2)=O C(=O)(C(C)S(=O)(=O)CCC)NC1C(C=C)CN(C(=O)CC2(C)OCCO2)C1 Nc1cccc(C(N2CCC(CNC(=O)C(c3cccnc3)O)C2)=O)n1 C1(C(N2CC(CCCCNC(C(C)CC3CC3)=O)C2)=O)CCS(=O)(=O)C1 c1(CC(=O)NC2C(SC)CN(C(C3CCC(O)C3)=O)C2)c(F)cc(F)cc1F c1(C(N(CCN(C(Cc2c(CC)con2)=O)C)C(C)C)=O)cc2ccccc2o1 Cc1c(C(=O)NC2CCCN(C(=O)CCC3CC3)C2C)oc(=O)c2ccccc12 C1(CC=C)(NC(=O)CC2(N(C)C)CCCC2)CN(C(c2c[nH]c(C)c2)=O)C1 N1(C(c2cnn(C)c2C#N)=O)CCC(F)(F)C(CNC(c2ccc(O)nn2)=O)C1 C1(S(C)(=O)=O)(C=O)CCC1.n1(C(C)C(=O)N(CCC)C2CC2)cc(Cl)cn1 c1(CC)ccc(OCC(=O)NCCC(C)NC(C2CCS(=O)(=O)N2)=O)cc1 N1(C(Cc2c(C)ocn2)=O)CC2(CCN2C(=O)C(C)Cc2cnn(C)c2)C1 N1(C(COC)=O)CCN(C(c2n[nH]c(C3CC3)c2Br)=O)C(c2cn[nH]c2)C1 C1(NC(C(C)CN(C)C)=O)CN(C(=O)CN2CCCCCC2)C2CCCC12 CC1(C)OC(=O)CC1C(N1CCC(O)(CCNC(=O)CCC2CCCC2)C1)=O c1(N(C(=O)CCc2cnco2)C(C)C2CC2)ccccc1.CCCCOCC=O C1(NC(c2nn(CC)c(O)c2)=O)CS(=O)(=O)CC1NC(C1(Br)CC1)=O n1(CCC)cc(C(=O)NC2(CO)CN(C(C3CCCN3C)=O)C2)c2ccccc12 C1CCCCC1.C1(C=O)C2(CC2)C12CC2.c1(CSCC(=O)N)ncc[nH]1.C C1(C2CCN(C(CN(C(C)=O)C)=O)C2)CCCCN1C(=O)C=Cc1cnn(C)c1 C(C)(C)(CCCNC(C1CCC(=O)N1)=O)NC(C(C)CC1CCCC1)=O Cc1cncc(C=CC(=O)NC23CC(C2)C3)c1.c1(C(=O)N)c[nH]c(C#N)c1 C(C(C(=O)N1CCC1C(C)O)NC(=O)CN1CC=CC1)OC c1(CN2C(C)(C(=O)NC(c3nccs3)C)CCC2)cccc2c1ccn2C C12(C(=O)NC3CC(C)(NC(C(C)OC)=O)C3)CCCC(CCC1)C2 C=CC1COCC1NC(C1CC2CC2N1C(C1(C#N)CC=CC1)=O)=O c1(NC(CC(C)NC(C2CCN(OC)CC2)=O)=O)ccn2nccc2c1 Cc1c(C(=O)NCCCN(C(=O)C(O)C2CCC2)C(C)C)nnn1C CC1=C(C(=O)NC2CCN(C(c3ccc4c(c3)NCC4)=O)C2C)CCS1(=O)=O CC1=NOC(CCNC(=O)CO)C1.C1CCN(C(=O)C(F)CC2CCOC2)C1 c1(C(=O)O)ccc(C(F)(F)F)cn1.C1(=O)CC(N)C2CN1C2 C(C1CCCc2ccccc21)C1N(C(=O)NC2CC(C3CC3)C2)CCC1 CCC(CC(C)C)C(=O)NCC(=O)NCC(N1CC(CO)C1(C)C)=O Cc1cc(C(=O)NCC2CN(C(C3CCCN(c4nccs4)C3)=O)C2)ccc1F N1(C(C(c2ccc(Cl)s2)C)=O)CCC2(CCCN(C(c3ccncc3F)=O)C2)C1 c1(CNC(c2c(C)scc2)=O)cccc2c1CCN(C(=O)CCOC1CCC1)C2 C(=O)(C1(C)CCc2ccccc21)NC(C)CCNC(=O)CC(C)(F)F C(CCC)(C(=O)NC1CCCCC1)=CCC.c1(CC(=O)N)cccc(C2CC2)c1 C#Cc1ccc(F)cc1C(=O)NCCCNC(C12CCCC1CC(=O)C2)=O Cc1ccccc1COC(C)C(=O)N(C(C)C)C.C1(=CC=O)CCCC1.N N1(C(c2cnc(CC)s2)=O)CC(NC(=O)CCN2CCC(O)CC2)CC1(C)CC c1(C(=O)NCC2C(CNC(C=C(CC)CC)=O)C2)ncc(C(F)F)s1 CC(C)CC(O)C(C)C(=O)NC1(C)CN(C(C2CCC([N+](=O)[O-])CC2)=O)C1 C(=O)(C1=CC2(CCOC2)C1)NC12CN(C(C3CCCC(OC)C3)=O)C(C1)C2 C(=O)(C1CCCc2sccc21)NC(CNC(CC(C(=O)OC)(C)C)=O)C N1(C(CCSCC)=O)CCC2(CC1)COC(CNC(C1CC1CO)=O)C2 CC#CC1CCN(C(=O)CC(CNC(=O)C(C2CC2)C2CC2)OC)C1 CCC(C)(CNC(=O)CN(C(=O)Cc1ccc(F)cc1)C(C)C)C(N)=O Cc1cc2occ(CC(=O)NCCC(C)N(C)C(C3CCC=CO3)=O)c2cc1C C(=O)(C#CC1CCOC1)NC1CN(C(CCOCCOC)=O)CC1n1ccnn1 C1(C(C(=O)N(CCCC)CC)C)CCN(C(=O)CCNC(N)=O)C1 c1(C(=O)NCCC(=C)CNC(C2CCC(C)(C)C2)=O)cc2n(n1)CCO2 N1(C(C2CC(=O)N2)=O)CCOCC(NC(c2sccc2C(F)F)=O)C1 c1(C(O)Cn2cc(CN3CCCC3c3cccs3)nn2)cc(Cl)ccc1Cl N#Cc1ccc(C(=O)NCCOCCNC(=O)CN2CC3C=CC2C3)cc1 C1(NC(c2nnc(C)s2)=O)C2CN(C(C3CC4CC3CO4)=O)CC12 c1(C(=O)NC(C)(CNC(=O)Cc2cncc(F)c2)CO)c[nH]c2nc(Cl)ccc12 c1(C(=O)NC(CCNC(c2nncc(C)c2)=O)C)cncc2ccccc12 c1(N2CCC(C(N3CCC(C4CCC4)C3)=O)CC2)nc2ccc(Cl)cc2s1 C#Cc1cccc(OCC(=O)NC2CC(CNC(=O)C(O)C3CCC3)C2)c1 c1(-c2nc(C3NCCC(=C)C3)on2)ccc2ccoc2c1 N1(C(C2C3C=CSC23)=O)CCC2C1CCN2C(c1cnc(O)nc1O)=O c1(N2CC(CC)OCC2)nc(N(C)Cc2c(C)noc2CC)nc2scnc12 C1(NC(c2cc(CC)nnc2C)=O)CCSC12CN(C(c1ccccc1C)=O)C2 C1(C(N2CCC(NC(CCc3ccn(C)c3)=O)C2)=O)CCC2(CCCCC2)CC1 Cc1nc[nH]c1C(N1CC(OCCNC(=O)Cc2ccn(C)n2)C1)=O S(=O)(=O)(c1c[nH]ccc1=NCC1(N(C)C)CCSC1)NC(CC)CN1CCCC1 N1(C(C(N)Cc2cc(Br)c(Br)o2)=O)CC(CO)CC12CCOCC2 CC1c2ccsc2CCN1C(=O)C(=O)NCC12CCC(CC1)NC2 CCC(C)C(C(=O)Nc1cncc(F)c1)NC(=O)CCNC(=O)CO CCC(C(N)=O)NC(=O)C(Cc1ccco1)NC(=O)CCc1cccs1 c1(NC(CCN(CC=C)C(C2CCC(O)C2)=O)=O)cnc(COC)nc1 c1(C(N2CC(C)N(C(=O)CC(C)(F)F)CC2)=O)ccc2ccn(C)c2c1 N1(C(C2C(C)OCC2)=O)CC2CCOC2(CNC(=O)C2=CCCOC2)C1 c1(C(N2CCCC(C)C2C)=O)ccc2c(c1)COC2.C1(CC(=O)N)CCC(=O)C1 c1(OC)nccnc1C(N1CC(O)CC1CC(=O)N(CC(C)(F)F)C)=O CN1CCCC(O)(CC(N2CCC(O)C(NC(=O)CCCN=[N+]=[N-])C2)=O)C1 OC1CC(C2CC(c3nnnn3C3CC3)(NC3CCOC3c3ccccc3)C2)C1 c1(C(=O)NC2CN(C(c3cc(C)ncc3)=O)CC23CC3)cc2cc[nH]c(=O)c2s1 C(=O)(C(C#N)C(C)C)NC1(C(=O)NCCc2nc(C)on2)CSC1 C12(C(N3CC(NC(CSCC)=O)C(C)CC3)=O)C3C4C1C1C2C3C41C C(C)(C)(CC(=O)NCc1cncn1C)NC(c1c(C)snc1)=O CC1C(NC(C2CN(C3CCCCC3)C2)=O)C(C)CCN1CC1CCCC2CC12 Cc1cc(C(=O)NC(CNC(=O)C#CC2(C)CC2)C2CC2)c2cnccc2c1 C1(CC)CN(C(c2coc3c2COC3)=O)CCC1NC(c1cnn(C(F)F)c1)=O c1(SCC)ccc(Cl)cc1NC(c1cc(Cl)c(Cl)[nH]1)=O C1(C(N(C2CCN(C(CC3(C=C)CC3)=O)C2)CC)=O)COc2ccc(F)cc2C1 N1(C(CN(C)C(C2CC23CC3)=O)=O)CCC(C(N2CCN(C3CC3)CC2)=O)CC1 C(=O)(C1=NOC(C)C1)N1C(C(C=O)(C)C)CCC1.n1(C)nccc1C.C1=CCC1 Cc1cn2cc(C(=O)N(CCCCN(C)C(c3ccncc3O)=O)C)nc2s1 C#CCCCCCC(=O)NCc1ccc(C(N2CC(N3CCOCC3)C2)=O)nc1 N#Cc1ccc(C(=O)NCCOCCNC(C23CC(F)C2C3)=O)[nH]1 C(=O)(CCCCCCN=[N+]=[N-])NC12CN(C(c3c(C)n[nH]c3)=O)C(C1)C2 CC1CCOC(C(N2CC(NC(=O)Cc3cc(Br)cs3)C(C)C2)=O)C1 c1(NCC(O)CC2(O)CCC2)cccc(-c2ccsc2)c1 N1(C(C(C)c2cccs2)=O)CCC(C)(C)C1CC(N1CC(C)(CF)C1)=O c1(C(=O)NCC2(F)CC(NC(CCSCCC)=O)C2)noc2c1CCCC2 C(=O)(C1=NN(C)C(=O)CC1)N(CC)C.C(=O)(CCC(C)(C)C#N)N1CCCC1 N1(C(CCCCC)=O)CC2CCCC(NC(=O)C=CC3CCCC3)C2C1 N1(C(C2CCC(=C)CC2)=O)CC2CN(C(=O)CCc3ccccc3C#N)C2C1 C(CC)(C(C)C)NC(CCc1onc(CC)n1)=O.n1(C2(C=O)CC2)ccnn1.N CC1(C(N2CCOC(c3cn(-c4ccccc4C(=O)O)nn3)C2)=O)SCCCS1 N1(C(=O)OCC)CCOC(C(N2CCCC2)=O)C1.C1(CC(=O)N)CN(C)C1 CC(C)P(=O)(CC(=O)N(CC(O)CNC(=O)CCCCC(C)(C)C)C)C(C)C C1(C)(OC)CCN(C(=NCC2C3COCC23)NC2CCCCC2)CC1 C1(CC)C(O)CCN1C(C1CCCCN1C(c1csc(Cl)n1)=O)=O c1(C(=O)NC2C(NC(c3cc4sccc4s3)=O)CC2)c[nH]c2ccc(F)cc12 c1(C(C(=O)NC(C(=O)OC)C)N(CCC#N)C)cc(C2(C)CC2)on1 c1(-c2ccc(C(=O)Nc3ccc(-n4cccn4)cc3)nn2)ccn2cnnc2c1 Cc1coc(C=CC(=O)NC2CCN(C(C3CC4C=CC3O4)=O)C2)n1 C1(NC(c2c(C)nc(-c3ncc[nH]3)s2)=O)CCCN(C(c2cncn2C)=O)C1C c1(CSC)ccc(C(=O)N(CC(O)C)C)o1.c1(C=O)ccn(C(C)(C)C)c1 N1(C(CCCC#C)=O)C2CCCC1CN(C(=O)C(c1ccc(N(C)C)cc1)C)C2 n1(CC)ncc(C(=O)NC2CCCC(N(C(=O)C=Cc3cccs3)C)C2)c1C C(=O)CC(CN(C)C)C(F)(F)F.c1(CC)c[nH]c(C(N2CC(CO)C2)=O)c1.N N1(C(c2cn(CCOC)nn2)=O)CC2CN(C(=O)C3=C(Cl)CCOC3)CC2(C)C1 c1(OC)cc(NC(C2CC2NC(=O)Cc2ccccc2Br)=O)cc(C)n1 c1(C(N(CC2N(C(C3C(C=C)C3)=O)CCCC2)CC)=O)ccc(C#N)cc1F c1(CNS(=O)(=O)CCC2CCCO2)ccc2cc[nH]c2n1 c1(C(=O)NCC(C)NC(=O)CC2COCCN2CC(F)F)ccc(Cl)nc1O C1(NC(C(C)C#N)=O)CCC12CCN(C(c1cc(O)nc(Cl)c1)=O)CC2 Cn1cc(Br)cc1C(=O)NC1CN(C(=O)CCN2CCOCC2)CC1F CCC(O)C(F)(F)C(=O)N1CC2CC(C1)N2C(=O)C(C)Cc1cccnc1 Cc1cccc(C(N2CC(C)C(C)C2)=O)c1N.c1(CC(=O)N)cnc(C2CC2)[nH]1 Cc1nc2c(C(N3CCC(C)C(N(C(=O)C(F)(F)F)CCO)C3)=O)cccc2o1 C#CC1CN(C(=O)C(C)OCC2CC2)CCN1C(=O)CS(=O)(=O)CCC c1(CC)c[nH]cc1C(=O)NC1CCCC1NC(=O)CC1COC(=O)C1 C1(OC)(CNC(=O)CC(O)CCSC)CCN(C(=O)CCN2CCCC2)CC1 c1(C(=O)NC(C(C)C)(C)CNC(C2CCCCN2C)=O)ccn2c1CSCC2 c12cccc(c1)CO2.C(=O)(C(C(C)C1CCC1)N(C)CCF)NCC C(=O)(CS(=O)(=O)C(C)C)N.c1(SC)ccccc1C(N1CCC(O)(CC)C1)=O c1(NCCC(N)=O)nc(=NC2CCC(N3CCCC3)CC2)[nH]c2cccnc12 c1(OC)cc(NC(C2CC(F)CN2C(C2(C)CC2)=O)=O)ccc1Cl N1(C(=O)CNc2ccc(C(=O)O)nc2)CCC(O)(CO)C1.C=CC1CCC1 c1(CCC(N2CCC(CC)C2)=O)ccc(F)nc1.C1(C(=O)N)(CN(C)C)CC1 c1cccc([N+](=O)[O-])c1.CCCC(C)(C)C(=O)NC(C)CCN(C(=O)CCO)C N1(C(CN2CCN(C)CC2)=O)CCCC(C)(NC(=O)CN(C2CCCC2)C)C1 c1(C(=O)NCC(CCOC)NC(=O)C=Cc2cccnc2)cc2ncccc2s1 C(=O)(CC(F)(F)CS(C)(=O)=O)NC(CNC(CC1(CSC)CC1)=O)C C1(CN(C(=O)C(C)(O)C2CC2)CC)CCN(C(c2cc(F)cs2)=O)CC1 Cc1oc(C(N2CC=C(C)CC2)=O)cc1S(C)(=O)=O.C1(C)(CC=O)CC1(F)Cl N1(C(C(C)N(CC)CC)=O)CCOC(CNC(C2(CC)CCCC2)=O)C1 C(=O)(C1CCC(=O)c2ccccc21)N.CC1(C)CC(C(=O)NCCC2CC2)=NO1 C(=O)(CS(=O)CCC(F)(F)F)N1C(CNC(c2cc(CO)[nH]n2)=O)CCC1 c1(CNC(=O)Nc2c(OC)cc(C3CC3)cc2)cnn2cnnc2c1 CC1C(C)N(C(c2ccc(CO)o2)=O)CCN1C(c1cc2c([nH]1)CCCC2)=O C(=O)(CCCC(=O)N1CCCN(C(C2CCC(O)C2)=O)CC1)NCC N(C)(C[Si](C)(C)c1ccccc1)C(c1n[nH]c(C)c1Cl)=O C1(C(N2CC(c3c(CNC(Cc4nnc(C)s4)=O)nco3)C2)=O)CCCCC1O C1(CC(=O)NC)COC(C)(C)CO1.C1CCCN1C(c1csc(C(N)=O)n1)=O N1(CC)CCOC(CNC(=O)C(CCF)NC(C2CCOC2C(C)C)=O)C1 C(CCCC(=O)NCC1(O)CSC1)NC(c1c(OC)n[nH]c1)=O C1(CC(N2CC=CC(NC(C(CCC)OCC)=O)C2)=O)CCCCC1(C)C CCC(CN(C)C)C(=O)NC(Cn1cccn1)C(=O)NCCCS(N)(=O)=O c1(C(N2C(CO)CC(NC(c3ccn(C)n3)=O)C2)=O)cc2n(n1)CCOC2 C1(C(N(CCCCCNC(=O)Cn2nccn2)C)=O)C2C3CC4C1C1C2CC3C41 c1(C(C)=O)cc(C(=O)NC2(CNC(=O)C(C)N(C)C)CCOC2)n(C)c1 Cn1ccc2c(C(=O)NC3CCC(NC(C4CNC(=O)C4)=O)C3)ccnc12 C(CN=c1[nH]nc(C(F)F)s1)C1CCC(CC(c2cn(CC(=O)OC)nn2)=O)C1 C1(O)(NC(CCC2(C)CN(C(C3C(OCC)CC3)=O)C2)=O)CC2CCC1C2 c1(C(=O)NCCNC(C(C)OCCOC)=O)cc(Cl)c(F)cc1C c1(CNC(C2C(CCC)CCC2)=O)cnn2c1CN(C(=O)C(C)(C)CO)CC2 c1(SC(C(=O)N(C(CCNC(Cc2cc(C)on2)=O)C)C)C)ccc(C#N)cc1 c1(-n2ccc(C(=O)NCCCN(C(C(C3CCC3)OC)=O)C)n2)cncc(F)c1 c1(C(=O)NCC2C(C)CN(C(=O)C=CC3CCC3)C2)cc([N+](=O)[O-])ccc1Cl C1(C(=O)NCc2c(C)occ2)COC2(C1)CN(C(c1ccc(O)cn1)=O)C2 C1(c2n(CCCOC)nnn2)(NCC2=C(C)CCC2)CCC(C2CC2)C1 C1(NC(Cc2cc(C)[nH]n2)=O)CC(O)CN(C(c2cc(C(F)F)ncn2)=O)C1 c1(C(=O)NC(C(C)NC(c2c(C)nn(C)c2)=O)CO)cnc(C2CCC2)nc1O c1(C(=O)OCC)ccc(Cl)nc1NC(C1CC(C)CN1C(=O)C(C)CC)=O N1(C(c2ccnc(CO)c2)=O)CCCN(C(C2CC3CCC2C3)=O)C(CO)C1 C1(CCCC)CN(C(=O)C(C(C)C)SCC)CCN1C(c1cc(Cl)cc(Cl)c1)=O c1(NC(N(C)Cc2cccc(N(C)C)c2)=O)cc(C2CCOCC2)ccc1F c1(OC)ccc(C(=O)NC(CC)C(C)C)c(F)n1.c1(CC=O)csc(C)n1.N c1(N2CC3C(NC(c4n[nH]c5cccnc45)=O)C3C2)ncnc2c1CCC2 c1(CNC(c2ccc(C)[nH]2)=O)ncccc1C(=O)N(C1CCC1)C1CC1 Cc1coc(C(=O)NCCC(C)NC(C2CCN(CC(F)(F)F)C2)=O)c1 C12(NC(C3CC(OCC)C3)=O)CCC1CN(C(C1CCNC1=O)=O)C2 CCCC(C(=O)NCC1COCCN(C(c2sccc2C(C)C)=O)C1)C(C)C C=CCN=C(NCc1nc(C#N)cs1)NCC(c1ccc(OC)c(OC)c1)CO c1(C(N2C(C)CC(CNc3nc(C)nc(O)c3)C2)=O)cc2n(n1)CCCO2 c1(C(=O)NCC2(CNC(CC(C)C)=O)CCCCC2)cnn(C)c1C#N c1(C(=O)NC(CC)CNC(c2csc(Cl)c2)=O)ccc(N2CCC(C)=N2)cc1 C(=O)(CCC1=NNC(=O)CC1)N1C(CNC(c2c(C)onc2O)=O)CN(C)CC1 Cc1cc(N2CCC3OCCCC3C2)nc(=NCCC2(CO)CC2)[nH]1 C1C2CC1N(C(=O)CC1CCOC1C)C2.C1(C(F)(F)F)(OC)CC(C=O)C1.N C(=O)(C1=CC(C)(C)C1)NCCN(CCC)C(C1(C(F)F)CCCO1)=O Cc1ccc(C(c2nnnn2CCC2CC2)NC2CCCC(C)(C)C2)c(Cl)c1 N1(C(C23CCC(OC)C2C3)=O)CCC2(C=C(C(=O)NC(C)CCF)C2)C1 C1(SC)CN(C(=O)C(c2cccnc2)C)CC1NC(=O)C=Cc1ccccc1 C#CCCC(O)CCNC(=O)NCc1c[nH]c(Br)c1 C1(CNC(CCCN(C(C)=O)C)=O)CN(C(c2cocn2)=O)CC1C.C1CC1.C c1(C(N2CC(CC)N(C(C3CCCN3N=O)=O)CC2)=O)cnc2[nH]nnc2c1 N1(C(c2cc(C)oc2)=O)C(CNC(c2ccc3[nH]ccc3n2)=O)CC2OCCC12 CS(=O)(=O)c1ccc(C(=O)NCC2=CCN(C(C3(F)CCCOC3)=O)CC2)cc1 Cc1ccc(CC(=O)NC2CC(CO)N(C(c3ccc(C)s3)=O)C2)c(Cl)c1 C#CCCCCC(C(=O)NC1CC(C(=O)OC)C1)N1CCSCC1c1ccccc1 c1(C(N(C2CCC(NC(C3CCC(C)(F)CC3)=O)C2)C)=O)cc2sccc2[nH]1 c1oc(C=O)cc1C.C1(O)(CC(N2C(CC)CC2)=O)CCOC1.C1CCC1 c1(NCC2(CC)CCOCC2)[nH]c(=NC(C)c2conc2CC)nc2sccc12 C1(C(=O)NC(C2CCCCC2)C#C)COCCN(C(=O)CCCCCC)C1.OC Cc1cccc(O)c1C(N1CC(O)(CC)C1)=O.C1(C=O)CCC1C(C)(C)C.N c1(-c2cc(C(N3CC(N(C)C(C4CC45CC5)=O)C3)=O)on2)cccc(Cl)c1F C1(CNC(COCCOC)=O)CN(C(=O)C(O)CC(F)(F)F)CCC1(C)C C(C1CN(C(=O)C(F)n2ccnc2)CC1C(=O)N)=CC.C1CCCC1(C)N(C)C c1(C(N2CC(NC(C(CC#C)C)=O)C(C)C2)=O)oc2ccccc2c1CN(C)C CC1=C(C(=O)N2CC3=C(C2)CN(C(=O)C(c2cccc(Cl)c2)C)C3)SCCO1 C1CC2CCC(C1)N2C(=O)CC1CC1(C)C.c1(C(C)C)ncc(C(=O)N)s1.C N1(C(C(CCCOC)C)=O)CCCC2(CNC(C3(Cl)CC3)=O)CCCCC12 c1(C(N(c2cccc(C)c2F)C2CCNCC23CC3)=O)cc2cccc(Cl)c2s1 c1(CNC(=NCC(=C)Br)NCC2CCCO2)c(S(N)(=O)=O)c(C)nn1C C1(CC(=O)N(C2CCN(C(=O)C(C)O)C2)CC#C)CCC(C)(C)C1 c1(C=O)cccn(C)c1=O.C1(CC(=O)NC(C(C)C)c2ncc[nH]2)CCC1O.N C#Cc1ccc(C(=O)NCC2N(C(=O)CCC(C)SC)CCC2(C)C)c(OC)c1 C(=O)(C1CCCc2nn[nH]c21)N1CCC(NC(=O)C2=CCCC2)C1 N1(C(C2C(C)C2)=O)CCC(O)(C(C)NC(=O)Cn2ccc(C3CC3)n2)C1 c1(C(N2CC(C(C)NC(c3cccc(=O)o3)=O)OCC2)=O)ccc2n[nH]cc2c1 C1(NCC2(C(C)(F)F)CC2)COCCC1.c1(C2(C=O)CC2)cccc(F)c1.N N1(C(=O)NC(CC=C)C)CCN(C(=O)OC(C)(C)C)CC1CSCC C1(NC(CC2C(C(=O)OCC)C2)=O)CCCCC1NC(=O)C(C)CC.O c1(C(=O)NC2(CNC(c3cnc(CC)s3)=O)CC2)cc2ccccc2cc1Cl c1(C(N2C3C(NC(C(C)(C)CF)=O)CC(C3)C2)=O)ccc2c(C#N)c[nH]c2c1 CCCC(CCCO)C(=O)NC(C)CCNC(=O)CCOc1ccc(OC)cc1 C(C(C)(C)C(C)(O)CCOC)Nc1cccc(CC(=O)NC)c1 Cc1cc(C(=O)NC(C)(C)CNC(c2cc(C3CC3)sn2)=O)cn(C)c1=O C#Cc1cncc(C(=O)N)c1.C1CC(C)CN(C(C2CC(=C3CCC3)C2)=O)C1.C c1(C(C)C)oncc1C(=O)NCC=CCNC(C1(c2cc[nH]n2)CC1)=O c1(C2(CNC(=O)NCC3CCN(C(CC)=O)C3)CC2)cc(C)ccc1Br C1(NC(CC2C(NC(c3cc(CC)[nH]n3)=O)CC2O)=O)CCOC12CCCC2 N1(C(=O)C=C2CCC2)CCC(C2(NC(=O)C(F)(F)c3cncs3)CC2)CC1 C=CC(CCC)CC(=O)N1C2CCC1CN(C(c1cn(CC)nc1C)=O)C2 C1(CCNC(=O)NC)CN(C(=O)C(C)(C)COC(C)=O)CCS1 C1(C(=O)NCC2N(C(c3c(C)n(C)nn3)=O)CC(O)C2)Cc2nnsc2S1 N1(C(C2(N(C(C3C(C)(C(C)C)C3)=O)C)CC2)=O)CCCCC1 CCC(C(=O)NCC1(C(=O)NCCC(C)C(C)C)CC=CC1)C(C)C CC(CC(F)(F)F)C(=O)NCC1CC2(CC2)CN1C(=O)C(O)CC(C)(C)C C1(CC=C)(C(=O)NCC2(CO)CCOC2)CCCN1C(c1cnccn1)=O C1(C(=O)NC2C(NC(c3c[nH]nc3C(F)(F)F)=O)C2)CCC12CCC2 C1(CC)CCCCC1OCC(=O)NCC1CN(C(C2CCC(C)C2)=O)CCO1 c1ccc(C)cc1.c1(CC)cnoc1C(N1CCC(CN(C(=O)CC)C)C1)=O.S c1(C(=O)NCC(CC(C)C)NC(c2cc(C)n(C)n2)=O)ccn2ccccc12 N1(C(=O)CC2CCOC2)CCC(NC(=O)C(F)(F)F)CC1 C(c1ccc(S(=O)(=O)N2CCOCC2)cc1)=CC(=O)OC1C(CC)CCCC1 Cn1c([N+](=O)[O-])cnc1C(=O)NC1CC(CCNC(c2cnsc2)=O)C1 C=CC(C)(C)CC(=O)N(CCN(C(C1CCCN1c1ccncn1)=O)C)CC c1(CC(=O)NC2CC(NC(C3C(C)(CC)C3)=O)C2)cc(Cl)cc(Br)c1 n1(CC(N2C(CN(C(=O)C(O)CF)C)CCCC2)=O)ccc(O)nc1=O C(CCC(=O)N(CCC(=O)Nc1cnn(CC2CC2)c1)C)C1C(C)C1 c1(C(N2CC(NC(C(CC)C)=O)C3(C2)CC3)=O)ccc2ncccn12 C(C)(C)(C(C)CC(=O)NC(C)(C)CCO)NC(C(C1CC1)OCC)=O CCN(CC(=O)NC)N1CC(C)C(C)C1.C(C)(C)(C)OC(=O)NCC [SH](=O)(=O)c1cccs1.C1(C)(C(N(C)CCNC(=O)CC)=O)CC(O)CN1C c1(C(N2CCCC(NC(c3nn(C)nc3Br)=O)C2)=O)cccn2cncc12 C(c1c(F)cccc1F)=CC(N1CCN(C(CC2CCC(=O)C2)=O)CC1CO)=O C1(C(=O)NC(C(=O)NCCCCC2CCCC2)C2CCOC2)CCC(C2CC2)C1 c1(C(C)N(C)C(C2(NC(=O)CCc3ccsc3)CCN(C)C2)=O)ccncc1F c1(CSCCOc2ccc(C(=O)OC)cc2)ccc(S(C)(=O)=O)cc1.O CC1(C)C(C(=O)NC2(CNC(C3CCCN3C3CC3)=O)CC2)C1C#N C1CCN(C(=O)C=CC2CCC2)CC1C1CC1.Cn1cnc(C=CC(=O)N)c1.C c1(C(C)NC2CCNC2)ccc(S(=O)(=O)NC2CC2)cc1 C(=O)(C(CNC(c1cc([N+](=O)[O-])n[nH]1)=O)C(C)(C)C)N1CC(C(C)C)C1 Cc1cc(C=O)ccc1S(C)(=O)=O.C1(C(N(CCC)C)=O)CCC1.C1CC1.N N1(C(C)C)CC(C(N2CC=CC(NC(=O)C(=CC3CCCCC3)F)C2)=O)CC1=O c1(C(N2CC(N(C(C3CC(C)CC(C)C3)=O)C)C2)=O)ccn2c1CSCC2 N1(CCCNC(C=CCC)=O)CCN(C(C2(C(=O)OC)CCC2=C)=O)CC1 c1(C(N2C(C(C)(C)C(=O)NC3CC(n4cncn4)C3)CCC2)=O)occ2c1CCC2 c1(OC)cnnc(C(=O)NCC2(C)CCCN2C(C2CC(C)=NO2)=O)c1 N1(C(C2C(C=C)C2)=O)CCN(C(C2C(C)C2C)=O)CC1c1ccc(OC)cc1 C(=O)(C(O)C(C)C)NCc1occ(C(N(C2CCCC2)CCCC)=O)n1 c1(COC)cccc(S(=O)(=O)NCc2cc3ccccc3cn2)c1 C(=O)(C(C)C(C)(C)C)NCc1cc(C)c(C)nc1.C(=O)C(O)CC1CCCC1.N CC(C)C(O)C(C)C(=O)N1CCC(N(CCO)C(c2cnc(C(F)F)nc2)=O)C1 C1(NC(CC(C)n2cccn2)=O)C2CC1N(C(c1ncccc1N)=O)C2 N1(C(c2cc(C)sc2C)=O)CC2CC(C1)N(C(C1CCN1C(C)(C)C)=O)C2 CCCCC(F)C(=O)N(CC(CC)NC(c1ccccc1C#N)=O)C c1(C(=O)NCC2(C(=O)NC(C(C)F)C)CCC2)ccc(Cl)cn1 CC1COc2ccccc2C1C(=O)N1CCN(C(=O)Cc2cncnc2)C(C)C1 N1(S(CC=C)(=O)=O)CC2CC1CN2C(c1ccc(C(F)(F)F)c(Br)c1)=O Cc1cc(C)c(C(=O)NC2CCN(C(C3CCC(C)CC3)=O)C2)cn1 CC1=CCC(C(=O)NCC(C)(C)CN(C)C(C2(C(C)(F)F)CC2)=O)CC1 c1(C(=O)NCC(=O)NC2CC2)cnc2c(-c3cccc([N+](=O)[O-])c3)cccc2c1 c1(C(=O)NCC(C)N(C(Cn2ccc(C)n2)=O)C)cc(C)c(O)nn1 C1(C(N2CCN(C(C3CSCCS3)=O)CC2)=O)CC2(CSC2)C1 N1(C(COC(CC)C)=O)CCC2(CC1)CN(C(=O)C(C)NC(N)=O)C2 c1(C(=O)NCCC2N(C(C(C(CC)C)O)=O)CCSC2)n[nH]c2nccc(Cl)c12 c1(OC)ccc(C(=O)NC2(C)CC(NC(c3cccnc3S)=O)C2)cn1 C=C(C)CC(C(=O)NC1C2CC(NC(=O)CC(C)n3ccnc3)CC12)OC N1(C(=O)Nc2nnc(C)o2)CC=CCC1C(=O)N(C1CCCCN1C)C(C)(C)C Cc1ccccc1CN(c1ccnc(NCCN2CCOCC2)n1)C Cc1cccc2c(CCC(=O)NC3CN(C(c4cccnc4)=O)CC3C)c[nH]c12 C(=O)(C(C)CC(C)C)NC(CNC(C1CC2(CC(C(=O)OC)C2)C1)=O)C O=C1CCC2(CN(C(C3(NC(=O)C#CC4CC4)CC(O)C3)=O)C2)O1 C(C)(CC(F)(F)F)NC(Cn1cnc(C(N)=O)n1)=O.C(=O)CCC1CC1(F)F c1(SC)ncc(C(=O)NC2(C)CCCC(C)C2)c(Cl)n1 C=C(Cl)CC(C(=O)NC1CCC(F)CC1)NC(=O)C(C)c1cc[nH]n1 C1(NC(=O)Cn2cncn2)COCCN(C(c2ccccc2CO)=O)C1 N1(C(C2C(C=C)CC2)=O)CCN(C(=O)C2=CCSC2)C(C)C1 C1(NC(c2cc(C)no2)=O)CC12CCN(C(=O)CC1=CCCC1)CC2 C12(CNC(c3c(Cl)c(C)n(C)n3)=O)CN(C(C3CC3C#N)=O)CC(F)(C1)C2 C1(C(=O)OC)CCOCCC1NC(=O)NCc1cocn1.C1CN1 N1(C(C=COCC)=O)CCC2(CC(NC(c3ccccc3C(N)=O)=O)CO2)C1 C1(NC(CC2CC(=C)C2)=O)CCN(C(c2ccsc2)=O)C1c1ccccc1 C1(C(CNC(C=CC(C)NC(=O)CSCCC#N)=O)O)CC(C)(C)C1 c1(C(C=O)N(CC=O)C(C)C)ccc(C(F)F)c(C)c1.C1(C)CC1.CC C1(NC(COCC(=C)C)=O)CCCCC12CCCN(C(C1(CC)CCC1)=O)C2 c1(CC)ccc(C(=O)N(CC(C)NC(=O)C=CC(C)(C)SC)CC)o1 C(=O)(C1(C)CCCc2ccccc21)N(C)CCNC(c1cccc(C#N)c1)=O C1(CNC(C2CC(F)C2)=O)CCCCN1C(=O)CCCc1cnccn1 Cc1csc2c(NC(N3CCSCC3CO)=O)ncnc12 N1(C(C(CCC)N(C)C)=O)CCC2CC1CN(C(C1(CC)CCCCC1)=O)C2 C1(CC(=O)NF)CC(F)CN1C(=O)CCCNC1CCOC1.N12CCC(C1)C2=O CCC(C)(CNC(C1CNC(=O)C1)=O)NC(=O)C=CCn1cncn1 c1(C=O)cn(C(C)C)nc1C.N1(C(C2(C(=O)OC)CC2)=O)CC(CC)C1.N CN(C)S(=O)(=O)N(C)CC(=O)NC1CCN(C(C2CCC3(CC3)C2)=O)CC1O c1(CC)ccccc1CC(=O)NCCNC(C1(n2cc(Br)nn2)CC1)=O C=C(C)CCC=O.C1(C=O)CC2(CC2)CN1C(=O)C=C(C1CC1)C1CC1.N n1(CC)ncc2cc(C(=O)NCC#CCNC(c3ccccn3)=O)c(C)nc12 Cc1cc(C(=O)NC2CN(C(=O)C(F)(Cl)c3ccccc3)CC2O)cnc1O c1(C(=O)NC(C(C)C)(C)c2nn[nH]n2)ccc2c(n1)OCC(=O)N2 c1(NCC(CCCC)NC(=O)CCc2ccon2)ccnc2nc(C)nn12 c1(C(N(C)CC2N(C(c3c(C)cno3)=O)CCC2)=O)c(Cl)sc2nnsc12 C1(NC(C2(C)CC=CCO2)=O)CCC2CCN(C(c3cc(N)ccc3O)=O)C1C2 C1(CC(=O)N(CC(CC)(C)OC)C)CC(C)(C)CN1C(C1CC(=O)CS1)=O c1(C(=O)NC2CCN(C(C3C(C)(C(F)F)C3)=O)CC2)coc2c1C(=O)NCCC2 C1(C(N(C)CC2(O)CN(C(=O)Cc3ccn(C)n3)C2)=O)CCn2cncc2C1 C1(C(N(C(C)(C)CC(=O)NC2COC(C(F)F)C2)C)=O)C2CCCCC12 c1(CNC(C(CNC(c2c(CC)cno2)=O)N(C)C)=O)cc(=O)cc[nH]1 C1(C(=O)NCC(C)NC(C2CC3(C2)CC(F)(F)C3)=O)CCCC(C)(C)CC1 C(C)(C(CC(=O)NCc1ccc(C#N)s1)NC(c1cc[nH]n1)=O)OC c1(OCC=C)ccc(C(C(=O)NC(C)C(=O)O)N(CCCO)C(C)C)cc1 N1(C(CCN(c2ccccc2)C(C)=O)=O)CCCN(C(=O)CC)CC1C.[SH](C)(=O)=O C1(C(=O)NC(C)C(CO)NC(=O)Cc2cnc[nH]2)C2CCCCCC12 C=CCCC(CC)(c1nnnn1CCCF)NCC(c1ccccc1)(C)C c1(CNc2c(CC(N3CCC(Br)CC3)=O)cccc2)cc(Br)cc(Cl)c1F C(CC(=O)Nn1cnn(C)c1=S)N(C(c1c(C)nc(C)o1)=O)C C1(O)CCN(C(=O)C=CC2CCC2)CC1.C1(C(=O)NC)CCS(=O)(=O)N1 N1(C(C(C2CCC2)OC)=O)CCCCC(N(C(=O)COCC2CCOCC2)C)C1 c1(C(=O)OCCCC2CC2)ccc(C(C2CC2)C2CC2)cc1 Cc1cc(C)c(CC(=O)NCC2C(O)C(O)CN2C(=O)CCCC(N)=O)c(C)c1 C1(C(=O)NCC(C2CCC(C(C)C)CC2)(C)O)(N)CC2CCC1C2.C1CC1.C c1(C(N2C(C(=O)Nc3cnc(C(N)=O)nc3)CCC2)=O)cc(Cl)ncc1F C1(C(=O)NCc2c(C(=O)NC(C)CN(C)C)nco2)CCC2(CC2)C1 C(=O)(C(CC1CCCc2ccccc21)N1CCC(c2ccccc2)c2ccccc21)NCCOC Cc1cnc(C(C)NC(=O)CCOCCN(C)C(C2CS(=O)C2)=O)s1 C1(C(C)C)CN(C(c2ncoc2CNC(c2cnn(C)c2N)=O)=O)CC(=O)N1 c1(C(=O)NCC(O)CC(F)(F)CO)cc(Br)c(O)c([N+](=O)[O-])c1 c1(NCC(C)CC(F)(F)F)nccc(=NCC2CCC(CO)O2)[nH]1 Cc1oc(C(=O)N(C)CC2(O)CN(C(=O)CSc3ccccc3Cl)C2)cc1.C N(C(=NCc1ccnc(F)c1)NC1CCCCC1)CC1C(C)CCO1 CCC(CCCC(=O)NCc1ccccc1Cl)NC(=O)CC1=CCCC1 CC1=C(C)CC(C(=O)N(CCC(=O)NC(C)Cn2cnnc2)C)CC1 C1(NC(c2nc(CCP(C)(C)=O)sc2)=O)CCCN(C(c2cn[nH]c2)=O)CC1F CCCCC(=O)C(=O)N1CCC(CC(=O)NCCC2NC(=O)NC2=O)C1(C)C C1(NC(C2C(CC)C2)=O)CC2(C1)CC2.C(=O)(CC(C)(C)C1CCCCC1)N c1(C(=O)N)c[nH]c2c(F)cccc2c1=O.C=CC1CC1C(=O)N(CCC)C1CC1 CCC(C)CC(C)C(=O)NC1CCC(Nc2ncnc(Cl)c2CO)CC1 C1(CNC(C2(OC)CCC2)=O)(CNC(C2OCC2(C)C)=O)CCCC1 c1(CC(=O)NCC(C)CNC(c2cccc(OC(F)F)n2)=O)ccc(Cl)nc1 C1(C(=O)NCCc2ccnc(O)c2)(NC(c2c(C)snn2)=O)CCC(C)(C)C1 c1(C(=O)NC(CCCC)CNC(c2cc(O)ncn2)=O)cnc2c(c1)COCC2 Cc1cc(Cl)ncc1S(=O)(=O)N1CCC(N(S(=O)(=O)CCc2ccccc2)C)C1 C(=O)(C1=NOCC1)NCC(C)C(=O)NC(C)C(N)=O CC(CC(N)=O)C(=O)NC1CC(F)CN(C(c2ccn(C3CCC3)n2)=O)C1 c1(-n2cc(C(N3CCCCC3CC34CC(CO3)C4)C)nn2)ccc(Cl)cc1F C(c1sc(Cl)nc1Cl)=CC(=O)NC(CN(C(c1nc(OCC)oc1)=O)C)C N1(C(CCC(=O)N(C)C)=O)CC(C(=O)N(C)CC2CCCS2)C2(CCC2)C1 C#Cc1cccc(CC(=O)NC(C)C(C)NC(C2(CCCC)CCCC2)=O)c1 Cc1oc(C(C)C)nc1C(=O)NC1CN(C(c2nn(C)cc2Br)=O)CC1C c1(CC(=O)NCCC(C)N(C(C2CC(C(C)=O)C2)=O)C)ccc(F)nc1 C(CC(CNC(c1c[nH]c(C(N)=O)c1)=O)NC(=O)CC(O)C1CCCC1)OC C(C)(CCC(=O)NC1CC1CNC(c1nn(C(C)C)cc1Br)=O)SC C1(OC(C)(C)C)CC2C1CCN2S(=O)(=O)N1CCC(c2cc(O)cc(F)c2)CC1 Cc1nc(C(=O)NC2CCCN(C(C3CC34CC4)=O)C2)c(C)n1C CC(C)CC(C(=O)NCCC1(NC(=O)C(O)C2CC2)CCCC1)c1ccccc1 N1(C(C(c2ccc(C)cc2)F)=O)CCC2C(NC(c3cccc(C)c3F)=O)C2C1 CC(C)(C)CCCCC(=O)NCC1(O)CN(C(c2ccc(F)c(CO)c2)=O)C1 CN1CCC(NC(N2CCC3CCC(O)C2C3)=O)c2ccccc21 N1(C(CCC(=O)OC)=O)CCCC(C2CCCN(C(c3coc(Br)n3)=O)C2)C1 C1(C(=O)NCc2c(C)ocn2)CCN(C(C2(CO)CCCO2)=O)CCO1 C(c1ccc(F)nc1)=CC(=O)NC1(C)CCN(C(c2c(C(C)C)occ2)=O)C1 c1(NC(C(C)C)CCO)nccc(=NCc2nnn(C(C)(C)C)n2)[nH]1 N1(C(c2cncc(SC)c2)=O)CCC(NC(c2ccc(N(C)C)cc2)=O)C(F)C1 CC(N=c1[nH]c(=NC2CC3CCCC(C3)C2)[nH]c2cc[nH]c12)c1cccc(Br)n1 c1(C(=O)NC2CC(N(C(C(CCCC)C)=O)C)C2)c(C)cc(C)nc1C CC(C)CC(C)(CO)NC(=O)C(F)C1CC(NC(c2[nH]nnc2C2CC2)=O)C1 C1(C(=O)NCc2c(C(=O)NCc3snc(C)n3)scc2)CCN(C)C1=O C1(C(N2CC(c3nncs3)C2)=O)(NC(c2cc(C(F)F)[nH]n2)=O)CCCCC1 C1(OC)CN(C)CC1NC(C1(NC(C2CCN(C)C2=O)=O)CSC1)=O c1(C(=O)NC2(CC(=O)NC(c3nc[nH]n3)C)CCC2)ccn2ccccc12 c1(C(=O)NC(CN(C(=O)C=Cc2nccs2)C)(C)C)cccc(O)n1 C1(c2nnnn2CC2CC2)(NC(CC)(C)C)CCCC(OC)C1 C1(O)(C(N(CCN(C(C(C=C=C)C)=O)C)C)=O)CCCC(C)(C)CC1 C1(NC(c2ccc(CC)o2)=O)CCN(C(=O)C(C)CC2CC2)C1C c1(C(=O)NCCC2OCCN(C(COCCC)=O)C2)cc(C)c2occc2c1 Cc1nc(C(=O)N(C)CCNC(c2cc(C(C)(C)C)no2)=O)nn1C CC#CCCCC(=O)N(C1CN(C(=O)Cc2csc(CC)n2)CC12CC2)C C=C1CCN(C(C2CC(OC)C2)=O)C(C(=O)NCCCn2cccn2)C1 c1(OC)ccc(C)cc1C(N1CC(C(=O)N)C1)=O.c1cnc(C(F)(F)F)cc1I Cc1ccnc(C(=O)NC2(C(=O)NCC3(C)COCCO3)CSC2)c1F C1(N(C(C(CO)N(C)C)=O)C)CCC2CN(C(=O)C3=CCSC3)CC12 c1(C(=O)NC2CC3CN(C(CC(C(C)C)C)=O)CC3C2)coc2c1C(=O)NCC2 c1(C(N2C(C)CN(C(C3SCCCS3)=O)CC2)=O)nn2cccnc2c1Cl C1(NC(c2onc(COC(C)C)n2)C)CC2CCC1C2 c1(C(=O)N)cc(F)c(F)cc1F.CCCC(C)NC(c1cc(C(F)(F)F)c[nH]1)=O N(C1CCNc2ccc(Cl)cc21)C(C(N1CCC(C)(CC(=O)OC)C1)=O)=O N1(Cc2ccc(COC)o2)CC(O)CC1C(=O)NCc1nccn1C c1(C(c2n(-c3c(C)cccc3)nnn2)NCCC2CC2)ccc2ncsc2c1 CCC(CC)(CCNC(=O)COC(F)F)NC(C1CCCC(F)(F)C1)=O c1(C(C)N(C)C(C2(C)CCCO2)=O)ccnn1C Cc1sc(C(N2CC(CCNC(=O)C(C)(C)C)OC(C)C2)=O)cc1S(N)(=O)=O C1CCC(C=O)CC1.c1(C(C)C)cc(C=O)no1.C1C=CC(C(=O)N(C)C)C1.N Cc1noc(C)c1C(C)C(=O)NC1CC(NC(=O)COCC(C)(C)C)C1 c1(C(=O)NC(CNC(c2cc(OC)nc(C)c2)=O)C(C)C)cccc2cnsc12 CC(CC(C)NC(c1cc(C2(C)CC2)n[nH]1)=O)N=c1[nH]c2cc(F)cc(F)c2o1 c1(C(=O)NCCC(C)N(C)C(C2CC3CCC2O3)=O)ccncc1.C(C)(C)C.S N1(C(c2cncc(C)n2)=O)CC(NC(=O)CC2CCCCO2)CC(C)(C)C1 C12(C(=O)NC3C(C)CCC3C)CCN(C(C3CNC(=O)N3)=O)CCC1C2 C1(OCCC)CCN(C(C2CN(C(C3CCCN3C)=O)CCS2)=O)CC1 C(N=c1ccnc(NCC2(CO)CC3CC3C2)[nH]1)C1S(=O)(=O)CCC1 C1(C(=O)Nc2cc(C(F)F)cc(F)c2)CC(C23CC(C2)C3)CN1 N1(CC(N2C3CC(CNC(=O)Cn4cccc4)C2CC3)=O)CCCCCCC1=O C(=O)(C(C)(C)CC(C)(C)C)NCCOC1CCN(C(C2CC=C(C)CC2)=O)C1 c1(C(=O)OC(C)(C)C)cnn(CC(N2CCN(C3CCS(=O)(=O)C3)CC2)=O)c1N N1(C(CCC#CC)=O)C(C)CC2CN(C(c3ccc(=O)oc3)=O)CC12 Cc1nc(C2CCCC2)sc1C(=O)NCC1CCC(NC(C2CCO2)=O)C1 CC(CNC(c1csc(CNC(=O)CO)c1)=O)C(C)(F)F.c1nc[nH]n1 C(=O)(CCCCc1ccccc1)N(C1C2CN(C(C3CC3C3CC3)=O)CC12)C N1(C(C(C)(C)F)=O)CCN(C(c2ccc(O)cc2F)=O)C(CC(F)(F)F)C1 c1(OC)ccc(C(=O)NCC2CCCCN(C(c3ccc(F)s3)=O)C2)cc1F c1(C(=O)NCC(C)(C)OCC)scc2c1CCCC2.C1(C=O)CCCC(F)C1.N N1(C(c2nn(C)c3c2CCC3)C(=O)NCC)CCN2C(=O)N(C)CC2C1 c1(C(N(C2CCC(NC(c3c(SC)snn3)=O)C2)C)=O)ccc(F)c2c1OCC2 N1(Cc2cnc(C(C)C)s2)CCSCC1C(=O)NCC(O)CO n1(CC(=C)CC)cc(CN(O)C(=O)C2CC(CC)C2)nn1.c1(C=O)ccccc1 c1(-c2cnc(CCC(=O)NC3CC3NC(c3n[nH]cc3F)=O)o2)ccccc1F N1(C(C(=O)NCCOCCCC)=O)CCC(NC(c2cocn2)=O)C12CC2 C1(CNC(C2CC2C2CC2)=O)CCCC2(CN(C(c3cc4occc4[nH]3)=O)C2)O1 C(N=c1cc(C)nc(C)[nH]1)C1CN(C(c2cc(CC)no2)=O)CC1(C)C C(=O)(CCCCCCCC(=O)N1CCCC(NC(C2CN(C)C(=O)N2)=O)C1)OC C1(C=O)CC2C=CC1O2.Cn1ccnc1C1(C(=O)NCC2(F)CCC2)CC1 C(=O)(C1=Cc2ccccc2OC1)N1CC2(CCN(C(CC(=O)NC3CC3)=O)C2)C1 Cc1cc(CNCC2COCCN2C(c2csc(C(F)(F)F)n2)=O)n(C)n1 c1(C(N2CC=CC(NC(CC=CC=C)=O)C2)=O)cnc(OC)nc1C c1(NC(=O)OCC)ccc(NC(=O)NCc2nocc2C)cc1 C1(Cc2cn(CCC3CC(NC(C=CSC)=O)C3)nn2)NC(=O)N(C)C1=O C1(CC)CCCC1C(=O)NCC(C)(F)CNC(=O)CO.C1(C)CCCC1 N1(CC)CCCC1C(F)F.n1(CCN(C2(CC=O)CC2)C(C)=O)cnnc1 C(=O)(CCS(C)(=O)=O)N1CC(C(=O)NCC(=C)C)C(N(C)C)C1 C(=O)(CCCCC(C)C)NC1CCN(C(C=CC(CC)=CC)=O)CC1O C1(C)(C(N2CCC(C)(C(=O)NC)C2)=O)CCOC(C)C1 C(C)(CCC(=O)N1CCOCC1C1CCOCC1)NC(C(c1ccccc1)OC)=O Cc1ccc([N+](=O)[O-])c(NCCC2CCN(C(C3(C)CCCO3)=O)CC2)c1 N1(CC(=O)NCCOC2CCN(C(C3CCC(=O)N3)=O)C2)C(=O)CNC1=O CC1(C)CN(C(=O)CC2CC2(Cl)Cl)CC1NC(c1c[nH]ccc1=O)=O C(=O)C(C)(C)CS(C)(=O)=O.c1(C(N(C(C)C)C)=O)ccnc(-n2cncn2)c1.N C1(C)(NC(C2CC(OC)C2)=O)CCN(C(c2ccc(-c3cscn3)cc2)=O)C1 C#CCCCCC(=O)N(C1CCN(C(=O)C(C)(C)c2cccs2)C1)CCO C=CCC(CNC(=O)CCc1cnn[nH]1)C(=O)N(CC(C)(C)OC)C N1(C(c2c(C)n(C)nc2)=O)CC2(CCC2)CC1C.c1(C(=O)N)ncsc1C(C)C c1(C(N2CC(CC(=O)N(CC(F)F)CCOC)OCC2)=O)ccc(C)c(C)n1 N1(C(C)(C)CF)CCN(C(=O)CNC(=O)CCC(=O)NC2CCCC2)CC1 c1(OCC)cc(CNC2CC(NC(=O)Cc3ccn(C)n3)C2)c(F)cn1 N1(C(CC2C=NN(C)C2=O)=O)CCC(C(=O)NC23CC(C)(C2)C3)CC1(C)C N1(C(C2CC(OC)C2)=O)CCC(NC(C2(CO)CCOC2)=O)C1C(C)(C)C N1(C(=O)NCC=Cc2ncn(C)c2)CCc2cccc(CO)c2C1 CC(C)C(C)CC(=O)N1CCC1CNC(=O)Cc1c[nH]nc1O c1(N(CCCNC(C2CC3CC2C2CC32)=O)CC)cc(S(C)(=O)=O)ncn1 c1(C(N(C(CNC(c2[nH]cc(C)c2)=O)C)C)=O)cc2n(c1)CCC2 Cc1cc(C(N2CC(C)(CCC(=O)N3CCC3CN3CC3)C2)=O)cc(Cl)c1 C1(C(=O)Nc2cc(C(C)(C)C)no2)CC2(CCN(C(=O)Cc3cc[nH]n3)CC2)C1 CCC(CC)(CC)C(=O)N1CCN(C(c2cnn(C3CC3)c2C)=O)C(C)C1 C1(CCNC(C2CCCC2)=O)CSCCN1C(=O)CCN1CCOC1=O C1(NC(c2sccc2F)=O)CCC2CC1CN2C(=O)CC1CCC(F)(F)C1 C1(CNC(c2csc(-c3ccco3)n2)=O)CCCCN(C(C2CCCS2)=O)CC1 Cc1cc(N)cnc1C(=O)NC(C1(CNC(=O)CC2CCCCC2)CC1)C c1(C(N(CC(CC)NC(c2cnn(CC)c2)=O)C)=O)ccc2nn[nH]c2c1 CC1CCCN(C(=O)Cc2ccco2)C1CNC(c1coc(C)n1)=O.C1CC1 C1(NC(C2CC(C)(CC)C2)=O)CCCCN(C(C2CCOC2)=O)C1 c1(N2CCC(C(C)NC(c3c(CCC)cccc3)=O)CC2)nc(C)nc(=N)[nH]1 CC(C)CCC.c1(C=O)occc1C1CC1.C1(C=O)CC1C=O.C(C)(C)C CC(C)(C)C(C(=O)NCC1(C#N)CCC1)NC(C1CN(C(N)=O)C1)=O CC1CC(CNC(c2ccc(NCCO)cc2)=O)CN1C(C1CCOC(C)C1)=O CCCCCCC(=O)NC1C=CCN(C(c2cnsc2C)=O)C1 Cc1nnc2cc(NC3CN(C(=O)Cn4cc(C(C)O)nn4)CC3C)ncn12 CC1CC(NC(C2CCCN2C=O)=O)CCN1C(c1cnn(C)c1Cl)=O N1(CC)CCN(CC(C)(C)NC(=O)NC(c2cncn2C)C(=O)O)CC1 O=S(=O)(c1cccnc1NCc1cscc1C(F)(F)F)N1CCC2CCC(O)C1C2 c1(NC2C(Nc3ncccc3Cl)COC2)ncnc(N2CCN(CC)CC2)c1C c1(C=O)cc(C(C)C)nc(O)c1.Cc1cc(C(=O)NC(C2CCCC2)C)n[nH]1.N C1(C=O)C2C3CCC(C3)C12.C(F)(c1ccccc1)=CC(N1C(CC)CCC1)=O C1(C(=O)NCc2ccncc2F)C2CCN(C(C3C=CCCC3)=O)CC12 CCC(C)(C(=O)O)NC(=O)CC(C1CC1)NC(=O)COc1ccccc1 O(P(C)(=O)CNC(=O)C(c1cnn(C)c1)NC(=O)C=CCF)CC C1(CC(N2CCC(C)(NC(C34CC(C)C3C4)=O)C2)=O)CCC2(CC1)CC2 c1(C(=O)NCCC(C(=O)NC2(C)CCC(C)(C)CC2)OC)ccc2nc[nH]c2c1 C1(NC(c2ccc(C(F)F)o2)=O)CCCCCN(C(=O)Cc2cccnc2Cl)C1 CCCS(=O)(=O)C(C)C(=O)N(CCCCN(C)C(c1c(N)sc2c1CCC2)=O)C N1(C(c2c(C)csc2)=O)CCC2CC2(C(=O)NCCC23CC(CCO2)C3)CC1 c1(C(=O)NCC(CN(C(C2(F)C(C)C2)=O)C)(C)C)cccc2ccoc12 c1(C(=O)OC)ccc(C(=O)N)s1.C1(F)CCC1.n1(CC=O)nnc(=O)[nH]1 N1(C(C(C)NC(C)=O)=O)CCCC(NC(=O)C(=O)Nc2ccc(C)cc2)C1C C1(NC(CC(C=C)C)=O)CCC(O)CN(C(c2coc(C(F)F)n2)=O)C1 C1(C(=O)NCCNC(Cc2c(Br)ccc(OC)c2)=O)CCC(=C(F)F)CC1 C12(C)CC(C1(C)C)N(C)C(c1ccc(CO)o1)C(=O)N2.C1(COC)CCOC1 C(=O)(CCS(=O)(=O)N1CCOCC1)NCC(CN(C(CC(=O)OC)=O)C)(C)C C1(NC(CC=CC=C)=O)CCCN(C(=O)C=CSc2nc[nH]n2)C1 Cc1ncc([N+](=O)[O-])n1CC(=O)NC.C1C(C)CCN1C(=O)C=C1CCC1 c1(C(=O)NC2CN(C(C(CC)(C)C(F)F)=O)CC2(C)C)nc2c(s1)CN(C)CC2 C=CCN=C(NCc1ccnc(C)c1)NCC1(OC)CCCC1 Cc1ccn(C)c1C(=O)NC1CN(C(C2(c3cccc(Cl)c3)CC2)=O)C1 C(C1(O)CCc2ccccc21)CN(S(N(C)C)(=O)=O)CC1CC1 n1(C(CC)CC)nc(C(=O)NCC2(O)CCN(C(C3CCC(O)C3)=O)C2)cc1C c1(C(c2nnc(N(C(CCSCC)C)C)n2CC)C)ccc(F)c(F)c1 Cc1c(NCC2CN(C(=O)C(C)C)CCC2C)cccc1C(=O)NCCC(C)C N1(C(Cc2c(C)cccc2)=O)CC2(C1)CN(S(=O)(=O)c1cncc(Br)c1)CCO2 N1(C(Cc2cc(OC)no2)=O)CCC(NC(c2ccc(N)cn2)=O)CC1C Cc1ccn2c(C(N3CCSC(C(=O)N=c4cc(CCO)[nH][nH]4)C3)=O)cnc2c1 Cc1ncc(NC(=O)C(CC(N)=O)NC(=O)CC2CCC(C)O2)cc1Cl C1(C(=O)N(CCC(N2CC(F)(CF)C2)=O)CCO)Cc2ccccc2C1 C1(C(=O)NC(C)CC)C(C)(C)C1(C)C.c1(C(=O)N)ccc(C(F)(F)F)cc1 C#Cc1cc(C(=O)Nc2ccc(OCC3CCCO3)cc2)cc(N)c1 Cc1cc(N)c(C(N2CC(NC(C3CCOC3)=O)C(C)(C)C2)=O)cc1F c1(C(=O)NCCCOCC(C)(C)NC(C(CCC)OC)=O)nccc(Cl)c1C c1(NC(=O)NCCC(C)SC)ccc(-c2ccc(CCCC)cc2)cc1 c1(-c2cccc(C=C)c2)cc(C(=O)Nc2cc(Cl)cnc2Br)cc2c[nH]nc12 CC1=C(C(=O)NCCC(C)NC(c2csnc2Cl)=O)CCC1 C1(C(=O)OCC)CC(F)(C(=O)N)C1.c1(CC=O)ccccc1.CC(O)C N1(C(CCCCCC)=O)CC(NC(=O)CC2CSC2)C(C2CC2)C1 C1(NC(Cc2cc(C)c(CO)cc2)=O)CC2CCC(C1)N2C(c1ccsc1)=O C(=O)(CC1CCOc2ccccc21)N1CC(NC(CCSC)=O)C(C2CC2)C1 C1(C(=O)NCC(C(C)O)C)C=CCN(C(=O)CN2CCC(C)C2)C1 C#Cc1cn(C)nc1C(=O)N(C1CCC(NC(C2CCC(C)(C)C2)=O)CC1)C N1(C(C2(CC=C)CCC2)=O)CCC(CCC(=O)NCC2CC3C=CC2C3)CC1 C(=O)(C(CNC(=O)CC1CC2CCC1O2)(CC)CC)NC(CCC)c1nn[nH]n1 C1(N(C(c2cnc(C)[nH]2)=O)C)CN(C(c2cccc(CO)c2)=O)CC1F c1(C(=O)NC(C(CO)NC(CCNC(=O)NC)=O)C)ccncc1.N(C)C N1(C(C(C)=CC2CC2)=O)CCC(NC(c2ccc(F)c(C(F)(F)F)c2)=O)CC1C N=c1nc2c(C(N3CCSCC3C3CC3)=O)cc(Cl)cn2[nH]1 N1(C(c2cccc(OCC)c2)=O)CC(N=c2[nH]c(Cl)ncc2C2CC2)CC1C c1(CCC(N2C(C)CCC2)=O)c(F)cccc1F.C(C(COC)C(=O)NC)OC CCC(C)C(C)(O)CNC(=O)CN(C)C(c1cc(C)c(F)cn1)=O N1(C(C2C(C)C(=O)C2)=O)CCOC(C(F)(F)C(F)(F)F)C1 Cc1cccc(C(=O)NC2CCC2NC(C2CC(F)CN2C)=O)n1 c1(C(=O)NC(C2(O)CCN(c3ncnc(C)c3F)C2)C)ccc2n[nH]cc2c1Cl C(=O)(CCCCCCc1ccccc1)NC1CN(C(C(C)OCC)=O)CC(C)C1 C1(C(N(CC(C)SC)C)=O)CCCCN1C(c1ncn(C(C)C)n1)=O N1(CCNC(CCC#C)=O)CCC(NC(c2cnc(C3CC3)[nH]2)=O)CC1 C#CC1(NC(c2ccc3c(c2)OCO3)C)CCC(C)(C)C1 c1(C(=O)NCC2CCCCN2C(c2cscn2)=O)cc(Cl)cc(I)c1 C(=O)(C(C)CC(=O)OC)NCCC(=C)CNC(=O)CCc1ccncc1Br Cc1cccc(CCC(=O)N(C2CCCC(NC(c3snnc3C)=O)C2)C)c1 N1(C(c2c(C)nsc2N)=O)CCCCC(NC(=O)C(c2cccc(Cl)c2)O)C1 C(C(C)(C)CC(=O)NC1CCCN(O)C1=O)NC(C(F)=CCC)=O c1(C(=O)NC2CCN(C(C(C3CC3)OC)=O)CC(O)C2)cccc2c1CNC2=O C(CN=c1[nH]c(=NCC2CCC(O)C2)[nH]c2c1CCC2)NC(=O)OC(C)(C)C c1(CC)onc(C(=O)N(C2CCC(NC(c3cnc(C4CC4)o3)=O)C2)C)c1C C1(NC(C(CSC)(C)C)=O)CC2CC1N(C(C1NC(=O)OC1C)=O)C2 C1(CNC(c2n[nH]c(C)c2Cl)=O)CCCN(C(=O)C#CC2(C(F)(F)F)CC2)CC1 c1(-c2nc(C(C)C3CC3)nn2Cc2cccnc2)ccc2cnnn2c1 N1(C(C2C(=C)CC2)=O)CC(O)CC1CNC(=O)CC(C)C Cn1cnnc1SCC(N1CCCC1CNCC1(N2CCOCC2)CCCC1)=O c1(C(N(C(CNC(C(S(CCC)(=O)=O)C)=O)C)C)=O)cc(C)c2nc(C)cn2n1 c1(N2CCC(Cc3cn(CC)nn3)C2)ncc([N+](=O)[O-])cc1C(F)F CC1CCC(C)(CNC(=O)CCCN(C)C(c2cnn(C(F)F)c2)=O)CC1 C1(CNC(Cc2cc(C)sc2)=O)CCCCC1NC(c1c[nH]cc1C1CC1)=O C1(CNC(CNC(CCC)=O)=O)(CO)CCN(C(=O)CCC(C)OC)C1 N1(C(CC2(OC)CCCC2)=O)CC(NC(c2cc(C)nn2C(F)F)=O)CC1.S CCCCC(O)C(C)C(=O)NCCN(C)C(C1CC=CC1)=O c1(C(=O)NCc2c(C)scn2)ccnc(C)c1.c1(C=O)cn(C(C)C)nn1.N n1(CC)nnc(C)c1C(=O)N(CCCN(C(=O)C=CC1(C)COC1)C)C N1(C(CC2CCCN(C(C(CC)(C)COC)=O)CC2)=O)CCC(C2CCC2)C1 C12(C(=O)NC(C=C)C)CC(C)(CN1C(c1c[nH]cc1CC)=O)C2 c1(C(=O)NC2C(OC)CCCC2)ccnc(OC(C)C)c1F C1(C(=O)NC(CNC(c2oc(C)c(CO)c2)=O)CO)CCS(=O)(=O)C12CCC2 CC1CC(NC(C2(CO)CC2)=O)CCN1C(C1CCCCS1(=O)=O)=O CC(O)(CC(=O)N1CCC2(NC(C3CC4C(C3)C4(F)F)=O)CCCC12)C(F)(F)F C(CCCCCNC(=O)CC(=O)N(C)C)N(C(CNC(CCC)=O)=O)C N1(C(CC=CCNC(CC)=O)=O)CC2C(=O)NC(=O)C2C1 C1(OC)CCN(N2CCC(Cc3ccc(F)cn3)C2)C1 C(CCN=C(NCc1cncn1C)N1CC=C(c2cccc(F)c2)CC1)OC N1(C(CCc2cc(C)n(C)n2)=O)CCC(NC(=O)COC2CCCC2)CC1C N1(C(C(CNC(Cc2cnc(C)s2)=O)CC2CC2)=O)CC(=O)NC(C)C1 N1(C(CC2CCC(=O)N2)=O)CCC(C(=O)NCCc2ccncc2)C(O)C1 C(=O)(C(Cc1ccoc1)NC(c1cc(Cl)n[nH]1)=O)NC(C(N)=O)C1CC1 C(=O)(CCC(C)N(C)C)NC(COC)C(=O)NC(C)CCO N1(C(c2cc(Cl)cnc2O)=O)CCN(C(C2(Cl)CC2)=O)CC(O)C1 c1(NC(C2CCC(NC(CC(C)(C)O)=O)C2)=O)cc(F)c(Cl)cc1F Cc1ncc(C(=O)NC2CCCC(NC(=O)CC3CC(O)C3(C)C)C2)n1C c1(C(=O)NCCCNC(C2C(CC)C2)=O)ccc(-c2ccco2)s1 CC(C)CCC(F)C(=O)NCC(C)(C)OCC(=O)NOC1CCOC1 c1(CN2CC(NC(N(CCN(C)C)C)=O)C2)ccc(N(C)C)nc1 c1(C(=O)NCc2ccc(C(=O)NCC(CC)C)s2)c[nH]c(C)cc1=O c1(C(=O)NCC(CC)NC(c2ccc(C)c(CO)c2)=O)cc(Cl)cnc1O C1(C(=O)NCC(C)(CC)NC(CCCOCCC)=O)CC(F)(F)C1(C)C C(=O)(C(F)C(F)(F)C(F)(F)F)N.Cc1cccc2c(C(=O)N(C(C)C)C)n[nH]c12 Cc1ccc(C(=O)NC(C)CCCNC(C2CCC(=O)C2)=O)c(C)c1 N1(C(C2N(C(C(C)OC)=O)CC23CCCC3)=O)CC(C)C12CCOCC2 C=CC(C(=O)NC1CCCC1)NC(=O)OC(C)(C)C.C1(C=O)CCCC1 c1(C(c2n(C(C)C)nnn2)NCCCCCF)cccc(S(N)(=O)=O)c1 CC(CN(C)C)CCC(=O)N1CCC(CC(N)=O)CC1.C(=O)CN(C)C1CC1.N c1(C(N2C(C)C(C)N(C)CC2)=O)cncc2nc(O)[nH]c12 CC1=NNC(=O)C1CCC(=O)N.C(C)(C)CC.c1(C=O)cnc(C(F)(F)F)s1 N1(C(c2ncnc(C)c2C)=O)CCCC12CCC(NC(C1CC1F)=O)CC2 C1(C(=O)NCC2(C)CCC(NC(=O)C3=CCCOC3)CC2)CCn2nnnc2C1 CC1CCN(C(c2sc(F)cc2Cl)=O)C1CNC(=O)Cn1ncn(C)c1=O N1(C(C2CC3(CCC3)C2)=O)CCC(C(=O)O)C(C(=O)O)C1 c1(OC)nccc(C(N2CCN(S(=O)(=O)CCCl)C(C)C2)=O)c1F Cc1ccc(C(=O)NC2CCN(C(=O)CCc3cnco3)C2(C)C)cc1CO C(=O)(CCCN=c1nccc[nH]1)N1CC(C(C)NC(=O)C=C2CCN(C)CC2)C1 c1(CC(=O)NC2CN(C(C=NOC)=O)CC2C2CC2)ccc2nc(O)[nH]c2c1 c1(CNC(C(CC2CN(C(c3cnc(CC)o3)=O)C2)F)=O)cccc(CO)c1 Cc1c(CN=C(NCc2ccco2)NCC23CC(C2)C(C)O3)cccc1F N1(C(C=C(CC)C)=O)CC(NC(c2ccn(CC)c(=O)c2)=O)C(C2CC2)C1 N1(C(c2ccc(CC3CCC3)cc2)C(=O)NCC(C)C)CCN2CCC1C2 C(=O)(CS(=O)(=O)C1CCCC1)N(CC(CC)NC(=O)CSc1nccn1C)C N1(C(Cn2ncc(C)c2)=O)CCC(NC(c2cc(F)c[nH]2)=O)C12CCC2 C1(CNC(C(C2CCCN(C(C3(C)CC(C)C3)=O)C2)C)=O)OCCCC1(C)C Cc1ncc2n1CC(C(N1CC(NC(=O)CCc3cn(C)nn3)C(C)C1)=O)CC2 O(NC(=O)C(F)C1(O)CN(C(c2cocc2C(N)=O)=O)C1)CCCCC N1(C(C2N(C(COC(C)C)=O)CCSC2)=O)CCOC(C)C1C C1(CC#C)(C(=O)NCCCCCNC(=O)COCCC(C)C)CCCO1 C(C1=NOC2CN(C(=O)CC3=NNC(=O)C3)CC12)NC(c1cc(C(C)C)on1)=O Cc1cccc(Br)c1C(=O)NC1CC2(C1)CN(C(=O)Cc1ccns1)C2 N1(C(C2(CC(C)C)CCC2)=O)CC2C=CC1C(C=O)C2.c1(C2CC2)nccs1.N C1(CCC)(NC(=O)C=Cc2nc(C)co2)CCCN(C(c2ccc(C)[nH]2)=O)C1 c1(C(=O)NC2CN(Cc3cncnc3)CC2F)cc2cc[nH]c2cc1Cl CCC(CC)C(CNC(=O)NCC(c1ccc(OC)cc1)OC)N(C)C c1(C(N2CC(O)(C(CNC(C=NOC)=O)(C)C)C2)=O)c2c(nn1C)CCCC2 N1(C(c2ccc(C(C)C)s2)=O)CC(C)CN(C(=O)C(F)CC2CCOC2)CC1C N1(C(c2c(C)ccc(C)c2N)=O)CCN(C(C2CCS2(=O)=O)=O)C2(CCC2)C1 N1(C(C(=O)NC2CC2)=O)CCC2(CCCN2c2ccnc(C(F)(F)F)n2)CC1 Cc1ccc2c(N3CCCCC3CCNC(C3CCOCC3)=O)ncnc2c1 N1(C(C(=O)NCC(C)(C)N(C)CC)=O)CCC(n2nc(C)nc2C)CC1 c1(C(N2CCC(NC(=O)CC(c3cccc(F)c3)O)CC2)=O)ccc([N+](=O)[O-])s1 N1(C(C2CC(C)(F)C2)=O)CC(NC(C2(n3cncn3)CC2)=O)C(O)C1 C1(C(N(CCSC)CC)=O)CN(C(C2CCC(=O)NC2)=O)CC1(F)F CN(C)N=Nc1ccccc1C(=O)NCC1(O)CN(C(=O)COC(F)(F)F)C1 CC1CN(C(c2cnc(C(N)=O)s2)=O)CC1NC(=O)C.C(=O)CN(C)C CCCC(C)CC(=O)NC1(CNC(c2cnn(C)c2F)=O)CCOC1 c1(C(N2C(CCCNC(c3c(C)c[nH]n3)=O)CCC2)=O)ccc2cnccc2n1 Cc1[nH]nc2c1C(Nc1ncc(C(F)F)cn1)CCC2 CC(=O)C(C)(C)CC(=O)N1CCCC(C)(CNC(=O)C=Cc2cnc[nH]2)C1 C(=O)(CCCC#N)NCC1CCC(C(N(CC#C)CCO)=O)O1 c1(C(N2CC3C(CNC(C(C(C)C)(C)C)=O)(C3)C2)=O)c(O)cnc2ccccc12 c1(C(=O)NC(CC)CNC(=O)CC(O)CC2CC2)nc(C)c(C)nc1O C(=O)(CC(C)CC(C)(C)C)NC1CCC(C)N(c2ncnc3ccccc23)C1 c1(C(N2CC(C(=O)NCCNC(CC(C)OC)=O)C2)=O)ccc(O)cc1F C1CCC2(CCN(C(=O)CSC(F)F)CC2)C1.CCS(=O)(=O)NC(C)C(=O)N C(=O)(C1CCCc2nncn21)N1CCC(NC(c2c(C)cco2)=O)(CF)C1 C1(NC(=O)CCC2CC2(F)F)COCCC1NC(=O)Cn1cc(CO)nn1 C(c1ccc(Br)o1)=C(C)C(=O)NC(C)(C)CNC(c1coc(C)c1)=O n1(CCC(N2CC3C(C)(CC3)C2)=O)c(CO)nc2ccccc12 c1(C(N(CCNC(CCC(=C)Cl)=O)CC)=O)cc(Br)c(C)c([N+](=O)[O-])c1 N(C1CN(C(=O)Cc2n[nH]c(=N)s2)CCc2ccccc21)C(C(C)=CC)=O c1(C(=O)NCC(C)CC(=O)NCCCCN2CCCC2)n[nH]c2c1COC2 CCC(C)C(C(=O)N1CC([N+](=O)[O-])C1)N(C(=O)C(n1ccnc1C)C)C c1(C(=O)NCC2C3CN(C(C4CC4F)=O)CC23)ccc(F)c(Cl)c1F C(=O)(C1=CC2C=CC1C2)N(C1CCCN(C(Cc2c(C)cccc2)=O)CC1)C c1(CC(=O)NC(CNC(CCCN(C(C)=O)C)=O)(C)C2CC2)c(Cl)cnn1C N1(C(C(CC)=CC)=O)CC(C(N2CC(C(C)CC)C2)=O)CCC1C c1(CC(=O)N(C)C)cn2cc(F)ccc2n1.C(C)(C(=O)NC1CC1)=C(C)C C=C(C)C(CC(=O)NCC1CC(C)CN(C(=O)Cc2sccc2C)C1)OCC C1(NC(c2c(CC)ncs2)=O)CN(C(=O)CN2CC=CC2)CC1C(F)(F)F C1(NC2(c3n(Cc4nnn(C)n4)nnn3)CC(C)(CBr)C2)CC2CCCCN2C1 C12(NC(c3c(C)noc3C)=O)CCCC1(F)CN(C(=O)Cc1c(C)n[nH]c1C)C2 c1(C(C)(C)NCc2cnn(C3CCC3)c2)ccc(Cl)cc1 Cn1cc(C(=O)NCC2CN(C(c3ccco3)=O)C2)c(C(F)(F)F)c1 c1(NC(=O)CC2COCC2O)cc(F)ccc1NC(c1cccs1)=O Cc1ccc2c(C(N3CCC(N4CCOCC4)(C(N)=O)CC3)=O)ccnc2c1Cl C1(CNC(=O)Cc2ccoc2)CC2(CO1)CN(C(c1ccncc1O)=O)C2 CC1(C)CC1(Br)C(N1CCC1CNC(=O)Cn1cccc1)=O Cc1[nH]nc2c1CC(c1nc(C(C)O)nn1-c1ccc(C(F)(F)F)cc1)CC2 C1(NC(c2ccc(C)o2)=O)CC(=O)N(C2CN(C(=O)C(C)SC(F)(F)F)C2)C1 C1(C)(NC(c2cc(CNC(C(CC)OCC)=O)sc2)=O)CCCCCC1 C1(C(=O)NCCCNC(c2c(SC)snn2)=O)CC1C1CCCC1 C1(NC(C2CC(OCC)C2)=O)CC2CC1N(C(c1ncc(Br)cc1N)=O)C2 N1(C(C(CCC)NC(N)=O)=O)CC2(CCCCN(C(=O)C(CCC)CCC)C2)C1 CCCC(C)(O)CC(=O)NCc1cccc(CN(C(=O)Cc2ccnn2C)C)c1 CCC(CC(F)F)C(=O)N1CC2CCOC2(CNC(=O)C=Cc2ccoc2)C1 c1(OC)ccnc(O)c1C(=O)NC1CN(C(c2onc(C)c2C)=O)CCC1O N1(C(c2ccc(N(C)C)nc2)C(=O)NC(C)(C)C)CC=C(c2ccncc2)CC1 c1(C(C)=O)cc(C(N2CC3C(NC(C4COCC4C(F)F)=O)C3C2)=O)ccc1O S(=O)(=O)(CC(=O)N1CCC(COC)(NC(C2CCCN(C)C2)=O)C1)NC C(CCCC(C)(C)C(=O)NNC(=O)C(O)CC(C)C)NC(CCC(CC)CC)=O c1(OC)cc(C(=O)NC(C)C(CO)NC(=O)C2CC2)cc2c1OCCO2 C=CC(C)(O)CC(=O)N(CC(=O)NC12CCCC1OCC2)C1CC1 c1(C(N(C)CCOCCN(C(=O)C(C)(C)Br)C)=O)ccc(Cl)cn1 C(C1=CCCC1)NC(=O)NCC1C(C)(Br)C1 c1(C(N(C2CCN(C(=O)Cc3cccnc3)CC2)CC#C)=O)cnc(F)cc1C C(=O)(C1=CC2(CCOC2)C1)NC1(CC=C)CCCN(C(=O)Cc2cnnn2C)C1 N1(C(c2c(C)occ2)=O)CCCC(C)(C)C1C(=O)NCc1cncn1C(C)C C1(C)(OC)CCCN(c2ncnc(NC(c3ccc(C)cc3)C)c2C)C1 c1(NC(C(CN(C)C(C2COCC2C(N)=O)=O)(C)C)=O)cccc2nccn12 c1(C(=O)NCCCN(C(=O)C=C2CCC2)CC)cc2ccccc2nc1C.O CC1CN(C(=O)C(N2CCOCC2)C)CC1(C)CNC(=O)CCC1CCC(=O)N1 c1(CN)sccc1C(=O)NC1CCC(NC(=O)C(F)CC2CCCCC2)C1 N1(C(C2CN(C(C)=O)C2)=O)CCN(C(C2(Cl)CC2(C)C)=O)CC1CC(F)(F)F C(CNC(C12CCC(C1)C2)=O)(C(C)C(C)C)NC(c1c(C)n(C)cc1)=O CC(C)(C)C(CCc1ccccc1)C(=O)NCCNC(=O)CC1(O)CCOC1 C1(O)(c2cn(CC(CC3CCCO3)OC)nn2)CCC(F)(F)CC1 Cc1cc(N(C)C)ccc1C(=O)NC12CC1CN(C(=O)CCNC(N)=O)C2 c1(C(N2CC3C(NC(c4occc4F)=O)C3C2)=O)cc2cccnn2n1 c1(C(=O)NC2(C)CCC2)ccc(F)cc1C#N.C(F)(c1ccccc1)=CC(=O)N c1(CC)cc(C(=O)NCC(CC(C)C)NC(c2ccoc2)=O)ccc1O C12(C(=O)OC)CCC(C(=O)NC(=O)CCCC(C)N)(C1)C2.c1ccccc1 c1(NC(C(CC(C)C)ONC(c2cc(C)[nH]c2)=O)=O)ccc2c(c1)OCC2 C1(C(N2CCC(F)(C(N(C)CC3CCN(C)C3)=O)C2)=O)CCCC1C1CC1 N1(C(c2[nH]cc(CC)c2)=O)CC(NC(C2CC2(Cl)Cl)=O)C(c2ccnn2C)C1 N#Cc1ccsc1C(=O)NCCCCCNC(C1CCC1F)=O c1(C=O)ccc(C#N)c(F)c1.C1COCC1.C(C(=O)N)=CCN(CC)CC Nc1cc(Cl)nc(C(N2CCC(F)(CNC(=O)C3=CCC3)CC2)=O)c1Cl C1(C(N2CC3C(c4cn(C(COC)COC)nn4)C3C2)=O)CCCC(C)(C)C1 N1(C(c2n(CC#C)ccn2)C(=O)NC)CC(C)(C)C1c1nccn1C CN1C2CCC1CC(NC(C1C=CCN(C(c3ccncc3N)=O)C1)=O)C2 c1(C(CNCCn2ncc(S(C)(=O)=O)c2)O)ccc(S(C)(=O)=O)cc1 Cc1cccc(C)c1-n1cc(C(C)N(C)C(C2(O)CCCCCC2)=O)nn1 c1(C(=O)NC2CN(C(c3c(C)c(C4CC4)[nH]n3)=O)CC2C)cc(F)c(F)cc1F Cc1ccc(Cl)c(C2CCCN2C(=O)C(F)(F)C2CCOCC2)c1 Cc1nsc(C)c1C(=O)NCC(C1CC1)N(C(=O)C(N1CCCC(O)C1)C)C c1(C=O)cc2c(F)cccc2s1.CCC(C)C(C(=O)NCC(O)C)NC(C)=O.N C1(C(=O)Nc2cccc(NC(C)=O)n2)CC(F)CN(Cc2cc(Cl)ccc2F)C1 N1(C(C2(NC(C3C4CCCOC34)=O)CSC2)=O)CCN2CCC1C2 Cc1nn(C)cc1CC(=O)NC1CN(C(C2(NC(N)=O)CCCCC2)=O)CC1C C(C1CCCCC1)=CC(=O)NC(C)CCCNC(=O)CC1CN(C)C1 c1(CC)cc(C(=O)NC2CCC(NC(c3ncn(CC)n3)=O)CC2)cc(F)c1 c1(C=O)cccc(N)n1.C1(C(F)(F)F)(C(N(C)CCO)=O)CCCCC1.CC c1(Cc2n(C)cnc2)ccc(C(=O)NC(C(F)F)C2CCCO2)cc1Cl c1(C(N2CC(C)CC2)=O)cc(N)ccc1C.C1(C(=O)NC)(OCC)CCCC1 C1(NC(C(COC)O)=O)CCCCN(C(c2csc(C3CCCCC3)c2)=O)C1 C1(CNC(c2csnn2)=O)CCC2CN(C(=O)C(C3CC(F)(F)C3)O)CC12 C1(Cc2ccccc2)CC(N=c2nc(CC3CC3)[nH][nH]2)CCO1 CC1(C)C=C(C(=O)NCCN(C2CCCC2)C(c2cc(Br)co2)=O)C1 N1(c2ccc(C#N)nn2)C2CCC1CN(C(C13CCC(F)(CC1)CC3)=O)CC2 C(C)(N=c1c(C)c(C)[nH]c2ccccc12)c1c(C)cccc1C CC1(C)CNc2ccc(C(=O)NC(C)(C)C3CCC3)cc21.c1(C(=O)N)cocn1 C1(F)CCN(C(=O)C=CC(c2ccccc2)=O)C1.C1(CC(=O)N)CC2CC2C1 c1(C(=O)NC(C=CC(=O)N(CCOCC=C)C)C)cn(C)c(=O)n1C C1(C(=O)NC2CCN(CC=C)CC2)N(C(=O)CCC(C)(F)F)CC12CCCC2 c1(C(N(CC(CNC(c2ncc(CC)s2)=O)C)C)=O)ccnc2[nH]cnc12 N1(C(C(CC2CC2)OC)=O)CC(N(C(=O)C)C)C(O)C1.C=O.C1CC1.N C1(CNC(CCCc2onc(CC)n2)=O)CN(C(C2CSC2)=O)CCO1 C1(C)(C(N2CC(NC(C=CCCC)=O)C3(C2)CC3)=O)CC(C(F)(F)F)=NO1 N1(C(CCC#CC)=O)CCC(C(N2CCC(C(=O)OC)C2)=O)CC1CC CCCCC(F)C(=O)NC1(C(N2CCC(CC)C2)=O)CCC(C)(C)C1 c1(CC(N2CC(CNC(CCCCSC)=O)C3C2C3)=O)c(C)nn(C)c1C C1(C(=O)NCc2ncc(C)s2)CC(C)CN(C(=O)C(c2cccn2C)=O)C1 c1(C(=O)N)cnc2ncnn2c1C(C)C.N1(C(C=CC)=O)C2CCC1CC(C)C2 N1(C(C(C=C)C)=O)CCC(C=C)(C(=O)NC(CO)CCCC)C1 N1(C(c2n(CCC)nc(C)c2Cl)C(=O)N)CCOC(C)(C)CC1.C1(C)(CC)CC1 N1(C(CSc2n(C)ccn2)=O)CC(NC(C2CC2C2CC2)=O)C(O)C1 N1(C(C2C(OC)CCCC2)=O)CC2(CCC(NCc3ccccn3)C2)C1 C1(S(C)(=O)=O)(C(=O)OC)CC(NC(C2(c3ccnc(C)c3)CCC2)=O)C1 Cc1cc(C(=O)N(C2CCCCC2NC(c2ocnc2C)=O)C)cc(C)c1 Cc1ccc(C(=O)NCC(C2CCN(C(=O)C(C)N(C)C)CC2)(C)O)c(F)c1F Cc1oc(C)c(C(=O)NC2COCC2NC(=O)C(C)N(C)C)c1Br N1(C(CN(C)C)=O)CCCC(N(C(=O)CCCCn2ccnn2)C)C1 N1(C(C(CC)SC)=O)CC=C(CCNC(=O)CC2CC2Cc2ccccc2)CC1 N1(C(c2cncc(NCC)c2)=O)CC(C2CN(C(=O)CCCC(=O)N(C)C)C2)C1 N1(C(c2cc(C)c(C)nc2C)=O)CCC2(CCC2)C(NC(=O)C(O)CN(C)C)C1 N1(C(c2n[nH]c(C)c2O)=O)CCN(C(=O)Cn2nccn2)CC1C1CCCC1 c1(OC(C)C)ccccc1C(=O)N(CCC)C.C1(C=O)CCCN(C(N)=O)C1.N C1(NC(C2(COC)C=CCC2)=O)CCCCC1.c1(CC=O)cnc(C)[nH]1.C N1(C(c2ccc(C(C)C)nc2)=O)CC2(CCCC2NC(=O)Cc2cnc[nH]2)C1 C1(CNC(c2c(C)ncnc2O)=O)CN(C(C2CSC2)=O)CCC12CCOC2 N1(C(C2N(C(C)=O)CSC2)=O)CCC(C(=O)NCc2ccn(C3CC3)n2)C1C C1(CCOC)(C=O)CCN(C(=O)C(F)C(C)(C)O)CC1.N(S(N)(=O)=O)CC N1(C(c2cc(Br)c(C)s2)C(=O)NCCCSC)CCN(C2CC2)CC1C c1(CC)cc(C(N2CC(NC(=O)CCN3CCC(C)CC3)CC2C)=O)c(C)nn1 C1(C(=O)NCC2N(C(c3c(C)nn(C)c3C)=O)CCC2)CCC2CC1C2(C)C c1(C(N(CC(c2ccc(F)cc2F)C)C)=O)ccc2c(c1)C(C)C(C)O2 N1(C(C2CCC(=O)NC2)=O)CC(NC(=O)CSC(F)F)C2(CCC2)C1 C(=O)(C1CSc2ccccc21)NC1CN(C(Cc2c(C)ccc(F)c2)=O)CC1O c1cccs1.c1(CC(C)NC(CNC(=O)NCC)=O)ncco1 C1(C=O)COCC1(C)C.N1(C(C)=O)CCCC1C.C(=O)(C)NC.CC(N)=O.N C1(C(N(C2CCCCC2)CC)=O)CCCNS1(=O)=O.CC1(C(=O)N)CC2CC2C1 C1(CCC)CN(C(=O)Cc2cc(C)ccc2C)CCN1C(C1CCCN1N=O)=O C1(NC(Cn2c(CCC)nnc2S)=O)CC12CCN(C(=O)C(COC)OC)CC2 Cc1c(C(N2CCN(C(=O)Cn3cnnc3)C3(CCC3)C2)=O)ccc2n[nH]cc12 N1(C2CN(C(Cc3c(C)non3)=O)C2)CCN(C(=O)CC2CC3COCC23)CC1 C=CC(CCC)CC(=O)N1CCN(CCN(C(=O)C(C)Cn2cccn2)C)CC1 C1(C(=O)OC)CN(C(=O)NCC2(F)CC(CO)C2)C2(CCC2)CO1 Cc1cc(C(N2CCCC2C(C)NC(c2cc[nH]n2)=O)=O)cc2ccsc12 c1(CCC)nc(C)c(C(N2CC(F)CC2)=O)o1.C(C(F)(F)F)C1(C=O)CC1.C N1(C(c2ccc(OCC=C)cc2)=O)CCCC(C)C1.C1(C=O)(N(C)C)CC1.C CN1CC(O)CC1(C)C(N1CCC(C(N2CC(O)(CCO)C2)=O)CC1)=O C1(CC)CN(C(C2(Cl)CC2(C)C)=O)CCN1C(c1cc(CCOC)on1)=O C(CC(C)(C)C)(C(=O)NC(C#C)CC1CC1)NC(c1ccc(C#C)o1)=O CC1(C)C2CN(C(c3cc([N+](=O)[O-])cs3)=O)C(C(=O)NCc3cn[nH]c3)C12 c1(C(N2CCCC3(CCCO3)C2)=O)cc2c(Br)cccc2c(O)n1 C1(O)(C(=O)NC(CCCNC(CCCOC)=O)C)CCCC(C)(C)C1 CC(C)CCCNC(C1(C)CC1C)=O.c1cccc(C(F)(F)F)c1.C(=O)C.N C1(C(N2CCC(C)C2C(N2CCCC2CN(C)C)=O)=O)CC12CCOCC2 C(=O)(C(F)(F)C(F)(F)F)NC1CC2CN(C(CCCC3(C)N=N3)=O)CC21 C(c1cnc(O)nc1O)=CC(N1C(CC(=O)NC(C#C)(C)C)CCC1)=O c1(CN(CC)CC)cc(F)c(C(F)(F)F)cc1F.C1(O)(CC=O)CCC1 c1(CNC(C)=O)nc2c(s1)CN(C(=O)CCC(C)c1ccccc1)CC2 C12(C(N(C(C#C)C)C)=O)COC(C1)C(NC(=O)C(C)n1ccnn1)C2 c1(C(C)NC(N2CCOCC(F)(F)C2)=O)nc2cc(Cl)c(Cl)cc2[nH]1 C1(C(=O)N)CC(C)CCC1C(C)C.C#CC(C)(C)C(=O)NCC(C)C1CCC1 C(C)(CC(C)(C)C)NC(c1cnc(CC)s1)c1nnnn1CCSC n1(CC(=O)N(C(C)CCNC(C2(C(C)(C)C)CCC2)=O)C)ccccc1=O CCC(CNc1ccc(C(N2CCCCC2)=O)cc1)(C(=O)OC)c1ccccc1 c1(C(N2CC(O)C2)=O)ccc2sncc2c1.c1(CC)sc(=N)[nH]c1C(=O)NC Cc1[nH]c(=NC(C)C(C2CCCC2)NC(=O)Cc2cc[nH]n2)ccc1C#N C(=O)(C(C)S(C)(=O)=O)N1CC(CNC(COCCCC#C)=O)OCC1 CCC(CC(=O)NCc1ncccc1C(=O)NCCSCCCO)SC c1(C(=O)NCCC2(O)CCN(C(C(CC)OC)=O)C2)csc2cc(OC)ccc12 O=C1NCC(C(=O)NCC=CCNC(C2(CC3CC3)CCCO2)=O)N1 c1(C(=O)OC)cccc2nc(NC(=O)C(C(C)(C)C)OC(C)=O)n(C)c12 c1(C(=O)NCC(C2CCC2)NC(C2C(C)C2C)=O)c[nH]c2cc(F)ccc12 CC(C)(C)CCN(C(=O)C(C)n1ccnc1)C.C1(CC=O)CCC1.C(C)=O.CO C=CCCN=C(NC1CCCN(C(=O)OC(C)(C)C)C1)NC1CC(=O)N(CC)C1 c1(C(N2CCN(C(C34CCC(OC)C3C4)=O)CC2C)=O)cc(Cl)c(F)cc1N CCC(C(=O)N1CCC(CCNC(C2(CF)CC2(F)F)=O)CC1)C(C)(F)F Cc1cc(C)n(-c2cnc(C(=O)OCc3csc(Br)n3)cn2)n1 N1(C(c2c(C(=O)OC)cncc2)=O)CCC(C)(C)CC1.C(=O)(CCC(C)(F)F)N N1(C(C(CC)SC)=O)CCN(C(c2cnc(C)nc2)=O)CC1CC1CC1 C(=O)(C1=NOC2(CCC2)C1)N.c1(CC)cc(C(=O)NC(C)C(C)C)n(C)n1 N=c1[nH]c(CCC(=O)NCCC2CCN(C(C3(n4nccn4)CC3)=O)C2)cs1 Cc1nc(CNC(c2cc(CNC(=O)Cc3cn[nH]c3)cs2)=O)cs1 N1(CCN(C2CCCC2C)CC)CCC(C(C)N(C(C2CCCCO2)=O)C)CC1 C#CCC(C)(C)C(=O)NC1CCC(CNC(=O)CC2COC(=O)N2)CC1 N1(C(c2ncc(C)nc2)=O)CCC2(CCCN2C(=O)CC2CCC(C)(C)CO2)CC1 N1(C(C(F)=CCC)=O)CC(NC(c2ccc3c(n2)CCC3)=O)CC12CCOC2 c1(C(=O)NCC2C(CNC(Cn3c(C)ccn3)=O)C2)ccnc2ncnn12 Cc1cc(C(=O)Nc2ccccc2-n2nccn2)ccc1[N+](=O)[O-] c1(C(N2CC(C)C(NC(=O)C(O)C3=CCCCC3)C2)=O)cccc2c1OCCO2 N1(C(C(c2ccccc2)C)=O)CC(C)CC(C)(C)C1.N(S(N)(=O)=O)CC(=O)N CC(C)(C)C(=O)CCC(=O)N1CCC(NC(=O)C=Cc2ccccc2)C1(C)C C1(NC(c2cc(OC)c(I)cc2)=O)CN(C(c2ccccc2)=O)CC(F)(F)C1 Cc1cnc(NC(C2CCCN(C(c3ccc(F)c(Br)c3)=O)CC2)=O)c(O)c1 C1(C=O)CC(S(C)(=O)=O)CN1C(=O)CC1CC1.C(=O)(C(C)N=[N+]=[N-])N S(=O)(=O)(c1[nH]c(=NCCCC(C)(C)CO)ccc1Br)NCCN(C1CC1)CC c1(C(=O)OCC)cc2n(n1)CC(C)N(C(=O)CCn1cnc(C)cc1=O)C2 c1(CC)cccc(C(N2CC(C)(NC(c3cncc(Br)c3)=O)C2)=O)c1N c1(C(C)C)nn(C)cc1C(=O)N(C)CCNC(c1c(Cl)nsc1Cl)=O C1(C(=O)NCC2N(C)CCN(C(=O)C3=CCC3)C2)CCc2nc(=N)[nH]cc2C1 N1(C(c2cc(C)sc2)=O)CCCC(C)C1CCNC(=O)CCOCC(F)F C(CC(C(=O)N1CC2CC1C2C(N1CCC(COC)C1)=O)OC)OC C1(Cn2cc(C(C)N(C)C)nn2)CCN(C(c2ncc(Cl)cc2F)=O)CC1(F)F C1(NC(=O)CCC2CC2(Cl)Cl)CCOC12CCN(c1ncnc3[nH]cnc13)CC2 c1(C(=O)NCC2(C)CCN(C(=O)C(Cl)=CCl)C2)cc(Cl)ncc1O C1(C(=O)NCC(N)=O)CC2OCCC2N(C(C2CCNC(=O)C2)=O)C1 N1(C(C2CCCC(OC)C2)=O)CCOCC(NC(C23CC(C2)C(C)(C)O3)=O)C1 N1(C(c2cc(OC)c(O)cc2)=O)CC2ON=C(CNC(=O)Cc3ccsn3)C2C1 c1(C(=O)NC(c2ccccc2Cl)COC)ccc(S(=O)(=O)C(F)(F)F)cc1 C1(NC(c2ccc(OC)o2)=O)CCCCCC1C(=O)N(CC(N1CCCC1)=O)C CC1(C(=O)Nc2cccnc2OC(F)F)CC(c2ccccc2Cl)=NO1 N1(C(c2c(CC)noc2)=O)CC(C)CN(C(=O)CC(=O)N(C)C)CC1C c1(NC(C(=O)NCCS(C=C)(=O)=O)=O)ccc2c(c1)NC(=O)CO2 C=CCCC(O)CNC(=O)C(O)CCNC(C1(C)CCOCC1)=O N1(C(c2c(C)nccc2)=O)CCC(CNC(c2nccn2C(C)C)=O)C(C)C1 C(CC(C)(C)C(=O)NC1CN(C)NC1=O)NC(CC(C)c1ccco1)=O C1(O)(CNC(C2(CC)CC2)=O)CCCN(C(=O)Cc2cccc(O)c2)CC1 N1(C(C(CCC=C)NC(c2sccc2CC)=O)=O)CC2CN(C)CC2(C)C1 c1(C(=O)NC(C2(C)CC2)C)ncc(Cl)cc1Cl.C12(CC=O)CCCC1C2.N CS(=O)(=O)C1CC(CN)C1.C12(Cc3nnnn3CC(F)F)CCCC1C2(F)F Oc1nc2cccc(CNC3CN(c4nc5cccnc5s4)C3)c2o1 C1(C2CC2)(CNC(C(CCC)OC)=O)CCN(C(c2c(Cl)ccc(O)c2N)=O)C1 C(CC(C(=O)NC1CC(O)C1)NC(C1CCC(CO)CC1)=O)OC c1(C(=O)NC(CC(=O)NC(C(C)C)c2nc[nH]n2)C)cc(N)cc(F)c1 C(C(C(=O)NCC(C)(O)CNC(=O)CC)c1ccccc1)OCC=C.CCC C1(NC(C2CCC(CC)CC2)=O)CN(C(c2cncc(OC)c2)=O)CC(F)(F)C1 c1(C(=O)NCC(c2ccccc2Cl)CO)cc(OC(F)(F)F)cc(Br)c1 CCC(CC)(CC(=O)OC)C(=O)NC(CNC(=O)CCC(C)C)C(C)C C(C(C=O)NC(=O)CN(C1CC(C#N)C1)C(c1cc(C)ns1)=O)OC.O C1(CCNC(C2C(C=C)C2)=O)CCCN(C(c2cn(C)[nH]c2=N)=O)CC1 C1(F)(C(N2CC=CC(NC(c3c(OC)scc3)=O)C2)=O)CCS(=O)(=O)C1 CC1CN2CCN1CC2C(=O)NCCC1(O)CCN(C(C2CC=CCO2)=O)CC1 CON(C)S(=O)(=O)c1cc([N+](=O)[O-])ccc1NCC(C)CC(C)C c1(C(=O)NC(CCN(C(=O)CSc2ccncc2)C)(C)C)ccc(N)c(N)n1 c1(CN2CCC(C)(N(C)CC)C2)cc(C)c2occc2c1 C1(O)(CC#C)CC(C(=O)N(C(CNC(=O)CCN(C)C)C2CC2)C)C1 N1(C(C(Cc2cc[nH]n2)NC(CN(CCOC)C)=O)=O)CCCC(O)CC1 Cc1ccnc(C(=O)NC(C)CCNC(=O)CN(C)S(N)(=O)=O)c1F C1(N(C(=O)C(C)(C)CCl)Cc2c(C)ccs2)CCNCC12CC2 c1(OC)cnc(Cl)c(C(=O)N(C2CCN(C(c3ccoc3)=O)C2)C)c1 C1(C(=O)NCc2cn(CCC)nn2)COCCN1C(C1CCCCS1)=O C(=O)(CCCC(C)C)NCc1c(CNC(C(C(C)OC)O)=O)cccn1 C1CN(C(C2(C#N)CC(C)C2)=O)CC1S(C)(=O)=O.Cc1nn(C)c(Cl)c1C=O Cc1noc(N)c1C(=O)NC(CCN(C(=O)Cn1cc(Br)cn1)C)C(C)C N1(C(c2n[nH]nc2C)=O)CC2=C(C1)CN(C(=O)C(=Cc1cnn(C)c1)C)C2.C N1(C(C(C(C)C)C2CCC2)=O)C(CNC(c2cccnc2)=O)CC2CCCC12 C(CCN=C(NCCC1CSCCO1)N1CC(=O)N(C(C)C)C(C)(C)C1)OCC CCCCC(C(=O)N1CC(O)(C(=O)OC)C1)NC(c1cccc(NC)n1)=O N1(CCOC)CCOCC(C)(F)C1.c1c(C#N)cnn1CCC(C)C CCCC(O)C(=O)N1CC2CC1(C(=O)NC(C)C(C)COC)C2 O=C(C1=CS(=O)(=O)CCC1)NCC1CCC1.c1(C(=O)N)ccc2cccnc2n1 N1(C(C2(C#N)CC(F)(F)C2)=O)CC2CCCC(C)C2C1.C1(C=O)CCC(=O)N1.N C1(NC(C2(NC(CN(C)C)=O)CCN(C)C2)=O)CCCCC12CC2 C1(CNC(=O)Cn2cnc(C(F)(F)F)c2)CN(C(=O)C=C2CC2)CCO1 c1(C(=O)NCc2scc(CNC(C(CCC)C)=O)n2)c(O)nnc(C)c1C N1(C(C(C(C)O)(F)F)=O)CC2(CNC(C3CCCN(C(C)C)C3)=O)CCC1CC2 N1(C(C2C(C)C2(F)F)=O)CCCC2(CCN(C(c3ccnc(Cl)c3O)=O)CC2)C1 C12(NC(C(C)c3ccco3)=O)CCCC1N(c1cc(C(C)(C)C)ncn1)CCC2 C1(NC(c2ccc[n+]([O-])c2)=O)CC2CN(C(=O)C=C3CCSCC3)CC12 c1(OC)ccccc1S(=O)(=O)N1Cc2[nH]nc(C(=O)NCC(C)O)c2C1 C1(C(=O)NCC2CN(C(c3c(C)con3)=O)CC2(C)C)Cc2c(C)cccc2O1 c1(OCC)ccc(Cl)nc1C(N1CC(O)(CNC(c2sccc2Cl)=O)C1)=O C1(N(C)C(c2cccc(OCCF)c2)=O)CCCN(C(C2CC2F)=O)CC1 N1(C(c2ccn(CCCC)n2)=O)CCCCC(N(C)C(c2cnc(C)s2)=O)C1 CC1CCN(CCOCc2ccccc2)CC1NC(=O)Cc1cccc(Br)c1 N1(C(c2cc(C)c(F)c(C)c2)=O)CCN(C(c2ccncc2)=O)C2CCCCC12 C=C(C)CCCC(=O)N1CCC(C(C)NC(=O)CCCn2cc(CO)nn2)CC1 C1(CNC(C2CCC(CC)CC2)=O)CC12CCN(C(=O)CN1CC(C)C1)CC2 C1(C(=O)NCC(F)(F)F)CCN(C(=O)CCO)CC1.C1(CC(F)F)CC1.C C(=O)(C(C(C)CC)NC(C1CCNC1=O)=O)N1CC(F)(C(=O)OC)C1 c1(CC(=O)OC)occc1C(=O)NC.C1COCC1.C1(CC=O)CCCO1 C1(C(N2CCC(C(C)OC)CC2)=O)CCCN(C(c2c(F)cncc2F)=O)CC1 C=CC(CC)CC(=O)N1CCOCC1C(=O)NC1(CO)CC(F)(F)C1 c1(C(N2CC3(CCN(C(C4(C#C)CCC4)=O)C3)C2)=O)c(C)ncc2ccccc12 N1(CCC)CCCC(C(=O)NCCCN(C(c2cc(C#N)on2)=O)CC)C1 c1(NC(C2CC(Oc3ccccc3)CN2C(c2cccs2)=O)=O)ccc(F)nc1 C(=O)(NNC(=O)C1CC(=O)N(C)C1)C1C(COC)CCO1 c1(C(=O)NCCc2nc(O)cs2)cnn2c1CN(C(c1ccccn1)=O)CC2 c1(C(=O)NC(CNC(C(CCC)OCC)=O)(C)C(C)C)cccc2c1SCCC2 CN1CCCCCC1C(=O)N(C(C)(C)CC(=O)NCCCC1(O)CC1)C N1(CC(COCC)O)CCOC(C)(C)C1.C1(CC=O)CCC(C(F)(F)F)O1 C1(NC(C(CC)C#N)=O)CN(C(c2cccc3nnn(C)c23)=O)CC2CCCC12 c1(NC(CC)CSC)nc2ccccc2nc1NCC1COC(=O)O1 C1(NC(C(=C(C)C2CC2)F)=O)CN(C(=O)C(C)CCOc2ccccc2)CC1C CC1(CNC(c2cn(Cc3cccs3)nn2)=O)CCN(C(c2ccccn2)=O)C1 c1(C(C)NC(=O)CNC(=O)CNC(=O)CN(C)C)nccc(O)n1 CC1(CC(N2CCCC2CCNC(=O)C(c2ccccc2)F)=O)NC(=O)NC1=O C1(C(N2CC3N(C(C#CC4(C)CC4)=O)CC(C3)C2)=O)Cc2c(F)cccc2O1 c1(C(=O)NCCC(=C)CNC(C2CCCO2)=O)cccc2c(Br)cccc12 c1(N(C)C(C2COCCN2c2ncc(C3CC3)cn2)=O)cccc(S(C)(=O)=O)c1 c1(C(=O)NC2CC(NC(C3C(C)(C)CCC3)=O)C2)cnc2c(c1)NCC2 C1(C(=O)NCC(=O)NC)CCCC12CCN(Cc1cncs1)C2.c1cc[nH]c1.C c1(C(N2C(C)CC(CC(=O)NCCCOC)C2)=O)cn2c(n1)CCC2 N1(C(C(c2ccc(F)cc2Br)C)=O)CCCN(C(=O)N(C)C)CC1 N#Cc1ccc(C(=O)NC23CC2CN(C(c2ncccc2C(F)F)=O)C3)cc1 Cc1cc(CNC(c2nnnn2C(C)C)(C2CCCC2)C)cc(Cl)n1 N1(C(c2c(CC)[nH]cc2)=O)CC2C(CNC(c3cnc(CO)[nH]3)=O)C2C1 N1(C(C(C=C)(C)C)=O)CC(OC)CC(NC(=O)C(C2CC2)C2CC2)C1 CCC(CCCC(=O)NCC1CCCCN(C)C1)NC(=O)C(N=[N+]=[N-])C(C)C C(=O)(C1CCCc2n[nH]cc21)N1CCCC(C)(CNC(=O)CSCCC#N)C1 C(CC(CC)C(=O)N1CCCC1(C(C)C)C)=CC.C12(C=O)CC(C)(CO1)C2 c1(C2N(C(=O)NC(C3CCCCC3)CCC)CCC2)ccc(Cl)nc1 N1(C(C(CN(C)C)O)=O)CCC2(CC(NC(c3ccc(CO)cn3)=O)C2)C1 N1(C(C2CC(C)N2C(c2c[nH]c(C(N)=O)c2)=O)=O)CCOCC2(CC2)C1 Cc1cc(C(N2CCCC(C)(C)C2)=O)c(C)nc1C.O(CP(C)(C)=O)CC(=O)N C(=O)(C(C)C(C)n1cccn1)NCC(C)NC(C1(n2cccn2)CCC1)=O c1(SC)nc(C)cc(=NC2CC(CCNC(c3ccc(C)nn3)=O)C2)[nH]1 C(CN=[N+]=[N-])(C(=O)N1CC(C#N)C1)NC(C1CCC(=C)CC1)=O C12(NC(=O)CC3CCCCO3)CCC(NC(C3C4COCC34)=O)(CC1)C2 CC1(C)CC(n2cccn2)(SCC=Cc2ccncc2)CO1 C(C(O)(CO)CO)NC(C1(NC(C(C)C2CCOC2)=O)CC1)=O c1(N(CCN(CC)CC)CCO)ncnc(N2CCC(C(F)(F)F)(C)C2)c1C c1(CC(C)C)ncc(C(=O)N(C)CCO)s1.C1(C=O)CCC1.CC.N(C)C C1(NC(=O)NC(c2nncn2C)C(C)C)CCN(C(N)=O)C1 C(=O)(C1=CCCSC1)NCC(CC)(CC)NC(C1CC2CCCC2C1)=O C1(NC(c2c(C)ocn2)=O)CCC2(CCN(C(=O)C(F)(F)C3CCCC3)C2)C1 C1(C(=O)NC2CCN(c3ccc(C(=O)OC)cn3)C2)CCc2cncn2C1 N1(C(C(C=C)O)=O)CCCC(NC(=O)C(C)(C)c2cnsc2)C1 c1(OCC#C)cc(CNC(Cc2ccc(O)c(O)c2)C(=O)OC)cc(S)c1 c1(C(N2CCCC3(NC(C4CC(SC)C4)=O)C(C2)C3)=O)c2ccccc2nn1C C#CCCC(O)C(=O)NCCC1(NC(c2coc(C3CCOCC3)n2)=O)CCC1 C(C)(C(=O)NC(CN(C(=O)CN(C(=O)COC)C)C)CC)=C(CC)C c1(C(N2CC(CC=C)(NC(=O)C(C)C(C)(F)F)C2)=O)cc(OC)ccc1F.O c1(C(=O)OCC)ccc(C)c(NC(CC(C)SC)c2nnnn2CCCF)c1 c1(C(N(C)C)=O)ccc2c(c1)CCCC2.C(C(N=[N+]=[N-])C(=O)N1CCC1)OCC C1(CC(N2CC(C=O)C2)=O)CC2CC2C1.CS(=O)(=O)SCC(=O)N.CC CC(C)CCCCCC(=O)NC1COC2(CCN(C(c3cc[nH]c(=N)n3)=O)C2)C1 C1(NC(C2C(C)(CC)C2)=O)CCC2(CC1)CN(C(=O)C1=CCCOCC1)C2 n1(CC)nc(C(=O)NCC2CCC2NC(c2ccnnc2O)=O)c(Br)n1 c1(C(C)=O)ccc(Br)cn1.c1(C(C=O)N(C)C(=O)OC(C)(C)C)ccccc1Cl c1(CC)cc(C)c(C=O)o1.C1(C)CCCN1C(c1csc(C(F)(F)F)c1)=O.N C1(C(=O)NC2(CCO)CN(C(CCSCCC)=O)C2)CCN(C)C1=O CCCC(C(O)C(=O)N1CCC2(C=CCO2)C1)NC(=O)COC1CC=CC1 C=C=CC(C)C(=O)NCC(CC1CCCC1)C(=O)NCCSC(F)F S(=O)(=O)(c1cccc([N+](=O)[O-])c1C(=O)O)NCC1CCC(CC)O1 c1(N2CCC(C(=O)NCCn3cc(CCC#N)nn3)C2)ccc(F)c(Cl)c1 Cc1ccc(C)c(NC(N2CCN(C(=O)C=Cc3ccc(C)s3)CC2)=O)c1 N1(C(CCCSC)=O)CC2CCCC(NC(=O)Cc3ccc4c(c3)CCO4)C2C1 c1(C(N(CCNC(C(C)C(=O)N2CCOCC2)=O)C2CC2)=O)ccc(O)nc1Cl c1(C(=O)NC2C=CCC(C(=O)NC(CC)C(C)(C)C)C2)cc(C)nc(C)c1 c1(C2C(C(=O)N)C2)ccccc1Cl.CC1C(=O)N2CC(C2)CCO1.C(C)(C)C c1(N2CC(N(CC=C)C)C2)ncnc2c1ncn2CC(O)C1CC1 N1(C(C2(C(N)=O)CC2)=O)CCCC(O)C1.C1(C(C=O)O)CCS(=O)(=O)CC1.C N1(C(CCN(CC)CC)=O)CC2(CC(C=O)CO2)C1.C12COC(C1)C(O)C2.N N1(C(C2(C)CC(=O)C2)=O)CCC(F)(C(N2CCC2CF)=O)C1 CC#CCC(C(=O)NC(CSCC)CC)NC(=O)C(=O)NCC1CC1 C(=O)(C(CCSC)OC)NCC(CC)NC(C1CCCN1C1CCCCC1)=O Cc1cc(C(=O)N(C2CCC(NC(c3csc(-c4ccco4)n3)=O)C2)C)ns1 C#Cc1ccc(C(=O)NCC2CN(C(=O)C=Cc3cccs3)CC2C)cc1F c1(CCC(=O)NCC2CCN(C(=O)CC3CC4CC4C3)C2)ccc(Cl)cc1 C(CC(O)C(=O)NCC1CC1CC(=O)Nc1cnn(CCO)c1)N(C)C CC(C)(CNC(=O)Cc1cncnc1)CNC(=O)C(O)c1ccco1 C(=O)C1=NNC(C(F)(F)F)C1.C(CCC(=O)N1CC2CC1C2)SC.C(N)(=O)N c1(C(N2CCN(C(CC)=O)C(CC#N)C2)=O)cc(F)c(F)cc1C(F)(F)F.CS N1(c2nnc(COC)n2CC(C)(C)COC)CCc2ccc(Cl)cc2C1C C1(CNC(CCSCCC)=O)COCC1NC(c1ccsn1)=O C1(NC(CCCOCC=C)=O)C(C)CCN(C(c2ccccc2CC)=O)C1C CC1OC(C)C(C(=O)NCC2CCN(C(=O)COc3ccccc3F)CC2)C1C N1(C(Cc2cc(C)no2)=O)CC(CNC(C2(C(F)(F)F)CC2)=O)C(C)C1 c1(CC(C(=O)NC2C(NC(c3cnc(CC)s3)=O)CC2)C)c(C)noc1C c1(NC(c2n(CC#C)ccc2)=O)c(C#N)c2c(n1-c1ccccc1)CCCC2 Cc1c(S(=O)(=O)N2CC3(C)CC2(C(=O)OC(C)(C)C)C3)cnn1C(F)F C12(C(=O)NC3CCN(C(CCc4onc(C)n4)=O)C3)CCCC(CCC1)C2 C1(NC(c2cn(C)nn2)=O)CN(C(C2CS(=O)C2)=O)CC2(CCC2)C1 C1(C(=O)NC(C)CNC(=O)CC2(C)CC2)CC2(CCO1)CC2 CC(C)(O)C(C)(C)CNC(=NCc1ccc(C(F)(F)F)cn1)NC1CCC1 O=C1COCC2(CCCN(C(c3ccc(C(F)F)cc3)C(=O)NCCCF)C2)N1 C12(OC)CCCC1(C(=O)N(C)CC1CCCN1C(=O)CCn1cncn1)CCO2 C(=O)(C(CC(C)C)n1ccnc1)NC1CCC(NC(COCC#C)=O)CC1 c1(NCc2c(OC)cccc2)ccc(Br)cc1C(N)=O C(c1ccccc1)=C(C)C(N1CCC(F)(C(N2CC(c3ncc[nH]3)C2)=O)C1)=O O=C1NCC2(CCOCC2)C1NC1(C(=O)O)CC(Cc2ccccc2)C1 C1(OC)CCCCC1C(=O)NCCCN1CCN(C(C2CCCCC2)=O)CC1 CCCCCC(C)CC(=O)N1CCCC(CN(c2ncc3ncn(C)c3n2)C)C1 CC(C)CC(C)C(=O)N1CCC(C(C)(C)NC(c2cc(C(F)F)cs2)=O)CC1 c1(C(=O)NCC2C=CC(NC(C(C(C=C)C)C)=O)C2)ccc2nnc(O)n2c1 C1(CNC(CSCC=C)=O)CCCCC1NC(C1CCCCN1CC)=O c1(C(=O)NC(CN(C(C(CC)N(C)C)=O)C)CC)ccnc(S(N)(=O)=O)c1 C1(NC(C(=O)Nc2cccc(C)c2)=O)CCN(C(c2ccc(CO)s2)=O)CC1C C1(NC(c2cccc(=O)o2)=O)CN(C(=O)Cn2cc(C3CCC3)nn2)CC1.C CCC(C)CCC(=O)NC1CCC(NC(=O)CC2CCOCC2(C)C)CC1 C1(CNC(C23CCCC(C2)NC3)=O)CCC2(CCCCCCC2)O1 O=C(C(Cl)=CCl)NC1CCN(C(c2csnn2)=O)C1 N1(C(C(C)(C)N(C)C)=O)CCCC(O)(CCNC(=O)CC2CSC2)C1 c1(C(N2C(CN(C(C(C)OCC(C)C)=O)C)CCC2)=O)cc(Br)cn1C Cc1ccc2c(c1)CC(C(=O)NC(c1nc(Cc3ccccc3)no1)C)S2 C1(C(=O)NCC2CCN(C(c3n[nH]c(C)c3Br)=O)C2)CN=C2N=CNN2C1 C(CCC(C)C)(C(=O)NCCOc1ccccc1)NCC(C1CCCCC1)OC C1(CC)CC(C(=O)NC(C2CCN(C(C3CCCN3C)=O)C2)C)CCC1=O Cc1cc(C(=O)NCC2CC2)cnc1C1CC1.C(=O)CC.CC(F)(F)F.C c1(CC(=O)NC2CCC(NC(C3OCC(C)(C)C3)=O)CC2)ccc2c(c1)CCC2 c1(C(N(CC(C)O)CCNC(=O)CC(=O)N(C)C)=O)cccc2cnsc12 N1(C(C(C)C2CCCO2)=O)CCC(C)(NC(=O)C(c2ccccc2)=O)CC1 C(=O)(CC(C)(C)C(C)=O)N(C(CC)C(=O)NC1CN(C)CCC1O)C C1(N(C(=O)CSCc2cccs2)CCO)CCN(C(=O)Cn2cccn2)C1 C1(C(N(CCN2CCCC2)CC)=O)CN(C(C2OCCCC2(C)C)=O)CC1(C)C C(=O)(CCCCC(F)(F)F)N1CCC(C(C)(C)C)(CNC(C#CC(C)(C)C)=O)C1 N1(C(CCNC(c2n(CC#C)ccc2)=O)=O)CC(O)C(O)C12CCC2 CCC(CC(F)(F)F)C(=O)NC1CCCC1CNC(C1(C)CCC(=O)N1)=O C(C(C)(C(=O)NC1CCC(=O)NC1)NC(=O)CC1(O)CCCC1)SC C(CC(C(=O)N)OC)OC.C(C)(C)CN(C)C(C1(C(=O)N(C)C)CC1)=O N1(C(C2(C3N(C(c4nc(Cl)cs4)=O)CCC3)CC2)=O)CCn2c(O)nnc2C1 N1(C(CC=CC)=O)CCC2CN(C(=O)C(C)(C)c3cscn3)CCC2C1 Cc1cccc(C2CC2)c1CNC(=O)CCC1CCCCN1 C1(C)CCCN(C(=O)Cn2ccc(C3CC3)n2)C1.c1(OC)cc(C(=O)N)ccn1 C(=O)C(C(C)(C)C)n1ccnn1.C(=O)(CC(=O)N(C1CCCC1)CC)N.CC c1(C(=O)NC2CCCC2NC(c2ccccn2)=O)cccc(-n2cccc2)c1 Cc1nn(CC(=O)NCCCC(C)(C)NC(C2CCCC2(C)C)=O)c(C)c1C N1(CC)CCN(C(CCc2ccc(Cl)cc2F)C(=O)NC(C)C)CC1C CC(CC(=O)NCCCC1CCCN1C(c1nnc(O)nc1O)=O)C(C)(C)C Cc1nc(C)n(CC(=O)NC)n1.C1(C)CCCC1.c1(C=O)cc(C(N)=O)c[nH]1 C(=O)(C(C(C)(C)C)C1CCCCC1)NCC1N(C(CCC#CC)=O)CC1 C1(C(=O)NCC2CN(C(c3cnc(CC)s3)=O)CC2C)CCCC(F)(F)CC1 N1(C(c2n(C(C)C)nnc2)=O)CCOC2(CCN(C(=O)CC3(C)CCCO3)C2)C1 c1(CN2CC(CC(=O)Nc3c(C(N)=O)nccc3)C2)sc(Br)c2c1OCCO2 C1(CC=O)CCC(=O)NC1=O.N1(CC(N2CC(O)(CC)C2)=O)CCN(C)CC1 c1(C(=O)NC(c2ccc(F)cc2)(C(=O)OCC)C)ccnnc1O c1(OC)ccc(C(=O)NC2(C)CCCN(C(C3(F)CCCCCC3)=O)C2)c(F)c1 c1(C(=O)NC2C(CNC(CC(=O)OCC)=O)C2)ccc(OC)c(O)c1 N1(C(CC)=O)CCC(C)(C(=O)NC2(c3nnc(OC)s3)CCOC2)C1 C1(NC(C(C2CC2)OC)=O)CN(C(=O)CC2(CSC)CC2)C2CCCCC12 C(=O)(CC(=O)N=c1cc(C)o[nH]1)N1C(COC)CN2CCCC2C1 C1(N(C(c2c(C)cns2)=O)C)C2CN(C(=O)COCC3CCC3)CC12 c1(C(=O)NCC23CN(C(CC=C(C)C)=O)C(C2)CO3)csc2c1CCC(C)C2 CCC(CCOC)C(=O)NCC(C(F)(F)F)N1CCN(C(=O)C2=CCOC2)CC1 CC1(C)CN(c2nnc(O)s2)CCC1NC(c1cn(C(F)(F)CO)nn1)=O C(=O)(C1=CCCC1)N.c1(CC(=O)OC)ccno1.C(=O)CC=O.C(C)(C)C N1(C(C(C)OCC)=O)CCN(C(=O)CSC(F)(F)F)CC2(CC2)C1 c1(C(=O)NC)cn(CC(=O)NC(C)(C)C(C)NC(=O)C(O)CSC)nn1 c1(C(=O)NC(C(C(=O)NCCc2ccnc(C)n2)C)C)cc(C)c(F)cn1 C12(C(=O)NCC(CNC(c3ccccc3)=O)F)COCC(C1)C2.C1CC1.O N1(C(c2ccc(OCCOC)cc2)C(=O)NC(C)C)CCC2CCCCC2CC1 N1(C(C2CCCC(C)CC2)=O)CC2CCC1C(NC(c1csnn1)=O)C2 CC1(C#CC(=O)NOCC(=O)NC2CC3CCCC(C2)C3)CCCO1 c1(C(=O)NC(C(C)NC(C(C)NC(CC)=O)=O)C)ccc2n[nH]cc2n1 C1(CNC(c2c(C)n[nH]c2)=O)CN(C(=O)C(C(C)C)c2ccn(C)n2)CC1(C)C c1(OC(C)C)ccc(NC(c2ncccc2)=O)c(Cl)c1.c1(C=O)cnc(Br)o1.N Cc1cc(=NC(=O)C(=O)N2C(C)CC3CCCC23)[nH]n1-c1ccc(Cl)cc1 N1(c2ccnc(NC3C(C)COC3)n2)CCCN(C(c2ccccn2)=O)CC1 C1(NC(CSCCOC)=O)CCN(C(C2CC2C2CCCC2)=O)CC1O CC1CN(C(c2cc(Cl)ccc2C(F)F)=O)CCN1C(=O)Cn1nnc(=N)[nH]1 c1(C(N2CCC(CNC(c3ccc(OC)s3)=O)CC2)=O)ccc2c[nH]nc2n1 c1(CNC(=NCCC(C)C)NC(C2CCOC2)C)ccc2c(c1)CCS2(=O)=O N1(CCCc2nc(CC(C)C)nn2-c2ccc(Br)nc2)CC(C)OC(C)C1 c1(C(=O)NCCC2(NC(c3cnsc3)=O)CC2)nc2c(s1)COCC2 C1(CNC(c2c(C)c[nH]n2)=O)CCCN(C(=O)CCc2ccc(Cl)nc2)C1 c1(C(C)C)cc(CC(=O)NCC(C)(C2CC2)NC(=O)CCC2CCCO2)on1 c1(C(N2CC(C(C)C)N(C(=O)C3=C(Cl)CC3)CC2)=O)ccc(N)cc1S(N)(=O)=O n1(-c2scc(CC(=O)OCc3c(C)con3)n2)c(C)ccc1C C(=O)(C(Cc1ccccc1)C(F)(F)F)N1CCCC(n2c(C(=O)OC)ncn2)C1 C1(N(C(c2ccc(OCC)nc2)=O)C)CCCN(C(=O)CCNC=O)CC1.N CCC(C)(C)CC(=O)N(C1CN(C(=O)C(c2cc(F)cc(F)c2)C)C1)C C1(NC(c2cnc(CCC)s2)=O)C2CC1CN(C(c1ccc(C)cc1OC)=O)C2 c1c(F)ccc(F)c1F.C1(c2onc(COC)n2)(C(=O)NC)CCOCC1 C1(NC(c2ccc(C(C)=O)o2)=O)CCCCC1C(N1CCC(F)(CO)C1)=O C1(NC(C2C=CCN2C(c2cc(Cl)no2)=O)=O)CC2C(C1)C2(F)F C1(CC=C)(NC(=O)C(n2nc(C)cc2C)C)CCN(C(C2(CC)CCCO2)=O)C1 c1(C(N2CCCCC(NC(CN(C)CC)=O)C2)=O)coc2c(Br)cccc12 C=CCC(CC)C(=O)N1CC(CC(=O)N(C)Cc2cn(C)cn2)CC1(C)C N1(C(C2CCCCN(C(CCCCCSC)=O)C2)=O)CCc2ccc(F)cc21 C1(C=O)CCC2(CCC2)O1.c1(CC=O)ccnn1C1CCC1.C(C)(C)OC.N c1(CNC(N2CC(CC(=O)OC)OC(C)C2)=O)cccc2nc(O)oc12 C1(C(=O)NC(C(C)C)C)CN(C(c2n[nH]c(=N)[nH]2)=O)CC(C)(C)C1 C1(C(=O)NCC(C)CNC(c2ncncc2N)=O)CCCC(=O)N1C C1(NC(=O)CC2CC2)CCCN(C(=O)CNC(c2ccccc2)=O)C1 C1(CN(C(CC=C(C)C)=O)C)COCCN1C(c1cc(C(F)F)ncn1)=O C(c1ccccc1)=CC(=O)NC(C(C)NC(C1C(OCC)C1)=O)CO CCC(CC(=O)N(C)CC1CCCC1O)NC(C1(Cl)CCCCC1)=O C1(CC(=O)NC(C2CCCO2)CC)CCCC1NC(c1cnsc1C)=O C1(NC(=O)CCCC2CC2)CCN(c2cc(Cl)nc(C3CCC3)n2)CC1F c1(C(=O)NC2CCC(C(=O)NC(C)(C)C)C2)cc(Cl)c(Cl)c(Cl)c1 CC1(C#CC(=O)N2CCC(O)(CNC(C34CCC(C3)C4)=O)C2)CCCO1 C1(NC(C(C)(C)CCl)=O)CN(Cc2ccnc(Br)c2F)CC(F)(F)C1 C(=O)(C(C)(C)C(=O)N1CCC(NC(c2ccnnc2C)=O)CC1)NC CC1(NC(=O)CC2CC(F)C2)CCCN(C(c2sccc2-n2ccnn2)=O)C1 c1(C(N2CC(O)(CN(C(C3(COC)CC3)=O)C)C2)=O)cccc2nn[nH]c12 c1(C(N(C)CC2N(C(c3cc(C)ns3)=O)CCC2)=O)cc(C2CC2)nn1C c1(C(COC)(C2CCC2)NCC(CO)OC)nnnn1-c1ccccc1 n1(CC(C)C)cc(C(=O)NCCCNCC)nn1.C1CCOCC1.C(=O)C.O C1(C2CC2)(NC(C2(OC)CCCC2)=O)CCN(C(C2CC2C)=O)C1 c1(NCCC2(OC)CN(C(c3cc([N+](=O)[O-])c[nH]3)=O)C2)ncnc2scnc12 c1(C(C(=O)NC(C)C(=O)OC)N(CCC)C2CC2)cc2cc(Br)ccc2o1 N1(C(CCOC)=O)CCC(O)(CNC(=O)C(F)(F)c2ccnn2C)CC1 c1(NC(C(C)NC(COc2cc(C)on2)=O)C(C)C)cc(C)c([N+](=O)[O-])cc1Br C1(NC(c2cc(CNC(C3(C)C(C)(C)C3)=O)sc2)=O)CCC2(CCCC2)C1 C=CC(CC)CC(=O)NCC(C)CN(C(=O)CCCc1cccnc1)C c1(C(N(C2CCN(C(=O)CS)C2)CC)=O)cccc2nonc12.c1cscn1.C c1(C(=O)N(C2CC3(CNC3)C2)CCC2CCO2)cccc2c1oc1ccccc21 c1(-c2n(CCCCC)nc(-c3ccnn3C)n2)ccc2ccncc2n1 O=C1Cc2cnc(NC34CC(N5CCCCC5CO)(C3)C4)nc2N1.CC(F)(F)F CC1CCN2N=C(C(=O)NCC3CCC(NC(C4(Cl)CC4)=O)CC3)NC2=N1 c1(C(N2CCCC(N3CCCCC3)C2)=O)cnc(F)c(Cl)c1 C1(NC(C(C)O)=O)C2CC1N(C(=O)CCN(c1ccccc1)C)C2C c1(C(=O)NC2C(NC(CN3CCP(C)(=O)CC3)=O)C2)c[nH]c2cccc(C#N)c12 C1(C#N)(NC(c2c(C)nn[nH]2)=O)CCN(C(=O)NCCCl)C1 c1(C(=O)NCC2CN(C(C3CCCN(CC)C3)=O)C2)cc(F)c(C)c(F)c1 CC(C)CC(=O)C(=O)NC1(C)CN(C(=O)CN(C2CCSC2)C)C1 C1(N(C(c2c(C)noc2)=O)C)CN(C(C23CC(CC(F)F)(C2)C3)=O)CCC1C Cc1ccc(C(=O)OCc2ncc(-c3ccc(F)cc3F)o2)cc1CN C1(c2n(-c3ccc(OC)cc3)nnn2)(NCCC(F)F)CCCC2CC12 c1(OC)ccc(Br)cc1C(N1CCC(NC(=O)CC(F)F)C(F)C1)=O c1(C(=O)NC2(CNC(C(CCSC)O)=O)CCCCC2C)cc2ccncc2s1 CC1=C(C(=O)NCCC2CN(C(=O)C3=COCCO3)CCO2)SCCO1 CC(Cc1cnc[nH]1)C(=O)NCC1CC(NC(c2coc(Cl)c2)=O)C1 C12(C(N3CCC(COC)(NC(C4CC45CC5)=O)C3)=O)CC3CC1C2C3O CC1=C(C(=O)N(CCCN(C)C(C2CC3COCC(C2)C3)=O)C)SCCO1 C1(C(=O)NC2(c3ccc(OC)cc3)CC2)(OC)CCC(F)(F)CC1 c1(C(=O)NCCn2cc(CC(C)O)nn2)nnn(C2CC2)c1C(F)F C(N=c1[nH]cc(-c2ccc3ncc(C(=O)OC)n3c2)cc1C)C1(COC)CC1 C1CCC(C(N2CC(O)(C(C)(C)C)C2)=O)C1.c1(C=O)ccn(C2CC2)n1.C Cc1ccc(C(N2CCOCC(NC(c3nsnc3O)=O)C2)=O)c(Cl)c1C N1(C(CCCC(C)NC(C)=O)=O)CC2CC=CCC2C1 c1(CC)nc(C)c(C(N2CCC(C(=O)Nc3cnn(C)c3C)(OC)C2)=O)o1 c1(CC)ccc(Br)cc1C(=O)NC1CCN(C(=O)CC(F)F)CC1CO CC(C)CC(CO)NC(=O)CC1CCCN(C(=O)CC2C(C)(C)C2(C)C)C1 N1(C(c2cn(CCCC)nn2)=O)CCC(CC)(NC(=O)CN2CCCC2C)CC1 c1(C(N2CCC(=CCNC(C(CC)(C)COC)=O)CC2)=O)ccncc1N=[N+]=[N-] c1(C(N2C(CNC(c3ccc(CN(C)C)o3)=O)C=CC2)=O)ccc(O)cc1F c1(CC)cccc(C(=O)NC2CCC2)c1.c1(C2(C=O)CC2)ccc(C)nc1.C C(CC(C)C(=O)NCC(C)(C)CN(C(c1c[nH]nc1OC)=O)CC)=CC C(CC(F)(F)C(C)C)NC(C1(CC=C)CN(C(=O)C(c2cccn2C)=O)C1)=O N1(C(C2=CC(C)(C)C2)=O)CCC2(C1)CN(C(c1ccnc(C(F)F)c1)=O)CCO2 C=CCCCC(=O)N1CCCC(CCC(=O)NOC)C1 c1(C(=O)NC23C(CCN(C(CSCC=C)=O)CC2)C3)cccc2ccn(C)c12 c1(CC(=O)OC2CCC(OCC)CC2)ccc(I)c(OC)c1 c1(CCN(C(C2CC3CCC2O3)C(=O)NC2CCCCC2)C)ccc(Cl)c(Cl)c1 N#CCCCCCC(=O)Nc1cccc(CS(N)(=O)=O)c1 C1(C(=O)Nc2cn(C)nc2Cl)C(C2CC2)CCN1C(c1n[nH]c2ccccc12)=O C1(NC(c2c[nH]cc2Br)=O)CCC(CNC(C2CCCC2C(F)F)=O)CC1 [N-]=[N+]=NC1CCC(C(=O)NCc2cc(C(=O)N)cs2)C1.c1cccc(F)c1O.C CC(C)CC(CNC(=O)C=C1CCC(C)C1)NC(c1cnn(C)c1Br)=O c1(C(=O)NCCCOC2CCN(C(=O)C3=CCCC3)CC2)snc2ccccc12 N1(C(C2CC(CCC)OCC2)=O)CC2(CCN(C(C3CCC(C)(CC)O3)=O)C2)C1 C(=O)(CC(F)(F)C(F)F)N(CC(CNC(c1c(C)scc1)=O)C)C C1(CN(C)C(C2(C)CCC2)=O)C2CN(C(C3C=CCS3)=O)CC12 C(CO)(CC(F)(F)F)NC(CC(CC)NC(CCCC)=O)=O C1(NC(C(CC)F)=O)CC2(C1)CC(NC(c1cccc(C(F)(F)F)c1C)=O)C2 c1(N(C)Cc2c(C)cccc2C)nc(=NCc2ccc(Br)cn2)[nH]c2ccsc12 CC(C)C(C(=O)N1CCC(CNC(C2CCC(c3ccccc3)O2)=O)C1)NC=O C1(CNC(C=C(C)C2CC2)=O)C(C)CCCN1C(=O)CCS(C)=O c1(C(=O)NC2C(CC)N(C(=O)C(OC)OC)CC2)cc2c(C)c(F)ccc2[nH]1 Cc1cc(C(F)(F)F)c(C#N)c(N(C(C)C)C)n1.C(C1CCOCC1)=CC=O.N C1(C(=O)OCc2ncc(C)cc2C(F)(F)F)CC2C#CCC(C1)C2 C(=O)(CC(C)(C)C(F)F)NC(C1CN(C(C2CC2CC(C)(C)C)=O)C1)C N1(C(CC2(OCC)CCC2)=O)CCC(C)C1C.C(C1CCCC1)=CC=O.N C1(C(N2CCC3CN(C(CSCCC#N)=O)CC32)=O)C2C3CC4C1C1C2CC3C41 C(CCCCC(=O)NC1CN(C(=O)C(C)C(C)(C)C)CC1OC)=CC Clc1ccnc(Cl)c1CCNCc1cccc(Oc2ccccn2)c1 C(=O)C1CCc2nccn21.c1(CC(=O)NCCC)cc(C(F)(F)F)cc(Cl)n1.N N1(Cc2c(-c3n(C)ncc3)n[nH]c2)CC2(CCCC2NC(=O)C(F)(F)F)C1 C12(NC(c3c(C)cc(C)s3)=O)CCC(C1)N(C(=O)CC1(O)CCCN(C)C1)C2 C1(C(=O)NCC(C)NC(C(Br)=C(C)C)=O)CCOC1C c1(CC(=O)NCC(C)CN(C)C(C2CCC2)=O)c[nH]nc1O.c1(C)cnn[nH]1 C1(CC=C)(NC(c2ccc(Cn3ccnn3)cc2)=O)CCCN(C(=O)C(C)O)C1 C(=O)(C(C1CN(C(c2cscn2)=O)C1)OC)NC(c1ccsc1)CC C(=O)(C(C)S(N)(=O)=O)N1C(CNC(c2cnc(C(C)C)o2)=O)CC2CC21 c1(C(=O)NCC2CC(NC(C(COC)O)=O)C2)ccnc(C(F)(F)F)c1F Cc1sc(O)nc1C(=O)NC(C)(C)CNC(C1CCC2CCC12)=O c1(OC)ncnc(OC)c1C(=O)NCC(C)N(C)C(C12COCC1C2)=O C1(OCC)CC2(C1)CC2C(N1CC(NC(c2ncc(Cl)s2)=O)CC1C)=O C(C)(C(=O)N1CCC1C)OCCOCC.C1(CC(=O)N)CC(=O)C1 c1(C(=O)NC(CC)CNC(=O)C(=Cc2ccccc2)OC)ncc(F)cc1F C(=O)(CS(=O)C(F)(F)F)NCCCC1N(C(CN(C)C2CC2)=O)CCCC1 C(CC(C)(C)C)(C(=O)NCC1(CC=O)CC1)OC.C1CCCC1C(C)C.N c1(Sc2cc(NC(=O)OC(C)(C)C)c(O)cc2)cc(N)ccc1S(C)(=O)=O C1(NC(C=CC)=O)CCN(C(c2cn(C(C)C)nc2Br)=O)CC1CO C1(COC)(C)CCCN1C(=O)C.C(=O)C(F)(F)CC1CCCO1.C(C)C C=CCC(CC(C)C)C(=O)Nc1ccc(NC(=O)CC2CC3CC3C2)c(C)c1 c1(C(N(C(C)CNC(=O)OC(C)(C)C)C)=O)c(F)cc(Br)cc1F c1(C(=O)NC2CN(C(C34CCC(OC)C3CC4)=O)CC2C)cncc2ccsc12 c1(CNC(C2CCN(C(C(C3CCCC3)OC)=O)C2)=O)ccncc1C N1(C(c2nc(C(C)C)sc2)=O)CCC2(C1)CN(C(C1(C#N)CC=CC1)=O)CCO2 n1(C(CC)C(=O)N2CC(C)(NC(c3ccc(F)s3)=O)C2)cnc(C#N)n1 C(=O)(C(C(C)(C)C)C1CCCC1)N1CCC(N(C(=O)C(O)C2CCC2)CC)CC1 n1(CCC(=O)NCC2C(C)CN(C(=O)CCC3CC3)C2)nc(O)c2ccccc12 C1(O)(CN(C(Cc2cc(C)ns2)=O)C)CCN(C(C23CCCC2C3)=O)C1 C1(CNC(C(C#C)(C)C)=O)COC(C(F)(F)F)CN1C(=O)C=CSC CC(c1cccc(Cl)c1)=CC(N1CC=C(CNC(=O)C(F)C(C)C)CC1)=O C(=O)(CC(C)C(F)F)NC(C1CCN(C(c2ccoc2Cl)=O)CC1)C(C)C N1(C(c2ccc(CCCCCC)s2)=O)CCN(C(=O)C=CCOC)C(C2CC2)C1 C1(C(=O)NCC2(C(=O)NCC=C=C)CC2)(CC)CCC1 C1(C)(C(=O)OC)CCCN1C(=O)CC(C)C1CCC1.c1(CC(=O)N)cc[nH]c1 C(=O)(C(C)C(=O)N1CCOCC1)N(CCN(C(C)C)C(=O)C1CC1)C c1(C(C)C)cccc(OC(C)C(N2CCC(NC(=O)C=CCO)C2C)=O)c1 n1(C2CCN(C(=O)NC3C(C(C)C)CCC3)C2)c(CO)nc2ccccc12 C(=O)(C#CC1CCC1)N1C(C(=O)N(C2CC2C2CC2)C)CC(OC)C1 C(=O)(CCC(=O)N)N(CC)CC.C1(CC)CCN(C(=O)CCc2cc[nH]n2)CC1 N1(C(c2n(C(C)C)ncc2)=O)CCC2CCCC12CNC(c1ccc(F)o1)=O C(=O)(CC1OCCc2ccsc21)NCC(C)N(C(=O)C1=CCCC(C)(C)C1)CC c1(C(N2C(C3CCCN(C(CCC(=O)NC)=O)C3)CCC2)=O)ccc(N)c(F)c1 N1(C(c2c(CC)scc2)=O)CCCC(CCNC(c2c[nH]nc2C(F)F)=O)CC1 C1(CNC(c2c(C)n[nH]c2)=O)CN(C(=O)CN(C2CCC2)C)CC1C C=CC1CN(C(c2nnn(C)c2C2CC2)=O)CC1NC(=O)C(C)C(F)(F)F C1(N(C(C(CCOC)C)=O)C)CN(C(=O)C(F)(F)c2nc(C)cs2)CC1(C)C N1(CC(C(C(=O)OCC)(F)C(=O)OC)C)CCCC(C2CCNCC2)CCC1 C1(C(N2CCC(CNC(CSC(C)(C)C)=O)(C)CC2)=O)CC2CCC1NC2=O CC1CCC(NC(=O)C)CN1C(c1ccc(F)c(Cl)n1)=O.c1(C=O)cscn1.N CC(=O)CC(C)(C)CC(=O)NCC(C1CC1)N(C(=O)C)C.c1ccccc1C.O c1(N2C(C)CC(NC(c3cnc4sccn34)=O)CC2)ncc2cccnc2n1 C#CC1(NC(=O)NCC2(N3CCSCC3)CCCCC2)CCCOC1 N1(C(CCC(C)C)=O)CC2(CCC2)CC1CNC(=O)C(C)(O)C(C)C C1(C(N2CC(N(C(c3ccoc3C)=O)C)C2)=O)Cc2c(C)cccc2O1.COC C(CS(=O)(=O)CC(=O)NCC1(CO)CCN(C(=O)C2=CCC(C)CC2)C1)OC N1(C(c2cc(OCC)ns2)=O)CC(NC(c2cc(C)[nH]n2)=O)CC2(CC2)C1 n1(CCNC(COCC)=O)cc(C(=O)NC2(C(N)=O)CC2)cn1 Cc1ccc(C(=O)NC(C)CCNC(C2CCC2)=O)c(N)c1C.c1cnn[nH]1.C CCCCCCC(=O)Nc1ccc(NC(C2CC(F)(F)CS2)=O)cc1C C1(N(CC#C)C(c2n[nH]cc2C)=O)CCN(C(=O)C(C)CCC)CC1 c1(C(=O)NC(C)(CNC(C2CC2F)=O)C2CCC2)ncc(C2CC2)cc1F C(=O)(C(C)C(F)(F)F)N1CCC(C)C1.Cc1ccc(-c2oncc2C(=O)N)o1.C N1(C(=O)C(F)n2ccnc2)CCOCC(C(=O)NOC2CCCC2)C1 N1(C(CN(CC)CC)=O)CCCCC(NC(c2ccc(O)c(Cl)c2)=O)C1 c1(OC(C)C)ccccc1.C1(C)(C(c2nnnn2C2(C)CC2)N)COC(=O)N1 n1(CC)nc(C(=O)NC2CC3CC2CN3C(=O)Cc2cc(C)[nH]n2)ccc1=O C(=O)(C#CC1CCOCC1)NC(=N)N.CC1CC(N2C(=O)NCC2=O)CCC1O CCCC(CC)C(=O)NCCCCN(CCCNC(=O)C(C)(O)COC)C C12(OC)CCC(c3cn(C4CN(C(=O)CN5C(=O)CCCC5=O)C4)nn3)(CC1)C2 C(=O)(C1CCCc2ccccc21)NCC(C)NC(C1Cc2c(C)[nH]nc2CC1)=O C=CC1(CC(=O)NCC(n2ccnn2)C)CN(C(=O)C(O)c2ccco2)C1 c1(C(=O)NC2C(C)CN(C(=O)C(O)CC3CC3)C2)ccc(Cl)c(N)c1 CC1(C)CC(CNC(=O)CN2CCCCCC2)CN1C(c1ccccn1)=O CC1Cc2ccccc2N(C(=O)COC(=O)CC2CCCCC2C)C1 c1(CC)cc(C(F)(F)F)ccc1C(=O)NCC(F)CNC(C1CCCO1)=O Cn1cnc2c1CCN(C(c1ccc3c(c1)CNC(=O)N3)=O)C21CCNC1 C1(NC(COCCNC(c2n(C(C)C)ccc2)=O)=O)CCCCCC1F Cc1cc(F)c(CC(=O)N(C)CCNC(C2CCC3CC2CO3)=O)cc1F C(=O)(C(C)(C)C(F)(F)F)NC1CC2CC(NC(Cc3cncc(C)c3)=O)C2C1 c1(CSC)cccc(C(=O)NC(C)CC)c1.c1(C(=O)N)cc(C(C)C)on1 c1(C(=O)NC2(CCNC(c3ccc(C)cc3)=O)CC2)cc(C#N)[nH]c1C C1(C(=O)NC2CCC(F)(C)C2)(CC)CCNC1=O.c1(C=O)nnn(C)c1C.N C(=O)(C1COc2ccc(F)cc21)N1CC2(CN(C(c3c(OC)scc3)=O)C2)C1 c1(OCC)c(CN2CCC(CNC(c3cc(C)c[nH]3)=O)C2)cc(C)cc1Br N1(C(Cn2c(C)ccn2)=O)CC2C(N(C(=O)CCOCCN(C)C)C)C2C1 c1(CC(N2CCN(C(=O)CSc3nc[nH]n3)C3CCC23)=O)ccc2c(c1)CCC2 C(=O)(CC1=Cc2ccccc2C1)N1CC(CNC(C=COCC)=O)C(F)(F)CC1 C12CC1CN(C)C2.C1(CCC=C)(C=O)CN(C(C)=O)C1.C1CCC(C=O)C1.N CCCCC(O)C(=O)NC(C)CCCNC(=O)C(C1CCC(C)CC1)CC CCC(O)C(C)(C)C(=O)NCC1(F)CC(CNC(=O)CCC(C)(C)C)C1 N1(C(C2C(CCC)CN(C(=O)C(O)C(C)C)C2)=O)CC(OC)CC(C)C1 c1(SC)ccc(C=CC(=O)NCC(C)C2CCC2)o1.C1(C=O)CCCC1(F)F C1(N(C)C(c2cc(C3CC3)ccc2F)=O)CCCN(C(C2(F)CC2)=O)CC1 N1(C(c2c(CC)con2)=O)C2CCC1(CNC(=O)CC(CC)C1CC1)CC2 C12(NC(c3nccc(Cl)c3F)=O)CCN(C(C3(n4cccn4)CC3)=O)CC1C2 N1(C(C2C(C)=CCS2)=O)CCN(C(=O)C=C(Cl)Cl)C(c2ncc[nH]2)C1 c1(C(=O)NC(CCSCC)C)ccc(CNC(C2C=CCS2)=O)s1 N1(C(CN(C)C(c2ccc(CO)cc2)=O)=O)CCOC(C2(C)N=N2)C1 N1(CC)CCC2(CCCN(C(=O)C(O)Cc3ccc(C)cc3Cl)C2)C1 CCCC(C)(CC)C(=O)N1CC(n2cc(CN3CCSCC3)nn2)C(SC)C1 N1(c2ncc(C#C)cn2)CCC(C2(NC(=O)C(N3CCCC(C)C3)=O)CC2)C1 Cc1ccc(=O)n(CC(=O)NCC(C)N(C)C(C2CC2Br)=O)c1 C1(NC(=O)NCCc2ccc(OC)c(OC(F)F)c2)CC12CCC1(CC1)CC2 C(=O)(C1CC(=O)c2ccccc21)N.N1(C(C2(CC)CC2)=O)CCC(O)(CC)CC1 C(=O)(C(F)(F)C(O)CC)N1CC(CC(C)NC(CCCCCC)=O)C1 c1(CC)cc(C(N2CCCC2C2(NC(c3cc(Cl)n(C)n3)=O)CC2)=O)ncn1 c1(OC)ccc(O)cc1NC(C1CCN(c2ncc(C3CC3)cn2)CC1)=O C(=O)(CCN=[N+]=[N-])NC1(C(NOCC2C(C)(C)C2)=O)CCOCC1 c1(NC(CC)C(N)=O)cc(Nc2nc(C)cs2)ccc1O C1(CCN(C(C2C(COC)C2)=O)C)CCCCN1C(c1ncc(C)s1)=O.O N1(C(CCSCCC)=O)CCC2(CC1)CN(C(c1nnsc1C)=O)C2C(C)C N1(C(c2ccc(OC)c(F)c2F)=O)CCOC2CN(C(=O)C(C)=O)CC12 CC(CCN(C)C)C(=O)N(CC(C)NC(=O)C(F)(F)c1nccn1C)C C(=O)(C(C(C)CC)N(C)C(c1cc(Cl)cn1C)=O)NCC(=O)NCC=C Cc1nc(-c2c[nH]c(C(=O)NCC(C)(O)CNC(c3ccc(Cl)o3)=O)c2)cs1 C1(NC(C(C)N(C(=O)CCc2cnoc2)C)=O)CC2(C1)CC(O)C2 c1(CC)cc(C(=O)NC(C)(CC)CC)c(C)nn1.C1(C=O)CCC(N(C)C)C1 c1ccc(Cl)c(Cl)c1.N#CC1CC(C(=O)NC2CCC(NC(=O)CCO)C2)C1 CP(C)(=O)C(CC(=O)NCC(Cl)C(F)(F)F)C(F)(F)F N1(C(C2(OC)CCC2)=O)CCC(CO)(NC(c2ccc(C(N)=O)s2)=O)CC1 c1(C(C)O)ccc(-c2noc(C3CC4CC4N3CCSc3ccc(F)cc3)n2)nn1 C1CN(C(C2CC(N3CCCC3)C2)=O)CC12CC2.n1(CC)ccnc1C(=O)N.C c1(C(=O)NC2C(C)CN(C(C3CCCCC3C)=O)C2)ccc2c(c1)C(=O)NC2 C1(C(=O)NC(CC)CNC(=O)Cc2cnoc2)CCc2nc(C)nn2C1 c1(C(N2CCCC(NC(c3c(C)noc3C)=O)CC2)=O)cccc2c1CCC2 Cc1cc(C(=O)NC2(CNC(c3c(Cl)n[nH]c3C)=O)CCC2)cc2ccoc12 Nc1ccc(CCNC(N2CCOC(C3CCCCC3)C2)=O)cc1 C1(C(=O)NC(CC)CNC(C2CSC2)=O)CCCN1C(c1ccccc1)=O C=CCC(C(=O)NCc1cc(C(=O)N)co1)C(C)C.C1CN(C(N)=O)C1.C N1(CCC(=O)N(C(CNC(CNC(=O)NC)=O)C)C)CCCC1C.N(C)C C1(OC)C(N=c2nc3c(cnn3C)c(N(CCCSC)C)[nH]2)CC12CCC2 C1(CC)CN(C(c2c(C)nn(C)c2Br)=O)CCN1C(c1csc(O)n1)=O C(=O)(CCC(F)(F)F)NCC(C1(O)CCN(C(c2ccc(N)c(O)c2)=O)C1)C N1(C(CCN(CCCO)C(C2CCC(C)(O)CC2)=O)=O)CC2(COCC(=O)N2)C1 C(C)(C(=O)N)SCCCC.C1(C)CC1C(=O)N(CC(=O)OC)CC c1(C(=O)NC2C(C)CN(C(c3ncsc3C3CC3)=O)CC2)cc2ccncc2s1 N1(C(C2ON=C(CC)C2)=O)CCCC(CO)(NC(C2CCC(=O)C2)=O)C1 N1(C(CC(C)C)=O)CC2CC1CN(C(=O)CC1CCNC(=O)C1)C2.C(=O)OC.N CCCC(CCC)C(=O)NC(CNC(c1sc([N+](=O)[O-])cc1Cl)=O)C1CC1 C1(CC(=O)N(C2CCN(C(=O)Cn3cncn3)C2)CCC)CCCCC12CC2 N1(C(C(C)O)=O)CCN(CC(C)NC(=O)CC2CCCO2)CC1 C1(C)(CNC(C2(C(C)C)COC2)=O)CN(C(c2cscc2Cl)=O)CC1C C=C(C)C(C)(O)C(=O)N1CCN(c2ccc(-c3nn[nH]n3)nc2)CC1 CCCCC(CNC(=O)CC1(C)CCN(C(=O)Cn2cc(C)cn2)C1)CC C(CS(=O)(=O)CC(=O)N)OC.C(=O)(C(C(C)C)C(C)C)N1C(C2CC2)CCCC1 N1(CC(=O)N(C(c2cccc(Cl)c2)C(C)C)C)C(=O)c2ccccc2S1(=O)=O c1(OCCC#C)ccc(OCCNC(C2CC2CC)=O)cc1.c1ccncc1 c1(C(=O)NC2CCC(C)N(C(c3csc(O)n3)=O)C2)cc2ccc(F)cc2o1 c1(OC)c(Cl)cc(Br)cc1S(=O)(=O)NCCCCC(C)C c1(CC)ncc(Br)cc1C(N1CC(NC(c2cnn(C)c2)=O)CCC1C)=O c1(CC(=O)NC(CNC(C2=C(C)CCC2)=O)C2CC2)csc2sc(C)cc12 C(CC(O)CC(=O)N1CCCC(NC(c2coc(C3CCOCC3)n2)=O)C1)SC C(=O)(C1CCCn2cnnc21)N1C(CNC(C2(CSC)CCC2)=O)CC(O)C1 C#Cc1ccc(=NCC2CCN2C(C)(C)C)[nH]c1C c1(OC)cc(Cl)cc2[nH]c(C(=O)N(C)Cc3cc(O)cc(Br)c3)cc12 c1(C(=O)OC)cc(S(=O)(=O)NC2CC23CCC3)on1 c1(C(N2CCC(OCCO)C2)C(=O)NC(C)C)cnn(-c2ccccn2)c1 Cc1cc2cc(NC(=O)N(C)Cc3nccn3C(F)F)ccc2[nH]c1=O Cc1nc(C(=O)N)c2ccnc-2[nH]1.c1(C(N2CC(F)C2)=O)cc(=O)cc(Cl)[nH]1.C C1(C(=O)NC(CC#C)(C)C)CCCCN1C(=O)CC(CC)C1CCC1 N1(C(c2ccc(C3(COCC)CCOCC3)cc2)=O)CC2NC(=O)OC2C1 c1(C(C(=O)OC)=O)cccnc1NCC1CCN(C(C2CNC(=O)N2C)=O)C1 c1(C(C)=O)cn(CC(=O)NCC(c2ccccc2)CNC(=O)C(C)CF)nn1 C(=O)(C(O)(C(F)(F)F)c1ccccc1)NCCCN(C(=O)C(O)c1ccsc1)C C1(CC)CCN(C(c2cnn(C3CCC3)c2)C(=O)NC2CC2)CC1OC c1(N(C2CCCCC2)C)ccc(NC(C2CC(OCCF)C2)=O)cc1 C(CCCC(=O)NCCN(C)C(c1cn(Cc2nn[nH]n2)nn1)=O)N(C)C C(=O)(C(C)(C)C1=CCS(=O)(=O)CC1)NC1CN(C(C(C)CF)=O)CC1O C1(NC(COCCCC(C)C)=O)CC2CC1CN2C(c1ccc(C#N)cc1)=O c1(OC)cnccc1C(=O)NC(C)CC(C)C.c1(C(=O)N)ccc(C(F)F)s1 CCCC(C(=O)NC1(C(=O)NC)CCN(C)C1)NC(C)=O.c1csc(C)n1 Cc1cc(C(=O)NC(C)CN(C(=O)Cn2ccnc2C)C)c(N)c(F)c1 C#CCCCC(C)C(=O)N1CCN(C)CC1C(=O)Nc1ccc(C)nc1OC N1(CC)CCC1C(=O)N(CCNC(=O)C(C)c1cncs1)C(C)C N1(C(C2N(C(CCNC(N)=O)=O)CCC2)=O)CCC2(CCC2)C(O)C1 c1(OC)ccc(OC)c2sc(=NCC3C(C)CCCN3C(c3csnn3)=O)[nH]c12 C=CC1OCCC1C(N1CCCC1CCCNC(=O)CCCN(C)C)=O C12(C(=O)Nc3ccc(CC)cc3)CCC(CC1)N(C(=O)CCc1cccnc1)C2 CON1CCC(N(C(=O)C(C)(C)NC(=O)C(C)ONC=O)C)CC1.C(C)(C)C.O N1(C(c2cnc(SC)s2)=O)CC(CNC(C2CCC(CN)O2)=O)CC12CCC2 CCC(CCC(=O)NC1COCC1N=[N+]=[N-])NC(C1CC1CC(C)C)=O N1(C(c2c(CC)nccn2)=O)CCCC(CCNC(C2CCCCS2)=O)CC1 Cc1ccc(CCCC(=O)N(C(C)CNC(c2coc(O)n2)=O)C)cc1C N1(C(c2c(CC)nn(C)c2)=O)CC(C2CN(C(C3C4CCCCCCC34)=O)C2)C1 N1(C(C(C)OCC#C)=O)CCC2(CCC(NC(=O)C(C)OCC=C)C2)CC1 CC1(C)CCN(C(c2cnc[nH]c2=N)=O)C1C(N1CCC(C)(C(N)=O)C1)=O C1(C(=O)NC(CNC(C(CCO)N(C)C)=O)CO)CCCCNC1=O N1(C(C(C(C)C)=O)=O)CC(C2CC2)(C(=O)NCCC(C)c2cn[nH]c2)C1 c1(CCC(N2CCC(O)(CN(C(CCOCC)=O)C)C2)=O)ccc(O)c(Cl)c1 C(CN=[N+]=[N-])(C(=O)NCCc1ccc(F)nc1)NC(CCC(C)OC)=O Cc1cc(C(=O)NCC(C)CNC(C2CCCN2CCC(C)C)=O)nc(O)c1 C(=O)(CCCC(C)(C)C)NCC(CNC(C=Cc1cn(C)nc1)=O)(C)F c1(CC(=O)NCC2(F)CN(C(C3C(C=C)OCC3)=O)C2)c[nH]c2cnccc12 C12(NC(c3ccc(C(CC)=O)cc3)=O)CCCC(C1)C2.C(=O)(C(C)CC(C)C)N C1(CC#C)(C(=O)N(CC(C)CCC)C)CCN(C(=O)CC2CSC2)C1 C1(CN(C)C(c2csc(C(C)(C)C)n2)=O)CCCN1C(C1COC(=O)O1)=O C12(C(=O)NCC(C)NC(Cc3nnc(C)o3)=O)CCC(CC1)C2 c1(OC)ccc(CC2CCN(c3nnn[nH]3)C2)nc1.C1(CC(N)=O)(C=O)CC1.C N1(C(c2ccn(CC)n2)=O)CCC(O)C(N(C)C(c2cocn2)=O)C1 C(=O)(CC1OCCc2sccc21)N1CCC(NC(Cc2nc(C)sc2)=O)C1 C1(C(=O)NC2(CC=C)CCCN(C(c3ncn(C)n3)=O)C2)CCn2ccnc2C1 c1(C(NOCC(=C)Cl)=O)ccc(N2CCN(C(C3C4CCCC34)=O)CC2)nc1 C1(C(=O)NC2CCC(C)N(C(=O)C=Cc3cscn3)C2)COC2COCC2O1 c1(C=O)ccc(C(F)(F)F)cn1.c1(OC)n[nH]cc1C(=O)N(CC)C1CC1 C1(C(N2CC(CCC#C)C2)=O)CCCN(C(c2cccc(CC#N)c2)=O)C1CC N1(C(c2c(CC)c[nH]c2)=O)CCC(C(N2CCC(OC)C2C)=O)CC1CC N1(C(C(CC#C)O)=O)CCCC(CC(=O)NC2CC(CO)C3CC23)CC1 C12(C(N3CC(C(C)NC(=O)CS)C3)=O)CCC(F)(CC1)C2.c1nnnn1C C1(C(=O)NCC2CC2C(=O)Nc2cc(C3CC3)on2)CCSCC1 N1(C(C2N3CC(C)N(CC3)C2)=O)CC2CCN(C(=O)CCc3ccoc3)CC2C1 CC(C)C(CC(=O)NCC(C)N(C)C1CC1)NC(=O)C(C1CCOCC1)=O CONS(=O)(=O)c1ccc(C(=O)NCC2CC2)cc1.c1(C=O)cnc(C)s1.N N1(C(C(C)(C)C)=O)CC2CCCC(NC(=O)C=Cc3cnc(O)nc3O)C2C1 CCC(CC(=O)NCC1C(C)CCCN1C(C1CCN(C2CC2)CC1)=O)C(C)C N1(C(C2(CCC)CC2)=O)CC2CC(C1)N2C(=O)C(C)(C)C1CCC1 N1(C(C2CC(C)SCC2)=O)CC2CC3CC2C1C3NC(c1ccncn1)=O c1(C(C(=O)NCCCF)N(C(C)C(=O)NC)CC)ccc(SC(F)F)cc1 N1(C(c2cc(C)c(C(=O)O)c(C)c2)=O)CCC2(C1)CN(C)C(=O)CO2 c1(NCCC(CC)NC(=O)OC(C)(C)C)cccc(-c2ccncc2)c1 C(N=c1ccc(Br)c(S(=O)(=O)NCCc2ccsc2)[nH]1)C1N(C)CCOC1 C1(CC(N2CCC(OC)C2C)=O)C2CCCC2N1C(=O)C(F)OC(F)(F)F N1(C(c2c(C)nc(CC)s2)=O)CCC(NC(C2CCC(=O)O2)=O)C(C)(C)C1 c1(C(=O)NC2CN(C(C3=C(C)CCCC3)=O)CC2F)cn2c(n1)C(C)CCC2 c1(OC)cc(C(F)(F)F)[nH]c(=NC(C)C2CCCCN2C(C2CCS2(=O)=O)=O)n1 N1(C(=O)C(F)(F)Cl)CCOC(Cn2cc(-c3cscn3)nn2)C1 Cc1ncc(Cl)cc1C(N1CC(N(C)C(C2CCC(O)C2)=O)C2(CC2)C1)=O Cc1ccc(C(=O)NC2CN(C(C3CC=CCC3)=O)CC2n2cccn2)cc1Cl CC1SCCCC1C(=O)NCC1(N2CCOCC2)CCCC1 CN=c1[nH]c(=NCc2cc(Cl)cn2C)[nH]c(=NC2CCCOC2)[nH]1 C12(NC(=O)COC3CC3)CCC(C(=O)NCC3CCC3(F)F)(CC1)C2 C(C)(CCC(=O)NCCCCNC(c1ccccc1Cn1cncn1)=O)SC C#Cc1cn(C)nc1C=O.c1(C(NCC)=O)cn(C)nc1C(C)C.C1CC1 c1(N(CC(=O)NCCNC(c2cc(C)no2)=O)C)ccnc(Cl)n1 Cc1cc(C(=O)NCC(C(C)C)NC(=O)CCCOC(C)C)c2n[nH]cc2c1 CC#CCCCC(=O)NC(C1CN(C(c2ccc(-c3cc[nH]n3)s2)=O)C1)C C(CN=c1[nH]c2c(c(=NCC(CC)(CC)CCO)[nH]1)CCC2)NS(CC)(=O)=O Cn1ncc(C(=O)NC23CC(C(=O)N)(C2)C3)c1C#N.CC(C)(C)n1cccn1 C1(C(N2CC(C)C(NC(=O)C3=CC(C)(C)C3)C2)=O)Cc2c[nH]cc2S1(=O)=O c1(C(=O)N)cnc2ncc(Cl)cn12.CC(C=O)C(=O)NCC.C(C)(C)(C)NC c1(C(=O)N)cccc(C2CCC23CCC3)c1.C(c1nccs1)=CC(=O)NCCC C1(CC(=O)NC(C(C)NC(C(CC)=CC)=O)CO)CCCS(=O)(=O)C1 c1(-c2c(C(N(CCCNC(C3(O)COC3)=O)C)=O)con2)ccc(Cl)cc1 c1(CC)sc(=N)[nH]c1C(N1CC(NC(C2CCCCS2)=O)C(F)C1)=O Cc1ccc(CCC(=O)NC2CCC(F)(C)C2)cn1.C(c1cc[nH]n1)=CC(=O)N CN1CCC(C(=O)NCC2COCCN2C(c2cnn(-c3nccs3)c2)=O)C1=O c1(C(=O)NC2CCC(N(C)C(c3csc(O)n3)=O)CC2)ccc(C#N)cn1 N1(C(c2ncoc2C)C(=O)NCC=C)Cc2ccccc2CC1C(=O)NC C1(C)(C(=O)NC(COC)C)CCCN(c2nccs2)C1 C1(CNC(=O)Cc2cccs2)CC(NC(C2CCC2)=O)C12CCC2 n1(C2CN(C(=O)NCc3ccccc3Cl)C2)ncc([N+](=O)[O-])n1 C1(NC(=O)C(O)CC2CCCCC2)CC12CCN(C(=O)CCc1cscn1)CC2 C=CCC(CC)C(=O)N1CCC(OCCCNC(=O)Cc2csnc2C)CC1 S(=O)(=O)(c1ccc(C=CC(=O)O)cc1Cl)NC(CCSC)(C)C n1(CC)ccnc1CNC(C1CCCN1C(=O)Cn1nccn1)=O N#Cc1cccc([N+](=O)[O-])c1N1CC=CC(NC(C2(c3ccccc3)CC2)=O)C1 CC1CCC(CNC(C2CC3CC2(COCc2ccccc2)C3)=O)OC1 N#CCCCCCC(=O)N1CCCC(CO)(CNC(=O)CCC(N)=O)C1 N1(C(c2n(C(C)C)ncc2Cl)=O)CC2CN(C(C3(Cl)CC34CCC4)=O)CC2(C)C1 N1(C(CCSCC)=O)CCCCCC(NC(=O)C=C2CCC(C)CC2)C1 C(=O)(C1=NOC(C)(C)C1)N1CC(NC(C(C2CCCC2)OC)=O)C(SC)C1 N1(C(c2cnn(CCC)c2Cl)=O)CC(C)N(C(=O)CC2(C(=O)OC)CC2)CC1C C1(C(=O)N)CCCC(F)(F)CC1.c1(C(=O)NCC(C)CO)ccc(C2CC2)cc1 c1(C(=O)NC2CN(C(CC#N)=O)CC2N=[N+]=[N-])cc2c(s1)CCS(=O)(=O)C2 N1(C(CCOCC)=O)CC2CCC1C(CNC(=O)C(F)n1cccn1)C2 C(=O)(C1=CC2(CCN(C(C3(C)CCCC3O)=O)C2)C1)N1C(C)(CCC)CC1 N1(C(CC(CN(C)C)O)=O)C2CCCC1CN(C(=O)CN(C)C1CC1)CC2 C#CC1(C(=O)NCCC(C)c2cn[nH]c2)CN(C(c2n[nH]cc2Cl)=O)C1 c1(C(N2C(C)CC2C(=O)NCC2CC2[N+](=O)[O-])=O)ccc(F)c(O)c1 CCCC(C(=O)N1CC(C)(NC(=O)Cc2ccoc2)C1)c1cccc(Cl)c1 c1(C(=O)NCC(CC)NC(=O)Cc2cccc(SC)c2)cnn2c(C)cccc12 c1(C(=O)NCC#CCNC(c2c(CC)c[nH]n2)=O)ncn2c1CCC2 c1(OC)c(C(=O)NCC2CCCC2NC(=O)CCC2CC2)cccc1Cl.O C(CSC)(C(=O)NC1(CCC(=O)NCC(=O)NCCO)CCCC1)OC Cc1ccc(CC(=O)NC2CC(C(F)F)(NC(=O)CC3CC3(C)C)C2)cc1C c1(COC)ncc(NC(c2ncccc2)=O)cn1.c1(C=O)cc(C(C)=O)[nH]n1 O=C1C=C2CN(C(=O)C3=CCCN(Cc4cccc(CO)c4)C3)CCC2S1 CON=Cc1ccc(C(=O)NC2CC2NC(c2cc(Br)c[nH]2)=O)cc1 c1(C(N2C(C(=O)NC)C(O)CC2)=O)cc(F)c(OC)c(Br)c1 O=C(C1=NOC2COCC12)NCCCc1ccccn1 c1(C(=O)NCC2N(C(C3C(C=C)C3)=O)CCOC2)ccc(Cl)nc1OC C1(CNC(CC=C)=O)CCCCC1NC(=O)C(c1cccc(OC)c1)O C(C(CC(C)(C)C)C(=O)OC)NC(c1cc(C)ccn1)CC C12(CNC(CC(=C=C)C)=O)CC(CC)(CN1C(=O)C(C1CCCC1)O)C2 N1(C(CC2ON=C(C)C2)=O)CCOCC1C(=O)NCC1OCCC1C N1(C(C)=O)CC(C(=O)O)CC12CCCC2.n1(CCC)cc(CCCC(C)=O)nn1 CC1(C)CC(NC(C2(CO)CCCCO2)=O)CN1C(c1cc(C2CCC2)no1)=O CCCCC(CNC(c1csc(Br)c1Cl)=O)NC(=O)CC(C)CC N1(C(C(CN(C(c2c(CC)ocn2)=O)C)(C)C)=O)CCSCC(C)C1 CCCCCC(O)CC(=O)NC12CC1CN(C(c1ccc(C(C)(C)C)nc1)=O)C2 N(C1CCCc2n[nH]cc21)C(C(C)NC(C1(COC)CCCC1)=O)=O c1(C(N(CC(C)O)CCNC(COCC(=C)C)=O)=O)nc2cccnc2s1 N1(C(c2c(CNC(CCN(CCC)C)=O)noc2)=O)CC(=O)NC2(CC2)C1 N1(C(C(C)(O)C2CCC2)=O)CC2(CCN(C(c3cc(Cl)on3)=O)C2)C1 C(C(C)(C)C=O)N(C)C(c1cccc(F)c1)=O.C1(C=O)CCC(N(C)C)CC1.O C1(C(N(C2CCCN(C(c3cncc(Cl)c3)=O)C2)C)=O)CCCCC1(F)F Cc1cc(C(N2CCC(C(F)C(=O)NCCCS(N)(=O)=O)C2)=O)cnc1O CCS(=N)(=O)c1ccc(N2CCCC2c2ccc(OC)cc2)nc1 C1(CC)(NC(C2CC2C(C)C)=O)CN(C(C2CC(C)(CO)C2)=O)C1 C1(NC(=O)CC2CC3CC3C2)CC2CCC(C1)N2C(c1ccc(CO)c(Cl)c1)=O CC(C(=O)NC1(CNC(=O)CC2CCC3(CCC3)O2)CCC1)C(C)(F)F N1(C(c2c(C(C)C)cco2)=O)CCCC(C(C)C(=O)NCC(C)N(C)C2CC2)C1 c1(C(=O)NC2C3CN(C(C4(C#C)CCC4)=O)CC32)ccc(C(=O)OC)c(Br)c1 CC1=C(C(=O)N2CC(C)(CCC(=O)NC3CC3(C)C(F)F)C2)CCO1 CC(=O)CCCC(=O)N1CC2CC1CN2C(=O)Cc1ccc(C#N)nc1 C1(NC(c2cn(CC(N)=O)nn2)=O)CCCCN(C(C2CCC3(C2)N=N3)=O)C1 c1(CC)cc(C(=O)NCC2CN(C(c3ccccc3)=O)C3CC23)c(C)o1 CC1(C)CCCN(C(=O)CC2CCCC(=O)C2)C1C(=O)NC1CCC(O)C(O)C1 C1(F)CCN(C)C1.C(Cc1cc[nH]n1)(C(=O)N)NC(C(N1CCNC1=O)C)=O.C S(=O)(=O)(CCCC(C)(C)C)Nc1c(C(=O)OC)ccc(CC)c1 N1(C(Cc2cccc(C#C)c2)=O)CC(C(=O)NCC(C)(O)C(C)C)C2(CCC2)C1 N1(CC)CCC(N(C(=O)C(C)CN(C(=O)CC2CSC2)C)C)CC1 N1(C(C2(CC#N)COC2)=O)CC(NC(c2cc3ccncc3s2)=O)CC2(CC2)C1 N1(C(Cc2cc(C)sc2)=O)CC(C(=O)NCC2CCC(C)C2)C(C2CC2)C1 c1(CNC(C(C)OC2CCCC2)=O)nc(C(=O)NC)co1.C1(C)CCOC1 CC(O)(C(=O)NCCCN(CCC)O)C(F)(F)F.C1(CC(=O)N)CC12CC2 Cc1cccc([N+](=O)[O-])c1C(=O)NC(C1CCN(C(c2n[nH]c(O)n2)=O)C1)C C(=O)(CC(F)(F)CC)N1CC(C(C)NC(C2CCN(CC)CC2)=O)C1 c1(CC(=O)N(C)Cc2cn(C3CCCC3O)nn2)cc(C2CC2)nn1C C1CC(=O)NOCC(=O)N1.CC(C)(CN1CCCC1)NC(N)=O C1(C(N(C)Cc2nc(C)on2)=O)CCN(C(c2cncs2)=O)CC1(C)C c1(C(N2CC(OC)C(NS(=O)(=O)c3cnoc3C)CC2)=O)cccc([N+](=O)[O-])c1F C1(C)(NC(C(C2CCCO2)NC(CCC(C)=O)=O)=O)CCC(C)(C)CC1 N1(CCC(=O)N(C2CCN(C(C3CCC(=O)NC3)=O)CC2)C)CCSC(C)(C)C1 C12(NC(c3cnccn3)=O)CCCCC1CN(C(C1CC3CCCCCC13)=O)C2 N1(C(c2c(C)cc(C)s2)=O)CCN2C(=O)C(NC(=O)C3=CCCSC3)CC2C1 c1(-n2cc(C3N(C(CC(CC)C(F)F)=O)CC3)nn2)ccc2c(c1)CCN(C)C2 c1(OC)ccc(C(=O)NC2CC(O)CN(C(=O)CC3(O)CC3)C2)c(Cl)c1 N1(C(CNS(NC)(=O)=O)=O)CCC2CN(C(c3cc(OC)ncc3F)=O)CCC2C1 O=S(=O)(c1ccc2ncsc2c1)NC1CN(Cc2cnc(Cl)s2)C1 C(CCCCCNC(c1ccc(C(C)C)o1)=O)NC(c1cnc(CC)[nH]1)=O c1(CC)ncc(C(=O)NC2(CNC(C3CC3(F)F)=O)CC2)c(C)n1 C(=O)(C(C(C)C)n1c(-c2cccs2)nnc1S)NC1CCC(NC(CC)=O)C1 C1(C(=O)OCC)CCCN(CC(=O)NCCC)C1.CCC.C1(C=O)CC1C.O CCC(CC(F)(F)F)C(=O)NCC1CC1NC(c1cnn2c1OCC2)=O c1(CC(N2CCCC2)=O)ccn(C)n1.c1(OC)ncc(C(=O)NC2CC2)s1 CC(C(=O)NC1CC(CO)N(C(c2cccn2C2CC2)=O)C1)S(C)(=O)=O N1(C(c2c(C)oc(CNC(=O)C(C(C)C)C(C)C)n2)=O)CCCC1C1CCCO1 c1(C(=O)NCC(C)CNC(=O)C(C)(C)C(C)(C)O)cc(O)nc2ccccc12 CC(C)C(C(=O)NC1C=CC(C(=O)NCC2(C)CCCC2O)C1)N(C)C C1CCCN(C(=O)C=C2CC2)C1C.n1(CCOC)ccc(NCC(O)C=O)n1 Cc1c(C(=O)N(CCNC(c2ncccn2)=O)C(C)C)cnn1C1CCCC1 c1(N(C)C)ccc(C(=O)NCC2CCC(NC(C3C4CCCC34)=O)CC2)nc1 N1(C(=O)Cc2cscn2)CCN(C(c2cc(C3CC3)no2)=O)C(C2CCCC2)C1 CC(C)(C)CC(F)C(=O)NC1CCCC1Cn1cc(C2C3COCC23)nn1 Cc1cc(C)c(C(N2CC(NC(C34CCCCN3CCC4)=O)C(C)C2)=O)c(C)c1 Cc1cc(CCC(=O)NCCC2(C(=O)NC3CCC(O)C3)CCCC2)on1 C1(NC(Cc2c(C)nc[nH]2)=O)CC(F)CN(C(c2c(C3CC3)noc2C)=O)C1 C=CCC(CC)C(=O)NC(CCC)CCCNC(=O)C=CC(=O)N(C)C C1(CNC(C2(SC)CCC2)=O)CCC2(CO1)CCC2.C1(C(=O)N)CCCO1 C1(NC(=NCC)NC(c2ncnn2C)C2CCCO2)CC2CCCCN2C1 N1(C(C(CC)C#N)=O)CCN(C)CC1CNC(=O)Cc1cc(C)[nH]n1 CCCCC(F)C(=O)NCC1CC(O)CN1C(C1CCC1c1nc[nH]n1)=O C=C(C)C(C)(C)C(=O)NC1COCC1C(=O)NC1CC2C(C1)C2(F)F N1(C2CC3N(C(c4cccc(OC)c4F)=O)C(CC3)C2)CCc2c(O)n[nH]c2C1 c1(OC)cc(NC(=O)C(=O)NC2CC(=O)N(C3CCCCC3)C2)ccc1C C1(NC(C=Cc2nc(C)sc2)=O)CCN(C(=O)CO)CC1C(C)C.C(C)C c1(CC)ncc(Cl)c(-c2nnc(C3CCCCN3)o2)n1 C1(NC(c2nc(CC)sc2)=O)CN(Cc2ccc(C(=O)O)cc2Br)CC1C#N N1(C(=O)OC(C)(C)C)CCCC(NC(c2ncccc2)=O)C(F)C1.CC(F)F.O C(=O)(C(CCCC=C)NC(=O)Cc1csc(C)c1)NC(C#CC#C)(C)C c1(C(N(C2CCCN(C(c3cccnc3N)=O)C2)C)=O)cnc2c(c1)ncn2C C1(CC(=O)N(C2(O)CCCC2)C2CN(C(N3CCCC3)=O)C2)OCCCC1(C)C C#CCCCCC(=O)N1CCC(NC(c2cnc(C)n2C)=O)C(C)C1 c1(C(=O)OC)cncc(-n2cc(C3CN(C(c4ncn(C(C)C)n4)=O)C3)nn2)c1 Cc1sc(C(=O)NCC2CN(C(=O)C(O)CC(C)C)CCN2C)cc1S(N)(=O)=O N1(C(C=CSC)=O)CC2CC(NC(c3ccccc3C)=O)C(C2)C1.C(C)(C)C.O CC1CC(c2cccs2)CN1CC1(CS(C)(=O)=O)CCC1 c1ccccc1.C1(NC(CN(C)C)=O)CC(NC(=O)C(=O)NC2CC2)C1 c1(-c2c(C)occ2)csc(=Nc2ccc(C(N)=O)nc2)n1CCCN(C)C N1(C(C2(OC)CCS(=O)(=O)C2)=O)CCCN(C(C2CC(C)(C)C2)=O)C(C)C1 c1ccc(C(=O)CC)cc1.CCCC.C(=O)(C=CC=O)N.C(C)(C)C.C=O C(=O)(CCCCCC(C)O)N1C2CC(CNC(CCSCCCC)=O)C1CC2 N1(C(C2C(NC(C(C)NC(=O)NC)=O)CC2)=O)CCC(CC(N)=O)CC1 Cc1cc(C)c(C(=O)N(C2CCCN(C(c3csc(C(C)C)n3)=O)C2)C)s1 N1(C(C2C(OC)CCC2)=O)CC2COCCC2(NC(=O)CC2CCOCC2)C1 C1(O)(CNC(CCCC)=O)CCN(C(=O)C(O)CN2CCCC2)C1 C1(=O)CCCCCCN1.c1(SC)nc(=NC(=O)C2CC(=O)C23CCCC3)s[nH]1 c1(NC(C(c2ccc(C)cc2)OC)=O)cccc(CNC(=O)C(C)O)c1 C1(NC(C2Cc3ccccc3O2)=O)COC2(C1)CN(C(c1cccnc1O)=O)C2 C1(NC(C(C(C)C)OC)=O)COCCN(C(c2cccc(F)c2)=O)C1 N1(C(c2ncsc2C)=O)CCCC1CNC1CC(C(=O)O)C1.c1ccccc1 N1(C(c2nc(C)sc2C)=O)CCC(NC(=O)C=Cc2ccc(F)cc2)C1(C)C CCCC(CCC)CC(=O)N1CCC2C(NC(c3c(C)noc3C3CC3)=O)CC12 c1(OC)ccc(CNC(=O)Nc2ccc(OC(F)(F)F)c(C)c2)cc1Br CN=C(NCC(C)OC(C)(C)C)NC1CC1(C)C Cc1nccc(C(N2CC(CNC(C3CCC(C(N)=O)CC3)=O)C(C)C2)=O)c1C c1(OC)cc(-c2cnc(C(=O)NC3CONC3=O)cc2OC)cc(C#N)c1 c1(C(=O)OC)cc(C(=O)NCC(O)C)ccc1F.C(=O)C(C)N(C)C(C)=O c1(NC(C2(C)CCN2C(C2(c3ccc(O)cc3)CC2)=O)=O)ccc(Br)c(F)c1 N1(C(CNC(CCC)=O)=O)CCCC(O)(CNC(c2cnn(C(C)C)n2)=O)C1 CCC(C)CCCCC(=O)C1CC(NC(C2CCC2Cc2scnc2C)=O)C1 CC1(C)CCC(C(N2CC(F)CC2CNC(C2CCCC(F)C2)=O)=O)O1 CC1C(=O)N(CC(N2CC(c3ccc(N)cc3)C2)=O)CN1C(=O)CO C1(NC(=O)OC(C)(C)C)Cc2ccccc2CN1Cc1nc(-c2cccs2)cs1 c1(C(C)C)ccc(Br)cc1NC(N1CCC(CCn2ccnc2C(=O)O)CC1)=O C=CC1OCCCC1C(N1CCN(C(=O)CC=CCC)CC1c1ccccc1)=O N1(C(C2CCC(=O)O2)=O)CCC(CCNC(c2cc(CO)ccn2)=O)C(F)(F)C1 O(NC(=O)C(CN(C)C)NC(=O)C(C1CCOCC1)O)CCOCC#C C1(NC(c2n[nH]cc2I)=O)CC2(CCN(C(c3nc4ccccn4n3)=O)C2)C1 c1(C(N2CCN(C3CCN(C(C(C)CF)=O)C3)CC2)=O)cc(Cl)cc(Cl)c1 C(=O)(C(C)(F)CC1CCCC1)NC1C(NC(C(C)(C)OC)=O)COC1 N1(C(C2(C)CCOC2)=O)CC2(CO)CC1(C(N1CCC(F)(CO)C1)=O)C2 c1(C(N(C2CCCN(C(C3(COCC)CCC3)=O)C2)C)=O)ccn2ncnc2c1 c1(C(=O)NC(CC)(CC)CCNC(C2(O)CCOC2)=O)ccc([N+](=O)[O-])cc1Cl C(=O)(C(CC)C(=O)NC(CNC(=O)CCCCCSC)CO)OCC CC1CN(C(c2cc(C(N)=O)co2)=O)CC(C)CN1C(c1cn(CCO)nn1)=O CC(C(F)(C(=O)O)C(=O)O)NCc1cc(Br)cc(F)c1N N1(C(C=C(C)CNC(=O)CC2(C)CCOC2)=O)CC=CC1(C)C Cc1cc(NC(C2CC(F)CN2C(c2ccccc2Cl)=O)=O)c(C)s1 C#Cc1cccc(C(=O)NCC(O)C(=O)NC(C)(CC)CC)c1 c1(C(=O)NC(CNC(C(C)n2cnnn2)=O)(C)C2CC2)ccc(-c2ccco2)s1 c1(C(=O)NC2C(NC(c3ncn(C)n3)=O)CC2)c[nH]c2ccc(F)cc2c1=O C1(CC(=O)NC2CC(CCC(=O)NC3(C(F)F)CCC3)C2)CC1C1CC1 O=C(CCCC(F)(F)F)N1CCC2(CC2C(N2CC(F)C(F)C2)=O)C1 Cc1cn(C)cc1C(=O)NOCC(=O)NCCc1cn(C)nc1C N1(C(c2nc(C(C)C)sc2)=O)CCC2CN(C(C34CC(CO3)C4)=O)CCC2C1 C1(NC(COCC#C)=O)CN(C(c2cc(C)sn2)=O)CCC1CO n1(C(CC)CC)nc(Cc2cccc(C(=O)N(C)C)c2)nc1-c1ccc[nH]1 c1(-c2ccn(CCC)n2)nc(C2CC2C)nn1CCCOCC1CC1 C(=O)(C(C)(O)C1CCC1)NCC(CC)NC(=O)CCc1noc(C)n1 C1(C(=O)O)Cc2ccccc2C1NC(c1cn2cnnc2cn1)=O C1(N2CCC2)(CC)CCN(C(c2ccc(-c3ccnc(C)n3)cc2)=O)CC1 C1CC12CCC2.c1(C=O)ccc[n+]([O-])c1.C(C)(C(=O)NC)(C1(C)CC1)OC c1(CC(=O)NCCC(CNC(CCSC)=O)O)cn2cc(C)sc2n1 Cc1c(Cl)c[nH]c(=NCC2(O)CCCN(C(c3n[nH]cc3C(C)C)=O)C2)c1C#N Cc1nc(C(=O)NC2CC2NC(c2conc2C2CCCO2)=O)c2ccnc-2[nH]1 N1(CC)CCCC1=O.C(=O)CC(F)(F)F.C1(C(N2CCC2)=O)C2CC3C(C2)C13 C1(CC)CCCC(C(=O)OC(CNC(=O)NC)C(=O)OC(C)C)N1 CCCC(F)C(=O)NC1(C(=O)N(CC(C)(C)N(C)C)C)CC1(C)C Cc1c(C(=O)NCC2CC2NC(c2sccc2F)=O)noc1C1CC1 c1(CN(C(C2C(C)(COC)C2)=O)C)ccccc1.N1(CC=O)CCOCC1 C1(CNC(CCOCC#C)=O)CCC2(CO1)CCC2.C1(C)(C=O)C=CCCC1 N1(C(C)C)CCCC1C(=O)NCCCN(C)C(C1C(C(F)F)C1(C)C)=O [N-]=[N+]=NC1(C(N2CC(O)(CF)C2)=O)CCN(C(c2cc(C(F)F)[nH]n2)=O)C1 C=CCC(C)(C)CC(=O)N1CCN(C(c2ccnnc2C)=O)C(CC2CC2)C1 C(CCC(=O)N(C1CC(SC)C1)C)N(C(C(C)SCC)=O)C Cc1ccc(C(C)C)cc1C(=O)NCCCN(C)C(C1(F)CCCN(C)C1)=O c1(C(=O)NC2CCN(C(c3csc(C(F)F)n3)=O)CC2O)onc2c1CCCC2 Cc1nc2c(C(N3CC4CC4(NC(=O)C(C4(O)CCCC4)F)C3)=O)cccc2o1 C1(C(N2CCc3c[nH]nc3C2)=O)CCN(C(C2CC2(F)F)=O)C12CCC2 C12(CCNC(CCOCC)=O)CCC1CN(C(=O)Cn1nnc(=N)[nH]1)C2 c1(CC)c(C(=O)NCC(CC)(CC)NC(=O)C(C)CCC)cnn1C(CC)CC c1(C(=O)NC2C(CNC(Cc3cc(C)ns3)=O)CC2)cccn(C)c1=O c1(C(=O)OCc2c3ccc(CC)cc3on2)ccc2[nH]c3c(c2c1)CC(C)CC3 N1(C(C2C(C)SCCC2)=O)CCC(C2CC2)C1C(=O)Nc1cc(F)ccc1O C(CCCC)N(C(C=CCN(C)CC)=O)C(C)C.C(=O)(C(C)C1CCC1)N CCC(CC(=O)N1CC=CC(C(=O)NCC2CCN(CC)CC2)C1)C(F)F c1(C(=O)NCC=CCNC(C2OCC(C)(C)OC2)=O)[nH]nc([N+](=O)[O-])c1Cl C1(NC(c2cn(CC3CCCO3)nn2)=O)CCCCN(C(=O)C2CC2)C1 C1(S(C)(=O)=O)(C)CC1.c1(C(C)C)ccoc1C(N1CC(C(C)(C)O)C1)=O C12(C(N3CC4C(CNC(=O)CSc5nncs5)C4C3)=O)CCCCC1C2(F)F c1(CC)ncc(Cl)c(C(=O)NC(C)CNC(c2ccc(OC)c(F)c2)=O)n1 c1(C(N2CC(C)CC(NC(C3(COC)CC3)=O)C2)=O)ccc2cc[nH]c2n1 C1(CCC)CCCC1C(N1CC(O)C1)=O.c1(C(NC)=O)nnn(C(C)(C)C)n1 c1(OC)cc(C)c(C(=O)NCC(C)CNC(=O)C=C(C)C)c(F)c1 c1(NC(c2cncc(NC(c3cscn3)=O)c2)=O)cc(Br)c([N+](=O)[O-])cn1 N1(C(C2N(C(C)=O)CC(O)C2)=O)CC(NC(=O)C2=CCOCC2)C(C2CC2)C1 C(=O)C1=CCCCC1.c1(C(C)C)cccc(C(N2CC(C(C)(C)O)(C)C2)=O)n1.N N1(C(CCNC(C)=O)=O)CC2CCCN(C(c3cn4cc(C)nc4s3)=O)C2C1 c1(C(=O)NC2CC(C)N(C(=O)COc3ccsn3)CC2)cc2c(cn1)OCCC2 c1(C(C)C(=O)OC2CC3(OC(C)(C)C)CC23)cn(C)nc1C(F)F C(=O)(C(O)CCNC(=O)CC1(C)CCN(C(C2CCC(C)O2)=O)C1)OC CCCCC(O)CC(=O)NCC1CCCN1C(c1ccccc1NC(=O)NC)=O C(=O)(CC(C)(C)O)NCC1(O)CC(C(=O)NCCc2cn(C)nc2)C1 c1(CC)ccc(C(N2CC(CN(C)C(C3COC(=O)N3)=O)C2)=O)cc1CC N1(C(CCCC(=C)C)=O)CCn2c(CNC(C3CC(N(C)C)C3)=O)nnc2C1 N1(C(C(C)(C2CCC2)NC(CCC2C(C)C2)=O)=O)CC2CC=CC1C2 C(=O)(CC1OCc2ccccc21)NC1CCCN(C(C2(C(C)C)CC2)=O)C1 c1(C(=O)NCCN(C(C2COC(=O)N2C)=O)CC)ccc(C2CC2)cc1 C1(N(C(=O)Cc2ccco2)CC)CCCN(C(c2n[nH]cc2F)=O)C1 C(=O)(C1=NNC(=O)CC1)N1CCC(N2CCC(NC(C(CC=C)C)=O)C2)CC1 N1(C(C(N2CCOC2=O)C)=O)CC(O)CCC1C(=O)NCC1(CCO)CCCC1 C1(NC(C(C)(C)OCC)=O)CN(C(=O)C(F)CC2CCOC2)CC1CO Cc1nc2c(N3CCN(CCNCC4(F)CCCCC4(F)F)CC3)ncnc2[nH]1 C1(NC(c2c(CC)onc2C)=O)CN(C(=O)Cc2nc[nH]n2)Cc2ccnn2C1 C12(C(=O)N)CC3CC(C1)CC(C)(C3)C2.C(CC(C)C(=O)N(C1CCC1)C)OC C1(CNC(c2c(OC)nsc2)=O)CC2(CCN(c3nc(C)ccc3C#N)C2)CO1 CN1CCN(C(c2cccn2C2CC2)=O)CC1CNC(=O)C.C1CCCOC1.O c1(C(N2c3cccc(OC)c3CCC2)=O)ccc2c(c1)C(C)(C)OC2(C)C CC1(CC(=O)O)CCN1C(=O)C(Cc1ccnnc1)C=O.CCC.C(C)(C)C.O C1(OC(C)C(=O)NC2CCCC(NC(c3coc(Cl)c3)=O)C2)CCCCCC1 C(=O)(C(F)C(F)(F)F)N.c1(CCNC(c2c(C(C)C)con2)=O)ccccc1F n1(CCOC)nc(C(=O)NC2CCOCC2NC(c2ncsc2C)=O)ccc1=O C1CCCC(CC(N2CC(C(=O)NOc3sccc3C(N)=O)C2)=O)C1.CC(=O)N C1(O)(C(C)NC(=O)CCc2cccnc2)CCCN(C(=O)CC(C)(C)O)C1 c1(C(N(CCCNC(=O)C(C)(C)CF)C(C)C)=O)cc2c(s1)CCC2 CC(C)(C)C(C#N)C(=O)N1CC(CNC(c2coc(Br)c2)=O)C(O)C1 CCCC(C)(O)C(=O)NCC(CC(C)C)NC(c1c(OC)noc1C1CC1)=O c1(C(N2CCCC(n3cc(C4CC4CO)nn3)C2)=O)ccc(F)cn1 CS(=O)(=O)c1ccc(C(=O)NCC2C3CCCC2NC3)cc1[N+](=O)[O-] C1(NC(CC2CC(C)(C)OCC2)=O)CC12CCN(C(=O)C1=NNC(=O)CC1)CC2 CC1(C)CN(C(c2ccc(C(F)(F)F)nc2Cl)=O)Cn2ncc(C#N)c21 C1(C(=O)NCC2CC(C#N)C2)CCN(C(=O)Cc2ccccc2)CC1O c1(NC(C23CC(NC(CC4ON=C(C)C4)=O)C(OC2)C3)=O)ccc2c(c1)COC2 c1(C(N2CCN(C(CC(C)F)=O)CC2CF)=O)ccc(S(C)(=O)=O)c([N+](=O)[O-])c1 CC1(C)CCC(C)(NC(C2C=CCN(C(=O)CCn3ccnn3)C2)=O)C1 c1(C=O)cncc2c1CCC2.C1(C(C)(C)C)CCCN1C(C12CC(F)(C1)C2)=O.N CCC(C)C(CNC(C1(CC)CN(C(C2CCCCC2O)=O)C1)=O)OC c1(C(N2CCCC(N(C(C=CC=CCC)=O)CC)C2)=O)cc2nc[nH]c2cc1N c1(OC)cc([N+](=O)[O-])cc(Br)c1NC(c1cc(F)ccc1I)=O CCCC(C)CC(=O)NC(C)(C)CNC(c1ccc(CC)c(CC)c1)=O CCC(C)CCCCC(=O)NCCCCC(C)NC(=O)C(F)C(C)(C)O Cc1ccc(C(=O)NCC2CCCC2NC(c2cc(CO)on2)=O)c(Br)c1 N1(C(c2c(COC)cc[nH]2)=O)CC(C(N2CCOC(C#N)C2)=O)CCC1C C1(C=O)CC2(CCC2)CO1.Cc1nsc(NC2CC2)c1C=O.C(C)C(C)C.N c1(C(=O)NC2CCC(CNC(C(C)(C)O)=O)CC2)cc(O)cc(F)c1 N1(C(C(C(C)C)n2cncn2)=O)CC(NC(=O)CCC2CCCC2)CC(C)C1 c1(OC)cnc(F)c(C(N2CCC(C)(NC(=O)CC3CC3C3CC3)C2)=O)c1 c1(C(=O)NC(C)CC2CCN(C(=O)CC3CC34CC4)CC2)ccc2nsnc2c1 CCC(C)CC(=O)C(=O)N1CC2CC1C2C(=O)N(C(C)CO)C C=CC1OCCCC1C(=O)N(CCCCNC(=O)C(N1CCCC1)C1CC1)C N1(C(c2ccc(C)c(C)n2)=O)CCc2nc(C(=O)NCC3CC(C)C3)ccc2C1 c1(CC)cc(CC(N2CCC(C)(CCNC(C3CCCC3)=O)C2)=O)n(C)n1.C C1(CCC(=O)NCCn2cc(C3(O)CCC3)nn2)CCCCC1 c1(C(=O)NC(CNC(C(C(C)C)F)=O)C)cc(OC(F)(F)F)ccc1F N1(C(c2cccc(CCC)c2)C(=O)NCC(F)F)CCCN(C)S1(=O)=O c1(C(=O)NCCC(=C)CNC(=O)C(C)CC)cccc(C)c1 C1(NC(Cc2cccc(OCC)c2)=O)CCN(C(=O)COC)CC1.C1CC1.C C(=O)(CC(C)(F)F)N1C(C2CC2)CCC1.C1(C=O)CC(F)(C=O)C1.CC.O c1(C(=O)NNC(=O)Cc2csc(-c3ccc(O)cc3)n2)cccc2nsnc12 c1(OC)ccc(C(=O)NCC2COC(CNC(C3(C)CC3)=O)C2)nc1 C#Cc1ccc(C(N2CC(N3CC(NC(C4CCC4(F)F)=O)CC3=O)C2)=O)cc1 CCCC(CCCNC(c1cnn(CC2CCCO2)c1)=O)NC(=O)CCC(F)F N1(C(C=CC2CCN(C(C(C(CC)C)C)=O)CC2)=O)CC2COCC2(C)C1 c1(C(C(=O)NCCCN(C(C2(CC)COC2)=O)CC)C)cccnc1 C1(NC(C(c2cccnc2)NC(CCCOC)=O)=O)CCCN(C)C1 Cc1cc(Cl)ncc1CC(N1CC(NC(C2CCCO2)=O)C(C)C1)=O Cc1ccnc(C(=O)NCC2CN(C(=O)Cc3cnoc3)CC2C)c1 C1(n2cc(-c3c(C)noc3C)nn2)(NC(Cc2ccc(C)s2)=O)CCOCC1 N1(C(C=Cc2cnc(OC)nc2)=O)CCCC(C)(C)C1.c1(C=O)ncc(Cl)s1.N n1(C(CC)C)ncc(C(=O)NCC(CC)(CC)NC(=O)C(O)C(F)F)c1C N1(CCNC(=O)C=CCO)CCCN(C(C2(F)CCCCCC2)=O)CC1 CCCCC(C(=O)N(CCCOC)C)NC(=O)CC1CCSC1 c1(NC(C2N(C(c3c(C)cc(F)s3)=O)CCSC2)=O)cnc(O)c(F)c1 c1(C(N(C2CCCN(C(c3cc[nH]c3)=O)C2)CCF)=O)ccc2c(n1)COCC2 N1(C(C(CC)O)=O)CC2C3CCC(C(NC(=O)C(=O)NC(C)C)C3)C2C1 c1(SC)ccc(-c2cn(C(C)C(C)(C)NS(=O)(=O)C(F)(F)F)nn2)cc1 C1CCN(C(=O)CCN(CC(F)(F)F)C)CC1.CC(C(=O)N)OCC1CC1 N1(C(C2CCN(CC)C2)=O)CCOC(CN(C)C(c2c(C3CC3)cnn2C)=O)C1 C12(C(=O)NCC3CCCN(C(CC=CC(C)(C)C)=O)C3)CCC(F)(CC1)C2 Cc1ccc(CC(=O)NC2CN(C(C3CC(O)C3)=O)CC2C)c(Cl)n1 C1(C(=O)NCc2ncccn2)(NC(C2CC(=O)C2)=O)CCSC1 c1(C(=O)NC2(C3CN(C(C4CC(=O)NCC4)=O)C3)CC2)n[nH]c2ccccc12 N1(C(Cc2nc(C)sc2)=O)CC2CCC(C1)N2C(c1cc(C(=O)O)ncn1)=O c1(C(=O)NCC(CC)NC(=O)CC)ncoc1C1CCOCC1.C(=O)C=CCl.N Cc1cc(=NC(=O)CC2CC2CNC(c2cnnn2C)=O)[nH]n1C c1(CNC(C(C2CC2)SC)=O)cc(O)ncn1.C1(CC=O)CCC2CC12.C N1(C(C(=C(C)C2CC2)F)=O)CCC2CN(C(c3cc([N+](=O)[O-])c[nH]3)=O)CC12 N1(c2c3nc(C)sc3ncn2)CCC2(CCCC2CNc2ncccn2)CC1 c1(C(N2CC(NC(CC(CC)(C)C)=O)C(CO)CC2)=O)[nH]cc2c1CCS2(=O)=O C(=O)(C(C)CC(F)(F)F)N1CCN(C(Cc2c(C)ccnc2)=O)CC1C1CCC1 N1(C(C=Cc2ccc(C)s2)=O)CC(NC(=O)CCN2CCOC2=O)CC(O)C1 Cc1cc(F)cnc1C(=O)NC1CC2(C1)CC2C(=O)N.C1CN(C(C)C)C1 N1(C(C2(C(=O)OC)CC2)=O)CCCC(F)C1.c1(C(C=O)(C)C)cccc(F)c1 N1(C(C(C#C)(C)C)=O)CCC(NC(c2c(C(F)(F)Cl)n[nH]c2C)=O)C(F)C1 n1(CCOCC)nnnc1C(c1csc(C2OCCO2)c1)N.C1CC(CCO)C1 c1(OCc2cccc(Cl)n2)cnc2[nH]cncc1-2 Cc1ccsc1C(N1CC=CC1Cn1cc(C(C2CC2)N(C)C)nn1)=O Cc1ccc(Br)cc1CC(=O)Nc1ccc(NC(c2[nH]cc(C)c2C)=O)cc1F C#CC1(C(=O)NC2CC(c3ncc[nH]3)C2)CCN(C(=O)CC2CCC(O)C2)CC1 Cc1nc2cc(Cl)cc(C(=O)NC3C4CN(C(=O)C5=C(Cl)CCC5)CC34)c2[nH]1 c1(NCC(N(C)C(C2(S(N)(=O)=O)CC2)=O)C2CC2)ncnc2ccccc12 S(=O)(=O)(c1c[nH]c(=NCC2COC(C)(C)O2)cc1C)N1CCCC(C=C)C1 C1(CC(=O)NC(CNC(c2nccc(C)c2)=O)C2CC2)CC2(CCCC2)CO1 CCC(C(=O)N1CC(NC(C2(O)CCC2)=O)CC2(CCC2)C1)C(C)(C)CC c1(C(=O)NC(C2CN(C(c3cc(Cl)cnn3)=O)CCO2)C)ccc(N)c(F)n1 c1(SC)cccc(NC(C2(NC(c3ccc(Cl)cc3)=O)CCCC2)=O)c1 C1(NC(C(C(=C)Cl)(C)C)=O)CC2CCC1CN(C(=O)C)C2.C1(C(=O)N)CC1C C(CCN(C)C(c1ccc(F)s1)=O)(C(C)C)NC(C(C)SC)=O Cc1cc2cc(NC(N3CCN(C(=O)C(N)=O)CC3)=O)ccc2o1 C1(C(N2CC(C(O)C(=O)N)C2)=O)(NC(N)=O)CCCCC1.C1(CC)CCCOC1 c1(C(N2C(CO)CC(NC(C3CC4CCCC4C3)=O)C2)=O)ncc2ccccn12 N1(C(C2N(C(C(C)N(CC)CC)=O)CC2)=O)CC(O)(C(F)F)C1 CC1(C)CC(C(N2CCCC2c2ncc(-c3ccccc3)[nH]2)=O)CO1 CC(C(=O)NCC(C1CC1)N(C)C(c1n[nH]c(C2CC2)c1Br)=O)C(C)(C)C N1(C(C(=O)NCC)CCC(C)C)CCc2cc(C(=O)OC)cnc2C1 c1(C(=O)NC2(C)CCN(C(CN(C3CC3)CC)=O)C2)cnc2oncc2c1.C CC1CC(C)CCN1C(=O)C(O)CC1CCCC1.n1(CC(=O)N)ncn(C)c1=O N1(C(c2cnc(S)[nH]2)=O)CC(CO)C2(C1)CN(C(C1CCN1C1CCCC1)=O)C2 C1(CC(N2CC=CC(NC(CC3CC(=C)C3)=O)C2)=O)CCC(=O)NC1=O C1(C(N(CC=C)CC)=O)(C(C)C)CCN(C(=O)CCCn2ccnc2)C1 C1(C=O)CCOC(=O)CC1.Cc1nc(CN(C(=O)Cc2cnn(C)c2)C)cs1.N c1(C(NCCNC(C2C(C)C2)=O)=O)n[nH]c2c1CS(=O)(=O)CC2.C1CC1 C(=O)(CCCC(F)(F)C(F)(F)F)N(CCCN(C(C1CCN(C(C)=O)C1)=O)C)C N1(C(c2ccc(C#C)cn2)=O)CCC(C=C)(C(=O)NC(C)CCC)CC1 Cc1cc(Cl)ccc1CC(=O)NC.C12(C=O)CCCC1C2(F)F.C12CC(C1)C2 C1(C(=O)NC2CCCC(NC(CC(=C)C)=O)C2)C2CC3C(C2=O)C13 Cc1nn(CC(=O)NC2CCC(CNC(C3(CO)CC3)=O)C2)c(C)c1Br N1(C(=O)C(O)CCCNC(C2(CO)CC2)=O)CCC2=C(CCCC2)C1 N1(C(CN(C)C)=O)CC2=C(C1)CN(C(C1(C)CC1Br)=O)C2 C1(NC(=O)Cc2cc(C(F)(F)F)n[nH]2)CC2CN(C(C3(Cl)CC3)=O)CC12 C1(NC(C2CCCN(CC(C)C)C2)=O)(C)CC2CCC1CC2.C(=O)C(C)C#N.N C1(F)(C(=O)NC(c2nc(C)on2)C)CN(C(=O)OC(C)(C)C)CC1(C)C c1(CCC)cc(C(N2CCC(c3n[nH]cc3CNC(C)=O)C2)=O)c(C)o1 CCCC(C)CC(=O)N1CCN(C(=O)C=Cc2ccoc2)CC1c1cnn(C)c1 c1(C(=O)NC2CCC(NC(=O)C=CC3CCOC3)CC2)ccc2n[nH]cc2c1Cl N1(C(C(=O)Nc2cccc(COC)c2C)=O)CC2(CCCCC2)CC1C(=O)OC C1(C(=O)NCC2(CCC=C)CC2)CCCN1C(=O)CC1(C)CCOC1.C c1(C(=O)NCC(CC=C)NC(c2ccccc2Cl)=O)cnn2c(OC)cccc12 C(=O)(C(Cc1cc[nH]n1)NC(=O)C(F)F)NC(C1(O)CCC1)C c1(CC)ccccc1NC(=O)C(c1ccon1)N(CCCC(C)(F)F)C c1(C(=O)NC2CC(CCNC(C3CCC(C)C3)=O)C2)ccc2nnc(S)n2c1 C1(C(N(CC(c2nn[nH]n2)C)C)=O)CN(C(=O)C2=CCOCC2)CC12CC2 n1(C(C)C)ncc(C(=O)N(C2CN(C(=O)Cc3cccc(C4CC4)c3)C2)C)c1N c1(SC)ncc(C(=O)NCCC2(C)CCN(C(C3(C)CCC3)=O)C2)n1C C(=O)(C1SCCc2sccc21)N(CCNC(=O)CN1CCCC1C)CC C12(NC(Cn3c(C)ncc3)=O)CCOCC1CN(C(=O)CN1CCCCC1=O)C2 N1(C(c2c(C)nccn2)=O)CC2CCN(C(c3ccc(C(F)(F)F)cc3)=O)C2C1 Cc1cccc(C(CC(=O)O)N(CCCCC(C)C)Cc2ccccc2)c1C C=CCC(C)(CC=C)NC(c1coc(C)n1)c1nnnn1C(C)(C)C C(=O)(C(C)(C)C(F)(F)F)N1CCN(C(CNC(C(C)OCC)=O)C)CC1 Cc1cc([N+](=O)[O-])c(C)cc1C(=O)NC1(CC(=O)NC2CNC2)CCC1 N1(C(C2N(CC)CCOC2)=O)CCC(C2CC2)C1.c1(C(=O)N)ccsc1C(F)F C1(CCOC)(OC)CCCN(C(c2c[nH]nc2C)C(=O)NC(C)(C)C)C1 CC1(CNC(C2CC23CCOCC3)=O)CCN(C(=O)C2=CSCS2)CC1 c1(CCCCC)ccc(CNC(=O)CC2CCC(NCc3ccccn3)C2)o1 C(=O)(C(C)(C)CNC(=O)CCC1CCCC1)NCC.c1(C=O)cncn1C C12(NC(=O)C3=CCOCC3)CCCC1CN(C(c1cc(CC3CCC3)c[nH]1)=O)C2 c1(C(N(C)CC2CCN(C(=O)C(c3ccccc3)SC)C2)=O)ccc(CO)cc1 CC1(C)CCC(C(=O)NCCC(C)(C)C(=O)NC2CC(F)(F)C2(C)C)CO1 C(=O)(C1=CC2CCC(C1)C2)NC(C(=O)N(CC(COCC)O)C)C(C)CC c1(N(C2CCCCC2)C)ccc(C(=O)N(C)C)cc1.N12CCC(O)(C1)C2=O CC(C)CC(O)CC(=O)N(C)Cc1ccc(CNC(C2CC3C=CC2O3)=O)cc1 c1(C(=O)NCCN(C(=O)CC(C)(C)C)CCC)ccc(OC)c(OC)c1C N1(C(CNC(C2C(C(=O)OC)C2)=O)=O)CCS(=O)CC1C.CC.C(=O)N c1(C(=O)NCC(c2ccccc2)NC)cc(O)no1 c1(C(=O)NC(CC)CNC(c2n[nH]c3c2CCOC3)=O)cccc2nn(C)cc12 N1(C(C(=Cc2ccccc2)CC)=O)CC(NC(=O)CS(=O)(=O)CC)CC(C)C1 CCC(O)C(F)(F)C(=O)N(CCCNC(c1occc1Br)=O)C1CC1 c1(CCC=O)nc(SC(F)(F)F)no1.C1(NC(CNC(CC)=O)=O)CCC1.C N1(C(Cc2c(C)cc(O)cc2C)=O)CCC(O)(C2CCN(C(=O)C(C)O)CC2)C1 CN1C(=O)CCC1C(=O)NC(C)C(C)(C)C.c1ccc(Cl)cc1.C(=O)(C)N c1(CNc2cc(NC3C(OC)COCC3)ncn2)cccc([N+](=O)[O-])c1N c1(NC(c2cc(OC)c(S(C)(=O)=O)cc2)C)ccc2c([N+](=O)[O-])cccc2n1 C1(NC(CSCC)=O)COCCC1C(=O)N(C)CCN(C)CC CCC(C(N)=O)(C(C)C)NCC1CC12CN(C(=O)Oc1ccccc1)C2 C(CC(C)(C)C)NC(C(C)SCC)=O.c1(C=O)cccc(C(C)(F)F)n1.N C1(C(=O)N)CC2COCC(C1)C2.C1(NC(CC2N(C(C)=O)CCC2)=O)CCCCC1 n1(-c2ccc(C)cc2)c(C)cc(C(=O)NCc2cccc(OC3CNC3)c2)c1C c1(NC(N2CCCN(Cc3onc(C)n3)CC2)=O)c2c(nn1C)CCC2 c1(C(N2CCCC(C(C)NC(c3cn(CCC)nn3)=O)C2)=O)ccc(Br)c(C)c1 CCC(C)C(O)C(=O)NC1CC(N(C)C(C2CC=CC(O)C2)=O)C1 N1(CCCc2ccc(OC)cc2)CCC(=O)N(CC2CCC(F)(F)C2)C1=O C12(C(=O)NC(c3nc(CC)[nH]n3)C)CCC(CC1)N(C(c1cnccc1C)=O)C2 c1(C(N2CC(C(C)C)N(C(=O)C=CCF)CC2)=O)cc(=O)n(C)cc1Br N1(C(c2ccn(C)n2)=O)CCN(C(=O)CCn2cncn2)C(CO)C1 C1(C=O)CCC(C)(F)CC1.C1(COC)CN(C(=O)C(C)(O)C2CCOC2)C1.N Cc1ncc(C(=O)NCC2CC(NC(C3COC(C)C3)=O)C2)cc1N N1(C(CC(CC=C)NC(C(C=C=C)C)=O)=O)CC2(CCC1CO)CC2 Cc1coc(CC(=O)OC(c2ccccc2)C(N2CCOCC2)=O)n1 N1(C(C2C(c3n(C)cnc3)C2)=O)CCCC(C2(NC(=O)CC3CCCO3)CC2)C1 C(CC)(CCCC(=O)N(C)Cc1cscn1)NC(C(CC)(CO)OC)=O O=C1OC(CNC(=O)NC2CC2)CC12CC2.c1ccccc1N1CCOCC1.C c1cccc(C(=O)N(C(C)C)C)c1.CC(C)[SH](=O)=O.c1(C=O)ccc(Cl)o1.N Cc1cnccc1C(=O)N(CC(C)CNC(C1CCCC12CC2)=O)C c1(COC)ccc(CNCc2c[nH]nc2-c2ccc(C)cc2)cc1C#N c1(C(=O)NCC#CC(=O)NCCC2CC(O)C2)cccc2nccn12 CC(C)(CO)C(=O)NC1CC(C)(NC(C2CCCCO2)=O)C1 C1(NC(CC2C(C)CCC2)=O)CCN(C(=O)Cc2ccno2)C1C C1(C(N(CCCSC)C)=O)(CNC(=O)C(F)=CC2CC2)CCC1 c1(CC(N2CCN(C(CNS(N)(=O)=O)=O)CC2CO)=O)cccc2ccoc12 c1(C(N2C(C)CC(C)C2)=O)ncnc2c1CCC2.C1(CC(=O)N)CS(=O)(=O)C1 c1(C(N2CCCC(Cn3cc(CS(C)(=O)=O)nn3)C2)=O)ncn2ccccc12 C(=O)(CCC(=O)NN(C)C)NCC1C(NC(C(CC)OC)=O)COC1 Cc1c(Cl)ccc(Cl)c1NC(c1ccc(O)c(F)c1F)=O C1(=CC(=O)N)CCOc2ccccc21.C(C)(C)(CC(=O)NC(C)C(C)C)SC Cc1cc(C(F)(F)F)cc(N2CCC(O)C(C(=O)NC(c3cccnc3)C)C2)n1 C#Cc1ccc(C(=O)NC(CNC(C2CCC2OC)=O)CC(F)(F)F)nc1 N1(c2cc(C(=O)OC)c(Br)cc2)CCC2(CC1)CC(C(=O)OC(C)(C)C)=NO2 CC#CCC(C(=O)NCC(C)C(=O)OCC)NC(=O)C(C)C(C)C C1(C(C(N2CC(C)(OC)C2)=O)C)CCCN(C(C2CN(C)C2)=O)C1 N1(C(C=CC(=O)N(C)C)=O)C2CCC1C(NC(=O)CC(O)c1ccccc1)C2 c1(C(=O)NC2C(C)CN(C(c3coc(CO)c3)=O)C2)c[nH]c2nccc-2c1 c1(CC(=O)NC2CN(Cc3cnc(O)nc3O)CC2F)ccc(F)cc1Br c1(C(=O)NC(CNC(CCC2CCC(C)O2)=O)C2CCC2)ccc(C#N)cc1 Cn1cc(C#N)cc(NC(=O)NC2CCN(C(c3ccccc3)=O)C2)c1=O c1(CC)cn2c(n1)CC(C(=O)NC(C)CC(F)(F)F)CC2.C(=O)CC(C)(F)F Cc1scnc1C(=O)NCCOCC(=O)NC1CCN(C(C)C)C1 CC(C)CCCNC(=O)CN1CCC(N(C)C)CC1.c1(C(=O)N)cncc(O)c1 CCCC(C)CC(=O)NC1CCCCCC1C(=O)NCCc1nc[nH]n1 C1(NC(C(COC)COC)=O)CCC(C)N(C(c2cc(Br)cnc2O)=O)C1 C(=O)(C(O)P(C)(C)=O)NCCCC1N(C(Cc2c(C)ccs2)=O)CCC1 N1(C(c2c(C#C)c[nH]n2)=O)CCCCC(CNC(=O)CC2CCCC2O)C1 N1(C(CNC(C2C(C)C2)=O)=O)CCCOC(CNC(=O)CCCC2CCC2)C1 C1(NC(=O)CCOc2ccccc2Cl)C2CCN(C(=O)CC3(CO)CC3)CC12 Cc1cccc2c1CCOC2C(=O)NC1CCOCC1NC(=O)C1=CCSC1 N1(C(c2onc(CC)c2C)=O)CCC(NC(=O)CC(F)(F)F)CC1C.C(C)=O.O CCCCCCCCC(=O)NC1CN(C(=O)CC(C)c2ccccc2)CCC1F n1(CC(=O)N(C2C3CN(C(COCC(C)C)=O)CC32)C)ccc([N+](=O)[O-])n1 C(CC(O)C(=O)NCC1CC(F)CN1C(C1CN(C2CCOC2)C1)=O)SC c1(CC)ncccc1NC(c1occc1CNC(c1ccsn1)=O)=O N1(C(COC2(C)CCC2)=O)CCOC(CC2CN(C(C3C4CCCOC34)=O)C2)C1 C1CC(F)(F)C(=O)N1.Cc1ccc(-c2cn(C(C)C(=O)NCC(C)C)nn2)s1.C c1(CC(N2CC3C(C(=O)NC(C)C(F)(F)F)(C3)C2)=O)cn(C)c2ccccc12 N#Cc1ccc(C(N2CC3CN(Cc4coc5ccccc45)C3C2)=O)c(Cl)c1 C12(C(=O)NC3C=CCN(C(c4c(C)ocn4)=O)C3)CCCC(C)(C1)OC2 c1(C(=O)NC2(C)CC(NC(C3(C(C)C)CCC3)=O)C2)cc(C#N)c[nH]1 CCCCCC(=O)NCCC(=O)NCCc1cn(CC)nn1 c1(C(N2CCN(CCCNC(CC3C(C)C3)=O)CC2)=O)cc(F)ccc1N N1(C(c2cc(Br)c(C(=O)OC)s2)C(=O)NCC)CCc2nc(Br)n(C)c2C1 N(C1COCc2cc(Cl)ccc21)C(=O)NCCC(=C)CO CCCCS(=O)(=O)CC(=O)NC12CC(NC(=O)OC(C)(C)C)(C1)C2 C1CC2COCC2N1C(c1nccnc1C(N)=O)=O.C(C)(C(=O)N)SCC.C C#CCCCC(C)C(=O)NCC1(O)CCCN(C(=O)COCc2ccccc2)C1 Cc1cccc(C(=O)NC)c1.C1CC(C(F)(F)F)CN1C(c1cnnc(O)c1)=O CON1CCC(C(=O)NCCOC2CN(C(C3CC3c3ccoc3C)=O)C2)CC1 C1(CNC(c2c(C)cc(C)nc2)=O)CN(C(c2ccc(O)cc2)=O)CC(C)(C)O1 c1(CN2CCC(C(c3n(C)ccn3)O)CC2)c(-c2cccc(Cl)c2)ccnc1O N1(C(C(C)(C)n2cccn2)=O)CC2=C(C1)CN(C(=O)CC1CCCNC(=O)C1)C2 Cn1nccc1C1(C(=O)N)CC1.CC(C)CO.C(=O)CC1(C(F)(F)F)CC1 C(=O)(C1=COCC1)NC1C=CC(C(=O)OCC)C1 C(C(=O)N(C1(C(=O)NC(c2cscn2)C)CC1)C)(C1CCOC1)OC c1(C(=O)NC2CC3C(NC(=O)CCc4csnn4)C3C2)cc2n(n1)CCC2 C12(NC(CC=Cc3ccc(C)cc3)=O)CCC(CN=c3nc(C)[nH]s3)(CC1)OC2 c1(NC(CNC(C=C(C)c2cccs2)=O)C(C)C)nc(C(C)C)ncc1Br CC1(C)CC(C(=O)NC)CN(C(=O)C)C1.C1CCCO1.C1(C(F)(F)F)CC1 c1(CNC(c2c(C)nn[nH]2)=O)ncc(C=O)cn1.C1CC(=O)N(C2CC2)C1.N C12(CC)CN(C(=O)CC3CCCO3)C(CNC(c3cccnc3)=O)(C1)C2 c1(CC(=O)NC2(COC)CN(C(=O)CC3CSC3)C2)cc(C)ccc1F n1(CC)cc(Cl)cc1C(N1CC(NC(=O)C(c2ccccc2)C)CC1C)=O CCC(CC(=O)N(C1CN(C(c2cc(C)c(F)cc2Br)=O)C1)C)C(F)F C(=O)(C(C)CC(C)CC)N1CC(C(N)=O)(CNC(C2CC(=C)C2)=O)C1 c1(CC)cnc(C(=O)NC(C2(O)CN(C(=O)Cc3ccco3)C2)C)s1 C(=O)(CC(C)CC(C)(C)C)NC1(CC(=O)NCc2c(C)cc(C)s2)CC1 N1(C(C(C=C)(C)CC)=O)CC(CO)C2(C1)CN(C(=O)CC(C)(C)CCC)C2.C1CC1 CN=c1[nH]c(=NCCc2ccn(C)n2)[nH]c(=NC2CCC3C4CCC(C4)C23)[nH]1 N1(C(CCC(C)SC)=O)CC(N=c2[nH]cnc3cnccc23)C(C)(C)C1 C12(C(N(CCCCCCNC(CNC(CC)=O)=O)C)=O)CCCC(C1)OC2 c1(C(=O)NC2C(OC)CN(C(c3cccc(N)c3)=O)C2)cn2c(n1)SCC2 c1(C(N2CC3(CN(C(c4c(C)[nH]cc4)=O)C3)C2)=O)cnc2n(c1=O)CCS2 C(=O)(CCC(N)=O)NC(C)(CNC(=O)COCCO)C1CCC1 N1(C(c2c(C)scc2)=O)CCCCC1C1CCN(C(C23CC(CF)(C2)C3)=O)CC1 N1(C(CC(C(=O)OC)C)=O)C(C(=O)NC(C)(C)C)C2CC(F)C1C2 N1(C(C(c2ccccc2)OC)=O)CC2CC(C1)C2NC(C1CCC2(CCC2)C1)=O C(=O)(CCCCC(C)C)NC(C1OCCN(C(c2ccc(C)s2)=O)C1)C [N-]=[N+]=NCCCCCCNC(c1cc(CNC(=O)Cc2ncccc2F)on1)=O N1(C(C=C(CCN(C)C)Cl)=O)CC2(NC(=O)C(O)C(C)(C)C)CCCC2(F)C1 c1(C(N2C(C=O)CCC23CC3)=O)cccc2[nH]ncc12.C1(C(=O)OC)CCC1.N C1(C(N2CCC2)=O)(CNC(COCCCC)=O)CC(F)(F)C1 CC1(C)CC(C(=O)NC2CC3(C2)CC(NC(=O)Cn2cnnc2)C3)CNC1=O c1(C(=O)N)cnc(O)c2cncn12.c1(SCC(=O)NC2CCC2)ccc(Cl)cc1 c1(C=O)cc([N+](=O)[O-])c(F)cc1N.Cc1ccc(C(=O)N(C)CC2CC2)cc1.N C1(c2onc(Cc3nc(=N)[nH][nH]3)n2)CC2(CCCCC2)C1 c1(SC)ncc(NC(c2ccc(N3CCC(OCCNC)CC3)nc2)=O)c(O)n1 c1(C(N(CCCC)C)=O)cc(F)c(F)c(F)c1N.C1(OCC)CC(C(=O)N)C1 c1(N(C)C)cccc(-c2ccnc(NC(c3cccc(C(C)(C)O)c3)=O)n2)c1 c1(NC(C2C3N(C(CNC(C)=O)=O)C(CC3)C2)=O)cnn2ccccc12 C1(c2ccn(CC(C)C)c2)NC(=S)N(C2CC2)C2=C1C(=O)NC21CCOC1 c1(OCC)cc(F)ccc1-c1ccc(NC(=O)Cc2cccc(OC)n2)cc1F C(=O)(CCC(N)=O)N(C(CN(C(c1ccn(CCCC)n1)=O)C)C)C.C(C)=O.N CC#CCCCC(=O)N1CCN(C(=O)CC2SC(=N)NC2=O)C(CC)C1 N1(C(C2C(C)=C2)=O)CC=CC(NC(=O)CCNC(=O)CC(C)C)C1 CC1CCCC1(C)C(=O)NCC1C2CN(C(=O)C(C)CCN(C)C)CC12 C1(CC)CCOCCN1C(CC1C=CCC1)C(=O)NCc1cccc(OC)c1 c1(C(C)=O)cc(C(=O)NC2(C=O)CC(F)C2)no1.C(=O)C(C)(C)C.CC c1(NCC(c2ccc(Cl)cc2)C)nccc(N2CCC(C(O)C(N)=O)CC2)n1 N(C(=NCCCCC1CC1c1ccccc1)NCC1C2CCCCC12)CC(F)F C1(C(N(CCCCCNC(c2cc(C)oc2)=O)C)=O)CN2CCN1CC2C CCC(CC(C)C)C(=O)N1CC(CC(=O)NCC[Si](C)(C)C)(OC)C1 CC(C)CCC(=O)NC1(CO)CN(C(=O)CCc2cncc(Br)c2)C1 CCC(C)C(=O)NCCOCCN(C(=O)Cn1ccsc1=N)C C#CCCCCC(=O)NCC(O)CNC(c1ccc(CSc2nncn2C)o1)=O c1(C(=O)NC2(C(N3CC(OCC(=O)NC)C3)=O)CC2)ccnnc1O N1(C(c2ccc(C)cc2N=[N+]=[N-])=O)CCCC(N=c2c(Br)c[nH]cc2[N+](=O)[O-])C1 N#Cc1ccc(NC(C2(F)CCN(C(c3cccnc3C(N)=O)=O)C2)=O)cn1 c1(CC(C(N2CCCC(CC(=O)NC)C2)=O)C)cncc2ccccc12 N1(C(CN(C(C)=O)C)=O)CCC2CCN(C(c3cnc4[nH]c(O)nc4c3)=O)CC12 Cc1cc(Cl)c(C(=O)NCCC(C)CCNC(c2n[nH]c(C3CC3)c2Cl)=O)s1 c1(C(N2CCC(OCCNC(C(C)(CO)OC)=O)C2)=O)cccc(F)c1Cl CCC(C(=O)NC(C1(O)CN(C(=O)Cc2cnnn2C)C1)C)n1nccc1C C1(C=O)C2CC3C(C2=O)C13.C1(C(=O)N(CC)C2CC2)CC1(F)F.CO c1(OC)ccc(F)cc1C(=O)NCC(O)CNC(=O)CC12CCCC1C2 c1(C(=O)NC2C(SC)CN(C(c3ccc(O)nn3)=O)C2)cncc(C)c1C C1(c2cn(CCCC(=O)OC)nn2)N(C(=O)C(C2CCC2)OC)CC1(C)C.OC C1(CCNC(CN2CC(C)(OC)C2)=O)CCCN(C(c2cc(C)ns2)=O)C1 C(CN=c1[nH]n2cc(C)nc2s1)N(C(c1cnco1)=O)CC C1(C(=O)NC2C3CN(C(c4ccc(C)nc4N)=O)C2C3)OCCOC12CCC2 CC(CC(=O)N(C)Cc1cn(C)cn1)C(C)(C)NC(=O)CSC(C)(C)C C1(NC(C2(NC(=O)COc3ccsc3)CC(O)C2)=O)CC(O)C12CCC2 C1(CNC(CC2(C)CCN(C(=O)C=CCO)C2)=O)CCC(C#N)CC1 c1(C(=O)OC)cncc(C(=O)N(C(C)CC)C)c1.c1(CC(=O)N)ncccc1F C12(C(=O)NC3CCCCN(C(=O)C(F)C4CCOC4)C3)C3CCC(CC13)C2(F)F Cn1ncc2c1CCC(C(N1CCN(CCCNC(c3cn[nH]c3)=O)CC1)=O)C2 C1(NC(CCCC#C)=O)CC(O)CN(C(c2cn(C)nn2)=O)C1 C(=O)(C(C(=O)N1CCOCC(NC(C23CCC2C3)=O)C1)C(C)(C)C)OCC C=C(Cl)CC(C(=O)NC(c1cn(C)cn1)C)NC(C12CC(F)(C1)C2)=O c1(-c2cn(CC(O)COC3CCOC3)nn2)ccc2c(c1)OCO2 CCC(O)C(C)C(=O)NC1(CC=CC(=O)Nc2cc(C)cc(C)c2)CCC1 CC1(C)CCCCC(C(=O)NCC2(F)CCCN(C(C3CSCCS3)=O)CC2)C1 c1(C(=O)NC(C)CCCNC(C2CS(=O)C2)=O)ccc(F)c(Cl)c1 CCCCCC(C)(CC)C(=O)NCCN(C(C)C(=O)NCC(C)C)CCC c1(C(=O)NC(C(C)NC(c2n(CCC)nc(C)c2)=O)C)cnc2ccnn2c1N C1(NC(c2c(C)scn2)=O)CCCCC12CCCN(C(c1cnn(C)c1N)=O)C2 Cc1cnc(F)c(CN)c1.c1(Cc2nnn[nH]2)cc(Cl)ncc1C1CC1.C1CC1 c1(C(N2C3C(CNC(COCCCC#C)=O)C(C3)C2)=O)cccc2[nH]ccc12 CP(C)(=O)CC(=O)NC1CCC1NC(=O)C(c1ccc(Cl)cc1)O CCC(CS(C)(=O)=O)NC(c1ncn(C)c1Cl)c1nnnn1C1CCOCC1 c1(NC(c2csc(CNC(c3cc(CO)on3)=O)c2)=O)cccc(F)c1O C(N=c1ccn(CCCO)[nH]1)(c1n(Cc2occc2)nnn1)c1cnoc1 C1(c2cccc(C)c2)CCN(C(C23CCCCC2C3)=O)C1(C)C C1(F)(C(=O)NCC(C(=O)NC)O)CCN(C(=O)CC(C)C)CC1 Cc1ccc(OCC(N2CCCCC2CCCNC(C2(C)CC2)=O)=O)cc1C c1(C(CNC(=O)C(=O)NCC(O)C2CCC2)OCC)cccc(Cl)c1 Cc1c(C(=O)NC2CCN(Cc3n[nH]cc3Cl)CC2F)sc2ccccc12 CC(C)CC(=O)C(=O)NC(C1CN(C(=O)Cn2ncn(C)c2=O)CCO1)C C1(NC(C(C2CCOCC2)OC)=O)CCN(C(c2cc(C)c(C)cn2)=O)CC1C Cc1cc(N(C)Cc2ccc[nH]2)nc(NC(c2cn(C)nc2C)C)n1 C(C(=O)N=S(C)(=O)C1CC(O)C1)c1c(C)cccc1 N1(C(C(C(C)OC)NC(c2cnc(O)cc2C)=O)=O)CC(C)(C)C2COCC12 c1(C(=O)NC2C(CNC(C3C(CC)OCC3)=O)C2)ccc(F)c(O)c1F C1(C2CC2)(C(=O)NC(C)C(=O)NCCC(=O)N2CCCC2)CC1 c1(C(=O)NC2CC(C)(CNC(C3C=CCC3)=O)C2)cc2c(nc1N)CCCC2 N1(C(C2=CCCC2(C)C)=O)CCOC2(CCCN(C(C3(C)CCOC3)=O)C2)C1 C1(CC)CN(C(c2cc(SC)c(C)s2)=O)CCN1C(=O)Cc1ccc(O)c(Cl)c1 c1(C(=O)NCC(C2CCC2)NC(=O)Cn2nccn2)cc(F)c(F)cc1Br N1(Cc2ccc(OCC)cc2O)CCC2(CCN(C(c3cc(C)no3)=O)C2)C1 C1(C(=O)NCC2(OCC)CC2)CN(C(C2CCOC2(C)C)=O)CC12CC2 C(=O)(C(C)(C)CC(C)C)NC1CCCC(C(N2CC(OC)CC2(C)C)=O)C1 C1(NC(Cc2c(C)ccc(F)c2)=O)CCCN(C(c2nc(C)n(C)n2)=O)CCC1 c1(-n2c(-c3nc(CC)sc3)nc(-c3ccc(Cl)s3)n2)ccc(S(N)(=O)=O)cc1 C1(NC(=O)CC2CC(C3CC3)C2)(CO)CCCN(C(=O)CS)C1.c1ccncc1 c1(N2CCC(CC)(CO)C2)ncnc(NCCCCCCC2CC2)c1C N1(C(c2cc(C)cc(Cl)c2)=O)CC2CCN(C(=O)C(C)NC(N)=O)C2C1 C1(OCC)CC2(C1)CC2.C1(C)(C=O)CCN(C(c2c[nH]c(=S)cn2)=O)C1.N C1CCC2(CC1)CC(O)C2.n1(CC(=O)N(C(C)C)CCNC)ccc(=N)[nH]1.C C1(NC(C(CC)C(C)C)=O)CCCOC12CCN(C(c1ocnc1C)=O)CC2 N1(C(c2cc(C)sn2)=O)CCN(C2CCN(C(C3CC4CCC34)=O)CC2)CC1 C1(NC(c2c(C)n(C)nc2)=O)C2CC3C(C2)C13C(=O)N(CCCO)CCO C=CC1CCCN1C(c1cc(CNC(C2COCCC2C)=O)on1)=O c1(C=O)ccccc1F.N#CC1(C(=O)NCC2CCCC2)CCC1.C(=O)(C)N c1(C(N2C(C(=O)Nc3ccc(C)cc3CO)CSCC2)=O)cccc2ccnn12 N1(C(CSC(C)C)=O)CCN(C(C2CC(N(C)C)C2)=O)CC1c1ccc(F)cc1 C=CCCCCN=c1cccc(S(=O)(=O)NC(C)C(CO)SC)[nH]1 c1(CC)cc(C(=O)NC2COCCN(C(c3ccc(N)cc3Cl)=O)C2)c(C)nn1 CC(c1cnn(C)c1)=CC(=O)NCC1CN(C(C2CC(C)(O)C2)=O)CCO1 N1(C(CC(CC)C2CCC2)=O)CCCC(C2CC2NC(=O)COC2CCOC2)C1 C#CC1(C(=O)NCC2(O)CCCC2C)CCN(C(c2ccc(C)cc2)=O)CC1 C(=O)(CC(C)SC)NC(C(N1C(CC)CC1)=O)c1ccoc1 c1(C(=O)NCC(C(C(C)C)O)(C)C)nc(Br)c2c(F)cccn12 N1(C(c2ncn(C)c2)=O)CCc2nn(C)c(C)c2C1.N(CP(=O)(O)O)CC(=O)N CC(CS(C)=O)N(C(=O)C=CCN(C)C(c1cnn[nH]1)=O)C Cc1ccc(CN2CC3C(C2)N3C(=O)CSc2ccccc2)cc1O N1(C(c2ccn(CCOC)n2)=O)CCC(CF)(NC(C2(C)CCSCC2)=O)C1 CCCC(CCC)C(=O)NC1CS(=O)(=O)CC1NC(c1cc(CCO)on1)=O C1(NC(CC(CCC)O)=O)CCC2CN(C(=O)CCCCCC#N)CC2C1 CC(=O)CCCCC(=O)N1CC=C(C(=O)Nc2cnsc2)CC1 C(=O)(CC(C)(C)C(=O)N1CCC1C)OCC.c1(C=O)ccnc(C(F)F)c1 C(=O)(CCCN=c1nccc[nH]1)NCC(CNC(c1ccc(C)nc1C)=O)(C)C Nc1cc(N2CC(O)CC2C(N2CCN(C(c3ccc(Cl)o3)=O)CC2)=O)ncn1 c1(NS(C)(=O)=O)cc(C(F)(F)F)ccc1F.C12(C)CCC(CC1)NC(=O)N2 C12(CCC(=O)NC(C)CNC(C3CCC(=O)C3)=O)CCC(CC1)C2 C(CCSC)(C(=O)NCC(C)N(C(=O)Cn1nccn1)C)NS(CC)(=O)=O C1(CC(=O)N(CC(=O)NC2CN(CC)C2)CCC)CC(O)C1(C)C C(CC(C)(C)CC(=O)N1CC(CC(C)(C)C)C1)OC.c1(C(=O)N)ccc(C)cc1F c1(CC)nccc(=NC2CCCCC2NC(=O)Cc2c(C)cccc2C)[nH]1 C1(CC=O)CCS(=O)(=O)CC1.Cc1cnc(C(=O)NC(C)C2CCC2)nc1.N c1(C(N2CC(N(C(c3c(C)cc(Br)cc3)=O)C)C2)=O)cc(F)c(F)c(F)c1 C1(N(C(C2C(=O)NCC2)=O)CCO)CCN(C(=O)CSc2cccc(F)c2)CC1 N1(C(CCC(=O)OCC)=O)CC(NC(=O)CCC(=O)N(C)C)C2(CC2)C1 C(=O)(C(F)CC(C)(C)NC(=O)CCC1CC1)NCCOC(CC)(C)C.O C(C1CCOC1)=CC(N1C(CC(=O)NCC(CO)C2CCC2)CC1)=O C1(O)(CCNC(C2C(OCC)C2)=O)CCN(C(=O)CCCn2cccc2)C1 C(=O)(N=c1cc2ccccn2[nH]1)C1CCN(C(CCCCC(C)(C)C)=O)C1 N1(C(COC(C)C)=O)CC(NC(=O)C(O)CC2CC2)C2(CC2)C1 C1(C(N2CC(CCNC(C3CC3(C)C)=O)(OC)C2)=O)CC=C(C)CC1 C12(NC(c3scc(C)c3C)=O)CCC(C1)N(C(c1ccncc1)=O)C2 c1(CC(=O)NC2CC(C)(NC(CN3CC(C)(OC)C3)=O)C2)cccnc1C c1(CN(CCCC)C)ccc(S(=O)(=O)NC2(C)CCOC2C2CC2)c(Cl)c1 c1(C(=O)N)c(N)cccc1F.c1(OCC)cc(C(=O)NCC2CCC2)sn1 CCCC(C(=O)OC)C(=O)NCC1CC(NC(c2cccnc2O)=O)C1 N1(c2ccc(S(=O)(=O)N3CCN(C)CC3)cc2F)CCC2(CC1)SCC(=O)N2C C1(C)(CC)CCC(C(=O)NCC(C)NC(=O)C=Cc2ncc[nH]2)O1 c1(CC(=O)NCCN(C(C(c2c(C)noc2C)CC)=O)CC)ccc(Cl)cc1 Cc1cc(C#N)cc(C(=O)NC2CC(CNC(=O)CCC=CBr)C2)n1 C1(CN2CCCC(c3c(C(=O)OCC)cn(C)n3)C2)CC(=O)c2ccccc2O1 c1(C(=O)NCCNC(C2CCC2F)=O)ccc(C(=O)NCCO)cc1 N1(CC)CCN(CC(=O)NCC2CCCCO2)CC1.C(=O)C(C)CC1CCC1.N c1(C(=O)NC2C(NC(c3n(C)nnc3)=O)CCCC2)coc2c1C(O)CCC2 Cc1nc(O)ccc1C(=O)NC(C1CCN(C(=O)CC2CCCC(C)C2)C1)C N1(C(c2nc(C)sc2)=O)CCC(O)(CN(C(=O)Cn2cccnc2=O)C)C1 N1(C(C2C(C(C)C)=NO2)=O)CCN(C(=O)CCC(N)=O)C(CC(F)(F)F)C1 c1(NC(C2CN(C(C(C(C)C)=O)=O)CC(F)(F)C2)=O)ncc2ccc(Br)cc2n1 C1(CC)CN(Cc2ccnc(OCC(F)(F)F)c2)c2cccc(Cl)c2O1 c1(OC)cnnc(C(=O)NCC2(O)CCN(C(C3CC3C(C)C)=O)C2)c1 N1(C(C=CCC)=O)C2CCCC1CC(NC(c1ccc(-c3ccco3)o1)=O)C2 c1(C(N(c2ccccn2)C)=O)cn2c(n1)CCC(N)C2.C1CCOCC1 C(=O)(C(=O)N=S(C)(C)=O)NCCC1(NC(CC(C(C)C)O)=O)CCC1 O=C(CCC(=O)NC(=O)N(C1CCCOC1)C1CC1)NC.c1ncco1.CC CCCC(C)CCNC(=O)COC1CN(C(C2CCCN2CC)=O)C1 CC1CC(CCNC(=O)CC2(NC(c3cc(CO)ccn3)=O)CC2)CCO1 Cc1ccc(Cl)cc1OCC(=O)NCCCNC(C1(CN(C)C)CC1)=O C1(CNC(CCN(C(C2(SC)CC(=O)C2)=O)C)=O)CCCCC1CO N1(C(C(CCCC)C)=O)CCCCC12CC(NC(=O)CC1CNC(=O)C1)C2 C=CCC(C(=O)N1CCOC(CC(=O)NCC2(C)CC2(F)F)C1)NC(C)=O c1(C(N2CC(CNC(c3c(C)[nH]cc3)=O)C2)=O)cccc(-n2cccn2)n1 Cc1cccc2c(C(=O)NCC(C)(F)CNC(c3cc(Cl)n[nH]3)=O)coc12 N1(C(C(CC#C)(C)NC(=O)C=Cc2ccnn2C)=O)C2CCC1CN(C)C2 c1(C(CC)C)cccc(NC(=O)CNC2CCC(N3C(=O)CCC3=O)CC2)c1 N1(c2ncc(OC)cn2)CCC(NC(c2cc(F)cc(Br)c2)=O)C(C)(C)C1 C(CCCC(=O)N1CC(C)(COC)C1)NC(c1cn(CC)nn1)=O C1(CC)C(NC(=O)CCOCCOC)CCN1C(c1nccn1CC)=O Cc1ccc(CC(=O)NCC2CN(C(=O)Cc3ncccc3C)CCO2)c(F)c1 N1(C(C2(COC)CCC(=O)N2)=O)CC2CC1CN(C(=O)Cc1cscc1)C2.O c1(C(N(CC(C)(C)C)C)=O)cccc([N+](=O)[O-])c1N.c1(CC)cc(C=O)no1.N c1(C(=O)NCC(C)(C)OCCNC(C2CC=CCO2)=O)cccc(C#N)c1 C(=O)(C(O)CCC(C)C)N1CCC(NC(c2c(C)n[nH]c2)=O)C(C(N)=O)C1 c1(-c2nc(-c3occ(C)c3C)on2)c(Cl)nc(Cl)n1C N1(C(c2cnc(CC)[nH]2)=O)CC(NC(C2CC(C)(C)C2)=O)C2(CCOCC2)C1 C1(NC(C(C=C)(F)F)=O)COC2(C1)CN(C(c1ccc(N)cn1)=O)C2 c1(C=O)cc(N)cc(O)n1.c1(N(C)C)ccc(C(=O)NCCC2CC2)cc1.C C(CCCC(=O)N)N(C(C)=O)C.C1(CC)CCCN1C(=O)C(CN(C)C)N(C)C N#Cc1cnn2cc(C(=O)NCC3C=CCN3C(=O)C=CC3CCCC3)cnc12 N1(CCCC(C)(F)F)CC(C2CC2)C1C1CC1 C1(C(N2C(CCCNC(c3c(C)sc(Cl)n3)=O)CCC2)=O)CCCCS1(=O)=O N1(C(c2cc(C(F)(F)F)ccn2)=O)CCN(C(C2CCCO2)=O)CC(O)C1 c1(C(=O)NC(CC=C)CNC(=O)C(O)C2CCC2)cc2cccnn2c1 O=C(C1=CCCN(Cc2nccnc2Cl)C1)Nc1cc(F)c(I)c(F)c1 C(=O)(C(O)CC(C)(C)C)N1CC(F)(C(=O)NC(c2ccccn2)CC)C1 C1(CC(=O)N(CCCCCNC(c2c(C)snc2)=O)C(C)C)CCCC1(F)F Cc1ccccc1C(F)(F)C(=O)NC1CC1NC(C1(C#N)CC1)=O c1(OC)nccc(N2CC(CN(S(=O)(=O)Cc3cccc(Cl)c3)C)C2)n1 Cc1cccc2[nH]c(=NC(C)C3CN(C(c4ccc(Br)o4)=O)CCO3)oc12 N1(C(C2(C(=O)NC)CC2)=O)CC=C(C)CC1.c1(C=O)cc(C2CCOC2)[nH]n1 c1(C(=O)NC2(CC(N3CC=C(COC)CC3)=O)CC2)cccc2occc12 C1(CNC(=O)CC2=CCCC2)CCC2CN(C(c3cc(O)ncc3F)=O)CC12 N1(C(c2cc(C)nn2C)=O)CC(CNC(=O)CCN)CCC1C.[SH](C)(=O)=O C1(CNC(Cc2c(C)nc[nH]2)=O)CCC(C)N(C(=O)Cc2cncs2)C1 CCCCCCCC(F)C(=O)NCC1CCN1C(c1ccc(CC)cc1)=O N1(C(Cc2cc(CC)no2)=O)CC(O)CC1C(=O)Nc1cccc(OC)n1 Cc1cc(Cl)c(C(=O)NC2COC3(C2)CN(CCC2CCOCC2)C3)cc1C C1(C(C)C(=O)N(C2CC(O)C2)C)CCN(C(=O)Cn2cc(C3CC3)cn2)CC1 c1(C(=O)NC(CNC(c2cncc(C(C)=O)c2)=O)C)c(C)nc(C)n1O c1(C(=O)NC(CN(C(C(C)Sc2ccc(C)cc2)=O)C)C)c(F)cc(F)cc1F c1(OC)c(C(N2CC3(C2)CN(C(=O)CSS(C)(=O)=O)C3)=O)c(C)nn1C C1(CNC(CNC(=O)NC)=O)CCC(C(N2CCC3CC23)=O)CC1 N1(C(C2N(C(C)=O)CSC2)=O)CC2(CCC2)CC1CNC(c1ncc[nH]1)=O C1(OCC)CC(NC(c2ncccc2C)c2nnnn2C(C)C)C12CCCCC2 O=C(C1=CCCSC1)N1CC(C(F)Cn2cc(-c3ccncc3)nn2)C1 C(=O)(CCCCC(F)(F)F)NC(C1CCCN(C(c2cocn2)=O)C1)C c1(NC(CC)C)[nH]c(=NC2CC(Sc3ccccc3)C2)nc2scnc12 N1(C(c2cscc2Br)C(=O)NCC=C)CCC(C2CCOCC2)C1 c1(C=O)cncc2c1CCC2.C(=O)(C(F)(F)c1cncs1)N(CCOC)CC.N C(CC(C)(C)NC(=O)CC)=CC(N1CC(N(C)CC)C1)=O.C(=O)CO.N Cc1ccc(C(C)NCCC(C)S(C)(=O)=O)cc1F C(=O)(NN1CCCC1C(=O)NC1CN(C)NC1=O)c1c(C)ocn1 Cc1sc(C(N2CCCC(CNC(c3coc(Br)c3)=O)C2)=O)nc1O Cc1cc(C(=O)NCC2(NC(c3ccc(-n4cccn4)cc3)=O)CC2)[nH]c1C C1(CN(C)C(C2(C)CCCC2O)=O)CCC(C)CC1.c1(C=O)c[nH]c(=N)s1.N C1(NC(c2c(C)coc2)=O)CC2CC(C1)N(C(c1nccc3c[nH]nc13)=O)C2 CN1C(=O)C(C)(C)c2cc(C=O)ccc21.C1(C=O)C2CCCC12.CC=CC.N C1(N(C(=O)Cn2cnnc2)C)CN(C(=O)CC(C)(C)C)CC12CC2 C(=O)(C(C)C(F)(F)C(F)F)NCC1N(C(c2c(C)sc(O)n2)=O)CCCC1 c1(C=O)ccccc1.c1(OCC)cncc(NC(C2CCCC2)=O)c1.C(C)=O N1(C(c2cncc(SC)c2)=O)CC2CC(NC(=O)C(C(C)C)O)C1C2.CC(C)C C(C(O)C(=O)NCC1CCC1C(=O)NC(CO)C(N)=O)=CC c1(C=O)cc(F)ccc1-n1cccn1.C(C(=O)NCC1CC1)SCC#C.N C1(CNC(C=C(CCC)C)=O)CCOC1C(=O)NCc1ccon1 C1(NC(c2n(C)ncc2Br)=O)C2CCN(C(=O)CN3CCCC3)CCC12 c1(C(=O)NCC2C(NC(c3cc(C)oc3)=O)CCCC2)cc2cccc(F)c2s1 N1(C(c2n(C)cnc2)=O)CCCC2CN(C(c3ccc(O)c(N)n3)=O)CCC12 CCC(F)(F)C(=O)NCc1ccc(CCNC(=O)CCCn2cccn2)cc1 Cc1cc(F)cc(CNC2CC2C(N2CCOCC2c2ccccc2)=O)c1O C1(CNC(C=C(C)C)=O)CCCN1C(C1CS(=O)C1)=O c1(C(=O)NC(C)CCCNC(C2C=CCS2)=O)cc(F)cc(F)c1N c1(C(=O)NC(C(CO)NC(Cc2nc(C)[nH]n2)=O)C)ccc(C)c2cccnc12 CN1CC(=O)N(CC(=O)N)C1=O.C1CC(C)(C)CN1C(=O)CC.CC(N)=O.C c1(CC(=O)NCC(CNC(CCOCC#C)=O)O)c(Cl)cc(Cl)cc1Cl Cc1oc(C#N)cc1C(=O)NCC(C)N(C)C(C1CCC1c1nc[nH]n1)=O N1(C(CCC(N)=O)=O)CCN(C(c2cc(-c3ccncc3)[nH]n2)=O)C2CCC12 c1(NC(C2C3CN(C(CC(CC)O)=O)CC32)=O)ccc(F)c(F)c1 C1(CNC(CN(CC)CC)=O)CCCCCN1C(c1cc(CO)oc1C)=O C#Cc1ccc(C(N2CC3CC3(NC(c3cc(SC)cc(SC)c3)=O)C2)=O)nc1 CC1CN(C(C2CCCN2C(C2CC2c2ccccc2)=O)=O)CC(=O)N1 CN1CCCC(F)(C(=O)NCC(C)(C2CCC2)NC(=O)CS)C1.c1nncs1 c1(C(N2CCN(C(c3nc(CC)oc3)=O)C3C2C3)=O)cnc(O)n(C)c1=O C(=O)(C1=Cc2ccccc2OC1C(F)F)OCC(=O)Nc1cccnc1 CC1CC(NC(c2coc(CNC(c3cccnn3)=O)c2)=O)C(C)CN1C c1(C(N2CCN(C(C3C(=C)C3)=O)C(C)CC2)=O)c(C)oc2ccc(OC)cc12 C(CCC(=O)N1CCC(CCO)C1)C1(NC(C2CCS2(=O)=O)=O)CCC1 C1CCC2(CC1)CC2.Cc1cc(CC(=O)NC(Cc2cnc[nH]2)C(=O)NC)on1 C1(NC(C(C2CCN(C(c3cc(C)n(C)c3)=O)C2)C)=O)CNC(=O)C12CC2 C1(C(n2cc(CC3CCN(C(=O)C(O)c4ccsc4)C3)nn2)C)COCCO1 N1(CCCNC(C2(C)CC(F)C2)=O)CCN(C(C2(C)COCCO2)=O)CC1 Nc1cc(F)c(CC(=O)NCC2CC2)cc1F.c1(C(=O)N)cnc(C2CC2)s1 c1(C(=O)NCC2N(C(C(C)NC=O)=O)CCC2)ccccc1N1CCOCC1 C1(c2cn(CCOCC)nn2)CN(C(c2ccnn2CCC(F)(F)F)=O)CCO1 C1(C(C)C)CCC(C(N2CCN(C(=O)CSc3ccccn3)CC2)=O)CC1 c1(C=O)cc([N+](=O)[O-])c[nH]1.C1(OCC)CCC(C(=O)O)CC1.C(CC)C(C)C CC1(C)CC(CNC(c2ncc(F)cn2)=O)CN1C(C1CCC(O)CC1)=O c1(C(=O)NCC(CN(C(CCC(=O)OCC)=O)C)C)cc2cc(O)cnc2[nH]1 Cc1nc(C(=O)NCCOC2CCN(C(=O)C(CO)N(C)C)C2)[nH]c1C Cc1c(C(=O)NCC(F)C)nn2ccccc12.n1(CC(=O)N)nnc(C(C)C)n1 N1(C(C(C)=CC=C)=O)CC(C)C1C(=O)N(C)CCNC(C)=O C1(C2N(C(c3nc(CC)oc3)=O)CCCC2)CCC(=O)NC1=O C(=O)(C1CCCc2cncn21)NCC1CC(NC(C2CCN(C(C)=O)CC2)=O)C1 N1(C(CCSC)=O)CCC(N=c2[nH]c(C3CC3)nc3[nH]ccc23)C(C)C1 Cc1c(C(=O)NCC2CCCC2)[nH]c2c1CCCC2.C1(C(=O)N)COC(C)(C)C1 C1(NC(C2CCN(CC(C)C)C2)=O)CCCCCC1NC(c1cnc[nH]c1=N)=O C1(C(N(CC#C)CC)=O)(OC)CCN(C(=O)CC2CC(=O)C2)C1 C1(C(=O)NCC2(CSC)CC2)(OC)CCN(C(C2CC23CCC3)=O)C1 CCCCC(C(=O)NC(c1ccccc1)C(N1CCC2CC1C(=O)O2)=O)C(C)C c1(C(N2CC(CNC(C3(OC)CCSC3)=O)OCC2)=O)ccnn2ccnc12 Cc1nc(C)c(C(C(=O)NC2(C)CC2)N(C2CCC(C)(C)C2)C)nc1C C(CC(C(=O)NCC#CC(F)(F)F)NC(=O)CCc1ccc[nH]1)SC c1(NC(C2N(C(C(=Cc3cn[nH]c3)C)=O)CC=C2)=O)ccc(C)nc1O C(=O)(C(C)(C)CCC#N)NC1CCN(C(COCc2cccc(C)c2)=O)C1 S(=O)(=O)(c1ccc2c(c1)CC(C)O2)N1CCCC(C(=O)OC)C1.C(C)(C)(C)O C12CC(CO1)C2.C1(C=O)CCCCC1.c1(C(=O)NC)ccc(C(F)(F)F)[nH]1 N1(CC(=O)NCC2COc3ccccc3O2)Cc2cc(Cl)ccc2C(C(=O)O)C1 c1(C(N2CC(CN(C(=O)CC(F)F)C)OCC2)=O)cc(N)c(Cl)c(O)c1 Cc1cc(C)c(C(=O)N)c(=O)o1.C(=O)(C(C)CC(C)(F)F)N1CCCC(C)C1.C C1(NC(CSCCCC)=O)CN(C(=O)CN(C)CCO)CC1CCC N(C1c2ccccc2CC1O)C(c1ccnc(OC(F)F)c1)=O N1(C(c2c(C)snn2)=O)CCC2(COC(CNC(=O)CC=C(Cl)Cl)C2)C1 C1(NC(c2ccc(CC)cc2)=O)CN(C(c2coc(CO)c2)=O)C2(CCOC2)C1 C=CCC(C)(CC)C(=O)N(C)CC=CC(N1CC2CC2C1)=O C(=O)(CCC(F)(F)C(F)(F)F)NC(CNC(COCC(=C)C)=O)(C)CC c1(CC)cc(N2CCCC2CN(C)C(c2cncc(C)c2)=O)nc(CC)n1 Cn1cc(S(C)(=O)=O)c(C(=O)NCCNC(C2(C)CCCCNC2=O)=O)n1 C1(c2cn(C(C)C(=O)O)nn2)CCCN(C(c2ccn(-c3ccncc3)n2)=O)C1 C(=O)(C1CCCc2ccnn21)N(CCCNC(C1CC1C1CCC1)=O)C CCCCC(CC)C(=O)N1CCC(O)(CNC(=O)CC2NC(=O)CNC2=O)CC1 c1(CC)ncc(C(=O)NOCC(=O)N(CC(C)C)CCO)s1 CS(=O)(=O)c1ncc(C(N2CC(CCn3cc(C4CCCCC4O)nn3)C2)=O)s1 c1(C(N2CCCC(NC(c3ccc(SC)o3)=O)CC2)=O)ccnc2ncccc12 CC(C)CC(C(=O)NCC1CN(C(=O)CC2CC(F)(F)C2)CC1O)N(C)C CC(C(=O)NC(C)(C)CO)C(C)(F)F.c1(C=O)ccc(F)cc1.C(=O)CC.N c1(OC)cccc2c1C(C(=O)NC1CC(NC(C3CC4CC4C3)=O)C1)CC2 C1(NC(c2cc(SC)ccc2)=O)CN(C(=O)CCF)CC(F)(F)C1.C(C)(=O)N Cc1c(CNC(=O)N(C)CC2CCCC3CC23)cccc1Cl C1(S)(CO)CCC1.C1(C2N(C(=O)CC3CC3)CC2)CC(F)(F)C1 C1(NC(CN(C(COC)=O)C)=O)CN(C(=O)CC(F)F)C2CC12 Cc1cc(C)n(C(C)C(=O)NC2CC(NC(=O)CC(C)F)C(O)C2)n1 CC(O)(CC(=O)N1CCCC1CCc1cn(C2CCCC2)nn1)C(F)(F)F N#Cc1cc(F)ccc1COC(c1cc(Br)c(N)c(Br)c1)=O C1(C(C)(C)C(=O)NCCCC2CCOC2=O)CCCN(C(C2COC(=O)N2)=O)C1 c1(OC)cc(NC(=O)COCCNC(C2CCCSC2C)=O)ccc1O Cc1ccc(Cl)c(O)c1C(N1CC2CC(NC(=O)CC(C)N(C)C)CC1C2)=O Cc1noc(C(=O)N(CCNC(=O)CC(F)(F)c2ccccc2)C2CC2)c1C c1(CNC(NCC)=S)cnc(-c2cn(CCN3CCCCC3)nn2)nc1 C(=O)(C1CCOc2ccccc21)NCC(C(C)(C)C)NC(C1CCCCC1O)=O CC(C)CC(C(=O)NC1CN(C(=O)Cc2csc(-c3ccccc3)n2)C1)N(C)C Cc1cccc2c1ccn2CC(N1CC2CC1CCN2C(=O)Cc1cc[nH]n1)=O O=C(C#CC1CCC1)NC12CCOC(C)(C1)C2.C1(C(=O)N)CCS(=O)(=O)C1 C1(N(C(C2CN(c3n(C)nnn3)C2)=O)CC)CN(C(=O)C=CS(C)=O)CC12CC2 Cc1cccc(Br)c1C(N1CC(NC(C2CC(C(C)C)=NO2)=O)C1)=O C1(C(=O)NCCCNC(C2CCC(N(C)C)CC2)=O)CCc2nc(O)[nH]c2C1 N1(C(c2scc(CNC(C=C(COC)C)=O)c2)=O)CCC(C)(N(C)C)C1 c1(-c2cccc(OCC)c2O)cnn2cc(C(=O)Nc3cncnc3Br)cnc12 Cc1[nH]nc(Cl)c1C(N1CC2C(C)C2C1)=O.c1(C=O)ccccn1.C(=O)(C)N C1(C(N(CC(=O)Nc2cc(C(CC)C)no2)C)C)Cc2ccccc2O1 N1(C(C(CC)=O)=O)CCC(NC(c2cncc(O)c2)=O)C(F)C1 CCC(CNC(=NCc1ccnn1C)NC1COC(C)C1)(CC)N(C)C CC(C)CC(O)C(=O)NCCN1CCC(NC(=O)COc2ccccc2F)CC1 C=CCCC(C(=O)NCCCOC(=O)NC)NC(=O)CCn1cnnn1 C1CN(C(c2cnc(C)c(C#N)c2)=O)CC2(CC2)C1.C1(CC#C)(C=O)CCC1.N C=Cc1cncc(C(=O)NCC2CN(C(c3csc(SC)n3)=O)CC23CC3)c1 N=c1nc2c(c[nH]1)CC(Nc1ncnc3c1nnn3-c1ccccc1)CC2 CC(C)C(C(=O)c1ccccc1)NC(c1cn(C)nc1O)=O c1(C(=O)NC2C(C)CN(C(COCCC#C)=O)CC2C)cc(C)c2[nH]nnc2c1 O=C1CC2(CCOC2)C(C(=O)NC2(CCC)CC2)CN1.n1(CC=O)ncnn1.N c1(OC)ncc(C(=O)NCC2(O)CCN(C(=O)CC(C)C(F)F)C2)c(C)n1 C1(N(C(C2CC(SC)C2)=O)C)CCC2CN(C(c3cc(C(F)F)ccn3)=O)CC12 Cc1cc(C(N2CC(NC(C3CC(C)(C)CCO3)=O)C(CO)C2)=O)cc(C)c1 N1(C(C(Cn2ccc(C)n2)C)=O)CCC2(CCCN(c3nnc(C(N)=O)s3)C2)C1 C1(OC)CC(O)CN(C(=O)C=CCN(C)C(c2sccc2C#N)=O)C1 C1(O)(CNC(C(C)=CC2CC2)=O)CCCN(C(c2ccccc2C)=O)C1 Cc1cc(=NCC2(O)CCCN(C(c3c(Cl)ccnc3F)=O)C2)[nH]c(C)c1C#N C1(NC(c2c(OC)scc2)=O)CCN(C(=O)Cc2ccnn2C)C(C2CC2)C1 N1(C(C(COC)O)=O)CCC2CN(C(C3(CF)CC(=O)C3)=O)CC2C1 CC1(C)OCCC1CC(=O)NCCC.C1(CC=O)CCCC(=O)C1.CC(C)C.O CCCC(O)CC(=O)NC1C2CC1N(C(=O)COCc1ccccn1)C2 c1(C(C)OC)ccc(C(C(=O)NCC(C)C)N(CC=O)C)cc1.C(C)(C)C.N c1(CCC(=O)NCCCNC(=O)COCC2CCCOC2)c[nH]c2ccccc12 C1(CNS(CC2(COC)CCC2)(=O)=O)CCC12CCCO2 c1(NC(C2(COC)CC2)=O)ccc2cn(C)nc2c1.N12CCC(O)C(C1)C2=O c1(C(N(C)CC2CN(C(C(C(C)C)O)=O)CC23CC3)=O)nc2cnccc2s1 c1(C(=O)NCC2N(C(CSCC(N)=O)=O)CC=C2)cc2cnccc2o1 CCCCCC(CCCCC)NC(=O)NCCc1ccc(S(N)(=O)=O)s1 C1(C(=O)NC(C)CN=[N+]=[N-])(CO)CCN(C(=O)CN2CSCC2=O)C1 c1(OCC(=O)N(C2CCC(NC(c3cc(C)oc3)=O)C2)C)ccc(F)c(C)c1 c1(NC(=O)NC(CC(C)=O)C)cn2cccc(Br)c2n1 Cc1c(Br)ccc(C(=O)N(C2CCN(Cc3ccccc3)C2=O)C)c1F N1(C(c2cc(C(C)C)on2)C(=O)NCC=C)CCOCC(C)(O)C1 CCCCCCCCCCC(=O)NC1CN(Cc2ccnc(C)n2)CCC1C Cc1occc(=O)c1OCC(=O)NC(c1cccc(C(F)(F)C(F)(F)F)c1)=O O=C(C1=CCN(C(C2CC3(CCC3O)C2)=O)CC1)NC1COCCC1(F)F c1(OC)cc(C)c(Br)cc1C(=O)NC(C1(O)CCN(C(=O)CSC)C1)C c12ccccc1C1CC1C(=O)NCC2.C(=O)C=CC=O.C1CC1.CC NS(=O)(=O)c1cnn(CC(=O)N)c1.C12CCC(CC1)C2.C1(C=O)CCC(=O)O1 Cc1coc(C(=O)NOCC(=O)NCC(O)C(C)C)c1 C(CC(C)(C)C)(C(=O)NCC1CCCCC1)OC.c1(C=O)c[nH]nc1[N+](=O)[O-].N c1(C=O)cc(F)n(C)n1.C1(C(N2CC(COC)(C)C2)=O)CN(C)CCO1.N C1(C(=O)NCCc2nccc(C)n2)CCCCCN1C(=O)CSC1CC1 C1(C)(CNC(c2nc(C)oc2)=O)CCCC1NC(=O)CC1CCCSC1 C1(NC(=O)CCC2CCC(O)CC2)CN(C(=O)COC2CCC2)CC1C1CC1 C1(NC(c2c(C)cnn2C)=O)CC(C)CN(C(=O)COCc2ccccn2)C1 N1(C(CNC(CC(C)C)=O)=O)CCC(F)(C(=O)NCC2(C)CCC2)C1 C1(NC(C=NOC)=O)CN(C(=O)C(C)(C)COCC(F)F)CCC1O N1(c2nnc(C)o2)CC(C)CN(C(C2(C)CC(C)C2)=O)CC1C c1(OCC)c(Cl)cc(C(=O)NC(=O)CC2CNCCO2)cc1Cl.c1ccc[nH]1.C Cc1cc(F)ccc1C(=O)NC1CC=C(C(=O)NC(c2nccs2)C)C1 CN=c1nc(C(=O)NCC(C)CNC(c2csc(Br)n2)=O)cc(C)[nH]1 c1(C(N2CC(NC(CCSCCC)=O)C(C)CC2)=O)cc2c(nc1O)CCCC2 Cc1ccn(CCC(=O)NC(Cc2ccoc2)C(=O)NCCN(C)C)n1 C1(C)(C(=O)NC2CN(C(C)=O)C2)CCCN(C(=O)CP(C)(C)=O)C1 C1(OC)C=CC(C(=O)NCC(C)N(C(=O)COCCO)C2CC2)C1 O=S(=O)(c1cccc(=NCCCOC2CCOCC2)[nH]1)NC1C2COCC12 C1(C(N(CCCO)CC)=O)CC12CCN(C(c1cc(OC)n(C)n1)=O)C2 C1(C(N(C)C)=O)CCN(C)C(=O)C1.N1(C(C2(CC#C)CCCC2)=O)CCCCC1 C1(CNC(C2(SC)CCC2)=O)CN(C(C2CC3(C2)CC3F)=O)C(C)(C)C1 C(CC(=O)O)(CC(C)C)NC=O.c1(CC(=O)NC)ccccc1Br.C(C)(C)C C1(C(=O)OC)CN(C(=O)CS(=O)(=O)N2CCN(C)CC2)CCS1 C1(O)(CCNC(c2nc(Cl)cs2)=O)CCN(C(C2CC3(CC3)C2)=O)C1 Cc1c([N+](=O)[O-])c(C(=O)NC2CC(Cn3ccnn3)C2)nn1C C1(CC(=O)NC23C(CN(C(CCCCNC(N)=O)=O)C2)C3)CCC(F)(F)CO1 N1(CC)CCC(C(=O)NC(C)(C)CC(=O)NCC2(CCO)CCC2)CC1 C1(C)CC(F)(F)CN1C(=O)C.CC(C)C(C)(O)C(=O)N.c1n[nH]c(=N)s1.C CC(C)C(CN(C(=O)CCCCN(C)C)C)C(C)C C(=O)(C1=NOC2(CCOC2)C1)N1CCC(O)(CNC(=O)COCCF)CC1 C#Cc1ccc(CC(=O)N(C)CC2CCCN(C(=O)C3=CCCC3C)C2)cc1 C1(CC(=O)N)CCCCCC1(F)F.Cc1cc(F)cnc1C(=O)NCC1CCC1 C(C(C)(CO)OC)NCC(c1ccccc1)OC CN1CCN(C(=O)C=Cc2nccs2)C(C)C1.c1(C(=O)N)nn(C(F)F)cc1Cl C(=O)(C(C)C(CC)CC)N1CC(CC=C)(NC(C2COCCO2)=O)C1 c1(C(N(C2CCC(NC(=O)Cn3cncn3)CC2)C)=O)onc2ccccc12 N1(CCCN(CCCNC(=O)CC2CC(F)(F)C2)CC)CC(=O)NC1=O C1(OC)CCCC(c2nnnn2CN)(NCc2ncn(-c3ccccc3)n2)CC1 N1(C(c2ccc([N+](=O)[O-])[nH]2)=O)CCCCC(C2CN(C(c3nncs3)=O)C2)C1 CCC(C)(C)C(N)=O.C(c1ccc(C)o1)=CC=O.c1(CC(=O)N)cccnc1 S(=O)(=O)(c1ccc(Cl)cc1)NCCC(=O)NC1CN(C(CCC#C)=O)C2C1C2 Cc1cnn(C)c1S(=O)(=O)NC(c1nc(C(C)(C)C)no1)C N#Cc1cc(C(=O)NCc2ccccc2CS(N)(=O)=O)ccc1C1CC1 C1(CC(N2CC(C(N3CC(CN(C)C)C3)=O)(CC)C2)=O)CCC(=O)C1C CC(C)CCCC(C)C(=O)N1CC(NC(c2ccc3ccoc3c2)=O)CC(F)C1 N1(C(=O)Cc2cccc(F)c2)CCN(Cc2ccc(O)cc2Br)CC1C(F)(F)F c1(C(=O)OCc2ccc3nonc3c2)cc(O)c(F)c(F)c1F N1(C(C2(C)CC2)=O)C2CCC(C(=O)NCCCO)C1CC2 N1(C(c2c(C)nc(=N)[nH]c2C)=O)CC2ON=C(C)C2C1.c1(CC(=O)N)ccns1 C1(C(=O)NCCCN(C(C(C)Cc2ccco2)=O)C)CCCCN(C)C1=O c1(C(N2CC(CNC(C(CC)C#N)=O)C(C)C2)=O)cc2cccc(C)c2s1 S(=O)(=O)(c1cc[nH]n1)N(CC(C)C(=O)OC(C)(C)C)CC1CC1 c1(C(N2CCC(NC(c3ccc(O)cn3)=O)C(CO)C2)=O)nc2c(s1)COCC2 c1(N(CCN(C)CCO)C)nc2ccsc2c(=NCC2CC(O)C2)[nH]1 c1(CC(=O)NCC2(NC(CC3N(C)CCOC3)=O)CC2)ccc2ncsc2c1 c1(C(=O)NCC(CN(C(c2cc(C)sc2)=O)C)O)cc(N)c(F)c(F)c1Cl Cn1cc(C(=O)NC2CCCC2NC(=O)C(C2CCOCC2)F)c(C2CC2)n1 N1(C(CCCNC(=O)OC)=O)CC2(NC(c3ccc(Cl)cc3F)=O)CCC1C2 C1(C(F)(F)F)(C(=O)NC(CNC(C2(C#C)CCC2)=O)C)CC=CCO1 C1(NC(C(CC#C)C)=O)CC(F)(F)CC1NC(C1CC1)=O.c1ccc(Cl)cc1 C1(C(N2C(CNC(CCOC)=O)C(OC)C(OC)C2)=O)CN2CCN1C(C)C2 O=C1CCC2CN(c3nc4ccccc4nc3NCCC(F)(F)CO)CCC2N1 C1(CCC)CN(C(C2CCCCS2)=O)CC1C(=O)NCc1ccnc(C)n1 CCC(CN(C)C)C(=O)NC1CCC(CCC(=O)NCC(C)(O)CN(C)C)C1 N1(C(C2CCC(CCC)CC2)=O)CCC2(CC1)CCN(C(=O)C(O)C(C)OC)C2 C1(C(C)=O)CC(C)CN(Cc2cscc2-c2ccc(Br)cc2C)C1 N1(C(C(CC=CC)C)=O)CCC2CCCC12C(=O)NC(C)Cc1nn[nH]n1 Cc1cc(C(=O)Nc2ccccn2)ccc1NC(C1COCC1C(F)(F)F)=O CCCCCC(F)C(=O)NC1CN(C(=O)CCCCCF)CC(F)(F)C1 N1(C(C=CC=CCC)=O)CCN(C)C(C(=O)NC2CC(CO)C3CC23)C1 N1(C(Cc2c(C)noc2Cl)=O)CC2CCCC(C1)N2C(c1cnc(O)c(Cl)c1)=O Cc1sc(C(=O)N(C2CN(C(=O)Cn3cc(C4CC4)cn3)CC2F)C)nc1O CC(C)CC(C)CC(=O)N1CCC(C(=O)NCCNC(=O)CO)O1 Cc1nsc(C)c1C(=O)N(C)CC1CCCN1C(C1CCCC1F)=O Cc1sc(C(=O)NNC(=O)NCC2(O)CC(C(=O)OC(C)(C)C)C2)nc1O Cc1[nH]cc(C(N2CCCC2C2CCN(C(c3cnsn3)=O)C2)=O)c(=O)c1Cl CC1=C(C(=O)NCC2C(C(N3CCC3C3CCOCC3)=O)C2(C)C)CCCO1 c1(C(=O)NC2CN(c3ncnc(OC)c3C)CC(C)C2)ccc2nc[nH]c2c1 N1(C(C(C2CC(NC(=O)CSc3cn[nH]c3)C2)F)=O)CCC(F)(CF)C1 c1(C(N2CCC(O)(CNC(C3CCC(=C)CC3)=O)C2)=O)ccc(NC)c(S)c1 C(=O)(C(CC)(CO)OC)NCCNC(C1CN(CCC)C(=O)C1)=O S(=O)(=O)(c1cccnc1OC(F)F)NCCc1ccc(NS(C)(=O)=O)cc1 N1(c2cncc(C(=O)C(F)(F)F)n2)CC2CC1CC2(F)F CC(F)(F)CN(C(=O)C(C)C1CCC1)C.C(=O)CC(C1CC1)C1CC1.CO CON1CC(C(=O)NCC2CCN(C(c3ccc(Cl)cc3Cl)=O)C2)CC1=O N1(C(c2c(C)noc2)=O)CCC(NC(=O)CCCN2CCCC2)C12CCC2 N1(C(c2nc(OC)c(C)s2)=O)CC2CC(CNC(C3(C)CC=CC3)=O)C2C1 Cc1cc(C#N)cnc1C(N1CC(O)(C)C1)=O.c1(C=O)ccsc1C(F)(F)F C1(C(=O)NC(C)CCCNC(=O)CC2CCCC(=O)N2)CCN(C)C(=O)C1 C(CCN=C(NC1CC1)N1CC(=O)N(CCC(F)(F)F)C1)SC Nc1cc(CNCCC(N2CCCCC2)=O)ccc1Cl C1(OC)CC(NC(c2cc3n(c2)CCSC3)=O)C12CCN(C(=O)CCCF)CC2 c1(C(N2CCC(NC(CC=CCCCCC)=O)C2C)=O)ccn2ccnc2n1 C1(C(N2CCC(N(C(=O)CN3CCCCC3C)CCC)C2)=O)CN2CCC1CC2 N1(C(C2CCOC2)=O)CCN(C(=O)C(c2ccc(Cl)cn2)(F)F)CC1 C1(C(N2C(C)C(NC(C3(CO)CCCCC3)=O)CC2)=O)CCC2(CC1)CC(O)C2 C1(NC(c2ccc(C)s2)=O)CC(CNC(=O)C)C1(C)C.C1(C)CCCC1.O c1(C(=O)NC(CCCCNC(CC2(C=C)CC2)=O)C)cc2c(C)cc(C)cc2[nH]1 N1(C(C(C)CN(C(=O)CC2(C)OCCO2)C)=O)CC(=O)NCC1C(N)=O C1(C(=O)NCC(=O)OC)CCCCC1NC(=O)C(=C1CCCCC1)F N1(C(C2(SC)CC2)=O)CCC(C2CCN(C(c3c(C)cncc3C)=O)C2)C1 C(=O)(C(F)(F)C(O)C1CC1)NC1CC(CNC(C=CCCC)=O)C(O)C1 c1(NC(C)=O)ccc(S(=O)(=O)NC2CC(C(F)F)(OC(C)C)C2)cc1F Cc1cc(C(=O)NC2CCC2NC(=O)CC23CCCC2C3)cc(Cl)c1 c1(C(=O)NCCNC(C2CCCC2C2CC2)=O)cc(Cl)cc(F)c1F c1(CC)c(C=O)csc1C.C(=O)C(C)n1cccn1.C1(CCC)CC1.C(C)=O.N C(=O)(C1CCc2cccnc21)NC(C1CC(NC(CC(C(C)C)C)=O)C1)C CN1CCC(C)(C(=O)N(CC(O)CN(C)C(C2(C(F)F)CC2)=O)C)C1 C1(NC(c2cc(C)oc2)=O)CCN(C(c2ccc(C(N)=O)c(F)c2)=O)CC1CO C(=O)(C(C)C(O)C(C)C)N1CCCCC(CCC(=O)NCC(CC)(O)CC)C1 Cc1ccc(CC(=O)NCC2CC2NC(c2ccn(C(C)C)c2C)=O)cn1 C#CCC(CC(F)F)C(=O)N1CCC(CC)C1C(=O)NC(CC)C(C)(F)F CCC(C)C.C1(CC=O)CCN(C(=O)C(C)C)C1.N1(CCC=O)CCCC1=O.N S(=O)(=O)(c1ccccc1Br)N1CC(CNC(CC(C)(C)C)=O)OCC1 C#CCCC(O)C(=O)NC12CCC(CNC(c3cc(N)cc(O)c3)=O)(C1)OC2 CC(O)C(F)(F)C(=O)N(CCC)C1CC1.c1(C=O)coc(CS(C)(=O)=O)n1 c1(CCC)ccc(S(=O)(=O)N2CC(CC(N3CCN(C(C)=O)CC3)=O)C2)cc1 C1(COC)(NC(c2ccncc2OC)=O)CCCN(C(=O)C2=COCC2)C1 Cc1c(C(=O)N)ccc(F)c1F.C1(C(N2CCC(F)C2)=O)C(F)(F)C12CCC2.C C1(C(N2CCC(C(=O)OC)(OC)C2)=O)CNc2cccc(Br)c2O1 CC(C)CC(F)C(=O)NC1CCN(C(c2ccccn2)=O)C1C(C)(C)C CC1CN(CC(O)CNC2(CNC(=O)OC(C)(C)C)CCC2)CCO1 C1(NC(C2C(C(=O)OC)C2)=O)CN(C(C2CCC2OC)=O)CC12CCCC2 C(=O)(CCP(C)(C)=O)NC(C(CO)NC(C(c1c(C)cccc1)(C)C)=O)C C1(C)CC(F)(F)CN1C(=O)Cc1ccc(F)cn1.Cc1scc(C(=O)N)c1C.C C(c1ccc(Cl)cc1)=CC(N1C(C(N)=O)(COC)CCC1)=O c1(NC(C(=O)N(C)CC2CCCO2)=O)cc2c(cc1F)CCNC2=O c1(OCC)ccccc1OCCN1CC(N2CCCC2)CC1C(C)C N1(C(C=COCC)=O)CC(NC(c2ccc(CS(N)(=O)=O)cc2)=O)C(C)C1 C1(CNC(c2c(C)ncs2)=O)CN(C(c2cc(F)cnc2O)=O)CCC12CCC2 C1(C(=O)NCC2C3CN(C(C(CCC)CC)=O)C2C3)CCOC2(CCCCC2)C1 N1(C(CC2C(NC(c3nc(C)sc3)=O)CCC2)=O)CC2CCC2(C)C1 Cc1cc(CNC2CN(C(=O)Cc3ccccc3O)CC2C)cc(C)c1 N1(C(CCCCN(C(C)=O)C)=O)CC2(C1)CN(C(c1csc(=N)[nH]1)=O)CCO2 C1(C(=O)OCC)CN(C(=O)C(C)C)CCN1C(c1ccc[n+]([O-])c1)=O C12(NC(c3nc(C)oc3)=O)CCN(C(C3CCCN3C(N)=O)=O)CC1C2 C1(NC(C2CCCC(N(C)C)C2)=O)CCN(c2nnc(C3CC3)o2)CCC1CO C1(CC(=O)NCc2c(CCNC(COC)=O)ocn2)CCC2(CCC2)CO1 C(=O)(C1=NOC(C)(C)C1)NCC1CN(C(c2nc(C)n(C)n2)=O)C(C)CC1 N1(C(c2c(C#C)cn(C)n2)=O)CCN(C(=O)COCC(F)(F)F)C2CCCCC12 C(=O)(CCCCC(C)(C)C)N1C(C)CCN(C(C2CC3(CCC3)CCO2)=O)CC1 CCCC(C(=O)NC1COCCC1OC)NC(C1CC(C2CC2)C1)=O CN1CCCC2(CCN(c3nc(N4CC5CCC4C5)nc4cccnc34)C2)C1 c1(CCC(=O)NCC)ccccc1C(F)(F)F.C1(C=O)CC1.C1CC1.C Cc1ccc(C(=O)NCC2(CCNC(C3COCCN3C)=O)CC2)c(N)c1Cl c1(OC)nc(C)c(S(=O)(=O)NC(=O)CC2CCOC2)s1.C(C#N)N c1(C(=O)NC(c2cn(-c3ccncc3F)nn2)(C)C)n[nH]c2cc(C#N)ccc12 c1(C(=O)N)ccc2c(n1)CCC2.C1(CC(=O)N(CC(C)O)CC)CN(C)C1 C1(CC(=O)NCc2n[nH]c3ccncc23)CCC2CNCCC2C1 c1(C(N2C3CCC(CNC(=O)CCF)(C3)C2)=O)ccc(S(=O)(=O)CF)cc1 c1(C(C)=O)cc(NC2CCC2CNC(c2cccnc2O)=O)ccc1[N+](=O)[O-] C1(C(=O)NCC2C(CC(=O)O)CCCC2)CN2CCN1CC2 Cc1cc(C)c(C(=O)N(CC(C)NC(c2cn(CC(F)F)cn2)=O)C)cn1 CCCC(C(=O)NCC1(F)CCN(C(C2CC(O)CN2C(C)=O)=O)C1)C(C)C c1(OC)cccc(-c2cc(C(=O)NCC=CCNC(=O)CC#N)no2)c1 C1(C(N2CC(=O)CC2C(=O)NCCCN2CCCC2)=O)(CC)CCCC1O C1(NC(C2CC2c2ccc(Br)cc2)=O)CCN(C(c2ccco2)=O)C12CCC2 N1(C(C(c2ccc(OC)cc2C)C)=O)CC(O)C(O)CC2(CCOCC2)C1 N1(C(C(C)N(C(C(C(=O)OCC)OC)=O)CC)=O)CCN(CC)CC1C C1(C(N2CC3CC=CC2C3)=O)CC2CCC1N2C(=O)C1=NOCC1 C1(CNC(c2sccc2Cl)=O)CN(C(=O)COC)CC1(F)F.c1cccnc1 C#CCCCCC(=O)NC1CCOCC1C(=O)NCC=CCOC CC1(C)CCN(C(C2(N3CCOCC3=O)CC2)=O)C1.C(=O)C.[SH](C)(=O)=O.N C1(C(C)NC(=O)C(=O)NCc2nc(C3CCCCC3)no2)CCc2nccn2C1 C1(N(C(C(CC)O)=O)C)CCC(CNC(=O)CSc2ccc(CC)cc2)CC1 c1(C(CC)(C)C)cn(CC2C=CCN2C(=O)COC)nn1 C(=O)(CS(=O)(=O)c1ccccc1F)N1CC(O)(CNC(C2CCCC2)=O)C1 CCC(CN(C)C)C(=O)NCc1occc1C(=O)N(CC(C)SC)C c1(OC)cc(C(=O)NCC(O)CN(C)C(c2[nH]c(C)nc2C)=O)cc(F)c1F CC(C)(C)C(C(=O)NC1CCC1)NC(C1CC(O)C1)=O N1(C(C(=O)NCC2N(C)CCCC2)=O)CCCC(N)(C#N)C1 N1(C(C(C)C2CCCC2)=O)CC(NC(c2ccc(Br)s2)=O)CC(F)C1 c1ncc(C(N2CCC(O)(C(F)(F)F)C2)=O)cn1.c1(C(=O)NC)ncccc1O CC1CCCC(CCN(C)C)N1CC1CC2CC(C1)C2 c1(C(=O)NC2CCN(C(CC(C)F)=O)CC2)ccc(S(=O)(=O)CC#N)cc1 CON=Cc1ccc(C(=O)NC2CN(C(C3CCC4(CC3)CC4)=O)CC2C)cc1 N1(C(=O)NC(C#C)CC2CCCC2)CCCC(CC)C1 CC1=C(C(=O)N2CCC(CCNC(=O)CC3(C)CC3F)CC2)SCCO1 C#CC1CCCN(C(C2CCCN2C(=O)C=CC(F)(F)F)=O)CC1 N1(C(CC2CCN(S(C)(=O)=O)CC2)=O)CCC2(CC2)C1.C1(C=O)CCC1(F)F.N Cc1cccc(CC(=O)NC2C3CN(C(c4[nH]cnc4C)=O)CC23)c1F c1(CN(C(CC)CSC(C)COC)C)ccc(C(=O)OC)cc1 C12(NC(=O)CCF)CCC(CC1NC(=O)Cc1cccc(Br)c1F)C2 c1(C(=O)N)cc2ccccc2nc1O.CC(CN(C)C)C(=O)NC1CC(C)(C)C1 C12(CNC(C(CCC)O)=O)CCCCC1N(C(c1cc3ccsc3[nH]1)=O)CC2 C1(NC(=O)C2=CCCC2)CS(=O)(=O)C12CCN(C(C13CCC(CC1)CC3)=O)CC2 c1(C(=O)N)ccc2occ(C)c2c1.c1(C(=O)NCCC(=C)C)cc(C)n(C)c1C C1(C(=O)N)CC12CCN(C(=O)C1=NOC(C)(C)C1)CC2.n1(CC)cc(CC)cn1 C1(NC(c2nc(COC)[nH]n2)=O)CN(C(C2(n3ccnn3)CC2)=O)CCC1C n1(CC)cnc2[nH]c(=NC(C)CC(N)=O)nc(N3CCOC(C)(C(C)C)C3)c12 O=C(CC1=CCOCC1)NC12CCN(C(c3snc(Cl)c3Cl)=O)CC1C2 CC(C)C(CC1CCCCC1)C(=O)NC1CC1c1ccccc1C(F)(F)F c1(C=O)c(Cl)sc(C)c1C.C1(OCC)(C)CN(C(=O)Cc2cccs2)C1.N N1(CCOC(c2ccnn2CCO)=O)CCC(F)(F)CC1 C(=O)(C1=C(C)OCCS1)N(CC(CNC(C1(CC)CCOCC1)=O)C)C c1(C(N2CC(C)C(C)C2)=O)nc2c(s1)CCCCC2 N1(C(c2ccc(C)n2C)=O)CCC(C2(NC(C3CCCC(O)C3)=O)CC2)CC1 CCC(N=c1[nH]c2c(c(=NCC(C)C(=O)NC)[nH]1)SCC2)C1CC1 N1(C(C2(NC(=O)CCC3CCOCC3)CCCC2)=O)CCC2(CCCO2)C1 N1(C(C2CC(OC)CN2C(=O)CO)=O)CC(=O)NCC12CC2.CCCN(C)C c1(OCCNC(=O)NC2CC(=C)C2)ccc2oc3ccccc3c2c1 C1(C#C)(C(=O)NCC(C#C)(C)C)CCN(C(=O)C=C(C)COC)C1 C1(NC(C2CN(CC)C(=O)C2)=O)CCC2(CC1)CCC2.C1(C(=O)N)CCNC1=O n1(CC)cc(C(=O)NC2CCC(N(C(=O)CCCSC)C)C2)cn1 c1(C(=O)N)c(F)ccc(F)c1F.c1(COC)ccccc1C(N1CC2CC1C2)=O c1(NC(C(=O)NCCc2nccn2CC(F)(F)F)=O)cc(Cl)c2c(c1)OCO2 C12CCCC(CN(C(c3ccc(C(F)F)s3)=O)C1)C2.C(C)(C(=O)N)OCC#C CCC(CCCO)NC(=O)C(Cn1cccn1)NC(c1cocc1C)=O n1(CC)ncc2c(NC3CCCN(C(C4(C)CC4)=O)CC3)ncnc12 C=C(C)CC(C(=O)NCC1CCN(C(=O)CC(C)C(F)F)C(C)C1)OC N1(C(C=CCC)=O)CC(NC(=O)CCCN2CCOC2=O)CC1C c1(OC)cc(Br)c(CNC(=O)C(C(F)(F)F)OC(C)=O)cc1OC C12(C(=O)NCC3CCCCN(C(Cc4ccc(C)s4)=O)C3)C3CC(CC13)C2(F)F C1(NC(Cc2cc(CC)no2)=O)CC2CCC1CN2C(=O)C(C)S(C)(=O)=O N1(C(CCC#C)=O)CC(NC(=O)CCC2CC(C)C2)C2CCCC12 C1(NC(C(CC)CN(C)C)=O)CC(C(=O)N(C)Cc2cn[nH]c2)C12CCC2 C1(CC(=O)NCCNC(C(CC)C)=O)CCCCN1C(C)=O CCCCCC(O)C(=O)NC1CCC(O)CN(C(c2ccc([N+](=O)[O-])cc2)=O)C1 N1(C(C(C)(C)C2CCC2)=O)CC2(CCN(C(c3cnn(C4CCCC4)c3)=O)C2)C1 C1(CNC(CNC(N(C(C)C(F)F)C)=O)=O)CC12CCc1ccccc12 c1(C(C)C(=O)N(CCCNC(=O)CCC2OCCO2)C)ccccc1C(F)(F)F C1(C(N(C)CC2C(C)OCC2)=O)C2CC3C(C2)C13.C1(C)(C=O)CCCN1C.N N1(C(c2c(C)cnnc2)=O)C2CCCC1CN(C(=O)CC1CC(C)(C)C1)C2 C(C(CO)(CO)NC(C1CC1F)=O)N(C(c1ccc(C(OC)OC)o1)=O)C N1(C(C(F)OC)=O)CCC2CN(C(c3ccc4nc(C)sc4c3)=O)CC2CC1 N1(C(c2c(C)nns2)=O)CCC(C(=O)Nn2cccn2)CC1C N1(C(CNS(CC)(=O)=O)=O)CCC(C(C)NC(=O)CN2CCCCC2)C1 c1(OCCC(=O)NCC2(O)CN(C(C3CC3Br)=O)C2)ccccc1F c1(-c2ccccn2)ccc(-c2nc(-c3ccccn3)nn2C2CC2)cc1 C(=O)(C(C)CCNC(C1CCCN(C(=O)CSCC(N)=O)C1)=O)OC C=CC1(C(N2CC(C(C)CC)C2)=O)CCN(C(c2cc(Cl)n(C)n2)=O)C1 Cc1ncnc(C(=O)NCc2ccc(C(=O)N(C(C)CN(C)C)C)cc2)c1C c1(C(=O)NCC(=O)NCC)occc1CNC(c1cc(=N)[nH][nH]1)=O c1(OC2(CC(=O)OCC(C)C3CCC3)CCC2)cccnc1Cl Cc1cc(C)c(NC(C2COCCN2C(=O)C=Cc2cnc[nH]2)=O)c(C)c1 C(=O)(CS(=O)(=O)C1CC1)NC(CCNC(C(C1CCC(C)CC1)CC)=O)C(C)C c1(C(N2CC(NC(c3c(CC)ccs3)=O)C(O)CC2)=O)ccc(N)c([N+](=O)[O-])c1 C(CCCCC(=O)NC1(C2CCCN2C(C2C=CCCC2)=O)CC1)OCC C1(C(=O)NC(CCC)C(=O)NC2CCN(CC)C2)CC(=O)OC1(C)C.C1CC1 c1(C(N(C2CCCN(C(C3CCCS3)=O)C2)CC)=O)cc2c(s1)CCCNC2=O c1(C(N2CCCC(CN(C(CC3(C=C)CC3)=O)C)C2)=O)ccc2ccnn2c1 C(=O)(C(C)(C)C(=O)N1CCC(CNC(=O)C2=CCOCC2)C(O)C1)OCC C1(C=O)CC2(CC(=O)N2)C1.C1(C(=O)NC(CCC)C)CCC(C(N)=O)CC1.N N1(C(CC(CC)C)=O)CC2CC1CN(C(c1cc3ccncc3[nH]1)=O)C2 C1(NC(C2(C)COC2)=O)COC2(C1)CN(C(c1nncn1C1CC1)=O)C2 N1(C(COCCNC(CC2C(C)OCC2)=O)=O)CC2(C1)CN(C)C2 c1(OC)cc(C(N2CCN(CC(=O)NC(C)CF)CC2)=O)cc(OC)c1Br n1(CC(=O)NC(Cc2cnc[nH]2)C(=O)NCCC(O)C2CC2)ncccc1=O N1(C(C(C(CC)C)N)=O)CC2CCCC(C(N3CCCC3C#N)=O)C2C1 CCC(CC)C(O)CNC(=O)C(C)(C)CCNC(c1ccoc1Cl)=O C1(C)(NC(C2CC(OC)C2)=O)CC(NC(=O)CO)C1.C1CCCCO1.C C1(NC(c2cc(OC)no2)=O)CN(C(c2ccc(C(F)(F)F)cn2)=O)CC1C N1(C(COCCCC#C)=O)CC2CC(C1)N(C(=O)C(F)CC1CCCC1)C2 N1(C(c2cc(C)cc(C)c2)C(=O)Nc2ccccc2)CC(C)(C)C12CCOCC2 C(=O)(CCC(C)C(C)=O)NCc1nccc(C(=O)OCC)c1 Cc1ccc(OCCC(=O)NCC2CCC2NC(C2(CCO)CC2)=O)cc1 N1(C(CSCCNC(CCc2onc(C)n2)=O)=O)CCOc2cc(F)cnc21 Cc1nsc2ncc(C(N3CC(N(C)C(c4ccns4)=O)C(C)(C)C3)=O)cc12 c1(N2CC(C)OC(C)C2)nccc(=NCCSc2ccc(F)cc2)[nH]1 c1(C(=O)NC2CCC(CNC(C=CC)=O)C2)cc2c(O)cc(Cl)cc2[nH]1 C1(CCC(=O)NCC(c2nccs2)C)CCN(C(=O)CC2(C#N)CC2)CC1 Cc1cnc(C2(NC(=O)CCc3cnc[nH]3)CC2)o1.C(=O)(C(C)n1ccnc1)N C#CC1(C(=O)NCCNS(N)(=O)=O)CCN(C(=O)C(C)C2CCCO2)CC1 c1(C(=O)NCC2CC(C)C(C)(C)CC2)cc2c(nc1O)CCC(F)(F)C2 N1(C(C2(C(C)C)CC2)=O)CCN(C2CCN(C(=O)CC3C=CCCC3)CC2)CC1 N1(C(=O)COCC2CC2)CCN(C(C2(CF)CC3(CCC3)C2)=O)CC(O)C1 c1(C(N(C2(c3cc[nH]n3)CC2)C)=O)n[nH]c2c1CN(C(c1ccon1)=O)C2 CC1CCN(C(C2CC3C(C2)C3(F)F)=O)CC1NC(C1CC12CCCC2)=O Cc1nn(C)c2sc(C(=O)NCC(C3CC3)NC(=O)C(O)CC[S+](C)C)cc12 C1(F)(CNC(CC)=O)CC(NC(C2(C)CCOC2)=O)C1 C1(CNC(c2cc[n+]([O-])cc2)=O)C2CN(C(=O)Cc3ccoc3)CC12 CC1CC(CNC(=O)CC2CCSC2)CN(C(=O)CCOCC(C)(C)C)C1 CC1CN(C(=O)CCC2CC2C)CCN(C(C2CC(C3CC3)=NO2)=O)C1.C1CC1 C(=O)(CCC(C)S(C)(=O)=O)NC(C)CNC(C1CCC=CCC1)=O Cc1ccc(F)c(Br)c1C(=O)NCCCNC(c1ncc(F)cc1N)=O c1(CC(=O)NC(C)(CNC(c2csc(Cl)n2)=O)CO)ccc2c(c1)OCCO2 c1(CCCC(=O)NCC2C(N)CCC2)ccc(F)c(F)c1 C1(C(=O)NCC2CCN(C(=O)Cc3cccc(Cl)c3)C2)CCn2ncnc2C1 Cc1cn(C)nc1C(=O)NCC1CC1CNC(c1cc(C)n(C)n1)=O N(C(=NCCC1CCSC1)N1CCOC2(CCCCC2)C1)CC(C)(C)C C1(COC(=O)NC)CCCCN1C(=O)CC1CCC(=O)N1 c1(NC(c2occc2Br)=O)ccccc1C1(NS(=O)(=O)CCCCl)CC1 N1(C(c2c(CNC(C(C=C)OC)=O)noc2)=O)CC2(C=CCO2)C1 N1(C(C(=O)NCc2ccc(-c3cn(C)nc3)cc2)=O)CCC(CSC)C12CC2 CCC(C)C(O)C(C)C(=O)NCc1cc(C(N2CCCC2(C)C(C)(C)C)=O)n[nH]1 C1(NC(C(C2CCC2)OC)=O)CCC2(CC1)CN(c1ncnc3c1SCCC3)C2 O=C(C1CCCn2ncnc21)NCC1CCN(C(c2cc3ccccc3s2)=O)C1 c1(C(=O)NC2CN(c3snc(CCOC)n3)C(C)CC2)cccc2cnccc12 c1(C(=O)NCC2(F)CC(NC(c3c(C)ocn3)=O)C2)nc(O)c(C)s1 Cc1cccc(CCC(N2C(C(=O)Nc3ccc(CCO)cc3)CC3CC23)=O)n1 c12nn(c(=O)c3ccccc13)C2.c1(C(=O)OC)ncncc1CCO C(CC(C)(C)NC(=O)C(C)N1CCCC1)=CC(=O)NC(CCSC)C CC(C)CC(C)(O)C(=O)N1CC(C(C)NC(=O)C(F)(F)c2ccncc2)C1 C1(C(C)C(=O)NC2(C)CN(C(C3OCCCO3)=O)C2)CCCCCC1 C1(CCNC(C2C(CC)C2)=O)CCN(C(c2nn[nH]c2C(F)(F)F)=O)C1 C=CCC(CC(C)C)C(=O)NCC1CCN(C(C2CC(C)(O)C2)=O)C1 C(=O)(C1=CCS(=O)(=O)C1)NC(CNC(C(C(C)C)c1ccc(F)cc1)=O)CO Cc1cc(=NCC2CCCN2C(=O)C2CC2)[nH]c(=NCc2ccc(Cl)c(Br)c2)[nH]1 c1(CCC)nc(C)c(CN(C)CCN(C(C2CC(C)CO2)=O)C(C)C)o1 N1(C(CN(CCC)C)=O)CCC(C(C)NC(=O)C(Cc2ccccc2)CC)CC1 c1(C(C(=O)NCCCCNC(CP(C)(C)=O)=O)O)cc(F)c(F)cc1F N1(C(c2cnn(CC)n2)=O)CC2CCCC1C2CNC(=O)C(C)C(C)C CC1(C)CCN(C(c2cnn(C3CCC3)c2)=O)CC1C.C1(C)(C=O)C=CCC1.N C1(C)(C(=O)NCCC)CCCN(C(CC2CCCSC2)C(=O)NC)C1 C1(NC(CC(C)CF)=O)CC2CCC1N(C(=O)Cc1ccc(F)c(Cl)c1)C2 N#Cc1csc(C(=O)NC2C=CCCC2C(=O)NC2CCC3CCC23)c1 C1(NC(CCCOC(C)C)=O)CCN(C(c2n[nH]cc2F)=O)CC1 N1(C(C(CC)O)=O)CC2(C1)CN(C(c1cn3ccccc3n1)=O)CC2CO N1(C(C2C(OC)C2)=O)CCC2CN(C(c3ccc(C)cc3SC)=O)CC12 c1(C(=O)NC2CCC(NC(C(C(C)C)OC)=O)C2)ccc2cncn2c1C N1(C(C(CC)NC(C)=O)=O)CCOC2CN(C(=O)C(F)CC3CCOC3)CC12 N1(C(c2cc(O)nc(Cl)c2)=O)CC2CCC(C1)N2C(c1ccnn1CC(F)F)=O CC1(C)CC=C(c2ccc(C(=O)O)cc2-c2nccn2Cc2cc(Cl)ccn2)CC1 N#Cc1cscc1C(=O)NC1CCCC(NC(=O)CCCCN2CCCCC2)C1 C1(C)(CNC(c2n(CCC)ccc2)=O)CN(C(=O)CC2(C)CC2)CC1C CCC(C)(CC)C(=O)N1CCN(C(=O)Cc2ccn(C)n2)C(CCO)C1 C(=O)(C1=C(C)CCOC1)N1C(CC)CCC1C(=O)Nc1cnn(CC(N)=O)c1 C(=O)(C1=CC(O)CC1)NC(c1ccn(C)n1)CC.n1(CC=O)cc(C)cn1.N C(CC(F)=C(F)F)NC(=O)CC1COCCN1C(=O)CC(F)(F)F N1(C(c2ccc(NC)cc2Cl)=O)CCC2CCN(C(=O)C=CC=C(Cl)Cl)CC12 c1(C(c2nnnn2C2COC2)NCC(COCC)C)ncc(I)s1 C(=O)(CCCN=[N+]=[N-])NC1CC(C(N2CC(C)(NC(C)=O)C2)=O)CC1O CC(C)C(C)CNC(c1cnn(C(F)F)c1)=O.N1(CC=O)CCC(O)CC1.N N1(C(C(C)SC)=O)CCOC2(CCN(C(C3CCC(=O)C(C)C3(C)C)=O)C2)C1 c1(C(=O)NCC2N(C(C(c3ccc(Cl)s3)C)=O)CC2)ccc(C2CCC2)nc1 C1(C(C)C)CN(C(=O)CC2OCCC2(C)C)CC1C(N1CC(O)(C(F)F)C1)=O C1(CNC(C(CC)SC)=O)(OC)CCN(C(C2CC(C)=NO2)=O)CC1 N1(C(c2cnc(C)[nH]2)=O)CCC(CNC(=O)COc2cccc(Cl)c2)CC1 C(=O)(C(C(O)C1CC1)NCc1cnc(C2CC2)o1)OCC c1(CCNC(=O)NS(C)(=O)=O)cn(CCSc2ccncn2)nn1 c1(C(N2CC(CNC(C3CC34CC4)=O)C2)=O)cc2cccc(Cl)c2s1 C(=O)(C(C)=Cn1ccnn1)N1C(CNC(CCC(C)OC)=O)C(C)CCC1 C(=O)(C#CC1(C)COC1)N(CCN(C(C1C(C=C)C1)=O)C(C)C)C c1(CNCC2N(C(C=CC=CC)=O)CCCC2)cc(OC)ccc1O C1(C(N(CCCC)C)=O)CCCN(C(C2CC(=O)N(C3CCC(C)CC3)C2)=O)C1 c1(C=O)cc(C)c(C)o1.N1(C(C)=O)CCCC1CNC(c1ncoc1)=O.C Cc1cc(N)cnc1C(=O)NCC1(NC(c2cccc(F)c2Cl)=O)CCCC1 N1(C(=O)Cc2c[nH]ccc2=O)CCC(NC(C2(CO)CC2)=O)C(CO)CC1 N1(C(c2c(C)n(C)nc2)=O)CCCC2(CCN(C(C3CCC4(CC4)C3)=O)C2)C1 N1(C(C(C2CCC(=O)N2)C)=O)CCC2(CCN(C(=O)CN(C)C3CC3)C2)C1 C1(F)(CNC(c2cc(C)[nH]c2C)=O)CCN(C(=O)C(O)P(C)(C)=O)CC1 C(=O)(C1CCc2nccn21)NCC1(C)CCCN1C(=O)CCc1ccc[nH]1 N1(C(CNC(CN(C(COC)=O)C)=O)=O)CCN(C(C2SCC=C2C)=O)CC1 n1(CC(=O)N(C(C(=O)O)C2CC2C(=O)O)C)cnc2c(N)ncnc12 Cc1cnc(NC2CCC(=O)NC2)c(S(=O)(=O)NCCn2cccnc2=O)c1 N1(C(c2c(C)n[nH]c2C)=O)CCN2C(=O)C(NC(=O)CCCC3CC3)CC2C1 CCCC(CCC)CC(=O)NC(COC)CC(=O)NCc1cnc2n1CCC2 c1(OC)cc(C(=O)NC(C2CN(C(c3cccnc3S)=O)CCO2)C)cc(C)c1 C(=O)(CC(C(F)(F)F)NC(N1CCC(OCC2CCC2)CC1)=O)NCC N1(C(C2(OC)CCC2)=O)CCCCC(C2CN(c3nccc(C)c3[N+](=O)[O-])C2)C1 c1(C(N(C(CNC(c2c(C)n(C)nc2)=O)C2CC2)C)=O)cc(Cl)nc(Cl)c1 c1(CC(=O)NCC(O)CNC(c2cc(F)n[nH]2)=O)csc(-c2cccnc2)n1 N1(C(CC(C=C)(C)C)=O)CC(C)CN(C(c2cccnc2F)=O)CC1C c1(NC)snc(C)c1C(=O)N.C1(C=O)CC(=O)N(C(C)C)C1.C1CC1.C c1(C(N(C2CC(NC(C34CCC(OC)C3C4)=O)C2)C)=O)ccc(C)c(Cl)c1Cl C12(C(N3CCCC(N(C(c4nc(C)sc4)=O)C)C3)=O)CC(C)(C1)OC2C CC(=O)CCCCC(=O)NC(C(N1CC2(C1)CC(C)(O)C2)=O)C1CCC1 CCC(CC(=O)N1CCC(CNC(c2cnc3ccnn3c2)=O)C(O)C1)C(C)C c1(COC(C(=O)NC(CN(C(CCC#C)=O)C)CC)C)ccc(F)cc1 c1(C(=O)NCCNC(C2CCCN(S(CC)(=O)=O)C2)=O)cc2sc(Cl)cc2[nH]1 c1(C(N(C2CCCN(C(c3cnnn3C)=O)C2)CC)=O)ncc(P(C)(C)=O)cn1 Cc1ccc(C(N2CCC(C(=O)NCC3CC3(C)C)C2(C)C)=O)nc1C C(C(COC)CC(=O)NC(C)(C)C=CC(=O)NCC1CCSC1)OC C1(O)CCC1.N1(C(C=O)C)CCNC1=O.C1(C(=O)NC)(C(=O)N)CCC1.C N1(C(C2(N(C)C)CC2)=O)CCOCC(C)(CNC(c2snc(Cl)c2Cl)=O)C1 CC(F)(F)CC(=O)NCCCCC1CCN(C(c2cncnc2)=O)CC1 N1(C(c2c(CCC)nco2)=O)CC2CCC1CN2C(c1c(O)cccc1Cl)=O O=CN1CCCC1C(=O)NC1CC(NC(c2cnc(-c3ccoc3)s2)=O)C(O)C1 C(=O)(C1=CCSC1)NCC(C1CCC1)NC(C1(COC)CCCO1)=O Cc1ncc(C(=O)NC2CC(C(N3CCC(O)C3(C)C)=O)C2)cc1C#N Cc1nn[nH]c1C(N1CC(O)(CNC(=O)CCn2cccc2)C1)=O C1(OC)CC(NC(c2ccc(C)n2C)=O)CN(C(C2CC3CCC3C2)=O)C1 Cc1cc(=O)c(C(=O)NCCCCC2CN(C(=O)CCC(C)(C)C#N)C2)cn1C C(CC(=O)N1CC(NC(=O)C=C=C(C)C)C2CCCC12)(C(F)(F)F)OC c1(OCC)ccccc1NC(C1CC(NC(c2ccsc2C#N)=O)CCO1)=O C(=O)CCC.C1(c2cccs2)(C(N(CC)CC)=O)COC1.C(=O)C1CC1.N CC1CN(C(C2CC3C=CC2O3)=O)CCN1C(=O)CSCCC#N c1(C(=O)NC2CCC(CNC(c3n(C)cc(C#N)c3)=O)C2)ccc2nc[nH]c2n1 c1(C=O)ccc2c(c1)COCC2.C(=O)(C(CC)C(=O)N)OCC.C(C)C1CC1 c1(N(C(N2CCN(C(Cc3c(C)con3)=O)CC2)=O)CCO)cc(C)c(Cl)c(C)c1 Cc1ncc(C(=O)N(CCCNC(=O)C(C)SC(F)(F)F)C2CC2)cc1N C(=O)(C(F)C(=O)NCCC(C(=O)NCCCCC(=O)OC)OC)OCC Cc1c(C(N2CC3CCN(C(=O)CC4CSC4)CC3C2)=O)c2ccccc2n1C C(=O)(CC1=CCCCC1)N1CCC(NC(=O)C=Cc2ccc(C(F)F)o2)C1 c1(C(N2CCCC(CN(C(C3C(CC)C3)=O)C)C2)=O)cc(C)c2ncccc2c1 c1(C(N2CC(O)C2)=O)cc(F)ccc1O.c1(C(C)OCC)nc(C(=O)N)cs1 c1(C=O)cc2ccccc2c(O)n1.C1(C(=O)NCC)(OC)CCS(=O)(=O)C1.N c1(OC)nc(C(=O)NC(CNC(c2cnco2)=O)C(C)C)co1 N1(C(=O)C(C2CCN(C(c3ccc(C(F)F)o3)=O)C2)F)CCn2nccc2C1 CN1CCC=C(CNC(=O)CCC2CC(NC(C3CC3(C)C(F)F)=O)C2)C1 C1(NC(C2CC(C)(C)OC2)=O)CN(C(=O)COC(F)F)CCC12CCC2 N1(C(C(C=C)CC)=O)CCCC12CCN(C(=O)C#CC1CCOC1)CC2 c1(N2CCC(CC)OCC2)nc(N2CCC(CC)C2)c2c(n1)COC2 C=CCCN=C(NCCc1sc(C)nc1C)NCc1ccco1 c1(C(N2CCC(C)C2CNC(c2cc(C3CC3)on2)=O)=O)cccn2nccc12 N1(C(C(CC)NC(N)=O)=O)CCOCC(NC(=O)Cc2c(Cl)cnn2C)C1 N1(C(C(N2CC=CC2)C)=O)CCCN(C(C2C3CCC2(c2ccco2)C3)=O)C(C)C1 C1(NC(C(CC)C)=O)C2COCC1CN(C(c1ccc(O)cc1F)=O)C2 C1(=CC(=O)NC2C(NC(C3N(C)C(=O)CC3)=O)C2)CCOc2ccccc21 C(=O)(CCCCC(F)F)NC1C(C)CCN(C(c2cc(Br)c[nH]2)=O)C1 Cc1ccc2c(c1)C(NCC(O)C(F)F)CCC2 c1(-c2cc(NC(C3SCC(=O)C3)=O)sc2)cc(F)cc(F)c1 c1(N2C(C)CCC(NC(C3CCS3(=O)=O)=O)C2)ncnc2c(Cl)cc(Cl)cc12 C1(NC(C2(NC(Cc3ncn(C)c3)=O)CC2)=O)CCN2CCCC2C1 C1(C(=O)NC(C(C)C)(C)CNC(c2cc(C(F)F)ccn2)=O)CCCCN1N=O c1(CCC(=O)NC2CCN(c3ccccc3)C2)nnc(C(F)F)o1 CCC(CCC(=O)N1CCN(C(C2CCCC2)=O)CC1CF)OC c1(OC2CCN(C(=O)NCC3CC4CC3(CO)C4)C2)ccc([N+](=O)[O-])cc1 C1(NC(C2N(C(c3cnc(C)s3)=O)C(C)C2)=O)CCCC(CO)C1 C1(NC(c2ccc(C(F)F)o2)=O)CCOCC1NC(c1cc(Br)co1)=O N1(C(c2noc(C)c2C)=O)CCC2C1CCN2C(c1cc2cccnn2n1)=O N1(Cc2c(CC)ccs2)Cc2ccc(OC)cc2C(C(=O)OC)C1 c1(C(N2CC=CC(NC(CC3(C=C)CCOCC3)=O)C2)=O)ccc(C#N)c(O)c1 N1(C(c2c(C)scn2)=O)CCN(C(=O)CNc2ccccc2Cl)CC1CC(F)F C(C(COC)CC(=O)NC(CNC(c1cncnc1)=O)C(C)C(C)C)OC.O N1(C(C2(NC(C(CC)=CCCC)=O)CC2)=O)CCC2(CCCC2)CC1 C(=O)(CCCCC(F)F)N1CCC(CN(C(=O)C(c2cncnc2)C)CC)CC1 c1(CC)cc(N)c(C(=O)NC(C)CN(C(=O)CSCC(N)=O)C)cc1F C(=O)(N=c1ccn(C(C)(C)C)[nH]1)C1(F)CCN(C(C2N(CC)CC2)=O)CC1 CCC(C)C(=O)NCC(=O)N(CCCCN(C)C(C1(CF)COC1)=O)C N1(C(c2ccc(SCC)nc2)=O)CCCC2(CCN(C(=O)CC3CC3(C)C)C2)C1 C(=O)(CC(CNC(C1CNC(=O)N1)=O)OC)NCCOC(CC)CC C(=O)(CCCCCNC(=O)COCCOCCO)N1C(C(CC)C)CCC1 C1(CN(C(C2(CCCC)CCC2)=O)C)CCN(C(=O)C(c2cncn2C)O)CC1 Cc1occ(C(F)(F)F)c1CC(=O)N(CCF)Cc1ccc(-c2ccccc2)nc1 C(=O)C(C)(C)CS(C)(=O)=O.c1(N(C)C)ccc(C=O)cn1.C(C)C(C)(C)C.N c1(C(=O)NC2CC3CN(C(CC4CC(=C)C4)=O)CC3C2)cnc2sccn2c1=O Cc1cc(C)nc(N2CCOCC(NC(c3nccnc3C(N)=O)=O)C2)n1 C1(NC(=O)Cc2cnoc2)CN(C(C2CC3C=CC2C3)=O)C2CCCCC12 N1(C(Cc2ccc(C)s2)=O)CC2(CC2)CC1C(N1CCC1(C)CCO)=O c1(OC)cc(C=CC(=O)NCc2nc(Br)cs2)ccc1F N1(C(=O)CNc2cccnc2)CC(C(N2CC3(CSC3)C2)=O)C(F)C1 N1(C(=O)OC(C)(C)C)CC(F)(F)CC1CC.C(=O)C(C)C.[SH](C)(=O)=O N1(C(CCc2ccc(C)o2)=O)CCCC(C(=O)N(C(C)C(F)F)C)C1 C1(NC(C2CSCCS2)=O)CCN(C(C23CCC(CC2)OC3)=O)CCC1(F)F c1(CC)nc(=N)[nH]cc1C(=O)NCCC(C)CCNC(=O)COC(C)C C(=O)(C(CC(C)C)N(C)C)N1C(CCNC(c2c(C)scc2)=O)CCC1 Cc1cc(C(=O)NC23CC(C2)N(C(C2CC(N(C)C)C2)=O)C3)cc(C)c1O C1(C(=O)NCCOCC(=O)NCC(C)OC)CCC=CCC1 C=Cc1cc(C(=O)NCC2CN(C(C3CCCC(F)(F)C3)=O)CC2C)cc(F)c1 c1(C(N2CCC(NC(=O)NC(C)(C)C)C2)CCOC)ccc(F)cc1Cl C1(NC(c2conc2C2CCCC2)=O)CCCC(NC(C23CCOCC2C3)=O)C1 N1(C(CCC)=O)CCCC(C2(NC(=O)CC3CCN(C(C)=O)CC3)CC2)C1 c1(N2CCc3c(nc(C)o3)C2)ccc(S(=O)(=O)NCC2C(C)C2(F)F)c(Cl)c1 C12(C(N3CC(C)(NC(c4cc[n+]([O-])cc4)=O)C3)=O)CC3CC(CC1C3)C2 c1(OC(C)C)ccc(C(=O)NCC2(C)CC2)nn1.c1(C=O)ccncn1.N C1(CC=C)CC2CCC(C1)N2C(=O)CC.C12(C=O)CC(F)(C1)C2.C(N)=O c1(C(C)=O)cnc(C)c(NC(=O)NC(c2ccc(N(C)C)cc2)C)c1 CC1CCCN1C(c1ccnc(C(F)F)c1)=O.c1(C(=O)N)cnc(S)n1C1CC1 C(CCCCC(=O)NC(C)C(C)C)NC(=O)OCC.C(=O)C.C(N)=O.N N1(C(C(=Cc2ccncc2)C)=O)CCC(N(C)C(c2nc(C)nn2C)=O)C(C)C1 C1(CNC(CSC)=O)CCCN(C(=O)Cc2c(C)n[nH]c2C)C1c1ccccc1 c1(C(N(CCNC(C2C(=C)C2)=O)CC)=O)n[nH]c2c(C)cc(Br)cc12 c1(-c2c(C(=O)NCC3C(NC(C(C)N(C)C)=O)C3)c[nH]n2)cccc(F)c1 c1(C(=O)OCCCOc2ccc(Br)cc2F)cc2c(nn1)CCC2 N1(C(C(=O)NCCC(N)=O)=O)CCCC(F)C1.C1(C(=O)N)CC1.C(N)=O C1(CNC(c2c(C)oc(C)c2)=O)CC2CCC1N2C(C12CCC(C1)OC2)=O C(=O)(C1CCCc2c[nH]nc21)N1CC(C(C)(C)O)(CNC(C2(C)CCC2)=O)C1 C=CCC(C)(C)C(=O)N(CCC(=O)Nc1cccnc1COC)C c1(CCC(=O)N(CCOCCN(C(CCC#C)=O)C)C)ccnc(C)n1 C#CC1(C(N2CCC(N=[N+]=[N-])CC2)=O)CCN(C(=O)CCC(N)=O)CC1 N1(C(C)=O)CCC(C(=O)NC)CC1.C1(CC=O)CCNC(=O)C1.C1C=CCC1 C(=O)(C1CCc2c[nH]nc21)N1CC2(CN(C(c3c(C)nc(N)cn3)=O)C2)C1 C1(CCNC(C2CN(CC)C(=O)N2)=O)CCCN(C(c2ccc(Cl)cc2)=O)CC1 N1(C(c2cnc(CC)s2)=O)CC(NC(=O)C(F)C(C)(C)O)CC12CCCCCC2 Cc1cc(C(=O)N)cc(C)c1F.C1C(C)CCCN1C(=O)CN(S(C)(=O)=O)C N1(CC(=O)N(CC=O)C2CC2)C(=O)CCCC1=O.c1(CC)nc(C)cs1 CCCCCC(O)CNC(=O)CCC1(NC(=O)CC2COC(=O)C2)CCCC1 c1(C(=O)NC2CC(CNC(CCCC#C)=O)C23CCC3)cnc2c(c1)COCC2 c1(N(C)Cc2nc(C)sc2)nc2c(c(=NCC34CCN(CC3)C4)[nH]1)COCC2 c1(CC(C)NCC(COCC(C)C)O)ccnn1C c1(C(=O)NC2CCN(C(C3=NOC(C)C3)=O)CC2O)ccc2cc(Cl)ccc2c1 Cc1nccnc1C(C)OC(C1(Cc2ccccc2)CCC1)=O C1(C(=O)NC2C3(CN(C(c4c(C)c(F)ccc4)=O)C3)CC2)CCc2ccnn2C1 N1(c2c(OC)cnc(SC)n2)CCN(Cc2cc(O)c(F)c(F)c2)CC12CC2 C1(CNCC(C2CC(F)(F)C2)(C)N)CCCCC1N c1(C(=O)NC(CNC(CC(COC)(C)O)=O)(C)C)ccc(=O)n2c1CCCC2 C(O)(CC(=O)N1CCN(c2cc(F)cnc2Br)CC1)(C(F)(F)F)c1nc(C)c(C)o1 CC(C)(C(=O)N)C(N)=O.C1(C=O)CCCN(S(C)(=O)=O)C1.C(C)C1CCC1 c1(Nc2c(Br)cc(C)c(C)c2)ccc(N=c2[nH]cnc3cnccc23)c(F)c1 C(=O)(C(CC(F)F)N(C(=O)CC)C)N(CCC(=O)OCC)CC=C C1(CNC(C(C)N(C(=O)CCC2CCCN2C)C)=O)CCOCC1 C1(CC(=O)NC(CCCC)CNC(=O)Cc2ccc(O)nc2)CCC(F)(F)CO1 c1(C(N(C(C)C(=O)NCC(C)CC2CC2)C2CC2)=O)cnc(O)c(F)c1 N1(C(CCSC)=O)CCC2C(NC(c3ccnc(N4CCOCC4)n3)=O)C12 C1(C=O)CCOC2(CCCC2)C1.C1CCCC1.C1(C(=O)NC)(COC)CCC1 C1(NC(COCCC)=O)CN(C(C2CCCOCC2)=O)CC(C)(C)C1 c1(N(C)C)ccc(Br)c(C(N2CCCCC2CCC2CCCN2)=O)n1 c1(CCNC(=O)OC(C)(C)C)ccc(-c2csc(C)n2)cc1.C1CCC2CC2C1 Cn1nc(CNC(c2cnc(N)cn2)=O)cc1C(=O)NCC1CC(C)C1 O=C1CC(C(=O)NC2C=CC(C)C2)CCN1.c1(C=O)cncc(C(F)(F)F)c1 CC(C(C)(C)C(=O)N1CCCC(CO)CC1)NC(=O)CCC1CCC(=O)C1 N1(C(C2C(C)CCC2)=O)CCOCC1C(=O)NCCCCO n1(CC(N2C(CC)CN(C(=O)C(C)SC(C)C)CC2)=O)nc(C)c2cccnc12 N1(C(CCOC(C)C)=O)CCC2CCCC12CNC(=O)C=Cc1cnccn1 N1(C(CC(C)SC)=O)CCC(NC(c2cc(C#N)c(O)nc2N)=O)C2(CCC2)C1 Cc1nc(NC2CCN(C(=O)Nc3cccc(C)c3C)C2)c2c3c(sc2n1)CCC3 C(=O)(C(C)(C)CCCNC)OCC(=O)OCC.C1(CC(N)=O)CCCC1 C(=O)(C(C)CC(C)(C)C)N1CCCC(CC=C)(NC(Cn2ncc(C#C)c2)=O)C1 c1(C(=O)NC(C(=O)NCCCC(C)(F)F)CCC2CCC2)cc2ncccc2[nH]1 Cc1cc2n[nH]cc2cc1C(=O)N(C)CC1(O)CN(C(=O)C(C)(O)C2CCC2)C1 Cc1cnc(NCC2CN3CCN2CC3)c(S(=O)(=O)N2CCC(C(F)(F)F)C2)c1 C(=O)(C(N)CCS(C)=O)N(C)Cc1ccc(Cl)c(C(F)(F)F)c1 c1(OC)ccccc1C(C(=O)NC1CCCC1NC(C1OCCCO1)=O)OC C1(C(=O)NCC(C2CCCCN2C(=O)CS)(C)C)CCOC(=O)CC1.C1CC1 c1(SCC(=O)NC23CC(NC(C(CC)C)=O)(C2)C3)cccc[n+]1[O-] C(=O)(C(C)(C)C(=O)NCCCC)N(C)C.c1ccc(Cl)cc1.C1(C(=O)N)CC1 CN=S1(=O)CCN(S(=O)(=O)c2nc(C(=O)OC)cs2)CC1 N1(C(Cc2scc(C)n2)=O)CCC(C)(CNC(=O)CN2CCOCC2)CC1 C(=O)(C#CC(=O)NCc1ccccc1)N(C)C.C1(C(N(C)C)=O)CC1(F)F N1(C(c2c(C)ocn2)=O)CCN(C(c2ccc(Br)c(Br)c2)=O)CC1CC#N c1(COC)ccccc1.C1(NC2CC(CC)(CC)C2)CCC(c2nc[nH]n2)CC1 C1(C(N(C2(C(C)=O)CC2)C)=O)CC2CCC(C1)O2.C1CC(=O)N1 C1(CC#C)(C(=O)NCC2CCC2)CC=CCC1.C1(C=O)CC1.C(C)C.N Cc1cc(C(=O)NC2CC2CNC(c2ccsn2)=O)n2ncnc2n1 N1(C(c2cc(C(=O)OC)[nH]c2)=O)CCN(C)CC1CNC(=O)C(C)(C)O CCCCC(C(=O)NCC(CCOC)NC(C1(O)CCOCC1)=O)C(C)C C1C2CCCCCC12.Cc1cc(CNC(=O)COC2CCOC2)oc1C(=O)N c1(C(=O)O)ccc(Br)c2nc(C=Cc3nccn3C(F)F)oc12 Cc1cc(C)c(C(N2CCOCC(C)(CNC(C34CC(O)C3C4)=O)C2)=O)cc1C Cc1ccc2ncc(C(=O)N(C(C)CNC(=O)CN3CCC(C)C3)C)n2c1 C=CCC(C)C(=O)NC(C1CN(C(c2cnc(C3CC3)[nH]2)=O)C1)C Cc1nc(C(C)NC(=O)NC(C)CN2CCCC2=O)cs1 Cc1cc(C)nc(CNC(=O)CC2CN(C(c3c[nH]c(C)c3)=O)CCO2)n1 C(C)(C(=O)NCCN(C(=O)CCC1CCCO1)C(C)C)OCCOC N1(C(C(c2ccc(C)cc2)O)=O)CCC(CO)(CNC(=O)Cc2cnsc2)CC1 C1(N(C(=O)CCc2nc(C)cs2)CC)CCN(C(=O)C(=O)NC(C)C)CC1 C1(CNC(CC2(C=C)CC2)=O)CC(NC(=O)C=Cc2cnccn2)C1(C)C CCC(CCCC(=O)NCCc1cnn[nH]1)NC(=O)C1CC1 C(C(=O)NCCN(C1CCCCC1)C(=O)CC)(C(C)C)OCC CCC(CNC(=O)CC1(OC)CN(C(=O)C=Cc2ccoc2)C1)CCO C#Cc1cccc(CN2CCNCC2C(=O)NCc2cc(C)nc(C)c2)c1 C(C(C)C(C)C(=O)NCC1CCCC1C(=O)N(CC=O)C1CC1)OC.O Cc1cc(Cl)cc(C)c1C(=O)NC1CCN(C(c2cn(C(C)C)nn2)=O)CC1 CN1CCOCC1C(=O)NCC1COCC1NC(=O)CCc1ccc(F)cc1 CC1(CNC(=O)CN2CCCCC2=O)CCCN1C(C1CC=CCC1)=O C(=O)(C1=NOC(c2ccccc2)C1)NC1CCC(N(C)C(C2CCCO2)=O)CC1 O=C(CCCCCCn1cc(CC2(F)CC2)nn1)NCc1ccccc1 C1(C(N2C(C)CC(NC(c3c(C)nc(C4CC4)o3)=O)C2)=O)CC2CC(=O)C1C2 Cc1cc(C(=O)N(C)CC2CCN(C(=O)CSC(F)F)CC2)[nH]c1C c1(OC)ccc(C(=O)NC(C)CCN(C(=O)CCC(F)F)C)c2ccncc12 Cc1ncnc(C)c1C(=O)NC1CC2CC1CN2C(c1nc(Cl)c(Cl)s1)=O C=CC1CC(N=c2cc[nH]cc2S(=O)(=O)NCc2ncn(C3CC3)n2)CCO1 C1(CC)CNC(=O)CN1C(=O)C(F)C(C)CNC(=O)CSC(C)(C)C C1(C(N2CCC(C)(CCNC(=O)CC3C=CCCC3)C2)=O)CC2(CCOCC2)C1 c1(C(=O)NC(C)CCNC(c2ccc(Cl)s2)=O)cnc(C2CC2)nc1 C=C(C)CC(C(=O)Nc1cc(C)cnc1C)NC(c1cc(C(C)C)on1)=O C#CC1(C(N2CCCC2CCN(C)C)=O)CN(C(c2ccccc2)=O)C1 N1(C(C(C)SC(C)C)=O)CCCC2(C1)CN(C(=O)CSc1nccn1C)CCO2 Cc1cncc(C(=O)NC2CC(C)N(C(c3cnc(C4CC4)nc3)=O)C2)c1 C1(CC=O)CC2(C1)CN(C(c1cncc(F)c1)=O)C2.c1(CCC)ncc(C)s1.N N1(C(CCc2cc(C(C)=O)c(C)o2)=O)CC(C)C(F)(F)C1.C(=O)C=C1CCC1 CCCCCCCCCC(CC)N1CCC(c2ccccn2)CC1 C1(C(N2CCC(c3cnn[nH]3)C2)=O)CC2(CCN1C(C1SCCS1)=O)CC2 N1(C(COC2(C)CN(C(C3(C)C(C)C3)=O)C2)=O)CCC(CO)C(C)(C)C1 N1(C(=O)CCF)CCCC12CCCN(C(C1(Br)CC13CCC3)=O)C2 C1(C)(C(=O)NCC2N(C(CCCCC)=O)CCC2C)CCC(F)(F)C1 C(c1c(C)noc1C)=CC=O.c1(CC)cnn(CC(=O)N)c1.C1(O)CCC1.C Cn1cc(C(=O)NC2CCCC23CN(C(=O)CC(C)(C)O)C3)c(=O)n(C)c1=O C1(C(=O)N)CNC(=O)N1.C1(O)(CC)CN(C(C2CN(C3CCOCC3)C2)=O)C1 c1(CNC(c2cc(OCC)no2)=O)ccccc1.C(=O)(CC(C)(C)C)NC N1(C(C2Cc3n(cc(C)n3)C2)=O)CC2(C1)CN(C(c1ccoc1Cl)=O)CC2CO N1(C(c2c(C)scc2)=O)CCC2CCC(NC(c3cccnc3OC(C)C)=O)C12 N1(C(C)=O)CC2(CC(NC(=O)CCc3ccn(C)n3)CO2)C1 N1(C(C=CCCC(C)C)=O)CC2CCC(C1)N2C(c1cnco1)=O O=C1NCCCc2occ(C(N3CCOC4(C3)CN(C(=O)CC(F)(F)F)C4)=O)c21 N1(C2CCCN(C(COCC(C)C)=O)C2)CCN(C(c2cccs2)=O)CC1=O c1(C(N(CC(O)CNC(C2CCCO2)=O)C)=O)cc(N2CCCC2)ccn1 N1(C(C)=O)CCC(C(C)C)CC1.C(=O)C(C)(C)c1ncco1.C(=O)(CS)OC C(=O)(C1(C)CCn2c(C)nnc21)NC1C(NC(CCCOCCC)=O)CC1 c1(C(=O)NCC2(OC)CN(C(c3cncc(Cl)c3)=O)C2)cnn2c1CCCN2 n1(C[Si](C)(C)C)ncc(F)c1CNCC1CCCCS1 N1(C(Cn2c(C)ncc2)=O)CC(C(=O)Nc2cnc(Cl)c(Br)c2)CC(F)C1 N#Cc1ccc(Cl)cc1S(=O)(=O)N1CCN(C2CCCC2C2CCCC2)CC1 C1(CNC(c2ccc(OC(F)(F)F)nc2)=O)CCC2CNCC12 C(=O)(C1CCCc2nn(C)cc21)N.C1(NC(COCCC(C)C)=O)CCCC1C C12(CNC(c3cn(-c4ncccn4)cn3)=O)CCC(CC1)N2C(C1CC1)=O c1(C(=O)OC)ccc(CNC(N2CCCCC2CC=O)=O)cc1F.C(C)(C)C c1(OC)cc(Br)ccc1C(N1CCC(C)(O)CC1)C(=O)NCc1ccco1 N1(C(C2CC(=C)C2)=O)CC(C)CCC1CNC(c1ccc(OC)c(Cl)n1)=O c1(Sc2n(C)cnn2)ccc(-c2nc(C(F)F)nn2CC(F)(F)F)cc1 C(C(C)(C)C)N(C(c1nc(Cl)cs1)=O)CC.N1(CCC(=O)N)CCC(F)C1 C1(C)(C(=O)NCCCN(C)C(C2(C3CCCO3)CCCC2)=O)CNC(=O)C1 C1(CNC(c2c(C)cco2)=O)CC2(CO1)CN(C(=O)C(c1ccc(F)cc1)F)C2 N1(C(C(C=CC)O)=O)CC2C(CC(=O)NCCOC3CCCC3)C2C1 N1(C(C2CCC(C)C2)C(=O)NC(CC)C)CCC(OC)CC1 Cc1ccc(C(=O)NC2CC3CC(NC(=O)CCC(N)=O)CC23)c2ccccc12 C1(C(N2CCN(C(CNC(=O)OCC)=O)C(C)C2)=O)CCn2nncc2C1 C1(CCC(=O)N(C2(C)CN(C(c3ccccc3CO)=O)C2)C)CCCCN1C c1(CCC(=O)NCC2(C)CCN(C(c3cnsc3)=O)C2)ccc(O)c(Cl)c1 C1(CC)(NC(=O)CC2CCOCC2)CCN(C(=O)C)CC1.[SH](=O)(=O)CC.O c1(C(N2CC(CNC(CC3C(C)=NNC3=O)=O)OCC2)=O)c(C)ccc(C)c1C C1(NC(CC2CC(=C)C2)=O)CN(C(=O)C(c2ccc(CC)s2)=O)CC1(C)C c1(C(N2CC3C(C(N4CCCC(C)CC4)=O)C3C2)=O)ccc2cc[nH]c2c1Br S(=O)(=O)(c1cccc(F)c1)N1Cc2c(-c3c(OC)c(F)ncc3)n[nH]c2C1 C1C(C2CC2)CCN1C(=O)C1=NNC(=O)C1.C1(C(C(=O)N)OC)CCCOC1.C C1(C(=O)NCCC(CNC(c2cnc(OC)nc2)=O)O)CCCC(C)CC1 N1(C(c2cnn(C)n2)=O)CC2CC(NC(=O)CC34CCC(CC3)C4(C)C)CC1C2 c1(N2CCC(CNC(C3CCCN3Cc3c(C)c[nH]n3)=O)C2)ccc(F)cc1 c1(CC(C)NC(C)C(=O)NC2CCCCC2)nc(-c2ccccc2)no1 N1(C(CC(C)(C)n2cc(C(=O)OCC)nn2)=O)CCN(C(=O)CC)CCC1C C1(C(=O)NC(CCC)C2CCCC2)CCN(C(=O)C=C(C)C2CC2)C1(C)C C(=O)(CC(C)C(F)(F)C(F)(F)F)Nc1c(CC)cccc1CC CCC(C(=O)NC1(CNc2cc(=O)n(C)cn2)CCOCC1)C(C)O Cc1noc(C)c1C(=O)NC1CCN(c2nccn2C)C1 C1(C#N)(C(N2C3C(NC(C4(COC)CC4)=O)C(C3)C2)=O)CCOCC1 C1(NC(c2csc(Br)c2)=O)(CNC(c2ccon2)=O)CC2CCC1CC2 c1(C(=O)NCC2(C)N(C(C3CC(CCC)C3)=O)CCC2)ncc2c(F)cccn12 C1(C(N2C(C=C)COCC2)=O)COC2(C1)CN(C(=O)CC(O)C(C)C)C2 C1(CC(=O)NC(C)CNC(=O)CCOCC2CCC2)CCCC(=O)N1 Cc1cc(-n2cc(C3CN(C(C4C=CCS4)=O)C3)nn2)cc(C)c1 N1(C(C(C)=CC(C)(C)C)=O)CC2(CC2)CC1CC(=O)NOCCCC1CC1 CC1CC(C(=O)N2CCC(CNC(c3cnc(C(C)C)o3)=O)C(O)C2)=NO1 Cc1nccnc1C(N1CC(NC(=O)Cc2cnns2)C2CC12)=O C1(C(C)C)CN(C(=O)Cc2ncncc2Cl)CCN1C(=O)CN(C)C C1(NC(CC=C)=O)(CNC(c2cc(O)nc(N(C)C)n2)=O)CC2CCC1C2 C(=O)(C1OCCn2ccnc21)NCC(C)NC(=O)C(C)Cc1ccccc1 C1(C(=O)NCCCCC(C)NC(C(c2ccc(C)s2)C)=O)C2CCC1(C)C2(C)C C(C)(N=c1cc(C)nc(N(CCCC(C)O)C)[nH]1)c1nc(COC)sc1 CS(=O)(=O)C(C(=O)N1CCC2C(NC(C3CC4(CCC4)C3)=O)C12)C1CC1 N1(C(C(C=C)O)=O)CC2CCC(N(C(=O)CSc3nc[nH]n3)C)C2C1 C(=O)(C1=NOC(C)C1C)NC1CC(CC(N2CC(C=C)C(O)C2)=O)C1(C)C c1(C(=O)Nc2ccc(C(=O)OCC)c(C)c2Br)csc2c(OC)cccc12 c1(C(=O)N)cc([N+](=O)[O-])cc(C)n1.c1(CC)sccc1C(=O)N(C(C)CC)C N1(C(C)=O)CCOC(CN(c2ccc(Cl)o2)C(=O)Cc2ncccn2)C1 C12(C(N3CC(CCNC(c4ncncc4F)=O)C3)=O)CCCN1CCC2 CCC(CC)(CO)C(=O)N1CCC(C(F)F)(CNC(=O)C(C)(C)c2ccns2)C1 c1(C(N2CC(CNC(C3C(C)CCC3)=O)N(C)CC2)=O)c(F)cc(O)cc1F Cc1cnc(NC(c2ccoc2)C)c(S(=O)(=O)N(CCS(N)(=O)=O)C)c1 CC(C)C#CC(=O)N(C1CCN(C(C2CC(C)(F)C2)=O)C1)C c1(C(N2CCC(NC(CC(C=C)CC)=O)C(CC)C2)=O)cc2c([nH]1)CCCC2 C1(NC(=O)CC2CCN(C(C3CCC=CCCC3)=O)C2)CNC(=O)C12CC2 CC(C(=O)NC1CC(N(C(=O)CC2CCSC2)C)C1)n1cnnn1 C1(OCCNC(CCOCCC)=O)CCN(C(=O)C=CBr)C1 CCCCCC(O)C(C)C(=O)NC(CC)(CC)CCNC(=O)CS.CCN(C)C C(=O)(CCCC(=O)N(C)C)NC1CCN(C(c2cnc(CC)s2)=O)C1 c1cnc(C#N)c(C(F)(F)F)c1.n1(CC=O)cc(C#N)c(C(=O)N=c2cc[nH][nH]2)n1 C(=O)(CCCOCCC)NC(C(=O)NCCOCCC#C)c1ccoc1 Cc1cnn(CCC(=O)N(C(c2cn(CCCC(=O)O)nn2)C)C)c1 c1(C(C(=O)N(CC(C)NC(=O)C(C)CC2CCCCC2)C)(C)C)ccc(Cl)nc1 C(=O)(C1CCCn2nccc21)NC(C(C)NC(Cc1nnc(C)o1)=O)(C)C c1(OC)cnnc(C(=O)NC2CC(C)(C=O)C2)c1.C1(CC)CC(F)(F)C1.N C1(NC(c2ccc(C)cc2)=O)CC(F)CN(C(=O)Cc2nncn2C)C1.CC(=O)N N1(c2n(CCCOC)c(-c3nc(O)sc3C)nn2)CCN(C)C(C)(C)C1 Cc1oc([N+](=O)[O-])cc1C(=O)NC.C1CCCN1C(C1(n2cccn2)CC1)=O.C C(=O)(C#CC1CC(F)(F)C1)NCC1(C)CCCN1C(c1ccc[n+]([O-])c1)=O C1(CC)(CO)CCCN(C(=O)CN(C(c2cc(Cl)no2)=O)CC2CC2)C1 C=C(C)CC(=O)NC(CNC(=O)C=C(CC)CC)CCC c1(C(N2CCC(F)(CNC(C3(CO)CCOC3)=O)CC2)=O)cccc(F)c1Cl N1(C(C2(NC(C3CCCN3C)=O)CCN(C)C2)=O)CCC(=C(F)F)CC1 N1(C(CNS(NC)(=O)=O)=O)CCC(CNC(=O)C=CBr)C(F)(F)C1 C1(NC(CCCn2c(C)ncc2)=O)CCC2CC1CN2C(=O)COC1(C)CCC1 C(N(C)N1CCC2CC(F)(F)CC2C1)c1ccc(N(C)C)cc1 CC(CN=c1[nH]c(N2CCc3c[nH]c(=N)nc3C2)nc(=N)[nH]1)S(C)(=O)=O C1(NC(C(C)C2CC2)=O)CCCCC1CNC(c1cc(=O)n(C)o1)=O O=C(C(O)CCc1ccccc1)OCCCOc1ccccc1 c1(CC)ccsc1C(=O)NC(c1ccccc1)CNC(=O)COC(C)C N1(C(=O)NCc2cocn2)CC(O)C(O)C12CCOCC2 N1(C(C23CC(OC)C2C3)=O)CCN(C(=O)CC2CC=CC2)C(CC2CC2)C1 C(=O)(C(O)CCCNC(=O)C=CC1CCCN1C)NCc1c(CC)con1 c1(C(=O)NC(CN(C(=O)Cc2ccon2)C)(C)C)cc2c(O)cc(Cl)cc2[nH]1 Cc1ccc(-n2cc(C(c3nnnn3C)NC3CCCN(C)C3=O)nn2)c(C)c1 Cn1c(C(N2CCCCC2CCn2cncn2)=O)nc2ccccc12 C(N=c1[nH]c2ccc(F)cc2o1)C1OCCCN(C(CSCCCC)=O)C1 N1(C(C(=O)Nc2cc(OC)c(Br)cc2OC)=O)CCOC2(CCC(C)(C)C2)C1 C1(Cn2cc(C(C3CCOC3)C)nn2)(C)CC12CCC2.C(=O)CC1(C)CC1 Cc1ccc(C(N2CCN(C(C3CCC(C)O3)=O)C(C)C2)=O)c(C)c1 CP(C)(=O)C(CC(=O)NC1CN(C(C2CC2F)=O)CC2(CCC2)C1)P(C)(C)=O N1(C(C(CCC)CC)=O)CC2CCC(C1)N2C(=O)C(C)(C)C1CCOCC1 Cc1ccc(C(=O)NC(C)C(C2CCCCC2)NC(=O)CCc2ncc[nH]2)o1 c1(CCC(=O)NCC2C(NC(C(COCC)C)=O)C2)ccc(O)cc1 N1(C(C(C(C)(C)O)(C)C)=O)CCC2CN(C(c3cnc4ccnn4c3)=O)CC2C1 c1(C(=O)NCC(CC)(C)NC(c2ccc(C(C)(C)C)cn2)=O)oc(C)cc1C CC(CCCCNC(c1ccnn1C(F)F)=O)NC(=O)CCCF c1(C(C)C)ncncc1C(=O)NC(C1CN(C(C)C(=O)Nc2nccs2)C1)C N1(C(C(=O)NCC(F)F)=O)CCOCC(C(=O)NC2(CO)CC(O)C2)C1 N1(C(c2cc(CNC(C(C)CC3CC3)=O)[nH]n2)=O)CCC2(CCSC2)C1 Cc1nsc(C)c1C(=O)NCC1CCC1.c1(C(=O)N)ccoc1CC(N)=O Cc1nn(C)c2c(NCC(c3ccccc3)F)nc(=NCCc3ccco3)[nH]c12 CC1CN(C(C2COCCN2C(c2sccc2F)=O)=O)CC2(CCC2)O1 C1(CNC(C(CC)NC(C)=O)=O)C2CN(Cc3ccc(OC)cc3)CC12 N1(C(c2c(CC)n(-c3ccccn3)nc2)=O)CCS(=O)CC1(C)C c1(CC(=O)NC2C(C)CCN(C(COC(C)C)=O)C2C)ccc2cccnc2c1 Cc1cc(Br)c(F)cc1C(N1CC(CNC(=O)CC(C)C)C1)=O.C(N)=O.N C1(CNC(C(CC)(F)F)=O)N(C(c2cc(F)c[nH]2)=O)CCCC1(C)C c1(C(=O)NCC2(C)N(C(Cc3n(C)ccc3)=O)CCC2)ccc(Br)c(Cl)c1 CCC(C(=O)N1CC(C2CC2)(C(=O)NCC(F)(F)C(C)(C)O)C1)C(C)(C)CC C(=O)C1=NOC(c2ccc(F)cc2)C1.C(C(C)=CC=O)NC(C)=O.C1CC1.N C#CCC(C)(C(=O)N1CC(OCC)C1)NC(c1cc(C#N)oc1C)=O CCCC(C)CC(=O)NC1(C)CCN(C(c2sc(SC)cc2C)=O)CC1 CC1CN(C(c2cnc[nH]2)=O)CCC1NC(C1CCOC(C)(C)C1)=O C=CC(CCC)CC(=O)NCCC1CN(C(=O)Cc2cc(O)nnc2O)CC1C C12(NC(C(C)OCCC(C)C)=O)CCCC1N(C(=O)Cc1nccs1)CCC2 c1(N(C)Cc2c(CC)cccc2)nc(N2CCN(C=O)CC2)c2ncsc2n1 N1(CC(=O)N(C)C)CCN(C(=O)C(c2ccccc2)n2cccc2)CC1 CN1CCCN(C(c2cccc(-c3ccc(O)nn3)c2)=O)CC1 c1(-c2c(C(=O)Nc3n(-c4c(OC)cccc4)ncc3)c[nH]n2)ccc(F)c(Cl)c1 c1(C(=O)NCC2(NC(=O)Cc3cnc[nH]3)CCOC2)cn2ccccc2n1 c1(C(=O)NCC(C(C)C)NC(=O)C(C)n2cccc2)cccc2sccc12 C1(NC(c2n(CCN(C)C)ncc2)=O)CC2CC(NC(=O)C3=CCCCC3)CC12 c1(CNC(=O)C(F)C2CCC2)ccc(Cl)c(C(F)(F)F)c1 C(C(Cl)C(C)(F)F)NC1(c2nnnn2C2CCOCC2)CN(C(C)=O)C1 c1(COC)nc(C(=O)NC(c2nc(C3CC3)n[nH]2)C)cs1 C1(C2CN(C(c3cnc[nH]c3=N)=O)C2)(NC(C(C)OCC)=O)CC1 c1(C(=O)NC2(CNC(C3(C#C)CCC3)=O)CCCCC2C)cnc2[nH]ccc2n1 C1(NC(CC(=C)Br)=O)CC2(CCN(C(C3(C)CC(C)C3)=O)CC2)C1 c1(C(N(CC(CN(C(C(C)C2CC2)=O)C)O)C)=O)ccc(CC#N)cc1 c1(C(N(CCN(C(CN2CCN(C)CC2)=O)C)C)=O)cc2n(n1)CCCO2 N#Cc1c(C(=O)NC2(CNC(=O)COc3ccccc3)CC2)cccc1F C1(NC(c2c(C)cncn2)=O)COCCN(C(=O)CCc2nc(=N)[nH][nH]2)C1 c1(NC(CCNC(C(CC)(C)OC)=O)=O)ccc(O)c(OC)c1 C12(CNC(CCc3c(C)ncs3)=O)CC(CN1C(c1nc(Cl)cs1)=O)C2 Cc1noc(CCCNC(=O)C(C2CCN(C(=O)Cc3cn[nH]c3)C2)C)n1 C1CC12CCN(C(=O)Cc1ccn(C(F)F)n1)CC2.C(C)(C(=O)NC)=CC C1(NC(C2(CC#C)CCC2)=O)CCN(C(c2ncc(F)cc2N)=O)CC1(C)C c1(C(N2C(CNC(c3coc(C)n3)=O)CC(OC)C2)=O)cc(C)c(N)cc1F C12(NC(=O)C=Cc3ccncn3)CCC(CN(C(C3CCCCC3(F)F)=O)C1)C2 c1(C(=O)NC(C)CCN(C)C(C2(S(C)(=O)=O)CC2)=O)cccc2cnsc12 C1(O)CCCCCC1.C(C)(C)(CC(=O)N)N(C(C(C)(C1(C)CC1)OC)=O)C.C N1(C(C=CC=O)=O)CC2COCCC2C1.c1(C=O)ncc(Cl)cc1F.CC(C)C.O N1(C(c2c(CC)occ2)=O)CC2CC1(C)C2.C1(C(=O)N)(N(C)C)CCOCC1 c1(NC(C(n2cc(C3(CC)COC3)nn2)C)=O)ccc2c(c1)CCCC2 CCC(CCOC)C(=O)N(C1CCCN(C(C2CC(F)(F)C2(C)C)=O)CC1)CC c1(N(C)CC2(CO)CC2)nc(NC2CCN(CC(F)F)C2)c2ncn(C)c2n1 N(C1CN(C(=O)CSS(C)(=O)=O)Cc2ccccc21)C(CC(C)F)=O C(=O)(C1CCCCc2ccccc21)N(CCCNC(=O)Cc1cncnc1)CC C(CN=C(NCC1CCC1)N1CC2CCCCC2C1)c1ccc2nc(C)[nH]c2c1 N#Cc1csc(NC(C2CCN2C(c2cccnc2)=O)=O)n1 c1(C(N2C(C)(C(=O)NCCc3cccnc3)CCC2)=O)cnn2ccccc12 C1(NC(c2oc(CC)c(C)c2)=O)C2CC1CN(C(C1CCCC1C)=O)C2 c1(CC(N(CCC)CCNC(=O)C(O)C(C)O)=O)cc(F)cc2c1OCOC2 N1(C(c2c(C(C)C)occ2)=O)CCC2CCC(C1)N2C(C1CC1C(F)F)=O CC(CNC(C1(NC(c2ccnn2C)=O)CC(CO)C1)=O)CCCO N1(C(C(C(CC)C)O)=O)CCC(NC(=O)CCc2cn(C)nc2C)C2(CCC2)C1 C12(COC)CC(NC(=O)Cc3cnc[nH]3)(CN1C(c1cc[nH]n1)=O)C2 C(=O)(CC(C)C(C)(C)NC(=O)CC1CCOC1)NCCCSCC c1(C(N2C(C(=O)NC(C3CCOCC3)CC)CC(=C)C2)=O)ccc2ncoc2c1 N1(C(C(N)=O)=O)CC2COCCC2(NC(=O)CCOc2ccc(F)cc2)C1 N1(C(C(=O)NCC2(c3ccc(C(F)(F)F)cc3)CC2)=O)CCNC2COCC12 C(=O)(C(CNC(C1CC(F)(CF)C1)=O)C(C)(C)C)NC(C)(C)CO C1(C(=O)N(C(CNC(C2CCCC2)=O)C2CC2)C)(OC)CCCOC1 CC(C)C(O)CC(=O)NCCC1(NC(C2C3CCCC23)=O)CCC1 C1(N(C(=O)Cn2nccn2)C)CCN(C(C2CC23CCCC3)=O)CC12CC2 Cc1csc(C(=O)NC2CC2NC(c2c(Cl)cnn2C)=O)c1C Cc1nc2c(F)cc(NC(=O)C(=O)NCCCCCO)cc2o1 c1(C(=O)N)cccnc1N1CCOCC1.C(CC(=O)NC1CC1)NS(C)(=O)=O Cc1ccn2cc(C(=O)NC(C)CCCNC(c3cccc(C)c3F)=O)nc2c1 Cc1ccc(Cl)c(C(=O)NCC(C)(C)NC(C2CC3(C2)CC(C)C3)=O)c1N C1(N(C(c2ccc(N(C)C)nc2)=O)C)CN(C(c2coc(Cl)n2)=O)CC1(C)C C1(C=O)CC2COCC2C1.c1(C(=O)NC(COC)C2CC2)coc(CC)n1.N N1(C(CC2C(CNC(C(CC)SC)=O)C2)=O)CC(C2=NOCC2)C1 c1(C(C=O)C)ccc(C(F)F)cc1.Cc1ncsc1COCC(=O)N.C(C)C C1(NC(CNC(C)=O)=O)CC(NC(=O)CO)C12CCOCC2.CC(F)(F)F C=C=CC(C)C(=O)N(CC)CC1CCN(C(=O)CCc2cccnc2Cl)CC1 C(=O)(C(F)C1=CCCCC1)N(C(C)C)CCN(C(=O)C(c1ccccc1Cl)O)C C1(C(C)C)C(NC(=O)CN(C)C(c2ccccc2)=O)CCN1C(=O)CC(C)F c1(C(=O)NCCCN(C(C2C(C)C2C)=O)CC2CCCC2)cncc(F)n1 c1(C(=O)NCCC2N(C(C(CC#C)C)=O)CCCC2)ccc(F)c(Br)c1 c1(NC(CC)CNC(=O)CC(C)OC)cc(C(F)F)nc2ncnn12 C1(NC(=O)CCSc2ccccn2)CC(O)CN(C(=O)C=Cc2ncco2)C1 c1(OC)ccc2c(C(=O)NC3(CCCNC(=O)CC(C)(F)F)CC3)c[nH]c2c1 Cc1nc(N2CC(C(=O)Nc3ncnc4ccsc34)C2)c2cc(Br)ccc2n1 C1(NC(c2scc(OC)c2)=O)C2CC3C1C3C2C(=O)NCC(C)(CO)OC C(CC(C)(C)C(=O)NC1(C)CCC1)SC.c1(C=O)cccc(C(N)=O)c1F.N n1(CC)c(C)cc(C=O)c1C.c1(N(CC=O)C(C)=O)ccccc1.CCC.N C1(C(N(CCN(C)C(c2cccc(-n3cccc3)n2)=O)C)=O)CCCC2CC12 c1(OC)ccccc1C(O)C(=O)NCC(C)CN(C(=O)C=Cc1cncs1)C N1(C(CCC#C)=O)CC(NC(c2cnn(C)c2C#N)=O)CC12CCOCC2 Cn1c(C(=O)NC2CCCC2NC(c2cnc3c(c2)NCC3)=O)cc2sccc12 Cc1cnn(C)c1CN(C)C(C1CCC=CC1NC(C1CC(=O)CCO1)=O)=O CC(C)CCC(=O)NCC(C)(O)CNC(=O)CCN1CCNC(=O)C1 C(C(C)(C)C#CC(=O)NCCOC(C)C)NC(c1cccc(C)n1)=O C1(C(N2CC(C)C(F)C2)=O)CCCN(C(c2cc(F)c[nH]2)=O)C1C c1(C(N2CCCC(N(C(c3cc(CC)[nH]n3)=O)C)C2)=O)nc(C)n(C)c1C C1(C(=O)NCC(CCOC)NC(C2(C(C)(C)O)CC2)=O)CCN(OC)CC1 C1CCC2(C1)C(CCNC1CC3CCC(C1)N3)CC2 CC1=C(C(=O)N2CC3CCCC2C3CNC(=O)C(C)(F)F)CCCO1 c1(C(N2CC(N(C)C(C3CCC=CCC3)=O)C(F)C2)=O)nccc2cccnc12 N1(C(C(CC)CC(F)(F)F)=O)CCC2(C1)CN(C(=O)C1=CCC1)CC(C)O2 c1(C(N2CCOCC(NC(Cc3c(C)nsc3)=O)C2)=O)cc2cc(Cl)ccn2n1 C1(C)(NC(COCCSCC)=O)CCN(C(=O)CS)C1.CC(F)(F)F C12(NC(C(CC)CC)=O)CCC(CN(C(=O)C=CCOc3ccccc3)C1)C2 C1(NC(C=C(C)c2ccco2)=O)C2CCN(C(=O)CCc3ccco3)CCC12 N1(C(C2C(=C)CC2)=O)CC(OC)CC(NC(c2c(C)c[nH]c2CC(N)=O)=O)C1 c1(CC)ncc(C(=O)NCCC(C)N(C(=O)CCC2CCC(C)O2)C)s1 Cc1ccc(C)n1CC(=O)N(CCC(=O)NOCC1CC1)C N1(C(c2nc(CC)oc2)=O)CCCC2(C1)CN(C(=O)Cn1cnc(=N)[nH]1)CCO2 c1(CC)ccc(C(C)CC(=O)NC(C)CN(C(=O)C=CCOC)C)cc1 C(CC(C(=O)NOCCC(F)F)NC(=O)C(C1CCOCC1)F)OCC n1(CC)[nH]c(=NC(=O)C(=O)N(C(CC)CO)C)cc1C1CC1 N1(C(=O)Cc2c[nH]nc2O)C2CCCC1CN(C(C13CSCC1C3)=O)C2 N1(C(c2n(CC)cnn2)=O)CCC(C)(CNC(=O)CC2CC(SC)C2)C1 C12(C(=O)OC)CC1CN(C(=O)CCNC(c1cc(C)[nH]n1)=O)C2 Cc1ccn2nc(C(=O)NC)nc2n1.C1(C=O)C2CS(=O)(=O)CC12.C1CCC1 n1(CCOC)nc(C(=O)NCC(C)CC)ccc1=O.C1(C=O)CCCC(=O)N1.N c1(C(N2CC(CNC(COC(C)(C)C)=O)C2)=O)cccc(-n2ccnc2)c1 c1(C=O)cc(N)ccc1F.Cc1ccc(SCC(=O)NCC2(O)CCC2)cc1.N N1(C(CCOCC)=O)CCN(CC2CC2)CC1.C(c1cccnc1)=CC(=O)N c1(C(=O)NC2CN(C(=O)CN3CC4CC4C3)CC2C2CC2)nccc2cc[nH]c12 N1(C(C=CCC)=O)CC2CS(=O)(=O)CC2(NC(c2cnn(CC)c2Cl)=O)C1 N1(C(C2CCCC(NC(CCC(N)=O)=O)CC2)=O)CCc2nncn2CC1 c1(C(N2CCC(N(C(CN(C)CC)=O)C)C(C)C2)=O)c[nH]c2ccccc12 N1(C(CCC(C)SC)=O)CCC2(CCC2)C(CNC(c2nn(CC)nc2C)=O)C1 Cc1cccc(C)c1NC(C1CCN(C(=O)CN2CCC(F)(F)C2)C1)=O C=CCCC(C(=O)NCC(C)SC)NC(C1CCCC(C#N)C1)=O Cc1ccc2c(c1)CCC2C(=O)NCCCN(C(=O)CCC1CCCO1)CCO c1(OC)cc(CO)ccc1C(=O)NC1CCN(C(C2CCC(=O)O2)=O)C1 N1(C(C(c2ccccc2)OC)=O)CC2CC2C1CNC(c1ncn(C)n1)=O N1(C(c2cnc(C)s2)=O)CC2(CCC2)CC1C(=O)NCCC12CCCC1C2 Cc1cccc(CC(=O)NC2(C)CC(NC(=O)Cc3ccsc3C)C2)c1F C12(NC(=O)COCCCF)CCCCC1CN(C(c1c[nH]c3nccc-3c1)=O)C2 CC(C)CC(C)(O)C(=O)Nc1cccc(NC(c2cnc(C3CC3)s2)=O)c1 N1(C(C(C(C)C)O)=O)CCC2(NC(=O)Cc3ccnc(O)c3)CCCC12 C1(C(N2C(C(=O)N(CC(C)(F)F)C)CC2C)=O)(OC)CCCCC1 C1(O)(CNC(CCNC(N)=O)=O)CCCN(C(C2CCC=CCCC2)=O)CC1 C1(NC(COC)=O)CC2(C1)CC1(CC(NC(C3(C)C=CCC3)=O)C1)C2 N1(C(COCCCC#C)=O)CCCC1C1(C(=O)NC2CC(C=O)C2)CC1.O Cc1cc2[nH]c(C(N3CCC4(C3)CN(C(=O)CCCn3ccnn3)C4)=O)cc2s1 c1(C=O)ccccc1F.c1(C(=O)OC)ccccc1CNC(=O)N.C1COC1 c1(C(N2CC3C(NC(CSCC)=O)(C3)C2)=O)cc(P(C)(C)=O)cs1 C=CCC(CNC(c1cc(OC)cnn1)=O)C(=O)NC(C)(CC)C(F)(F)F c1(CCC)ccc(N)c(C(=O)NC2(C)CCN(C(c3cnsc3C)=O)C2)c1 c1(C(=O)OC)cccc2c(CNC(=NCCO)NC(C)C)c[nH]c12.C1(C)CCC1 c1(C(=O)NC(C2CCN(C(c3c(CC)[nH]nc3Cl)=O)C2)C)cn2cccnc2n1 Cc1cc(C(N2CC(C)(C)CC2CNC(c2cscn2)=O)=O)c(C)cc1Br N1(CCC(C)C)CCCC1C(=O)NCC(C)(O)CNC(c1cncs1)=O CCC(C)C(CNC(=O)CCN(C(=O)CCc1ccnn1C)C(C)C)CO C1(CNC(C2CC3COCC3C2)=O)CC2CCC1N2C(c1csc(Cl)c1)=O c1(C(N2C3CN(Cc4cccc(OC)c4F)C(C3)C2)=O)ccc(C#N)c(Cl)c1 N1(C(CSCC(C)C)=O)CCC(CCNC(=O)C(C)Sc2ccccc2)C1 N1(C(C(C=C)c2ccccc2)=O)CCC2(CC1)CC2NC(=O)CC1CCCC1 CC1COCC(C(=O)NCCC2(NC(C3CC=CC3)=O)CCC2)O1 C=CC(CC)CC(=O)NC(C)C(C)NC(c1cnc(-c2ccccn2)nc1)=O CC1(C)CC(COC(c2cccc(OC(F)(F)CC(F)(F)F)c2)=O)OC1=O c1(CC)ncncc1C(N1CC(O)(C(C)(C)C)C1)=O.C(=O)CCC(=O)N(C)C C1(N(C)C(C2CC23CCC3)=O)CN(C(=O)C=O)CC2(CC2)C1.CC(F)(F)F.N c1(C=O)ccc2nc(O)[nH]c2n1.CCCCN(C(=O)COCc1nc[nH]n1)C.N c1(C(=O)NCC2(F)CC(NC(C3C(C)CCC3)=O)C2)ccc2nnnn2c1 c1(-n2ccc(C(=O)Nc3c(C(=O)OC)cc(C)[nH]3)n2)cc(C)c(OC)c(C)c1 c1(C(N2CC(NC(c3nc(CC)oc3)=O)C(C)CC2)=O)cnc2sc(C)nc2c1 c1(NC(C(=O)NC(C)Cc2ccc(C(=O)O)cc2)=O)ccc(F)c(F)c1 c1(C(=O)NC2C(NC(C(CC)OCC)=O)CC2)cn(C)c(=O)cn1 N1(C(c2c(CC)scc2)=O)CC(CNC(=O)CC2CCCOC2)OC(C)(C)C1 Cc1ccccc1C(N1CCOCC1c1ccc(Cl)cc1)C(=O)NCCC1CC1 c1(C(=O)NC(c2ccc(Br)cc2)C(=O)O)cnc2cc(Br)ccn12 c1(C(CNC(C=CCCC)=O)N(C(=O)C(C)Cc2ccco2)C)ccccc1 N1(C(c2n(C)nc([N+](=O)[O-])c2)=O)CCC2CN(C(c3coc(CO)c3)=O)CC2C1 N1(C(C)=O)CSCC1C(N1CCCC1C(C)NC(C1(n2ccnn2)CC1)=O)=O CC1(C)CCC(CNC(C2SCCS2)=O)N(C(=O)C2=NOC(C(C)(C)C)C2)C1 CC1(C)CN(C(C2CCN2C(C2CC(=O)C23CCC3)=O)=O)CCS1 CC(=O)C(C)CC(C)C(=O)NCC(C)(F)CNC(=O)CC1CCC(C)C1 c1(CC)cc(N2CCC(N(C(c3ccn(C(C)C)n3)=O)C)CC2)ncn1.C1CC1 Cc1cc(C(=O)NC(C)(C)C(C)C)c2occc2c1.c1(C(=O)N)cn(C)[nH]c1=N C1(F)(C(N2CCC(N(C(C(C)OCC)=O)C)CC2)=O)CCCN(C)C1 c1(OC)cccc(C(=O)NC(C(C)NC(c2ccnc(C)n2)=O)C(C)C)c1F N1(C(c2cc(C)ns2)=O)CC2CCCN(C(C3C=CCCC3)=O)C2C1 N1(C(=O)CCN2CCC(O)CC2)CCC2CN(C(C3CCCCO3)=O)C2C1 c1(NC(C(C)=O)=O)ccc(C2CCN(C(c3ccc(CO)o3)=O)CC2)c(F)c1 N1(C(C(C2CCOC2)OCC)=O)CCC2(C1)CN(C(=O)C(C(C)C)OC)CCO2 C1(CC(N2CC(O)(CNC(CC3(C=C)CC3)=O)C2)=O)CCC(F)(F)C1 N1(C(c2ccc(C(C)=O)[nH]2)=O)CC(NC(=O)C(C)C2CCC2)C(C)C1 C1(NC(CC(CC)OC)=O)C(C)CCN(C(=O)Cc2[nH]cnc2C)C1C C1(C(N2CC(SC)C2)=O)CC(C)(C)CN1C(c1cc(C#N)n(C)n1)=O Cc1cc(S(N)(=O)=O)sc1C(=O)N.C1(CCC)CCCCN1C(=O)CC(C)(C)O C1(C(N2OCC(n3cc(-c4c(C)nccc4)nn3)C2)=O)CCC2(CCOCC2)O1 C(=O)(C1=CCS(=O)(=O)C1)N1CCC2(CC2)C1.Cc1c(C(=O)N)cnn1CCO C1(CC(=O)N)SC2=NCCN2C1=O.c1(C(C)C)nnnn1CC(N1CC(C)C1)=O CCCCCC(O)CC(=O)NCC1CCN(C(=O)CC(C)O)C(C)C1 C(=O)(C1=CC2C=CC(C1)C2)N1CCC2(C(C(=O)NC3CN(C)NC3=O)C2)CC1 C1(CNC(CCOC)=O)CCN(C(c2coc(C(F)F)n2)=O)C12CC2 O=C(C#CC1CCOCC1)NCC1CCC2CN(C(c3cnn(CC)c3)=O)CC12 C1(C(=O)NCC23N(C(c4c(C)oc(CO)c4)=O)CC(C2)C3)CCN2CCCC2C1 Cc1cc(C)c(OC(C)C(=O)Nc2ccc(C(C)C)cc2)c(Br)c1 C(CC(C)C(=O)N1CCN(CC(=O)NCc2ccc(CC)cc2)CC1)=CC c1(OC)nccc(C(=O)NCC2(C)CCN(C(C34CCC3C4)=O)CC2)c1F.O C(=O)(CCCC(C)(C)C#N)N(C1CCN(C(=O)CCOC(C)C)CC1)CC N1(C(C2CC3(CC(OC)C3)C2)=O)CC2CC1CCN2C(=O)C(C)N(C)C CCN=c1ccc(C(=O)NC2CCCC(NC(c3[nH]c(C)nc3CC)=O)C2)c[nH]1 C1(CCNC(=O)NC(C)COc2ccccc2F)CCCC1(C)C Cc1csc(C2(NC(=O)CN(C)Cc3ccccc3)CCCC2)n1 N1(C(COC(C)C)=O)CC(C(=O)NCC2OCCCC2(C)C)CC1(C)C C1(C(=O)N(C)CCOCCNC(=O)C(C)OC)(OC)COC1 N1(C(CCC(C)(C)C)=O)CCC2CCC(NC(=O)Cn3cc(C4CC4)nn3)C12 C=C=CC(C)C(=O)NC1C2CC(NC(c3cn(C)nc3C(C)C)=O)CC12 c1(-n2c(C(C(C)C)(C)C)nc(CCCO)n2)ccc(Cl)cc1Cl C#Cc1ccc(C(=O)NC2CC(NC(C3CN(C(C)=O)C3)=O)CC2O)c(F)c1 N1(C(CC(C(C)C)O)=O)CC2OCCN(C(c3ccc(Br)cc3N)=O)C2C1 C(=O)(C1=CC(O)CCC1)NCC(C1CCN(C(C2(Cl)CC2(F)F)=O)CC1)(C)C c1(C(N2CC(F)CC(NC(C(CC=C)(C)C)=O)C2)=O)ccc(Cl)cc1[N+](=O)[O-] C1(CNC(C(C)N=[N+]=[N-])=O)CCN(C(=O)C(F)CC2CCOC2)CC1C CCCCC(CNC(c1nnsc1SC)=O)NC(C1(C)CCCN1C)=O c1(OC)ccc2[nH]ccc2c1NC(=O)NC(c1cccc(-n2ccnc2)c1)C N1(C(C23CSCC2C3)=O)CCc2c(Br)cc(Cl)cc2C1 C(=O)(C1=CCCCCC1)N1CC(NC(=O)C=Cc2ccc[nH]2)C(F)CC1 C#CCCCCCC(=O)NCC12CCCC(CN1C(=O)CC=CCC)C2 CCCCCCCCCC(C(=O)NC)N1C2CCC1CC2 c1(NC(C2CCCN2C(c2ccccn2)=O)=O)cc2ccc(F)cc2o1 C(=O)(CS(=O)(=O)C1CC1)N1CCCC(CNC(C2CCC(CC)O2)=O)CC1 CCCC(C(=O)N(CC(O)CO)C(C)C)NC(=O)C(C(=O)OCC)OC C1(OC)CN(C(C2(NC(=O)C=Cc3cc(C)no3)CC2)=O)CC1OC CC(CC=O)C(C)(C)C.C1(=CC)CCN(C(c2cscc2C(F)(F)F)=O)CC1.N CS(=O)CCC(=O)N1CCCC(n2cc(CNC(c3c[nH]c(Br)c3)=O)nn2)C1 CS(=O)(=O)c1ccsc1C(=O)NC.C1(C(N2CC=CC2)=O)OCCOC12CCC2 N1(C(CCCCOC)=O)CCCC2(CCCN2C(C2OCCOC2C)=O)C1 C(C(C)C(=O)NC1(C(=O)NCC(CC)N(C)C)CC(CO)C1)OCC c1(OC)cccc(CN)c1[SH](=O)=O.C(=O)C(C(C)C)c1cccc(C(F)(F)F)c1.N Cc1c(C(N2CCCC(NC(C3(CO)COC3)=O)C2C)=O)cnc2ncnn12 C1(CNC(C=COCC)=O)CCC12CCN(C(=O)CCc1csc(C)n1)CC2 C=C1CC(C(=O)NCCCC(C)C)(CNC(C2OCCC2CC)=O)C1 C(C1=CCCOC1)NC(C1CC(O)CN1C(=O)C(O)c1ccsc1)=O CC1(CNC(=O)C(N)=O)CCCN1C(=O)CN1CSCCSC1 c1(C2(NC(=O)NC(C=C)CO)CC2)c(OC)cccc1Cl Cc1nc2ccccc2n1CC(N1CC2(C1)CN(C(=O)C(F)C1CCOC1)C2)=O C=CCCCCCNC(C1(NC(c2cnsn2)=O)CCN(C)C1)=O C(CC(C(=O)NCC(C1CC1)N(C)C)NC(c1ccc(C)n1C)=O)OC N1(C(Cc2cc(C)[nH]n2)=O)CCCC(NC(C2OCCCC2(C)C)=O)CC1 CCC(O)(CC)c1cn(CC(=O)NC(C)(C)CNC(N)=O)nn1 C#CCC(CC(F)F)C(=O)N1CC2C(CC(=O)N(C(C)C(C)C)CC)C2C1 c1(CCCC)ccc(CC(=O)NCC(CO)NC(=O)CCCCSC)cc1 C1(C(=O)NCCCCCCC)CC2C=CC1N(C(c1ccc(OC)o1)=O)C2 C(C(=O)N1CCC(CC(C)(C)C)C1)(C(C)O)NC(C)=O.c1(C=O)ccoc1C.N CCC1=NOC(C(N2CC3C(N(C)C(c4coc(O)n4)=O)C3C2)=O)C1 c1(C(N2CC(N(C)C(c3ccnnc3)=O)C2)=O)cc2cccnn2n1 C1(O)(C(=O)NC(CC)CN(C(=O)CCCN2CCOCC2)CC)CC(C)(C)C1 C1(C)(C(N2CC(NC(C(=O)NC(C)C)=O)C2)=O)CCOC1C C1(NC(C(C)=C2CCC2)=O)CC12CCN(C(=O)C(C)NC(N)=O)CC2 N1(C(C2=CC(C)(C)C2)=O)CCC(C2(NC(c3[nH]nnc3C3CC3)=O)CC2)C1 c1(CC(C(=O)NCC(N(C(C2C(C)C2)=O)C)C2CC2)=O)cccc(Cl)c1 C1(C(C)(C)C)CCC(CC(=O)NC2CN(C(C3CC3(F)Br)=O)C2)CC1 Cn1cc([N+](=O)[O-])c(C(=O)NCC2=CCN(C(C3COC(=O)O3)=O)CC2)n1 C12(NC(CCCS(N)(=O)=O)=O)CCCC1N(C(c1cccs1)=O)CCC2 c1(OC(C)C)ccc(OCC(=O)N)cc1.C1(C=O)CCCC(C(N)=O)C1 Cc1ccn2cnc(C(=O)NCC3(NC(C4CN5CCCN4CC5)=O)CC3)c2c1 N1(C(CCOCCCNC(C(n2c(C)ccn2)C)=O)=O)CCCOC(C)(C)C1 c1ccc(F)c(C)c1.N1(CCOC)CCCC1C=O.C(=O)(CCO)NCCC C1(CC(=O)NC2CC(F)(CNC(C3(C)CCCS3)=O)C2)NC(=O)NC1=O CC1(C)CC(C(=O)N)CCN1C(=O)Cn1cc(C#N)cn1.CC(O)CC1CCC1 C=Cc1cncc(C(=O)N2CC(n3cc(-c4cccnc4C)nn3)CO2)c1 c1(C(N2C(CNC(C3ON=C(CC)C3)=O)C=CC2)=O)cc(N)c(OC)cc1.O N1(C(c2c(CC)n[nH]c2)=O)CCCC(C2CCCCN2C(C2CCOCC2)=O)C1 C=CCC(C(=O)Nc1ccccc1N(C)C)NC(=O)C(C)OCC(C)C C1(CNC(COC(CC)C)=O)CC(F)(C)C1.C1(CC=O)CC(C)(C)C1 N1(C(C(C)(C2CCC2)NC(C(CC(CC)C)=O)=O)=O)CC2(C1)NC(=O)NC2=O C(=O)C1=NN(C)C(=O)CC1.c1(SC)ccc(C)o1.C(=O)(CCc1ccoc1)N c1(OC)ccc(C)nc1C(N1CC(CCCCNC(C2COCCO2)=O)C1)=O N1(C(C2CCC(OC)C2)=O)CCC(C(=O)NCCC(=O)NC(C)(C)C)CC1 Cn1ncc(C(=O)NC2CCC(CCNC(c3cc[nH]n3)=O)C2)c1C1CC1 CC1CC(C(N2CC(F)(C)C2)=O)CC(C)O1.C1(S(N)(=O)=O)(C=O)CCC1.N C1(C(=O)NC2CC(NC(CC(CN(C)C)O)=O)C2)CCC12CCOCC2 C(=O)(C(C(C)NC(c1sncc1C)=O)C(C)C)NCc1n(CC)c(O)nn1 C1(O)(C(C(=O)N(CC(C)O)C)F)CN(C(C2(CC(C)C)CC2)=O)C1.CC.O C12(CNC(COC)=O)CC1CN(C(C1OCCCC1c1ccccc1)=O)C2 c1(C(N2CC(CCn3cc(-c4cccnc4Cl)nn3)C2)=O)c(F)cccc1F c1(OC)ccc(C(=O)N)c(F)n1.C1(CC)CSCCN1C(=O)Cc1cnn(C)c1 N1(C(c2c(CC)nc[nH]2)=O)Cc2ccccc2C1CNC(C1CC2CC2C1)=O c1(CN(C(=O)C(=O)NCC2CC(F)(F)CN2)CCC)ccccc1Br c1(C=O)cc2n(n1)CCC2.Cc1nc(CC)no1.C1(CC=CC=O)CCC1.N Cc1ccc(CC(N2CC3CC2C3CNC(=O)C(c2ccccc2F)C)=O)cc1 C(=O)(C(C#N)C(C)C)NCC=CCC(=O)N(CC(COC)O)C Cc1nc(Cl)c(C(=O)NC(c2cn(-c3ccnc(C(=O)O)c3)nn2)C)c(C)c1C c1(NC(CC)=O)cccc(NC(=O)C(=O)NC2CC3CC(N)C3C2)c1C C=CC1(C(=O)NC(C2(CO)CC2)C)CCN(C(=O)C=CC2CCCN2C)C1 N1(C(C2(CC)CN(C(=O)C=Cc3cccc(C)c3)C2)=O)CCS(=O)C(C)C1 C1(CC)CCCC1(C)C(N1CC2(NC(=O)C(c3ccc(Cl)cc3)=O)CC1C2)=O C1(C(=O)NCCS(N)(=O)=O)CC12CCN(C(c1ccc(C(F)F)o1)=O)C2 N1(C(C(C)C(F)(F)F)=O)CCC2(CC1)CC2C(=O)NCc1cncn1C C(CC(C)C(=O)NC1(CF)CN(C(=O)Cn2cccnc2=O)C1)=CCC C(=O)(C(C)CC(=O)OC)NCC(C(C)(C)C)NC(c1cccc(CC)c1)=O Cc1cc(C)nc(SCC(=O)NC)n1.C1CCCCN(C(=O)CC2(O)CCC2)C1 C#CC1(NCC2CC2c2ccccc2)CCCC(C)(C)C1 c1(C(C)=O)ccc(F)c(NC(C2CN(C(=O)C(C)Cc3ccccn3)C2)=O)c1F N1(C(C(N(C)C)C2CC2)=O)CCCOC(CNC(=O)CCCc2ccccn2)C1 C(CCC(C)C(=O)NCC(C)N(C)C(c1snnc1C1CC1)=O)OC CCCC(C(=O)NC1(C)CC(C)(C)C1)NC(=O)C=CC(F)F C1(NC(C(CC)(C)C)=O)COC2(C1)CN(C(c1cc(C(F)(F)F)cs1)=O)C2 N1(C(CSCCOC)=O)CCCC2(CCN(C(C3CCS(=O)(=O)N3C)=O)C2)C1 C(=O)CC(C)C.C1CCC1.C(C=O)NC(=O)OCC=C.[SH](C)(=O)=O.N c1(C(=O)NC(CNC(c2cc(CC)sn2)=O)CC)cccc2nccnc12 n1(COC)ccc(C(=O)N(C(C)CCNC(c2cnoc2-c2cccs2)=O)C)n1 Cc1c(CN2CCC(NC(=O)CCc3ccc[nH]3)C(F)C2)[nH]c2ccccc12 N1(C(=O)CSC(F)F)CCC(C2(O)CN(C(C34CCCC3C4(F)F)=O)C2)CC1 C1(CNC(c2c(SC)ccs2)=O)CN(C(C2CCCCNC2=O)=O)CC1(F)F N#Cc1cncc(C(=O)NC2(CNC(=O)C=C3CCC3)CCOC2)c1 CC1CCn2cc(C(=O)NCC3(F)CC(NC(C4CCCOCC4)=O)C3)nc2C1 N1(C(C(n2ccccc2=O)C)=O)CC2(CCC(Nc3cnc(O)[nH]3)CC2)C1 C(C)(CCCCNC(C1CC1c1ccccc1)=O)NC(CN(C1CCSC1)C)=O n1(CCC(=O)NC(CNC(C(CC)NC(C)=O)=O)(C)CC)ncn(C)c1=O C1(COC)CC(C)N(C(=O)C)C1.c1cccc(C)c1.C1(C=O)CC(C)=NO1 C1(F)(C(N(CC(c2ccco2)O)C)=O)CCCN(C(C2(C(N)=O)CC2)=O)C1 C1(O)CCCN(C(c2ccc(Cl)c(I)c2)=O)C1.c1(C(=O)N)cc(O)nc(O)n1.C C1(NC(C(Cn2cccn2)NC(C2C(C=C)OCC2)=O)=O)CCC(C#N)CC1 O=C1CS(=O)(=O)CC(C(=O)OCC(C2CCCCC2)F)N1 N1(C(CC(CC)SC)=O)CCCCC(NC(=O)C=C(C)c2ccco2)C1 N1(C(c2cccnn2)=O)CC2OCCN(C(c3cc(Cl)c4n[nH]cc4c3)=O)C2C1 C1(NC(c2c(C)n(C(C)C)nc2)=O)CCN(C(C2CC2(F)F)=O)CC1C N1(C(C(C)OCC)=O)CCCC(C2(NC(c3n[nH]cc3[N+](=O)[O-])=O)CC2)C1 CC1C(NC(=O)CCc2cnn[nH]2)CCCN1C(=O)Cn1ccc([N+](=O)[O-])n1 C(=O)(C1CCCc2c1ncn2C)NCCC1(NC(c2cc(CC)on2)=O)CC1 N1(C(Cn2c(C)ncc2)=O)CC(NC(=O)COC2CCOCC2)C2CC12 c1(C(C)C)c(C(=O)N(CCCOCCNC(C2CCNC2=O)=O)C)cnn1C C1(NC(C(C)N(C(C2CC2C#N)=O)C2CC2)=O)CCC(CCO)CC1 Cc1c(O)c(=O)ccn1CC(N1CCC(C)C(NC(=O)CC2CCNC2=O)C1)=O N1(C(C2CN(C(CNC(N)=O)=O)C2)=O)CCC(OCCF)CC1.c1ccccc1.O Cc1cc(C(=O)NCc2ncoc2CCNC(=O)C(C)n2cncn2)cnc1F N1(Cc2c(C(=O)OCC)ccs2)CC2CC2(C(=O)Nc2cnccc2Br)C1 C1(C(N(CCOC)CC)=O)C(C2CC2)CCN1C(c1ccc(O)cc1F)=O n1(CCC(=O)NC2CCCN(C(C3=C(C)CCC3)=O)C2C)cc([N+](=O)[O-])nc1C C1(CC(=O)NCC2(NC(CCCC(C)O)=O)CCC2)CCCC2CCCCC12 OC1CC2CC(N=c3[nH]c(N4C5CCC4COC5)nc4c3CCC4)C1C2 C1(CC(=O)NOCC(O)CO)C2CCCC2N1C(=O)C(O)CC1CCCC1 C1(C(=O)NCC2N(C(COCC#C)=O)CCCC2)CC2C=CC1CC2 N1(C(CC2CCCN(C(c3cn(CC=C)nn3)=O)C2)=O)CC2(CCOC2)C1 CCC(CCCC(=O)N(C(C)CC(C)C)C)NC(c1n[nH]c2ccccc12)=O Cc1cc(C)c(C(=O)NC2CCCC2C(N2CCC3(CCCO3)C2)=O)c(Cl)n1 c1(CCC(=O)NC2CN(C(c3ccc(C)s3)=O)CC2O)cc(F)cc(F)c1 N1(C(Cc2ccn(C(C)C)n2)=O)CCCC(N(C(=O)C=Cc2ccn(C)c2)C)C1 c1(CC)ccc(C(=O)N(CCCNC(c2c[nH]nc2C2CCCO2)=O)C)cc1F Cc1cc(C(N2CCCN(C(C3CC3(C)C)=O)CC2)=O)c2c(c1)CCCN2 Cc1cc(N2CCC(NC(c3ccc(Cl)cc3Cl)=O)C(O)C2)nc(C2CC2)n1 c1(C(=O)NC(CCN(C(C(CCC)OCC)=O)C)C(C)C)cc(Cl)cc(Cl)c1O Cc1cn2c(n1)C(C(=O)N1CC(NC(=O)CP(C)(C)=O)C(C)(C)C1)CCC2 C1(C)(NC(C2CC(CCC)C2)=O)CCCCC1C(=O)N(CCCCC1CC1)C O=C1NC2CN(S(=O)(=O)c3ccc(NCc4ccoc4CO)c(Cl)c3)CCC2CO1 c1(N2CCCC(=C)C2)nc2c(c(=NC(C)C3CCOCC3)[nH]1)CCC2 N1(C(CCC(=O)N(C)C)=O)CC2CCCN(C(c3cc(O)cc(C#N)c3)=O)C2C1 C1(CC(=O)NCC#CCNC(C2CC(OC)C2)=O)CCCCN1C(C)=O N1(C(c2ncn(C)c2)C(=O)NCC2CC2)CCC(c2nc(C(C)(C)C)cs2)CC1 O=C(NN1CC2CCCC2C1)c1cc(C(F)F)on1 N1(C(Cn2nnc(C)n2)=O)CCC(F)(CNC(=O)C(C)Sc2nncn2C)C1 N1(C(CCCC#C)=O)CC(C)(C)CC1CNC(C1(C)CCC(N(C)C)CC1)=O c1(CC(=O)N)c[nH]c2ccc(Cl)cc12.C12CCC(CC1)N2C(=O)C(O)C1CC1.C Cc1cc(=O)ccn1CC(=O)NCCC(C)NC(c1cnccc1Br)=O n1(CC=O)ncc2ncccc12.C1(CC(=O)NCCC2CCC2)CCC(=O)N1.N C1(CNC(C=C(C)C(F)F)=O)CCCCC1.C(C)(c1ccsc1)=CC(=O)N c1(OC)cc(C(N2CCC3CC(N)C23)=O)ccc1-n1ccnc1 c1(C(=O)OC)ccc(=NCCC2CCC(NC(=O)C(F)(F)C(C)(C)O)C2)[nH]c1 C1(CNC(C(C)NC(C(C)(C)OCCC)=O)=O)CCCN(C)C1=O c1(C(N2CCCC(C)C2CNC(=O)CCc2cn[nH]c2)=O)nccc2cc[nH]c12 c12cccnc1C(=O)N2C(C)C.Cc1nc[nH]c1C(CC(C)(C)C)=O Cc1nc(C(=O)NC(C)CCN(C(=O)CC2CNC(=O)C2)C)cc(O)n1 c1(C(N2C3CCC(NC(c4ccc(OC)cn4)=O)(C3)C2)=O)ccc(Cl)c(F)c1O CC(CC(F)(F)F)C(=O)N1CC(OCC(=O)NCCc2ccc(F)cc2)C1 C=CC(C)(CCOC)C(=O)NC1CCCN(c2cc(C(=O)O)ncn2)C1C.C1CC1 c1(C(=O)NC2CC(NC(CSCC=C)=O)C2)ccc(N=S(C)(C)=O)s1 CC1(C#CC(=O)NCC2C3CN(C(c4c[nH]nc4C(F)F)=O)CC23)CCCO1 c1(C(=O)NC2C(NC(Cc3ccc(OC)cc3Cl)=O)C2)ccc(C#N)cc1O CC(CC(=O)NCC(C)(CO)NC(c1cc(C2CCC2)[nH]n1)=O)C1CCCCC1 C1(NC(CCc2n(C)cnn2)=O)CN(C(c2ccc(=O)n(C)n2)=O)CC1C1CC1 N1(C(C23CCC(CN(C(C=C=C(C)C)=O)C2)C3)=O)C2CCC1CC1(CC1)C2 C1(CN(C(C2(CCOC)CCCC2)=O)C)CCCC(NC(=O)C2CC2)C1 c1(C(=O)OC)cc(Cl)c(SC)c(Cl)c1.C1(S(C)(=O)=O)CC1C(F)(F)F N1(C(C2(CC#C)CC=CCC2)=O)CC2(CC(NC(=O)C3=NOCC3)C2)C1 C(=O)(N=c1cc(Cl)nc(O)[nH]1)C12CN(C(C(CCC)OC)=O)C(C1)CCO2 N1(C(Cn2c(=O)sc(C)c2C)=O)CC2(CCCC2NC(=O)Cc2csnn2)C1 C(C(C)(C)C)NC(c1ccnn1CCF)=O.C1(CCC=O)CCC(=O)C1.CC C1(C(=O)Nc2c(C)nn(C)c2)CC2(CC(NC(=O)C3=CCCSC3)C2)C1 C1(NC(c2cc(OC)ns2)=O)CN(C(=O)C(C)(C)SC)CC2(CC2)C1 N1(C(c2c(CC)scn2)=O)CCN(C(=O)Cc2ccno2)CC1CC N1(Cc2ccc(OC(C)=O)c(Cl)c2)CC2CN(C(=O)CCCCCl)CC2C1 c1(OC)ncc(Cl)cc1C(=O)NCC(CNC(C1CCCOC1C)=O)OC C1(NC(C2CCOC2C2CC2)=O)(C)CCOCC1.C1(O)(C(=O)N)CCOCC1 c1(C(=O)Nc2cc(Br)cc(I)c2)n[nH]c2c1CN(C(=O)CCCCBr)CC2 c1(CCC(=O)NCCC2CC2)ccc(O)cc1.c1(CC=O)nc(C2CC2)cs1 C(C(=O)N(CCC(=O)N1CCCC(C)C1CCO)OC)C1ON=C(CC)C1 Cn1cncc1C(=O)NC1(C2CCCN2C(c2coc(Br)c2)=O)CC1 N1(C(Cn2nc(C)c(Br)c2)=O)CCN(C(=O)C2=CCCS2)C2CC12 C1(NC(C=C(C)Cl)=O)CCC2(CCCN(C(=O)Cc3cc(F)c(N)cc3F)C2)C1 Cn1cnc2cc(C(=O)NCC(C)(C)NC(c3nc4cccnc4s3)=O)cnc12 C1(CC(N2CC(C)(NC(CC(CN(C)C)(C)C)=O)C2)=O)CCCCCC1 C(=O)(CC(C)(C)O)NC(CC=C)CNC(C1(c2cc[nH]n2)CCC1)=O C1(C(N(C2CCC(NC(C3CC(OC)C3)=O)CC2)C)=O)CCC2(CCCCC2)C1 C1(N(C(Cn2c(C)ccn2)=O)C)CN(C(=O)C(F)=C2CCCC2)CC1(C)C C1(C(C)NC(C(C=C)O)=O)CCCN(C(=O)Cc2sc(S)nc2C)C1 C1(NCC2(CO)CC2(F)F)CC2CC1C(O)C2O C(C(C(=O)NCCC1CC(NC(c2cccnn2)=O)C1)N(C)C)N(C)C N1(C(C2CC3CCC2CC3)=O)CC2CC(C1)N(C(=O)Cc1cnccn1)C2 C1(C(=O)NCC(C)OCCC)CCCN(S(=O)(=O)Cc2cccc(Cl)c2)C1 c1(COC)cc(C(=O)NC(C2CCCN2C(C2CC(CF)C2)=O)C)on1 CC(C)C(F)(CNC(C1CCCCC(=O)C1)=O)C(=O)N(C)CC1(CO)CC1 c1(C(=O)NCC2(O)CCC2)cc2ccoc2cc1F.C1(C=O)(CCF)CC1.C C1(C(=O)Nc2c(C(C)C)n[nH]c2)CCc2[nH]nc(C(F)F)c2C1 O=C1CCCCC(C(N2CCC(CC3CCCCC3)CC2C(=O)O)=O)N1 Cc1cccc(C(N2CCC3(CCN(C(=O)CC(C)C)C3)C2)=O)c1[N+](=O)[O-] C=CC1(CC(=O)NCCCCN(C(=O)CC2(C#N)CCCCC2)C)CCOCC1 C=CC1(NC(C2COCC2NC(=O)C=Cc2ccn(C)c2)=O)CCCCC1 N1(CC)CCOC(C(=O)NC(C)C(CO)NC(C2CC(OC)C2)=O)C1 c1(CC)nn(C)cc1C(=O)NC1CC(C)N(C(c2cnn(C)c2Cl)=O)C1 N1(C(c2cc(C(C)=O)sc2)=O)CCN(C(c2cc(Br)n(C)n2)=O)C2CCC12 C(CC(C)C)(C(=O)NCCNC(=O)C(O)Cc1cn(C)cn1)OC C#CCCCCCCC(=O)N1CCCCC1C1(NC(C2CC(N(C)C)C2)=O)CC1 c1(CC)cc(C(=O)NCC2CC2C)ccc1F.c1(C(=O)N)cc(C)ccn1 c1(OC)ccc2c(C)c(C(=O)N(C3CCCN(C(=O)C(C)O)C3)C)[nH]c2c1 n1(C(C)C)ccc(C(N2CCC(CC(=O)NC(C)CCO)C2)=O)n1 N1(C(c2n(C)c(S)nn2)=O)CC(O)C(O)C1C.C1(CC(=O)N)CCCNC(=O)C1 CC1CCCCCCN1C(=O)CONC(=O)CS(C)(=O)=O C(CCC(C)C(=O)N1CCCCC1CNC(c1cc(Br)cnc1N)=O)OC N1(C(c2c(OC)nsc2OC)=O)CC(NC(C)(C)C)CC(F)C1 CCCC(CCC)C(=O)NC1CC(CC(=O)NCc2nncn2C)C1(C)C c1(OC)cc(F)c(C(=O)NC2CC(C)C2)c(F)c1.C(=O)C#CC(C)(C)C.N Cc1c(F)cc(C(=O)Nc2ccc(NC(=O)C(C)(C)O)cc2F)cc1F c1(C(=O)NC2C(C)CN(C(c3ccncn3)=O)CC2)cn2ccc(F)cc2n1 N1(C(CN(S(CC)(=O)=O)C)=O)CC2CC1CN2C(C1CCN1S(C)(=O)=O)=O C(CC(C(=O)NCc1ncccc1Cl)NC(C1CCC2CC12)=O)SC c1(C(N2CCC(CC)C2)=O)cc(C)cc(F)c1N.C(C)(C(C(=O)N)N(C)C)OC c1(C(=O)NCC23CCC2CCN3C(=O)C2=CCCC2)cnc2ccsc2c1 c1(NC(C2CC3CC3N2C(=O)CC2CCC2)=O)c(I)cc(Cl)cc1[N+](=O)[O-] c1(C(N(CC(CN(C(C(CC(C)C)O)=O)C)O)C)=O)ccc2c(Cl)nccc2c1 Cc1cnncc1C(=O)NC1(C)CC(NC(C2CC2(F)F)=O)C1 c1(NC(C)=O)ccc(C(=O)OCc2scnc2C2CC2)c(F)c1 N1(CC(=O)OC)CCN(C(=O)CSc2cc3c(s2)CCNC3)C(C)C1=O c1(C(N2CCC(NC(c3csc(Br)c3)=O)C2)=O)ccc2ncccc2c1 c1(OC)nc(C)cnc1C(=O)NC1C2CN(C(=O)CN3CC4CCC3C4)CC12 c1(NC(C2CCC(C)N2C(c2nccnc2Br)=O)=O)ccc2cnccc2c1 c1(C(=O)NCCCN(C(C2CC(C)(O)C2)=O)C2CC2)c(Cl)ccc2c[nH]nc12 C12(C(C)NC(CC(C)NC(c3ccccc3)=O)=O)CC(F)(CO1)C2 c1(C=O)ncncc1C#N.Cc1[nH]c(C(C)(C)C)cc1C(=O)NC1CC1C.N n1(CC(=O)NC(C)CNC(=O)CCc2csnn2)cc(Cl)cn1 C1(N(C(c2cnc(CC)[nH]2)=O)C)CN(C(=O)C=Cc2cncc(O)c2)CC12CC2 C1(C)(C=O)CC2(C1)CC(F)(F)C2.C1(C(N(C(C)C)CC)=O)CCSC(C)C1 C(=O)(C(CCC)C(=O)OC)NC(CC=C)C(=O)N1CC(C)(O)C1 c1(C(=O)NC(c2c(OC)cccc2)C(F)(F)F)ccn2nccc2c1 S(=O)(=O)(c1ccc(C)c(C(F)(F)F)c1)N(c1cc(C)c(=N)[nH]c1)c1ccccc1 C(=O)(CCS(N)(=O)=O)N(C(C)C(=O)NC1CC2(CCC2)C1)CCC CC1CCCCC1C(=O)NCCOCCC.c1(C(=O)N)csc(-c2nc[nH]n2)n1 c1(NC(CC2N(C(CCc3cncc(OC)c3)=O)CCC2)=O)cnc(Br)c(Br)c1 N1(C(c2n(CC)cc(Cl)c2)=O)CCC(C)C(C)C1.c1(C=O)ccnn(C)c1=O.N C#Cc1cc(F)cnc1NC(C1CC1NC(=O)C(O)C(C)C)=O C(C(C)(C)C(=O)N1CC(NC(C2(CF)CCC2)=O)C(SC)C1)OCC C1(NC(C2(Cl)CC2)=O)CCCC(N=c2[nH]c(Cl)ncc2Cl)C1 C(C)(CC(C)N=c1nc[nH]s1)NC(C(c1ccc(F)cc1)OC)=O C1(CNC(C2CC(F)C2)=O)CC2CCC(C1)N2C(=O)C=Cc1ncc[nH]1 C1(C(=O)NCc2nc(CNC(=O)COCCF)sc2)CC1C1CCOCC1 CCC(CC(=O)N(CC(O)CN(C)C(c1cnoc1C1CC1)=O)C)C1CCC1 N#Cc1cc(F)ccc1C(N1CCN(C(C2CC(=O)N(O)C2)=O)CC1)=O c1(C(c2n(CCCCCC)nnn2)NCC(=O)N(C)C)n[nH]c2c(F)cccc12 O=C1NCC2(CCCC2)C(=O)N1CCN1CCN(CCNc2ccc(Cl)cc2)CC1 CC1=C(C(=O)N)S(=O)(=O)CCO1.C1(C=O)C2CCC1(c1cncs1)C2.C(C)C N1(CC)CCOCC1C(=O)NCC1CCC1.c1(CC(=O)N)ccc(F)nc1 C1(CCC)CN(C(c2occc2C)=O)CC1C(=O)NCCCC(=O)OC C1(NC(c2cc([N+](=O)[O-])cs2)=O)COCCN(C(c2ccc(Br)cc2F)=O)C1 c1(CC(C(=O)OC(C)C)NC(=O)CNCc2ccccc2)ccc(O)cc1 N1(c2nc(N(CCOCCOCC)C)c3c(n2)CSC3)CCN2CCOCC2C1 c1(C(=O)NC2(C)CCN(C(CS(CC)(=O)=O)=O)C2)cncc2c1CCNC2=O c1(N2CCC(NC(CCS(C)=O)=O)C(F)(F)CC2)nnc2c(c1C#N)CCCC2 C1(CC(=O)NCCCN(C(c2sccc2COC)=O)CC)OCCC1C C1(F)(CNC(c2ccc(CCC)s2)=O)CCCN(C(=O)C=C(Cl)Cl)C1 C1(C(=O)NCCNC(=O)NC)CSCCN1C(c1ncncc1C)=O C1(N(C(CC=C=C)=O)C)CCCCN(C(C2CC2c2ccccn2)=O)C1 Cc1cccc2[nH]c(=NCC3CCCC3NC(c3ccc(Cl)cc3)=O)sc12 C1(CC(NOCCS(C)(=O)=O)=O)CCNC12CCC2 C(C)(C)(CCCCC(=O)N(CCCNC(=O)CCNC1CCC1)CCO)OC c1(NC)cncc(CNC(C2CCN2C(=O)CC2CC3(CC3)C2)=O)n1 N1(C(c2cn3ccccc3n2)C(=O)NC)CCC(CC#N)C(F)(F)CC1 N1(C(CN(CCC)C)=O)CCC2C(C1)CN2C(=O)CC(F)(F)Br O(N1C(=O)c2ccccc2C1=O)CCOCCNC(c1cc(C(C)C)no1)=O c1(C(=O)NC2CN(C(c3cccc(C)c3O)=O)CC2C)ccc2c(c1)CCCS2 Cc1nn(C)cc1C(N1CC2CC1C2C(N1CCC(O)(c2cnn[nH]2)C1)=O)=O N1(C(C=CCN(C2CCOC2)C)=O)CC2CC(N(C)C(c3cn[nH]c3)=O)C1C2 C1(NC(c2c(CC)cccc2)=O)CC2(CCC(C)OC2)C1.C(=O)C1=COCC1.N c1(C(N(CCC)CCNC(C2CCCCNC2=O)=O)=O)csc2c(O)ccnc12 N1(C(C(c2scc(CC)n2)(F)F)=O)CCCOC(C)C1.C(=O)(C(C)(C)CC#N)N C1(NC(C2(C)CC(F)C2)=O)CC2CCC1CN2C(c1ncn2c1CCC2)=O C1CCc2nncn2CC1.C1(ONC(C2(C)CN(C(C)=O)C2)=O)CC2(CC2)CO1 c1(C(=O)Nc2scc(C#N)n2)cc2cc(-c3cccc4ccsc34)ccn2n1 O=C(CC(C(F)(F)F)NC(=O)C(=O)NCC(F)F)NCC1CC=CCC1 C1(C)(CC)CC(C(=O)NCC2(O)CCN(C(C3CCOC3C)=O)C2)CCO1 CCCC(C(=O)NCCCCCC(=O)NCC1CCCCCC1)C(C)C C1(C(=O)OC)CCOC1C(=O)NCCN(C(=O)CCc1ncc(C)[nH]1)C C1(c2nnnn2Cc2nnn(C)n2)(NCCCn2ncc(C)c2)CCC(=O)NC1 c1(OC)cccc(NC(=O)C(C)Oc2ccc(Br)c(C)c2)c1F c1(C(N2CCC(NC(c3cscn3)=O)CC2C2CC2)=O)cnc2[nH]ccnc1-2 C(=O)(C1=NOC2COCC12)NC(COCC)C(N1CCCC(O)(CO)C1)=O N1(C(c2ccc(F)s2)=O)CC2(CCCN(C(c3cc4n(n3)CC(F)C4)=O)C2)C1 C1(NC(c2ncc(Cl)cc2Cl)=O)CCN(C(c2cc(Br)cs2)=O)CC1F N1(CCCC)CCC(C(N2CCCCC2C(=O)NC(C)C(=O)OCC)=O)CC1 c1(C(N(C)CCOCCC(=O)NCC2(CO)CCCC2)=O)ccc(C#N)[nH]1 C1(C(N(C)CCNC(=O)Cn2nnc(-c3ccsc3)n2)=O)CCC=CCC1 CC(C)(CO)CCNC(=O)CCCC1(NC(=O)C(O)C2CC2)CCC1 c1(OC)nc(C(N2CCCCC2C)C)sc1C.c12ccc(cc1)c(=O)o2 N1(C(c2c(C)ocn2)=O)CC2CCC1C(CNC(C1CCN3CCCC3C1)=O)C2 c1(NC(=O)NCC(N2CCOCC2C)C)c[nH]c2cc(F)ccc12 C1(C(N2C(c3cn(CC(CC)CC)nn3)CCCC2)=O)CCn2nnnc2C1 C1(NC(C(CCC=C)NC(=O)CN2CCC(O)CC2)=O)CCCCC12CCC2 C1(OCC)CC(N(C(c2cc(F)ccn2)C(=O)NC2CCOC2)C)C12CCC2 C1(CC(=O)NC2(C(=O)NCCc3ocnc3CO)C(C)C2)COCCN1C C1(NC(=O)CCN=c2[nH]ccs2)CCC12CCN(C(=O)C(O)C(F)(F)F)CC2 C(CC1CCc2ccccc21)OC.N12C=CC(=NC(=O)NCCCC1)N2 Cc1ccc(F)c(Br)c1C(=O)NCC1CC(C)N(C(=O)CSC2CC2)C1 C1(NC(CSCCCC)=O)CC(CNC(c2nnc(O)cc2C)=O)C12CCC2 C1CCCCC1.c1(CCC=O)cccnc1.C(C(O)C)NC(=O)OC(C)(C)C.N C(C(C)CC(=O)OC(C)(C)C)OC.C1(CCNCCCC=O)CCCC1.N CCCCC(C)CCC(=O)N1CCC2(CC(NC(c3[nH]cnc3CC)=O)C2)C1 CC(CCCC(=O)N1CCOC(C2CC2)CC1)NC(c1n[nH]cc1Cl)=O c1(CNC(=O)NC(Cc2ccc(C)cc2C)C(=O)O)cc2cncc(Br)c2o1 C1(NC(C(CC#C)O)=O)(COC)CCN(C(=O)CCSC2CCCC2)CC1 C12(CNC(C3(CC=C)CCCC3)=O)CCC(CC1)N(C(=O)C(C)N(C)C)C2 C12(NC(C=C(C)C)=O)CCCN(C(=O)CN(C)CCO)CC1C2 C1(C(=O)NCC2CN(C(=O)CCc3ccc(CO)cc3)C2)CCc2cncn2C1 C1(C(N2CC(CN(C(C=C(C)C)=O)C)C2)=O)COc2ccc(F)cc2C1 N1(C(CC(C=C)(C)O)=O)CCC2(CCC2)C(NC(=O)CC(=O)NC)C1.C1CC1 N1(C(C2(C(C)C)CC2)=O)CCC(NC(=O)CN2CCCCC2)C(C)C1 C(=O)(CC1COc2ccccc21)NC1CN(C(c2scc(OC)c2)=O)CC1C Cc1cc(C(=O)NC2CN(C(=O)CC3CCCCCO3)CC2O)c2[nH]cnc2c1 Cc1nc(COC(=O)CSCC(=O)Nc2cccc(Cl)c2)oc1C C1(C(N2C(C)CC(CNC(c3c(C)cccn3)=O)C2)=O)CNC(=O)C(C)(C)C1 N1(C(c2ccc(C)nn2)=O)CCC(NC(=O)Cc2ccc(Cl)cc2C)C(CO)C1 C1(NC(CS(C(C)C)(=O)=O)=O)CC2CC(C1)CN(C(C1CCC(C)(C)OC1)=O)C2 c1(C(C(=O)OCC2=CCN(C)CC2)(F)F)cccc2ccccc12 N1(C(C2CCC(OC)C2)=O)CC2CC1CCC2NC(c1csc(C2CC2)n1)=O CCC(CNC(C1CC2CCC1CC2)=O)(CC)C(=O)NCC(C)(Cl)CC O=C(C1CCCc2nncn21)NCC1COCCN(C(=O)COCC(F)(F)F)C1 C(CN=c1[nH]c2cccc(C)c2s1)(CC(C)C)NC(CCC(=O)NCCC)=O c1(C(=O)NC(CC2CC2)C(=O)NC2C3CCCCCC23)cccc2ccoc12 N1(C(COc2cccc(C)c2)=O)CCC(C)C(CNC(c2cncc(Cl)c2)=O)C1 C1(C(=O)N)CC2CC(=O)C1O2.C1(CCC)CN(C(=O)C=Cc2ccnn2C)CC1 C1(NC(C2C(OCC3NC(=O)OC3)CC2)=O)CCCN(c2nccs2)C1 c1(OC)ccc(C(=O)NC(C)(C)C(C)C)c(C)n1.C1(Cl)(C=O)CC12CCC2 c1(C=O)c(F)cccc1F.N1(C(C=CC(=O)OCCCC)=O)CCC1C.N Cc1c(Cl)ccc2[nH]c(C(=O)NCCCCCNC(=O)C(C)O)cc12.C1CC1.C N1(C(C2(Cl)C(C)(C)C2)=O)CCC2(CC1)CCN(C(C13CCCC1CC(=O)C3)=O)C2 Cc1[nH]c(C#N)cc1C(=O)NC(C(=O)NCCCCCC(C)C)C1CCCC1 C1(OC)CC2(CCN(C(=O)C(O)CCNC(c3c[nH]nc3[N+](=O)[O-])=O)C2)C1 c1(C=O)cc(C)cc(C#N)c1.C1(CSC)(NC(=O)CC2CCOC2)CCC1 c1(NC(N(C)CC2CC3CCC2CC3)=O)ncnc2ccnn12 c1(C(=O)NCC(CO)NC(CCN(C(CCC)C)C)=O)ccc2c(c1)OCCC2 Cc1sc(O)nc1C(N1CC(CNC(=O)C(C)O)CC1C)=O C1(NC(c2c(C)nn(CC(F)(F)F)c2)=O)CC(N2CCOCC2)C12CCC2 CCCC(C(=O)N1CCC(O)C1C(=O)NCCc1ccc(F)cc1)C(C)C c1(C(=O)NC(CCOC)CNC(=O)C(C)c2ccsc2)c(OC)cccc1O c1(C(=O)NCC(CNC(c2cn(C)nc2O)=O)O)cc2c(nn1)CCCC2 c1(NC(C(N2CCCN(CC=C)CC2)=O)=O)cc(Cl)c(OC)cc1F CCC(C)C(C)(O)CNC(=O)CN(C(=O)CC1CCCN(C)C1)C1CCC1 c1(OC(CC)C(=O)N)cccc(C)c1.C12CC(C1)N(C(C1CC3(CC3)C1)=O)C2 c1(CNC(N(C)Cc2cc(Cl)ccn2)=O)cc(Br)cnc1Br C1(C(=O)OC)CSCCN(C(=O)CC2CC3(CNC3)CO2)C1 N1(C(C(C(=O)OC(C)(C)C)(C)C)=O)C2CCC1CN(C(C1COCCO1)=O)CC2 C=CCCCCCN(c1cc(NC2CN3CCC2C3)ncn1)C c1(C2(C)CC2)nc(N2CCC(NC(c3cnn(C)c3Cl)=O)CC2)cc(Cl)n1 Cc1ccc(C(=O)N(CC(C)NC(c2c(C)noc2C)=O)C)c(F)c1F Cc1cc(=O)c(C(=O)NCC2CCCCC2NC(c2n[nH]c(O)n2)=O)c[nH]1 N1(C(CNC(C)=O)=O)CCC(C2CC(NC(=O)CCN3CCCC3)C2)C1 c1(C(N2CC(OC)CC2)=O)cc2n(n1)CCCO2.C1(CC=O)NC(=O)NC1=O.N c1(-n2cc(CC3CN(C(c4scnc4I)=O)C3)nn2)cc([N+](=O)[O-])ccc1Cl C#CCCC(C(=O)N(CCC(=O)NC)CC)NC(c1ccccc1O)=O C1(CS(CC)(=O)=O)CC(C)N(C(=O)Oc2ccncc2Sc2ccccc2F)C1 N1(C(C(C)OCCOCC)=O)CC2CC1CN(C(c1ccc[nH]1)=O)C2 C1CN(C(=O)CC2CC3CC3C2)C(C)(C)C1.C(C=CC(=O)N)(CC)=CC C1(NC(C(CCOC)C)=O)(CNC(c2cc(OC)ncn2)=O)CCCCC1C c1(C(=O)NCCC2(O)CN(C(=O)C=CI)C2)cccnc1OCCO C(=O)(CC(C(C)CC)NC(=O)C=C(C)C(C)C)N(CCCC)CC(N)=O Cc1sc(C)c(C(c2nnnn2C2CCCC2)NCCc2ccc(Cl)cc2)c1Br c1(N(CC(C(C)C)OC)C(=O)NC(COC)C)ccc(-c2ccccc2)cc1 CC(=O)CCCC(C)C(=O)NCC(CC(=O)NC(c1cnsc1)C)C1CCC1 C(=O)(C#CC1CCCCC1)N1CCC(NC(c2cc3occc3s2)=O)(CF)C1 C1(NC(c2cnnc(O)c2)=O)CC2CC(C1)N(C(=O)CCO)C2.CC(F)(F)F c1(CNC(=O)C=CCNC(=O)Cc2ncccc2F)ncc[nH]c1=O C1(N(C(c2c(C)cc[nH]2)=O)CCO)CCN(C(c2ccc(C3CCCO3)[nH]2)=O)CC1 N1(CCc2cn(CC(=O)N(CCN(C)C)CC)nn2)CCC(C)(C)C1 CCCCC(C(=O)NC1(C(=O)Nc2cnn(CCO)c2)CCSC1)N(C)C c1(CNC(C2C(C(N(CCCO)C(C)C)=O)C2)=O)cccc(O)c1F CCCN=C(NCCc1ccc(F)cc1Cl)NCC1CCOCC1C C(C(O)CC(=O)NCc1cc(CC)no1)NC(COCCCCC)=O CN1CCC(C(=O)NC(C2CCOC2)C)CC1.C(=O)C(C1CCC1)C1CCC1.N Cc1csc(=NCC(=O)N(C(C)CNC(C2CC3CC3CC2C)=O)C)[nH]1 CC(CC(F)F)C(=O)NC1CCC1CNC(=O)COc1c(Cl)cccc1Cl CC(C)CCCCCCNC(=O)C(C)N(C)C(c1ccc(CO)cc1)=O N(C1CCc2cccnc21)C(CC(CNC(c1cnc(CC)nc1)=O)(C)C)=O c1(C=O)cccc(Cl)c1F.C1(C(=O)OC)C=CC1C(=O)NCC1CC1.N CCC(CC(=O)NC(C1(C(=O)N(C2CCOCC2)C)CC1)C)C(F)F c1(C(=O)NC(C2CCOC2)C#C)ccn2ncc(Br)c2c1 C(=O)(C(C(F)(F)F)C(F)(F)F)N1CC(C(C)C)CCC1.c1(CC(=O)N)cn[nH]c1 C1CCCCC1.c1(CC(N2CC(C)(N(C)C(=O)C3CC3)C2)=O)cnc[nH]1.C CCC(CC)C(=O)N(CCN(C(c1[nH]nnc1COC)=O)CC)CC N1(C(C2C(C)(C)CC2)=O)C2CCC1CC(NC(c1cnn3ccncc13)=O)C2 C#CC1(OCC(N2CCC(OCC(N3CC(=CC)C3)=O)C2)=O)COC1 Cc1csc(C2CCN(C(C3(CO)CCNC3)=O)C2)n1 C1(NC(C(=O)OCC)(C)C)CCC(C)(C)N1C(=O)OC(C)(C)C C(c1nc(C)c(C)[nH]1)=CC(N1CCC(O)C1)=O.Cc1coc(C=CC=O)n1.N CC1CN(C(c2ccccn2)C(=O)NCCC2(C)CC2)CC1N=[N+]=[N-] Cc1oc(C)c(C(=O)NC2CC(O)(CNC(=O)C3=COCCO3)C2)c1C C1(C(COCCC)(C)C)CCCCN1C(C)C.C12(CC1)NC(=O)N2 c1(C(=O)NC2C=CCN(C(c3ncn(C)c3)=O)C2)cnc2cccnc2c1 C1(C(=O)NC(CC)C(F)(F)F)CCN(C(c2ccn(C)c2)=O)CC1O C12(CCOCC1)C(=O)OC2.C1(C(C(=O)OC)(F)F)CCCC(=O)C1 N1(C(c2c(C)nc(CC)o2)=O)CCC(O)(CC)CC1.O(C(F)(F)F)CC=O.N CCCC(C(=O)NCc1cn(C2CN(C(=O)C=CSC)C2)nn1)C(C)C c1c(C)occc1=O.C(=O)(C(F)(F)CC)N(C1CCN(C(=O)CO)CC1)CCC Cc1nsc(N)c1C(N1CCN(CC(=O)NC(c2ccncc2)C)CC1)=O C1(NC(CCOCC#C)=O)C2CC3CN(C(=O)Cc4ccsn4)C1C3C2 C1(NC(C(C)NS(C)(=O)=O)=O)(C)CCCCC1C.C1(C=O)CCC2CC12.N c1(SC)cccc2c1CN(C(=O)C(O)C(C)c1ccccc1)CC2 C1(CC2N(C(c3cn(CCC)nn3)=O)CCC2)CCCCN1C(c1cc[nH]n1)=O C=C(C)CCC(=O)N1CCCC1CN(C)C(c1cc(C)c(CC)s1)=O C(=O)(CC(F)(F)C(F)F)N1CC(NC(c2nc(C)oc2C)=O)C(CO)CC1 CS(=O)c1cccc(C(=O)NC2CC3CC(NC(c4cncc(F)c4)=O)CC23)c1 c1(C)ccnc(C(F)(F)F)c1F.C1(S(C)(=O)=O)(C(NC(C)C)=O)CC1 c1(OC)nn(C)c(Br)c1C(=O)NC(C)C(CO)NC(=O)CCC1CC1C C1(C(=O)OC)CCN(C(=O)CN2CCCCCC2)C(C2CC2)C1 Cc1c(C=CC(=O)NCCC2CC2)cnn1C.C(=O)CC.C1(C=O)CCC1 C(=O)(C1Cc2ccccc21)NC1CC2CN(C(c3c(OC)cccc3)=O)C1C2 N1(C(C(COC)N(C)C)=O)CCC(CCCCNC(=O)C(CCO)N(C)C)CC1 c1(NC(=O)NCc2cc(Br)c[nH]2)nc(N2CCCCCC2)ccc1Cl C(C1CCCCC1)=CC(=O)NCCOCC(=O)N(C)CC1CCCOC1 C1(NC(C2CN(CC)C(=O)C2)=O)CC(F)(F)CC1.c1(C=O)cc(F)cnc1O.N C1(NC(C(Cc2ccoc2)NC(COCCCN=[N+]=[N-])=O)=O)CCCC1N=[N+]=[N-] N1(C(CCc2ccc(CC)cc2)=O)CCC(F)C(NC(c2nccnc2C)=O)C1 C1(C(N(C2CCCC2)CC)=O)CCN(C(=O)Cn2ccc(C)n2)CCO1 c1(C(N2CC3C(NC(C4C(COC)C4)=O)C3C2)=O)ccc2cnc(C)cc2c1 c1(C(=O)N)cnnc(C)c1C.c1(CCC)ccc(NC(C2(C)CC=CC2)=O)cc1 CCCCC(CC(=O)Nn1cnn(C)c1=S)NC(=O)CSCC(F)F c1(C(C(=O)NC2C(NC(c3n(C)cnc3)=O)C2)O)cc(F)c(F)c(F)c1 N1(C(C(Cc2ncn(C)c2)O)=O)CCOCC(NC(=O)CN2CC3CC3C2)C1 C1(NC(c2n(C)cnc2)=O)C2CCN(C(=O)Cc3ccccc3)C12.CC(C)(C)C c1(OC)cc(N2CCCC(C(=O)NC3(C)CCOCC3)C2)nc(OC)n1 c1cc(C)c(O)cc1C.c1(COC)ccc(CNCC2(CS)COC2)cn1 C1(N(C(=O)CSCc2cscn2)C)CCC(C)CC1.C(=O)CCC1CCC1 C(=O)(CCCCC1CC1)N1CC(c2cnco2)C1.C(=O)(CC(=O)N)NCC.C c1nc(C(F)(F)F)cs1.C1(NC(=O)OC(C)(C)C)CC(C(=O)OC)C1 CS(=N)(=O)C1CN(C(C2CCCN(C(C3CCO3)=O)CC2)=O)C1 c1ccccc1[N+](=O)[O-].c1(OC)ccc(OCCCC(C)C)cc1.c12ccc-1s2.CC c1(CC(N2C(CNC(C=C(CCC)C)=O)COCC2)=O)ccc(C#N)cc1 O=C(C1=NOC(c2ccccc2)C1)NCC1(NC(=O)COC(F)F)CCCCC1 C(C[Si](C)(C)C)NC(=O)NCC(COC)OC CCCC(CNC(C1CC1(F)Cl)=O)C(=O)NCC1(C)CC=CCC1 c1(N2CC(O)(CCNC(C3C(C)=C3)=O)C2)cc(Cl)nc(C(F)(F)F)n1 C(=O)(C(F)C(CC)CC)N1C(CC(=O)NCc2ccc(CC)s2)COCC1 N1(C(c2cc(COC)[nH]n2)=O)CCCCC1.c1(CC=O)cccc(C(F)F)c1.N N1(C(C=C(CC)C)=O)CCCC(C)(C(=O)NCc2ccon2)C1 C1(C(c2nc(-c3ccccc3)nn2Cc2ccccc2)CCC)CCCCCC1 N1(C(Cc2ncc(C)o2)=O)C2CCCC1CC(NC(C1CN(C(C)C)C1)=O)C2 c1(C(=O)NC(CN=[N+]=[N-])C(=O)NC2CCS(=O)CC2)cc[nH]c2nccc1-2 C(=O)(C(F)C(C)(F)F)N1CC(C)(C(=O)NCC(C2CCCC2)OC)C1 CC1(C(N2CCC(CC(N3CCC(n4cccn4)C3)=O)C2)=O)CC(C#N)C1 C1(NC(c2c(C)c(F)cnc2)=O)CC2COCC(C1)N2C(=O)Cc1cn(C)cn1 C1(C)(C(N2CCC(C3NC(=O)N(C)C3=O)CC2)=O)Cc2ccccc2C1 c1(C(=O)OC)ccc(C(=O)NCC2(C=O)CC2)cc1.N1(CC)CC=CC1 N1(C(C(C)CN(C(=O)CCc2cnccn2)C)=O)CCSCC(C)C1 C1(NC(=O)CC2CCCC2)CC2(C1)CC(NC(=O)CCCCBr)C2 c1(C(C(CN2CC(C(=O)OC)C(O)C2)=O)=O)ccc(O)c(F)c1 C1(C(=O)NC2CN(C(c3sc(C)c(O)n3)=O)CC2C)CN2CCN1C(C)C2 C1(C)(C=O)CC=CCC1.N1(C(CNC(=O)OCC=C)=O)CC(CCC)C1.N c1(OC)ccnc(O)c1CNC(=O)N(C1CCC1)Cc1ccc(Br)cc1 C1(OC)C2CC1CN(C(c1n[nH]c(=N)n1C1CC1)=O)C2 N1(C(c2cc(C)[nH]c2)=O)CCC2(CC1)OCCC2NC(C1CCCC1(C)C)=O C=C(F)CN=c1nc2c(ncn2CC)c(NC2(CC)CCCCC2)[nH]1 Cc1ccc(C2(C(=O)NCC=CC)CCC2)cc1.C1(C(=O)N)CC(O)CN1C C1(C(N(CCC)C)=O)CCCCC1(C)C.c1(CC(=O)N)ccc(C(F)(F)F)nc1 Cc1scnc1C(N1CCC(CCC(=O)NCC(c2cnn(C)c2)O)C1)=O c1(N(CC(C)CNC(C2CCOC2)=O)C)nnc(C2CC2)o1 C(CC(=O)N1CC(C)(O)CO1)N(C(C1C(C)(C)CCCC1)=O)CCO c1(CCC)cccc(C(=O)NCC2(O)CN(C(c3cc(OC)ns3)=O)C2)c1 n1(CCN(C(CC)C)C)c(N2CC(C)CC2C)nnc1-c1cnc[nH]1 n1(COCC)nnc(C(=O)NCC2(F)CC2)c1N C(=O)(C1CCc2nccn21)N1C(C(=O)NC2CCCCC2)CCC12CC2 C1(C=O)CN2CCC1C2.c1(C(N(CC(C)(C)C)CC(C)C)=O)cc(CC)on1 Cc1cc(F)c(N)cc1C(=O)NC1CCN(C(C2(CC(F)F)CC2)=O)CC1C Cc1cc(C)c(C(=O)N(C2(C(=O)NCC(C)(CO)CO)CCC2)C2CC2)s1 C1(C(=O)NCCOCCC)CCN(C(=O)C=CC(C)C)C1CC C1(CC(=O)Nc2cc(Cl)ccc2C(c2ccccc2)=O)CCCC2CCCCC12 C1(C(=O)NC(C(C)C)CO)CCCN(C(c2cc(CO)ccn2)=O)C1 c1(C(N(C)CC2(O)CN(C(CCCCSC)=O)C2)=O)ccn2ccnc2c1 Cc1cc2ccc(C(=O)NCC3CN(C(C45CCC(C4)C5)=O)CCO3)cn2c1 C(C1=NOC2CN(C(=O)C=CCO)CC12)NC(c1cc2n(c1)CCC2)=O C1(NC(C2(OC)CC(CF)C2)=O)CN(C(=O)CN=S(C)(C)=O)CC(C)(C)C1 c1(CNc2nc(CC)on2)cn2ccsc2n1 C1(C(=O)NC(C2CCN(C(C3CC3F)=O)CC2)CO)CC2(CCOCC2)C1 Cc1nccc(C(=O)N(CCCCN(C(=O)Cc2ccc(Br)cc2)C)C)n1 c1(C(N2CC(NC(C)=O)CC3(C2)CC3)=O)cc2n(n1)C(C(F)(F)F)CC(C)N2 N1(C(C2CC(C)(F)C2)=O)CCC(CCNC(C2(C3CCCO3)CC2)=O)CC1 N1(C(C=Cc2ccn(C)c2)=O)CCN(C(=O)Cc2ccns2)C(CCO)C1 C(=O)(C=C1SCC(=O)N1C)N1CCCC(O)(CNC(C(C)CC(C)(C)C)=O)C1 Cc1cccnc1C(F)(F)C(=O)NC1CCCN(C(C2CCC(C)(C)C2)=O)C1 Cc1cc(C(N2CCC(N(CCO)C(C3CCN(C)C3)=O)C2)=O)nnc1C Cc1ccc2c(c1)C(N(C1CC1)Cc1ccc([Si](C)(C)C)cc1)CCCO2 c1(N(CCCNC(c2cc(Cl)c[nH]2)=O)CC)nc2cc(C)ccc2o1 CCCCC(C(=O)NC12CCC(C1)N(C(C1CN(S(N)(=O)=O)C1)=O)C2)C(C)C C1(c2n(C(C)C)nnn2)(Nc2ccc(O)c(Cl)c2)CC2CC1CC21CC1 C(=O)CCC(C)(C)C.c1(C(N(CC)CC)=O)ccc(N)cc1C(C)(C)C.N c1(OC)n[nH]c(C(=O)NCC2C(C)CCN2C(c2coc(O)n2)=O)c1Cl N1(C(COCCOC)=O)CC(NC(=O)CC(=O)N(C)C)C(C)C1 Cc1cc(C(=O)NC(C)C(C)(C)NC(C2CC(C)CC(=O)N2)=O)cc(F)c1 N1(C(C(=O)N(CCNC(C=C(CCC)C)=O)C2CC2)C)C(=O)CCC1=O C1(C(=O)N)CC12CCOCC2.C1(CNC(C(C)c2cccs2)=O)CC(F)(C)C1 C=C(C(=O)N1CCC(c2cccc(C)n2)C1)C1CC1 C1(NC(N)=O)CCN(C(=O)CC(C2CC2)NC(c2csc(O)n2)=O)C1 C1(NC(c2c(OC)cc(C)s2)=O)CC2CCCC(C1)N2C(c1sccc1Cl)=O N#Cc1ccc(S(=O)(=O)NCC(=O)Nc2ccc(F)c(Cl)c2)cc1 N1(C(C2C(NC(C(CCC(C)C)F)=O)CCOC2)=O)CC2(C1)CC1(CCC1)C2 C1(C(=O)NC(C(C)C)c2nc[nH]n2)CC(C)CN(C(=O)C(O)C2CC2)C1 N1(C(Cc2cn(CC)nc2)=O)CC(C)(C)CC1CNC(C1(F)CC1C)=O n1(CC(C)NC(C(C)NC=O)=O)cc(CNC2CCCCC2)nn1 Cc1cc(C)c(C(=O)N(C(=O)CN(C)C)CC)c(O)c1.c1ccc(Cl)cc1.S CN=c1nc(N(C)CC2CC(O)C2)[nH]c(=NC2CCCC2C#N)[nH]1 N1(C(c2ccn(CC)n2)=O)C(C)CC2CN(C(c3ccc4cnnn4c3)=O)CC12 c1(C2(CC)CC2)cccc(-c2nc(C(=O)NC3CCCCC3N(C)C)no2)c1 c1(CC)nccnc1C(=O)N(CCC)C(C)C.c1(C2(C=O)CC2)cc[nH]n1.N c1(OC)cc(C(=O)Nc2cc(Cl)ccc2Cl)c(Cl)cn1 N1(CC=O)CCC(C)CC1.c1(CC(C)C)nc(C(=O)N)cs1.C1(F)CCC1.C c1(C(=O)N)ccc(-c2ccccn2)o1.C(C)(C(=O)N(CC(C)C)C)N(C(C)=O)C c1(-c2c(OC)ccs2)ccnc(NC(C2CCCC(C=O)C2)=O)c1.C(C)(C)C.O c1(OC)ccc(C(N2CCC(NC(C3CCSC(C)C3)=O)C2(C)C)=O)c(F)c1N c1(CCCCCC)ccc(CSC(CCSC)C(=O)NCCOC)cc1 CCC(C)C(O)C(=O)N1CC(CNC(=O)C=Cc2cccc(O)c2)C1 C(CO)(C(=O)NCC=CCC(=O)N(CC(F)F)CC1CC1)N(C)C CC1CN(C(=O)Cc2ccnn2C)CCC1CNC(c1sc(C#N)cc1Cl)=O C(=O)(C(C#N)(CC)CC)N(CCNC1(O)COCCC1O)CC C1(C(N2CC(N(C)C(C3CC(O)C3)=O)C(F)C2)=O)(COC)CCOCC1 c1(COC)nc(NC2CCCN(C(=O)C3=CCCS3)CC2)cc(O)n1 C1(CC(=O)NCCC2CCCN(c3nnc(CO)s3)C2)CCCC2(CCC2)O1 n1(CC=C)c(SCCNC(=O)CCc2nnc(C3CCCOC3)o2)nnc1S N1(C(C2C(CC)CC2)=O)CCC(C(=O)N(CC(C)(O)C2CC2)C)C1C(C)C Cc1cccc(CCNC(c2n[nH]cc2CNC(=O)C)=O)c1.C1CCOC1.O c1(C(N(CC(CN(C(CCCC(C)=O)=O)C)O)C)=O)c(Cl)ccc(F)c1C c1(CC)nc(CNC(N2CC(OC3(OCC(F)F)CC3)C2)=O)n[nH]1 c1(-n2ccc(C(N3CCC3)=O)n2)ccc(F)cc1.C(=O)(CC(=O)N)NCC#C Cc1cc(C(F)(F)F)nn1C(C)SC(C)C C1(CCC(=O)NCC2COCCN2C(=O)CC2CCCO2)CCCCCC1 N1(C(C=CC(C)=O)=O)CCC(F)(CNC(=O)C(C2CCOCC2)F)CC1 C1(C(N2CC3C(NC(C(C4CCCC4)OCC)=O)(C3)C2)=O)CC2CCC1CC2 c1(C(=O)NCC2C(C)CCN(C(C(CC)OC)=O)C2)cnc2ncnn2c1N CCCC(CCNC(C1CC(=O)CN1C(=O)CCCSC)=O)CCC c1(CC)ccc(CNC(=O)NC2CCC(=O)NC2C)cc1F C(=O)(CC1CCc2ccccc21)NCC1CCCCN(C(C(F)=CCC)=O)C1 C(N=c1ncc(Cl)c[nH]1)C1C(NC(c2cc(C3CC3)no2)=O)CCCC1 C1(NC(C2CC(=O)NC2)=O)CCOCC1NC(=O)CSc1nnc(S)s1 C1(C)(CCC)C(=O)NCCN1C(c1ccc(CCn2cnc([N+](=O)[O-])n2)cc1)=O c1(C(=O)NCC2=CCN(C(C)=O)CC2)cc2c(C)n[nH]c2nc1O c1(OC)cc(C(=O)NCCC2CCC2)c(F)c(Cl)c1.c1(C=O)ccnc(C)n1 N=c1ccc(C(=O)NCC2CCCCC2NC(C2CCC(CO)CC2)=O)c[nH]1 CC1(C)NC(=O)N(CCC(=O)N(c2ncc(C(=O)O)cc2Br)C2CCOC2)C1=O N1(C(C(CC)SC)=O)CC2(CCNC(c3cc(OC)cc(F)c3)=O)CCC1CC2 N1(C(CC(C)OC)=O)CCCC(C2CC2NC(=O)CC2(O)COC(C)(C)C2)C1 C1(CC=C)CCCCC1NC(C1CCC(n2cc(CN)nn2)CC1)=O c1(C(N2CC(CNC(c3ccc4c(c3)CCO4)=O)C2)=O)ccc2[nH]cc(Br)c2c1 c1(C2(CNC(C(C)NC3CCCC3)=O)CCC2)cc(Cl)ccc1F c1(C2C(C)C2)c(C(=O)OCc2nnnn2C2CC(F)(F)C2)cnn1C Cn1ncc2c(N(c3ccc(C#N)nc3OC)C3(C#N)CCNC3)ncnc12 Cc1cc(C(=O)NC2(C)CCCCC2C(=O)NC(C)(C)CCCO)ncc1N N1(C(c2nc(SC)sc2)=O)CCC(N(C(=O)C=C(C)c2ccco2)C)CC1 C1(CNC(C2(CC)CC2)=O)CCCN(C(=O)CCc2cccc(OC)n2)CC1 c1(C(=O)NC2C(CNC(C=CCC)=O)C2)ccccc1.[SH](=O)(=O)CC c1(C(N2CC(O)(C(C)NC(COCCCCC)=O)C2)=O)ccc(O)c(F)c1F Cc1cc(C(N2CCOCC(NC(=O)Cc3ncc(Cl)s3)C2)=O)c(N)c(Cl)c1 n1(CC(=O)NC2CN(C(C=C(C)C(C)(C)C)=O)C2)cccc(C)c1=O C1(NC(N2CC(C)N(CC(F)F)CC2)=O)CC2(CCOCC2)CO1 N1(C(CC=CCC)=O)CCCC1(C)CC=C.C1(C(F)(F)F)(C=O)CC(=C)C1.N c1(CC(N2CC3C(N(C)C(C4CCO4)=O)C3C2)=O)cc2ccccc2nc1O c1(C(N2CCC(C(C)NC(C3CCC4CC4C3)=O)C2)=O)cccn(C)c1=O Cc1cc(N2CCC(CCC3CC3)CC2)ncc1S(=O)(=O)NC1CC1(C)C(F)F c1(C(N(CCN(C(CC2C(CC)C2)=O)C)C)=O)sccc1.[SH](C)(=O)=O.N CCS(=O)(=O)c1cccc(C(=O)NCC#CC)c1.c1(C=O)c[nH]nc1C(F)F.N C1(C)(CC)CCC(C(=O)NCC(C)C)O1.C1(CC=O)(N(C)C)CCC1.N N1(C(c2cc(Br)cs2)=O)CCC(F)(C(=O)Nc2cc(CO)ccn2)CC1 c1(CC(=O)N)cc(Cl)ccc1[N+](=O)[O-].c1(OC)csc(C(=O)NC2CCC2)c1 C(=O)(C(CC(C)C)ONC(C1COCCN1CC(C)C)=O)NCCOC(C)=O C1(C=O)CCCC1(F)F.CC(Cc1ccccc1)C(=O)NCC1(C)CC1(F)F CC1CCCC(N=c2cc[nH]cc2S(=O)(=O)NCCCCCCCC(F)(F)F)CC1 C=CCCCC(=O)NCC(CNC(c1cc(C)n(C(C)C2CC2)n1)=O)OC CCC(O)C(C)(C)C(=O)N1CC(C2CN(C(=O)C(F)C3CCCC3)CCO2)C1 N1(C(c2c(SC)nccn2)=O)CCC2C(CCCN2C(c2cc(C)cs2)=O)C1 N1(C(C(COC)C)=O)CCCN(C(=O)CCc2ccccc2F)C(C(C)C)C1 NS(=O)(=O)c1ccc(F)c(C(N2CC3CN(C(=O)C(F)(F)F)CC3C2)=O)c1 c1(SC)ccc(C(=O)NC2CCC2CNC(=O)Cc2cc(Cl)cs2)o1 C1(NC(Cc2nnc(C)o2)=O)CCCCC1.c1(CC(=O)N)cnn(C(C)(C)C)c1 Cc1cnccc1C(C)C(=O)N(C(C)CNC(=O)C=CC=C(Cl)Cl)C C1(CC)CN(C(C2CC(C)CO2)=O)CCC1NC(c1cc(F)cnc1Cl)=O c1(CN2CCC(O)(C(=O)NCc3ncn(C)c3)C2)c(I)ccnc1F Cc1cc(N)c(F)c(C(N2CCC(CN(C(=O)CCN(C)CCO)C)C2)=O)c1F Cc1cccc(C)c1-n1nc(-c2ccc(Cl)nc2)nc1C1CCC1F c1(OC)cccc2c(C(N3CCC(F)C(NC(C4(F)CC4)=O)C3)=O)n[nH]c12 Cc1cc(C(N2CC(=O)NCC2C(=O)Nc2cc(F)ccc2O)=O)c[nH]c1=N Cn1cccc1C=CC(=O)NCC1CCCN1C(c1cc(CF)on1)=O c1(C(=O)NCC(CC)NC(=O)C(O)CSC)ccc2nc(S)[nH]c2c1 N1(C(c2ccc(F)cn2)C(=O)NC(C)C)CC2(CCCC2)CC1C Cc1[nH]nc(C(N2CCC(C)C2CNC(=O)C=Cc2cccnc2)=O)c1F Cc1ccc(CN=C(NCC(C)(C)F)NCC2CCCCO2)c(C2CC2)c1 c1(C(=O)NC2CCN(c3cc(CC)nc(C)n3)CC2C)cnc2ccnn2c1O O=C1CC(C(=O)NC(CNC(C2(C(F)F)CCCC2)=O)C2CC2)CCN1 CC1C(C(=O)NC(C)(CNC(c2cccc[n+]2[O-])=O)C2CC2)=Cc2ccccc21 CCCCCC(C)(C)CNC(=O)C=CC(C)NC(=O)C(C)(C#N)CC c1(OC)ncnc(C(=O)NCC2CCN(C(=O)C(C3CCC(=O)N3)C)CC2)c1F N1(C(c2nc(C#C)sc2)=O)CC(C)CN(C(c2cc(C)ccc2N)=O)CC1C C(CC1CCOCC1)(C(=O)NCCCN=[N+]=[N-])NC(COCCC#C)=O c1(C(N2CC(CC(C)NC(c3cnc(O)o3)=O)C2)=O)ccc(C(C)O)cc1 CC(C)(C#N)C(=O)N1CCC(C)(CCNC(=O)CCc2nc(C3CC3)no2)C1 CC(CC(=O)NCC(F)CNC(c1ccc(Cl)[nH]1)=O)NC(C1CCCC1)=O CCC(CC)CC(=O)N(CC(C)NC(=O)Cn1ccc(Br)cc1=O)C CC(C)CC(C(=O)O)NC(C1CCCN1C(c1cc(Cl)ccc1Cl)=O)=O c1(C2(C(C#C)(C)NC(=O)NC3COC3)CC2)ccccc1O N1(C(c2cc(CC)on2)=O)CCN(C(=O)CSC)C(C(C)C)C1.C1CCCO1 C1(CNC(c2n(C)cnn2)c2nnnn2CC2CC2)CCC2(CO1)CC(O)C2 N1(C(C(CC)C)=O)CC2(C1)CN(C(=O)Cc1c(C)nn(CC3CC3)c1C)C2 N1(C(C(C)C)=O)CCCCC1C(=O)NCC(CO)NC(C1CC(F)(F)C1)=O CC1(CC#N)CCN(C(=O)C(F)(F)c2ccncc2)C1 C(C(C)C)(C(O)C(=O)NCC(C)(C)CC(=O)N1CCCNC(=O)C1)OC C1(C(N2CCCC(CF)C2)=O)CC2CCC(C1)C2O Cc1cc(C)n2ncc(CNC3(c4nnnn4C(C)(C)C)CCOC(C)C3)c2n1 C1(CC(=O)N(CC(C)C)C(=O)C2CC2)(CCN)COCCO1 Cc1ccc(CC(=O)NC2CN(C(=O)C(c3ccccc3)C)CC2F)c(C)c1 CC(C)S(=O)(=O)CC(=O)NCC(C)(C1CCC1)NC(=O)C.c1ccccn1.O C1CC2CCC(C1)N2C(=O)Cn1cc(C2CC2)cn1.C=C(C)CC(C(=O)N)OC c1(C(=O)NC(CNC(C(C(CC)C)C)=O)(C)C)cc2sc(=O)n(C)c2s1 Cc1nc(N2CCC(NC(=O)CO)C(C)C2)ncc1[N+](=O)[O-] c1(C(=O)NCCC(C(=O)Nc2ccccc2)OCC)ccn(C)c(=O)c1.S n1(CC(CC)CC)nc(-c2ccccc2Cl)nc1-c1cc(CO)on1 c1(CC)nonc1C(=O)NCc1csc(C(=O)N)c1.C1(CCC)CCCO1 c1(CC(=O)NCC(n2cc(CNc3nccs3)nn2)C)cncn1C1CC1 Cc1cc(C(=O)NC2CCN(C3CCN(C)CC3)C2)cc(=NCC(F)(F)F)[nH]1 CC1CN(C(=O)CC2CCC(C)(C)O2)CCN1C(c1cc(Cl)no1)=O c1(NCC(N2CCC(NC(C(CC)COC)=O)C2)=O)ccc(C#N)cc1 c1(C(=O)NC2C(C)CN(C(c3cccn3C3CC3)=O)C2)cc(C#N)c(O)nc1N c1(N(C)Cc2ccc(OC)c(F)c2)nc2ccsc2c(=NC2COCC2C)[nH]1 c1(C(=O)NCC(COC)O)cc2c(s1)CCOC21CCN(Cc2c[nH]nc2C)CC1 c1(C(=O)NCC2(F)CN(C(CC3CC(C)OC3C)=O)C2)nn(C)c2c1CSCC2 C1(CN(CCN(C)C)C(=O)N)COc2ccccc2C1.C1(S(C)(=O)=O)CCC1 C=CCCCCC(=O)N1CC(C)CCC1CNC(=O)C=CC(=O)OCCCC c1(NC2CC3CN(C(C(CCOC)C)=O)CC32)nc2c(cc1Cl)C(=O)OC2 C1(C(=O)N)CC(C(C)(C)C)=NO1.CC1CCCCN1C(c1cnn(C(F)F)c1)=O c1(CCNC(C(CC=C)C)(C)c2nnnn2CC=C)c[nH]c2cccc(C)c12 CCCC(C(=O)NC1(C2CCN(C(=O)Cc3cscn3)C2)CC1)C(C)C c1(CNC(CNC(C(CC)C)=O)=O)nnc2c(=O)[nH]ccn12 C1(NC(C(C2CCC(C)CC2)CC)=O)CCCN(C(c2ccn(CC)n2)=O)C1C Cc1cccc2[nH]cc(C(=O)NC(C)(C)CNC(C3(C)CCNC(=O)C3)=O)c12 C1(C(C)C)C(NC(C2(C3CCCCO3)CC2)=O)CCN1C(c1cncc(N)n1)=O CC1OC2(C(=O)NCC3(CCNC(=O)CC)CC3)CC1C2.c1nncn1C N1(C(C(CC(C)C)F)=O)C2CCCC1CC(NC(c1cc(F)c[nH]1)=O)C2 N1(C(C(C2CCCO2)NC(C(C(C)C)OC)=O)=O)CCC(C)(OC)CC1 c1(C=O)cc(S(C)(=O)=O)cs1.C1CCCCC1.C1(N(C)C)CC(C(=O)N)C1.C C(=O)(C1CCCc2nncn21)NC1CCN(C(c2c(C)nccn2)=O)CC1F c1(C(=O)NC2(CNC(C3(C)CCCNC3=O)=O)CC2)onc2ccccc12 CCC(C)C(C(=O)N1CC2CC1(C(N)=O)C2)N(C)C(c1cnn(C)c1N)=O C(=O)(C1COc2ccccc21)N1CC(C(C)NC(c2sncc2Br)=O)C1 C12(C=O)CCC(C)(CO1)C2.C1(COC)CN(C(=O)C(C)(C)C2CCCO2)C1 c1(C(N2CCC(CN(C(C3C(C=C)C3)=O)C)C2)=O)cc(N)ccc1[N+](=O)[O-] N1(C(C(C)SC)=O)CC2CN(C(=O)CCC(C)c3ccccc3)CC2C1 Cn1cnc2cc(C(=O)NCCNC(=O)CCOC3CCOCC3)cnc12 C(=O)(C(C)CC(C)(C)C)NC1(C2N(C(CNC(CC)=O)=O)CCC2)CC1 c1(C(N2CCCC2C2(C)CC2)C=O)ccnn1CC(F)(F)F.CC(C)C.CC Cc1cc2cc(C(=O)NCCC3CCCN3C(c3cnsc3)=O)c(Cl)cc2[nH]1 N1(C(C2CC(C)OC2)=O)CCN(C(c2cc3n(n2)CCCC3)=O)C2(CCC2)C1 N1(C(c2ccc(COC)[nH]2)=O)CCCN(C(c2cccc(CF)c2)=O)CC1 c1(OC)ccc(C)cc1C(=O)NC1CCC(NC(C2COCCC2C)=O)CC1 C12(C=O)CC1COC2(C)C.c1(C(N(C)CCOCC)=O)ncsc1C1CC1 c1(NCC(N2CC3C(C(=O)NCC4(CCO)CC4)C3C2)=O)ccccc1Cl N1(C(CCC=CC)=O)CCOC2(CCN(C(c3cc(C)sn3)=O)C2)C1 CC(C)CCCN(C)C(c1snc(Cl)c1Cl)=O.c1(CC(=O)N)cc(C2CC2)on1 c1(-c2c(CNC)cccc2)c(C(=O)Nc2cc(Br)ncc2C)nc2ccccn12 C(=O)(CN=S(C)(C)=O)NC1C(OC)CN(C(C2CCC2(C)C)=O)C1 CCCCCCCC(=O)NC1(CCCC(=O)NC2CC(O)C(O)C2)CCC1 c1(OC)cc(OC)c(C(N2CC(NC(C3CCCO3)=O)C(C)C2)=O)c(OC)c1 c1(OC)ccc(C)nc1C(N1CCC(C)C(NC(=O)CCc2cnn[nH]2)C1)=O CCC(CC(C)C)C(=O)N1C2CCC1C(CNC(=O)COc1ccccc1F)C2 C1(C(N(C(C2(O)CN(C=O)C2)C)C)=O)CC2CCC1(C)C2(C)C.C(C)(C)C C(C(=O)N=c1cc(C)n(C)[nH]1)(C1CCCC1)OC.c12cc(no1)C(=O)NC2 N1(C(c2ccc(C)nc2C)=O)CC2CN(C(=O)CCCC(N)=O)CCC12 C1(C(=O)NCC(C#C)C(C)C)CC(C)(C)CN1C(C1CC1C1CCC1)=O CCC(CC(F)F)C(=O)N1CCOCC1CN(C)C(c1ccc(C(C)C)s1)=O C1(C(=O)NC(C)CCCCNC(c2ccn(C)n2)=O)CCCC2(CCC2)C1 c1(C(C2CC2(C)C)NC2(C#C)CC2)ccc(C2CC2C)o1 C1(C=O)CCCC2(C1)CC2(F)F.C1CCOCC1.C1(CC=C)(C(=O)NC)CC1 Cn1nc2c(c1C(N1CC3CC1CN(C(=O)C(F)C1CCCC1)C3)=O)CCC2 c1(OCC)ncc(C=O)cc1Cl.C1(C(N2CCC2)=O)CC(=O)N(C2CC2)C1.N C(=O)(CCCN=c1nc(N2CCCC(OC(C)(C)C)C2)c2c([nH]1)CCS2)NC Cc1ccc(C)c(N(C)C(C2CCN(C(=O)c3cocc3C)O2)=O)c1 N1(C(C=Cc2c(C)ccs2)=O)CC2(CCC2NC(=O)CC2CCN(C)C2)C1 C(=O)(C#CC(C)(C)C)Nc1ccc(CC)nc1C.C(=O)C(C)S(N)(=O)=O.N C(=O)(CCS(C)(=O)=O)NCCCC(c1ccccc1)NC(C(C)O)=O N1(C(c2c(C)ocn2)=O)CCC(C2CCCN(C(C34CCC(C3)C4(C)C)=O)C2)C1 c1(C(=O)NC2C=CCN(C(Cc3cc(C)on3)=O)C2)nccc2ccsc12 c1(C(=O)NC(C(C)NC(c2ccc(C)cc2C)=O)C(C)C)ccnc2[nH]cnc12 C1(NC(C2CN(C(C)C)C(=O)C2)=O)CCCCN(C(c2ccnc(F)c2N)=O)C1 n1(CC)nnc(C(=O)N(C)CC2(CNC(=O)C(O)COC)CC2)c1C C1(C)(CNC(C(CC)NC(C)=O)=O)CCN(C(=O)COC2CCCC2)C1 N1(C(c2n(CC#C)ccc2)=O)CCCC(C2CCCN2C(=O)CCCN(C)C)C1 N1(C(C2=C(C)CC2)=O)CC(CNC(c2cc(Cl)cs2)=O)C(F)(F)C1 c1(CC)c(Br)c(C(N2CCN(C(c3cc(C)[nH]c3C)=O)C3CC23)=O)nn1C Cc1nc(CCCC(=O)NCC2CC(CNC(C3(CO)CCCC3)=O)C2)cs1 C1(O)(CCNC(c2c(C)cccc2)=O)CCCN(C(=O)C(C)(C)n2cnnn2)C1 C(=O)(CCC(F)(F)C(F)F)NCCCCNC(C1OCCN(C(C)=O)C1)=O C1(N(C(=O)CC2CC3CCC2O3)C)CCCN(C(c2cocn2)=O)CC1 C(C)(C)(CN=c1c(Br)c[nH]cc1[N+](=O)[O-])C1CCN(C(C2(CC)CCCCC2)=O)CC1 C(C(CC(F)(F)F)NC(c1sc(CC(C)C)nc1C)=O)NC(C(CC)N(C)C)=O N(C1CCc2ccccc21)C(c1ccc2c(Cc3nn[nH]n3)cnn2c1)=O CCC(C)CCC(=O)N1CCCC(CN(C)C(C2CCCCC2O)=O)C1 C=CCC(CC=C)NC(=O)C(Cc1cn[nH]c1)NC(c1cc(OC)ccn1)=O C1(NC(C=CC=CC)=O)CCN(C(c2cnn(CC(F)(F)F)n2)=O)C1.C C1CC(=O)N(C)C1=O.c1(OCC)ccccc1-c1cc(CNC(=O)O)on1 c1(C(=O)NCC2C3CN(C(CCC(N)=O)=O)C2C3)cc2sc(Br)cc2s1 c1(C(=O)NC(CCN(C(C(C)(CO)OC)=O)C)C(C)C)ccc(N)c(Cl)c1 CCCCC(C(=O)NCc1cnc(C)cc1C)NC(c1cnc(OC)s1)=O C1(CC)(CC)CCCN(C(=O)C(C)CN(C)C(C2COCOC2)=O)C1 Cc1cc(C(=O)NCC(C)CNC(C2(C)CC2)=O)nn1-c1ccc(F)cc1 N1(C(C(C)=CC2CC2)=O)CCC(NC(C23CC4CC2C3C4O)=O)CC(O)C1 c1(OC)cnnc(C(=O)NC2CCC2C)c1.c1(C(=O)N)coc(C2CC2)n1 c1c(Cl)cccc1Cl.N1(C(C2(CNC(C3CC3)=O)CC2)=O)CC(O)C1.C C(=O)(C(C(=O)NC12CC(NC(=O)C(C)SC)(C1)C2)C(C)C)OCC N1(C(C(C)n2cncn2)=O)CCCC(C)(C)C1CNC(=O)CN1CCCCC1 c1(OC)cccc2c1N(C(c1csc(C#N)c1)C(=O)NCC1CCOC1)CC2 C(C)(C)(CC(=O)NCC1CCN1C(=O)C(CCN(C)C)N(C)C)OC c1(C(N2CCCC2Cc2ccc(F)cc2)=O)c(-c2ccccc2)nc2sccn12 CCCC(C(=O)OCc1ncoc1CSC1CC1)OCC N1(C(COCC=C)=O)CCC(c2ccc(OC)cc2)C(NC(=O)CCS(C)=O)C1 c1(CC(c2c(C)nccc2)NC(C2CC23CCNC3)=O)ccc(C#N)cc1 C#CCCCCCC(=O)N(C1CN(C(=O)CCc2cnn[nH]2)CC1F)C O=C(CCCCC(F)F)NC1(CO)CCCN(C(c2ccnnc2O)=O)C1 n1(CC=C)cc(C(N2CC(N(C(=O)C(c3ccc(C)o3)C)C)C2)=O)nn1 C(N=c1[nH]c(=NCCCCCCCO)[nH]c2c1COCC2)C1(OC)CCCSC1 Cc1cc(C)c(C(=O)NCC2CCN(C(c3ncn(C)c3C)=O)C2)c(O)c1 c1(C(C)N(C)Cc2cccc(C(O)C(F)(F)F)c2)cccc([N+](=O)[O-])c1 S(=O)(=O)(c1ccc(F)c(F)c1)N1CCCC(O)C1.c1(C(=O)N)nc(Cl)sc1Cl.C c1(OC)cc(F)ccc1-c1cn(CCCNC(c2nc(C)no2)=O)nn1 C1(O)(C=O)CN2CCC1CC2.C1(NC(=O)NC)CCC(C=O)CC1.C1CC1.N O=C1NCC2CCC1N2C(=O)NCC12CCOCC1C2 C1(CNC(CCCC)=O)CN(C(c2cnncc2C(F)(F)F)=O)CCN1C Cc1cc(Cl)c(C(=O)OCc2ccc(Br)cc2Cl)cc1[N+](=O)[O-] N1(C(CC2CC(NC(Cc3cc(C)[nH]n3)=O)C2)=O)CCC2C(=O)NCC2C1 C1(CC(=O)NC(C(CCC)C)C)C2CCCC2N1C(c1nccnc1C)=O C1(CC(=O)NCCCCCNC(C2(N(C)C)CCCC2)=O)CC(O)C1(C)C C1(C(=O)NCC(C2CC2)NC(C(CC)=CC)=O)CC2(CCC2)CO1 C1(CNC(COCCOC)=O)CC2(CC2)CN1C(C1C=CCC1)=O CCC(CC(=O)NC(CC(C)C)C(=O)NCCCCN=[N+]=[N-])C(F)F Cc1nn(C)c(C)c1C(=O)NC1CC(CCNC(C2CC(C)CO2)=O)C1 c1(-c2cnc(CCC(=O)NCC(C)NC(c3cnco3)=O)o2)ccccc1Cl N1(C(CCCOC)=O)CCN(C(c2cc(OC)c(Cl)s2)=O)C(CCOC)C1 CC1OC2CCC1(C(=O)NCC(C1CCC1)NC(=O)Cc1ccco1)C2 C(=O)(C1CN(CC)c2ccccc21)N1CCCN(C(C(CC)(C)OC)=O)CC1 C(=O)(C1=NOC(C)(C)C1)NC1CN(C(c2c(SC)cccc2)=O)CC1C Cc1ccc(C(=O)NC2CCCC2C)c(N)c1C.C12(C=O)CC(C1)C(C)O2.N N1(C(C=CCCC)=O)CC(NC(c2cn(C)cn2)=O)CCC1C CCCC(C(=O)NC1CC2CC1N(C(c1c(F)cc(C)cc1F)=O)C2)S(N)(=O)=O c1(C(N2C(C)CCC(NC(=O)CCn3cccn3)C2)=O)ccnc2ccnn12 c1(C=O)cn(C)c(=O)n(C)c1=O.Cc1ccn(C(C)CC(=O)NC2CCC2)n1.N C(CC(F)F)(C(=O)Nc1cccc(C(N)=O)c1)N(C)C(C1C=CCCC1)=O N1(C(CC(C=C)(C)C)=O)CCC2(CCC2CNC(=O)Cn2cncn2)CC1 c1(C(C)=O)c(Cl)nc[nH]c1=NCC1CN(C(C2CC(C)(C)CO2)=O)CC1(C)C c1(SC(C)C(N2CC(F)CC2C=O)=O)ccccc1F.C12CC(C(=O)O)(C1)C2 C1(NC(c2c(OC)csc2)=O)COC2CN(C(=O)Cc3ccc(SC)cc3)CC12 c1(CC)ccc(COC(C2CCC(CC)CC2)=O)cc1C Cn1nnc(CNC(C2CCSCC2)=O)c1C(=O)N.C1CCN(C(C)(C)C)C1 CC1(C)CC(NC(C2CCn3nnnc3C2)=O)CCN(C(=O)C=CC=C(Cl)Cl)C1 CC1(NC(=O)C=CC(F)(F)F)CCN(C(C2CC2(Cl)Cl)=O)C1 c1(SCC(=O)NCC2(O)CN(C(C(C(C)O)C)=O)C2)ncnc2[nH]cnc12 Cc1ncc(Cl)cc1NC(C1CCCN(Cc2cnc(Cl)nc2)CC1)=O c1(CC)ccccc1C(=O)N(C1CN(C(=O)C(C)(F)CC2CCCC2)CC1O)C c1(OCC)ccc(CC(C)C(N2CC(F)(F)CC2CC(=O)OC)=O)cc1OC C1(CCNC(C(C2CC2)OCC)=O)COCCN1C(=O)CN(C)CC C#CC1COCCN1C(c1cc(-c2ccc(OC)cc2)on1)C(=O)NC(C)C N1(C(Cc2cncc(C)c2)=O)CCN(C(C2CC3(CCC3)C2)=O)CC12CC2 c1(C(N2C(C(=O)Nc3ccc(Cl)cc3C)CC(=C)C2)=O)ccc(F)cc1[N+](=O)[O-] C1(C(=O)NCC(C2CC2)OC)C=CCN1C(c1csc(C)c1)=O O=NN1CCCC1C(N1CCN(CCNC(C2CCS2(=O)=O)=O)CC1)=O C1(OC)CN(C(=O)Cc2ccccc2)CCC1NCc1ccnc(O)c1 N1(C(CCC(=C)C)=O)CC(CNC(=O)CCCc2ccsc2)OC2(CCC2)C1 N1(C(C(CO)OC)=O)CCN(C)C(C(=O)NCc2ccco2)C1 C(=O)(CS(=O)(=O)c1ccc(Cl)cc1)NCCNC(CCC1C(=O)NC(=O)N1)=O C(=O)(C(C)(C)CCCNC(c1oc(C)cc1C)=O)N1C(COC)CCCC1 Cc1cc(C(=O)N)c(O)nn1.C12(C(N3CC4CC4C3)=O)CC(C1)S(=O)(=O)C2 c1(C(N2CCC3CC23C(=O)NC)=O)ccc(C2CC2)cc1.C1(O)CC(O)C1 C1(NC(C(Cc2ccc(C)cc2)C)=O)CN(C(=O)C=Cc2ncc[nH]2)CCC1C CC1(CNC(C2(C)CCCCO2)=O)CCCN(C(C23CC(CF)(CO2)C3)=O)C1 N1(C(=O)NCc2cn3ccsc3n2)CCC2(CC1)CC(O)CCO2 N1(C(C2(CCOC)CC2)=O)CC(C2CCCCN(C(c3cc(C)nn3C)=O)C2)C1 CC1(C)CC(NC(c2cc3c[nH]nc3s2)=O)CN(C(C2(C#N)CCCC2)=O)C1 C1(NC(CCSCC)=O)CC2CC(NC(C3(C(F)F)CCCC3)=O)C2C1 c1(N2CCN(C(c3c(C#N)cn[nH]3)=O)CC2)cncc2ccccc12 Cc1nc(CN2CCC(CCC(=O)Nc3cccc(C(=O)O)c3)CC2)oc1C CN1CCc2[nH]nc(C(=O)NC3CCN(C(c4ccnn4C)=O)CC3CO)c2C1 C(=O)(C(O)C(C)CC)N(CC(N1CCOCC1CC)=O)CCC C=CC(C)(O)CC(=O)NC1CCCCC1CNC(=O)CS(C)(=O)=O c1(SCC)cc(Cl)ccc1C(N1CC(NC(=O)CC2CC2)C(C)C1)=O.O c1(C(=O)NC2C(C)CCN(C(=O)C(C)(C)NCCC#N)C2)n[nH]c2c1COCC2 C12(C(=O)OC3COCCN(C(=O)OC(C)(C)C)C3)OCCCC1C2(F)F c1(NC(=O)C=CCBr)cnc(F)cc1C(=O)Nc1ccc(O)cc1F c1(SC)cscc1C(=O)NC(C)CC.C(=O)(C(C)N(C)C)N.C(C)(C)C C1(C=O)C2CS(=O)(=O)CC12.C1(OC)(C)CCN(C(c2cncnc2C)=O)C1.N Cc1cn2c(n1)CC(C(=O)NCC(C)(O)C)C2.c1(CC=O)csc2nccn12.N CC1(C(=O)NCC2CC2c2ccccc2)CCCN1C(=O)COCC(F)F CC(CNC(=O)C#CC1(C)COC1)CC(=O)N=c1ccn(CCO)[nH]1 c1(C(=O)NC(CN(C(CC2CC(CC)C2)=O)C)C)ccc2nc(Cl)nn2c1 C1(c2nnnn2C2CCOCC2)(NC2CCN(CC)CC2C)COC(C)(C)OC1 C1(CCNC(CC2CC(=C)C2)=O)CCCN(C(=O)CCc2nnc(C)n2C)CC1 N1(C(=O)NCC(C(C)C)c2cccnc2)CC(=O)NCC1C N1CCC(C)(C=O)C1.c1ccc(C(N)=O)cc1.c1(C(=O)OCC)ccc[nH]1.C CC(C)CC(CC(=O)NCCN1CCCCC1C)NC(=O)CC1(N(C)C)CCC1 C1(C)(CC)C=C(C(=O)NCC(C)CNC(=O)Cc2ccc(OC)cn2)C1 N1(C(C(C(C)C)O)=O)CCC2CC(CNC(=O)CCC3CCC3)CCC2C1 C(=O)(C(F)(F)C(O)C1CC1)N1CCC(C)(CNC(C2CCC(C)(C)C2)=O)C1 c1(OCC)ccc2cc(C(=O)NCC3CN(C(=O)C(C)OC)CCN3)[nH]c2c1 N1(C(C(=O)NCc2cn(-c3ccccc3)nn2)=O)CC2(C(=O)O)CC1CO2 N(C(=NCCO)NC1CCS(=O)(=O)C1)CC(C)(C)C(O)C1CCC1 c1(C(=O)NC(CCC)C(=O)NCCc2cnn(C)c2)cnc2n1CCC2 C1(NC(c2nnc(C(C)C)s2)=O)C2CC1N(C(c1nn(C)cc1N)=O)C2 c1(CC)ccc(C(=O)NC(CC)C(C)C)c(F)c1.c1(C=O)cncn(C)c1=O.N C(c1c(C)nn(C)c1Cl)=CC(N1CC(F)C1)=O.c1(OC)ncccc1C(=O)N c1(-n2ncc(NC(=O)NCc3scc(CC)n3)c2)cccc(F)c1 N1(C(C23CC(C)(OCC2)C3)=O)CCC(F)(F)C(CNC(c2csnn2)=O)C1 CC(C)C(CCN(C(=O)CN1CCCC1CO)C)NC(c1cn(CCF)nn1)=O S(=O)(=O)(c1cc(C(=O)NCCC)co1)N(CC)C.C(=O)CC(F)(F)F Cc1cc(F)c2ncc(C(=O)NCCN(C)C(c3ccccc3F)=O)cc2c1 c1(C(C)NC(=O)CC2(C)CC2(Cl)Cl)cccc(OC(F)(F)Cl)c1 c1(OC)cc(C(=O)NCC2CC2)ccc1O.c1(C=O)cnn(C(C)(C)C)c1 C(=O)(C(F)CC(C)(C)NC(c1ccc(C)cc1O)=O)NC(C1CCOC1)C#C C1(NC(c2c(C)nc(CNC(=O)C(C)(C)CN(C)C)o2)=O)CCCCCC1 Cc1ccc(OCCC(=O)NC2CCN(C(C3CCNC3=O)=O)C2C(C)C)cc1 C1(C2CCOCC2)(CNC(C(CC=C)CC)=O)CCN(C(=O)C=CC(C)(C)C)C1 c1(C=O)cc(O)nn1C.C1(COC)(C)CN(C(=O)Cc2cnn(C)c2)C1.N c1(N2CC3CC(NC(=O)CC(F)(F)F)C3C2)ncc2ccccc2n1 C1(C(=O)NCCCC(C)(C)O)CCN(C(C2CC23CCCCC3)=O)CCO1 CCC(F)(F)CC(=O)N1CCOC(CC(=O)Nc2cn(C)nc2C)C1 c1(C(N=c2c(C(C)=O)c[nH]cc2)=O)cc(F)cc2nc(S)[nH]c12 C(=O)(C1=CCC(C)(C)CC1)N1CC2C(C(N3C(C)CC(CS)C3C)=O)C2C1 N1(C(CN(C(=O)C(c2ccccc2)C)CCOC)=O)CCCC(C(=O)OC)C1 c1(C(=O)NCC#CCNC(C2C(C)(C)C2)=O)ncc(C(F)(F)F)cc1N CC(C(C)(C)C(=O)N(C)C1CC1)NC(=O)CCn1ccnn1 N1(C(CC2OCCN(Cc3cccc(C=C)c3)C2)=O)CCCC2CCCCC12 Cc1ccc2nc(C(N3CCCC3CNC(=O)CC3CC4CC4C3)=O)ccc2c1 c1(C(=O)NC2CC(NC(CC(C(=O)OC)C)=O)C2)ccc2nc(O)[nH]c2n1 c1(C(C=O)C2CC2)ccc(C)cc1.c1(C=O)nccn1C(C)C.C(C)C.C C(CC(C(=O)NCC(O)CF)NC(=O)C(C)N(C)C)OC c1(OC(C)C)ccccc1NC(=O)NC1CNCC1c1cnn(C)c1 c1(CC)ncccc1C(=O)N(CCCCC(=O)NCC1CCC(C)C1)C c1cc(C=CC=O)ccc1F.c1(C(N(CC)C2CC2)=O)nccc(C)c1N.CO Cc1cc(C(=O)NC(C)CCC)ccc1[N+](=O)[O-].C1(C(=O)N)C(C)(C)OC1(C)C CCCCCC(C(=O)N1CC2(CCC2NC(c2cncn2C)=O)C1)C(C)C C12(c3ccn(C)n3)CCC(C1)C2C(=O)NCC1COC(C)(C)C1O C1(C=O)CCCCCS1(=O)=O.CC(CNC(=O)CCNS(C)(=O)=O)C.N C1(C(N2CCC(CN(C(c3[nH]c(CC)c(Cl)n3)=O)C)C2)=O)COCCC1(F)F C#Cc1cccc(C(=O)NC2(C(=O)Nc3cc(O)ccc3C)CCCC2C)c1C Cn1cncc1CC(=O)NC1CC(NC(C23CC(C)(C2)C3)=O)C1 N1(C(CCN(C(C)=O)C)=O)CCC(NC(=O)COCc2cccc(C)c2)C1C c1(CC(=O)NC2CCCC2C(=O)NCC2COC2)ccc([N+](=O)[O-])cc1 c1(CC(=O)NCC(CN(C(c2c(C)cccn2)=O)C)C)c[nH]c2ccc(Cl)cc12 N1(C(c2ccnc(F)c2)=O)CC2CC1CN2Cc1cc(C(F)(F)F)cc(Br)c1 C(c1cc(F)c(F)c(F)c1)=CC(=O)NCC1CCN(C(CC(C)O)=O)C1 C#CC1(NC(=O)CC(C)(C)CNC(=O)CC2CCC(C)O2)CCCOC1 Cc1cc(N)cc(C(N2CCN(C(=O)C=CBr)C3CC23)=O)c1F c1(NCC(CC(C)C)NC(c2n[nH]c(C)c2O)=O)c(Br)cccc1[N+](=O)[O-] N1(C(C(C)C2CCCC2)=O)CC(CNC(=O)C(F)=CCCF)C(C(F)(F)F)C1 C(CC1=CCN(C(c2occ3c2CCCC3)=O)CC1)NC(=O)C1=COCCO1 C1(NC(C2C(C)(C)C2(C)C)=O)CCCN(C(c2ncncc2Cl)=O)CCC1 C1(NC(=O)C(O)C(F)F)CC2(C1)CC(NC(C1(C3CCCCO3)CC1)=O)C2 N1(C(C(C)(C)N(C)C)=O)CCCN(C(=O)CC2CC(C)(C)OC2=O)CCC1 c1(C(N2CC(C3OCCN(C(CS(CC)=O)=O)C3)C2)=O)c(F)ccc(F)c1Cl C(=O)(C#CC1(C)CCCO1)N(C1CCN(C(=O)C=Cc2cocn2)C1)C CC1(CNC(c2cc(O)nc(Cl)c2)=O)CCN(C(C2CC2C2CC2)=O)CC1 C1(C(N2CC(O)(CC)C2)=O)CCCCCN1C(c1cc(C)nnc1O)=O c1(C(=O)OCC)cccc(C(=O)NCC2C=CCN2C(=O)COC)c1 Cc1ccc(C)c(OCC(=O)NCC(C)N(C)CCF)c1 C1(O)(C(C)NC(=O)CO)CCN(C(=O)CC(C)(C)C#N)CC1.C1CCCCO1 c1(C(N(C2CCC2)C)=O)cc(Cl)cc([N+](=O)[O-])c1.c1(C2(C=O)CC2)ccno1 c1(CNC2C(C)CN(C(c3cc4n(n3)CCC4)=O)CC2)sc2ccccc2c1Cl Cc1nn(C)cc1C(=O)NC(C)C(C(C)C)NC(c1cn(C)c(C)n1)=O N1(C(C2N(C)CC(F)C2)=O)CCCC(C(=O)NCCNC(N)=O)CC1 N1(C(C)=O)CC(NC(c2ccc(NC(C3CCCOC3)=O)cc2)=O)CC1(C)C C1(NC(C(C2CCC2)OCC)=O)C2CC(O)C1N(C(c1cn(C)nc1)=O)C2 N1(C(C2CC(C)(C)N(C(=O)Cc3ccco3)C2)=O)CC2CC(O)CC1C2 c1(OC)ccccc1.CCC(=O)N(C)CCOCCNC(=O)CO.C=O C1(C(N(CC)Cc2ccc(C)cc2)=O)CC(F)CN(c2nc(C)cc(C)n2)C1 CC1CN(C(c2csc(Br)n2)=O)CCS1 c1(C(N(C2CCN(C(c3ccnnc3S)=O)CC2)CC)=O)ncccc1N c1(C(=O)OC)sc(C(=O)NC2CCC2NC(=O)C(O)C2CC2)cc1N C1(C(=O)NC(C2CCCN2C(C2C3CN(C)CC23)=O)C)CCC=CCCC1 C(=O)(CCCC(F)F)N(C)CC1N(C(C2C(=C)C2C(=O)OC)=O)CCCC1 N1(C(c2ncc(C)nc2)=O)CCC2(COCC(CNC(=O)Cc3cc[nH]n3)O2)C1 c1(N2CCC(NC(c3cc(CC)c(C)s3)=O)C(C)C2)nc(Cl)nc2c1cnn2C C1(C(N2CC(C)OCC2)=O)CC(F)(F)CN1C(C1C2CCCC(=O)C12)=O Cc1ccc([N+](=O)[O-])c(N2CCCC(NC(c3cc(C)n(C)c3)=O)CC2)c1 C(C(CC(C)C)NC(=O)Cn1nc(C)cc1C)NC(C(C)OCC)=O c1(C(N2CCC(N(C(COC(CC)C)=O)CC)C2)=O)ccc(C)c(CO)c1 C(=O)(CCCCCS(N)(=O)=O)NC(CNC(c1c(C)cc(C)nc1)=O)(C)C N1(C(C2C(C)C2)=O)CCC(C2CCN(C(=O)CSc3ccc(Cl)cc3)CC2)C1 C1(NC(CC(CC)C)=O)CN(C(C2(OC)CCSC2)=O)CCC12CCC2 CCCCC(C(=O)NC1CC1CC(C)(C)C)NC(c1cc(OC)nn1C)=O C1(C(N2CCN(CCOC)CC2)=O)N(C(=O)C(C2CC2)OC)CCC1(C)C C12(C(=O)NCC(CC)C#N)CCC(F)(F)CC1CN(C(=O)OC(C)(C)C)C2 c1(C(=O)NCCCC)cc(C(F)(F)F)cc(N)c1C.C(=O)(C(C)C1CCCC1)N N1(C(c2c(COC)cc[nH]2)=O)CC(C)CN(C(C2(F)CCOCC2)=O)CC1C C1(CCNC(CC(C)=C(C)C)=O)CN(C(=O)Cc2c(C)ncnc2C)CC(C)O1 CC1(CCC(=O)Nc2csc(C(c3ccc(F)cc3)=O)n2)CCC(=O)N1 c1(OC)ccccc1C(=O)C(=O)NC(C)C1CC1.C1(C(=O)N)CCC(C)O1 C1(NC(=O)CCCc2ncco2)CC(CO)N(C(c2cc(Cl)ns2)=O)C1 c1(OC)ccc(CC(=O)N(c2ccccc2Cl)C2CC3CC2CN3)c(C#N)c1 CC1CCC(C(N)=O)CN1C(=O)C(C)(C)CN(C)C(C1CCSC1)=O c1(C(N(CC(C)NC(C2COCC2C(F)F)=O)C)=O)cccnc1-n1ccnc1 N1(c2nc(C)cc(OC)n2)CCC2CCN(C(=O)C(C)NC(N)=O)CC2C1 c1(C(=O)NCC(CNC(c2cc(O)nn2C)=O)OC)ncc(C#N)cc1Cl C(C(C)C)(C(O)C(=O)NC1(C(=O)NCC2CC2C2CC2)CCSC1)OC N1(CCCNC(=NCC)NCCN2CCNC2=O)CCCC(C)(C)C1 c1(C(C(=O)NC2C(NC(c3c(C)n(C)nc3)=O)C2)O)ccc(Cl)cc1F C(C(C)CN=c1[nH]c(=NCC(C)(CC)OC)[nH]c2c1SCC2)OCC c1(C(=O)OCCCCOC)c(C#N)ncn1C C(CS(=O)(=O)CC(=O)NC(C1(O)CN(C(=O)C(C)CC2CC2)C1)C)OC CC1=CCC(C(C)NC(c2cncc(Br)c2)C)CC1 Cn1ccnc1C(N1CCCC1C1(O)CN(C(c2ccnn2C2CCC2)=O)C1)=O C(C(CC1CC1)C(=O)NCC=CCl)NC(=O)CCC1OCCO1 CC(CC1=CCCCC1)NC(=O)C(O)CNC(=O)C(F)=CC1CC1 CCC(C)C(O)C(=O)N1CCC(CC(C)NC(=O)Cc2c(C)cccc2F)CC1 C1(CCC)CN(C(=O)CC2NC(=O)NC2=O)CCO1.C1(CC=O)(COC)CC1 Cc1cc(O)ccc1C(=O)NC1CC(CC(=O)NCc2ccc(F)c(Br)c2)C1 N1(C(C=CCOCCOC)=O)C(C=O)CC2CC12.C1CC(O)C1.CC.N c1(OCCOC)cccc(CNC(C)CC(N)=O)c1 Cc1cc(C(=O)NCC(C2CCOC2)NC(=O)CC(C)C)c(C)n1NC(N)=O Cc1ccc(Cl)c2[nH]c(C(=O)NC)cc12.C1CC2(CO1)CN(C(=O)C(C)(C)F)C2 C1(C(=O)NC(CN(C(c2ccc(CC)cn2)=O)CC)C)COCCC1(F)F c1(C(=O)NCCCCNC(CC2CC(OCC)C2)=O)c(F)cncc1Br Cc1cccc2ncnc(N3CCCC(NC(c4cccc5c4CCC5)=O)C3)c12 C1(NC(C(C(C)O)(C)C)=O)CC2(CCN(C(c3cc(C(F)F)nn3C)=O)CC2)C1 C1(NC(Cc2cn(C)nc2)=O)CN(C(c2nnc(O)cc2O)=O)CC1N=[N+]=[N-] C1(NC(C2CCCC2C2CC2)=O)CCCC12CCN(C(C13CC4CC1C3C4)=O)CC2 N1(C(CC2CC(C)C2)=O)CCN(C(=O)CNC(=O)C(C)C(F)F)CC1 c1(NCC2C(C)CN(C(=O)CCS(N)(=O)=O)CC2)cc(C#N)c(F)cc1[N+](=O)[O-] N1(C(C(C)=CC)=O)CCC(C2(NC(C3CCCC(C4CC4)O3)=O)CC2)CC1 Cc1ccnc(O)c1C(N1CCC(C)C(NC(=O)C(c2ccnn2C)C)C1)=O Cc1c(C(=O)NC2CCC2)cnn1C1CC1.c1(C=O)cnn(C(C)(C)C)c1C C(=O)(C1CCc2c[nH]nc21)N(CC(C)N(C(CCOc1cccc(C)c1)=O)C)C n1(Cc2cn(C3CN(C(C4(Cn5ccnc5)CCC4)=O)C3)nn2)cccnc1=O C#CC1(O)CCCN(C(=O)CC23CCC2CN(C(=O)COC(C)C)C3)C1 C(=O)(CCCCCN(C(=O)C#CC(C)(C)C)C)NC1CCCC(CC)C1 N1(C(C2CCN(C)C2)=O)CCC(O)C(NC(C2CCN(C3CCCCC3)C2)=O)C1 N1(C(CC(=C=C)C)=O)CC2COCC(C1)C2NC(C1Cc2ccc(C)cc2S1)=O c1ccc(F)cc1O.C1(NC(c2nc(CCC)sc2)=O)CC(C)N(C(=O)CO)C1 Cc1ccc(CC(C)C(=O)NCC(O)CNC(=O)CCc2cnccn2)cc1 c1(OC)n[nH]c(C(=O)NCC2CC2)c1Cl.c1(CC=O)csc(NC=O)n1.C N#Cc1c[nH]c(C(N2CCCCC2C(=O)NC2CC23CC(O)C3)=O)c1 C1(NC(C(C)(C)CO)=O)CCC2CCN(C(C3CCCC4CCCCC34)=O)C1C2 C1(NC(Cn2c(C)cc(C)n2)=O)CC2CCC1(C)C2.C(=O)(CCc1cnoc1)N Cc1nn(C)c(Cl)c1C(=O)NCC1CCCC1.c1(C=O)ccc(C(N)=O)s1 c1(C(=O)NC23COCC(N)(C2)C3)cc(Br)n2ccccc12 c1(NC(C)=O)cnccc1C(N1CCCC(CNC(=O)CC#N)C1)=O Cc1nnc2n1CC(C(N1CCC(NC(=O)CN3CCCCC3C)C1)=O)C2 C(=O)C1c2ccccc2OCC1(C)C.C(CCC(=O)NC1CC1C)SC(C)(C)C.N CC(CC(=O)N1CCCC1C1CCN(C(C2(C)CCN(C)C2)=O)CC1)C(F)(F)F c1(CN(CC)Cc2ccncc2Br)ccc(F)c(OC(F)F)c1 C1(NC(C2CCC(CN(C)C)O2)=O)CCCCC1NC(c1c[nH]nc1Br)=O C1(C(=O)NC(CC(=O)NC)C2CC2)CCCN(C(c2cnc(Cl)s2)=O)CC1 C1(NC(=O)CCn2ccnn2)C2CC3CN(C(C4CC4c4ccco4)=O)C1C3C2 C(=O)(C(C(F)(F)F)C(F)(F)F)NC(C1CCCN(C(=O)CN2CCCC2)C1)C c1(C(N2CCC(C)(NC(c3n(C)c(Cl)c(Cl)c3)=O)C2)=O)cccc2cccnc12 c1(C(=O)N)ccc(C)c(C)c1.N1(C(=O)NC(C(=O)OCC)C)CCOCC1 c1(C(=O)NC2(C)CN(C(C(COC)C)=O)C2)coc2ccccc12 C1(C(=O)NC)C2CN(C(=O)C(C3CN(C(c4nccs4)=O)C3)OC)CC12 C1(C(=O)NC2C(CC(=O)NC(CC)C(C)C)C(O)C2)Cc2ccccc2C1 C1(C2C(n3cc(-c4c(C)ocn4)nn3)CCO2)CCCC(CC(=O)N(C)C)O1 C(=O)(C1CCCn2nccc21)NC1(C)CN(C(C23CCCC(C2)C(=O)N3)=O)C1 Cc1cnc(C(=O)NC2CCN(C(C3(Cl)CC34CCC4)=O)C2)c(C)c1 C1(NC(Cc2nc(C)sc2C)=O)CC2CC1CN(C(=O)C(C)n1ccnc1)C2 c1(C(CC)C)ccc(C#N)c(NC2(CO)CCN(C(C3CCC3OC)=O)CC2)n1 N1(C(C=CCCC=C(C)C)=O)CCCC(C2CN(C(c3cc(C)sn3)=O)C2)C1 c1(C(=O)NC(COC)C(=O)N(C)C(C)C2CC2)cc(=O)cc[nH]1 CCCS(=O)(=O)C(C)C(=O)NC1CCCC(NC(c2c(F)ccc(F)c2N)=O)C1 C(CN=c1ccnc(-c2ccccc2)[nH]1)=CCNC(c1c2c([nH]n1)C(C)CC2)=O C12(CNC(c3cncc(N)n3)=O)CCCC1CN(C(c1ccc(Cl)s1)=O)C2 C=CCCC(CC(C)C)C(=O)NCCCC1CCCN1C(C1CC(CC)=NO1)=O c1(C(N(CCCNC(=O)CC2CCCC2O)C(C)C)=O)cc2ccccc2o1 CCCC(C(=O)NC1CCCC1NC(C1CC(n2cnnc2)C1)=O)NC(C)=O N#CCCCCC(=O)N1CCCC(F)(C(N2CCCCC2CO)=O)C1 N1(C(c2c(OCC=C)cccc2)=O)CC2CCC1CN2C(=O)CC(C)OC N1(C(c2nccc(-n3c(C)ncc3)n2)=O)CC(NC(=O)C2=CCOC2)C2(CC2)C1 CCCC(CNC(C1(CNC(c2ccnn2C)=O)CCC1)=O)OCC c1(C(=O)NC23CC(NC(c4cc5cnn(C)c5s4)=O)(C2)C3)c[nH]c2cccnc12 CC1Oc2ccc(C(=O)NCCC(C)(C)Nc3nccc(CO)n3)cc2C1C C1(C(N2CC(CCCNC(C(F)=CCC)=O)OCC2)=O)CC12CC(F)(F)C2 CCCC(C#N)C(=O)NC1C2CC3C1C3C2C(=O)NCCc1ccc(F)cc1 c1(C(N(CC(C)NC(c2cncc(C#C)c2)=O)C)=O)c(C)nc(C2CC2)nc1C C(C(C(=O)NC(C)C)N(C)Cc1ccc(Cl)cc1)(C1CCCC1)OCC C=CC1(NC(C2(NC(=O)C(C(C)CC)OC)CC(O)C2)=O)CCOCC1 N1(C(C(C)N(C(C2CCC(O)CN2C)=O)C2CC2)=O)CC2CC=CC1C2 C=CC(O)C(=O)NCc1cc(CNC(=O)CCC2(C=O)CCCC2)c[nH]1 c1(OC)nccc2c(C(=O)NCC3C(C)CCCN3C(=O)CCF)c[nH]c12 c1(NC(C(CNC(c2ccsc2)=O)OC)=O)ccc2nccn2c1 C(=O)(C(C)(C)CC(=O)N1CCCC1C(=O)NC(c1snnc1C)C)OC c1(OC2(C(=O)NC(CC)CNC(C34CCC3C4)=O)CC2)ccc(C)cc1 C1(CC(=O)NC(c2cncn2C)C)CCCC(NC(=O)Cc2cn[nH]c2)C1 n1(Cc2cn(C(C)CN3CCNC3=O)nn2)cnc2ccccc12 CC1(C)CCC(C(N2CCC2)=O)CN1C(C1CCCO1)=O CC1CCN(C(c2cc[n+]([O-])cc2)=O)C(C)C1NC(c1c[nH]c2ncccc12)=O c1(C(N(CCNC(CCCCC=C)=O)CCOC)=O)cc(F)c(F)c(N)c1Cl N12CCC(CC1)NC(=O)Cn1cc(nn1)C2.C1(C(=O)NCC)CCCC1.C CC1CN(C(C2CNC(=O)CC2(C)C)=O)CC(C)CN1C(=O)CC.[SH](C)(=O)=O.N CCC(CN(C)C)CC(=O)N1CCC(NC(=O)Cc2cc(C)ccc2OC)C1 C(=O)(C(CC)(CC)CC(=O)OC)N(CCNC(C1C(C#C)C1(C)C)=O)CC c1(C(N2CCCC(O)(CN(C(COCCC#C)=O)C)C2)=O)cc[nH]c2nccc1-2 C1(NC(=O)CCC2CCC(O)CC2)CCCCN(C(=O)C)C1.C(=O)(C(F)(F)F)N c1(C(=O)NC(C(C)C)(C)CNC(=O)C(C)c2ccon2)cc2cc(F)ccc2o1 Cc1cc(OCC(C)NC(=O)C(=O)Nc2ccc(-c3cccs3)cc2)cc(C)c1 C1(CNC(CC(C)SC)=O)CCN(C(=O)Cn2nnc(=N)[nH]2)C1(C)C C=CCCCCC(=O)N(C(C)(C(=O)N(C)CC1COCCO1)C1CC1)C C(=O)(C(F)(F)C(O)C(C)C)N1C2(C(=O)NCc3c(C)scn3)CC(C1)C2 c1(NCc2ccc(C)c(Cl)c2)ccc(S(=O)(=O)NCC(C)(C)CCCO)c(Br)c1 N1(C(C2CC2F)=O)CCCN(C(=O)C(O)Cc2ccncc2Br)CC1 C12(CNC(CC(C)O)=O)CC(C1)C(NC(=O)CCN1C(=O)CCC1=O)CO2 C1(CC(=O)NC(CC)C(=O)NCC=CC2CC2)CCCC(=O)N1 O=C(C1CCCn2c(O)nnc21)N1CC2(CCOCC2)CC1CO C(C)(C)(CC(=O)NCCc1cc(C)ns1)N(C(C(C)(C1CC1)OC)=O)C C1(CC#C)(C(=O)N(CCNC(=O)C(C)(C)O)C)CCCO1.c1ccccc1 C=Cc1ccc(C(=O)NC2CC(F)CN(C(c3cc(Cl)nnc3O)=O)C2)cc1 C#CC(C(C)(C)C)NC(=O)C(CC1CCC1)NC(=O)CCC1CC1(C)C C1(N(C(=O)CC2(C)CC2)C)CC2CCC(C1)N2C(c1cc(N)cc(O)c1)=O CC1(C2CCCN(C(N3CCCC(n4ccc(CN)n4)C3)=O)C2)NC(=O)NC1=O CN1CC(NC(=O)C(C2(C)CC2)NC(=O)CCCC2CCCO2)CC1CO C1(NC(C(c2ccco2)NC(C(C)n2ccnc2)=O)=O)CCn2cnnc2C1 CC1(C)NC(=O)CC1C(=O)NC1CN(C(=O)C=CCO)CC1C(F)F c1(N2CCC(NC(Cc3c(C)con3)=O)C2)ncnc2sccc12 C1(C(=O)NC(C(=O)NC2CN(C(C)=O)C2)c2ccco2)CCCCN1C C(=O)(CCC(=O)C(C)(C)C)NC(C(=O)NCC(CCCC)O)CO CCC(C)(C)C(C)CC(=O)N1CCC(O)(CNC(=O)COC(C)(C)C)C1 C(=O)(CCCC(F)(F)F)NCC(CC(=O)NCC1(S(C)=O)CC1)O C1(C(N2CCC(N(C)CC)CC2)=O)CCCN(C(C2(OC)CC(C)C2)=O)CC1 N(C1CCc2cccnc21)C(C(CCNC(C(C)(C)CC#N)=O)O)=O C#CCCCCC(=O)NCC1CN(C(=O)C2=CCCCO2)CCC1C(F)(F)F c1(OC)cc([N+](=O)[O-])c(C)cc1NC(C1CN(Cc2cc3ccccc3[nH]2)C1)=O c1(C(C)C)cc(C(F)(F)F)ccc1NC(N1CC(n2ccnn2)C(N)C1)=O C1(CNC(CN(C2CCSC2)C)=O)CCN(C(c2csc(Br)n2)=O)C1 CC(C)CC(O)C(C)C(=O)NCC1(CC(=O)O)CCCC1 C1(CNC(CCC#C)=O)CN(C)CCN1C(c1cc(F)cc(F)c1)=O c1(CC)cc(=NCC2(O)CCCN(C(C3(C)CC3(F)Cl)=O)C2)[nH]cn1 c1(C(=O)OC)cnc(N(C)C)cc1C.c1(CC(N2CCC2)=O)cc(F)cc(Cl)c1 Cc1ccc([N+](=O)[O-])cc1C(N1CC(C)(C(=O)Nc2ccc(Br)cc2C)C1)=O C1(CC=C)(NC(c2ccoc2)=O)CCN(C(C2CC(CC)C2)=O)C1 N1(C(c2nccc(C)c2)=O)C2CCCC1CN(C(=O)Cn1nc(C)ccc1=O)C2 Cc1cnc(C(=O)NC(CO)CCCCNC(C2(C#N)CCCC2)=O)c(F)c1 C=C(CNC(=O)C(C)Sc1nncn1C)CCNC(c1ccc(CC)[nH]1)=O CC(C)C(O)C(F)(F)C(=O)N1CCN(C(c2cccc(F)c2)=O)C(C2CC2)C1 Cc1cc(O)ccc1CC(N1CCC(CCNC(=O)Cn2cccn2)CC1C)=O O=C(C1=CCN(C(C2CC3CC3C2)=O)C1)NC1CCCCC1O Cc1cc(F)c(CC(=O)N(C(C)CCNC(c2nn(C)c(N)c2C)=O)C)cc1F c1(C(N2CC(CCC(N)=O)OCC2)=O)ccc(S(=O)(=O)N2CCCC2)cc1 C(=O)(C(C#N)CC)NCCC(=C)CNC(=O)C(C)Oc1ccc(Cl)cc1 c1(NCCC(N2CCN(C(C3(NC(C)=O)CC3)=O)CC2)=O)oc(C)nc1C#N C(=O)(CCCC(C)C)NCc1c(OC)cccn1.C1(C(=O)N)CCC1.C1CC1 c1(C(=O)NC2CC(NC(c3cnc(C(C)=O)s3)=O)C2)cc2cc(C)ccc2o1 Cc1cc(C(N2CCN(C(c3cc(C(C)(C)C)nn3C)=O)C3CC23)=O)ccc1O C1(C(=O)NC2CCCC(C(N(C)Cc3n(CC)ncc3)=O)C2)CN2CCC1CC2 c1(C(=O)NC2(C)CCN(C(C3CC(O)(C#N)C3)=O)C2)ccc(F)c(CO)c1 C12(C=O)C(=O)C3CC1C2C3.C1CCN(C(=O)Cc2cc(C)nn2C)C1.CO.C CC(C)C(CO)CCNC(=O)NC1CC2(CC2)C12CC2 c1(CCN(C(C(=O)NC(C)C)C(C)C2CCCOC2)C)ccc(C#N)cc1 Cc1ccnc(C)c1CNC(C1CCCCC1(C)NC(c1ccc(CO)s1)=O)=O N1(C(CN(C(COC)=O)C)=O)CC(Nc2nccc(C)n2)C(C)(C)C1 C(=O)(C(C)=Cn1ccnn1)N1CCC2(C1)CC2.C(C)(C(=O)N)OCCOCC C=CCC(C(=O)N1CCOC(CCNC(=O)C=C=C(C)C)C1)C(C)C c1(OC)c(C(N2CC(C3CN(C(=O)C4CC4)C3)C2)=O)ccc(Cl)c1C C1(CC)CN(C(=O)CC(C)C)CCS1(=O)=O.C(C)(C=O)OCC#C.C(C)=O c1(CC(=O)NC(C)CN(C)C(C2CCCN2C)=O)csc2c(Cl)cccc12 c1(C(=O)NCC(CNC(=O)CC2CCCS(=O)(=O)C2)O)cc2nc[nH]c2cn1 C1(CCC)CN(C(c2cnc(CC(C)(C)C)o2)=O)CCN1C(=O)Cc1ccon1 c1(C(=O)NC(C(=O)OC)CC2CCOC2)cnn(-c2ccccc2F)c1C C1(NC(C(N2CCNC2=O)C)=O)CC2CC1CN(C(c1nc(CO)cs1)=O)C2 C(C1=NOC2CCCC12)NC(c1c(CNC(c2c(C#C)c[nH]n2)=O)c[nH]n1)=O c1(C2CCN(CC(c3cccc(Cl)c3)O)C2)cccc(Cl)c1 C1(C(=O)NCC(C)(C)NC(c2occ(OC)c(=O)c2)=O)CCc2nnnn2CC1 N1(C(CSC(C)C)=O)CC2(CCCCN(C(c3cc4ccccc4o3)=O)C2)C1 C1(C(=O)NCCC(C)(C)OC)CN(C)CCN1C(=O)C1=CC(C)(C)C1 c1(OC)cnc(C(=O)NCCC2CC2)nc1.C1(C(O)CO)(NC=O)CC1 c1(C2(N(C)CCn3ccnc3-c3cn(CC(=O)O)nn3)CC2)ccc(F)cn1 c1(C(=O)NC2CC(C(=O)NCC3=C(C)CCC3)OCC2)cnc(C)cc1C C1(NC(C(CCCCC)F)=O)CN(C(C2CC(OC)C2)=O)C2(CCCCCC2)C1 c1(C(N2CCC(NC(CSCCC)=O)C(C)C2)=O)c2ccccc2nn1C C=CCC(CC(C)C)C(=O)NC1CCCC1CC(=O)NCC1(O)CCOCC1 C(=O)(C1=CCCOC1)N(C1CCN(C(C2OCCCO2)=O)CC1)C CC1(C)CC(C(=O)NCCOCC)=NO1.c1(C(=O)N)cccc(S(C)=O)c1 C1(NC(CCSC)=O)CC2(C1)CC(NC(=O)C(C(C)C)n1ccnc1)C2 N1(C(c2ccc(O)cc2)C(=O)NCc2cccs2)CCC2CCC(O)C1C2 c1(C(N2CC(CN(C(C(CC=C)C)=O)C)C3(C2)CC3)=O)cc2ccccc2nn1 Cc1c(-c2cn(C(C)C(N3CCN(C(C)C)CC3)=O)nn2)cccc1F C(N=c1nn[nH]n1-c1ccccc1)C1C(NC(C2CCS(=O)(=O)CC2)=O)CCC1 N1(C(C(C)CNC(c2ccccc2)=O)=O)CC(CO)C(O)C1 C(=O)(C1=C(C#N)CCC1)N1CCCC(CNC(C2C(C)C2)=O)(CO)C1 C(=O)(C1=NOC(C2(O)COC2)C1)NC1CC(N(C)C(c2cc(O)nn2C)=O)C1 N1(C(CCn2cc(-c3cnc(OC)c(C)c3)nn2)=O)CCC(O)CC1(C)C c1(OC)cc(C)c(C(N2CCC(C(C)NC(=O)CC(O)C(C)C)CC2)=O)c(F)c1 C=C(Cl)CC(C(=O)NCC=CCl)NC(c1cc(C)nc(O)c1)=O C(=O)(C(F)CC(C)(C)NC(=O)CCC)NCC1C(CCC)C1.C(C)=O.N c1(C(=O)NC2C(NC(C=NOC)=O)C2)cnc2c(cnn2C)c1O C1(F)(CNC(C2(CC=C)CC2)=O)CC2CCC(C1)N2C(=O)C.C(C)C c1(CN2C(C(=O)NC3C(C)COCC3)CSCC2)c(F)cc(Br)cc1Br Cc1c(C(N2CC(O)CC2CNC(=O)CO)=O)[nH]c2ccccc12.C1CCOC1 C1(CCC)CC2CCC(C1)N2C(=O)Cc1ccc(F)cc1.C=C1CC1C=O.N CC1CN(C(C2CC(CF)C2)=O)CCC1CNC(=O)CCCNC(N)=O Cn1ncc(C(=O)NC(CNC(c2ccc(C#N)s2)=O)CO)cc1=O CC1CC(CNC(c2cnc(Cl)s2)=O)CN(C(C2COCC2(C)C)=O)C1 N1(C(C(C)NC=O)=O)CCC(C(=O)NCC2(n3cccn3)CC2)C(C)C1 C1(NC(c2ncn(CC)n2)=O)CCCCC1C.C(=O)C(F)(F)c1csc(C)c1 Cc1[nH]nc2ccc(C(=O)NC3CC4CCC(C3)N4C(c3cc(Cl)c[nH]3)=O)cc12 c1(C(N(c2cnn(CC(=O)N(C)C)c2)CC)=O)ccc2[nH]ccc2c1 C(=O)(C(O)CC(F)(F)F)N(CCNC(C=CCN(CC)CC)=O)C c1(OCC(=O)NC2CCC2NC(c2ccncn2)=O)ccc2ccc(=O)oc2c1 c1c(F)c(F)cc(F)c1F.Cc1ccccc1C(=O)NC1(C)CN(C(=O)C)C1.O C1(CC(=O)NCC(CC)(C)NC(=O)C(C)Cc2cccnc2)CN2CCC1CC2 Cc1c(C(=O)NCC2CCCN(C(=O)CC(F)(F)C(F)F)C2)nn2c1CCCC2 N1(C(C2CC(SC)C2)=O)CC2=C(C1)CN(C(C1(C3CCCO3)CC1)=O)C2 N1(C(C2(C)CC3C=CC2C3)=O)CCN(C(c2cccc(C3CC3)n2)=O)CC12CC2 CCCC(=O)NNC(=O)C(=O)Nc1c(I)cnn1C1CCCC1 C(=O)(C1=COc2ccccc2O1)NC(CNC(C=CC1(C)CCOCC1)=O)(C)C C1(NC(=O)CC2CCC2)CCN(C(C2CCS(=O)(=O)N2)=O)CCC1(F)F c1(C(=O)NCCC(C)N(C(=O)Cc2cnccc2Cl)C)nn(C)cc1Cl CC1CCN(C(C2(C(c3ccc(O)cc3)=O)CC2)=O)CCN1C(=O)Cn1nccn1 CCC(CC)(CO)C(=O)NCC(CNC(C1CCC1C(F)F)=O)OC N1(C(=O)COCC2CCC2)CCC2CC2(C(=O)NCC2=CCCOC2)CC1 C1(C)(C(=O)NC(C)CC2CCC2)CC(O)CN1C(=O)CC1CCCSC1 N1(C(C=CCC)=O)CC(NC(c2ccccc2COCCO)=O)C2CCCC2C1 N1(C(c2ncc(OC)nc2)=O)CCCC2C1CCCN2C(=O)Cn1[nH]cnc1=N Cc1cnc2c(C(=O)NC34CCCC(CN(C(C5CCOC5)=O)C3)C4)cnn2c1 C1(CNC(c2ccc(CNC(=O)CCc3cnoc3)o2)=O)CCC2(CC2)C1 C(=O)(CCC(C)(C)NC(N)=O)N1CC(C(N(C2CC2CO)C)=O)C1 S(=O)(=O)(c1ccccc1CF)N(C(c1ccccc1C(=O)OC)=O)CC C1(COC)COCCN1C(C1COCC1NC(=O)C(C)(C)O)=O c1(C(NOCC(=O)NC(CC=CC)CO)=O)cncn1C(C)C Cc1cc(C(=O)N(C(CNC(c2cc(Br)cn2C)=O)C2CC2)C)cnc1O c1(C(N2C(CC(=O)NC3CN(CC)CC3C)COCC2)=O)cnn2cccc2c1 c1(CN(C(=O)C(n2cc(CCC(C)O)nn2)C)CCC)ccc(Cl)c(Cl)c1 C(=O)(C(C)CC(F)F)N1CC(F)(CNC(c2cc(C)n(C)c2)=O)C1 c1(CCC)cnnc(C(=O)NCCCCCCNC(c2cccnc2S)=O)c1 C1(NC(c2cnc(C(C)C)s2)=O)CC(NC(=O)C(c2ccccc2F)O)C(O)C1 CCCC(C(=O)OC)C(=O)NC1CCCN(C(=O)CC23CCC(CC2)CC3)CC1 c1(CC=O)ccc2cnccc2c1.c1(COC)nc(C(=O)NC)cs1.C1CC1 N1(C(c2cc[nH]c(=N)c2N)=O)CC2CCC1C(C)C2.C(=O)C(C1CC1)C1CC1.N C(=O)(CCCC(C)(C)C)N1C(C)CCC(NC(=O)C(c2ccccn2)O)C1 C12(NC(C3N(CC)CC3)=O)CCCC1(F)CN(C(c1cc(OC)ns1)=O)C2 C12(C(=O)NCC(C)NC(c3ccc(N)cn3)=O)CCCC(C)(C1)OC2 C(CCCCC(=O)NC(C1(O)CN(C(=O)CN2CCCNC2=O)C1)C)OCC Cc1c(C(=O)Nc2cc(C(C)(C)C)no2)[nH]c2cc(C(=O)NCCCO)ccc12 n1(CC(=O)NCC(C)C(N2CCC(O)(C(F)F)C2)=O)ccccc1=O Cc1cc(=NCC2CCN(C(c3cc(Cl)c(Cl)s3)=O)CC2C)[nH]c(Cl)n1 c1(C(C(=O)NC2CC(C)(NC(C(COC)OC)=O)C2)C)ccncc1C c1(OC)ccc(CCC(N2CCSCC2C(N2CCC(F)C2)=O)=O)cn1 C(c1ccccc1C#N)=CC(N1CC(CC(C)NC(C(CCC)OC)=O)C1)=O C(C)(C)(CCC(=O)Nc1ncoc1-c1cccc(C(F)(F)F)c1)NC(C)=O N1(C(C=Cc2c(C)n(C)nc2)=O)CCCN(C(=O)C(F)(F)CC2CC2)CC1CO c1(C(=O)NC2CC(C)(NC(COCCCCCC)=O)C2)c(C)nsc1N c1(NC(=O)C(=O)NC2CCCC2CO)ccc(Cl)c([N+](=O)[O-])c1 C1(C(=O)NC2C(n3cc(C4(C)CC4)nn3)CCC2)CC(=O)N(C2CC2)C1 N1(C(CSC)=O)CCCC(N(C)C(c2cc(Cn3ccnc3)on2)=O)C1 N1(C(c2cc(C)nc(C)c2O)=O)CCC2(CC1)CC(NC(=O)C(F)C(C)(F)F)C2 Cc1cc(CN(CC(F)F)C(c2ncoc2C2CCCCN2)=O)cc(C)n1 c1(C(=O)NCc2ncc(C(=O)OC)n2C)ccc(OC)c(F)c1F CN1CC(C(N2CCC(N(C)C(C3CCOC(=O)N3)=O)CC2)=O)CCC1=O N1(C(C2(C(N(C(C)C)C)=O)CC2)=O)CC(C2CC2)C1.c1(C=O)scnc1Cl.N c1(C(=O)NCCCCNC(c2ccc(F)s2)=O)scc2c1CCCC2 N1(C(c2cnn(CC)c2Br)=O)CC2CCN(C(c3oc(C)nc3C)=O)CC12 C=C=C(C)CC(=O)NC1(C(=O)NCc2nccs2)CCOCC1 c1(C(=O)OC(C)C(=O)NC(c2ccccc2)C2CC2)ccc2nnn(C)c2c1 N1(C(c2c(SC)n(C)nc2)=O)CC2CCN(C(=O)CCn3ccnc3)CC12 N#Cc1cn[nH]c1C(N1CCC(CNC(=O)C=Cc2ccncn2)C1)=O c1(C(N2CC(CCn3cc(C(C=C)(C)O)nn3)C2)=O)ccnc(OC)c1F c1(OCC)ccccc1C(=O)NC(C)CCNC(C1CSC(C)=N1)=O C1CCOCC1.c1(CC(C)C)cc(C(=O)NC)n[nH]1.C1(CC=O)COC(=O)N1 c1(CN2CCOCC(C(=O)NC(C)C(=O)OC(C)(C)C)C2)cccc2[nH]ccc12 C1(CNC(c2ccc[nH]2)=O)CC(F)(F)CN1C(=O)C(F)F.c1ccccc1.C C=Cc1ccc(C(=O)NCC(=O)NCc2cn(-c3ncccn3)nn2)cc1 O=C1CC(C(=O)NCCCOC2CCC2)N(C(=O)C=Cc2ccncn2)C1 C(=O)(C(F)(F)C(O)CC)N1CCC(C(CNC(C=COCC)=O)C)CC1 C1(C2CCCOC2)(NC(CCC2(NC(c3c(C#C)c[nH]n3)=O)CCCC2)=O)CC1 c1(C(=O)NCCCC(C)NC(C2(C)CCC(=O)N2)=O)cc2nc[nH]c2cn1 C1(CNC(CCNS(C)(=O)=O)=O)CCCCC1NC(=O)CC=O.C1CC1 c1(SC)cc(F)ccc1C(N1CCCC(N(C)C(c2cccc(=S)n2O)=O)C1)=O N1(C(=O)CCOC2CC2)CCC(CNC(C2(C3CC3)CC2)=O)C12CC2 C1(C(C)(C)NC(c2n(CC)cnn2)=O)CCN(C(c2n[nH]c(C)c2O)=O)CC1 C(=O)(CCCCCC(C)C)N(C(C(=O)NCCc1cc(C)ncc1)C)C N1(C(c2ccc(CC)[nH]2)=O)CCC(C)C1.c1(CC(=O)N)cn(C2CC2)cn1 c1(C(=O)NCC2N(C(C(CC(C)C)C)=O)CCCC2)ccc2c(c1O)CCC2 C(=O)(N=c1nc2n([nH]1)CCC(=O)N2)c1ccc(S(C)=O)c(Cl)c1 C1(C(N2CC(OCCNC(C3CN(C(N)=O)C3)=O)C2)=O)OCC2CCCC12 C(N=c1ccn(C2(C(F)(F)F)CC2)c(O)n1)c1c(OC)ncc(-c2ccsc2)c1 C1(CC)(NC(=O)C(C(C)(C)C)SC)CCCN(C(=O)CCc2scnc2C)C1 Cc1cc(C(N2CCC(C(=O)NCC3C=CCCC3)(CF)C2)=O)cnn1 CCCC(C(=O)N1CC2(CCC2)CC1C(=O)NCCC1CCCOC1)C(C)C CC1CCN(C(C2CCC2)=O)CC1CNC(c1ccnc(O)c1)=O C1(NC(CCC=CC)=O)CS(=O)(=O)C2CN(C(=O)C=CC(C)CC)CC12 CC(CC(O)c1cccs1)NC(N1CC(OC(F)F)C1)=O c1(C(N(C(C)CNC(c2cc(N3CCCC3)ccn2)=O)C)=O)ncc(F)cc1F c1(C(=O)NCC(CNC(c2c(OC)c(Cl)ncc2)=O)O)c(C)ccc(C)c1C c1(C(C)=O)cc(C(=O)NC2(C)CC(NC(=O)CO)C2)c[nH]1.c1cccnc1 c1(C(=O)NCC(C)NC(c2ncc(F)cn2)=O)ncc(Br)cc1O C1(NC(C(n2cc(C)nc2)(C)C)=O)C2CC1N(C(=O)C(C)O)C2C N1(C(C2C(C)C3CCC2C3)=O)C2CCC1CC(NC(C1(c3ccsc3)CC1)=O)C2 c1(C(N2CC(C)C(CNC(c3occc3F)=O)CC2)=O)cc2c([nH]1)CCCC2 Cc1cc(C(N2CC(NC(C3(C)CC(C(F)(F)F)C3)=O)C(O)C2)=O)c(C)[nH]1 c1(OC)ccc2cc(C(N3CCC3)=O)[nH]c2c1.c1(C(=O)N)c(Cl)n[nH]c1C1CC1 N1(C(C(CC)C)=O)CCN(c2ccc(C(=O)NCCC(=O)NC3CC3)cn2)CC1 CC1(C)CCN(C(C2CCCCC2(C)C)=O)C1CC(=O)NCC1CCC1 C1(C(N2CC(CNC(CC3C(C)(C)CCO3)=O)OCC2)=O)CCc2nncn2C1 c1(C(=O)NC2C(NC(CCC)=O)CCCC2)nc(Br)n2c1CCCCC2 Cc1cnc(C(=O)NC2CCC(C(C)C)CC2)c[n+]1[O-] N1(C(C=Cc2cc(OC)ns2)=O)C2CCC1CC(NC(=O)Cc1nccn1C)C2 CCCC(C)(c1nnnn1C1CCCC1)NCCc1ccn(CC(F)(F)F)n1 C(=O)(CC(C(F)F)NC(=O)CN1CCC(C)C1)N(c1cccc(OC)c1)C c1(C(=O)NC2CC(C(=O)Nc3cccc(F)c3)C2)cc(Cl)ccc1OC(F)F C1(CC)CN(C(C2(F)CCC2)=O)CC1C(N1CCOC(CC(N)=O)C1)=O N1(C(C2CC(F)(F)CN2C(C2CC(NC=O)C2)=O)=O)CCCN2CCCC2C1 Cc1nc(NC(c2nnnn2-c2ccc(F)cc2)(C)CC2CCCC2)[nH]c1C C1(C(=O)Nc2cc(F)cnc2I)CC1C1CC(F)(F)C1 C1(SC)CCN(C(c2c[nH]nc2OCC(F)(F)F)=O)C2(CC2)C1 N1(C(C(CC=C)C)=O)CCN(C(=O)Cc2cccc(SC)c2)CC1COC N1(C(CCC(C)N(C)C)=O)CC2CC(C1)N(C(c1ccc(N(C)C)cc1F)=O)C2 C(=O)(C1CCCn2ccnc21)NC(C(C)C)CNC(c1cccc(C2CC2)n1)=O N(C1CCCn2cnnc21)C(C1(NC(C(C)C2CC2)=O)CC(F)(F)C1)=O C(c1c(F)ccc(Cl)c1F)=CC(N1CCOCC1)=O.C(C)(C(=O)N)OCC#C CN1CCN(C(=O)COC2CCN(C(=O)CCc3cccn3C)C2)CC12CCC2 C12(C=O)COC(C1)CC2.Cc1noc(C)c1C.C1(C=O)(C(N)=O)CCC1.N N1(C(C(C2(C)CC2)NC(=O)CN2CCSCC2)=O)CCOCC1CCO CCCC(CC)C(=O)N1CC(O)C(O)C1CNC(c1ccnc(C2CC2)c1)=O C1CN(C(c2ccc(Cl)s2)=O)C2CC12.c1(C(C(=O)NC)O)ccc(C2CC2)cc1 c1(N(C)CC2N(C(C(n3cc(Br)cn3)C)=O)CCC2)ccc(C#N)nc1 C1(C#N)(C(N(C)C)=O)CC12CCC2.c1(C2CC2)cccnc1.N1(C(C)=O)CCC1 Cc1cccc2oc(C(=O)NCC3=NOC4(CNC4)C3)cc12 C(CC(C)C(=O)NCc1cccc(C(=O)NCC2CCCOC2)n1)=CCC N1(C(c2c(C)cc(=N)[nH]c2)=O)CCC2(CC1)CCN(C(C1CC1CF)=O)C2 CC1(C(=O)NCCCCCNC(C2CC3C=CC2O3)=O)COCCO1 c1(OC)cncc(Br)c1C(=O)NC1CN(C(=O)C(C)(C)CC2CC2)C1 Cc1nc(Cl)nc(N2CC=CC(NC(c3ccc(C(F)F)o3)=O)C2)c1Cl Cc1cc(Br)c(NC(=O)NC2CCN(C(=O)C(C)(C)C)CC2)cc1Cl N1(C(CC(=C)Br)=O)CC(NC(=O)CNS(=O)(=O)CC)CC(O)C1 C1(C(=O)NC2CCC(F)(CNC(=O)CCCC)C2)(OCC)CCOCC1.S C1(CCC)(NC(=O)CCC(N)=O)CCN(C(C2CCN(C)C2CC)=O)CC1 C#Cc1ccc(C(=O)NCc2cccnc2CNC(C2CCC2)=O)cc1 C1(CNC(Cc2c(O)ccc(C)c2)=O)CCN(C(=O)C2=CCCCO2)CC1(F)F N12CCc3cc(ccc3C1)NC2=O.C1(CC)CCCC(CNC2CCCC2)CC1 C1(CC)C(NC(c2ccc(N)cc2F)=O)CCCN1C(=O)Cn1cc(C)cn1 C1(NC(C2CC3(CCOCC3)CN2)=O)(CO)CCc2cc(Br)ccc2C1 c1(OCC#C)ncccc1C(N1CCC(O)C1)=O.C1(C=O)CCCS1(=O)=O.C C(=O)(CC1=Cc2ccccc2C1)NC(CNC(C(C)C1CCC1)=O)C1CC1 c1(N2C(CC)CN(C(C3CC(O)C3)=O)CC2)ncnc2sc(Br)cc12 c1(C(=O)NCC2CCC(NC(Cc3cc(OC)no3)=O)C2)cc(C)ccc1Cl c1(C(=O)NCC(C)(C)F)cc(-c2cc(F)c(F)c(F)c2)c2n[nH]cc2c1 C(=O)(C(CCC1CCCO1)N1CCCC(C(=O)NCCC)C1)NCC=C CC1=C(C(=O)N2CC(NC(=O)CS(C)(=O)=O)C2)Cn2ncnc2N1C C(=O)(C1CCc2cccc(Cl)c21)N1C2CN(C(c3cncc(OC)c3)=O)C(C2)C1 C1(C(=O)NCC2(C=O)CC2)CCC2(CCOCC2)CO1.C1CC1.C1CC1.N c1(-n2c(CNCCC3OCC(C)(C)C3)nnn2)ccc(Cl)cc1F N1(C(C(SC)SC)=O)CCCC1(C)CNC(c1scc(C)c1Cl)=O Cc1cccc(C(=O)NC(C)C=CC(=O)NCC(C)(O)C(C)(C)C)c1C#N Cc1cnc(C=CC(N2CCC(CC(C)NC(C3NC(=O)CC3C)=O)CC2)=O)[nH]1 c1(C(=O)N)ccc(C(C)(C)C)nc1.c1(CC=O)cc(Cl)n(C)n1.CCC(C)C c1(CC)ccc(C(=O)NC2CCCN(C(=O)CC3CC=CCN3C)C2C)c(C)n1 N1(C(c2c(CC)nco2)=O)CCC2(CC2)CC1C(=O)NC.c1ccc(F)cc1C C1(O)(C(C)C)CCN(C(=O)CCN(C)C(C2CC(=O)CS2)=O)C1 N1(CC(=O)Cc2cc(F)cc(F)c2)CCOc2cccc(Cl)c2C1 c1(C(CC(=O)NCCCCc2cn(C3CCCC3)nn2)O)cccc(F)c1 C1(CNC(c2c(OC)ccc(Br)c2)=O)CC2CCC1N(C(=O)CCC1CC1)C2 C1(C(=O)NCC2ON=C(C)C2)CC12CCN(C=O)CC2.C(CC(=O)O)C=O.N C(=O)(C1=CCN(C(c2nocc2Cl)=O)C1)N(C(C=C)C)C CON1CC(C(=O)NC2CCCC(NC(=O)CCc3cnc(C)s3)C2)CC1=O c1(C(=O)NC2CCN(C(CCCCCC)=O)C(C)C2)cn2ccc(OC)cc2n1 C(CN=c1nc2sccc2c(NCC2SCCS2)[nH]1)c1nc(C)nc(O)c1 CCC(C)C(O)CC(=O)N(C(C)C(=O)NC1CCCNC1=O)CC n1(CCC(=O)NC(CC)CNC(=O)Cc2ccno2)ncn(C)c1=O CCC(C)C(C(=O)N1CCN(CC(N)=O)CC1)NC(=O)C=C(C)C(C)C C(C(=O)N1CC(C(O)C(=O)N(C2CCC3(CC2)CC3)C)C1)(C(C)(C)C)OC c1(OC)cc(C(=O)NC2CC2NC(c2cc(C(F)(F)F)n[nH]2)=O)ccn1 C1(CC(=O)N(C)CC2CCN(C)C2)(OC)CN(C(=O)CC2CC=CCC2)C1 CCC(C)C(C(=O)N1CC(O)(CSC)C1)N(C)C(c1ccc(F)c(F)c1)=O N1(C(c2cccc(C)n2)=O)CC2CCC2(CC(=O)NCc2ccc(O)nn2)C1 c1(C(=O)OC)nc(=NC2CC23CCC(NC(=O)C(C)C(C)O)CC3)cc[nH]1 C=CCC(F)(F)C(=O)N1CCC(CO)C(NC(c2ncccc2OC)=O)C1 C(=O)(C(CC(C)(C)C)OC)N(CCC(=O)NC1CC2CC1CC2CO)CC CCC(CC(F)F)C(=O)NCC(CNC(c1cc2ccccn2c1)=O)CO C1(CC)CCN(C(=O)C2=CCSC2)C1C(=O)NCC1(C)CC=CCC1 c1(C(=O)NC(C(C)C)(C)CNC(=O)CCc2ccncn2)cn2cnnc2cn1 CC(C)C(C)C(=O)N1CCOC(C(=O)N(CCCF)C)C1 C1(C(N(CC(=O)NCC(O)CNC(N)=O)CCC)=O)CN(C)CC(C)O1 c1(OCC=C)cc(Cl)ccc1C(N1CCN(C(C2COC2)=O)CC1)=O CC1CN(C(=O)CCCCC2CCCCC2)CCN1C(=O)C=Cc1ccccc1 C(=O)(N=c1ccnc(CO)[nH]1)c1cc(CNCc2cc(C)nn2C)ncc1 C=C(C)C(CC(=O)NCC=CC(=O)NCc1ncccc1C)OCC Cc1cc(CC=O)cc(C)c1.c1(C(C=CC=O)=O)ccc(F)cc1.CC=CC Cn1ncc(C(=O)NCCC(C)(C)NC(=O)COC2CC=CC2)c1N c1(OC)ccc(C(=O)N)cc1.C1CC(F)CN1C(c1ccn(CC(C)C)n1)=O.C C1(COC)CN(C(c2nnc(S)n2C)=O)CCN1C(c1ccc(C)cc1)=O C1(C(N(CC(=O)OCC)C)=O)CN(C(c2cc(O)nn2C)=O)CC1(C)C CCN=c1[nH]c(C)c(C(N2CC3CC(C2)C3NC(c2c(Cl)cnn2C)=O)=O)s1 N1(C(C(CNC(=O)CCOCC2CCC2)CC2CC2)=O)CCn2ccnc21 N1(C(CCOC(C)=O)=O)CCCC2CN(C(=O)Cc3ccsc3)CCC12 Cc1cc(CC(=O)NCC2(C)CCN(C(c3ncncc3Cl)=O)C2)cc(F)c1 c1(C(=O)NC(CCCNC(C=CCCC)=O)CO)nc(C)ncc1Cl C=C(C)C(C)(C)C(=O)NC1CC(CNC(=O)CCc2ccc(Cl)cc2)C1 C(=O)(CC(C)(C)C)N1CCC1.c1(OC(C)C(=O)N)ccc(F)cc1.C(C)(C)C c1(CCC)cc(C(=O)NC2(C)CCC2)cc(O)n1.C(=O)(CCCC1CCCC1)N C=C(C)CC(C(=O)N1CC(N(C)C(c2ccc(O)nn2)=O)C1)OC C(=O)(CCC(=O)NCCC1CC(NC(=O)C=Cc2ccc(C)o2)C1)NC Cc1ccc(Cl)c(C(N2CC3C(NCc4cccc(-n5cccn5)c4)C3C2)=O)c1 Cc1nc2c(N3CCCC(C(=O)NCCNc4cccnc4)C3)ncnc2o1 c1(OC)ccnc(C(N2CCC(O)(CCNC(=O)C(C)CC(F)F)C2)=O)c1O N1(C(CC2CCN(C(C)=O)CC2)=O)CC(NC(=O)C=C2CC2)CC(C)C1 CC(CC(=O)NCCN(C)C(c1cc[nH]c2nccc1-2)=O)CC(F)(F)F N1(C(CC(CC)C(C)C)=O)CC(C2CCCN(C(=O)C(C3CCCCC3)O)C2)C1 Cc1ccc(Br)c(C(=O)NC2CC2CNC(C2CCC(O)C2)=O)c1N C1(NC(C(COC)C)=O)CCCCC12CCN(C(c1cnc(C#N)s1)=O)CC2 CCCCCC(CC)C(=O)N(C(CNC(c1cc(C(F)F)n(C)n1)=O)C1CC1)C CC1(C)CC(NC(C2(F)CC2)=O)CN(C(=O)CC2CCCCC(=O)N2)C1 Cc1ccc(C)n1C(C)C(=O)NCCn1cc(C2(c3ccccc3)CC2)nn1 c1(C(=O)NC(C)CN(C)C(C2CC2(C)C)=O)cc(C2CCC2)on1 C(CCC(C)(C)NC(c1cn(C)c(C)n1)=O)NC(c1cnc(C)[nH]1)=O c1(C(=O)NCC(CC=C)NC(=O)Cc2ccno2)ccc(Br)c(F)c1C N1(C(c2cn(CC(C)C)nc2)=O)CCC(NC(C23CCCN2CCC3)=O)CC1C c1(C=O)c(Cl)cnn1C(C)C.C1(CC#C)(C(=O)NCC(C)CO)CCOC1.N C1(C(=O)NC(COCCOC)C)C2CCN(C(=O)COCC(F)F)CC12 N1(C(C2CC(CC)C2)=O)CC(O)CC1CC(=O)NCC1CCSC1 N1(C(C2(COC)CCCO2)=O)CCOCC1C(C)(C)O C(=O)(C(C(C)C)n1cnnn1)NCCN(C(c1c(C)scn1)=O)C1CC1 Cc1coc(C=CC(=O)NCCN(C)C(C2CC2O)=O)n1.c1ccccc1 c1(C(=O)NC(C)Cn2cc(-c3ccc(N)cn3)nn2)ncnc2ccsc12 c1(CC)ncc(C(=O)NC(C2CCN(C(=O)Cc3ccoc3)C2)C)c(C)n1 c1(OCC)n[nH]cc1C(=O)NC1CN(C(=O)COC2(C)CCCC2)C1 c1nc2cc(F)c(F)cc2[nH]1.c1(N2CCCC(C)(C(=O)O)C2)ncc(C#N)cc1F N1(C(C(F)=CCC)=O)CCC(C2CC2NC(c2conc2C)=O)CC1 O([Si](C)(C)C(C)(C)C)Cc1ccc(C(N(S(CC(=O)OC)(=O)=O)C)C)cc1 c1(N2CCCC(CNC(c3cnc(O)nc3O)=O)C2)nc(Cl)ncc1Br C(=O)(C1=CCC2CCC1N2C(=O)C(O)C(F)(F)F)N1C(C(=O)NC)CC1 C1(NC(CCOCCNC(C(CCC)C)=O)=O)CCOCC12CCC2 CC(N=c1cc[nH]c(=NCCc2c[nH]c3ccc(F)cc23)[nH]1)c1nncs1 C=C1CCN(C(C2CC23CCC3)=O)C(C(N2CCCOCC2C)=O)C1 C1(NC(c2c(C)n(C3CC3)nc2)=O)CCN(C(c2cn(C)c(=O)n2C)=O)CC1C N#Cc1ncc(NC(=O)C(=O)NCC2COC(=O)O2)cc1Cl C1(NC(CC(=O)OCCC(C)C)=O)(C)CCCCC1.c1(C=O)coc(O)n1.N Nc1ccc(C(=O)NCc2csc(C(N3CC(O)CC3C(N)=O)=O)c2)nc1 Cc1c(C(N2CC(F)(CNC(=O)C(C)(c3cccs3)N(C)C)C2)=O)ncn1C C1(CC)C(NC(c2snnc2C)=O)CCCN1C(=O)Cc1ccc(C)s1 Cc1c(Br)sc(C(N2CC(N(C(=O)CC3COCC3O)C)C2)=O)c1C C1(C(=O)NCc2ccc(OC)cn2)CCN(C(C2NC(=O)OC2C)=O)CC1O C1(CC(=O)NC2C=CCN(C(c3ncncc3Cl)=O)C2)CCC2(CCC2)CO1 C=CC(C(=O)N(CCCN(C)C(C1CSCN1C)=O)C)c1ccccc1 C=CCCCC(C(=O)NCC1=NOC(C)C1)NC(=O)C(O)CC1CCCC1 CC(C)(C(O)C(F)(F)F)NCc1ccc(F)cc1 c1(C(=O)NCC2(C)CCN(C(c3csnn3)=O)C2)cnc2ccnn2c1N Cc1ccc([N+](=O)[O-])cc1NNC(=O)NCC1(O)CCCC(C)C1 N1(C(CC)=O)CC(CC(=O)NOCCCCF)(C(N2CCC(NCC)C2)=O)C1 C=CCC(C(=O)NCCC1CC1)C(C)C.c1(C=O)c(C(F)(F)F)coc1C.C CCC(C)(CNC(c1cc(C(N)=O)[nH]n1)=O)C(=O)N1CCN(C)CC1C C(=O)(C1CCc2nccn21)N1CCCC(C(=O)NCCN2CCC2)C1 C1(CCNC(C2CC2C)=O)(NC(CSCC#C)=O)CCC1 C#Cc1cccc(C(c2nnnn2C)NCCOCCn2cc(Br)cn2)c1F c1(C(N2C3CCN(C(C4(N(C)C)CC4)=O)CC3C2)=O)cc(Cl)cc2c1OCC2 c1(C(N(CCCNC(C2(C)CCC2)=O)C)=O)c[nH]c2cccc(F)c12.C1CC1 C=CCC(C(=O)N1CC(O)(CCO)C1)NC(=O)CC1CCC(=O)NC1 N1(C(C(C)OCOC)=O)CC(O)C(O)C1CNC(=O)COCCC(C)C Cc1cc(C)c(C(=O)NC2COCCC2NC(C2CC2)=O)cc1C.C1CCC1.C Cc1cnn(C)c1C(=O)NC(C)(C)CNC(C1CC(N(C)C)C1)=O C=CCC(CNC(c1ccsc1)=O)NC(c1cc(Cl)c[nH]1)=O CC1CC(C(N2CCOCC2CC(N)=O)=O)N(C(=O)CC23CCCC2C3)C1 C(N=c1[nH]cnc2c1CCC2)C1(CNC(CNc2cn(C)nc2)=O)CCC1 Cc1cc(C)n2nc(C(=O)NC3CN(C(=O)CC(C)(C)C(F)F)C3)cc2n1 C1(CN(C(c2cnn(CC)n2)=O)C)COCCN1C(=O)CN(c1ccncc1)C C(=O)(CCCNC(c1cccs1)=O)NC(C#C)(C)C1CCOC1 C(=O)(C(CC(F)F)N(C(=O)CCCOC(C)C)C)NCc1c(OC)nsc1 c1(C(C)=O)c(NC(C2CN(C(=O)Cc3ccccn3)CCS2)=O)cccc1F c1(NC(C2CCCCN2c2ncccn2)=O)cncnc1O C(CC(C)(C)CC(=O)NCC(CC(C)C)C(=O)N1CCCCC1CO)OC c1(C(N2CCOCC2CC2CCC2)C(=O)NCC2CCCC2)cccc(F)c1F c1(CC)ccc(CN2CCC(CNC(=O)CC3CCCCO3)CC2)c(O)c1 c1(OC)cc(F)c(S(=O)(=O)NC(C2CC3(C2)CC(CN)C3)=O)cc1Br N1(C(c2ncn(C)c2)=O)C2CCC1CC(NC(=O)CO)C2.C(F)(F)C(F)(F)F C=CCC(CC(C)C)C(=O)N1CCC(F)C(NC(c2n[nH]c(C3CC3)c2Cl)=O)C1 c1(NCC(=O)NCCc2cn(CC34CC(C3)C4)nn2)ccc(Br)cc1 Cc1nn(C)cc1N(C(=O)C(C)(C)C1CCNCC1)c1ccncn1 C1(C(N2C3C(NC(C4(F)C(C)OCC4)=O)C(C3)C2)=O)CC2(C1)CC21CC1 O=C(CCc1nncs1)NCCOCCCNC(c1cnn[nH]1)=O CC1=C(C(=O)NC(CNC(=O)Cc2cccs2)C(C)C(C)C)CCO1 C1(NC(c2cnc(-c3ccccc3)nc2)=O)CCCN(C(C2CC2CF)=O)CC1 c1(C(=O)NCC(CC(C)C)NC(=O)CC2CCCCO2)cc2n(n1)CCNC2=O N1(C(c2c(CC)nn(C)c2)=O)CCC(C)C12CC2.C1(C=O)CCOC1C1CC1 c1(C(=O)NC(CNC(CN(C)CC)=O)C2CCC2)csc(=NC)[nH]1 N1(C(c2c(OC(C)C)nccc2)=O)CC(NC(C2CCCCN2C)=O)C(C)(C)C1 C[Si]1(C)CCC(CNC(=O)CCC2CCCN2C(c2ccc(F)s2)=O)C1 C(CC(C(=O)N(CC(O)CF)C)NC(=O)CC1(C#N)CC1)N(C)C c1(CCC(=O)N(C2CCN(Cc3ncc(C)s3)C2)CCO)ccccc1F c1(C(=O)N)cc(F)c(O)c(Cl)c1.C1(C(N2CCOCC2)=O)CC2(CCCC2)C1.C CN1CC2(CCN(C(c3ccccc3)C(=O)NCC(F)F)CC2)OC1=O CC(CC(C)(C)C)C(=O)NC1CCCCC1NC(c1ccnnc1)=O C1(NC(C2C(CN(C)C)C2)=O)COCCN(C(c2cn(C)[nH]c2=N)=O)C1 c1(OC(C(=O)NC)C)cccc(CNC(c2cccnn2)=O)c1 c1(C(=O)NC2CCC(N(C(CCN(CCCCC)CC)=O)C)C2)c(C)ncn1C c1(C(N(CC(CNC(C=CSC)=O)C)C)=O)cc(C)cc(C)n1 C1(F)(CNC(c2ncc(C)cc2F)=O)COCCN(C(=O)CO)C1.C1CCOC1 C=CC1(C(=O)NCC2CCC(NC(=O)C(c3cccnc3)C)C2)CCOCC1 c1(C(=O)N)cc(S(N)(=O)=O)n(C)c1.c1(C(=O)NCCC)ccc2n[nH]cc2n1 c1(CC)cc(F)ccc1C(=O)NC1CCCC1CNC(=O)CC.C=O.N c1(OC)cccc2c1CCCC2NC(=O)N=c1cc(C)[nH][nH]1 c1(C(=O)NC2CCC2NC(c2cnoc2C2CC2)=O)ccccc1.CCF.O C(=O)(CCCCCn1cnnn1)NC1C(OC)CN(C(COCCC#C)=O)C1 N1(C(c2cc(C)[nH]n2)=O)CC2CCC2(CCNC(c2ccc(CO)nc2)=O)C1 CC1(C)C(NC(=O)Cn2cccn2)CCN1C(=O)CCn1cnccc1=O C1(NC(=O)C(C2(O)CCCC2)F)CCOC12CCN(C(c1ccoc1Cl)=O)CC2 C1(NC(C(CC)CC)=O)CN(Cc2c(Br)cnn2C)CC1(F)F C(CC(C)(CC)NC(=O)C(F)C1CCCC1)NC(Cc1c(CC)con1)=O C1(CCC)CN(C(C2CC(=C(F)F)C2)=O)CCN1C(=O)CCNC(C)=O c1(N(C)C)ccc(NC(C2CCCC(N)C2)=O)c(F)c1 CC1(C)CCCC1C(=O)NCC1CC1CNC(C1CC(O)C1)=O C1(O)CCN(C(c2cc[nH]c(=N)c2N)=O)CC1.C(CC(=O)NC)OCCCOC N1(C(C(C)(C)O)=O)CC(CNC(=O)COCC2CCCCO2)C(F)(F)C1 c1(OCC)nc(Cl)cc(=NC(=O)C2CC2NCc2cccc(OC)c2C)[nH]1 c1(C(=O)NCC(C)N(C(CSCCC(C)C)=O)C)cc(S(N)(=O)=O)c[nH]1 N1(C(CCCCCCCC)=O)CCC2(CC1)CCN(C(C1CCOCC1)=O)C2 C1(NC(Cc2scc(C)n2)=O)CCCN(C(C2CCCCO2)=O)CC1 C1(CCn2c(N3C(C)COCC3)nnn2)OCCN(C)C1c1cnn(C)c1 C(=O)(C1CCc2snnc21)N(CCCn1cc(CCC2CCCCO2)nn1)C c1(C(N(C2C3CN(C(=O)Cc4cccc(Cl)c4)CC23)C)=O)nnc2ccccn12 C1(NC(CCN(CC=C)C(c2cscn2)=O)=O)CN(C(C)C)CC1C N1(Cc2ccc(S(C)=O)cc2)C(=O)NC2(CCN(C(=O)O)CC2)C1=O.C(C)(C)C c1(COC)ccc(C(=O)NC2CCCN(C(C3CCC4CC4C3)=O)C2C)cc1F C(=O)(CCCC(C)CCC)N1C2(CN(C(C(CCCC)O)=O)C2)CC1 C1(C(=O)NC2CN(C(c3cc(C(C)C)[nH]n3)=O)CC2F)CC2CCC(C1)O2 C1(CNC(C(=O)NCC(n2cccn2)C)=O)CCOC2(CCC2)C1 c1(C(N2CCN(C(c3n(CC)ccn3)=O)C(C)C2C)=O)csc2ncnc(O)c12 Cc1cccnc1C(=O)NC1CCC1NC(=O)C(C(C)C)N(C)C.C(=O)C CC1(C)CC(NC(=O)CC2C=CCC2)CCN(c2ncncc2Cl)C1 C(CS(=O)(=O)c1ccc(C(=O)Nc2ncsc2C(=O)OC)cc1)OC N1(C(CC(CC)C)=O)CC2OCCN(C(c3cc(F)cnc3O)=O)C2C1 Cc1cc2c(C(N3CC4(CCN(C(=O)C(F)C(C)C)CC4)C3)=O)nccn2n1 c1(C(=O)NC2(c3ccc(Cl)cc3)C(CCC)C2)c(F)c(N)cc(Cl)c1F N1(C(Cc2ccc(C)s2)=O)CCC2CC12C(=O)NCc1cnccn1 c1(C(N2CC(NC(=O)C(F)(F)C3CC3)CC(F)C2)=O)ccc2ccncc2n1 C=CCCCCCC(=O)NC1CCOCC1NC(C1COC(=O)N1)=O C(=O)(CN=c1ccc(C#N)c[nH]1)N1CC(C(C)NC(C2CC(C)CC(C)C2)=O)C1 N1(C(CCC(=C)Br)=O)CCn2c(CNC(C3(C)CC4CC4C3)=O)nnc2C1 N1(CC)CCCC1CCNC(=O)NC1CC(F)C1.C(C)(C)C.C(=O)N C1(NC(C(C2CCN(C(c3cnco3)=O)CC2)C)=O)CCN2CCC1C2 Cc1cc(C)c(C(=O)NCCN2CCCCC2)[nH]1.C(=O)(C(C)CC1CCCC1)N C1(NC(Cc2ncc(C)o2)=O)CC(C)N(C(=O)C(C(C)C)n2cnnc2)C1 C12(NC(CSCCC)=O)CCOCC1CN(C(=O)Cc1c(F)cc(F)cc1F)C2 C1(NC(c2ccc(OC)nc2)=O)C2CC1CN(C(C13CC(C)(C1)C3)=O)C2 C1(C(N(CCCNC(=O)CCC2CC2C)CC)=O)CC2(C1)CC2F Cc1[nH]nc2ccc(C(N3CCC4CN(C(c5ccoc5Cl)=O)CC34)=O)cc12 C(=O)(C(F)(F)COC1CCC1)NCC(n1cc(CC(c2ccccn2)O)nn1)C C(=O)(C1=C(C)CCOC1)N1CC(NC(c2c(OC)cccn2)=O)(CO)C1 Cc1cc(Cl)ncc1NC(=O)CC1(C)CCN1C(=O)C=CC=O.C1CC1 c1(C(N2C(CCNC(CCCOC)=O)COCC2)=O)ccc(S(N)(=O)=O)o1 C(CC=O)(C(C)C)NC(C1(CCOCC)CCC1)=O.C1(C(C)C)CC1.N c1(C(N(CCCNC(c2ccc(OC)cc2)=O)C)=O)nccn2ccnc12 c1(C(=O)NCC2CC(C)N(C(=O)CC3CC3)C2)cc(C(F)(F)F)ncc1Cl c1(C(=O)NCC2CN(C(CCCCOCC)=O)C(C)C2)cc2ccccc2o1 Cc1cc(C(F)(F)F)ncc1C=O.C1(C(N(CC)C)=O)OCCC1C(C)C c1(OC)cc(C(=O)NC(Cn2cncn2)C(=O)N)[nH]n1.C(C)CO.C(C)=O N1(CC=O)CCN(C)C(=O)C1.C(C(C(=O)NCCCO)NC(C)=O)OC.N CC(C)C(O)CNC(=O)C(C)(C1CC1)N(C)C(C1CCC(=O)O1)=O N1(C(Cc2nc(CC)sc2)=O)CC2(NC(=O)Cc3ccc(O)nc3)CC1C2.C CC(C)(O)C#CC(=O)NC1CN(C(=O)Cc2cc(F)cc(Cl)c2)CCC1CO c1ccccc1[N+](=O)[O-].c1(OC)ccc(CNC(N2CCC2C(=O)N)=O)cc1 C1(CC=O)CCC(O)C1.c1(CC)n[nH]cc1C(=O)NCC.C1(Cl)CC1(F)F C1(NC(CC(=C)C)=O)CC2CN(C(=O)C(CCC)Oc3ccc(Cl)cc3C)CC12 C(C(=O)NC(C)CC(C)C)(C(C)C)SCC.C(=O)C=CC(=O)N(C)C N1(C(C2C(CC)CCC2)=O)CCC(CCCNC(c2ncn(C)c2C)=O)CC1 c1(C(C)Nc2cc(NCC3CCSC3)ncn2)ccccc1[N+](=O)[O-] c1(C(=O)NC2(C)CCN(C(C3(C(F)(F)F)CC=CCO3)=O)C2)cc2cscc2s1 N1(C(c2c(C)csc2)=O)CCCC(N2CCN(C(C3(S(C)(=O)=O)CC3)=O)CC2)C1 C1(CN(C(=O)CCn2ccc(=N)[nH]2)C)CN(C(C2CC23CC(O)C3)=O)CCO1 N1(C(=O)CCN2CCCC2)CCC2CN(C(C3(Br)CCC3)=O)CC12 CCCC(CCC)=CC(=O)NCCN(C(=O)CCS)CCOCC.CCCC C1(CNC(CC(=C)C)=O)CC(O)CN1C(=O)CC1C(CC)C1(F)F N1(C(c2cc(C)c(N)cn2)=O)CCC2(NC(c3coc(Br)c3)=O)CCCC12 C(CCC(=O)C(C(N(CC(C(=O)O)N(C)C)C)=O)CC)NC(C)(C)C C1(C)(NC(=O)NC2C(c3ccc(C)cc3)C2)CCc2ccccc2C1 Cc1cc(Cl)ccc1C(=O)NC(C)CCN(C)C(C1(C)CC1C)=O c1(CCC=O)ccc(C(F)(F)F)o1.N1(C=O)CCC1C=O.CC(C)C.CC Cc1nnc2n1C(C(=O)NCCNC(=O)CC1(n3cccc3)CCOCC1)CC2 C(CC1=CCOCC1)NC(C1C(NC(Cc2c(CC)con2)=O)COC1)=O Cn1cc(N)c(C(=O)NC2CCCC(NC(c3nn[nH]c3Cl)=O)C2)n1 S(=O)(=O)(c1ccc(Br)cc1)N1Cc2c(-c3cc(C)c(N(C)C)cc3)n[nH]c2C1 C(=O)(C1CCCn2cnnc21)N1C(C)CC(CNC(c2ccsc2C#N)=O)CC1 c1(CCC)nc(C)c(C(=O)NC2CCN(C(=O)C(C)OCC3CC3)CC2)s1 Cc1cc(C(=O)NCCN2CCN(C(C3COCC3(C)C)=O)CC2)c(F)cc1F O=C1NC(=O)C(CCC(N2CCN(CCNC(=O)C(F)(F)C3CC3)CC2)=O)N1 c1(N(CCCCC=C)C)ccncc1S(=O)(=O)NC(C)CNC(=O)NC C(CCCC(=O)N1CC(CF)(NC(=O)C(C)CN(C)C)C1)SC CCS(=O)(=O)CC(=O)N1CCOCC1C(=O)NCC(CO)C(C)C C1(NC(C(C)=CC2CC2)=O)(CNC(c2csnn2)=O)Cc2ccccc2C1 c1(-n2c(C)cnn2)ccc(C(=O)NCCCC(C)NC(=O)C(O)C(C)C)cc1 S(=O)(=O)(c1ccc(Br)cc1NCc1cc(Cl)ccc1Br)NC1C(C#N)CCCC1 C1(NC(=O)C=Cc2cccs2)CCCCC1NC(=O)COC1CCCCCC1 CC(C)(C)C(CNC(C1CS(=O)(=O)C1)=O)C(=O)N1CC(N2CCOC2=O)C1 N1(C(c2ccn(C(C)C)n2)=O)CC(O)CC1(C)C(=O)N(C)Cc1cccc(O)c1 C1(NC(CC(C=C)(C)C)=O)CN(C(c2cc(C)c(C)[nH]2)=O)CC2(CC2)C1 C1(O)(C(=O)COC(C2(C)CCCCO2)=O)C2C3CC4C5C3CC2C5C14.C1CC1 N1(C(c2c(C3C(C)C3)noc2)=O)CC2CCC1CN2C(c1cc([N+](=O)[O-])c[nH]1)=O c1(C(N(CCOCCN(C)C)CC2CC2)=O)ccc(-c2nc[nH]n2)cc1 C1(OC)CC2CCC(C1)N2C(C1CCCCN1C(C1CCCCC(=O)N1)=O)=O CN=c1nc(N(C)Cc2ccc(Br)cn2)[nH]c(=NC2CCCC2CF)[nH]1 C(=O)C(F)(F)C(F)(F)C(F)(F)F.C(=O)(C(O)C(C)(C)C)N1CC(CC)C1.N c1(C(=O)NCC2CCCCN(C(c3cc(=O)cc[nH]3)=O)C2)cc2ncccn2n1 C1(N(C(c2c(C)nc(CO)o2)=O)C)CCCN(C(=O)CCc2cscn2)CC1 C1(C(=O)NC(CC=C)C(=O)OCC)CCCCCC1NC(=O)C(F)C(C)(C)O C(=O)(C1CCCc2c(O)cccc21)NC(CNC(c1cc(CC(C)C)on1)=O)C c1(N2CC(NC(C(C)C3CC3)=O)C(C)CC2)ncnc2c1CCO2 N1(C(=O)Nc2cncc(C(F)(F)CF)c2)CCS(=O)CC1c1ccccc1 N1(C(C(CC)F)=O)CC2(C1)C(NC(c1ccn3nncc3c1)=O)CCS2(=O)=O C(=O)(C(O)C1=CCCCC1)N1CCC(NC(CCn2c(C)ncc2)=O)CC1 C(C(CCC)NC(=O)CCc1cnn(-c2ccccc2)c1)NC(C(C)=CC)=O N1(C(C(CC)SC)=O)CCCC(C)(NC(c2cc(OC)nc(C)c2)=O)C1 C1(NC(C(C)OCOC)=O)CC12CC(NC(C1(CO)CCC1)=O)C2 C12(C(=O)NC(c3ccccc3O)C)CC(CO1)N(C(c1cnc(N)cn1)=O)C2 CCCC(C)C(c1nnnn1CCSC)NCC(=O)N(C)OCC(=O)OCC n1(CC(=O)NC(c2ccsc2)CC)ccc2ccccc12 N1(CC=O)CCS(=O)CC1.c1(C(C(=O)NCC2CCCC2)O)ccc(Cl)cc1.N C1(CC)CCN(C(=O)C)CC1.C(=O)CCC(C)C.C(=O)(CSC(F)F)C=O.N C(CCCCC(=O)N(C)CC1CCCC1NC(=O)CCc1ccn(C)n1)=CC C(c1ccccc1)=CC(=O)NCCNC(C=C)=O.C1CCN(C(C)=O)C1.N c1(OCCC(N2CCC3CCC23CNC(C2CC2)=O)=O)cc(F)ccc1F.C C(C(C)S(C)(=O)=O)NC(CC1(C)CCOC1)=O.C1(C(=O)N)CS(=O)(=O)C1 C(=O)(CS(=O)CCC(F)(F)F)N1CC=C(CNC(c2cn(C(C)C)nc2)=O)CC1 N1(C(CCCC(C)O)=O)CCCC2(NC(=O)C=Cc3cn(C)nn3)CCCC12 C1(NC(C(CSC)O)=O)CCCN(C(c2cc(-c3ccccc3)ns2)=O)C1 Cc1[nH]nc(Br)c1CNCC1CC2CCC1O2 N1(C(c2nc(C)oc2)=O)CCCCC1CCNC(c1ncc(Cl)n1C)=O c1(C(N(C(CCNC(C(C(C)C)CO)=O)C)C)=O)cc2c(F)cccc2[nH]1 C(=O)(CCCCCF)NCCN(C(CC(CC)C)=O)C1CCCCCC1 c1(C(=O)NCC2(F)CC(NC(CCC#CC)=O)C2)c(Cl)ccc(C)c1O c1(-c2c(C(=O)NC3CCN(C(C)C)C3=O)nccc2)ccc2nn(C)cc2c1 CC(C)(C)C(CO)C(=O)NC1CCC1NC(=O)C(O)CC1CCCC1 C1(CCC)CN(C(=O)Cc2cccnc2)CCN1C(c1coc(C(N)=O)c1)=O N1(C(CCCOC)=O)CCC(C(N2CCN(CCO)C(C)(C)C2)=O)C12CCC2 Cc1nc2nccc(C(N3CCC(CNC(=O)CC4CC4(Cl)Cl)C34CC4)=O)n2n1 c1(C=O)ccc(C(F)F)cc1F.C1C2CN(C(=O)CC3CC4(CCC4)C3)CC12.N Cc1ccc(Br)c(C(=O)NC(C2CCCN2C(C2CCS2(=O)=O)=O)C)c1 c1(C(=O)OC)ccc(F)c(NC(C2C=CCC2)=O)c1.c1(C=O)ccnc(C)c1 CC(c1cccnc1)=CC(=O)NC1CN(C(c2n[nH]cc2Cl)=O)CCC1CO C1(C)(C(=O)NCc2nc(CC)sc2)CCN(C(=O)CCn2cc(C)cn2)C1 O=C(C1CCc2nccn21)N1CCC(N(C(=O)Cc2ccc(F)cc2)CCO)C1 C1(C(=O)NCCC(C)N2CCC2)CN(C(=O)C(N)=O)CCN1C C1(NC(Cc2nc(C)sc2)=O)CCCC2CN(C(C3CN(C)C(=O)N3)=O)CC12 C(=O)(CCCCNC=O)N(C)Cc1cnccc1C(F)(F)F.C(C)(C)C.N C(CC(C)(C)C)NC(c1c(OCC)scc1)=O.C(=O)C(C)SC(F)(F)F.N C(N=c1[nH]c(=NCC2CCCCC2O)[nH]c2c1SCC2)c1nccc(C)c1F C1(COC)(NC(=O)CCC(C)N(C)C)CCCN(C(=O)CCSC(F)(F)F)C1 CCCC(C(=O)NC1CCC(CNC(C2CC(O)C2)=O)C1)S(N)(=O)=O C(=O)(C(C(C)(C)C)n1cc(CNC(=O)OC)nn1)NCCC(CCC)O N1(C(c2c(C)nn(C)n2)=O)CC(CNC(C2CC2(Cl)Cl)=O)C(F)(F)C1 CCCC(C)(O)CC(=O)N1CC(C)N(C(=O)CCC=CC(C)C)CC1C c1(COC)ncccc1C.N12CCCC1OCCOCC(=O)NC2=O S(=O)(=O)(c1ccc(N2CCOC(CO)CC2)cc1Cl)NC(CSC)C COC1OC(=O)c2c(F)c(C(=O)OC(C)C(c3ccc(C)c(C)c3)=O)cc(F)c21 C1(CCC(=O)NCC(C)OCC#C)CCCCN1C(c1cnc(C)nc1)=O N1(C(CNC(CN(C)C)=O)=O)CCC(C2CCN(C(c3nocc3Cl)=O)C2)CC1 C(C(C)C)(C(O)C(=O)NC(C)(C)C(=O)N1CC(c2nc(C)no2)C1)OC CC1CN(C(=O)COCCF)CC(C)CN1C(c1cccc2cc[nH]c12)=O Cc1cc(O)c(C(=O)NCCC2CCN(C(c3ccncc3C)=O)C(C)C2)nn1 Cc1ccc(CC(=O)NCC2C(C)CCN2C(c2cnn[nH]2)=O)cc1 CC(CCCCNC(c1ccc(C2CC2)cn1)=O)NC(=O)C(CCO)N(C)C Cc1c(C(=O)NCC2CCCCN2C(=O)C(Cl)=CCl)cccc1C1CC1 c1(CC)cc(C(=O)N)ccn1.C1(C)CCN(C(=O)Cn2cc(C3CCC3)nn2)C1 c1(NCC(CC)(CC)NC(=O)C(F)CC2CC2)ncccc1S(C)(=O)=O c1(C(=O)NCCCC)ccc([N+](=O)[O-])c(N)n1.c1(C(CC=O)C)ccc(C)cc1.N c1(NC(=O)NC2CCC(S(C)(=O)=O)C2)cccc(Cl)c1S(C)(=O)=O N1(C(C(Br)=C(C)C)=O)CCC(NC(c2ccc(C(C)C)nc2C)=O)C(F)C1 C(CCC(C)C(=O)N(C1CCCC1)CCNC(=O)C(CO)N(C)C)OC N1(C(C2CC(CC)OCC2)=O)CCCOC(CNC(=O)C(C2CCCCC2)O)C1 c1(OC)ccc(C)cc1C(N1CC(C(=O)NC23CC(C2)C3)C1)=O C(=O)(C#Cc1ccc(Cl)cc1)N1C2CC(CN(C(c3ccc(Br)cn3)=O)C2)C1 C1(N(C(C(C(C)C)n2ccnc2)=O)C)CCC2CN(C(=O)CSC(F)F)CC12 N1(C(c2c(C)cc(F)s2)=O)CC(CNC(c2cc(N)cnc2Cl)=O)CCC1C CC1(C)CCN(C(C23CC(CN(C(=O)C4=CCOCC4)C2)C3)=O)CC1 C(=O)(C(CO)C(C)C)NCCN(C(=O)CCOc1ccccc1C)CCC N1(C(C)=O)CCN(C(=O)C(c2cn(C)nn2)N)CC1C N1(C(C(CC(C)C)OC)=O)CC(NC(c2cc(C#N)c[nH]2)=O)C2(CCOCC2)C1 N1(C(CCOCCCOC)=O)CCC(CO)CC1.C1(C(=O)N)(C(N)=O)CCC1 C1C2CN(C(C3C(C)(C)C3(C)C)=O)CC12.c1(C(C)(C)C)[nH]cnc1C(=O)N C1(C=O)CC(=O)N(CC(C)C)C1.N1(C(C2CC(SC)C2)=O)CCCC1CC.N CC1(C(=O)NC(c2ccccc2)C)COC(=O)C1.C12(C(=O)N)CCC(CC1)C2 c1(C(NOCc2cn(-c3ccc(C)cc3C)nn2)=O)ccc2c[nH]nc2n1 C1(C)(C(=O)N)CCCC1(F)F.N1(C(c2nc(C(C)C)sc2)=O)CCCC1C1CC1 CC(CO)C(=O)NC(C)CC1CN(C(C2(Cc3ccccc3)CCCC2)=O)C1 C1(NC(C=CCN(C)C(c2cn(C)nn2)=O)=O)CCC2CC12 c1(OC)cc(CNC2CC(C(=O)Nc3cn4ccccc4n3)C2)cc(O)c1O CC1(F)CCCN(C(=O)CCC2(NC(=O)CN3CCCNC3=O)CCCC2)C1 C(=O)(CCCC(=O)c1ccc(F)cc1)N(CCC(C)NC(=O)CC)C.C(N)(=O)N N1(C(C)=O)CCCC(N(C(c2ccn(C3CC3(F)F)n2)=O)C(C)C2CC2)CC1 C(=O)(C1=CCC2CCC1N2C(=O)CC1(O)CCC1)N1C(C)CC(F)(F)CC1 C1(NC(c2ccc(Cl)c(C)c2Cl)=O)CCC2(CC1)CN(C(C1CCC1)=O)CCO2 N1(C(C)(C)C)CC(CNC(=O)NCC(O)COc2ccc(Cl)cc2)CC1=O C1(CCC(=O)NC(C)CCN(C)C)CCN(C(C2C3CC4C(C3)C24)=O)CC1 C1(CC(=O)N(C)CC2(NC(c3cccc(C)c3)=O)CC2)CN2CCC1CC2 CCCCC(CC)C(=O)N(CCNC(C1OC2CCC1CC2)=O)C(C)C Cc1cccn2cc(C(=O)OC3CCC(C)C(C)C3)nc12 c1(C2CC(=O)NC2)cccc(C(=O)NCCC(=O)Nc2cccc(F)c2)c1 c1(NC(C2CC2NCc2cc(F)c(O)c(F)c2)=O)cc2c[nH]nc2cc1F C=Cn1nncc1C(=O)NC1CCC(NC(=O)C(C2CCCC2)OC)CC1 c1(C(=O)NCCN(CCC)C(C2CC2Cl)=O)cc(C(=O)OC)ccc1N c1(C(=O)NC2(C(=O)O)CC3(CCOC3)C2)cc(Br)cc2ccccc12 N1(c2ccnc(C)n2)CCC(CNC(=O)C=CC(N)=O)C(F)(F)CC1 C1(C(C)NC(C(C2CCCCC2)OC)=O)CCN(C(=O)C(C)SC(C)C)CC1 c1(C(=O)NC2C(CNC(c3c(C)nn(CCO)c3)=O)CC2)ccn2nncc2c1 C(CN=C(NCCc1cccs1)NC1CCCC1)c1c(C)nc(C)s1 C(=O)(C1=C(Cl)CCOC1)NCC1CCN(C(C2(CC#C)CCC2)=O)C1 C(=O)(C(C)CC(C)C)NC(CCC)C(=O)NCc1cc(=O)cc[nH]1 c1(CC(=O)NCC2C(C)CN(C(=O)CNC=O)CC2)csc2ccccc12 C1(CNc2ncc(C)c(O)n2)N(C(=O)COCc2ccncc2)CCCC1(C)C C=CCCC(C(=O)NC(c1nnc(O)n1C)C)NC(c1cc(O)ccc1C)=O Cc1ccc(C2=NOC(CNC(=O)NCc3nc(Br)cs3)C2)cc1 C1(C(N(C(C=C)C)C)=O)(NC(c2cnc(N)cn2)=O)CCCC1C c1(CCC(=O)NC2CC(NC(C=C3CCC(C)C3)=O)C2)cccc(F)c1Br n1(CC(=O)NCCN(C(c2c(C)nsc2)=O)C(C)C)cnc([N+](=O)[O-])c1 c1(-c2nc(C)sc2)cc2c(s1)CCN(Cc1cc3cc(Cl)cnc3o1)C2 C(CC1CCC1)(C(=O)NC1(CO)CN(C(=O)C=CBr)C1)NC(C)=O Cc1ccc2scc(CC(=O)NCc3cccs3)c2c1 c1(CC(N2CCC(O)(CC)C2)=O)cc(S(N)(=O)=O)cn1C.CCCC(C)C(=O)N CC(C)(Cl)C(=O)NCCC1CC(C(=O)NCc2cocn2)C1 c1(C(=O)NC2C3CN(C(C45CC(C#N)(C4)C5)=O)C2C3)cc2n(n1)CCCC2 CC1CCN(C(c2c[nH]c3cnccc23)=O)CCN1C(=O)C#CC1CCOC1 CC(C)C(O)C(C)C(=O)NCCC1(O)CCCN(C(=O)CS(=O)(=O)N(C)C)C1 N1(C(CSc2cc(C3(C)COC3)no2)=O)CCCCC1(C(=O)O)CO C1(C(=O)NC(CC)CNC(=O)CC2CC(C)=NO2)CCC(C)(O)CC1 C1(CNC(C2C(C)C2)=O)CCN(c2nncs2)CC1 C1(C)(C=O)CC2(C1)CC(F)(F)C2.c1(OC)cc(CC(=O)N)c(F)cc1O.CC C1(CC)CN(C(=O)CCC(=O)NC)CCC1NC(=O)CC1CCC(F)(F)C1 c1(NC(C2CN(C(c3cc(C#N)c(F)cc3)=O)C2)=O)c(F)cccc1[N+](=O)[O-] C1(C=O)COCCN1C(C1CCC1)=O.C(C(F)C)NC(C1(C(N)=O)CC1)=O n1(C(C)C)ncc(C(=O)NCC(O)CNC(C2(F)CC2C)=O)c1Br CC1CCCN(C(=O)C(=O)N(CC(C)NC(=O)Cc2ccccc2O)C)C1 C1(NC(C2CCN(C)CC2)=O)CCN(C(=O)C(=O)C(F)(F)F)CC1(C)C c1(C(=O)NCC(n2cc(-c3nc(C4CCC4)no3)nn2)C)ccc(Cl)c(Cl)c1 c1(C(N(CC(C)NC(C2(SC)CCC2)=O)C)=O)ccc(C)c([N+](=O)[O-])c1 N1(C(c2cc(C)c(Cl)s2)=O)CCC2CN(C(c3csnc3C)=O)C2C1 N1(C(COCC)=O)CCC(N(C(=O)Cc2coc(-c3ccc(Cl)cc3)n2)C)CC1 C=C(Br)CCC(=O)N1CC(NC(c2ccccc2SCC(=O)NC)=O)CC1C c1(NC(C2CCC(NCc3ncc(N(C)C)nc3)CC2)=O)cncc(C#N)n1 C(=O)(C(CC(C)(C)C)NC(=O)Cc1ccccc1F)N(C)Cc1nccc(C)c1 c1(C=O)cc2c(O)cccc2n1C.C12(NC(CSCCCC)=O)CC(C)(C1)C2 C1(C(=O)NC2(C)CCSCC2)CNC(=O)CN1C(=O)CCC1CCCO1 Cc1cc(F)c(Cl)cc1C(=O)N(CCC(C)NC(c1csc(CO)n1)=O)C c1cccc(N2CCOCC2)c1.c1cncc(CNC2CC2)c1.C1CCCO1.C(C)O CC(C)CC(O)CC(=O)N1CC2(C1)CN(C(C1C3C4CCC(C4)C13)=O)C2 C(=O)(C1=CCC(C)CC1)N1CCCCC1.c1cnn(C)c1.C(=O)(C)N(C(C)C)C N1(C(c2ccc(C)s2)=O)CCN(C(C2CC3(CCO2)CC3)=O)CC1C1CC1 CCCCCC(O)C(=O)NC(C(=O)Nc1cn(C)nc1Cl)c1ccoc1 C1(N(C(c2c(C)cno2)=O)CCO)CCN(C(C2(CO)CCCO2)=O)CC1 C#Cc1cc(C(=O)NC(C)C(C)C)cc(F)c1.c1(C(=O)N)cc(F)cc(Cl)c1N c1(CC(=O)NC(Cc2csc([N+](=O)[O-])c2)C(=O)O)cc2ccccc2oc1=O C(N=c1cc(C)nc(NC2CCOC(c3cccs3)C2)[nH]1)c1c(NC)cccc1 Cc1nsc(C)c1C(N1CCC(OCCNC(=O)C(Cl)=CCl)C1)=O N1(C(c2n(CC=C)ccc2)=O)CC(NC(c2ccn(CC)c2C)=O)CC1(C)CC CCCC(C(=O)NC1CCCCC1CNC(C1C=C1C)=O)N(C)C C(=O)(C#CC1CCCCO1)N1C2CN(C(c3c(OC)c[nH]n3)=O)C(C2)C1 c1(CC)cccc(C(N2CCC(C(=O)N(C)Cc3nccn3CC)C2)=O)n1 c1(CC(=O)NCc2cn(C3CN(C(C4CCC4)=O)C3)nn2)ccccc1Cl c12cc(O)nc(n1)-c1ccc(s1)N2C.N1(CC2CN(CC)C2)CCN(C)CC1 c1(C(=O)NCC2(O)CCN(C(c3n(C)ccn3)=O)C2)ccc2ccoc2c1 Cc1cccc(C(N2CCC(C(=O)N(C)CCOCCCO)C2(C)C)=O)c1C C(CCC(C)CC(=O)NC1CC(CNC(=O)CCC2CC2(Cl)Cl)C1)=C(C)C N1(C(C2C(C(=O)OC)C=C2)=O)CCOCC(C=O)C1.C(C)(C)C(O)C(F)F.N C1(NC(C2(COC)CN(C(c3cccs3)=O)C2)=O)CCC([N+](=O)[O-])CC1 N1(CC)CC(C(=O)NCC2(F)CCC2)c2ccccc21.c1(C(=O)N)ccccn1 C1(NC(CCC=C)=O)CC(CNC(c2ccn(CC(F)F)n2)=O)C1(C)C C(C(C(=O)N1C2CCC1CC2)C(C)C)NC(C=CCCC(C)C)=O N1(C(c2c(OC)cnnc2)=O)C2COCC1CN(C(=O)Cc1cc(C)[nH]n1)C2 CCC(CC(=O)N1CC(C(O)C(N2CC(O)(C(F)F)C2)=O)C1)CC(C)C CC(C)C(CC(=O)N1CC(NC(C2CCCCN2C)=O)C(C)C1)C(C)C Cc1nc(C(N2CC3(CCC3NC(C3CCCC4(CC4)C3)=O)C2)=O)c(=O)[nH]c1C c1(CCC)cc(C(=O)NC(C)(C)CNC(=O)C(C)NC(C)=O)no1 c1(OC)cc(=NC(=O)CN(C(=O)CCSC)C(C)C)[nH]n1C C(=O)(CCCC(C)(C)NC(c1cnncc1O)=O)N(C)CC1CCOCC1 c1(C(=O)NC2C(NC(C3(C#N)CCOC3)=O)CCC2)ccnc2c(F)cccc12 CCC(C)CCCC(=O)NC(CNC(c1cnn(CC)c1)=O)C(C)C n1(CC(N2C3CC(NC(CC=C)=O)C(C3)C2)=O)cc([N+](=O)[O-])ccc1=O CCCCCC(F)C(=O)NC(C)C(=O)NC1(CC)CCCC1 c1(C(=O)NC(C)C2CC2)cnc(O)c(Cl)c1.c1(C=O)cnc(C2CC2)[nH]1.N C1(C#N)(OC)CC(C(=O)NCCNC(C2CC2C(C)O)=O)C1 O=C1c2ccccc2CN1NS(=O)(=O)c1ccccc1C(=O)NC1CC1 N1(C(CCOc2cccc(C)c2)=O)CC2(CCCC2NC(C2CC(C)(C)O2)=O)C1 C1(C(N2CC(CNC(c3cnn(CCC)c3C)=O)C(O)C2)=O)CC2CCC(C1)C2 CC(CN(C)C)CC(=O)N(C1CCN(C(C2CC2c2ccccc2)=O)CC1)C N1(C(c2c(C)con2)=O)CC2(CCC2)CC1CNC(=O)Cc1ccccc1Cl C12(C(=O)NC(CC)CN(C(=O)C(C)N(C)C)C)CC(O)C1C2 c1(NC(C2CN(Cc3cc(Br)ncc3F)CCC2O)=O)nc(Br)ccc1Cl C1(NC(c2cnc(COC)nc2O)=O)CC1C1CCCN(c2ncc(Cl)cn2)C1 C(=O)(C1CCc2c[nH]nc21)NCC1C(NC(c2cc(C)c(Cl)cc2F)=O)CCC1 C=CCCCCCC(=O)NC1C2CCC1N(C(c1cnn(C(C)(C)C)c1C)=O)C2 N1(CC(N2CC(C(C)NC(c3ccnc(OC)n3)=O)C2)=O)CCCCCCC1=O C(C)(C(C)C(C)C)NC(C1C(OC)CCC1)=O.C12(CC=O)COC(C1)C2 C=C(C)C1OCCC1C(=O)NCCC1CN(C(=O)CCn2ccnn2)CCO1 C=CC(CC)CC(=O)NCC(CCOC)NC(c1ccc(N)c(F)c1)=O c1(CC(C)C(=O)NCC(O)CNC(c2ccnnc2)=O)ccccc1Cl C(=O)(C(C)(C)C(F)(F)CC)N1CC(NC(C2(OCC)CCC2)=O)N(C)CC1 Cc1c(C(=O)N(CC(C)C(=O)Nc2cncnc2O)C)[nH]ccc1=O N1(C(c2c(CC)cno2)=O)CC2(CCN(C(c3nc(O)[nH]c(=O)n3)=O)C2)C1 C1(C2CCN(C(=O)C(O)C3CCCC3)C2)(NC(c2cnc3[nH]nnc3c2)=O)CC1 c1(C(N2CCCC(N(C(C(C)C3CCC3)=O)C)C2)=O)cc2ccc(F)cc2o1 C(=O)(C1CCc2c[nH]nc21)N(C(CNC(=O)C=Cc1cocn1)C1CC1)C C(C#Cc1cn(CCC2CC3(CCC3)CO2)nn1)C(C)=O.N1CC(C)(C)C1 N1(C(C(C)=C(CC)C)=O)CC2CCN(C(C3(CCCF)CC3)=O)CC12 N1(C(CCc2onc(C)n2)=O)CCN(C(C23CCCC2OCC3)=O)CC(C)C1 c1(CC)nn(C)cc1C(=O)N(CCCOCCN(C)C(C1CCCO1)=O)C c1(NC(CC2CCC(=O)NC2=O)=O)cccc2c1COC(=O)N2 Cc1[nH]nc2c1CCC(C(=O)NCCC1(O)CCN(C(c3cnnn3C)=O)C1)C2 C(c1ccc(=N)[nH]c1)=CC=O.C1(CNC(C(CC)=CC)=O)CCCCC1.N C12(C(=O)NC3C4CN(C(CC(C)N(C)C)=O)C3C4)CCCCC1CCC2 c1(C(N2C(C(N3CCC(O)C3)=O)CC3CC32)=O)ccc(Cl)c(Cl)n1.c1ccccc1 c1(CN2C(C(N3CCCC(CC)C3)=O)COCC2)ccc(Cl)cc1[N+](=O)[O-] S(=O)(=O)(c1ccc(C(=O)NCc2ccn(C)n2)cc1)N1C(CCC)CNCC1 c1(N2CCCC(F)(CC)C2)nc(=NC2CCCCC2C(N)=O)[nH]c2c1CSC2 C(=O)(C#CC1CCCOC1)NC1CN(C(C2(C)CC=CC2)=O)CC(F)C1 c1(C(N(C(C)C)CCO)=O)cccc(O)c1O C1(C(N2C(CNC(=O)C3=COCCO3)COCC2)=O)CCCCC12CCC2 Cc1ncn(O)c1C(=O)N.C12(CC)CCC(CC1)C2.C(CCC(C)C)=CC=O C(CC(C)C(=O)N1CC(N(C)C(c2cc(C3CC3)sn2)=O)C1)=CC C1(CNC(C2(CC#C)CCC2)=O)CC2CCCCC2N1C(c1ccccc1C)=O CC(C)C(C(=O)NCC1(NC(c2sc(Br)cc2F)=O)CC1)C1CCC1 c1(CC(=O)NCC=CCNC(c2cn3c(n2)CCC3)=O)cccc2c1OCO2 C1(C(N(C2CC(=C)C2)C)=O)CCCN1NC(=O)C(F)C(CC)CC CC(=O)CCCC(=O)NC1CCN(C(=O)C(C)(C)OC(C)=O)CC1O c1(C(N2CC(NC(=O)C=Cc3ccccn3)C2)=O)ccc2ncnc(O)c2c1 N1(C(c2cnc(OCC)nc2)=O)CCC(CNC(=O)C2=COCCO2)C12CC2 Cc1c(F)ccc(CN2CC3CCN(S(=O)(=O)c4ccc(Cl)s4)C3C2)c1F c1(C(=O)NC2CCC(NC(C3(C)CC3)=O)C2)cccc(N)c1 Cc1nc(Nc2ccc(F)c(N3CC(C)(C)C3=O)c2)ccc1[N+](=O)[O-] C1(OCC)CN(C(=O)C(CC)OC)CC1CNC(=O)Cc1cnccc1Cl c1(CN(C(CC(C)F)=O)C)ccc(CNC(=O)CCN2CCCC2=O)cc1 C12(NC(C3CCC(=O)OCC3)=O)CCC(CC1)N(C(=O)CN1CCCC1CO)C2 C(C)(CCC(=O)NCC(C)C(=O)OCC)NC(CSCCC)=O C1(C(=O)NC2CC=C(C)CC2)CCCCC1(C)NC(C1CC2(CC(=O)C2)C1)=O C1(C)(C(=O)NC2CCC(NC(c3c(C)nc(C)n3O)=O)C2)Cc2ccccc2N1 Cc1cc(C(N2CC(O)CC2C(=O)N(C(C)CN(C)C)C)=O)c(C)nn1.C N1(C(C)=O)CCC(CC(=O)N(C(C)C)CC2(c3cc(C)on3)CC2)CC1 c1(C=O)cccc(CS(N)(=O)=O)c1.CC(CNC(=O)CCOC1CC1)C CCC(CC(=O)N(CCNC(=O)CNc1ccncc1)C1CC1)C(C)(C)C CCC(CC)C(F)C(=O)N(C1CC(NC(C2OCC3CCCC23)=O)C1)C C12(NC(c3cnc(C)s3)=O)CCCC1CN(C(=O)C=CC1CC1)C2 CCCCC(CC)C(C(=O)NCC)N1CCC(CC2CCCO2)C1 C(=O)(C(C)CCCC(C)C)NC1(C)CC(C(=O)NCC(N(OCC)C)=O)C1 C1(C(=O)NC(CC=C)C(=O)OC)CCN(C(=O)CC2CC(SC)C2)CC1C Cc1ncn(C)c(=O)c1C(N1CCC(O)(C)C1)=O.C1(C#N)(C(=O)N)CCCO1 C=CCC(CC(=O)N(C1CCCCC1(C)C)C)NC(=O)C(C)N=[N+]=[N-] c1(C(=O)NCC2CN(C(C(C)C(C)c3ccc(Cl)cc3)=O)C2)ccnc(O)c1F C1(NC(c2ccc(CC)cc2)=O)CC12CCN(C(=O)CCC1CCOCC1)C2 n1(CCOC)ccc2cc(C(N3CC(C)(NC(=O)CCCC(C)C)C3)=O)ccc12 O=C1CCC(C(=O)NCC2CCCN2C(c2cscn2)=O)CN1 C1(NC(COCC(=O)NC)=O)CCCC(C)C1.C1(C=O)CCC(=O)C1.N N1(CC)CCC(CN(C)C(C2CCCN2C(c2sccc2OC)=O)=O)C1 C1(C2CN(C(=O)C)C2)CC1.c1(CC)cccs1.C(C=O)N(C)C(=O)C1CC1 O=C(CCCCCc1cccs1)NCC1CCN1C(c1ncc(F)cn1)=O c1(CC)occc1C(N1CC(CNC(=O)C(C)(C)c2ccc(Cl)s2)C1)=O Cc1cc(Br)c2cc(C(N3CCCC(O)(CC(=O)OC(C)(C)C)C3)=O)[nH]c2c1 c1(C(=O)NCC2COCCN(C(c3ncn(CC)c3)=O)C2)cc(F)c(F)cc1F C1(NC(c2nc(C)sc2C)=O)CCN(C(=O)CCc2cccnc2F)C(C)C1 C(=O)(CCCC(=O)NCC)NC(C1CCOC1)CNC(C=CCC)=O C1(NC(C2N(C(C3(C(=O)OCC)CC3)=O)C2)=O)C(O)CC1O n1(C(C)C)c(O)nc(N2CC(=C(F)CNC(C3CNC(=O)N3)=O)C2)cc1=O N1(C(CNC(C2CC=CCO2)=O)=O)CCCCC1C(F)F C1(NC(CNC(C(C)(C)C)=O)=O)CC2(CCN(C(C3CCCC3)=O)CC2)C1.C N1(C(C2NCCN(C(C3N(C)CCC3)=O)C2)=O)C2CCC1CC1(C2)OCCO1 C1COC(C)(C)CN1C(c1ncc(F)cc1C)=O.C(C=CC(=O)N)(CC)=CC n1(C(C)C2CC2)nc(-c2ccc(-c3ccco3)cc2)nc1C1CCCc2c[nH]nc21 c1(C(=O)NC2CN(C(C3CC(C)(C)C3)=O)CC2(C)C)ccc(Cl)c(C#N)c1 c1(C(=O)NC(Cc2cn[nH]c2)C(=O)NCc2cnco2)ccc(O)cc1 C1(NC(C2C(OC)C2)=O)CC2CCC(C1C)N2C(C1(C2CCCO2)CCC1)=O C1(NC(C(CC=C)NC(=O)C(CC)=CC)=O)CCC2(CCC2)CC1 C(=O)(CC(C)(C)CC(=O)N)OCC.C(=O)CC(C)CN(C)C.C1CC(F)C1 CON1CCC(CC(=O)NCC2(C)CCN(C(c3cc(N)cnc3C)=O)C2)CC1 c1(OC)ccc(C(=O)N(C2CCCN(C(=O)CN(C3CCC3)C)C2)C)c(F)c1 c1(C(N(C2C(C)CCN(C(c3c(C)nccn3)=O)C2)C)=O)coc2c1CCCC2 Cc1ccncc1C(=O)NCC1CCC1NC(c1c(Br)cnn1C)=O C(=O)(C(C)CN(C)C(c1ncn(CC)n1)=O)N(CCC)C c1(C(=O)NC(C)(C)CC=CC(=O)NC2CCC3(CCC3)C2)ccc2cccnn12 c1(NCC(=C)F)ccc(S(=O)(=O)NCC2(CSC)CCC2)c(Br)c1 Cc1cc(F)c(C(N2CC3CC(C2)C3NC(=O)CC2C(C)C2(F)F)=O)cc1F Cc1cc(CNC(=O)C(CC2(C)CC2)c2ccccc2)sc1C C(C)(c1cccnc1)=CC(=O)N(C1CCC1)C.C1(C(=O)N)CC1.C1CCC1 C#CC1(C(=O)N(C2(CC(=O)NCC(C)(C)n3cccn3)CC2)C)CC(=O)C1 C1(C(=O)OCCC2CCC2)COc2cc(O)ccc2C1 CCC(C)C(O)C(C)C(=O)NCCC1CCCCN1C(=O)C1=COCC1 N1(c2nc(C)nc(C)c2F)CCC2C(CCCN2C(c2[nH]c(C)c(C)c2C)=O)C1 c1(C(C(N2C(CNC(C(F)=CCC)=O)C=CC2)=O)CC)ccc2c(c1)OCO2 C12(C(CNC(C(Cn3cccn3)N(C)C)=O)O)CC3CC(CC(C3)C1)C2 c1(C(N(C2CCCC(N(C(=O)CCC3CC3)C)C2)C)=O)ccc2c(n1)NCCO2 C1(CC(=O)NC)CN(C(c2cnc(O)c(C)c2)=O)CCN1C(C1C=CCCC1)=O C1(C(=O)NC(CNC(c2cccc(N(C)C)n2)=O)C(C)(C)C)CCC=CCCC1 O=S(=O)(Oc1ccc(C(F)(F)F)cc1F)c1ccc(Br)cc1 CCCC(C(=O)NC(CO)C(=O)NCCOCCN=[N+]=[N-])C(C)C Cc1cc2[nH]c(C(=O)NCCC3CC(NC(=O)Cc4cnns4)C3)cc2s1 c1(C(=O)NCC2CCCCN(C(c3n(C)nc(O)c3)=O)C2)cccc2nncn12 CN1CCC(=CC(=O)NC2CCC(N(C(=O)Cc3ccnn3C)C)CC2)CC1 C(C)(CCC(=O)NC(C)CC(=O)NCC1(C(=O)NC)CCCCC1)OCC O=S(=O)(c1ccc(NCC2CCSCC2)c(F)c1)NC1CCC1O c1(C(=O)OCC)cc(N2CCC(C)CC2)nc(C)n1.C(=O)C(C)CCN(C)C O=S(=O)(c1ccc(Cl)cc1)NCC1CCCN(c2ncnn3cc(Br)cc23)C1 C(=O)(CCS(=O)(=O)c1ccc(Cl)cc1)NCC(C(C)(C)C)NC(CCC#C)=O C(C)(C)(C(=O)NC1(CNCc2ccnn2C(C)C)COC1)OCC Cc1c(C(N2CC(NC(C3C4C5CCC(C5)C34)=O)C(C)C2)=O)c[nH]c2nccc1-2 c1(OC)cc(NCC2CC(NC(c3ccsc3Cl)=O)C2)nc(OC)n1 c1(C(=O)NC2C(CC(=O)N(C3CCN(C)C3)CC)CCC2)cc(O)nn1C N#Cc1sccc1C(N1CCN(CCNC(C2CCOC2C(F)(F)F)=O)CC1)=O CCCCCC(CC)C(=O)NC1CCC(C)(NC(C2CC(F)(CO)C2)=O)CC1 c1(CC)cn2c(n1)CC(C(=O)NCCC)CC2.c1(C(C(=O)N)C)ccc(F)cc1 C=CCC(C)(C)CCNC(=O)CC(O)CNC(C1COCC(C)O1)=O n1(CC)cnc2c(NC(C)CN3CCCCC3)nc(N3CCC(CC#N)C3)nc12 Cc1nc2nccc(C(=O)NCC3CCCC3)n2n1.C1(C=O)(C(C)C)CCC1.N N(C(=NCCC(=O)N(C)C)NCC1(C)CC1(Cl)Cl)C(COC)C c1(NC(C2C3CN(C(c4c(C)nn(C)c4C)=O)CC32)=O)ccc(Br)cc1[N+](=O)[O-] N1(C(C(C(C)C)CNC(=O)CC2CC2(C)C)=O)CC2C=CCC(C2)C1 CCN=C(NCc1ccc(OCCOC)cc1)N1CCC2OCCCC2C1 N1(C(C(F)OC)=O)CC(C)(C)CC1C.c1(C(=O)N)cccc(F)c1C(C)C N1(C(=O)Cc2c[nH]nc2O)CCC(CO)(CNC(C2CC2C2CCCC2)=O)CC1 N1(C(c2nc(CC)oc2)=O)CC(NC(=O)C(CC)OC)C(c2cnn(C)c2)C1 c1(NC2C(C)CC2)ccc(S(=O)(=O)NCCc2nncn2C)c(Cl)c1 N1(C(c2cncc(COC)c2)=O)CC23CCCCC2(C1)CN(C(=O)C(F)OC)C3 N1(C(CCC(=O)N(C)C)=O)CCC(C(N2CCC(C3(C)N=N3)C2)=O)C1(C)C C1(NC(CSCCOC)=O)CC2CC1CO2.c1(CCC=O)c(C)n[nH]c1C.C c1(C(N(CC(C)N(C)C(C2CCn3nccc3C2)=O)C)=O)ccc2[nH]ccc2n1 C1(NC(c2ccc(CC)o2)=O)CCC(N(C(=O)CCc2cc(C)sc2C)C)CC1 C1(C(N2CC(COC)C2)=O)CC2(CCC(F)(F)CC2)C1.C(=O)(C)N.CCF Cc1onc(Br)c1C(=O)NC1(CO)CN(C(C2CC3C=CC2C3)=O)C1 N1(C(CCOCCC)=O)CCCCC12CC(NC(c1nc(SC)ncc1N)=O)C2 Cc1noc(C(N2CCCC(NC(=O)CCCc3cnn[nH]3)C2)=O)c1C N1(C(=O)CC2CCC(O)C2)CCOC2(C1)CN(C(=O)CCc1nc(O)n[nH]1)C2 O=C1CC(C(=O)NC2CN(C(=O)C3=NOC4(CCOC4)C3)C2)c2ccccc2N1 c1(C(C)NCCSC2(C)CC2)ccnc(C(F)F)c1 C(=O)(CS(C)(=O)=O)NC1CC(NC(c2cc(-c3ccn(C)n3)on2)=O)C1 CCCCCC=CCC(=O)NCCCNC(=O)CCc1ccccc1.C(N)(=O)N C(=O)(C1=CCN(C(=O)CC2CCC(=O)N2C)CC1)NCCN1CC(C)OCC1 c1(C(=O)OCC)ccnc(NC(C2COCCN2C(=O)C(C)=O)=O)c1 Cc1cn2c(n1)CN(C(=O)NC1(Cc3ccccc3)CC1)CC2 C(=O)(C(C)CC(C)(C)C)N1CC(C(=O)NCCCC)C(C)(C)C1 C#CCC(C)(C)C(=O)NCC(C)(CC)NC(c1cc(F)cc(Br)c1)=O C1(CCOC)CCCC1NC(C1(N(C)C(C2(Cl)CC2)=O)CC1)=O c1(C(N(C)CCNC(c2cnn(C(C)(C)C)c2)=O)=O)cccc2sccc12 C1(NC(CCCn2c(C)ncc2)=O)CC2CCC1N(C(c1ccc(N)cn1)=O)C2 C1(CCC)(NC(=O)C2=CC(C)CC2)CCCN(C(=O)C(C)C)C1 CON(CCC(=O)N1CCCC(C)CC1)C(=O)C1CCN(C)C(=O)C1 C1(OC)CN(C(c2cc(=O)cc[nH]2)=O)CC1.C1(C=O)CCC(=O)N1C(C)C.N Cc1ccc(C(N2CCCC2(C(=O)NC(c2nc[nH]n2)C)C(C)C)=O)c(C)n1 Cc1c(C(=O)NCCC(C)NC(c2nncs2)=O)oc2c(F)cccc12 C1(C(N2CC(N(C(c3cc(CCC)[nH]n3)=O)C)C2)=O)CCCC(O)C1 c1(C=O)cc2scnc2[nH]1.C1(NC(C2CCN(C(CC)=O)C2)=O)CC2(C1)CC2.N N1(C(C(C(CC)C)O)=O)CCCC2CN(c3nn4cc(C)nc4s3)CC12 C(=O)(CCC(=O)NC(C1(O)CCCCC1)C(=O)NCC(O)C1(Cl)CC1)NC C(=O)(CCC(F)(F)F)N(C1CCN(C(C2CCC(=O)N2)=O)CC1)C n1(CC)cc(C2OCCC2C(=O)NCCCCC)cn1.C(=O)(C=CC1CC1)N Cc1cc(CCC(=O)NC(C)CCN(C(=O)CC2CCOC2)C)no1 c1ccc2c(c1)OCO2.c1(C2(CNC(=O)NCCO)CC2)ccc(Cl)cc1 CC1CN(C(c2cccc(F)n2)=O)CCC1CNC(=O)CCn1cncn1 C(=O)(C(C)CSC)NCCCCN(CCCNC(CCC)=O)C c1(OC)cc(OC)[nH]c(=NCC(C2CC2)NC(=O)C(c2c(C)noc2C)C)n1 c1(CNC(C(C)(C2CCC2)NC(=O)CC2CCCC2O)=O)cncc(F)c1 c1(C(CC)C(=O)NC2CC(N(C)C(c3ccsc3CC)=O)C2)ccc(OC)cc1 C(=O)(C1OCCn2ccnc21)NC(C(C)NC(=O)CCCn1cncn1)CO c1(OC)cc(O)c(CNC2CC(C(=O)NC(c3cccnc3)C)C2)c(Br)c1 c1(N2CCCC(c3n[nH]c(=N)o3)C2)cc(F)c(N)cc1F C1(C(=O)NCC2(NC(c3[nH]n(C)c(=O)n3)=O)CCOCC2)C2CCCCCCC12 C=CCN=C(NCCc1cnccc1C)NCc1cccs1 Cc1cccc(CC(C)NC(N2CCOC(CNC(N)=O)C2)=O)c1 CCS(=O)(=O)c1ccc(C(N2CCN(c3cnccn3)C(C)C2)=O)cc1C Cc1cc(C(=O)NC(C)(CNC(=O)C(C(C)C)C2CCC2)C2CC2)ncc1 C(CO)(CCCCNC(=O)CCC(C)(F)F)NC(Cc1ccc(CCC)cc1)=O C1(C(C)C)CCN(C(=O)CN(CC(C)(C)C)C)CC1.C1(CC(=O)N)CCCC1O c1(NC(=O)OC(C)(C)C)ccc(-c2nnc(-c3cccc(Br)c3)o2)c(O)c1 C=CC1(C(=O)NCC2CC2NC(c2cc(C)n(C)n2)=O)CCOCC1 C(=O)(C1=CCCOCC1)NCCCNC(CCOC(CC(C)C)C)=O CC(C)C(F)(F)CCNC(=O)N(c1ccc(I)cc1)C C(CCCC(C)(F)F)(C(=O)NCc1cccc(Cl)c1)N1CCN(CC#C)C(=O)C1 CC1CC(C(=O)N(CCCNC(=O)Cc2cccc(Br)c2)C)CC(C)C1 CC1CCN(CC(=O)NCC(c2ccccc2)CNC(=O)CC(Cl)Cl)C1 c1(C(N2CC(N(C(c3c(COC)cc[nH]3)=O)C)C(O)C2)=O)cc2cccnc2o1 C1(CNC(C(C)OCC=C)=O)CCC(O)C1.c1(C=O)ccccc1.CC=C CC(C)C(C(=O)NC1CN(C(C2C=CCC2)=O)CC1C)N(C)C Cc1cc(OCC(=O)NC(C)CCCNC(c2nocc2C)=O)ccc1Cl N#CC1CCC2(CCOCC2)C1NC(=O)CCSc1ccc(F)c(F)c1 c1(CC)ccc(C=CC(=O)NC2CCC2)o1.N(S(=O)(=O)NC)CC=O.C c1(OC)cscc1CC(=O)NC1(CCNC(=O)C=Cc2ccco2)CC1 N1(C(CCc2cc(C)no2)=O)CCCC(C(=O)NCC(O)C(C)(C)O)CC1 Cc1cc(C(=O)NCC(C)(C)NC(=O)C=Cc2nccs2)oc1Br CCCC(C)CCNC(=O)C(C)(C)CN(C(=O)CCc1ccncc1)C C1(NC(=O)CCn2cnnn2)CCCN(C(C2CC(N(C)C)C2)=O)C1 N1(C(c2cn(CC=C)nc2)=O)CC2(NC(=O)CS(=O)(=O)NC)CCC1CC2 c1(C=O)cc2n(c1)CCCC2.n1(CCC)cc(C(=O)NC2CCC(C)C2)cn1.N Cc1sc(C(N2CCC(O)(CC)C2)=O)cc1S(N)(=O)=O.c1(C=O)cn(C)nn1.N C(C1=CCN(C(=O)C(F)(F)c2ccnn2C)CC1)NC(CN(C(C)=O)C)=O C(=O)(C1=C(C)CCC1)NCCC1(C)CCN(C(c2ccc(NC)cc2)=O)C1 c1(SC(C)C(=O)N(C2CN(C(c3c(Cl)cnn3C)=O)C2)C)c(F)cccc1F C(=O)(C#CC1(C)CCCO1)NCC1CC(Nc2ccnc(C(CC)C)n2)C1 Cc1cccc2c(C(=O)N(C3CCCN(C(=O)CCNC(N)=O)C3)C)nccc12 CCC(C)C(C)C(=O)NNC(=O)C1CC(n2cc(CC3(O)CCSC3)nn2)C1 C1(ONC(CN(C(=O)CCC2OCCO2)C(C)C)=O)CCC(O)C1O Cc1ccc(F)c(C(=O)NCCCC2CN(C(=O)Cn3nnc(C)n3)CCO2)c1 C1(CCOC)(NC(COC(CC)CC)=O)CCN(C(=O)C(=O)CC(C)C)CC1 C#Cc1ccc(C(N2CCC(C)C(CC(=O)NCC3(CC)CCCC3)C2)=O)cn1 N1(C(C)C(=O)NC2CCC(NC(C3CC(C)(C)C3)=O)C2)C(=O)CCC1=O n1(CC)nc(C)c([N+](=O)[O-])c1N.C1(C)(C(N2CCCC2)=O)CCCNS1(=O)=O N1(C(c2c(C)noc2)=O)CCN(C(=O)CC2CCCC(F)(F)C2)CC(C)(F)C1 c1(C(=O)NC2(C)CCN(C(C3ON=C(CC)C3)=O)CC2)cc(OC)c(O)cc1F Cc1cc(C(=O)NCC(C2CCN(C(C3CCCCN3C)=O)CC2)F)ccc1Cl C1(C(N(C2CN(C(C(C)NC(COC)=O)=O)C2)C)=O)CC(OC)C(OC)C1 CCCC(C)(O)CC(=O)N1CC(C(=O)NCCCc2cncnc2)C(CCC)C1 c1(C=O)cc(C(F)(F)F)n(C(F)F)n1.CC(C)CC.C1(C=O)CCS1(=O)=O C1(C(CNC(C2(COC)CC2)=O)(C)O)CCCN(C(c2ccc(Cl)o2)=O)C1 C1(CNC(COCCCCC)=O)C(C)CCCN1C(c1cc(F)cc(F)c1)=O C(=O)(C1=CCS(=O)(=O)C1)NC(C)C(C)(C)NC(=O)C1=NNC(=O)C1 Cc1cnc(NC(C2CC3(CC(NC)C3)C2)=O)c(C#N)c1.c1cc(C#N)ccn1 N1(C(c2cc(CC)[nH]n2)=O)C(C(=O)NC2(C(O)C)CC2)CCC1C1CC1 c1(SCC(N2C(CNC(c3c(CC)cco3)=O)CC2)=O)ccccc1Cl Cc1nc2c([nH]1)CC(C(=O)N(C)CCn1cc(CN3CCOCC3=O)nn1)CC2 c1(C(=O)NCC2(NC(C=C(CC)C)=O)CCOCC2)cc(F)ccc1F c1(OCCC)ccc(Nc2nc(N(CC(F)F)C)cc(C)n2)c(C)c1 N1(C(C)=O)CCC(C2CCC2)C1.c1(C=O)nc(C)sc1C.C(COCC)OC.O C(CC)(CCCC(=O)NC(c1cccnc1C)C)NC(C(CCC)C#N)=O N1(C(c2cc(C)nc(C)n2)=O)CCN(C(C2CC2C2CCC2)=O)C2(CCC2)C1 N1(C(C(COCC)(C)C)=O)CCCC(C2(NC(c3cnoc3)=O)CC2)C1 c1(CC(=O)N(CC(C)NC(=O)Cc2cnccc2Cl)CC)cccc(F)c1Cl c1(CCOC)nc(=NC=O)s[nH]1.C1(CC)CCCN(C(C)=O)C1.C1(C=O)CCC1 N1(C(CCC2(C)N(C(CCCOCC=C)=O)CCC2)=O)CCOC(C)(C)C1C C(=O)(C1CCSc2ccccc21)NCC1C(NC(CC2CCN(C)CC2)=O)C1 C(=O)(CCCCCc1cccs1)NC(CNC(CC1CC(OC)C1)=O)CCOC C=C(F)C1(CC(=O)NC)CCC1.C1CN(C(=O)C(C)(C)n2cnc(C)c2)CC1C N1(CC)CCC(C(N2CCC(C(=O)NC3(CN(C)C)CC3)C2C)=O)CC1 N1(CC=C)CCCC(CNC(c2nnc(C3CC3)s2)=O)C1 c1(OC)ccc(SCC(=O)N(CC(C)CNC(c2cc(C)no2)=O)C)cc1 N1(C(CCCSC)=O)CCN(C(=O)CCC2(C)CC2)CC1C1CCC1 CCC(CC)C(C)C(=O)NC1CCN(C(=O)Cc2ccc(C)cc2)CC1(C)C c1(C(=O)NC(CCOC)CNC(c2[nH]ccc2COC)=O)cc(Br)ccn1 c1(C(N2C(C(=O)Nc3cc(CO)ccn3)CC(F)C2)=O)c(Cl)ccc(Br)c1F Cc1sc(C(N2CCC(NC(C3CCN(C)S3(=O)=O)=O)C2)=O)cc1[N+](=O)[O-] c1(C(=O)NC2CC(NC(c3cnc(C)s3)=O)C2)cncc(S(C)(=O)=O)c1 CCCC(C(=O)NCC(O)C1CCC1)NC(c1cn(CCO)nn1)=O C1(NC(CCc2cc(C)no2)=O)CCCN(C(=O)CCC2(C)CC2)C1 C12CC3CCC(C1)N3c1cc(ncn1)NCC2.c1(C(C)O)n[nH]c(CO)n1 C1(CC=O)CC(C2CC2)C1.C1(CC(=O)NCCN(CC=C)C)CCC1O CCC(C)CCC(=O)N1CC(O)CC1C(=O)NC1CCC(CCO)CC1 N1(C(c2c(OC)ccnc2)=O)CCCN(C(=O)C2=CS(=O)CCC2)C(C(C)C)C1 C(=O)CCC(F)(F)F.c1c(O)cccc1C#N.CC(C)C.C1(C=O)CC1C=O.O C=Cc1cncc(C(N2CCOCC2CC(=O)NCC2CCCC3(CC3)C2)=O)c1 N1(C(C2C(C=C(C)C)C2(C)C)=O)CCCN(C(c2ccc(C#N)[nH]2)=O)C(C)C1 Cc1cnccc1C(=O)NCCC(C)(C)CNC(=O)Cc1csc(Cl)n1 Cc1nc(C(N2CC(C)(NC(c3ccc(CO)cc3F)=O)C2)=O)ccc1Br N(C(=NCCF)NC1CCCN(C(=O)OC(C)(C)C)CC1)CC(C)CN(C)C Cc1[nH]c(C)c(C(N2CCC(F)(CNC(=O)CCc3cnn(C)c3)C2)=O)c1C c1(C(N2C3CC(CNC(C(CC)(C)CO)=O)C2CC3)=O)cc2c(nn1)CCCC2 C(CC(C)(C)C)(C(=O)NCCCC(=O)NC(C)(C)C(O)C(F)F)OC C1(C(N2CCC(NC(=O)COC3CC3)(CO)C2)=O)CNC(=O)CC12CCC2 N1(C(c2cncs2)=O)CC2CC(C1)N(C(=O)C=Cc1ccc(C)o1)C2.CCO c1(C(N2CCC(NC(c3ccc(C(=O)OC)nc3)=O)C2)=O)cc(C)c(F)cc1Br c1(C(N2C3C(NC(C(COCC)C)=O)CC(C3)C2)=O)ccnc2c1CCC2 CCCC(C(=O)OC)C(=O)N1CCC(C)(CNC(=O)C(C)(C)OC(C)C)C1 N1(c2ccnc(NCC3NCCC3C3CC3)n2)CCCN(c2ccncc2)CC1 C#CCC(C(=O)NC(CC1CC1)CC1CC1)NC(=O)C(c1ccccc1)C C=CC(C)(CC)C(=O)NCc1cc(C(=O)NCC(C)(O)C(F)F)on1 C(=O)(C(C)(C)CO)N1CC(O)(CCNC(C(C2CCCCC2)N(C)C)=O)C1 C1(NC(=O)CN2C(=O)CCC2=O)CC2CCC1N2C(C1CCCCC1(F)F)=O C1(O)(CNC(CC(C)SC)=O)CCCN(C(C23CC(CO)(C2)OC3C)=O)C1 c1(CN2CC(NC(c3cccnc3CO)=O)C2)ccc(Cl)nc1Cl C=CCC(C)(C)C(=O)N(CCCNC(C1CCCC12CCC2)=O)C C(=O)(CCC#Cc1ccccc1)N1C(C)CC(NC(c2ccc(C#C)cc2)=O)C1 c1(C=O)cnc(O)c(Cl)c1.c1(CCC)ncoc1C(=O)NC(C)(C)C1CCC1 C1(CCNC(CCOCCC)=O)CN(C(c2cc(C)cs2)=O)CC(C)O1 n1(CC(N)=O)ccc(=NC(=O)C(CC(F)F)NC(c2cccs2)=O)[nH]1 CCCC(C)C(=O)N1CC(NC(c2cc(OC)ns2)=O)CC1C c1(C(=O)NC2C(OC)CN(C(C3CC3(C)C)=O)C2)cc(Cl)cc([N+](=O)[O-])c1O C(=O)(C(C)C(C)C)N(C1(C(=O)NCCc2cnc(C)s2)CC1)C C1(C=O)CCCCC12CC2.N1(C(CN(C=O)C)=O)CC(O)(C(C)(C)C)C1.CO c1(C=O)cc(O)ccc1F.n1(CC)cc(C(=O)NCC2CC2)c(C(C)C)n1 C1(C(=O)NCC(CC)NC(=O)CC(C)(C)CC(F)F)COc2cc(F)ccc2C1 N1(C(c2nn(CC)c(O)c2)=O)CCCC(NC(c2cnn(C)c2N)=O)CC1 C(C(C)C(C)C(=O)N1CCC(C2CCCN2c2ncncc2Br)C1)OC CC1CCCC1C(=O)N(C)CCNC(c1cscc1C(F)(F)F)=O C1(C(N(C)CCc2cnccn2)=O)CCN(C(C2CC23CCOC3)=O)CC1 C=CCC(C(=O)NC(C1(C(N2CCCCC2CC)=O)CC1)C)C(C)C N(C(=NCCCCl)NCC1CC1)CC(=O)NC(c1ccc(N(C)C)nc1)C.C N1(C(c2ccc(COC)cc2)=O)CCC(NC(=O)C=CC(C)(C)S)CC1C C=CCCCCCCC(=O)N1CCN(C(=O)C(C#N)CCC)CC1c1cn[nH]c1 CCCCCC(O)C(=O)N1CCC(O)(CNC(=O)Cc2sccc2Cl)C1 C1(C(=O)NC(C=C)(C)C)CC(N=[N+]=[N-])CN1C(c1ccnc(C)c1C)=O Cc1ncc(Cn2cc(CN3CCCC3=O)nn2)c(O)n1 C=C(Br)CC(=O)N(CC(C)N(C)C(c1csc(Br)c1)=O)C C12(NC(C3CC(C)(C)C3)=O)CCCC1N(C(=O)CSC(C)(C)C)CCC2 N1(C(C(n2cc(C)nc2)(C)C)=O)CCC(C)(C)C1.C1(C(=O)N)CC(=O)C1(C)C c1(C2CC(=O)C2)ccc(CC2CCN(C(=O)CN3CCC(F)(F)C3)C2)cc1 N1(C(CCc2cccc(OC)c2)=O)CCN(C(=O)CCn2ccnn2)CC1CF c1(C(=O)NC(C2CCN(C(C(CSC)O)=O)CC2)C)cc2ccc(F)cc2s1 C1(C(=O)NCC(CC)OC)CC2(CC(NC(c3cscc3C)=O)C2)C1 c1(OC(C)C)ccc(CC(N2CCC(N(C3CCN(C)C3=O)C)CC2)=O)cc1 C=CCCCC(=O)NC1CCCCC1NC(=O)COC(C)CC N1(C(CC(CN(C)C)O)=O)CC2CC(NC(c3cc(C4(C)CC4)n[nH]3)=O)C2C1 N1(C(Cc2n(C)ncc2Cl)=O)CC2CCCCC2(CNC(=O)CO)C1.C1CC1 N1(C(c2nn(CC)nc2C)=O)CCC(C)N(C(=O)C(c2csc(C)n2)=O)CC1 C1(OC)CN(C(=O)CCc2cn(C)cn2)CC1NC(=O)CC1CC(OC)C1 C(=O)(C1CCCn2nccc21)NC1CC(C)(NC(c2cccc(F)c2F)=O)C1 Nc1cc(C(=O)NC23CCC(CN(C(C4(F)CC4)=O)C2)C3)c(F)cc1F CON=Cc1ccc(C(N2CC(NC(=O)CC(C)C(C)C)CC(F)(F)C2)=O)cc1 C1(NC(c2nnn(CC)c2C)=O)CC12CCN(C(C1COCCN1C=O)=O)C2 C(=O)(C(CC)NC(C1(CF)CC(=O)C1)=O)N(C1CC(OC)C1)C C1(COC)CCN(Cc2cn(CCN(C)CCO)nn2)CC1 Cc1snnc1C(N1CCC1(C)CC(=O)NCCN(C(C)C)C(C)C)=O CCC(COC)(CC)C(=O)NCc1nocc1C(=O)N(C)C(C)C1CC1 C(=O)(C(C)(C)CCNC(=O)C(C)CO)N1CC2(C(C(=O)OC)C2)C1 C1(CNC(c2ccn(C)n2)=O)CC(O)CN1C(=O)CCc1ccoc1 Cc1cn2c(n1)CCC(NC(C(C)(C)C(C)(F)F)c1nnnn1C1COC1)C2 C1(NC(c2nc(I)cs2)=O)CCN(c2ncccn2)CC1 N1(C(c2cc(CCC)on2)=O)CC(NC(C2(C)CC2(F)F)=O)CC1C C1(N(C)C(c2cccn2C)=O)CCCC(NC(c2ccc(O)nn2)=O)C1 C1(C(=O)NC(c2cc(C)no2)(C)C)CC2CCC1N2C(c1ncn2c1CCC2)=O C1(C(C)=O)C(C(=O)NCc2nc(C(=O)NCCN=[N+]=[N-])co2)C1(C)C C(=O)(CC(C)(C)C(F)F)NC1CCN(C(c2cncc(C)n2)=O)C(C)C1 C(=O)(C1=C2CCCN=C2NN1)NCCC(CNC(CCc1n(C)ccn1)=O)(C)C CC1CC(C)(C(N2CC(=C(F)CNC(c3cnccc3Cl)=O)C2)=O)CCO1 CCCCCS(=O)(=O)CC(=O)NCC(C)NC(c1cn(C)nc1-c1nccs1)=O c1(OCC)ccc(F)c(C(N2CCOC(C)C2)=O)c1F.c1(C=O)ccn(C)c1.N Cc1[nH]c2ccccc2c1CC(=O)NC1CC(C)CN(C(=O)Cc2cn[nH]c2)C1 CC1CN2CCN1CC2C(=O)NC1(C2CCN(C(=O)COc3ccsc3)C2)CC1 Cn1c(NC(=O)Cn2nnn(C3CC3)c2=O)nc2cc(Br)c(Cl)cc12 c1(C(=O)NC(C)C(C)NC(c2ccc(Cl)cc2)=O)nn(C)c2ccccc12 C1(C(=O)NCC(C2CCC2)NC(=O)COCCCF)(CN(C)C)CC1 Cc1ccc2cc(C(=O)NCC(F)CNC(C3(C)CCN(C)C3)=O)ccc2n1 N1(C(C2CC(CC)C2)=O)CCC(C)(C(=O)NCC2CCNC(=O)C2)CC1 c1(C(N2CCC(C(=O)NCC3CC3(Cl)Cl)(CF)C2)=O)cc2occc2[nH]1 C1(CNC(=O)C2=CCC2)CCN(C(c2cn(CC3CC3)nn2)=O)CCC1(F)F C12(C(=O)NCC(CN(C(CC3CCCC(OC)C3)=O)C)C)CCC(CC1)CC2 N1(C(C)=O)CC2CC(C1)CN(C(=O)CCC(=O)Nc1sccc1C(N)=O)C2 C1(C)(OC)CC(N(C(=O)C(F)(F)CCn2cc(CC(C)C)nn2)C)C1(C)C C=CC(F)(F)C(=O)NC1CC(C)N(C(=O)CCCNC(C)=O)C1 N1(C(C(C)(C)C2CC2)=O)CCCC(O)(CNC(=O)CCP(C)(C)=O)C1 c1cc2c(NCC3CCCS3)[nH]c(=NCc3nc(C4CC4)cs3)nc2s1 C1(C(=O)NC2CC(N(C(=O)CC(F)F)C)C2)CCCCN1C C(CCCC(F)(F)F)NC(C1(C)CCN(C(=O)CCN=[N+]=[N-])C1)=O CCCC(C(=O)NCC12CC1CN(C(c1snnc1C)=O)C2)NC(C)=O N1(C(CC(CNC(C(C=C)O)=O)C)=O)CCC2CC1C(=O)O2 C1(CC(=O)NC(C=CC(=O)N(CCCCO)CC)C)CCCOC1 C(=O)(C1=CCCCC1)N(CC(CC)NC(C1CCN(CC)C1)=O)C N1(C(C(C=C)(C)C)=O)CCC2CC(NC(=O)C3CCCc4c[nH]nc43)CCC2C1 C1(N(C)CC)CCN(N2CCC(CC(=O)NC)CC2)C1 CCC(C)(C(=O)NCC1CC(C)(C)CN1C(=O)C=Cc1ccco1)C(F)F N1(C(CNC(C)=O)=O)CCN(C(=O)CC2(N(C)C)COC2)C(C2CCCC2)C1 c1(OC)ccc(C)cc1-c1cn(C(C)C(=O)NCC23CC2(C)C3)nn1 C(=O)(CCCCC(C)C)N1CC(CC)C(C(=O)NC2CCC(C(C)O)CC2)C1 c1(C(=O)N)ccc(O)c(Cl)n1.c1(CCCCC)cc(C(=O)NCC2CC2)n[nH]1 c1(C(=O)NC2(CC=C)CN(C(C(C#C)(C)C)=O)C2)ccc2cc(F)c(F)cc2n1 C12(C(N3C(Cc4cn(-c5ccc(C)cc5)nn4)CCC3)=O)CCCC1OCC2 C=CCCC(C(=O)OC)NC(=O)CC1CCN1C(=O)C(n1nccc1C)C C1(O)(C(N(C(C)CNC(c2cnc(S)n2C)=O)CC)=O)CN2CCC1CC2 C=C(C)CC(C(=O)N)NC(=O)C(C)OCCOC.C1(CC)CCC(C)(C)C1 CCCC(C(O)C(=O)NCC12COC(C1)C(O)C2)NC(=O)Cc1cc[nH]n1 CCCC(C#N)C(=O)NCC1C2CN(C(=O)CCn3ccnn3)CC12 c1(SC)ccc(NC(c2cnc(C(C)O)s2)=O)cn1 C(=O)(C(CO)C(C)(C)C)N1C(CC(N2CC3C(CC)C3C2)=O)CC(O)C1 c1(C(N2CCC3(CCCN3C(C3CC3F)=O)CC2)=O)ccnc2ccc(F)cc12 N1(C(C(N2CCC(N(C(=O)C(=O)N)CC)C2)=O)=O)CCCC(C)C1.C1CC1 c1(C(C(N2CC3C(CNC(C(C)(C)CO)=O)(C3)C2)=O)O)cccc2c1OCC2 CC1CC(CNC(=O)CCCC#N)CN1C(=O)C=Cc1ccccc1 C1(CNC(c2c(CC)cccn2)=O)CN(C(=O)C(CO)C(C)C)CC(C)(C)C1 CC(C(C)(C)C)NC(=O)C(Cc1ccoc1)NC(=O)C=Cc1ccoc1 c1(NC(C2C3(CCN(Cc4cc(C)cc(Cl)c4)C3)C2)=O)cc(Br)ccc1[N+](=O)[O-] CC1CCC(C)(NC(C2CC=CCN2C(c2cnn(CCF)c2)=O)=O)C1 C(=O)(C(C)CC(=O)NC(C1CCN(C(=O)CC2OCCC2(C)C)C1)C)OC C(=O)(CC(C(=O)NCc1ccccc1)C1CC(c2ccccc2)(C(F)F)C1)OC c1(C(N2CCC(F)(CNC(C(C)SC)=O)C2)=O)cnc2nc(Cl)ccc2c1 C1(C(=O)NCc2ncc(C)s2)CC2CC2N1Cc1cnc(N2CCCC2)s1 CN(CCCC(=O)N1CCCCC1CCNC(c1n[nH]c2cccnc12)=O)N=O c1(C(N2CCC(NC(=O)CSC3CCCCO3)C2)=O)ccccc1OC(F)F N1(C(CSCC=C)=O)CC(NC(c2ccc(-n3cncn3)cc2)=O)CC(F)C1 c1(C(=O)NCC2CCN(C(CC(=O)OCC)=O)C(C)C2)cncc2nc(O)[nH]c12 N1(C(C2(NC(=O)C(=O)NCC(F)F)C(C)(C)C2)=O)CCc2sccc2C1 N1(C(C(CCCC)F)=O)CCC2(CCCCN(C(c3cc(C)ns3)=O)C2)C1 c1(C(N(CCCN2CCCOC(C)C2)CC)=O)cc(=NCCc2cccs2)[nH][nH]1 C1(NC(c2ccc(C)nc2)=O)CN(C(=O)CSC2CCOC2=O)CCC1CO c1(C=O)ccc2c[nH]nc2c1.c1(SCC(=O)NCC2CC2)cccc(F)c1.C c1(Nc2scc(C(=O)NCCN(CC(C)C)CC)n2)cncc(O)c1 C1(CC(=O)OCC)(C(N2CCC2C)=O)CCCC1.C(=O)CC.C(N)=O C1(C(=O)NC2CC(n3cc(COCCN(C)C)nn3)C2)CCCC12CCOCC2 Cn1nc(CNC(=O)CC2(O)CC2)c2c1CCN(C(C1CC1F)=O)C2 Cc1nc2ccc(C(=O)NC3(C)CCN(C(=O)C(O)C4CC4)C3)cc2o1 CC(C)CC(CNC(c1ncc[nH]c1=O)=O)NC(=O)C(C)CC1CCCC1 O=S(=O)(c1ccc(NCC2(F)CCC2)c(Br)c1)N1CCOC(C(F)(F)F)CC1 c1(NC(=O)NC2CCC(CCC(C)C)C2)cccc(-c2cnco2)c1 CN1CCN(C(c2c[nH]c(=S)cn2)=O)CC1CNC(=O)CC1CCCC12CC2 C(C)(C)(C(C)C)NC(c1c(C)cno1)=O.C(=O)(CC)N.C(C)(C)C.C=O c1(C(=O)NCC(C)CNC(C2CCC3CCCCN23)=O)coc2ccccc12 C1(C(=O)OC)CCCN(C(C2CCCSC2)C(=O)Nc2ccc(OC)cc2)CC1 c1(C(=O)N)cnc2c(cnn2C)c1.[SH](=O)(=O)c1cccs1.C(=O)(C)N(C)CC Cn1nc(C(=O)NCC23CC2CN(C(=O)CCc2ccc(O)cc2)C3)cc1Cl C1(NC(=O)Cc2cncs2)COC2(C1)CN(C(=O)C=Cc1cncc(F)c1)C2 C(=O)CS(=O)(=O)N(C)C.c1(CN2CC(O)(CC)C2)cc(C(C)(C)C)on1 C1(C(=O)NC(C(C)OC)C)(NC(C2(c3cccnc3)CCC2)=O)CCCC1 CCCCCC(C)(C)C(=O)NC1CCCC(NC(=O)CNS(=O)(=O)CCCC)C1 N1(C(C2N(C)CCC2)=O)CCCC(C2(NC(=O)CC3CC(=O)NC3=O)CC2)C1 c1(OC)cc(F)c(CN2CCOC(CCC(=O)O)C2)cc1Cl C1(CNC(C2(OCC)CCCC2)=O)CN(C(=O)C=C(Cl)Cl)C2CC12 Cc1cccc(NC(=O)C=CC(C)(C)NC(=O)C(N2CCNC2=O)C)c1 C1(C(F)(F)F)(C(N(C2CN(Cc3ccccc3Br)C2)C)=O)CCC(=O)CC1 C(=O)(C1=CC2C=CC1C2)NC1(C)CC(NC(C2CCCCS2)=O)C1 n1(CC)cnc2c(N3CCCCC(NC(c4cccc[n+]4[O-])=O)C3)nc(Cl)nc12 N1(C(c2ccccc2)Cc2cccc(OC3CC3)c2)CCOc2ccccc21 C1(N(C(=O)COC(C)C)CC)CCCN(C(c2csc(C(F)F)n2)=O)C1 c1(C(=O)NCCC2CC(NC(c3cccs3)=O)C2)cn(C2CCOC2)nn1 N1(C(C(C(CNC(C2(C=C)CCCC2)=O)C)F)=O)CCCC2C(O)CC12 N1(C(C2(CC)CCN(C(=O)CC3(C)CCOC3)CC2)=O)CC2CCCCCCC12 C1(NC(c2cnnn2C(F)F)=O)CCCN(C(=O)COc2ccccc2)C1 c1(OC)cc(F)c(C(=O)N)c(Cl)c1.C1(C=O)CNC(=O)CC1C.C1(CC)CC1 c1(-n2c(C)cc(C(N3CC4CC(c5ccccc5)CC34)=O)n2)cn2ccsc2n1 Cc1noc(C)c1NC(C1CCC(C2CC2)N1C(c1cc(Cl)no1)=O)=O C(CC(C(=O)NC(COCC)C(C)C)NC(c1ccc(O)cn1)=O)=CC C(=O)(CC1NC(=O)c2ccccc21)N(CCNC(=O)C(C)CCOC)CC c1(NCCCC)ccccc1C(N1CCC(NC(=O)C(C)(C2CC2)SC)C1)=O CC(C)(C)CCC(=O)NC1CCCC1NC(=O)C(CC1CCCCC1)C1CCC1 c1(C(N2CC(C)(C)C(c3ccc(F)cc3)C2)=O)cc2n(n1)CCNC2=O c1(CC(=O)NCC(O)CCNC(=O)Cc2cnns2)c[nH]c2ncccc12 CC(C)CC(C)CC(=O)NC(c1ccccc1)CNC(=O)CC1C=CCC1 C(CCCC(C)NC(=O)CSCC(C)C)NC(C1CN(C(=O)NC)C1)=O C1(NC(c2n(CC=C)ccn2)=O)CN(C(=O)Cc2ccccn2)CC2(CC2)C1 C(=O)(NNC(=O)NC1(O)CCCCC1)NC1CCC(C)C1 CC1(C)CCN(C(c2[nH]c(=N)sc2C(F)(F)F)=O)C1.c1(C(=O)N)c[nH]nc1F c1(N2CCOCC(NCc3c(C)c(Br)ccc3)C2)ncc2sccc2n1 Cc1cccc(Cl)c1C(=O)NC(C)CCCNC(=O)CO.c1(CC)cccs1 c1(C=O)ccc2c(c1)CC(C)O2.C(CC)(C(=O)N(C)CCO)OCC.CCC c1(C(N2C(CCNC(C3C(C=C)C3)=O)CSCC2)=O)cc(OC)cc(OC)c1 N1(CC(C)C)CCN(C(=O)NCCc2ccc(NS(C)(=O)=O)cc2)CC1 Cc1ccc(C(N2CCCCC(NC(C3(N(C)C)CC3)=O)C2)=O)c(F)c1Cl Cc1cc[nH]c1C(=O)NC1CCC1CNC(c1cn(C(C)(C)C)nn1)=O C1(NC(CCS(N)(=O)=O)=O)CCCC12CN(C(C1(c3cccc(Cl)c3)CC1)=O)C2 C1(C2CCN(C(=O)CN3CCC3)CC2)(NC(=O)C=CC2CCOCC2)CC1 C1(CCNC(C2(CCCC)CCC2)=O)CN(C(=O)Cc2nccn2C)CCCO1 C=CC(C)C(C)C(=O)NCC1CCC1.n1(CC=O)cc(C(F)(F)F)nn1.N CCC(CCC(=O)N1CCCC(CCNC(C2CCCC(O)C2)=O)C1)OC C1(N(C(=O)CCOC2CCCCC2)CCC)CCN(C(c2ccnc(C)n2)=O)CC1 O1NC(=O)C=CC(C)NC(=O)C1.N1(C(C)C)CC(CF)C1 C1(C(=O)NCCc2ccns2)(NC(=O)Cn2ncnn2)CC(F)(F)C1 C(=O)(CC1NC(=O)c2ccccc21)NC(C(C)NC(C(CCC)(C)C)=O)C Cc1[nH]c(=N)nc(O)c1CC(=O)NCC1CCCN1C(C1CCC2CC2C1)=O N(C1CCCc2cc(CNC(C3CCCCC3O)=O)ccc21)C(C=CC=CC)=O C1(C(=O)NCCCC(=C)C)CCC(C)CN1C(=O)C(F)CCCC c1(C(N2CCC(N(C(c3occ(C)c3)=O)C)C2)=O)ccc(C2=CCCC2)cc1 CC1CCN(C(=O)CCCc2ccc(O)c(F)c2)CC1NC(c1cn(C)cn1)=O c1(C(=O)NC2CC(CNC(CC(C)O)=O)CC2O)cnc2n1CCOC2 CC(C)(C)C(C)(C)O.Cn1nnc(C)c1C=O.c1(C=O)cnnn1C1CC1.N c1(CC)cc(NC(c2nc3ccccc3s2)C)n2ncnc2n1 C1(NC(c2ccc(CC)o2)=O)CC(NC(c2cnncc2OC)=O)CC1O C1(NC(C2N(CC)CC2)=O)CN(C(=O)Cn2ncnn2)CCC12CCOCC2 n1(CC)ncnc1CC.C(=O)CCN(C(=O)CCC1(C)N=N1)C(C)C.N c1(C(N(CCOC)CC)=O)cc(Cl)cnc1.C1(CC=O)CC(C)(C)C1.N N1(c2nnn(C)n2)CCC2CCC(C1)N2C(c1cncc(C(C)(C)C)c1)=O C1(CNC(COc2c(C)cccc2)=O)CN(C(=O)CCC#N)CCC1C c1(C(N2CCN(C(C=C(C)Cl)=O)C(CO)C2)=O)ccc2c(c1F)CCC2 c1(C(=O)NC2(CF)CCN(C(c3cc(CCC)[nH]n3)=O)C2)ccc(F)c(Cl)c1F C(=O)(C(O)C(F)(F)F)NCCCN(C(CC(C)O)=O)CCO C(C(C)(O)CC(=O)N(CCC(N1CCC(CC(F)F)C1)=O)CCO)OC C=CCCCCCC(=O)NCC1(NC(c2nnc(Cl)cc2N)=O)CCC1 C1(C)(NC(C2N(C(=O)NC)CCC2)=O)CCCN(C(c2cccnn2)=O)C1 N1(C(CN(C(=O)OCC)C)=O)CC(NC(c2cccc[n+]2[O-])=O)CC(C)C1 C1(NC(c2cscc2C(F)F)=O)CC2CC1N(C(=O)C(c1ccc(F)cc1)O)C2 N1(C(c2[nH]c(CC)c(Cl)n2)=O)CCC2CCN(C(=O)C=Cc3cn[nH]c3)CC12 CS(=O)(=O)c1ccc(-c2nc(CCOC3CCCCC3)nn2C2CSC2)nc1 c1(C(N2CCC2C)=O)cc(Cl)cc(Cl)c1[N+](=O)[O-].C12(C=O)CCC(CC1)O2.N N1(C(c2cc(C)no2)=O)CC(C(=O)NC(c2cccnc2)CO)CC(C)C1 C(=O)(C(F)CC1CCOC1)N.C1(C(=O)NC2(CCC)CC2)CC1C(F)F N1(C(CCCC(=C)C)=O)CCC2(CC1)CC(NC(=O)C(C)(O)c1ccccc1)C2 C(CCCCC(=O)NCC=CCl)NC(Cn1ccc(C)n1)=O CC1CCC(=CC(=O)NCCC2CCCCN2C(C2C(C)C2(F)F)=O)CC1 CCCC(C(=O)NC(C)(C)CN1CCN(C(=O)CCC(C)CC)CC1)C(C)C c1(NC(c2n(CCSC)nnn2)C(C)(C)C)ccc(-n2cncn2)cc1 Cc1nonc1.C1(CC(=O)NCC=C(C=O)F)CCCC1.C(C)(C)C.C=O N1(C(C2ON=C(C)C2)=O)CCCC2(C1)CN(C(=O)CC1CCCCC(=O)N1)C2 c1(OC(C2CCC(c3ccccc3)O2)=O)ccc(C(N2CCOCC2)=O)cc1 N1(Cc2ccc(C(=O)OCC)o2)CCN(C(=O)C(c2ccccc2F)C)CC1 CC1=NOC(CC(N2CCC2(C)CC(=O)NC(C2CCCC2)C)=O)C1 C=CCC(C)(CC)C(=O)NCC1CC2(CC2)CN1C(c1nccc(C)c1N)=O CCCCCC(=O)NCC=CC(=O)NCC1CN(C(N)=O)C1 C(=O)(C(C)CS(C)(=O)=O)N(CCCCN(C(C(COC)COC)=O)C)C c1(OC)n[nH]c(C(=O)Nc2cccc(NC(C3(C4CCCO4)CC3)=O)c2)c1Cl c1(C(=O)NCCC2COCCN2C(c2ccco2)=O)cc(Cl)c2[nH]c(O)nc2c1 c1(C(N2CCC(NC(C=C(COC)C)=O)C(C)C2)=O)ccn2c1CSCC2 O=C1CS(=O)(=O)CC(C(=O)NC2CCN(Cc3ccc(Br)cc3)C2)N1 c1(C=O)cnc(N)c(N)c1.C1(NC(c2ccc(C(C)C)s2)=O)CC(C)C1(C)C Cc1cnc(F)c(NC(=O)C(=O)NCc2nc(CN(C)C)cs2)c1 C1(CC(C)NC(c2ncn(CC)c2)=O)CCN(C(=O)CC(C)OC)CC1 C(=O)(CCCCC(C)=O)NCCC(CNC(=O)CN1CCC(F)CC1)OC C(C)(C)(CC(=O)N1CCCC(C(C)NC(c2cnccn2)=O)C1)OC.C(C)C.O O=C1CCC(CCC(=O)NC2CC(NC(c3cc(Br)cnc3O)=O)C2)=NN1 C(CC(O)CNC(c1cc(C2CCOC2)[nH]n1)=O)NC(CCN(C)CC)=O C1(CN(C(c2c(C)csc2)=O)C)CCCC(NC(=O)C(=O)N(C)C)C1 C1(CN(C(=O)C(=Cc2c[nH]cn2)F)CC)CCN(C(C2CC2F)=O)CC1 C(=O)(CCC(=O)NC(C)CNC(c1scc(C)c1C)=O)OCC N1(C(C(C)S(N)(=O)=O)=O)CC2CCCC1C2.n1(CC=O)cnc(C(N)=O)n1.C C1(C(=O)NC2C(C)C2C)CC2(CCN(C(c3cccc(O)c3)=O)C2)C1 C1(C(=O)NCC(c2ccccc2F)N2CCOCC2)CC2CC1CC2(F)F N1(C(C(CCOCCO)NC(=O)C2=CCSC2)=O)CC2CCC(C1)C(=O)O2 c1(CC)ccccc1-c1ccccc1C(N(C(C)C)Cc1cnccn1)=O Cc1cnc(C(=O)NCCCOCCC(=O)NCC(F)Br)c[n+]1[O-] C(=O)(C1=NN(CCO)C(=O)CC1)N1CCN(C(c2c(OC)cccn2)=O)C2C1C2 CC1(OCC(=O)NC)CCCC1.C(=O)C(F)(F)c1ccccc1.C1(CC)CC1 C(=O)(C(F)(F)C(F)F)NC1C(CNC(C2ON=C(C)C2)=O)CCCC1 N1(C(C(C)O)=O)CCC(O)(CNC(=O)C(C)(C)Cc2cccc(Cl)c2)CC1 CN1C(=O)N(CCC2CCCOC2)C(=O)C1c1ccc(Br)cc1F c1(C(N2C(CC)CSCC2)=O)cc(S(=O)(=O)N(C)C2CC2)ccc1C.CC(=O)N CCCCC(O)C(C)C(=O)NC1CCN(C(=O)CC#N)C1C(C)(C)C CCC(CNC(=NCC(C)SC)NC)(CC)C=O.C1CCCO1.C(C)(C)C.C(C)=O c1(C(N2C(C3(O)CN(C(Cc4c(C)ocn4)=O)C3)CCC2)=O)cc(Cl)cc(Cl)c1F C1(OC)CC(CO)N(C(c2cn(CC)nn2)=O)C1.C1(C#N)(C=O)CC1(C)C.N c1(OCCC)ccc(CNCC(O)CC2(C#N)CCOCC2)cc1OC Cc1cccc(OC(C)C(=O)NCC(C)(CO)NC(c2cnc(Cl)[nH]2)=O)c1 C12CC(C1)C2.c1(C2C(C)C2C(=O)N)ccccc1.C1(C=O)CC1C(F)F CCC(C)C(CC(=O)N1CCCOC(C)C1)NC(=O)CCN(C)C N1(C(C(C)SC)=O)CCC(C)(NC(=O)CC2OCCCO2)CC1 c1(NC2CCC(CCC(=O)OC)O2)cccc2nc(C(F)F)[nH]c12 c1(C(=O)NCC(C)NC(CC(CC)c2ccccc2)=O)c(C(F)F)nn(C)c1C C(=O)(CC(C)C(C)(C)NC(=O)CC(=O)NCC)NCC(C#C)C(C)C C1(CC)CN(C(c2cc(-c3ccoc3)[nH]n2)=O)CCN1C(=O)C(F)C1CC1 C1(OC)CC2C1CCN2C(=O)CCC(C)NC(c1cnc(C)nc1C)=O C1(N(C(CN(C(=O)OC)C)=O)CC(C)C)CCN(C(C2(C)CCOC2)=O)CC1 N1(C(C2C(C)(C)C2C#N)=O)CCC(O)(CC)CC1.c1(C=O)cc(C(F)F)no1.N c1(CNC(c2scc(-c3cnc(SC)nc3)c2)=O)ccc(I)c(F)c1F c1(C(=O)NC2CC(NC(c3cccc(OC)n3)=O)C2)cc(OC)c2occc2c1 C1(CC(=O)NC(C)C)OCCC1(C)C.c1(C=O)cnn(C)c1C1CC1.CC CCCCCC(F)C(=O)NCC12CC(NC(=O)CCC(C)OC)(C1)C2 N1(CC(C)C)CCCC1C(=O)NC1CCC1NC(c1cnc(Cl)s1)=O c1(C(=O)OC)cnc(NCC(O)Cc2ccc(OC)c(OC)c2)c2ccccc12 CCCCCC(O)C(=O)N1CCCC1C1(C(=O)NCC2(CC(=O)O)CC2)CC1 N1(C(CC2(C)CCN2C(C23CSCC2C3)=O)=O)CCc2nn[nH]c2C1 c1(C=O)cccc(=O)o1.C(=O)(CCn1cccn1)N(CC)Cc1ccoc1.N c1(N2CCC(CN3CCC(CC(=O)NC(C(C)C#N)=O)C3)C2)ncccc1N c1(CN(C)C(C2CC(=O)C23CCC3)=O)c(C(F)(F)F)cccc1Cl C=CC1(C(N2CCCC(CCC)C2)=O)CCN(C(=O)C(=O)NC(C)C)C1 C(=O)(C(C(C)C)n1cnnc1)NC1(CCO)CN(C(c2c(C)csc2)=O)C1 c1(NCC2(C)CC(C)(C)C2)cc(Br)ccc1S(=O)(=O)N1CCC2CCCC2CC1 CCCC(C#N)C(=O)NC1CCCCC1NC(C1(Cc2ccc(F)cc2)CC1)=O C#Cc1cc(C(=O)NC(CCC)C(O)C(=O)NC2(C=C)CCOCC2)ccc1C c1(C(N(C(C(=O)NCc2n(CCC)ccn2)CC)C)=O)cc(CO)ccn1 C1(NC(c2c(C)ncn2O)=O)CC2CCC(C1)N2C(C12CC(C)(CCO1)C2)=O C=CCCC(C(=O)NCCC1(O)CCCCC1)NC(C1CCS(=O)CC1)=O CC(F)(F)C(F)C(=O)NC(C)(CNC(=O)CC1CC1)CO.c1ccccc1 C1(CC#C)CN(Cc2cccc(OC)n2)C12CCC2 C1(OC)CN(C(=O)C(C2CCOCC2)OC)CC1NC(=O)C(C)=C1CC1 c1(OCC)cc(CN2CC3CN(C(C4(c5ccccc5)CC4)=O)CC23)cc(Br)c1 c1(C(=O)N)coc(S(C)(=O)=O)c1.Cc1cccnc1C=CC(=O)NC(C)CC Cc1c[nH]c(=NCCNC(=O)NC2CCS(=O)(=O)C2)nc1SC(C)C C(=O)(CC(O)(c1ccccc1)C1CC1)NC1(C)CN(C(c2ccc(Br)cc2)=O)C1 c1(C(=O)NC(CCCC)CNC(=O)C(C)CC(C)(C)C)coc2c(F)cccc12 Cc1ccc2c(c1)cc(C(=O)NCCC13CCC(CC1)CC3)n2C c1(C(=O)NCC2CCCN(C(C3C(C4(C)COC4)C3)=O)C2)ccc2c[nH]nc2n1 c1(C(N(CC(C)NC)C)=O)cc(S(N)(=O)=O)n(C)c1.C1CC2CCC(C1)O2.C N1(C(C2CCCC(C)C2)=O)CC2C3CCC(C2C1)N(C(=O)CSCCN(C)C)C3 C1(C(=O)NC2CC(CNC(=O)CN3CCC(O)CC3)C2)CC12CC2(F)F N1(C(C2(C)CCC(OC)CC2)=O)CCC2(C1)CN(C(C1CC3CCC1C3)=O)C2 Cc1ccc2snc(C(N3CCC(CN(c4nnco4)C)CC3)=O)c2c1 C12(c3n(C(C)C4CC4)nc(-c4ccccn4)n3)CCCCC1C2(F)F C(=O)(C(C)S(N)(=O)=O)N.c1(COC)cc[nH]c1C(=O)NC1(C)CCC1 CC1(C)CC(CNC(C2(NC(c3csc(O)n3)=O)CC2(C)C)=O)CO1 c1(OC)c(C(=O)NC2(CC(N3CCC(C(C)C#N)CC3)=O)CC2)cnn1C C#CCCC(C(=O)NCCCC1CCCC1)NC(=O)C(C)C1CC1 N1(C(C(C2CCC2)OCC)=O)CC=CC1(C)C(=O)N(C)CC1(O)CCOC1 C1CC2(C1)CC2C=O.C1CC12CCC2.c1(CC(=O)OCC)cn(C)nn1 C(=O)(C(C)CC(F)(F)F)NCC(C1CCN(C(c2nccc(C)c2F)=O)CC1)C c1(C(=O)NC2C(NC(C(CCC)N(C)C)=O)COCC2)cc(Cl)ccc1Cl C(CCC(=O)N1CC(C(N)=O)(CNC(c2ccncc2)=O)C1)=C(C)C C1(C(=O)NCCCNC(c2cc(C)on2)=O)(OCCOC)CCOCC1 N1(CC(=O)NCC2(NC(C3CCO3)=O)CCOCC2)CC(=O)Nc2ccccc21 C1(CCC(=O)N(CCO)CC)CCN(C(c2cocc2C)=O)C1 CC1(C(N2CCN(C(C3(Cl)CC3(F)F)=O)CC2)=O)CCN(c2ccncc2)CC1 c1(NC(CCN(C(=O)Cn2cnnn2)CC#C)=O)cncc(C)c1 Cc1c(Cl)ccc(C(=O)NCC(C)(O)CNC(C2COC3CCCCC23)=O)c1O N1(C(C(C)N(C)C)=O)CCC(NC(C2(c3cc(F)ccc3F)CC2)=O)C(F)C1 C12(C(N3CCC(CN(C(=O)C(C4CCCCC4)O)C)C3)=O)CCCCC1C2 CC1CC2CN(C(C3CCOC3C3CC3)=O)CC2N1C(=O)CC1(N(C)C)CCC1 C1(NC(C(CC)C(C)O)=O)CC2CCCC(C1)N2C(C1COC(C)(C)O1)=O c1(C(=O)NCC2(CNC(CCNC(N)=O)=O)CCC2)cc(Cl)cnn1 CC1CCN(C(=O)C2=NOC(c3ccccc3)C2)C(CNC(c2ccon2)=O)C1 C1(CCC)CN(C(=O)CCc2ncccc2C)CC1NC(c1cccn1C)=O C=C(CC(C(C)C)NCC=O)C(=O)N1CC2CCC(O)C2C1.C(C)(C)C.C=O.O CCCCC(CNC(c1nc(C2CC2)no1)c1nnnn1C(C)C)CC C1(C)(C(=O)NC23C(CN(C(CNC(CC)=O)=O)C2)C3)CCC(=O)NC1 C1(CN(C(=O)Cc2cc(C(F)(F)F)n[nH]2)C)CN(C(=O)CCS(C)=O)CCO1 c1(C(=O)NCC(C(C)C)NC(C(C)SCCCC)=O)ccn(C2CC2)c1C C(=O)(CCCC(=O)N1CCN(C(C2CCOC2CC)=O)CC1C)OCC N1(CCC(=O)NCCCCN(C(C=C(CC)C)=O)C)C(=O)C2CCCCC2C1=O CCCC(CCNC(=O)C(CNC(=O)C(C)C(=O)OC)SC)C1CC1 C12(NC(CC3(C)OCCO3)=O)COCCC1CN(C(=O)CCc1nccs1)C2 NS(=O)(=O)c1cncc(C(N2CC(NC(=O)Cc3ccco3)C3CC23)=O)c1 C(=O)(C(C)CC(C)C)N1CCC(O)(COC)C1.C1(C(=O)N)CC2(CCC2O)C1 N1(C(c2c(C)scc2)=O)CCC2(CNC(C3CC(N(C)C)C3)=O)CCCCC12 c1(CC(=O)NC(CCNc2nc(SC)c(C)cn2)(C)C)ccc2cnccc2c1 N1(C(c2cncc(C#C)c2)=O)CCC2CC1CN(C(c1csc3cncn13)=O)C2 C1(N(C(Cc2c(C)n[nH]c2)=O)C)CCCCN(C(c2ccc(C(F)F)s2)=O)C1 C#CCC(C)(C(=O)NCc1cccnn1)NC(c1c[nH]c(=NC)o1)=O C1(NC(c2cn(C)nc2Cl)=O)CCC2(CC1)CCC2.C1(C=O)C(C)(C)C1(F)F N1(C(Cc2ccc(OCC=C)cc2)=O)CCC(NC(C2(C)CCCC2)=O)C(O)C1 N1(CC=O)CCC(=O)NC1=O.c1(OCC)cncc(C(N2CC(CO)C2)=O)c1 c1(C(C(=O)NCC)N(C)C)ccccc1.C1CCCOCC1.C(C)(C)C.C=O CCC(C)C(C(=O)NCCCCc1ncc[nH]1)N(C)C(c1cccc(=O)o1)=O Cc1cccc(C)c1C(=O)NCC1CCN1C(C12CC(C1)C(C)O2)=O C1(C(=O)NCCOCC#C)C2CCC1CN(C(c1cccc(C)n1)=O)C2 C1(C(=O)NCC2(C(N3CCCC3)=O)CC(=C)C2)CC12CCOC2.C1CCC1.C C1(CC(=O)N(C2CC2)CC2CCCN2C(c2cc(CCO)on2)=O)OCCCO1 c1(C(=O)NCC(C2CCCCC2)NC(CCC(C)OC)=O)c(Cl)cccc1Cl C1(NCCC(COC)OC)CCC(C)N1C(=O)OC(C)(C)C N1(C(C2(C)C(C)CCCC2)=O)CCCc2c(Br)cccc2C1 n1(C(C)C)ncc(Cl)c1C(=O)NCC1C(C)CCN1C(C1CC(O)C1)=O N1(C(CC=C=C)=O)CC(OC)CC1C(=O)NCC1(CC2CC2)CC1 N1(C(CCOCC(C)C)=O)CCC(O)(C)C1.C1(C=O)CC(O)CN1C(N)=O Cc1c(C(=O)NC2CCOC(C(=O)NCCCCN(C)C)C2)ncn1C Cc1cc(C=CC(=O)N(CC(C)NC(c2nc(F)ccc2Cl)=O)C)ccc1F Cc1cc(F)cc(C)c1C(=O)NCC1CC2(C1)CN(C(C1CC(F)C1)=O)C2 C1(OC)CN(C(c2cccn2C)=O)C(C)(CNC(=O)CCC(C)(C)F)C1 N1(C(CC(C)C)=O)CC(NC(=O)C=Cc2ccc(C(N)=O)o2)C2CC12 c1(C=O)ncc2ccccn12.c1(C(=O)NCCCOC2CC2)conc1C.N c1(C(N2CC(CNC(=O)Cc3nncs3)OCC2)=O)ccc2nncn2c1 c1(C=O)cc2n(n1)CCOC2.c1(C=O)cc(Cl)c([N+](=O)[O-])[nH]1.CCC1CC1.N C(C#CC#CCO)NC(c1c(CNC(C2(CC)CCC2)=O)cco1)=O c1(NCC2CCCC(NC(c3cc(CCC)on3)=O)C2)ncnc2c(C)csc12 C1(NC(C2C(F)(F)C23CC3)=O)CC2(CCN(C(C3(CF)CCC3)=O)CC2)C1 O=C(C1COc2ccc(Cl)cc21)NCC12CCC(CC1)N2C(c1cc(Cl)c[nH]1)=O N1(CC)CCOC(C(N2CCCC2Cn2ccnn2)=O)C1.C(=O)CC1CC1.C C1(NC(c2ccnnc2Cl)=O)CC2CN(C(c3cccc(C4CCC4)c3)=O)CC12 CCCCCCC(C)C(=O)NCC1CCCC1NC(c1csc(O)n1)=O c1(Nc2cc(OC)nc(C)n2)cccc(S(=O)(=O)NC)c1.c1cccc(C#N)c1 c1(C(=O)NC2CC(NC(C(C=C)(F)F)=O)C23CCC3)ccc(OC)c(Cl)c1F N1(C(Cn2c(C)ncc2)=O)CCNC(C(=O)N(CC(C)(C)O)CC(C)(C)O)C1 C(=O)(CC(C)(C)N(C(=O)CCCn1cccc1)C)NCC1C(C)C1 C1(C(=O)NC(c2cccc(C)n2)CCC)CC(C)CN1CCOc1ccccc1 c1(C(=O)NCCCC2N(C(C3C(C)C3)=O)CCCC2)cccc2c1C(=O)NC2 N1(C(C=C(C)CNC(C2CC3CC(=O)C2C3)=O)=O)CCC(C2CC2)C1CO c1(C(=O)NC(c2cccc(OC)c2)CNC(=O)C(C)O)cc2nc[nH]c2cc1F N#Cc1ccccc1OC1(CN2CC=C(Br)CC2)CC1 c1(-c2cn(C(C)C(N3CCCC4CCCC34)=O)nn2)cccc(P(C)(C)=O)c1 c1(C(=O)NCC(=C)CCNC(=O)Cc2ccsc2C)cc2cc(OC)ccc2o1 CCCC(O)CC(=O)NC1CC2CC(NC(c3ccc(CO)cc3F)=O)C1C2 c1(C(N2CC(CC(C)C)C(O)CC2)=O)ccc(I)cc1C#N C(c1cc(Cl)cc(Cl)c1)=CC(=O)NC(CNC(C=COCC)=O)(C)CO c1(SCc2nc(-c3cn(CC4CCC(=O)O4)nn3)on2)ccnc(Cl)c1 c1(OC)cccc2c1CC(C(=O)NCC1CN(C(=O)CC)C1)CO2.C(N)=O.N N1(C(C2(CC=C)CN(C(=O)Cn3[nH]cnc3=N)C2)=O)CC(C)C(C)C1C C1(CNC(c2ccc(C)n2C)=O)CN(c2cc(C(C)C)nc(Cl)n2)CC(C)(C)O1 c1(C(N2C3CCC2CC(O)C3)C(=O)NC(C)(C)C)ccc2c(c1F)CCC2 C1(C)(CC)CCC(C(=O)NCc2c[nH]nc2C(=O)NCCF)O1 NS(=O)(=O)c1csc(C(=O)NCC2CCCC2)c1.C1(C=O)CC12CCCC2.C c1(C(N2CC(C(=O)NOCCCOCC)(CCC=C)C2)=O)cnc(OC)nc1 c1(C(=O)NCC2N(C(C(C)OC)=O)CCOC2)cc(Cl)cc(Cl)c1Cl c1(OC)ccc(CCNC(C2(C)CCC2)=O)cc1.c1(C(=O)N)c(Cl)cnn1C C1(C(N2CC(O)(C(C)NC(C=CC=CC)=O)C2)=O)CC2CC1CO2 C1(C(=O)NC(C=CC(=O)N(C)CCN2CCOC2=O)(C)C)CCCOCC1 C1(NC(CC(C)(C)O)=O)CC2(C1)CC1(CCC1)C2.c1(C=O)ccsc1C(F)F N1(C(c2ncc(Br)cn2)C)CCC(C2(CO)CCC2)CC1 Cc1ccc2c(c1)C(C(=O)NCC1CCC(C)CN1C(=O)Cn1nccn1)CC2 c1(C(=O)NCC=CCNC(C(CC)F)=O)sc2cccc(F)c2c1COC C=CCC(F)(F)C(=O)NC(CNC(=O)CCCn1nc(C)nc1C)C(C)C c1(C(N2CC=CC(NC(COCCC=C)=O)C2)=O)cc(S(N)(=O)=O)co1 C1(NC(CNC(c2ccc(C)s2)=O)=O)CCC2CCN(C(=O)C3=CCC3)C1C2 n1(CC(=O)NC2CC(OC)CN(C(=O)C(O)CSC)C2)c(C)cc(C)nc1=O N1(C(COc2cc(C)nn2C)=O)CCN(C(C2CCCCC2)=O)CC1CC(F)F C(C)(C)(CCC(=O)C(C#N)c1ccccc1Cl)c1c(SC)cccc1 C(C(=O)NCC(F)F)(C1=C(C)C=CCC1(C)C)N(CCCO)CCC CC1(C)Cc2cccc(C(N3CC4OCC(NC(c5ccco5)=O)C4C3)=O)c2O1 c1(CN(C2C(OCCOC)CCCC2)C)ccccc1[N+](=O)[O-] C1(C(=O)NC(CC2CC2)CO)CCOCCN1C(=O)C=C1CCOCC1 c1(C(=O)NCC(C2CC2)NC(c2cc(C)c(O)cc2)=O)cc2c(Cl)cccc2[nH]1 O=C(N=c1[nH]oc2cc(Br)ccc12)C1C(O)CCN1Cc1cc(Cl)c(Cl)cc1Cl C1(NCC2(O)CCC2)C(OCc2ccccc2)C2CCCC12 Cc1cc(C(N2CCC2CNC(=O)C(C)NC(C2CCCCC2)=O)=O)no1 Cc1cc(F)cc(C)c1C(=O)NC(C)CC(C)NC(C1OCC1(C)C)=O Cc1nc(O)ccc1C(N1CC(C)(C)CC1CO)=O n1(CC)ccnc1C(C)NC(=O)NCCCCCSC c1(C(N(CCCCCNC(c2c(C(C)C)n[nH]c2)=O)C)=O)cnn(C(C)C)c1F CS(=O)(=O)c1ccc(F)cc1C(N1CCCCC(NC(=O)CCCC(F)F)C1)=O c1(CC(N2CC(CC(=O)N(C3CC4(CC4)C3)C)(OC)C2)=O)c(C)noc1C c1(C(=O)NCC2(F)CN(C(C(CC)OCC)=O)C2)ccc(Br)cc1 Cc1cnc(CCNC(=O)C(C2CCC2)NC(=O)Cc2ccns2)cn1 Cc1nn(C)c(C(N2CCN(C(C3CC3Br)=O)CC2)=O)c1Br C1(CN(C(C)=O)CC)CN(CC(O)CC2CC3CCC(C2)N3)CCC1O N1(C(C2(NC(c3ncc(C)[n+]([O-])c3)=O)CC(F)C2)=O)CC2CCCCC2C1 N1(C(C(C=CC)O)=O)CC(NC(c2ccc(-n3cnnc3C)cc2)=O)C2(CC2)C1 c1(C(=O)Nc2ccnn2CC2CCOC2)cnc(C2CCNCC2)nc1 C(N=c1[nH]c(=NCCCC2CC2)[nH]c2c1COC2)c1ccc(C)nc1 C1(COC)(C)CN(C(C2CC(=O)C2C)=O)C1.C(=O)(CCCN1CCCC1)N CC1=CCC(C)(C(N2CCCC(CO)(NC(c3ncccc3O)=O)C2)=O)CC1 Cc1nc(C(F)(F)F)c(C(=O)NCC2(NC(c3oncc3C)=O)CCC2)o1 C#CC1(C(=O)NCCC2CC2C)CCN(C(c2ccn(C)c2C)=O)CC1 c1(C(=O)NCC2(CNC(CC(C)F)=O)CC2)cc(N2CCOCC2)ccn1 C1(C=O)CN2CCC1C2.C1(CNC(C2CC(=C3CCC3)C2)=O)CC1(F)F c1(NC)ccc(C(=O)NCC(CC)NC(=O)COCC2CCCO2)cc1 C1(NC(C(C)N(C)C(C23C=CC(CC2)C3)=O)=O)CCC(CCO)CC1 Cc1sc(=O)n(CC(=O)NC2(C)CCCN(C(c3occc3C(C)C)=O)C2)c1C C1(CC(=O)NC(CCSC)C(=O)O)CS(=O)(=O)CCO1 Cc1cnn(C(C)C(=O)NC(C)C=CC(N2CCC(OCCF)C2)=O)c1 c1(C(N2CCCCCC2c2ncon2)=O)c(F)ccc(I)c1Cl C12(NC(c3csc(C)c3C)=O)CCOCC1CN(C(c1ccnn1C(F)F)=O)C2 C(C(C)(C(=O)NCC1CC=CC1)NC(=O)COC(C)C)SC c1(OC)ccc(C)nc1C(N1CC(CCNC(c2ccc(F)s2)=O)(O)C1)=O C1(NC(C(C(C)C)n2cnnc2)=O)(CO)CCCN(C(=O)C(F)(F)C(C)O)C1 C(=O)(CC1=CCN(C(C2CC2CC(C)C)=O)CC1)NCC(CC)(F)CC C1(NC(c2cc(C)nn2C(C)(C)C)=O)C2CC1N(C(=O)O)C2C.C(C)(C)C C1(OCCN(CC)CC2CC2c2ccccc2)CCN(C)C1 Cc1[nH]nc(C(N2CCC(C(C)C(=O)NCC3C=CCCC3)C2)=O)c1C C1(c2cn(C3(c4cc(C)on4)CC3)nn2)CN(C(=O)C(O)CF)CCO1 CN1CCOc2ccc(C(=O)NCC#CCNC(C3COC(=O)N3)=O)cc21 Cc1cccc(C)c1C(N1CC2(C1)CN(C(c1cn(C(C)(C)C)cn1)=O)C2)=O c1(C(C)NCC(=O)NCC23CC(F)(CO2)C3)cccc2ccccc12 CCC(C)(O)C(=O)NCc1cn(C2CCN(C(C3(CC(F)F)CC3)=O)C2)nn1 CN1CCCCC(C(N2CCN(C(c3nn(C)cc3N)=O)CC2CF)=O)C1=O N(C(=NCCc1noc(C(C)(C)C)n1)NC1CCS(=O)(=O)C1)CC(=C)CC O=S(=O)(c1ccc(Br)cc1N)NCCc1cnc(Cl)s1.C1CC2C(C1)C2(F)F c1(C(=O)NCC2N(C(c3cn(CCC=C)nn3)=O)CCC2)cc2nc(C)sc2[nH]1 C1(CC)C(C(N2CCC(O)(CN(C(=O)C(C)=C3CCC3)C)C2)=O)CCN1C C1(C#N)(C(=O)NC(C(=O)N2CC(n3ncc(C)c3)C2)C(C)C)CCCCC1 c1(CC(C=O)O)ccc(Cl)cc1.C=CCCCNC(c1cnn(C2CC2)c1)=O.N C1(C)(NC(c2c(C)cc(CNC(=O)C(F)C3CCOC3)o2)=O)CC2CCC1C2 CCCCC(=O)C(=O)N(C)CCC1CCN(C(C2CCCC2O)=O)CC1 C=C(Cl)CC(C(=O)NCc1cc(C)ccc1O)NC(=O)CC1CCCC(=O)N1 c1(C(C)C)cc(C(=O)N)n(C)n1.c1(C(N2CCCC2)=O)ccc(C2CC2)cn1.C C1(CNC(CCc2ncc(C)[nH]2)=O)CN(C(c2ccc(Cl)c(N)c2)=O)CCN1C N1(C(CCNC(=O)C=CCl)=O)CCC(CF)(NC(=O)CS)C1.c1ncc[nH]1.C C=CCC(CC(=O)N1CCCC(CCCO)C1)NC(=O)CCC=CC(C)C C#Cc1ccc(C(=O)N(CCC(=O)NC2(CCCF)CC2)CC=C)c(C)c1 C(CC(F)F)(C(=O)NC)N(C(=O)CCCC1CCCO1)C.C12CC=CC(C1)OC2 C12(CNC(C3CCCO3)=O)CN(C(=O)CC3=CCCCC3)CC(F)(C1)C2 C#Cc1cccc(C(=O)NC2(CN(C)C(C3CCCCC3C)=O)CC2)c1Cl c1(C=O)c(C#N)cnn1C.N1(C(C=CC(CC)=CC)=O)CCC(C)C1C.N C#Cc1ccc(C(=O)NCC2CCCN2C(=O)Cn2nc(O)ccc2=O)c(C)c1 c1(C(N2C(COC)CN(C(=O)C(C)(C)CF)CC2)=O)cccc2cncn12 N1(C(c2nc(OCC)oc2)=O)CCCC(C(=O)N(CC(C)COC)C)CC1 c1(CC)nn(C)cc1O.c1(CNC(C=C(COC)C)=O)cc[nH]c1C(=O)N c1(OCC)nc(NC2CCCN2C(c2cnc(Cl)cn2)=O)ncc1Br CCCC(CC(=O)NC(c1nnc(O)o1)C)NC(C12CCN(CC1)C2)=O c1(OC)cccc(C(C(=O)NCC2CCCN2C(C2CCN(C)C2C)=O)OC)c1 CCC(CC)CCC(=O)N1CC(C(=O)NCC2CCC(C)(C)CO2)C(F)C1 C(=O)(C(F)C(=O)N(C1(C(=O)NC)CC1)C)OC.C1(C=O)(NC)CCC1.C C1(NC(CCCCC)=O)CCCC12CN(C(=O)C(F)(F)c1cnnn1C)C2 N1(C(COC2(C#C)COC2)=O)CCN(C(c2nccc(OC)c2OC)=O)C(C)C1 C1(C(=O)NC2C(N(C)C)COC2)CCOCCN1C(c1ccn(C(F)F)n1)=O c1(N(C)Cc2cn(C3CC(O)C3)nn2)ccc(Cl)cc1F c1(CC(=O)NCC2CCN(C(C(=Cc3cccs3)C)=O)CC2)cc(C)ccc1C Cc1ncc(C(=O)NCCN(CCCN(C)C)C(c2ncccn2)=O)s1 C1(NC(c2ccc(C(C)=O)s2)=O)CC(O)CN(C(C23CC(C)(C2)C3)=O)C1 C1(C(=O)NCC2(CC)CCC2)COC(C)C1.C1(CC(C)C)(C=O)CCC1 C1(CN(C(c2n(C(C)C)ccc2)=O)C)CCCCN1C(c1csc(C#N)c1)=O N1(C(CNC(CC)=O)=O)CC(C)CCC1C(=O)NCCc1noc(C)n1 C(C)(CCCCNC(C1CC(F)C1)=O)NC(CCOCCOCC)=O.C c1(C(=O)NCC(C)(C)NC(C2CCCCO2)=O)cc2cncn2c(O)n1 c1ccc(Cl)cc1.C1(C=O)C(C)CN1C(=O)N.CCC.CC=CC=CCBr N1(C(c2cn(CC)cn2)C(=O)NCC)CCn2c(cnc2C2CCC2)C1 C(=O)(C(C(C)C)NC(=O)CN1CCC(=O)CC1)N1CC(CSC)C1 c1(CCC)ncc(C(=O)N(CCC)Cc2ccncc2)s1.C1(C)(C=O)CC1.N N1(C(C(C(=O)OC)C)=O)CCN(C(=O)C(=CC2CCCC2)C)CC(CO)C1 C1(C(=O)NCC(CC=C)NC(c2ncoc2C)=O)COc2ccc(Cl)cc2C1 N1(C(C=NOC)=O)CCC(CNC(=O)CSCc2ccncc2)C(C2CC2)C1 c1(CN(CCOCC)C)cc(C(C)(C)C)cc(C(C)(C)C)c1 Cc1cc(C(=O)Nc2cn(C)c(C(=O)Nc3nnc(Cl)cc3Br)n2)cnc1C CC1=C(C(=O)N2CCN(C)C(CNC(=O)C(C)(C)c3cccs3)C2)CCO1 N1(C(CCCN=[N+]=[N-])=O)CCC(C2CC2)C1CNC(C1CC(F)(CO)C1)=O C1(OC)CCCCC1C(=O)NCC(=O)NCC(C1CC(C)(C)C1)O.C1CC1 c1(C(=O)NC(CCNC(C(C=C)(C)CC)=O)C)noc2c1CCc1ccccc1-2 N1(C(CC(CCC)(C)O)=O)CCC2(CCC(NC(c3cscn3)=O)CC2)CC1 c1(C(N2CCc3ncncc3C2)=O)n[nH]c2cc(-c3cc(O)cc(F)c3)ccc12 CC1CCN(C(c2cnc(C(F)(F)F)s2)=O)CCN1C(C1CCC1C)=O c1(C(N2CC3(CC(CC(=O)Nc4cncc(Cl)c4)C3)C2)=O)cc(I)c(F)cc1F C1(C(N(CCCN(C)C)CC)=O)CCN(C(c2ccc(CC#N)cc2)=O)C1C C1(NC(COC)C(=O)OC)CCN(c2cc(C(=O)OC)nc(C)n2)CC1F N1(C(CC(C(C)C)C)=O)CCN(C(C2CN3CCC2CC3)=O)C2CCCC2(C)C1 N1(C(C2CCC(=C)CC2)=O)CC2CC(NC(C3CC=CCC3)=O)C2C1 N1(C(CCn2c(=O)cc(C)nc2)=O)CC2CCC(C1)N2c1ncnc2c1COC2 N1(C(c2c(C)scc2)=O)CCCC(NC(=O)C(CC(F)F)C2CCC2)CC1 c1(C(=O)NC2(CNC(=O)C(C)C(C)O)CC(OC)C2)cc(C)c(C)nn1 C(=O)(C(CNC(c1ccc(F)c(F)c1)=O)C(C)(C)C)N1CCC(OCC)C1 N1(C(c2cc(CC)n(C)n2)=O)CCC(NC(c2ccncc2F)=O)C(C)C1 N1(C(C)CNC(C2CCC(F)CC2)=O)CCN(C(C2COC(=O)N2C)=O)CC1 c1(C(N2C(C#N)CCC2)C(=O)NCC2CCCO2)ccc(Cl)c(Cl)c1 C(=O)(C1=CSCCO1)NCC1CC(C)N(C(c2cnn[nH]2)=O)C1 c1(C(N2CCC(CC)C2)=O)cc(N(C)C)nc(Cl)c1.C(C=O)(C(C)C)SCC Cc1cnc(C(=O)NC(C2(O)CCN(C(C3CC=CC3)=O)CC2)C)cc1C N1(C(C2CN(CC)C(=O)CC2)=O)CCC(C)=C(c2ccco2)C1 C1CCCCCN1C(=O)C=Cc1cocn1.C1(C(=O)N)(COC)CCC(=O)N1 N1(CC(=O)NC2CC(NC(=O)C(C3CCOCC3)F)C2)C(=O)CNC1=O Cc1cccnc1CC(=O)NC(C)(CNC(C1CSCC(=O)N1)=O)C1CCC1 c1(N2C3C(C(=O)Nc4nccc(F)c4F)C(C3)C2)nc(Cl)c2c(n1)COC2 C(=O)(CCCN(C)N=O)N.C1(NC(Cc2c(OC)nccc2)=O)CS(=O)(=O)CC1 c1(C(N2CC(NC(CC(=C)C)=O)C(c3cnn(C)c3)C2)=O)cc2ccccn2n1 N1(CCC(=O)NCC(C)(C)CNC(=O)CCC2CCC(=O)N2)CCCCCC1 C1(C)(OC)CCCN(C(=O)C(O)C2CN(C(=O)CC3C(C)(C)C3(C)C)C2)C1 N1(C(C2(COC)CC2(F)F)=O)CCC2(CC2)C1.c1(C=O)cc(O)cc(Cl)c1 c1(C(C)NC(C2N(C(c3cccc(C)c3)=O)CC2)=O)ccc(S(C)(=O)=O)cc1 c1(CCNC(=O)NC(C2ON=C(C)C2)C2CC2)cn(C)c2c(C)cccc12 c1(C(=O)NCCC2(O)CCOC2)ccccc1CSC1=NCCS1 Cc1cc2nc(C(N3CCN(C(c4csc(Cl)n4)=O)C4CC34)=O)cn2cc1C C1(c2n(CCOCC)nnn2)(NC(c2nncs2)C)CC(C)CC(C)C1 C1(CNC(C(N2CCC(NS(CCC)(=O)=O)C2)=O)=O)CCC=CCCC1 N1(CC(C)NC(=O)Cc2csc(S)n2)CCN(C(=O)Cn2nnc(=O)[nH]2)CC1 C1(C(=O)N(C)C)(CC)CCCN1C=O.n1(CC)cc(N)nn1.C(C)(C)C c1(C(=O)NCC(C)N(C(c2n(C=C)ncc2)=O)C)cccc([SH](=O)=O)c1.N C(CC1CC1)(C(=O)NC(C1CCCCO1)(C)C)NC(C(=O)NC(C)C)=O N1(C(C2(C)CC2)=O)CCC(C2CC2)(NC(c2cnsn2)=O)C1 CCCCC(O)C(=O)NC(C(=O)NC1CCCC1)c1ccco1 C1(CC(=O)NC(C=C)COC)(NC(C2C=CC2C=O)=O)CCCCC1.O N1(C(COCCOCC#C)=O)CCN(C)CC1C.C1(C=O)CCCCCCC1.N C(c1ccc2[nH]ccc2c1)=CC(=O)NCC1N(c2nnc(C(C)(C)C)s2)CCC1 N1(C(C2N(C(c3onc(C)n3)=O)C3CCC2C3)=O)CCC2(CCC(O)CC2)CC1 N1(C(c2c(C)coc2C)=O)CC(N(C)C(C2CCCS(=O)(=O)C2)=O)C(C)(C)C1 c1(OC)ccccc1C(C)CC(N1CCC(NC(=O)C=CCN(C)C)C1)=O c1(C(=O)N)c(N)cc(F)cc1F.C1(C(N(CC(C)O)CC)=O)CC12CCOCC2 C1(CC(=O)N(C)CC2(NC(C3CCN(CC)C3)=O)CC2)CCCN(C)C1 C1(NC(C(C2(O)CN(C(C3(C)N(C)CCC3)=O)C2)F)=O)CCn2cnnc2C1 c1(OC)cc(C(C)NC=O)ccc1S(C)(=O)=O.c1(CC(C)O)cccc(F)c1.N c1(-c2nc(C3CCCN(C(=O)OC(C)(C)C)C3)on2)cc2c(nc1O)CCC2 N1(C(C(C)CC(N)=O)=O)CC(C)CN(C(C2(N(C)C)CCC2)=O)CC1C c1(SC)cc(C(=O)OCc2csc(C)c2C)ccc1N CCCC(C)(CC)C(=O)N(C1CC(NC(=O)CCc2ccncn2)C1)C N1(C(C(C)OCCCC)=O)CCCCCC1.n1(CC(=O)N)nnc(C(C)(C)C)n1 C(=O)(CCCCNC(c1c[nH]nc1CNC(=O)Cc1ncccn1)=O)OC CCCCCC(F)C(=O)N(CCCCN(C)C(C1CCCCN(C)C1=O)=O)C CCC(C)CCCC(=O)NC(C)(CNC(c1cc(CO)ccn1)=O)CC c1(C(=O)NCc2cnc(C)s2)ncccc1NCc1cccc(CO)c1 c1(C(N2CC(O)(C(C)NC(Cc3c(C)ncs3)=O)C2)=O)ccc(CO)cc1 c1(C(=O)NC2CCC(N(C(CN(C(C)C)C)=O)C)C2)cccc2ncccc12 c1(C(N(C)CCN(C(=O)C(O)c2ccco2)C)=O)cc(Br)co1 C1(OCC=C)CCN(C(=O)CC(C)NC(C2(CC)CC2)=O)C1 C1(COC)(NC(=O)CC)CCN(C(=O)CCC2CCC(O)CC2)CC1.C(C)C c1(CN2CCC(C)(C(=O)Nc3c(Br)ccc(C)c3)C2)ncn2ccccc12 C(=O)(C1CCc2c[nH]nc21)N1CCCC(C(=O)NCC(COCC)O)CC1 c1(C(=O)N)cccc(C2(S(C)(=O)=O)CC2)c1.C1(C(N(C)CC)=O)CCOC1 N1(C(C2CC3(CN(C(c4cc(C(C)(C)C)n[nH]4)=O)C3)C2)=O)CCC(O)C(F)CC1 CCCCC(C)C(=O)N1CC(NC(=O)CN2CCN(C)C(=O)C2)CC(F)C1 C12(C(N3CC(CCC)N(C(=O)CC(O)C(C)C)CC3)=O)CCCN1CC(OC)C2 c1(C(=O)NC2CN(C(c3c(C)oc(C)c3C)=O)CC2C)cc(O)cc([N+](=O)[O-])c1 c1(CC)cc(C(=O)NCC2CC(F)CN2C(=O)C(O)CCSC)cc(F)c1 C(=O)(C(O)(C(F)(F)F)C1CC1)N1CC2(CN(C(COc3cn(C)nc3)=O)C2)C1 N1(C(C)C)CCCC(C(=O)NC2CCC(NC(=O)C=O)CC2)C1.CCC(N)=O.N CCCC(C(=O)NC1CCN(C(=O)CSCc2ccncc2)C1C)N(C)C Cc1nc([N+](=O)[O-])cn1CC(=O)NC(C)C1CCC1.C1(CC=O)CCN(C)C1 C1(CCNC(COc2cccc(CC)c2)=O)CC(F)(F)CN1C(=O)C(O)C C1(n2cc(CCCSCC)nn2)CN(C(=O)CCc2scnc2C)CC1O c1(C(=O)NC2CC(N(C(c3c(C)scc3)=O)C)C2)noc(-c2ccccc2)c1C Cc1cccc2[nH]c(C(N3CCC(=CCNC(C4CC4(Cl)Cl)=O)CC3)=O)cc12 C1(NC(c2cn(C)nc2O)=O)CN(C(C2(C#N)CCOCC2)=O)CC12CC2 c1(C(=O)NC2CCCN(C(C(C(CC)C)O)=O)CC2)cc(F)cc2nn(C)cc12 C1(OC)CN(C(c2nn(C)cc2Cl)=O)CCC1NC(C1CCCC1F)=O N1(CC(=O)NC(C(=O)NCCSC(C)C)c2cccs2)CCOCC1=O N1(C(C(CC)CC)=O)CC2CCOC2(CNC(c2c(OC)ccnc2F)=O)C1 c1(C(C)C)cccc(CN2CC3C(CNC(c4ccc(C#N)s4)=O)C3C2)c1 CC1CN(C(=O)Cc2cnsc2)CCC1CNC(c1cnn(C)c1Cl)=O c1(-n2c(C)nnn2)ccc(C(N2CCC(NC(C3CCC(=O)C3)=O)C2)=O)cc1 C#CCCCCCCC(=O)NC1CCN(C(=O)C(C)(C)C(O)C(C)C)CC(O)C1 C1(C(=O)NC2C(NC(c3cn(C)nc3)=O)CC2)CCCC1C1CC1 c1(C(C)NCC(=O)N(C2CC2)Cc2ccc(C#N)cc2)nc2cnccc2s1 C1(NC(C=C(CCC)C)=O)CN(C(C2CCN(C(C)C)CC2)=O)CC2(CC2)C1 C1(C)(CNC(c2nnc(C)s2)=O)CCCN(C(C)C(=O)NCC(C)C)C1 N(C(=NCC)N(C)CCOC)C(C#C)Cc1ccccc1OC.c1cccc(F)c1 Cn1cc(Cl)c(CC(=O)NCCc2ccc(CNC(=O)C(C)(C)CO)cc2)n1 C(=O)(C1CC(=O)Nc2cc(F)ccc21)N1C(CNC(CCCC)=O)CCC1 C12(C(N3CCC(N(C(C=CSC)=O)C)C3)=O)CC(C)(CCO1)C2 Cc1nc(CCNC(C2CC2C(C)NC(=O)CCN2CCOCC2)=O)cs1 Cc1cc(C(=O)NCC2(NC(C3CC4C=CC3C4)=O)CCCCC2)c(C)s1 c1(C(N2CCC(NC(C(COC)NC(C)=O)=O)C2)=O)cccc2nncn12 c1(N2C(C)CC(CNC(=O)CC3CCC(=O)NC3=O)C2)ncc([N+](=O)[O-])cn1 c1(OC)ccc(O)c(C(N2CC3CC3(C(=O)NCc3c(C)noc3C)C2)=O)c1 C1(C(=O)Nc2ccc(F)s2)CCCN(C(=O)C2CC2)C1 C1(C(=O)NCC(c2ccccc2)CNC(=O)Cc2ccccn2)CC(F)C(=O)N1 N1(C(c2nncn2CCO)=O)CC(C=O)C2CC12.c1ccccc1.C1(C)CC1.N c1(OC)cccc(S(=O)(=O)N2CCSC(C(=O)Nc3cnc(Cl)cc3C)C2)c1 C(=O)(CCC(=O)CC)N1CC(C(C(=O)NC(C#C)C(C)C)O)C1 N1(C(c2cc(C)nc(O)c2)=O)CCC(C)(C)C(C(=O)NC2CCCC2N(C)C)C1 CC1(C)CC(C)(C(N2CCC(N(C(=O)C3CC3)CC)CC2)=O)C1.C1CC1.N c1(C(N(C2CCN(C(C(C)C)=O)CC2)C)=O)cc(F)cc(S(N)(=O)=O)c1.CC.O C(C(C)N=c1[nH]c(=NC2CC(CF)C2)c2cc(Cl)ccc2[nH]1)SC CC(CC(=O)NCC(C)CN(C)C(c1cnc(Cl)[nH]1)=O)CC(C)(C)C c1(C(=O)Nc2cc(C)no2)cc2n(n1)CCCN(Cc1cccnc1O)C2 C(c1ccccc1Cl)=CC(N1CC2C(NC(c3cc(Br)co3)=O)C2C1)=O c1(OCC)cccc2[nH]c(C(N3CCCC3)=O)cc12.C(=O)C(C)(O)C(F)(F)F.N n1(CC(=O)OCc2cn3ccccc3n2)cnc2ccccc2c1=O c1(C(N2CCC(O)C2)=O)cnn2c1CC(F)(F)C2.CN(S(N)(=O)=O)CC(=O)N c1(OC)ccc(C(=O)NCC(C)NC(c2nn(CC(F)(F)F)cc2Cl)=O)cc1O C1(C2CCN(C(c3ccc(Cl)[nH]3)=O)CC2)(NC(c2n(CCC)ccc2)=O)CCC1 Cc1cc(C)c(CC(=O)NC2CC2CNC(=O)CSc2ccccc2F)s1 c1(C(=O)N)cnc2sc(C)nc2c1.c1(CC(=O)N(CC)CC)cc(Cl)ccc1O C(=O)(NNC(=O)CC1CCC2CNCC12)c1ccc(N(S(=O)(=O)c2cccs2)C)cc1 n1(CC(=O)N(C2CCCC2)C)c(C)c(C)sc1=O.c1(CC)cnc(C=O)nc1.N C1(NC(C=CC(CC)=CC)=O)CN(C(c2cnn3c2OCC3)=O)CCC12CCC2 N1(C(Cc2ccc(OCC)cc2)=O)CCN(C(=O)CSCC)CC1COC N1(C(C(C(C)C)NC(c2ncc(C)nc2)=O)=O)CCCC(C)(C#N)C1 C(=O)(C(C)(C)CC#N)NC1CCCN(C(C(C)CCc2ccc(F)cc2)=O)C1 C1(OC)CC(NC(c2cccc(CCO)c2)=O)CN(C(=O)CC2CC2)C1 c1(C(N2CCOCC2c2ncn(CC(F)(F)F)n2)=O)cc2c(O)ccc(F)c2[nH]1 C1(C(=O)NC(C)CNC(C2(N3CCOC3=O)CC2)=O)Cc2ccncc2C1 c1(OC)cc(C)ccc1CNc1ncc(OC)s1 c1(C(=O)NC(CN(C(=O)C2=CC(C)(C)C2)CC)C)cc(OC)nc(C)c1 N1(C(CCc2cc(C)[nH]n2)=O)CCCOC(CNC(C2(C)CC(=O)N(C)C2)=O)C1 C1(NC(C(c2n(C)cnc2)O)=O)CCCCC1NC(=O)CO.c1ncnn1C.C CN1CC=C(CC(=O)NCCC(O)CNC(c2cnc(C3CC3)[nH]2)=O)CC1 Cc1ccc2[nH]cc(C(=O)N(CC)C(C)C)c2c1.C(=O)C(C)C(C)S(C)(=O)=O N1(C(c2cnn(CC)c2Cl)=O)CCN(C(c2ccc(C3CC3)nc2)=O)C2CCC12 N1(C(C2CCN(C(c3ccn(CCC)n3)=O)C2)=O)CCC12CCC2 C=C(CC)CN=c1cc(C)nc(NC(c2cccc([N+](=O)[O-])c2)C)[nH]1 C(CC(O)C=O)N(C)C.C(=O)(C(C=O)C1CC1)N(CC)C1CC1.C(C)(C)C c1(C(=O)NCC(CNC(C2(SC)CCC2)=O)(C)C)cc2c(nc1O)CCC2 NS(=O)(=O)C1(C(=O)NC2COCC2NC(=O)C(O)C2CC2)CC1 c1(C(=O)NCC(C)CN(C(=O)CCc2nc(=N)[nH][nH]2)C)cnc(C2CC2)s1 c1(CNC(C2C=CCCC2)c2nnnn2C2CCC2)noc2c1COCC2 Cn1cc(NC(=O)C(Cc2ccoc2)NC(=O)C(O)C2CC2)c(O)nc1=O N1(C(CC(CC)C)C)CCC2(CC1)CC2(C)C(=O)NCC1CN(C)CCO1 N#Cc1ccncc1C(N1CCC1C(N1CCCC(C(F)F)C1)=O)=O c1(C(=O)OCC=CCC)ccc(CC)s1 C1(C(=O)NC(c2ccccn2)CC)CC(O)CN1C(=O)CCC1CCCCCC1 C1(C#N)(C(=O)NCCC(C)N(C)C(c2ncc(F)cn2)=O)CC2CCC1CC2 c1(CC)cccc2[nH]c(C(N3CCC(CNc4ncn(C)c(=O)c4Br)C3)=O)cc12 N1(C(C(C)SCC)=O)CCC(O)(C(=O)NCCc2ncccc2C)CC1 c1(C(C)(C)C)cccc(CC(=O)NCC2CCCCN2C(c2csnn2)=O)c1 c1(CC(N2CC3C(NC(CN4C(C)CC4)=O)C3C2)=O)ccc2c(c1)COCC2 c1(C(=O)N)cc2n(n1)CCC2.N1(C(c2ncn(CC)c2)=O)CCC(CO)(C)C1 Cc1ccc(O)c(CC(N2CC(C)(NC(c3ccn(C4CC4)n3)=O)C2)=O)c1 CCC(CC)C(=O)NC1COCC1NC(=O)COc1ccccc1C(F)(F)F c1(NC(=O)CCC2CC2(Cl)Cl)cccc(CNC(C2C3CCCCC23)=O)c1 C(CC(=O)NCCCCNC(C1CC(F)(CO)C1)=O)(OCC)OCC C=Cc1ccc(C(=O)NCC(C)(CC)C(=O)NCc2csc(C)n2)cc1 c1(C(c2n(CC)nnn2)Nc2cc(C)cnc2C)c(F)cc(C)cc1Br N1(C(CC(CC)N(C)C(C2CCC(=O)N(C)C2)=O)=O)CCC12CC(C(N)=O)C2 N1(C(C(C)N(C(C2CC(CCC)C2)=O)CC)=O)CCCC(O)(CC)C1 C1(C(N2C(CNC(CCCC#C)=O)CCC2)=O)CCC(O)CN1C Cn1[nH]c(=NC(C2CC3CCC2CC3)c2nnnn2-c2ccc(F)cc2)cc1Br N1(C(c2ccc(CNC(C3CCC(F)CC3)=O)nc2)=O)CCS(=O)(=O)CC1 C1(CNC(c2c(C)coc2)=O)CCCC(CNC(C2CCN(C)C2C)=O)C1 c1(C(C)NC(N(CCC(C)CO)C)=O)cn(C)c2cc(Cl)ccc12 c1(N2CCCC(CNC(c3ccon3)=O)CC2)nc2c(cc1[N+](=O)[O-])CCCC2 C(=O)(C1=C(Cl)CCC(C)C1)N1CC(CC(C)C)C(NC(=O)Cc2cncnc2)C1 C(=O)(N1CCC(C(=O)NCc2nc(=O)o[nH]2)O1)c1cnc(C)s1 N1(C(Cn2c(C)ccn2)=O)CC(CC(=O)NCC(O)C2CC2)CC1(C)C C1(NC(=O)C(c2ccncc2)O)CCN(C(c2cnc(Cl)s2)=O)CC1F C=CCCCCC(=O)NN1CCCC1C(N1CC2CC1C1CC21)=O Cc1cc(C(=O)NCC(C2CCCCC2)NC(C2CCSCC2)=O)cc(N)c1Cl C(CC(C)(C)CC(=O)N1CCCC1CN(C)C(c1nnc(C(C)C)s1)=O)OC c1(N(CCC(=O)OC)C(=O)CC2CC3CC3C2)ccc(Br)cc1 c1(OC)cc(OC)c(S(=O)(=O)N2C3CCC(C3)C2CO)cc1Cl C=CCC(C)(CC)C(=O)NCCNC(c1ccon1)=O Cc1nc(C(=O)NCCCNC(C2C(C(F)F)C2(C)C)=O)sc1C c1(C(=O)N)ccc2nnn(C)c2c1.CC(C(=O)NC1CCC1)OCCN(C)C c1(C(C)(C)C)ccc(-c2nc(Cn3cnnn3)n(C34CC(C3)C4)n2)cc1 CC1CC(NC(=O)CCF)CCN1C(c1ccc(Sc2cnc(=N)[nH]c2)cc1)=O c1(OCC#C)ccccc1C(c1nnnn1C)NC(C)Cc1cccc(Cl)c1 c1(NC(CC2N(C(C3=C(C)OCC3)=O)CC2)=O)cc(C)c(O)cc1C C1(NC(=O)NC(CCC)C(=O)N)CN(C(=O)OC(C)(C)C)C2(CCC2)C1 C(=O)(C#CC(C)(C)C(F)F)N1CCCC(NC(c2ccc(C)cc2C)=O)CC1 c1(C(CNC(=O)COCc2ccco2)(F)F)cccc(C(=O)O)c1 C=C(CNC(C1CCN(C(=O)C2C(C)(C)C2(C)C)O1)=O)c1ccccc1 C(=O)(C1=C(Cl)CC1)NC(CC)C(=O)Nc1cncc(F)c1 C1(C)(C(=O)NC2(CF)CN(C(CCSCCCC)=O)C2)CCN(C)C1=O N1(C(C(CC)NC(C)=O)=O)CCCC2CN(CC3CCCCCC3)CCC12 c1(C(=O)NC2CCCC(NC(C3(c4cc[nH]n4)CCC3)=O)C2)cnn2ccsc12 C#CCC(CC#C)C(=O)N1CCN(C(c2c(C)noc2C)=O)CC1CC(C)(C)C Cc1cc(CN2CCOC(CC(=O)Nc3sccc3C#N)C2)cc(Cl)c1 N1(C(=O)CC23CCCC2C3)CCCCC(CNC(c2coc(C3CC3)n2)=O)C1 C(=O)C1=C(C)OCCS1(=O)=O.C#Cc1cc(C(=O)NCC2CCC2)ccc1C.N N1(C(C(c2cccc(C)c2)=O)=O)CCN(C(=O)CC(F)(F)Cl)C2CCCC12 C1(CC=O)CCC(F)(F)CO1.N1(CCC(N2CC(CC)C2)=O)C(=O)CCC1=O.N CN1CCn2ncc(Cn3cc(-c4cc(F)c(F)cc4N)nn3)c2C1 c1(NC)ccc(C(N2CCCC(CCNC(C3CCC(=O)N3)=O)C2)=O)cc1F N1(C(CCC(=O)N(C)C)=O)CCC(O)CC1CNC(c1ccc(C#N)[nH]1)=O C(C(F)C(=O)N1CCCc2ccnn21)C1CN(C(c2ccncn2)=O)C1 c1(C(N(CC(O)CNC(=O)CC2COC(=O)N2)C)=O)cccc(Cl)c1 N1(C(CC(CC)C)=O)CC2CCC1C(NC(=O)COc1cc(C)ccc1F)C2 c1(CNC(C2(C#C)CCCC2)=O)nnc2n1CCN(C(=O)C(F)C1CCC1)C2 C1(CNC(c2csc(C)c2C)=O)CCN(C(=O)CC#N)CC1C C1(NC(c2nc(C3CC3)cs2)=O)CCN(C(=O)Cc2cccs2)CC1 c1(CN(Cc2ccc(C3C(C)C3)o2)CC)cc2cc(F)c(F)cc2nc1Cl N1(CCC)CCCC1C(=O)NCC1(O)CCC1.c1(CC=O)csc(C)c1.N C1(CNC(C(CCN(C)C)NC(c2c[nH]c(C#N)c2)=O)=O)CCCCC1(C)C N1(C(CC2(C)CCOCC2)=O)CCC(C2CN(C(C3CCC4CC34)=O)C2)CC1 CC1=C(C(=O)NCC(c2ccc(F)cc2)NC(=O)CCCN2CCCCC2)CC1 N1(C(=O)CC2CC3(CC3)CO2)CC(C2CCN(C(=O)C(O)CC(F)(F)F)CC2)C1 C1(CNC(=O)C(=O)Nc2n[nH]c(C3CC3)n2)CCC(C(F)(F)F)CC1 N1(C(COc2ccc(C)cc2)=O)CC(F)(F)CC1(C)CNC(C1CCCC1O)=O c1(NC(CC)=O)cncc(C(=O)NC2CCCC(C)C2)c1.C1(C(=O)N)CCC1 c1(C(N2C(CNC(c3n(CCC)ncc3)=O)C=CC2)=O)cnc2n1CCCC2C N1(C(C(C)(C)O)=O)CC2(CO)CC1(C(=O)NC1(CC3CC3)CC1)C2 N1(C(C(c2cc(Cl)cc(Cl)c2)=O)=O)CC2CCC1CN2C(=O)C1=NOCC1 c1(OC)ccccc1C(CC)NC(=O)CS.n1(CC=O)cnnc1.CC(C)C C(=O)(CCC(=O)c1ccc(C)s1)NCC(CNC(=O)CC1CCCO1)OC Cn1c(C(=O)NC2CCCC2C)cc2ccccc12.C(C(F)(F)F)=CC=O.N C1(SC)CCCCC1C(=O)N(C(C1CCN1C(C)(C)C)=O)C.C1(C)CC1 N1(C(c2cncc(C)c2)=O)CC(C2(NC(=O)CC(O)C3CCCC3)CC2)C1 C=CC(CC)CC(=O)NC(C)CNC(c1cnc(-c2ccoc2)[nH]c1=N)=O C(=O)(C(C)CS(C)=O)NCC1(NC(Cc2cc(C)ns2)=O)CCC1 C1(NC(C2(COc3ccccc3)CCC2)=O)CC2(C1)CC2N=c1[nH]ccnc1F C1(NC(C(CC)=CCCC)=O)CC2(CCCN(C(c3ccc(Cl)c(Cl)c3)=O)C2)C1 C=C(C)C1OCCC1C(=O)NCCNC(c1noc(-c2cccc(Cl)c2F)n1)=O c1(C=O)cccc2ncn(C)c12.c1(CC)nc(C(=O)NCC2CCCC2)n[nH]1.N N1(C(C2(CC#C)CC2)=O)CC2(NC(=O)C(=O)NC)CCC1CC2.C1CC1 N1(C(c2cc(CC)c(C)s2)=O)CCCCC(N(C)C(c2cnn3ccsc23)=O)C1 O=S(=O)(c1ccc(NC(c2nnnn2C2CC2)CC2CCOC2)cc1)C(F)F Cc1cc(C(N2CCC(C)(c3cn(C4(C(N)=O)CC4)nn3)CC2)=O)cc(Cl)c1 c1(C(=O)NC(CNC(C2N(CCC)CCC2)=O)C)cncc(C(F)F)c1 C(=O)(CS(=O)(=O)N(CCCNC(=O)CCSC)CC)NC1CCCOC1 c1(C(=O)NCCCNC2C(C)CCNC2)ccc2c(c1)OCCO2 C1(NC(Cc2ccc(SC)cc2)=O)CCN(Cc2cccc(C#N)c2)CC1(C)C C(=O)(C1CCc2ccccc21)N(C1CC(C(N2CCc3ccccc3C2)=O)C1)C c1(OC)cnc(C(=O)NC2CC(C)N(C(=O)C=Cc3nccs3)C2)c(OC)n1 C1(F)(CNC(c2c(C)oc(CO)c2)=O)CCCN(C(=O)C(c2cncn2C)O)C1 Fc1c(C(c2nnnn2CC(F)F)NC2CCSCC2)cccc1Br C1(CNC(=O)Cc2ccc(Cl)cc2)CN(C(C2CCC2(F)F)=O)CC12CC2 O=S(=O)(c1ccc(Br)cc1N1CCCC(CF)C1)NC(CO)CC(F)(F)F c1(CNC(c2ccc(Oc3ccc(F)cc3)nc2)=O)ccccc1SC(F)(F)F N1(C(c2cnn(C(C)C)c2Cl)=O)CC(C2CC2)C1.c1(C(=O)N)cnn(C2CC2)c1 Cc1nc2ccc(C(N3CC4CC4(CNC(=O)C(C)(F)F)C3)=O)cc2n(C)c1=O c1(C(=O)NCC(C)(CO)NC(=O)C#CC2CC2)ccc2ccc(Br)cc2n1 C(C(O)C(=O)N(C)Cc1ccsc1)NC(C(C)OC(C)=O)=O N1(C(c2c(CC)occ2)=O)CC2(C1)CN(C(c1ccc(Br)o1)=O)CC2CO c1(CC)nc(NC2(C3CN(C(c4cnc5n4CCS5)=O)C3)CC2)cc(C#N)n1 c1(OC)ccc(OC)c(CC(=O)NC2(C)CN(C(C3CCOCC3)=O)C2)c1 CS(=O)(=O)c1ccccc1C(CO)NC1CCCCC1c1ccc(Cl)cc1 CCCCCCOCC(=O)NCC(C)(C)CNC(=O)C=CC1CCCO1 c1(C(=O)NCc2c(C(N(CCS(C)(=O)=O)C)=O)n[nH]c2)cnc2ccccn12 Cc1ccc2n1CCN(CC1CN(C(=O)CSc3ccccc3)C(=O)CO1)C2C C#Cc1ccc(C(=O)NC(C)C(C)(C)C(=O)N2CCCC(N3CCC3)C2)cn1 CC(N=[N+]=[N-])C(=O)N1C(C(=O)NCC2CNC(=O)O2)CCC1C1CC1 c1(OC)ccc(CNC(C)(CC(C)C)C(=O)O)c(OC(F)F)c1OC CC1(O)CC2(CCN(C(C3COCCN3Cc3cnco3)=O)CC2)C1 c1(CC2(C(=O)NCC3CCN(C(CN(CCC)C)=O)C3)CC2)ccccc1Cl c1(C(N2CCN(CCCNC(=O)CO)CC2)=O)ccc2c(c1)COC(=O)N2 CC1OC2(CO)CC1(C(N1CCC(NC(C3(C)CC3)=O)C1C1CC1)=O)C2 C1(C)(CC)CCC(NC(=O)C(C(C)C)NC(c2ncnc(O)c2F)=O)CC1 C1(NC(C(c2cn(C)nc2)(F)F)=O)CN(C(c2cnc(C3CC3)[nH]2)=O)CCC1F N1(C(CCC(=O)NCC)=O)CCC(C(=O)NC2CCCC2)C1(C)C.N(C)C.C CC1CC(NC(c2ccccc2CC#N)=O)CCN1C(c1n[nH]c2c1COC2)=O CC1(F)CN(C(c2ccoc2)=O)CCN(C(c2ccccc2OC(F)F)=O)C1 c1(C(=O)NCC2(NC(C3Cc4nccn4C3)=O)CCC2)ccc2ncccc2c1 N1(C(CCOCC)=O)CCC2(NC(c3ccc(F)cc3SC)=O)CC2C1 c1(C(N(CC(CC)NC(=O)CNC(=O)NC)C)=O)coc2cc(F)ccc12 N1(C(C(C)Sc2ccco2)=O)C(=O)CCC1COC(c1ccc(C)cc1)=O C(=O)(C1=CCCOCC1)NC1(C)CN(C(=O)C(c2ccc(Cl)s2)=O)C1 C12(C(=O)NC3CCC(NC(C4CCC(C)(CC)O4)=O)CC3)CC=CCN1CCC2 n1(CCC)c(=O)nc(O)c2cc(NCC(O)COCc3ccccc3)cnc12 c1(C(=O)NCC(CC=C)NC(=O)C(C)OC2CCOC2)cnc(CC)nc1 CC(C(=O)NC1CCCCC1NC(c1ncoc1C1CCCCC1)=O)C(C)(C)C N1(C(c2cn[nH]c2)=O)CC(NS(=O)(=O)c2ccccn2)CC(F)(F)C1 C(=O)(C(C1CCC1)OC)NCCN(C(=O)CC1(OC)CCC1)CC C(=O)(C1CCCc2nc(C)[nH]c21)NC1CC(NC(C2CN(CC)C(=O)C2)=O)C1 c1(C(N2CC(CCOC)N(C(=O)CC(O)C(C)C)CC2)=O)ncn2ccccc12 N1(C(C(CC=C)NC(=O)OC(C)(C)C)=O)CC2CCCC(C1)C2O C=CC(F)(F)C(=O)NCC(C)(C)NC(c1cc(I)on1)=O c1(C(N2CCC(CCOC)(C(=O)NC3(CF)CC3)C2)=O)cc(OC)cnc1F C(C(CCC)CCC)NC(CCN(C(=O)C1=CCCSC1)CC#C)=O N1(C(COC2(C)CN(C(C(CCC)C#N)=O)C2)=O)Cc2ccnn2CC1C CC(C)(CO)C(=O)NC1CCC(OC2CCCCC2C)CC1.C(=O)C.C1CC1 Cc1cccc(C=CC(N2CC(C)CCC2C(=O)N(C)CCO)=O)c1 c1(C(=O)OC(c2cc(F)c(F)c(F)c2)C)ccc2c(c1)OCCC2S(N)(=O)=O C(=O)(C(O)C(C)(C)CC)N1CCC(NC(c2cccc(C(C)=O)c2)=O)C(CO)C1 S(=O)(=O)(c1cccc(=NCc2sc(C)cc2Br)[nH]1)NCCC(CC)C CC(C)C(CC(=O)NC1CC(CNC(=O)C(=O)N(C)C)C1)c1ccccc1 C#CCCCCCC(=O)N1CC2CC(NC(C3C4CCC(F)(F)C34)=O)C1C2 N1(C(c2cc(SC)c(C)o2)=O)CCC2CCCN(C(c3ccncc3N)=O)C2C1 N1(C(C(CNC(C(CCCC#C)C)=O)(F)C(C)C)=O)CCc2nc(O)[nH]c2C1 N1(C(C(C2CC2)OCC)=O)CC(C)(C(N2C3CSCC2C3)=O)CC1(C)C CC1C(=O)NCCCN1C(=O)CC1CC(O)CN1C(=O)COCC1CCC1 c1(CS(=O)(=O)N)ccc([N+](=O)[O-])cc1.C1(NC(C2CCCC2)=O)CCCOC1 C=CCC(F)(F)C(=O)N1CC(C2(NC(C3CCN(CCO)C(=O)C3)=O)CC2)C1 c1(C(C)C)ncsc1C(=O)NC(C1CCN(C(=O)CCc2cc[nH]n2)C1)C C(C(CNC(c1ccc(C)c(F)c1)=O)S(C)(=O)=O)NC(C(C=C)C)=O C1(NC(c2c(C)[nH]cc2)=O)CCC2CCN(C(C3CCC(N(C)C)C3)=O)C12 N1(C(C(CC)c2ccccc2)=O)CCN(C(c2oc(C)cc2C)=O)CC1C(F)F c1(C(N2C(C(=O)NC3(C#N)CCCC3)CCC2)=O)ccc(Br)cc1CO c1(CC)ncc(C(=O)NC2(C)CC(NC(=O)C(O)c3ccco3)C2)[nH]1 CC(CCC(=O)NC1CC(C)(NC(=O)CC2CC23CC3)C1)N(C)C N1(C(C(CC=CC)C)=O)CCCC(NC(=O)Cc2noc3ccccc23)CCC1 C1(C2CCC2)(C=O)CC1(F)F.CC1(C)CC(C(=O)NC2(CC)CC2)CCO1.N C1(NC(COC(CC)C)=O)CC2CCCC(C1)N2C(c1c(N)cccc1Cl)=O C(=O)(C(CC1CCC2CC12)N1CCC(Cc2ccnn2C)C1)NC(CC)(C)C c1(CN(c2ccc(-c3ccnc(C)c3NC)cc2)CCC)ccc(Cl)cc1OC CC1CC(C(=O)NCCc2ccco2)N1C(c1ccsc1)=O N1(C(C2CCCN(C)C2)=O)CCN(C)C(CNC(c2occc2Br)=O)C1 C1(C(=O)NC2(CNC(C3(C)CC3(F)F)=O)CCC2)Cc2ccccc2S1 c1(CCCC(=O)NCC2C(NC(CC(C)OC)=O)CC2)ccc(F)c(F)c1 CCCC(CCC)CC(=O)NCc1ocnc1-c1cn(C(C)C(=O)OC)nn1 C1(C(=O)NC2(C(N3CC(c4nncs4)C3)=O)C(C)(C)C2)CC2CC(=O)C1O2 c1(NC(CC#C)C)cccc(OC2CCCC2)c1 C1(CCNC(C(c2ccsc2Cl)C)=O)CCCCC1CN1CCCC1CO C(C(C)(O)CCO)CC.N1(CC(=O)OC)CCOC1=O.C1CC1CC(=O)N.C CC(O)CC(C)(C)CNC(=O)CC(C)(C)CNC(C1CC=CCO1)=O c1(C2CN(C(C)=O)C2)ocnc1C.[nH]1cc(C(N)=O)cn1.C1(C=O)CCC1.N C1(NC(CCC=CC)=O)CCCN(Cc2cn(C(C)C)nn2)C1 C(CN=c1[nH]c(=NCC=C(Cl)Cl)[nH]c2c1CSC2)C1OCC(C)(C)C1 Cc1cc(Br)c(C(=O)NCCCCNC(C2CCC2(C)C)=O)nc1C Cc1nn(CC(F)(F)F)c(C)c1CN1C(C(=O)NC(C)(C)C)CCC1C CC1CCC2(CCC2)CN1C(=O)NC1CC2CCC(C1)C2=O c1ccccn1.C1(OC)CC(C(=O)NC(C2CC(NC(=O)CCS)C2)C)C1 CCCCCCC(F)C(=O)N1CCC(NC(c2cc3c(nn2)CCC3)=O)CC1C N1(C(CCC(CC)C)=O)CCC2CN(C(c3cc(=O)cc(Cl)[nH]3)=O)C2C1 c1(C(=O)NC2(C)CCC2)ccc([N+](=O)[O-])o1.c1(C=O)cc(C(F)F)ccc1F.N C1(CCCCCC)CCCN(N(C)CCCC(=O)NC(=O)C(F)(F)F)C1 C12(NC(CCCC(=O)NC(C)(C)C)=O)CCC(CC1)C2(C)C C1(C(=O)NCC(C)F)C2CCC(C2)N1C(=O)Cc1cn[nH]c1 c1(CN2C(C(N3CCC4(CCC4)C3)=O)CCCC2)cc(F)cnc1Cl c1(C(N2CC(C)(NC(C3CC(C(F)(F)F)CO3)=O)C2)=O)ncncc1F C(=O)(C(O)CCNC(=O)C(CNC(=O)C(C)N=[N+]=[N-])OC)OC S(=O)(=O)(c1ccc(C#N)c(N2CCc3nc[nH]c(=N)c3C2)c1)NCCC(=C)C Cc1ncccc1CC(=O)NCC(C)C(=O)NC(c1c(C)n[nH]c1C)C N1(C(c2ccsc2Cl)=O)CCC2C(C1)CN2C(=O)CCN1CCCC1 C(CC(C)C(=O)NC(Cc1cnc[nH]1)C(=O)NC1CCN(C)CC1)=CCC CC1(C)CCC(C(=O)O)(NC(=O)OC(C)(C)C)C1.c1cc(C#N)ncn1 c1(CC=C)cccc(C(N2CC(C)C2C(=O)NC)=O)c1.C1CC(=O)N(C)C1 c1(-c2cc(C(N(CCNC(C=CCCC)=O)CC)=O)on2)c(Cl)cnn1C C1(CCC(=O)N(C2CN(C(c3cnc(Cl)s3)=O)CC2F)C)CCCCCC1 c1(C(=O)NCC(CC(C)C)NC(C=CSC)=O)ccc(Br)c(O)c1 c1(C(C)N(C(=O)C(n2cc(C3(c4ccccc4)CC3)nn2)C)C)cnnn1C C1(N)(C(=O)NCCC(C)(C)c2ccccc2)CC(F)(F)C1 C1(NC(C2CC(C)(NC(CC(=O)OC)=O)C2)=O)CCC2CCC1C2 c1(C(=O)NCc2cc(C(=O)NC(c3onc(C)n3)C)no2)cccc(O)c1 C1(NC(C2CC2(F)F)=O)CCC12CCN(C(c1ccc3ccncc3c1)=O)CC2 N1(C(Cc2ccc(C#N)cc2)=O)CC2CCCC(C1)N2C(=O)C(F)F C1(O)(CNC(CC2(C=C)CC2)=O)CCN(C(c2ccc(-n3cnnc3)cc2)=O)C1 c12c[nH]nc1C(c1nnnn1CCCF)NCC2.C(C)SC.CC C1(CN(C(C(C)N(CCC)C(c2cncnc2)=O)=O)C)CN(C)CCO1 Cc1nccc(C(N2CCN(C(C3(C)CCN(C)C3=O)=O)CC2)=O)c1N CC(CC(=O)NC1CCCCN(C(c2ccc3nccn3n2)=O)C1)C(C)(C)C Cc1c(NCc2ccccc2-c2ccncc2)ncnc1NC1CCC2CC12 c1(C(=O)OC)n[nH]c2c(C(=O)NCC(O)C)cccc12.C1(C=O)CC=CCC1.N C12(NC(CCC(=C)Cl)=O)CC(CNC(c3cnc(SC)s3)=O)(C1)OC2C N1(C(c2c(C)[nH]cc2)=O)CC(C)CN(C(c2c3c(nn2C)CCC3)=O)C(C)C1 N1(C(C(CCOC)(C)C)=O)C2CCCC1CC(NC(c1cccc(O)n1)=O)C2 C(=O)(CN=c1[nH]c2ccccc2s1)N1CCN(C(CCCNC(C)=O)=O)C2C1C2 c1(C(N2CCC(C)(NC(C(C)n3cccn3)=O)C2)=O)cnc2c(=O)[nH]ccc2c1 C1(NC(C2CCC(C)(C)CO2)=O)COC2(CCN(C(=O)CCF)CC2)C1 c1ccccc1[N+](=O)[O-].CC1(NC(=O)Cc2cc[nH]c2)CC(NC(=O)CO)C1 Cc1c(C(=O)NCCNC(C2CC3CCCC3C2)=O)cc(C2CCCC2)n1C C(=O)(CC(O)CC(C)(C)C)N1C(C(=O)NC(C2CCC2)C)C=CC1 Cc1ncc(C(=O)N)n1C.C1(C(N)=O)CN(C(=O)Cc2nc(C3CC3)n[nH]2)C1 Cc1ccc(CC(=O)NC(C2(CNC(=O)Cc3cc[nH]n3)CC2)C)cc1O Cc1cc(=NCC(C)C#N)[nH]c(N2CCC(CN(C)CC3CC3)C2)n1 C=C1CCN(C(=O)OC(C)(C)C)C(C(=O)NC2(COC)CCCCC2C)C1 Cc1cc(CNCC(O)Cc2ccc(Cl)cc2)c2ccccc2n1 Cc1cc(O)c(C(C)C)cc1C(N1CC2CCC1CN2C(C1CCOC1C)=O)=O N1(C(C2N(C(c3cc(C)sc3C)=O)CCOCC2)=O)CC2(CCN(C)CC2)C1 CC1CCCC(N(CCO)C(c2ccccc2OCC(F)F)=O)C1 C12(C(N3CCCC(N(C(COCC#C)=O)C)CC3)=O)CCC(N=[N+]=[N-])C1C2 C(=O)(C1=CCC(F)(F)CC1)N1CCC(O)C1.C1(CC(=O)N)CC2(CCC2)CO1.C N1(C(COC(CC)(C)C)=O)CCC(C)(C)C1.C1(N(CCC=O)C)CCCCC1.N C(=O)(CCCC(=O)NC1CCC(NC(c2ccc(C)c(F)c2)=O)CC1)NC Cc1cc(Br)cc([N+](=O)[O-])c1.c1(CCC)cnc2cc(Br)ccc2c1.C1(C=O)CCCCC1 c1(NC(C2CCN(C(C(CC)n3ccnc3)=O)C2)=O)ccc(OC)nc1 C(=O)(CC=CCNC(=O)Cn1cccn1)NCC(c1nccs1)C c1(CC=O)cc(C(F)(F)F)nn1C.C(=O)(C(C)CC1CCC1)NCCCC.N CC1(C(=O)NCC2(Nc3nccc(-n4ccnc4)n3)CCOCC2)CC=CCC1 C1(CNC(=O)C=CCF)C2CN(C(=O)Cc3cc(C(F)(F)F)n[nH]3)CC12 N1(C(C2CCN(C)S2(=O)=O)=O)CC2CCN(C(c3ccc4c(n3)CCC4)=O)C2C1 c1(C(=O)NC2CC(C)(NC(c3c(C)scn3)=O)C2)cccnc1C1CC1 N1(C(C(C)NC(=O)NC)=O)CCC2(CCC2)C1.c1(C=O)ccc2ncccn12.N n1(CCC)cc(C(=O)NCCC2(NC(=O)C(n3nccc3C)C)CC2)nn1 n1(CCC)nc(C)c(C(=O)N)c1C.C1CCN(C(C2C3CCC(=O)C23)=O)CC1.C CCCC(CNC(c1occc1C(C)C)=O)C(=O)N1CC(CC(=O)OC)C1 N1(C(c2cc(OC)c([N+](=O)[O-])cc2)C(=O)NC)CCN2C(=O)CCCC2C1 Cc1cc(NC(c2cnc(Cl)cc2N)=O)ccc1NC(C1(C)CC=CCC1)=O C1CC(C)(C)CN1C(=O)CN1CC(=O)NC1=O.C1(CC)CCC(C(=O)N)O1 N1(C(C(C)=C2CC2)=O)CCC(C2CC2)C1C(=O)NC1(CCCCO)CC1 C(=O)(C(CC(C)SC)N(c1cccc(C2CCCC2CO)c1)C)OC CC1C(=O)CCC(C(N2CCCC(NC(C3CC3(C)C)=O)CC2)=O)C1(C)C CN1CC2(CCN(C(=O)C(CN=[N+]=[N-])NC(c3coc(C(F)F)c3)=O)CC2)C1 C12(C(N(CCCNC(c3c(CC)[nH]nc3Cl)=O)CC)=O)CCCCC1OCC2 c1(C2(C(=O)NC(CC)CN(C)C(C3C=CCS3)=O)CC2)ccccc1Cl C(C(CC(C)C)C(=O)N1CCC2(CSC2)C1)NC(c1n(CC)ncc1)=O c1(COCC(=O)N(C2CC(SCC)C2)C)ccccn1 n1(CC(=O)NC(C(C)C)CCN(C)C(C2CCCN2C)=O)nc(O)ccc1=O C(=O)(C1=CCN(C(=O)CSC(F)F)C1)NC1(CC)CCOCC1 Cc1ccc(C(N2CCC(CNC(=O)CCc3ccon3)C2)=O)c2c1NCCC2 CC(CC(C)(F)F)C(=O)NC1CN(C(=O)CCN2CCN(C)CC2)CC1(C)C c1(C=O)cc(C#N)c(O)nc1N.CC(C(=O)NCC1(C)CCC1)N1CCC1.N c1(C(N2CC(F)C2)=O)ccc(F)cc1O.c1(C(=O)NC)cc(C2CCOC2)[nH]n1 C=CCCCCN(C(=O)CC1CCN(C(C2(OC)CC2)=O)C1)C C(C(C)(C)C(=O)NCC1C(CO)C1(C)C)NC(Cc1nc(C)[nH]n1)=O C1(N=[N+]=[N-])(C(=O)NCC(C(C)(F)F)Cl)CCN(C(=O)CC2OCCO2)C1 C(=O)(C1c2c[nH]nc2CN1C(c1cnco1)=O)NC(C=C)C1CCC1 c1(C(=O)NCC(CCC)NC(c2cc(CCOC)on2)=O)cc2n(n1)CCO2 N1(C(C2CCCN(CCC(=O)N(C)C)C2)=O)CC2CC1CCN2C(C1CCC1)=O C1(C(=O)NC2CC(C(=O)OC)CC2O)CC(P(C)(C)=O)CN1 CCCC(O)CCN=c1[nH]c(=NC(C)CCCC2CC2)c2ncccc2[nH]1 Cc1cc(C(N2CCOCC2CNC(c2cncc(C(N)=O)c2)=O)=O)nc(O)n1 C1(N(C)C)CCCN(CC(N2CC(C)(NC(C3CC3F)=O)C2)=O)C1 c1(COC)cc(-c2cn(CC)nn2)no1.c12cncn1CC(=O)NOCC(=O)N2 CCCCC(C)C(=O)NCC(C(C)(C)C)NC(c1nsnc1O)=O C(C)(CCC(=O)N1CC(CNC(=O)CC2(n3cccn3)CC2)C(O)C1)SC C1(C(=O)NCc2cccc(C(N(C)CCc3ncon3)=O)n2)CC12CCOCC2 C#CC1(C(=O)NCC2CC2NC(=O)CCC)CCCC1.C1CCC(C)CC1.O C(=O)(C(CCNC(c1sccc1Cl)=O)NC(=O)OC(C)(C)C)OC Cc1cc(C(N2CC3(CCC3NC(c3cnc(S)n3C)=O)C2)=O)cc2nc[nH]c12 CCCCC(O)C(C)C(=O)N1CC2CC(C1)N2C(c1ccn2cncc2c1)=O c1(COC)cc(N2CC(O)(CCNC(C3CCOC3C)=O)C2)ncn1 S(=O)(=O)(c1cccnc1NCc1cccc(CO)c1)NC1(C)CCC(F)(F)CC1 C(C(CNC(C1CCCCCC1)(c1nnnn1C1COC1)C)C(C)C)OC Cc1c(CNC2CN(C(c3cc(O)cc(O)c3)=O)CC23CC3)ccnc1Cl CC(C(=O)NCC1(N(C)C)CCC1)N(C(=O)Cc1cnc[nH]1)C CC1CC(NC(=O)C2=C(Cl)CC2)CN1C(c1ccc(CC2CCC2)cc1)=O c1(NC(CCNCc2cc(C)[nH]c2C)=O)cccc(S(=O)(=O)N(C)C)c1 c1(N(CCCNC(C2(O)CCOC2)=O)CC)cc(Oc2ccccc2)ncn1 c1(C(=O)NCCOC2CN(C(COC(C)(C)C)=O)C2)scc2c1OCCO2 N1(C(CSSC)=O)CCCC(C2CCN(C(=O)Cc3ccnn3C3CCC3)C2)C1 CCCCCCCCCC(=O)N1CCCCC1CCCNC(C1(C)CCCC1)=O N1(C(C(CSC)(C)C)=O)CC(C(=O)NC(C)(C)CCF)C(C2CC2)C1 c1(C(N(CC)C(C)C)=O)cccc2sccc12.N1(C(C)=O)CCOCC1C(=O)N Cc1cc(C(N2CCC(NC(c3cncc(Cl)c3Cl)=O)C2C)=O)cc2nc[nH]c12 N1(Cc2cccc(-c3nnc(C)o3)c2)CCC(C2CCN(C)C2)CC1 CCC(C)(CO)C(=O)NCC1C(CNC(c2cccc(O)n2)=O)C1(F)F N1(C(C(C)=CC)=O)CC(N(C(=O)Cc2cc(C3CC3)no2)C)C(O)C1 CC(C)(F)CCC(=O)N1C2CCC(C2)C1CNC(=O)CCC1CCOC1 N1(C(c2c(Cl)c(C)nn2C)C(=O)NCCOC)CCC2(CCN(C)C2)C1 C1(NC(c2n(CC)c(O)nc2)=O)CCN(C(c2cncn(C)c2=O)=O)CC1O c1(C(=O)NC23CCN(C(c4cnc(Cl)s4)=O)CC2C3)cccc2cc(O)ccc12 C(CC1=CCCCC1)NC(C1CN(C(C2CCCO2)=O)CCN1)=O CCCCC(CC)C(=O)NCC(C1(O)CN(C(=O)CCCC(C)CC)C1)(C)C N1(C(C(C)C)=O)CCCC(C(N2CC(NC(=O)CCc3cncs3)C(C)C2)=O)C1 CC(CC(=O)NC1CC(CNC(=O)Cn2cnnc2)C1)C(=O)c1ccccc1 C1(NC(=O)CC2SCC2)CC(CNC(=O)CS)C(O)C1.c1cccs1.C N1(C(CC(CC)CC)=O)CC2CC(C1)N(C(=O)C(CC)OC1CCCC1)C2 C(=O)(C(F)C(C)CNC(=O)CCc1cn[nH]c1)NC(C)Cc1ncn(C)n1 Cc1cc(C(=O)NCC2(C)CCN(C(c3cc(C)c(C)nn3)=O)C2)nc(C)n1 c1(C(=O)NC(C2CN(C(c3cnco3)=O)CCO2)C)ccc2c(n1)CCC2 CC(N)C#CC(=O)OCC(=O)NC1CCN(Cc2ccccc2)C1 CC1(C)CN(C(=O)C=CCN2CCC2)CCO1.n1(C(C=O)C)cc(Cl)cn1.C CCC(CCC(=O)NC(CCN(C)C(c1cncc(OC)c1C)=O)C(C)C)OC C(=O)(C1=C(Cl)CCOC1)N1CC(N(C(CCCn2ncc(C)c2)=O)C)C(C)CC1 C(=O)(C(C(C)(F)F)c1ccccc1)N1C(CNC(COC(C)=O)=O)CCC1 C(=O)(C(C)Cn1cccn1)NC(CC)CNC(C1(CCN=[N+]=[N-])CC1)=O c1(C=O)ccc2c(c1)OCC(=O)N2.C(=O)(C(F)C(=O)N)OCC.C1COCC1 c1(C2(C(N(CCNC(c3c(CC)occ3)=O)C)=O)CC2)cccc(F)c1F c1(C(C(=O)NC(CNC(c2ncn(CC)n2)=O)C)O)ccc(Cl)c(Br)c1 N1(C(C(C)NC(=O)NC)=O)CCCCC1C1CCN(C(=O)CC2CCCOC2)C1 C(C)(C(=O)N)(C(C)C)OC.C1CC(F)(F)CN1C(=O)CCc1csc(=N)[nH]1 Cc1cc2nc(Cl)nc(N3CCC(CNC(=O)CC4CCC5CC45)C3)c2s1 C1(CC)CN(C(C2(C)CCNC2=O)=O)CC1NC(=O)C.C(=O)CC(C)(C)C CC1(C)CC(C(=O)NC(C2CCCC2)C)CO1.c1(C=O)nc[nH]c1C(F)(F)F C(=O)(C1CC(=O)N(C)c2ccccc21)N(CCNC(CC(CC)C(C)(C)C)=O)C C#Cc1cncc(C(=O)NC2CC2NC(=O)C(c2ccccc2)C2CC2)c1 N1(C(c2c(C)cn(C)n2)=O)CCC(CNC(C2CC(F)C(=O)N2)=O)CC1C c1(C(N2CC(OC)C(NC(C3CNC(=O)N3)=O)C2)=O)cc2ccnn2cn1 C1(NC(C2CC(CCO)C2)=O)CC2CCC1N2C(=O)Cc1cc(Cl)cc(Cl)c1 c1(C(N2CC3(CCN(C(C4C5COCC45)=O)C3)C2)=O)cc2c(s1)CCSC2 C(=O)(CC(O)CNC(C1(F)CCCC1)=O)NCC1CC(OCC)C1 c1(C(C)(C)NCC2CC2c2cccc(Br)c2)ccc(OCC(F)(F)F)cc1 C(=O)(CC(C)(C(F)F)N(C)C)N(C)CCNC(=O)CN1CCCCCC1 C1(C(C)C)CN(C(C23CCC(CO2)C3)=O)CCN1C(c1ccnc(CO)c1)=O C=CCCC(=O)N1CC(CC(F)C(=O)NC2CC(C)(CO)C2)C1 C1(CC)CN(C(c2cn(C3CCC3O)nn2)=O)CCN1C(=O)CCSCC(N)=O N1(C(CCCCC=C)=O)CC=C(C(C)(C)C(=O)NCCN(C)CCF)C1 C(=O)(C(O)C(F)F)N.C1(OCC(=O)NCCc2ccccc2)CC(F)(F)C1 N1(C(C(CO)NC(C(C)C)=O)=O)CC2(CCN(C(=O)C=CI)C2)C1 C(=O)(C(CC(=C)C)NC(C1CC=CCC1)=O)NC(CC#C)C(=O)NC C(=O)(CCCC1CC1)NC(CCN(CC)CC)C.n1(CC=O)cc(Cl)cn1 c1(N2CC(SC)C(N3CCCC3)C2)nc2ccsc2c(=NCC2(C)CC2)[nH]1 N1(C(C(C)OC)=O)CC2CCC2(CNC(c2ccnc(CN(C)C)c2)=O)C1 N1(C(Cc2cnc(C)s2)=O)CCCCC(NC(=O)C(C)Sc2ccc(Cl)cc2)C1 C1(C(N2CCC3CCC23)=O)CC(C2CCNCC2)CN1 Cc1ccc(C(N2CCOCC(NC(c3ccccc3F)=O)C2)=O)c(C(C)C)n1 N1(C(c2nc(C)sc2C)=O)CCN(C(C2(O)CC(CF)C2)=O)CC1C1CCC1 Cc1ccc(C(N2CCCC(N(C(C3CNC(=O)O3)=O)CC3CC3)C2)=O)nc1C CC(CC(=O)c1ccccc1F)C(=O)N1CCC(C(O)C(F)(F)F)CC1 C1(NC(c2c(C)ncc(C)c2)=O)CCCCN(C(=O)C(=O)Nc2ncc[nH]2)CC1 CC1CCSC1C(=O)N(CCCN(C)C(c1cc(C(C)(C)C)on1)=O)C CC1SCCCC1C(N1CCC(CCCCNC(=O)Cc2cnnn2C)CC1)=O C1(NC(C(COC)OC)=O)CC2CCC1N(C(=O)Cn1cnc(=N)[nH]1)C2 CC1CN(C(C2(C)COCCO2)=O)CC1NC(c1ccnn1C1CCCCC1)=O N1(C(C2(OCC)COC2)=O)CCCC(CCCc2ccccc2)C1 N1(c2nc(C)cc(OC)n2)CC2CCC(C1)C2NCc1cnc(C2CC2)s1 C(=O)(C1CC(C)Cc2c[nH]nc21)N(CCCNC(c1cc(OC)nc(F)c1)=O)C c1(NC(=O)NC2C(C)C2C)ccnn1C1CCOC1 N1(C(C2NC(=O)OC2)=O)CCC2(C1)CN(C(C1(C3CCCCO3)CC1)=O)C2 C1(NC(C(C)NC(N)=O)=O)CN(C(c2cccc3nccn23)=O)CC12CCC2 CCCCC(CC)C(C(=O)NCCCF)N1CCOC(C(F)(F)C(F)(F)F)C1 CCC(CNC(=O)C(=O)Nc1nc(-c2ccc(C#N)cc2)cs1)(CC)C(F)(F)F C(C(C)(C(=O)NCC1(F)CCC1)OC)OC.n1(CC=O)ncc(Cl)c1C.C N1(C(C2CCC(C)O2)=O)CC(O)CC1C(=O)Nc1c(Cl)cnn1C N1(C(c2cc(C(F)(F)F)no2)=O)CCC2(CCN(C(C3CC4CCC34)=O)CC2)C1 N1(Cc2n(C)nc(Br)n2)CCC2CCCC2CC1 C1(NC(c2c(CC)ccc(F)c2)=O)CN(C(C2CCNC2=O)=O)C2(CCC2)C1 c1(C(=O)NC2CC(NC(Cn3c(C)cnc3)=O)C2)ccc2[nH]c(=N)[nH]c2c1 C1(O)(CCNC(C=CC(C)C)=O)CCN(C(=O)C(C)Oc2ccccc2)C1 c1(SC)ccc(Cl)c(C(=O)N(C)CC2CCCN(C(=O)C(C)c3cc[nH]n3)C2)c1 c1(C(N(C2CCCN(C(=O)C(C)(C)c3cnco3)C2)C)=O)ccc(C2CC2)nc1 N1(C(CCN(CCCCC)C(C)C)=O)CC(NC(=O)C(C)CCCC)C(C)(C)C1 N1(C(CC(CC)SC)=O)CCC=C(C(=O)NCCc2nnc(C)s2)C1 c1(N(C)CC2CCN(C(CCCCN(C)C)=O)CC2)ccc(Br)cc1[N+](=O)[O-] S(=O)(=O)(CCC(=O)NC1CN(C(=O)C(F)C2CCC2)CC1c1ccccc1)NC C(C(N=c1[nH]c(Cl)ncc1[N+](=O)[O-])C(C)C)NC(C1CN(CCC)C(=O)C1)=O c1(C=O)c(C)nn(C)c1N.c1(CSC)cc(C(=O)NC2CCCC2)ccn1.C Cc1cccc(C(N2CC3(CC3)CC2C(=O)Nc2cnc(C#N)cn2)=O)c1I C(N=c1nc2ncccc2c[nH]1)C1CN(C(=O)C2=CCCC2)CC12CCC2 CC1(C(=O)NCC2C3CN(C(c4cnn5c4CCC5)=O)CC23)CCC12CCC2 C1(F)(C(N(CCC#C)C)=O)CCCN(C(=O)C(Cl)Cl)C1 C1(C(N2CCC(NC(C(C)C(C)(C)C)=O)C(C)C2)=O)CCn2ncnc2C1 N1(C(C2ON=C(CC)C2)=O)Cc2ccccc2CC1CNC(C12CSC(C1)C2)=O c1(CN2CC3C(C(=O)NC(C)(CO)CO)C3C2)c[nH]c2ccncc12 c1(NC(=O)NCC2CCC3(CC3)C2)nc2cccc(OC(F)F)c2s1 CC(C)C(C)CCNC(c1cncs1)=O.c1(C(=O)N)ccccc1CC(F)(F)F C1(C(=O)NC2CC3(CN(C(CC(=C=C)C)=O)C3)C2)Cc2nn[nH]c2C(C)C1 C1(C(=O)NCC2N(C(c3c(C)nc[nH]3)=O)CCCC2)C2CCN(CC2)S1(=O)=O c1(CC(=O)NCC2(C)N(C(C3C(CC)C3)=O)CCC2)ncn2c1CCCC2 CCC(C(=O)NCC1CC(C)C1)C(C)(C)CC.c1(C(=O)N)c[nH]c2ncccc12 N(C(=NCC(=O)OCC)N1CCC(C2CCCC2(C)C)C1)CC(CC)(CC)CO C1(CNC(c2ccncc2)=O)CC(CNC(C2CCSCC2)=O)CO1 c1(NC(C(C(C)SC)N)=O)cccc(Cl)c1N1CCCCC1 N1(C(Cn2c(C)nc(C)n2)=O)CCN(C(C2CNC(=O)N2)=O)C(C2CCC2)C1 C(=O)(C(C)CC(C)CC)NC1C2CN(C(c3nc(CC)sc3N)=O)C1C2 C1(C)(CC)CCCCC1.C1(F)(C=O)CCN(C(=O)CC2CC(=O)NC2=O)CC1.N N1(C(COC)=O)CC(NC(c2csc(Cc3ccc(F)cc3)n2)=O)C2(CC2)C1 C1(C(=O)NCCN(C)C(c2cc(Cl)cs2)=O)CCNC(=O)C1 c1(CC(=O)NC(C)(CNC(=O)C(C)(O)C2CC2)CO)ccc(O)nc1 c1(C(N2CCC(F)(F)C2)=O)cc(Br)cc(F)c1F.c1(SCC=O)n[nH]c(O)n1.N c1(C(N2CCC(N3CCC(NC(C)=O)CC3)C2)=O)cccc(I)c1O C(N=c1cc(C)c(C#N)c[nH]1)c1cc(OC)n[nH]1 c1(CNC(=O)CC2CC2CNC(c2coc(CO)c2)=O)ccc(Cl)nc1 c1(C(=O)NC(CN(C(=O)Cc2csc(NC=O)n2)CC)C)ccc(C)n1C N1(CC(=C)C)CCC(C(=O)O)(NCC)C1.c12ocnc1C(=O)N1CC2C1 c1(C(N2CCN(C(c3ccc(OCC)c(C)c3)=O)CC2)=O)ccc(C)c(C)c1O c1(C(c2cccnc2)NC(Cn2c(C)ccn2)=O)ccc([N+](=O)[O-])cc1 C1(O)(C(N(CCCNC(C2CC(n3ccnn3)C2)=O)CC)=O)CCSC1 C1(C(=O)NC2C(C)(C)C2)CC2CC2N1C(=O)Cc1ccsn1 c1(C(CN(C2CCOCC2)CCC)OC)cccc(OCC)c1 C=CC1(C(N2CCC(C)(CC)CC2)=O)CCN(C(C2CC2(F)Cl)=O)C1 c1(OCC)ccc(C(=O)NCc2[nH]c(C)nc2C)cc1S(=O)(=O)N.C1CC1 C(=O)(CC(C(F)F)c1ccccc1)NCCCNC(C(CC)NC(N)=O)=O N1(C(C2C=CCC2)=O)CCC2CCN(C(c3cccc[n+]3[O-])=O)C2C1 C(=O)(CCCCCF)N1CCC(CC#C)(C(=O)Nc2cnn(C3CC3)c2C)C1 N1(C(=O)CC2CCCN(C(C3(CO)CCOC3)=O)C2)CC2CCCC1C2CO c1(C(=O)NC(C2CCN(C(Cc3nc(C)oc3)=O)C2)C)sc(O)nc1C C1(C(=O)NC2CCC(CNC(Cc3c(C)nccc3)=O)CC2)CC2CC(=O)C1C2 N#CC1(F)CN(C(C23CC(C2)N(C(=O)OCc2ccccc2)C3)=O)C1 c1(CNC(N(CCSC)CC)=O)cnn(C2COC2)c1 C1(OC(c2onc(C)c2-c2ccc(F)cc2)=O)C2CC3C(=O)OC1C3O2 CCCC(CCCS(C)(=O)=O)C(=O)NC1CC2CCC1C2.C(=O)(C=CC(C)C)N CCC(C)C(C(=O)NCC(=O)OC(C)C)NC(=O)Cc1csnc1C C1(CC(=O)N(CC(=O)OC)CC#C)CN(C(C2CCCN(C)C2)=O)CCO1 C=CC1CN(C(=O)C=CCOc2ccccc2)CC1.c1(C(=O)N)cc(F)cs1 N1(CCN(C)CC)CCN(C(=O)OC(C)(C)C)CC1.C12CCN1C2 c1(C(C)C)ccc(C(=O)NC(C)(CNC(c2ccnnc2S)=O)C2CCC2)nc1 c1(OC)cc(C(C)(C)NC(C2CC3CCC2CN3)=O)cc(Cl)c1 c1(CC(=O)NC2CN(C(c3c(OC)nsc3)=O)C3C2C3)ccc2c(c1)CCCO2 C1(NC(c2ccc(CC)cn2)=O)CCCN(C(=O)COc2cc(C)on2)C1.C C1(NC(C2N(C(CC3ON=C(CC)C3)=O)C3C(C2)C3)=O)CN(C)CCN(C)C1 C(CCC(C)(C)NC(c1cc(C)oc1CC)=O)NC(CNC(CCC)=O)=O C(CC(C(=O)NCCCC1CC(C)C1)NC(=O)C(C)SCC)OCC N1(C(C=Cc2cc(C)no2)=O)CCC(C)CC1CNC(=O)C(C)C CC1C(=O)N(CC(N2CCC(NC(C3OCCOC3C)=O)C2)=O)C(=O)C1C c1(C(=O)NCC23N(C(c4ccc(C)s4)=O)CCC2CC3)ncnc2c1ccn2C C1(C2CCCC2)CCCN(C(=NCC(C)N2CCCC2)NC2CCOCC2)C1 N1(C(C(OC)OC)=O)CCN(CC2CC2c2ccc(C(=O)O)cc2)CC1 c1(C(=O)NC(C)CCO)cnc2c(-c3cccc(CN4CCCC4)c3)cnn2c1 CC1CN(C(=O)CN2CCC(C)(C)C2)CCC1NC(=O)CN1CCCNC1=O N1(C(CN2CC(C)C2)=O)CCC2CN(C(c3ccc4cncn4c3)=O)CCC2C1 c1(CC)cc(C(=O)NC2(C(=O)N(C(C)C(N)=O)C)CC2(C)C)nn1C CCC(C)CC(C(=O)NCC1CCC(C)(C)CC1)NC(=O)CCOC1COC1 Cc1cc(NC(C2CN(C(c3cc(=O)cco3)=O)CCC2O)=O)ccc1Br C1(n2cc(C(CC)(C)O)nn2)(C(=O)NC2CCCCO2)CCSCC1 CCC(CO)C(=O)NCCC(C(C)C)NC(c1cnn(C)c1C(F)F)=O C12C3C4C1C1C2C3C41C(=O)O.Cc1ccc(C(=O)N)cc1N.C1(C=O)CC1 CC1CC(CO)(NC(=O)COc2ccc(Cl)cc2N2CCCCC2)CC(C)(C)C1 C1(C)CN(C(=O)C=Cc2ccccc2C#N)C(C)(C)C1.C=CC1(C(=O)N)CC1 C(N=c1ccc([N+](=O)[O-])c(O)[nH]1)C1N(C(C2(OC)CCS(=O)(=O)C2)=O)CCCC1 c1(C(=O)NCC2C(CC(=O)NC3C(O)CCC(C)C3)C2)ccn2nccc2c1 N1(C(c2scc(C)n2)=O)CC(NCc2c(O)cccc2O)CC(C)C1 Cn1ccc(=O)c(C(=O)NCc2nnn(C)c2C(=O)NC)c1.C1CCSC1 c1(OC)ccc(OC)c(C(O)C(C)NC(c2cnc(C)s2)C)c1 c1(C(=O)NCC(CC)NC(c2ccc(Cl)c(F)c2F)=O)cccc2c1CNC2=O CCC(C)CCC(O)CC(=O)NCC(C)N(C)C(c1cnc(F)c(C)c1)=O c1(C(N2C(C)C(C)N(C(C3CC(O)C3)=O)CC2)=O)cc2c(cn1)CCCC2 N1(C(C(C)(O)CC(F)F)=O)CCOC2(CCN(C(c3ccncc3F)=O)CC2)C1 N1(C(C2CC(C)(O)C2)=O)CCN(C(c2cnn(-c3ccc(Cl)cc3)c2)=O)C2CC12 c1(C(C(=O)NCCC2N(C(c3nc(OC)oc3)=O)CCC2)OC)ccccc1Cl C=CCCCCCNC(=O)CCC1CCCCN1C(=O)Cc1csc(C)c1 C1(CNC(Cc2ccn(CC)n2)=O)CC2CCC1N2C(=O)COC(F)F N1(C(C=Cc2n(C)ccc2)=O)CCOC2(CCCN(C(c3cc(Cl)no3)=O)C2)C1 c1(CNC(N(CC)Cc2cccnc2N2CCOCC2)=O)cc(O)ccc1Cl c1(C(N2C(CC(=O)NCC3CC3(F)F)CCC2)=O)cc2sccc2s1 C(CCCCCC(=O)NCC1CCCC1O)NC(c1cncc(OC)c1)=O N1(C(C(CSC)O)=O)Cc2ccccc2C(NC(=O)CCCCCF)C1 C12(C(N3CCOCC(NC(C4CC(C)(CC)C4)=O)C3)=O)CCC(=O)N1CCS2 N1(C(C=CCOC)=O)CC2CC(NC(C3CCC(C)(C)OC3)=O)C1C2 N12CCC(C1)CCC2.n1(CCNC(=O)Oc2ccsn2)cc(Br)cn1 O=C(CC(c1ccccc1)n1cnnn1)NCc1ccc[nH]1 CN1CC(O)CC1C(N1CC(NC(=O)C(F)n2cccn2)C1)=O N1(C(CNC(C)=O)=O)CC2C(NC(C3(C)CC(F)C3)=O)CS(=O)(=O)C2C1 c1(OC)ccnc(C(=O)NCC2CC3CC3N2C(C2C=CCCC2)=O)c1O c1(C(N(CC(CN(C(C(CSC)O)=O)C)O)C)=O)csc2ccc(F)cc12 N1(C(c2cn(CCCC)nn2)=O)C2CN(Cc3ncc(C)s3)CC12 CCC(C)(C)CCCC(=O)NC(C)(C)CCNC(=O)C(C)C(F)(F)F N1(C(C(C)N(C)C)=O)CC2(CC(NC(=O)C(c3ccc(F)cc3)O)CO2)C1 c1(N2CCC(NC(c3[nH]cc4c3CCC4)=O)C(F)C2)ncnc2ccc(F)cc12 c1(C(N2C(CN(C(COC(CC)C)=O)C3CC3)CCC2)=O)ccnc2ccsc12 Cc1cc(N)c(C(N2CC(CO)(NC(=O)CC3CC3C)C2)=O)cc1F N1(CC(N2CCOC(CC(N3CCC(CF)CC3)=O)C2)=O)CCCCC1=O N1(C(=O)CC2CC=CC2)CC2COCC2(C(N2CCOC3CCC23)=O)C1 C1(C(=O)NC(CNC(CC(=C)Br)=O)(C)C2CCC2)C2CC3C(C2=O)C13 C=C(C)CCC(=O)NCC(C1CCN(C(c2cnccc2C)=O)CC1)F CC1(C)C(NC(=O)Cc2ccc(F)cc2Br)CCN1C(c1ccncn1)=O Cc1ccc(C(=O)OCC(c2ccc(I)cc2)=O)c(N)c1F CC(C)C(O)C(F)(F)C(=O)NC(C)CNC(C1SC2C=CC1CC2)=O c1(NC(C(C)N(C(CCOCCC)=O)CC)=O)ccc(Cl)nc1C N1(C(C2CC23CCC3)C(=O)NCCC(=O)OCC)Cc2nccn2CC(C)C1 C1CC2CCC(C1)N2C(c1ccc(C(N)=O)cn1)=O.CC(C1CC1)=CC(=O)N C(=O)(C1=CCc2ccccc21)N1C2CN(C(CC3ON=C(CC)C3)=O)C(CC2)C1 Cn1cc(NC(=O)CC2(C)CCN2C(=O)C(O)Cn2cncn2)cn1 Cc1ccc(C(=O)N(C)CCNC(=O)Cn2nnc(=O)[nH]2)c(O)n1 N#Cc1ccc(S(=O)(=O)N2CC3(CC3C(=O)Nc3ccc(Br)c(Br)c3)C2)cc1 c1(C(C(C)C)NC(=O)NCC2(CCO)CCC2)ccc(OC(F)F)cc1 c1(N2CCC(N(C(=O)C3=CCC3)CCC)CC2)ccc(S(C)(=O)=O)cc1[N+](=O)[O-] S(=O)(=O)(c1ccc(N)c(F)c1)NC(c1cc(C)cc(C)c1)CC.C1CCC1.C CC(C)C(CC(=O)NCC1(CO)CCC1)NC(c1ncc(F)cn1)=O C1(NC(C(c2ccccc2)NC(C)=O)=O)CCCCC1.c1(C(=O)N)nnc(C)s1 CC(C(C(=O)NC1CCOCC1)N1CCSC(C)C1)C(C)(C)C C(=O)(C(C)S(=O)(=O)C1CCOCC1)NCC(C)(C)NC(C(CC)F)=O C1(NC(C(CC)SC)=O)CC(C)CN(C(c2c[nH]nc2OCC(F)F)=O)C1 c1(C(N(CCC(C)NC(COC)=O)C)=O)cc(C)n(CC(F)(F)F)n1 C1(C)(C(=O)NC2CC(CNC(COCC)=O)C(O)C2)CCC(=O)N(C)C1 c1(NC(CC)CC2CC2)ccccc1C(O)CC c1(C(=O)OC)nn(C)cc1C(=O)NC1CC(NC(=O)C(O)CF)C1 c1(CCC(=O)N(CC(CNC(CCc2ncc(C)[nH]2)=O)O)C)ccc(C)c(C)c1 C1(C(=O)NCc2cnn(C)c2N)CCCN(C(=O)OC(C)(C)C)C12CC2 c1(CC)cc(C(=O)NC2CCC(C)CC2)cc(O)n1.C(=O)CCCCC1CC1.N c1(OCC)ccc(C(=O)NC2CCC2NC(C2CCC(OC)CC2)=O)cc1F n1(CCC)cnc(NCc2ccnn2C(F)F)c1 C(C(C)(C)C)N(C(c1cnn(CC(F)F)c1)=O)CC.C(=O)CC1CC1C.N C=CC(C)(O)CC(=O)Nc1cccc(CNC(=O)CCC(C)(F)F)c1 CC#CCC(CO)NC(=O)CNC(=O)CNC(=O)NC c1(C(N2CCC(CNC(C(C)CC3CCC3)=O)C23CC3)=O)cc2cc[nH]c2cn1 C1(CNC(C2OCC(C)C2)=O)CN(C(=O)CC2OCCO2)CCN1C c1(C(c2ccc(C)cc2)NC2COCC2N(C)C)cc(C)c(C)cc1C c1(OC)cc(OC)c(CN2CC(C(=O)Nc3cnnc(Cl)c3)CC(F)C2)c(Cl)c1 c1(C(=O)NC2(CC(N(CC)OC)=O)CCC2)cc2ccccc2o1 c1(C(N2CCCCC2c2ccccc2)=O)ccnc(-c2cnn(C(F)F)c2)c1 C1(NC(C(C2CN(C(=O)C(C)(F)c3ccon3)C2)OC)=O)CC(O)C1(C)C C12(C(=O)NC34C(CN(C(CC=C)=O)C3)C4)CCC(C(=O)OC)(CO1)C2 O(NC(=O)CN=C(NCc1cccs1)NC1CCN(CC(F)F)CC1)CC CC(F)(F)CCCC(=O)N1CC2CC(C1)N(C(=O)C(CC(F)(F)F)c1ccccc1)C2 C=CCCCC(C)(C)CNC(c1ccoc1CNC(C1CC1C=O)=O)=O C12(CC(=O)NC3(C(=O)NC4(CO)CCC4)CC(O)C3)CCCC1C2 N1(C(CCC=C)=O)CCC(NC(=O)C=Cc2cnccn2)C(CO)C1 c1(-c2occ(CC(=O)NC(C3CCCCC3)C(C)N)n2)ccc(F)cc1 C1(C(N(CC(C)C)CCO)=O)CC2CCCC2N1C(=O)Cc1ccn(C)n1 CC1(C)Cc2cccc(C(=O)NC3CCCC(NC(=O)O)CC3)c2O1.C(C)(C)C CC(CNCC=Cc1ccco1)CS(N)(=O)=O c1(C(=O)NCC(CC)(CC)NC(c2nccc(Cl)c2F)=O)ccc(S(C)=O)cc1 Cc1cccc(COc2ccc(C(C3CCCCC3O)=O)cc2)c1 N1(C(CCC)=O)CSCC1C(=O)NC1(CCNC(C2(C)CCCO2)=O)CCC1 CCC(CN(C)C)CC(=O)NC(CNC(c1cnc2sccn12)=O)C1CC1 CC(C(=O)NCCCC1CC1)C(C)(C)c1ccccc1.C(=O)(C)N.CC(N)=O CC1=C(C)C(OC(C2CN(C3CCOC3)C2)=O)CCC1 CCC(C)C(O)CC(=O)NCCC(O)C(=O)NCc1cccnn1 C1(C(=O)N)CC2OC(C)(C)OC2C1.C1(CC)CCN(C(=O)CS(=O)(=O)CC)CC1 C1(NC(CC2C(C)C2)=O)Cc2ccccc2N(C(C2CCCC3CCCN23)=O)C1 C1(CNC(CC(C)n2cccn2)=O)CC2(CO1)CN(C(c1ccccn1)=O)C2 C1(COC)CCN(C(c2cnccn2)=O)C1.c1(C(=O)N)ccc(Cl)o1.C(C)C N(C1CCCc2ccccc21)C(CNC(COC(C1CC(OC)(OC)C1)=O)=O)=O CCCS(=O)(=O)C(C)C(=O)N1CCOC(CCNC(=O)CSCC(C)C)C1 N1(C(c2c(C)ncn2O)=O)CCC2(CC1)CC2CNC(C1CC=CC1)=O c1(C(=O)NC(CNC(Cc2scc(C)c2)=O)CO)nccc2cccnc12 c1(CCC(=O)NCC(C)NC(c2c(CC)ocn2)=O)n[nH]c2c1CCCC2 N1(C(C2CC(OC)(OC)C2)=O)CCN(C(c2sccc2Cl)=O)C2CC12 N1(C(CCC(CC)CC)=O)C(C)CC2CN(C(=O)CCN3CCC3)CC12 c1(C(N2CC(O)(CCNC(C(C)C3CCC3)=O)C2)=O)cc2cc(Br)cn2cn1 n1(CC)c(C)nn(CC(=O)NCC2CN(C(c3cnc(C)cc3C)=O)C2)c1=O N1(C(CNC(=O)Cc2ccsc2)=O)CCN(C(=O)CSC(F)(F)F)CC1 CC1(C(=O)NCC2(C)CC23CCC3)Cc2ccccc2C1.C1(C(=O)N)CC1 C(CN=c1nc(OC2CCC2)cc[nH]1)C1CCN(C(C2C(C)C2)=O)CC1 C(=O)(C(C1=CCSC1(C)C)N1CCOCCC1C)Nc1c(C)cc(C)cc1C O=S(=O)(c1ccc2ccccc2n1)NCc1cc2c(s1)CCC2 C=CCC(CC(C)C)C(=O)NCC1CCCN1C(c1ccc(C(C)O)cc1)=O c1(OC(C)C)cccc(C(=O)N)c1.n1(C2(C=O)CC2)cc(Cl)cn1.C(C)CC Cn1nc(C(F)(F)F)c(CN2CCC(c3ccccn3)CC2)c1Cl C1(C(=O)NCC(n2cc(C3(CC)COC3)nn2)C)CC2(CC(=O)C2)C1 c1(C(=O)NC(C2CCC2)C)cccc2ccncc12.C1(C(=O)N)CCC(C)(C)C1 C1(C(=O)NC2C(NC(C(C(C)(C)O)(F)F)=O)C2)CCCN2CCCCC12 c1(C(=O)NC(CC)C(=O)NCCOCCOCCO)cc(Br)c(Br)o1 N1(C(Cc2ccc(C)s2)=O)CCOC2(CCN(C(=O)CCCC3CCCO3)C2)C1 N1(C(c2sc(C)c(O)n2)=O)CCC2(CCCN2C(c2cccc(N(C)C)c2)=O)C1 N1(C(COCC(C)C)=O)CCN(C(C2CCCN(C(C)C)C2)=O)CC(O)C1 C1(C)(C(N2CC(CC(=O)NCC3CCCCS3)(OC)C2)=O)CCCCC1 N1(C(c2c(NC)scn2)=O)CC2(C)CC1(C(=O)N(C1COCC1O)C1CC1)C2 N1(C(c2cc(C)cc(C)c2)=O)CC(NC(=O)CCC(C)C)C2CCCC12 CC1CC(NC(=O)Cc2cnns2)CCN1C(c1cnc(Cl)cn1)=O C1(NC(C2(CNC(C3C(CC(C)C)C3)=O)CCC2)=O)C2CCCCCC12 C1(NC(c2c(C)nc(CCCC)s2)=O)CCN(C(c2c[nH]c(=N)s2)=O)C12CCC2 C1(C(=O)NC)CCC2CN(C(c3cnc(C)c(C)c3)C(=O)NCCOC)CC2C1 C(=O)(C(CNC(C1CC(F)C(=O)N1)=O)C(C)(C)C)N(C(C#C)C)CCCC c1(C(=O)N)ccn2c(C)cnc2c1.c1(OC)ccc(C(=O)NC2CCC2)c(C)n1 c1(C(=O)NCC23CC(NC(CCC(=C)Cl)=O)(C2)C3)ccc2nn(C)cc2c1 N1(CC=O)C(=O)NC(C)(C)C1=O.C1CCCCC1.C1(CC=C)(C(=O)N)CC1 c1(-c2cc(C(=O)NCC(C)N(C(=O)CC3(O)CCCC3)C)on2)ccccc1Cl Cc1nc2ccc(C(=O)NCCC3(NC(=O)Cc4ccoc4C)CCC3)cc2o1 N1(C(CCCC#C)=O)CC2CC(NC(c3sccc3F)=O)C1C2 c1(C(N2CC(NC(C(C=C)O)=O)C(O)CC2)=O)c(F)ccc(C#N)c1F N1(C(CN(C(C)C)C)=O)CC(C)C(NC(c2cccc(Cl)c2Cl)=O)C(C)C1 N1(CCC)CCCC(C(=O)N(CCC)C2CC2)C1.c1(CC=O)ccc(F)cc1.N c1(CN(C)C(C2CCCN(Cc3cc[nH]n3)C2)=O)ccc(Br)cc1 n1(CC)cc(-c2cn(CCSCC)nn2)cn1.c1(C=O)csc(C(C)=O)n1.N N1(C(c2c(C)cncc2)=O)CC2CCC1C1CN(C(=O)C=CC=C(Cl)Cl)CC21 c1(C(=O)NC2CN(C(CCOC)=O)CC2O)ccc2c(c1)OCCC2 c1(CNC(c2cccc(C(F)(F)F)c2)CC)cn2c(n1)CCCC2 C=C(Br)CC(C)(C)C(=O)NCCC1CCN(C(C2(F)CC=CCC2)=O)C1 c1(N(C)Cc2ccoc2)[nH]c(=NCCCCn2ccnc2)nc2c1ncn2C c1(C(=O)NC(C)CNC(c2c(Cl)cncc2Cl)=O)ccc(F)cc1C#N CN1CCC(OCCC(=O)NCCC2CN(C(=O)C=CC3CC3)CCO2)CC1 CC1(C(=O)NCCCc2ccc(F)c(F)c2)CC(c2cc(Cl)cc(Cl)c2)=NO1 C1(OC(C)C)CCCN(C(=O)C(C)OC2CCCC2)CC1.c12ccc(nc1)o2 C(CO)(C(=O)NCC1(NC(=O)CC2CC(CF)C2)CCOC1)N(C)C c1(C(=O)NCCN(C(=O)CC2OCCCO2)C(C)C)ccsc1C(F)F n1(CC=C)c(N2CCC(COc3cccc(C)c3)CC2)nnc1CSC c1(C(=O)OC)cc(Cl)nc(NC(=O)NC(c2ccc(Br)cc2)C)n1 CN1CCC(C(=O)NCC=C2CCN(C(=O)CC3(CO)CCC3)CC2)CC1=O C=CCCCC(C(=O)N(C)CP(C)(C)=O)NC(=O)CC1CCCC2CC12 n1(CC)cc(C=O)c(C(C)C)n1.C1(C(N2CC(F)C2)=O)CC(=O)N(C)C1.N C1(NC(C(c2cn(CC)nc2)=O)=O)CCCCC1.c1(C=O)cc(C(N)=O)no1 C1(CNC(c2sccc2C(F)F)=O)CC2CC2N1C(=O)C.c1cn[nH]c1.S C1(CC)C(=O)NCCCN1C(C1CCCCN1C(c1cc(F)c[nH]1)=O)=O N1(C(CCC(=O)NCC)=O)CCC(C)N(C(C2CC=CCC2)=O)CC1 S(=O)(=O)(c1ccc(F)c(F)c1)NC1CCC(C(=O)Nc2cn[nH]c2)OC1 C(=O)C1CCCc2nn[nH]c21.c1(CC)cc(C(=O)NCC2COC(C)C2)no1.N C(=O)(C1=CCCCC1)N(CC(C)NC(c1cc(-c2c(Cl)cnn2C)no1)=O)C c1(OC)ccc(CC(=O)NCC(C)N(C(=O)Cn2nc(C)oc2=O)C)nc1 Cc1cc(C(N2CC(C)C(O)C2)=O)c(C)n1-c1ccn(C)n1.C(=O)(C(C)O)N N1(C(C(C)(C)n2cncn2)=O)CCOCC(C(=O)NCCCCO)C1 c1(CC(N2CC(C)C(C(F)(F)F)C2)=O)cc(F)cc2c1OCOC2 CC1CCN(C(C23CC(C)(CO2)C3)=O)CCN1C(c1cc(F)cnc1Cl)=O C1(NC(C=C(C)C(C)(C)C)=O)CN(C(c2cccc(N(C)C)n2)=O)CC1N=[N+]=[N-] CCCCS(=O)(=O)CC(=O)N1CCN(C(C2CC(n3cnnc3)C2)=O)CC12CC2 c1(CC(N2CC(C)CC2)=O)cc(F)ccc1F.C1(CC(=O)N)CCCS(=O)(=O)C1 C1(C(N(CCNC(=O)C(c2ccccc2)O)CC)=O)CCCNC1=O CC(C)C(CN(C)C)C(=O)NC(c1nc(C(N2CC3CC3C2)=O)co1)C C#Cc1ccc(C(F)(F)F)c(C(N2CC3(CCN(C(C45CCC4C5)=O)C3)C2)=O)c1 C(=O)(C(CC)(CC)CO)N1CCOCC(NC(c2c(CCC)[nH]cc2)=O)C1 C1(C(=O)NCCC2CCCN(C(=O)C3CC3)CC2)CC2(C1)CC1(CCC1)C2 CC1CCC(NCc2ccccc2)CN1CCOc1cncc(Cl)n1 C(C(=O)NCCC(O)C(=O)NCC1(OC)CCCC1)(C(C)(C)C)OC CC1CCCC(OCC(=O)N)C1.C1(O)(CC)CN(C(C2(C(N)=O)CC2)=O)C1 CC(C)(C)C(CC(=O)NC1CC2CCCC(C1)N2C(C1CCCCO1)=O)C(F)F Cc1ccc(CCC(N2CCCC2C(C)NC(=O)CN2CCCC2=O)=O)cc1 N1(C(CC2C(CC)C2(F)F)=O)CC(C2CN(C(=O)C(C)(F)C(=O)OC)C2)C1 C1(N(CC(=O)NCC)C)CCCN(C(=O)Cc2ccc(C)cc2)C1 c1(C(=O)NC(CNC(C2(CCC)CCC2)=O)CC)cnc2cc(C)ccn12 C(C(C(C)C(C)C)NC(c1coc(Br)n1)=O)NC(Cc1cc(C)on1)=O Cn1ncc2c1CCC(C(=O)NCC1(F)CC(NC(=O)C)C1)C2.c1ccsn1 N1(C(C(CN(OCC)CC)F)=O)CCCCC1C.c1ccc(-c2cccs2)o1.N N1(C(c2cccc(CC)c2)=O)CC2CC(C)C2C1.C1(C(=O)N)CCCC(C)(C)O1 C1(CNC(C(C)(O)C2CCC2)=O)COCCN(C(c2ccc(CC#N)cc2)=O)C1 N1(CC)CC(C(=O)NCCCOCCN(C(=O)C(C)O)C)CC1=O.CCF c1(C(=O)NCC(CN(C)C(C2(Cl)CC2(F)F)=O)O)c[nH]c(=N)s1 N1(C(C(C)OCC)=O)CCCC(C2CN(C(c3n[nH]c(C)c3O)=O)C2)C1 S(=O)(=O)(c1cc(C(=O)Nc2n[nH]c3cccc(F)c23)ccc1Cl)NCC=C Cc1ccc2c(c1)N(C)CCN2S(=O)(=O)c1cn(C)nc1Br c1(C(C)NC(c2c(NC(CCCC)=O)c[nH]n2)=O)ccc(Cl)c(Cl)c1 CCC(C(=O)NCC(CC)N(C)C(c1nocc1C)=O)C1CCOCC1 c1(N(C(CCO)c2cccs2)C)ncnc2c([N+](=O)[O-])csc12 C1(C(=O)NCCc2ccc(CNC(C3CCC(C)O3)=O)cc2)CCOCC1(C)C CC1=CCC(NC(=O)NCCCN2CCCC2)CC1 Cc1nnccc1C(N1CCCC(N(C(=O)C(C)OCC(C)C)CCO)C1)=O C(=O)(C(C(C)O)NC(=O)C(CC)OC)N(C)CC1CC(=C)C1 c1(C(=O)NCCCN(C(C(COCC)C)=O)C)cnc(O)c2cncn12 N1(C(CC2=NNC(=O)C2)=O)CC2CCC1C1CN(C(c3[nH]ccc3C3CC3)=O)CC21 CC1=CC(NC(=O)C(c2ccnn2C)NC(C2CCOC2(C)C)=O)CCC1 C(=O)(CCCC(F)(F)F)N1CCC(C(CNC(C(COCC)(C)C)=O)C)CC1 C1(NC(=O)CN2CCOC2=O)CC12CCN(c1ncnc(C(F)(F)F)c1Br)CC2 c1(CC)cccc(C(=O)NCC(CNC(C2(C)COC(C)CO2)=O)CO)c1N c1(C(N2CC(OC)(CNC(=O)C(F)C3CCOC3)C2)=O)cc(N)c(F)cc1C c1(OC)nn(C)cc1NC(C1CCN(C)C1)=O.c1(C=O)ccc(C(N)=O)[nH]1 c1(C(=O)NC2C(NC(=O)Cc3ccno3)CC2)cc2cccc(F)c2s1 c1(C(N2CCC2)=O)cc(S(N)(=O)=O)c[nH]1.Cn1cc(OCC=O)cn1.CC.N c1(N2CCCC(NC(c3ccnn3CC(F)F)=O)CC2)c(Cl)cncc1[N+](=O)[O-] N#Cc1ccc(C(N2CC(O)(CNC(=O)CO)C2)=O)c(F)c1.C1CCOC1 c1(C(=O)NCCCCCNC(C(COC)OC)=O)ccnn2ccnc12 C1(C)(NC(CNS(CC)(=O)=O)=O)CC(NC(C2CC2(F)Cl)=O)C1 CCC(C)CC(C)C(=O)NC1CN(C(=O)CC2(NC(C)=O)CC2)CC1C Nc1c(Br)ccc(F)c1C(=O)NC1CN(C(C23CCC(CO2)C3)=O)CC1O C1(O)(CC(=O)NC(c2cncnc2)c2ccccc2)CCCOC1 c1(NCC(CC)CCO)ncc(C)cc1S(=O)(=O)NC1C(O)C2CCCC12 CCCC(C(=O)NCC(O)COC(C)C)NC(=O)CCC1CC1(C)C CCCC(C(=O)NCC1(NC(c2cnn(C)c2C2CC2)=O)CCC1)OC C1(CNC(c2ccc(SC)s2)=O)CCC(C)CN1C(=O)CC.C(=O)(CO)N C(=O)(C1CCCc2c[nH]nc21)NCCC(C)N(C(c1c(C(C)C)noc1)=O)C C12CC(C(=O)O)(C1)C(C)O2.CC(C(C)C=O)NC(=O)OC(C)(C)C.N c1(C(=O)NC2CCCCC2NC(c2ncccc2O)=O)cnc2[nH]nc(O)c2c1 c1(C(=O)NCC(n2cc(CSC)nn2)C)cccc(Br)n1 C#CCC(C)(C(=O)NC1(CCF)CCC1)NC(=O)CC(C)(O)COC C(CC(C)(C)CO)NC(C(Cc1cc[nH]n1)NC(CCN(CCC)C)=O)=O C(=O)(C(C)CC(C)C(C)=O)NC(CCCC)CC(=O)NCC(=O)N(C)OCC N1(CCC#C)CCC(C(=O)NCCC(O)CNC(C2CC(F)C2)=O)CC1 C1(C(=O)NCC(CNC(c2cccc(F)c2Cl)=O)F)CCc2nc[nH]c2C1 N1(C(C2N(C(=O)NC(C)C)CCC2)=O)CCCC2CN(C(=O)CP(C)(C)=O)CC12 N1(C(COCCOC)=O)CC(C2CN(C(c3cc(OC)ns3)=O)C2)C1 Cc1c(NC(c2ccc(Cl)c(Sc3nccn3C)c2)=O)cccc1Br C(N=c1[nH]c(=NCC2CCCSC2)c2c(F)cccc2[nH]1)C1CCN(C(C)=O)C1 c1(C(CNC(c2nnnn2CCCSC)C2(CC)CCC2)F)ccc(Cl)c(F)c1 N1(C(CC2C(C(=O)OC)C2)=O)CC(N(C(=O)C(F)=CCCF)C)C(C)(C)C1 c1(C(N(CC(C)NC(c2ncoc2Br)=O)C)=O)ccc(C2=CCCC2)cc1 c1(C(C)=O)cc(Cl)nc(Cl)c1NC(C1CCN(C(c2scnc2C)=O)CC1O)=O c1(NCC)nnc(CSc2cnn(C)c2)n1CCCOc1ccccc1 N1(C(CC2(CC)CC2)=O)CCC(CNC(=O)CCCC(=O)N(C)C)C(C)C1 C(=O)(CCC(C)(C)[N+](=O)[O-])N1CC(F)C1.c1(C(C(=O)NC)OC)ccccc1F c1(C(N2CCC(=CC(N3CCC(F)CC3)=O)CC2)=O)cc(Cl)c(Cl)cc1F c1(C(=O)NCC(CC)NC(C2CC3C=CC2O3)=O)cccc(CCCCO)c1 c1(COc2ccc(C)cc2OC)nc2ccccc2c(=O)n1C(C)C.C1CCCO1 c1(CC)ccc(C(=O)NC(C)CCCNC(=O)C=Cc2scnc2C)c(Cl)c1 N=c1[nH]c2ccc(C(=O)NC3CC3NC(=O)CCc3ccncn3)cc2[nH]1 c1(CC)cccc(C(=O)NC2CCCC(N(C)C(C34CC(C)(C3)C4)=O)C2)n1 Cc1oc(C(C)(C)C)cc1C=O.c1(C=O)cnn(C(C)(C)C)c1.C(C)CO.N C(=O)(CC(C)(C)C(F)(F)F)N1CCC(CCCNC(C2C(CC)CCC2)=O)CC1 n1(CC(=O)NC2(CNC(C3C4COCC34)=O)CCOC2)ccc(O)nc1=O Cc1cc(Cl)c(C(=O)NC2(CNC(=O)C=Cc3ccoc3)CCCCC2)s1 Cn1cc2c(n1)CC(C(=O)NCC1(F)CCC1)NC2=O.n1(CC=O)cncn1 CC1CCN(C(=O)CCN2C(=O)CCC2=O)C(C)C1NC(=O)C.C(N)(=O)N C1(CC(=O)N)CN(C(C2CC23CCC3)=O)CC12CC2.C(C(C)(C)C)OCC CC1CN(c2ncc(C(=O)NCC3CCN(CC(F)(F)F)CC3)cn2)CC(C)O1 C1(NC(c2ncncc2Cl)=O)CC2CC1N(C(c1cccc(C3CC3)c1)=O)C2 C(CC(=O)NC1C(C)CCC1C)(C(F)(F)F)NC(C(C)C)=O Cc1cc(NC2(CNC(=O)C(C)n3ccnc3)COC2)nc(C(C)(C)C)n1 c1(C(N2CCN(C(C(CCC)NC(C)=O)=O)CC2C)=O)ncc2cc(Cl)ccn12 C(=O)(C(F)(F)CC(=O)N1CCOC(C)C1)OC.c1(C2(C=O)CC2)ccccc1.N C(=O)(C1Cc2ccc(Cl)cc21)N1CC(NC(=O)CC2CCCC(F)(F)C2)(CO)C1 N1(c2nccc(NC(C3CCCCC3)CC)n2)CCC2(CCC(OC)C2)C1 N1(C(c2cc(CCC)[nH]n2)=O)CCC(NC(c2ccc(OC)cc2)=O)CC1 C#CCCCCCCC(=O)N1CC(CNC(=O)C(C)(O)C2CCOC2)C1 Cc1nc(C(=O)N(CC(CO)(CO)NC(=O)CC2CC3CCC2C3)C)cc(O)n1 C1(C(N2CC(OCC(=O)NCC3CCC4CC34)C2)=O)Cc2ccccc2C1 C1(NC(c2c[nH]c(=NC)s2)=O)CN(C(=O)COC2CC=CC2)C2(CCCC2)C1 c1(CN(C)C(c2cc[nH]n2)=O)ccc(CNC(=O)CC2CCC2)cc1 C(=O)C1=C(C)OCC1.c1(CCC(=O)OC)cccc(C(N2CCC3CC23)=O)c1.N Cc1cc(C(C(=O)NC(C)(C)C)N(CC#N)C2CC2)nnc1C C1(C#N)(OC)CC(C(=O)NCC(C)CC(=O)N2CCN(CCO)CC2)C1 c1(C(=O)N)nccnc1C(N)=O.CCCCN(C)C(C1CN(c2nncs2)C1)=O C1(CNC(c2cccc(NC)n2)=O)CCN(C(=O)C(O)C(F)(F)F)C1(C)C Nc1ccc(O)cc1C(N1CCCC(CNC(=O)Cc2ccco2)C1)=O C(=O)(CC(C)(C)O)NC(C1CCN(C(=O)Cc2ccccc2)C1)C.C1CC1.C c1(CC)cnccc1C(=O)NCC(C)N(C(=O)C(CN(C)C)N(C)C)C Cc1ccc(Cl)c(C(=O)NC2CCN(C(=O)Cc3cccnc3O)CC2C)c1N C(c1ccc(C2CC2)cc1)=CC(=O)NCC#CCNC(c1cc(C)on1)=O CCC(C(=O)N(C)CCN(C(=O)C(F)=C(C)C1CC1)C)n1cccn1 Cc1nn(C)c(C)c1CN1CCC(O)C(C(=O)NC2(C)CC2)C1 CC1(C)CC(c2cn(CCOCCON)nn2)CN1C(=O)CC1CCCNC1=O CC1c2ncc(C(=O)NCc3nccnc3Cl)n2CCN1C(c1cnc(O)[nH]1)=O C(CN=c1[nH]cnc(C)c1F)C1N(C(c2c(CC)noc2)=O)CCCC1C Cc1cc(C(=O)NCC2CN(C(c3cn(C(C)C)cn3)=O)CCC2C)nc(O)c1 N1(C(c2cc(CC)nn2C)=O)C2CCC1C(C(=O)NCc1cccnc1C)C2 C1(CNC(C(C)SCC)=O)(CO)CCN(C(C2(OC)CCSCC2)=O)CC1 c1(C(N(C2CN(C(c3cc(OCC)no3)=O)CC2F)C)=O)ccc2n[nH]cc2c1 c1(C(=O)NCC2(O)COC2)cc(-c2cc(CO)ccc2F)cc2cc[nH]c12 C(C(O)CC)NC(C(C)=C1CC1)=O.c1(CCC(=O)N)ncc(C(C)(C)C)o1 C1(C)(CNC(C(C)(Cl)Cl)=O)CN(C(c2ccoc2C2CC2)=O)CCO1 Cc1ccc2nc(C(=O)NC3CCCN(C(=O)C(F)C4CCOC4)C3C)cn2c1 c1(C(=O)NC2CCCN(C(C(C)(C)C#N)=O)CC2)cc2n(c1)CCOC2 c1(C2(C(=O)NCCC3C(C(=O)OC)C3)CC2(F)F)ccccc1Br c1(N2CC(C(C)C)OCC2)nc2c(c(=NCCn3cccn3)[nH]1)CC(C)CC2 C(=O)(C(C)CN(C(=O)C(CN(C)C)NC(=O)CNC)C)OCC.C C(CC(C)C)(C(=O)NC1CCN(C(C2(C)CCOCC2)=O)C1)OC C#Cc1ccc(C(=O)NC2CN(C(=O)C(C)OCOC)CC2CC(C)(C)C)nc1 C(Cc1ccoc1)(C=O)NC(COCCC#C)=O.C(CC1CC1)C1CC1.N c1(CN2CCN(C(=O)NC3(COC)CC3(F)F)CC2)nc2ccccc2[nH]1 Cn1cnc2c1CCCC2C(=O)NC1CC2CC1N(C(c1ccccc1F)=O)C2 C1(CC(N2CC(COC)(NC(c3cn[nH]c3)=O)C2)=O)SC2=NCCN2C1=O N(C(=NCC(C)C)NC(c1ccc(Br)cc1)C)Cc1c(C)ccs1 N(C1CCCc2ccoc21)C(C1CCC(CNC(CC2(OC)CCC2)=O)O1)=O C1(C(N2CCC(N(C)Cc3ncc(C)o3)C2)=O)CC(=O)N(C(C)C2CC2)C1 N1(C(CCC(=O)NCCC)=O)CCN(C(=O)C(CC)SC)CC1CC(=O)NCC N(C1c2ccccc2CC1O)C(C1CSCCN1Cc1c(Cl)ccc(Br)c1F)=O N1(C(CCCOCC)=O)CCN(C(c2nc(C)c(C)s2)=O)C(c2cnn(C)c2)C1 N1(C(CCCSC)=O)CCN(C(=O)C(C(C)C)N)CC(C)(C)C1.[SH](=O)(=O)C1CC1 n1(CCC=O)nc(O)c2c1CCCC2.C(C(=O)NC1(C)CC1)(C(C)C)SC.N Cc1cc(C(=O)NCCCCC(C)NC(=O)CSC(F)F)nnc1C N1(C(=O)Cc2cccc(Cl)c2)CC2CC(C1)N(C(=O)CC1CCC(O)C1)C2 C(=O)(CC(C)CC(=O)NC1(C(=O)Nc2cnc(F)nc2)CCSC1)OC C12(C(=O)OC)CC1CN(C(c1cc(C(N)=O)cs1)C(=O)OC)C2 c1(OC)ccc(-c2nccc(NC(=O)C(=O)NC3CC(F)(CN)C3)n2)cc1 N1(C(C(c2ccccc2)OCC)=O)CCOCC1C.C1(C(=O)N)CCCC(=O)N1 C1(C(N2CC(C(C)NC(c3cscn3)=O)C2)=O)CC1C1CCCC1 C1(F)(C(=O)NCC(CC)NC(=O)CO)CC=CCC1.C(C)(C)C(F)(F)F C(=O)(C1=COc2ccccc2O1)NCC(CN(C)C(C1(CO)CCCO1)=O)O CCN=C(NCc1ncc(Br)s1)NC1CCN(CC2CCCO2)CC1 CCCCC(C(=O)NCCC1CC(NC(=O)C(C)(C)CF)C1)ON=C(C)C N1(C(C(=O)NCCOC)CCC2(C)CC2)CC2CC(OC)C(C2)C1 C(=O)(CCC(C)CCCC)N1C(C(N2CCC(C#C)C2)=O)CCC(O)C1 c1(C(N2CC3C(CO)C3C2)C(=O)NCCCSCC)cc(Br)cnc1OC c1(-c2n(CC(=C)C)nc(-c3cnn(C)c3)n2)ccc(S(=O)(=O)CC)cc1 Cc1cc(CNC(c2nc(-c3cccs3)no2)c2nnnn2C)nnc1C CCC(C)(COC)C(=O)NCC1CC2(CC2)CN1C(c1cscn1)=O c1(OC)c(C(=O)N(C)CC2C3CN(C(c4cncc(F)c4)=O)CC23)ccnc1Cl C12(CNC(C3CCC(C)C3)=O)CC(CO1)N(C(c1scnc1Cl)=O)C2 Cc1c(C(=O)NC2(CF)CCN(C(C3CCC4CC34)=O)C2)cnn1CC(C)C C1(NC(C(CNC(c2cnc(CC)nc2)=O)O)=O)CCCCNC1=O c1(CCC(=O)NC2C3CCN(C(C4CC(F)(CO)C4)=O)C23)ccccc1Cl N(C1CSCc2ccc(Br)cc21)C(CNC(C(CC[S+](C)C)O)=O)=O c1(NC(CC#C)COCC2CC2)ncn2ccc(C)cc12 C(CC(C(C)(C)C)NC1(C2CCCO2)CC1)NC c1(C(=O)NCCOCCNC(C(CC(CC)C)C)=O)cc2ccccc2cc1F C=CC(C)(C)CC(=O)NC(C)CN(C(c1ccc(N2CCNC2=O)cc1)=O)C N1(c2nc(OC)nc(OC)n2)CCCC2(CCN(C(=O)CC3CCC4CC34)C2)C1 C1(C(c2n(CC=C)nnn2)NCCCOCCOC)CCC(C)(C=O)CC1 c1(C(N2C(CNC(C(C(C)O)N(C)C)=O)CC2)=O)cccc2cnccc12 C(C1CN(C(C2CCC3(CCC3)C2)=O)CC1C(=O)Nc1c(C)cccc1C)=CC N1(C(C)=O)CCc2cc(-c3ccccc3C)ccc21.N12CCN(C)C(C1)C2=O C1(NC(C(F)OC)=O)C(C)(C)C(NC(=O)CCCc2cc(C)no2)C1(C)C C(=O)(CS(=O)C(F)(F)F)NC.N1(C(C2(NC(C)=O)CCC2)=O)CCC(O)C1 C1(C(=O)N)CC12CCC(=O)CC2.CN1CC(O)CCC1C(=O)NC1CC(C)C1 c1(OC)ccnc(OC)c1C(=O)NC(CO)C(C)NC(=O)Cc1ccccc1C N1(C(C(c2cn(CC)nc2)=O)=O)CCC2(C)C(C1)C2(Cl)Cl Cc1cnnc(O)c1C(N1CCC(CNC(c2coc(Cl)c2)=O)C1)=O C1(C)(NC(CCC=CC(C)C)=O)CCCN(C(c2ccn(C3CC3)n2)=O)C1 C=C=CCCC(=O)NC(CCF)C(=O)NC(c1cc[nH]n1)C N1(C(C=CC2N(C(C(C(=O)OCC)OC)=O)CCC2)=O)CCC(OC)C(O)C1 C1(NC(Cc2ncc(C)o2)=O)CN(C(=O)C(F)(F)c2cnccn2)CC1C C(=O)(C1=C(C)OCCS1)N(C1CCN(C(C(CCC)NC(C)=O)=O)CC1)CCC C1(N(C)C(c2cnc(Cl)cn2)=O)CCCN(C(c2ncccc2F)=O)CC1 c1(C(N(CCCC(=O)NC2(CCC)CCC2)C)=O)ccn2ccccc12 N1(C(C(C2(O)CN(C(=O)C(O)c3ccsc3)C2)F)=O)CCOCC12CC2 N1(C(CCc2ccc(OC)nc2)=O)CCCC(NC(C23COCC(C2)C3)=O)CC1 c1(C(=O)NC2C3(CC(NC(Cc4nc(C)oc4)=O)C3)C2)cc(Cl)c(Cl)cc1N CCC(C)C(C(=O)NC1(CO)CC1)NC(=O)CC1CCCN1C c1(C(=O)NCC(CN(C(C(CC=C)(F)F)=O)C)(C)C)ccc2c(c1)CCCC2=O Cc1nn(C)c2c(NCCC3CCSC3)nc(N3CCC(CS(C)(=O)=O)C3)nc12 c1(CCN(C(C(C)NC(c2cccs2)=O)=O)CC2CC2)c[nH]c2ccccc12 c1cccc(Cl)c1F.c1(C(C)=O)ccc(NC(=O)C(=O)NCC(O)C2CCC2)cc1 C1(NC(C(C=C)(C)CC)=O)CC2CC(C1)N(C(c1ccc(=O)n(CCF)n1)=O)C2 C1(C(=O)NCC(C)NC(C2C(OCC)C2)=O)CCCN1C(=O)OC c1(C(=O)Nc2cc3sc(C#N)c(C)c3cc2)sc(S(N)(=O)=O)c(C)c1Cl N1(C(c2scc(C(C)=O)c2)=O)CC(NC(=O)CSC(F)(F)F)CCC1C c1(C(C(=O)NC2CCC2)N(C)CCN2CCCC2=O)cnc2c(c1)COCC2 C(=O)(C(C)(C)C(O)C(C)C)N1CCC(CNC(CCCC)=O)(OC)C1 C12(NC(CCCC(=O)OC)=O)CC3CC(C1)CC(NC(c1cnn[nH]1)=O)(C3)C2 c1(C(N(C(C)CF)C)=O)cn2cccnc2n1 O=C1CC2(CCOCC2)C(CN2CCC(F)(F)C(F)C2)O1 c1(-c2nc(CC(=O)Sc3nncn3-c3ccc(Cl)cc3)sc2)cc(F)ccc1F C1(C(=O)NC)C2CCC(O2)C1C(F)(F)F.C1CCCCC1.C(=O)C.C(C)=O N1(C(C(C)NC(=O)OC)=O)CCN(C(=O)C(C(C)C)SC)C(c2ccccn2)C1 N1(C(CCCC(=O)NC)=O)CC2CCC(CNC(c3ccc(SC)s3)=O)(C2)C1 CC(C(=O)N1CCCc2nncn21)NC(=O)C(C)(C)C1CCOC1 N1(C(COc2cc(C)on2)=O)CCN(C(=O)C(C)Cc2cnc[nH]2)CC12CCC2 C(=O)(C1=CCC(NC(=O)C(C)C(F)(F)F)C1)N(CCC(F)(F)F)CC c1(OCCC(=O)NC2CCC23CN(C(C2COC(=O)N2)=O)C3)c(F)cccc1Cl O=S(=O)(C(F)F)C1CCN(CC23CNCC2CCO3)C1 c12cc(C)ccc1NC2C.C(C)(CCC1CCCC1)(c1nnnn1C(C)C)OC Cn1ncc2c(N(CCc3nn[nH]n3)Cc3ccsc3I)ccnc12 N1(C(Cc2c(C)nc[nH]2)=O)CCC2(CCC2)C(NC(=O)C(O)CC[S+](C)C)C1 CN(C1CCCc2c1cnn2C)C(=O)NCc1nc2cccc(F)c2[nH]1 C1(NC(CCCCC)=O)CC(OC)CN(C(=O)CCc2ccccc2Cl)C1 c1(C(c2n(CC=C)nnn2)NC(COC)C2CC2)cccc(-c2cc[nH]n2)c1 Cc1cc(OC(C)(C)C)ccc1NC(=O)NC(c1ccccc1)(C)CO N1(C(C(N(C(=O)CCc2cnn(C)c2)C)C2CC2)=O)CC(C#N)(CCF)C1 CC1(C)CN(C(=O)Cc2ccns2)C1C1CCN(C(=O)C=CSC)CC1.C1CC1 C(=O)(C1COc2ccccc21)N(C1CCN(C(c2cc3sccc3n2C)=O)C1)C C1(C(=O)NCC(C2CC2)SC)(CC)CCN(C(=O)CC2CCOC2)CC1 C1(N(C(=O)Cc2sc(O)nc2O)C)CCCN(C(C2CCC2C(F)F)=O)CC1 c1(CNC(CNC(N)=O)=O)ccc(CC)cc1.C(=O)C(O)Cc1ccccc1 CCCCCCCCNC(=O)C(=O)NC1C=CC(NCC2CCC(C)(C)O2)C1 N1(C(CC2(C(=C)F)CCC2)=O)CC2CC(C(=O)N(CC(C)C(F)(F)F)C)CC2C1 c1(OC)cc(-c2cccc(C3(C(=O)Nc4cccc(F)c4F)CC3)c2)cnc1Cl N1(C(c2ncn(C(C)C)n2)=O)CC=CC(C(=O)NC(C)C(O)C(F)F)C1 C1(C)(C(N(C(c2ccccn2)C)C)=O)CCCN(C(=O)C#CC(=O)N(C)C)C1 C1(NC(CCc2cnc(C)o2)=O)CC2CC(NC(c3ccns3)=O)C1C2 C1(CCNC(C(C)(N)C2CCC2)=O)CCS(=O)(=O)C1 C(c1cccs1)=C(C)C(=O)NCC(C)NC(=O)C(C1CC1)C1CC1 C1(NC(C2(C(C)(C)OC)CC2)=O)CC12CCN(C(=O)C=CC1CC1)CC2 c1(C(N(CCOC)CC)=O)cnn2cc[nH]c12.c1(CC(=O)N)ccc(C)nc1 Cc1scc(C(=O)NC2CN(C(C3CCC(N(C)C)CC3)=O)CC2C(F)F)c1C N1(C(C2CC2C(F)(F)F)=O)CCC(C=CC(N2CCC2CF)=O)CC1 c1(C(=O)NC2CCN(C(Cn3c(C)ccn3)=O)CC2C)cc2c(=O)cc[nH]c2s1 c1(C(=O)NCCCC(C)NC(C23CC(O)C2C3)=O)ccc2nc(O)[nH]c2c1 c1(C(C)NC(c2ccc(C)c(C)c2)c2n(CC(=C)C)nnn2)c(C)cccc1C CC(C)C(N=[N+]=[N-])C(=O)N1CCC(NC(C2(N(C)C)CC2)=O)C(CO)CC1 N1(C(=O)CC2C=CCC2)CCC2(CC1)CCN(C(c1cccnc1)=O)CC2 N1(Cc2ccc(OC)c(F)c2F)CCNC2CCCC2(C)C1 n1(C(C(=O)Nc2ncc(C(=O)OC)cn2)C)c(C)cc(O)cc1=O C1(C(=O)NCC23C(CN(C(c4cc(C(N)=O)oc4)=O)C2)C3)CC12CCSCC2 CC(c1ccsc1)=CC(=O)Nc1ccc(C2CCC23CCC3)cc1 C1(F)(CNC(C(C)=CC)=O)CCC(NC(=O)C(C)C)C1.c1ccccc1 N1(C(c2c(C)nncc2)=O)CC(NC(=O)C(C)(F)CC2CCCC2)C(C)(C)C1 c1(OC)ccc(Cl)c(CNC2COCC2C(=O)NC(c2cccs2)C)c1F N1(C(CCCOC(C)C)=O)CCC(NC(=O)C(C)(C)F)C2(CCC2)C1 c1(CCC(CC)C)nc(C(C)O)nn1-c1cnn(C)c1 C1(C)(C(=O)NCCCCNC(C(C)(c2ccccc2)N(C)C)=O)COC(=O)C1 CCCC(C)(O)C(=O)N1CCC(NC(=O)COc2ccc(C)cc2C)C(C)C1 Cc1nc(C(N2CCC3(CC2)CC3NC(=O)C2=CC3CCC2C3)=O)ccc1C#N N1(C(C2N(C(CC)=O)CCCC2)=O)CC2CCN(C(=O)Cc3sccc3Cl)C2C1 C1(NC(c2cc(C)n(C)c2)=O)CCN(C(=O)C(C)C)C(C2CC2)C1 CN=c1[nH]cc(C(N2CCCC2C2(O)CN(C(=O)CC3CCC(=O)NC3)C2)=O)o1 c1(NC(CCN(C(=O)CCN(C)C)CC)=O)cncc(NC(N)=O)c1 c1(CC=O)ccc([N+](=O)[O-])cc1Cl.C1(C(N(CCC)C)=O)(C(F)F)CCCO1.N c1(C(=O)NC(CN(C(c2ccc(CC)cc2C)=O)C)C)nccc2nn[nH]c12 N1(C(c2c(C)onc2C2CC2)=O)CCC2(CC1)CC2NC(=O)C=O.CC(F)F C1(O)CCN(C(c2c(C)noc2C(F)F)=O)C1.C(C)(C(=O)NC)NC(C)=O C1(C=O)CN(C(=O)CC2(O)CCOCC2)CC1C1CC1.C(=O)(CC)NCCC.N c1(CC)noc(C)c1C(=O)NC1CC1CNC(=O)CCC.C(N)=O.N C1(C(N(CC)CC2CCN(C(C)=O)CC2)=O)CCn2cncc2C1 C1(C(=O)OC)CN(C(C2CCC3(CC2)CC(C(=O)O)C3)=O)C2(CCCCCC2)C1 N1(C(c2n(C)ncc2)=O)CCCCC1CCNC(c1ccc(F)s1)=O Cc1ccc(C(=O)N)nc1O.C1CC2(C1)CN(C(C1CCC(=O)N1C1CC1)=O)C2 c1(C(=O)NC2CN(C(CC3OCC(C)(C)C3)=O)CC(F)C2)cccc2ccoc12 CC(C)C(CN(C)C)NC(C1(NC(C2CCOCC2)=O)CC(F)C1)=O C1(NC(c2cnc(CCCC)s2)=O)CCCN(C(=O)C=Cc2cnc(C)s2)C1C N1(C(C2C(C)(C)COC2)=O)CCC(F)CC1C(=O)NCCCN=[N+]=[N-] Cc1nnc2n1CC(C(=O)N(C)CCN(C)C(c1ccnnc1)=O)C2 C(=O)(C1(C)COc2ccccc21)NC1CC(NC(C(C)OCC2CC2)=O)C1 c1(C=O)cc2c(s1)-c1ccccc1CC2.C(CC(=O)NCC1CC1)SCC.N c1(C(N2CC=CC(NC(COC)=O)C2)=O)ccc2scc(C)c2c1 C(=O)(C(C)C(F)(F)F)NCC(C)=CC(=O)NCC1COC(=O)C1 C1CC12CCN(C(=O)Cc1cc(C)[nH]n1)CC2.c1(CC)ccc(C(=O)NC)nc1 Cn1cc2c(C(=O)NC3CC(CCNC(=O)C4=COCC4)C3)cccc2n1 C(=O)(C(C)C(O)C(C)C)NC(CC)CCC(=O)N1CCC(C)(C)C1 O(P(C)(=O)CNC(C1(CC)CN(C(c2coc(C3CC3)n2)=O)C1)=O)CC c1(C(N2CC(C)N(C(c3cncc4c3CCC4)=O)CC2)=O)cnc2[nH]cnc2c1 c1(C(=O)NC(CCN(C(CCOC(C)C)=O)C)C)cc2n(c1)CCCC2 C1(C(C(N2CCC(NC(c3ccc(SC)o3)=O)C2)=O)O)CCS(=O)(=O)CC1 c1(OC(C)C(=O)N2CC(NC(=O)CSC(C)(C)C)C2)cccc(C#N)c1 C(C)(C)(CCCNC(=O)CCOC)NC(Cc1c(C)cco1)=O.C1CCCO1 c1(NCc2ccc(C)nc2O)c(F)cc(F)c(Br)c1[N+](=O)[O-] c1(C(=O)NCC(C)(C2CC2)NC(c2ccc(C)cc2)=O)cnc2c(c1)CCC2 C1(C)(CNC(C(C)NC(C2CCOCC2)=O)=O)CCCCO1 Cc1ccccc1C1(NCC(c2cn(C(C)CN(C)C)nc2C)=O)CC1 c1(CC(=O)NCC2(C)CCN(C(C3(F)CC3)=O)C2)ccc2ocnc2c1 C1(CF)CCN(C=O)CC1.N1(C(COC)=O)CC(F)(C(=O)OC(C)C)C1.O C1(NC(c2ccoc2)=O)C=CCCC1C(=O)NC1CCCSC1 Cc1cc(F)ccc1CN1CCC1C(=O)NCC1CCCCC1 c1(C(N2CC(CCC)N(C(c3cc(C)c[nH]3)=O)CC2)=O)cccn2ccnc12 C(=O)(CN=c1cc[nH]cc1)N1CCCC(F)(C(=O)NC(C)CC(N)=O)C1 N1(C(C2(c3ccc(CC)cc3)COC2)=O)CC(C2CCCN(C(C)=O)C2)C1 N1(C(c2nc(C)n(C)c2C)=O)CC2CCC1CN2C(c1cc(C)n(C)c(=O)c1)=O c1(C=O)cnc(O)c(C(C)=NO)c1.C(=O)C(C)(O)C1CCC1.C(C)(C)OC.N C1(C(N(CCC)C)=O)C(C(F)F)C1(C)C.CCS(=O)(=O)NCCC(=O)N c1(C(N2C(C(=O)N)CC(O)C2)=O)ccc(O)c(C#N)c1.c1(OC)cccc(F)c1 C1(CNC(c2cc[n+]([O-])cc2)=O)CN(C(c2cc(Cl)c[nH]2)=O)C2(CCOCC2)C1 C1(NC(C2OCCN(C(C(CCC)C#N)=O)CC2)=O)C2CCC3C(C2)CC13 N1(C(C2C(c3c(C)cccc3)C2)=O)CC(NC(=O)C2=CCOC2)CC1(C)C C1(CNC(Cc2cnc(C)o2)=O)CN(C(C2(C#N)CC2)=O)CC(C)(C)C1 c1(C(=O)NCC(CC)NC(=O)C(C)S(C)(=O)=O)cc(O)ncc1F C1(C(F)F)(CNC(CCCc2c(C)ccs2)=O)CCN(C(=O)CC2CCCC2)C1 C1(CCNC(=O)C(F)CC2CCCCC2)CCCN(C(c2cc(O)no2)=O)CC1 CC(C(=O)N1CCC(N(C(C2(c3ccccc3)CC2)=O)C)CC1)C(F)F.C1CC1 Cc1cc2c[nH]nc2cc1C(N1CCC(O)C(NC(C2CC2C2CCC2)=O)C1)=O CC(C)(O)C(C)(C)C(=O)NCC1COCCN(C(c2cnn3ccncc23)=O)C1 C=CC(C)(CC)C(=O)NC1CCC1NC(c1ccc(-c2ncon2)cc1)=O C1(C(N(C(CNC(c2ccc(COC)s2)=O)C)C)=O)CC(=O)NC(=O)C1 C1(C)(C(N2CC3C(CNC(C(CC)(C)O)=O)C3C2)=O)CCC(C)(C)CC1 N1(C(CCCOC(C)=O)=O)CCCC(CN(C(=O)CC(C)(C)F)CC)C1 c1(NC(C)=O)cc(C)c(S(=O)(=O)Nc2ccnn2CCC(F)(F)F)cc1Br C1(CNC(CCSC)=O)CC12CCN(C(C13CCC(C1)C3(C)C)=O)CC2 C(CC(C(=O)NCC(O)C1CC1)NC(C1CC(C)(O)C1)=O)SC C(=O)(C(C)(C)CS(C)(=O)=O)NC1CC(C)(NC(c2ccc(C)c(Cl)c2)=O)C1 C#CC1(O)CCN(C(C23CCC(CC2)C3)=O)CC1.C(=O)(CC=CC(C)(C)C)N C12CCC(C1)N(C(C1CCCC3(CC3)C1)=O)C2.CC(C)(C=O)N.[SH](C)(=O)=O C1(CCNC(c2cnn(C3CCC3)n2)=O)CCN(C(=O)C=Cc2ccc[nH]2)C1 C#CCC(C(=O)NCC12CC(CO)(CO1)C2)NC(c1ccccc1Cl)=O N1(C(CC(=C)C)=O)CCN2CCN(C(=O)CC3CC3CC)CC2C1 Nc1c(C(N2CCCC(NC(=O)C(O)CC(F)F)CC2)=O)cccc1Cl c1(CC=O)cc(=O)n(-c2ccccn2)[nH]1.CC(C)CC.C(=O)C=C1CCC1.N C1(CC(=O)OCC)CCN(S(=O)(=O)N2CCCC(SCC)C2)CC1 C(C1CN(C(=O)C=Cc2ccccc2C)CC1C(=O)NC(CO)C=O)=CC.O Cc1nc(NC(C2CC2C(=O)Nc2cnc(C(F)(F)F)cn2)=O)nc(Cl)c1Br N1(C(C(CC)SC)=O)CC2OCCN(C(c3ccco3)=O)C2C1 C1(CNC(CCCNC(C)=O)=O)CC2CCC1N2C(c1c(C)csc1C)=O Cc1cnn(CCC(=O)N(CCC(C)(C)NC(c2cn(C3CCC3)nn2)=O)C)c1 C1(C(=O)NC(CSCC)C(=O)N(C)Cc2ccccn2)CCC=CCCC1 c1(NC(N2CCC(c3ccccc3)(CC(N)=O)CC2)=O)cc2cc(Cl)ccc2o1 C(=O)(C#CC1(C)CCCO1)N1CC(C(=O)Nc2cc(C)sc2)C2(C1)CC2 N1(C(=O)C(F)OC(F)(F)F)CCC(C(N2CC([N+](=O)[O-])C2)=O)CC1 c1(C(=O)NCC2CN(C(C3C4C5CCC(C5)C34)=O)CCO2)cc2ccccn2n1 CC(C)CC(CC(C)C)C(=O)NCC1CN(C(C2CC(O)C2)=O)CCC1C c1(C(=O)NC(CC(=O)O)c2ccccn2)ccc2ccccc2n1 N1(C(C2C(C)SCCC2)=O)CC2(C1)CN(C(c1ccnnc1O)=O)C2 N1(C(=O)NC2C(C)CN(S(C)(=O)=O)C2)CCc2c(cnn2C)C1C(N)=O C1(NC(C(CC)SC)=O)COC2C(NC(C3SCCS3)=O)COC12 C1(C(=O)NC2(CCNC(Cc3cc(C)no3)=O)CCC2)COCCC1(F)F N1(C(c2c(C)cco2)=O)CCCC(NC(c2ccncc2Cl)=O)C1C c1(CC(=O)NC2CN(C(C3C(C)C3)=O)CC(O)C2)ccc2c(c1)CCCN2C N1(C(c2cnc(CC)o2)=O)C2CC1CN(C(=O)Cn1cc(C)ccc1=O)C2 C1(NC(C(C)Oc2ccccc2)=O)CN(C(C2(C)CCCCO2)=O)CC1CO CCCC(C)(C)C(=O)NC1CCC(C(N2CCC(N3CCC3)CC2)=O)C1 C=CC(C)(C)CC(=O)N1CCC(C(N2CCN(C)CC2C(C)C)=O)C1 c1(OC)cc(CCC(=O)NCCC2CC(NC(=O)C(F)C3CC3)C2)ccc1O Cn1nc(C(F)(F)F)cc1CCNC(=O)N.c1nccs1.C1CC1CC=O Cc1ccc2c(N(C)CCOCCO)nc(N3CC(C(N)=O)OC(C)C3)nc2c1 c1(OC)ccc(C=CC(N2CC(NC(C34CCN(CC3)C4)=O)CC2C)=O)cc1Cl N1(C(C2(C#N)CC3CCC2C3)=O)CCC2CC(NC(C3(O)CCC3)=O)CCC2C1 CN1C2CCCC1CC(NC(c1cc(-c3ccc(N)cc3)cs1)=O)C2 N1(Cc2ccc(OC)cc2)CCn2cc(C3=CCN(C)CC3)nc2C1 Cc1nc(N2CCCC2)cc(SC(C)C)n1.c1(C(N(C)C)=O)ccc(=O)n(C)n1 c1(CC(=O)NCC(C(C)(C)C)NC(C2CCCCC2O)=O)cnc2cccnn12 N1(C(=O)C(O)CN2CCOCC2)CCC(NC(C2(C(F)(F)F)CCCC2)=O)CC1 N1(C(C(NOC)=O)=O)CCC(C2(C(N3CCCC(CF)C3)=O)CCOCC2)CC1 C1(NC(c2c(C)nn[nH]2)=O)COCCC1NC(C1(C2CCCCO2)CC1)=O N1(C(C(F)=CCC)=O)CCC(C)C1CNC(c1ccccc1)=O.C1CC1.O C1(CNC(CC2N(CC)CCC2)=O)(OC)CCN(C(=O)C=CCOC)C1 C1(C(N2C(CCC)COCC2)=O)CC(F)(F)CN1C(C1C2CCCCC12)=O Cc1cc(C(=O)NCC2CCCN(C(C3CC3(C)C(C)C)=O)C2)cc(O)n1 Cc1cnc2c(C(N3CCC(NC(=O)C=C4CC4)CC3C)=O)cccn12 C(c1cccc(O)c1)=CC(=O)N(C1CCN(C(=O)C(C)(C)O)C1)C CCCCC(C)C(=O)N1CCN(C(=O)Cc2cc(COC)no2)C(CC(F)F)C1 n1(CCC=C)c(N(CC(C)C#N)C)nnc1-c1ccco1 N(C1c2ccccc2CCC1C)c1ccc(N2CCC(C)CC2)cc1 c1(C(=O)NC(CNC(C(C)OCC(C)C)=O)C)c[nH]c2cc(F)ccc12 CC1C2CC(C2)N1C(c1n[nH]c2c1CCC2)=O.C1(C=O)CCN(S(C)(=O)=O)C1 C(=O)(C1=NN2CC(C)CN=C2N1)N.C1(C(=O)N(CCC)C)(COC)CCCCO1 N1(C(C(CNC(C(COC)OC)=O)C(C)C)=O)CCC(CO)C(C)(C)C1 Cc1ccc(CCC(=O)N(CCNC(=O)CCSCC(N)=O)C2CC2)cc1 C(=O)(C1=CC2C=CC(C1)C2)NCC(CC(=O)N(CC(C1CC1)OC)C)O C1(NC(CC(=O)NCC)=O)CC2CN(C(=O)C(CC)OCC(F)(F)F)CC12 c1(OC)ccc(I)c(CCNS(=O)(=O)CC(C)(C)C)c1 C1(NC(C(=Cc2ccco2)C)=O)C2CCN(C(=O)CC(F)(F)Cl)C12 c1(C(=O)NCCCCNC(C(C)OCC)=O)c(C)nn(C2CCCCO2)c1C N1(C(C(C)C2(O)CCC2)=O)CC=CC(C(=O)NCC2(F)CCCCC2)C1 CC1(C)CC(C=O)C1C(F)(F)F.C1C=CCN(C(c2nc(C3CC3)cs2)=O)C1 C1(CCC(=O)NCC(C2N(C(CCOC)=O)CCC2)(C)C)CCC(=O)NC1 C1(O)(C(CNC(C2(CC#C)CC2)=O)C)CCN(C(=O)C(C)=CC)C1 C1(C(=O)NC(CC=C)CC=C)CCCCC1(C)NC(=O)CC1(CSC)CC1 c1(C(=O)NCc2cc(OC)c(C)cc2)ccc(N)c(C)c1C N1(C(CC2C(=O)OCC2)=O)CC2CCCC2(C(=O)N(C2(C3CC3)CC2)CCO)C1 S(=O)(=O)(CCC(=O)N1CCC(C2OCCCC2)CC1)NC.C(=O)(C=C(C)Cl)N C#CCCCCCNC(c1cccc(CNC(=O)C(CCOC)OC)n1)=O C#CC1(C(=O)NC(C#C)C(C)C)CCN(C(c2cc(CC)[nH]n2)=O)CC1 C(=O)(C#CC1CCCOC1)NC1C(CNC(c2c(C(C)C)scn2)=O)C1 N1(C(C(CCC)=CCC)=O)CCC2(CC1)CN(C(c1ccsc1Cl)=O)CCO2 Cc1c(C2(C(=O)NCC3CC3)CC2)cccc1F.c1(C=O)ccnc(S)c1.C c1(C(N2CCC(C(C)NC(C(C=C)(C)C)=O)CC2)=O)cnc(Cl)cc1N CCCC(C)(O)CC(=O)NC1CC2CN(C(=O)CCc3cnccn3)CC12 N1(C(COCc2cc(C)on2)=O)CCN(C(C2CC(C)(C)CO2)=O)CC12CCC2 c1(C(N2CCC(C)(C(=O)Nc3n(CC)nc(C)c3)C2)=O)ccc2sccc2c1 c1(NCCCC(CC)O)nc(N2CC3CC2C(F)(F)C3)nc2sccc12 c1(C(N(C(C(=O)NC(C)C(C2CCCCC2)C)=O)C)C)ccc(Cl)cc1 C12(C(N(C(CCNC(CCCCOC)=O)C)C)=O)CCCCC1(C(=O)OC)CC2 N1(C(C(=O)NC(CC)C)CCSC)CC2CC(C1)C1CCCC(=O)N1C2 CCC(C)(CNC(C1CC(CC)(CC)C1)=O)C(=O)N1CCC1CF C(c1ccccc1)=CC(N1CCC(O)(C(=O)NCCCN2CCOCC2)C1)=O N1(C(c2c(CC=C)cccc2)=O)CCC(C2CC(NC(c3ccnnc3)=O)C2)C1 C(CC(C)(C)C(=O)NCCCNC(c1cc(C(=O)OC)ccc1N)=O)OC.O c1(C(=O)NC(C)CC2CN(C(c3c(F)ccnc3Cl)=O)C2)c[nH]c2cccnc12 CC1CCC(CNC(c2cc(N)ccn2)=O)CN1C(=O)CC1CC=CC1 O=C(CCCNC(=O)C1CC1)NCC1(F)CCC1.C1(C=O)CSCCS1.N c1(C(=O)Nc2cc(C)nn2Cc2ccccc2)ccc(S(C)(=O)=O)nn1 n1(CC)cnc2nc(=NC3CCCC(F)C3)[nH]c(NCCN3CCCS3(=O)=O)c12 c1(CC(=O)NC2CCN(C(c3ccco3)=O)C2)csc2ccc(Br)cc12 C1(N(CC(=O)NC2CCCCC2)CC)CCN(C(c2ccc(F)o2)=O)CC1 CC1(C(=O)NC2C=CCC(C(N3CCCC(C)(F)C3)=O)C2)CC2C=CC1C2 Cn1cc2cc(NC(=O)CN3CCNCC3=O)ccc2n1 c1(CNC(C2C3CN(Cc4cnc(C)s4)C2C3)=O)ccc(C(=O)O)c(F)c1 N1(C(c2ccc(C=C)cc2)=O)CC2CCN(C(=O)CSC(F)(F)F)C(C2)C1 c1(CC)ccccc1CC(=O)N(C)CCOCCCNC(=O)C1=CCOC1 Cc1c(F)ccc(Cl)c1C(=O)NC1CCCCC1NC(=O)CCC(=O)N(C)C Cc1c(NC(c2cc(CNC(c3ccccn3)=O)[nH]n2)=O)cccc1CO Cc1c(O)c(=O)ccn1CC(=O)NCCC1CN(C(C2CCCC2C)=O)C1 C(=O)(CC(C1CC1)NC(=O)CCc1nc[nH]n1)N(C(C)C(N)=O)C C(=O)(CCCN=[N+]=[N-])N1CC(NC(CC2C(C)C2(F)F)=O)(CO)C1 N1(C(C2(NC(C)C)CC2)=O)CCCC1.c1(C(N(C)C)=O)ccnn1C(C)C C(=O)(CCCC(=O)N1CCCC(C(=O)NC23CCN(CC2)C3)C1)OC Cc1c(CNCC23CCCC2C3)cnn1C(C)C C12(CNC(C(CC=C)C)=O)CC(CO1)N(C(=O)C(c1cccc(Cl)c1F)(C)C)C2 c1(CC(=O)NCC(C)NC(=O)CN2CCCNC2=O)c(Br)ccc(F)c1F c1(C(N2CC(C)N(C(C3CC3F)=O)CC2)=O)ccc(-n2ccnc2)c([N+](=O)[O-])c1 n1(CC)nccc1C=CC(=O)N.C1CN(C(c2ccc(C3CC3)nc2)=O)C2CC12 c1(OC)cccc(C(=O)NCC2CCCC(NC(=O)CC(C)C)C2)c1 C1(CC=C)(C(=O)NCC2CCCC(C)(C)O2)CCCN(C(=O)CCCOC)C1 Cc1c(C(=O)N(C(C)CN(C)C(C2CC(C(C)C)C2)=O)C)nn(C)c1Br c1(CNC(CN(C(CC2C(CC)C2)=O)CC2CC2)=O)csc(O)n1 c1(C(N2C(CNC(CC(=C)C)=O)COCC2)=O)nc(C2CC2)ncc1Cl N1(C(C2C(C(=O)OC)COC2)=O)CCOC2(C1)CN(C(C1CCOC1)=O)C2 C1(C(N2CC3CC(C2)N(C(=O)Cc2ccon2)C3)=O)Cc2ccccc2CO1 c1(C(=O)NC(CC)CN(C)C(C2(C)CCCCO2)=O)cc(C)cc(C)c1O N1(C(c2cccc(OC)c2O)=O)CCC2(CC1)OCCC2NC(c1cnn[nH]1)=O C1(C(=O)NCCCCCCN(C(=O)CN2CC(C)(C)C2)C)CN2CCC1(C)CC2 CN1CC2CCN(C(c3cnn(CCNC(C4(C)CC4(C)C)=O)c3)=O)CC2C1 C1(CNC(C2(C(=O)OC)CC2)=O)CC(C(=O)N)C1.CCCC1CC1C Cc1c(N)ccc(C(=O)N(C)CC2(O)CCCN(C(=O)CC(F)F)C2)c1C c1(-c2n(CC)nc(-c3cccc(C(F)F)n3)n2)cn2cc(F)ccc2n1 c1(NC(CONC(c2ccc(C)nc2)=O)=O)cncc([N+](=O)[O-])c1 c1(NC(C2N(Cc3c(C#N)cc(Br)cc3)CC2)=O)cnc2ccc(Br)cc2n1 C1(C(N2C(C(=O)NC3C(C)OCC3)CCCC2)=O)CC2(CCC2=O)C1 N1(C(C2C(NC(C(C=C)OC)=O)CC=CC2)=O)CCC(C)(C2CC2)C1 C1(CC#C)(C(=O)NC2CC2NC(c2ccco2)=O)CC=CCC1 c1(OC)ccc(-c2cc(F)ccc2C)cc1S(=O)(=O)N1CC(N(C)C)C1 c1(C(=O)NCC2CC(NC(c3ccncc3O)=O)C2)ncnc2c1OCCO2 CCCC(C)(O)CC(=O)N1CCN(C)CC1C(=O)Nc1ccc(O)c(C)c1 C(C)(C)(CCCC(=O)N1CCC1CC1CC1)NC(C1C(CC)C1)=O N1(C(C(CSC)(C)C)=O)CCC2(CC1)CN(C(=O)CC1OCCCO1)CC2CO C(C)(CC(=O)N)NC(C1(CCC=C)CC1)=O.CC(O)C.C(N)=O.C1CC1 CC1CCN(CCC(=O)NCC2(c3ccccc3)CC(NC(=O)C3CC3)C2)CC1 c1(C(=O)NC(CCOC)CNC(C2CCCN2C)=O)cc(Cl)c(F)cc1F c1(C(=O)NCCCN(C(C2C(CCC)CCC2)=O)C)cc(F)c(O)c(Cl)c1 N1(C(C=CC(C)C)=O)CC(C)C(NC(=O)CCc2ccc(CO)cc2)C(C)C1 C1(CC(=O)N(CCCC(C)(C)C)C)C2CC3CC(C2)CC1C3.C1(C)(C=O)CC1 C1(CNC(CCCC)=O)CC2CC(C1)N(C(=O)Cc1c(C(F)(F)F)coc1C)C2 N(C(=NCCF)NCc1cccc(OCC(F)F)c1)C1CC(OCC)C1 CCC(CCOC)C(=O)N(C(C)CNC(=O)C=Cc1cnn(C)c1C)CC c1ccc(C(N)=O)cc1C.N1(C(C2C(C(=O)OC)C2)=O)CCC2(C=O)CC2C1 c1(C(N2CC(NC(Cc3cc(C)sc3C)=O)C(CO)C2)=O)n[nH]c2ccccc12 C1(NC(C(CNC(C)=O)(C)C)=O)CC(F)CN(C(=O)OC(C)(C)C)C1 N1(C(C(=O)NCC)=O)CC=CC(NC(=O)CC2CCC(C)(C)C2)C1 N1(C(C(C)(C)OC(C)=O)=O)CCN(CCNC(C2CC23CCC3)=O)CC1 c1(C(C)(F)F)ccc(C(=O)NC2(CF)CCN(C(C3CCCO3)=O)C2)nc1 C1(C(N2CCC(CNC(C(C)(C)C3CCC3)=O)C2)=O)COc2cc(Cl)ccc2C1 c1(C(N2CCC(CC)C2)=O)ccc2cn(C)nc2c1.C(C=O)NC(=O)OCC C1(C(=O)NC2(CNC(C3C(C)(C)CCC3)=O)CC2)CCc2nncn2C1 C1(C(=O)NCCc2cc(C)on2)CCN(C(C2C3CCC(C3)C2C)=O)C12CC2 Cc1n[nH]c(C)c1CC(=O)NCCC(O)CNC(C1CC12CCCC2)=O C1(NC(=O)CCCC2CC2)CC(C(=O)Nc2ccc(F)cc2)=CC1O Cc1nc(N2CCC(NC(C3CCCC(C)C3)=O)CC2)c(C)c(Cl)n1 c1(C(N2CCCC(NC(C(=O)NCC)=O)CC2)=O)nn(C)c(C)c1[N+](=O)[O-] C1(C(C=O)C)CCC(=O)N1.C1(N(C(=O)CC2CC2)CC#C)CCCCC1.C C=CC(CC)C(=O)N1CCC(C(C)C(=O)NC(C)CCC)CC1 CC1CCC(CNC(=O)C(N2CCC(C3CCCCC3)C2)=O)Cc2ccccc21 N1(C(c2n(C=C)nnc2)=O)CCOC2(CCN(C(c3coc(Cl)n3)=O)C2)C1 C1(CC(N2CC(NC(=O)Cn3ncnn3)C(C)C2)=O)CC2CCC1CC2.C1CC1 C1(NC(CN(C2CCC2)C(c2cnn(CC)c2C)=O)=O)CCC(=O)NC1C CCCC(C(O)C(=O)N(C)CC1(CO)CC1)NC(C1CC2CCC1CC2)=O CC(C)(CONC(=O)NCCN1CCCS1(=O)=O)CC#N N(C(=NCCC1(O)CCOC1)NCC1CC2CCC1CC2)CC(C)(C)C C1(O)(CCNC(CSCC(N)=O)=O)CCN(C(=O)CCc2cnoc2)C1 c1(C(N(CCCNC(c2cc3ncccn3n2)=O)C)=O)ccc(S(N)(=O)=O)nc1 N1(CC(=O)NC(N)=O)CCC2(CCN(C(C3CCC(F)C3)=O)C2)C1.CCO c1(C(=O)OCC)ccnc(N2CC=CC(NC(C3C=C3C)=O)C2)c1[N+](=O)[O-] c1(C(N2CCC(C)(NC(c3nsnc3O)=O)CC2)=O)cc2ccccc2o1 c1(C(=O)NCC2(F)CC(C)C2)nnc(O)c(Br)c1O.c1(C=O)cocn1.N c1(C(=O)NC2CCCC(NC(CC3C(C)=NOC3=O)=O)C2)ccc(F)c(C)c1Cl C(=O)(C1CCc2ccccc21)N1CC(O)(CNC(C2CC23CCCC3)=O)C1 C(=O)(CCCCN(C(=O)CC1NC(=O)NC1=O)C)NCC1(CC)CCC1 Cc1cc(Br)ccc1CNC(C1CC(C)CN1C(c1ccc(I)cc1Cl)=O)=O N1(C(C2(C(C)(F)F)CC2)=O)CCN(C(C)C(F)F)CC1.C(=O)C.C(N)=O.N C(CCCC(=O)N1CCCC(NC(C2CCC2(F)F)=O)CC1)(OC)OC c1(CC)cc(C(=O)NC2CCC(CNC(=O)CC3CCCC3O)CC2)nn1C Cn1ccc2c(NCC(O)CNC(c3cn(C(C)(C)C)nn3)=O)ncnc12 CC1ON=C(C(=O)NCCN(C(=O)CCc2nc(-c3ccoc3)no2)C)C1C Cc1cccc(Br)c1C(=O)NC1(CNC(=O)CC2C=CCC2)CCOCC1 c1(C(=O)NC2CN(C(c3ccc(F)cc3F)=O)CC2O)ccc2nc(O)oc2c1 Cc1c(F)cccc1S(=O)(=O)NC1CCC(CNC(C2CC2C2CC2)=O)CC1 C1(N2C(COC(c3cc(CC(C)C)[nH]n3)=O)CC2)CCCSCC1 Cc1cc(C(=O)NCCn2cc(C(=O)NOCCN(C)C)nn2)ncn1 O=C1CC(N=c2nc(N3CCOCC3)[nH]c(=NC3COCCOC3)[nH]2)CN1 Cc1ccc2c(c1Cl)N(CC(=O)Nc1ccc(C(C)(C)C)cc1)CCC2 C1(CNC(=O)CCC(F)F)CC2(CCN(C(c3cc(O)ncn3)=O)CC2)C1 CC(O)(CC(F)F)C(=O)NCCCNC(c1cc(Cl)cs1)=O Cc1cccc(C(C)C(=O)NC2(CO)CN(C(C3CCCC3F)=O)C2)c1 c1(NC(CCCOC)c2nnnn2CCCF)ccccc1CCO c1(CN(C)C)cc(CNc2cc(COC)ccn2)ccc1Cl c1(C(N(C)CC2(CNC(COC(C)=O)=O)CC2)=O)cncnc1 C(=O)(C1=C(C2(C)CC2)N(CCF)C(=O)NC1c1cc(C2(C)CC2)on1)O.CC CC1CN(C(c2c[nH]nc2C2CC2)=O)CC(C)C1NC(c1coc(Br)n1)=O c1(CCC)ccc(CC(=O)NCC2CC2)cc1.c1(C=O)ccn(C(F)F)n1.C C1(CNC(C(C)N(CC)CC)=O)CCN(C(=O)C(O)C2CCCC2)CC1 C1(CC)CC(F)(F)CN1C(C1CC12CC(O)C2)=O.Cc1noc(C)c1C(=O)N C1(NC(=O)CC2CCOC2)CC1C1CCN(C(=O)C=Cc2ccco2)CC1 N1(C(C(C)n2ccnc2)=O)CCC(NC(=O)C2Cc3ccccc32)C12CCCC2 C1(C(=O)NCC2(CC(=O)NC3CCSCC3)CC2)CCCCCCC1 c1(C(N)=O)ccc(O)c(C(N2CC(C(=O)N)C2)=O)c1.C(=O)C1=CCSC1.CC C1(NC(CCS(C)=O)=O)CCCCN(C(c2[nH]c(=N)sc2C(F)(F)F)=O)CC1 C(=O)(C1=CCCOCC1)N1CCC(NC(CCCc2ccc(C)cc2)=O)C1(C)C c1(C(=O)N)cnn2c1OCC2.N1(C(CCNC(C2C(C)C2)=O)=O)CCCC1CC C1(N(c2snc(C)n2)C)CCN(C(C2CC23CCCC3)=O)CC1 N1(C(c2nc(CC)oc2)=O)CCC2(CCN(C(C3OCCC3C)=O)CC2)C(C)C1 c1(CSC)cc(Cl)cnc1F.c12cc(co1)C(=O)NC1COCC1n1cc-2nn1 C1(C(N2CCC(CC=C)(NC(c3cccs3)=O)C2)=O)CCC12CCOCC2 N1(C(CCn2ncn(C)c2=O)=O)CC2COCCC2(NC(c2ccncn2)=O)C1 c1(CC(N2C(C(=O)NCC3CCCOCC3)CCCC2)=O)ccc(F)c(Cl)c1 C=C1CON(C(=O)CNC(=O)CNC(C23CCCN2CCC3)=O)C1 CCC(O)C(C)(C)C(=O)N(C)CC1(CNC(C2COCCOC2)=O)CC1 C(CS(=O)(=O)c1ccc([N+](=O)[O-])cc1)N1C(C)CN2CCCC2C1 C1(NC(C2C(NC(CN(CCC)C)=O)CCO2)=O)C2CCC1CC2 CC1CN(C(c2cc(C(F)(F)F)n(C)n2)=O)CCCN1C(=O)CC1CC1(C)C c1(C(=O)NCC2C(O)CCN(C3C(C=C)OCCC3)C2)cc(Br)c(F)cc1OC C1(C)(C(N(CCCO)CCC)=O)CCCN(C(C2CC3(CC3)CN2C)=O)C1 Cc1cc(C)cc(C=CC(=O)NC2CCCN(C(=O)C(C)CN3CCCCC3)C2)c1 N1(C(Cn2cccc(C)c2=O)=O)CC2CCOCC2(NC(=O)C(=O)NC2CC2)C1 C1(NC(c2c(OC)nsc2)=O)CCCN(C(=O)CC2CCC(=O)N2)C1 C1(C(=O)NC(C)CNC(C2CCCSC2)=O)CCC2(CCCC2)C1 c1(COC)cc(NNC(=O)c2cc(C)oc2CC(=O)O)nc(C)n1 N1(C(c2cc(C)[nH]c2)=O)CCC2(CCN(C(c3ccc(F)c(Cl)c3)=O)C2)C1 Cc1ccc(C(N2CCCC2CN(C)C(C2CC(CF)C2)=O)=O)cc1Br c1(C(=O)NC(C)CNC(=O)CNC(N)=O)cccc(S(C)(=O)=O)c1F C#Cc1ccc(CC(=O)NCC2CCN(C(=O)CC3CC(F)C3)C23CC3)cc1 c1(OC(C)C)cc(CNC(C23CC(C(=O)O)C(C2)C3)=O)cc(C#N)c1 CC1(C)CC(NC(=O)C=C2CCCC2)CN(C(c2ccc(F)cc2)=O)C1 CC(C)(C(=O)NC1CCCC1NC(c1ccc(F)cc1F)=O)C(F)(F)F c1(C(=O)NCC2C3CN(C(CCCCC)=O)C2C3)cnn2c1S(=O)(=O)N(C)CC2 C(N=c1nnn(C)[nH]1)c1cccc(NC(COC2CCCC(C)C2)=O)c1 C(CC(C)(C)C)(C(=O)NCC1(C(=O)Nc2cccc(OCF)c2)CC1)OC C(C(C)(C)C(=O)OC)c1cn(C(COCC)C)nn1.N12CCC1C2=O n1(CC)nc(C2CC2)cc1C(=O)N.c1nccs1.N1(CC=O)CC(C)C1.C C=CCCCCCC(=O)NCC(O)CCNC(c1c(F)cc(N)cc1F)=O c1(C(=O)NC2(C)CCCCC2)ccc2ncsc2c1.C12(C=O)C=CC(CC1)C2.N C1(NC(CNC=O)=O)CN(C(C2CC(n3ccnn3)C2)=O)CCC1F CCCCC(=O)N1CCC(CNC(=O)C=CCNC=O)C1.C(C)(C)C Cc1noc(Cl)c1CCC(=O)NC(C)CNC(=O)CC1CCC(=O)O1 C(CCCCC(=O)NC(c1ccccc1)C(C)NC(=O)Cc1ccccc1F)SC c1(C(N(C(CCNC(C(c2cccc(C)c2)(C)C)=O)C)C)=O)ncc(F)cc1F N1(C(C2CCN(C)C2)=O)CC2=C(C1)CN(C(=O)C(F)(F)CC1CC1)C2 C1(CNC(C2N(C(C)=O)CCC2)=O)CCCN(C(=O)CC2CCCCCC2)CC1 N1(C(C(CC)CN(C)C)=O)CCC(F)CC1C(=O)NCc1nnc(C)s1 c1(OC(C)C(=O)NC2(CNC(c3ccon3)=O)CCC2)cccc(N)c1 N1(C(C(C=O)C)=O)CCC(O)(CC(=O)N(C)CCC2CC2)CC1.C(C)=O.CO CCC(C#N)C(=O)N1CC=CC1C(=O)NOCC1CCOCC1 c1(OC)ccc2c(c1)OCCC2C(=O)Nc1nc2ccccn2n1 c1(N2CCCC(N(C(Cc3c(C)nc(C)s3)=O)C)CC2)ncnc2[nH]ccc12 Cc1cc(C(=O)N(C)C(C2CCC2)C)nn1-c1ccc(F)cc1 c1(C(N2C3CC(NC(CCc4cc(C)[nH]n4)=O)C2CC3)=O)cnn2ccccc12 C(=O)(C(O)C(C)c1ccccc1F)N(C)CC1N(C(C2CC(SC)C2)=O)CCC1 N1(C(CCC(=O)NC)=O)CCCN(C(=O)CC2NC(=O)CN(C)C2=O)CC1CO c1(C=O)ccc2nc(C)oc2c1.N1(CCNC(C2C(CC)C2)=O)CCNCC1.N C1(C(=O)N)(N(C)C)CCC(F)(F)CC1.C1(NC(c2cc(C)sc2)=O)CCCCC1 Cn1cnc2ccc(C(=O)NC3(CNC(C4CCCCS4)=O)CCOCC3)nc12 CN1CCCC1CCC(=O)OCc1csc(CCc2ccccc2)n1 C1(OC)CCCCN(CC(=O)NCC2CN(C(=O)CC)CC2O)C1=O.C(C)=O.N CC1(C)C(C(=O)NC(C)(C(=O)NCC2CCCCS2)C2CCC2)C1(C)C c1(-n2c(C(C)Cc3cnn(C)c3)nc(CCOC)n2)nc2ccccc2n1C C1(NC(C2CC(OC)C(OC)C2)=O)CN(C(c2nncs2)=O)C2(CCOCC2)C1 C1(NC(C2CC(C)OC(C)C2)=O)CCSC12CN(C(C1CC3(C1)CC(F)C3)=O)C2 C1(CN(CCN(C(=O)CCn2cncn2)C)C)CCN(S(=O)(=O)C(F)F)C1 C=CCC(CC(=O)NOCC(C)C)NC(=O)C(C)N1CCCC1 c1cn2ccc(Br)cc2n1.c1(OC)ccc(C#N)cc1NC(C1CC1C=O)=O.N Cc1ccc(SCC(=O)NC(C)(C)C(C)NC(=O)CCc2cncnc2)cc1C CC(C)C(CNC(c1ncnn1C)=O)NC(c1cc(C2CCC2)no1)=O S(=O)(=O)(c1cccc(S(C)(=O)=O)c1)N1CC2N(S(CC=C)(=O)=O)C(C2)C1 c1(CC)cc(NC(C2CCN(C(c3cnc(C4CC4)o3)=O)CCO2)=O)ccc1F C1(NC(=O)CC2C=CCCC2)CCCCC1NC(c1ccnc(OCCO)c1)=O C(CC(=O)NCc1ncc(C)cc1C)(C(C)CC)NC(C(CCCC)O)=O C(C)(CO)(C(=O)NCCCC(C)(C)OC)NC(CCCOC)=O c1(CCC(N2CC(OC)(C)C2)=O)c(N)cnn1C.c1(C=O)occc1C(C)C n1(CC(=O)NCC(CNC(CN2C(C)CC2)=O)O)cc2ncccc2n1 c1cccc(F)c1.C1(OCC)(OC)CC(C(N2CC(C)C2)=O)C1.C(=O)C.N C(=O)(C1=C(F)CN(C(=O)C(=O)CCC(C)C)CC1)NC1C(OCC)CCCC1 N(C(=NCCCC1CCOC1=O)NCC1CCCCO1)C1CCN(C(C)=O)CC1 c1(N(C(=O)C(O)CNC(CC2(CC(=O)OC)CC2)=O)C)ccc(O)cc1 c1(C(N(C2CN(C(=O)CC(C)(C)N(C)C)CCC2O)C)=O)ccc2n[nH]cc2c1 C1(C)(CNC(C(C)(C)SC)=O)CCCN1C(C1CC(C(C)C)C1)=O c1(C(=O)NC2CC3CC(NC(=O)CSC(F)(F)F)CC32)cn2ccccc2n1 c1(N2CCC(N(C(C(CC)(C)O)=O)C)CC2)nc2ncc(Cl)cc2s1 CC1(C(=O)NC2CN(C(=O)Cc3coc(C(F)F)n3)CC2O)COCCO1 C1(C(=O)NC(CC#CC)C(=O)NC2CC2(C)C(F)F)Cc2ccccc2C1 C(c1ccccc1)=CC(=O)N.c1(CC)ccc(C(=O)NCCC2CCOC2)s1 N1(C(Cc2cn(CC)nc2)=O)CC2(CCN(C(=O)CC3CC(OC)C3)CC2)C1 c1(N(C)C)cc(NC(c2cccc(CN)n2)=O)cc(F)c1 c1(OC)ccc(NC(=O)C(c2cn(C(C)C)nc2C)N2CC3CC3C2)cc1 c1(C(N2CC(OC)CC(Cc3n(CC)nnn3)C2)=O)ccc(C)c(OC)c1 C1(C2(C(N(C(CNC(C3C=CCC3)=O)C3CC3)C)=O)CCC2)CCCCO1 c1(C(N2CCC(NC(CC(CCC)C)=O)C2C2CC2)=O)cccc2oc(C)cc12 S(=O)(=O)(c1cccnc1)N(CC(=O)NC(CC(C)NC(C(CCC)C)=O)C)C Cc1ccc(Br)cc1CN1CCC(NC(=O)CCc2ccc(F)cc2Br)C(F)C1 C1(C(C)C(=O)NC2(CC3CC3)CCC2)CCCN(C(c2cccnc2)=O)C1 N1(C(Cc2nnc(C)s2)=O)CCCC(C(C)NC(=O)CCOCC(C)C)C1 C(=O)(Nn1ccccc1=O)C1CC2CN(C(C(C)(C)C3CCC3)=O)CC1C2 C#Cc1ccc(Cl)c(C(=O)N(C)CC2CCCN2C(=O)C(CC)CCC)c1 C1(NC(=O)OC(C)(C)C)CCOCC1C(=O)NCCC.c1cccc(Br)c1.N Cc1ccc(-n2cnnc2SCC(=O)N(CC(C)O)CC)cc1.C(=O)(CC#N)N CC(C)CC(C)CC=O.C(CC#CBr)OCO.C1C(=O)O1.C(COCC)O.O c1(C(=O)NC2C(N(C(c3cn(CC)nn3)=O)C)CCCC2)ccc2ccoc2c1 CCCCCC(CCCCC)C(=O)N1CC(NC(c2cocc2C)=O)CC(C)C1 c1(CCC(=O)N)cnc(C)o1.C(=O)(CCC1CCC1)N(CCCC)CCOC CCCC(O)CC(=O)NCC1(C)CCCN1C(c1coc(C2CCC2)n1)=O C1(NC(CCCNC(C)=O)=O)COC2C(NC(=O)C(c3cccnc3)O)COC12 Cc1cc(NC2CC(NC(c3occc3Br)=O)C23CCC3)ncc1[N+](=O)[O-] C#Cc1ccc(OC)c(NC(c2oc(CN)nc2C)=O)c1 C(C(CC(C)C)C(=O)NCc1cc(C(=O)NCCCC(=O)N(C)C)co1)OC N#Cc1cc(F)ccc1C(N1CC(F)(C)C1)=O.C1(CCC=O)CCCC(=O)N1.N c1(CCC(N2CCC(C(C)NC(=O)Cc3nccn3C)C2)=O)cccc(F)c1Cl C1(C2CCN(C(=O)CCc3cncs3)C2)(NC(=O)CN2CC3C=CC2C3)CC1 C1(NC(C2CCCN(CCC)C2)=O)CN(C(C2CC2(C)C)=O)CCC1C c1(C(C)=O)sc(C(=O)NCC(=O)Nc2ccc(Oc3ccccc3)cc2)cc1C N1(C(C2C(C=C)CC2)=O)CCC2(CC1)CCN(C(c1oc(Br)nc1C)=O)C2 C=CC(CC)C(=O)N(CC(=O)NC(Cc1ccccc1Br)C(=O)NC)C1CC1 C1(C(=O)NCCCC(C)(C)OC)CN(C)CCN1C(c1n[nH]c2c1COC2)=O C(CC(C(=O)N1CCC1CC)NC(=O)Cc1csc(C)c1)OCC Cc1cc(C)c(C(=O)N(CC(C)NC(c2cnnn2C)=O)C)s1 CC1COc2c(C(=O)NC3CN(C(C4CC(=O)OC4(C)C)=O)C3)cccc21 c1(C(N2C(CNC(=O)NCCCCl)CCC2)=O)cc2cc(Br)ccc2s1 N1(Cc2cc(OC(CC)C)c(OC)cc2)CCOc2ccccc2C1C(=O)O C(C)(CCC(=O)NC1CCN(C(c2ccoc2CC)=O)C1C1CC1)OCC O=C(CCCF)NC1CC(CNC(C2CSCCS2)=O)C1 S(=O)(=O)(c1cccc(Cl)c1)N1CCN(C(c2cc(Br)cc(OC)c2N)=O)CC1 C(=O)(C(C)CC(C)C)NC1CN(C(C=Cc2ccc(C(=O)OC)o2)=O)C(C)C1 n1(CC(=O)N(C(=O)Cn2cc(C)cn2)CCN(C)C)nc(C=O)cc1C Cn1cnc2c[nH]c(=NCC=CCNC(=O)CC(c3cccc(F)c3)O)nc12 CCCC(C)N=c1cc(NCc2ccc3c(n2)OCCO3)nc(C(C)C)[nH]1 c1(CNC(C(C)SCC)=O)nc(C)cc(O)n1.c1(C=O)cnc(C#N)s1 c1(C(=O)N)cnn2c1NCC(C)C2.c1(OC)ccc(C(=O)NC(C)CC)c(Cl)c1 c1(C(=O)NC(CNC(CCCN(C)C)=O)CO)cc(C2CC2)oc1C1CC1 C1(C)(NC(C2C(C)C2)=O)CC(NC(=O)CCc2cnc[nH]2)C1 C(C)(C)(CCCCC(=O)N(C(C)CCNC(=O)CN1CCNC(=O)C1)C)OC c1(C(N2CCC(C)(NC(c3c(CC)non3)=O)C2)=O)c(Cl)nc2cc(Cl)ccn12 c1(C(N2CC(CCNC(c3ccc(-c4ccccc4)[nH]3)=O)C2)=O)cncnc1 N1(C(c2c(C)scc2)=O)CC2(CCC(C)O2)C1.N1(C(C(=O)N)=O)CCCC(C)C1 C1(C(N2CC3C(NC(c4cc(C)n(C)n4)=O)(CC3)C2)=O)CCc2nncn2CC1 O=[N+]([O-])c1cccc2c1CCN(S(=O)(=O)C1CCOCC1)C2 Cc1ccc(Cn2nccc2NC(C2CC23CCOCC3)=O)c(C)c1 c1(C(N2CCC(NC(c3cc(C)c(C)s3)=O)C2)=O)cc(C2CC2)cc(F)c1 c1(OC)ccc(C(N2CC(O)CCC2C)C(=O)NCC2CC2)c(OCCO)c1 N1(C(CC2CC(OCC)C2)=O)CCCC(CC(=O)NCC(F)CO)CC1 C1(NC(C(C)CC2CC2)=O)CCCC(NC(=O)CSc2cccc(F)c2)C1 C(=O)(CC(=O)O)NCCOC1CN(C(=O)OC(C)(C)C)C1.C1CCC1 C1(C(N2C(C)CC(NC(c3c(C)coc3)=O)C2)=O)CC(C)(C)SC(C)(C)C1 C(=O)(C(C)(CC)CCC)NC1C(NC(C(CCC)O)=O)COCC1 c1(C(N(CC(=O)Nc2sccc2C(N)=O)C)=O)cc(Br)ncc1F N1(C(C2N(N=O)CCC2)=O)CCC2CCC(C1)N2C(=O)COCc1ccncc1 c1(OC(C(=O)NCCCNC(C(C=C)(C)C)=O)CC)ccc(Br)cc1F C1(CC(=O)N(C(CNC(CC2CC(CC)C2)=O)C)C)CC(=O)NC1=O C1(C(N2C(C(N3CC(OCC)C3)=O)C=CC2)=O)CCC(O)CC1 C1(NC(c2n(CC)c(O)nc2)=O)CCC12CN(C(c1ccc(F)cc1C)=O)C2 Cc1cc2scc(CC(N3CCCC(NC(c4ncccc4Cl)=O)C3)=O)c2s1 Cc1cc(=NCc2ccncc2)[nH]c(=NCC2CCCC2N2CCCC2)[nH]1 CC1CCC=C1C(=O)N1CC(C)(NC(c2cccc(C3OCCO3)c2)=O)C1 c1(C(C(N2C3CN(C(=O)CC4CCCOC4)C(C3)C2)=O)O)cccc2c1OCC2 CCCCCCC(=O)N(C1CCCN(C(c2cc3n(n2)CCC3)=O)C1)C C(=O)(C(CO)CC(C)C)NC1CC2CN(C(C3(CC)CC(C)(C)C3)=O)C1C2 N1(C(CCCCC#N)=O)CC2CCC(NC(c3ccc4ccnn4c3)=O)(C2)C1 c1(CC=O)n[nH]c(=NC)s1.C(C)(C)C.C1(CC)CC1C(=O)NCCO c1(C(N2C(C)CC(NC(C3C4COCC34)=O)C2)=O)cccc2c1NCC2 N1(Cc2cccc(C#N)c2)CCC2(CC1)CC2C(=O)Nc1ncncc1Cl c1(C(CNC(c2n(CC)ncc2)=O)NC(=O)C)ccc(F)cc1.CCC.O CC1(C)CNCC(CN2CCC(O)(C(N)=O)CC2)C1 c1(C(=O)NC2CCN(Cc3nnc(CC)s3)CC2O)cnc2[nH]c(O)nc2c1 C=Cn1nncc1C(=O)NC1CCOC1C(=O)Nc1cscc1CC CCC(C)(C)C(O)C(=O)N(CC(=O)NC1CN(C)CC12CC2)C1CC1 CC1CCCC=C1C(=O)NCCOC1CCN(C(=O)CS(=O)(=O)N)C1.C1CC1 C(CCS(C)(=O)=O)(C(=O)N1CCC1C(F)(F)F)SC CC1(C)CCCN(C(c2cnnn2C2CCCNC2)=O)C1 N1(C(C2(CC(C)C)CCCC2)=O)CC2CCN(C(=O)C3=CC(C)(C)C3)CC2C1 C(N=c1nc(N2CCC(N(C)C)CC2)c2c([nH]1)CSC2)c1c(C)ocn1 C(=O)(CN=c1ccc(C#N)c[nH]1)NC1CCC(NC(C=C(C)c2ccco2)=O)C1 c1(OCCC)ccc(C(=O)NCCCCCNC(=O)CSC)cc1OC C1(CNC(CCCC)=O)CC2(CN1C(c1sccc1SC)=O)CC2(F)F C1(CC(=O)NCC2(NC(=O)CCc3cnccn3)CCOC2)CC(=O)NC1=O n1(CCC)ncc(C(=O)NC2CC(C)N(C(c3cc(C(C)=O)cs3)=O)C2)c1C C1(NC(CCNS(C)(=O)=O)=O)CCCC(NC(=O)CN2CCC(O)CC2)C1 c1(C(C2CCN(C(=O)N)CC2)C(=O)OCC)ccc(Cl)cc1.c1ccnc(C)c1 CC1CCN(c2cc(C(C)(C)C)nc(Cl)n2)CC1NC(=O)COC1CCOCC1 CCCC(C(=O)NC(C)(CNC(=O)Cc1sc(O)nc1O)C1CC1)OC C(c1cccc2cccnc12)=CC(=O)NCC1(C)CCC(F)(F)CC1 N1(C(CSc2n(C)cnn2)=O)CCC2(CNC2)C1 N1(Cc2c(C)nc(C)[nH]2)CCn2c(Cc3ccccc3F)nnc2C1 c1(C(=O)NC(C)CCCNC(c2ccc(C(F)F)cn2)=O)cccc2nncn12 c1(C(C(=O)NC(CCNC(C2CC(C(=O)OC)C2)=O)C)CO)ccc(Cl)cc1 N1(C(C=C2CCN(C)CC2)=O)CC(CNC(=O)Cn2cncn2)OC2CCCC12 N1(C(CCC=CC)=O)CCC2CCN(C(=O)CSc3cnn(C)c3)CC2C1 N1(C(CCSCC)=O)CC2CC(C1)N(C(=O)CCNC(c1ccccc1)=O)C2 N1(C(CCC)=O)CCCC(C(C)NC(c2cc(C3CC3)on2)=O)C1 C(=O)(C(F)(F)c1cncs1)N(CCCCNC(C(=C(C)C1CC1)F)=O)C N1(C(c2c(OC)cccc2OC)=O)CC2(CCCN2C(c2cscc2Br)=O)C1 C1(COC)CCCN1C(=O)CCCC1CCC1.C1(C#N)(CCC(=O)N)CCC1 CC1(C)CCCN1C(c1ccc(C(N)=O)cc1)=O.C1(C=O)CC(F)C(=O)N1.N Cc1cc(=N)[nH]cc1C(N1CC(N(C)C(C2COC3(CCC3)C2)=O)C(C)(C)C1)=O c1(C(N2CCCC(NC(C3CC4CC4N3)=O)C2)=O)ccc(Br)c(C(F)(F)F)c1 c1(CCCNC(=O)C(F)n2cccn2)cn(Cc2ccccc2)nn1 c1(OC)ccc(CN2CCCC(C(=O)NCCC#N)CC2)cc1C C1(CC)(NC(c2ccc(Cl)cc2Cl)=O)CCN(C(c2nc(=N)cc[nH]2)=O)CC1 C(N=c1nc[nH]s1)C1CC(NC(c2ocnc2CC2CC2)=O)C1 Cc1ccc(C)c(CN2CCC(NC(c3cccc(=O)n3O)=O)C(F)C2)c1 C(=O)(C1CCc2nccn21)N1C(C)CN(C(c2ccc(F)o2)=O)CCC1 c1(C(N2CCC(NC(C(CC)NC(C)=O)=O)C(C)C2)=O)nccc2ncccc12 C1(NC(c2c(CC)ncs2)=O)CCCN(C(c2ccncc2N)=O)CC1 CC1CCN(C(c2cccnc2C(F)F)=O)CC1NC(C1CC(O)(C#N)C1)=O CC(C)C(CO)C(=O)NC1CCN(C(=O)COC2CCCCC2)C1(C)C c1(OC)c(Cl)ccc(C(=O)NCCN(C)C(C2CCCCCC2(F)F)=O)c1N c1(CN2C(C(N(C)Cc3ccc(CC)cc3)=O)C=CC2)cc(C)cc(C)c1 Cc1oc2ncnc(O)c2c1C(=O)NCCNC(=O)CC1CCc2ccccc2N1 n1(CC2N(C(CC3CC(CC)C3)=O)CCC2)cc(CCNC(C)=O)nn1 c1(CC=O)ccc(Cl)c(C)c1.C1CCN(C(=O)C=C(C)C2CC2)C1.CO.C C(=O)(CC1CCOc2ccccc21)OC.N12CCC(C1)NC(=O)OCC2=O c1(CN(C)C(c2cnc(C3CCCN3)nc2)=O)ccncc1Cl C12(NC(CC(=O)OC)=O)CCCCC1CN(C(C13CCCC1OCC3)=O)C2 Cc1cnc2n1CCCC2C(=O)NC(C)CCNC(C1CCCCC1)=O C(=O)(C(CC(C)C)NC(C1CC(C)(O)C1)=O)N(CC(C)(C)OC)C c1(OC)ccc(C(=O)NC2CCCC(NC(=O)CN3CCOC3=O)C2)cn1 C=CC(CC)C(=O)N1CCC2CC12C(=O)NCc1ncn(CC)n1 N1(C(C=C2CCN(C)C2)=O)CCN(C(c2ccc(C(N)=O)c(Cl)c2)=O)C2CC12 C1(C(=O)NCC=CCC(=O)NC(C)CCOC)(CC)CNC(=O)C1 c1(CC(C)NCc2cnc(-n3cccn3)s2)ccc2nonc2c1 c1(CNC(=O)C=C2CCN(C(c3cc[nH]c3)=O)CC2)ccc(Br)cc1F N1(C(c2nc(CCC)sc2)=O)CCC(O)(C(C)NC(=O)Cc2ccon2)CC1 N1(C(C(C(C)C)C(C)NC(=O)CC2=NN(C)C(=O)C2)=O)CCC2(CCC(O)C2)C1 C1(NC(C=C(CNC(c2cncc(NC)c2)=O)C)=O)CC2CCCCCC12 Cc1ccc(C(N2CCCC2CN(C(=O)CCC2CCC(=O)NC2)C)=O)c(Cl)c1 C(c1cccc(F)c1Cl)=CC(N1CCN(C(C2C(CC)OCC2)=O)C(C)C1)=O c1(CC2(NC(=O)C3CC3)CC2C(F)(F)F)cnn(C2CC2(F)F)c1 c1(C(N(C2CCN(C(=O)C(F)C3CCC3)C2)C)=O)ccc2nnn(O)c2c1 c1(C(N2CCC(C)(C)C(C)C2)=O)n[nH]c2c1C(=O)CCC2.C(=O)(C)N.C(N)=O C(CC(CC)C(=O)N(CCCNC(c1ncccc1O)=O)CCO)=CC CCC(C)(F)C(=O)NCc1cccnc1CNC(=O)Cc1cncc(C)c1 C(=O)(C(CC)C(C)C)NCc1ccc(C)c(C)c1.C(=O)C=CCN1CCC1.N c1(C(=O)NC(C2CN(C(=O)CC3OCCO3)C2)C)cccc(CCO)c1 C(=O)(C(C)S(C)(=O)=O)N1CC(CC(=O)NC(C(=O)OC(C)C)C)OCC1 N1(C(C(=O)NCC(C)NC(=O)CCc2csc(-c3ccco3)n2)C)CCOC1=O C(=O)(C(=O)CCc1ccccc1)NCCCOC(=O)NCC.C1CCSCC1 Cc1ccc(-c2ccc(C(=O)N)s2)s1.C1(F)CN(C(=O)CC2COC(=O)N2)C1 N1(C(C2CN(C(C(C)OCC=C)=O)CC2F)=O)CCCC(C)(C)C1 c1(C(N(C)CCNC(=O)COCC2CCCC2)=O)cnc2ccccc2c1 c1(C(=O)N)cc(C(F)F)cc(Cl)c1.C1(OC)CCC(C(N2CC3CC3C2)=O)CC1 C1(C(N2CC(CN(C(CCC(=C)C)=O)C)C2)=O)Cc2cc(F)ccc2O1 C1(C(=O)NCCC(C)N2CCC2)CCN(C(=O)C(C)(C)C(C)O)CC1(C)C C(=O)(C(O)C(F)(F)F)NC(C(C)C)CCN(C)C(c1cc(Cl)ns1)=O c1(-c2cn(C3CCN(C(C4(CC=C)CC4)=O)CC3)nn2)cc(C(C)=O)ccc1C Cc1ccc2occ(CC(N3CCC(NC(C4(O)CCC4)=O)C(CO)C3)=O)c2c1 S(=O)(=O)(c1ccccc1F)Nc1scc(-c2cc(C(C)C)c(F)cc2)c1 Cc1c([N+](=O)[O-])c(C(=O)NC2CCC2)nn1C.C1(C=O)C(C)(C)C1(F)F.C C=CCCCC(C(=O)N1CC(CC2CC2)C1)NC(c1cscc1OC)=O c1(C(=O)NC(CNC(C(C(C)(C)O)F)=O)(C)C2CC2)cccc2[nH]ncc12 C1(CC)CN(C(c2cc(Cl)n[nH]2)=O)CCC1C.c1(C=O)cnn(CC(F)F)c1.N C1(CNC(=O)CNC(N2CCCC2)=O)CN(C(C2CCC=CCC2)=O)CC1O c1(-c2cn(Cc3c(CNC(CCCCSC)=O)ocn3)nn2)cc(F)ccc1F C(=O)(CC1=CCCCC1)N1CCC(C(=O)NCCCC(C)(C)C)C1(C)C c1(CC)nc(N2CCCCC2CNC(C2CCc3c[nH]nc3C2)=O)cc(C#N)n1 c1(CC)nc(N2CCC(CCNC(c3cncc(F)c3)=O)C2)c(C)c(Cl)n1 c1(CC)cccc(C(N2CCCC(CN(C(=O)CC)CC)C2)=O)c1.C(=O)N C(=O)(CCN1C(=O)C(C)Oc2ccccc21)NC(CCN(C(CCOC)=O)C)C N1(C(CC)=O)CC2CCC(C=O)(C2)C1.CC(C(C)C)C(C)C.C(C)OCC.O C1(NC(c2n(C)nnc2CNC(C2C3COCC23)=O)=O)CC2CCCC(C1)C2 Cc1cc(NC(=O)C=CCN(C(=O)CC2(N(C)C)CC2)C)n(C)n1 C(=O)(CCC(C)NC(=O)C(C)(C)CN(C)C)NCC1C(CC)OCC1 N1(C(C=CCCC)=O)CCN(C(C2(Sc3ccccc3)CC2)=O)C2(CCC2)C1 C1(C(=O)NCc2ccc(SC)o2)CN(C(c2ccc(F)cc2F)=O)CCC1(C)C C1(CC(N2CC(C=O)C2)=O)CC2(CC2)CO1.CC(C(=O)N)C1CCCC1.CC c1(C(=O)NCC(CNC(C(C2CCC2)OC)=O)CO)c(Cl)n[nH]c1C1CC1 CCC(C)C(C(=O)N1CCN(CCNC(c2cc(C(N)=O)co2)=O)CC1)OC N1(C(c2cc(C3CC3)nn2C)C(=O)NCC)CCCC(N2CCOCC2)CC1 CCCC(O)C(CO)NC(c1[nH]ccc1CNC(=O)CO)=O.CCN(C)C C1(CC)CN(C(C2CCC2c2nc[nH]n2)=O)CCN1C(c1n[nH]c(C)c1O)=O C1(NC(C(CC)(C)CO)=O)CC2CCC1C(NC(=O)CCc1nnc(C)n1C)C2 C1(C(N2CC(C)(C#N)C2)=O)CC12CCN(C(c1sccc1Cl)=O)C2 N#Cc1cnc(NC2CN(C(=O)CSC(F)(F)F)CCC2C(F)(F)F)c(Cl)c1 C(=O)(C(C)CNC(c1ncoc1CNC(C1CC1(Cl)Cl)=O)=O)NC c1(C(N(C)CC2(O)CCN(C(c3cc(C)ns3)=O)C2)=O)ccc(C)c(C)n1 c1(C(N2CCN(C3CN(C(CCN(C(C)=O)C)=O)C3)CC2)=O)ccc(F)c(O)c1 N1(C(c2c(CNC(C(C)N3CCCC3)=O)c[nH]n2)=O)CC(C2CC2)C1C1CC1 c1(C(N2C(C)CCC2)=O)cc(O)nc(Cl)c1.c1(C(C)=O)ccc(C(=O)N)nn1.C CC1CCCN(C(c2ccc(F)s2)=O)C1C.c1(CC(=O)N)cccc(C2CC2)c1 C1(C(=O)NCC(C)NC(=O)C(F)(F)Sc2cnn(C)c2)CCCC(C)CC1 C(=O)(C1Cc2ccc(F)cc21)N1CCC(NC(c2c(C)nccc2Cl)=O)C1C c1(CC)nc(C(=O)NC(CNC(=O)C(O)C(F)F)C2CCC2)c(N)s1 CCCC(C)OCCC(=O)NCC=CCNC(C1CC(C(C)C)C1)=O C1(NC(C=CCOC)=O)CCN(C(=O)C(Cc2ccccc2)OC)CC12CCC2 c1(C(=O)NCCC(C)NC(C(CC)COC)=O)cc2c(cn1)NC(=O)CO2 n1(CC)cc([N+](=O)[O-])c(COC(=O)CSC2CCOC2=O)n1 c1(C(N2C3CC(CNC(C(CCOC)C)=O)(OC3)C2)=O)cnc2sccn2c1=O N1(C(=O)C=Cc2cscn2)CCC2CN(C(=O)Cn3cnnn3)C2C1 N1(C(C(C)OC2CCCC2)=O)CCC(C)(C(=O)NC2CCN(C)C2)CC1 N1(C(C2CCC(NC(C)=O)CC2)=O)CCc2c(ncn2C)C12CCN(CC#N)C2 C1(C(N2C(C)(CC(=O)NCc3nc(C4CC4)no3)CC2)=O)C2CC(=O)CC12 C1(CC=C)(NC(c2ccc(C)cc2O)=O)CCCN(C(=O)C=CC2CCOC2)C1 C1(C(=O)OC(C(=O)OCC)C2CC2)Cc2cc(Cl)ccc2C(=O)O1 CC(C(=O)NCC(C1CCN(C(c2ccncc2)=O)CC1)F)C(F)(F)F.N(C)C.C n1(C(C)(C)C)ccc(=NC(=O)C(O)C2CN(C(=O)CC3CC(=O)C3)C2)[nH]1 c1(C(C(=O)NC(C)CCNC(C2(O)CCSC2)=O)(F)F)cccc(Br)n1 c1(NC2CCCCC2)cc(NC)ncn1.Cc1cc(C2CCC2)no1.[SH](C)(=O)=O Cn1ccc2c(-c3ccc(CNCc4ccc([N+](=O)[O-])cc4Cl)cn3)cccc12 c1(C(C(=O)N(C)CCNC(C2(C(=O)O)CC2)=O)N(C)CC)ccccc1 C1CN(C(C2CC(=O)N(C(C)C)C2)=O)CC1(C)C.C(C(=O)N)=CC=CC C(=O)(C(CC(C)(C)C)NC(=O)CCC=C(C)C)N1CC(O)CC(OC)C1 C1(C(C(=O)NC2C(OC)COC2)C)CCN(C(c2ncccc2O)=O)CC1 N1(C(=O)CCN(CCCO)C(C2CC2Cl)=O)CCC2(CCO2)C1 c1cnc(C(c2nnnn2C2COC2)OCCN(C)C)s1.C1(NC)CCCN1C c1(C(C)C)ccc(C(=O)NCCCNC(C2CCCC2n2cccc2)=O)c(O)n1 c1(C(=O)NCCNC(C2(O)CCC(CCC)CC2)=O)nc[nH]c2ncc(C)c1-2 N1(C(CCC2CCC(C)O2)=O)CCC(F)(CNC(=O)CCCn2cncn2)CC1 c1(OC)cc(CC(=O)NC2COCC2NC(=O)CCCC(=O)N(C)C)ccc1F C(=O)C1=CNC2=NCCC2=C1.C1(NC(C(=O)NCC(F)F)=O)CCCC1C.N N1(C(C(C)Oc2ccc(Cl)cc2)=O)C2CCC1C(NC(C1(O)CC1)=O)C2 c1(C(=O)NCC2CC3CN(C(=O)CC(F)(F)F)CC23)cc(F)c(O)c(Cl)c1 Cc1cncc(C(=O)N(CCCNC(C2CC(F)C(=O)N2)=O)CCO)c1 N1(C(C2C(C#C)C2)=O)CC2=C(C1)CN(C(c1cc(OC)c(Cl)cc1OC)=O)C2 c1(CC(=O)NCCCCCCNC(C(F)=C(C)C)=O)c(F)cccc1Br Cc1cc(C(N2CCC(NC(C3CC3C(F)F)=O)C2(C)C)=O)c(N)c(Cl)c1 C=C1CC2CCCC(C1)N2C(C1(NC(C2CNC(=O)C2)=O)CCC1)=O C(CC(CC)C(=O)N1CC(CC(=O)NC2CCC(CO)C2)(OC)C1)=CC c1(C(N2CC(C)CC(NC(CCSC)=O)C2)=O)cnc2cccnn12 C(=O)(C(CNC(C12CCC(CC1F)C2)=O)C(C)(C)C)N(CCN=[N+]=[N-])C c1ccccc1.c1(OCC)n[nH]cc1C(=O)NCC1CN(C(=O)CC)C1.O C1(C(N2CC(N(C(=O)CCCc3ncco3)C)C2)=O)CCc2nnc(O)cc2C1 c1(SC)cc(C(N2CCC(C)C2CNC(=O)Cc2cnco2)=O)ccc1F C1(NC(CC2(OC)CCC2)=O)CC2CCC(C1)N2C(=O)CC1(C)CC1(F)F C1(NC(C2N(C(CCNC(C)=O)=O)CC=CC2)=O)CC2(CCOC2)C1 C1(C(=O)N)CN(S(N)(=O)=O)C1.c1(CC)sc(C(N2CCC(C)C2)=O)cc1C O=C1CCC1C(=O)NC1CC(CCNC(C2(C(F)(F)F)CCO2)=O)C1 C1(CC(N2CC3C(NC(c4ccn(COC)n4)=O)(C3)C2)=O)CC2(CCC2)CO1 C1(C(N2CC(CC)C2)=O)CC2(C1)C(F)(F)C21CC1.CC(C(=O)N)c1ccco1 S(=O)(=O)(CCC(F)(F)F)NC1C(F)CCN(C(c2cncc(OC)c2)=O)C1 c1(C(N(C2CCC2)C)=O)ccc(S(C)(=O)=O)cc1Cl.CC1=CCC(C(=O)N)CC1 CN1CCN(C(c2ccc(C(F)(F)F)o2)=O)C(CNC(=O)C#CC(C)(C)C)C1 CCC(C)CC(C(=O)N1CC(C)(COC)C1)NC(c1ccnnc1O)=O c1ccc(C)cc1.C1(CCNC(C2(CCCC)CC2)=O)CN(C(=O)CCO)C1 Cc1cncc(OCC(=O)NC2CCC2NC(c2cnn(C3CCCC3)c2)=O)n1 Cc1cc(CC(N2CC(NC(=O)CCCC(C)C)C3(CC3)C2)=O)cc(F)c1 c1(-c2ccc(C(=O)OCC)cc2)ccc2cc(-c3ccnc(OC)c3F)sc2c1 Cc1nc2ncccc2cc1CCC(=O)NCC#CCNC(=O)CNC=O c1(CC)cccc2[nH]c(C(=O)NC3CCCN(C(=O)C(C)=CC(C)(C)C)C3)cc12 C(=O)(C(C)CC(C)C(C)=O)NCC1CCC(C(N(CCF)CC)=O)CC1 CC1(C(=O)NCC2CCCN(C(c3csnc3Cl)=O)C2)CCCOC1 C(=O)CS(=O)(=O)C(C)(C)C.Cc1cccn(CC(=O)NCC2CCC2)c1=O.N C#CCC(C)C(=O)NCC1CC(COC)CN1C(c1cc(CC)c[nH]1)=O c1(CNC(CN(C(=O)C(C)C(F)F)CC)=O)ccnc(Cl)c1 C=CCCC(F)(F)C(=O)NCC1CC12CCN(C(=O)CC1SC(=N)NC1=O)CC2 CC1(F)CCCCN(C(C2CCN(Cc3cccc(-n4cncn4)c3)C2)=O)C1 c1(NC(COC)C2CC2)cc(NC(c2ccc(C)o2)C)ncn1 C=CCCCCCCCC(=O)NCC1C2CN(C(=O)CC3CC34CC4)CC12 CC#CCCC(=O)N(CCCNC(=O)CC1CCC(=O)N1)C(C)C CC1CCN(C(c2c[nH]c3ncccc23)=O)CCN1C(c1cn2c(n1)SCC2)=O C(CCN(C(=O)Cc1ccccc1C(C)C)C)C(C)(C)C.C(C=O)SCCC c1(N(CCC(C)CO)C)ccnc(NCCC(C)N(c2ccccc2)C)n1 O=S(=O)(N1CCC(C(F)(F)F)CC1)N1Cc2ccccc2C2CCC1C2 c1(C(=O)NC2CC(C)N(C(c3ccc(O)cn3)=O)C2)cc2c[nH]cnc-2n1 C(=O)(C(C)CS(C)(=O)=O)NCC1CCN(C(CNC(C(CC)C)=O)=O)CC1 Cc1ncccc1C(=O)NC1(C(N2CCC2C(C)O)=O)CC1(C)C c1(CC=O)ccc2c(cnn2C)c1.c1(C(C)=O)cc(C(=O)NCCC)c(C)o1.N N(C(=NCCN1CCOCC1)NC1CC2CCC1O2)CC1(CO)C(C=C)C1 c1(C(=O)NC(CN(C(c2coc(C)n2)=O)CC)C)ccc(OC(F)F)cc1 C(=O)(CC(C)(C)C(F)(F)F)NC1C2N(C(Cc3scc(CC)n3)=O)CC(CC2)C1 CN1C(=O)CCC1CC(N1CC(O)CC1C)=O.c1(C=O)csc(C(F)(F)F)n1 N1(C(C2(C)CC(OC)(OC)C2)=O)C2CCC1C(NC(=O)C(F)(F)C(F)F)C2 c1(C(=O)NCCCN(C(C(N2CCC(C)C2)=O)=O)CCO)cc(C#N)on1 C(C)(C)(CNCCC1CCN1)OCCOC CC1(C(=O)NCCNC2CCSC2)CCCN1C(=O)Cc1ccco1 N1(C(CC2(OC)CCC2)=O)C2CCC1CN(C(=O)CC1(O)CC1)C2 c1(N2CC3(C(C(N(C)Cc4ccc(C#N)cc4)=O)C3)C2)ncc2[nH]ncc2n1 CC1(C)CCC(C(N2CCCC2CC)=O)C1.C(=O)(CC(C1CCC1)C1CCC1)N N1(CCC)CCCCC1C(=O)NCCOCCNC(=O)CCc1cncs1 c1(C(=O)NC2CCC(NC(=O)C=CCN3CCCC3)CC2)cccc2nonc12 C1(CNC(C(C)(C)c2ccno2)=O)CN(C(c2nncs2)=O)C2(CCC2)C1 c1(N(CC(N2CC=CC(NC(CCN(C)C)=O)C2)=O)C)ccc(C#N)cc1F C1(C(=O)NCCCc2n(C)nnn2)CC2(CCN1C(=O)CC1=CCCCC1)CC2 C(=O)(CN=c1cc[nH]cc1)N1CC2N(C(c3cc(C)c(C)[nH]3)=O)CC(C2)C1 C(CC(C)C(=O)N1CCC(C)(CC(=O)NC(C)(C)CC(N)=O)C1)=CCC c1(C(=O)OC)ccc(-c2cn(C3CC(C(=O)NC4CC=CCC4)C3)nn2)c(C)c1 c1(C(=O)NCC(C)CNC(C2CC3(CCCO3)C2)=O)cc(Br)c2cccnn12 N1(C(C=CC=O)=O)CCOCC1.CC(C=O)NC.C1(C=O)CC1.C1CC1 c1(C(=O)N)cc2ccc(N(C)C)cc2[nH]1.C(C)(C)(CC)NC(CCOCC)=O N1(C(C2(CCOC)CCC2)=O)CC2(CCN(C(C3(C)C=CCC3)=O)CC2)C1 c1(CNC(c2nc(C(C)C)sc2)=O)ccc(N2CCC(O)C2)cc1 c1(C(=O)NC2C=CCN(C(c3cc(COC)[nH]n3)=O)C2)cnc2ncc(Cl)cn12 C(C(=O)NCc1conc1CSC)(C(C)CC)N(C(CC(C=C)C)=O)C CCCCCCC(C)CC(=O)N(CCC)CCNC(c1c(C)nc(C)nc1C)=O c1(OCCC)cccc(CC(=O)NCC2CCN(C(c3nncn3C)C)CC2)c1 c1(C(=O)NCC2N(C(CSCCCC)=O)CCOC2)cc(C(F)(F)F)ccc1C C1(C(=O)NC(C(C2CCCCC2)NC(COCCC)=O)C)CCCCC1O N1(C(COCC)=O)CCC(C2CCN(C(C3COC(=O)N3C)=O)C2)CC1 N1(C(C(CC)N(C)C)=O)CC(NC(c2c(C)[nH]c(C)c2C)=O)C2(CCC2)C1 c1(C=O)cc2n(n1)CCCC2=O.C1(NC(c2ccsn2)=O)CC(C)C12CCC2.N CCCC(C(=O)OC)C(=O)NC1CCCC1NC(c1cnc(SC)s1)=O C1(C(N2CC(CC(CNC(C(CCC)C)=O)(C)C)C2)=O)CCc2nc(C)cn2C1 c1(C(=O)NCCCC(C)NC(C(C)SC(C)C)=O)ccc2nc(Cl)nn2c1 C1(O)CCCC1.C1(C(C)C(=O)N(C2(C(=O)N)CCC2)C2CC2)CCC(=O)N1 C#CC1CN(C(C2CCCC23CCC3)=O)CCN1C(=O)COC1CC1 CCCCCCCC(=O)NCC1COCCN(C(c2csc(C(=O)OC)n2)=O)C1 CC#CC1CCN(C(=O)C(C2(C)CC2)NC(c2ccc(C#N)cc2)=O)C1 c1(N2CCCC(CNC(C)=O)C2)cccc(S(=O)(=O)N2CCC(F)(C#N)C2)n1 C12(C(N3CC(C)C(O)C3)=O)CCC1CN(C(=O)C(=O)Cc1ccc(O)cc1)C2 N1(C(c2cccc(OC)c2)=O)CCC(N=c2[nH]c(Cl)ncc2F)CC1C N1(C(c2ncc(CSC)s2)C(=O)NCCOC)CCC(N(C)C)C(C)C1 C(CCC(F)(F)F)NC(C1(OC)CCCOC1)=O.C(C)(C(C)(C)C)=CC=O c1(NC(c2n(CC)cnn2)C)[nH]c(=NCC(=O)NCC2CC2)nc2scnc12 c1(C(=O)NC(CNC(C(C=C)O)=O)(C)C2CCC2)cnc(N)c(N)c1 C1(CCC)CCN(C(=O)OC(C)(C)C)CC1.c1nnc(S)n1C.C(=O)(C=O)N C1(NC(COCCC(C)C)=O)CCOC(C(=O)NCC(=O)NCCO)C1 CC(CCc1cccc(F)c1)C(=O)NCC#CCNC(c1cn(C)[nH]c1=N)=O N1(C(CN(C(COC)=O)C)=O)CC2CCC1C1CN(C(=O)C(C)COC)CC21 N1(C(c2nc(C)nc(O)c2)=O)CC(C)OC2(CCN(C(c3cc(F)c[nH]3)=O)C2)C1 N1(C(=O)CNCC2CC2(F)Cl)CC(O)(C2(CN3CCOCC3)CC2)C1 c1(C(N2CCC(C(=O)Nc3cn(C(C)C)nc3)CC2)=O)ccc(F)c(Br)c1F CCCC(C(=O)NCC1CC(CNC(c2cnn(C)c2CC)=O)C1)C(C)C C(C(C)N=c1nc(N2C3C=CCC2CC3)c2[nH]ccc2[nH]1)SC C(C(C)C(=O)N1CC(CNC(C2(CC3CC3)CCC2)=O)C1)OCC CC(C)CCC(C(=O)N(C)Cc1nc[nH]n1)NC(=O)CCC1CC1C N1(C(=O)NC(c2ncco2)C)CCOC2CCCCC12 c1c[nH]cc(Cl)c1=O.N1(C(C2CC(CF)C2)=O)CCCC1C1(C(=O)N)CC1.C C1(CNC(=O)C=C(Cl)Cl)CCC2(CO1)CC(NC(=O)CS(=O)(=O)CCO)C2 C1(C(N2CCC(NC(=O)C(COC)OC)C2)=O)(OCC)CCCC1 C(C)(C(O)C(=O)NCCN(C)C(C1CCCCC1)=O)SC.c1ccc(Cl)cc1.S Cc1ccc(C)c(-n2cc(C3C(C)CCN3C(C3(CCCF)CC3)=O)nn2)c1 C#CC(C(C)OC)NC(C1(N(C(=O)CC2CSCCO2)C2CC2)CCC1)=O C1(NC(c2c(CC)ncs2)=O)(CO)CCN(C(=O)C(c2cccnc2F)(C)C)C1 c1(C(N(C2CC3CCC2O3)C)=O)sc(Cl)cc1Br c1(C(=O)NC2C(NC(CC3CCC(=O)O3)=O)CCCC2)cnc2c(c1)CCOC2 C(=O)(CCCN(C)C)NC(c1cnn(C)c1)C.C1(C=O)CC(=C2CC2)C1 CC1CCCC(C)N1NC(=O)Cc1ccc(F)cc1 C1(C(=O)NC2CC(C)SC2)CCCN1NC(=O)c1ccn(C)c1 N1(C(C2(C)CC3CC3C2)=O)CCC(O)(CCNC(c2ccn(CCF)n2)=O)CC1 Nc1cc(C(=O)N)cc(Cl)n1.C12CC(C1)N(C(=O)C(c1ccc(Cl)nc1)(F)F)C2 N1(C(C(c2ccc(Cl)s2)C)=O)CCCCC(NC(c2nnc(C(C)(C)C)s2)=O)C1 Cc1nc(C(F)F)cc(=NCC2(O)CCCC(C)C2)[nH]1 c1(C(=O)NCC2(F)CCN(C(C(C)CC(C)(F)F)=O)C2)cnnc2ccccc12 Cc1ccc(C(N2CCC(F)(C(=O)NC3CS(=O)(=O)C3)CC2)=O)cc1F c1(C(N2Cc3c(-c4cn(COC)nc4)n[nH]c3C2)=O)c(C)cccc1[N+](=O)[O-] c1(NC(=O)NC(CCCC)C(=O)NC)nc(Br)ccc1C#N c1(C(=O)NC23CC(C(N4CC(CC)C4C(C)C)=O)(C2)C3)cnn(C)c1C C1(NC(c2nsnc2O)=O)CCN(C(c2cc([N+](=O)[O-])ccn2)=O)CCC1CO N1(C(C(CC)CC)=O)CCC2(CC1)CC2NC(=O)C(O)c1ccsc1 N1(C(C(CC)(C)CC)=O)CCCCC(C2CN(C(C3(C)C=CCC3)=O)C2)C1 N1(C(C(C(=O)OCC)OC)=O)CC2CC1CN2C(=O)CC=CC(C)(C)C CC1CC(CC(N2CCC(n3cnnn3)C2)=O)CN1C(C1COC(=O)N1C)=O C(=O)(N=S(C)(=O)C1CC(O)C1)c1c(C(n2cccc2)C)ccs1 C1(C)(CC)CC(C(N2CCCCC(NC(C3CSCC(=O)N3)=O)C2)=O)CCO1 C(=O)(C(C)C(C)(F)F)N1C2CC(NC(C3CN(C(CCC)C)C(=O)C3)=O)(C2)C1 CCC(CCC(=O)NCc1ccnc(C)n1)NC(c1nccnc1C)=O N1(C(C=COCC)=O)CCN(C(=O)Cc2n[nH]c(=NC)s2)C(c2cn[nH]c2)C1 c1(N(C(=O)C(C)Cn2ccc(C)n2)CC(=O)OCC)ccc(F)cc1 N1(C(N(c2cccc(C(N)=O)n2)CCC)=O)CCCN(CC(N)=O)CC1 c1(C(N(CC(COC)O)C)=O)c[nH]nc1CNC(=O)C.C(=O)C1CC1 CC(=O)CCCC(=O)N1CCN(C(c2cncc(C(F)F)c2)=O)C(C)C1 N1(C(C(C)NC(=O)NC2CCC2)=O)CCCN(C(c2cccn2CC)=O)CC1C CCCS(=O)(=O)C1CCCC1NC(c1ccccc1)C(C)O c1(C(=O)NCCN(C(=O)C)CC)ccc(N2CCCC2=O)cc1.C(C)C.O c1(CC)nc(=N)[nH]cc1C(N1CC(NC(=O)Cc2ccccc2C)CC1CO)=O C(=O)(C(C)CCOC)N(CCCNC(C(F)=CC)=O)Cc1ccccc1 C1(CCNC(c2n(C)ncc2)=O)CC(F)(F)CN1C(=O)CC(O)c1ccccc1 N1(C(c2n(C)ccc2)=O)CC2CCN(C(C3CC(CC(C)(C)C)C3)=O)CC2C1 Cc1cc(C)c(C(=O)N)c(C)n1.C1(CC)CCN(C(=O)CN(C)C(N)=O)CC1 N1(C(C=CC(C)(C)SC)=O)CCCCC(CNC(c2scnc2C)=O)CC1 C(CC(O)C(=O)NCC(C1CCCC1)NC(c1ccccc1)=O)SC.C(CF)O Cc1cc(=N)[nH]cc1C(=O)NCC1CCC1.c1(C(C=O)O)cc(F)cc(F)c1 c1(NC(=O)CC2CN(C(=O)C=Cc3ccc(Br)cc3)C2)ncc([N+](=O)[O-])cc1O C1(C(N2CCC(C(C)NC(c3c(C)nc(O)[nH]3)=O)C2)=O)C2C3CCC(C3)C12 CCC1=NOC(C(=O)NCC2(F)CCN(C(c3occc3COC)=O)C2)C1 NC(=O)CCCNC(C1(CNC(C2SCCS2)=O)CCC1)=O CCC(C)(C)CC(=O)NCC1CCC(N(C(=O)C(C)O)C)CC1.CCN(C)C N1(C(COCCC=C)=O)CCCN(C(C2(C)CCCO2)=O)CC1c1ccccc1 c1(-n2cc(C3(C)CN(C(=O)CC4CC5CC5C4)C3)nn2)ccc(S(C)(=O)=O)cc1 C1(C(=O)NC2C(C)(C)C2(C)C)CCCN(C(C2CCCNC2=O)=O)CC1 c1(C=O)cc(C2CC2)ccn1.C1(C(C)NC(C2(CC#C)CC2)=O)CCC1.N Cc1cc(C(N2CCN(C(c3cc(F)ccc3O)=O)C3CC23)=O)cc(C#N)c1 c1(CC(=O)NC(C)C)sc(C)cc1C.C1(C=O)CCN(CC(F)(F)F)C1.C N1(C(=O)NC2CCN(c3ccc(C(C)(C)C)cc3)CC2)CCc2cc(Br)sc2C1 C(=O)(C(CC(C)C)n1ccc(C2CC2)n1)N1C(C)(C(=O)OCC)C=CC1 C1(CCNC(C=CC=CCC)=O)C(C)CCCN1C(=O)CC.CC(C)C.O c1(C(N2C3CC(NC(C(CSC)C)=O)C2CC3)=O)coc2c1CCCC2 c1(OC)cccc(C(=O)N(CC(C)O)CCNC(C2CCC(=O)N2)=O)n1 c1(CC(=O)OC)ccc(F)c(C(F)(F)F)c1.C(c1ccccc1)=CCC(=O)N C#CC1(CNC(C2CCN(C(=O)CC3CCCC3O)CC2O)=O)CCOCC1 c1(C=O)cn(C)nc1Cl.c1(CC=O)csc(C)c1.C1(CC)CCCN1C(=O)C c1(C(N(C2CC2)CC2N(C(c3cc(C)no3)=O)CCC2)=O)c[nH]c(=O)cn1 Cc1cc(C(N2CC(C)(C(=O)NC3CCC(=O)NC3)C2)=O)cnn1 N1(C(C2(COC)CCC2)=O)CCN(C(c2c(C)cc(C)nc2C)=O)CC(C)(F)C1 c1(CCNC(C2C(C)CC2)=O)n[nH]cc1C(=O)NCC(=O)O.C1CC1.C [N-]=[N+]=NCCCCC(=O)NCC1(C(N2CCC=C(F)C2)=O)CC=CC1 Cc1cc(C(=O)NCC(C)(C)Cn2cc(-c3ncc(C(=O)O)o3)nn2)c(Br)cn1 O=C1CCC(C(N2CC(=C(F)C)C2)=O)CCO1.c1(C(=O)N)[nH]nnc1C(F)F C1(C(=O)NCc2[nH]nc(N3CCC(C)CC3)c2C)CC2(C1)CC(CN)C2 C(=O)(C1=C(C)CCC1)NCCCN(C(C1CN2CCC1CC2)=O)CC CC1CC(C(=O)NC2CC(CCNC(=O)CCCc3cccs3)C2)C(=O)O1 O=S(=O)(c1cc(F)c(Br)c(F)c1)NCCCCc1ccccc1 c1(CC)cc(NC(C2CCC(O)CN2C(c2cn(C3CC3)nn2)=O)=O)ccc1F N1(C(c2c(C(C)=O)ccs2)=O)CC2CC(C1)CN(C(=O)CCc1ncnn1C)C2 N1(C(CCOC(CC(C)C)C)=O)CCC(NC(C2CCCS2)=O)C12CCCC2 N1(C(CCCOCCC)=O)CCN2CCN(C(c3cnc(C)cc3C)=O)CC2C1 c1(C(=O)NCC2(NC(C(C)OC3CCCC3)=O)CCC2)ncnn1C c1(C(N2CCN(C(c3ccc(C)cn3)=O)C3C2C3)=O)n[nH]c2c1CSCC2 N1(C(C2C(C(=O)NCc3c(CC)onc3C)C2)=O)CCC(O)CC1C N(S(=O)(=O)N1CCC(C(C)(C)O)CC1)(CCC)CCC c1(C(=O)NC(CCSC)C(=O)NC2(c3cnn(C)c3)CC2)c[nH]c2cnccc12 N1(C(COCC=C)=O)CCCC(NC(C2(CCN(C)C)CC2)=O)CC1 C1(NC(CCc2n(C)ncc2)=O)C2CC1CN(C(=O)CC1CCOC1)C2 N1(C(C(C2CCCCC2)=O)=O)CCC(C(=O)NCCC(F)(F)Cl)C(O)C1 CC1C(NC(C2(C)CC(C#N)C2)=O)CCN1C(c1ccc(C(F)F)cn1)=O CCC(C(=O)N1CC2CN(C(=O)CC3CCOC(C)(C)C3)CC2C1)C(C)(C)CC N1(C(c2c(COC)cc[nH]2)=O)CCC2(C1)CN(C(C1CC=CC1)=O)CCO2 N1(C(Cc2c(C)nsc2)=O)C2CCCC1CN(C(C1(C)CCCS1)=O)CC2 Cc1ncn(C)c1C(N1CCC(C(C)NC(c2cc(C#N)cs2)=O)C1)=O S(=O)(=O)(C1CC1c1cccc(F)c1)NCCCNC(C)C N1(C(C2CC(C)(CC)C2)=O)CC2(CCN(C(=O)C(c3cncc(F)c3)C)CC2)C1 C=C=C(C)CC(=O)N(C1CN(C(c2cn(Cc3ccccc3)nn2)=O)CC1F)C C1(C)CC(F)(F)CN1C(=O)Cc1cnoc1.C(CCCC(=O)N)OCCC=C.C Cc1noc(CCC(N2CCC(CCNC(c3cncs3)=O)C2)=O)n1 c1(C(C)C)ccc(C(=O)NC2CC(=O)N(C3CN(C(=O)CCCF)C3)C2)c(O)n1 c1(OC)cccc2oc(C(N3C4CCC3C(NC(=O)C(N)=O)C4)=O)cc(=O)c12 c1(OCC(N2CC(NC(CCSC)=O)C2)=O)cncc(C)n1 c1(C(N(CCC(C)C)C(C2CC3CC3C2)C(=O)NC2COC2)C)ccccc1 C(=O)(C1=C(C)N(C)c2nnnn2C1)NC(CC=C)CNC(c1cc(C#N)c[nH]1)=O C1(CC)OCCC1C(=O)NCC#CC(=O)NC(C)Cn1cnnc1 c1(CC)nc(Cl)c(F)c(=NC2CCN(C(=O)CC(n3nc(C)cc3C)C)C2)[nH]1 C1=CCN(C)C(=O)COc2ccc1cc2OC.C(=O)(C(C)NC(=N)N)NC C=C(C)CCCC(=O)N1CCN(C(C2CCC(=O)N2CCC)=O)C(C(C)(C)C)C1 c1(CC)occ(C)c1C(N1CC2CC2(C)C1)=O.c1(C=O)n[nH]cc1C1CCC1 C1(C(N2CCC(n3ccnn3)C2)=O)(NC(COC(C)=O)=O)CCOC1 c1(CCC=O)ccc(O)cc1.C(=O)CC=C(C)C.C(C)C1CC1.CC=O.N C(=O)(C1CC(=O)Nc2ccccc21)N(CC(=O)NCCC)C C1(NC(c2nncc(OC)c2)=O)CC(C)CN(C(=O)CCc2cn[nH]c2)C1 C1(C(N(C2CCN(C(c3ccc(C#C)cn3)=O)CC2)C)=O)CCn2nccc2C1 C(C(=O)N1CC(NC(C2C(C)OCC2)=O)C(CO)C1)(C(C)C)SC.C(C)=O Cc1ncc(Cl)cc1C(=O)NCC1CCN(C(=O)Cc2cccs2)C(C)C1 c1(C(=O)NC2CC(NC(C3(C#N)CC4(CC4)C3)=O)C2)nc(O)nc(O)c1F CCC1=C(C(=O)NCCCCC(C)NC(=O)C(F)n2ccnc2)CCCO1 C#Cc1ccc(C(N2CCC(N(C)C(c3cc(S(N)(=O)=O)cs3)=O)C2)=O)cc1C c1(C=O)ccn2c1CSCC2.C(C)(CCNC(=O)C)OC.C(=O)CN(C)C c1(C(=O)NC(C)CNC(C2OCCC2C)=O)ccn2ncnc2c1 Nc1ccc(C(N2CCC2CNC(=O)CS)=O)nc1F.C1CCS(=O)(=O)C1 N1(C(C2CN(OC)C(=O)C2)=O)CCC(C(=O)NCC(C)(C)CC(C)C)C(C)(C)C1 C1(NC(c2cc(C)c(F)cc2)=O)CC2CCCC(C1)N2C(c1ccc(I)cc1)=O c1(C(=O)NC2CN(C(=O)NCc3ccc(C)cc3)CC2F)cccn(C)c1=O C1(NC(c2c(OC)cccc2)=O)CCC(O)CN(C(=O)CC(C)P(C)(C)=O)C1 c1(OCC#C)ccc(C(=O)NC23CC2CN(C(=O)CN2CCOCC2)C3)cc1 c1(CNC2CCC(NC(CSCC)=O)C2)cccc(-c2ccccn2)n1 C1(CNC(C(C)(O)C2CC2)=O)CCC(C(=O)NCCCN2CCCC2=O)CC1 N1(C(C2C(CC)CCN2C(c2cnccn2)=O)=O)CC2CC2C2CC12 c1(CNC(C(CC)C#N)=O)cc(C)ccc1F C1(NC(CNC(CC)=O)=O)CCCCC1CNC(C1(N=[N+]=[N-])CC1)=O C(=O)(C(CO)N(C)C)NCC(C)NC(=O)C(C)(C)C1CCC1 C(=O)(C1=NNC(C(F)(F)F)C1)NC12C(CN(C(CCCn3ncc(C)c3)=O)C1)C2 c1(C(=O)NC)ccc([N+](=O)[O-])s1.c1ncoc1C1CN(C(c2ccno2)=O)C1 N1(C(C(C(COC)C)C)=O)CC2CC(C1)N(C(C1CNc3ccnn3C1)=O)C2 c1(CNC(c2ccc(C)c(C#N)c2)=O)nc2ccccc2n1C(C)C Nc1ccc(C(N2CCCC(CNC(C3CCCO3)=O)C2)=O)c(Br)c1F c1(OC)cc2c(cc1F)CCC2NC(=O)C(=O)NCCC1COC(C)(C)O1 CCC(CC(C)O)Nc1ncc(OCC(F)F)cn1 O=C1CCC2(C(=O)NCC3CCCN3C(C3CC34CCOCC4)=O)CCCC2C1 c1(N(CCN(CC)CC)C)nc(=NCC2CCC(C(C)C)CC2)[nH]c2ccsc12 C1(NC(C2CCN(C(CC)=O)C2)=O)CN(C(=O)C#CC(=O)N(C)C)CCC1F CC(C)CC(CN=c1ncc(Cl)c[nH]1)NC(c1cnc2n(c1=O)CCS2)=O N1(C(c2n(CC)ccn2)=O)CC(NC(c2oc(C(=O)OC)cc2C)=O)CCC1C c1(CC)nc(C)ncc1C(=O)NC1CN(C(c2nn(C)c(Cl)c2Cl)=O)CCC1C CN1CCCC(F)(C(=O)NCC(F)CNC(c2cccc(F)c2Br)=O)C1 C1(CCCC)(C(=O)NC2CCC(CNC(c3cnc(Cl)s3)=O)C2)CCCC1 CC(C)CCC(=O)NCC(N1CCC(C(C)C(=O)NCC(C)(O)CO)C1)=O N1(C(C2(C#C)CN(C(C34CCCC3C4(F)F)=O)C2)=O)CCC(F)(C#N)C1 C(CCCCCNC(=O)CC1CC(n2cnnc2)C1)N(C)C(C1(CO)CCC1)=O CC1=CCC(C)(C(N2CCN(CCNC(C3CCC(=O)N3C)=O)CC2)=O)CC1 C(=O)(C(F)CNC(=O)C(=O)NCC(=O)N(c1ccccc1)C)OC Cc1nn(C)nc1C(=O)NCCN(C(=O)CCC1CCOCC1)C C1(NC(=O)CCC2CC2)CCC(NC(c2cncn2C2CC2)=O)CC1 c1(CC)c[nH]nc1C(=O)N(CCNC(=O)C(C)(C)C1CCCO1)CC c1(OC)cc(C(N2CCC(NC(=O)C=CC3CC3)C3CC23)=O)c2ccccc2n1 C1(c2n(CCCC(=O)OCC)nnn2)(NCC2(OC)CCC2)CCOCC1.C CCCCC(C)CCC(=O)N(C)CCNC(=O)C(F)(F)C(C)O C(C(C)(C)CN(C(c1ccnn1C)C(=O)NCc1cccs1)C)N(C)C N1(C(C2CCC(O)C2)=O)CCN(C(=O)CC2CCCCCC2)C(CF)C1 Cc1cc(N)cnc1C(=O)NC(CNC(C12CC=CC(C1)OC2)=O)C1CC1 C(=O)(CCC(=O)NN(C)C)NC(C(=O)NC(C#C)CCC)CC(C)C CCS(=O)(=O)C1CCN(c2ncnc(NC3CN(C(=O)OC)C3)c2C)CC1 C1(CC(=O)N(C(C)CNC(c2cnc(C(F)F)cn2)=O)C)Cc2ccccc2N1 C12(NC(c3ccc(F)c(F)c3F)=O)CCCC1N(C(c1ccc(Br)o1)=O)CC2 C1(C(N2C(CN(C(C3(C)CCC(C)C3)=O)C)CCC2)=O)CC2(C1)CC(O)C2 C1(C(C)C(N2CCC(c3nn[nH]n3)C2)=O)CCN(C(c2cc(Cl)cs2)=O)CC1 c1(CC)nc(C)ccc1NC(C1CC(NC(C2(C)CCCN2C)=O)CCO1)=O C1(NC(CCOCC)=O)C=CCC(C(=O)Nc2cccnc2C2CC2)C1 c1(C(C)=O)ccc(C(=O)NCCN(C)C(C2(SC(C)C)CCC2)=O)nn1 CN1CC=C(C(=O)N2CCC(CO)(CNC(c3cccc(Cl)c3N)=O)CC2)C1 C(C)(CCCC(=O)NC(c1cncs1)C)NC(C1(CC)COC1)=O c1(C(=O)NC(C(C)NC(C(C)(C)OCC)=O)C)c(C)nsc1Br C1(NC(CCC(N)=O)=O)CCC2CC1CN2C(=O)CC1(C#N)CCC1 C1(CNC(COC(C)C)=O)CCCC2CN(C(=O)CC3COCCOC3)CC12 C1(NC(C(n2cc(COC(=N)O)nn2)C)=O)CCN(c2ccccc2)C1C CC(C)CCC(C(=O)N1CCCC(F)(F)C1)NC(=O)CCCC1CCCO1 C1(CCC)(CO)CCN(C(c2ncnn2C)C(=O)NC(C)C(=O)OC)C1 C1CCOC1.C(=O)CC.n1(CC=O)cncn1.C1(C(C)C)CC1C(=O)NC c1(C(=O)NCC23C(CN(C(C(CCOC)C)=O)C2)C3)ccc2ncn(C)c2n1 Cc1nc(C)c(CCC(N2CC(NC(C3CC4CC4C3)=O)C3(CC3)C2)=O)c(O)n1 C1(C(N2CCCC(NC(C(CC#C)C)=O)C2)=O)C2COC(C)(C)OCC12 C1(NC(CCn2ccc(C)n2)=O)CN(C(C2CC2c2ccc(F)cc2)=O)CC1C S(=O)(=O)(c1ccc(NC(c2ccc3ncsc3c2)C)cc1Br)NCC(CC)OC C(=O)(CC1CN(C)c2ccccc21)NC1C2OCC(NC(C(CC)CC)=O)(C2)C1 C(CC(F)F)(C(=O)NC1CC(C)(C)C12CC2)N(C)C(c1csnn1)=O Cc1ccnc(C(=O)NCC2CCCC(NC(=O)CO)C2)n1.c1cc(C)on1 C1(CC(=O)NC)CCN(C(C2(NC(=O)CC3CCSC3)CSC2)=O)C1 C(=O)(CC(C)CCCCC)N1CC(CC=C)(NC(c2ncc(C#C)cc2C)=O)C1 c1(C(N(C2CCCN(C(CC(CC)SC)=O)C2)C)=O)cc(N)ccc1O N1(C(COCCCC)=O)CC2COCCC2(NC(c2cn3c(n2)SCC3)=O)C1 C1(CCNC(CCN(C(CCC)C)C)=O)CCCN1C(c1cnn(C(C)C)c1)=O C1(NC(=O)CCCn2ccnn2)C2CC1N(C(=O)Cc1nc(C3CC3)cs1)C2 C1CCCN1C(=O)C(=O)N(C)CC.C1(C(=O)N)CC(n2ccnn2)C1 N1(C(C)=O)CCN(CC(N2CCC(CN(C)C(c3n[nH]cc3Cl)=O)CC2)=O)CC1 N1(C(C2(F)CN(C(c3ccco3)=O)C2)=O)CC2OCCOC2C1 C(=O)(CCCCC(F)F)N1CCC(NC(CC2C(C)=NOC2=O)=O)C(F)C1 C(=O)(C(C)(C)C(F)(F)F)N1CC2CC(Nc3ccnc(C)n3)C2C1 Cc1cc(F)ncc1CNC(C1CC(NC(C2C(C)(C)C2(C)C)=O)C1)=O c1(C(=O)N)cc2c(nc1N)CCCC2.CC(C)C(C)(O)C(=O)NC1CC2(C1)CC2 CCC(C(=O)NC1(CC=CC=O)CCC1)NC(C)=O.C1(O)CN(C)C1.N c1(C(=O)NCC(N(C(CC(=C=C)C)=O)C)C2CC2)ccc(OC)c(N)c1 C1(CNC(C(CC)C)=O)(CNc2nccnc2N2CCCC2)CC12CCC2 C=C=C(C)CC(=O)NCC(CCCC)NC(c1ccccc1-c1ncn(C)n1)=O N1(C(C=O)=O)CC2(CCC(=O)NC2)C1.c1(OCC(=O)OC)ccccc1C c1(NC(C2C=CC(NC(c3cnc(C)nc3C)=O)C2)=O)cnn2cccnc12 N1(C(c2ccc(C(=O)OC)o2)=O)CCC(C2CC2)C1.C1(C(=O)N)CCCN1C=O CCC(CC)CC(F)C(=O)N1CCC2(C)CN(C(=O)CC3CC3C3CC3)CC12 c1(C(N(C2CC(NC(C(n3c(C)ncc3)C)=O)C2)C)=O)cc(Cl)c(Cl)s1 N1(CC(N2CC(C(C)NC(CCc3onc(C)n3)=O)C2)=O)CCC(C)CC1 c1(C(N2CC(CCCNC(CCC#C)=O)OCC2)=O)cc2c(F)c(Cl)ccc2[nH]1 c1(C(=O)NC2C(NC(C(C)(O)C3CCC3)=O)COC2)sc2ncccc2c1Cl CC1(C)CCOC(C(=O)NC(CC2CCC2)C(=O)NCCC(F)F)C1 N1(C(=O)CCCCN2CCOCC2)CC(CNC(C2CC(=C)C2)=O)C2(CC2)C1 Cc1cncc(C(=O)N(C)Cc2ccccc2I)c1Cl c1(C(=O)NCC2(O)C(C)(C)COC2)ccc2[nH]c(=N)sc2c1 CC1CN(C(=O)C(F)C2CCC2)CC1NC(c1ccnc(C2CC2)c1)=O C1(CC)(CC)CC(NC(C2C3CCCCC23)=O)CN1C(=O)CCC1CCC1 c1(C2N(C=O)CC(O)C2)ccc(F)c(F)c1.C12CCOC1c1ncnn12.C1CC1.N C(=O)(C(C)CCCC(C)C)NC1(C)C(C(=O)NCc2cc(OC)no2)CCCC1 C(CC(F)=C(F)F)NC(C(CC1CC1)NC(c1n(CC#C)cnn1)=O)=O N1(C(CCN(C(C(CC)C#N)=O)CCO)=O)CCC2(C1)CC2(F)F Cc1cc(CC(=O)N(C2CCN(C(=O)CCc3csc(=N)[nH]3)C2)C)ccc1CO c1(C(N2CC(N(C(C3CCN(CCC)CC3)=O)C)C(F)C2)=O)c[nH]cc(F)c1=O c1(C(C)NC(C2(CNC(=O)C=CC3CC3)CC2)=O)nc(O)n[nH]1 N1(C(C(C)OCCCCCC)=O)CCN(C(c2ccc(F)cn2)=O)CC1CCO c1(NCCC(C=C)(C)C)nccc(=NCc2cn3ccccc3n2)[nH]1 Cc1ccc(Cl)c(C(=O)NCC2CN(C(=O)C(O)P(C)(C)=O)CCO2)c1N N1(C(c2c(C)nns2)=O)CC(CO)C2(C1)CN(C(=O)C1=NOC(C)C1C)C2 C1(NC(C(CSCC)NC(=O)Cc2nccn2C)=O)CC(C2CC2)C1 N1(C(CCCOCC=C)=O)CCC2CCC(C1)N2C(c1ccco1)=O N1(C(C(CC)=CC)=O)C2CCC1CC(F)(CNC(=O)C(C)CO)C2 N1(C(C(CC(=O)OC)C)=O)C2CCC1CN(C(C13CCC(CC1(F)F)C3)=O)C2 c1(CC(=O)NC(C)C(CO)NC(C2(c3ccc(F)cn3)CC2)=O)cnccc1Cl C1(NC(c2c(C)nc(CC)o2)=O)C2CC1CN(C(=O)C1=CC(C)(C)C1)C2 Cc1ccnc(C)c1C(=O)NC1CCCC(C(=O)NCC(N)=O)CC1 C1(NC(C(c2cc(C)sc2)(C)C)=O)CCN(C(=O)C(=O)NC2CC2)CC1 N1(C(CCC(=O)NCC)=O)CCN(C(C2CCN(C)C(=O)C2)=O)C(COC)C1 CC1(CNC(=O)CCCC2CC2)CCN(C(c2cccc(CO)n2)=O)C1 C(=O)(CC(F)(F)Cl)N(CC(C)NC(c1ccccc1SC(F)F)=O)C N1(C(C2(C)C=CCC2)=O)CC2CC(NC(=O)C(O)Cc3ccccc3)CC(C2)C1 CCC(CC)CCC(=O)N1CC(F)CC1CNC(=O)C(c1cccc(OC)c1)=O C1(OC)COc2c(C(=O)NC3CN(C(c4c[nH]c(=N)s4)=O)CC3(C)C)cnn2C1 C=C(C)C(CC(=O)NCc1cn(CCc2c(Br)cc(Br)cc2Br)nn1)OCC c1(C(N2CC(CC)OCC2)=O)cc2c[nH]nc2s1.C(C(C)(C)C)N(CC(=O)N)C N1(C(C(C)OCCOC)=O)C(C(=O)N)C2CC(O)C1C2.C1CC1.C1CC1 CC1(C#CC(=O)NC2COCCC2NC(=O)C(C)(C)c2cscn2)COC1 c1(C(N2CC(CC(C)NC(C3CN(S(CC)(=O)=O)C3)=O)C2)=O)n[nH]cc1Cl C(CC(C)(C)CC(=O)N1CCCCC1CN(C(=O)C(O)C(F)F)C)OC C1(C(C)C)CCC(C)N(C(=O)NC2CCCC(C)N2)C1 C1(C(=O)NC2C(CC(N3CCCC(CCC)C3)=O)CCC2)Cc2nccn2C1 c1(CC(=O)NCC2N(C(C3C(C)CCCC3)=O)CC2)c[nH]c2cccc(F)c12 N1(C(C(C)N(C(=O)C)CCc2cccnc2)=O)CC2(CC(C)CO2)C1.CC.O c1(C(=O)NC2C(C)CN(C(C3(C(=O)N(C)C)CC3)=O)C2)ccc2oncc2c1 CC1CN(C(c2cnc(S)n2-c2ccccc2)=O)CCN1C(C12CCCC1C2)=O N1(C(c2cccs2)=O)CC2(C(=O)NCCC3CCCCCC3)CC1CCO2 c1(CC)cc(=NC2CN(C(=O)CN3CCC3)CCC2C(F)(F)F)[nH]c(CC)n1 C1(CNC(C(C)CC2CCCC2)=O)CC(C(=O)NC)=NO1.c1ccnc(F)c1 C1(NC(c2cc(F)cc(F)c2)=O)CC2CC(NC(C3(CF)CCC3)=O)CC2C1 N1(C(CNS(NC)(=O)=O)=O)CCC2(C1)CN(C(c1n[nH]c3c1CCC3)=O)CCO2 N1(C(C2(C=C)CC2)=O)CCCC(N(C(C2CCCC(C(N)=O)C2)=O)CC)C1 c1(OC)ccc2[nH]c(CNC3CCC4(C3)CC4C(=O)NC(C)C)cc2n1 N1(C(C(CC=C)NC(C)=O)=O)CCCC(F)C1.c1(C(=O)N)nccc(C(F)F)n1 Cc1cnc(C(N2CCC(CCNC(=O)C(C)(C)c3cscc3Cl)C2)=O)cc1C N1(C(CC2CCC(C)CC2)=O)CCC2(CC2)CC1C(=O)NCC(C)(C)F C(=O)(CCCC(F)(F)F)N1CCCC(C)(CNC(c2c(SC)ccs2)=O)C1 C(=O)(C1=CCCCO1)NC(CSC)(C)C(=O)N(C(C)CN(C)C)C CC(C)CCC(=O)C(=O)N1CCC(C)(C)C(C(N2CC(N=[N+]=[N-])C2)=O)C1 c1(OC)cc(C(N2CCC(C(C)NC(C3CC(=O)N3)=O)C2)=O)c(F)cc1N CCCCCCC(C)NC(=O)CC(O)CNC(C1C2CC(=O)CC12)=O C12(C(=O)NC3(C)CCN(C(c4c(SC)csc4)=O)C3)CCCC1C2(F)F C1(O)(C(C)C)CCN(C(c2ccc(C#N)s2)C(=O)NC(C)(C)C)C1 N1(C(C)=O)CCCC1C(=O)N.c1cc(C(C)(C)C)c[nH]1.C1(C=O)CC1.CC C1(C=O)CN(CP(C)(C)=O)C1.C(C(C)C(F)(F)F)NC(COC(C)C)=O.N C1(NCC2CC(CC(CC)OCC)C2)CC2(C1)CC(C(=O)O)C2 N12C(CCC13CCC3)CC1(O)CCN(CC1)CC2=O.c1(CO)ccccc1F c1(C(N2CCC(N(C(=O)Cc3cnsc3)CC)C2)=O)ccc2cnoc2c1 Cc1cnc(C(N2CCCC(OC(C)C)C2)C(=O)NCC2CCCO2)cn1 CC1CN(C(=O)CC2C=CS(=O)(=O)C2)CCN1C(=O)CCc1ccc(F)cc1 c1(C(=O)NC2(CC=C)CCN(C(=O)C(F)=CCCF)C2)ccc2nnc(O)n2c1 C1(OC(=O)CCc2ccc(F)cc2)CCCCN(C(C2CCCCO2)=O)C1=O CC1(C)CN(Cc2ccc3[nH]ccc3c2)CCC1NC(=O)CCC1CCOCC1 C(=O)(C(C)(C)CCC(=O)NC(C)C)OC.c1(C=O)ccc(-n2cnnc2)cc1.N c1(C(N2CCC(C(C)NC(C3COCCO3)=O)C2)=O)ccnc(-n2ccnc2)c1 CCCS(=O)(=O)N(C1CCN(C(c2nc(CN3CCCC3)cs2)=O)C1)C c1(C(N2C(CC)CCC2)=O)cnn(C(C)(C)C)c1Cl.n1(CC)ncnc1C=O.N CC(C)C(O)C(C)(C)C(=O)NCC(O)C(=O)NC(C1CSC1)C Cc1ccc2cccc(NC(c3nc(C(=O)NCCCCCO)cs3)=O)c2n1 N1(C(c2ccc(C(C)C)cc2)=O)CCC2(CC2)C1.C(c1cn(C)cn1)=CC=O.N C1(C2(C(=O)OC(C)(C)C)CCC2)(OC(=O)NCCCOC)CCC1.O CCC(CCC(=O)N1CC(NC(=O)CN2CC=CC2)C2(CC2)C1)OC C1(NC(c2n(C)ncc2)=O)CCC2(CCN(C(=O)C(C)(O)C3CC3)CC2)C1 C1(NC(C(CC)O)=O)CCC(F)(CNC(c2ccc(OCCO)cc2)=O)C1 c1(CC)ccc(C)c(NC(=O)C(F)CC2CN(C(=O)CN3CCNC3=O)C2)c1 CCC(CC)C(F)C(=O)NCC1COCCN1C(=O)C(O)CC(F)(F)F N1(C(CC2C(C)=NOC2=O)=O)CCCC2(CCN(C(c3ncc(F)cn3)=O)C2)C1 CCC(CC(=O)NCCCCCn1cc(C(C(C)C)N(C)C)nn1)SC C1(C2(NC(=O)C3=CCN(C(=O)CC4CCOC4(C)C)C3)CC2)(OC)CCC1 c1(NC(c2scc(-c3ccc(N4CCN(C)CC4)cc3)n2)=O)nc(Cl)ccc1O c1(OC)ccc2nccc(C(=O)NC3CN(C(C4CCOCC4)=O)CC3F)c2c1 C1(C(=O)N(C)OC)(COC)C=CCN1C(=O)CC1CCCN(C)C1 C12(C(=O)NCCCCCOC)CC(CO1)N(C(=O)CCCCc1ccccc1)C2 c1(OC)ccc(CN2CCC(C#N)C2)c([N+](=O)[O-])c1.c1(C(=O)N)ccnc(Cl)c1 c1(C(=O)NCCOC2C(C)CCCC2)nn(C)cc1S(N)(=O)=O N1(C(c2ccn(CC)n2)=O)CC2CCCCC2(NC(=O)CCc2cccs2)C1 c1(NC(C2C(CNC(c3c(C)scn3)=O)CCC2)=O)ccc(O)c(Cl)c1 C(C)(CCCCO)NC(C(C1(O)CCCCC1)NC(CCSCCC)=O)=O c1(C(=O)NCC(C)NC(C2N(CC)CC2)=O)cn(C)nc1-c1cccs1 Cn1c(-c2ccccc2)nc2c1CCN(C(c1cc3ccccc3oc1=O)=O)C2 N1(C(C(C2CCCC2)OCC)=O)CCC2(CC2)C1.N(S(=O)(=O)NC)CC=O c1(OC)nc(C(=O)O)ccc1-c1cn(C(C)C(=O)N2CCCC2)nn1 N1(Cc2c(C)cccc2)Cc2[nH]nc(C3=CCS(=O)(=O)CC3)c2C1 S(=O)(=O)(c1ccc(F)cc1)NC1C(F)CCN(C(C2CC2F)=O)C1 C=C1CCN(C(C2CC3CC(=O)C2C3)=O)C(C(=O)NC(C)CC(N)=O)C1 N1(C(CC(=O)N(C)C)=O)CCOCC1CNC(=O)Cc1ncsc1Cl C(=O)(C(C)(C)CC)NC(C=CC(=O)NCCc1cn(CC)nc1)C c1(NC(C#C)=O)ccc(NC(=O)OC(C)(C)C)cc1O C(=O)(C1=CCOCC1)NCCC1CCC(NC(CCN2CCN(CC)CC2)=O)C1 c1(C(c2n(C)c(N3CC(CC#N)C(O)C3)nn2)O)ccc(Cl)c(Cl)c1 CCCC(F)(F)C(=O)NCCn1cc(-c2cc(C)cnc2C(=O)OC)nn1 c1(OC)nc(C)nc(Cl)c1NC(C1CCCCC1NC(c1nccs1)=O)=O N1(C(CCCCCC)=O)CCCC2CCN(C(=O)C=Cc3cccn3C)CC12 c1(C(C)=O)ccc(C(=O)N(C2CN(C(=O)Cn3nc(C)cc3C)CC2F)C)cc1 CCC(F)(C(=O)OC)C(=O)OCc1cc(F)cc(Br)c1 n1(CC)cc(C(=O)NCCCO)c(C(F)(F)F)n1.c1(C(=O)N)ccnc(C)n1 CC(C)(CCl)C(=O)N1CCN(c2ccc(-c3cccc(I)c3)cc2)CC1 N1(C(C2(CN(C)C)CC2)=O)CCCC1CNC(=O)CC1CC(CF)C1 c1(SCC)cc(C(=O)NCC2CCN(C(=O)C)CC2)ccn1.c1cscn1.S CP(C)(=O)C(O)C(=O)N1CCN(C(=O)Cc2ccccc2Cl)C(c2cn[nH]c2)C1 C1(NC(C2CC2c2cccc(-c3ccc(CO)s3)c2)=O)CCS(=O)(=O)C1 c1(C(C)C)cc(N2CCC(c3ncc(-c4ccccc4F)[nH]3)C2)n2ncnc2n1 c1(C(=O)OC)ccc(F)cc1NC(C)(CCCO)c1nnnn1C1CCCC1 Cc1nccc2c(NC(=O)CCCCCCBr)cccc12 C1(C(N(CCN=[N+]=[N-])CC)=O)CC12CC(NC(=O)C=C(C)COC)C2 Cc1cc(C(N2CCC(N(C(=O)CN3CC(=O)NC3=O)C)C2)=O)cc(O)n1 c1(N(C)C)ccccc1NC(=O)C(F)CC1CN(C(=O)C(F)(F)C2CC2)C1 C(=O)(C#CC1CCCOC1)NC1(C)CCC(NC(=O)C=C2CCSCC2)CC1 C(C(CC(C)C)C(=O)N(C1CCCCC1(C)O)C)NC(CCOCCOCC)=O c1(CNC(C2(C)CCCN2C(=O)CC2COC(=O)C2)=O)ccc(F)cc1F CCCC(C(=O)N1CCCC1CCC)NC(c1cccc(=O)o1)=O C#CC1(C(=O)NCCCc2ncn(C)n2)CN(C(=O)C(C)Cn2ccnc2)C1 N1(C(CC2(C=C)CC2)=O)CCC2CN(C(c3n[nH]c4ccccc34)=O)CCC2C1 C1(CC)CCN(C(C2CCC2C#N)=O)C(C(=O)NC23CC2COC3(C)C)C1 N1(C(COCC)=O)CCOCC1CCNC(C1(CC(C)C)CC1)=O C(=O)(CC1=CCCCC1)N(CC(C)(C)NC(C12COCC1C2)=O)C C(=O)(CS(=O)CC)NC(CC)CC1CC1.c1(C(=O)NCC)cncnc1 c1(OC)ccnc(-c2cn(CC3CCN(C(=O)Cc4cc[nH]n4)C3)nn2)c1 c1(OC)ccc(C(=O)Nc2ccccc2CN(CC(F)(F)F)CCO)cc1 C(=O)(C(F)CC(C)(C)C)NC(CCC)CNC(C1(C(F)F)CCCC1)=O C1(O)(C(N2CC(C)(NC(C3C(C(=O)OCC)C3)=O)C2)=O)CCOCC1 CC(CO)(CS(C)(=O)=O)NCC(N1CCSC1)=O C1(C(N2CCC(CCNC(c3n[nH]c(=N)[nH]3)=O)CC2)=O)CCC(C2CC2)CC1 c1(OC)ccccc1-c1ccc(NS(=O)(=O)CCc2ccc(F)cc2)s1 C12(CC(=O)N)CC3CC(CC(C3)C1)C2.CC(C)CCCC(=O)NC(CC)C(C)C C1(C(=O)NCCCCNC(C2(C)CNC(=O)C2)=O)CCCC12CCOCC2 c1(C(=O)N)cnccc1N(C)C.C1(C(N(CC(C)O)CC)=O)CCC(F)CC1 N1(C(=O)NC(CC)CC(F)(F)F)CCn2[nH]c(=N)cc2C1 C1(CNC(C2CC3(CCC3)C2)=O)CCCN(CCc2ccccc2)C1 C1(C(=O)OC)CN(c2nc(C3CC3)no2)CC1(F)F c1(N2CC(C)SC2)ccn2ncc(S(=O)(=O)N(CCCCN(C)C)C)c2n1 C1(O)(C(C)C)CCN(C(=O)C=CC(F)(F)F)C1.c1(C=O)ccco1.N(C)C C1(C(=O)NC(CC)CN(C(=O)CN2CC3CC3C2)C)Cc2nccn2C1 n1(CC)nnnc1C(c1cnn(CCSC)c1)NCCC(O)COC N1(C(C2CCN(C(C)=O)C2)=O)CCCC(NC(c2n[nH]cc2C2CCC2)=O)C1 C(N=c1[nH]c(=NCc2cccc(Br)c2)[nH]c2c1CSC2)c1cnc(COC)[nH]1 c1nccnc1C(=O)NC1CCN(C(=O)C)C1.CCCN(C)C.C1CC1.CC c1(CC)onc(C(=O)N(C2CCCN(C(=O)CC3CC(=O)C3)C2)C)c1C O=C1CC(C(=O)NC2CC3C=CC2C3)N(C(=O)C(O)Cn2cncn2)C1 C1(C(=O)NC(c2ccoc2)C)CN(C(c2cccc(=O)o2)=O)CC1(F)F CC(C)C(F)C(=O)NCC1(C)CCN(C(c2cc(Cl)cnn2)=O)C1 c1(C(=O)NC23CC(NC(c4nn(C)c(O)c4)=O)(C2)C3)cc2n(n1)CCCC2 C1(NC(C(=O)NC2CC2)=O)C2CN(C(=O)C(F)(F)c3ncc[nH]3)CC12 N1(C(C2C(CC)CN(C(c3ccc(C)cc3F)=O)C2)=O)CCCN2CCCC2C1 c1(NC(C(=O)NCC2CC(C)(C)OC2)=O)ccccc1S(=O)(=O)C1CC1 C1(N(C(c2cc(F)c[nH]2)=O)CC)CCN(C(c2ccon2)=O)CC1.N(C)(C)C C1(NC(C(CC=C)OC)=O)CCC2(CC1)CC(NC(=O)C1=CCOCC1)C2 N1(C(CC2C(C)(C)OCC2)=O)CCC2CCN(C(c3ccnn3C3CC3)=O)CC12 C(=O)(C(CC(C)(C)C)NC(=O)C(C)C(F)F)N1CCCN(CCC)CC1 c1(C(=O)NC2CCN(c3nc(SC)nc(C)c3)CC2C)cnc2c(cnn2C)c1 Cc1ccnc(Cl)c1C(N1CCC(CNC(c2c(C)ncn2C)=O)C1)=O c1(C(=O)NCC(C)CC2CC2)ccc(CNC(=O)Cc2cncnc2)s1 N1(C(C(C)=CC)=O)CCC(NC(C23CC(C(C)(C)C)(C2)C3)=O)C1C C=CC(C)(C)CC(=O)NC1CN(C(c2ncccc2OC)=O)CC1n1cccn1 C12(NC(CSCCC(C)C)=O)CCCC1(F)CN(C(=O)CCc1cn(C)nn1)C2 c1(NCC#Cc2c(N)cccc2)[nH]c(=NC2CC=CC2)nc2scnc12 C(=O)(CC(O)(C(F)(F)F)c1nc2ccccc2s1)N(C)CC1COC(C)(C)O1 CCCCCC(O)C(=O)N1CCOCCC1C(=O)Nc1ccccc1O CC(=O)CCCC(=O)NC1CC(NC(c2cc(C)ccc2O)=O)C1 C1(C(=O)NC2CC(NC(C(CC)(C)OC)=O)C2)CC(C(C)(C)C)=NO1 N1(C(CNC=O)=O)CC=C(C(=O)NSC(F)F)C1 c1(CC)cccc(C(=O)NCCCCC(=O)NCCCCC(=O)OC)c1 C#CCCCCC(=O)N(C1CC(C(=O)NCC(C)(O)C2(C)CC2)C1)C C1(COC)COCCN1C(C1CN(C(=O)CCCn2cccc2)CC1C)=O N1(C(C(C)(C)OCC)=O)CCCC(NC(=O)CSc2cn[nH]c2)CC1 c1(NC(C2N(C(C3(COC)CC3)=O)CSC2)=O)cnc2ccc(Br)cc2c1 N1(C(CC(CNC(c2c(CC)nn[nH]2)=O)C2CCC2)=O)CC2(CCCC2)C1 C1(CC(=O)N(CC(=O)N(C(c2ccco2)C)C)C2CC2)CCCCC1C c1(C(=O)NCC(CCC)NC(=O)Cc2cccnc2C)ccc2cc[nH]c2c1 c1(CC2(C(=O)NCCCC)CC2)ccccc1F.n1(CC(=O)N)cnccc1=O CCCCC(C(=O)NCC1(CO)CCN(C(C2(CO)COC2)=O)CC1)C(C)C C(C1C(C(=O)NC2(C)CCC2)C1(C)C)=C(C)C.c1(C=O)cc(C#N)on1.N Cc1ccc(CCC(=O)NC2CC(CNC(C34CC(F)(C3)C4)=O)C2)cc1 N1(C(Cc2cc(C)no2)=O)CCCCC12CN(C(C1CN(S(C)(=O)=O)C1)=O)C2 N#Cc1csc(-c2ccccc2-c2ccccc2CCO)c1 Cc1cc(C(=O)N(CC(=O)NCC2C3CCCC23)C)cn1C C1(C(N2CCC(CCNC(c3scc(Cl)c3Cl)=O)C2)=O)CC12CCCC2 CC1(C)CC(C(=O)NCC)CCO1.c1(CC=O)cc(C(F)(F)F)cc(F)c1.N C1(CC=C)(C(=O)NCC(C2(O)CCCC2)O)CCCC1 C12(NC(c3n(CCC)nc(C)c3)=O)CCCCC1N(C(c1c[nH]cc1C)=O)CC2 CC1CN(C(C2C3CCC(=O)C23)=O)CCC1NC(c1cc(C2CC2)[nH]n1)=O c1(C(NCCNC(C2CCCC(F)C2)=O)=O)ccc2c(c1)COCC2.C1CC1 C(CC(C)C)(CS(=O)(=O)Nc1ccc(CN2CCN(C)CC2)cc1)OC c1(NC(C2CCN(Cc3ccncc3Cl)CC2O)=O)cc(F)c(F)c(F)c1 Cc1cc(CCC(=O)N(C)CC=CC(N2CC(CC(N)=O)C2)=O)no1 C1CC2CC(C1)N(C(=O)CS(N)(=O)=O)C2.Cn1cc(C=O)c(C(C)(F)F)n1.N N1(C(C(F)=CCC)=O)CCCC(CN(C(=O)COC(C)(C)C)C)C1 N1(CC(COC(COC)C)O)CCCC(N(C)C(c2cnc(C(C)C)s2)=O)CC1 C=CCC(C)(C)C(=O)NCC(O)CNC(c1cnc(OC)s1)=O N1(C(c2cnnc(O)c2)=O)CCCC2(CC(NC(C3(F)CCC3)=O)CO2)C1 C#CCCCS(=O)(=O)NCc1ccc(C(C)CC)cc1 c1(C(=O)NCCN(C(=O)CC(C)c2cccnc2)CCC)cnc(Cl)s1 c1(C(N2CC(O)(CNC(C(CC(N)=O)O)=O)C2)=O)cc2ccc(Br)cc2o1 N1(C(C=C(CCC)C)=O)CCCC(C2(NC(c3c(Br)cnn3C)=O)CC2)C1 Cc1cc([N+](=O)[O-])c(C)cc1NC(c1ccc(-n2cccn2)c(F)c1)=O c1(-n2c(CSc3cc(Cl)ccc3Cl)nc(C3C(C)C3)n2)ccc2ccccc2n1 N1(CC(=O)NC2CCCC23CCN(C(=O)CO)C3)CCOc2ccc(Cl)cc21 C(N=c1[nH]c(=NCC2CCN2C(C)(C)C)[nH]c2cccc(F)c12)C1C(C)(C)C1 C(=O)(CC(C(F)F)NC(=O)C(N1CCNC1=O)C)NC(C)Cc1cn[nH]c1 c1(CC)cc(N)ccc1C(N1CCCC(C2CCCCN2C(=O)C(O)CF)C1)=O CC1(C)CCN(C(=O)C(C)(C)C(C)(C)C)CC1C(N1CC2CC1CC2CF)=O N1(C(C2(C)CCC(=O)N2)=O)CC(CNC(c2ccnc(Cl)c2O)=O)C2(CC2)C1 c1(CC)cc(C(N2CC3CC2C3C(=O)Nc2ccc(I)cc2C)=O)cc(C)n1 c1(C(=O)NCC(CO)NC(c2c(C)nc(CC(C)C)o2)=O)cnc2ccccn12 Cc1ccc(C(=O)NC2(C)CC(NC(=O)C(C)N(C)C)C2)c(O)c1C C1(C(=O)NCCCN(C(C2(C(C)C)CC2)=O)CC)CC2CCC2C1 c1(CC(C)C)nnc2c(C(=O)N)cccn12.C1(C(N(CCC)C)=O)CCC1(C)C c1(CC)ccc(C(=O)NC2(CNC(=O)C(c3cnccn3)C)CC2)cc1F c1(C(=O)N)cc(F)cc(S(N)(=O)=O)c1.c1(C(=O)NC(C)CC)ccc(O)cn1 C1(CNC(=O)COC2CCC2)C2CC2CN1C(=O)CCCN1CCCC1 c1(C(=O)NC2CCN(C(c3c(C(C)C)nn(C)c3)=O)C2)ccc(F)c2ccsc12 N1(C(CSCC#C)=O)CCC(F)C(NC(=O)C=CC2CCCO2)C1 c1(C(N2CCC(C(=O)NCCC3C(=O)OCC3)OCC2)=O)cc2ccccc2[nH]1 C1(C(N(CCCCNC(C2CCCN2C2CC2)=O)C)=O)CCc2nnn(C)c2C1 C1CCOC(C2CCN(C(=O)CC(C)(C)O)CC2)C1.C(=O)(COCC=O)NC.N N1(C(C2(CCOCC)CCC2)=O)CC(C2CCCCN(C(=O)CCS(C)=O)C2)C1 c1(C(=O)NCC(CCNC(Cc2cc(C)nn2C)=O)O)c(C)cc(C)nc1S N1(C(c2cccc(CCC)c2)=O)CCCCC(N(C)C(c2ccc(O)nn2)=O)C1 c1(-n2cc(C3N(C(C4CC5CCC5C4)=O)CCCC3)nn2)ccc(Br)cc1F C1(C(NCCCN(CC)CC)=O)CCN1C(C)=O.C1(C=O)COC1.C CC(C)C(C#N)C(=O)NCC1(F)CC(NC(=O)CCCN=[N+]=[N-])C1 C1(CNC(CC=C)=O)C(C2CC2)CCN1C(c1cccn2nncc12)=O N1(C(c2cc(Cl)ncn2)=O)CCN(C(=O)C2=CCCC2)C2(CC2)C1 N1(C(Cn2c(N)cc(C)n2)=O)CC2(C1)CN(C(=O)C(F)(F)CC1CC1)C2 C1(CC(N2CCN(C(C(=O)N3CCC3)=O)CC2)=O)CC(F)(F)C1(F)F c1(C(=O)OC)cc2c(cc1OC)CN(C(=O)CCC1CCN(C)CC1)CC2 N1(CCCCCNC(C2(CCC=C)CC2)=O)CCN(C(C23CC(C)C2C3)=O)CC1 CC1CCC(C(N2CCC(CCNC(c3ccnn3C(C)(C)C)=O)CC2)=O)CC1 C1(C(N2C(C)C(C=O)CC2)=O)C2CC3C(C2=O)C13.c1cncn1C.C(=O)(C)N CC(CC(C)NC(c1ccnn1C1CC1(F)F)=O)N=c1[nH]nc(CO)s1 CCC(CC)CC(=O)NCC1CCOC1C(N1CCOCCC1C)=O CCCCN=C(NCCN1CCOC(C)C1)NCC(C)CC1CCOCC1 c1(OCCNC(=O)NC2(O)COC2)cccc(O)c1 N#CC1CC(F)(F)CN1C(=O)COC1CCCCC1 N1(CC2CCCN(C(c3ccc(F)cc3)C(N)=O)C2)CCc2ccccc21 C(=O)(C(CC)(CC)CCCCCC)N1CC2(CN(C(CCCOCC=C)=O)C2)C1 N1(C(C(C)NC(CC)=O)=O)C2CCC1C(C)CC2.c1(C=O)cnn(C(F)F)c1.N C1(C(=O)N)CN(C(=O)C(C)(C)C2(O)CCC2)CC(C)(C)C1.CCC(C)C(C)CO C(=O)(C(C)(C1CC1)N(C)C(c1csc(CO)n1)=O)NC1(CCC)CC1 N1(C(C(C)SCCCC)=O)C2CCCC1CN(C(c1cscc1C(=O)OC)=O)C2 C1(N(C(c2cc(C)sc2)C(=O)NC(C)C)C)CCC(C)(C)C1 N1(C(c2scc(Cl)c2Cl)C(=O)NC2COC2)C2CCCC1CC(F)(F)C2 N1(C(C=C(C)C(=O)O)=O)CCCC2(CCCN2C(c2ccc(Cl)cn2)=O)CC1 N1(C(CSCCN(C)C)=O)CCN(C(c2cc(C3CC3)nn2C)=O)C2CC12 c1(CCNC(C2CCC(CNC(=O)CC3CCC4CC34)C2)=O)ccccc1O C1(NC(c2ncccc2Cl)=O)CC2CN(C(c3ccn4ccnc4c3)=O)CC2C1 c1(C(=O)N)cc(C)c(C#N)cn1.C(C)(C(=O)NCC1CCC1)OCC=C C12(NC(c3c(Cl)cn(C)n3)=O)CCC(CC1)N(C(C1CC1C1CCCC1)=O)C2 Cc1cn2cc(C(=O)NC3CCCN(C(=O)C(F)C4CCC4)C3)sc2n1 C1(SC)CC(CC(=O)NCC2CC2CNC(=O)C=CC2CC2)C1 C(CCC(=O)N(CC(Cc1ccccc1)NC(=O)Cn1cccn1)C)OC(C)C C(CCCCC1CC1)NC(C(C)NC(C=C(COC)C)=O)=O N1(C(c2c(C)nc(C)s2)=O)CC(NC(=O)CC2(C)CC2(Cl)Cl)CC(C)C1 N1(C(C(CCOC)C)=O)CC(NC(=O)C=Cc2c(F)cccc2F)CCC(O)C1 C1(NC(c2c(COC)noc2)=O)CCN(C(c2ccc(NC=O)cc2)=O)CC1O c1(CC)cc2c(N3CC(NC(c4ccoc4C(C)C)=O)CC3C)ncnc2s1 C1(C)(C(=O)Nc2c(SC)cccc2)CCCN(C(c2n[nH]c(Br)n2)=O)C1 O=C(C1=CCC2(COC2)OC1)N1CC2CCCCCC2(C#N)C1 CC(C)C(C)C(CNC(c1cnc(O)n1C)=O)NC(=O)CCc1cnc[nH]1 c1(CC)cncc(C(N2CCC(OCCNC(=O)CCC3CCCN3C)C2)=O)c1 C(CN=C(NCCc1ccccc1Br)NCC1CCCCO1)=CC CC(C)C(C(=O)N1CCOC(CS(C)(=O)=O)C1)c1cn(C)nn1 C(C(C)(C)CNC(=O)NCCc1cscn1)N(C)C c1(C(=O)NC2CCCC(N(C(c3cc(C)ncn3)=O)C)C2)ccc(C)c(F)c1 C(=O)(CC(C(C)C)NC(=O)CC(C)C1CC1)N(C)Cc1onc(CC)n1 N1(C(CC)=O)CC2CS(=O)(=O)CC2(CNC(c2ccncc2NC)=O)C1 C1(NC(C2(CSC)CC2)=O)CCC(C)N(C(=O)CCc2ccc(F)cc2)C1 C1(C(N2CCC(CN(C)CC)C2)=O)CC=CCN1C(c1cnnc(C)c1)=O C1(C(=O)NC2CC3(CC(NC(C4N(C)CCC4)=O)C3)C2)CCOC2(CCC2)C1 c1(C(=O)NC2(C)CCN(C(C3(CCCC)CC3)=O)CC2)ccc2nccnc2n1 C1(CNC(C(C)(C)N(C)C)=O)CN(C(c2cnc(=N)[nH]c2)=O)CC1O C(=O)(CC(C(F)(F)F)NC(C1(C)CC1(C)C)=O)N1CCCN(C(C)C)CC1 CCCCC(O)C(=O)N(CC(C)N(C)C(C)=O)C.c1(C(=O)N)cnc(C2CC2)o1 Cc1nc(O)nc(O)c1CCC(=O)NCC1CCN1C(=O)C(=O)C1CCCC1 Cc1cc2ccc(C(N3CC4CN(S(=O)(=O)c5ccccc5F)C4C3)=O)cc2[nH]1 CCCCN=C(NCCC1COCCO1)NCc1ccncc1 N1(C(C=C(C)C)=O)CC2(CCC2)CC1C(=O)NCC1CC2CCC2C1 N1(CCC2CC(OC)C2)CC(=O)N(CC23CCC(CC2)C3)C1=O Cc1cc(F)c(C(=O)NCCCC(C)NC(c2[nH]nc([N+](=O)[O-])c2Cl)=O)c(F)c1 C(=O)(C#CC(C)(C)C)NCCC(C)NC(C(n1c(C)nnn1)c1ccccc1)=O N1(C(=O)CCOC2CCOC2)CCN(C2CCN(C(=O)Cn3cccn3)C2)CC1 C1(C#CC(=O)NC2COCCN(C(c3csc4nnsc34)=O)C2)(CC)COC1 Cc1cccc2[nH]cc(C(=O)NC3CN(C(c4ncncc4Cl)=O)CCC3C)c12 C(=O)(C(C)(C)C(C)(F)F)N1CCCC1.Cc1cccc(C(=O)N)c1C(F)(F)F C12(CC(=O)NCCC(C)OC)CCC(CC1)C2.C1(C)(C=O)CNC(=O)N1 C1(C(=O)NC(c2cccnc2F)C)CCN(C(=O)C(O)C(F)(F)F)CC1O N1(c2cc(OCC)nc(C)n2)CCC(C)C(NC(C)=O)C1C C1(CNC(COC(CC)C)=O)C=CCN1C(=O)CCSCC(N)=O Cc1nnc(O)c(C(=O)NC2CC(NC(=O)CC(O)CC(C)C)C2)c1C c1(C(=O)NC2(CCNC(C3N(C)CCOC3)=O)CC2)cc(O)cc(Br)c1 c1(C(N2CCC(C)CC2CNC(=O)Cc2ccno2)=O)ccc2c(c1)CCC2 C1(NC(CC2(CC)CCOCC2)=O)CCN(C(=O)CC(C)(C)O)C12CC2 c1(C(C)C)nc(-c2c[nH]cc2Br)n(C(c2ccncc2)C)n1 Cc1conc1CC(=O)NCCC(=O)N(C)C.C12(CCCC1)C(=O)N2 C#Cc1cnc(C(=O)NC2CC(C(N(C)C[Si](C)(C)C)=O)C23CCC3)c(C)c1 N1(C(C2(C)COCC2(F)F)=O)CCC(C2CN(C(=O)Cc3ccccc3)C2)CC1 N1(C(C(CCCC)O)=O)CCC2(CC1)CC(NC(=O)C(=O)N(C)C)CCO2 c1(C(N(CCCF)C)=O)ccc2c(n1)CN(C(=O)C(C#N)C(C)(C)C)CC2 c1(C(N2CC(O)(CC)C2)=O)cc(-n2cccn2)ccn1.C1(SC)CC(C=O)C1.N CC(CCCCNC(=O)C(CN(C)C)CC1CCCC1)NC(c1cccs1)=O C1(NC(c2c(C)con2)=O)CCCC12CN(C(=O)CC(c1c(C)n[nH]c1C)C)C2 Cc1cnc(C(=O)NCCCC(C)NC(=O)CCOc2cccc(F)c2)c(F)c1 Cc1noc(CCC(=O)NCCNC(=O)C(F)(F)c2cscc2Br)n1 c1(C(=O)NC2CCN(C(C(C)C34CC(C3)C4)=O)CC2)ccc(=N)[nH]c1Cl C1(CC(=O)NCC2C=CC(NC(C(COC)C)=O)C2)CCCCCC1 C1(CN(C(=O)COc2ccsc2)CC)CCCCN1C(C1CCCO1)=O c1(OC)ncc(Cl)cc1C(=O)NCC(c1ccccc1)N(C)C(=O)C1CC1 C1(NC(C=C(C)C2CC2)=O)CN(C(=O)CC2CC3(CCC3)CO2)CC2(CC2)C1 C1(CNC(COC(CC)C)=O)C(C(=O)NC2(C(N)=O)CC2)C1(C)C C12(NC(c3ccc(SC)o3)=O)CCCN(C(c3ccc(C(F)F)nc3)=O)CC1C2 N1(C(Cc2ncc(C)o2)=O)CCN(C(=O)C(C)(C)C2CC2)CC1c1ccncc1 CC1CCCC(C(=O)COC(c2c(Cl)nsc2Cl)=O)C1 c1(C(=O)NCCN(C(CC(CC)C2CCC2)=O)C)c(Cl)cncc1Br C1(CC=C)(C(=O)NCC2(F)CN(C(=O)CCc3ccc[nH]3)C2)CCCCC1 c1(C(=O)NC2C3CC2CN(C(c2cn(C(F)F)cn2)=O)C3)cccc2nccn12 c1(CCC(=O)NC2CC(NC(C(C)=C3CCC3)=O)C2)nc(O)c2ccccc2n1 C#Cc1cccc(C(=O)NC(CC(=O)NCc2ncccc2F)C(F)(F)F)c1C C1(C(=O)NC2C3CN(C(=O)COC)CC23)CCC(C2CC2)C1.C1CCOC1 C(=O)(CCCNC(C)=O)N(CCCNC(=O)CC1CCC(C)C1)CCC N1CCOCC1.C1(C=O)CSC1.C1(C)C(=O)N(C2CC2)C(C)C(=O)N1C.C Cn1cccc(C(=O)NCc2cccc(C(=O)NCC3CCC=CO3)n2)c1=O CC1(NC(=O)CCCN2CCCCC2)CC(NC(C2CCCCC2)=O)C1 N1(C(C2N(C(C)C)CCCC2)=O)CCOCC(NC(c2c(F)cccc2Cl)=O)C1 Cc1cc(C2(C=O)CC2)cc(C)c1.c1(CC=O)ccn(C)n1.C1(CC)CC1.N C1(NC(C(CC)(CC)OC)=O)CC2CCC1CN2C(C1CCC2(CC2)C1)=O c1(-n2cc(C3(C(=O)OC)CN(C(=O)C=O)C3)nn2)cccc(Br)c1F.C1CC1.N CCC(CC(=O)NCC(O)CNC(c1csc(Cc2ccccc2)c1)=O)C(F)F CCC(C)(C(=O)NCC1(C(=O)NCCC2CCCOC2)CC1)OC C#CCC(CC#C)C(=O)NC1(C2CC2)CCN(C(=O)CSS(C)(=O)=O)C1 O=C1CCc2nc(NCC3CN(C(=O)CC(F)(F)C(F)(F)F)CCO3)ccc21 C=C=CCCC(=O)NC(C1CCCCC1)C(C)NC(C1(CO)CCCC1)=O c1(NC(CC(C)NC(=O)C=C2CCC2)C)ncnc(Cl)c1C(C)(C)C c1(CC)cncc(C(=O)NC(C)CC(C)NC(c2cnc(C=O)cn2)=O)c1.O n1(CC)nc(C(=O)NC2CC3(C2)CC3C(=O)N)c(C)n1.C1CNC(=O)C1 C=CCC(C)(C)C(=O)NC1CCC1NC(c1nccc(Cl)c1C)=O c1(CC(=O)N(CCCNC(C(C)Cn2cccn2)=O)C)ccc2nn(C)cc2c1 c1(C(=O)NC(C(=O)OCC)Cc2cccnc2Cl)ccc(C)nc1O C1(C(=O)NCC2(F)CCN(C(C(c3c(C)nn(C)c3)C)=O)C2)CCCCCCC1 C1(C(=O)NC2C3CN(C(CNC(=O)OCC=C)=O)C2C3)CCCCCCC1 N1(C(C=C(COC)C)=O)CCC(NC(c2cccc(O)c2Cl)=O)C2(CCC2)C1 C(=O)(C(CC(C)C)C(C)C)NCCCN(C(c1ncc(OC)nc1)=O)CCO O=S(=O)(c1c[nH]ccc1=NCC1COC(CCN)C1)NCCCCCCO.c1ccccc1 C1C2CCC1N(C(=O)CCn1ccnc1)C2.C1(N(CC=O)C)CCS(=O)(=O)C1.N c1(OC)ncnc(NCC2CCN(C(=O)C=Cc3cnc(C)s3)C2)c1OC C1(C(=O)NCCCCSC)COCCC1NC(c1c(C)nsc1C)=O C1(N(C(=O)CC(C)(C)C2CC2)C)CCCC(NC(=O)CC(C)(C)C)C1 C1(C(=O)NCC(C(=O)N2CCCC2CN(C)C)OC)CCCC(=O)N1C CC1(CNC(=O)C(O)C2CC2)CC(F)(F)CN1C(=O)C(C#N)=CC1CC1 c1(C(N(CC(CNC(C(CC)CC(C)C)=O)C)C)=O)cc2ccc(C)cn2c1 c1(CN2CC(C(=O)NC(c3cccc(C#N)c3)C)OCC2)cc(Br)c(F)cc1O N1(C(C=C(CC)C)=O)CC2CCC(C1)N2C(=O)CS(=O)(=O)NC1CC1 CC(CC(=O)NCC1CCN1C(c1nc2cc(F)ccc2s1)=O)CC(C)(C)C c1(C(=O)NCCNC(C2(Cl)CC2(F)F)=O)c(F)c(F)cc(F)c1F c1(C(C)C)cnc(Cl)c(NC(=O)C(N2CCCC(Cc3nccn3C)C2)=O)c1 c1(C(=O)NCCNC(COCC#C)=O)cc(C)nc2cc(F)ccc12 c1(NCCOCCOC)cc(=NCC2CC(C)C2)[nH]c(C(F)(F)F)n1.O O(NC(=O)C(Cn1cncn1)NC(C1C=CCS1)=O)CCCC O(NC(=O)C(Cc1ccccc1Br)NC(=O)CCOC(C)=O)C(C=C)C N1(C(C)C)CCC(C(N2CCC(CNC(=O)CC3CC34CC4)CC2)=O)CC1 C1(CC=C)(NC(c2scnc2Cl)=O)CCCN(C(C2(CCF)CCC2)=O)C1 c1(C=O)cc(S(C)(=O)=O)co1.c1cnn(C)c1.CC(C)CN(C(=O)C)C.N CC(C)(C)C(=O)C(=O)N1CCN(C(=O)C)C(c2cn[nH]c2)C1.C(=O)(C1CC1)N c1(C(N2CC(OC)(CNC(=O)Cc3ccno3)C2)=O)noc2ccc(Cl)cc12 c1(C(N2C(CC(=O)NCC3(OCC)CCOC3)CCC2)=O)ccc(N)cn1 n1(CC)ncc(C)c1CN1CCCC(NS(=O)(=O)C2CC2)C1 c1(C(=O)NC2(C)CC(C(=O)NC3CCCC(O)C3)C2)cc(F)ccc1F Cn1ncc(C#N)c1C(N1CCN(CC2CCN(C(C3CC3Cl)=O)CC2)CC1)=O C1(NC(=O)CC2CCC(F)(F)C2)CC2(CCN(C(=O)Cc3ccccc3Cl)C2)C1 S(=O)(=O)(c1ccc2[nH]c(=NCCCNC(C)=O)sc2c1)NC1CCN(OC)CC1 N1(C(C=C(COC)C)=O)CCC(CNC(C2SCCS2)=O)C12CCC2 c1(OC)ccnc(O)c1C(=O)NC1CCN(C(=O)CCc2cncn2C)CC1C C1(C2CN(C(C3(C#N)CC34CCC4)=O)C2)(NC(c2cnc(N(C)C)o2)=O)CC1 C1(COCC)CCCN(Cn2nc(CC)n(C)c2=S)C1 C1(OC)CCn2cc(C(N3CCC(C4(O)CC4)CC3)=O)nc2C1 C1(NC(c2ncoc2CNC(C2(CO)COC2)=O)=O)CC12CC(O)C2 N#Cc1ccc(CCC(=O)NCC(=O)NC2CCC(O)CC2)c(Br)c1 C(c1cccnc1)=CC(N1CCC(C(C)C)C1)=O.C1(C(C)=O)C(C=O)C1(C)C C1(NC(CC=CC=C)=O)C2CC(O)C1N(C(=O)C(CC)CC=C)C2 CC1(C)CCN(C(=O)CCOC2CC2)CC1C(=O)NC1CCCC(F)C1 CCN=C(NCCC(F)F)N1CCn2c(nn(CC(F)F)c2=O)C1 N1(C(c2coc(C3CC3)n2)=O)CCC2(CCCN2C(c2ccn(C3CC3)n2)=O)C1 N1(C(C(C(C)C)OC)=O)CC2CCCC(C1)N2CC(=O)Nc1ccc(Cl)cc1 C1(C#N)(CNC(CCOCCN(C(=O)C(C2CCCCC2)F)C)=O)CCC1 n1(CCOC)nnnc1C(c1ccc(Cl)s1)NC(c1scnc1C)C N1(C(CCC=CC)=O)CCC(C2CCN(C(c3nccn4c(C)nnc34)=O)C2)C1 N1(C(C2N(c3ncc(CC)cn3)C(C)CC2)=O)CCCN(C(C)C)CC1 Cc1nc(C(=O)NC2CN(C(=O)Cc3csc(Cl)c3)CC2C)c(C)o1 c1(C(=O)NC2C(NC(CCC(C)SC)=O)C2)ncc(Br)cc1O N1(C(C(C)OCC=C)=O)CC(OC)C(C(=O)N(C)Cc2nc(CC)no2)C1 c1(OC)ccc(C(=O)NC2CC2CNC(=O)CCCCCF)c(Cl)n1 C1(CCC)CN(C(c2ccn(C3CC3)c2C)=O)CCN1C(=O)Cc1ccoc1 C#CC1(OCC(N2CC(NC(=O)C(C)c3cncs3)C2)=O)COC1 C1(C=O)CC2CC1CN(C(=O)Cc1cnn(C)c1)C2.C1(C(=O)O)CC1C.CC C1(CSC)CCCN1C(=O)Cn1cc(CNC(=O)Cn2nnnc2C)nn1 C1(NC(CN(C)CC)=O)CN(C(C2CCC(C)(C)C2)=O)C2(CCCC2)C1 CC1(C)C(C)CCN1C(=O)C(F)CC1CC1.c1(C(=O)N)coc(C2CC2)n1 c1(N(CC(C)CNC(=O)CCS(C)(=O)=O)C)ccc([N+](=O)[O-])c2cccnc12 C=C(C)C(C)(C)C(=O)N(C)CCN(C)C(C12CC1COC2(C)C)=O C=CC1(CC(=O)NCC2(N3CCCC3)CCCCC2)CCCCC1 c1(C(N(CCC)C)=O)ncoc1C1CCC1.C1(C=O)CCN(CC(F)(F)F)C1.N C(CC(C)(C)CNC(c1cnc[nH]1)=O)NC(c1ccc(OC)s1)=O c1(C(=O)NCCCN2CCN(Cc3n(C)ccc3)CC2)cc2n(n1)CCCO2 N1(C(CC(CCSC)O)=O)CC(C)(CNC(c2c(CO)noc2C)=O)CC1(C)C c1(N2CC(C(C)NC(C3CCc4cncn4C3)=O)C2)nc(=N)[nH]c(Cl)c1[N+](=O)[O-] C#CCCCC(=O)N(C1CCC1NC(c1cc(-c2ccccc2)nn1C)=O)CC c1(C(C)=O)cc(Br)ccc1NC(C1(C)CCCN1Cc1csc(Br)c1)=O c1(C(=O)NC(C)CN(C)C(c2ccc(C(O)CF)cc2)=O)cc(N)ccc1Cl N1(C(C(CC)OC)=O)CCC2(CCCCC2NC(c2nnc3n2CCCC3)=O)C1 C1(CC)CN(C(c2cn(CC)nc2C)=O)CCN1C(=O)C(C)OCCN(C)C C1(C=O)CCCC2(CC2)C1.C1(OCC)(C)CN(C(C2CCC2(F)F)=O)C1.N C12(CCCCC1)C(=O)NC2.C1C=CC(NC(C2(OC)CC(C)C2)=O)C1.O C(=O)(C1CCc2cccnc21)NC(COC)CNC(c1nsnc1O)=O C(=O)(C1CCc2c[nH]nc21)NC(CCOC)C(=O)NCc1ccc(SC)o1 N1(CC)C(C)CN(C(=O)C(CCSC)NC(=O)C(n2ccnc2C)C)CC1C Nc1c(F)c(F)cc(C(=O)NCC2CC2)c1Cl.C1(C(=O)N)CC12CC2(F)F C(CC(C(=O)N(C)Cc1nnc(O)o1)NC(C1CC1COC)=O)=CC C(=O)(CCCOCCO)N(C)CCC1CCCN1C.C1(C=O)CCC2(CC2)C1.N CC(C)CC(C)(CNC(c1cc(=N)[nH]cc1Br)=O)NC(C1CC1C)=O C#Cc1ccc(C2CC2)cc1.C(=O)(C(F)CC1CCOC1)NCC(CNC)O.C CC(C)CC(F)C(=O)NC.C1CC2(CC2)CN1C(c1cc(C(F)(F)F)cs1)=O C1(C(=O)NCC2(C=C)CCCCC2)CC12CCC(N=[N+]=[N-])CC2 C=C(CNC(C1(C)CCCN1C(=O)CSC(C)(C)C)=O)C1CCOCC1 c1(NC(C2CC(=C)CN2C(=O)CN(C)C(C)C)=O)ccc(OC)c(Cl)c1.O Cc1nc(CC(C)C)sc1C(=O)NCC1CN(C(c2cnc(Cl)[nH]2)=O)C2CC12 N1(C(c2c(C)oc(Br)c2)=O)CCCCC1C1(C(F)(F)F)N=N1 N1(C(c2cnn(C)n2)=O)CCC(F)(F)C(CNC(C2(C3CC3)CCOCC2)=O)C1 N1(C(=O)OC(C)CN(C)C(=O)OC(C)(C)C)CCN(C)C(=O)C1(C)C c1(C(C(=O)NCCOCC2CC2)N(C(C=C)C)C)ncc(C)o1 C1(S(C)(=O)=O)(C(=O)N)CCCCC1.N1(C(C2(OC)CCC2)=O)CCC(C)C1 c1(C(N2C(CNC(CCCCC=CC)=O)C=CC2)=O)cc(S(=O)(=O)N)c[nH]1 c1(CC(=O)NCC2(C)CCN(C(C(C(CC)C)=O)=O)CC2)csc2nc(C)cn12 N1(C(C2(CC#C)CC2)=O)CC2C=CC1C(C(=O)NCCCCCN(C)C)C2 C(=O)(C1=CCCCCC1)NC(C)CNC(C1(O)CCOC1)=O C1(C(=O)NC(C)C(=O)NC23CC2COC3(C)C)CC2(CC2)CN1C C1(C(C)C)N(C(=O)CC2CC(=O)NC(=O)C2)CC12CCN(C(=O)C1CC1)CC2 C1(Nc2ccnc(SC)n2)CCc2[nH]nc(C(F)(F)F)c2C1 N1(C(CC(CNC(C(C)(C)C2CCOC2)=O)C2CCC2)=O)CCOC(C#N)C1 C1(NC(C(CNC(Cc2ccn(C)c2)=O)CC2CC2)=O)CC2OC(=O)CC12 C#Cc1ccnc(C(=O)NCc2csc(CNC(C3(O)CCC3)=O)n2)c1 N1(C(C(C)Oc2cccc(Cl)c2)=O)CC2(CCN(CC3CCCC3)CC2)CC1C N1(C(C2(C)CCCS2)=O)CCC(NC(c2cc(CCO)on2)=O)CC(O)C1 N1(C(C(C(C)NC(=O)C(C)(C)N=[N+]=[N-])C)=O)CCOC2(CCCC2)C1 C1(NC(c2c(CC)nc[nH]2)=O)C=CCN(C(C2(O)CC(c3ccccc3)C2)=O)C1 CC1CCCC(NC(c2nc(C(=O)Nc3nccnc3Br)cs2)=O)C1 CC(C(=O)NC1C2CCC(C2)C1C(N1CC2CCC=CC12)=O)S(C)(=O)=O c1(C(N2CCN(C(c3c(C)coc3)=O)C3C2CC3)=O)ccc(Cl)c2cccnc12 C12(C(=O)NC3(CC#C)CCC3)CC(C)(CN1C(c1sccc1OC)=O)C2 c1(NC2CCC(NCc3c(C)cccc3O)C2)ncnc2c(C)csc12 C1(C(N(CCCC)CC(N)=O)=O)CC1C1CN(C(c2cc(Cl)no2)=O)C1 C(C)(c1ccccc1Cl)=CC(=O)NC(C1N(C(C(COC)OC)=O)CCC1)C c1(N(CCOCC=C)C)cc(NCc2cc(C)cc(F)c2)nc(COC)n1 Cc1nc(C(N2CCOCC2C(=O)N(C)C)C(=O)Nc2ccc(F)cc2)oc1C c1(NC2C(C)CC=CC2)cc(=NCc2cc(Br)ccc2OC(F)F)[nH]c(CO)n1 Cc1nc(C=O)c(C)n1CC.C(=O)(CC(C1CC1)C1CC1)N(C1CCC1)C [N-]=[N+]=NCCCOCC(=O)NCC1(NC(=O)C(F)C2CCC2)CC1 CC(N=[N+]=[N-])C(=O)OC1CC2CC2C1 C=Cc1cc(C(=O)NC(C)(C)C(C)NC(=O)Cc2cccnc2Br)cc(F)c1 c1(CNC(c2cn(C)c(=O)cc2)=O)n[nH]c2c1CN(C(C1C=CCCC1)=O)CC2 c1(CC=O)cc(C2CC2)on1.C1(CC)CCCN1C(c1ccc(C2CC2)s1)=O CCCC(C(=O)NC(CCSC)C(=O)NCc1ccc(Cl)cn1)N(C)C c1(-c2ccc(CN(CCCOC)C=O)o2)ccc(F)cc1C CCCCCC(C)(CC)C(=O)N(CC(C)N(C)C(c1cnc(O)n(C)c1=O)=O)C c1(C(N2CC(C)CC2)=O)nn(C)c(Cl)c1Cl.CC(C)C(C(=O)NC)c1cccnc1 c1(C(=O)NCC(C)N(CC(=O)Nc2ccccc2)C)cc2ccccc2[nH]1 CC1(C2CC2)CN(C(C2COC(C(F)(F)F)CN2)=O)C1 Cc1nc2ccc(NC(=O)CN(C)Cc3ccc(Br)s3)cc2[nH]1 c1(C(N(CC(CNC(C(CC)NC(N)=O)=O)C)C)=O)cc(F)ccc1OC C1(C(=O)NC(CCC)C2CC2)(NC(C2CC=CCC2C)=O)CC(F)(F)C1 c1(NC(C(N2CCC(CC)CC2)c2sc(C)nc2C)=O)cccc([N+](=O)[O-])c1 C1(C(=O)NCCc2ccnc(O)c2)CCN(C(=O)C(c2ccccc2)F)C12CC2 N1(C(C(CC=CCC)C)=O)CC2(C1)CN(C(=O)C(C(C)(C)C)N(C)C)C2 CCCCC(CNC(=O)C(C)OC(C)(C)C)NC(c1cc(C)sn1)=O c1(C(=O)NCC2CN(C(c3c(SCC)nccn3)=O)C(C)C2)cc2occc2s1 C(=O)(CS(=O)c1ccc(Cl)cc1)N1C(CNC(=O)C(O)c2ccsc2)CC1 N1(C(c2c(F)ccc(N)c2)=O)CCN(C(c2cncs2)=O)C2COCC12 S(=O)(=O)(c1ccc2c(c1)CCC(C(F)F)O2)NC(c1ccc(Cl)cc1)CCOC c1(C(N(C(C)C)CC)=O)csc(C#N)c1.C(=O)(C(C)CSC(F)(F)F)N CC1CN(C(=O)CCOCCNC(C2CC2C(N)=O)=O)CCCO1 CC1CC(NC(C2CCOCC2)=O)CN1C(=O)CCNC(C1CCCCCC1)=O Cc1cnoc1COC(=O)C1CC1(c1ccccc1)CC C=C(C)CC(C(=O)N1CCC(CN(C(=O)C(C)(F)F)CC)CC1)OC Cn1c(C(=O)NCCC2(C)CCOC2)cc2c(Br)cccc12 C1(CC)CC2CCC(C1)N2C(C1CCCN(C(C2(CF)CC2)=O)CC1)=O c1(CC)nn(C)c(Cl)c1C(=O)Nc1ccccc1C(N)=O C1(F)(CNC(C(c2ccccc2)SC)=O)CCCN(C(c2csc(C)c2C)=O)C1 C1(c2nnnn2CC2CCOCC2)(NC(C)C)CCC(C)SC1 C1(C(N2C(CNC(c3cc(C4CCOCC4)no3)=O)CC2)=O)CCCS1(=O)=O c1(CCC(=O)NC2CCCN(C(C(C=CC)O)=O)C2)nnc(S)nc1O c1(C(N2CCC(C(F)(F)F)C2)=O)ccc2c(c1)CCO2.C(CC(=O)N)=CC.C C12(NC(=O)CCc3cc(F)cc(F)c3)CCN(C(c3cc(O)cs3)=O)CCC1C2 C1(C(=O)NC2(CC(=O)NC(CCSC)C)CC2)CN(C)CCO1 CC1OCCCC1C(=O)NC1(CO)CN(C(c2ccnc(-c3cc[nH]n3)c2)=O)C1 C1(NC(CCCCSC)=O)CC2(C1)CN(C(=O)C(C)Cc1cccc(F)c1)C2 C1(NC(CC(C)(C)C)=O)CCC(C)(C)CC1CNC(=O)CC.C1CCCO1.O C1(NC(c2c(CCC)nns2)=O)CCC12CN(C(=O)C=Cc1cccn1C)C2 c1(CNC(C2CC(OC)C2)=O)ccc(C)cc1F.C1(CC(=O)N)CCC1C Cc1cc(C(N2CCC(C(C)C(=O)Nc3cccc(O)c3)CC2)=O)nnc1C c1(OCC=C)ccc(C(=O)NCC2CCCC2)cc1.C(=O)C(F)(F)C=C.N c1(CC)ccccc1OCC(=O)NC(CNC(c1occc1C)=O)(CC)CC C#CCCC(C(=O)Nc1cnn(CC(C)C)c1)NC(C1CCOC1CC)=O c1(CC)c(C(N2CC(C(N)=O)C2)=O)csc1C.C1(CC=O)CC2C=CC1C2.C C1(O)(C(C)NC(COC(CC)(C)C)=O)CCN(C(c2cnc(C)s2)=O)C1.O C1(NC(c2c(CC)nco2)=O)CC(F)CN(C(=O)C2=NOC(C)C2)C1 c1(C(=O)NCCC2CC(NC(=O)C(F)C3CCCC3)C2)sccc1F c1(C(N(C2CCCN(C(=O)CC3CCCCO3)C2)CC)=O)cn(C)nc1Br c1(C(N2CC(NC(c3cc(C(C)=O)on3)=O)C(C)C2)=O)cc(N(C)C)nc(Cl)c1 C=C1CN2C(=O)CCC2(C(N2CCC3(CC2)CC3)=O)C1.c1(C(=O)N)cc(Cl)c[nH]1 C1(COC)CCCN1C(=O)CC1CCCC1(F)F.C(=O)CCN(C)C(C)=O C1(NC(C)=O)C2CN(C(C3CC3C(C)NC(=O)C(C)NC=O)=O)CC12 C(=O)(C(C)(C)CC)NC(CNC(c1n(CCOC)ncc1)=O)C1CCC1 C1(NC(C2(COC)CC2)=O)CCN(C(=O)C(c2ccc(F)cc2C)C)C(C)C1 C(=O)(CCCCCCCCCO)NCC1(NC(C=COCC)=O)CCOCC1 C(=O)(C1CCCc2cn(C(C)C)nc21)NC1(C)CCN(C(COCC=C)=O)C1 c1(NC(CC(C)NC(c2cccc(Cl)c2)=O)C)ncc([N+](=O)[O-])cc1Cl C(=O)(C(CC(C)C)C(N)=O)NC(CC)CCC(=O)N(CCC(C)(C)O)C CC1CN(C(c2ncn(-c3ccccc3)n2)=O)CC(C)CN1C(=O)CC1CSC1 C1(C(=O)NCCCCC)(C(F)F)CCCCC1.N1(CCC(=O)N)C(=O)CCC1=O C(C1c2ccccc2CCN1C(c1cc[nH]c1)=O)NC(=O)C1=CC2CCCC12 N1(C(C)=O)CCC(O)CC1C(=O)NC(c1snnc1C)C N1(C(C(c2ccc(C)s2)C)=O)CCC=C(CNC(=O)CCC2CC(F)(F)C2)C1 C1(NC(C2(C)CC2)=O)CCC(CNC(C2CC(n3ccnc3)C2)=O)C1 C12(NC(CC3CC(SC)C3)=O)COCCC1CN(C(=O)C(C)(C)N1CCCC1)C2 C#CC1(O)CC(C(=O)NC(C2CCN(C(=O)CCc3nccs3)CC2)C)C1 N1(C(CSc2n(C)ccn2)=O)CC(CNC(=O)CC2CCOC2)CC12CCC2 CC(CCCO)NC(=O)C(C)(C1CC1)N(C)C(c1ccco1)=O N1(C(COC)=O)CCN2CCOCC2(CNC(C2(c3ccc(Cl)cc3)CC2)=O)C1 N1(C(CCCn2cc(CC(OC)OC)nn2)=O)CCC2(CCN(C)CC2)C1 c1ccccc1.CC1CCC1CC(=O)NCCC(C)NC(C1CC(OCC)C1)=O C1(C(=O)NCC2(OC)CN(C(C3(c4cc[nH]n4)CC3)=O)C2)COCCN1C ON=C1CN(Cc2cn(CC3CC3)nn2)CC2(CC2)N1 c1(CC(N2CCCC2)=O)ccccc1OC(F)(F)F.C1(C(C)C)CC1C(=O)N C(=O)(CC(C)C(C)(C)NC(c1cc(CC)no1)=O)N1CC(CC#C)OCC1 C(=O)(CCCCCCS(N)(=O)=O)NCC(CNC(C1C(C)N(C)CC1)=O)O c1(CC(=O)NCC(CC)NC(c2cc(-c3ccccn3)c[nH]2)=O)cc(CO)on1 N1(C(c2c(C)cc(C)s2)=O)CCC2(CC(NC(=O)C(C)N3CCC3)C2)C1 C#Cc1ccnc(C(=O)NC(c2cn(C)nn2)C(=O)NCCOC)c1.C1CC1 c1(CN(C(c2ocnc2C)=O)CC)c(OC)cc(OC)cc1OC C1(F)(CNC(C(CC=C)(F)F)=O)CC2CCC(C1)N2C(=O)Cn1cnnc1O C1(N(C(CN(C)C(c2ccco2)=O)=O)C)CCN(C(=O)C=C(Cl)Cl)CC12CC2 Cc1ccc2snc(C(N3CC(N(C)C(c4cc(O)ncn4)=O)C3)=O)c2c1 C1(=CC=O)CC2CCC(C1)N2C.CCC(C(=O)NCC=CC)n1ccnc1.N C1(N(CCCOCC2CCC2)C)CCNCC1.C(C)(C)C.CCN(C)C=O c1(C(=O)NC(CC)(C)CCNC(=O)CC2C=CCCC2)cc(C)cc(F)c1 S(=O)(=O)(c1ncccc1OC)Nc1ccc(SCC)c(C)c1 C1(NC(COC(C)C)=O)CN(C(=O)C(N2CCP(C)(=O)CC2)C)CC1N=[N+]=[N-] C1(NC(C2(CC)CN(C(c3ccc(CC)cc3)=O)C2)=O)CC(C)(C)OC1(C)C c1cnn2c1CC(C)CC2.C(=O)(CC(CC)C(C)C)N1C(C(=O)OC)SCC1CO c1(C(N2CCC(N(C(C3C(C(=O)OC)CCC3)=O)C)C2)=O)ccc(CO)nc1 C12(NC(CCCC)=O)CCCC1N(CC(=O)NCC(N1CCC(C)CC1)=O)CC2 c1(C(N2CC3C(C(N4CC(C)CC(C)C4)=O)C3C2)=O)cccc2ccoc12 CC1(C)OCCC1(O)C(=O)NCC1CC(O)CN1C(C1CNC(=O)C1)=O C1(C)(C(=O)NC2C(OC)C(O)C2)CC(O)CN1C(=O)CC(=O)N(C)C c1ccc([N+](=O)[O-])cc1.c1(CC(=O)NC(C)C(C)NC(=O)C)cn(C)nc1Cl c1(C(N2C(CNC(c3c(C)con3)=O)CCCC2)=O)cc2cccc(Cl)c2o1 S(=O)(=O)(c1ccccc1F)NCCC(N1C(CNC(CSC)=O)C=CC1)=O C=CC(C)(C)C(=O)NCC(C)NC(C1CC(=O)N(CCN(C)C)C1)=O c1(C=O)cc(S(N)(=O)=O)c(Cl)o1.Cc1cnncc1C(=O)NC1CCCCC1.N c1(C(N(C2CCN(C(=O)CC3CC(CF)C3)C2)C)=O)cccc2c1NC(=O)CC2 c1(C(=O)NC(C)C(C)(C)NC(C2CC2(C)C)=O)ccn2c1CCCC2 n1(CCOC(C)C)nc(C(C2CC3CCC2C3)C)nc1-c1cnsn1 c1(OCCOC)ccc(N)c(CNC(c2cccc(-n3cncn3)n2)=O)c1 CC(CC(=O)NCC(c1ccccc1)N(C)C(c1cn(C)c(=O)cn1)=O)C(F)F c1(C(=O)NC2CCCC(Nc3ncc(Cl)cn3)C2)cnc2[nH]nnc2c1 c1(C(=O)NC2C(NC(C(C)c3cc[nH]n3)=O)CCC2)ccc(OCC(F)F)cc1 C1(CC(=O)N(CCCC)CCCC)CN(C(C2(CSC)COC2)=O)CC1C c1(OC)ccc(NC(C2CC(F)(F)CN2C(=O)CCN2CCOCC2)=O)cc1Br C1(NC(C2N(C(CC=C)=O)CCC2CC)=O)CC2(CCCCC2)C1 C(=O)(C1=CC2(CN(C(=O)CC3CCC(C#N)C3)C2)OC1)N.Cc1cc(CC)n[nH]1 C1(F)(CNC(=O)CN2CCC(F)CC2)CCCN(C(C2CC2F)=O)CC1 O=C1OC(CC(=O)N(C2CCCNC2)Cc2cnn3ncccc23)c2ccccc21 C1(CNC(=O)Cn2cnnn2)CN(C(c2cn(C3CCOC3)cn2)=O)CC1(F)F CC(C)S(=O)(=NC(=O)C12CC(CN)(C1)OC21CCC1)C1CCNC1 c1(C(=O)NCC2(C)CCCN(C(C3(C)CCC(=O)N3)=O)C2)ncc(C#N)cc1Cl c1(C(=O)N)ccc(C(F)F)cc1.C(CCCC)NC(C(C)NC(=O)NC)=O CS(=O)(=O)c1cnn2c1CN(C(=O)NCC1CCC3C(CC1)C3(F)F)CC2 CCC(C(=O)N1CC=CC(C(=O)NCCCOC(=N)O)C1)C(C)C C1(NC(C(C=C)O)=O)CCCC2CN(c3cc(C(=O)OCC)nc(C)n3)CC12 c1(C(N2CC(C(C)C)CCC2C)C(=O)NCCOC)nc2c(s1)CC(C)CC2 C#CC1CCCN(C(=O)CC2(C)CN(C(=O)C=Cc3ccc(Cl)cc3)C2)C1 Cc1nc2cc(C(=O)NC3(C)CCCN(C(=O)CC(O)C(C)C)C3)cnc2s1 C(=O)(C1=CNS(=O)(=O)N=C1C)N(CC(C)NC(=O)C)CC.C1CCC1.O n1(CC)ncnc1C(=O)N(CCCNC(c1coc(Br)c1)=O)CCO C1(C(=O)NCC(CNC(C(c2ccccc2)SC)=O)O)CCCCN1N=O C(=O)(CCCCC(C)(C)C)NC1C(C(=O)Nc2cc(OC)cc(O)c2)CC=CC1 C(=O)(C(O)CCCNC(C1CS(=O)C1)=O)NC(C#C)CC c1(NCC(C)(C)NC(C(=Cc2cnc[nH]2)C)=O)cc(=O)n(C(C)C)c(O)n1 c1(OC)ccc2[nH]c(C(=O)NC3CCN(C(C4CNC(=O)N4)=O)C3C)cc2c1 C1(NC(c2cn(C)nc2)=O)CC(Nc2cc3c(s2)CCC3)C12CCC2 c1(CC2(NC(C=CCNC(CCC)=O)=O)CCC2)cccc(Cl)c1 c1(C(=O)NC2CCC(C(N3C(CC)CC(C)C3)=O)C2)cccn2cncc12 N1(C(CSCCC)=O)CCC2CN(C(C3(OCC)CCCCC3)=O)CCC2C1 C(=O)(C1=NOC2(CCOC2)C1)N(CCCNC(C1(C)CC(=O)N(C)C1)=O)C CCCCC(CCCC)C(=O)NC1CC(CNC(c2ccc3ccnn3c2)=O)C1 Cc1occc(=O)c1OCC=O.C1(C)(C(N2CC=CCC2)=O)CCC(F)(F)C1.N CC(CCC(C)(C)C)C(=O)N1CCC(C(F)(F)F)C(NC(C2COC(=O)N2)=O)C1 N1(C(CCS(N)(=O)=O)=O)CCN(C(C2CC23CC(F)(F)C3)=O)CC(O)C1 N=c1nc2cc(C(=O)NC3CCOC4(CCC4)C3)ccn2[nH]1 CC(CN(C)C)CC(=O)N(CCCCNC(C1C=CC=CC=C1)=O)C C1C(C2CC2)CCN1C(C1CC(O)C1)=O.c1(C(=O)NC)cc2c([nH]1)CCOC2 C(=O)CCC(C)(C)C.C1(CNC(CCOCCCOC)=O)(C)CC12CCC2 CCC(F)C(=O)NC(CNC(c1cc(-c2ccco2)c[nH]1)=O)CO c1(C(N2CCC(NC(C3(OC)CCCC3)=O)(CF)C2)=O)cc2occc2[nH]1 c1(CC)ncc(C(=O)NCCCOCCNC(=O)C(O)CSC)[nH]1 C1(NC(=O)NCC2(c3ccc(-c4cccc(O)c4)nc3)CC2)CCCCC1(F)F C(c1cccnc1)=C(C)C(=O)NC1CN(C(C2CC23CCCC3)=O)CC1C c1(C(N(C(C)CNC(C2CC=CCC2)=O)C)=O)ccc(OC2CC2(F)F)cc1 C(C1c2ccccc2CCN1C(c1c[nH]ccc1=O)=O)NC(C(C=C)(C)CC)=O C1(CC)C(C(=O)NCC(C)(F)F)CCN1C(=O)CN1CCOCC1 CC1CN(C(c2nc3c(s2)COCC3)=O)CCCN1C(=O)C(C)P(C)(C)=O n1(CC(=O)NCC(CNC)(F)F)cnc2c1c(=O)n(C)c(=O)n2C C1(C(=O)NCCOC2CN(C(Cc3ncc(C)[nH]3)=O)C2)(N(C)C)CCCSC1 C1(C(=O)NCC2N(C(=O)CCCN=[N+]=[N-])CCC(C)C2)CCc2ncncc2C1 N1(C(c2nccc(C)c2)=O)CC2CC(NC(c3ccc(C(F)F)cn3)=O)C(C2)C1 c1(OC)cccc(C(=O)NCC2CC23CCC3)c1F.n1(CC=O)nccn1.C C(CCC(F)(F)C(F)(F)F)N1C(=O)CC(CN2CCC(C(=O)OC)CC2)C1 c1(C(=O)NCCCC)cnc(OCC)c(Cl)c1.C(c1ccncc1C)=CC=O.N N1(C(COCCNC(CC2CC(CC)C2)=O)=O)C(C(=O)OC)CCC1C Cc1c(C(N2CCC(CNC(C3(C)CCC34CCC4)=O)C2)=O)nn2ccccc12 CC1CCC(C)N1CC(N1CCCC(CCNC(=O)CN2CSCC2=O)C1)=O N1(C(C(C(C)C)OC)=O)CC2CC(C)N(C(c3cnc(C#N)s3)=O)C2C1 CCCC(C(=O)N1CCC(C(=O)N(C)CC2CC2C)C1CC)N(C)C c1(C(=O)NC2CN(C(c3c(CCC)nns3)=O)C(C)C2)cc2c(nc1O)CCC2 N12CC3C(C3C1)NC(=O)C2C.c1(OCC(=O)N(CC)CC)ccsn1 N1(C(c2cnc(SC)n2C)C(=O)NCCC)CCOC2CCN(C)CC12 c1(C(=O)NCCN(C(c2ccn(-c3ccccc3)n2)=O)CC)ccccc1O C1(CNC(c2c(C(C)C)ccs2)=O)CCCCC1.C1(=C(C=O)F)CCCCC1.N CC1SCCCC1C(=O)NC(C)(C)CNC(=O)CCCSc1ccccc1 N1(C(C(N2CCCC(O)C2)C)=O)CC2CC(C1)C2NC(=O)CCN(C)CCO c1(C(CC)NC2(Cn3ccnn3)CCC2)cccc([N+](=O)[O-])c1 N1(CC)CCOCC1C(=O)NC1CCC(CC)C1.c1(CC=O)nc(C)sc1C.N c1(C(N2CCN(C(c3nc(C)oc3)=O)C3C2C3)=O)cc2c(Br)cncc2s1 C1(C(=O)NC2(C)CC(NC(=O)C(O)C(F)(F)F)C2)CCC2(CCC2)C1 c1(NC(C(=O)NCCCN(CC)CC)=O)ccccc1[Si](C)(C)c1ccccc1 c1(CC)cccnc1C(=O)OC.N1(C=O)CCN(CC)CC1.N12CCC(CC1)CC2=O CC(CC(=O)N(c1nnc(-c2cccs2)o1)C)c1cnn(C)c1 N1(C(c2ncn3cccnc23)=O)CC2CCCC(C1)N2C(C1(C(F)F)CC1)=O CC1CN(C(C2(C)CCN(C)C2)=O)CC1n1cc(-c2cncs2)nn1 c1(OC)ccc(O)cc1C(=O)NC1CC(CNC(=O)C(O)CF)C1 c1(C(=O)NC(CNC(C=C(CC)CC)=O)C(C)C)ccc(F)c(OC)c1 c1(CC)ccc(OC)c(C(=O)OCCOC2CCCC2)c1.c1(N)cccc(F)c1 CCCC(CNC(=O)CC1(O)CCCOC1)C(=O)Nc1csnc1OC c1(NC(C2CC(O)CCN2C(C2CC2(F)F)=O)=O)nc(Cl)ccc1F c1(CC)ccc(F)cc1C(=O)NCCOC.N1(CC=O)CN(C)C(=O)C1C N1(C(Cc2c(C)ocn2)=O)CCC(CNC(=O)CC2CC3CCC2C3)CC1 N1(C(c2cnc(CC)[nH]2)=O)CCN(C(C2CSCCS2)=O)CC1CC1CC1 C(=O)(C(CCC(C)C)NC(=O)CCCNC=O)NCCN(CCO)CC C1(NC(c2nc(C)oc2C)=O)CN(C(c2ccc(C(F)(F)F)s2)=O)CC1(C)C C(=O)(C#CC(C)(C)CNC(C1(CCOC)CCC1)=O)N(CC(CCC)C)C Cc1ccnc(-n2cc(C3CCN3C(=O)C(C3CCCO3)C3CC3)nn2)n1 c1(N2CCC(Cc3cc(C(C)=O)no3)C2)ncccc1S(N)(=O)=O C1(CC(C)C)CCCN(C(=NCCCCC(F)(F)F)NC2CCCC2)C1 CC(C)(O)CC(=O)N1CC(O)CC1CNC(c1csc(-c2ccoc2)n1)=O Nc1ccc(C(=O)NCC2CC2NC(C2(F)CCCCC2)=O)cc1Cl c1(C(=O)NCC(C)(O)CNC(c2cccnc2O)=O)cccnc1O CC1CCOCC1C(N1CC(F)CC1C(N1CCOC(CC(N)=O)C1)=O)=O c1(-c2cc(C(=O)NCC(C)NC(=O)CC3CCC(=O)O3)n[nH]2)ccccc1F C(=O)(C(C(C)C)NC(c1ccc(Cl)cn1)=O)N1CCC(=C)C1 c1(C(=O)NC(CC(C)NC(CSCC(C)C)=O)C)ccc2oncc2c1 c1(C(N2C3CC(NC(C(C)NS(C)(=O)=O)=O)C2CC3)=O)cccc2c1ncn2C N1(C(Cc2cc(C)sc2)=O)C2CCC(C2)C1CC(=O)NOCCC(C)C N1(C(c2ccnn2CC(F)F)C(=O)NCCC#N)CCCC2(C1)C(O)CC2O c1(C(N2CCC(C(C)(C)C)C2)=O)cc(F)cnc1O.CC1CCC(C(=O)NC)C1 c1(C(=O)NCC(CNC(c2c(C)snn2)=O)F)ncc(Br)cc1F N1(C(C=C(COC)C)=O)CCC(NC(C2CC23CCCC3)=O)C1C1CC1 C1(C(N2CC(C)(NC(CCc3ccc(C)o3)=O)C2)=O)CCCCC12CC2 N1(C(=O)OC(C)(C)C)CCC(C2CC2)(NC(N2CCOC(CF)C2)=O)CC1 N1(CC(=O)NCC2CC2)CC2CC2C1.c1(C(=O)N)cnc(C(F)(F)F)s1 Cc1nc2cc(Cl)cc(C(=O)N(C(C)CN(C)C(c3cc(=O)cc[nH]3)=O)C)c2[nH]1 CCC(C)C(C)N=c1nc(NCCCS(=O)(=O)NC)c2c([nH]1)c(C)nn2C c1(SC)cccc(C(=O)N(C2CCN(C(C3CC3c3ccncc3)=O)CC2)C)c1 c1(C(N2CCC(C)C2CNC(=O)Cc2cnccn2)=O)cnn2cc[nH]c(=O)c12 C1(C=O)CCN(C(C)C)CC1.C1(CC)CCCC1C(N1CC(C(N)=O)C1)=O.C C1(C#N)(C(=O)NC2CC(NC(Cc3onc(C)n3)=O)C2)CC1(C)C c1(CC(=O)N(CC(CC)NC(C2CC(F)C2)=O)CC)nc2c([nH]1)CCCC2 c1(OC)c(NC2CC3CN(C(c4cc(Cl)cs4)=O)CC23)ncnc1C CC(C)(F)C(C)(F)C(=O)NC1C=CC(CC(=O)NC(C(N)=O)C2CC2)C1 C1(C(C(=O)OC)N)CCN(C(c2ccc(-c3ccc(Br)s3)s2)=O)CC1 C1(NC(CC(CC)C2CC2)=O)(CO)CCCN(C(=O)COc2ccc(Cl)nc2)C1 C1(N(C(CCCOCC=C)=O)C)CCCN(C(=O)C(F)(F)COC)CC1 c1(C(N2CC3(C(C(=O)NC(C)C(F)(F)F)C3)C2)=O)cc(O)cc(F)c1 c1(C(=O)NC2CCC(CNC(CCC(=C)Br)=O)C2)ccc(=O)n(CC)n1 c1(NC(C2C(NCc3cnc(C)s3)C2)=O)ncc(Br)nc1C(N)=O c1(OCC)ccc(Cl)c(C(=O)NC2CCCC(NC(=O)C(C)OC)C2)n1 c1(C(N2CC(NC(Cc3nnc(C)o3)=O)C(C)C2)=O)c(C)cc(=O)oc1C C(=O)(C#CC1(C)CC1)NCC1(OC)CN(C(=O)C(N2CCC(O)CC2)C)C1 c1(C(C(=O)N(C(C)C(C)C)Cc2ccco2)NC)ccc(Cl)cc1 c1(C(N2CC3OCCOC3C2)C(=O)NCCCSC)nc(Cl)cc(Cl)c1C c1(C(=O)NCC2(CO)CCN(C(C(CC)F)=O)CC2)c(Br)ccc(C)c1F C(=O)(C(C)CC(F)(F)F)N1CCCC(O)C1.Cc1noc(C(=O)N)c1C(F)(F)F CC1NC(=O)C(C)N(C(=O)Cc2cn(C)nn2)C1C N1(C(C2C(C=C)CC2)=O)CC2=C(C1)CN(C(=O)C(C1CCC1)OCC)C2 C=CCCCCCCC(=O)N(C(C)(C(=O)NC(C)COCCOC)C1CC1)C c1(C(C2CCC2)N(C2CC2)CC)cccc(C(F)(F)F)c1 C1(NC(CCS(C)=O)=O)CCOC12CCN(C(=O)CNS(=O)(=O)C1CC1)CC2 N1(Cc2c(C)cn(C)n2)CCC2(CC1)CC2(C)C(=O)N(CC(N)=O)C Cc1cc(C(=O)NC2(C)CCCCC2)cnn1.c1(C=O)ccnn1C(C)(C)C.N C(CC(O)C(=O)NC(c1ccnn1C)C)NC(Cn1ccc(C)n1)=O Cn1nc(C(=O)NC2COCC2n2ccnc2)c2c1CCC(F)(F)C2 C(=O)(C1=NN(C)C(=O)CC1)N1CC(C(N2CC(C(C)C)C2)=O)C2(C1)CCC2 N1(C(c2nc(CC)sc2)=O)CC2CC1C2NC(C1CCC(OC)C1)=O c1(C(N2CCCC(NC(CCSCCC)=O)C2C)=O)ccc2c(=O)ccoc2c1 C(=O)(CCC(CC)CCC)N1CC2C(CNC(C3(C#C)CCC3)=O)C2C1 C1(CNC(C2(OC)CCC2)=O)CCC2CN(C(C3OC4CCC3C4)=O)CC12 n1(C(C)C)cc(C2(N(C3CCC3(F)F)C(C3(C(=O)O)CC3)=O)CCC2)nn1 C1(C(N2C(C(CNC(C(C)(C)CF)=O)(C)C)CCC2)=O)CCc2nccn2C1 c1(OC)ccc(C)c(C(=O)N)c1.c1(C2(C=O)CC2)ccnn1C.C(C)C1CC1 C1(C(C)(C)C)CCN(C(C2(C)CS(=O)(=O)C2)=O)C1.C=C1CC1C(=O)N N1(C(CC(C)(F)F)=O)CCC(C2(NC(=O)CO)CC2)CC1.c1cc(Cl)cc(Cl)c1 CCS(=O)CC(=O)NCCOC1CCN(C(C2C=CCCC2)=O)CC1 c1(C(C)C)ccccc1OCCC(=O)NC1C2CN(CCC3CCCCO3)CC12 C1(C(=O)NCC(C)(C2CC2)NC(c2nccc(C)c2)=O)COC2(C)CC1C2 C(=O)(CCCCCCCC(=O)OC)N1CCC(CNC(CCCOC)=O)(OC)C1 C(CNC(C1CCN(C)C1)=O)(C(=O)N1CC(O)(CN(C)C)C1)OC N1(C(C(n2c(C)ccn2)C)=O)CCOC(CCNC(=O)CCCc2cnn[nH]2)C1 c1(C(=O)OC)snc(C(=O)NC(c2ccc(C(F)(F)F)cc2)CC(=O)O)c1I N1(C(C(CC)NC(=O)C(C2CCCCC2)C)=O)C2CCCC1CC2 Cc1ccc2c(CC(=O)NCc3c(C)noc3C(=O)O)coc2c1C CC1=C(C)CC(C)(C(=O)NC2CC(CO)N(C(c3cc(Br)n[nH]3)=O)C2)CC1 CCCCCCC(C)C(=O)NC(CNC(c1ccc(O)cc1F)=O)C1CC1 C1(C(=O)N(CC(F)(F)COC)C)(NC(CCOC)=O)CCN(C)C1 c1(CC=C)ccccc1C(=O)NCC1CN(C(=O)CC2CSC2)CCO1 c1(C(=O)NCCC(C)(C)NC(C23CCC2C3)=O)cc(N)ccc1[N+](=O)[O-] C(CCCCCNC(=O)C(C1CC1)C1CC1)NC(C(c1cnn(C)c1)C)=O N1(C(CCC)=O)CC(CNC(=O)C(CC)NC(N)=O)OC2(CCC2)C1 N1(C(c2c(OC)c(Cl)sc2)=O)CC2CC(NC(c3cn(C)c(O)n3)=O)C1C2 N1(C(C2N(C(c3ccncc3CC)=O)CCC(=C)C2)=O)CC(C)NC(=O)C12CC2 c1(-c2ccc(C(=O)NCCCC)cc2)ccn2nc(C(=O)NC3(C)CC3)cc2c1 N1(C(c2nc(N(C)C)oc2)=O)CC2CCN(C(=O)CCn3cncn3)CC12 C=CCC(C)C(=O)N1CCC(c2n[nH]cc2CNC(=O)CCc2cnccn2)C1 c1(-c2nnc(C)o2)ccc(OCc2cnc(Cl)s2)cc1 Cc1cc(C(=O)NC(CNC(=O)C(c2cncn2C)O)CO)cs1 N1(C(C(C)CC2CC2)=O)CCC(C)C12CC2.C1(C)(C(=O)N)CS(=O)(=O)C1 C(=O)(C(CCOC)NC(=O)Cc1nonc1C)N1CCC(OC)C1 N1(C(c2nnc(C)s2)=O)CCN(C(=O)NC(C2CC3(CCC3)C2)C)CC1 C(C)(C(=O)NCC1CC1NC(=O)C)(c1ccccc1)OC.c1cccnc1 C(=O)(C1=NOCC1)NC(C(=O)NCC(C)(C)CO)Cc1cc[nH]n1 c1(CCCC)ccc(CC(=O)OCC=CCl)cc1.C12CCCN1C(=O)C2 N1(C(C(CC)(C)C)=O)CC(CC(=O)NC2(C)CCCC2C)C2(CC2)C1 N1(C(Cc2c(C)ccs2)=O)CC(C(N2CCCC(CCCO)C2)=O)CCC1C CC(CNC(=O)CC1(O)CCC1)CC(=O)N1CCC(c2nn[nH]n2)C1 C1(C(N2CC(C)(CCC(=O)NC(c3cncs3)C)C2)=O)COCC1(C)C C(=O)(C(C(F)(F)F)C(F)(F)F)N1CC(NC(c2cncc(Cl)c2)=O)CC(C)C1 c1(CNC(C(C2CCOC2)OC)=O)ccc(C(C)NC(C2SCCS2)=O)cc1 c1(OC)ccc(NC(=O)CC2(C)CCN(C(=O)C(C3CCOCC3)F)C2)cc1F N1(C(C2CC(C(C)C)C2)=O)Cc2[nH]nc(C(=O)Nc3cccc([N+](=O)[O-])c3)c2C1 Cc1ccc(CCC(=O)NC2CCC(C)N(C(c3c[nH]c(=N)s3)=O)C2)cc1Cl Cc1c(C(=O)NC23CC(NC(C4CC5CC4CC5O)=O)(C2)C3)nc2sccn12 C1(C)(NC(C2N(C(CCC(CC)C)=O)CCC2)=O)CCC(C)(C)CC1 n1(CCC)ccc(=NC(=O)C(C)(C2CC2)N(C(=O)C(C)NC(=O)CC)C)[nH]1 Cc1cc(Br)cc(C)c1C(=O)NC(C)CNC(=O)C(F)(F)CC(C)C C1(C(=O)NC2C3CC4C(C3)C24C(N2CC(CO)C2)=O)CC2(CCC2)CO1 C1(=O)CCC(=O)N1C(C)(CO)C1CCC1.C(=O)(CC)NCCCO.C1CC1 C=CCC(C(=O)N1CCN(C(c2cccc3c2NCC3)=O)CC1C1CC1)C(C)C CCCC(C)(CC)C(=O)N1CCCC(N(C(=O)COC2(C)CCCC2)CCO)C1 C1(C(N2CCC(O)C2)=O)CN(S(N)(=O)=O)C1.CC(C(=O)N)NS(C)(=O)=O N1(C(c2ccc(C)c(Cl)c2N)=O)CCC2CN(C(=O)CCc3ccoc3)CC2C1 C1(C(c2nnnn2C)NC2(CN3CCOCC3=O)CC2)(SC)CCCCC1 N1(C(c2ccc(C)nc2)=O)CCC(NC(C2(C)CNC(=O)C2)=O)C(C(N)=O)C1 c1(C(=O)NC(C(C)NC(C(C)Oc2ccc(C)cc2)=O)CO)ccc(C)nc1N CN1CCC(C(=O)NCC2(F)CC(CNC(c3cncnc3)=O)C2)C1 C#CC1(NC(=O)CC=CCNC(=O)Cn2ccnc2)CC2CCCC12 N1(C(CC)C(=O)Nc2cc(Br)cs2)CCN(C2CN(c3ncccn3)C2)CC1 CC1(C)CCC=C1C(=O)NCC1(F)CN(C(=O)CC2CCCC(F)(F)C2)C1 C(=O)(CC(CC1CC1)NC(c1cc(Cl)cn1C)=O)N(C)CC1(F)CCC1 C1(CCNC(C2CCCC3CCCCC23)=O)CC(N=c2[nH]nc(C(F)F)o2)C1 C1(O)(CNC(C2CCC(O)C2)=O)CCCN(C(c2ccccc2F)=O)C1 CC1CN(C(=O)COC2CCCCC2C)CCC1C(N1CCCC1C(N)=O)=O N1(C(=O)C(c2cccc(F)c2)O)CCN(C(c2ccncc2)=O)C(CO)C1 CC(CF)CC(=O)NCCC1(O)CCN(C(=O)Cc2csc(Cl)n2)C1 C1(C(=O)NCCC(CC)(C)C)CCN(C(=O)CCC2CCCO2)CC1O C1(NC(C(C)C2CCC2)=O)CCCCN(C(C23CC(CF)(CO2)C3)=O)C1 Cn1nc(C(N2CCCC(CCNC(C3CCC34CCC4)=O)C2)=O)ccc1=O CS(=O)(=O)CCC(=O)NCC1(CO)CCN(C(=O)C(F)F)CC1 Cc1c(C(=O)N(C2CN(C(=O)C(C)(C)F)C2)C)oc2ccccc2c1=O C1(NC(CN(C2CC2)CC)=O)CN(C(C2CCC=CCCC2)=O)CC12CCCC2 c1(C(N(CCN(C(C=CCCC)=O)C(C)C)C)=O)ccn(C2CC2(F)F)n1 c1(OC)nccnc1C(=O)NC(C)CC(C)(C)c1ccccc1 C1(CNC(C2(N(C)C)CCCC2)=O)CC(NC(C2SCCS2)=O)C12CCC2 C#CC(C)(C1CCC1)NC(=O)CCC1CC(NC(=O)C)C1.C1CC=CC1.O N1(C(CC=C(C)C)=O)CC(O)(C2(CNC(C3CCCOC3C)=O)CC2)C1 CC(C)S(C)(=O)=O.c1(CC)nc(C(=O)N)co1.c1(C=O)ccon1.C1CC1 C(CC(C)C(=O)N1CCC(C(C)CNC(C2CC2)=O)CC1)OC.N1CCCC1.C Cc1[nH]c(CN2CC3CCC2CN3C(=O)C=Cc2ccsc2)c(C)c1[N+](=O)[O-] Cc1ccc(C)c(C(=O)NC2CN(C(c3ccc(-c4ccncc4)s3)=O)C2)n1 c1(C(=O)NC2C(CNC(C3(N=[N+]=[N-])CC3)=O)C2)ccccc1.[nH]1cccn1 C1(C(N(C)C)=O)CCC(NC(=O)C(N2CCC(c3ccncc3)C2)=O)CC1 c1(C(=O)NC(C)CNC(c2occc2F)=O)ccc(=O)n(C)n1.c1ccccc1 c1(CN2CCC(C)(NC(c3ccccc3)=O)C2)c(C(F)(F)F)[nH]c2ccccc12 c1(NCCCNC(C2CC(=O)N2)=O)c(Cl)cc([N+](=O)[O-])cc1Cl CON(CCO)C(=O)C(CCC1CC1)NC(=O)C(C)S(N)(=O)=O N1(C(CSC)=O)CCN(C)C(CNC(=O)C=CI)C1 Cc1cc(NC(C2CCCN2C(c2ccccc2C2CC2)=O)=O)c(O)cc1F C(C)(CCN=c1cc(C)nc(S(C)(=O)=O)[nH]1)NC(c1nc(OCC)oc1)=O C(C)(CO)(C(=O)NCC1CC(O)(C)C1)NC(C)=O.C(=O)(CC(C)F)N Cc1nsc(C)c1C(N1CCC(N(C)C(c2cc(CF)on2)=O)C1)=O c1(C(=O)NCC(C)CNC(c2cscc2C2CC2)=O)cnc(N(C)C)cn1 N1(C(c2cc(Br)cc(C)c2N)=O)CCCC2(CCN(C)C2=O)C1 N1(C(CSC(C)C)=O)CCC2(CCCCC2NC(C2CCC(C)(C)O2)=O)CC1 c1(C(N(C2CCCC2)CCNC(CC2N(C)CCOC2)=O)=O)cc([N+](=O)[O-])c[nH]1 C1(NC(CCNS(CC)(=O)=O)=O)CCCCCN(C(=O)C(C)OCCOC)C1 C(=O)(CCCn1ccnc1)N1CC(C(C)NC(C(F)OC)=O)C1 N1(C(CC2(C)CCOCC2)=O)CC(NC(C2C(Cl)(Cl)C23CC3)=O)CC(O)C1 c1(OC)cccc(F)c1C(=O)NC1CC(NCc2ncsc2C)C1 N1(C(=O)NC(c2cccc(Cl)c2)COC)CCC(C2COCCO2)CC1 c1(N(CC(=O)NCCOC2CCN(C(CCC=C)=O)C2)C)ccc(Cl)nn1 Cc1ncncc1C(=O)NCC1CCCCC1NC(C1CCN(C)CC1)=O C12(C(=O)NCCCNC(COCC(C)(C)C)=O)CCCCC1C2 c1(C(=O)NCC(CNC(C(CC)NC(c2ccco2)=O)=O)O)cnc(N)cn1 C1(NC(C=C(COC)C)=O)CN(C(=O)C(=C2CCCCC2)F)CC1C c1(C(N2CC(NC(C=CSC)=O)CC23CCOC3)=O)nn(C)c2ccc(F)cc12 N1(C(C(CCC)F)=O)CCCCC(N(C(=O)CCOCCOC)C)C1 CC1CCC(C(=O)N(CCCNC(c2coc(C(F)(F)F)n2)=O)C)O1 C#CCC(CC#C)C(=O)NC1CN(C(c2ccc3c(n2)CCO3)=O)CC1O c1(N2c3cccc(CC)c3CCC2)nc(=NC2CC(Cl)(Cl)C2)[nH]c2c1SCC2 N1(C(c2ccc(COC)s2)=O)CC2CCC1C2NC(C1CCOC1)=O c1(COC(C2CCCN(CC(C)C)C2)=O)ccc(F)c(F)c1 C1(NC(C(N2CC(C)C2)C)=O)CN(C(=O)C(O)CC2CCOCC2)CCC1O N1(C(C(C)CN(C)C)=O)CC2CCN(C(C3(c4ccncc4)CC3)=O)CC12 C12(C(=O)NCCCCN(C)C(C3CC(C4CCCC4)C3)=O)CCCC(C)(C1)OC2 C1(CN(C(=O)CCSC2CCCC2)C)CCN(C(C2CCC2(F)F)=O)C1 C1(C(=O)NCC2(OCC)CN(C(C3CCCC3)=O)C2)CCCC(=O)N1.O C=CC1(C(=O)N(CCCN(C(=O)C(F)(F)c2cscn2)C)C)CCC1 Cc1ccc(C(=O)NCCOCCNC(=O)CSCCC(F)(F)F)nc1 N1(c2c(C#N)c(Cl)ns2)CCC2CC(NC(c3ccncc3F)=O)CCC2C1 Cc1cccc(CC(=O)NC2CN(C(=O)Cn3nccn3)CC23CC3)c1Br c1(C(N2CC=CC(NC(C3CN(CC)C(=O)CC3)=O)C2)=O)nccc2occc12 c1(NC(=O)OC(C)(C)C)cc(CNc2ncc(C(N)=O)cc2Br)ccc1Br C(CCCCCCC(=O)NC1CN(C(=O)CCc2nc[nH]n2)C1)SC Cn1ncc(C(F)(F)F)c1C(=O)N.C1(O)CCN(C(C2CC(F)(F)C2)=O)C1 c1(C(=O)NC2CC=C(C(N3CC(C#C)C(OC)C3)=O)C2)ccc(C#N)c(C)c1 O=[N+]([O-])c1ccc(CCCNC2CC3(COC(CO)C3)C2)cc1 c1(C=O)ccnc(-n2ccnc2)c1.c1(C(=O)OC)ccc(CNC(C)C)s1.N N1(C(C2N=C(C)SC2)=O)CC2(CCN(C(c3n[nH]c(C)n3)=O)CC2)C1 C(CC(O)C(=O)NCCCN(C)C(C1CCC(C(F)(F)F)CC1)=O)SC Cc1cnc(C(=O)NC(CNC(c2ccc(Br)o2)=O)CC(C)C)cc1Cl c1(C=O)cc2n(n1)CCCO2.CN(S(N)(=O)=O)CC(=O)NCC1(F)CCC1 c1(C(N2C3(CN(c4nc(SC)c(Br)cn4)C3)CC2)=O)cc2ccccn2n1 c1(C(N2CC(NC(CC3N(C(C)=O)CCC3)=O)C(O)C2)=O)cc(Cl)c(Cl)n1C CC1CCN(C(C2CC(N3CCCC3)C2)=O)C1CNC(=O)CS.c1nc[nH]n1 C1(O)(CNC(C2NC(=O)OCC2)=O)CCN(C(C23COCC2C3(F)F)=O)CC1 C#Cc1c[nH]nc1C(N1CC(O)CC1C(=O)N(C1COC(C)(C)C1)C)=O C1(NC(c2cnc3cccnn23)=O)CCC2(CCN(C(c3cc[nH]c3)=O)C2)C1 C1CN(C(=O)CC2(N3CCCC3)CC2)CCN1C.C(C)(C)(C=CC=O)SC.N N1(C(CC2(OC)CN(C(=O)Cn3ccnc3)C2)=O)CCC(F)(F)C(O)C1 c1(CNC(C(=O)OC)c2ccoc2)cn2ccc(Br)cc2n1 CC1CC(NC(=O)CCc2cn(C)nn2)CCN1C(c1ccsc1)=O C(CC(C(=O)N1CCCO1)NC(C1CC1C(F)F)=O)OCC N1(C(C(C)c2ccsc2)=O)CCC(C)(C)C(NC(=O)CCS(=O)(=O)N(C)C)C1 Cc1cc(C(N2c3cnn(C)c3CCC2C(F)F)=O)c2ccc(F)cc2n1 C#CCC(CC(F)F)NC(C1(COC)C=CCN1C(c1cc[nH]c1C)=O)=O C(=O)(C1SCCc2sccc21)NCCCN(C(C1CCCC1(F)F)=O)CC N1(C(C=CC(C)C)=O)CCCN(C(C)C)CC1.C1(C=O)(OCC)CCC1.N c1(CC(=O)N(C2CCN(C(=O)Cc3ccsn3)C2)CCC)scnc1C.C=O C=CCC(C(=O)N1CC2CC1(C(=O)N(C1CCC3CC13)C)C2)C(C)C N1(C(c2c(CNC(C(CC)N(C)C)=O)nccc2)=O)Cc2nc(C)sc2C1 C12(NC(COc3ccc(C)cc3)=O)COCCC1CN(C(C1(C)CC=CC1)=O)C2 C1(NC(CN2CC(C)(OC)C2)=O)CCOC(CNC(C2CCCNC2=O)=O)C1 N1(C(C23CC(NCc4ccc(CC)cc4O)(C2)C3)=O)CCCC2(CCO2)C1 N1(C(C(C(C)C)C)=O)CC(NC(c2nnn(-c3ccccc3)n2)=O)CC(C)C1 c1(C(=O)NCC2CCCN(C(CC(CC)O)=O)C2)ccc(F)c(OC(F)(F)F)c1 Cc1ccc(-c2c[nH]cc2C(=O)N(C)CCNC(=O)C(C)CN(C)C)s1 c1(N(C)CC)ccnc(C(=O)NC)c1.N12CCN(CC1)CC21CCC1 n1(CC(=O)NCC2N(C(C(C(C)(C)O)(C)C)=O)CC2)nc2ccccn2c1=O C1(CNC(C(CSC)O)=O)CCCC(C)(C)C1.C12CCCC(C1)C(=O)N2 c1(C(=O)NCc2ccc(COC)o2)ccc(F)c2ccoc12.N1(C)CCOCC1 C12(CNC(C3CN(C(C)=O)C3)=O)CC(CO1)C2.c1(C=O)cc(C)[nH]n1.C N1(C(C(C)=O)=O)CC(CO)C2(CCN(C(=O)CN(c3ccccc3)C)CC2)C1 O=C(C(F)C(F)(F)F)NCC1CCCCN1C(=O)CCOc1ccccc1Cl CC1(CNC(C2CC(O)(CNC(=O)C(C)(O)CO)C2)=O)CCCCO1 N1(C(c2ccc(C(N)=O)s2)=O)CCN(C(C2(C(F)F)CCCC2)=O)CC(O)C1 C(C(CC(C)C)C(=O)N1CC(CC)(CO)C1)NC(C1(CC#C)CC1)=O CCC(CNC(c1csc(C)n1)=O)(CC)C(=O)NC(CC1CC1)CO C(CN=c1[nH]c(=NC(C)C2CCCC2O)c2cc(Cl)ccc2[nH]1)=CCOC C1(NC(c2n(CC=C)ccc2)=O)CCC(C)N(C(c2cccc(CC)c2N)=O)C1 CC1CCC2CCC1N2C(=O)CC(C)(O)C(F)(F)F.C1(C=O)(C(N)=O)CCC1.N N1(C(C=CC)=O)CCC2CCN(C(c3cn4cc(C)sc4n3)=O)C2C1 c1(NC(CC(=O)NC)C)cc(N2CCS(=O)CC2)nc(C(F)(F)F)n1 c1(C(N2CCN(C(C(CC)C)=O)CC2CF)=O)cc2cc(C)cc(C)c2[nH]1 N1(C(C=CCOC)=O)CCCC(CNC(C2C=CCCC2)=O)CC1 C12(C(N(C3CCN(C(c4cncc(C)c4)=O)C3)CCC)=O)CC(C)(CO1)C2 C1(O)(CNC(=O)OC(C)(C)C)CCN(C(=O)C=O)C1.CCCOC(F)F C(CCCCCCn1cc(CCC2CC2)nn1)NC(=O)C(O)Cn1cncn1 c1(C(C)(C)OC)cn(C(C)C(=O)NCCC(C2CCCCC2)O)nn1 n1(CC2(N(C)CC)CCC2)ncc2c(Br)cc(C)cc2c1=O Cn1cnc2cccc(C(=O)NC3CC3CNC(C3CCC(C)(F)CC3)=O)c12 C(=O)(C(O)C1=CCCCC1)N1C(CC(N2CC(CC(C)C)OCC2)=O)CC1 C1(CNC(C(C)n2cnnn2)=O)C(C2CC2)CCN1C(c1cc(C#N)cs1)=O C1(c2nnnn2C2CC2)(NCc2nc(COC)[nH]n2)CCc2cccnc2CC1 c1(CC)cccc2[nH]c(C(N3CCN(C(C4CC4(F)F)=O)C(C4CC4)C3)=O)cc12 Cc1cc(C(=O)N(CCCCN(C)C(C2NC(=O)CC2C)=O)C)c(F)cc1F C1(NC(c2n(CCCOC)nnn2)c2ccc(I)s2)CCC(=O)NC12CCC2 c1(C(CCC)N(C(=O)C=Cc2scnc2C)C)cccc(C(F)(F)F)c1 c1(C(=O)NCC2OCCN(C(c3ccc(C)c(C)c3)=O)C2)ncc2n1CCCC2 C(=O)(C1=CC2CC(C1)CC2O)NCC1(NC(CCCNC(C)=O)=O)CCC1 C1(C(N2CCCC(CC)CC2)=O)CC2(C1)C(F)(F)C21CC1.C(C(=O)N)=C(C)Cl C(=O)(CC(O)CC(C)C)NCC(C)(C)NC(Cc1cccc(C)c1C)=O Cc1cccc(NNC(=O)Cn2ccnn2)c1F c1(C(=O)NC(C)(CNC(=O)CCC(N)=O)C2CCC2)cncc2c(Cl)cccc12 CN1CCOC(C(=O)NCC2(C)CN(C(c3cncn3C)=O)CCO2)C1=O c1(C(=O)NCC2N(C(c3c(C)onc3)=O)CCCC2)nccc(Cl)c1C C=CCCCCCC(=O)NC1CC2CC(C1)N(C(=O)CCSc1ccccc1)C2 O(S(=O)(=O)c1cccc(F)c1C)c1c(=O)cc(C)oc1 C1(CC)CCCC(C(=O)NCC2CC(F)C2)C1.n1(C2(C=O)CC2)cncn1 c1(C(=O)NC(CC)CN(C(=O)C(C)NS(C)(=O)=O)C)ccc(C#N)s1 C(C(CCCC)NC(C1(CCOC)CC1)=O)NC(CCC#C)=O C(=O)(CCCCCCC)NCCC1CCN(C(C(CC#C)(C)C)=O)C1 c1(-n2ncc(NC(Cc3c(C)nc[nH]3)=O)c2)ccccc1F c1(C(N2C(Cc3cccc(OC)c3)CCC2)C(=O)NC(C)C)cncc(Cl)c1C C1(CNC(CC=CCNC(C2C3CN(C)CC32)=O)=O)CCC2(CC2)CO1 c1(CN2CCC(N(C(C3CC(=C)C3)=O)C)C2)cccc2nc[nH]c12 O=C(N=c1ccn(Cc2ccncc2)[nH]1)N1CC2(CO)CCC1CC2 C(=O)(C(C)C(O)C(C)C)NC(C(=O)NCC(CCC)CCO)CC1CC1 N1(C(C2C(C(=O)OC)C2)=O)CCCC1(C)C.C(c1ccccc1Cl)=CC(=O)N c1(OC)cccc(F)c1C(C)NC(=O)C(=O)NCc1cc([N+](=O)[O-])sn1 C(=O)(C(C)CCN(C)C)N(CCC(N1CCC(NC(C)=O)C1)=O)CC C1(NC(=O)CSCC(F)F)CN(C(c2nocc2Cl)=O)CC1C1CC1 CCC(F)(F)CC(=O)N1CC(C)(C)CC1C(N1CCC12CC(C(N)=O)C2)=O C1(C(=O)NCC2CCN2C(c2cn(CCF)nn2)=O)CCCCCCC1 c1(C(=O)NCC(C)(CO)NC(C(CC)SC)=O)c(OC)cccc1F c1(C(N2CC(NC(c3cc(C)sc3)=O)C2)=O)cc2c(s1)CC(C)(C)C2 C1(C)(NC(C2CN(S(CC)(=O)=O)C2)=O)CCCN(c2cc(C(F)F)ncn2)C1 c1(C(N2CC(CNC(C(C=CC)O)=O)C(C)(C)C2)=O)cnc2c(c1)COCC2 Cc1cc(C(=O)NC2(CNC(C3(C#N)CC3C)=O)CCCCC2)cn(C)c1=O C(=O)(C(C)S(N)(=O)=O)N(CCNC(CCc1nnc(C)o1)=O)CC1CC1 N1(C(CC)CC)CC(C(=O)NCCC(C)(C)NC(=O)C=CBr)CC1=O Cc1nn(C)c(C)c1C(C)C=O.C1(CC)CCCN(C(C23CC(F)(C2)C3)=O)C1 C=CC(O)(C(=O)N1CCC2(CC1)CN(C(=O)CCCC(C)CCC)C2)C(F)(F)F CCC(C(=O)N(C(CNC(=O)CC)C1CC1)C)Oc1ccccc1.C1CC1.O C1(C(N2CC(NC(CC3(C)CC3(F)Cl)=O)C2)=O)CCN(C2CC2)CC1 C1(C(=O)NCC2C(CC#C)C2)CCCCN1C(=O)CC1CC(=C)C1 n1(CCCC)ncc(C(=O)N(CCNC(=O)C#CC(C)C)C2CC2)c1CC c1(NC(CN2CCCC(CSC)C2)=O)cn(C)c(=O)cn1 c1(OC)ccc(C(C)=CC(=O)NC(CC)C(C)C)cc1.C1(C)(C=O)CC1C.N C1(NC(c2cc(C)no2)=O)CN(C(c2cc(O)nc(O)n2)=O)CCC1O C1(CNC(c2c(C(C)C)nn(C)c2)=O)CN(C(=O)C(=O)C(F)(F)F)CCN1C c1(C(C)C(=O)NCC2CC3CC3N2C(c2nnn(C)n2)=O)cc(Cl)cc(Cl)c1 Cc1ccc2ncn(CC(=O)NC(CNC(C3CC34CCC4)=O)C3CCC3)c2c1 C(CC(C)(C)C(=O)NCc1nc(C(=O)NCC(C)OC)c(C)o1)OC Cc1cnc(NCc2cc(Cl)cc(Cl)c2F)c(S(=O)(=O)N2CCOC(C)CC2)c1 CC(C)CC(CC(C)C)C(=O)NCCNC(=O)C=Cc1cn[nH]c1.C1CC1.C C1(COC)C=CCCN1C(=O)C(c1cn(C)nn1)NC(=O)C(C)N=[N+]=[N-] C1(NC(Cc2c(CC#N)cccc2)=O)CC2CC1CN2C(c1cnco1)=O N1(C(C2N(C(C(C(CC)(C)C)O)=O)C3CCC2C3)=O)CC2OC(=O)N(C)C2C1 c1(C(C)=O)ccc(C(=O)NC2CCCC2NC(=O)C#CC2CC2)c(F)c1 C1(NC(CONC(Cc2scc(C)n2)=O)=O)CCCC1C#N C(C)(C(C(=O)NCCN=[N+]=[N-])NC(c1coc(C)c1)=O)OC C(=O)(C1CCc2cccc(O)c21)N1C2CCC(NC(CCC)=O)C(C2)C1 C(C(C(=O)NC1(C(=O)N(CC(C)(C)C)CCO)CC1(C)C)OC)OC C1(C(N2CC(C)(C#N)C2)=O)CC(N=[N+]=[N-])CN1C(=O)CCS(C)(=O)=O C(=O)(C(O)P(C)(C)=O)N.c1(C(=O)NCCC(=C)C)ccccc1NCCO c1(C(N2CCCC(C3CCCN3C(=O)CC(F)(F)F)C2)=O)ccc(F)c(I)c1 c1(C(C(=O)NCC2CCCO2)N(C)Cc2cnc(C)s2)c2ccccc2nn1C C(=O)(C1CCc2ccccc21)NC(C(=O)Nc1c(OC)cc(O)cc1)CC(C)C C1(NCCOC)CCN(C(=O)C(=O)NCc2ccc(C3CC3)cc2)CC1 c1(C(=O)NCC(C(C)C)NC(C2(C=C)CC2)=O)ccnc2cc(C)ccc12 C#CC1(C(N2CC3CC(C2)C3(C)C)=O)CCN(C(C2CCCCC2O)=O)CC1 C1(CCC(=O)NC(CCNC(C2CC(OC)(OC)C2)=O)C)CCC(O)CC1 Cc1ncc(C(=O)NCc2ccsc2C(=O)NC)c(C)n1.c1cc(O)ncn1 Cc1cc(=NC(=O)C(=O)N2CCN(C(=O)CCCc3cccs3)C(CO)C2)[nH]o1 N1(C(C2CN(C(N)=O)C2)=O)CCC2CC12C(=O)NCC(C1CC1)N(C)C c1(NC(C2C3(CC(C)OC3)C2)=O)cnc2ccc(C#N)cn12 N1(C(COC(C)(C)C)=O)CC2CC1C2NC(=O)CC1CCSCC1 N1(C(CS(CC)=O)=O)CCC2(CCC(NC(=O)CN3CCCNC3=O)C2)CC1 N(C1CN(C(C2C3CCC2(C)C3(C)C)=O)Cc2ccccc21)C(CSCC=C)=O C#Cc1cnn(CC(N2CC(C)(OCC(=O)NCC3(C)CC(C)C3)C2)=O)c1 c1(N2CC3CC3C2)nc2ccc(F)cc2s1.C=C(C)CC(C(=O)NC)OC.C(C)=O N1(C(c2c(CC)ncs2)=O)CCC(F)(C(=O)N(CCC(=O)OC)CC)CC1 Cc1cc2n(n1)CCN(C(=O)C1=C(F)CN(C(C3CCCOC3C)=O)CC1)C2 c1(SC)nc(N2CCCC(F)(C)C2)cc(C)n1.c1(C=O)csc(C(C)(C)C)n1.N C1(C(=O)NCCCCNC(C(C=CC)O)=O)CCCN(CC(C)C)C1 C(=O)(C1CC(=O)Nc2ncccc21)OCc1cncc(OC)c1 N1(C(C2N(CC)CCC2)=O)CCC(CCC(=O)NCC(O)C(C)(C)O)CC1 N1(C(Cc2cccc(C(C)C)c2)=O)CCC2CN(C(C3CCC(=O)N3)=O)CC12 C1(=CCNC(C2CC3CC3C2)=O)CCN(c2ccnc(-c3nccs3)n2)CC1 n1(CC)cc(NC2(c3nnnn3CC(F)F)CCCC2OC)ccc1=O C1(O)(C(=O)NC2CC(C(N(CC#C)CCF)=O)OCC2)CCOC1(C)C N1(C(Cc2cnc(C)s2)=O)CCCC(CCNC(=O)Cc2cnsc2)C1 N1(C2CC(C=O)C2)CCOCC1.CC(C)COCC(=O)NCC1CC1C C1(NC(=O)OC(C)(C)C)CCS(=O)(=O)C1C.C1C(C(=O)NC2CC2)N1 C1(CC(=O)NCC(C)N(C(=O)CN(c2ncccn2)C)C)CC2(CC2)CO1 Cc1nc(NC(C2CC2C(=O)Nc2ccc(Cl)c(C#N)c2)=O)ccc1[N+](=O)[O-] c1(OC)cc(C)c(C(N2CC(C)C2(C)C)C(=O)NCc2ccccc2)cn1 c1(C(N2CCC(NC(CSC)=O)C2(C)C)=O)ccc2c(n1)CCC(C)C2 c1(C(C(=O)NCC2CCN(C(c3cc(C)[nH]n3)=O)C2)(F)F)ccccc1F C(=O)(C1CCCc2scnc21)N(C1CCN(C(=O)Cc2sc(C)cc2C)C1)CC O=C1CN(C(C2CC(F)(F)C2)=O)C(C(N2CCC2CC2CC2)=O)CN1 N1(CC(N2CCC(C(C)CNC(=O)C=CBr)CC2)=O)OC(C)(C)CC1=O N1(C(CC(C)(C)C2CC2)=O)CC2CCC2(CNC(c2cnc(O)o2)=O)C1 C(=O)(C1Cc2c(Cl)cccc21)NC1CC(CNC(=O)CC2CCCC2(F)F)C1 N1(C(C(c2ccccc2)OC)=O)CCC2(CCCN2C(=O)C(O)CSC)C1 N1(C(C#C)=O)CCC2C1CCN2C(=O)CNC(c1cccnc1)=O Cc1ccc(=O)n(CC(=O)NCCC(C)NC(c2cccc(=O)n2C)=O)n1 c1(SC)nccc(=NCC2CCN(C(c3cc(Cl)cc(Cl)c3O)=O)CC2)[nH]1 N1(C(C(C)(C)CF)=O)C(C(=O)NC2CCN(CC3CC3)C2)C2CC(O)C1C2 N1(C(CCN(C)C(c2cc(C#N)cs2)=O)=O)CCCC2(C1)N=N2 C1(C(=O)NC(COC)C)(CCNC(C2CCC(OC)C2)=O)CCCC1 N1(C(C2C(CC)CCC2)=O)CCCC2(CCCN2C(=O)CCCC(OC)OC)C1 N1(C(C(Cc2ccc(C)cc2)C)=O)CC2(NC(=O)Cc3cc(C)ns3)CCC1C2 N1(C(C(C)(C)F)=O)CCC(CO)C(NC(c2cccc(SC(F)(F)F)c2)=O)C1 N1(C(C=CCC)=O)CCCN(C(c2nc(-c3cccs3)oc2C)=O)C(C(C)C)C1 N1(C(C(c2cn(C)c(=O)cc2)(F)F)=O)CCCC2(C1)CN(C(C1CC1(F)Cl)=O)C2 CCC(CC(=O)N1CC(C)C(C)(CNC(=O)CSc2nncn2C)C1)C(C)C O=CCCC(=O)NCC1CCC1.C12CCN(C1)C2=O.C1(C=O)CC1.C1CC1 Cc1ccc(-n2nc(Cc3cccc(Cl)c3)nc2C2CC2F)c(C)c1 C(CN=c1cc(C)[nH]c(=NCCCCCF)[nH]1)OC c1(OCC#C)ccc(C(=O)NCC(CCCC)NC(C2CC2(C)Br)=O)cc1 C1(NC(c2cn(CC)nc2)=O)C2CC1CN(C(c1cc(C(C)C)ccc1F)=O)C2 O=Cc1ccncc1-c1ccc(-c2nccn2C2CC3CNC2C3)c(F)c1 C=C(C)CN=C(NCC1CC2CCC(C1)O2)N1CCn2c(COC)nnc2C1 C(=O)(C(F)CCC(C)C)N1CCC(CC=C)(C(=O)NCc2cccn2C)C1 c1(C=O)cnn2ccsc12.c1(C(=O)NCC2CC2)csc(C(F)(F)F)n1.N C#Cc1c[nH]nc1C(N1CC(O)CC1CNC(C1CCOC1C=C)=O)=O c1(C(N2CC(C)N(C(=O)COCC3CCOC3)CC2)=O)cccc2c1CNC2=O N1(C(C(C)(C)OC)=O)CCC2CC(NC(=O)CCc3c(C)noc3C)CCC2C1 C(=O)CC(O)CC(C)(C)C.N1(C(C(C)NC(N)=O)=O)CCC(C)C(F)(F)C1.N C1(NC(CCN(C(CSCC=C)=O)CC2CC2)=O)CCCOC1 CC(C)CCC(C(=O)NCc1cnc2n1CCC2)NC(C1C(C)C1C)=O C1(NC(=O)C=CI)CCC2CN(C(=O)CC3CNc4ccccc4O3)CCC2C1 S(=O)(=O)(c1ccc(C)s1)N1C(C=O)CCC1.c1(C(=O)OCC)nncs1.C c1(NC(C(=O)NCCCCCC2CCNCC2)=O)cc2n(n1)CCC2 c1(C(=O)NCc2ccc(C(=O)NCC=CC)s2)ccc2[nH]ccc2c1 N1(C(C2(CNC(C(CCC)NC(C)=O)=O)CC2)=O)CCC2CC1C(=O)O2 CC(c1ccccc1)=CC(=O)NC1CCC1NC(=O)C=Cc1cnn(C)c1 c1(NC(c2nccc(OC(C)C)c2)=O)ccc(S(C)=O)c(F)c1 c1(SC)ccc(Cl)c(C(=O)NC2CCCCC2C)c1.C(=O)C.[SH](C)(=O)=O CCCCC(CC)CC(=O)NC1CN(C(=O)Cn2nnnc2C)CC12CCC2 C#CCCCCCCC(=O)N1CC2CCC1CN2C(c1ccc2nccn2c1C)=O c1(CCC)cc(C(=O)NCC2CC(NC(=O)CS)C2)n[nH]1.c1ccccc1 CC1(C(=O)NC2(CO)CCCS(=O)(=O)C2)CC2CCC(C1)S2 C(C(=O)N(C)CC1CCOC1)(C(C)(C)C)NC(CSCC)=O N1(C(C(=O)NCCCSc2ccccc2)=O)CCCC(Sc2cccc(Cl)c2)C1 c1(C(=O)NC2C(NC(=O)CCc3cc(Cl)no3)CCC2)ccc2nnc(O)n2c1 C(=O)(C1CCCc2nn(C)cc21)N.C(=O)(C(F)C1CCC1)N(C)CCOCCC CCCC(C)(O)C(=O)N1CCC(C(C)(C)C)(CNC(C2(S)CCCCC2)=O)C1 C1(CC(=O)OC23CCC(C(=O)OC)C2C3)SC(N2CCCC2)=NC1=O C(C(C(=O)NCC1CC12CCN(C(C1CCCC1)=O)CC2)C(F)(F)F)OC CC1CC(C(=O)N2CCN(CC3CN(C(c4ccc(CO)nc4)=O)C3)CC2)=NO1 C1(CC=C)(NC(C2CCC(n3cc(CCOC)nn3)C2)=O)CCCC1 c1(C(=O)OC)cc(C(=O)NNC(=O)c2cccc(Br)c2)sc1S(N)(=O)=O CC1CCCC(=O)O1.C12(C(=O)OC(C)(C)C)CC(c3ccccc3)C1C2 C1(CC)CCCCC1C(N1CCC1Cn1cc(-c2ccc(OC)nc2)nn1)=O c1(OC)nc(N2CCC(NC(c3sc(CC4CC4)nc3C)=O)C2)cc(C)n1 Cc1cncc(C=CC(N2CC(C)CCC2CNC(c2ccc(F)s2)=O)=O)c1 C1(C#N)(C=O)CCSCC1.Cc1onc(C2CC2)c1C(=O)NC1CC2CC2C1.N N1(C(c2cncc(O)c2)=O)CC2CCN(C(c3cncc(O)c3)=O)C2C1 c1(NCCc2c(C)noc2C)cccc(S(=O)(=O)NC(c2cn(C)nn2)=O)c1 C1(CNC(c2n[nH]c(C)c2C)=O)CCC(C)CN1C(=O)CCN1CCC1 C1(NC(C=NOC)=O)CC2C(NC(=O)CC(C)C3CCCC3)C2C1 N1(C(C(CC)SC)=O)C2CCC1CN(C(=O)COc1c(C)cccc1Cl)C2 N1(C(=O)CCCn2ccnc2)CCC2(CCCC2CN=c2cc(Cl)nc[nH]2)CC1 N1(C(C(n2cc(Cl)cn2)C)=O)CCCC(CNC(=O)CS(C)(=O)=O)CC1 C1(NC(C=C2CCN(C)CC2)=O)CC(NC(c2cnn(C)n2)=O)C12CCC2 C1(C(N2CCC3(N(C(CSCC=C)=O)CCC3)C2)=O)CSC(c2ccccc2)=N1 C1(C(=O)NCC2(NC(CN3C(=O)CN(C)C3=O)=O)CC2)CC2COCCN2C1 CN1CCCC(C(C)(C)C(N2CCC(F)(C)C2)=O)C1.C1(CC=O)CC(F)(F)C1 C1(C(=O)N)COC2(C1)CN(C(=O)C(O)CCN(C)C)C2.C1(OC)CN(C)CC1 N1(C(c2c(C)scn2)=O)C(C(=O)NC(C)C(=O)N2CCCC2)CC2CC12 n1(CC(N2C(CN(C(CC3C(CC)C3)=O)C)CCC2)=O)nc(C)oc1=O C1(C(N2CC(NC(c3ncn(C(C)C)c3)=O)C(CO)C2)=O)CCOC(=O)CC1 N#Cc1cc(C(N2CCCCC2C(=O)Nc2cc(F)c(Cl)cc2F)=O)ccc1Br N1(C(C(CC)OCC)=O)CC(CC(=O)NCC(C)C(=O)OCC)CC1(C)C C1(NC(CCC=C(C)C)=O)CCC12CCCN(C(c1cn(C)[nH]c1=N)=O)C2 c1(NC2CCN(C(C3(CC)CCOCC3)=O)C2)nnc2c(c1C#N)CCCC2 C1(NC(COCCCC(C)C)=O)CC2CN(C(c3cccc(N)c3)=O)CC12 c1(CC)ccc(O)c(C(=O)N(CCCNC(=O)C(N2CCOCC2)C)CC)c1 C(=O)(C1Cc2ccccc21)NC1CN(C(c2ncn(C(C)(C)C)c2)=O)C(CO)C1 c1(N(C(C(C2CCCC2)OC)C(=O)NCC(C)C)C)ccc(F)c(F)c1 C1(CC(=O)NCC2C(NC(C(C)=CC3CC3)=O)C2)CC(C)(C)CO1 c1(C(=O)NC(C)C(c2c(F)cccc2F)O)cc(Br)cc2[nH]ncc12 c1(C(=O)NCCC2(C(N(CC)CC3(O)CCC3)=O)CC2)scnc1C Cc1cc(OCC(=O)NC2CC2NC(c2cc(CO)n(C)n2)=O)ccc1Cl CC(C)C(C)(CNC(=O)CC1CCN1C(=O)CCC(C)(C)N(C)C)C(C)C C1CCC(C(=O)N(C(C)C)C)CC1.C(C)(C)C(F)(F)F.C(=O)C.CC=O.N C=C(C)C1CN(C(=O)CCCCN(C(=O)CCC2OCCO2)C)CCO1 C12(C(=O)NC(C3(O)CCN(c4nccc(OCC)n4)C3)C)CC=CC(C1)OC2 C1(OC)CN(C(=O)C(C2CCC(O)CC2)(C)C)CC1NC(c1cc(Cl)cnn1)=O c1(OC)ncc(F)c(=NC(=O)C2CC(C)CN2Cc2ccc(Cl)cc2OC)[nH]1 C(=O)(CS(=O)(=O)C1CC1)NCC1CCN(C(c2c(C)nc(CO)s2)=O)C1 N1(C(C2(C)CCN(C(C)=O)C2)=O)CC2CC(C1)C2N=c1cncc(Cl)[nH]1 c1(C(=O)N)cnc(O)cc1C(F)(F)F.N1(C(CC(C)C2CC2)=O)CCOC(C)C1 C#CC1CC2(CC2)CN1C(=O)C(O)CNC(c1ccn(CC)n1)=O c1(NC)cc(Cl)ccc1C(=O)NCC1CCCC1.C1(C=O)CC(N(C)C)C1 C1(NC(c2ccc(C(C)C)nc2)=O)CC(NC(C2CC=CC(O)C2)=O)C12CCC2 C=Cn1nncc1C(N1CCCC(CCNC(=O)C(F)=CCC)C1)=O Cc1cccc2[nH]c(C(=O)NCC3CCN(C(C4CCC5CCC4O5)=O)C3)cc12 C(CC1=CCN(c2ncc(O)cn2)CC1)NC(c1cn(CC)nn1)=O C(=O)(CS(=O)(=O)C1CCCC1)N1CC2(C(NC(C3CC(C)(C)C3)=O)CCS2)C1 c1(CC)cc(C(=O)NCC(O)CN(C)C(C2CCCS2)=O)cc(Cl)c1 c1(CN2CCCC(CNC(c3ccc([N+](=O)[O-])o3)=O)C2)cc(Cl)ncc1Cl n1(CCCC)nc(Cc2cccc(F)c2)nc1-c1ccc(Br)cc1 CCC1=C(C(=O)NCC2CC2CNC(=O)Cc2conc2C)CCCO1 c1(C(=O)NCCC2CC(NC(c3nccc(C)n3)=O)C2)cccn2c(C)cnc12 c1(C(=O)NCC(=C)Br)ccc2c(=O)ccoc2c1 Cc1cc2nc(N3CCOCC(CNC(C4(C)CCCO4)=O)C3)cc(=O)n2o1 c1(C(N2CC(NC(C3(CO)CCC3)=O)CC(C)C2)=O)cc2ccc(F)cc2s1 C(=O)(C(C)(O)CC(C)C)NCc1c(C(=O)NC(CCC)C(C)(C)C)cco1 N1(C(Cc2c(C)nc(Cl)cc2)=O)CC2CCCN(C(=O)CC3CCCOC3)C2C1 c1(CC)cc(C(N2CCN(C(=O)CCc3ncc(C)[nH]3)C(CC)C2)=O)cc(O)n1 c1(C=O)ccc(Cl)cc1C(F)F.Cc1c(C(=O)NC2CCC(C)C2)cnn1C.N C(=O)(C(CC(F)F)NC(C1CN2CCN1CC2)=O)N1CC(CCC)C(CO)C1 c1(C(=O)NC23CN(C(C4(OC)CC4)=O)C(C2)C3)cccc2oc(C)nc12 Cc1nc(N2CCC(CF)(NC(=O)C(C)C3CCC3)C2)ncc1Br CCCC(C(=O)NC1CCC(NC(c2cc3n(n2)CCOC3)=O)CC1)C(C)C C12(NC(CCC(=O)NC)=O)CCC(C(=O)Nc3cscc3SC)(CC1)C2 c1(NCC(C(C)O)C)ccc(S(=O)(=O)NCCCSC(F)(F)F)c(Br)c1 C(C(CC(C)C)C(=O)N1Cc2ccccc2CO1)NC(C(CCC)OC)=O C1(CC(N2CCC(OCC)CC2)=O)CC2CCC1C2.C12(C(=O)N)CCC(CC1)C2 O(NC(=O)C(CCNC(=O)CC=C(C)C)OC(C)=O)C(COC)COC c1(C(N2CC(C(=O)NCC(=O)N(C)C)C(O)CC2)=O)cc2ccc(Cl)nc2[nH]1 C1(CNC(c2cnc(OC)s2)=O)C(C)CCN1C(=O)CO.c1ccccc1Cl C1(NC(C(CO)NC(N)=O)=O)CN(C(c2cc(Cl)ccc2N)=O)CCC1O CC1=C(C(=O)NC2CCC(NC(=O)CCCCCc3cccc(O)c3)C2)CCO1 c1(C(C)NC(c2c(NC(CC3C(CC)C3)=O)nccn2)=O)c(C)cccc1F C(=O)(C(O)P(C)(C)=O)N1C(C2CC2)CCC1.Cc1oc(C(C)C)cc1C=O.N C1(NC(CSC(C)(C)C)=O)CN(C(=O)Cc2cnccn2)C2(CCCCCC2)C1 c1(OC)ccc(-c2cc(-c3nc(-c4cn(C5CCOCC5)nn4)no3)n[nH]2)cc1 N1(C(C2C(CC)N(C)CC2)=O)CCCCCC1C(=O)NC(CCF)C(=O)OC C(CN=c1[nH]c(=NCCc2ccsc2)[nH]c2c1CCCC2)N(C1CC1)CC CCCCC(CC(=O)NCC1OCCC1(C)C)NC(=O)CCN1CCOCC1 C(=O)(C(CNC(=O)CCCOC(C)(C)C)CC(C)C)NCC(CC)CO N1(C(c2cc(C)oc2C(F)(F)F)=O)C2CCC1CN(C(C1CCC1)=O)CC2 N1(C(C2CCCN(Cc3n(COC)ccn3)C2)=O)CCC(C)(C)CC1 N1(C(C2CN(S(CC)(=O)=O)C2)=O)CCCC12CCCCC2.c1(C(=O)N)coc(Cl)n1 C(CN=c1ccc(S(=O)(=O)N(CC(O)CF)C)c[nH]1)N(C)C(C1CCOC1)=O C(=O)CN=S(C)(C)=O.C1(CC#C)(C(=O)NC(C)Cc2ccccc2)CCCO1 c1(C=O)ccccc1Cl.c1(C(C)N(C(=O)CN2CC(CC)C2)C)cnn(C)c1.N C1(CNC(C2(CC)CC2(F)F)=O)CC2CCC1N(C(c1ocnc1C)=O)C2.C C(N=C1NS(=O)(=O)c2ccccc21)C1CC(N2CC(=O)Nc3c2ccc(F)c3)C1 C(=O)(C(C)CC(C)(C)C)NC(CC=C)CC(=O)NCCNC(=O)C(C)(C)C N1(C(C(COCC)C)=O)CC(NC(=O)Cc2ncc(C)o2)CC12CCCC2 C=CC(C)(CC)C(=O)NC(C)C1CCC1.c1(CC(=O)N)ccn(CC(C)C)n1 C1(CC(=O)NCCC(C)(C)NC(C(CC)n2cncn2)=O)CC2CCC(C1)N2C C(c1cc(C)no1)=CC(=O)N.C(=O)(CC(C)NC(=O)CCC1CC1)OC c1(C(NCC)=O)cccc2c1OCC2.n1(CC=O)ccc(C2CC2)n1.C1CC1.N C(=O)(C(C)(C)C(F)c1ccccc1)NCC(C)(CO)NC(C=C(C)C)=O N1(C(CSCC=C)=O)CCC2(CCN(C(c3cc4cccn4cn3)=O)C2)C1 C1(C(=O)OC)CN(c2nnnn2CCC23CCC(CO2)C3)CCC1(F)F N1(C(C(F)=CCC)=O)CCC(C)(C)CC1C(=O)NC1(CF)CC1 c1(C(N2CC3C(NC(C(COC)(C)OC)=O)C3C2)=O)cc(Cl)ncc1O C(Cc1ccoc1)(C(=O)N(C)Cc1cocn1)NC(C(C)n1cccc1)=O Cc1cc(C#N)c(O)nc1C(=O)NCC1CCC(NC(=O)CCC(C)C)C1 N1(C(C2CC2C2CC2)C(=O)NCC)CCC(C(c2cccs2)=O)CC1 CC1OC(=O)NC1C(N1CC(O)(CCNC(C2CC3(CC3)C2)=O)C1)=O N1(CC(=O)NCCC2(O)CCN(C(c3ocnc3C(F)F)=O)C2)CCCCC1=O CC(C)C(C)(C(N)=O)NC(=O)CCN(C)C(C1CCC2(CCC2)C1)=O c1(C(N2CC(CNC(=O)C(=O)Nc3ccccc3)OCC2)=O)ncc(F)cc1F C1(C(=O)NC)CN(C(C2CC(O)C2)=O)CCC1(F)F.c1cc(-c2cccs2)on1 c1(C(C)OC)nc(N(C(C)CNC(C2C3CCCC23)=O)C)cc(Cl)n1 C(=O)C(C(C)C)c1ccc(C)cc1.C(=O)(CN(C)C(C)=O)N(CC)CC C(=O)(CC(C)C(=O)N1CCC(C(=O)NCCCC(C)(C)C)(CF)C1)OC c1(CNC(CC(CNC(CC2C(C)=NNC2=O)=O)C)=O)c(F)cncc1F C(c1cc(Cl)ccc1Cl)=CC(N1CCC(CNC(C2C(C)C2(F)F)=O)C1)=O c1(C(N(CCCNC(CC(=C)Br)=O)CC)=O)nccc(C)n1 O=C(C1=C(Cl)CCOC1)NCC1C2CN(C(=O)Cc3ccnc(O)c3)CC12 N1(Cc2ncc(C)nc2)CCCC(C)(C(=O)N(C)C(c2cccs2)C2CC2)C1 C1(C(=O)N)CN(C(=O)C(C)(C)CO)CC1C1CC1.C(C)(C)(C1(C)CC1)OC CCCCCCC(CC)C(=O)NCC(CCCC)NC(=O)C(c1ccc(Cl)s1)C C1(C)(C(=O)NCCNC(C2N(C(C)=O)CCC2)=O)CC2CC2C1.C1CC1 CCC(CNC(C1(C)CCC1)=O)N(C(=O)CCOCCOC)C CC(C1Cc2ccccc21)NCc1cnc(C(F)F)s1 Cc1cc(NC(c2c(C)ncn2O)=O)ccc1NC(=O)CCCc1ccncc1 N1(C(C(CCC)OC)=O)CC(S(=O)(=O)N2CCN(C(=O)C(C#N)CCC)CC2)C1 C(=O)(CC1=CCN(C)CC1)N.C(C(=O)NC1CCC1)(C(C)C)NC(=O)OC C1(C(=O)NC2CCN(CC(=C)Br)C2)CC(=O)N(CC)C1 C1(C)(COC)CN(c2ncnc(NCC3SCCS3)c2C)CCO1 C1(CNC(C(C=C)(C)C)=O)C2CCC(C2)N1C(c1cccc(Br)c1C)=O C=C(C)CCCC(=O)N(CCNC(c1cnc([N+](=O)[O-])s1)=O)C1CC1 Cc1c(N(C)C(C2(F)CCN(C(c3csc(F)c3)=O)C2)=O)cccc1F c1(C=O)cccc2nn(C)cc12.C1(C(=O)NCCC2CCCC2)(CC)COC1.N Cc1cc(C)c(C(N2CCC=C(CNC(=O)Cn3cnnn3)C2)=O)c(C)c1 c1(C(N2CC3(CCC3)C2c2ccco2)C(=O)NCCCSC)nc(Cl)ccc1Br CC1CN(C(=O)COCc2ncno2)C(C)CN1C(c1cn(C)[nH]c1=N)=O.C C1(C(=O)NC(COC)CNC(C2CC(OC3CC3)C2)=O)CC=CCO1 N1(c2ncc(C)c(C)n2)CCC2CC(C(=O)NC(C)Cc3ccncc3)C2C1 c1(C(N(CCCNC(=O)CCc2ccccc2F)CC)=O)ncc2n1CCCC2 CCCCCCCC(=O)N1CCCCCC1CNC(C1CCC(C)CC1)=O c1(CC(C)C)nc2cccc(C(=O)NCCC3CC3)c2[nH]1.C1(C=O)CCCO1.N C1(C(N2CC(CNC(C(CC)N3CCCC3=O)=O)OCC2)=O)C(F)(F)C12CCC2 C1(C(=O)NC(C=C)COC)(NC(c2cc[nH]c2CC)=O)CC1(C)C CCCCCCC(C)(C)C(=O)NCC(C)(CC)NC(=O)CC(C)C(=O)OC C1(N(C(c2cc(O)cs2)=O)CC)CCN(C(=O)CC2(CO)CCCC2)CC1 c1(C(N2C3(C(N(CCC=C)CC)=O)CC3CC2)=O)cc[nH]c2nccc1-2 N=c1cc[nH]cc1C(=O)NC1CCC1NC(c1ccnc(C2CCCC2)n1)=O C(=O)(CC(C)(C)CC(=O)NC1CCC1NC(C1(CF)CC1)=O)OC Cc1nn(CC(N2CC(C)C3(CC3)C2)=O)c(C)c1[N+](=O)[O-].C(=O)C.C(C)C.N CN=c1[nH]cc(C(=O)N(C)CC2CCCCC2)o1.N1(CC=O)C(=O)CNC1=O.N c1(N2CCC(C#N)(NC(c3ccc(Cl)c(C)c3Cl)=O)C2)ncc2cc(Br)ccc2n1 c1(C(=O)NCCCN(C)C(C23CC(O)C2C3)=O)ccnc2ccnn12 CCCCS(=O)(=O)NC(C)C(=O)NC(C)(C)CNC(c1n[nH]cc1Cl)=O c1(C(=O)NC)cc(C=O)on1.C(=O)C(O)C.c1ccco1.CCC1CC1 c1(C(=O)OCC)ccc(C)c(NCc2nnc(C3CCC3)n2C)c1 c1(C=O)cc2ccsc2c(O)n1.N1(C(CN(C)C(N)=O)=O)CC(C)CC1(C)C.N C=CCC(C)(C)CCC(N1CC(O)(c2cn(-c3cnc(OC)n3C)nn2)C1)=O CCC(CC)(C(=O)N1CCC(C(F)C(=O)NCC2(C(F)(F)F)CC2)C1)OC C12(C(N)=O)CCCC1(C(N1CCCCC1CNC(C1CCC1)=O)=O)C2 C(C(C)C(C)C(=O)NC1CC12CC(NC(c1cc(C(N)=O)co1)=O)C2)OC C(=O)(C(CC(C)C)ONC(=O)C(C)(c1ccccc1)OC)OC c1(NC(C2CC2C(=O)Nc2cc(Cl)ccc2CO)=O)ccc2occc2c1 CCC(CC(=O)N1CCC(NC(=O)C2CCc3snnc32)C1C)CC(C)C N1(C(c2cc(CCC)c(C)s2)=O)CCN(C(c2cc(C)nn2C)=O)C(CO)C1 C(=O)(C1=CCCOC1)NC1CC(NC(c2n(CC)nc(C(C)C)c2)=O)C1 N1(C(C(C2CCCC2)NC(c2cc[n+]([O-])cc2)=O)=O)CCC(O)C(O)C1 N1(C(COCCC)=O)C2CC1CN(C(C1C(C=C(C)C)C1(C)C)=O)C2 C(=O)(CCCC(C)C)NC(Cc1cn(CC(c2cccc(C)c2)O)nn1)C(=O)O C1(N(C(C(COCC)NC(c2sccc2OC)=O)=O)C)CCOC(C)(C)C1 N1(C(CCC=CCC=C)=O)CCCC2(NC(c3nccc(C)c3F)=O)CCCC12 CC(C)CC(C(=O)NC1CC2CC1CC2CO)ONC(=O)CC1CC2CCC1O2 CC(C)(CC(F)F)C(=O)NCC1CC(C)C1.C1(C=O)CCS(=O)(=O)C1.N N1(C(C2CC3(C2)CC3F)=O)CCC2C(C1)CN2C(c1ccc2c(c1)OCC2)=O N1(C(C=COCC)=O)CCC(NC(C2(CO)CCCCC2)=O)C1C(C)C C=CCC(C(=O)NCCc1cc(C(=O)NC2CC(CC(N)=O)C2)no1)OC c1(C(N2CCC(C)(NC(C3CCC(F)C3)=O)CC2)=O)cn2ccccc2n1 CC(CC(=O)NC(Cc1ccoc1)C(=O)NCC(CO)N(C)C)C(C)(C)C C(=O)(C1=CC(C)(C)C1)N.c1(COC)nc(CC(=O)NCC(C)(O)C)cs1 c1(CC(=O)NC2CN(C(c3c(C)c[nH]n3)=O)C(C)C2)c(O)nc(=N)[nH]c1C CC1(C)OCC2CC12C(N1CCN(C(=O)C)CC1)=O.C1(C#N)(C(=O)N)CCC1 C1CC2(CC2)CN1C(c1c[nH]c(C(N)=O)c1)=O.CC(C(C)(C)C)=CC(=O)N c1(OC)ccncc1NC(C1(NC(C2CC=CCC2C)=O)CCSC1)=O c1(NC(C)=O)ccc(OC(=O)CC2NC(=O)NC2=O)c(C)c1 c1(C(=O)NC2C(OC)CN(C(=O)CCc3cn(C)nn3)C2)nc(C)n(C)c1C C1(CC)CN(C(c2ccc(C(N)=O)cn2)=O)CCO1.C1(C(=O)N)(OC)CCSC1 C(C(O)C(C)C(=O)OCC1(c2cc(Cl)ccc2Cl)CCCC1)NC N1(C(C(COC)N(C)C)=O)CCCC(NC(=O)Cc2cccn2C)CC1 C1(C(=O)N)OC2CCC1C2.c1(C(=O)NCC(N(C)C)C2CC2)coc(C)c1 C12(O)CCCN(C1)C(=O)C=CC2.c1sc(C(F)(F)F)cc1Br.C(C)(C)C.N c1(C(c2nnnn2CCC2CC2)NCC=C)cccc2sccc12 Cc1scc(C(=O)NCC2(C(=O)Nc3cnn(CC(N)=O)c3)CCCC2)c1C C1(NC(c2c(CC)[nH]c(=N)s2)=O)COC2(C1)CN(C(=O)CC1COCCO1)C2 c1(C(=O)N)cnc2c(c1)COC2.c1(C(C)C)ccsc1C(=O)NC(C)C1CC1 N1(C(CC=CCC)=O)CCC2(NC(=O)CCn3c(O)nnc3O)CC2C1 N1(C(c2cc(NCCN(C)C3CC3)cc(Br)c2)=O)CC(N)CC12CCOCC2 N1(C(CC=CC=C)=O)Cc2occ(C(N3CC4CCC=CC34)=O)c2C1 c1(C(N(CCNC(C(CC)n2cncn2)=O)C2CC2)=O)c(C)ccc(F)c1N C1(N(C(Cc2ncc(CC)[nH]2)=O)C)CCCN(C(=O)Cc2ccn(CC)n2)C1 C1(COC)Cc2cc(NC(C3(O)CC(C)CCC3C)=O)ccc2O1 c1(OC)cccc(C(N2CCCC2(C)C(=O)NCC2(CF)CCC2)=O)n1 N1(C(c2n[nH]c(C)c2C)C(=O)NCC=C)CCN(C(=O)C(F)(F)F)C(C)C1 C1(C2CC2)(NC(CC(C)(C)C)=O)CCN(C(=O)Cc2ccccc2F)C1 CCCC(CC)N=c1[nH]c(=NCC(C)Cn2cccn2)[nH]c2ncn(CC3CC3)c12 C(C(C)C(C)C(=O)NC1CC(F)(CNC(=O)CN2CCCCC2)C1)OC c1(N(CC(CCC)C)C)nc(N(C)Cc2nn(C)nc2Br)nc2c1ncn2C C=C(Br)CCC(=O)NC(C1CCCC1)CNC(=O)CC(C)(C)C C12(CC)CC1CN(C(C1(NC(C3CCCOCC3)=O)CSC1)=O)C2 N1(C(CCCCN(C)C)=O)CC2CCC(N=c3nc(C(C)(C)C)[nH]s3)C2C1 c1(C2C(C(N3CC4CC(O)CC4C3)=O)CC=CC2)nc2ccccc2s1 c1(N2C(CNC(c3c(C)cc(F)cc3)=O)CCCC2)ccnc2ncnn12 C1(C(=O)NC(COC)(C)C)CCC2COCCC2C1 c1(SC)csc(=Nc2cnn(C)c2)n1C1CCCCC1C(c1ccccc1C)=O c1(C(=O)NCC2CC(NC(c3ccc(F)nc3)=O)C2)cc2ccc(O)cc2[nH]1 N1(C(CCC(=C)C)=O)CCCC(C2CCCN(C(c3cc(OC)cs3)=O)C2)C1 N1(C(c2c(C)nc(O)s2)=O)CC2(CC(C(N3CCCCC3C)=O)CO2)C1 c1(C(=O)NC2CCC(C(=O)Nc3nc(Br)cs3)CC2)ccc2c(n1)OCCO2 N1(C(CC(c2ccccc2F)C)=O)CCCC1(C)CNC(=O)COc1cn[nH]c1 N1(C(c2c(C)oc(C(C)(C)C)c2)=O)CCN(C(c2cnc[nH]c2=N)=O)CC1C CC1(C)CC(CNC(=O)C2=NOCC2)N(C(=O)C2=COCC2)C1 c1(OC)cc(CNC(=O)C(=O)NCc2csc(C)n2)ncn1.C1CCNC1 c1(C(=O)NCC2C(C(F)(F)F)CN(C(C=CSC)=O)C2)cc(F)ncc1C N1(C(C(n2c(C)ccn2)C)=O)CCC(CF)(NC(=O)COC2CCCC2)C1 N1(C(Cc2c(CC)con2)=O)CCC(C(=O)NCCc2cscn2)C1(C)C N1(C(C=C(C)c2ccccc2)=O)CC(NC(C2CCN(C)C2=O)=O)C2(CCC2)C1 c1(NC(C2N(c3nc(OC)c(C#N)cn3)C(C)CC2)=O)cnc2ccc(Br)cc2c1 CCC(CNC(=O)C(C)Cn1ccnc1)(CC)NC(c1cc(C)sn1)=O c1(C=O)ccc(Cl)c(Cl)c1C.c1(C(=O)OC)cn(CC(N2CC(C)C2)=O)nn1.N N1(C(C=NOC)=O)CC(NC(=O)Cc2ccc(-n3nc(C)cc3C)cc2)CC1C C(CC(C)C(=O)NCC1CC1CNC(=O)CC1(O)CCOCC1)=CC c1(OC(C)C)cnccc1C(N1CC(N(C(=O)Cc2ccco2)C)C(O)C1)=O c1(C(=O)NCC(CNC(C(C)O)=O)C)ccc(C(F)(F)F)[nH]1 c1(C(=O)NC(CN(C(C(C(C)C)C(C)C)=O)C)C)cc(F)cc2nccnc12 C(=O)(NN=c1cc[nH]cc1F)c1c(O)nn(C)c1C(F)(F)F c1(CC=O)cc(S(N)(=O)=O)ccc1.c1(CC)ccc(C(=O)NC(C)C)[nH]1 c1(C(=O)NCC(C2N(C(C(C(C)C)C#N)=O)CCC2)(C)C)cnc2occc2c1 C1(NC(CCN(CC=C)C(c2ccnn2CCC)=O)=O)C(O)CC1O C#Cc1cnn(C)c1C(N1CC(C(=O)NCCC2CCC(C)C2)(SC)C1)=O CC1=C(C(=O)N2CCC3(C2)CN(C(C2(n4nccn4)CC2)=O)C3)COCC1 Cc1c(C(N2CCOCC2CNC(c2ncc(Br)cn2)=O)=O)cnn1CCO C1(NC(c2cc(C)n(C)n2)=O)CC2CN(C(C3CCC(C)CC3)=O)CC2C1 CC1(C)CCC(NC(c2cccnc2C)=O)C1.C1(C=O)CCCN1C(N)=O.N c1(C(C)O)ccc(-c2ccnc(SCc3ccccc3Cl)c2)cc1 C1(CNC(c2c(SC)cco2)=O)CN(C(c2nc(C3CC3)cs2)=O)CCN1C C(c1cnn(C)c1C)=CC(N1CC2C(CNC(CCc3nc(C)sc3)=O)(C2)C1)=O c1(OC)cncc(Br)c1C(=O)NC1CCC1.C1(C(=O)N)CCC(C(N)=O)O1 S(=O)(=O)(c1cccc(N2CC3CC2CO3)n1)N1CCC(C)(CN(C)C)CC1 C1(C(N(C(c2ccccc2)CNC(C(C(C)C)O)=O)C)=O)CC12CCC(=O)CC2 c1(CN2CCC(CNC(CCS(=O)(=O)N(C)C)=O)C2)ccc2ccccc2c1 C(CCC(N)=O)(C(=O)NCCCN1CCCC1C)n1cc(COCC)nn1 N1(C(c2c(CNC(Cc3c(C)nccc3)=O)ccs2)=O)CCC12CCCSC2 C1(C(=O)NC(C(C)(C)C)CO)CC(O)CCN1Cc1cccc(C(=O)O)c1F N1(C(c2ccc(N)c(C)c2Cl)=O)CCCC2(NC(c3cccs3)=O)CCCC12 CC12CCC1(C)CN(C(C1CN(C(c3cccc(F)c3)=O)CC13CCC3)=O)C2 C#CCC(C)(C)C(=O)N1CCC(N(C(c2ccn(C)n2)=O)CC2CC2)CC1.O CN1CCOC(C(=O)NCCC2CN(C(C3CCC(C(C)(C)C)CC3)=O)C2)C1=O Cn1cc(C(F)(F)F)cc(NC(c2cccc(N3C(=O)CCC3=O)c2)=O)c1=O C1(CN(C(=O)CC2CC3(CC3)C2)C)CN(C(C2CCOC2(C)C)=O)CCO1 C1(C(=O)NCC2(COC)COC2)CCCC1NC(C1CC1F)=O c1(C(=O)NC(C2CCCN(C(=O)C3=COCCC3)C2)C)cnc2c(F)cccn12 C(=O)(C(C)C(C)(F)F)N(CC(CC)NC(=O)Cc1cnccc1Cl)CC C1(NC(C(c2ccc(F)cc2)C)=O)CCC2CCN(C(=O)C(C)(C)CO)C1C2 C1(N(C)C(c2cnc(S)[nH]2)=O)CN(C(c2cnco2)=O)CCC1O C(=O)(C(CCC1(C)CC1)N(C(c1cccc(Cl)c1)COC)C)NCCOC N1(C(C(=O)NC)C)CCN(C(=O)CCN2CCCCC2)CC1 C=CCC(C(=O)OCCc1cn(CC(=O)NCCC)nn1)c1ccccc1 c1(OC)cc2[nH]nc(C(N3CCCCC3CN(C(=O)CSC)C)=O)c2cc1OC Cc1nc(NCc2ccc(O)c(C)c2)cc(NC2CCCN(C)C2)n1 Cc1nc2cc(C(N3CCSCC3CCNC(=O)C(F)=CC3CC3)=O)cnc2s1 c1(C(N(C(C2CCN(C)CC2)C)C)=O)cc2ccc(Br)cn2n1 Cc1ncc(Cl)cc1CC(=O)NC(c1ccccc1)CNC(=O)Cc1cc[nH]n1 C1(c2cn(C(CNC(c3cc(C)c(C)s3)=O)C)nn2)CCCS(=O)(=O)C1 c1(C(=O)NC(C(C)NC(C2(CC(C)C)CC2)=O)CO)cccc2cc[nH]c12 N1(C(c2cc(C)oc2C)=O)CCC(O)C(NC(c2cn(C3CCC3)nn2)=O)C1 C1(OC)(OC)CC(C)(CNC(N2CCCC(CCN)C2)=O)C1 C1(CNC(CN(C(CN(CCC)C)=O)C)=O)CCN1C(C)(C)C N1(c2c(C)cccc2[N+](=O)[O-])CCC2(CCCN(C(c3ccsc3Cl)=O)C2)C1 C(c1cccc(Br)c1)=CC(N1CCC(CCNC(C2(CF)CCC2)=O)C1)=O C1(C(N2CC(C(N3C(COC)COCC3)=O)OCC2)=O)CC12CCOCC2 C(=O)(C(C)(CSC)NC(c1ccsc1C)=O)NCCC(=O)OC C1(CN(C(CN(C(C)=O)CC)=O)C)CCN(C(c2cc(C)on2)=O)CC1 C(N=c1[nH]c(=NCc2ccc(F)cc2C2CC2)c2[nH]ccc2[nH]1)c1c(C)nn[nH]1 CC1(C)CCC(C(=O)NCCc2cccc(-c3cccc(Cl)c3)c2)NC1 C(=O)(CCC(C)(C)NC(c1c[nH][nH]c1=N)=O)NCCC1CCN(C)C1 C(=O)C1=NOC(C(C)(C)C)C1.Cc1ccc(C(=O)NCC2(F)CCC2)o1.N c1(C(N2CC(F)(CNC(C(COC)N(C)C)=O)C2)=O)[nH]nc2c1COC2(C)C N1(C(CC(C)C2CC2)=O)CCCN(C(=O)C(C)OC2CCCCCC2)CCC1 c1(CC(N2CCC(C(C)NC(CCC#C)=O)C2)=O)c(Cl)ccc(O)c1Cl C(CN=c1[nH]c(N2CCC(C)(C)C2)nc2c1CSC2)(C(F)(F)F)OC C1(NC(c2cnc3sccn23)=O)CC(O)CN(C(c2nc(Cl)cs2)=O)C1 C(=O)C1=CC2(CCOC2)C1.C12(C(N3CC(C)(C)C3)=O)CC3CC(CC(C3)C1)C2 N1(C(C(CCC)C)=O)CCC2(CCN(C(C)=O)C2)C1 C1(C(N(C(C)C(=O)NC2CSC2)C2CC2)=O)CS(=O)(=O)C1 C1(NC(c2ccc(CC)s2)=O)CN(C(=O)C(CO)NC(N)=O)CCC1C C1(C#N)(OC)CC(C(=O)NS(=O)(=O)CCC2CC2)C1 c1(CCC)c(-c2nc(C3CC3C3CCCCC3)no2)nnn1COC N1(C(c2onc(C)n2)C)CCC(C)C(NC(=O)CCc2c(C)noc2Cl)C1 C1(C(N2C(C)CC(NC(c3ccc(O)cc3)=O)CC2)=O)CCc2ccccc2O1 C1(O)(CN(C)C(c2cc3n(n2)CCC3)=O)CCCN(C(c2cccc(F)c2)=O)C1 C(C(CC)(CC)NC(=O)C)NC(c1ccc(COC)s1)=O.c1nccn1C.S c1(OC)ccc(C=CC(=O)NC(C)CCCC)cc1.S(S(C)(=O)=O)CC=O c1(C(N(CCCNC(C2CC3(CC3)C2)=O)C2CC2)=O)ccc(Br)c(O)c1 c1(C(=O)NCC2CN(C(c3c(C)nsc3C)=O)C3C2C3)ccc(F)c(F)c1 C(C)(C(C)C(=O)N(C)Cc1nc(=O)o[nH]1)NC(COCCCC#C)=O CCCC(C(O)C(=O)NC1CC1c1ccn(C)n1)NC(=O)C=Cc1ccc[nH]1 c1(C(=O)NC2(CNC(C(C)C3CCC3)=O)CCC2)ccnc(C(C)(C)C)c1 c1(OC)ccc(C)c(C(N2CCCC(O)C2)=O)n1.c1(C(=O)N)csc(C2CC2)n1 CC1(C)CN(C(C2CC(=O)NC2(C)C)=O)CC(CNC(=O)C(O)C2CCC2)O1 N1(C(C2CCCCC2)C(=O)NCC(=C)C)CC2CCC(C1)N2C(C)C c1(C(N2C3CC(CNC(C(C)OCC)=O)C(C3)C2)=O)ccc2nccn2n1 CCCCCS(=O)(=O)CC(=O)NCC1CC1CNC(=O)CCS(=O)(=O)N O=C1Nc2ccccc2CCC1N1CCC2CCCC2C1 c1(C(N2CC(CCC)C2)=O)ccc(Cl)c(Cl)c1.C1(C(=O)N)CC(n2cccn2)C1 n1(C(C)C)cc(C(=O)NC(c2ccccc2)C(=O)NCC2CCC=CO2)cn1 c1(N(C(=O)C(=O)N(c2ccccc2)C2CCCNC2)C)cn(C)cn1 c1(OC)ccc(N(C)C(C2CCCC2C)=O)cc1.c1(C(=O)N)cnn(CCF)c1 c1(NC)cc(C(N2CCCC(CO)(NC(=O)C)C2)=O)cc(Cl)n1.CC(N)=O.S Cc1cc(C(=O)N(C)CCNC(=O)Cn2c(C)cc(O)cc2=O)ccc1C#N CC1(CNC(=O)C(O)Cc2ccccn2)CCN(C(=O)CCn2cccn2)CC1 n1(C(COC)C)cc(CSCC(=O)NC2CC2)nn1 C(=O)(C(C)CC(F)(F)F)NCC(CCCC)NC(c1ccc([N+](=O)[O-])o1)=O Cc1c(Br)cc(NC(C2C3CN(S(=O)(=O)CCBr)CC23)=O)cc1Br CCC(C(=O)NC1CCC1C)Oc1ccccc1.C(C(C)(C)C)=CC=O.N N1(C(C(N2CCC(C)CC2)=O)=O)CCC2(CCCN2C(C2COCC2(C)C)=O)C1 N1(C(Cc2cnc(C)s2)=O)CCC(C(=O)NCCC2CCC3CC23)CC1 Cc1nc2c(C(=O)NC3CCCC(NC(=O)CS(=O)(=O)C(C)C)C3)cccc2o1 c1(C(C(=O)NC)N(C(C)C(=O)OC)C)cc(OC)cc(C(=O)OC)c1 C1(NC(C(C2CC2)OC)=O)CN(C(=O)C(c2ccc(F)cc2)C)CC(C)(C)C1 c1(OC)nc(C)cc(=NC2CC3CCC2N(C(=O)C(C)C2CC2)C3)[nH]1 N1(C(c2n(C)ncc2Br)=O)CCC2(C1)CN(C(c1cc(F)c(Cl)cc1F)=O)C2 C1(OC)C(NC(=O)CCCN(C)C(c2cc(Cl)no2)=O)CC1(C)C c1(OC)ccc(F)cc1CCC(N1CCC(NC(C2C3CCN2CC3)=O)CC1)=O N1(C(C(c2ccoc2)NC(CN=[N+]=[N-])=O)=O)CCCC(F)C1 CCCCC(C(=O)NC(C12CCC(CC1)C2)C)NC(c1[nH]ccc1C)=O C12(CNC(C=C(C)c3ccco3)=O)CCCCC1N(C(=O)Cc1ccon1)CC2 Cc1cccc2[nH]cc(C(N3CC(NC(c4ccnc(Br)c4)=O)C(F)(F)C3)=O)c12 C1(O)(C(=O)NC(CC2CN(C(C(C)OCC=C)=O)C2)C)CCCC1 N1(C(C2CCN(C(C)=O)CC2)=O)CCC(NC(=O)CSC2CC2)C12CCC2 c1(CC(=O)NC(C(C)NC(C=CC)=O)CO)cccc2ncccc12 C1(C(=O)OC)CN(CCC2CC2)CC1C(=O)OC1(C(N)=O)CC1 C1(NC(C=CCCC)=O)Cc2ccccc2C1NC(=O)CCCC1(C)N=N1 c1(C(N(C2CN(C(c3n(CC=C)ccc3)=O)CC2F)C)=O)cnn2cnnc2c1 c1(C(c2n(C(C)C)nnn2)NCC2CCCOC2)cc(F)cc(I)c1 C1(CC)C(=O)N(C)CCN1C(c1sc(C)c(C)c1C)C(=O)NCC(F)F O=C(CC1=CCCC1)NCC(O)CNC(C1CC1c1ccccc1)=O N1(C(C)C)CC(NC(C2CCC(C(C)C)N2C(=O)CC2CCSC2)=O)C(C)C1 N1(C(C2C(CC)CCO2)=O)CCC=C(CNC(=O)C(C)n2cccn2)C1 c1(C=O)ccc2c(c1)NC(=O)CCC2.C1(C)CCC1.C(C(C)=CC(=O)N)OC CCCCC(O)CC(=O)NCCC(O)CNC(c1ccnn2ccnc12)=O CCCCCCNC(c1conc1C(C)NC(c1cc(C(C)C)no1)=O)=O C1(CNC(C2(CC)CC2)=O)CN(C(C2(C(C)(C)C)CCC2)=O)CC1O C1(C(C#C)C)CCN(C(C2CC23CC(NC(=O)C(=O)C2CCCC2)C3)=O)CC1 CC(C)C(O)C(F)(F)C(=O)NCC(C)(C)NC(=O)Cc1ccc(Cl)nc1 c1(C(N2CC(C)C(NC(C3CCCC(C)(C)O3)=O)C2)=O)cc([N+](=O)[O-])n[nH]1 C1(CC)CCCCC1OCC(=O)NCCCC.c1(C(=O)N)ccnc(C2CC2)n1 C(N=c1ccn2ncc(S(=O)(=O)NC(C)C(C)CO)c2[nH]1)c1c(C)ccnc1 C1(NC(C(C)CC2CCC2)=O)CN(C(C2CCC=CCC2)=O)CC(F)(F)C1 C1(OC)CCC(C(=O)NC2(C)CCC(C)C2)CC1.C12(CC(O)C1)C(=O)N2 C1(C(C)C)OCCC1CNC(=O)COCCNC(=O)CC(C)F c1(C(=O)NC(CC=C)CNC(=O)CCSCC)cnc(OC)c(C)c1 Cc1csc(=O)n1CCC(=O)NC1CC(CCNC(C2CCN(C)C2)=O)C1 CC(C)C(C)(O)C(=O)N(C)CCN(C(=O)CCc1cncc(O)c1)C C(C(C(=O)NC(C)Cc1cccn1C)n1ccnn1)OCC.OCP(C)(C)=O.C CCS(=O)(=O)CC(=O)N1CC(N(C)C(c2cccc(C)c2)=O)C1 C(CNC(c1n[nH]cc1)=O)(C(C)(C)C)OC.C(c1cnccn1)=CC=O.C N1(C(CC2CC(CC)C2)=O)CCCCC1CCC(=O)NCc1cnccc1C c1(C(=O)NC(C)CNC(c2cn3c(n2)SCC3)=O)cnc2c(c1)NCC2 N(C1CCOc2ccc(OC)cc21)C(C1(C=C)CCCCC1)=O c1(C(=O)N)ccc(C)cc1F.C(=O)(CCCC1CCC1)N(c1cnn(C)c1)CC Cc1ccc(C#N)c(NCC2C3CN(C(c4cccc(C5CC5)c4)=O)CC23)n1 N1(C(CC2CC(NC(C(C3CC3)SC)=O)C2)=O)CC(C)=CC(C)C1 c1(C(=O)NC2C(NC(c3n(C)nnc3)=O)CCCC2)cnc2c(F)cccc2c1 C#CCC(CC)NC(=O)CCN(CCCO)C(C1CC1(C)C(C)C)=O N1(Cc2ccc(C(=O)OC)o2)CCC(C)(C(N2CC(O)C2)=O)C1 c1(OC)cc(C(=O)NC2CC(C)CN(C(c3ncc(F)cc3N)=O)C2)cc(F)c1 C1CC2CCC1CC2.C1(C(=O)NC2CC2)CCC(C)O1.C1(F)(C=O)CC1.N c1(C(N2CCC(C)(NC(=O)C(=O)NCCC(N)=O)C2)=O)cccc2ccoc12 C1(NC(=O)CO)CCCC12CCN(C(C1CC13CC(F)(F)C3)=O)CC2 CCCCC(O)C(C)C(=O)NC(c1cccnc1)C(=O)NCc1cc(O)ccc1C c1(C(=O)NC(C)CCNC(=O)CCc2ccc[nH]2)cn(CC(N)=O)nn1 c1(C(=O)NCC2(c3nn[nH]n3)CC23CCC3)ccc([N+](=O)[O-])cc1Cl CC#CCCCC(=O)N1CCC(CCNC(C2CC(F)C(=O)N2)=O)C1 C1(N(CC#C)C(C2CC2Cl)=O)CCN(C(=O)Cc2ccnn2C)CC1 N1(C(C(CCC)C)=O)CCC(C)N(C(=O)Cc2cccc(CC)c2)CC1 c1nccc2ccccc12.C1(NC(C2C(C=C)C2)=O)CC2(C1)CC2NC(=O)C CC(C)C(F)(CNC(c1cn(C2CC2)cn1)=O)C(=O)N.C1CCC(F)(F)C1 CC(C)CCCN(C)C(C1CC(=O)N(c2cn[nH]c2)C1)=O.C(=O)(C(C)C(C)O)N N(C1CCCc2ccoc21)C(C1C2(CCN(C(c3c(C)nsc3)=O)C2)C1)=O C1(CN(C(=O)CN(C)C(C2CC2(C)C)=O)C)CC1(F)F c1(C=O)[nH]cc2c1CCC2.C1(N(C(C(C)OCC(C)C)=O)CC)CCCCC1.N N1(C(C(=O)NCCCOCC)C)CCN(Cc2cccc(OC)c2)CC1 CC(C(=O)N1CC2(CNC(=O)Cc3sc(O)nc3O)CC1CO2)C1=CCCC1 C(CCCCCO)(c1nnnn1CCN1CCOCC1)NCC1(C)COC1 C1(C(=O)NC2(CNC(C(CC)NCC)=O)CCOCC2)CCCC(=O)N1C.C Cc1[nH]nc(C(=O)NC2(CCNC(c3nscc3Br)=O)CCC2)c1O C(=O)(C1CCc2c[nH]nc21)NCC=CCNC(c1c(C)cccc1C(C)C)=O c1(C(=O)NCCCNC(C2CCCC2O)=O)cccc2occc12 Cc1cc(C(C)N(C)C(C2CC2C)=O)no1.C1(CCC(=O)N)CCC(=O)C1 C1(C#N)(C(N2CCC(CCOC)(NC(c3cccc(C)n3)=O)C2)=O)CCSCC1 c1(CN(C(C2CC(N)(C(=O)OC)C2)=O)Cc2cccs2)cc(C)ccc1C C1(C)CCC(=O)N1C.C1(C=O)C=CCN1C(=O)CC1CC(C)=NO1.COC N1(C(CNC(CC)=O)=O)CC(NC(c2cc(C)c(C)s2)=O)C(n2cccn2)C1 c1(C(=O)NCC(C)OC)ccccc1.c1(C=O)ccncc1.CCN(C)C.O CC(C)C(CCN(C)C(c1ncccc1C1CC1)=O)NC(c1cncs1)=O C1(NC(CC=CC)=O)CN(C(=O)CC2CCCC2)CC(C)(C)C1.C(C)=O.N CC(CC(=O)NC1CC(CCNC(C2CC2F)=O)C1)N(C)C c1(NC(C(=O)NCC(C)NC(=O)C=CS(C)=O)=O)ccc2c(c1)OCCO2 C1(C)(C(N(C2CN(C(=O)CC3CC(C(C)(C)C)C3)C2)C)=O)CCCCNC1=O Cc1cnn(CC(=O)NCCC2(O)CCCN(C(=O)CC(C)(C)C)C2)c(=O)c1 CC(C)(C)CC(=O)CNC1(c2cn(-c3cncc(F)c3)nn2)CCC1 Cn1nnnc1C(c1ccns1)NC1CC(CCF)C1 C(C(=O)N=c1cnn(C2CC2)[nH]1)NCc1ccc(CS(=O)(=O)N(C)C)cc1 CS(=O)(=O)C1CN(C(=O)C(N2CCCCC2c2nccs2)=O)C2(CCCC2)C1 C1(C(=O)OC)CCCC(C(=O)NCC(C)NC(=O)CC(C)c2cnn(C)c2)C1 C(=O)(CC1CCC(=O)c2ccccc21)NC1(C)CC(NC(c2n(C)ncc2)=O)C1 C(=O)(C(CCS(C)=O)NC)NC1CCN(C(C(=O)N(C)C)=O)CC1.C1CCCO1 C(=O)(C=CS(F)(F)(F)(F)F)NC1(C)CCCN(C(=O)C(C2(O)CCCC2)F)C1 C(C)(C(CC(=O)N1CC(C2CC2)(OC)C1)NC(C1CN2CCN1CC2)=O)OC c1(C(=O)NCC2(CNC(CN3CCC(C)C3)=O)CC2)cnn2cccc2c1 c1(OC)cccc(C(O)C(=O)NC2CCN(C(=O)CCc3cncnc3)C2C)c1 c1(CC=O)cccnc1C(F)(F)F.c1(C(N(CCC)C)=O)scnc1C1CC1 C(=O)(C(C)(C)NC(=O)CCn1cncn1)NCC(C)N(CC)CC C1(CC#C)(C(=O)NCC2(CC(C)C)CC2)CCN(C(=O)C)C1.C1CCC1 C(C(CC(=O)NC(CCO)C1CCC1)OC)NC(CCOC)=O N1(C(CCCC(=O)NCC)=O)CCC2(CC1)CN(C(c1csc(Br)c1)=O)CCO2 C(=O)(C(CCCOC)NC(=O)C=C1CCC1)NCC.C1CSC1 Cc1c[nH]cc1C(=O)N(CCC)CCC.n1(C2(C=O)CC2)ccc(C2CC2)n1 c1(C(=O)NC2CCC(OCC)CC2)ccc(C)cc1-n1cc(CCCC#N)nn1 C#CC(CC(C)(C)C)NC(C1CN(C(c2cnn(C(C)C)n2)=O)CC1(F)F)=O c1(C(=O)N)ccc(-n2cnnn2)cc1.c1(C(C)=O)ncc(C(=O)NC2CCC2)s1 C1(C(N2C(C3CCCN(C(CCOCC)=O)C3)CCC2)=O)CC12CCCCC2 CS(=O)(=O)c1cc(Cl)cc(Cl)c1.c1(-c2cn(CC(=O)N)nn2)ccc(F)c(F)c1 C1(O)(CNC2CCN(CC=C)CC2)CCCN(C)C1=O c1(N(C2CCCN(C(c3nccc(OC)c3)=O)C2)C)ncnc2n[nH]c(C)c12 C(=O)(C#CC(C)C)N1CCC(N(C(c2ccn(CCC)n2)=O)C)C1 Cc1cc(C(=O)NCC(C)N(C)C(c2nncn2C2CC2)=O)nn1CCO C1(NC(c2c(C(C)=O)cn(C)n2)=O)CCCN(C(=O)C(O)C2CCC2)CC1 C1(C(=O)NCCCCCCF)CC2(CCC2)CN1C(=O)Cn1cnnc1 C1(COC2CCN(C(CC(C)OC)=O)C2)CCN(C(c2ccns2)=O)CC1 C1(CNC(C(CC=C)C)=O)CC(F)(F)CN1C(c1c[nH]cc(C)c1=O)=O c1(C(=O)NC(C)C(C)C(=O)N(C)C(C2CCCC2)C)ccc(N)c(F)n1 CCCCCC(C)(CC)C(=O)NCC1CCN1C(c1cnc(O)nc1O)=O C1(CNC(c2c(C)occ2)=O)CC(F)CN1C(c1ccc(-c2ccccc2)o1)=O Cc1ccnc(C(=O)NCC2(C(=O)N)CC2(F)F)n1.c1(C2CC2)ccccc1 c1(C(N2CCC(C(=O)OC)C2(C)C)C(=O)NC2CCCC2)cc(C)c(C)cc1C c1(OCCCC)c(OC)cc(C(N2CCN(CC(O)COC)CC2C)=O)cc1Cl CCCC(C)CC(=O)NCC1(CNC(c2ccc(F)cn2)=O)CCOCC1 C1(C2(O)CN(C(C3CCn4ncnc4C3)=O)C2)CC1.c1(C(=O)N)coc(O)n1.C c1(C(N(C2CC(S(C)(=O)=O)C2)C2CCC(=O)NC2=O)=O)cnc2c[nH]nc2c1 c1ccc(Cl)cc1.C1(C=O)CCCN1.C1(C(=O)NCCC)(CSC)COC1.N c1(CC(=O)NC2CC(CCNC(=O)CC3CCC3)C2)ccn(C(F)F)n1 c1(OC)ccc(CN2CCC(N3CCS(=O)(=O)CC3)C2)cc1-c1cccc(N)n1 c1(OC)cc(C(=O)NC2CC(C(=O)NC3CCOCC3CO)C2)ccn1 N1(C(c2cnn(C)c2N)=O)CCC(CNC(C2(C)CC3CCC2O3)=O)C(F)(F)C1 Cc1c(C(N2CCCC(CC)C2)=O)cc(C(C)C)n1C.C(=O)CN(C)C(C)C.N C1(C(=O)NC(CCC)C(=O)NC(C)C)CCN(C(=O)CC)O1 c1(OC)cnc(-c2noc(-c3ccc(I)nc3I)n2)c(OCc2ccsc2)c1 C(=O)(C1c2c[nH]nc2CN1C(C1CC1C#N)=O)N(C1C(OC)COC1)C C1(N(C(COCC=C)=O)CCO)CCCN(C(C2(C)CCNC2=O)=O)C1 c1(NCc2c(C)non2)ccc(S(=O)(=O)NC2CCCc3sccc32)cc1F Cn1c(N2CCC(CNC(C3(O)CCOC3)=O)C2)c(C#N)c(=O)n(C)c1=O CCC(CC(=O)N1CC(CNC(=O)C(C2CC2)C2CC2)C(C)C1)C(C)(C)C Cc1csc(C(=O)N(CC(C)CNC(c2csnc2C2CC2)=O)C)c1 C#Cc1cncc(C(N2CCCC(C(N3CCC4C(C(N)=O)C4C3)=O)C2)=O)c1 Cc1ccc(O)c(CC(N2CCC(NC(c3c(C)noc3C)=O)C(CO)C2)=O)c1 C1(C(N2CCC(C(=O)NCC)(CC)C2)=O)C2CCCC(=O)C12.CC(N)=O.O Cc1cnc(C(=O)NC2CC2C(=O)Nc2cccc(O)c2)cc1Br C(c1cn(C(c2ccc(C)cc2)CC)nn1)=CC [SH](=O)(=O)c1ccc(C(=O)N(CC(=O)O)CC(C)C)cc1.C1(OC)CCC1.N CCCC(C(=O)NC(CNC(=O)C(C)CC1CC1)C1CCC1)NC(N)=O c1(CC)nn(C)cc1C(=O)NCC1CCC1.C1(C(=O)N)C2CC2C2CC12 C1(C(=O)NCC(CN(C)C(c2cc(Cl)n[nH]2)=O)O)CCC2CC12 CC1(C(=O)Nc2ccc3cccc(F)c3n2)CCOc2ccccc21 C(=O)(CCC(F)(F)F)N1CCC(CCOC)(NC(c2ccncn2)=O)C1 CC1=NS(=O)(=O)N(C)C=C1C(=O)NC1CCCCN(C(c2cn(C)cc2C)=O)C1 c1(C(=O)NC2CN(C(C3N(N=O)CCCC3)=O)CC2CO)cc2c(s1)CCOC2 c1(OC)cccc2c1CC(C(N1CCc3ccccc31)=O)CO2 CC1COCCC1N(C)C(C1(C(=O)NCC2CC2C#N)CC1)=O c1(C(=O)NC(C(=O)NCC(C)C)C)cc(C(N)=O)ccc1C(F)(F)F C=CCC(C)(C(=O)N1CCOC(CN(C(=O)CC(C)(C)O)C)C1)N(C)C c1(CC)nc(CNCC2(F)CN(C(C)C)C2)cs1 C=C(C)CCCC(=O)N1CCC(O)(C(C)NC(c2cccc(OC)c2F)=O)C1 N1(C(c2cc(C)on2)=O)CCOC(C)(CNC(c2cc3sccc3[nH]2)=O)C1 CCCCS(=O)(=O)NCC(=O)NC1CCC(NC(C2(CC)CC2)=O)C1 C1(C(=O)NC2CN(C(c3c(C)ccc(Cl)c3F)=O)C2)C2Cc3ccccc3C12 CS(=O)(=O)C1(C(=O)NC2CC2C)CCOCC1.C(=O)(CCC1OCCO1)N N1(C(c2nc(CCCC)sc2)=O)CCN(C(c2ccn(C)c2C)=O)C(CCO)C1 Cc1cc2c(C(N3CCC(NC(=O)COCCCC(C)C)C3)=O)ccc(C)c2[nH]1 N1(C(C(Cc2cnc[nH]2)NC(c2cc(C)sc2C)=O)=O)CCC2(CCCC2)C1 N1(C(Cc2cc(C)on2)=O)CC(CNC(=O)C(C)c2ccco2)OC2CCCC12 C1(CCNC(=O)CCC2CC2)CSCCN1C(C1CCCC2CC12)=O c1(C(N2C(CC)CCC2)=O)cc(Cl)c(F)cc1Cl.c1(COC)cc(C=O)on1.N C1CC2CCC(C1)N2C(=O)CCC1(C)CC1.c1(OC)ccc(C)nc1C(=O)N Cc1c(C(N2CC=C(CNC(C3CCCC(C)C3)=O)CC2)=O)cccc1O C=CCCCCCC(=O)NCC(C1CCOC1)NC(c1cc(C(N)=O)cn1C)=O CC1(C)CN(C(C2COC(=O)C2)=O)C1C1CCN(C(=O)CC2(C)CCC2)CC1 Cc1ncc(C(=O)N(C(C)CCNC(C2(C(F)F)CC(O)C2)=O)C)s1 C#CCC(C(=O)NCCN1CC(N(C)C)C1)NC(=O)C1CC1 C(CC(C)(C)C(=O)Nc1ccc(NC(c2cncc(C)c2C)=O)c(C)c1)OC N1(C(COCCOCC)=O)CCN(C(=O)C=Cc2cnn(C)c2)CC1C Cc1nn(C)cc1NC(=O)CC1CC(C)N(C(C2CCC2)=O)C1 c1(C(C(=O)NC2(CO)CCN(C(=O)CCCF)C2)=O)c[nH]c2ccccc12 CN=c1nc(N(CCCc2ccccc2)C)[nH]c(=NC2CCCCC2OC)[nH]1 CCCCCC(=O)N(C(CNC(=O)Cc1cnn(C)c1)CC)C C(=O)(N=c1nc[nH]n1C)C1N(C(c2c(OC)cc(Br)cn2)=O)CC1 Cc1[nH]nc2c(C(=O)NC3CCC(NC(=O)C(C)c4ccon4)CC3)cccc12 N1(C(c2n(COC)ncc2)=O)CCN(CCNC(C2OCCCO2)=O)CC1 C1(NC(Cc2ncc(C)s2)=O)CCN(C(=O)C(c2ccc(F)c(F)c2)C)C1(C)C c1(CC=O)ccccc1.c1(C(=O)NCCCC)cnc(C(F)F)s1.C(C)=O.N C(=O)(C(CO)C(C)(C)C)NC1C(NC(c2c(OCC)nccc2)=O)CCC1 CC1(C(=O)Nc2cncc(CO)c2)CC(O)CN1C(c1ccncc1N)=O C1(CC)COC(C)(C)CN1C(C1CCC(C)N1C(c1cnc(OC)s1)=O)=O C(=O)CCC(N)=O.c1(CC)cnoc1C(=O)NC(C)(C)C1CC1.C(C)=O C12(NC(c3c(C)cc(Br)o3)=O)CC3CCC(C1C2)N3C(c1c[nH]nc1F)=O c1(C(=O)N)ccncc1F.C12(NC(c3cnc(-c4ccccc4)s3)=O)CC(C1)C2 C(=O)(C(CNC(=O)C=Cc1cc[nH]c1)OC)NC(C#C)(C)C1CCOC1 N1(C(C(N2CCOC(c3ccc(F)c(F)c3)C2)=O)=O)CC2(CCC(C(F)F)O2)C1 C1(c2n(C)ncc2)CN(C(C2C3CCC2CC3)=O)CC1NC(C1(C)CC1(F)F)=O N1(c2c(C)cnc(Cl)n2)CCC2CCC(C1)N2C(c1cccc2ncoc12)=O C1(NC(c2c(C(C)C)occ2)=O)CN(C(C2(CC(F)F)CCC2)=O)CC1O c1(NC(CCc2nc(COC)nn2-c2nccn2C)=O)ccccc1C(C)C CCC(C(=O)NCC1C2CN(C(C3C4CCCC34)=O)CC12)C(C)C Cc1[nH]c(=N)nc(O)c1CC(=O)NCC1CCN(C(=O)C(C)C)CC1C N1(C(C2C(OC)CN(C(c3nc(Cl)oc3C)=O)C2)=O)CCC(N(C)C)C(C)C1 C1(C(N2CC=C(CO)CC2)=O)CCC2(CC2)N1C(C1CC1(F)Cl)=O Cc1ncc(C(=O)NC(COC(C)C)C(=O)N2CC(n3cnnn3)C2)c(C)n1 N1(C(c2cnc(C(C)OC)s2)=O)CCOC(C)C1.N1(CCC(=O)N)CCOC1=O c1(OC(C)C)cccc(C(=O)NCC2CC(F)CN2C(=O)C)c1.C1CCC1 Cc1cn(-c2ccc(F)cc2)[nH]c1=NC(=O)NC(C1(O)CCOCC1)C c1(OC)nc2ccccc2cc1C(N1CCC(Oc2cccnc2)C1)=O C(O)(CC(=O)NCCc1cn(C2CCOCC2)nn1)(C(F)(F)F)c1scc(C)n1 C(c1cnc(-c2ccc(Br)cc2)s1)=CC(N1CC(C(=O)NC)C1)=O N1(C(C(C)N(C(c2ccnn2COC)=O)CC)=O)CCCC2COCC12 C12(NC(C3CC(C)OC3)=O)CCCC1N(C(=O)C(C)C(C)(F)F)CCC2 N1(C(Cc2ccc(OC)cc2)=O)CCC(NC(C2CC(=O)C2)=O)C(C)C1 C(=O)(C(C)CNC(C1(C#N)CC1)=O)NCCCCN(C(C)C)C c1(C(N(CCOC(C)(C)C)C2CC2)=O)cn2c(Br)cnc2s1 C1(NC(CC(COC)C)=O)CN(C(=O)Cc2cc(F)c(F)cc2F)CC(C)(C)C1 C1(NC(C2CC(C)(O)C2)=O)CCCCC1.c1(C(=O)N)ccnc(OC(F)(F)F)c1 O=[N+]([O-])c1ccccc1N1CC(NCC2=CCOCC2)C1 c1(CN(C)C(c2cnc(N3CCNCC3)s2)=O)ncc(Cl)n1C N1(C(COC(CC)C)=O)CCC(NC(=O)CCc2ncc[nH]2)C2(CCC2)C1 c1(NC(C2CCCC(C(F)(F)F)C2)=O)ncnn2cccc12 C1(CC)CN(C)CCCN1C(c1cn(C)c(=O)n1C)C(=O)NC1CC(F)(F)C1 N1(C(=O)Nc2c(SCC=C)cccc2)CC(C)OCCC1C c1(N(C2CCCCC2)C(C)=O)cccnc1C(N)=O.C1(C=O)(C=O)CC1.CO c1(SC)cccc(C(=O)NCCC(C)NC(=O)CC2(C)CC(F)(F)C2)c1 c1(C(N2CC=CC(NC(C(C(C)C)N(C)C)=O)C2)=O)cccc2cc[nH]c12 C1(C(N2CCCC(C(N(CC(F)F)CCC)=O)C2)=O)CCCC(C#N)C1 C1(NC(C2C(=C)C2)=O)CCN(C(c2csc(SC)n2)=O)CC1C N1(C(C=NOC)=O)CC(C(=O)NCc2cn(C)nc2OC)C2(CCC2)C1 CC1(C)CCC(C(=O)NCC2(C)CCCS2)CN1C(=O)CCc1nncs1 N1(C(c2c(C)nccc2)C(=O)NC(C)C)CCCSc2ccc(F)cc21 c1(CC)ccnc(SCN(c2ccc(SC(F)(F)F)cc2)C(C)(C)C)n1 c1(C(N2CCC(NC(c3c(C)scn3)=O)(CF)C2)=O)cc2cccnc2s1 N1(C(=O)C2=COCCC2)CC23CCCC2(C1)CN(C(c1snc(Cl)c1Cl)=O)C3 C1(C)(CC)CCN1S(=O)(=O)NC1C2(CC2)C12CC2 N1(CC(C)C)C(=S)NC(c2c[nH]nc2-c2ccccc2)C2=C1C(C)(C)NC2=O C1(CCN)CCCN(C(=O)CCC(=O)N2CCN(c3ccccc3Cl)CC2)C1 C(=O)(CC(C)C(C)C)N1CCC(N(C(C(COCC)C)=O)C)CC1 CCC(CC(=O)NC1(CNC(c2c[nH]nc2-n2cnnn2)=O)CCOC1)C1CC1 Cc1cc(C(N2CC(C)(NC(c3sc(CC(F)(F)F)nc3C)=O)C2)=O)cc(C)c1 c1cccc(O)c1.CC(CC(C)NC(C1(N2CCCC2)CCC1)=O)NC(=O)C.O N1(C(CC(CNC(C(C)N(C(C)=O)C)=O)(C)C)=O)CCN2CC(F)CC2C1 C1(C(=O)OC)C2CN(C(C3CCN(C(c4csc(C)c4)=O)C3C)=O)CC12 Cc1cc(C)c(C=CC(=O)N)c(C)c1.C1(C)CCN(C(c2cnnc(O)c2)=O)C1 Cc1nc(C(=O)N(C(C)CNC(=O)Cc2cncc(O)c2)C)c(C)o1 Cc1cc(N)ccc1C(=O)N(C1CCN(C(c2c[nH]nc2Br)=O)C1)C C1(CC(=O)NCC(=O)NCC(=O)NCC(C(C)O)C)COCCOC1 N1(C(C2(CC#C)CCOC2)=O)CC2CCN(C(=O)Cc3c[nH]ccc3=O)CC2C1 C(CC)(C(C)(C)O)NC(C(CN(C(C1(CCC)CCC1)=O)C)C)=O C(=O)C(O)CC(F)(F)F.c1(C(C(=O)N(CC(C)(C)C)C)=O)ccc(F)cc1F.N C1(O)CCCN(C(C2CCCCNC2=O)=O)C1.S(=O)(=O)(CC(=O)NC)NCC.C Cn1ccc2c(N(C3CCC(N)C3)Cc3ccc(S(N)(=O)=O)cc3)ncnc12 c1(C(N2C(CNC(CCSCC)=O)CCCC2)=O)cc2nc[nH]c2cc1N c1(C(=O)NCC2CCCCO2)cc2c(s1)CCN(C(c1c(Br)cccc1Br)=O)C2 Clc1cc(C(c2nnnn2C2CCC2)NCc2ncc(Br)s2)sc1Cl c1(N(C)C(c2ccsc2Br)=O)ccc(C#N)c(I)c1 c1cc(C)c(C=O)cn1.C1(CC(=O)N(CC)C(C)C)CCCC(F)(F)C1.C c1(C(=O)NC2COCCC2NC(C2CCC23CCC3)=O)cc(F)c2cn[nH]c2c1 C=C(Cl)CC(C(=O)NCCC1=CCCCC1)NC(C1C2CCC(C2)C1C)=O CC(CC(=O)N1CCC(C)(CNC(c2ccc(N)c(N)n2)=O)CC1)CC(C)(C)C C1(NC(c2nc(C)oc2)=O)CC(CNC(c2cncc(O)c2Cl)=O)C12CCC2 C(c1nnc(C(C)C)o1)=CC=O.C(=O)(CCCC1CC1C)N.C1CC1.CC Cc1cc(C(=O)NCC(O)C(=O)NC(C)Cc2nc[nH]n2)no1 N1(CC(N2CCCC2)=O)C(=O)CCCC1=O.C1(OCC(=O)N)CC(F)(F)C1 c1(C(=O)NC2CC(=O)NC2)n[nH]c2c1CN(C(=O)CCBr)CC2 S(=O)(=O)(c1ccc(-c2cccc(C(F)(F)F)c2)s1)N(C(C(CCC)C)C)C c1(OC)cc(C)c(Cl)cc1C(=O)N.C1(CC)CCN(C(=O)C)C1.C(C)(C)C C(C)(C)(CCCF)NC(C(C)NC(CC1(OCC)CC1)=O)=O Cc1cnc2c(C(=O)N(C3CCN(C(=O)C(=C4CCCCC4)F)C3)C)cccn12 CCCC(C#N)C(=O)NCCn1cc(CNC(C2CCCC(=O)N2)=O)nn1 C12(C(N(C)C)=O)CC(C)(C1)OC21CCC1.C(C(=O)N1CCCC1)(C(C)C)SC Cc1cc(C)c(C(=O)N)c(C)n1.C1CC2(C1)CC2.N1(CC=O)CCS(=O)CC1 C1CCC(O)CN(C(c2cc(C)c(Cl)c(C)c2)=O)C1.C(C)(C(=O)N)N(C(C)=O)C N1(C(CCc2ccc(C)o2)=O)CCC(CNC(C23CCN(CC2)C3)=O)C(C)C1 n1(CC)cc([N+](=O)[O-])c(N2CCC(CCNC(c3ncoc3C)=O)C2)n1 Cc1c(CC(=O)NCC2COCCN(C(=O)C(C)C#N)C2)ccc(Cl)c1Cl c1(C(N)=O)cc(C(N2CCC(CCNC(=O)CNC=O)C2)=O)co1 C1(CC)CN(C(c2ncc(C(F)F)s2)=O)CCC1NC(C1CC1CC)=O c1(C(=O)NC(CN(C(=O)C=Cc2ncc[nH]2)C)(CO)CO)cnc2cccnn12 N1(C(c2c(OC)ccs2)=O)CCCCC(NC(c2cnc(N)c(O)c2)=O)C1 c1(C(N(C)CC2CCCCN2C(=O)Cc2cnnn2C)=O)noc2c1CCCC2 C(CCCC(=O)NC1CC12CCCC2)N(C(=O)CC1(O)CCCCC1)C C1(C)(C(=O)OC)CCCN(C(=NCCC(C)=O)NCC2(CC(N)=O)CC2)C1 N1(C(C(CC)SC)=O)CCC2(CC1)CCN(C(c1cnc(OC)cn1)=O)CC2 c1(C(=O)NCC(n2cc(-c3c(C)cccn3)nn2)C)ccc(C#CC(C)(C)O)o1 Cc1cnc(Cl)c(C(N2CCCC(CCNC(C3(C)CCCC3C)=O)CC2)=O)c1 c1(C(N2CCCC(CCNC(C3C(CCC)CCC3)=O)C2)=O)c(F)ccnc1F N1(C(c2cnsn2)=O)CCC(C2CCN(C(c3cc4nc(Cl)ccc4o3)=O)C2)C1 CCC(CC(=O)N1CCCCC1CN(C(=O)CCC1OCCO1)C)SC c1(C(=O)NC2CC(NC(c3n(CC)nnc3)=O)C(O)C2)ccc(F)c(F)c1N c1(C(=O)NCC(COC)NC(=O)CCC2CC2C)nccn2cnnc12 Cc1coc(C)c1C=CC(=O)NCC(CO)NC(=O)Cc1c(F)cncc1Cl N1(C(c2ccnc(C)c2C)=O)CCC(C)(C)CC1C(=O)NC1CC(C)C1 CN=S(C)(=O)CCCC(N1CCC(Cn2cc(-c3ccc(C)cc3)nn2)C1)=O C(CC(C)(C)C)(C(=O)NC1C(C)CN(C(=O)CC2CC3C=CC2C3)CC1C)OC CC(C)C(C(=O)N(C)CC1CCN(C(c2ccc3nccn3n2)=O)C1)C(C)C Cc1cccc(C(N2CCOCC(CNC(c3cncn3C3CC3)=O)C2)=O)c1F C1(CONC(c2occc2CNC(c2csc(F)c2)=O)=O)(C)CC12CCC2 c1(C(=O)NCC2C(C(=O)NCCN(OC)C)CCC2)nccc2cc[nH]c12 c1(C(=O)NC2CCCC(NC(C34CCCC3OCC4)=O)C2)cnc2[nH]ccnc1-2 C(=O)(C(C)C(O)CC(C)C)N(CCC(=O)N(CCC(N)=O)CC)CC#C C#CC1(O)CCN(C(=NC)NCC2COC(C)(C)C2)C1 N1(C(C(c2cccc(C)c2)C)=O)CC(NC(c2cccnc2N)=O)CC1(C)C Cc1ccc(I)c(C(=O)NC2CC(NC(c3ccccc3)=O)C2)c1.C(C)(C)O Cn1cc(C(=O)NCCC(C)(C)NC(=O)CC2CC3CCC2C3)c2cccnc12 c1(C(=O)NC(C2(O)CCN(c3ccc(C#N)nn3)C2)C)cccn2nncc12 C(=O)(CS(=O)(=O)C(C)(C)C)NC1CC(C)N(C(c2ccc3nc(S)[nH]c3c2)=O)C1 c1(C(N2C(C(=O)NCC3CCC(F)(F)C3)CC2)=O)cc2ccccn2n1 CC1CN(C(=O)COc2cccc(Cl)c2)CCC1CNC(c1coc(O)n1)=O C(N=c1[nH]c(=NCC2(C)CC3CC3C2)[nH]c2ccsc12)C1N(C)CCCC1(C)C C(=O)(C1CCc2cc(Br)ccc21)NCCC(C)(C)CNC(C1CCC1)=O C1(C(=O)NC(CCC)(C)CO)Cc2ccccc2CN1C(=O)CN C1(COC)C(CN(C(c2cccnc2)C(=O)N)C)C1(C)C.C1(C=O)CC1 N1(C(C(C)NS(C)(=O)=O)=O)CCOC(CCNC(C2CC(C)(C)C2)=O)C1 c1(NCC(CN(C)C)(C)C)ccc([SH](=O)=O)cc1Br.C1CCCC1C(C)(C)C.N C1(C(=O)NC(C(=O)N(CC)CC)C)C=CCN(C(c2cn(C)cn2)=O)C1 C1(N(C(=O)CC(C)(C)O)C)CCCCN(C(C2COCC(C)(C)O2)=O)C1 c1(C(=O)NC2(C)CN(C(=O)COc3ccccc3Cl)C2)c[nH]c(C#N)c1 C1(CNC(c2c(CC)cco2)=O)(CO)CCN(C(C2SCCC2C)=O)CC1 c1(CNC(=O)N)sc(Br)c2c1OCCO2.C1(C(c2ccccc2)=O)CCOC1.C O=C1CCCC(CCCC(=O)N2CCC(CCNC(C3C4CCC3CC4)=O)C2)N1 C1(C(N2CC(C)CC(NC(C(CC#C)(C)C)=O)C2)=O)CC2CCC(C1)N2C C1(NC(C=CC)=O)CN(C(=O)CCOCC(F)F)CCC12CCOCC2 c1(C(N2CC3(CNC(CSCC)=O)C(C2)CCO3)=O)ccc2nc(CO)[nH]c2c1 C(CC)(C(=O)N1CCC(CNC(c2ccc(OC)s2)=O)C1)OCC C(=O)(C(O)CCC(C)C)N(C1CCN(C(c2[nH]cc(C)c2)=O)C1)CCO N1(C(C2(C)CN(C)C(=O)C2)=O)CC2CN(C(c3sccc3C3CC3)=O)CC2C1 C1(NC(C2=CCC(NC(C(C)c3ccco3)=O)C2)=O)CN(C)CCN(C)C1 C1(NC(CC)=O)CC2CCC(C1)N2C(=O)CCCCCN1CCSC(C)(C)C1 c1(C(C)C)nnc(CNC2COC(C)(C)C2)n1C c1(NCCCCCCN(C(CN(CC)CC)=O)C)ncc(C#N)cc1Br C1(C(C)CNC(=O)NCc2ccc(CS(C)(=O)=O)o2)CCCC(=O)N1 C(c1ccc(C(N)=O)o1)=CC(=O)NC(C)C.C1(C=O)CCN(C)C1.CC C1(CNC(C(=CC2CCCC2)C)=O)CN(C(c2nc(Cl)sc2C)=O)C(C)(C)C1 c1(C(=O)NC(C)CNC(c2cc(CO)on2)=O)cc2n(n1)CCNC2=O C1(CC)CCN(C(=O)CC2CCCC(NC(c3ccc(F)s3)=O)C2)CC1O Cc1ccc2nonc2c1C(N1CC(NC(c2nccc3ccn(C)c23)=O)C1)=O N1(Cc2ccc(OC)cc2)CCC(CNC(c2cccnc2O)=O)C(F)(F)C1 c1(OC)ccc(CC(=O)NCC2CC(NC(C3(OC)CCC3)=O)C2)cc1F c1(C(N2CC(NC(CC(C)C)=O)C2)=O)ccncc1N(C)C c1(N2CC(C)(NC(C3(OC)CCCCCC3)=O)C2)ccc2c(n1)CCCC2=O C1(CNC(c2n(C3(C)CC3)nnn2)c2csnn2)CCOCC12CCCC2 N1(C(c2ccc(C#C)nc2)=O)CCC2(C=C(C(=O)NCCc3nncs3)C2)C1 C(=O)(CC(C=C)CC)N1C(C(=O)NC(C#C)CC2CCCC2)CC(F)C1 c1(NCC(COCCOC)O)ccc(S(=O)(=O)N2CC(CO)CC2C)c(Cl)c1 S(=O)(=O)(c1cnc(N(C)CCn2ccnc2)c(Cl)c1)N1CC=C(C)CC1 C(CCC(=O)N(C1(C=O)CCC1)C1CC1)=CC.c1(C2CC2)ccc(C)o1.N c1(C(C)C)cncc(C(=O)NC2CCC(F)(CNC(=O)CO)C2)c1 O(NC(=O)CCC1CCCCN1C(C1CC2(CC2)CO1)=O)CCOC N1(C(C(=O)Nc2ccc(C(=O)OC)cc2C)C(C)CC)CC2CC=CCC2C1 S(=O)(=O)(c1cccc2ccccc12)N1CC(NC(c2cc(O)no2)=O)CC(C)C1 Cc1nc(N(CC(C)NC(=O)C(C)n2cncn2)C)ccc1[N+](=O)[O-] C(=O)(N=S(C)(=O)C1CN(C=O)C1)c1nc(C)c(C(=O)NC)cn1.C(C)(C)C C(C)(CC(F)(F)F)NC(c1c(C)nc[nH]1)=O.C(=O)(C(CN(C)C)N(C)C)N C1(c2n(CCCCCC)nnn2)(NC(c2ccc(Br)o2)C)CC(C)(C)CC1C C1(C(=O)NCC(=O)NCC2(F)CC(CO)C2)(CO)CCCO1 CN1C(=O)OCC1C(=O)NC1CCCC1(C)CNC(=O)CC1CCC(O)C1 c1(C(=O)NC(C2CCCO2)(C)C)cn(CC)cn1.C(C(F)(F)F)=CC=O.N C12(C(N(C(C(N)=O)CCC)C)=O)CCC(CC1)C2.C1(C=O)CC(C)N(C)C1 c1(C=O)ccc2c(c1)CCN2.C(=O)(CCC(=O)NC)NCC.C1(CC)CC1 n1(C(C)C)cc(Cl)c(C(=O)NCC(=C2CCCCC2)F)n1 C(C)C=O.C(=O)(C(F)Cc1ccccc1)N.C1(CSC)CC(C)C1.C=O c1(NC(C2CCN(C(C(CSC)(C)C)=O)CC2O)=O)c(Cl)cc(Cl)cc1I C1(C)(C(N(CC=C)OC)=O)CCCN(C(=O)C(C)C(C)(C)C)C1 C1(O)(CNC(C2N(CC)CCC2)=O)CCCN(C(=O)C=Cc2ccoc2)C1 N1(C(C(CCC)O)=O)CCC(CNC(c2scc(C)c2Br)=O)C1(C)C CC1=NNC(=O)C1CC(=O)NC1(C(=O)NCC(C)CC2CC2)CC1(C)C CCC(C)(F)C(=O)NCC(c1ccccc1SC)NC(c1cnc(C)nc1)=O C1(NC(c2nn(C)c(Cl)c2)=O)CN(Cc2ncccc2Cl)CC2(CCOCC2)C1 c1(CC)ccc2[nH]c(C(N3CCCN(C(=O)CS(=O)CC)CCC3)=O)c(C)c2c1 c1(CC)cccc(C(=O)NC2CC3C(NC(=O)C4=CCCCO4)C3C2)c1F c1(C(C)=O)ccc(C(=O)NC2CC(C)C2)c(O)n1.C1(C)(C=O)CCSCC1.C c1(C(=O)NCC(CC)(C)NC(c2nnn(C)n2)=O)c(C)cc(C)nc1C C1(C(=O)NCC(N)=O)CC2CCC1N2C(c1ccc(F)nc1)=O O=C(C1CCCc2nncn21)NCCC1COCCN1C(=O)C1=CCCS1 CN1CCN(c2ncc(C(=O)NCC3CC(n4cccn4)C3)s2)CC1 CS(=O)(=O)CCN(c1nncn1C1CC1)CC(N1CCCC1)=O c1(C(=O)NC23CC(C2)N(C(c2cscn2)=O)C3)cc(Br)cn(O)c1=O C1(NC(C(CC)SC)=O)CCN(C(c2cnc(C(C)(C)C)[nH]2)=O)C1CC C(=O)(C(O)CCC(C)C)N(CCOC)CC.c1(C(=O)N)ccn(C2CC2)c1C c1(OC)ccc(C)cc1NNC(=O)Nc1cc(Br)cc(Br)c1N C1(C(=O)NC)CN2CCCN1CC2.C1CC(F)CN1C(c1cscc1C(F)F)=O C1(NC(c2csc(CO)n2)=O)CCOC1C(=O)NCC(c1ccncc1)O Cc1cc(CO)oc1C(=O)NC1(C)CCN(C(=O)C(c2cnccn2)C)C1 C1(NC(C)CC2CCCNC2)CCCc2ccccc2C1 c1(NC(C2CN(C(c3ccc(S)cc3)=O)C2)=O)ccc2c(n1)CCC2 C1(CNC(c2n(C)ncn2)=O)CCN(C(=O)Cn2cnc(=N)[nH]2)CCC1(F)F C1(CCNC(C(CCC)=CCC)=O)CN(C(=O)C=CC2CCC2)CCCO1 n1(CC)ccc(C(=O)NC2CCN(C(c3cc(C(F)F)no3)=O)CC2F)cc1=O C1(NC(c2n(CC)nnc2)=O)(CF)CCN(C(C2(OC)CCC2)=O)C1 c1(CN2CC(CNC(CCSC)=O)OCC2)cnc(Cl)c(C)c1 C(c1ccccn1)=C(C)C(=O)NC1(CN(C(=O)CCc2ccsc2)C)CC1 C(=O)(CC(C)C(C)C)NCCN(C(C(OCC)OCC)=O)C N1(C(c2c(SC)snn2)=O)CCCCC(NC(c2ccnn2C2CC2)=O)C1 C1(CC(=O)NCC(C)NC(C2CC3CCCCC23)=O)CC2CCC(C1)N2C C(=O)(C(F)C(F)(F)F)NCCC(=O)NCC(=C)C C(=O)(CC(C(C)OCC)NC(=O)C=C1CCC1)Nc1cn(CC#C)nc1 C1(CC(=O)NC2C(C)CN(C(=O)Cc3cccnc3)C2)CCCC(C)(C)C1 N1(C(C=NOC)=O)CCC2(CC1)CC(NC(c1n[nH]c3c1CSCC3)=O)CO2 CCC(CC(=O)NCc1cc(O)ns1)N(C(=O)C=Cc1cscn1)C c1(OC)cncnc1NC(c1ncc(-c2ccc(Br)cc2)[nH]1)C c1(NC(=O)NCC(C)OCC=C)cc(C(F)(F)F)cc(Cl)c1 C12(CNC(=O)C3=CC4C=CC3C4)CCCC1N(C(=O)Cc1cc(Cl)cs1)CCC2 C(=O)(CC(C)CF)N1CCC(NC(C(=O)NCCOCCCC)=O)C1 N1(C(C(CSC)(C)C)=O)CCCC2(CCN(C(C3CC4CCC3C4)=O)CC2)C1 C(=O)(C(F)CCC(C)(C)C)NC1C2OCC(NC(C=COCC)=O)C2OC1 C1(n2cc(CCC(=O)NCC(CCC)=O)nn2)CCCCCC1O C(=O)(C(=O)N=c1cc(C)o[nH]1)N1C(CNC(c2[nH]c(CC)c(Cl)n2)=O)CC1 c1(C(N(CC)C)=O)cnc2c(ccn2C)c1.c1(OCC)ccc(C)cc1C=O.N C1(C(N2CCCCC(NC(Cc3cnc(C)o3)=O)C2)=O)CCC(=C(F)F)CC1 N1(C(C(c2ccc(OC)cc2)=O)=O)CCCCC(NC(C2(F)CCOC2C)=O)C1 CCC(O)C(=O)NC(c1ccccc1)C(=O)NC1CC(N2CCC2)C1 c1(C(N(C2CCN(C(c3ccccc3Cl)=O)C2)CCO)=O)nnn2c1CCCC2 N1(C(C2CCS(=O)CC2)=O)CC(C2CC2)(C(=O)Nc2cnc(O)c(F)c2)C1 C1(NC(=O)CCOCC(F)F)COCCN(C(=O)Cc2nnc(O)s2)C1 c1(C(CNC(c2ccc(C(C)=O)cc2)C)C)ccc(F)c(Cl)c1 N1(C(c2ccc(CCC)s2)=O)CCC(C2CC(NC(=O)C(F)(F)C3CC3)C2)C1 C1(NC(c2cn(CCOC)nc2)=O)CCC(C)N(C(=O)C)C1.c1cc(C)on1 c1(C(=O)NCCN(C(CC(CCCC)O)=O)CC(C)O)cccc2c1OCCO2 CC1CC2CN(C(=O)CCN(C(=O)Cc3cc(CN)no3)CC3CC3)CC12 c1(C(=O)NCCC(=C)C)cc(O)cc(=O)o1.C1(C=O)CC(N(C)C)C1.C C(=O)(C(F)CC(C)(C)NC(c1ccsc1)=O)NC1CCN(C(C)=O)CC1 CC1(C)C2CCC(C(=O)NCC3CCN(C(c4cc(C)on4)=O)C34CC4)C1C2 C(=O)(CCC(C)(C)C)N1CCC(CCC(N2C(COCC#C)CCC2)=O)CC1 CC(C)C(C(=O)N1CC(O)(C(C)NC(=O)CCC(=O)N(C)C)C1)n1ccnc1 C1(C(NOCCC(=C)C)=O)COCC1C(=O)NOCC.C(=O)CC(O)C1CCCC1 C1(NC(C(CCC)OC)=O)CC2CCC(C1)N2C(c1coc(CS(C)(=O)=O)n1)=O C1(n2cc(CC(C)(C)C)nn2)CC2CCC(C1)N2C(=O)COc1ncccn1 C(=O)(C(C)(C)c1cnco1)NCCN(C(C=C(C)C(C)C)=O)C C(=O)(C(CCCC)N(C)C)NCC1N(CCCC)CCC1 CC(C)(C(=O)N)S(C)(=O)=O.C1CC2(CO1)CN(C(C1COC(=O)C1)=O)C2.C C1(C(=O)NCC(C)NC(c2cc(CO)on2)=O)CNc2ccccc2O1 Cc1c(C(=O)N(CCCCCC(=O)NCc2ncc[nH]c2=O)C)cccc1C#N Cc1ccc(C(=O)NC2COCC2NC(c2cc(C)n(C)c(=O)c2)=O)cc1C#N N1(C(c2cc(C3CC3)ccc2F)=O)CCCC2(C1)CN(C(c1cscc1F)=O)C2 c1(C(N2C(CNC(C(C)(CO)OC)=O)C=CC2)=O)ccc(C#N)cc1 C1(CNC(C(CC(=C)C)C)=O)C2CCC1CN(C(c1cc[nH]c3nccc1-3)=O)C2 N1(C(C2CCC3C(C)(C)C2C3)=O)CC2(CCOCC2)C1C(=O)O c1(NC2(CNC(=O)COc3cccc(F)c3)COC2)ncnn2cccc12 c1(C(=O)NC2(C)CC(NC(C(C3CCC3)OC)=O)C2)ccc(=O)n(C)n1 c1(OC)cc(CC(=O)NC2(C)CCN(C(=O)CC3CCC(C)O3)CC2)ccc1Cl C1CCCCC1.C1(C(=O)OCC)(C=O)CC=CC1.C1(CC=O)CC12CC2.N CC1CC(CNC(=O)C(F)(F)c2cnn(C)c2)CN1C(=O)CCCCF C=C1CC2CC1CN2C(c1ncc(Cl)cc1Br)C(=O)NCCN1CCOCC1 C(=O)(C1=CCCCC1P(C)(C)=O)N1CC(NC(c2c(C)nn(C)c2Cl)=O)C1 c1(C(N2CCCOC(C(C)C)C2)C(=O)NC(CC)C)ccc(Cl)c2c1CCC2 c1(CC(=O)NCCN(C(C2CCNC2=O)=O)C2CC2)ccccc1F C1(CC(=O)NC(c2ccccc2)C#C)COCCN1C(C1CCC(=O)N1C)=O C1(Cc2cn(CC(C)NC(c3cc(C4CCCCC4)on3)=O)nn2)CCCCN1C C#Cc1ccc(F)cc1C(N1CC(NC(C2CC(=O)N(C)C2)=O)C2(CC2)C1)=O N1(C(c2c(C(=O)OC)c(C)[nH]n2)=O)CC(NC(=O)CC(C)C(F)F)CCC1C N1(C(c2c(C)cc(C)[nH]2)=O)CC2(CCN(C(C3(C4CC4)CC3)=O)CC2)C1CC c1(OC)cccc(CCNC(=O)Cc2ccno2)c1.c1(CC=O)csc(S)n1 c1(-n2ccc(C(=O)NC3CC(NC(C(N(C)C)C4CC4)=O)C3)n2)ccccc1F c1(C(=O)NCC(C(=O)NCC2CN(CC)C(=O)O2)OC)ncn2ccccc12 C1(C#N)(C(=O)NCCN(C)C(C2(O)CC(C)(C)C2)=O)CC12CCC2 C1(NC(C(CSC)O)=O)CN(C(c2oc(SC)cc2C)=O)CC12CCOCC2 C(C)(C)(CN=C(NC(C)C1CC1)N1CCC(C)(F)C1)SC c1(C(N2CCC(NC(C3C(C)C3C)=O)C2)=O)cc(F)ccc1-n1cccn1.CC N1(C(C=CC(C)C)=O)CCCCC1.C(=O)C=CC=O.C(N)=O.C1CC1.N Cc1cnc2c(cnn2CC(N2CCC(NC(=O)CCC#N)C(C)(C)C2)=O)c1 O=C(CCC1CCc2ccccc21)NC1CC(NC(=O)Cc2c[nH]ccc2=O)C1 N1(CCC(=O)NC(CNC(c2c(CC)nn(C)c2)=O)CO)Cc2ccccc2C1 C(CC(C)(C)C)(C(=O)NCC1([Si](C)(C)C)CC1)NC(CC(C)N(C)C)=O Cc1cnc2n1CC(C(=O)N(C(C)CNC(=O)C(C)(C)C(N)=O)C)CC2 C(=O)(C(C#N)C(C)(C)C)NC(C1CCCN1C(=O)CC(=O)N(C)C)C N#Cc1ccc(NC(=O)C2=CCCN(Cc3ccc(N4CCCC4)o3)C2)c(Cl)c1 C1(CC(N)=O)(NC(=O)C=Cc2nc[nH]n2)CCN(C(C2CCOC2)=O)CC1 CCN=c1ccc(C(=O)NC2CCCC(NC(=O)Cc3cn[nH]c3)C2)c[nH]1 c1(C(N(CC)CC)=O)cc(-c2csc(C)n2)c[nH]1.C1(CC(=O)N)C=CCC1 C1(CCC)CN(C(C2CC2F)=O)CCN1C(=O)Cc1cc(OC)cc(F)c1 CCCCC(C)CCC(=O)NCCCCCNC(=O)C(c1ccc(Cl)cc1)CO C1(NC(C(=O)N(C)C)=O)CC2CCCC(C1)N2C(=O)COCC1CCOC1 C1(C=O)CC1C1CCCC1.N1(S(C)(=O)=O)CCC(C(=O)NCCOCC)C1 c1(C(N2C(C)CC(CNC(=O)CC3(O)CCCC3)C2)=O)ccc2cc[nH]c2c1F c1(C(=O)NC2CCC(NC(c3cn(C)nc3)=O)CC2)c(N)cccc1Cl N1(C(C2C(=C)CC2)=O)CC2(C1)SCCC2NC(c1ccc(=O)n(C)c1)=O C(=O)(CCCC(C)(C)C)N1CCC(CCC(=O)N(CC(c2ccccc2)O)C)C1 N1(CC)CCC(N=c2[nH]c3ccc(S(=O)(=O)NC4CCS(=O)(=O)C4)cc3s2)C1 C(=O)(N(CCC(=O)N1CCC(CO)C(C)C1)OC)c1cccc(CC=C)c1 C=CC(C)(C)CC(=O)NCC1CC(C)N(C(c2coc(CO)c2)=O)C1 Cc1cc(O)c(C(N2CC=CC(NC(=O)C(C)(C)n3cnnn3)C2)=O)nn1 CC(C)CC(C)CC(=O)N1CCN(C(c2cc(F)c(O)c(F)c2)=O)CC1CCO c1ccccc1Cl.C(C(O)C(=O)NC(C)C(CO)NC(=O)CSC)=CCCC C(=O)(CCCCN(C)C(C1CC2C=CC1O2)=O)NCCSCCC=C C(C(C)(O)CC(=O)NC(C)(CNC(c1ncc(Br)cc1C)=O)CO)OC N1(C(c2cncc(C#C)c2)=O)CCCC12CCN(C(=O)CC(C)C(C)C(C)C)C2 N1(CCC(=O)NCCCCOC)CCOCC1=O.c1(C=O)csc(C(N)=O)n1.N C#Cc1cncc(C(N2CCC(C)C2CNC(C2(COC)CC2)=O)=O)c1 C1(O)CCCN(C(=O)CCN2CCCC2)C1.n1(CC(=O)NC)nnnc1C1CC1 CCC(C#N)C(=O)N1CCC2C(NC(=O)CC3CN(C)C3)C12 N1(C(C=Cc2ccc(OC)cn2)=O)CC2CN(C(c3n[nH]cc3F)=O)CC2(C)C1 c1(CC)sc(C(N2CC(O)(CN(C(=O)C(C)Cc3cnco3)C)C2)=O)cc1C C(=O)(C(F)C(C)(F)F)NC1C=CC(CC(=O)N(CC(CCC=C)O)C)C1 N1(C(CCC=C=C)=O)CCN(C(c2cc(C(F)(F)F)ccc2OC)=O)CC1CC CCC(C)(CNC(c1conc1COC)=O)NC(=O)Cc1nc(=N)[nH][nH]1 C1(C(CNC(CCC=CC)=O)O)CCN(C(=O)C(=Cc2ccccc2)CC)CC1 C1(C(N(CCCN(C(Cn2cc(C(N(C)C)=O)nn2)=O)C)C)=O)CC2CCCC12 C1(NC(CCOCCN(C(c2c(CCC)n[nH]c2)=O)C)=O)CC12CCCCCC2 c1(C(N(C(CC#C)C)C)=O)cc(CNC(C2CCOC2C(C)C)=O)cs1 C1(C2CCN(c3cc(CC(C)C)ncn3)CC2)(NC(C2=CC(C)(CC)C2)=O)CC1 C(=O)(C1=C(C)OCCC1)N1CCC(OCC(=O)Nc2ccc(C(CC)C)cc2)C1 c1(-n2cc(CNC(C(=O)OC)c3ncc[nH]3)nn2)ccccc1Cl C1(OC)CN(C(=O)Cc2cnccc2C)CC1NC(C1CC(F)(F)CS1)=O c1(OC)ccc(NC(C2C3CC(O)C(C3)N2C(c2sccc2Cl)=O)=O)c(C)c1C C#CC1(O)CC(C(=O)NCC(C)N(C(=O)CC2CCNC(=O)C2)C)C1 C(C(CC(=O)NC(C)CN1CCCC1=O)NC(c1nccn1C)=O)OC C(=O)(CC1COCc2ccccc21)N(C(C1CCC(C)(O)CC1)=O)CC.CC1CCC1 C1(C2(CNC(CNS(CC3CCC(C)C3)(=O)=O)=O)CC2)CCC2(CC2)C1 C(c1ccccc1C)=CC(=O)N(CC(CC)NC(=O)CC1CCN(C)C1)C C1(NC(c2n[nH]c(C)c2Br)=O)CC2(C1)CN(C(c1cn(C)nc1O)=O)C2 C12(NC(CC(C)OC)=O)CCCC(CN(C(c3nn[nH]c3Cl)=O)C1)C2 C12(C(=O)OC)CN(C(=O)C(c3cccc(C)c3)O)CC1CCCO2.C1CO1 c1(C(N2C(CNC(C3NC(=O)OC3)=O)CCC2)=O)cc(C(F)F)ccn1 C(CN=c1nc2scnc2c(N2CCC(C(C)(C)C)C2)[nH]1)(C(F)(F)F)OC CC(C)(F)C(C)(F)C(=O)NCCC1CC(C(N2CC3CCCCC3C2)=O)C1 CN1CCN(C(=O)C=Cc2ccccc2-n2cccn2)C(CNC(=O)CO)C1 C=CC(C)(C)CC(=O)NC1(CF)CCN(C(=O)C=CC(c2ccccc2)=O)C1 C(=O)(C(C)(C)S(C)(=O)=O)N1C2CC(NC(Cc3c(C)cccc3)=O)C(C2)C1 c1(OC)ncc(Cl)c(=NC2CCC(NC(C3COC(C)C3)=O)c3ccccc32)[nH]1 c1(CC)cc(C(=O)N(C(CC)C(=O)NC(C2CCC2)C2CC2)C)c(C)o1 C1(CC(=O)NCCCC=C)COCC(C)(C)O1.c1(C=O)sc(C2CC2)nc1C.N C1(C(=O)NC2CC(Cl)(Cl)C2)(NC(=O)CC2OCCO2)CCOCC1 C1(OC)CCC(C(=O)NCC2C3CN(C(c4cc(Br)cn4C)=O)CC23)CC1 CCCCCC(O)C(=O)NCC(C(C)(C)C)NC(=O)Cc1ccnc(O)c1 Cc1cc(C(=O)NC2CC(CNC(c3cccn(C)c3=O)=O)C2(C)C)nnc1C N1(C(CCN(C(C(CC#C)O)=O)CC2CC2)=O)CC23CCC2(COC3)C1 O=C1CC2(C1)CC(C(N1CCC(O)CC1C(=O)N)=O)C2.C1CC1C(F)(F)F c1(OC)c(NC(=O)CCC2CCC(NC(C3CCCOC3)=O)C2)cccc1F c1(SCCC)ccc([N+](=O)[O-])cc1C(=O)NC(C)C.C(=O)CC(CC)C(F)F C1(C(N(CCNC(C2C(CCC)C2)=O)CC)=O)CCC(C(F)(F)F)O1 O=C(CCN1CC(CC2CC2)C1)N=c1[nH]cnc2cc(-c3ccc(Br)cc3)sc12 N1(C(CN=S(C)(C)=O)=O)CCC(=O)NC2CN(C(=O)C(O)C3CC3)CCC12 S(=O)(=O)(c1cncc(Br)c1)Nc1scc(C(=O)Nc2cccc(OC)c2O)n1 N1(C(C2(CC#C)CCC2)=O)CCCC(N(CCF)C(c2cnnc(C)c2)=O)C1 C(=O)(C(CC)C(F)(F)F)NC1C(OC)CN(C(c2cc(CC)c(C)s2)=O)C1 N1(C(CC(CC)(F)F)=O)C(C)CC2CN(C(=O)C(C)C(C)C3CCCCC3)CC12 C1(CNC(C2(c3ccc(Cl)nc3)CCC2)=O)COC2(CCC2)CO1 c1(C(N2CC(C)C(n3cc(-c4ccccn4)nn3)C2)=O)cc(N)cc(O)c1 CCCC(C#N)C(=O)N1CC(OCCNC(c2[nH]cc(C)c2C)=O)C1 C=CC(C)(C)CC(=O)NC(CN(C)C(C1CCC(C)(C)C1)=O)CC c1(CCNC(=O)NC2(C)CCOC2)cc(C(F)(F)F)ccc1Br CC1CCCC(C(N2CCC(CC(=O)NCCN3C(=O)CCC3=O)C2)=O)C1 C(CCC(N)=O)(C(=O)N)NC(C)=O.C1(CC)CCCN(C(c2ncc(C)s2)=O)C1 C12(N(C)C)CCC(C(N3CC4(CCN4C(c4cccnn4)=O)C3)=O)(CC1)CC2 C1(N(C(CCC(=O)NC)=O)C)CCCN(C(=O)CC2CCNC(=O)C2)CC1 c1(C(N2CC(CCCCNC(C3(COC)CCOC3)=O)C2)=O)ccc(N)cn1 Cc1ccc(F)c(C(=O)NCC2CN(C(c3ccc(Br)nc3C)=O)CCO2)c1 c1(CNC(C2(Cl)C(C(C)=O)C2)=O)ccccc1CNC(c1cnsc1)=O c1(C(=O)NC2C(CNC(CCC#C)=O)CC2)ccn(C(C)C)c1C N1(C(c2c(C)cno2)=O)CC(CNC(c2occc2C(C)C)=O)CCC1C c1(Nc2c(OCC3S(=O)(=O)CCC3)cccc2)nc(Cl)nc2cc(I)sc12 C1(C(=O)N(CCCCCCNC(=O)Cc2csnn2)C)(OC)CCCOC1 C1(N2CCC(NC(C3C(=C)C3)=O)C2)CCN(C(C2CC2c2ccccc2)=O)CC1 C(CC(F)F)(C(=O)NCC1CCC(F)(F)C1)N(C)C(C1CCCC(C#N)C1)=O c1(CN(C)C)ccc2c(c1)CCN2C(C1CC2CC(=O)C(C1)C2)=O C1(NC(=O)OC(C)(C)C)CC(Sc2nc(-c3ccc(F)cc3)no2)C1(C)C c1(C(N(CCNC(C2CCC2)=O)CC)=O)ccc(C2(C)CC2(F)F)cc1 C1(NC(C)=O)(CNC(=O)Cn2ccc(=N)[nH]2)CCCCC1C CC1(C)NC(=O)CC1C(N1CCN(C(=O)C=Cc2nccs2)CC1CCO)=O Cc1cc(C(=O)N(CCC(C(C)C)NC(=O)CC2CCCC2O)C)c(C)nc1C c1(NC(C2N(C(C#CC)=O)CC(Oc3ccccc3)C2)=O)ccc(OC)c(O)c1 c1(C(N2CCC(C(CNC(CCC=C)=O)C)CC2)=O)c(F)ccc2nc[nH]c12 N1(C(CN(C)S(N)(=O)=O)=O)CCN(C(C2CCn3nnnc3C2)=O)C2(CCC2)C1 C1(NC(c2c(OC)ccs2)=O)CCN(C(=O)C(F)C(C)C)C1C(C)(C)C C1(NC(C(C)n2cccn2)=O)C2CC(O)C1N(C(=O)CSc1ccccc1Cl)C2 CC1CC(CNC(C2(C)CC2(C)C)=O)CN(C(=O)C(N2CCCCC2)C)C1 N1(C(c2c(Cl)cn(CC)n2)=O)CCC2(CCN(C(c3n[nH]c(=N)s3)=O)C2)C1 C(=O)(C(C)(C)C(C)NC(C1CC(CF)C1)=O)NCCc1ncn(CC)c1 C(C(CCNC(=O)C(C)(C)Cl)OC)NC(C(C)=C(CC)C)=O Cc1ccn2cc(C(=O)NCCC3CCCN(C(C4CCOC4C)=O)C3)nc2c1 C1(C(N2CCCC2)=O)(C(N2CC3C(C(F)(F)F)C3C2)=O)CCOCC1.CCO C1(N(C(=O)Cc2cc(C)nn2C)CC)CCCN(C(C2(O)CC2)=O)CC1 C1(C(N(C)CC2(CNC(CCc3ccc(C)s3)=O)CC2)=O)CCCCC1C1CC1 c1(C(=O)NC(CSCC)C(=O)NCCn2c(CC)cnc2C)nnccc1C N1(C(CCNC(=O)NC)=O)C2CCC1CN(C(c1cc([N+](=O)[O-])oc1C)=O)C2 c1(C(N2CCN(C(CNC(C)=O)=O)C(C)CC2)=O)cc(C)cc2c1NCCC2C CCCC(C)(O)CC(=O)NCC(F)CNC(=O)CCC1CCCCCC1 CCC(C)C(CC(=O)N1CCOCC(C)C1)NC(c1cnc(C)s1)=O N1(C(CN(c2c(C)cccc2Cl)CC)=O)CC2(CCN2C(C2CCCCO2)=O)C1 c1(C2(C(=O)NCC3CN(C(C(C#C)(C)C)=O)C3)CCC2)cc(F)ccc1F C1(NC(c2ccc(Cl)c(C)c2C)=O)CC2CCC1CN(C(C1CCO1)=O)C2 C1(C(N(C)CCOCCNC(=O)CC2CCSCC2)=O)CN2CCC1CC2 N1(C(c2cc(F)c[nH]2)=O)C2CC1CN(C(=O)C(F)(F)C(F)F)C2 C1(CC(=O)N(CCNC(=O)CC(C)SC)C2CC2)(COC)CCOCC1 CCC(Cc1ccccc1)CC(=O)N1CCCC(NC(=O)CN(C)CC)C1C C1(C(=O)NC2(c3ccccc3)CCN(C(=O)C(F)F)C2)CC2CCC(C1)C2O N1(C(CSc2ccc(C)cc2)=O)CCC(NC(C2CC(=C3CC3)C2)=O)CC1C Cc1c(Cl)[nH]c(-c2ncccn2)nc1=NCCCCCCCCc1ccccc1 Cc1[nH]nc2cc(C(=O)NCC(F)CNC(C3CCC(C#N)CC3)=O)ccc12 N1(C(C2CC(=C)C2)=O)CCN(C(CNC(C2CC2(F)F)=O)C(F)F)CC1 N#CC1CN(C(C2(NC(c3cccc(CO)c3)=O)CC(O)C2)=O)CCO1 c1(C(=O)NC(C)CC(C)NC(=O)Cn2ccnn2)cn(C)cc1C(F)(F)F C1(CNC(c2ccns2)=O)CCC12CCN(C(=O)C=CCO)CC2 N1(C(CC(=O)NC)=O)CCC2CCC(C1)N2C(C1(C)CCCNS1(=O)=O)=O C1(NC(c2cccc(C)c2)=O)CC12CCN(C(=O)C(C)Cn1cccn1)C2 c1(C(N2CCC(NC(C3(CCOC)CC3)=O)CC2)=O)cn2c(n1)C(C)CCC2 C(=O)(C(C)CC(C)C(C)=O)NC(CCOC)C(=O)NCC1CC2C=CC1O2 N1(C(CCNC(C)=O)=O)CCOCC1C(N1CCN(c2cncc(Br)c2)CC1)=O C1(CC(=O)N(CC(=O)NCCC2(OC)CC2)C)CCCC(=O)N1 N1(C(CCC(=O)N(C)C)=O)CC(NC(=O)CC2CCC(C)(O)CC2)CC2(CC2)C1 N1(C(C2(C=C)CCN(C(=O)CN3CCCCC3C)C2)=O)CCc2nccnc2C1 c1(C(=O)NC2CCC(NC(=O)CCc3ccncc3)C2)n[nH]c2c1CSCC2 C(C1c2ccccc2CCN1C(C1(F)CCCC1)=O)NC(C(CO)N(C)C)=O Cc1ncc(C#N)c(N2CCN(C(=O)Cc3cnc(C)s3)C3CC23)n1 CCCCC(C(=O)NC(CCOCCO)C(=O)NCC1CCC1(F)F)N(C)C N1(C(C(=O)NCCC2CN(C(C(C3CCOCC3)C)=O)C2)C)CCNC1=O n1(CCC)c(C)nc2ccccc12.N1(c2ccccc2)C(=O)CS(=O)CC1=O c1(C(=O)NCCCC2(NC(CCC3CC(OC)C3)=O)CC2)cnnc(C)c1C Cc1cc(O)ccc1C(=O)N(C(C)CC)C.c1(C(=O)N)cnn(C(C)(C)C)c1Cl Cc1cc(C(N2CC3CC2(CNC(C2CCSCC2)=O)C3)=O)cc(Cl)c1 N1(C(c2c[nH]c3cccc(C)c32)=O)CCOC2(CCCN(C(=O)C=CCF)C2)C1 c1(C(C)NCC(c2ccc(F)cn2)C)c(Br)cnn1C CNS(=O)(=O)NCC(=O)N(CCC(C)NC(C1CCOC1)=O)C C(=O)(C(C)CC(C)(F)F)NCC(CC)(C)NC(c1cccnc1)=O.C1CC1.O c1(C=O)cc(=O)ccn1C.C1(C)(COC)CC1C(=O)NCC1CCC1 C1(NC(C(CC2CCC2)OC)=O)CCC(C)(NC(c2cc[nH]c2)=O)CC1 C1(C(N2CCN(C3CCN(C(CC(=O)NCC)=O)C3)CC2)=O)CCC(=O)C(C)C1 C1(CC(=O)N(CC(C)N(C(=O)CN(C)C(N)=O)C)C)C(C)(C)C1(C)C C1(NC(CC(CCCC)O)=O)Cc2ccccc2C1NC(C1(C)CC1)=O c1(CSC)nc(C(=O)NC2CCC2C(=O)N(C)CCc2cnc[nH]2)co1 C1(N(C(C(C)N(C(C2CCCC(=O)C2)=O)CC)=O)C)CCCC(C)(C)C1 N1(C(c2ccc(OC)c(N)c2)=O)CC2CCC(N(C(=O)C=CCO)C)C2C1 CCC(C)(C#N)C(=O)N(CCC)C1CC1.c1(C=O)ccc(C(F)(F)CF)cc1.N c1(C(=O)NC(C2CCCCO2)C(=O)O)ccn(CC(F)(F)F)c(=O)c1 Cc1cc(F)ccc1C(=O)NCC1N(C(C2CC(F)CN2C)=O)CCC1(C)C C12N(CC13CCC3)C2=O.C(C)(C(=O)N1CC(CC)C1)SC.C(C)(C)C.C=O CC1CC(=O)NC(C(=O)NCCC2CCN(C(=O)CN3CCCCCC3)CC2)C1 c1(C(N2CC3C(NC(COC(CC)C)=O)(C3)C2)=O)cn2cc(C)sc2n1 c1(C(=O)NCCC#C)coc(CNC(c2cncn2C(C)C)=O)n1 c1(C(=O)NCC(CN(C(c2scc(COC)c2)=O)C)O)ccn2c1CSCC2 C1(OC)CCC(C(N2CC(O)(C(F)C(=O)NCC(=O)N(C)C)C2)=O)C1 C(=O)(C(F)CC(C)(C)NC(=O)C(C)O)NCCOCCC#C.CCC(C)C C(=O)(C(C)(C)CCCNC(c1cnc(Cl)s1)=O)NCCS(CC)=O c1(C(=O)NCCC2CC(OC)CN2C(=O)CO)ncc(Cl)cc1Cl C1(C(=O)NCC(=C)F)CC(C)CN(C(C2(CCSC)CCC2)=O)C1 N1(CC)CC(NC(=O)CC2(NC(=O)CC(C)C)CCCCC2)C(C)(C)C1.O N1(C(=O)CC2CCCCO2)CCC2(CCCN(C(=O)C=CC3CCCO3)C2)C1 N1(C(CCOCCC)=O)CCC(F)(C(=O)NCCC(C)C(C)C)C1 Cc1ccc(CC(=O)NC2(CNC(c3ccco3)=O)CCC2)cc1C CCC(CNC(c1nnnn1C1CC1)CC1CCCCC1)CC(C)C Cc1cccc(CCNC(c2ccc(C)s2)=O)c1.C1(CCC=O)CNC(=O)N1.N N1(C(c2cscc2OC)C(=O)NC(C(=O)OC)C)CCCC2CCCCC12 CN1CCC(C(=O)NC2CC(O)C2(C)C)(NC(=O)Cn2cnnc2)C1 Cc1nc2ncnn2cc1C(=O)NCC1CCCN(C(C2C(F)(F)C23CC3)=O)C1 C1(NC(C(C)(C)NC(CCCN(C(C)=O)C)=O)=O)CCCC1(C)O C(=O)(C(CC(C)C)NC(C1C2CC3C(C2)C13)=O)NC1CCN(C(C)=O)C1 c1(C(=O)NC(CNC(C(CC(C)C)C)=O)(C)C2CC2)sc([N+](=O)[O-])cc1Cl n1(C(C#C)CC)c(-c2cc(C)c(F)cc2Cl)csc1=Nc1ccc(Br)nc1 c1(C(N2CCC(N(CCO)C(C3CCSCC3)=O)C2)=O)n[nH]c(C2CC2)n1 N1(C(c2cc(C#N)sc2)=O)CCC2(C(=O)NCC3CC34CC4)CCCC12 C(=O)(CCCCCCNC(=O)C(C)NC(C)(C)CC)NCC(COC)(C)CO C(=O)(C1CCc2cccc(O)c21)NCC1N(C(C(C(=O)OC)(C)CC)=O)CC1 C(CCCCC(=O)NCC1(F)CCCCC1)NC(C1CC(C)(CC)C1)=O c1(OC)ccc(O)cc1C(=O)NCCC1CCN(C(=O)C(c2ccnn2C)C)C1 C1(CNC(C2CC(OCC)C2)=O)CCCCC1.C1(CC=O)OCCC1(C)C C(=O)(C1CCCn2nccc21)N1CCC2(CC(NC(C=C(CC)C)=O)C2)C1 C1(NC(COC(CC)C)=O)CC(C)(C)CN1C(=O)C1CC1.c1ncccc1O.C c1(C(N2CC(CNC(CN(CCC#C)C)=O)C(C)C2)=O)ccc(C2CC2)nc1C c1(C(N(C)CC2CCN(Cc3ccc(C)s3)C2)=O)ccc(Br)c(F)c1F n1(CCC(=O)NCC2CN(C(CSCC(C)C)=O)C(C)C2)cnc2ccccc12 C1(C(=O)OC)CCN(C(=O)C(C2(C)CC2)NC(=O)Cn2nccn2)C1C N1(C(Cc2ccc(OC)nc2)=O)CC2(CCC2NC(=O)CCc2nncs2)C1 c1(C(=O)N)cc(C(F)F)ccc1Cl.Cc1occc1C(=O)NCC1(O)CCC1 c1(C(N2CCCC(C)(NC(C(C=C)O)=O)C2)=O)cccc(S(C)=O)c1 c1(C(N2CCC(C)(CC(=O)N(c3c(OC)cccc3)C)C2)=O)cccc(C)c1F C(=O)(C(C)CCCCCC)N1CC(C(C(=O)NC2(CC#C)CCC2)O)C1 Cc1cc(N2CC(C(C)NC(=O)C(C3CCOCC3)F)C2)nc(C(C)(C)C)n1 C(CCC(C)C(=O)NCCCN1CCN(C(c2n[nH]cc2Cl)=O)CC1)OC N1(CCCCCNC(c2ccccn2)COC)C(=O)c2ccccc2C1=O c1(C(N(CCNC(=O)C(O)c2cnc[nH]2)CC)=O)[nH]cnc1C CC1(C)CN(C(=O)CCC2CC2(F)F)CC1NC(c1cc[nH]n1)=O C(=O)(CC1=CCN(C(c2[nH]nnc2C2CC2)=O)CC1)NC(C(=O)OC)CCF C1(C(=O)NCCCN(C(CCc2c(C)noc2C)=O)C)COC2(C)CC1C2 C=C=CCCC(=O)NCC1CC(OC)CN1C(c1cc(COC)cn1C)=O C(=O)(CC(C(F)(F)F)n1cccn1)N.O=C(COCCCF)NC1(CC)CC1 N1(C(C=CC=CCC)=O)CCCC1C(C)NC(=O)COCC(C)C Cc1cc(NCCC(=O)N)cc(C)c1.C12(CC)CCC1CCN2C=O.C(C)(C)C C(=O)(C1=Cc2ccc(Cl)cc2OC1)NCC1(C)CCN(C(C2CC2Cl)=O)CC1 c1(C(N2CCC(NC(c3cnc(C)[nH]c3=N)=O)C(C)C2)=O)cc2c(s1)CCCC2 C1(N(C)C)(C(=O)NC(C2CCCC2)CNC(=O)CCc2cnn[nH]2)CCCSC1 Cc1c(NC(=O)CC(C)CNC(=O)CCCc2cnn[nH]2)cccc1C#N c1(CC(=O)NCCCOCCN(C(C=COCC)=O)C)cc(C)nn1C N1(C(CCCCNC(C)=O)=O)CC(C(=O)NCC(C)(O)C(C)C)CC1(C)C c1(C(N(CCCOCCN(C(=O)C=Cc2ccsc2)C)C)=O)cc(F)c[nH]1 Cc1cc(O)c(C(=O)NC2CCCCN(C(c3sccc3C#N)=O)C2)nn1 CC1(C)COCC(C(=O)NC2CC(F)CN(C(C3(O)CCCCCC3)=O)C2)O1 C(=O)CC(F)(F)C(F)(F)F.C1(C(N(C(C)C)CC)=O)CC1C(F)(F)F.N C1(C(=O)NCC2CCS(=O)(=O)C2)COCCN(C(c2cccc(F)n2)=O)C1 c1(C(N(CCCNC(C2(C)CCOC2)=O)C2CC2)=O)csc2cnccc12 c1(OC)ccc(C)c(C(F)(F)F)c1.c1(C(C)=O)ccnn1C1CCC1.C(=O)N c1(C(N2C3C(CNC(CNC(=O)NC)=O)C(C3)C2)=O)cc(N)nc(Cl)c1 c1(C(N2CCN(C(COCc3n(C)ncc3)=O)C(CO)C2)=O)ncc(C#N)cc1Cl C1(NC(CCCC=C)=O)(CNC(=O)CC2CCC(OC)CC2)CCC(F)(F)CC1 C1(NC(C=C(C)Cl)=O)CN(C(=O)Cn2ccc(=N)[nH]2)C2CCCCC12 CC1(C)OCC2CC12C(=O)NC(CNC(c1c[nH]c(=N)nc1O)=O)C1CC1 C1(CCNC(c2cnc(C3CC3)[nH]2)=O)CCN(C(c2c[nH]nc2Br)=O)CC1 C(CC1=CCN(C(=O)C(C)Sc2ccc(C#N)cc2)CC1)NC(CC=CCC)=O C1(NC(COCCCOC)=O)CCC2CC1CN2C(c1cc(C)c(C)cc1N)=O N1(C(C(C(C)C)C)=O)CCCC2(C1)CN(C(c1cnc(O)s1)=O)C2 c1(CC=O)cccc(C(F)F)c1.CC(C)(C(=O)NCC=CC)c1cncnc1 c1(OC)nc(C(=O)N(CC(O)CNC(C2CN(C)C2)=O)C)cc(O)n1 N1(C(CCCn2c(C)ncc2)=O)CC2C(CC(N3CCN(CCF)CC3)=O)C2C1 N1(C(c2c(Cl)ccc(C)c2)=O)CCC2(CCC(NC(c3cccc[n+]3[O-])=O)C2)C1 C(C(CO)NC(=O)CC1CCN1C(=O)CSC1CC1)OCC N1(C(C(C(C)C)N(C)C)=O)CCCC(NC(c2c(F)cc(F)cc2Cl)=O)CCC1 C1(NC(CC(C)N2CCCC2=O)=O)CC(F)CN(C(C2(C)COC2)=O)C1 Cc1ncccc1NC(C1C(CN)CCN1C(=O)CN1CC2CCC1C2)=O C(=O)(C1CC(=O)Nc2ncccc21)N(CCC(C)NC(=O)CS(=O)(=O)C1CC1)C c1(OC)ccc(C(=O)NC2CCCN(C3CCNC3=O)CC2)cc1Cl Cc1cccc(N(C(=O)CCCCCBr)Cc2ccc(C3CCCN3)cc2)c1Cl CC(C)S(=O)(=O)CC(=O)NC1CC12CCC2.c1(C=O)cc(C(C)C)cnc1O.N Cc1[nH]nc(C(F)(F)Cl)c1C(N1CCC(NC(c2n[nH]cc2Cl)=O)CC1)=O c1(CC(=O)N(CCN(C(=O)CCF)CC)CC)c[nH]c2ccc(OC)cc12 O=C(C1=CC2(CCOCC2)C1)NCC1CCCN1C(C1CCCC2(CCC2)O1)=O C1(C(=O)NC(C)C)CC(C)N1C(=O)Cc1cc[nH]n1 Cc1cc(CC(=O)Nc2cccc(F)c2Br)ccc1C(F)(F)F c1(NC(C2C(NC(c3cc(O)ccc3I)=O)CCC2)=O)c[nH]c2ncc(Br)cc12 C1(NC(Cc2c(CC)cccc2)=O)CN(C(=O)Cc2[nH]cnc2C)CC12CCC2 CCC(F)(F)C(=O)NCCCN(C(=O)CC1CSCCS1)C1CC1 c1(C(=O)OC(c2ccc(OC(C)C)cc2)C(F)(F)F)ccnc(F)c1Cl C#Cc1ccc(F)c(C(=O)N)c1.c1(C(N(CC(C)C)C)=O)ccn(C2CC2)n1 CCCCCC(O)CC(=O)N1CCCC(NC(c2c(C)coc2CC)=O)C1 c1(CN2C(CNC(CC)C(=O)OCC3CC3)CC2)c(OC)cccc1F C(=O)(C(CNC(c1nc[nH]n1)=O)CC(C)C)N(C)Cc1c(C)noc1C c1cc(F)cc(Cl)c1.Cn1nccc1CC(=O)N(C1CCN(C(=O)C)C1)CCO.O CCC(CC)C(C)C(=O)N1CC=CC(NC(c2cc3nccnc3[nH]2)=O)C1 c1(C(C)C)ccccc1-n1cc(CN(C)CCc2cccnc2Cl)nn1 CC(C)(C)CC(F)C(=O)NC1COCC1NC(=O)CCn1cnnn1 c1(C(=O)NCCC(C)NC(C2CCC(C)(C)OC2)=O)cc2ccncc2[nH]1 C1(C)(C(N(C)Cc2cncnc2)=O)C=CCN1C(C1CC12CCC2)=O C1(NC(c2c(C)ocn2)=O)CC2CC(NC(C3CC4(CCCC4)C3)=O)CC2C1 C1(CC(=O)N(C2(C(N3CCC(N4CCCC4)C3)=O)CC2)C)CCN(C)C1=O C(=O)(N=c1[nH][nH]c2ccc(Br)cc12)C1CCC(NCc2c(OC)ccc(Br)n2)C1 C(=O)(CS(=O)c1ccc(Cl)cc1)N1C(CNC(CCOC)=O)C(C)(C)CCC1 C1(CNC(C(CCC)OC)=O)CCC2(CCN(C(c3cc(C)cs3)=O)CC2)CO1 c1(CC)nonc1C(=O)NCC(CC)NC(=O)CCOC1CCC1 c1(NC(c2nnnn2C2(C)CC2)COCC=C)ccccc1OC.C1CCCO1 N1(C(C(C)CC2CCCC2)=O)CCC(CNC(C2C3CC(=O)CC23)=O)C1(C)C c1(C(=O)NCCC(C)NC(C2CC2C2CCCCC2)=O)ccc(Cl)c(F)c1O C(CCN(C)C)(C(=O)NCC1(O)CSC1)NC(C(CN(C)C)O)=O c1(C(=O)NC2C(CNC(c3cn(CCC)nn3)=O)CCC2)c(C)cccc1C C1(OC)CN(C(c2cc(OC)nn2C)=O)CC1NC(c1ncccc1C)=O Nc1cc2c(cc1C(N1CCC3(CCC3NC(C3CC3CF)=O)CC1)=O)OCO2 C(=O)(C(F)C(C)(F)F)NCCCC(C)(C)NC(c1nn(CC)c(O)c1)=O c1(C(=O)NCC(c2cn(CC)nc2)=O)cccn2cncc12 N1(C(c2cc(=O)cc[nH]2)=O)CCC2CCC(C1)N2C(=O)C(F)=CC1CC1 C1(CC(=O)NC2C(C)(CC)C2)CN(C(c2cnn(C)c2OC)=O)CCCO1 Cc1cc(C(N2CC(NC(=O)CC3CCOC3(C)C)C3(CC3)C2)=O)cc(C)c1F C1(C)(CC)CC(C(=O)N)CCO1.C1CCCCN(C(C23C=CC(CC2)C3)=O)C1.C N1(C(CONC(C(C(=O)OC)OC)=O)=O)CCc2nocc2C1 C(=O)(C(F)CC(C)(C)NC(c1coc(N(C)C)n1)=O)N(C1CCCC1)CCC CC(C)CCC(F)C(=O)N1CCCC(C)(C(=O)NCC2CC(=O)N(C)C2=O)C1 C1(C(CNC(c2c(C)scn2)=O)C)CCN(C(=O)C(C)Cc2cnco2)CC1 C1(CC(=O)NCCN(C)C(c2ccc(-n3cccn3)cc2)=O)CCC(=O)NC1 c1ccccc1C=O.C12(C(N(CC)C3CC3)=O)CCC(C1)OC2.CCC=O.N c1(C(N2C3CN(C(Cc4ccn(C)c4)=O)CC2CC3)=O)cn(C)c2ncccc12 C1(CC(=O)NC(CC)C(F)(F)F)CN(C(C2CCCSC2C)=O)CC12CC2 c1(C(=O)NC2CC2C(=O)NCC(O)CO)ccccc1C(F)(F)F c1(CNC2C(C(=O)NC(CC)C)C2)ccc(F)cc1O c1(CC)c[nH]c2nc[nH]c(=NCC3CN(C(=O)CCC(C)(F)F)CC3C)c12 c1(OC)cncc(C(=O)NCCN2CCCCC2)n1.C(C1CCCC1)=CC=O.N C1CC2CC1N(C(=O)C(F)CC1CCC1)C2.c1(NC(C)=O)cccc(C=O)n1.N C1(CC)CN(C(=O)CCC2CCOCC2)CCC1NC(c1c[nH]cc1C)=O C(=O)(C1CCCc2sccc21)N1C2CN(C(c3cncc(F)c3Cl)=O)C(C2)C1 C1(OCC)CN(C(c2ccccc2)=O)CC1.n1(CC=O)ncnn1.C1(S)CC1 N1(C(CCNC(=O)NCC)=O)CC(C)(C)CC1C.c1(C=O)cncs1.N C(CCCN=[N+]=[N-])NC(C(C1(C)CC1)NC(c1c(CC)ncs1)=O)=O N1(C(c2cc(OC)cc(C3CC3)c2)=O)CC(C)N(C(=O)C(F)=C2CCC2)CC1C CC1(C(F)(F)F)CCN(C(C2(CO)CC2(F)F)=O)CC1 c1(C(N2CCC(CC)C2CNC(=O)CC(C)C(C)(C)C)=O)ccn2nccc2n1 Cc1c(C(N2CCC(C)N(C(c3cc(Br)co3)=O)CC2)=O)sc2nccn12 C(CCN=C(NC1CCC1)N1CCC(O)C(CO)C1)OCC(C)C C1(CNC(c2c(C(C)C)c[nH]n2)=O)CCCCC1.C1(CC=O)CCC(C)O1.C Cn1c(C(F)F)nc2cncc(C(=O)NC3CC3)c12.C1(C=O)CC1(C)C(F)F C1(C(N2C(CC(N3CCC(C=O)C3)=O)CCCC2)=O)CC2(CCC2)CO1.CC.O C(C1CCN(C(=O)C(C)(C)CCN(C)C)CC1)=CC=O.N1(CCC)CCCC1=O CCCCCC(C)(CC)C(=O)NCC(CC)n1cccn1.c12occc1NC2=O N1(C(C=CCCC(C)C)=O)CC2CC1C2C(=O)NCCN1CCCCC1C C(CC(C)(C)NC(C1(C)CCCS1)=O)N(C(=O)CCc1cccs1)C c1(OC)cccc2c1C(C(=O)N1CCC3(CCCN(C(=O)OC(C)(C)C)C3)C1)CC2 N1(C(Cc2n(C)ncc2)=O)CCC2(CC2C(N2CCCC(C(=O)OC)C2)=O)C1 C1(C=O)CC(=O)NC(=O)C1.C(CC(C)(C)C)NC(C(c1ccc(N)cn1)C)=O.N c1(C=O)cc2ccccc2o1.C1(F)(CNC(C(C)C)=O)CCC1.C(=O)(CC)N c1(CN2CCC(N(C(C3(C(C)C)CC3)=O)C)C2)ccc(F)c(Br)c1 C1(C(N(CC(C)NC(c2cccc(C#N)c2F)=O)C)=O)CCc2n[nH]cc2C1C C(CCCN=c1cc(Cl)nc(C2(C)CC2)[nH]1)NC(C1C(C(=O)OC)C1)=O C(CS(=O)(=O)CC(=O)N1CCC(F)C(NC(c2cnn(CC(C)C)c2)=O)C1)OC C12(C(N3CCC(C(C)C(=O)N(C(CC4CC4)CO)C)C3)=O)CCC(C)(CC1)C2 C1(C(N(C2CCN(C)C2)C)=O)C(O)CCN1C(=O)CCn1cnnn1 C=CC(C)(C)CC(=O)NCC1(C)CCC(NC(c2cc(C)c(C)cn2)=O)C1 c1(C(N(C(CC)CNC(=O)C(C2CCOCC2)F)C)=O)coc2c1COC2 C1(COC)CCN(C(C2CCC(=O)N2C(C)C)=O)C1.C(=O)C(C)(C)CF.C C1(N(C(=O)CC2CCC2(C)C)CCC)CCN(C(c2cc(CN)co2)=O)CC1 n1(CC)c(C(=O)NC(C)C(C)NC(C2(C)CC2)=O)cnc1O C=CC(C)CC(=O)N(CCCCCNC(C1CCC1c1nncn1C)=O)C N1(C(C(F)OC)=O)CCN(CCNC(=O)Cc2cncn2C2CC2)CC1 N1(C(CN(C)C(N)=O)=O)CCCC(NC(=O)Cc2ccc(-c3nnco3)cc2)C1 C1(C(=O)NC2C(CC(=O)N(C(CC)C)CC)CCCC2)CN2CCN1CC2 c1(OC(CC)C)ccccc1C=CC(=O)NCC(F)CNC(c1ccccn1)=O N1(C(CC=C)=O)CC2(C(=O)NC(c3nccn3C)C)CC1CCO2 CC1(C)CCC(C(N2CCC(NC(c3ccc(C4CC4)s3)=O)C2)=O)CC1 C=CCCCCCCC(=O)N1CCC(C(=O)NCc2cc(C)[nH]n2)CC1CC C1(NC(c2cnc(C)[nH]2)=O)COCCC1NC(=O)CC(C)O.C(=O)N(C)C.N c1(OC)cccc(-c2cc(C(=O)NCC(C)NC(C3(C)CCCC3)=O)on2)c1 n1(CCN(C)C)cc(C(=O)N(C(C)C2CC2)C)cn1.C1(C=O)CC1(F)F.N Cc1cnc2ccccc2c1C(N1CCOC2CN(C(=O)C3=CCSC3)CC12)=O Cc1nn(C)c(C)c1C(N1CCC(C(=O)NC2CC2)C1(C)C)=O Cc1nc2c(Br)cc(C(=O)NC(C)(C)CN(C)C(c3ccccc3)=O)cc2o1 c1(CC(c2ccccc2)NC(=O)NC(C)CCN2CCCC2=O)ccc(O)cc1 C(C)(CCC1CC1)(c1nnnn1-c1ccccc1)NCCCC(C)C.C1CC1.C C(C(=O)N(CC(C)N(C(=O)CCc1cccnc1Cl)C)C)(C(C)C)OCC(C)C C1(C)(C(N(CCCCCCNC(C2N(CC)CC2)=O)C)=O)CCCN(C)C1 C1(C(N2CCC(NC(C(C(C)(C)C)=O)=O)(CO)CC2)=O)CCc2nnnn2CC1 C(=O)(C#CC1CCOC1)N(CC(CNC(COc1c(C)ccc(C)c1)=O)O)C N1(C(C(C)Cc2ccnn2C)=O)CC2(C1)CN(C(c1c[nH]c(=O)cn1)=O)C2 c1(C(=O)NC(C#C)C)n[nH]c2cc(C(N3CCC(=O)C(C)C3)=O)ccc12 C1(C(=O)NC(CCC)CO)CCN(C(=O)C(=O)Nc2c(C)cccc2C)C12CC2 C=CCCCCC(=O)N1CCCC(F)(C(=O)NCc2cc(F)cc(F)c2)C1 C1(NC(c2n(CCOC)ncc2)=O)CC(NCc2c(Br)cnn2C)C12CCC2 C(=O)(C(O)CC(F)(F)F)NC12CC(NC(c3cc(C)nnc3O)=O)(C1)C2 N1(C(C(c2ccccc2)NC(CCC(CC)OC)=O)=O)CCCC(C2CCC2)C1 C1(CC(=O)NC(C)C2CC2)CC2(CCC2)CO1.C12(C(=O)N)CCC(CC1)C2 N1(CCC)CCC(C(N2CCC2CNC(C2CC3(C2)CC3F)=O)=O)CC1 C(=O)(C1CCc2ccccc21)N1C2C(CNC(C(CC(C)C)C)=O)C(CCC2)C1 CCC(C(=O)NC1COCCN(C(C2CCCCN2C)=O)C1)C(F)(F)F N1(C(c2c(C)ccs2)=O)CC2CCN(C(c3cc4c([nH]3)CCCC4)=O)C(C2)C1 C(CC(CC)C(=O)NCCCN(C)C(c1ccc(C2CCC2(C)C)cc1)=O)=CC c1(SC)ccc(C(=O)NC)c(C)c1.C12CC1CN(C(c1cc(C#N)c[nH]1)=O)C2 Cc1nc(S(=O)(=O)NC2CC2C2(C)CCOCC2)c2n1CCCC2 n1(CCC(N2CCC(CNC(c3c(C)non3)=O)C2)=O)c(C)nc2ccccc12 c1(OC(C)C)ccc(C=O)c(Cl)c1.CCC(C)(C)C.C1(=CC=O)CCCC1.N Cc1cc(C(c2nnnn2C)NCCCP(C)(C)=O)cc(C)c1.c1cccc(Cl)c1 c1(C(N(CC(C)(C)NC(c2cc(C)[nH]n2)=O)C)=O)ccc2[nH]c(=O)cnc2c1 C1(C)(CC)CC(C(N2CC3(C2)CN(C(=O)CO)C3)=O)CCO1.c1cc(C)on1 c1(C(C(=O)NC2CC(CNC(CCC=CC)=O)C2)(F)F)cccc(Br)c1 c1(C(=O)N)cnc(Cl)n1C.C1(CC(=O)NCCC2CCC2)(OCC)CCC1 c1(C(=O)NCC2(C)CCN(C(C(CC)C)=O)C2)cc(-c2c[nH]nc2C)ccc1F CC1C(CC(=O)NCC(O)CN(C(=O)CCCc2cnn[nH]2)C)C1(F)F c1(CC(C)NC(N2C(C(=O)NC)CC2)=O)ccc(O)cc1 c1(C2(C(=O)N)CCC2)ccc(Br)cc1.CC(C)C=CC(=O)NC1(C)CC1 c1cccc(C#N)c1.C(CSC)(C(=O)NCC1CCC1)OC.C(=O)(CC)N C12(OC)CCC(CNC(=O)OCC3CCN3C3CCCCCC3)(CC1)CC2 O=C(C1=COc2ccccc2O1)NCC1CC(NC(=O)C(F)C2CCC2)CCO1 CCCC(C(O)C(=O)NC1(C)CC(N(C)C)C1)NC(C1CN(C2COC2)C1)=O CCC(C)CCC(=O)NCC1(C)CCCN(C(=O)CC2(C#N)CC2)C1 N1(C(c2c(C)scc2)=O)CC2CN(C(=O)CCS(C)(=O)=O)CC12 c1(C(=O)NCC)cc2ccncc2[nH]1.C1(C(=O)NCCN2CCCC2)CCCC1 C1(CNC(C=Cc2ccc(C)o2)=O)CN(C(C2CC(Cl)(Cl)C2)=O)CC1(F)F CCC(O)C(C)(C)C(=O)NCC1(NC(=O)CC2CC3(CCC3)CCO2)CC1 Cc1cc(C(N2CC(NC(c3cncnc3)=O)C(O)C2)=O)ccc1N(C)C C1(C(N2C(C)(C3(C)CC3)CCC2)=O)CC2CCC1N2C(=O)CCCC(=O)C1CC1 C1(C(N(CC(CC)NC(=O)Cc2cnc(Cl)cc2C)C)=O)CC2C(C1)C2(F)F N1(C(Cn2nnc(=N)[nH]2)=O)CCCC(CNC(=O)CCC2CC2(Cl)Cl)CC1 c1(C(N2C(CNC(C3C=C(C)CS3)=O)CN(C)CC2)=O)ccc([N+](=O)[O-])n1C C1(CC)CN(C(=O)C(C)(C)CF)CCN1C(c1cnn(C2CCCCC2)c1)=O c1(CSC)cccc(C(=O)NC2C3CC2N(C(=O)C=CS(C)=O)C3)c1 c1(C(=O)NC23C(CN(C(c4c(C)cc(CC)o4)=O)C2)C3)cc(F)cc(O)c1N C(CCC(=O)NC1CCCC1CC(N1CCC(C(=O)OC)C1)=O)OCCC C=C1CCC(C(N2CCC(OCCNC(=O)C=CC=C(Cl)Cl)C2)=O)CC1 C(=O)(CCC(F)(F)F)NCCC(C)N(C(=O)CC1CCCS1(=O)=O)C CCCC(C#N)C(=O)N1CCCC1CCCNC(=O)C=Cc1cccc(OC)c1 N1(C(CC2OCC(C)(C)C2)=O)CCCCC(CNC(c2ccc(C#N)[nH]2)=O)C1 C#CCC(C)(C(=O)N1C2CSCC1C2)NC(=O)CC1CCCNC1=O c1(C(=O)NC(CC)CNC(=O)C(C(C)C)C2CCC2)cc(COC)ccc1F N1(C(CC2(C(=C)F)CCC2)=O)C2CCC1C(C(N1CC3C(C(N)=O)C3C1)=O)C2 Cc1ccc2ncnc(N3CCC(C(C)NC(C4(F)CCC4)=O)CC3)c2c1 c1(C(=O)N)ccc(C2CC2)nc1O.N#CC1(C(=O)NC2CC(CC)C2)CCOC1 CC(C)CC(CC(C)C)C(=O)N1CCN(C(=O)Cn2ccc(=N)[nH]2)CC(O)C1 c1(C(=O)NC(CNC(C(C=C)c2ccccc2)=O)C)ncc2ccccn12 C1(NC(c2n(C)nnc2)=O)C=CCCC1C(N1CCC(C(N)=O)C1)=O c1(OCCC(=O)NC2C(NC(CC=CCC)=O)C2)ccc(C)cc1 c1(C(=O)NCC(CCOC)NC(C(CCCC)C)=O)cc(Cl)c(Cl)cc1C N1(C(C(C)NC(CC)=O)=O)CC2(CNC(c3n[nH]c(C)c3F)=O)CCC1CC2 C(=O)(CC(O)CC(C)C)N1C(C(N)=O)CCC1C1CC1.C1CCC1.C1CC1.C C1(c2nnnn2C)(NCc2c(C)n(C)nc2)CCCCC1C1CCCCC1 C#Cc1cccc(C(=O)NC(CC2CCC2)C(=O)N2CCC2C2CCC2)c1C CC(CCCCNC(=O)COc1ccccc1F)NC(=O)C=CC1CCCN1C c1(C(C)C)nc(NC(c2cccnc2)C2CC2)cc(N2CCCC(CO)CC2)n1 C1(C(=O)N)C2CCC(F)(F)C12.c1cccc(-c2cn(C3CN(CC)C3)nn2)c1.C C#Cc1cn(C)nc1C(=O)NCC1(CO)CCN(C(=O)CS)CC1.C1CC1 C1(C(=O)N)CC12CC(F)(F)C2.Cc1ncc(C(=O)NCCC)n1-c1ccccc1 c1(C(=O)NC2C3OCC(NC(CN4CCC(C)C4)=O)(C3)C2)ccc(Cl)c(F)c1O CCCS(=O)(=O)c1ccc(-c2cc3c[nH]nc3cc2C(=O)Nc2ccns2)cc1 c1(C(N(C(C)CCNC(c2cc(F)cc(F)c2)=O)C)=O)cc(Cl)c(F)cc1N c1(CNC(COC)(C)C(N)=O)nc(C)c(C)nc1C c12cccc(c1)NC2=O.C1(OC(=O)CO)CCC(Oc2nccs2)C1 c1(C(N(C2CCC(NC(=O)Cc3cscn3)C2)C)=O)cccc2nonc12 O=C(CC(F)(F)C(F)F)NCC1CN(C(=O)CCc2ncccn2)C2CC12 C(=O)(C(C)C(O)C(C)C)N(CC=CC(=O)Nc1ccc(C#C)nc1)C C(=O)(C(C)=NOCC#N)NCCCOCCC(=O)NCCSCC#C C12CN(CCCO1)CC2.CN1CCC(CO)C1 N1(C(c2n(C(CC)C)ncc2)=O)CCC(NC(c2cc(C)n(C)n2)=O)CC(O)C1 CCCCC(CO)NC(C1C=CCN1C(C1C(C(C)=O)C1(C)C)=O)=O.CS C1(NC(=O)CC2CN(C(=O)CCCn3cccc3)CCO2)CC2CC1CC21CC1 c1(C(=O)N)cccc(N)c1.C(C(=O)NC1CC(C)C1)(C1CCC1)OCC C(=O)(C(C)(C)CCF)N1C(C)(CC(=O)N)CC1.C(=O)(CC)N(CC)CC c1(OCCN)ccccc1C#N.C1(OC)CCCC(CC(N2CC(C)(OC)C2)=O)C1 C(C)(CC(F)(F)F)NC(c1cc(C)n(C)n1)=O.C(=O)(C(C(C)(C)C)N(C)C)N N1(C(C2N(C(C=CC3(C)COC3)=O)CC23CCCC3)=O)CCC2(CCC2)C(O)C1 C=CC(CCC)CC(=O)NCC(CC(C)C)C(=O)NC1CC1C(C)(C)C C1(C(N(C)Cc2cc(C)n(C)n2)=O)CC2CCC1N2C(=O)C(C)NC=O c1(SC)cc(C(N2CCC(C3CCCN3C(C3CCC3(F)F)=O)CC2)=O)n(C)n1 N1(C(c2cc(C#N)on2)=O)CCN(C(C2CC2[N+](=O)[O-])=O)CC1CC(F)F N1(C(COCCCC(C)C)=O)CCC2CN(C(=O)C(C)CCN(C)C)CC2C1 C1(NC(Cn2c(C)ccn2)=O)C2CC1N(C(=O)C(O)C(C)c1ccccc1F)C2 O=C1CC(CC(=O)N2CC(NC(C34CCC(C3)C4)=O)C3CCCC23)=NN1 C#CCC(O)C(=O)N1CC(NC(C2(C)CCCCC2)=O)CC1CO C1(CC)CC(C)CN1C(C1OCCC1CNC(C12CC(C)(C1)C2)=O)=O C(=O)(C(O)C(CCC)NC(c1ccc(C)nc1O)=O)NC(C#C)(C)C1CCCC1 C=CC1CN(C(=O)CSC(F)(F)F)CC1NC(c1n[nH]c(CC)c1C)=O C1(S(=O)(=O)N2CCC(CC(=O)Nc3ccccc3C)C2)(CC=C)CC1 C1(CC(=O)NC(C)C(F)F)CCCN(C(C23CC(C#N)(C2)C3)=O)CC1 c1(OCC)cnc(C(=O)NC(CO)CCC)cn1.C1(C(=O)N)CC1C(F)F C1(C(NOCCC)=O)CCC(C)N1C(=O)C(O)CC1CCCC1 C(=O)(C(O)CC(F)(F)F)NCC=CCNC(c1c(N)c(Cl)ccc1)=O CC1CC=C(C(=O)Nc2ccc(-c3cn(Cc4ccc(Br)s4)nn3)cc2)CC1 Cc1cncc(C(=O)NC(C)CCC(=O)N2CCC(CC(C)O)CC2)c1 C1(NC(C2CC(CN(C)C)C2)=O)CN(C(=O)COC2CCC2)CC12CC2 c1ccc(C=CC(=O)O)o1.C1(C(N)=O)CC(C2CC2)C1 C1(N(C(C2CCC(C)O2)=O)C)CN(C(C2CC2C(F)(F)F)=O)CCC1C C=CC(C)(O)CCCC(C)C(=O)N1CCC(N(C)C(C2(SCC)CC2)=O)CC1 N(C1CCc2cc(C(=O)O)ccc21)C(=O)NCC(C)Oc1ccccc1 CC1c2ncc(C(=O)NCc3cnn(C)c3)n2CCN1C(C1(C)CCCN1)=O C1(NC(c2ncc(C)nc2)=O)C(C)CCN(C(=O)CN2CSCCSC2)C1C C(C)(CCCC(=O)N1CC(C)C(F)C1)NC(c1c(C)oc(CO)c1)=O Cc1nc(C)c(C(=O)NC(C)CCCCNC(c2cc(C)c(C)o2)=O)c(C)n1 CCC(F)(F)CC(=O)NCC1CC(F)CN1C(=O)CCCn1cccc1 c1(OC)ccc(CO)cc1C(N1CC(C)C1)=O.C1(CC(=O)N)CC12CCOCC2 C1(C(N2CCC(C(N)=O)C2)=O)C2CCC(C2)N1Cc1cncc(Cl)c1Cl c1(OC)ccc(C)nc1C(=O)NCC(O)CN(C)C(c1c(C)n[nH]c1C)=O O=C1CCCC(C(N2CCC2C(N2CC(CC(F)(F)F)C2)=O)=O)N1 c1(CC(C)C)ccnc(C(=O)NC2C3CN(C(=O)CC4CCOCC4)CC23)c1F c1(C(C(=O)NC2COC2)N(c2ccc(CC)cc2)C(C)C)ccc(Br)c(Cl)c1F Cc1cc(C(N2CCC(O)(CNC(C3CCC(C#N)CC3)=O)C2)=O)c(F)cc1F Cc1cnc(NCc2cncn2C(C)C)c(S(=O)(=O)NCC(C)C#N)c1 N1(C(C(CCSC)NC=O)=O)CCC(CNC(=O)C=C2CCSCC2)C(C)C1 N1(C(C2(CC)CCNC2=O)=O)CC2CCN(C(=O)CC(F)(F)C(F)F)CC(C2)C1 C(=O)(CCC(=O)NN(C)C)NCCCC(C)NC(c1c(C(C)C)ccc(C)c1)=O C=C1CCC(C(=O)NCc2cc(C(=O)NCC3CCOC3=O)n(C)n2)CC1 c1(OC(C)C)ccc(C(N(CCCN(C)Cc2ccnc(F)c2)C)=O)cn1 N1(C(c2n(CC)nnc2)=O)CC2CC(C(=O)NOCCOC)(C2)C1 c1(CN2C(C(=O)Nc3ccc(C(C)C)nc3)CC3CC32)ccc2n[nH]cc2c1 C1(CC)CCCC(NC(c2ccn(CCNC(c3cnnc(O)c3)=O)c2)=O)C1 C1(C(=O)NCCCC2(NC(c3c(C)noc3)=O)CC2)CCCCN1N=O C1(NC(C(C)CCO)=O)CCCCN(C(c2c[nH]nc2OCC(F)F)=O)C1 N1(C(c2c(CC)c(C)sc2)=O)CCN(C(=O)Cc2coc(C)n2)C(CC)C1 O=C(C#CC1CCOC1)N(CC=CC(=O)N1CC(O)CO1)C1CC1 CCC(CC)C(C(=O)N1CC(F)CC1CN(C)C(C1CC(C)(C)CCO1)=O)OC c1(COC)n[nH]c(CNC(=O)C=CC(C)(C)NC(=O)CN=[N+]=[N-])n1 Cc1c(C(=O)N(C2CCCN(C(=O)Cc3ccno3)C2)C)cncc1Cl C(=O)(C1CCCn2ncnc21)N1CC(C(Cn2cc(CNC(CC)=O)nn2)F)C1 C1(C(=O)NC(CCC)C)CC12CN(C(C1CN(C)CCO1)=O)C2 C(C)(CCC(=O)NC(C)C(CO)NC(=O)CSCc1ccccc1C)SC C1(CNC(c2c(CC)scn2)=O)CN(C(c2nc(Cl)sc2C)=O)CCC1C c1(C(=O)NCCN(C(c2cncn2C(F)(F)F)=O)C2CC2)ccccc1 C1(CNC(C2CC2CF)=O)COCCN1C(c1ccc(CO)s1)=O c1(C(=O)NCC2N(C(c3nc(CC)oc3C)=O)CC=C2)cc(C)ccc1.O C1(CNC(c2cc(C)c(C)[nH]2)=O)CN(C(=O)Cn2ccsc2=N)CC(C)(C)O1 C(C)(C(C)C(=O)Nc1cncc(Cl)c1)NC(C1(OC)CCCC1)=O c1(C(=O)NC2CCN(C(CCc3cnc(C)o3)=O)C2)ccc(S(C)(=O)=O)cc1Cl C12(NC(Cc3c(C)n[nH]c3)=O)CCCCC1CN(C(C1C3CCCCCC13)=O)C2 N1(C(c2cn(CCC)nn2)=O)CCN(C(C2CCCN(C(N)=O)C2)=O)C(CC)C1 c1(C(=O)NC(C)(C)CCCNC(=O)Cc2cnoc2)cncc2nc[nH]c12 C#CCC(CC(F)F)NC(=O)CC(C)NC(=O)C(C)(O)C(C)C CC1CC(Nc2nc(=N)[nH]c(=NCCC3CC(F)C3)[nH]2)c2ccccc21 c1(C(N2CC(F)(CNC(C3(CC=C)CCCC3)=O)C2)=O)cc(O)nc(Cl)c1 N1(C(=O)OC(C)(C)C)CC=CC(NC(=O)CC2(c3ccccc3)CCCC2)C1 c1(C(=O)NC(C)CCNC(=O)C(c2ccccc2)O)ncc(F)cc1F N1(C(C(CC)N(C)CC)=O)CCC(F)(C(N2CC(NC(=O)C3CC3)C2)=O)C1 C(C1CCCCCC1)=CC(=O)NC1CC2(C1)CC2NC(c1ccoc1)=O CC1C(NC(c2ncccc2F)=O)CCCN1C(C1OCCCO1)=O CC1(C)CC(CNC(C2CC3CC3N2C(C2CC2c2ccccc2)=O)=O)CO1 S(=O)(=O)(c1ccc(NCC2(C)CCOC2)c(Br)c1)NCC1CCCCN(C)C1 c1(OCC)cccc(C(=O)NCC(C)NC(=O)CNC(N)=O)c1 C(=O)CCC=O.CC(C)CC(=O)NCC1CC1.C1CC(=O)N1.C(C)(C)C.N c1(SC)ccccc1C(=O)NCCCNC(=O)C(F)(F)c1cccnc1 c1(N(CCCNC(=O)CC2CCC(F)(F)CC2)CC)nc(OC)cc(OC)n1 C1(CNC(CCC#C)=O)CC12CCN(C(=O)COC(=O)CO)CC2 c1(C(C)C)ccc(C(=O)NC23CC(C(=O)NCCC4CCCCC4)(C2)C3)o1 O(C1CCCc2ccccc21)c1c(C)cc(-c2ccc(Cl)cc2)cc1 c1(OC)ccccc1C(C)C(=O)NCC(O)CCNC(c1ccccn1)=O N1(C(=O)OC)CCC(F)(c2ccccc2OC)CC1 c1(OC)ccccc1SCC(=O)N.C1CCN(C(=O)CCn2cc(C)cn2)C1.C c1(NC2CC(NCC3C(F)C3)C2)cc(N2CCCC2)nc(C)n1 c1(CNC(C2(c3ccc(Cl)cc3)CCNCC2)=O)ccc2ccc(O)nc2n1 C12(C(=O)NC(CNC(CC(CC)C(C)C)=O)C)CCC(C)(C(=O)O1)C2(C)C C1(CC=C)CC(O)CC(CC(=O)NC2CC(F)CN(C(=O)C(CC)CCC)C2)O1 C1(NC(C2=CC(C)(C)C2)=O)CC2CC(NC(c3cc(O)cc(Cl)c3)=O)CC2C1 c1(C=O)cc2c(ncn2C)s1.Cc1nn(C)c(C(F)F)c1C(N1CC(C)C1)=O.N S(=O)(=O)(C(C)CN=c1[nH]c(=NCC2OCCOC2(C)C)c2ncccc2[nH]1)NC C(=O)(C1=CC(O)C(NC(=O)CC2(C#N)CCC2)C1)N(CCO)CC N1(C(=O)C=CC2CC2)CCC2(CC1)CC2NC(C1(CC(F)F)CCOCC1)=O CC1CN(C(=O)COC2COCCN2C(=O)OC(C)(C)C)C(C)CN1 C1(CC(=O)N(C(C=C)C)C)C2CCCC2N1C(C1CC=CCC1C)=O CCCC(CCCNC(=O)C(C)(C)C1CCCC1)NC(=O)C1=NNC(=O)C1 N1(C(C(C)C)=O)CCCCC(CNC(=O)CC(C)c2ccccc2)CC1 c1(C(=O)N)cncc(P(C)(C)=O)c1.C1(CNC(CC2CC(C)C2)=O)CCOC1 C1(C(N2C(CN(C(c3c(C)nn(C)c3)=O)C)CC(F)C2)=O)CC2CCC(C1)C2O N1(C(CC)=O)CCN(C(=O)CC2CNC(=O)O2)CC1C1CCCC1.C(=O)(NC)N CC12CN(C(c3cc(Cl)ns3)=O)CC1CN(C(=O)C(c1ccccc1)F)C2 N1(C(c2cc(CC(C)C)on2)=O)CCOCC(CNC(=O)C(C)(F)F)C1 Cc1cc(C#N)cc(C(=O)NC2CCCCN(C(C3CC3C(C)O)=O)C2)n1 N1(C(C2C(C)CCS2)=O)CCN(C(c2cc(N3CCCC3)ncn2)=O)CC1 C1(NC(C(C=C=C)C)=O)CCC2(CC1)CN(C(=O)C(C)C)C2 C=CCCC(C(=O)NCC(C)(F)F)NC(c1c[nH]c(C#N)c1)=O N1(C(c2nc(C)n3c2cccc3)=O)CCCC2(CCN(C(=O)C3=CCCC3)C2)C1 CCCCC(O)C(C)C(=O)N1CCC(CF)(NC(c2ccc(OC)s2)=O)C1 C1(O)(C(C)NC(c2ccn(CC(C)C)n2)=O)CCN(C(C23CC2C3)=O)CC1 N1(CC)CCC2(CCC2)CC1.c12cc(nc(C)n1)N1CCCC(C1)N2 C(=O)(CCCCCC(C)O)N1CCCN(C(CC2(OC)CCC2)=O)CC1C N1(C(COC(C)=O)=O)CC(CNC(C2CCCC(=O)N2C)=O)OC(C)(C)C1 N1(C(CC=CC=C)=O)CC(C(=O)NCc2ccccc2Cl)CCC1C C1(C(=O)NCCCN(C)C(C2CCN(S(C)(=O)=O)C2)=O)CCC(=O)O1 Cc1nn(C2CCCCO2)c(C)c1C(=O)N.C1(C(N2CCC2)=O)CC2(CCC2)CO1 C(=O)(C(CCO)N(C)C)NCCCOCCN(C(c1ccn(CCC)n1)=O)C c1(C(=O)NCCNC(C(C)NC(=O)NC)=O)cnc2c(Br)cccn12 Cc1cc(NC(C2(C)CN(C(=O)Cn3ccnn3)C2)=O)nc(C)c1 C1(CN(C(=O)CNC(N)=O)C)CCN(C(c2occc2Br)=O)C1 C(=O)(C(O)CC(F)(F)F)NCC(CC)NC(=O)Cc1csc2nc(C)cn12 CC1CC(N=c2[nH]nc(C(C)(C)C)s2)CCN1C(C1CC(C2CC2)=NO1)=O c1(CN2C(C(c3ccc(-c4ccncc4)cc3)=O)CCC2)c(F)ccc(Br)c1F CCCC(CNC(=O)C(C)(F)c1ccon1)C(=O)N(C)CC1CN(C)CCO1 C1(C(=O)NCC2C(C(=O)NCC(CCC)O)OCC2)CCCCN1C C(=O)(C1CCCc2n[nH]cc21)N(C1CCCN(C(CN(C)C2CC2)=O)C1)CCO c1(C(=O)NC(CC)(CNC(=O)Cc2nc[nH]n2)CC)cnn2c1OCC2 CCCC(C(O)C(=O)NCC1(C2CCC2)CC1)NC(=O)C(O)C(C)(C)C C=CCC(C)(CC)C(=O)N1CC(C(=O)NC)C2(CCC2)C1.n1(C2CC2)ccnn1 C1(C(=O)NCC2CCN(C(c3ccnnc3O)=O)CC2)CCn2nnnc2C1 C1(F)(CNC(C2CCCCC2O)=O)CCCN(C(=O)CCn2cncn2)CC1 C1(CNC(C(C)(C)C#N)=O)CC2CN(C(c3cnc(O)c(F)c3)=O)CC12 Cc1nc2cccnn2c1C(=O)N(CC(O)CN(C(=O)CC1CCSCC1)C)C C1(C=O)CCCC(C)(C)CC1.C1(N(C(CNC(=O)NC)=O)CC)CCCCC1 C1(NC(c2cccc(Cl)c2Cl)=O)CCCCC12CCCCC2 Cc1cc(C(=O)NC2CCC(C)CC2)c(C)n1C1CCOC1.C1(F)(C=O)CC1 C1(CNC(c2c[nH]nc2Br)=O)CN(C(=O)C#CC2CCC2)CC12CC2 N#CC1(C(=O)NC2CCC(NC(c3ccco3)=O)C2)CC=CC1 C(C1CCCC1)=C(C)C(=O)NC1CC(C)(NC(C2(F)CCOC2)=O)C1 C1(NC(c2c(C)nc(C(C)C)s2)=O)CCN(C(C)C(N)=O)CC1C c1(-c2scc(C(=O)NCCCCN(C(C(CC)(C)O)=O)C)n2)ccc(F)c(F)c1 c1(C(=O)NC2CCC(NC(c3cccc4[nH]ncc34)=O)C2)onc2ccccc12 N1(C(c2c(C)[nH]c(=N)s2)=O)CC2CCCC(CNC(C34CC3CNC4=O)=O)C2C1 Cc1nc2cncc(C(=O)NCCC(C)NC(C34CCCCC3OCC4)=O)c2[nH]1 N(C1c2ccccc2CC1NC(=O)C1=CS(=O)CCC1)C(C(CC)C#N)=O N1(C(C=C(COC)C)=O)CC2(C1)CN(C(=O)CC1CN3CCN1CC3)CCO2 C(N=c1[nH]nc(C#N)s1)C1(O)CCCN(C(C(C)OC2CCCC2)=O)C1 c1(C(C)C(=O)NC2CC(OCC(=O)NCC3SCCS3)C2)ccn(C)n1 c1(OC)ccc2cc(C(N3CCC4(C3)CN(C(=O)NC(C)C)C4)=O)c(C)nc2c1 c1(C(N(C2CCCN(C(C3CC4CCC4C3)=O)C2)C)=O)ccc2c(c1)CCCO2 C(=O)(CC(O)CCC)NCCCN(C(CC=C)=O)C1CC1 C(C(C(=O)NC(COC)COC)NC(c1[nH]ccc1C)=O)SCC C1(CNC(c2nc(C)oc2)=O)CC2CCC1N(C(c1nc3cccnc3s1)=O)C2 c1(CC(=O)N(CCC(C(C)C)NC(CC(CC)C)=O)C)ccc([N+](=O)[O-])cc1F C=C(C)CN=c1[nH]c(=NCc2nnc3ccccn23)c2[nH]ccc2[nH]1 c1(C(=O)NCC2CC(NC(C(C)CF)=O)C(O)C2)nn(C)c2ccccc12 N1(C(C)=O)CC2(CCC(C(=O)NCC=O)O2)C1.c1ccc(Cl)cc1C(C)=O.N c1(C=O)ccc(C=O)cc1.N1(C(CSCCOC)=O)CC(O)C1.C1CC1.C C#CCC(C)(CC)C(=O)NC(CC)CC(=O)NCC1CCCC1(C)C c1(C(N(C2CC3CC2N(C(C2CCCCCCC2)=O)C3)C)=O)ccc(Cl)c(F)c1 O=C1CCC(NC(=O)C(c2ccccc2)NC(=O)C(O)C(F)(F)F)C(=O)N1 CCC(CC)CC(F)C(=O)NCC(C)NC(=O)CCc1cn(C)cn1 CC(CCCC(=O)N(CC(F)F)CCO)NC(C1CC(N=[N+]=[N-])C1)=O N1(C(C2C3CN(Cc4c(OC(C)=O)cccc4)CC32)=O)CC(C)N(C)C(C)C1 CCC(CCCC(=O)N1CCOCC1C(=O)NC)NC(c1coc(N(C)C)n1)=O C#Cc1cc(NC(c2cncnc2)c2nnnn2CC)cc(C#C)c1 C=CCC(C(=O)NCCSCC(=O)NCc1cc(C)on1)NC(C)=O c1(C2CCN(CC3C(NS(C)(=O)=O)CCCC3)CC2)nc2c(s1)CCCC2 C#Cc1ccc(C(=O)NC2C3CC(NC(=O)C(C)OCC(C)C)CC23)nc1 C(C(=O)N1CCCCCO1)(c1cccs1)NC(CC1CCC(C)(C)C1)=O c1(-n2c(C(CC)n3cccn3)nc(C3CC34CC4)n2)cc(Cl)cc(Cl)c1 C(=O)(CCCCCCN=[N+]=[N-])N1CC2C(CNC(CSCC#C)=O)(CCCC2)C1 C(=O)(C1OCCc2c(Br)cccc21)NC1C(CNC(CCC)=O)C1 c1ccc(Cn2cc(CO)nn2)cc1.C1(OC)CCC1CC=O.CCN(C)C c1(OC)cc(Cl)ncc1C(=O)NC1CN(Cc2ccc(F)cc2Br)CC1O c1(CC)nn[nH]c1CNC(=O)Cc1cccs1.C12(CC=O)CCCC1C2.N Cc1c(Br)noc1C(=O)N(C(C)CNC(=O)C(c1cnn(C)c1)C)C CC(=O)NNC(=O)CCCc1ccc(Cl)cc1 CC(C)CC(C)(CNC(c1ccoc1)=O)NC(c1cc(CC(C)C)[nH]n1)=O C1(N(CCC(=O)NCC(F)(F)F)C)(COC)CCC1 c1(C(N2C(CC(=O)Nc3cccc4nsnc34)CCC2)=O)cccc2ncsc12 C1(NC(=O)CC2CCOCC2)C2CCN(C(C34CCCCC3C4)=O)CC12 C1(CC(N2C(C=C)CCC2)=O)CCCN(C(C2(C)CCCO2)=O)CC1 CCCC(CCC)C(=O)NCCC1(NC(=O)CO)CCC1.c1c(C)nn(C)c1C C(=O)(C#CC1CCCCC1)N1CCC(O)(C(C)NC(c2ccc(OC)nn2)=O)C1 C(=O)(CS(=O)(=O)C(C)(C)C)N(CCCCCNC(C(c1c(C)cccc1)C)=O)C C1(NC(C(C)(C)NC(C)=O)=O)C2CN(CC(Cl)=CCl)CC12 c1(NC(C2CC2C(=O)NCCCn2cccn2)=O)cccc(-c2cncnc2)c1 N1(C(C(C(CC)C)O)=O)CCC(O)(C2(NC(=O)CCCCCC(C)O)CC2)CC1 CC(C)(C)C(CNC(c1cscc1C#N)=O)NC(C1CNC(=O)C1)=O CCCC(CNC(C1CC(=O)N(CC)C1)=O)C(=O)N1CCC(CC)(CC)C1 C(=O)(CC(C(F)(F)F)NC1CC1)N1CC(CCNC(=O)CCc2cscn2)C1 c1(CNC(C2CN(c3cccc(C#N)c3)C2)=O)cn2cc(Cl)ccc2n1 c1(C(=O)NCCC(C(C)C)NC(c2nccc(CC)c2)=O)coc2ccccc12 c1(C(C)C)ccc(C(=O)NCC2(NC(=O)Cc3cscn3)CCC2)cn1 N1(C(C2C3CN(C(CCC(CC)OC)=O)C2C3)=O)CCn2nc(C)cc2C1.C1CO1 N1(C(C2CCC(CC(C)(C)C)CC2)=O)CCOCC(C(=O)N)C1.C(C)(C)C(=O)O CC(C)C(C)NC(=O)C=CCC1(NC(c2ccon2)=O)CCC1 C1(C#N)(C(N2CC3C(CNC(c4c(SC)scc4)=O)(CC3)C2)=O)CCCCCC1 C(=O)CCO.C(=O)C(F)(F)F.C1(C=O)CC1C=O.C#CC.CC=CC N1(C(C2C(C(N)=O)C2)=O)CC2OCCN(C(=O)CCCc3ccsc3)C2C1 Cc1cc(N)ccc1C(N1CCOCC1CCNC(=O)C#CC1CCC1)=O N1(C(Cc2cccc(OC)c2)=O)CCC(NC(=O)Cc2ccccc2F)C1(C)C C1(N(C(CC2(C=C)CC2)=O)C)CC2CCC(C1)N2C(=O)CO.C1CCOCC1.C C(CO)(C(=O)NCCC1(C(=O)NC2CC(O)C2OC)CCC1)OC c1(CCn2cc(C(C3CCCCC3)NC3(CO)CC3)nn2)c(F)cccc1Cl Cc1cc(C)c(C(N2CC3CN(C(=O)CC(C)Oc4ccccc4)C3C2)=O)c(C)c1 C1(CNC(CC(C)n2cccn2)=O)CN(C(=O)CS(C)(=O)=O)C2COCC2O1 C1(C(=O)NCCCN(C(=O)C=CBr)CC)CN(C)CC1C(F)(F)F CCC(C)C(=O)NC1C=CC(C(=O)NCC2(CF)CCC2)C1 c1(CNC(C=CCN(C(=O)C)CC#C)=O)ccccc1.C(C)(=O)OC CCCCCCCCC(C)C(=O)NC1CC2CN(C(=O)C3=CCCCC3)CC12 C(=O)(C(O)C=C)N(CCC(=O)NCc1n[nH]c(CC)n1)CC=C Cc1ccsc1CNC(c1conc1C(C)NC(c1ccccn1)=O)=O Cc1cc(C(=O)NC(C)(CNC(C2CC3CC2CO3)=O)CO)c(C)s1 c1(C(=O)Nc2nc(C(=O)Nc3ccc4c(c3)OCO4)cs2)cc(Br)cc(Br)c1F C1(C(=O)NCCN(CCOC)C(c2csc(C)c2)=O)CCCS1(=O)=O n1(CC(=O)O)cc(Br)cc(C(N2CCC(N3CCCOCC3)C2)=O)c1=O Cn1nccc1C(=O)NC1(C(=O)NCCOCC2CC2)CSC1 Cc1sc(S(N)(=O)=O)cc1C(N1CC(CNC(=O)CCCC#N)CC1C)=O c1(CC(C)C(=O)NCC(=O)NCCOCCC=C)cccs1 N1(C(C(C)SCCCC)=O)CCC(CC(=O)NCc2ncc(Cl)cn2)C1(C)C CC(C)(C)C(C(=O)NCc1ccnc(Cl)c1)NC(c1cc[nH]n1)=O C(=O)(C(C=O)OC(C)(C)C)NC1(CCNC(CCOCC)=O)CC1 c1cc(F)cc(F)c1.C1(C(=O)NCC2CCC2)(CC)CCC1.C(=O)CC.N C1(NC(C(=O)c2ccco2)=O)(CF)CCN(C(=O)CC2(CO)CC2)C1 CCS(=O)(=O)CCCNC(=O)CC(F)(F)c1ccnc(Br)c1 c1(C(N2CC(C(=O)OC)N(C)CC2)=O)sc(=NCCc2ccccc2)[nH]c1C c1(N2CCC(N(C(C3(CC)CCCCC3)=O)C)C2)ncc(C#N)cc1F C#CCC(C(=O)N(CC(C)(C)C#N)C)NC(=O)C(COC)N(C)C N1(C(C=Cc2ccc(C)s2)=O)CC2CN(C(=O)CCc3cnn(C)c3)CC12 c1(CC(=O)N(C2(CC(=O)NC(CO)C(N)=O)CC2)CC)csc(C)n1 C1(NC(CCc2cc(C)no2)=O)CN(C(=O)Cc2csnn2)C2(CCCCC2)C1 C1(NC(c2c(C)nc(CCC)o2)=O)CN(C(=O)C(C)CSC)CC12CC2 C(=O)(C1Cc2ccc(F)cc21)N1C(CNC(CN(C(=O)OC)C)=O)CC1 c1(C(=O)NC(CC)CN2CCOCC2)ccnc2c(C(F)(F)F)cccc12 c1(CC(N2CCCC(N(C(c3ccnnc3)=O)CC)C2)=O)ccccc1NC c1(NCCOC)nnc(C2CC(SC(=O)CC(C)C)C2)s1 C(=O)(CCNC(=O)C=CC=O)NCCC(C)N(CCC)C.CCC.N c1(-n2cc(-c3cncc(CNC(C(N)=O)=O)c3)nn2)ccc(Cl)c(F)c1 CCC(CO)(C(=O)NC(CNC(=O)Cc1cc(F)cc(F)c1)C1CC1)OC C12(CNC(CC(CC)CC)=O)CCCC1CCN2C(c1cc(C(F)(F)F)n[nH]1)=O C1(C(=O)NCc2nnc(O)o2)C(C2CC2)CCN1C(c1ccnc2cc[nH]c12)=O N1(C(c2cc(C)[nH]c2)=O)CC2CCC2(C(=O)N(C2CCC3(CC2)CC3)C)C1 N1(Cc2c(C)ncs2)Cc2ccc(O)cc2CC1C(N1CC2C(C1)C2(F)F)=O c1(OC)ccc(-c2noc(CCC(=O)NC(C(=O)O)c3nn[nH]n3)n2)cc1OC c1(C(N2CC(N(C(C(C(C)C)O)=O)C)C(O)C2)=O)cc2cc(Br)ccc2o1 C#Cc1cn(C)nc1C(=O)NCC=CC(=O)NCC1(O)CC(O)C1 CC(C)CC(C)(O)C(=O)NCCN(C(=O)C(CC(F)F)c1ccccc1)C(C)C c1(CC)ccccc1C(=O)NCC(CNC(C1CC(F)(F)CS1)=O)OC c1(C(=O)NCC(C)(CO)NC(C(C(C)C)SC)=O)ncc(C2CC2)cc1F c1(C(=O)NC2C(CNC(c3c(F)ccc(C)n3)=O)C2)ccc2sncc2c1 N1(C(CS(CC)=O)=O)CCC2(CC1)CC(NC(=O)Cc1cnc(C)[nH]1)CCO2 C1(NC(COCCCOCC)=O)CC2CC1CN(C(c1oc(C)nc1C)=O)C2 c1ccc2c(c1)CN(C(=O)C(C)(C)C#N)C2.c1(CCC)ccc(C(=O)NC)cc1 c1(C(=O)NC2C=CC(C(=O)NCCCN(CC)CC)C2)ccc(O)cn1 N1(C(C)=O)CC(C(=O)Nc2ccc(-n3nccn3)nc2)Oc2ccccc21 n1(CC)cc(NC(c2c[nH]nc2CNC(C2COCCO2)=O)=O)c(C#N)n1 c1(OC)cc(C(=O)NC2CN(C(c3nccnc3Br)=O)CC23CC3)cc(F)c1 c1(OC)ncc(NC(=O)CN(C(=O)CCOCC(C)C)CC(C)C)cc1C C1(CC)(NC(=O)C(C2CCCCC2)OC)CCCN(C(=O)C(C)(C)CO)C1 C(C(C(C)C)NC(=O)CCc1cnccn1)NC(C(c1cnn(C)c1)OC)=O N1(C(c2c(C)n[nH]c2)=O)CCOC(CCNC(=O)C(=C2CCCCC2)F)C1 c1(C(N2CCC(CCC)C2)=O)cccc2ccc(Br)cc12 c1(CNC(C=CC)=O)ccc2c(c1)CCCC2NC(c1cncc2ccsc12)=O C1(NC(C2OCCN(C)C2)=O)CCN(C(C2CC2(C)C)=O)CC1(C)C c1(OC)cc(F)c(CN2CC3C(C2)N3C(c2cc(C)nc(Cl)c2)=O)c(F)c1 C1CCCN1C=O.C(=O)CC.CCC(C)C.C(C=O)N(CC=C)CC=C(C)C Cc1ccc(C)n1CC(=O)NC1CCCC1NC(=O)COC.c1ccccn1 C1(CNC(c2c(C)scc2)=O)CCCN(C(=O)CCCn2cncn2)C1 C(=O)(C(C)(C)C(F)(F)F)NCC1CCN(C(C(N2CCSCC2)C)=O)CC1C C1(C)(NC(CC2CCN(C(C(C)NC(C)=O)=O)CC2)=O)CCC(C)=C(C)C1 c1(C(N(C)Cc2ccncn2)=O)coc2c1CN(C(=O)CCNC(=O)CO)C2 N(C1CC(C)n2ccnc21)C(C1(n2cc(CCNC(C)=O)nn2)CC1)=O C(c1cccc(F)c1)=CC(N1CCC(O)C1)=O.C(=O)(C=CC=O)OCC CC1CN(C(c2cc(Cl)ncc2N)=O)CCS(=O)C1 c1(C(C)N(C(=O)CC)CCO)cn(CC2CCOCC2)nn1.C(=O)C(F)(F)F Cc1c(CC(=O)NCCCC(C)NC(C2CCCCN2S(C)(=O)=O)=O)ncn1C C1(NC(C2N(CC#C)CCC2)=O)CC(C)N(C(=O)CCc2ccc(OC)cc2)C1 c1(C(N2C(C(=O)NCc3nccc(C)c3)CCC2)=O)cc(N(C)C)ccc1F CC1(C)CC(CN=c2[nH]c(-c3cccc(Cl)c3Cl)cs2)CCO1 CC1(C)CCC(C(=O)NCC=CCNC(=O)COC2CCCCCC2)O1 N=c1[nH]c(=NCC#CCCO)[nH]c(=NCC(C(F)F)c2ccccc2)[nH]1 C1(C2(O)CCOCC2)(C(N(CCCN(C)C(c2ccc(F)c(Cl)n2)=O)C)=O)CC1 C1(CC)C(=O)NCCN1C(=O)CCNC(c1ccc(C#N)s1)=O CCC(CC(F)F)C(=O)NCC1CC2COCC2N1C(c1cc(CO)c(C)o1)=O C(=O)(CC(F)(F)C(F)F)NC1(CO)CCCN(C(CCC(=O)NC)=O)C1 c1(C(N2CCCC(O)(CCNC(CCC#CC)=O)C2)=O)ccc(S(C)=O)cc1 C1(C(C)(C)NC(C(C)OC)=O)CCN(C(c2ccc(C(C)C)cn2)=O)CC1 c1(OC)ccc(NC(C2CC(NC(=O)CCc3cc(C)no3)C2)=O)c(C)c1 c1(C(N(CCC(=O)OCC)CCC(=O)NC)=O)c(Br)cnn1C CC1(C)CCCN(CC(N2CCCCC2c2n[nH]cc2C(N)=O)=O)C1 c1(C(=O)OC)cccc2c1CN(C(C1CC13CCN(C(C1CC1F)=O)C3)=O)CC2 c1(C(=O)NC(C)CNC(c2ccc(CCO)cc2)=O)cnc(=NCCF)[nH]c1 c1(SC)ccnc(N(C(C)C)CC2CCCN(C(c3c[nH]c(Br)c3)=O)C2)n1 CCN=C(NCC1CCCN(CC)C1)NC1CCCN(c2cc(C)nn2C)C1 C1(NC(C2(CC=C)CC2)=O)CN(C(C2(C)CCN(C(C)=O)C2)=O)CC1F C=CCCC(C(=O)N1CC(OC(=O)N(C)C)C1)NC(=O)C=Cc1ccsc1 CC(C)C(C)(C)CNC(C1CCC(NC(=O)C(c2ccccc2)C)CC1)=O N1(Cc2ccc(NC(C3(C)COC(c4ccccc4)O3)=O)o2)CC2C=CC1CC2 c1(C(N2CC=CC(O)C2)C(=O)NC(c2ccccc2)C)cc(F)c(F)cc1F C(=O)(C#CC1CCOC1)N(CCCCNC(c1cccc(-c2nc[nH]n2)c1)=O)C C12(CNC(C3C(CC)C3)=O)CCC(CC1)N2C(c1ccnc(C)c1)=O N(C1CCC(NC(=O)C(C)C)c2ccccc21)c1nc(C#N)cc(C)n1 N1(C(Cc2c(C)non2)=O)CC2(CCN2C(C2CC2c2ccsc2)=O)C1 CN1CCC(NC(c2cc(CF)on2)=O)C12CCCN(C(=O)C(F)(F)C(F)F)C2 N1(C(CCC=CC)=O)CC2(CCCCN(C(C3CCNC3=O)=O)C2)C1 C1(CC(=O)OCC)COCCN1C(C1CCCN(C(N)=O)C1)=O C1(NC(C2CCN(C(C)=O)C2)=O)CC2CN(C(=O)CC3NC(=O)NC3=O)CC12 CC(C)(C)C(=O)C(=O)NCCCN(C(=O)CC1CC2CC2C1)CCO C1(CC(=O)NC(CN(C(c2c[nH]c(=NCC)s2)=O)C)C)C2CC3CC(C2)CC1C3 c1(C(=O)NCC23CC2CN(C(C2(Br)CC2)=O)C3)noc2c1CCCC2 c1(C(CNC(C(N2C(C(C)(C)CN)CCCC2)=O)=O)=O)ccc(F)c(F)c1F CCC(C)CC(=O)NC1CC(CNC(=O)C(O)CCc2ccccc2)C1 c1(CC)ncoc1C(N1CCC(C(C)(C)NC(=O)C(C)c2cncs2)C1)=O N1(C(c2cc(COC)on2)=O)CCC(C2CN(C(C3CCCOC3C)=O)C2)CC1 c1(C(=O)OC)ccncc1NC(c1cc(-c2ccc(=N)[nH]c2)[nH]n1)=O n1(CC(N2CC(NC(CC(C)N(C)C)=O)C(CO)CC2)=O)ncc2cccnc12 c1(OC)ccc(C(N2CCCC(C(=O)Nc3cncc(C)n3)C2)=O)c(OC)n1 Cc1cc(C(=O)NCC(C)(C)NC(=O)C2=CC3CC=CCC23)cc2nn[nH]c12 C1(C(=O)NCC(CNC(CCOCCOC)=O)(C)F)CC=C(C)CC1 c1(C(=O)N)cccc([N+](=O)[O-])c1.c1(CC(=O)NCC2(C)CCC2)ccco1 Cc1cccc(C(=O)N(C)CC2CN(C(=O)C(c3cccc(F)c3)O)CCO2)c1 C(=O)(C(O)CCC(C)C)N(CCN(C(c1ccc(COC)[nH]1)=O)C(C)C)C O=C1CS(=O)(=O)CC(C(=O)NC2CC3CCC2CC3NC(C2CCC2)=O)N1 C1(C(C(=O)NCCN(C(C(F)OC)=O)CCOCCO)C)CCCCCC1 Cc1nc2ccccc2cc1C(=O)NC1CCCCN(C(=O)C(O)C2CC2)CC1 C=CCC(C)(CC)C(=O)N1CC2CC(C1)N(C(c1cc(C)n(C(F)F)n1)=O)C2 C1(CC)CN(C(=NCc2ccc(C)cc2)NCC(=O)NC(C)C)CCN1C c1(C(=O)NCC(CCNC(=O)C2=C(C)CC2)OC)ccc2ccccc2c1 c1(NC(CC(CC)C)=O)[nH]nc(C(C)(C)C)c1C#N C(=O)(C(CC(F)F)NC(C1OCCC1(C)C)=O)NC(CCC)CCO N1(C(CCCOC(CCC)=O)=O)C2CCC1N(C(C1OCCN(C)C1=O)=O)C2 C1(C)(C(N(C(CNC(CN(C(COC)=O)C)=O)C)C)=O)CC(C)=NO1 n1(CC)nc(C)c(C(N2CCOCC(NC(=O)C(O)c3ccco3)C2)=O)c1C N1(C(c2cc(CC)on2)=O)CC2CC(NC(=O)CSC(F)(F)F)CC2C1 N1(C(c2ccc(C)cc2C)=O)C(CNC(c2scnc2C)=O)CC2COCC12 C(=O)(C(C)(CC)CO)N(C1CC(NC(CC(OCC)OCC)=O)C1)C C12(C(=O)NCC34N(C(COCCCC)=O)CC(C3)C4)CCC(CF)(C1)OC2 c1(C(N(C2(CC(=O)N(CC(COCC)O)C)CC2)C)=O)conc1C c1(CCN(c2ncnc(NC3C(C=C)COC3)c2C)C)cccc([N+](=O)[O-])c1 Cc1nc2c(o1)CCCC2CC(=O)NC1(c2cncc(Br)c2)COC1 C1(CCNC(c2cc(C3CCC3)[nH]n2)=O)CSCCN1C(=O)CCc1ncco1 n1(CC)nc(C)c(C(N2CC(N(C(=O)C(C)c3ccsn3)C)C3(CC3)C2)=O)c1Cl C(C(CC(C)C)C(=O)NCC(O)C(F)F)NC(c1cccc(CC)n1)=O N1(C(C(C)=C(C)C)=O)CCOC2(CCC(NC(C3CC(O)C3)=O)CC2)C1 CC(C)CC(F)C(=O)N1CC(O)(C(C)(C)C)C1.N1(C2(C(=O)N)CC2)CCCC1 CC1CCOCC1C(=O)NCC1(O)CN(C(c2ccc(C(N)=O)s2)=O)C1 c1(C(C)=O)cc(C(=O)Nc2ccccc2C=O)n(C)c1.N1(CCC)CCOCC1.N c1(C(N2CCCC(N(C(=O)C3=CC(C)(C)C3)C)C2)=O)cc(O)nc2ccccc12 Cc1noc(Cl)c1CCC(N1CCC(NC(=O)CCN2CCN(C)CC2)CC1)=O c1(C(=O)NCC2OCCN(C(C3N(N=O)CCCC3)=O)C2)cccc2occc12 c1(NC2(C3CCN(C(C(CC#C)(C)C)=O)CC3)CC2)cc2c(cn1)C(=O)CCC2 N#Cc1cnc2c(Cl)cc(Cl)cc2c1NCc1ccncc1 C12(C(=O)NCCCCCNC(c3cncc(Cl)c3)=O)CCCCC1CCC2 c1(-n2cc(C34N(C(C5CC6CCC5O6)C)CC(C3)C4)nn2)cc(N)ccc1Cl N1(C(c2ccc(C=C)cc2)=O)CC(NC(c2cc(Cl)ncc2Cl)=O)CC2(CC2)C1 Cn1cc(Br)cc(NC(=O)C(=O)NC2CCC(O)CC2)c1=O C1(C(N2C(C(=O)OCC)CC2)=O)CCN(C(=O)C(C(C)O)N(C)C)CC1O C1(NC(=O)CCCCBr)CCN(Cc2cc(Cl)cnc2F)CC1F c1(OC)ccc(C(=O)NCC2(C)CCC2)nn1.C1(=CC=O)CCN(C)C1 Cc1cc(C(N2CC(CO)(NC(=O)CCO)C2)=O)cc(C(F)F)c1.C(N)=O.N C1(O)(CNC(C(c2cccc(Cl)c2)CC)=O)CCN(C(=O)C#CC(=O)N(C)C)C1 N1(C(CNC(C2C(C)C2)=O)=O)CC(C(=O)N)C(F)C1.C1CCS(=O)(=O)C1 c1(C(=O)NC(C2CCCN2C(=O)CC2(C)CC2(Cl)Cl)C)ccn(C)c1 CCC(C)C(C(=O)NC1CC(F)(F)C1)N(C(=O)CC(C)(C)C)C.C(C)(=O)N c1(C(=O)NC2CN(Cc3cccc(C)c3F)CC2O)c(F)cc(Cl)cc1Cl c1(CC)cc(C(=O)NC(C)CCC(=O)NCCS(=O)(=O)NC)nn1C c1(C=O)c(C)cc(Cl)cc1C.C1(NC(CC2C(CC)C2)=O)CC2(C1)CCC2.N C1(NC(C2CCCN(C(=O)CCc3cnoc3)C2)=O)CCCOC12CCC2 N1(C(c2cnc(C)o2)=O)CC=C(CC)CC1.C1(C)(C=O)CC1C(F)(F)F.C C1(O)(CC)CCCN(C(C2(C(F)(F)F)CC2)=O)C1.[nH]1cc(C=O)c(C)n1.C c1(C(=O)NC2CCCN(C(C3(C(C)(F)F)CC3)=O)CC2)cccc2c1CCOC2 c1(CNC(C2C(C)C2)=O)nn(C)c2c1CN(C(C1CCCC(=O)O1)=O)CC2 N(C(=NCCCCl)N1CCC(CCOC)C1)Cc1c2ccc(OC)cc2[nH]c1 CCC(C)(C)C(=O)NCC(CC(C)C)NC(=O)Cn1cc(C(C)O)nn1 CC1(C)C(C(=O)NC(c2ccc(Br)cc2)CF)CC1(F)F c1(C(=O)NCC(CNC(CCC(C)O)=O)O)ccnc2[nH]cnc12 Cc1cc(C(=O)N(C2CCN(C(=O)Cc3cccs3)CC2C)C)ncc1C(N)=O C1(CC=O)CN2CCC1CC2.N1(C(C2CCC(CC)O2)=O)CCC(COC)C1.N C1CC2(C1)CC2.c1(C=O)csc(CC(F)(F)F)n1.C1(N(C)C)(C=O)CCC1.N C=CC1(CC(=O)NC2CCN(C(=O)CCc3cnc(C)o3)C23CC3)CCOCC1 C1(CC)CCN(Cc2nc(Br)sc2C)C(CN)C1 c1(C(NC(C=C)=O)=O)ccc([N+](=O)[O-])cc1-n1cnnn1.c1nc(C)c(C)s1.C C1(C(=O)NC2CN(CC)CC2C)CN(C(=O)C(C2CCCCC2)C)CC(C)(C)C1 c1(NC(=O)C2=COCC2)ccc2cc(O)ccc2c1 C1(NC(c2n(C(C)C)ccc2)=O)CCC(C)N(C(c2cnc(C(C)O)s2)=O)C1 C1(OC)CC(NC(C2OCCN(C)C2=O)=O)CN(C(c2cn(C)ccc2=O)=O)C1 Cc1cc(OCC(=O)NC(C)(C)CN(C)C(C23CC(O)C2C3)=O)ccc1F C1(C)(C=O)CCC(F)(F)C1.N1(CC)CCCC1C(=O)NCCC1CCCCC1 C1(C)(C(=O)NC(c2n[nH]c(=N)s2)C)CC2(C1)CC(F)(F)C2 O=C(CCC(F)(F)C(F)F)NCC1(O)CCN(C(C23COCC2C3)=O)C1 N1(C(CCCOC)=O)CCC(C2CCCN(C(=O)Cn3nnc(C)n3)C2)C1 c1(C2(C(N3CCCC3)=O)CCC2)ccnc(Cl)c1.c1(C(=O)N)cnn(C2CC2)c1 c1(C(N2CCC(CC=C)(NC(C3CCC(CC)O3)=O)C2)=O)ccc(OC)cc1C CCCC(C)(O)C(=O)N(CCCCNC(C1CCCOC1C)=O)C C1(NC(C(n2cc(CCN3CCOC3=O)nn2)C)=O)CCC(N2CCCC2)CC1 CC1SCCCC1NC(=O)N(C)CC1CCC(=O)NC1 c1(C(=O)NCCC2CCC(NC(c3c(C)noc3)=O)C2)cc(C(C)C)cnc1O N1(C(CN(CCC)C(c2cc[nH]n2)=O)=O)CCC(F)C1 c1(C(=O)NCCN(C)C(c2nnn(C)c2C(F)F)=O)ccc(N(C)C)cc1 CC1(C(N2CC(O)(CCNC(=O)CN3CC4CCC3C4)C2)=O)CC=CCC1 C1(CNC(c2c(CC)sc(=N)[nH]2)=O)CCCN(C(C2CC23CCCCC3)=O)CC1 c1(CC)ccc(C(=O)NCC2(C)CCN(C(=O)C=CC3CC3)C2)cc1.O c1(C(N2CCC(OCCC(N)=O)CC2)C(=O)NCC)cc2occc2s1 C(CN=c1cc[nH]c(=NCCC(O)C2CCC2)[nH]1)c1c(Br)ccc(C)c1 N1(C(C(C)(C)O)=O)CCCC(N(C(=O)C=CC=O)CC)C1.c1ccc(F)cc1 Cc1ccc(CCC(=O)NCC2(NC(c3csc(C(C)C)n3)=O)COC2)nc1 N1(C(c2ccc(=N)[nH]c2)=O)CCC2(CCCN(C(=O)CC3CCCO3)C2)C1 c1cc(Cl)c([N+](=O)[O-])cc1O.c1(NC(=O)NC2CC(C(=O)N)C2)ccccn1 c1(C(=O)NC2(CF)CCN(C(C3CC(CCC)C3)=O)C2)cc(O)nc(Cl)c1 N1(C(c2cc(OC)ns2)=O)CCN(C(c2cccc(CN=[N+]=[N-])c2)=O)CC(O)C1 C=C1CCC1(C(=O)NC1CC(NC(=O)C)C1)C=O.C1(C=O)CCCC1 CCC(CCCC(=O)NC1CCS(=O)CC1)NC(=O)CC(C)(C)CC CC1CC(NCCC(O)C(F)(F)F)c2ccsc2S1(=O)=O c1(C(N2CC(NC(C34CCC(F)(CC3)C4)=O)C2)=O)ncn2cc(Br)sc12 c1(OCCCCC)ccc(CN2CC(NC(C3(C)CCCCC3)=O)C(F)C2)cc1 CC(C)(C)C(C#N)C(=O)NCCCOCCC(=O)NCC(F)F n1(CC)ncc(C(=O)NC2CCCCC2)c1Cl.C(C(C)(C)C)N(CC=O)C.C c1(CC(N2CCCC2)=O)noc2cc(F)ccc12.C1(C(=O)O)(C=O)CC1.CC c1(C(=O)NCCN(C(=O)C(F)F)CCOCCCCCC)c(N)cccc1F CC1CN(C(=O)CCc2ccn(C)n2)CCN1C(=O)C=Cc1ccc(Cl)s1 N1(C(C(C)C(F)F)=O)CCC2CCC(NC(c3ccc(O)nn3)=O)C12 c1(COc2c(C(N=c3cc(OCC)o[nH]3)=O)nccc2)ccc2ccn(C)c2c1 C(=O)(CC(C)C(C)C)NCCC(C(=O)N1CC=CC1CF)OC C1(CNC(CC(CNC(C2C(C)CC2)=O)O)=O)CC12CCOCC2 c1(CC(=O)NCC(C)NC(C2(CC)CCCCCC2)=O)c(F)cccc1C#N N1(C(Cc2nc(C)sc2)=O)CCCC(CC(=O)NCC2CCN(C)C2)C1 c1(C(N2CCN(C(C(C)OCCCC)=O)CC2C2CC2)=O)cnn2c1CCCC2 N1(C(c2nc(CC)[nH]n2)=O)CCOC(CNC(=O)CCc2ccccc2)C1 CN1CCn2cc(C(N3CC4CCCCCCC4C3)=O)nc2C1=O Cc1sc(Cl)nc1C(=O)N(C)CCN1CCN(C(c2nnn(C)c2N)=O)CC1 c1(C(N(CC(C)NC(c2c(CC)n(C)nn2)=O)C)=O)c(C)cccc1N C(=O)(C1=NOCC1)N(C(CNC(c1cnc(C(N)=O)s1)=O)C1CC1)C N1(C(C(c2cnn(C)c2)C)=O)CC(CNC(=O)C=CI)OC(C)(C)C1 C(=O)(CCCCNC(=O)C1CC1)N(CC(C)N(C(C)=O)C)C c1(C(C)C)ccc(O)cc1C(=O)N(CCCNC(=O)C(C)(C)N(C)C)C c1(C(=O)NCCOC(CNC(C2CC(CC)C2)=O)(C)C)ccccn1.O C(c1ccccc1)=CC(=O)NC1CCCC1NC(=O)CC1CCCCO1 N1(C(CC2(C)N(C(C(COC)(C)OC)=O)CC2)=O)CCC2(C=CCO2)C1 C(=O)(C(C(C)C)NC(=O)CO)NC1C(NC(C)=O)CCC1.c1ccccc1 N1(c2nc(OCC)c(OC)cn2)CC(NC(=O)Cc2ccncc2)CC(F)(F)C1 c1(CCCC(N2CC3C(C3)C2)=O)ccc(C)c(C)c1.C(C(=O)N)(C(C)C)OC.C c1(N2CCC(OCCNC(c3nc(C)sc3)=O)C2)ccnc2ncnn12 CCCCC(O)CC(=O)NC12CC(NC(C3(C)CN(C(C)=O)C3)=O)(C1)C2 Nc1cccc(C(=O)CCC(=O)NCCNC(C23C=CC(CC2)C3)=O)c1 c1(C(N2CCC(C)(NC(=O)CN3CCCCS3(=O)=O)C2)=O)cc[nH]c2nccc1-2 c1(NCCOC)cc(=NCc2cnccc2SC)[nH]c(C(C)C)n1 c1(-c2cc(C(=O)NC(C(C)NC(c3cnc(C)[nH]3)=O)CO)on2)cccc(F)c1 Cc1cc(C=O)nc(C)n1.C1(C(C)C)CCN(C(=O)C(C2CC2)N(C)C)C1.N C1(N(C)C(c2ccc[nH]2)=O)CCCCC1NC(=O)CC(C1CCC1)C1CCC1 Cc1nccc(C(=O)NCC2CN(C(=O)Cn3ncc(Br)n3)CCO2)c1C c1(C(=O)NC2C(NC(C(C)Oc3cccnc3)=O)CCC2)ccc(C#N)[nH]1 C(CCCO)N(C(=O)C(C1CC1)NC(=O)C=CC(F)(F)F)CC c1(OC)cc(C(=O)NCC2CC2(F)F)nn1C.C1(C)CCCC1.C(=O)C.C C1(C(=O)NC2CC3(C(C(N(C4CSC4)C)=O)C3)C2)CC2CC(=O)C1C2 C(=O)(CC(F)(F)Cl)NCC1(OC)CN(C(=O)COc2ccsc2)C1 S(=O)(=O)(n1ccnc1)N(C(c1cccc(OC)c1)COC)C C=CC(C)(O)C(=O)N1CCCC(CC(=O)NCCN2CCCC(C)C2)C1 C1(C(N2CCCC(NC(=O)C(F)(F)CC3CC3)C2)=O)Cc2ccc(F)cc2O1 N1(C(c2c(CC)noc2C)=O)CC2OCCN(C(=O)CCc3nc(C)cs3)C2C1 c1(C(N2CCC3(CCC3)C2)=O)cccc([N+](=O)[O-])c1.C1(C=O)(C(F)F)CC1.C C1(C=O)(NC(Cc2c(CC)con2)=O)CCC(C)(C)C1.C1(C)CCN(C)C1.N [nH]1ccnc1C(=O)N(CCC)C(C)C.c1(C(C=O)N(C)C)cccnc1.CC Cn1nc(C(=O)NC(CNC(C2CC2c2ccccc2)=O)C2CC2)cc1F c1(C(N2C(C3CCN(C(CC(CC)O)=O)CC3)CCC2)=O)cn(C)c(=O)cn1 N1(C(CCCCOC)=O)CC(C2CC2C(N2CC=CC2(C)C)=O)C1 C1(NC(c2c(CCC)cccc2)=O)CN(C(=O)C(C2CC2)C2CC2)CCC1C C1(N(C(C(c2scc(C)n2)C)=O)C)CCCN(C(=O)C=Cc2nc(C)co2)C1 Nc1c(C(N2CC3CC2CCN3C(c2cn[nH]c2)=O)=O)cc(F)c(F)c1F C(CC(=O)Nc1cnn(C(C)C)c1C)(C(F)F)NC(C1(CC)CCNC1=O)=O c1(C(=O)NCC2CN(C(=O)COc3cccnc3)C2)cc(O)cc(Br)c1 Cc1ccc2c(C(N3CC4CC3CC4C(=O)O)=O)[nH]nc2n1 C1(CNC(c2occ(C)c2C)=O)CCN(C(=O)C(=O)C2CCCC2)C1(C)C c1(C(C=O)C)c(F)cccc1F.N1(C(C2(CC#C)CCC2)=O)CC(O)(CC)C1.N C1(COC(CCNC(=O)Nc2ccc(C)cc2C)=O)CCCC2(CCC2)C1 c1(N2CCN(C(c3cc(C(C)C)n(C(C)(C)C)n3)=O)CC2)ccc(C#N)cc1 C1(CNC(C2SCCS2)=O)CC2(CC2)CN1C(=O)CCOC1CCCOC1 CC1CCC(CC(N2CCCC(NC(c3n[nH]cc3Cl)=O)C2)=O)CC1 N1(C(C(C2CCCC2)NC(c2cnn3ccccc23)=O)=O)CCOCC2(CC2)C1 C(CC1CCCC1)(C(=O)N1CCCC1)OC.C1(C=O)CN(S(C)(=O)=O)C1.C CCN=c1cc(-c2nc(CC3CCC(C)C3)n(C3CCCC3)n2)cc[nH]1 c1(C(=O)NC(C)(C)CNC(c2ccc(F)s2)=O)ccc(C(F)F)nc1 C=CC1(C(N2CCC(CNC(C3CCC(=O)NC3)=O)C2)=O)CCOCC1 C1(C=O)CCN(C(=O)CC2CC2)C1.C1(CC=O)CCOCC1.C(C)(C)C.CO C=CCC(CC)C(=O)N1CCC(O)(CNC(=O)C(=Cc2ccncc2)C)C1 C1(C(=O)NCC(N(C(c2c(OC)c[nH]n2)=O)C)C2CC2)CCCN1C=O C1(c2nnnn2C2CCCC2)(NC(CCCC)(C)C)CCN2CCCC12 N1(C(C2CCCOC2)=O)CCC2CCN(C(c3cnc(O)s3)=O)C2C1 C1(C2CCCN(C(C3CC=CCC3)=O)C2)(NC(C(CC)=CC)=O)CC1 Cc1ccc(F)cc1C(N1CCC(CF)(NC(C2C(F)(F)C23CCC3)=O)C1)=O N1(C(c2c(C)cc(O)nc2)=O)CC2CC(C)N(C(=O)CCCc3nccs3)C2C1 C1CC2(CCOCC2)CN1C(=O)C(C)(C#N)CC.CCC(C(=O)N)NC(N)=O.C C1(NC(CNC=O)=O)CCCCC12CCN(C(c1ccc(O)c(Cl)c1)=O)C2 c1(N(C)Cc2cscn2)cc(Br)ccc1S(=O)(=O)NC1CCCC1C1CCCC1 CCCCC(CCCC)C(=O)N1CCC(NC(C2CN3CCCC3CO2)=O)C1 N1(C(C(c2ccn(C)n2)C)=O)CC(C)(C)CC1C(=O)NCc1cnnn1C N1(C(C2C(Cl)(C(=O)OC)C2)=O)CCC(NC(c2cncc(OC)c2)=O)CC1 C1(NC(C(CC=CC)C)=O)CCSC12CN(C(=O)Cc1ccc(F)cc1C)C2 C1(C(=O)NC(CC)C)CC(N=[N+]=[N-])CN1C(=O)C=Cc1cncn1C c1(C(=O)NC2CC3CC(NC(CN4CCC(C)C4)=O)C2C3)cscc1S(C)(=O)=O c1(C(=O)NC2CCC2NC(C2(Cl)CC2)=O)cc([N+](=O)[O-])c[nH]1 c1(CC(N2CC(CCC)C2)=O)ccn2cncc2c1.C(=O)(C)N.C(=O)C1CC1 C1(NC(C(c2ccn(C)n2)C)=O)CC2CCCC(C1)N2C(c1cscn1)=O CC1CC(C(=O)NC2CCCC2CNC(c2ccc(N(C)C)cc2F)=O)=NO1 Cc1cccc2[nH]c(C(=O)N(C3CCNCCC3C)Cc3cnccn3)cc12 N1(C(=O)OC)CCCN(C(C2CN(Cc3cnc(N(C)C)s3)CCC2O)=O)CC1 C12(CNC(C3=C(C)CCC3)=O)CC(CCO1)N(C(c1ncccc1F)=O)C2 c1(OC)ccc(F)c(CC(=O)NCC2CCCCN(C(=O)CC(C)OC)C2)c1 N1(C(C2(CC=C)COC2)=O)CCC2(CC1)CN(C(=O)CCc1cccc(C)c1)C2 Cc1ccc(=NC(=O)C=CC(=O)NCc2cc(Cl)cnc2Cl)[nH]c1Br C1(C(N2CCC(C=O)C2)=O)OCCCC1(C)C.c1(NCC)ccc([N+](=O)[O-])o1.N S(=O)(=O)(c1cnn2ccc(NCC)nc12)N1C(C)c2nncn2CC1.[SH](C)(=O)=O.N c1(CCC)nc(C)c(C(=O)NC(C)C(CO)NC(=O)CC2CN(C)C2)o1 C1(NC(C(C)N(CC)CC)=O)C=CCCC1C(=O)NC.C1CCC1(F)F C1(C(=O)NC(CC)CN(C)C(C2(C)COC2)=O)CCn2ccnc2C1 c1(C=O)cc(=O)c2ccccc2o1.C12(CNC(C(CC)C)=O)CC(C)(CO1)C2 N1(C(C=Cc2ccc(C(C)C)cc2)=O)CC2CCN(C(c3ncn(C)n3)=O)CC12 c1(OC)ccc(C(N2CCN(C(c3cn(C)c(C)n3)=O)C(CO)C2)=O)nc1OC c1(C=O)cc(F)cc2cnccc12.C1(COC)(C)CN(C(c2cc[nH]n2)=O)C1.N C1(C=O)CC(O)C1.c1(C=O)cn(C2CC2)nn1.C(C)(C)N(CC)CC.N Cc1cc(CC(=O)NC(C)CN(C)C(C2CC(C)CC(C)(C)C2)=O)cc(C)c1Br C1(NC(=O)C(F)=C(C)C)CCCN(C(=O)CC(C)Cc2ccc(Cl)cc2)C1.C C1(CNC(C23CC(C(=O)OC(C)(C)C)(C2)C3)=O)CCCC2(CCC2)C1O Cc1cccc(F)c1NC(C1C2CC3C(C2)C13)=O.C1(C=O)CCCC2(CC2)C1 n1(C(CC)C)nccc1C(=O)NC1CCN(C(c2ccccc2)=O)C1 N1(C(c2cc(SC)oc2)=O)CC(NC(C2CCC(=O)N2)=O)CC12CCC2 c1(CC(N2C(C(=O)Nc3cnn(CCO)c3)CC2)=O)ccc(Cl)s1 CC(C)(C)CCCC(=O)NCC12CCC(NC(c3ccc(CO)o3)=O)(CO1)C2 N1(C(C(CCC)OCC)=O)CCC2(C)CN(C(c3ccnc(O)c3)=O)CC12 c1(C(N2C3C(NC(=O)CCN4CCCC4)C(C3)C2)=O)nc2n(c1Br)CCC2 c1(C(N2CCCC(CN(C(=O)Cc3ccns3)C)C2)=O)cc(F)c2[nH]nnc2c1 C1(CCN(C(=O)CCCCC2CC2)C)CCCCN1C(=O)Cc1cnc[nH]1 c1(NCC2N(C(C(c3cccc(F)c3)C)=O)CCC2)ncnc2c1c(Br)nn2C N1(C(c2cc(C)cc(F)c2)=O)CCN(C(c2[nH]nc3ncccc23)=O)CC(O)C1 C1(C(C(=O)NCC(=C)C)F)CCN(C(=O)CC2(CSC)CC2)C1 N1(C(C2CCCN(CC)C2)=O)C2CCC1CC(CNC(=O)C)C2.c1cccs1.S N1(C(CC(CC)(F)F)=O)C2CCC1CN(c1nc(Cl)ncc1C(N)=O)CC2 c1(C(N2CC(F)(CNC(C(C)(C)N(C)C)=O)C2)=O)ccc2occc2n1 c1(N2CCCC(COCC)C2)[nH]c(=NC2CCCSCC2)nc2c1ncn2C c1(NC(=O)C(N2CCOCC2c2ccc(Br)cc2)=O)ccccc1-n1cncn1 C(=O)(CC(C)(C)C1CCCC1)NC(C1CCCN1C(=O)C(N1CCOCC1)C)C c1(C(=O)NCC2CCN(C(c3ccccc3)=O)CC2)ccc2c(c1)OCCNC2 Cc1cc(=NCC2CC(n3cccn3)C2)[nH]c(N2CCC3(CC2)CSC3)n1 n1(CCC=C)c(N2CC(C(=O)OC(C)(C)C)C(C)C2)nnc1-c1sccc1Cl N1(C(C2CC2(F)F)=O)CC2CCC(N=c3[nH]c4ccccc4o3)C2C1 c1(C(=O)NCCN(CCOc2cccc(Cl)c2)CC)ccnc(C2CC2)c1 Cc1ccoc1C(=O)NCC(C1CCOC1)NC(=O)Cn1ccnn1 C1(OC)(C)CCN(C(c2oc(C)nc2C)=O)C1.N1(CC=O)C(=O)CNC1=O.N C1(C(N2C(CNC(C3C(N(C)C)CCCC3)=O)CCC2)=O)Cc2ccccc2C1 c1(C=O)c[nH]nc1S(N)(=O)=O.N1(C(CC2(C)OCCO2)=O)CC(C)C2(CC2)C1.N N1(C(c2cccc(N)c2O)=O)CCC(C2CC2)(CNC(c2cccc[n+]2[O-])=O)C1 c1(C(=O)OCC)ccccc1N(C(=O)CCc1ccccc1Br)C c1(C(C(=O)NC2CCN(C(Cc3cc(C)sc3)=O)C2C)C)cccc([N+](=O)[O-])c1 CC1CC(NC(=O)CCC2CCC2)CCN1C(c1cc(OCC(F)F)ccn1)=O O=S(=O)(c1c[nH]ccc1=NCC1CCCN1CC1CC1)NC(C1CCCC1)CO N1(C(C(C)CF)=O)CC(NC(=O)CN(C)C(N)=O)C2(CC2)C1 c1(C(N2CCC(C)(NC(=O)CN3CSCC3=O)C2)=O)cc2ccccc2c(O)n1 N1(C(CC2(NC(CC(COC)C)=O)CC2)=O)CC2CCC2(C)C1 c1(CC)noc2ncc(C(=O)NCC3CCCC3)cc12.c1(CC=O)cnoc1.N C1(NC(CCc2nnc(C)o2)=O)CN(C(C23CC(F)(C2)C3)=O)C2CCCCC12 CCC(C(=O)N1CCCC(NC(c2cnc(N)c(N)c2)=O)C1)C(C)C C1(N(C)C(C2CCCS2)=O)CCCN(C(c2cccnc2)=O)CC1.S(C)(=O)(=O)N C1(NC(C=CCOC)=O)CN(C(=O)C(C)C(C)C)C2(CCCC2)C1 N1(C(Cc2cc(C)ns2)=O)CC(NC(C2(C)CCN(C)C2)=O)C(C)C1 C(C(C)(C)C)N(C(C1C(COC)CC1)=O)C.C(c1cnc[nH]1)=CC(=O)N Cc1cn2ccc(C(=O)NC3CCC34CCCC4)cc2n1 c1(C(=O)NCCCNC(c2cnc3scnc3c2)=O)c(F)ccc(Cl)c1F C1(NC(C(C2CCCC2)OC)=O)CN(C(=O)Cc2csc(Cl)c2)CCC1O c1(OC)ccc2[nH]nc(C(=O)NC3CCCN(C(=O)CC4CC5CC5C4)C3)c2c1 c1(C(=O)NC2CC(CNC(C3C(C)C3C)=O)C2)cc2c(Cl)ccnc2s1 Cc1cc(C(=O)NCC2(F)CCCN(Cc3cccnc3)C2)cnc1F N1(C(c2c(C)noc2)=O)CCc2ccccc2C1CNC(=O)CN1CCSCC1 c1(C(N2CC(NC(C(C(C)C)F)=O)C(C)C2)=O)cc(Br)cc2c1OCC2 Cc1ccc(C2CCN(C(=O)N(C3CCCCC3)CCc3ccccc3)C2)nc1 c1(CNC(CC2CC(CC)C2)=O)ccccc1.C1(C=O)CN(C2COC2)C1.C c1(NC)cnc(F)cc1C(N1CCN(C(=O)OC)CC1)=O.C1C(C)(C)C(=O)N1 c1(SC)cc(=NC(=O)CCCNC(C2CC3C(C2)C3(F)F)=O)[nH]n1C Cc1cc(CCN2C(=O)CCN(CC3COC(=O)O3)C2=O)ccc1[N+](=O)[O-] Cc1cc(NC(C2(C)CCN(C(c3cc(O)no3)=O)C2)=O)c([N+](=O)[O-])cc1Br c1(C(=O)NC2C(NC(C(COC)(F)F)=O)C2)ccc2c(c1)nc(CO)n2C C1(N(CC#C)C(c2ccc(C(C)C)s2)=O)CCN(C(C2CC3CCC23)=O)CC1 c1(C(=O)NCCN(C(C(c2ccccc2)OC(C)=O)=O)C)ccc(F)cc1.C C(=O)(C1=CCCC(C)(C)C1)N.C1(NC(c2c(C)nccn2)=O)CC(C)C12CCC2 c1(C(N2CCC(C3N(Cc4n(CC)ncc4)CCC3)CC2)=O)c([N+](=O)[O-])cnn1C C(=O)(C(C)CN(C)C(c1cscc1Cl)=O)N(CC(c1nn[nH]n1)C)C c1(C=O)cc2nc(Cl)ccc2o1.c1(OC)nn(C)cc1C(=O)NCC1CCC1 Cc1c(C(N2CCN(C(C3CC34CC4)=O)C(CCO)C2)=O)[nH]c2cc(Cl)ccc12 CC1CC(NC(C2C(C)C2C)=O)CN(C(=O)C(C)(C)CC2CC2)C1 C=Cc1cc(-c2nc(CO)nn2-c2ccnc(C(F)(F)F)c2)cc(F)c1 N1(C(c2nc(OC)c(C)s2)=O)CCC(CNC(=O)C(CSC)OC)C1(C)C C1(NC(c2c(C)noc2)=O)COC2(CCN(C(c3ccn4nccc4n3)=O)C2)C1 c1(C(N2CCC(C)C(NC(=O)Cc3c[nH]nc3O)C2)=O)ccc(N)c(F)c1F C=CCC(C(=O)NC1CCN(C(c2cccnc2N)=O)C(C)C1)C(C)C C=CC1(NC(C23CC(CN(C(=O)COC4CCOC4)C2)C3)=O)CCOCC1 C(=O)(N1CCCc2ccnn21)C1N(C(CC2CC(=O)C2)=O)CC2CC21 c1(C(N(CCC)CC)=O)cc2ccccc2nc1C.C1(P(C)(C)=O)(C=O)CC1.N C(=O)(C(CC(C)C)CC(C)C)N1C(C(CC)O)CCCC1 C(C1CN(C(c2cc3n(n2)CCCN3)=O)Cc2ccccc21)NC(C(C)SC)=O S(=O)(=O)(c1cnc(-c2ccccc2)nc1)NCC1NCCC(C)C1 CC(C)CC(F)C(=O)NCC1CCCC1NC(=O)CCCOc1ccccc1 c1(C(=O)NC(C)(C)CNC(C2CCC(CCO)CC2)=O)cc(N)c(F)cc1F C(=O)(C#CC1CCC1)N1C(CNC(C=C(CC)CC)=O)C(C)CC1 c1(C(=O)NC(CC)(C)CNC(=O)C(C)(CC)CO)cc2ncccn2n1 c1(C(=O)N)cc2cccc(C)c2o1.Cc1coc(C(C)C)c1C(=O)NC(C)CC c1(C(N2CCCN(C(C(C)NC(N)=O)=O)C(C)C2)=O)nc2cc(O)ccc2[nH]1 N1(C(CNC(=O)NC)=O)CCC2(NC(c3snnc3C)=O)CC2C1 c1(C(=O)NC(CC)CNC(c2cc(C(N)=O)co2)=O)[nH]c2cc(C)ccc2c1C C1(C(N2CC(C#N)(COC)C2)=O)CCCCCN1C(c1cccs1)=O CC1CN(C(c2ccc(-c3cccs3)s2)C(=O)NC2COC2)C(C)(C)CO1 N1(C(C(C)O)=O)CC2CCC2(CNC(=O)CCN(S(C)(=O)=O)C)C1 C1(C(=O)NC(C#C)C(C)OC)C2CCC(C2)N1C(=O)CN1C(=O)CNC1=O C1(OC)CC(CNC(C2CCN(C)C2=O)=O)N(C(c2ncc[nH]c2=O)=O)C1 C(=O)(CCC(=O)NN(C)C)N(CC(=O)NCC(C)C)CCC CCCCCCCCCC(=O)N1CC(CN(C(=O)C=CC2CCC2)C)C1 CC(C)CC(C(=O)NC(CN(C(=O)CSc1ccccn1)C)(CO)CO)C(C)C Cc1cc(C)c(NC(N2CC(=O)N(Cc3ccccc3)C2)=O)c(Cl)c1 C1(NC(CC(CCC)C)=O)CCCC2CN(C(=O)CN3CSCCSC3)CC12 C=CCC(F)(F)C(=O)N1C2CCC1C(C(=O)NC1CC3(CCC3)C1OC)C2 Cc1nc2cc(C(=O)NC(c3ncsc3C)C)ccc2s1 C1(CC(=O)NC(C)CC(C)NC(C2(CC(F)F)CCC2)=O)CCCC(C)(C)O1 N1(C(C(CC)(C)O)=O)CCOC2(C1)CN(Cc1cccs1)C2 Cc1ccc(CC(=O)NCC2(F)CN(C(=O)C3=CCCSC3)C2)c(F)c1 Cc1cc(Cl)nc(N)c1C(N1CCC2(CC1)CC2NC(=O)COCCF)=O c1(C(N2CCC(C3(C)CC3)C2)C(=O)NC)ccc(Cl)c(F)c1F c1(CC)ccc(OC)cc1CNC(c1ccc(OC(C)C)c(Br)c1)=O c1(SC)ccc(O)c(C(=O)NC2CC2NC(c2cccc(F)c2F)=O)c1 N1(C(c2ccc(CC)s2)=O)CCN(C)C(CNC(C2CCOCC2)=O)C1 CCC(CN(C)C)CC(=O)NCC(C1CCC1)NC(=O)CO.C1CC1.C N#CCCN=c1[nH]c(N2CCOC(c3cccs3)C2)nc(=N)[nH]1 N1(C(C2C3N(C(C=CC=CC)=O)C(CC3)C2)=O)CC2C3CCC(C3)C12 c1(CC(N2CC(NC(C3(C)CC4CC4C3)=O)C(O)CC2)=O)cc(F)c(F)cc1F N1(C(=O)CC2CN(C(=O)C(=O)NCC(F)F)CC23CC3)CC2CCC(O)CC2C1 c1(CC(=O)N(CCCN(C(c2c(C)nc(C3CC3)s2)=O)C)C)c[nH]c2ccccc12 C1(C(=O)NCC(=C)F)CC2(CC2)CN1C(=O)C=CC1CCCCC1 C1(C(N2CCCC(CCC(=O)OC)C2)=O)CN(CCN2CCCCC2)CCC1O CCCCCCC(C)C(=O)NC1CCCCC1NC(=O)CC1(C#N)CCCCC1 c1(CCC(=O)NCCC2CCN(C(C3(C)CC3Br)=O)CC2)ccc2c(c1)CCO2 c1(CNC(CSCC=C)=O)ccsc1C(=O)N.C1CCCC1C(C)(C)C c1(C(N(CCC)C(C)C)=O)cccc(Cn2cc(CCCCO)nn2)c1 C(CN=c1nc2c(ncn2C(C)C)c(NCC2(C)CC2(F)F)[nH]1)=CC C1(NC(C2CN(C(N)=O)C2)=O)CC2CN(C(=O)CC3CCC3)CCN2C1=O C(=O)(C(C)(C)CC(C)C)N(CC(C)NC(C(CC#C)O)=O)C C(CC(C)(c1nnnn1Cc1ccco1)NC1(CC)CC1)N(CC)CC C(CCCCC(=O)NC(C1CN(C(c2cncc(N)c2C)=O)CCO1)C)OC N1(C(CCCCCOC)=O)CC2(CC(NC(c3c(C)noc3C3CC3)=O)CO2)C1 Cc1cccnc1-n1cc(-c2nc(-c3ccco3)nn2-c2ccnc(Cl)c2)nn1 N1(C(c2ccc(Cn3ncc(C)c3)cc2)=O)C(C)C2CC1C2NC(=O)C(C)O C1(C(=O)NCCC2(COC)CC2)C=CCCN1C(=O)Cc1c[nH]nc1C c1(C(C)=O)c[nH]c(C(=O)NC(CC2CC2)C(=O)NCC(c2ccccc2)F)c1 c1(C(N2C(CCC)CNCC2)=O)ccc(Cc2ccc(C(F)(F)F)cn2)cc1F C(=O)(CS(=O)(=O)CCO)N(C)CC1CCCN(C(C2(COC)CCCO2)=O)C1 C(CCCC(=O)N1CCN(C(C2CCCN(CC(F)(F)F)C2)=O)CC1)N(C)C C1(NC(c2cnc(CC)[nH]2)=O)CCN(C(=O)C(C)CC(C)C)CCC1(F)F C1(CN(C(=O)CCCF)C)COCCN1C(c1ccnc(N(C)C)c1)=O c1(C(=O)N)cc2c(s1)C1(CCN(C(C(=O)O)C(F)(F)F)CC1)OCC2.NC(=O)C C1(C(=O)NC(c2ccc(C)s2)C)N(C(c2cccnc2C)=O)CCCC1(C)C c1(SCC(N2CCC(C(CNC(CCC#CC)=O)F)CC2)=O)ccsc1[N+](=O)[O-] C1(CCC(=O)N2CCCC2)(NC(C(N)=O)=O)CCCC1.C1(CC=O)CCC2CC12 CC1CCN(C(c2nnn(C3CC3)c2C(F)F)=O)C1.C1(C=O)CS(=O)(=O)C1 C1(NC(C(C=C)(F)F)=O)CN(C(=O)C=CC=CCC)C2(CCC2)C1 C1(CC#C)(NC(C2CC=CCN2C(=O)C(F)C2CCCC2)=O)CCOCC1 C(=O)(CCN(OC)C(=O)C(C(C)(C)C)OC)NC(CC)CC(=O)OC S(=O)(=O)(c1ccc(SC)cc1)Nc1ccc(C(C)OC)cc1.C(C)=O N1(C(c2[nH]c(=NC)sc2)=O)CCCN(C(=O)Cc2cc(Cl)cc(Cl)c2)CC1C C(CC(C)CCNC(C1CC(C)(C)O1)=O)NC(C=C(C)C)=O c12cc(nc(C)n1)NC(C)C1CN2C1.c1(C(C(=O)OC)C)ccnn1C c1(COC)ccc(C(=O)N(C(C)CNC(C2COCOC2)=O)C)s1 c1(OCC)cc(C(=O)NC)ccc1.C1CC1.C(=O)(C=C(C)Cl)NC c1(OC)cc(CN2CCCC2C(=O)NC(c2cncnc2)C)ccn1 N1(C(=O)OC(C)(C)C)CC2CCOC2(C(=O)NC2C3CCC2CC3)C1 C#CCC(N)CC(=O)N(C(c1ccccc1OC)C(=O)OC)C C1(O)(CNC(c2c(C(C)(C)C)[nH]cn2)=O)CCN(C(c2cc(Cl)c[nH]2)=O)C1 Cc1cc(C(F)(F)F)c(N)c(O)n1.c1ccccc1Cl.c12ccnn1CC(=O)N2.C CC(C)C(CO)CCNC(C1CCN(C(C2CC(N(C)C)C2)=O)CC1O)=O C1(NC(C2(O)CC2)=O)CN(C(=O)Nc2ccccc2)CC1.c1ccccc1C.C Cn1cncc(C(N2C3CCC(C3)C2C(=O)NCC2CC2(Cl)Cl)=O)c1=O c1(C(C(=O)NCC=C)N(c2csnc2C)C)cccc(-c2cccs2)n1 O=C(CC1C(=O)Nc2c(F)cccc21)NC.C(=O)(C(O)CN1CCCC1)N1CCC1 N1(C(C2(C)C(C)C2)=O)CCn2c(C(N3CCc4ccccc4C3)=O)cnc2C1 O=C(C1SCc2cccnc21)N1CC(OC2CC3CC(C2)CC(F)(F)C3)C1 C1(C(=O)NCC(CN(C(C(C(CC)C)OC)=O)C)(C)C)CCC2(CCC2)CC1 c1(NC2CCC(CCCC)CC2)ncc(S(=O)(=O)NCC(CO)OCC)cc1Cl C(C(C)(C)CC(=O)N1CCN(C(C2CC(=O)N(C)C2)=O)C(c2cn[nH]c2)C1)OC O=C1CCC(C(=O)N2CCC(NC(c3cncnc3)=O)CC2C2CC2)=NN1 C1(C(N(C)Cc2scc(C)c2)=O)CCOCCN1C(=O)CC1(N(C)C)CC1 C(=O)(C(C)(C)CC(C)(C)C)NCC1CCC(NC(C=C(C)Cl)=O)C1 C(CO)(C(C)NC(=O)NCC(c1ccccc1)CO)SC Cc1cc(C)n(C(C)C(=O)NCCO)n1.C1(C=O)CC2CC2C1.C(C)(C)C C1(C(=O)NC2CCC(N(C(c3nnc(C)s3)=O)C)C2)CCC(=C2CCC2)CC1 C=CCC(C)(C)C(=O)NC1CCN(CC2CCC2)CC1C C1(OC)CN(C(C)=O)CC1.c1(CC=O)csc(C2CCCC2)n1.C(=O)(CC)N c1(C(=O)NC2CCN(C(CCC(=O)OC)=O)CC2C)cnc2[nH]nc(O)c2c1 C(=O)(C(C)CCCC(C)C)N(C)CC1N(C(COCC(=O)NC)=O)CCC1 N1(C(COCC=C)=O)Cc2nccn2CC(NC(c2cc(OC)cnn2)=O)C1 N1(C(CCCC=C)=O)CCCC(C)C1CCNC(c1n[nH]c2c1COC2)=O C1(NC(c2cc(C3(C)CC3)on2)=O)CCCCN(C(c2c(Cl)nsc2Cl)=O)C1 C#Cc1cccc(NCC(=O)NC2CCN(C(=O)COC(F)F)C(C)C2)c1 C1(C(=O)NCC(CSC)(C)O)CC12CCN(C(=O)CCC(C)(C)N(C)C)CC2 N1(C(c2nccc(OC)c2O)=O)CCC2CN(C(=O)C3CC3)CC12 Cn1cc(C(=O)NCC2CC(NC(c3cccnc3N)=O)CC2O)c(C2CC2)n1 c1(C(=O)NCC2(NC(C(CO)OC)=O)CCCCC2)ccc2ncn(C)c2c1 C1(NC(CCC=C)=O)CN(C(C2(CCOC)CCCC2)=O)CC1C1CC1 Cc1cc(S(=O)(=O)O)ccc1C(=O)N(C1CC2CCC(C1)N2)C1CCOCC1 C(=O)(CC(C)CC(C)C)N1C(CNC(CN(CCC)C)=O)C(C)CCC1 c1(C(N2C(CC)CC2C)=O)cc(S(C)(=O)=O)ncc1Cl C1(CCNC(c2n(C)ncc2)=O)COCCN1C(=O)CCCCN1CCOCC1 c1(CCC(=O)NCCC(CNC(CC2CC(=C)C2)=O)O)ccc(Cl)c(C)c1 c1(CC)oc(C(=O)NCC(CNC(c2sc(=N)[nH]c2CC)=O)OC)cc1C c1(OC)cc(O)ccc1NC(=O)C(CNC(C1CC2CCCC2C1)=O)N(C)C c1(C(=O)NCC(CNC(C2CC(=O)NC2)=O)CO)ncccc1O Cc1ccccc1OCC(N1CC(O)(CN(C(=O)CC2CCCO2)C)C1)=O N1(C(C2C(NC(c3nc(C)oc3C)=O)CC2)=O)CCC2CC1C(=O)O2 c1(C(CC(=O)NC2CC(NC(C3CC4(C3)CC4F)=O)C2)O)cccc(F)c1 C1(NC(C2C(C=C)CC2)=O)(C)CC(C(F)(F)F)C1.c1(CC=O)cscn1 CCCC(CNC(=O)C=Cc1ccncc1)C(=O)NCc1ncc[nH]c1=O c1(C(N(CC(C)NC(C(C(C)(C)C)SC)=O)C)=O)c(C)ccc(Cl)c1O C1(C(=O)NCC(N(C(CCc2ccc(C)nc2)=O)C)C2CC2)CCCC(=O)N1C C12(CNC(C(C(C)C)C)=O)CC(CO1)N(C(=O)CC1C=CCC1)C2 c1(C(N(C(C)CCNC(c2ccn(C)c2C2CCC2)=O)C)=O)cccc(=O)n1C S(=O)(=O)(C=Cc1ccccc1)N1C(CC)CN(C(=O)Cn2cc(Br)cn2)CC1 C(=O)(C(F)(F)C(O)C1CC1)NC(CC)CNC(=O)CC1CC(OC)C1 N1(C(c2nc(C#C)sc2)=O)CCN(C(=O)CC(C2CC2)C2CC2)CC1C(C)C C1(C(=O)NCC#C)CN(C(C2(Cl)CCC2)=O)CCN1C N1(C(C2CN(C(C)=O)C2)=O)CC(CNC(c2nn(C)cc2Cl)=O)C2CCCCC12 C1(NC(C(C)Cc2ccccn2)=O)(CF)CCN(C(C2CC2)=O)C1.C(N)=O.N c1(CN2CCC(Nc3c(Cl)cccc3)CC2)ccc2c(c1)OCCO2 c1(C=O)ccc(C)c(F)c1.C1(C(=O)NC2(CC#C)CCC2)CC2(CC2)C1.C N(C(=NCCC(=O)N(C)C)N1CCC2(CCC2)CC1)CC1COCC(C)O1 C(=O)(C1=CCC(C)CC1)N1CCC(CC)CC1C(N1CC2(CC2C=O)C1)=O.O C(C(C)(C)CNC(C1(C)CC1(F)F)=O)N(C(C1CC=CCC1)=O)CC c1(NC)ccccc1C(N1CC2CC2(NC(=O)Cc2ccnc(Br)c2)C1)=O N1(C(COCC=C)=O)CCC(NC(c2nc3ncccn3n2)=O)C(CO)CC1 c1(C(c2nnnn2C(C)C)NCCNC(C)=O)cnc(C2CC2)nc1 N1(C(c2ccc(N(C)C)cc2)C(=O)Nc2ccccc2)CC(O)CC(C)(C)C1 CC(C)C(C)CC(=O)N1CC(NC(c2cc(C(F)(F)F)on2)=O)C(C)C1 N1(Cc2nc(COC)sc2)CCN(C(c2ccc(OC(C)C)cn2)=O)CC1 C(C)(CC(F)(F)F)NC(C1(COC)CC1)=O.c1(C=O)cc(C)cc(F)c1 N1(C(C2N(C(C(C(C)C)C#N)=O)C3(CC2)CC3)=O)CC(CO)CC12CCC2 N1(C(C(OC)OC)=O)CCN(C(c2cc(O)ccc2O)=O)CC1C(F)(F)F N1(C(C(CC=C)CC)=O)CC2CN(C(c3csc4c3CCCC4)=O)CC2C1 c1(-c2nnc(NC(CNC(CNC(C(CC)C)=O)=O)=O)s2)cccc(F)c1 C=CCCCC(C(=O)NCCOC1CCC1)NC(C1CC(N=[N+]=[N-])C1)=O S(=O)(=O)(c1cccc(=NCCc2sc(=N)[nH]c2C)[nH]1)NCCCCSC C1(C(N2C(CNC(C(CC)(C)C)=O)C3CCC2C3)=O)CCn2cnnc2C1 C1(C(=O)NCC(CC)N(C(=O)CCC(C)C)C)CCCC(F)C1 c1(C=O)cc2c(ccn2C)[nH]1.N1(CC)CCOC(C(=O)NC23CC(C2)C3)C1.C Cc1cc(C(=O)NC2(CCC(N3CC(F)CC3C)=O)CCC2)c(C)[nH]1 C12(C(=O)NC(C)OC)CCC(C(=O)NCCCCc3ccccc3)(CC1)C2 c1(CN(C)C(C2C(C(=O)O)C2(F)F)=O)ccc(Cl)s1 N1(C2CCN(S(=O)(=O)C3CC3)CC2)CCN(N2CCCN3CCCC3C2)CC1 Cc1cccc(Br)c1C(=O)NCC1CC2(C1)OCCO2 C1(NC(C2CCCCO2)C)CCCC(C(C)(C)C)CC1 Cc1cccc(C(=O)NC2CC(CNC(c3cccc(O)c3)=O)C2)c1F N1(C(c2c(OC)cc(C)cc2)=O)CC2(CCCC2NC(c2ccn(C)c2C)=O)C1 C1(C(=O)NCCC2CN(C(c3cc[nH]n3)=O)C2)CC2CCC1O2 N1(C(COC2CN(C(CCCCCOC)=O)C2)=O)C2C=CCC1CCC2 c1(NCC)ncc(C(=O)NC)cc1Cl.C12CC1CN(C(=O)CC1CCC1)C2 C1(C(=O)NC(CNC(C2(CSC)CC2)=O)CO)OCCN(C)C1=O C(CCCCC(=O)N1CCC(CNC(c2nonc2N)=O)C1(C)C)SC C(=O)(C(CC)CC(F)(F)F)NC1C(CCC)CN(C(c2ccn(CC)c2C)=O)C1 c1(-c2cncc(C(=O)O)n2)cnn2c1CN(Cc1cccc(O)n1)CC2 C(C(=O)NCC1C=CC(NC(c2ccncc2)=O)C1)(C(C)C)NC(C)=O C(C)(C(C(=O)NCc1cnns1)C(C)C)NC(CCC)=O Cn1cc(C(N2CC(CC(C)(C)C)C(N)C2)=O)c(O)nc1=O c1(OC(C)C)ccccc1C(=O)NC(C)Cc1ccccc1.C(=O)(C(F)F)N c1(C(N(CC(=O)NC(C)Cc2ncn(C)n2)C2CC2)=O)cncn(C)c1=O c1(CC(N2C3CC(NC(c4cc(CO)on4)=O)C3CC2)=O)ccc2nonc2c1 C1(CC(=O)NCCCC2(NC(CC3CN(C)C3)=O)CC2)CCCOC1 c1ccccc1.N1(CC(C)C)CC(C(=O)NC)C1.C(=O)(C(C)N1CCC1)NC C(=O)(C(F)C(F)(F)F)NC1CC(N(C(CCCn2c(C)cc(C)n2)=O)C)C1 C1(N(C(=O)C(n2cc(C)cn2)C)CC)CCCN(C(=O)CCCC2CC2)CC1 N1(C(CN(C(=O)CN2CC3CC3C2)CC)=O)CCC(C)(CO)C1 Cc1ccc(C)c(C(=O)CCC(=O)N(C2CCC(C)CC2)CCO)c1 N1(CCN(C)C(C2(C3CC3)CCC2)=O)CCN(C(c2cc(F)n[nH]2)=O)CC1 c1(CC(=O)N(C)CCOCCN(C)C(C2CC23CC3)=O)cccc(Cl)c1F O=S(=O)(CC1CCCCCC1)CCc1cccc(Cl)c1 c1(C(=O)NC2C3CC2N(C(c2ccncc2)=O)C3)ccc2c(c1)CCC=C2 C1(CC)(C)CCCO1.C1(O)(C(C(=O)N)F)CN(C(=O)C(C)N2CC(C)C2)C1 CC(C#N)CN(C(C(=O)NC1COC1)C1CC(CC(N)=O)C1)C N1(C(CCOC)=O)CCC(CC(=O)NC(CO)CC(C)C)C1(C)C N1(C(c2cncc(NCC)c2)=O)CCN(C(C2CC2F)=O)C(CC2CC2)C1 C1(CNC(c2c(CCC)cccc2)=O)CCN(C(=O)C(C)=CCO)CC1C c1(C(N2CC(C)(CCC(=O)NC(C(CO)SC)C)C2)=O)ccn2ccnc2c1 C(CCCCCNC(=O)C(C)OCC(C)C)NC(C1CCC(CC)O1)=O c1(CCC(=O)NCC(C)N(C(=O)C(O)CC(F)F)C)nc2ccccc2s1 CC1CCC1C(=O)NCCN(C(=O)CCSC1CCCC1)C1CC1 CC1(C)OCC2CC12C(=O)NC1(C)CCCCC1.c1(C(=O)N)cc2occc2s1 N1(C(=O)CCc2nccs2)CCC2CC2(C(=O)NOCC2CCCC2)CC1 C(C(C(=O)Nc1cnc(F)nc1)C(C)C)NC(CCc1ccc(C)o1)=O C1(NC(CCc2ccc(C)nc2)=O)CCCCN(Cc2ccc(O)cn2)C1 C1(C(N2CCCC2)=O)CCCC2(C1)CC2(F)F.C1(C(=O)N)(COC)CC=CC1 CC(C)CCC(CO)N=c1cccc(S(=O)(=O)N(CC(=O)NC2CCCC2)C)[nH]1 Cc1cccc(CN2CCC(OC(C3COCCN3C(=O)C3CC3)=O)C2)c1 c1(NC(c2nc(C(=O)NCc3ccc(Br)nc3)sc2)=O)ccc(Cl)c(F)c1 n1(CC)cnc2c(NCC3(F)CC(NC(C4CCNC4=O)=O)C3)nc(Cl)nc12 C(=O)(C(C)(CC)C(=O)NC1CCN(C(c2cocn2)=O)CC1CO)OCC C(=O)(C(CCCOC)NC(C1CCC(C)(C)C1)=O)N(CCCC=C)CC C1(=CC=O)CCOCC1.C(C(=O)NCCO)(C1CCOC1)OCC.CCC c1(OC)cc[nH]c(=NCCCCC(C)NC(=O)C=C2CCCCC2)n1 CC(C)CC(C)(CNC(C1(C#N)CCC1)=O)NC(=O)CCC(=O)N(C)C c1(C(=O)NC2C(CNC(c3scc(C)c3)=O)C2)ccn2ncc(Br)c2n1 c1(CC)cc(F)ccc1C(=O)NC1(C)CC(NC(c2cc(Cl)ncc2)=O)C1 C1(NC(c2c(C)c(N)cc(O)c2)=O)CCN(C(=O)C=CC(F)(F)F)CCC1(F)F CC(C)C(C(=O)N(C)CCNC(=O)CC1CSCCS1)NS(C)(=O)=O c1(C(N2C(CC(=O)N(C)Cc3cccc(C)c3)CCC2)=O)ccc(F)c(C#N)c1 c1(CC=O)ccc2nsnc2c1.Cc1ccc(CCC(=O)NCC2CC2C)o1.N c1(OC)cc(C(N2CCC3CCC23CNC(c2cnn[nH]2)=O)=O)c(N)c(C)c1 N1(C(C(CC=CC)C)=O)CCOCCC1C(=O)NC1CCC(C)(C)CC1 c1(C(C)(C)C)ccc(C(N2CCC2C)=O)[nH]1.c1(C=O)cc(C2CCCC2)[nH]n1.N c1(C(N(CP(C)(C)=O)CC(=O)OC)C(=O)N)cc(OC(F)(F)F)ccc1F.C Cc1c(C(=O)OCC2C=CCOC2)ccc(Br)c1F C1(NC2CC(CCC)C2)CCN(C2CNC2)CC1 CCCCCCC(C)C(=O)N1CCN(C(c2cc(CCC)on2)=O)CC1CC C(=O)(CN1C(=O)COc2ccc([N+](=O)[O-])cc21)NC1CCC(C(C)C)CC1 c1(C(=O)NC(C2CC2C)C)cn(C2COC2)nn1.c1(CC=O)cscn1 N1(C(C=CC=CC)=O)CCCCC2(C1)CN(C(c1nccn3cc(C)nc13)=O)C2 C1(NC(CC(COC)C)=O)CN(C(c2ccnnc2)=O)C2(CCCCCC2)C1 Cn1cnc2cnc(N3CCN(CCNC(C4CC5CCCC45)=O)CC3)nc12 N1(S(CCCOC)(=O)=O)CC2CN(Cc3ccccn3)CC2C1 C#CCC(C)(C(=O)N1CCC1(C)C(C)C)NC(=O)CCN1CCCCC1 N1(C(CC2CCC(C)CO2)=O)CC2(CCC2NC(=O)C(=O)N)C1.CCN(C)C Cc1n[nH]c(=NC2(CNC(c3cnc(C4CC4)nc3C)=O)CC2)o1 C1(C(N(C(CC)C2CC2)C)=O)CCCN(C(c2cc(C)nc(O)c2)=O)CC1 n1(CC(=O)NCC(C)C)ccc(C2CC2)n1.c1(C=O)scnc1C1CCCC1 c1(OC)cc(F)ccc1C(=O)NC(Cc1cccs1)CC(=O)NC(C)(C)C c1cnc(O)c(C(N2CC(O)C2)=O)c1.c1(C(NC)=O)cn(C)[nH]c1=N.CCS c1(C(=O)OC)cc2cccc(NC(=O)C(=O)NC3(CCCO)CC3)c2s1 c1(C(=O)NCCCN(C)C2CC2)ccnc(CNC(=O)CC2CSC2)c1 C(=O)(CC(C)CCCCC)NC(CC=C)C(=O)N(CC(N)=O)CC(N)=O N1(C(CC(COC)C)=O)CCC2(CC(NC(c3sccc3C(C)C)=O)CO2)C1 Cc1cc(C(C)N(C(=O)CCC2CC2)C)no1.C1(C=O)COCC1C(N)=O.N N1(C(C2(C=C)CCC2)=O)CCC(NC(c2cnoc2CC(C)C)=O)CC1 c1(C(=O)NCC2(CNC(C(CO)OC)=O)CC2(F)F)cncn(C)c1=O C(=O)(CCC(C)S(C)(=O)=O)NC1C(NC(CCS(=O)(=O)NC)=O)CC1 c1(C(=O)NC2(CNC(CC(C)C3CCCO3)=O)CCC2)nccc(Cl)c1F CP(C)(=O)C1CCCC=C1C(=O)N1CC(C2CN(C(C3(CO)CC3)=O)C2)C1 C(CN=c1nc2c(ncn2C)c(NCc2nc(C)cs2)[nH]1)(C1CCCCC1)OC N1(C(c2ccc(Cl)nc2)C)Cc2ccc(O)cc2C1 C=CC1(C(=O)NCC(O)C2CCC2)CCN(C(c2ncccc2O)=O)C1 O=C1CCCN1CC.C1(C2(C(=O)N)CC2)CCCN1C(=O)C=Cc1cn[nH]c1 c1(CC(=O)N(CC(=O)NC(COC)C(C)C)CCOC)cccc(C)c1 n1(C(C)C(=O)NCCC2CCC3(CC3)CO2)cnc2c(N)ncnc12 N1(C(CN(C(=O)CCC2CCCCO2)CC(C)C)=O)CCNC(=O)C1CCO CC(C(=O)NCCC(C)N(C(=O)CCc1cocn1)C)n1ccnc1 CC1(C)C(C(N2CC(NC(C3CCCOC3c3cn[nH]c3)=O)C2)=O)C1(C)C c1(C(=O)NCc2cc3[nH][nH]c(=N)c3cc2)cccc2c1OCCCO2 CC(C(F)(F)C(F)(F)F)=CC(N1CC(C)N(C(=O)CCCC(C)(C)C)CC1C)=O Cc1ccc2nc(C(N3CCN(C(=O)C(C)C)CC(CO)C3)=O)c(N)n2c1 c1(N(C(=O)CC2(CN)CCOC2)C)ccc(Cl)cc1Cl.c12cnccc1CN2 c1(CC(N2CCC(NC(CCC=C)=O)C(C)C2)=O)cn2c(C)csc2n1 c1(C(N2C(COC)CN(C(=O)C(O)CC3CC3)CC2)=O)cccc2ncnn12 C=CCC(CC)C(=O)NC(c1cccc(C(F)(F)F)c1)C(=O)N1CC(F)C1 N1(C(CN2CCCC(CC)C2)=O)CCC2(CC(NC(=O)C(C)C(C)O)C2)C1 C1CC2(CCCOC2)C1.CS(=O)(=O)SCC=O.C1(C(F)(F)F)(C=O)CC1.N C1(NC(C2CN(C)C(=O)C2)=O)(C)CC2CCC1CC2.C(=O)C(C)(O)C1CCC1.N C1(C)(c2cccc(NC(c3ccc(COCC)cc3)=O)c2)NC(=O)NC1=O C(=O)(C(F)C(C)(F)F)NC1CC(CCC(=O)N(CCC)C)C1 c1(CC)nc(Cl)c(C)c(=NC2CC(C)N(C(=O)CC(C)n3cccn3)C2)[nH]1 c1(NC(C2C(NC(c3ccc(OC)c(Br)c3)=O)C2)=O)cc(Cl)c(C)cc1Br c1(OC)cncc(C=CC(=O)NCCC)c1.c1(C=O)sccc1-n1cccc1.N C1(C)(CC)CC(NC(c2cc(C)cs2)=O)CN1C(=O)CC(F)(F)Cl N1(C(c2c(C(C)C)ocn2)=O)CCN(C(C2CC(C)(O)C2)=O)C(C)C1 C(CCN(C(=O)C(C)C)C)C(C)(C)C.c1(NC(CC)=O)cccc(C(=O)N)c1 n1(CC(C)C)ccc(=NC(=O)C2CCCCN2C(C2CCCCC(=O)N2)=O)[nH]1 N1(c2ccc(C)cc2)CCCC(NC(=O)Nc2ccsc2C)C1=O.C(C)(C)C.O Nc1cc(Cl)cc(F)c1C(N1CCC(NC(C2CC2F)=O)C1)=O N1(C(c2scc(OC)c2)=O)CCN(C(C2CC(C)(C)CCO2)=O)CC1C1CC1 N1(C(c2nc(OC)cc(OC)n2)=O)CC(C)N(C(c2ccc(C)cc2)=O)CC1C CCC(CNC(C1(OC)CCC1)=O)(CC)NC(c1oc(CO)nc1C)=O N1(C(C(=O)NC(C)C)=O)CC(C(N2CCc3nocc3C2)=O)C2(CCC2)C1 O=C(CC(F)(F)C(F)F)NCC1CN(C(c2ccc3c(c2)COC3)=O)CC12CC2 C12(NC(C3C(C)(CC)C3)=O)CCCN(C(C3COC(C)(C)C3)=O)CC1C2 C(=O)(C1CCCn2cnnc21)NC1C(NC(c2c(SC)nn(C)c2)=O)CCC1 c1(CC)cc[nH]c1C(N1CCCC1CNC(=O)CN(C)C)=O c1(C(c2n(CCCCCC)nnn2)NC2COC2)cc(F)c(F)c(F)c1 c1(C=O)ccc(CCC)c(S(N)(=O)=O)c1.N1(C(CNC(CC)=O)=O)CCC1.C c1(C(N2CCC(NC(COCCC)=O)C(C)C2)=O)csc2cccc(OC)c12 Cc1noc(C)c1C(=O)NCC1(C)CCCN1C(=O)C=CCN(C)C c1(CCC)ncoc1C=O.C12CC(C1)C2.C(=O)CCN(S(C)(=O)=O)C.N C(CCN=c1ccc(Br)c(S(=O)(=O)NC(C)(CC(C)C)C(N)=O)[nH]1)OC=C c1(NC(=O)NCCc2cnn[nH]2)ccc(S(F)(F)(F)(F)F)cc1 c1(CC(C)C(=O)N2CC(C(N)=O)C2)ccc(Cl)cc1.C1(C)(CC=O)CCC1.C N1(C(CCn2c(C)ncc2)=O)CCC2CCN(C(=O)COC3CCCCC3)CC12 c1(C(C)C(=O)NCC2CCCC2)cccc([N+](=O)[O-])c1.C(=O)CC.C(N)=O.N C1(CC(=O)NC(c2ccccc2)CO)CCN(C(=O)CCCF)CC1 N1(C(c2ccc(C)[nH]2)=O)CC=C(C(C)(C)C(=O)NC2(C)CCCC2C)C1 CN1CCCC1CC(N1CC(CCc2cn(Cc3ccoc3)nn2)C1)=O C1(CC(N2CC(C(C(=O)N(CCn3c(C)ncc3)C)O)C2)=O)CCCN(C)C1 CCC(CC(=O)NCC1(F)CCN(C(c2ccncc2O)=O)CC1)CC(F)(F)F c1(C(=O)NC(C(=O)NC2(CO)CC(C)C2)c2cccs2)ccc(Cl)cc1 c1(CC)cc(N)c(C(N2CCN(C(=O)CC(C)CF)CC2)=O)c(F)c1 c1(C(=O)NC(C)CCNC(C2CC23CC3)=O)cnc(C2CCOCC2)nc1 c1(CC)cccc2[nH]c(C=O)cc12.C(=O)(CS(=O)(=O)C1CC1)N(CC(C)C)C.N Cc1c(C(=O)N)ccn1CCO.C12(CC)CCC(CC1)C2.C1(O)(C=O)CCSC1 Cc1nc(Cl)ccc1C(N1CCOCC1CC(N1CC(C)C1)=O)=O c1(C(=O)NCCOCC(C2CCCCC2)F)ccc(CS(=O)(=O)C(F)F)cc1 N1(C(COCC)=O)CCC(C2OCCC2NC(c2csc(C3CC3)n2)=O)CC1 C1(C(=O)Nc2c(CC)nsc2)CCC(C2CC2)N1C(=O)C(C#N)CC N1(C(C(CNC(C2(C)CC(=O)C2)=O)OC)=O)CC(CO)C(O)C1 C(=O)(C1CCCc2ncccc21)NCC1CCN(C(C2(N(C)C)CCCC2)=O)C1 c1(CCOC)n[nH]c(=NCCC2CCN(C(=O)C(C)NC(C)=O)C2)s1 C(CCc1ccccc1)(CC(F)(F)F)NCc1n(CCC2(C)CC2)nnn1 c1(NC(C2N(Cc3c(SC)cccc3)CCC2O)=O)ccc([N+](=O)[O-])c(Cl)c1 C(=O)(CCC1=CCCCC1)N1CC(CCNC(C2C(C(=C)C)OCC2)=O)OCC1 c1(SCCC)ccc(C(N2CC(OCCNC(=O)C(O)CC)C2)=O)cc1.S CS(=O)(=O)c1cnc(N2CCC(OCCNC(C3CCOCC3)=O)C2)c(Cl)c1 c1cc2nc(SCC3CC3)nc(NC3CCNC4(CCC4)C3)c2s1 C1(NC(CSC(C)C)=O)CCC(NC(=O)CCc2cnn(C)n2)CC1 CN1CCN(C(C2CCN(C(=O)CO)C2)C(=O)NCCCC2CC2)C(C#N)C1 C1(C(N2CCN(C(CCC(=O)N(C)C)=O)CC2CCO)=O)CN2CCC1(C)CC2 O(NC(=O)C(C)CNC(=O)CC1OCCC1(C)C)CC=C C1(NC(c2cc(CC)nc(O)c2)=O)CCSC12CN(c1cc(C)nc(SC)n1)C2 C(C(CNC(=O)C(c1ccc(F)cc1)F)C(F)(F)F)NC(c1cc(C)ns1)=O Cc1ccc(C)c(C(=O)NCCCCNC(=O)CC(C)F)c1C N1(C(Cn2c(C)csc2=O)=O)CC2CCC2(C)C1.c1(C=O)coc(C(C)C)n1.N C1(C(=O)NCCCN(C(c2c(SC)snn2)=O)C(C)C)CC(=O)N(C)C1 c1(N(C(c2cn(C(C)C)nn2)C(=O)NC2CCOC2)C)ccc(I)cc1.C1CC1 CC(C)(CCCF)C(=O)N1CCN(C(c2ns[nH]c2=O)=O)CC(O)C1 Cc1cc(C)c(CNC2(c3nnnn3C3CC3)CSC3CCCC23)c(C)c1 N1(C(C2CC(C)(F)C2)=O)CC=CC(NC(=O)CN2CCC(C(F)(F)F)CC2)C1 NS(=O)(=O)c1ccc(Cc2nnc(N3CCC34CCCC4)n2CCC#N)o1 C1(C)(C(=O)NCCCCCN(C(C(CC)C(C)C)=O)C)CCC(=O)N(C)C1 O=C1CCC(C(=O)NC2CC2CNC(c2ccnn2C2CC2(F)F)=O)O1 C1(O)(CNC(C(C)CSC(F)(F)F)=O)CCN(C(C23CC4CC2C3C4)=O)C1 C1(NC(C(=C(C)C2CC2)F)=O)CCN(C(c2cc(C(F)F)ccn2)=O)C1C c1(CC(=O)NC2CC(NC(C3CCC(C)S3)=O)C2)ccccc1[N+](=O)[O-] c1(C(N2CCN(C(C(CC3CC3)OC)=O)CC(O)C2)=O)ccc2c(n1)CCC2=O Cc1nc(NC(c2cc(Cl)c(Cl)s2)=O)sc1C(N1CCCC(C)C1)=O C1(C(=O)NC)CCCC1(C)NC1CCCN(CC(F)(F)F)C1 C1(C)(C=O)CC1C(=O)N.C1(C=O)CC1.CCC.CCC.C(C)C.CC Cc1c(C=O)noc1C1CC1.C1CN(C(C2(C=O)CC2C)=O)C1.C(C)(C)C C(CC(O)C(=O)NC1CCC1NC(c1cc(Br)cs1)=O)N(C)C N1(C(C2CCC(C(=O)OC)O2)=O)CC2(CCN(C(=O)C(C)C3CCCC3)CC2)C1 C(=O)(C1=C(C)OCCS1)N1C(C(N2C(CC)CCOCC2)=O)CC=CC1 C1(C=C)(C(N2C(C(=O)NCC#C)CC(O)C2)=O)CCOCC1 c1(C(=O)NCC(CC)NC(C2CC(SC)C2)=O)cc(C)ncc1C CC1OC2(C)CC1(C(=O)NC1CCC(C)N(C(=O)CCn3cccn3)C1)C2 Cc1noc(C)c1C(N1CCC(C(C)NC(c2cncn2C)=O)C1)=O C(=O)(C1=NOC(CNC(C2C3CCC(C3)C2C)=O)C1)NCC(C)CCCO Cc1ccc(C(=O)NC2CCCCN(C(=O)C(C)O)C2)nc1C Cc1cnccc1C(=O)NCC1CCCN1C(C1CCCOCC1)=O N1(C(C(C)CC(F)F)=O)CCCC2C(O)CC12 C(C(C(=O)NCCC1CCC(C)(C)C1)C(C)(C)C)NC(CCCC#CC)=O C(=O)CC(C)CC(C)C.C(C)(CCC)NC(CCNC(COC)=O)=O.C(C)=O C1(C(C)(C)NC(CC=C)=O)CCCN1C(=O)CN(C)C(N)=O c1(OCC2CCN(C(=O)NCCSCC(C)C)C2)ccc(Br)cn1 c1(C(=O)NC2CCC2NC(C2CC(N3CCOCC3)C2)=O)cnc2n1CCOC2 N1(C(C(C)(C2CC2)OC)=O)CC2(C1)CN(C(=O)CCC(C)N(C)C)CCO2 c1(CC(N2CCC(CCNC(c3nocc3Cl)=O)C2)=O)ccc(F)c(F)c1 Cc1cc(C(=O)NCC(C2(O)CCN(C(c3c(C)csc3C)=O)C2)C)cnc1O CCC(C)(C)C(O)C(=O)NC(C)CCN(C(=O)C(C)(C)n1cnnn1)C C=CCCCCCC(=O)NC1CCCC(N(C)C(c2cncc(C(C)C)c2)=O)C1 N1(CC(CC)O)CCN(C(=O)C(N2CCCC(OC)C2)=O)CC1 c1(CNC(c2nnn(C)n2)c2nnnn2CSc2ccccc2)ccccc1F C12(NC(c3c(CC)cno3)=O)CC(C1)OC21CCC1.C(=O)CC(C)(C)CC.C C=C(C)CC(C)C(=O)OCCC1CC(C(=O)OCC)C1 N1(C(c2cn(CCC)nn2)=O)CC(C)OC2(CCN(C(=O)CS)C2)C1.CC(C)=O c1(C(=O)NC2CC(N(C(c3cc(OC)nn3C)=O)C)C2)ccc2cncn2c1 N(C)(S(=O)(=O)N(C)C)CC(=O)N(CCC)C.C1(C=O)CC1.CCO C1(C=O)CC2CCC(C1)O2.c1(C(CNC(c2csc(C)n2)=O)F)ccccc1.N C1(C(C(=O)NCSc2ccc(F)cc2)NCc2cc(C)sc2C)CC12CCOCC2 C1(O)(C(=O)NCC(CNC(C(C)C(C)(C)C)=O)F)CCC(C)(C)CC1 c1(N2CC(C)C(NC(=O)C(C(C)(C)C)NC(N)=O)CC2)ncnc2c1COC2 N#Cc1cccc(C(=O)NC)c1.C12CC(CO1)C2.C1(CC=O)CCC(=O)NC1 C=C(Cl)CCC(=O)NCCC1CCCN1C(=O)CCOC1CCCC1 N1(S(CCC)(=O)=O)CCCC12CCCN(C(c1cccnc1)=O)C2 c1(C(=O)N)ccc2c(c1)nnn2C.C1(NC(c2c(C)occ2)=O)CCC(C)(C)C1 N1(C(=O)CC2CC3CC3C2)CC2=C(C1)CN(C(c1cn(C3CCC3O)nn1)=O)C2 c1(OC)cccc(C(=O)NC(C2CCCN2C(=O)C=Cc2ccco2)C)c1.O c1(OC)ccc(I)c(NC(=O)NCc2cn(CCCN(C)C)nn2)c1 c1(N2C(CCNC(=O)Cc3ccc(Cl)c(F)c3)CCCC2)ncnc2[nH]cnc12 N1(C(C(c2ccccc2)SC)=O)CCC(C)C(NC(=O)COC(C)=O)C1C CC(C)(C)C(C(=O)NCCCNC(c1cc[nH]n1)=O)N1CCCC1=O CC1(C(=O)NCC2CCNC(=O)C2)CCCN1Cc1ccc(C(=O)O)[nH]1 C1(NC(C2CC3(CCOC3)C2)=O)CCC2CC1CN2C(C1CCC2(CCC2)O1)=O N1(CC(CNC(=O)NC(c2c(C)nccc2)C)(C)C)CCc2ccccc2C1 C1(CNC(CC(C)n2cccn2)=O)CC2CCC1N(C(C1CCCC1(C)C)=O)C2 N1(C(c2c(CC)nn(C)c2)=O)CCC(NC(c2cncn2C(C)C)=O)C(O)C1 c1(C(=O)NC2CC(C)N(c3ccncn3)C2)cc2c(F)c(F)ccc2[nH]1 CCS(=O)(=O)CC(=O)N(CC(C)C(=O)NCC1(O)CCCCC1)C C(=O)(N(CCC(=O)Nc1ccc(F)nc1)OC)C1(CC)CCCO1 C=CCCCC(C(=O)N(C)Cc1ccncn1)NC(C1SCCS1)=O c1(C(C)Nc2nc(CCC)c(Br)s2)cccc2cc[nH]c12 N1(C(c2ccn(C(C)C)n2)C(=O)NCC=C)CC2CCC2(CO)C1 Cc1[nH]nc2ncnc(NC(C)CNC(=O)CSC3CC3)c12 N1(C(C(C)OCc2cccc(C)c2)=O)CC2CN(C(=O)COC(F)F)CC2C1 C(=O)(CC(CC)CC(C)C)NC(c1cnn(C)c1)C(=O)NC(CCC)CC C(=O)(C(C(C)(C)O)NC(c1n[nH]c2c1CCC2)=O)N(CC(N1CCCC1)C)C CCC(C)C(C)C(=O)NCCC(CC)(CC)NC(c1cc(C(F)F)ccc1Cl)=O c1(OC)ccc(C)nc1C(=O)NC1CCCN(C(c2ccc([N+](=O)[O-])o2)=O)C1C C(=O)(C1CCCc2cncn21)NC(C1N(C(CC(=C=C)C)=O)CCC1)C O=C1CC(c2nc(CC3CC3C(F)(F)F)no2)CN1C1CCCC1 C(=O)(C(C(=O)N(CCO)Cc1ccc(C(=O)O)cc1)C(C)(C)C)OCC C(=O)(CCS(C)(=O)=O)NC(C1CCCN1C(C1CC2CCC1O2)=O)(C)C c1(OCCC(=O)N(CCC2CCN(C(CCC)=O)CC2)C)cc(C)ccc1C c1(NC(C(CNC(C2(C)CCC(C)CC2)=O)C(C)C)=O)cnc2[nH]cnc2c1 N1(C(=O)C=Cc2ccccc2)CCCC12CN(Cc1cccc(Cl)n1)C2 N1(C(C)C)CC(C(=O)NCCCC(C)NC(c2ccccc2CC#N)=O)CC1=O c1(C(N2CC(CN(C)C(c3cnc(S)nc3)=O)OCC2)=O)cnc2[nH]ccc2n1 Cc1cc(CC(=O)NC2CCCC(CNC(=O)CO)C2)cc(F)c1.C1CCC1 c1(OC)ccc2c(C(=O)NCCC(C)NC(c3cnn(C)c3C#N)=O)n[nH]c2c1 C=CCC(C)(C)CC(=O)NC1C=CCN(C(C2CCCC23CCC3)=O)C1 C1(NC(CC(CC)SC)=O)CCN(C(=O)Cc2ccc(C(=O)OC)nc2)C(C)C1 c1(C(=O)NC(C(C)C)C(C)NC(C2CCC=CCC2)=O)cc2c(cn1)CCCC2 Cc1ccc(C(=O)NCc2ccc(O)cn2)c(C(C)C)c1 C1(C(N2CC(OCC(C)C)C2)=O)(OC)CCN(C(=O)CC2CCCC3CC23)C1 c1(C(N2CCC(NC(CSCCOC)=O)C(C(C)C)C2)=O)ccc2occc2c1 c1(OC)ccc(C(=O)NC(C)CCC)c(F)c1.C1(N(CC=O)C)CCCC1O.N c1(C(C(=O)NC)N(C2CCCC2)C(c2ccc(F)cc2)C)ccc(C)c(OC)n1 Cc1nnc(CCC(=O)NCC2CCCC2NC(c2cnn(CC(C)C)c2)=O)o1 C=Cc1ccc(C(=O)NC2CCOC(C(=O)N(C)CCOC)C2)cc1 c1(C(N2CCC(CC)C2)=O)ccc(C#N)cc1.N1(S(C)(=O)=O)CCC1C(=O)N c1(-c2cn(CCC#N)nc2)cc(CN2CC(=O)NCC2C(=O)O)cc2c1OCO2 c1(CC=O)ccc(Br)cc1Cl.c1(COC)ccccc1CN1CC(F)(C)C1.N Cc1cccnc1-c1cn(CCCCNC(=O)CC(C)n2cccc2)nn1 C1(CC(=O)NCC2N(C(Cc3ccc(C)o3)=O)CCC2)CC(C2CC2)C1 C1(C(=O)NCCCC)C2CC3C(C2)C13.c1(C(=O)N)ccccn1.C(C)(C)C c1(CNC(Cc2cnc(C)[nH]2)=O)cccc(NC(=O)NC2CCN(C)C2C)c1 C1(C(N(C2CCN(C(COc3cccc(CC)c3)=O)C2)C)=O)CCC(F)(F)CC1 c1(C(N2CCC(C(C)NC(CCOCC#C)=O)C2)=O)cc(O)c2oc(C)nc2c1 c1(C(N2CC(CC(C)NC(C(CC)n3ccnc3)=O)C2)=O)sc(N(C)C)nc1Cl C=CC(CC)CC(=O)NC(CSCC)C(=O)NCC(C)(O)C(F)F N1(C(CCC2CC(OC)C2)=O)CCCCC1CCNC(=O)CCCCF N1(C(CCOC(C)C)=O)CC(CC(N2CC3CC2C3)=O)CC1C CC1COCCN1C(=O)COC1CCN(C(c2cn(C)cn2)=O)C1 N1(C(C(N2CCNC2=O)C)=O)CCC(NC(c2cccn2C2CC2)=O)C1(C)C CC1Cc2ccccc2N1C(=O)COC(=O)CC1CCC(=O)N1C C1(NC(c2cc(CC)no2)=O)CC2(C1)CC2NC(c1cc(C)c(Br)o1)=O C1(OCC)(CNC(c2csc(CO)n2)=O)CN(C(=O)C(C)N(C)C)C1 C(=O)C1=CC2C=CC(C1)C2.CC1(C)C(C(=O)NC2(C)CCC2)CC1(F)F.N N1(C(c2c(C)nn(CC)c2Cl)=O)CCCN(C(=O)CCn2ccnc2C)C(C)C1 C(=O)(NNc1ccco1)NC(CC)C(=O)Nc1nc(=N)[nH][nH]1 CC(C)C(O)CC(=O)N1CCC(C)(C(=O)NCCc2cc(O)ncn2)C1 c1(C(=O)NCC(C)(C)NC(c2c(CC)cno2)=O)ccc(C#N)c(F)c1 c1(CCC(N2CCC(CCNC(=O)C3=CCCC3)C2)=O)cc(F)cc(F)c1 c1(C(N2CC(CC)OCC2CC)C(=O)NC2CCOC2)cccc([N+](=O)[O-])c1C C(CNC(c1cc(C(C)C)[nH]n1)=O)(C(=O)NCCCc1cncnc1)OC C(=O)(C#CC1CCCO1)N1CC(OC)(C)C1.c1(N(CC=O)C)ccc(Cl)cn1.N c1(NC(C2C(NC(c3cnn(C(F)F)c3)=O)C2)=O)csc2nccnc12 C(=O)(C(F)(F)CO)NCC(C1CCC1)NC(c1c(CC)noc1)=O CCC(C)(CCNC(c1c[nH]c(=NC)s1)=O)NC(c1cocn1)=O c1(C(C(=O)NCCOCC)OC)ccc(Br)cc1.C(c1ccc[nH]1)=CC=O CCC(C#N)C(=O)NC(CC1CC1)C(=O)NCCOC1CCC1 C12(C(N3CCC3C3CCCCC3)=O)CC1CN(C(=O)CCc1nncs1)C2 N1(C(C2CC(=C)C2)=O)CCC(NC(C2CCCC2C(F)(F)F)=O)CC1 Cc1ccc(Cl)c(C(=O)NC(C2CCOC2)C)c1.C(=O)C(C)(C)CC1CC1.N N1(C(=O)Cn2nccn2)CCC(NC(C2CC(OC(F)F)C2)=O)C2(CCC2)C1 C(C(C(=O)N(C(C)C)C)C(C)(C)C)OCC=C.c1(C(=O)N)cccc(O)c1C CC1CCSCCN1C(=O)NCC1(c2ccccc2)CC1C(F)(F)F C1(COC)CCN(C(=O)C(F)(F)C(C)O)CC1.N1(CC=O)CCN(C)CC1.C CCC(CCC(=O)NCCCNC(=O)CC1CCCNC1=O)NC(C)=O c1(OCC(=O)NCC(C)NC(=O)CCP(C)(C)=O)ccc2cc(Br)ccc2c1 c1(CC(=O)NCCCNC(c2noc(CC)c2C)=O)c(F)cc(F)cc1F.C c1(C(N2C(CNC(c3cnc(SC)s3)=O)C=CC2)=O)cc(C)c(N)cc1Cl N1(C(C(c2cc(C(F)(F)F)ccn2)C)=O)CC(C(C)C)c2ccccc21 Cc1scnc1C(=O)NC(C1CCCN1C(c1ccncn1)=O)C C1(C)(CC(=O)N(C(C)(C(=O)N)C2CC2)C)CCCCC1.C1COC(=O)N1.C N1(C(C2CC(C)OC2)=O)CCC(OC2CN(C(=O)C3=C(Cl)CC3)C2)CC1 c1(NC(CCSCCNC(=O)CC2(CO)CCC2)=O)cccc(OCF)c1 C1(C(=O)NCc2cc(OC)nn2C)CCN(C(=O)C(O)C(F)(F)F)C1(C)C C(CC(=O)N(CC(C)(C)CN(C)C)C)(CC(C)C)NC(C=C(COC)C)=O c1(CC(=O)OC(CC#C)Cc2ccccc2)cn2ccccc2n1 C(=O)(C(F)(F)CCn1cccn1)N(CCNC(c1cnco1)=O)C1CC1 C1(OC)CC(NC(=O)CC2CCCCC2)CN(C(c2ccc(C)cc2)=O)C1 Cc1nn2c(C(N3CCNC(=O)C3)C(=O)NCCOC(F)F)c(C)nc2s1 C(CC(C)C)(C(=O)NC1CC1C)OC.c1(C=O)ccccc1C(C)(F)F.N C1C(C)C(=O)N1.N1(C(N(CC(=O)OC)C2CCC2)=O)CCCCC1 C1(N(CCNC(c2sc(Br)cc2Br)=O)Cc2ccccc2)CCc2nn[nH]c2C1 C(CCCCCCCO)=CC(=O)NCCCC(C)NC(=O)CC1C=CCCC1 n1(CC)ncc2c1CCCC2NC(=O)CCOc1cccc(F)c1C N1(C(C(CCC)C)=O)CC2CCC(C1)N2C(c1cc(C)ns1)=O Cc1ccc(NC(C2CN(C(C3CS(=O)(=O)C3)=O)CCC2(C)C)=O)c(F)c1F c1(C(C)(F)F)cncc(NCc2cc(Cl)on2)c1 N1(C(CCOCC)=O)CCOC2(CCC(NC(=O)CC(C)(C)C(F)(F)F)CC2)C1 N1(C(c2nc(C)sc2)=O)CC(C2CCCCN(C(c3c(Cl)nn(C)c3Cl)=O)C2)C1 c1(SC)ncc(C(=O)NC(CNC(c2c[nH]nc2F)=O)C2CC2)c(O)n1 c1(C(N(CC(C)NC(C2CCCN2C=O)=O)C)=O)ccn2c(O)nnc2c1 CC1(NC(=O)CC2(O)CCCCC2)CC2(CCC2)C1.C(=O)CCC1CCOC1.N c1(CC)noc(C(=O)NC2(CNC(N)=O)CCCCC2)c1C C1(C(N2CCC(C(CO)NC(C3CCC(OC)C3)=O)CC2)=O)CC2C=CC1CC2 C1(CNC(N2CC3(CSC3)C2)=O)CCCC(CO)C1 c1(NCC(=O)N(CCC=C)CC)cccc2c1OC(C)(C)C2 C1(CNC(C2N(C(C3C(C)CC3)=O)CC=CC2)=O)CCC2(CCC2)O1 CC1(C)CCN(CC(N2CC(NC(c3cn(CCO)nn3)=O)CC(F)C2)=O)CC1 c1(CC(=O)N(C2CCC(NC(C3CC(C)(C)C3)=O)C2)C)ccc(Cl)nc1 N1(C(c2cc(C)cc(C)c2)=O)CCC(NC(c2csnn2)=O)C(CO)CC1 N#Cc1cc(NC2CCC(NC(C3CCCCO3)=O)CC2)ccc1[N+](=O)[O-] C#CCC(C)C(=O)NCC1COCC1NC(=O)Cc1occc1C Cn1cc(C(=O)NCCCNC(C2(NC(N)=O)CCCC2)=O)nc1O c1(N2C(C)CN(C(C3Cc4nccnc4C3)=O)CC2)nc2c(cc1Cl)C(=O)OC2 c1(CC(=O)NCC2CC(NC(C3C(C)OCC3)=O)C2)c[nH]c2ccccc12 N1(CC(=O)NC(C)CC(C)NC(C2CCCCS2)=O)C(=O)CCC1=O C1(C(F)(F)F)(C(=O)NCCOCCNC(=O)CC2CCC2)CCC1 C1(C(N2CC(O)(CNC(CCc3n(CC)ccn3)=O)C2)=O)CC(O)C(F)C1 C1(O)(CNC(C2N(C(C(C)OCC(C)C)=O)CCC2)=O)CCC(C)(C)C1 Cc1cc2ncc(C(=O)NCCCCN(C)C(c3cnc(S)n3C)=O)c(C)n2n1 c1(N2CCC(CCOC)(NC(c3oncc3C)=O)C2)ncnc2sc(C)c(C)c12 C1(C(=O)NCC(COC(C)C)O)CN(C(=O)C=Cc2ccco2)CC1F C1(CCC)(C(=O)NC2CC(CCNC(=O)C(C)NC(C)=O)C2)CCC1 CC1(NC(=O)CC2CCCO2)CC(NC(c2cnn(C(F)F)c2)=O)C1 C(=O)(C1=C(Cl)CCOC1)NC(C(C)(C)NC(C(F)OC)=O)C N1(C(=O)Cc2ccsn2)CCCC(C2CN(C(=O)C3CCCc4ccnn43)C2)C1 N1(Cc2c(C)ncs2)CCC(C(=O)Nc2ccncn2)C(O)C1 C1(C(=O)NCC2(F)CCCN(C(c3n(CC)ncn3)=O)C2)CCCCN(C)C1=O c1(OC)ncc(Cl)c(C(=O)N(C)CCN(C)C(c2conc2C2CC2C)=O)c1Cl C1(C(=O)NCCC(=O)NCC(C)C)CSCCN1C(C1CCN1C)=O c1(CCC(=O)NC2CCC(N(C(CCOCC)=O)C)C2)ccc(Cl)c(OC)c1 N1(CCc2ncc(C(C)C)o2)CCN(C2CNC2)CC1.C(C(C)(C)C)=CC=O.C c1(C(N(CCCCCNC(=O)CO)C)=O)cc(OCC(F)F)ccn1 CC1CN(C(c2cscc2C(F)F)=O)CCC1CNC(=O)Cn1cccc1 C1(C(=O)NC(CC)C)CN(C(c2cnc(N(C)C)o2)=O)CCN1 C12(C(=O)NCC(C)N(C)C)CC(CCO1)N(C(=O)CCCC#N)C2 N1(C(c2n(COC)ncc2)=O)CCC(NC(=O)C(C)(C)c2cncs2)CC1C C=CC(CC)C(=O)N(CC(C)NC(C1(C)COC(=O)N1)=O)C c1(-c2cc(C(N(C3CCOCC3)CCC)=O)n[nH]2)ccc(OC)c(OC)c1 C(c1cccc(F)c1)=CC=O.Cn1nccc1C=CC(=O)NCC1C=CCC1 CC1CCC(=CC(=O)N)CC1.C1C(C)CCN1C(=O)CC1(N(C)C)CCC1.C CCCCCCC(CC)NC(C1(CF)CCN(C(C2CCCC(=O)CC2)=O)C1)=O CC(C)CCC(F)C(=O)NCC1C(C(=O)N)C1(C)C.C1C2CCC3C(C2)CC13 C1(CC(=O)N)CCCC(F)(F)C1.C1(C(=O)NC(C)C)(COC)CCCC1 c1(SCC)cc(C(=O)NCCCN(C(C2CC(C)CO2)=O)CC)ccn1 C12(NC(CCC#CC)=O)CCCC1(F)CN(C(=O)COc1c(C)n[nH]c1C)C2 C(c1ccccc1Cl)=CC(=O)N(C)CC1CN(C(=O)CC23CCCC2C3)CCO1 N1(C(c2c(CC)[nH]cc2)=O)CCSCC1CCNC(c1cccc(SC)c1)=O N1(C(CNC(C)=O)=O)CC2CC1CCC2NC(=O)CC(F)(F)Br C1(NC(C2C3(c4ccc(C)cc4)COC2C3)=O)CCC2(CCN2)CC1 C1(c2noc(C=Cc3cnn(-c4cccc(OC)c4)c3)n2)(NC)CCOCC1 C1(CNC(c2cnc(CCC)s2)=O)CN(C(=O)Cc2cn(C)nc2C)CCC1C c1(OC)ccc(NC(C2CCC(NCc3cccc(Br)c3O)C2)=O)c(C)c1 CC1Oc2c(NC(N3CC(CS(=O)(=O)C(F)F)C3)=O)cccc2C1C c1(C(N2CCC(N(C(COCc3ncc(C)o3)=O)C)C2)=O)scc(C)c1C c1(C(NCC)=O)ccc2c(c1)S(=O)(=O)NC2.C=CCC(C=O)NC(C)=O C(=O)(C(CCC(C)C)NC(=O)Cn1cc(C#N)cn1)NCCCC(=C)C c1(C(=O)NC(c2ccccc2)CN(CCCC)C)cn2cccc(C)c2n1 N1(C(C)C(=O)Nc2cc([N+](=O)[O-])ccc2Cl)Cc2cccc([N+](=O)[O-])c2C1 N1(C(c2c(C(C)(C)C)noc2)=O)CCC(F)(C)C1.c1(C=O)ncc(C(F)F)s1 C1(F)(CNC(C(C)c2ccco2)=O)COCCN(C(c2cc(Cl)ncc2O)=O)C1 C(=O)(C1=Cc2ccccc2OC=C1)NCC#CCNC(CCCC(C)C)=O C(=O)(C1=COCCO1)NC(C)C(c1ccccc1)NC(C12CCC1CC2)=O CON(C)S(=O)(=O)c1ccc(C(=O)NCc2ccnn2C2CC2)cc1 N1(C(CCn2ncc(C)c2)=O)CC(NC(=O)Cc2cnc[nH]2)CC(C)C1 CC1(C)CCC(C(=O)NCCNC(=O)C(c2ccccc2)F)OC1 C(=O)(CCC(C)C#N)N1C(CCNC(c2c(CC)occ2C)=O)COCC1 CC1(NC(c2ccccc2)=O)CCN(C(=O)Cc2cncc(O)c2)C1 N1(C(C(CC)N(C)C)=O)CCC(CO)(NC(C2CCC3(CC3)C2)=O)CC1 c1(C(C)(C)C(=O)N)ccc2c(c1)OCO2.C1(C=O)CN(C(N)=O)CCO1.C1CC1 C1(CC=O)CCCC2(CC2)C1.CC(C)C(C=O)NC(N)=O.C(CC)C(C)C.N c1(C=O)cc(OC(F)F)cc(F)c1.C(C(=O)NC1CCCC1)(C(C)C)OCC c1cnccn1.O=CCCN(C(=O)CCNCCCO)C1CC1.C1CCC1.C N1(C(C(CN(CC)CC)F)=O)CCC(C2CC2)CC1.C1(CC(=O)N)CCCC1O n1(CC)nc(C(=O)NCC(C)NC(C2CC(N(C)C)C2)=O)cc1C Cc1ccc(F)c(C(=O)NC2CC(C)(NC(=O)CN3CCC(=O)CC3)C2)c1 Cc1cc(C(=O)NC2CC2C(=O)NC2(c3ccsc3)CC2)cc(C#N)c1 C(CC1CCC1)(C=O)NC(C1(CCOC)CCC1)=O.C1(C(C)O)CCCC1.N c1(OCCNC(C(CCC)CCC)=O)ccc(S(=O)(=O)N2CCOCC2)cc1 N1(C(c2nc(C)c(C)s2)=O)CCN(C(c2cc3cscc3s2)=O)C(C)C1 c1(OC)ccc(C(N)=O)cc1C(N1CCCCC1)=O.C(=O)(CC)N.C(C)(C)C c1(C(=O)NCC(CN(C(c2c(CC)nccn2)=O)C)O)nnn2c1C(=O)NCC2 c1(C(=O)NCC(CCCC)NC(c2cnn(C(F)(F)F)c2)=O)c(F)ccnc1F N1(C(C(CC)=CC)=O)CCCC(C)C1CCNC(=O)Cc1ccc(F)cc1C C(=O)(CCCCC(C)C)NC(C1CCN(C(CSc2ccc(C)cc2C)=O)C1)C C1(CC)C(NC(c2[nH]cnc2C)=O)CCN1C(c1ccc(C2OCCO2)cc1)=O C1(O)(CC(C)C)CCN(C(=O)C(C)(C)C)C1.c1(C(=O)N)c[nH]c(C(N)=O)c1 c1(OC)cc(C(N2CCC(NC(=O)C(F)n3ccnc3)C(O)C2)=O)cc(F)c1 C12(CNC(CS(=O)(=O)NC)=O)CC(C1)CCO2.c1(C(=O)N)ncccc1Cl Cc1c(C(=O)N)noc1C1CC1.C12CC1CN(C(C1CC(F)(F)C1)=O)C2.C C12(C(N(C3CCSCC3)C)=O)CCC(n3cc(CNc4cc[nH]n4)nn3)(CC1)C2 C(=O)(CC(CC#N)c1ccccc1)N1CCC(N(C(=O)Cc2cnnn2C)C)C1 C=CCC(CC=C)C(=O)NCC1=CCCN(C(c2cc(OCC)ns2)=O)C1 Cc1cc(C(O)CN(C)C(c2ccc(=N)[nH]n2)=O)ccc1O CCC(C)(CC)C(=O)N1CCC(C)(CNC(=O)C(C(C)C)c2ccncc2)C1 CN=c1nc(C(=O)NC2CN(C(c3ncncc3Cl)=O)CC2C)cc(C)[nH]1 C(C)(CC(F)(F)F)NC(c1cnn(-c2nccs2)c1)=O.C1(C(=O)N)C=CCC1 c1(NC)ccc(C(=O)NCc2ccnc(Oc3ccccc3)c2)c(Cl)c1 c1(C(=O)NC2(C#N)CCN(S(=O)(=O)c3cn[nH]c3)C2)ccc(O)c2ncccc12 c1(C(=O)NC(C)C(=O)NC2(CO)CCC2)ccc(CO)nc1 c1(CC)nc(C(=O)NCCCN(C(=O)C)CC)cs1.C1CCCCC1.C=O C12CCC(F)(CC1)C2.c1(C(C)C)cc(C(=O)NC(C(=O)N)c2ccoc2)no1 N1(Cc2cc(C(=O)NC(C)C)no2)CCS(=O)(=O)CC1C c1(OC)ccc(C(=O)NC(C)CN(C)C(C2(CO)CC2)=O)c(Br)c1F N1(C(CCCOC(C)=O)=O)CCC(NC(c2cc(CO)on2)=O)CC(C)(C)C1 c1(SC)nc(N2CCCC(CNC(c3c(O)cccc3Cl)=O)C2)ncc1Br N1(C(C2CCN(C)C2)=O)CCC2(CCC2)C(CNC(=O)CCC2CCC2)C1 CCCCC(CNC(=O)CN(C1CCSC1)C)NC(C1(CCO)CCCC1)=O Cc1cc(C)c(-n2cc(C3(F)CN(C(C4CCCC5CC45)=O)C3)nn2)c(C)c1 CC1CCCCC1C(=O)NCC1(F)CN(C(=O)Cn2cnccc2=O)C1 C1(NC(C2(NC(c3cocn3)=O)CCSC2)=O)CCCC(F)(F)C1 N1(C(C2CC(SC)C2)=O)CCC(C)(C)C(CNC(C2CCCC(O)C2)=O)C1 c1(C(N(CCNC(=O)Cc2ccco2)CCOCCO)=O)cccc[n+]1[O-] Cc1oc(C)c(C(=O)NC(C)CC(=O)NC2CCCC2N=[N+]=[N-])c1C c1(C(=O)NCC(CC)(C)C(N2CCC(CO)=C(F)C2)=O)ccc2cncn2c1 c1(-c2ccc(SCC3CCC(C(=O)O)O3)s2)ccc(Br)cc1 c1(N2CC(C)C(C(=O)O)C2)snc(Cl)c1C#N c1(C(N2CC(N(C(C3CN(C(C)C)C3)=O)C)C(O)C2)=O)ccc2cnoc2c1 CN(C)S(=N)(=O)N1CCCC1C(=O)NC1CCCC1NC(c1cnnn1C)=O N1(C(C(C)Cc2cnc[nH]2)=O)CCC2CN(C(C3(C(F)(F)F)CCC3)=O)CC2C1 C1(C(C)C)CN(C(=O)COCCN(C)C)CCCN1C(=O)CC(O)c1ccccc1 N1(C(c2cncc(C)n2)=O)CCC(NC(=O)C(C(C)O)N(C)C)C(O)C1 C(=O)(CC(O)CC(C)(C)C)N1CCCN(C(c2ccc(C#C)cc2F)=O)CC1C c1(C(N2CCC3(C2)CC3)=O)cc2c(s1)CCOC2.C1(C)(C(NC)=O)CC1(F)F.C O=C1COc2ccc(C(N3CCCC3C(=O)Nc3cncnc3I)=O)cc2N1 CCC(CC)CCNC(C1CC2C(C1)C2(C)C)=O.C1(C=O)CCN(C)C(C)C1.N O=C(C(O)CCCc1ccccc1)NCCN(C(C1(CCO)CC1)=O)C1CC1 C1(C2CCCCO2)(C(=O)N)CCCO1.C1(NC(=O)C(F)=C2CCC2)(C)CCCC1 Cc1noc(C(F)(F)F)c1C(=O)NC1CCCC1.c1(C=O)cnc(C(C)C)[nH]1 C1(C(=O)NCCCC=C)(COC)CCOCC1.n1(CCCC=O)c(O)nnc1O.N CC(C)C(C)(C)C(=O)N1CC(C)(NC(=O)Cc2cccc(Br)c2)C1 Cc1cccc(C(=O)NC(C2CCN(C(=O)C(O)C3CCCC3)C2)C)c1C N1(CCNC(C2CCC(C)C2)=O)CCCCC1.C(=O)(C(O)CN1CCCC1)N N1(C(C(C)OCC)=O)CCN(C(=O)CN2C(=O)CCC2=O)CC1C N1(C(CCC=C)=O)CCC(OCCNC(C2CCOC2c2ccccc2)=O)CC1 c1(CCC(=O)OCC)nnc(CNC=O)s1.c1nc(-c2cccnc2)cs1.N O=S(=O)(c1cccc(N2CCCCC(F)(F)C2)n1)NC1CCC(CO)CC1 CCC(CC)C(F)C(=O)N(CCC(N1CCC(C2CC2)C1)=O)CCO c1(C(N2C3CC(CNC(c4c(C)cccc4)=O)C2CC3)=O)occ2c1CCCC2 N1(C(CCC(=O)NC)=O)CC2CC1CCC2NC(C1(N(C)C)CCC1)=O CC(CF)C(=O)NC(C1CCCN1C(c1cc(-c2ccccc2)n[nH]1)=O)(C)C C#Cc1cc(NC(=O)C(C)N(C(c2cc(C)cc(C)n2)=O)CC)cc(F)c1 c1(C(=O)NCC2N(C(C=CC)=O)CCCC2)ccc2c(cnn2C)c1 CCC(C)(C)CC(=O)NCCC1CCN(C(=O)C(CC(C)C)OC)CC1 C(c1ccn[nH]1)=CC(N1CCC(N(C(=O)CCNC(=O)O)CC)C1)=O CC1(C)CC(C(=O)NC2CCOCC2F)(CNC(c2ncc[nH]2)=O)C1 c1(CCC(=O)OC(C2(O)CCOC2)C)nc(-c2ccco2)no1 C=CC1OCCC1C(=O)NC1(C)CN(C(C2CCCN(C(=O)COC)C2)=O)C1 CCCC(CCCNC(c1cnnc(O)c1)=O)NC(c1cc2sccc2s1)=O c1(C(=O)NCCCCCC(N2CC(C(C)C)NC(=O)C2)=O)cccc2c1OCO2 C(=O)(C(C)(C)S(C)(=O)=O)N.Cc1ccoc1CC(=O)NCCc1ccccc1 C1(C(N2C(C3CCCN(C(=O)C(F)(F)CO)C3)CCC2)=O)CC2(CCO1)CC2 c1(OCC(O)C(F)F)ccc(SC(F)(F)F)cc1 C(=O)(C(CC=C)CC(C)C)N1C(CC(=O)NCC(C)OCC=C)CCCC1 C1(C(=O)NCc2cn(C)nc2Cl)CCC(=O)CC1(C)C O=C(C1=CCCOC1)NCCN1CCN(C(c2cc(Cl)no2)=O)CC1 CC1(F)CN(C(c2cocn2)=O)CCN(C(=O)CCc2nc(=N)[nH][nH]2)C1 C(C(C(=O)NC(C1CCCN1C(=O)COC1CC=CC1)(C)C)OC)OC C1(NC(CCCCCn2cc(C(n3cccc3)C)nn2)=O)CC(C)(C)OC1(C)C C1(CN(C(C(CC)O)=O)C)CCC(CNC(=O)C(C)NC=O)CC1 C1(CS(C)(=O)=O)CCCCN1C(c1cnnn1C1CC1)C(=O)NC1CCC1 C=C=CCN=c1nc(N2CCC(c3nc(=N)[nH][nH]3)C2)c2cc(F)cc(F)c2[nH]1 C1(CC(=O)NCC(O)CNC(=O)C2CC2)CC(C(F)F)C1 c1(C(=O)NCCCC(C)(C)NC(c2cnc[nH]2)=O)ccc2c(c1)OCC2 N1(C(CC(CC)C)=O)CCC(NC(=O)Cc2ccns2)CC1c1ccccc1 N1(C(c2nccc(N)c2)=O)CCCC(CO)(NC(=O)Cc2c(F)cccc2Cl)C1 c1(OCC(=O)NCCCC)cccc(C#N)c1.c1(C(C=O)C)cccc(F)c1.N N1(C(C2(C#C)CCN(C(=O)COCCF)CC2)=O)CCOC2COCC2C1 C1(C(N(C2CCN(C(c3c(Cl)cnn3C)=O)CC2)CC)=O)CC2(CCC2)CO1.C Cc1cc(C)c(C(=O)NCC2(NC(=O)C#CC(C)C)CCCCC2C)c(N)c1 Cc1n[nH]c(C)c1C(C)C(=O)NCCC1CSCCN1C(=O)CO.c1cn[nH]c1 c1(CNC(CCCNC(C=CC(CC)C)=O)=O)cc(C)ccn1 C1(CC=C)(C(=O)NC)CCN(C(=O)CC2CN(C)C2)C1.C1(C=O)CC1 C1(C(N2C(CN(C)C(c3cccc(=O)n3C)=O)CCCC2)=O)Cc2cscc2C1 c1(N2CC(NC(C3C(C)CCC3)=O)C(C)CC2)ncnc(Cl)c1C#N N1(C(c2cc(F)cc(N)c2F)=O)CCC2(CC1)CN(C(c1ccncn1)=O)C2 N1(C(c2n[nH]c3c2CN(C(=O)OC(C)(C)C)CC3)=O)CCCC2(CCC2O)C1 Cc1cc(C(=O)NC(C)CC(C)NC(c2ccc(C(N)=O)[nH]2)=O)cc(C)c1O C(=O)(C1=CCC(F)(F)CC1)N1CC(NC(c2ncc(C)nc2)=O)C(C)C1 C1CC2(CCN(C(c3ccccn3)=O)CC2)CO1.C(C(=O)N)NC(=O)OCC C#Cc1ccc(C(=O)N(CC(C)NC(=O)CCC(C)C#N)C)c(C)c1 N1(C(c2cnn(CC)c2C)=O)CC2(COC)CC1(C)C2.C(=O)C(C)(CC)CO N(C)(C1CCc2cc(Cl)ccc21)C(c1cc(C)c(F)cc1)C(=O)NC(C)(C)C C(CCN(C(=O)C(C)CSC(F)(F)F)C)C(C)(C)C.Cc1nccn1CC=O.N c1(CC)ccccc1OCCC(=O)NC1CCCC1CNC(=O)C(F)CC c1(C(=O)NC2CCN(C(c3cnn(C)c3F)=O)CC2F)cnc2ncccn12 C#CC1(OCC(=O)NC(C)(C)CNC(C2CC2COC)=O)COC1 N1(C(C2C(C(C)O)C2)=O)CCC2(CC1)C(NC(c1nncs1)=O)CS2(=O)=O C1(C(=O)NCCN2CCCN(C(CC=CC=C)=O)CC2)Cc2cc(C)ccc2S1 c1(CC(=O)OC)ccccc1C=O.C1(CC=O)NC(=O)NC1=O.C1CC1.N O=C1CCCc2ccc(NC(C34CCN(C(c5cscn5)=O)CC3C4)=O)cc21 N1(C(CC(C)(C)O)=O)CCC2CN(C(C3(O)CCSCC3)=O)CCC12 c1(C(=O)NC2CCC(NC(c3cc(Cl)cnc3F)=O)C2)ccc2nc(Br)sc2c1 C1(NC(CCC=C)(CC)c2nnnn2C(C)C)CCN(S(N)(=O)=O)C1 C(=O)(C(C(C)O)N(C)C)NCC1C(C(N(CC(CCC)C)C)=O)OCC1 C1(NC(C2(C)CC2Br)=O)CCN(c2nn[nH]n2)CC1 N1(C(C2C(SC)CCC2)=O)CCCC2(CCN(C(C3(Br)CC3)=O)CC2)C1 C(=O)(C(C)CC(C)CC)N(C1CCN(Cc2nc(C(C)OCC)sc2)C1)C N1(C(C(C)OCOC)=O)CC2(CNC(=O)CCc3cn(C)nc3C)CCC1CC2 C(=O)(C1CNC(=O)c2ccccc21)c1nccc(C(C)(C)C)n1 c1(C(N2CCCC(NC(C3C(=C)C3)=O)C2)=O)cccc2c(Br)cccc12 C1(Nc2cc(NCC(C3CCCO3)OCC)ncn2)CC2(CCC(NC)CC2)C1 N1(C(C(C(C)C)=O)=O)CCC(C)(C)C1CC(=O)NC12CC(C1)C2 c1(C(N2C(C)CCC2)=O)cc(C)c(O)nn1.c1(CNC)cc(C(=O)N)nn1C N1(C(CCCCCC#C)=O)CCC2(CCC2NC(=O)Cc2cnc[nH]2)CC1 C#CC(CC(C)(C)C)NC(=O)CC(CNC(=O)CC1(C)CCOCC1)OC N1(C(c2cnc(C)nc2C)=O)CCN(C(c2cccnn2)=O)C2CCC12 C(=O)(C(C(C)CC1CC1)N1CCCN(c2ccccc2OC)CC1)NC N1(C(C(=O)NCC)C)CCC(C(=O)N(C)CC2CCN(C)C2)CC1 n1(C(C)C)ncc2c(NCC3CC(C(F)F)C3)[nH]c(=NCc3nc(Cl)cs3)nc12 c1(C(=O)NCC(CC=C)NC(c2[nH]cnc2C)=O)cc2c(C)nn(CC)c2s1 CC1(CNC(c2csc(-c3ccoc3)n2)=O)CCCN1C(=O)Cc1sccc1Cl C(=O)(CCC1=CCCCC1)NCC(C(C)C)C(=O)N1CCOC(CN=[N+]=[N-])C1 c1(CCC(=O)NC(C(=O)OC)Cn2cncn2)n[nH]c2cc(OC)ccc12 C(C(C(=O)N1CCC1)n1cc(CNC2(N3CCCC3)CCC2)nn1)OCC c1(C(=O)NCCN(C(C2(C#C)CC2)=O)C2CC2)cc(Br)ccc1F C1(C=O)CS(=O)(=O)CC(=O)N1.C1(C)(C(N2CC(C)CC2)=O)CCC(=O)CC1.N C1(CNC(C(n2cc(C)nc2)(C)C)=O)CC(O)CN1C(=O)CC(C)(F)F Cc1ccc(O)cc1C(N1CC(C)CC1C(=O)NCC1CC1(F)F)=O N#Cc1ccc(C(=O)NCCNC(=O)CN(c2ccncc2)N)nc1 C1(CC(=O)NCc2onc(C)n2)CC(O)CN1C(=O)C=Cc1ccco1 C(=O)(C1=Cc2ccccc2C1O)NC1(CNC(C(COC)OC)=O)CCC1 C(=O)(C1CCCc2c[nH]nc21)N1C(CNC(c2c(OC)nccc2)=O)CCC1 Cc1nn(C)c(N)c1C(N1CCC1(C)CC(=O)NCCCCN=[N+]=[N-])=O c1(OCC)ncc(C(=O)NC2CN(C(=O)CC3(C)CC3(Cl)Cl)C2)cn1 c1(C(=O)NC2CCN(C(C=C)=O)CC2F)ccc(N=[N+]=[N-])cc1 N1(C(C2CCN(C(c3cccc(C)c3)=O)CC2)=O)CCN(C)CC1(C)C c1(C(N(CCCNC(C2CC3(C2)CC3F)=O)CC)=O)cc(F)ccc1F N1(C(=O)NCc2cccc(Nc3nc(Br)cs3)c2)CCc2ccc(O)cc2C1 C(=O)(C(F)(F)CC(C)C)NC1C(NC(c2c(CC)ncnc2)=O)CCC1 c1(C(C(=O)NCCCF)N(CC)CC2CCCO2)ccnc(N(C)C)c1 Cc1cncc(NC(=O)N(C2CC(O)C2(C)C)C)c1 C1(NC(C(n2c(C)ccn2)C)=O)CC(NC(c2cnn(C)c2Br)=O)C(O)C1 C1(C(N(C)CC2(NC(C3CCCOCC3)=O)CC2)=O)CSc2ccccc2O1 c1(C(=O)OC)ccc(C(=O)NC2CN(C(=O)C(c3cnn(C)c3)C)CC2C)nc1 C(CC(C(C)C)NC(c1coc(C(F)F)c1)=O)N(C(C=C)=O)C c1(CC=O)cc(C)cc(F)c1.C1(N(C(=O)C(C)=O)CC)CCN(CCO)C1 C(C(C)(C)C(=O)NCC1CCCN(C)C1)N(C(=O)COC1CCOCC1)C CCCC(O)CC(=O)NCC(C)CN(C)C(c1ccoc1)=O [N-]=[N+]=NCC(=O)N1CC(C(O)C(=O)NCCC2CCCC2)C1 C1(NC(C(C(C)C)SC)=O)C2CCC1N(C(C1CC(O)C1)=O)C2 c1(C(C)C)ccc(C(N2CCC2CNC(=O)CC2CC(F)(F)C2)=O)cc1Cl c1(C(=O)NCC2CN(C(C3(C4CCCO4)CC3)=O)CCO2)occ2c1CCOC2 N1(C(c2c(CC)ocn2)=O)CCC(NC(c2ccnc(C)c2)=O)C(CO)CC1 N1(C(C(CO)NC(C(C)SCC)=O)=O)CCc2sccc2C1 N1(C(C(C(=C)Cl)(C)C)=O)CC2CCC1C1CN(C(c3c(C)cc[nH]c3=N)=O)CC21 C1(CC=C)(NC(CCC=C)=O)CCN(C(C2CCCNC2=O)=O)C1 C=CC1(C(=O)NCC2(OC)CCN(C(C3(C)CNC(=O)C3)=O)C2)CCOCC1 Cc1cc(C(=O)NC2CC2NC(c2cc3[nH]ccc3s2)=O)ncc1C(N)=O c1(C(N(CCN(C(=O)C2=NNC(=O)CC2)C(C)C)C)=O)cnn2c1N(C)CC2 CN1CCN(C(=O)CSCCN(C)C)CC1.c1(C=O)conc1C1CCCC1.N c1(CCC(=O)NCCN(CCOC)Cc2nnc(C)s2)cnn(C)c1C c1(OC)cnc(C(=O)NCCCC2(NC(=O)CC(O)C3CCCC3)CC2)cn1 c1(NC(C2CCN(C(CC3(OCC)CC3)=O)CC2C)=O)ccc2n[nH]cc2c1 C=CCC(CNC(=O)CCC1CCCN1C)C(=O)N1CC(O)(CC=C)C1 C1(NC(C(COC)COC)=O)CC12CCN(C(=O)CC1COC(=O)C1)CC2 C1(NC(C2N(C(C(C)n3cnnn3)=O)CCC2)=O)CNC(=O)OC1 N1(C(CCC2OCC(C)(C)C2)=O)CC2CC(NC(=O)C(F)C3CCOC3)CC2C1 C1(NC(CCCC=C)=O)CN(C(c2cc[nH]n2)=O)C2CCCC12 c1(CNC(C=C(CC)CC)=O)cc[nH]c1C(=O)OC(C1CC1N(C)C)C O=C1CCCCC(C(N2CC3CC3(NC(c3ccc(F)cc3F)=O)C2)=O)N1 C1(C(=O)NCC2N(C(=O)CC(C)(C)F)CCC(C)C2)CN2CCCN1CC2 c1(N2C(C)CC(CNC(c3cnc(C)s3)=O)C2)nc2cc(F)cc(F)c2o1 CCCCC(C)C(C(=O)NCC(F)F)N1CCC(NS(=O)(=O)N(C)C)CC1 C(C(C)(C)CC(=O)NC1CN(C)NC1=O)NC(C(CC)=CC)=O N1(C(C2(O)CCC(CC)C2)=O)CCOC2(C1)CN(C(=O)C(C)(C)C(F)F)C2 C(=O)(C(C)(C)c1cscn1)NCC(C)N(C(=O)CN1CC=CC1)C CCCCC(CC)CC(c1nnnn1C1CCCCC1)Nc1ccc(Br)nc1C Cc1cc(=N)[nH]cc1C(N1CC(NC(=O)C(C)c2cccs2)C(C)(C)C1)=O Cc1cc(NC(C2(F)CCN(C(C3C4CCC(F)C34)=O)CC2)=O)cnc1O Cc1nc2c(N3CCCCC(NC(c4csc(Br)c4)=O)C3)ncnc2[nH]1 CN1CCN(C(c2sccc2C#N)=O)CC1CNC(C1CC2(CCC2)C1)=O c1(C(=O)NC(C)CCNC(=O)C(F)(F)C2CCOCC2)cc(Cl)cc(Cl)c1O c1(C(N2CC(OC3CCN(C(c4cnc(C)o4)=O)CC3)C2)=O)[nH]c(=N)ccc1C c1(C(N2CCC(NC(CSCC(C)C)=O)C(C)C2)=O)cnc2[nH]nnc2c1 c1(C(N2CCC(O)C2)=O)ccc(F)c(C(F)F)n1.C(C)(C(=O)N)OCC.C C(c1cncc(O)c1)=CC(=O)NC(C1OCCN(C(CC(=C)C)=O)C1)C C1(C(N2CCC(NC(c3c(C)cco3)=O)CC2)=O)CC12CCS(=O)(=O)CC2 c1(CNC2(c3nnnn3CCOC)CCC(C#C)CC2)ccc(S(=O)(=O)CC)s1 N1(C(C(C)CSc2ccc(F)cc2)=O)CC(NC(=O)C(CO)N(C)C)CC(F)C1 C1(C(=O)NCC2OCCN(C(C)C)C2)CCC2(C1)CC2(F)F c1(CCC(=O)NC(CC(C)NC(=O)CC2CCCOC2)C)ccnc(Cl)c1 C1(C(=O)NCC(CC)OC)C2CC(O)C(C2)N1C(c1cncc(F)c1C)=O C1(CC(=O)NC(C2(CO)CC2)C)CCCN1C(=O)Cc1cn(C)nn1 C1(CC#C)(C(=O)NCC(C)(C)F)CCN(C(=O)C#CC2CC2)C1 C(=O)(N=c1[nH]oc2cc(Br)ccc12)C1C(C(N=c2cc(C)[nH][nH]2)=O)C1 C(N=c1ccc(Br)c(S(=O)(=O)N(CCO)CC)[nH]1)c1c(CC)con1 c1(CCC(=O)Nc2c(OC)nn(C)c2)ccc(Br)cc1F NC1CCCN(C(c2c[nH]nc2CN)=O)C1CCO C(CC(C)C)(CC(C)C)NC(c1cc(CNC(CN(C)CC)=O)sc1)=O C(c1ccc(O)cc1)=CC(=O)NCC(C1CC1)NC(=O)CC1(C)CC1 CC(C)(CCNC(c1sccc1C(F)F)=O)NC(=O)Cc1nc(=N)[nH][nH]1 C=CC1(C(=O)NC2CC(NC(=O)CC3CCN(CC(F)F)CC3)C2)CCOCC1 N1(C(=O)NCC(c2ccc(Cl)cn2)(C)C)CC(=O)NC2CCCC2(C)C1 C1(S(=O)c2ccccc2)(C(=O)NC2CC(NC(=O)C(F)F)C2)CCC1 C1(NC(c2c(C)cnnc2)=O)CN(c2ncncc2I)CC(F)(F)C1 Cc1ccc(C(=O)NCCN2CCN(C(C34COCC(C3)C4)=O)CC2)c(O)n1 C(=O)(C(O)C(C(C)C)S)NC1(COC)CCN(C(C(C(C=C)C)C)=O)CC1.C c1(C(N2CCN(C(CN(C(C)C)C)=O)CC2CF)=O)cc2n(n1)CC(C)(C)CO2 C(=O)(C1CCCc2nccn21)N1CCC2(CN(C(C(C)NC(C)=O)=O)C2)CC1 C1(NC(C2N(C)C(=O)CC2)=O)CN(C(c2ncsc2S(N)(=O)=O)=O)CC1N=[N+]=[N-] N1(C(COCCC=C)=O)CC(NC(c2nc(C(C)C)ncc2Cl)=O)CC(O)C1 C(=O)(C1COc2ccccc21)NCC1(C)OCCN(C(c2ccc(OC)o2)=O)C1 c1cccc2cccnc12.C1(CN(C)C(C2(F)CC2)=O)CCCN1C(=O)C=O.N Cc1[nH]ccc1C(N1CC(CC(C)NC(=O)C(C)(C)c2cscc2Cl)C1)=O N1(C(c2c(C(=O)OC)c[nH]n2)=O)CCOC2CN(C(=O)C(=O)NC3CC3)CC12 Cc1ccc(F)cc1C(N1CCC(n2cc(CN3CC4CC4C3)nn2)CC1)=O c1(C(=O)NCCC2(O)CCCN(C(C3(F)CC=CC3)=O)C2)ccc2cccnn12 C(=O)(CC(CC)C(F)F)NC(CCC=C)C(=O)NCC(C)CC1CCC1 O=C(NOCOC1CC(F)(F)CO1)C1COc2cc(F)ccc21.c12cn(nn1)C2 C(=O)(C(CCSC)NC(C1COC(=O)N1)=O)NC1CCN(CCC)C1 c1(C(N2CC(NC(C3C(C)OCCO3)=O)C(O)C2)=O)c(C2CC2)nc2sccn12 c1(C(N2CCCC(F)(CNC(C3(F)C(C)C3)=O)C2)=O)cc(F)c(F)cc1O n1(CC(=O)NC2CN(C(CC(C=C)(C)C)=O)CC2(C)C)cc2ncccc2n1 Cc1ccc(C(N2CCC(C(C)C(=O)NCC(O)CC3CCC3)C2)=O)c(F)c1 C(=O)(CCCCC(C(F)(F)F)N)OC.C12(C=O)CCC(CC1)C(C)O2 N1(C(c2occ(C(C)=O)c2)=O)CC(NC(=O)CC)C(C)C1.c1(C=O)cccs1 C(=O)(CC(C)C(C)C)N1CC(SC)C(NC(c2occc2C)=O)C1 C1(NC(CC(COC)NC(=O)CC2CCOC2=O)=O)CN(C)CCC1O C12(NC(C3CC(=O)N3)=O)CCCC1(F)CN(C(c1oc3ccccc3c1Cl)=O)C2 CC1CNC(=O)CN1C(C12CC(CO)(CN1C(C13CCCCC1C3)=O)C2)=O c1(OC)ccc(CNC(=O)Cc2cnc(Cl)cc2C)cc1N1CCCC1=O c1(NC(=O)C(=O)N(c2ccc(Cl)cc2)CC2CCCN2)cc(Br)c2c(c1)OCO2 C(=O)(C1=CCCOC1)N1CCC(C)(CCNC(Cc2c(C)cc(C)s2)=O)C1 N1(C(C2C(C)(C)C2NC(c2ccc[nH]2)=O)=O)Cc2ccccc2C1 N1(C(c2nn(C(CC)CC)c(C)c2)=O)CCN(C(C2CC2C(N)=O)=O)CC1CC CC(C(C)(C)C)=CC(=O)NC1CCN(CCC)C1.C12(C(=O)N)CC(C1)C2 C1(C(N2CCC(C)(CC)CC2)=O)CN(C(=O)C(n2cc(C)cn2)C)C2(CCC2)C1 C1(C)(NC(CNC(CNC(C)=O)=O)=O)CC(C)C1.C(=O)CC1CC1 C1(C(C)C)OCCCC1CNC(=O)CC1(c2ccc(Br)cn2)CCC1 C1(CC)CC(C)CN(C(C2CCN2C(=O)CN2CCCC2)=O)C1 c1(C(=O)NC2C3(CCN(C(C4C(=C)C4)=O)C3)CCC2)cc(O)c2[nH]c(C)nc2c1 N1(C(C(CCCC)N(C)C)=O)CCC(C)(C)CC1C(N1CCC(CCF)CC1)=O C1(C(=O)NC2CC(CNC(CCCCCSC)=O)C2)CCCC12CCOCC2 c1(C(=O)NC2CC(C(N(C(C)C3CC3)CC)=O)OCC2)ccc(C)c(F)c1 c1(NCC2CCN(C(C3C(CC)CCCC3)=O)C2)ncc(C#N)cc1Br N1(C(C(CCC)N(C)CCc2ccccc2)=O)CC(c2ccccc2)CC1(C)C c1(-c2c(C(N3CCC(Cc4ccccc4)CC3)=O)nccc2)c[nH]c2nccc-2c1 C1(NC(c2c(C)cc(CNC(c3cnn(C)c3N)=O)o2)=O)CCCN(O)C1=O Cc1[nH]c(Cl)nc(=NCC(C)(C2CC2)NC(C2CC(C)OC2C)=O)c1C#N n1(CC)ncc2c(C(N3CC(F)CCC(F)C3)=O)cc(C3CC3)nc12 C1(CNC(C=C(C)Cl)=O)N(C(c2cccn2C)=O)CCCC1(C)C CC1CCN(C(c2cc(C3CCC3)[nH]n2)=O)C(C)C1.C1(C=O)C(C#N)C1(C)C.N C=CCCCC(C(=O)NC1CCCOC1)NC(=O)CCC(C)OCC N1(C(C2C3(CC(NC(C(CC=C)C)=O)C3)C2)=O)CCC(F)(CF)CC1 c1(C(N2CC(CC(N3CCC(NCC)C3)=O)C2)=O)c(C)cccc1[N+](=O)[O-].C C=CC(C)(O)C(=O)NCC1CC(C)N(C(c2nn(CC)nc2C)=O)C1 CC(F)C(C)NC(=O)C(C1CC1)N(C)C(c1nc[nH]n1)=O N1(C(CN(CCC)C)=O)CCN(c2nccc(N(C(C)CO)C)n2)CC1 CC1C2CCCCC2CN1C(c1ccn2c1CSCC2)=O N1(C(C(C(C)(C)O)NC(C(C(C)C)C#N)=O)=O)CC(=O)NC(C)(C)C1 Cc1cnc(C(N2CCC(n3cnnn3)C2)C(=O)NC2CCOC2)s1 N1(C(C2(F)C(C)OCC2)=O)CC2CC(C1)N2C(c1ccc[n+]([O-])c1)=O Cc1cc(C#N)c[nH]c1=NC1CCCCC1CNC(=O)CC1OCCC1(C)C N1(C(c2cc(-c3ccc(Cl)cc3Cl)on2)=O)CCC2(C1)CC2(F)F c1(OC)cc(=O)n(C)cc1C(=O)NCC1CCN(Cc2cccc(F)c2)CC1 C(=O)(CCCS(C)(=O)=O)N1CC(CC)C(NC(C2CC(C(C)C)C2)=O)CC1 C1CCN(C)C1=O.c1(COC)cc(C(=O)NC(C)(C(=O)N)C2CCC2)no1 C1(C(N2CCOC(C(=O)NCCCCN3CCC3)C2)=O)(OC)CCC(C)C1 CCC(CC(=O)N1CCCC1CN(C(=O)C(C)(C)COCC(F)F)C)SC C1(NC(c2cc(C)ncn2)=O)(CNC(=O)CC(O)C2CCCC2)CCCCC1C C1(NC(C2CC=CCO2)=O)CCOC12CCN(C(C1CCC3(CC1)CC3)=O)CC2 c1(C(=O)NCC2CN(C(C(COC)C)=O)C(C)(C)C2)ccc(OC)c(OC)c1C N1(CC)CC(C(=O)NC)CC(C)(C)C1.C(C)C=O.C(COCCO)OC N1(C(C2(OCC)CCC2)=O)CC2(C1)CN(C(C1CC(O)C1)=O)CCO2 c1(C(N(CC(C)NC(C2CC(CC3CC3)C2)=O)C)=O)cncc2[nH]ccc12 C1(C(N2CCC(C(C(C)C)NC(c3csnn3)=O)CC2)=O)CCCCC12CCC2 C(C(=O)NCc1ncc(C)cc1C)(C(C)CC)N(C(c1ccc(C#C)o1)=O)C C(=O)(C(C)C(C)NC(c1csc(F)c1)=O)NCCCn1ncc(C)c1 c1(C(=O)NCC2(O)CN(C(C3CCC(CO)CC3)=O)C2)c[nH]c2ncccc12 c1(CCC(=O)NCC(C)NC(c2n(C(CC)C)ncc2)=O)ccc(Cl)nc1.C C1(NC(CC(C)OC)=O)(CNC(=O)C(O)P(C)(C)=O)CCCCCC1 c1(NCCCC(C)(C)NC(c2cc(C)n(C)n2)=O)[nH]c(=O)n(C)c(=O)c1C#N CC(=O)C(C)CC(C)C(=O)NCC(CC1CCCC1)C(=O)Nc1cn(C)nc1O CC1(C)CN(C(c2ccsn2)=O)CC1NC(=O)CCc1cccc(C#N)c1 CCCCC(CC)C(=O)NCc1cc(O)nc(CNC(c2nnccc2C)=O)n1 O(NC(=O)C(C1(O)CCC1)NC(=O)CCc1cnn(C)c1)CC(C(C)C)O C#Cc1ccc(C(=O)NCC(C)(C)C(=O)N(C2CC(=C)C2)C)o1 C1(C(N(CC)C)=O)CC2COCC(C1)C2(F)F.CC(C1CC1)=CC(=O)NCC C(C#CC(C)NCCCc1cccn1C)(OCC)OCC N1(C(C=CCN(C(COCCC#C)=O)C)=O)CCCC2CC12 CC(C)(C(=O)NC1CCCC1NC(C12CCCC1C2)=O)c1ccns1 C12(NC(C(C)n3cnnn3)=O)CCCC1(F)CN(C(c1cn(C3CC3)cn1)=O)C2 C(=O)(C#CC1CCOC1)NCC1N(C(c2cncc(N)c2)=O)CCC1 CCC(C)CCC(=O)N1CCCC(CNC(=O)C(C)(C)c2cnco2)CC1 C1(NC(c2cnccn2)=O)CN(C(c2ccoc2Br)=O)CC2(CC2)C1 c1(OCC(=O)NCC2CC(NC(=O)Cn3cnnn3)C2)cncc(Cl)n1 Cc1nc2c([nH]1)C(C(=O)NC(C)CCCNC(=O)C(F)(F)C(F)(F)F)CCC2 C1(C)(CC=O)CCCCC1.C1(C(=O)NCC=CCOC)(C)CCCO1.N C1(NC(c2cc(C)nnc2)=O)CC2CC(NC(C3C=CCS3)=O)C1C2 N1(C(c2c(C(C)C)ocn2)=O)CCC(C)C(NC(C2(C)CS(=O)(=O)C2)=O)C1 c1(C=O)ccccc1.C1(=O)C(C)O1.C(=O)(CC=C(C)C)NCC C(C1C(C)C1(Cl)Cl)=CC(=O)NC(C(C)NC(=O)Cc1cncnc1)(C)C C1(NC(=O)C(c2ccc(F)cc2)CO)CCCN(C(=O)CCC2CCOCC2)C1 C1(C(=O)NCC2N(C(C(CC)CC(F)F)=O)CCC2C)CC2CC1C1C2C1(F)F N1(C(C2CC(OC)C2)=O)CC(C)C(C)(C)C1.c1(CC=O)cccc(O)c1F.N C1(CNC(c2ncn(CC)n2)=O)C2CN(C(=O)CN3CC(C)C3)CC12.O CC1CCCN(C(=O)Cc2cnns2)C1CCNC(=O)C(C)(C)C1CCOCC1 c1(C(N2CCCC(c3occ(C(C)(C)C)n3)C2)=O)cnc2n1CCCCC2 C12(C(=O)NC(C)CN3CCN(C(=O)C(F)(F)CO)CC3)CCCC(=O)N1CCC2 Cc1ccnc(C(=O)N(C)CC2(CNC(=O)CCC)CC2)n1.C(N)(=O)N c1(C(=O)NCC2(O)CN(C(CC(C(=O)OC)C)=O)C2)cccc2scnc12 C1(OCC#C)CCCN(C(c2c(C)ccn2C)=O)CC1 c1(-c2cnc(CC)s2)nc(CCC2CCCN2C)nn1CCOC CC1(NC(=O)C(c2ccccc2)F)CCN(C(=O)CCN2CCCCCC2)CC1 C=CCCCCCN(C)C(C1CC=CCC1NC(C1C=CCC1)=O)=O C1(NC(C(N2CCC(C)C2)=O)=O)C2CC1N(C(=O)CCOC1CCCC1)C2 N1(Cc2cn(CC(C)NC(c3cnc(C(=O)O)nc3)=O)nn2)CCOCC1=O c1(OCC)cccc(CC(=O)NC2CCC(NC(c3cccc(F)c3)=O)CC2)c1 Cc1cc(C(=O)NC2C3CC2N(C(=O)CCc2ncccn2)C3)cc(C)c1 c1(NCC(=O)NCCCc2cn(CCCCCCO)nn2)ccc(O)cc1 c1(COC)nc(C)ncc1NC(C1CCCN1C(=O)OC(C)(C)C)C=O Cc1ccc2cc(C(=O)NCC(C(C)C)NC(=O)C=Cc3ncc(C)[nH]3)[nH]c2c1 Cc1cccc(CSCC(=O)NC2C3CC2N(C(=O)CCC2OCCO2)C3)c1 CCC(CC(=O)N1CCC(C2CCCO2)C1)OC(=O)Nc1ccnn1C C(N=c1nc2c(ncn2C)c(NCC(F)CO)[nH]1)c1c(CC)nn(C)c1 N1(C(c2cc(C(C)C)on2)=O)CC2(CC2C(=O)NOCc2ccc(O)cc2)C1 CC1CN2CCN1C(C(=O)N(C)CC1(NC(=O)Cc3sc(O)nc3O)CC1)C2 C1(CC)CCOC1C(=O)N(C)CCOCCCNC(C1CCOCC1)=O N1(C(CSCC=C)=O)CC2CCC2(CCNC(=O)C=CBr)C1 c1(C2C(C(=O)NC3C(NC(c4cnc(C)s4)=O)COCC3)C2)c(F)cccc1F c1(C(=O)NCCC2(O)CN(C(C(C)OC)=O)C2)ccc(CO)c(Cl)c1 C(CC(C)C)(C(=O)NC1CN(C(=O)C2=CCCOC2)CCC1C)NC(C)=O CC1CN(C(c2ccon2)=O)CCC1C(=O)NCC1(O)CN(C)C1 C1(C(N2C(CNC(c3cccc(C)n3)=O)C=CC2)=O)CS(=O)(=O)CCO1 N1(C(C(=O)NCCOC)CCC2CC(F)(F)C2)CC(C(=O)OC)OCC1(C)C C1(NC(c2c(C)nsc2NC2CC2)=O)CCN(C(=O)CC)CC1C.C(N)=O.N C12(OC)CCCC(C(=O)NCCCCNC(c3cccc4occc34)=O)(CC1)C2 C=Cc1ccc(C(N2CCN(C(=O)C(O)CSC)CC2CC(=O)NC)=O)cc1 c1(C(N2CC(CCOC)N(C(=O)C3=CCSC3)CC2)=O)cnc2cccnc2c1 O=C(C1=CCSC1)NC(c1ccc(F)cc1)CNC(=O)CC1NC(=O)NC1=O c1(C=O)cc2sc(=O)n(C)c2s1.Cc1cc(CCC(=O)NCC2CC2)nn1C.N C(=O)(C1=C(C)CCOC1)NCCCN(C(C1(OC)CCC(C)C1)=O)C1CC1 C1(CNC(CC)=O)CCN(C(=O)Cc2cc(C)nc(C)c2)CC1C N1(c2n(CCC=C)c(C3(C)CCCO3)nn2)CCN2C(=O)C(=O)NCC2C1 c1(C=O)nc(C2CC2(F)F)cs1.c1(CC(=O)N(CCC)C)cc(C2CC2)no1 N1(C(Cc2nnc(C)o2)=O)CCN(C(=O)Cn2cc(C3CC3)nn2)CC1.C(C#N)S c1(C(=O)NCC(C(=O)NCc2ncc(C)o2)N(C)C)cn(C)ccc1=O c1(-n2c(C(C)OCCC=C)nc(C3CCCC3)n2)ccc(Cl)c(Br)c1 N1(C(C2CCCCCN2C(=O)CN2CCCCC2=O)=O)Cc2ccncc2C1 C1(NC(c2c(C)noc2C)=O)CC2CC(C1)N(C(=O)CC1=CCOCC1)C2 c1(CC)cnc(C(=O)NCC2CCN(C(c3cccc(C4CCC4)c3)=O)C2)cn1 c1(OC)ccc(CC(=O)NC2CC(CCNC(C3CC3C)=O)C2)cc1OC c1(NC(C(CCN(C)C)NC(c2cn(C)c(=O)cn2)=O)=O)ccc(N=[N+]=[N-])cc1 C1(CC#C)(C(=O)NCCC2CN(C(c3c[nH]ccc3=N)=O)CC2C)CCCCC1 N1(C(=O)Cc2ccc(Cl)s2)CC2CCN(C(C3CCCC3)=O)C(C2)C1 N1(c2nc(C)nc(COc3ccc(F)c(F)c3Br)c2)CCCC2(CCC(=O)NC2)C1 N1(C(c2ccc(F)c(Cl)c2)=O)CCc2c(C(N3CCC(O)C3)=O)cccc2C1 C1(NC(Cn2c(C)cc(C)n2)=O)CC2CC(C1)CN(C(C1CC1C)=O)C2 Cc1csc2ncc(C(N3CCN(C(=O)Cc4cccc(C(N)=O)c4)CC3)=O)n12 CC1(C)CN(C(=O)CCC2CC2(F)F)C(CNC(c2ncccc2F)=O)CO1 c1(C(=O)NCC(CCC)NC(C2C3CN(C)CC23)=O)cn2ccsc2n1 C(=O)(CC(O)CC(C)(C)C)NCCC1CN(C(c2c(C3CC3)ccc(C)c2)=O)C1 O=c1c2ccccc2ccn1CCCN1CCN(NC(=O)c2cscn2)CC1=O CC1=C(C(=O)NC2CN(C(C3COCC3(C)C)=O)C(C)(C)C2)CCO1 N1(C(C2(C#N)CC2)=O)CC(C2CCCCN(C(c3ccn4nnnc4c3)=O)C2)C1 C(C(CC(=O)NC1(CO)CCSC1)NC(=O)C1=CCCC1)OC N1(C(COc2cn(C)nc2)=O)CCN(C(=O)COCC2CC2)C2CCCCC12 c1(C(=O)NCC2CN(C(c3c(C)ccc(C)c3)=O)CC2O)cnc2scnc2c1 C1(N=[N+]=[N-])(C(=O)NCc2ccc(C)c(C)c2)CCN(C(=O)C=CC(F)F)C1 CN=c1ccc(C(N2CC=CC2CNC(c2cc(C)cc(Cl)c2)=O)=O)c[nH]1 N1(CCSC(C)C)CCCC1c1ccon1 c1(CN2C3C(C(=O)NC4CC(=C)C4)C(C3)C2)c(F)cc(C)cc1F C1(CC(N2CCC(OCC)CC2)=O)CN(C(=O)CCCF)CCC1C Cc1cc(I)c(C(N2CCC(CC(=O)NC3CSC3)C2)=O)cc1C Cn1nnc2c1CCC(C(=O)NCCNC(=O)COCC(c1ccccc1)F)C2 C(=O)(CC(CC)C(C)C)NC(CC#C)(C)C(=O)N(C1CCN(C(C)C)C1)C c1(C(=O)NC(CC)CNC(C2CCNC2=O)=O)ccc2c(c1)OC(C)(C)CC2=O C1(CNC(CCC=CCC=C)=O)CCC(C)CN1C(=O)Cc1cccnc1C N#Cc1ccccc1NC(C1CC1CNCc1nc(Cl)ccc1F)=O C(=O)(C(O)CCCC)NCCC(=O)NCC1N(C(CCCC=C)=O)CCCC1 C1(Cc2cn(C(CNC(C3C(CCC)C3)=O)C)nn2)(OC)CCCCC1 N1(C(CCc2ccc(C)cc2)=O)CC(CN(C)C(c2cocn2)=O)C2(CC2)C1 C(C)(C(=O)N1CC(C(N)=O)(CNC(=O)C(N)=O)C1)(c1cccs1)N(C)C n1(CC)c2ccccc2c2cc(C=CC(=O)NC(C3CCCC3)C3CCC3)ccc12 c1(C(N2C(CCOC)CCCC2)C(=O)NCCSC)ccc(S(C)(=O)=O)o1 c1(OC)ccc(I)c(C(N2CC3CC2C3C(=O)NCc2ncccn2)=O)c1 c1(C(=O)NCC(C)N(C(=O)Cc2ccno2)CC)cnc(C2CCC2)o1 c1(CC)ccc(C(N2CCC(C(F)C)CC2)=O)cc1.C(=O)C.C(=O)C1CC1.N c1(C(N(CCC)C2CC2)=O)ccc([N+](=O)[O-])c(O)c1.CCCC=O.C(N)=O.N C1(CC=O)CC(F)(F)C1.C1CCN(C(=O)Cn2cc(C3CC3)nn2)C1.CC.N N1(C(CCC(=O)NCCC)=O)CC2(CCN2C(c2[nH]ncc2C#N)=O)C1 C(=O)(C1=CCC(C)(C)CC1)N1CCC(C)C(CNC(c2ccc(Cl)cn2)=O)C1 Cc1nn2c(c1C(=O)NCC1(F)CCCN(C(=O)C(C)N(C)C)C1)CCCC2 C#CC1(C(=O)N(C2CC2C)C)CCN(C(C2CC3C(C2)C3(C)C)=O)CC1 c1(C(=O)NCCN(CC(F)F)CC)c[nH]c2c(C(F)(F)F)cccc2c1=O c1(C(N(CCOC)CCNC(=O)C2=NOC(C)C2)=O)n[nH]c2c1NCCC2 C1(C(N(CC(C)N(C(C=CC(C)C)=O)C)C)=O)CCc2nc(=N)[nH]cc2C1 CN1CCC(CC)CC1.C1(CC(=O)N)CCC1(C)C.C1(CC=O)CC2(CC2)C1 C(CC(C)CC)(C(=O)NCC(C)(C)OCCO)NC(C(CCC)=CCC)=O c1(COC)ncsc1C(=O)NCC(C)(C1CC1)NC(=O)C(C)N(C)C C1(O)(CN(C(c2ccc(Br)cc2F)C(=O)O)C)CCCNCC1 N1(CCCNC(C2CC(N(C)C(c3ccoc3)=O)C2)=O)CCCC1=O N1(C(CCc2scc(C)n2)=O)CCCCCC1CNC(=O)CN1CCC(C)C1 C1(C)(C(N(CC#C)CCOC)=O)CC(O)CN1C(=O)CCSCCCC CC1CN(C(c2cc3ccncc3[nH]2)=O)CC2(CCN(C(c3cncs3)=O)C2)O1 CC(C)(C)C(C#N)C(=O)NC1CC2CCC1(C(=O)N)C2.C1CC(C)(C)C12CC2 C(=O)(C1=CC2CC=CCC12)NCC1(OC)CN(C(=O)C)C1.C1CCCCC1.O N1(C(CC(C=C)CCC)=O)CCC(C2(NC(=O)C(N3CCNC3=O)C)CC2)CC1 CC1CC(C#N)(C(=O)NCC=CC)C1.c1(C=O)ccc(C2CCCO2)nn1.N C1(C(=O)NC2CCN(C(C3(F)CC3(Cl)Cl)=O)C2)CC2(C1)CC21CC1 c1(CNC(=O)NC(c2cccnc2)(C)C)ccc(C#N)cc1 CC1CN(C(=O)C#CC(=O)N(C)C)CC1CNC(=O)C(C)(C)CC1CC1 c1(C2(C(=O)Nc3ccc(C(C)C)nc3)CC2)cc(C(F)(F)F)ccc1Cl c1(-c2c(C(N3CCCC(CN(C)C)C3)=O)n[nH]c2)cccc(S(=O)(=O)N(C)C)c1 CC(C)(C)C(C(=O)NC1CC1NC(=O)CCOC1COC1)N1CCNC1=O c1(NC(C2CCN(C(c3cncc(OC)c3)=O)C2)=O)nc(Br)ccc1Cl C(CN=c1[nH]cc([N+](=O)[O-])c(=N)[nH]1)C1CCCN(C(C(CC)C(C)C)=O)C1 C1C2CC1CN(C(c1ccc(C)nc1C1CC1)=O)C2.C(=O)(CS)OC.CC=O C(=O)(C1CCCc2c[nH]nc21)NC(CCN(C(CC=CC=C)=O)C)c1cccs1 c1(SC)cc(=NC(=O)C2CCCN2C(=O)Cn2nc(C)nc2C)[nH]n1C CCCCC(O)C(C)C(=O)N1CC(N(C(=O)CCCCC(=O)OC)C)C1 c1(C(=O)NCCC2CSCCN2C(=O)CO)sccc1S(=O)(=O)N1CCOCC1 c1(C=O)ccc(I)nc1.CCC(=O)N(CC)C(C)C.N(CC)(CC)CC.S C1(N(C)C(C2(C)CC2)=O)CCCC1NC(C1(Cc2cnn[nH]2)CCCC1)=O Cc1ccc(C(N2CC(CC(C)(C)CNC(c3cn[nH]c3)=O)C2)=O)cc1Br C12(C(N3CCCC(OC(C)C)C3)=O)CCC(CN(C(=O)CC(C)C(F)(F)F)C1)C2 C(=O)(C1=CC2CCC1C2)N1CC(C)C(NC(=O)C2=COCCC2)C1 N1(C(c2ccc(C)[nH]2)=O)CCCC2CN(C(c3ccnc(CN(C)C)c3)=O)CCC12 C(C)(c1cccs1)=CC(=O)NCCCNC(C(F)=CC)=O C1(C(=O)NCC(C2CCCC2)NC(c2nc(C)[nH]n2)=O)Cc2ccccc2CO1 Cc1ccccc1C=CC(=O)NCC1(CO)CCN(C(C2(C)CC2)=O)CC1 C(CC1=CCN(C(C2CCCC2O)=O)CC1)NC(c1c(C)cnc(F)c1)=O CCC(CCC(=O)N1CCC(F)(C(N)=O)C1)NC(c1ccc(C(N)=O)[nH]1)=O C#CCC(C)(C(=O)NCC(C)CC(=O)OC)NC(=O)CCC1(C#N)CCC1 c1(CC(=O)N(CCC)C(C)C)c(C)cccc1Cl.C1(C)(OC)CN(CC=O)C1 c1(OC(C(=O)NCCC(=C)C)C(C)C)ccccc1C#N.C(=O)(C(C)CC#N)N C=CC(C)(CC)C(=O)N1CCCC(CCNC(c2cnc(OC)cc2C)=O)C1 c1(C(=O)NCC(CO)NC(C(c2cncnc2)C)=O)c(Cl)ccc(O)c1Cl C1(C(=O)NOCC(=O)N(C)C)(CC)C=CCN1C(=O)CN(C)C(C)=O c1(-n2cc(CN(C)Cc3nccs3)nn2)ccccc1Br C=CCC(Cc1ccccc1)NS(=O)(=O)CC1CNC1 c1(C(=O)NCC2(NC(C3C(C)C3)=O)CCC2)c[nH]c(=NCC(F)(F)F)cn1 C1(NC(c2cncc(N(C)C)c2)=O)C2CCN(C(c3cn(C4CC4)nn3)=O)CC12 c1(C(C(=O)NCC2CCOC2)N(C)Cc2nnn(C)n2)ccc(F)c(Cl)c1 CC(C)C(CCNC(=O)C=C1CCC(C)C1)NC(=O)CCF C=CCN=C(NCCCC(=O)OC(C)(C)C)N1CCCC(C)(F)C1 C1(O)(CNC(c2cnc(C)[nH]2)=O)CCCN(C(c2cc(N)nc(Cl)c2)=O)C1 c1(C=O)c(O)nnc2c1CCC2.N1(C(C2(CC=C)CC2)=O)CC2CC(C)C2C1.N Cc1cc(CNC(=O)C=CCNC(C2CCCSC2C)=O)cc(F)c1 C(CS(=O)(=O)c1cn[nH]c1)NC(C1(CN)CCCC1)=O Cc1ccc(Cl)c(NC(=O)C(=O)N(CCC(F)(F)F)C(C)C)c1 Cc1cc(CNC(=O)C(O)C2CN(C(=O)CC3CC=CCC3)C2)co1 Cc1cnc(C(=O)NCC2(NC(c3ccccc3CO)=O)CCCC2)cc1C#N CC(CN=C(NCC1(C(F)(F)F)CCOCC1)NC1CCCC1)c1ccncc1 N1(CCNC(N(C2(C#N)CCOCC2)C)=O)CC23COCC2(COC3)C1 C1(CN(C(=O)CCC)C)CCN(C(=O)COC2(CC#C)CC2)C1.CC.O c1(N(C)C)nc(C(N2CC3CC2CN3C(c2csc(Cl)n2)=O)=O)cc(O)n1 N(C1COc2cccc(Cl)c21)C(c1c(N)[nH]c(=O)c(Cl)n1)=O C(=O)(CCCS(N)(=O)=O)NC(CN(C(C=Cc1occ(C)n1)=O)C)(C)C c1(OC)ccc(Br)cc1C=CC(=O)NC1CC(C)C1.C1(C=O)CC1(C)C.N C1(C(N2C3CCC2CSC3)=O)CCCCC12OCCO2 C1(CC(N2CC(C)(CCC(=O)NC3CC(OC)C3)C2)=O)CCCC2CC12 c1(C(N(C)C)=O)cc(F)ccc1.N1(C(C=CCN(C)CC)=O)CCC(O)C1 Cc1nc(C(=O)NCCC2CCN(C(C34CCCC3CCC4)=O)C2)c(C)n1C C1(CC=C)(NC(c2csc(=NCC)[nH]2)=O)CCCN(C(c2sccc2C)=O)C1 CC(F)(F)CCCC(=O)NC(C)(C)Cn1cccn1.C1(CC(=O)N)CC1(C)C c1(C(N2C(CN(C)C(C3CC3F)=O)CCC2)=O)ccc2c(c1)CCC2 c1(CC(=O)NC2CC(O)(Cn3cc(C4(C)CCCC4)nn3)C2)c(O)ncnc1O CCC(C)CCCC(=O)N1CCC(CNC(c2cc(C(N)=O)ccc2F)=O)C1 Cc1ccc(I)c(C(N2CCC3(CC3C(=O)Nc3ccc(Br)nc3)C2)=O)c1 C(=O)(CCCC(C)(C)C)NC(C(=O)NC(CCOCC)C)CCC1CC1 Nc1ccc(F)c(F)c1C(N1CCOCCC1c1ccc(F)cc1)=O N1(C(CN(C2CC2)CC)=O)CC2CCC(C1)N2C(=O)C=C1CCOCC1.C CC(C)CC(CC(=O)N1CCCC(N=[N+]=[N-])C1)NC(=O)C(C)(C)C1CCCO1 C1(C(=O)NC(CC)C(=O)NCC(c2cnn(C)c2)C)CC2(CCO1)CC2 C#CC1CN(C(=O)CCC2CCC(NC(=O)C(C)(C)C(F)(F)F)C2)CCN1C CCC1=C(C(=O)N(CCNC(=O)Cc2cnccn2)CC)SCCO1 C1(C(=O)NC(C(F)(F)F)C2CC2)(NC(c2n(CC)ncc2)=O)CCOCC1 N1(C(C(c2cnn(C)c2)C)=O)CC2CC(NC(=O)CN(CC(C)(C)C)C)C1C2 c1(C(=O)NCCC2(O)CN(C(C(CC(N)=O)O)=O)C2)nccc2n[nH]cc12 c1(C(N2C(C)(C)C(NC(c3ccccc3Br)=O)CC2)=O)cnc2[nH]ncc2c1 c1(CN2CC(C(N)=O)OCC2)cc(OCC2CCCC2)cc(F)c1 Cc1ccc(C(=O)NCCC2CC(NC(C3CCCN3C=O)=O)C2)cc1C N1(C(C(=O)N)=O)CC2CN(C(C3CCS(=O)(=O)N3)=O)CC2(C)C1.C(C)OC C12(CNC(c3n(C)ncc3)=O)CC(CN1C(c1c[nH]nn1)=O)C2.C1CCCO1 c1(N2CC(C)C(NC(C3CC3C3CCCCC3)=O)CC2)nccc(S(C)(=O)=O)n1 C#CC1(C(=O)N(CC(C)COC)C)CN(C(c2ccoc2Cl)=O)C1 C1(c2c[nH]nn2)(NC(c2cc(COC)sc2)=O)CCCCC1.c1(C=O)cccs1 C1(CC)CCCN(C(c2n[nH]c(C(C)(C)C)n2)=O)C1.C1(CC(=O)N)CCCCO1 CC(C)CC(F)(F)C(=O)N1CCN(C(=O)CC2CCOC2)C(C2CCCC2)C1 C(CC(C)C(=O)NC1(C(=O)NCC2(C#N)CCC2)CC(CO)C1)OC C1(CC(=O)NC(C)CNC(C2(c3nccs3)CC2)=O)CCCCC1 CC1CCCC(C(=O)Nc2cccc(NC(=O)CCNC(N)=O)c2)O1 c1(C(=O)NCC(C)NC(C2(C(C)C)COC2)=O)c(Cl)ccc(Br)c1F CCC(CC)(CCNC(=O)CCN1CCOCC1)NC(=O)C(O)CC1CCCC1 C1(NC(c2cn(CCOCC)nc2)=O)CN(C(C2CN(C)C2)=O)CCC1F C1(NC(C23OCC(CC)(C2)C3)=O)COC2(CCN(C(=O)CCCCCF)C2)C1 c1(C(=O)NC2CC2)conc1C(F)(F)F.C(=O)C(C1CC1)C1CC1.N c1(C(=O)NCC2C(C)CN(C(=O)CC3CCSCC3)CC2)ccc(Cl)c(F)c1F C(=O)C(C)(C)CS(C)(=O)=O.N1(C(CC)=O)CCOCC1CC.C(C)OCC C1(C(N(C(CCC)C)C)=O)CCN(C(c2ccc(CO)cc2)=O)C(C)(C)C1 c1(COC)cc(C(=O)N(C2CN(C(c3c(Br)cnn3C)=O)C2)C)c(C)o1 C1(F)(CNC(=O)CC2C=CCCC2)CCN(C(=O)C=Cc2cocn2)C1 c1(C(=O)NCC2CC2c2ccco2)n[nH]c2c1CN(C(c1cncnc1)=O)C2 N1(C(C(=O)c2ccco2)=O)CC2CCC1C(NC(C1CCCCC1)=O)C2 c1(C(=O)OCC)cc(Br)c(C(N2CCCC2C2CCOC2)C(=O)N)o1.C(C)C Cc1cccc2c1CCOC2C(=O)NCc1cccc(NC(C2CC(C)C2)=O)c1 C=CC1CN(C(c2cn(C)c(=O)cn2)=O)CC1NC(c1[nH]nnc1COC)=O Cc1c(C(=O)NC2(C)CN(C(c3cnc(C4CCOC4)s3)=O)C2)cccc1Cl c1ccc(Cl)cc1Cl.CC1(C(N2CC3CC3(CNC(=O)C)C2)=O)CC=CCO1.O CCC(C)CCC(O)CC(=O)N1CCC2(CC1)CC2NC(=O)COCCN(C)C C=CCCCC(C)(C)C(=O)N1CCN(C(=O)CC2COCCN2C)CC(O)C1 C1(C(=O)NC2CC(NC(C(C)Cc3ccco3)=O)C2)CCC(=O)N1C1CC1 C1(CNC(CNC(C)=O)=O)CC(C)CCN1C(=O)C(C)c1ccsc1 C(CCN=c1[nH]c(N2CCC(P(C)(C)=O)C2)nc2cccnc12)OC(C)(C)C c1(CC(=O)N)ccc(Cl)nc1.c1(C(C)C(=O)NC(C)C2CCC2)cncc(F)c1 Cc1ccc(C(N2C3CCC2(CNC(=O)C2=CCC(C)CC2)CC3)=O)c(N)c1Cl C1(CCNC(C(C)OCCC(C)C)=O)CCCN(C(c2ccn(CCF)n2)=O)C1 c1(OC)cc(OC)c(CNC(=O)C(N2CCC(C#N)(SC)CC2)=O)c(Br)c1 c1(N2CCCC(C)(NC(C3C(=C)CC3)=O)C2)ccc([N+](=O)[O-])cc1Cl c1(C(N(C(CNC(CC(C(=O)OCC)(C)C)=O)C)C)=O)cnc2ccccc2n1 c1(C(=O)NCC2(NC(c3c(C)oc(CO)c3)=O)CC2)cc([N+](=O)[O-])n[nH]1 N1(C(C(CCCC)C)=O)CC2CN(C(c3cc(Cl)n(C)n3)=O)CC2(C(F)(F)F)C1 c1(NC(CCSCC)C)cc(Br)ccc1S(=O)(=O)N1C2CCC1COC2 Cc1nccc(CCC(N2CC=CC(NC(=O)C(C)(C)c3cc[nH]n3)C2)=O)n1 C1(C)(C(=O)OC)CC(N=c2ccnc(C3CCC3)[nH]2)CCO1 C(=O)(C(C)C(C)(C)C)NCC1(C)N(C(C(C=C=C)C)=O)CCC1 N1(C(C(C(C)C)C)=O)CCC(C(N2CCC(CO)C(C)C2)=O)C12CC2 C(=O)(CC1c2ccccc2Oc2ccccc21)NCc1[nH]nc(C(=O)OCC)n1 c1(C(N2CCC(CCNC(C(CC)O)=O)C2)=O)cnc2cc(OC)ccc2c1 C=CC1CCN(C(C2(OC)CCN(C(c3cncc(O)c3)=O)C2)=O)C1 N1(C(CC(=O)NCC)=O)CC(NC(c2cnn(C)c2Cl)=O)C2(CC2)C1 C(c1cocn1)=CC(=O)NC(CN(C(=O)CCc1cc(C)[nH]n1)CC)C C(CC(C(C)(C)C)NC(c1cc(C)sn1)=O)N(C(C(CC)(F)F)=O)C C12(C(N3CCC(CN(CCCC(C)(C)C)C)C3)=O)CCCCC1OCC2 Cc1cc2ncc(C(=O)NCC3(NC(c4ccc5ccnn5c4)=O)CC3)cn2n1 c1(CCC(N2C(CNC(C3C(C)OCCO3)=O)CC(F)C2)=O)ccc(F)c(F)c1 c1(N2CCCC(CNC(c3cncc(OC)c3)=O)CC2)ccn2c(Br)cnc2n1 N1(C(CCCC)=O)CCN(C(=O)CC2CCOCC2(C)C)CC1CC(F)(F)F C1(NC(C(C)=CC=C)=O)CC=C(C(=O)NCC2(Cl)CC2(F)F)C1 Cc1cc(C(N2CCOCC(NCc3ccc[nH]3)C2)=O)cc([N+](=O)[O-])c1 C(=O)(CC1=CCCC1)NC(c1cn(C)nc1)C(=O)N1CC=CC1 c1(C(=O)NC2C3CN(C(c4ccc(=N)[nH]c4)=O)C2C3)cccc2c1C(=O)NC2 C1(C(=O)NC(CC)CN(C)C(c2nc(OC)ccc2Cl)=O)CNC(=O)CC1(C)C c1(C(N2CCOC(c3cn(CC4CC5CC5C4)nn3)C2)=O)cc2ccsc2[nH]1 c1(C(=O)NCC(CNC(C(C)CS(C)(=O)=O)=O)F)cnn2cc[nH]c(=O)c12 C1(NC(C2(C)CCC2)=O)CCC(NC(=O)CC(c2ccccc2)C2CC2)CC1 C(=O)(C(C)CCCC(C)C)NCc1cccc(NC(CC2CC(N(C)C)C2)=O)c1 C1(NC(CCc2cc(OC)no2)=O)CC(O)CN(C(=O)CC2(OC)CCCC2)C1 C(=O)(CCCC(F)(F)F)NC1CC(NC(c2cc(N)cc(O)n2)=O)C1 N1(C(C(C)(C2CC2)OC)=O)CCCCC(NC(=O)CCSc2ccccc2Cl)C1 CN1CCC(C#N)(C(=O)N(C)CCO)CC1.C1(CC(=O)N(CC)C)C=CCC1 CC1CCN(C(=O)C(Cc2ccoc2)NC(C23CC2CNC3=O)=O)CC1O c1ccc(C2CC2)cc1.C1(C=O)CCC(=O)O1.C1(C(N)=O)(C(=O)N)CC1.C c1(NC(N2CCCCC2C2(O)CC2)=O)ccnc(OCc2ccccc2)c1 CC1=C(C)CC(C(=O)NCCCC(C)NC(=O)C(C)NS(C)(=O)=O)CC1 N1(C(C=C(C)C2CC2)=O)CCC2(C1)CN(C(=O)Cc1c[nH]nc1C)CCO2 C(=O)(C1=CC2(CCOCC2)C1)N1CC(O)(CC)C1.CC1CCC(C(=O)N)C(=O)N1 N1(C(CCC)=O)CCC2CN(C(c3ccc(F)cc3C(F)(F)F)=O)CC2C1 N1(C(Cc2n[nH]c(=NC)s2)=O)CC2CC(NC(C3(C)CC(F)(F)C3)=O)CC1C2 c1(N2CCCC(NC(C(CC)C)=O)(CO)C2)ccc([N+](=O)[O-])c(C)n1 C1(C(=O)NC2CCN(C(C3N(CC)CCOC3)=O)C2)CCCCCC(=O)C1 S(=O)(=O)(c1c[nH]c(C(=O)NCC(C)(CO)NC(=O)CC)c1)NC.C(C)C C(C)(C(=O)NC1CCC(NC(=O)CCP(C)(C)=O)CC1)(C(C)C)OC C1(C(N2CCOCC(NC(c3cc(N)c(Cl)cc3)=O)C2)=O)CCOC2(CCC2)C1 N1(C(c2ccc(C(C)(C)C)s2)=O)CCCCC1C(=O)Nc1ccccc1C1CC1 CC1(CCNC(=O)COCC2CC2)CCN(C(c2ccc(Cl)cc2)=O)C1 C1(NC(CCc2nnc(C)n2C)=O)CC2(CCN(C(=O)CN3CCC(C)C3)C2)C1 N1(C(CC(=O)OC)=O)CCCCC1CCC(=O)NCC1CC1(Cl)Cl N1(CCN(CCC(=O)NCC(C)C(=O)O)CC)CCCC(OC)C1 N1(C(C(C)=CC)=O)CCCN(CCNC(C2CC3(CCOC3)C2)=O)CC1 C1(CC(N2CC(CC)(CC)C2)=O)CC2(CC2)CN1C(C1COCOC1)=O Cc1ccc(CNC(C2CCCC2C)=O)cc1C.C(=O)(CC(C)CN(C)C)N N1(C(CCSCC)=O)CC(NC(=O)CCc2nccn2CC)C(SC)C1 N1(C(C2C(C)(C(C)C)C2)=O)CCC(C2(NC(=O)CC3=CCCCC3)CCC2)CC1 C12(NC(CN3CCN(CC)CC3)=O)CCN(C(=O)CCc3cncs3)CC1C2 C1(N(C(c2cc(C)ns2)=O)CC)CCN(C(C2(F)CCOC2)=O)CC1 c1(C(N(C)CC2CN(C(C3CC3F)=O)CCO2)=O)ccc2c(cnn2C)c1 N1(CC=C)CCCN(c2cc(NC(c3ncc[nH]3)C)ncn2)CC1 CCCCC(C(=O)N(C(C)CSC)C)NC(=O)C(C#N)CCC Cc1noc(C)c1C=CC(=O)NC(C1CN(C(=O)C=CC(C)C)C1)C C1(NC(CCc2cncc(C)c2)=O)CCN(C(C2CCOC2)=O)C(C)C1 C1(C(=O)NCC23CC(CN)(OC2)C3)CC(c2cccc(F)c2)=NO1 C=C1Cn2c(C(=O)NCC3CN(C(=O)CC(C)(O)CO)CC34CC4)nnc2S1 C12(CC(=O)NCC3N(C(CCCc4ccc(C)s4)=O)CC3)CCCCC1C2(F)F C1(NC(c2ccns2)=O)CC2CC(NC(c3c(O)cccc3Cl)=O)C1C2 CCCCC(CC)C(=O)N1CCC(NC(=O)CN(CC(C)(C)C)C)C1(C)C CC1C(NC2(C)CCC(C)(C)C2)CCCN1C(=O)OC(C)(C)C c1(C(N2CC(CC=C)(NC(C3CC3C(=O)OC)=O)C2)=O)cnc2n1CCS2 Cc1cccc(C(=O)NC(C2CCCN2C(=O)CSC(C)C)C)c1C N(C(=NCC1CC1(Cl)Cl)NC1CCCC1)CC1(OC)CCOC1 C(C(COC)CC(=O)N1CCCC(C(=O)NCC(=O)N(C)O)CC1)OC CN1CCN(C)CC(NC(C23CC2CCN3C(c2ncccc2O)=O)=O)C1 Cc1cnc(N2CC(CNC(c3nc(C)sc3C)=O)CC2C)nc1O Cc1cnn(C)c1C(N1CC(C)(CCC(=O)N(C)CCOCC2CC2)C1)=O c1(C(N(C2CCN(C)C2)CC)=O)ncoc1C.C(=O)C(C)=C1CCCC1.N C1(NC(C(CCF)NC(c2ccc(OC)o2)=O)=O)CCCCCC1CO C1(CS(=O)(=O)NC2(CCOC)CCC2)CCOC(C)C1 Cc1cc(=O)n(C)cc1C(=O)NCCN(C(=O)C(CCCO)c1ccccc1)C c1(C(N2CCC(NC(c3ccc(OC)cc3)=O)CC2)=O)ccc2ncn(C)c2c1 C1(C(=O)NC(CC2CC2)C2CC2)CCC2(CC2)N1C(C1CC12CCC2)=O Cc1ccc(N)cc1C(N1CCC(CO)C(NC(c2ccc(Cl)s2)=O)C1)=O C(=O)(CC(O)CCCC)NCC(CC=C)NC(c1cnc(O)n1C)=O C1(NC(C(CC2CC2)NC(c2cnc(O)o2)=O)=O)CCC2(CC1)CC2 c1(CNC(c2c(N)nccn2)=O)nnc2n1CCN(C(=O)CC1CCCC1O)C2 C(=O)(CC(CC)C(F)F)N1CC(CCC)C(C(=O)NC(c2cnccn2)C)C1 N1(C(C(C)OC)=O)Cc2occ(C(=O)NCC3(O)CC(C)(C)C3)c2C1 CCCCCCC(F)C(=O)NC1CCC(CCNC(c2sc(CO)nc2C)=O)C1 c1(NCCCOCCNC(C2(COC)CCC2)=O)cncc(C#N)n1 C1CCN(C(=O)C(CC2(C)CC2)c2ccccc2)CC(O)C1.C(C(=O)N)OCC C1(N(C(C2C(CC)C2)=O)CCO)CCC1.C(=O)C(C1CCC1)C1CCC1 c1(OCC(c2cc(C)c(F)cc2F)=O)cc([N+](=O)[O-])c(C)cc1C C1(c2nnnn2C)(NCc2cc(SCC)no2)CCCN(C(C)(C)C)C1 c1(CCC(N2C(CNC(C(CC)OC)=O)CC2)=O)c(C)n[nH]c1C Cc1nn(C(F)F)c(C)c1CC(=O)NCC(CNC(=O)CC1CC1)CO O=C(C1=CCCNCC1)NC1CCCCCCC1F Cc1cncc(CC(=O)N(C)CC2CC(F)CN2C(=O)C(C)CSC(F)(F)F)c1 C1(C(=O)NCC(CCC)(C)O)CCCCCCN1C(=O)CCC(C)(C)N(C)C C1(Cc2cn(C)nc2)CCCN1N1Cc2cnc(C(F)(F)F)nc2C1 C1(N(C(CCn2c(C)ncc2)=O)C)CN(C(C2(N3CCOCC3)CC2)=O)CC1O Cc1cc(C)cc(C=CC(=O)NCC(C)N(C)C(c2cccc3nn[nH]c23)=O)c1 c1(C(=O)N)cccn2nncc12.CC12CCC(CC(=O)NCCC3CC3)(CO1)C2 c1(OC)ccc(C(=O)CCC(=O)NC2CCC2NC(=O)CC)cc1.C(=O)CO C1(CNC(C2(C)CCCCC2)=O)CN(C(=O)C(C)(C)F)CCC12CCOC2 N1(C(c2ccc(=N)[nH]c2)=O)CCCC(O)(CNC(C2CCCN2C=O)=O)CC1 N1(C2C(OC)CN(CC)C2)C2CCC1CC(CO)C2C=O.C(C)(C)C.C(=O)N N1(C(=O)OC(C)(C)C)CC2CCC(Nc3ccc(OC4CC4)cc3F)C2C1 C12(Cn3cc(COC(C)C)nn3)CCCCC1CN(C(c1ccc(=O)oc1)=O)C2 C1(NC(c2nc(Br)c[nH]2)=O)CN(C(=O)C(Cl)=CCl)C2(CCCOC2)C1 C1(C(=O)NCC2CN(C(C(CC)SC)=O)C2)(N(C)C)CCCCC1 c1(C(=O)NCCOCCCNC(CC2N(C)CCCC2)=O)c(F)ccc(F)c1Cl C(C(C)CC(=O)NC1CC(C)(NC(c2cc(C3CCCC3)[nH]n2)=O)C1)OC c1(NC(=O)C(=O)NC23CCC(CC2)OC3)cc(N2CCNCC2)cc(Br)c1 N1(C(c2c(C)nc(CO)s2)=O)CCC(C)C(C)C1.n1(CC=O)cnc(C#N)n1.N CCCC(C(=O)NCc1nnn(C)c1C(=O)N)C(C)C.C12CCC(CC1)C2.C N1(C(=O)CC(F)(F)Cl)CCC2CCC(C1)N2C(c1csc(C(F)F)c1)=O CC1COC(C(=O)N(C)CCOCCN(C)C(c2ccc(CO)s2)=O)C1 C12CCCC1CCN2C(C1CC(=C2CC2)C1)=O.Cc1cnc(C=CC(=O)N)[nH]1 C1(CNC(C2CCCN(C(=O)OC)C2)=O)CCOCC1(C)C.C1(C=O)CCC1 c1(OC)cc(C(=O)O)c2cc(-c3ccc(S(=O)(=O)C(F)F)cc3)[nH]c2c1 c1(C(=O)NC2CN(C(=O)Cc3cc(Br)cc(Br)c3)CC2F)cc(Cl)cnc1O c1(CNC(C(CCC#C)O)=O)ccc2c(c1)CN(C(C1(CC(C)C)CC1)=O)C2 C(C1CCOC1)=CC(N1CCC1CNC(C1(c2ccc(Br)s2)CC1)=O)=O Cc1cc(=NC(C)C2CC(N(C)C)C2)[nH]c(=NCCCC2CCCCO2)[nH]1 c1(C(=O)NC2(C)CCN(C(Cc3n(C(C)C)ncc3)=O)C2)ncc(Cl)cc1Cl C1(C(=O)N)C2CCC1(c1ccc(F)cc1)C2.C1CCC1.C1(C=O)CC1(Cl)Cl.C c1(NC(C(CSCC)NC(C2CCC2C#N)=O)=O)ccc2cncn2c1 C(=O)(C1CCCc2c[nH]nc21)N1CCC(N(C(c2c(C)noc2)=O)C)CC1 Cc1cc2ncc(C(=O)NCC3CN(C(c4ccc(Cl)c(C#N)c4)=O)C3)cn2n1 C1CN(C(c2ccc(C(F)F)nc2)=O)CCC12CCC2.C1(COC)CC1C=O.N N1(C(C2C(CC)N(C(=O)Cn3ncccc3=O)CC2)=O)Cc2cccc(O)c2C1 Cc1c(O)nc2ccccc2c1C(N1CCC2(CC(NC(=O)CNC=O)C2)C1)=O CCC(C)C(C)C(=O)NC(C12CCC(CC1)C2)C.c1(C(=O)N)cc(C)c(C)o1 C1(OC)CCn2cc(C(=O)NC3CCC3)nc2C1.C(=O)C1=CC2C=CC(C1)C2.N c1(C(N(C2CCN(C(COC(C)C)=O)C2)CCO)=O)cc(C#N)on1 c1(C(C)NCC2(OC)CCC23CCC3)ccc2c(c1)NC(=O)CO2 C(=O)(C1=NOC2COCC12)N1CC=C(C(=O)NC(c2ccnn2C)C)C1 CC1CNCCC(NC(c2ccccc2)CN2CCCCC2)C1 CCC(C(c1nnnn1CC(F)F)NCCNC(=O)C(C)C)C(C)C n1(CC)nnc(C(=O)NCCC2(C(=O)N(CC(Cl)Cl)C)CCCC2)c1C C1CCN(C)CC1.C(C)(CC(C)NC(=O)C)NC(C(C)OCCN(C)C)=O N1(C(=O)CCCN2CCOCC2)CC2CC(C1)CN(C(=O)CC1C=CCC1)C2 c1(C(N2CC(O)CC2C(C)C)C(=O)NCCCC)ccc(OC)c(C)c1C N1(C(COCC#C)=O)CC(NC(c2ccc(OC)c(Cl)n2)=O)CCC1C c1(C(=O)NC(C(C)NC(CCC2CC(OC)C2)=O)(C)C)ccc2n[nH]cc2c1 C1(CC)(CC)C(OC)CC1OC(C1COCC1C(N)=O)=O c1(CC(=O)NCC(C2CCCC2)O)cnn(-c2ccccc2)n1 Cc1nc(C)c(CNC(=O)CC2CC(C)OC2C)o1 c1(CCC(=O)N(CC(C)(C)NC(C2CN(C(C)=O)C2)=O)C)cc(C)nn1C C1(N(C(CC(C)n2cccn2)=O)C)CCC(NC(c2cnc(Cl)[nH]2)=O)CC1 C1(C(=O)NC(CN(C(c2c(CCC)[nH]cc2)=O)C)CC)CC(=O)CCO1 O=C1CCC(C(=O)NCC2(O)CC(C(=O)NCC3CCC3CO)C2)N1 C1(OC)CCCC(C(=O)NCC2(O)CN(C(c3cncnc3)=O)C2)C1 Cc1cc(C)c(C#N)c(NCC(C)NC(=O)CCS)n1.c1nnnn1C.C(N)=O C(=O)(CC(CC(C)C)NC(=O)CSCCC(C)C)NCC(COCC)C C=CCCCCC(c1nnnn1C(C)(C)CC)NC(C)CCOc1ccccc1 CC1CCCCC1CC(=O)N(C1CN(C(=O)Cc2nc(C3CC3)nn2C)C1)C Cc1cc(CNC(=O)CC2C3CN(C(=O)CC4CCCSC4)CC23)c(C)s1 C(=O)(C(CC(F)F)NC(=O)C=CC(F)F)Nc1c(C)nsc1 CN1CCN(C(=O)CCc2ccnc(O)c2)CC1CNC(=O)C(=O)N.C1CC1 N1(C(CC2(C)CCC2)=O)CC2CCC(C1)C(NC(=O)Cc1ccoc1)C2 C(CC(=O)NCCN(CCCF)C)(C(F)(F)F)NC(C1(C=C)CCCC1)=O CC1=C(C(=O)N2CC(NC(C3(c4ccc(C5CC5)nc4)CCC3)=O)C2)SCCO1 C(c1cncc(OCc2nc(C3CCCCC3)cs2)c1)=CC(N1CCCC1)=O C1(C(=O)NCCc2ccnc(O)c2)CCN(C(=O)CN2CC3CC3C2)C12CC2 c1(C(=O)NCC2CCCCN2C(=O)CC2CC2)c[nH]c2c(Cl)cccc2c1=O N1(C(CC2CC(NC(CNC(=O)OC)=O)C2(C)C)=O)CC2CC2C2CC12 CCC(C)CC(=O)NC1CCC1CNC(=O)C(F)=CCCF c1(C(=O)NC(CC(C)NC(c2c(CC)nc(C)[nH]2)=O)C)cccc2cncn12 Cn1nnc(=NC2CCC(NC(=O)C(C)(F)C(C)(C)F)CC2)[nH]1 CCC1=C(C(=O)N2CCCC(N(C(=O)Cc3noc(C)c3C#N)C)C2)SCCO1 C(C)(CCCCCC)NC(C(=O)OC)CC(C)C CC1(C)CC=C(C(C)(C)CNC(C2(C(=O)O)CC2)=O)CC1 C1(C(C)(C)C)CC(C)CN(C(=O)CC2CCCCC2)C1.c1(C(=O)N)ccc(F)o1 C1(C(N2C(CCNC(C(C)=C3CCCC3)=O)CCC2)=O)CC2CCC2C1 N1(C(Cc2c(Cl)ccc(OC)c2)=O)CC(C)CN(C(c2c[nH]nc2C)=O)C(C)C1 C1(NC(NNC(=O)Nc2ccc(C)cc2Cl)=O)CCS(=O)(=O)C(C)C1 CC(C)C(=O)C(=O)N1CCCC1C(N1CCC(NCc2ccc(F)cc2)CC1)=O N1(C(CC2(C#N)CC2)=O)CCC2(C1)CN(C(c1ccnc(CO)c1)=O)CCO2 Cc1ccc(S(C)(=O)=NC(=O)CNC(=O)C(C)NC(=O)CC(F)(F)F)cc1 c1(NC(C2C(CNC(c3cc(O)ncn3)=O)CCC2)=O)ccc2n[nH]cc2c1 C1(NC(N2CCC(C(O)CO)C2)=O)CCN(CC(F)(F)F)CC1.c1ccccc1F CC(N=c1ccn2ncc(S(=O)(=O)N3CCCC4(C3)OCCO4)c2[nH]1)C1CC1 c1(OCC)ccc(C(=O)NCC(C)(C)NC(C2CCC(CC)C2)=O)s1 C(=O)(C#CC1CCCCO1)N1CCCN(C(CCC(=O)OC)=O)CC1C(C)C Cc1nc2ccccc2c(C)c1C(N1CCC2CCN(C(=O)C(N)=O)CC2C1)=O C(C)(C(C)(C)C(=O)NCC1CC(F)(F)CO1)NC(Cc1nc(C)sc1)=O CC1C(NC(c2c(F)cccc2F)=O)C(C)CCN1C(=O)Cc1c[nH]ccc1=O c1(CNC(CC2CC(=C)C2)=O)ccc(C(N2CCCCC2C(=O)NC)=O)nc1 CCC(O)C(C)(C)C(=O)NCCC1(O)CN(C(c2ncc([N+](=O)[O-])n2C)=O)C1 CCCC(C)CC(=O)N1CCCC(C)(NC(=O)C(F)(F)c2nccn2C)C1 c1(CNC(C2CCC2n2ccnc2)=O)cncc(C)c1.C1(C(=O)N)CC1 c1(C(=O)NC2C3(CC(NC(c4c(C)sc(Cl)n4)=O)C3)C2)ccc2ncncc2c1 N1(CC(CCCCC)C)CCC2(CC1)CC(N1CCC(CO)C(F)(F)C1)C2 c1(C(=O)N)cc2ccccc2nc1O.CC1(C)C(C(=O)NCCC2CC2)C1(F)F Cc1ccc(N2CCCC(NC(=O)NCCCCN3CCCCCC3)C2)cc1 c1(C(=O)NC2CC(CNC(=O)C#CC3CCCO3)C2)ccc2ccccc2n1 C1(C#N)(CC(=O)OC(C)(C)C)CCN(C(=O)OCC2CCC(=O)N2)CC1 c1(CN2C(C(=O)Nc3ccnc(C4CC4)c3)CC(O)C2)c[nH]c2c(F)cccc12 Cc1ccc2c(c1)CCN2C(c1ncc(C)s1)C(=O)NCC1CCCO1 CC1=C(C)CC(C(=O)NCCC2CCC2)CC1.c1(CC=O)cccc(O)c1F.N CC(O)C(C=O)NC.C(=O)(C(C)(C)F)N1CCC1.C(=O)CC.C(=O)C=CCl C12(COC)CC(C(N3CCC(CC)CC3)=O)(CO1)C2.c1(C=O)cncc(N)c1 c1(C(=O)NC(c2ccccn2)C(F)F)cc2c(F)cccc2s1 O=C(C1CCCn2ccnc21)NCC1CCC2(CN(C(c3n[nH]cc3Br)=O)C2)O1 C12(C=O)CCC(C)(C1)C(=O)N2.C1(C)(C(=O)OC)CCCN1.c1ccccc1.O O=S1(=O)CC2(c3ccc(F)cc3)CN(CC(c3ccc(Cl)cc3)O)CC12 N1(C(C2(CC=C)CCOCC2)=O)CCN(C(=O)CNC(=O)OC)C(CO)C1 CCC(C)(O)C(=O)N1CCCC(CNC(=O)CCNS(C)(=O)=O)C1 c1(C=O)ccco1.N1(C(C)C)CC(C(=O)NCCC2CC2)C1.C1CCCC1.N Cc1cccc2nc(C(N3CCN(C(c4cn(C)nc4Cl)=O)C4(CC4)C3)=O)cn12 Cc1c(N2CCC(CC#N)C2)ncnc1N1CCC(CCO)CC1 Cc1ccc(S(=O)(=O)NC(C(=O)NCc2ncccc2C)C(C)C)cc1C C(=O)(CC(C)C(F)(F)F)N1CC(C#C)(C(=O)NCc2cnc(C)n2CC)C1 c1(NCC(Br)=C(C)C)[nH]c(=NCCCCCCCCO)nc2scnc12 C(C(=O)N(C)CCNC(c1cnn2c1OCC2)=O)(C(C)(C)C)NC(C)=O Cc1cc(C(=O)N(C)CC2CN(C(C3CCCN(C)C3)=O)C2)nc(O)n1 c1(CC)nc(C)oc1C(=O)N(CC(C)(C)C(=O)NC1CCCCCC1)C C1(NC(C2CC(CNC(c3cn(CC)nc3)=O)C2)=O)CCC(C)NC1=O c1(-n2cc(CNC(C3N(C(C)=O)CC(O)C3)=O)nn2)ccc(Cl)cc1F N1(C(CN2CCC(C)CC2)=O)CCC2(NC(=O)CC(F)(F)F)CC2C1 c1(NC(N2CC(C(C)C)OCCC2)=O)cc2ccccc2c(Cl)n1 C(=O)(C(CC)(CC)CCO)NCc1c(CNC(C(COC)C)=O)nccc1 c1(C(=O)NC(CCOC)CNC(C2(F)CCC2)=O)n[nH]c2cc(C)ccc12 N1(C(C=CC=CC)=O)CCC(C2CCN(C(C3(C)CCNC(=O)C3)=O)CC2)C1 C1(N(C(=O)C2=COCCO2)C)CCN(C(=O)CC2CC2(Cl)Cl)CC12CC2 CC(C)C(C(=O)N1CCCC1)NS(=O)(=O)C1CC1.c1(C=O)ccc(Cl)cc1.C C1(C(=O)NCCN(C(C=CC(CC)C)=O)CCO)CCC(N(C)C)CC1 N1(C(c2cc(C(C)C)[nH]n2)=O)CCCC(C)(CNC(=O)C=O)C1.CC(F)F.N C1(C(CNC(CCc2cc(C)[nH]n2)=O)O)CCN(C(=O)CC2CCCCC2)CC1 [N-]=[N+]=NC1CCC2(C(=O)NC3CC(C)C3)CC12.c1(C(=O)N)cnn2cnnc2c1 C12(C(N(CCC#C)CC)=O)CC1CCN2C(c1ccc(C#N)[nH]1)=O c1(OC)cnc(Cl)nc1N1C2CCC1C(CNC(=O)C=CCN(C)C)C2 O=C(N=c1c(Br)c[nH]c2ccccc12)NC(c1ccccc1)C1CCOC1 C(C(O)CNC(=O)CC1(NC=O)CCC1)N(C(C)=O)C.C(C)(C)C.O C(CCCCC(=O)N1CC(=C)C1)NC(C1CC(O)(CC#C)C1)=O C1(NC(c2cc(C(C)=O)on2)=O)CN(C(=O)C(C2CC(F)(F)C2)O)CC1(C)C C(=O)(CC(O)CNC(c1ccns1)=O)NCC(CC)O CC12CN(C(c3cc[nH]c3)=O)C(C(=O)N(C3CC3)CC3CCOC3)(C1)C2 N1(C(C2(SC)CC2)=O)CCCC(C(=O)NCC2CCC(F)(F)C2)C1 CC1CNc2c(C(=O)NCCCNC(c3cncc(C4CC4)c3)=O)cnn2C1 C(CCC(=O)N(C)C)(C(=O)OCC)N1CC(CCC)OCC1 N1(C(c2c(C)n[nH]c2C)=O)CCN(C(=O)CC2CCCC(C)(C)C2)CC(C)(F)C1 Cc1cc(C(N2CCC(O)C(NC(=O)CCc3ncccn3)C2)=O)c(C)nc1C C1(NCC(C(=O)OC)Cc2ccccc2F)CCc2nc(C(F)(F)F)nn2C1 CC(F)(F)CCCC(=O)NCC1CCN1C(C1(CCO)CC1)=O C#CCCC(C(=O)NC1COC(C(C)C)C1)NC(C1CC2CCC2C1)=O c1(C(N2CCC3(CCCN3C(C3CCO3)=O)C2)=O)nc2ccccc2cc1Br C1(C(N2C(C(C(N3CC(O)(CC=O)C3)=O)(C)C)CCC2)=O)CC(=O)CCO1 c1(CC(=O)NC(c2ccc(C)cc2)CNC(C=C(C)C)=O)cccc(N)c1 Cc1cc(C(N2CCN(C(c3csc(O)n3)=O)CC2C(F)F)=O)c(C)n1C C(=O)(C(C(C)CC)NC(=O)C(c1ccnn1C)C)NC(C=C)C1CCC1 C1(CNC(C(C)(C)C2CCCCN2)=O)(CF)CCCOC1 c1(C(=O)NC(CC2CCCC2)C(=O)NC2(CCF)CC2)cccc(Cl)c1 C(=O)(C1=Cc2cc(F)ccc2OC1)N1C(CNC(c2c(C)snc2)=O)CCCC1 C1(CC(=O)N(C)CCNC(=O)C(=O)NCC2CC2)CC(C)(C)C1 C1(C(=O)NCCCC=CC)CCCC1CNC(=O)Cc1coc(C)n1 C1(OCC(=O)NC(C#C)(C)C2CCC2)CCCCO1 C1CN(C(=O)C=C2CC2)CC(C(F)(F)F)O1.N1(CC(=O)N)CCCCCC1.C N1(C(C(CC(=C)C)C)=O)CCCC(C2(NC(c3ccc(OCC)cc3)=O)CC2)C1 C1(CNC(=O)CCC2CC2)COCC1NC(=O)COCCF C=CCCC(O)CNC(C1CCC(C(C)C)N1C(=O)CN(C)CCC)=O c1(SCC)ccc(Cl)cc1C(=O)NC(C)C(C)NC(=O)CCn1ccnc1 N1(C(CC=C)=O)CCC(NC(=O)C(CC)OCC)C1(C)C CC1(CCC(=O)N)CCC(=O)N1.C1(C=O)C2CC3C(C2)C13.c1cn(CC)nn1 c1ccc2cc(OC3CCCN(Cc4ncc(C5CC5)o4)C3)ccc2c1 c1(CC(=O)N(C2CCN(C(=O)C(F)C(F)(F)F)CC2)CC)cc(F)ccc1F C1(C(C)C)CN(C(=O)CNC(=O)C(C)(C)C)CCN1C(=O)CCc1cnc[nH]1 C(C(Cl)C(C)(F)F)NC(CC1(CNC(c2c(C(C)C)noc2)=O)CC1)=O c1(C(N2CC(NC(c3cc(SC)c(C)o3)=O)C3C2C3)=O)cccc2nn[nH]c12 c1(N2C3CN(C(C4(F)C(C)OCC4)=O)CC2CCC3)nc(Cl)nc2ccccc12 S(=O)(=O)(c1ccc(F)c(F)c1F)Nc1c(C#N)ncc(C)c1 c1(C(=O)NCC(C#C)OC)ccc(CC(F)(F)F)cc1F N1(C(CCSC)=O)CCN(C(C2CCC(=O)C2)=O)C(CC(C)(C)C)C1 C(C(C(=O)NC(C)CC1CN(C(c2cnn(CC(F)F)c2)=O)C1)OC)OC c1(N2CCC(C)(CSC)CC2)cc(C)[nH]c(=NCc2cn(C)nc2C(F)F)n1 C(=O)(CCC(C)c1ccccc1)N(CC(CNC(c1cn(CC=C)nn1)=O)C)C C1(N(C(CCC)CC)Cc2sc(C)nc2C)CCC(=O)N(Cc2ccccc2)C1 C(=O)(C(C)C(C)C(C)(C)C)N1CCC2(CN(C(Cc3ccc(C)o3)=O)C2)C1 Cn1cc(Cl)cc1C(=O)NCC(C(C)(C)C)NC(C1C=CCC1)=O CC(C)CC(CNC(c1sccc1-c1ccccc1)=O)NC(C1CC12CCC2)=O N1(C(=O)C=C2CCC2)CCC2CN(C(C3(Cl)CC3(F)F)=O)CC12 Cc1nc(C(N2CC3CC2C3NC(c2cccs2)=O)=O)c(C)s1 C(=O)(C(C)N=[N+]=[N-])N1CC(C(C(=O)NCC(=O)NCC)OC)C1 Cc1cccc(Br)c1C(C(=O)NCc1cn[nH]c1)NC(c1cscn1)=O c1(SC)cc(C)[nH]c(=NCC2CN(C(=O)C(F)(F)CO)CC23CCC3)n1 CCC(C)(C)C.C1(CC(C=O)NC(C(OCC)OCC)=O)CCCNC1=O c1(CC(NCCN(C(C2C(C)CC2)=O)C)=O)ccc(Cl)nc1.C1CCC1 c1(C(=O)NCCCC(C)C)cc(O)cc(C#N)c1.c1(C=O)ncc(C(F)F)s1.N C1(C(=O)NC(C)CC2CCN(C(C3CC(C)(C)C3)=O)CC2)C(C)OC(C)C1C Cc1cc(C(=O)NCC2(NC(C3CC3C)=O)COC2)cc(C)c1O Cc1c([N+](=O)[O-])ccc(Br)c1C(=O)NC1CC(C(=O)Nc2ccccn2)C1 C=CCN=C(NCC(c1ccc(F)c(F)c1)O)NCC1CNC(=O)O1 N1(C(C2(C)N(C(C(C(C)(F)F)F)=O)CC(O)C2)=O)CCC12CCCCC2 C12(NC(C3CC(C)C3)=O)CCOC(C)(C1)C2.c1(C=O)cnn(C(C)C)c1.N C#CCCC(O)C(=O)NCCCN1CCN(C(c2ncc(N)cc2C)=O)CC1 C1(NC(COC(C)C)=O)CC12CCN(C(=O)CC1(C)CC1(Cl)Cl)CC2 N1(C(c2ccnc(C)c2C)=O)CC2CCCC1(CNC(c1ccncc1F)=O)C2 Cn1cc(C(=O)NC2COCCC2)c(O)nc1=O.C1(CC(=O)N)CC2(CC2)CO1 c1(SCC)cnc(O)c(C(N2CC3CC3C2)=O)c1.c1(C=O)cnc(C(C)C)s1 N1(C(CC(C)(C)N(C(=O)CC2CCC=CCC2)C)=O)CC2CC1CS2=O CCCC(C)(C)CC(=O)NC1CC(NC(=O)Cc2cc(F)cc(Br)c2)C1 C1(C(=O)NC(CC)(C)CCNC(C2C(C)(C)C2(C)C)=O)CC2CCC(C1)C2 C=CC(C)(O)C(=O)N1CCCC(C(=O)NCC(=O)NCC(C)C)C1 c1(C(=O)NC2CCN(C(=O)C(O)c3ccsc3)C2)ncc(F)cn1 C1(F)(C=O)CCS(=O)(=O)C1.C(C)(c1ccco1)=CC(=O)NCCC.CC C=C(C)CN=C(NCc1cn(-c2ccc(OC)cc2)nn1)NCC1(OC)CCOC1 C1CC2(C1)CC2C=O.C1CN(C(=O)C(C2CC2)C2CC2)C1.CC(C)C.O C(CCCC(=O)N1CCSCC1CCNC(=O)C(N1CCCC(C)C1)=O)OC C1(C(C(=O)NCc2cc(C)no2)C)CCCN(C(C2COCOC2)=O)C1 N1(C(CC2CCC(C)CC2)=O)CCC(CCNC(c2cncn2C)=O)C(F)(F)C1 S(=O)(=O)(c1ccc(C)cc1)Nc1cccc(-c2onc(C3(COC)CCC3)n2)c1 Cc1ccc(S(C)(=O)=O)cc1C(=O)NC1CCCC1NC(C1CCCS1)=O N1(C(c2ccc(Cl)s2)=O)CCC(NC(C23CCCC2C3)=O)CC1 c1(OC)cc(C(=O)NC2CC(O)CN(C(=O)C)C2)cc2cnn(C)c12.C(C)=O c1(C(=O)OC)cn(CCNC(c2n[nH]cc2-c2ccccc2)=O)nn1 N1(C(c2c(C)n(C)nc2)=O)CCN(C(=O)C(C)N(C)C)C(CC(F)(F)F)C1 Clc1cnc(CNCn2cc(I)cn2)c(Br)c1 c1(C(N(CCCNC(C(CC)(CC)CO)=O)C2CC2)=O)coc2c1C(=O)NCC2 O=C(C1=COCC1)NCC1CCN1C(=O)COCc1ccccc1Cl c1(COCC(C)C)ccc(C(=O)NC2CC2)cc1.C(=O)C.C1CC1.C c1(C(=O)NCCCNC(C(C)C(F)F)=O)cnc2[nH]c(C(F)(F)F)nc2c1 Cc1ccc([N+](=O)[O-])c(OCCC(=O)NC2CC(NC(c3cscn3)=O)C2)c1 Cc1nc(CNC(C2CCOC2C)=O)oc1C(=O)NCC1CC(F)(C)C1 c1(NC(=O)C(=O)C2CC2)ccc2c(c1)CN(Cc1ccc(O)cc1Cl)C2 CC(C)C(C(=O)N1CCN(C(=O)CO)CC1)C(C)NC(c1ccc(F)cc1)=O C(C(F)(C(=O)Nc1ccc2ccoc2c1)C(C)C)NC(C=C(C)C1CC1)=O c1(C(N(C)CC2CCN(C(C3OCC3(C)C)=O)C2)=O)c2c(nn1C)CCSC2 c1(C(=O)NCC23CCC2CCN3C(=O)CCN2CCCC2)ccccc1[N+](=O)[O-] Cc1occ(-c2ccccc2)c1C(=O)NCCN(C)C(c1ccncc1Cl)=O S(=O)(=O)(c1ccc2c(c1)CCO2)N1CC(C(=O)NCc2ccc(C)nc2)OCC1 Nc1c(C(=O)NC2CC(O)CN(C(c3cccc(Cl)c3F)=O)C2)cc(F)cc1Cl Cc1ccncc1C1CC1C(N1CC(N(C(=O)CC(C)c2ccccc2)C)C1)=O Cc1cc(N(C)C)nc(CNCc2ncc(-c3cccs3)o2)n1 Cc1nn(C)c(C)c1CC(=O)N(CCNC(C1CCC2CC2CC1)=O)C1CC1 Cc1cc(CN2CCCC2C(=O)NC)cc(C)c1.c1ccc(N(C)C(C)C)nc1 CP(C)(=O)CN1CCCC(C(=O)N(C2CCS(=O)(=O)C2)Cc2ccccc2)C1 C1(C(C(=O)NCCOCCNC(C23CCC(C2)C3)=O)O)CCCCCC1 C(=O)(N=c1ccn(C2CCC2)[nH]1)C1C(NC(C2(C)CCC(=O)NC2)=O)CCC1 C1(NC(COC(CC)C)=O)CN(C(=O)CSCCNCC)CC1(C)C.C O(NC(=O)C(CCF)NC(C1C2CCCOC12)=O)CCN(C)C c1(OC)cnc(C(=O)NCC2CCN2C(=O)Cc2csc(Cl)n2)cn1 C1(C#N)(C(=O)NCc2cn(C3CCN(C(C(C)C)=O)CC3)nn2)CCOCC1 CCCCC(O)C(=O)N1CCCCC1C1(NC(C2CCC(=O)N2)=O)CC1 C1(O)(C(C)NC(C2CCC3CCC23)=O)CCN(C(c2ccc(O)nn2)=O)CC1 N1(C(C(C(CC)C)O)=O)CCC2(C1)CN(C(C1CC(S(C)(=O)=O)C1)=O)C2 C1(F)(C(=O)NCC(CNC(C2C(COC)CC2)=O)F)CC=CC1 c1(C(N2CCC(NC(CC(=O)NCC)=O)C(C)C2)=O)cc(OC)c(N)cc1F c1(C(CO)NC(=O)Cc2coc(-c3ccc(Cl)cc3)n2)cccc(C(F)(F)F)c1 C1(C(N(c2snc(C)n2)C)=O)CC(F)(F)CN1C(c1ccc(Cl)cc1)=O c1(C=O)ccc(O)c([N+](=O)[O-])c1.C(C(C)(C)CC(=O)NC1(C)CCOC1)OC C(=O)(C(C)C(C)(F)F)NCC(C)N(C(c1cccc(C(C)C)n1)=O)C C1(C(=O)N(CC(C)(C)C#N)C)(OC)CCN(C(=O)CO)C1.CCCN(C)C CC(C)C(C(=O)N1CCC(C2CCCCN2C(=O)Cn2cnnn2)C1)N(C)C C1(NC(c2ccc(NC)cn2)=O)C(C)CN(C(=O)Cc2csc(C)c2)CC1C CCC(CNC(=O)C(C)=CC(C)(C)C)(CC)NC(c1ccsc1SC)=O c1(NC(C(c2ccco2)NC(COCCC)=O)=O)cncnc1O c1(C(c2n(C(CC)C)nnn2)Nc2cnc(SC)nc2)cc2ccccc2o1 CCCC(C(O)C(=O)N1CCSC(CC)C1)NC(=O)C=CC1CCCN1C c1(C(C)=O)cccc(C(=O)N)c1.C1C2CN(C(=O)CC3CCC34CCC4)CC12.C Cc1ccncc1C=CC(N1CCCCC(N(C)C(C2CC=CC2)=O)C1)=O C1(NC(C2N(C(C)=O)CCCC2)=O)CC2(CCN(C(=O)C(O)C3CCCC3)C2)C1 C(C)(CCCCNC(C1CC1)=O)NC(c1c(C)nns1)=O.C(C)C.C(N)=O C(=O)(CC(F)(F)C(F)(F)F)N1CCC2C(C1)C2.C(=O)(C(C)(C)C)NC(C)C=O c1(C(=O)N)cn(C)cn1.C(CNC(C1(C)CCC1)=O)(CC1CC1)OC C12(C=O)CC(CN1C(=O)C=CC(=O)N(C)C)C2.C1(OC)CCCC1C C1(C(N2CCC(CC(=O)NCCN(OC)C)C2)=O)CCC(C)NC1 C1(NC(CC(CC)NC(c2ncccc2F)=O)=O)CCCN(C)C1=O C1(CNC(C(C#C)(C)C)=O)CN(C)CCN1C(=O)CCC(=O)c1cccs1 c1(C(=O)NC(CC)CNC(=O)C(C)C2CCC2)conc1C(F)(F)F C1(NC(c2ccc(CCF)cc2)=O)(CO)CCN(C(c2cccc[n+]2[O-])=O)CC1 c1(OC)ccc2cnc(C(=O)N(CCCNC(C3CCCC(F)C3)=O)C)cc2c1 N1(C(COCP(C)(C)=O)=O)CCCC2(CCCN2C(c2cn3ccsc3n2)=O)C1 n1(CC)ccc(CC(=O)NCC23CC(NC(c4nnsc4C)=O)(C2)C3)n1 C(=O)(CS(=O)(=O)CCO)NCc1nc(CNC(C(C(C)C)C)=O)sc1 N1(C(C=C(COC)C)=O)CCN(C(C2CC2C(C)(F)F)=O)CC12CCC2 C1(CNC(c2c(C)coc2)=O)CC2CC1CN2C(c1cccnn1)=O N1(C(CC(C)C2CC2)=O)CCN(C(c2cc(Cl)cs2)=O)C(C2CCC2)C1 C=CCC(CNC(c1c[nH]nc1C)=O)CC(C)C.C1(C)(C=O)CC(C)=NO1.N C12(NC(c3cn(CCC)nn3)=O)CCCC1N(C(c1ccnc(OC)c1)=O)CC2 c1(C(=O)NC(CNC(C(CC#C)C)=O)C2CCC2)cc2c(OC)cc(Cl)cc2[nH]1 C12(C(N3C(C)(C)CC(CO)C3)=O)CCC(CN(C(=O)CC3=CCCC3)C1)C2 C(=O)(CCC(=O)c1ccc(Cl)s1)N(CCNC(=O)Cc1cn(C)nn1)CC N1(C(c2nccc(C(N)=O)c2)=O)CCN(C(C2CC(=C3CCC3)C2)=O)C2CC12 C1(SCC)CCC(C(N2CC3CC3(CNC(=O)CCC3CC3C)C2)=O)CC1 CC(C)CCN=c1nc(N2CC(CC(F)(F)F)OC(C)C2)c2sccc2[nH]1 C1(C(=O)NCC(c2ccccc2)C)CC12CC(NC(=O)C(C1CCOCC1)C)C2 C1(C(=O)NCC(CC)NC(=O)Cc2cc(C)no2)CC2CCC2C1 c1(C(=O)NCC(CNC(C2C(CC)C2)=O)O)cc(C)c(O)nn1 CC(C)(C(=O)N(CC(F)(F)C(F)F)CC1CCCOC1(C)C)C(N)=O CON1CC(C(=O)NC2CCCC2C(=O)N(C2CCCC2)C)CC1=O N1(C(COC)=O)CCN(C(C2(c3cc(C)no3)CC2)=O)C(Cc2ccncc2)C1 C1(C(=O)NCC(CC)N(C)C)CCCCCN1C(c1cccc(=O)n1C)=O C1(C(N2CCC(C)C2)=O)(OC)CC(C)(C)C1.C(=O)C(C)Cc1ccnn1C.C c1(C(=O)NCCc2cc(C(=O)OC)no2)nccn2c(Br)ccc12 N1(C(C(C)S)=O)CCC(N2CCc3n[nH]cc3C2)C(C)CC1 CCCCC(C)C(=O)NCC12CC(CNC(=O)CC(C)n3cccn3)(CO1)C2 Cc1ccc(C2CCCC2NC(C2CC2C)C)cc1 c1(CN2CC(Oc3cn(C)nc3)C2)cc(Br)cc([N+](=O)[O-])c1O c1(CCC)cc(C(N2CCC(C(F)CNC(=O)C(=O)N(C)C)CC2)=O)sc1C N1(C(c2nc3cccnc3s2)=O)CC2CC(N=c3[nH]nco3)C2C1 C1(NC(=O)C=Cc2ccccc2Br)CC2CC(C1)N(C(=O)C(F)F)C2 c1(C(C)(C)C)nsc(N)c1C(N1CCC(O)(C)C1)=O.C(=O)(CC)N.C1CC1 c1(C(=O)NCCC(C)NC(=O)C(C)c2cncs2)c2c(nn1C)CCC2 C1(C(=O)NC(CC)CC(=O)OC)CC2CCC1N2C(=O)C(C)(C)C(F)F n1(CC=O)cc([N+](=O)[O-])c(C)n1.N1(C(C=CCC)=O)CCC(COC)C1.N N(C1CCOc2c(C)cc(F)cc21)(C(=O)CCc1cscc1Br)C(C)=O C(=O)(N=S(C)(=O)c1cccc(C)c1)c1c(OC)cc(CO)cc1 C(=O)(C1=C(F)CN(C(C2(CO)CCCO2)=O)CC1)NCC(C(C)(C)F)(C)F O=C(C1=CCSC1)NCCN(C(c1nn[nH]c1C(F)(F)F)=O)C1CC1 CC1(C)CN(C(c2cccc3nccn23)=O)CC(C)(C)C1NC(=O)COC(F)F C(=O)(C1CCNc2ccccc21)NCC1CN(C(C2CCC(C)C2)=O)CC1C N1(C(=O)OC(C)(C)C)CC2CC1CCC2NC(=O)Nc1cccc(CF)c1 c1(C(N2CCOCC(NC(C(CCSC)O)=O)C2)=O)ccc([N+](=O)[O-])c(O)c1C C12(C(=O)NC3COCCN(C(C=C(COC)C)=O)C3)C3C4C1C1C2C3C41.C C(=O)(C(C)(CO)CO)NC1CC(C)CN1C(=O)CN(CCO)CCO C1(C(=O)NCC(CCNC(COCCC(C)C)=O)O)CC2C=CC1C21CC1 CCCCC(C)(F)C(=O)N1CCN(CC2CN(C(=O)Cn3cnnc3O)C2)CC1 c1(OCCC(N2CCC(N(C(C3C(C(C)C)CCC3)=O)C)C2)=O)cccc(F)c1 c1(CC(N2CCC(CCOC)(NC(=O)COC)C2)=O)cnn2c1OCCC2 c1cccc(F)c1C(N1CCCC1c1noc(C2CC2)n1)=O.O=C(CC1CC1)N C1(NC(=O)CC2C=CCC2)CC12CCN(C(c1ccns1)=O)C2 c1(CCC(=O)N(C)CC)ccc(O)c(F)c1.c1(C(=O)N)c[nH]nc1-c1cccs1 c1(C(=O)NCC(C)OC)ccc(F)cc1.c1(C=O)ncccc1C(C)=O.C c1(CC(=O)OC)ccnc(NC(=O)C(=O)NCc2cnn(C3CC3)n2)n1 c1(CC)cc(C(C(=O)NCCC2(C)CC2)N(C)Cc2cnco2)sc1C N1(C(c2cnc(OC)nc2)=O)CCCC12CN(C(c1ccc(C)o1)=O)C2 C1(NC(c2c(CNC(c3ccc(C)s3)=O)ccs2)=O)(CO)CC2CCCC12 Cc1ccc2c(N(C3CCN(C(C4CNC(=O)N4)=O)C3)C)ncnc2c1 N1(C(C(c2cn(CC)nc2)=O)=O)CC(NC(=O)Cn2cncn2)CC1C CC1CCCn2c(C(=O)NCC(C)(CO)NC(=O)C(C)(F)F)cnc21 N1(C(c2cccc(CC)c2)=O)CCC2CN(Cc3cncc(F)c3)CC12 c1(C(N(CC(O)C2CC2)C)=O)c[nH]nc1CNC(=O)C(C)(C)C1CCCO1 c1(CC(N2CCC(C(=O)NCC3(O)CCC3)C2)=O)ccc2c(c1)OCO2 C1(C(=O)NCCN(C(c2cn(CCOC)cn2)=O)CC)COCCC1C N1(C(=O)CCCNCCCCCCCCF)CCC=C(c2ccccc2)C1 c1(C(N2CC(c3n[nH]c4c3CCC4)C2)=O)cc2ccncc2o1 c1(SC)cnn(C)c1C(=O)NCC1(NC(c2cccc(F)c2)=O)CCOC1 CCC(C)(CNC(c1nnnn1C(C)C)(C1CCOCC1)C)OC n1(CC)cc(Cl)cc1C(N1CCN(C2CCN(C(c3cn[nH]c3)=O)C2)CC1)=O C=CC1(CC(=O)N(C)CCOCCNC(C2CCCOC2C)=O)CCOCC1 C1(CC)CN(C(c2cnn(C)c2OC)=O)CCN1C(=O)C(O)C1CCCC1 C1(C(=O)NCCN2CCN(C(C(CCOC)C)=O)CC2)CCC2(C1)CC2(F)F c1(C(C(=O)N(C2CC2(C)C)C)NC(c2n(CC)nnc2)=O)c(C)cccc1Br CC(CS(C)(=O)=O)C(=O)NCCC1CC(NC(c2cc(Cl)sc2Cl)=O)C1 N1(C(C2C(C)(C)C2)=O)CCC(CCC(=O)NCCN2CC3CCC2C3)CC1 N1(C(c2nc(N(C)C)oc2)=O)CCC(C(=O)NCc2ccc(Cl)cn2)C12CC2 C(=O)(C(O)C(C(C)C)OC)N(CC(=O)NCC(c1cnn(C)c1)O)CC C(c1ccccc1[N+](=O)[O-])=CC(=O)NCC1C(NC(C=CSC)=O)CCC1 c1(N2CCOCC(C(=O)NCCSc3ccc(F)cc3)C2)ncnc2[nH]cnc12 Cc1[nH]nc(C(=O)NC(C)CN(C)C(c2cncnc2)=O)c1N Cc1cc(O)cc(O)c1CN1CC(C)(CNC(=O)C(C)Cn2cccn2)C1 C=CC(C)C(=O)NCCCN(CCO)C(c1ncnn1CC)=O N(C1CCC(C(=O)N=c2ccn(C)[nH]2)c2ccccc21)C(c1c(C)ocn1)=O c1(C(=O)NC2CC(NC(=O)CCN3C(=O)C=CC3=O)C2)cc(Br)cc(Br)c1 c1(C2C(C(N3CC(CCCCNC(COC(CC)C)=O)C3)=O)C2)ccccc1C c1(Nc2n(C)nc(CC)c2Br)ccc2c(n1)OCCC2=O C1(CNC(=O)C(c2ccccc2Cl)O)C2CN(C(c3csc(O)n3)=O)CC12 N1(C(CC2CCN(C)CC2)=O)CC2CCN(C(=O)CC3CCOC(C)(C)C3)CC12 c1(C(=O)N)cc(C)nc(O)n1.N1(CCC)CCCC(C(=O)NC(CC)C(C)C)C1 C1(NC(c2c(C)con2)=O)CCN(C(=O)CN(C2CCCC2)C)CC1(C)C C=CCCC(=O)NCC(C1CC1)NC(C1CC12CC2)=O CC1CCNCCC1CN(CC(C=O)C)C(c1cc(F)ccc1Cl)=O.C(C)(C)C C(C(C(C)C(C)C)NC(=O)C(c1nc(F)ccc1Cl)C)NC(CCC=CC)=O C(=O)(CC1COc2cccc(Br)c21)Nc1c(CC)nn(C)c1 CCC(C(O)C(C)C)NC(=O)CN(CCOC)C(c1ocnc1C(C)C)=O N1(C(c2cc(C(N)=O)[nH]n2)=O)CC2CC1C2NC(C1CCC(CO)CC1)=O Cn1cc(C(F)F)c(CNCC2COC2)n1.c1(CC(=O)N)ccc(O)cc1 c1(C(=O)NCC2C(NC(CC(=C)Br)=O)C2)ccc(-c2ccccc2)n1C c1(-c2cnc(NC(c3cnccc3I)=O)c(C(F)(F)F)c2)ccc2ccoc2c1 C1(CCC=C)(C(N2CC3CC2C3)=O)CN(C(=O)CC(C)C2CC2)C1 C=C(Br)CCC(=O)NCC1CCN(C(c2n[nH]cc2C2CC2)=O)C1 C1(C(F)(F)F)(C(=O)O)CCN(S(=O)(=O)Cc2c(Br)cccc2Br)CC1 CC(CCCCNC(=O)C=Cc1ncc[nH]1)NC(C1(CF)CC(=O)C1)=O N1(C(C2C(C)(C)CN(C(c3ccc(C#N)s3)=O)C2)=O)CCCC(N=[N+]=[N-])CC1 c1(C(C)N(C)C(C2(N(C)C(C3CCOCC3)=O)CC2)=O)cnn(C)c1 C1(C(=O)NC(C(=O)NC(CC=C)(C)C)Cc2ccoc2)C=CC=CC=C1 c1(C(N(CCCNC(c2cc3sccc3[nH]2)=O)CC)=O)ccnc2c1CCC2 Cc1ccc(C=CC(=O)NC2CCCCC2)cn1.c1(C(=O)N)cnn(C2CC2)c1 CC1Cn2nccc2CN1C(C1C(NC(=O)CC(C2CC2)C2CC2)C1(C)C)=O N1(C(C(C=CC)O)=O)CC2CCN(C(c3cc4n(c3)CCC4)=O)CCC2C1 C1(C(=O)NCc2occ(C(=O)NC(C3CC3)C)n2)CC(=O)NC1(C)C c1(CC)cc(C(N2CC3CC3(C)C2)=O)ccc1Br.c1(C=O)ccc([N+](=O)[O-])o1.N C12CCC(CC1)N2C(c1ccnc(O)c1)=O.c1(C(=O)N)ccon1.C1CC1.C C12(C(=O)NC(c3nc(C)no3)CC)COCC1CN(CC(F)(F)C(F)F)C2 c1(CC(C(=O)Nc2nnc(C)s2)C)ccccc1OC(F)(F)F S(=O)(=O)(CCCCF)N1C(c2occ(C)n2)COCC1 C(=O)(C(C)Cc1ccco1)N(CCOCCCN(C(CCOC)=O)C)C C(=O)(CS(=O)(=O)C1CCCC1)N.N1(C(C(C)OCCC(C)C)=O)CC2CCC1C2 C=CCCCC(C)(C)CNC(=O)CCCN(C)C(c1coc(CO)c1)=O c1(C(=O)NCC(CN(C(C(C(C)C)n2cnnn2)=O)C)(C)C)ccc(F)c(N)c1 CCCCCC(CC)C(=O)NC1CCN(C(c2ccc3cc[nH]c3n2)=O)CC1F C=C(Cl)CCC(=O)NCCCCC1CCN(C(=O)C(c2cccs2)SC)CC1 N1(C(c2nn(CC)c(C)c2)=O)CCC=C(C(=O)NC(C(F)(F)F)C2CC2)C1 C(=O)(CS(=O)(=O)CCO)NC(CN(C(CCOCCC)=O)C)C CCC(CN(C)C)CC(=O)NC1CCN(C(c2cnc(OC)c(Cl)c2)=O)CC1F C1(C2CC2)(NC(c2c(OC)ccs2)=O)CCN(C(=O)CC2CCOC2)C1 N1(C(c2cnns2)=O)CC2(CC(C=O)C2)C1.C1CON(CC(F)(F)F)C1=O.CC c1(C(=O)NCC(C2CCOC2)NC(C=C(C)Cl)=O)ccnn1CC#N N1(C(c2cnc(C)[nH]2)=O)CC=CC(NC(C2(F)CCOCC2)=O)C1 N1(C(c2cc(CCCCC)[nH]n2)=O)CCOCC1CNC(c1sc(C)cc1C)=O C1(NC(C(=Cc2ccncc2)C)=O)COCCN(C(C2CC=CC2)=O)C1 C1(C#N)(C(=O)NCCc2cn(Cc3c(C)c[nH]n3)nn2)CCCC1 Cc1ncccc1C(=O)NC1CCCN(c2ccc(-c3ccccc3O)cn2)C1 N1(C(C2CC(C)(CC)C2)=O)CCC(CNC(c2ccc(C#N)o2)=O)CC1C Nc1cc(F)c(Cl)cc1C(N1CC(NC(C23CCCC2C3Br)=O)C1)=O c1(C(N(CCC#C)C(C)CC)=O)cnc(N(C)C)nc1 N1(C(C(CC)F)=O)CC(OCC)C(CNC(c2ccc(Br)o2)=O)C1 C(CC(C(C)C)NC(=O)C(C)n1cccn1)N(C(CC1CC(OC)C1)=O)C C1(NC(C2CC(C)(NC(C(C)N(C)C)=O)C2)=O)CCCCCC1F c1(OC(CC)C(=O)NC(C)CC(C)NC(C2CCCO2)=O)ccccc1F N1(C(CCC)=O)CCCC(C)C1.c1(C=O)ccccc1.C(=O)C=CCN(C)C.N C1(C)(C(N(C2CCCC2C#N)C)=O)CC(O)CN1C(=O)CN1CCOC1=O Cc1cc(C(=O)N(CC(C)O)CCNC(c2nc(O)c(C)s2)=O)cc(C)c1Cl Fc1ccccc1N1CCC(CNCc2cnc(C3CCCCC3)s2)C1 N1(C(c2n(C)nnc2)=O)CC2CCC(C1)N2C(=O)NC(c1ccccc1)=O C1(OCC)CCN(C(c2ccc(C(N)=O)[nH]2)=O)C1.C1(F)(C=O)CCOC1C.C Cc1cc(C(=O)NCC2CC(C)CO2)c(Cl)cc1F.C(=O)(C1=C(Cl)CCC1)N CCC(CC(C)C)C(=O)NCC1CC2CCC1N2C(=O)CC1C=CCC1 c1(C(C)NC(c2csc(-c3cccc(F)c3)n2)=O)ccc(Cl)c(F)c1 N1(CCC(=O)NCC#CCNC(C2CCN(C)C2)=O)C(=O)CCC1=O N1(C(CC2CCN(C(C3CCN(C)C3=O)=O)C2(C)C)=O)CCC12CCC(C)CC2 C=CC1(C(=O)NCC2(O)CCCC2(C)C)CCN(C(=O)CC=C(Cl)Cl)C1 c1(C(C(N2CC(CNC(C(C=C)O)=O)C2)=O)C)ccc(Cl)cc1 c1(CNC(CC2(NC(c3c(C)ncnc3)=O)CC2)=O)cccc(F)c1F C1(NC(c2occ(C)c2)=O)CCN(C(c2c[nH]c(=N)o2)=O)CC1F N1(C(CCC=C=C)=O)CC(NC(c2ncoc2C)=O)CC(F)(F)C1 C1(C(=O)NCC(C)(C)NC(C2CCC=CCCC2)=O)CCCC2(CCCCC2)C1 c1(OC)nn(C)cc1C(N1CCN(CCCNC(=O)CC2CC=CC2)CC1)=O Cn1ncnc1CCC(=O)NCC1CCN1C(=O)CC1CCC1 Cc1nn(C)c(C(F)(F)Cl)c1C(N1CCN(C(=O)C2=CCCC2)C(C)C1)=O N1(C(CCNC(=O)NC)=O)CC(C)CC1(C)C.c1(C=O)cnn(C(C)C)c1N c1(C(c2n(C(CC)C)nnn2)NCc2cscn2)sc(Cl)cc1Br N#Cc1ccc(C(N2CCCC2C2(CNC(=O)CC)CC2)=O)o1.CC(F)F.O CC1CCN(C(=O)CC=CCNC(=O)C(C)(C)C2(O)CCC2)CCS1 c1(CC(=O)NCCOCCCNC(c2ccns2)=O)ccccc1Cl C(CCCCC(=O)N(C)CC1C2CN(C(c3c(C)ncnc3C)=O)CC12)SC CCC(C)CCN=c1[nH]c(=NCc2cc(C)c(C)nn2)[nH]c2c1CSC2 c1(N(CCC)CC)ccc(C(=O)NC2CC2)cc1.C1(CC=O)COCC1O.N C1(COC)CCCN(C(=O)CC)C1.c1(C=O)ccoc1.C(=O)C=CC(C)C c1(C(C)C)oncc1C(=O)NCC1CC(CNC(=O)CC#N)C1 c1(C(N2CC(O)C2)=O)ccc(S(C)(=O)=O)[nH]1.Cc1cccc(C(=O)NC)c1C C(=O)(CCCS(C)(=O)=O)NCCCC(C)NC(C1(C2CCCCC2)CC1)=O c1(N2Cc3c(cccc3)C2)nc2c(c(=NC(CC3CC3)C3CC3)[nH]1)CCC2 C1(NC(C2CC(OC)C2)=O)CCC(CN(C)C(C2CC(C)OC2=O)=O)CC1 C1(COC)(NC(C2CCC(F)(F)C2)=O)CCN(C(C2CCC(C)C2)=O)CC1 C12(C(N(CC)C)=O)CC(CN1C(C1CC(F)C(=O)N1)=O)C2.CC(C)C=O C(=O)(CCCC(=O)NC1CN(C(c2cc(Cl)ccn2)=O)CCC1C)NC(C)C Cc1ccc(C)c(C(=O)NCCC(O)CNC(C2CC3CCC2O3)=O)c1C Cc1ncc(C)c(N2CCC(C)(CNC(=O)Cn3ncnn3)CC2)n1 CC1CCC(CNC(=O)COC2(C)CCOCC2)N(C(=O)C)C1.c1nc[nH]n1 c1(C(N2C(CCCNC(C=C(CCC)C)=O)CCC2)=O)cccc2c1OCCN2 C#Cc1cnc(NC2(CNC(C3CCCO3)=O)COC2)nc1 C1(CCC)CCCC1C(=O)N(CCCN(C)C(c1n[nH]c(C)n1)C)C c1(N(C(C23CC(n4cc(-c5cc(OC)ns5)nn4)C2C3)=O)C)ccc(Br)nc1Cl N1(C(CN(C(C(COC)O)=O)C)=O)CCN(C(=O)C=CC(C)C)CC1 C1(NC(CCC(C)(F)F)=O)CCN(C(c2cnn3c2CCC3)=O)C12CCC2 c1(C(=O)NC2C(C)CN(C(C)=O)CC2C)nc[nH]c2ncc(Br)c1-2 C1(C(N2CCC(CN(C)C(c3ccnc(O)c3)=O)C2)=O)Cc2ccc(F)cc2C1 c1(C(N(C2CCN(C(c3cccnn3)=O)C2)CC)=O)cc(C2CC2)n(C)n1.O C(=O)(C(C(C)(C)C)c1cc[nH]n1)NCC(CC(C)C)NC(c1cc(C)nnc1)=O C(C)(C)(CC(=O)N(CCCC(=O)NCc1n[nH]cc1C)C)OC CCCC(C)(O)C(=O)NCC1(CCC)CCCC1.C(=O)(C(C)(C)c1cccs1)N NS(=O)(=O)c1ccsc1C(=O)NCC1CC1.c1(C=O)ncnc2cc[nH]c12.N C(C1CC1)(C1CC1)=CC(N1CC(C(N2CC(OC(F)F)C2)=O)C(F)C1)=O N1(C(CC(=O)N(C)C)=O)CCN(C(=O)CCC(=O)c2ccncc2)C2CC12 C1(NC(C(N2CCN(c3cccc(F)c3)CC2C)CCC)=O)CC(C)CC(C)C1 C1(C(=O)NC(C(C)C)CNC(=O)CC2(C)CC(F)(F)C2)CCCCC1(F)F C1(CC(=O)NCC2(C(=O)NC(CC)CSC)CC=CC2)CCCC(=O)C1 C1(NC(COCC#C)=O)CN(C(C2(C)CC2(F)F)=O)CC12CCC2 C1(NC(=O)C(=Cc2c[nH]cn2)F)CCC2(CCN(C(C3C4CCCCC34)=O)C2)C1 N1(C(C2C(C)CC(=O)NC2)=O)CCn2c(C3CC3(C)C)nnc2C1 n1(C(C)C)ncc(C(=O)N(C2CCNCC2O)CCSc2ccccc2)c1N n1(CCC(C2CCC2)=O)nc(-c2nccs2)nc1-c1cccc(OC(F)(F)F)c1 N1(C(C(CCC)NC(N)=O)=O)CC(C)(C)OC2(C1)CN(C(C1CC1(C)C)=O)C2 N1(C(c2c(OC)nccn2)=O)CCN(C(c2ccc(I)cc2)=O)C2CC12 C1(OCCCNC(C(C)(C)OC)=O)CCN(C(C2(CC(C)C)CC2)=O)CC1 C#CCCC(O)CCNC(C1(CC=C)CCCN1C(=O)CCC(F)(F)F)=O C1(N(C(=O)CCC)CCOC)CCN(C(=O)CCc2ncc[nH]2)CC1 N1(C(c2nn[nH]c2-c2ccccc2)=O)CCCN(CCOCCO)CC1 Cc1c(C(=O)NCC(C)N(C(=O)Cn2[nH]cnc2=N)C)ncn1C N1(C(C2CCC(C)(C)O2)=O)CCCC(C)(NC(=O)C(=CC2CCCCC2)F)C1 C1(NC(C2CC(C)(C)C2)=O)CN(C(c2scnc2C(F)(F)F)=O)CCC12CCC2 N1(C(c2nc(C)oc2)=O)CCNCC1C(N1CCOCC1c1ccccc1)=O n1(CC(=O)N(CCCC)C)cc(CNCc2cccnc2)nn1 C1(C(N2CCC(CNC(=O)CC3CCOC3)C2)=O)CCC2(CCCCC2)CC1 C1(C2CC2)(C(N2CCCC(NC(c3cn(CCCC)nn3)=O)C2)=O)CC(=O)C1 N1(C(CC(CC)SC)=O)CCC2C(CCN2C(c2[nH]nc3c2COC3(C)C)=O)C1 c1(C(=O)NC(CN(C(C2CC(SC)C2)=O)CC)C)csc(C#N)c1 n1(CC(=O)N(C2CN(C(=O)CC3CNC(=O)O3)CC2O)C)ncc(O)nc1=O C(=O)(C#CC1(C)COC1)N(CC(C)N(C(=O)CCc1c(F)cccc1Cl)C)C C(=O)(C(CC1CC1)NC(=O)C(CO)N(C)C)NC1C(CCC)C1 c1(CC)ccnc(C(=O)N)c1.C1(CC(=O)N(CCC)CCO)CCC(C)(C)O1 c1(CC(N2CC3(CN(C(C4(C)C(C)OCC4)=O)C3)C2)=O)c[nH]c2cc(F)ccc12 c1(C(=O)NCC(C(C)C)C(=O)N2CC(c3ccncc3)C2)cccc2ccoc12 C1(C(=O)NC2C(C(=O)Nc3c(SC)cccn3)CCCC2)CCc2nc[nH]c2C1 C1(CC)(NC(C2CC=CC2)=O)CCN(C(=O)Cn2nc(O)ccc2=O)CC1 C1(C(N2CCC(NC(c3cn(C)c(O)n3)=O)CC2)=O)(CC)CCC(O)CC1 C=CC(CC)C(=O)N1CCC(C(N2C(C(=O)OC)CC2C)=O)(OC)C1 C1(OC)(CNC(c2ccncc2)=O)CN(C(=O)C(F)CC2CCOC2)C1 C1(NC(CCCC)C)CCC2CCC(C1)N2C N1(C(=O)CSCc2ccccn2)CCN(C(C2CC(O)C2)=O)C2CCCCC12 c1(-c2c(CN(C3CCCOC3)CC)cn(C)n2)c(F)cccc1F Cc1cc(NC(=O)CC2CCC(NC(=O)C=CC(F)(F)F)C2)cnc1Cl n1(CC(=O)NC(C)CN(C)C(C23CC(N=[N+]=[N-])C2C3)=O)cc2ccccc2n1 C1(NC(c2[nH]n(C)c(=O)n2)=O)CN(C(C2C=CC=CC=C2)=O)Cc2nccn2C1 C(C(=O)N=S1(=O)CCC(CN)C1)Nc1c(C)ccc(-c2cncc(F)c2)c1 C(=O)(CC1=CCOCC1)NC1CN(C(c2n(CC)ncc2Cl)=O)CC1CO C1(C(=O)NC(CC)(CC)CO)CC(C(C)=NO)C1(C)C c1(OC)ccc(-c2nnc(S)n2CC(=O)NCCC)cc1.C(=O)(C(O)C(F)F)N C1(CC(=O)N(CC(C)O)CCNC(c2nn[nH]c2)=O)CCC(=O)NC1 N1(C(c2c(C)noc2C)=O)CC2CCC(C2)C1.c1(CC=O)cnn(C(C)C)c1.N C(=O)C(C(C)(C)C)C1CCC1.c1(CC)[nH]ccc1C(N1CCC(OCC)C1)=O C(C)(C)(CCCN=c1[nH]c2cccc(Br)c2o1)NC(C1CN(C)CC(C)O1)=O c1(C(=O)Nc2cccc(-c3nnco3)c2)cnc2n1CCNC2 c1(C(=O)N)cc(Br)cc(S(N)(=O)=O)c1.c1(CC(=O)OC)ccc(C)c(F)c1 Nc1ncc(C(=O)N)cc1.N1(CC=CC(=O)N(CC)C2CC2)CCCCC1 C1(F)(C(=O)Nc2n(CC)ncc2)CCN(C(=O)C(c2cccn2C)=O)C1 C1(CNC(c2ccc(NC)cn2)=O)CC2CCC1N(C(=O)CC1CC=CCC1)C2 CC1(C(=O)NC23CC2CN(C(c2cc(Cl)c[nH]2)=O)C3)CC=CCO1 C1(CC(=O)NCC(CCCC)NC(C23CCC(C2)C3)=O)CCn2cncc2C1 N1(Cc2c(O)cc(C)c(Cl)c2)CC2(CN(C(c3scc(C)c3C)=O)CC2CO)C1 N1(Cc2scc(C)c2)CCN(CCCNC(=O)C(C)O)CC1 C1(C(C)NC(=O)CCC2(C)CC2)CCN(C(c2cc[nH]c2C2CCC2)=O)CC1 c1(C(C)C(=O)N(CCNC(C2CCC2)=O)C2CC2)ccccc1F.C1CC1.C C1(CCNC(=O)COC2CCOCC2)(NC(Cc2nc(C)oc2)=O)CCOCC1 N1(C(c2cc(C)n(C)c2)=O)CCC(F)(F)C(CNC(C2CC3CCCCC23)=O)C1 C1(NC(C(Cc2cn(C)nc2)O)=O)CC12CCC(NC(c1cccs1)=O)CC2 C1(CC(=O)N(C2CCN(C(=O)CCCc3ncco3)C2)C)COCC1O c1(C(N2CC(CC(C)NC(=O)CC(C)CF)C2)=O)cc(C(C)(C)C)ccn1 C1(C=O)C2C3CCC(C3)C12.N1(C(C(C)OCC(F)(F)F)=O)CC(F)CC1C N1(C(C(CCC)O)=O)CCCC(C2CC2NC(C2(C)CCC(C)C2)=O)C1 c1(C(=O)OC)coc2c1C(NC(C1(C)C=CCCN1)=O)CCC2 c1(N2CCCC(C)(OC)C2)nccc(=NCCN(C)C)[nH]1 CCC1=C(C(=O)NC(C)CN(C(=O)C(C(=O)OCC)OC)C)SCCO1 c1(NC(=O)NC2CC(CC(N)=O)C23CCC3)ncc2c(n1)CCCC2 O=NN1CCCC1C(=O)N.C1C2CN(C(C3CC3)=O)CC12.C(=O)N1CC1.C N1(C(=O)NCC2(OC)CCOC2)CCS(=O)(=O)CC1C1CC1 c1(C(=O)NCCCN(CCO)C(c2cnns2)=O)ccc(F)cn1 c1(C(N2CC(CC)C(C(N3CC(N(C)CCO)C3)=O)C2)=O)c(C)cccc1C Nc1c(C(=O)NCCNC(=O)Cc2cccnc2)cc(Cl)cc1Cl C(=O)(CC(C)C)NCC1N(CC)CC1.n1(C)cc(-c2cnn(CCF)c2)nn1 C(=O)(N=c1cc(C(N)=O)n(C)[nH]1)C1CCC(NC(C(CC)SC)=O)CC1 Cc1cccc(O)c1C(=O)NCC(CNC(c1ncc(F)cc1F)=O)C(F)(F)F c1(C(N2CC(OC)C(NC(c3cc(C)nc(O)c3)=O)C2)=O)nc(C)ccc1F C(=O)C1=CN(C)S(=O)(=O)N=C1C.c1(NCC)cccnc1C(=O)N(C)CC C1(CS(C)(=O)=O)(CNC(=O)NCC2C(C)OCC2)CC(F)(F)C1 C(C)(CO)(C(=O)NCC#CC(=O)Nc1ccc(OC)nc1)OC CC(C)CCCC(C)C(=O)NC1CC1CNC(=O)C1=CCCC1C c1(SCC(=O)NCC(C)NC(=O)C(F)(F)C2CC2)ccc(C#N)cc1 c1(CNC(C(=O)N(C)CC2(C)CCCO2)=O)cccnc1C(F)(F)F Nc1cncc(C(=O)NCCC2CN(C(c3cn(C4CCOC4)nn3)=O)C2)n1 Cc1cnc2n1C(C(=O)NCCC1(C)CCN(C(c3ccncn3)=O)C1)CCC2 c1(C(=O)NCC2CCC(NC(C3CC(F)C3)=O)CC2)nccc2occc12.C c1(C(=O)NCC2CN(C(CC(=O)OCC)=O)C(C)C2)cccc(F)c1CC c1(C(N2CC(NC(C3CCC(OC)CC3)=O)C(SC)C2)=O)ccc(C)c(C)c1F C1(C(=O)Nc2c(C)ccc(Br)c2F)C2CCCC1CN(Cc1cnccc1Cl)C2 C(C)(C(CO)NC(=O)Cc1cnnn1C)NC(C(c1ccccc1)OC)=O c1(C(N2C(C)CCC(NC(c3cc(CO)[nH]n3)=O)C2)=O)cnc2ncccn12 C12(C(=O)NCC3(F)CC(NC(CSCC)=O)C3)CC1Cc1c[nH]nc12 C1(Nc2ccc(CC(=O)OC)cn2)CCCC(NC(=O)OC(C)(C)C)C1 c1(C(=O)NCC(CCNC(c2cc(OC)no2)=O)O)cc(C)ncc1C CCC(F)(F)CC(=O)N(CCNC(=O)C(C)Cc1ccc(F)cc1)C1CC1 c1(C(N(CCC(C)NC(C(CC2CC2)OC)=O)C)=O)cc2ccsc2n1C C1(C(=O)OC)CCC(CC(=O)N(CC(O)CN(C)C(C2CCOC2)=O)C)CC1 CCC(C)C(O)C(=O)N1CC(CO)(NC(=O)CCCCC2CCCCC2)C1 C1(NC(C(CC(C)C)O)=O)CN(C(c2c(N)cc(Cl)nc2Cl)=O)CC2(CC2)C1 N1(C(c2c(NC(C=C)=O)cccc2)=O)CC2CCC1C(NC(C1CC1C=C)=O)C2 Cc1cccnc1C(=O)NCC12CC1CN(C(C1(CO)CCC1)=O)C2 C12(Cn3cc(C(C4(O)CCCOC4)NC(C)=O)nn3)COC(C1)C(O)C2 Cc1nc(CC(=O)N(CCCO)C)cs1.c1(C(N(CC)C)=O)[nH]nnc1C1CC1 N1(c2n(C)nnn2)CC2CCC1C(NC(C1CCC3CC3C1)=O)C2 CCC(C(=O)NCC(C)(C1CCC1)NC(=O)CC1CS(=O)(=O)C1)OC CC1CN(C(c2ccsn2)=O)CCN1C(=O)Cn1ccc(Br)n1 c1(C(C)(C)C(=O)NC2CC(F)(CC3CC3)C2)cccnc1F.C(=O)(CCCF)N C(=O)(CC(CN(C)C)C(F)F)NCCCN(C(C(CC)F)=O)C.c1cccnc1 C(c1nc(C)cs1)=CC(=O)NCC1C(NC(C2(OC)CCC2)=O)CC1 c1(OC)ccc2cc(C(=O)NC(C)C(C)NC(=O)C(C)OC)n(C)c2c1 O=C(CC(C(F)(F)F)NC(c1cccn2nccc12)=O)NC1CCOCC1F c1(N(CC(C2CCCCC2)C)C)nc(=NC2CC2)[nH]c2cc[nH]c12 C1(C(=O)Nc2cccc(SC)c2)CN(C)CCN1C(c1cc(O)nc(O)n1)=O C1(C(=O)NC(CC)(C)CNC(=O)C=C2CCC2)CCc2n[nH]cc2C1 C1(CCC)CCC(C(=O)NCCCNC(=O)CCCc2ccncc2)CC1 C1CCCC12CCN(C(=O)CN1CC(C)(C)C1)CC2.C1(C)(CC)C=C(C=O)C1.N c1(CC)[nH]nc(C(=O)N(C2CCCC(NC(C3(CSC)CCC3)=O)C2)C)c1Cl CC1CCCN(CC(=O)C(N)C2CC2)C1CCc1ccc(Cl)c(Cl)c1 CCCC(CCCNC(c1nn(C(C)(C)C)cc1Cl)=O)NC(C1CC(O)C1)=O O=C(C(C(F)(F)F)C(F)(F)F)NC1(CC)CC1.C1(C=O)CC2CCCCN2C1.N C1(C(C)NC(CC(=O)OCC)=O)CCCN(C(C2(CO)CCCCC2)=O)C1 C(=O)(C(CC)C(=O)N1CCC(C(=O)N(CCC(C)C)C)(CC)C1)OCC C(=O)(CCCCCN(C)C)NC(C1CCN(C(CC(=C)C)=O)C1)C c1(C(N2CCN(C(CC=CCC)=O)C(CO)C2)=O)cnnc2ccccc12 c1(C(=O)NC2CCC(F)(CNC(=O)Cc3cnc[nH]3)C2)c[nH]c2ncccc12 CC#CC1CCN(C(c2ccn(CCNC(=O)CCCC(=O)NCC)c2)=O)C1 S(=O)(=O)(CCC(=O)NC1CCN(C(C2C=C2C)=O)C1(C)C)NC CC1CCN(C(c2cc(F)c(F)cc2O)=O)CCN1C(c1cccc(F)c1Cl)=O C(=O)(CCC(C)(C)NC(c1ccnc(C)c1)=O)NC1CCN(CCC)C1 N1(C(=O)CCc2nc[nH]n2)CCCN(C(C2CC3(CCC3O)C2)=O)CCC1 Cc1c(Br)cc(Br)c(NC(C2CC2C(=O)NCC2(O)CCCC2)=O)c1Br c1(OCC(N2CC(C)(NC(C3CCCCO3)=O)C2)=O)cc(Br)ccc1Cl N1(C(C2(C)CCCN(Cc3c(OC)c(C)ccc3)C2)=O)CCC2(CCCO2)CC1 C1(OC)CC(CNC(c2cnc(OC)nc2)=O)N(C(=O)CCC2CC2)C1 c1(C(=O)NC2CCC(NC(c3ccn(C(C)(C)C)n3)=O)C2)ccc(O)cc1 N1(C(C(C)N2CCC2)=O)CC(NC(c2ccc(C(C)(C)C)nc2)=O)C2(CCC2)C1 Cc1ccc(C(Cc2ccccc2Br)NC(=O)NCc2ncccc2Br)cc1C Cc1cccc(F)c1CC(=O)NC1CC(C)CN(C(c2ncc(F)cc2F)=O)C1 N1(C(C(C(=O)OCC)F)=O)CC(C=O)C(C)(C)C1.C1(C)CC(N(C)C)C1 N1(C(C(=O)NC(C)C)=O)CCC2CN(C(=O)CC(C)CN(C)C)CC2CC1 N1(C(c2c(C)snc2)=O)CCN(C(c2cc(=O)n(C)cn2)=O)CC1CC(F)(F)F C1(CNC(C2(C(F)(F)F)CCCCC2)=O)COC2(CCOCC2)O1 Cc1cc(C(N2CCOC(CCCNC(c3coc(C(N)=O)c3)=O)C2)=O)c(C)[nH]1 c1(C(N2CC(CC=C)C2)=O)ccc(F)c(Cl)n1.C1(=CC(=O)N)CCC(C)C1 c1(CC(=O)NC(C(C)(C)NC(CS(CC)=O)=O)C)c(C)nc(O)nc1O C(=O)(CCCCCC=C)NC(C1(O)CCCCC1)C(=O)NC(C#C)CC1CCCO1 C(=O)(C(F)(F)C(F)F)NC(C1CCC1)C.c1(CC=O)cc(F)cc(Cl)c1.N C1(NC(CCSC)=O)CCC(C)(C)CC1CNC(c1cccc(O)n1)=O N1(C(CCc2nnc(C)o2)=O)CCC(O)CCNCC1 CCC(C(=O)NC(C)C(C)OC)NCc1ccccc1 c1(CC)ncc(C(=O)NC2COCCC2NC(=O)CCOCCCOC)n1C c1(C(=O)NCC2OCCC(NC(C3CN(C)C3)=O)C2)c([N+](=O)[O-])cnn1C Cc1scnc1C(=O)N(CC(O)CNC(C1(CN2CCCC2)CC1)=O)C c1(C(C)N(C)C)cn(CC2CCCN2C(c2cc(C(F)F)cs2)=O)nn1 c1(C(N(CC(C)NC(C)=O)C)=O)ccc2c(c1)CN(C)CC2 CCCCC(O)CC(=O)N1CCC(C(N2CCC(F)C2)=O)(OC)C1 C12(NC(c3nccnc3Cl)=O)CCCN(C(=O)CC3CC4CC4C3)CC1C2 CCC(O)C(C)C(=O)NCC(C)(C)CN(C(=O)CCc1ccc(Br)cc1)C c1(C(=O)NCC(CO)NC(c2cc(C(CC)C)no2)=O)cc(OC)c(N)cc1F C1(C(N(CCC)C(C)C)=O)COCCN(C(=O)C(F)=CCCF)C1 Cc1nc(C(C)(C)C)nc(O)c1C(=O)NC1CNCC(C)C1 c1(C(=O)NCC(C)(C)O)cnc2[nH]cncc1-2.c1(CC=O)csc(Cl)c1.CC c1(C(=O)NC2CC(C)N(C(=O)CCc3nncs3)C2)cc2ccccc2cc1O c1(OCC)cc(C(=O)NC2(C)CCOCC2)ccn1.C(=O)CC.C(N)=O.N c1(C(N2CCCOC(CCO)C2)C(=O)NCCN2CCCC2)cc(Cl)ncc1Cl Cc1ccc(Cl)c(C(=O)NCC(C)(C)OCC)c1.c1(C(=O)N)ccc(C)o1 N1(C(C(C(C)C)OC(C)=O)=O)CC2CC1CN2C(c1cccc(Cl)c1)=O c12cc(n(C)n1)C1(CN(C(c3cc(OCC)no3)=O)C1)C2.N(C)(C)CC C(=O)(C(C)(C)C(C)(F)F)NCC#CCNC(c1c(C)nns1)=O C1CCCCN1C(C1C(Cl)(Cl)C12CC2)=O.C(C1CCCCC1)=C(C(=O)NC)F.C N1(C(C(C)OCC)=O)CCC2C(NC(c3cc(C(N)=O)[nH]n3)=O)C2C1 C1(C(=O)NC(C)CC(N)=O)CC2(CCC2)CN1C(=O)C=CC1CCC1 C(CCN=C(NCC1CCS(=O)(=O)N1C)NCC(C)(O)c1cccs1)OC CC(CC(C)(C)C)C(=O)N1CC(C)C1.c1(CC=O)ccccc1CS(N)(=O)=O C12CN(CCO1)CC(=O)NC2.CC(C)CCSC(C)C c1(CC)ccc(C)cc1NC(C)(CCOC)c1nnnn1CCC1(C)CC1 c1(C(=O)NCCC(F)(F)c2ccccc2)c[nH]nc1[N+](=O)[O-] C1(C(CC)O)CCCCN1C(c1ccc(CCCN)cn1)=O C#CC(C)(C)C(=O)NC(C1CCCN(C(=O)Cc2c[nH]nc2C(F)(F)F)C1)C N1(CC)CC(C(=O)NC(C)CCNC(=O)Cc2ccoc2C)CCC1=O C1CC(F)(F)CN1C(=O)Cc1ccncc1F.c1(CCC)nc(C(=O)NC)cs1 CCCC(C)(O)CC(=O)NC(CC(=O)N(C)CCn1ccnc1)C(F)(F)F c1(CC(=O)OC2CC(CC#N)C2)csc2ccccc12 C=CC(C)(O)CC(=O)NCc1ccc(C(=O)NCC(C)(C)C2CCC2)o1 C1(OCC)CC(N(S(=O)(=O)CC2(C(=O)O)CC(F)(F)C2)C)C1(C)C CC1(NC(=O)CN2CC3CC3C2)CCCN(C(c2cn3c(n2)CCC3)=O)C1 C(=O)(CC(C(F)F)n1cccn1)NCC12C(CN(C(=O)C#CC3CC3)C1)C2 C1(NC(CCCCCCSC)=O)CCC2(CC1)CC(NC(=O)CC1CCSC1)C2 C=CCC(CC=C)C(=O)N1C2CCC(C2)C1C(N1CCCC1(C)C1CC1)=O CC(O)CCC1CC1.C1(CC(=O)N)C=CC(NC(C2(O)CC(CF)C2)=O)C1 c1(C(N2CCOC(C)(C)C2)=O)sc(S(N)(=O)=O)cc1C.C=CC(O)C(=O)NC CC1CCN(S(=O)(=O)CC(=O)NCCN(C(=O)CC(C)F)C)CC1.C1CC1 c1(CC(N2CC(NC(c3ncccc3Br)=O)(CO)C2)=O)cnc2ccccn12 C1(CC(=O)NC(c2ncnn2C)CC)CCC(NC(c2c[nH]nc2CN)=O)CC1 N1(C(C2(C=C)CCCCC2)=O)CC=C(CC(=O)N2CCCC(CC)C2)CC1 c1(C(N2CCC(N(C(c3ccsc3C)=O)CC)C2)=O)ccnnc1Cl CC1(C)CC(C)(c2nc(C3CC3)no2)CN1CC1CC(F)(F)CO1 N1(C(C(CC)SC)=O)CCCC(O)(CNC(c2ccc(C3CC3)c(F)c2)=O)C1 Cn1ncc(CNC(C2(C3CCCN3C(=O)CN3CCCCC3)CC2)=O)c1Cl C12(CCOC(CNC(C(C)SCC)=O)C(=O)NCC)CC(CCO1)C2 N1(C(CCc2nc(C)c(C)o2)=O)CCCC(C)C1CCNC(C1SCCS1)=O c1(OC)ccc(Cl)c(C(=O)N(C2CCNCCC2C)Cc2cnc[nH]2)c1F CN1CCC(C)(C(N2CCC(C(O)CNC(C3CC3(Cl)Cl)=O)CC2)=O)CC1 C1(C(C)NC(=O)CC2CC2(Cl)Cl)CCN(C(=O)CCOC2CCC2)CC1 c1(CC)cnccc1C(C(=O)NC1COC1)N(C)Cc1cnn(C)c1 c1(C(=O)NC2CN(C(c3c(C)cccc3C)=O)CC2C)c(F)cc(F)cc1Cl C1(CNC(CN(CCC)C)=O)CCC2CN(C(c3cccnc3N)=O)CCC2C1 CC(C)CC(CNC(C12CC(C#N)(C1)C2)=O)C(=O)N1CC(C#N)C1 C(CCC(C)C)(C(=O)NCc1cn[nH]c1)NC(CSC)=O C1(CNC(CC(=O)NCC)=O)CN(C(=O)CCc2ccsc2Cl)CCC1(F)F c1(-c2cn(C(C)CNC(=O)CC3CC=CCC3)nn2)cnn(C)c1C(N)=O C(C)(C)(CCC(=O)NCC(CO)C1CCC1)NC(C(C1CC1)OC)=O C(=O)(C(C)(O)C(F)(F)F)N1CCN(C(C(C)C2CC2)=O)CC1 CC1(C)C(NC(=O)C(C2CCCCC2)F)CCN1C(=O)COc1ccon1 C(CCN(C)C(c1n[nH]c(C)c1C)=O)(C(C)(C)C)NC(c1c(CC)nco1)=O n1(CC(=O)NC(C2N(C(c3ncc(CC)cn3)=O)CCC2)C)ccc(C)cc1=O N1(C(CN(C)C2CC2)=O)CCC(NC(=O)CCc2cccs2)C1C1CC1 c1(C(=O)NCCC(C)NC(=O)C=CC)cc2ccsc2n1C.C1CCOCC1.O N1(C(c2ccc(C)cc2)C)CCC(F)(F)C(CNC(=O)CCCc2cccs2)C1 c1(C(N2CCN(C3CCN(C(c4c(C)ccs4)=O)C3)CC2)=O)c(C)cccc1N c1(C(N(CCCNC(CCC#CC)=O)C(C)C)=O)ccn2ccnc2n1 C(CN1CCCOP1(N)=O)NC1CCC(CC#N)C1 NS(=O)(=O)CCCCCC(=O)N1CCC(NC(c2nccc3c2CNC3=O)=O)C1 c1(C(C)NCCCN=[N+]=[N-])ccc2c(c1)C(C)C(C)O2 C1(NC(C2CCN(C)C2)=O)CC=CCC1C(=O)NCC(F)CO n1(CC(=C)C)nc(COC(C)C)nc1-c1ccc(C)nn1 c1(CC)ccc(C(N2CCC(CNC(=O)C(C)OC)(OC)C2)=O)cn1 CC(C(=O)N1CCC(C(F)CNC(=O)C=Cc2nccs2)CC1)S(N)(=O)=O C1(NC(C=CCCC)=O)CC12CCN(C(=O)Cc1cncc(F)c1)CC2 c1(C(N2CC(NC(C3CCS3(=O)=O)=O)C2)=O)ccc([N+](=O)[O-])cc1Cl N1(C(C2(C#C)CC2)=O)CCCN(C(=O)C(CC)C(C)O)CCC1 c1(CCC)cc(C(N2CC(F)CC2C)=O)c(C)o1.c1(C=O)cc(C)c(C)[nH]1.N CC1CCCN(C(=O)Cc2ccnn2C)C1CNC(=O)C(C)(C)c1ccnn1C C1(CN(C)C(c2cc(C)no2)=O)CN(C(=O)OC(C)(C)C)CCC12CCC2 c1(CNC(=O)NC(Cc2c(C)cc(F)cc2)C)cn(C(C)C)c(=O)nc1O C(=O)(CCC(C)(C)C#N)N1CCC(NC(C(C(C=C)C)C)=O)CC1 C(=O)CCS(=O)(=O)C(F)(F)F.C(=O)(C(C)(F)C(=O)N)OC.C1CCCC1.C c1(C(C)C(=O)N(c2ccnc(Cl)n2)CC2CCCNC2)ccc(F)cc1F C(=O)(CC(C)P(C)(C)=O)N1CCCN(C(C#CC(C)C)=O)CC1 c1(CC)cc(NC(=O)C(c2cccs2)NC(=O)C(O)C(C)C)ccc1F CC(C)(CC(F)C(=O)Nc1ccccc1O)NC(C1CCC(C2CC2)C1)=O O=C1CCCc2ncc(C(N3CCCC(C(O)C(F)(F)F)C3)=O)cc21 C1(NC(c2cc(C)c(Cl)s2)=O)COCCN(C(c2c(C)nsc2N)=O)C1 c1(C(N2C(c3scc(C(=O)NC)n3)CCC2)=O)cn(C)cc1C1CC1 c1(C(N2CC(C(N3CCC(C(=O)NC)C3)=O)(SC)C2)=O)cncc2[nH]ccc12 N1(C(c2n(C)ccc2)=O)CCC2(CC1)CC(NC(=O)Cc1cccs1)C2 c1(C(OCC)OC)cc(=NC(=O)c2cncnc2C2CC2)[nH]o1 CCN(OC)C(=O)CN=c1[nH]c2c(c(=NC(C)C3CCCCC3)[nH]1)CC(C)CC2 N1(C(C2C(C(C)(C)C)C2)=O)CC2CCC1CN2C(C1CC(Cl)(Cl)C1)=O N1(C(c2onc(C(C)S)n2)=O)Cc2ccnn2CC(C(=O)O)C1.c1ccc(F)cc1 C1(C)(C(N(C)CC2CCN(CC)C2)=O)CCCN1C(=O)C(c1ccccc1)C c1(C(=O)NC2C(OC)CN(C(c3ccn(CC)c3C)=O)C2)cc(Br)ccc1C C1(C(N2CC(NC(COCCSC)=O)C(C)(C)C2)=O)CCc2nnc(O)n2C1 c1(CNCC2(C(=O)Nc3nccc(OC)c3)CC2)ccc(C)nc1Br CON1CC(C(N2CCCC(C(=O)NCC3CCCC3)CC2)=O)CC1=O Cc1nc(C(N2CCCC(NC(C3(Br)CC3)=O)C2C)=O)cc(O)n1 Cc1nc(Cl)c(C)c(=NCC(C2CC2)N(C(=O)C(c2ccc(F)cc2)(C)F)C)[nH]1 c1(CNC(C2(c3cccc(C(F)(F)F)c3)CC2)=O)cc(F)ccc1Br N1(CC)CCC(N(C(=O)C(=O)NC(c2sc(C(C)C)nc2C)C)C)C(C)C1 c1(C(=O)NC(CN(C(=O)C=CCCC(C)C)CC)C)cc2ccc(O)cc2[nH]1 N1(C2CCN(C(CC=C=C)=O)C2)CCN(C(C2(C)CC=CC2)=O)CC1 N1(C(c2c(Cl)cnc(C)n2)=O)C2CCC1CC(CNC(c1cn(C)nn1)=O)C2 c1(C(N2CC(C)C(C)(CNC(C3(C)CC=CCO3)=O)C2)=O)cc(F)c(Cl)cc1F C1(NC(C(C)N2CCC2)=O)CC(NC(c2ccncc2F)=O)CC1O c1(OC)cccc(F)c1C(=O)NCC1CN(C(=O)C(C)CN(C)C)CCO1 c1(C(=O)NCC(CCNC(CCC=C)=O)OC)cc(Br)ncc1OC C1(NC(C(c2cnn(C)c2)C)=O)CN(C(c2cc(O)cc(F)c2)=O)CC2(CC2)C1 CCCCCCCC(=O)N1CCC(C)CC1C(=O)NC1(CSC)CC1 Cc1ccc(C)c(NC2CC2C(=O)NCCN)n1.c1ccccc1C=O.C c1(C(=O)NCCOCCNC(c2c(C#N)ccs2)=O)nccc2ccccc12 c1(C(=O)NC2C3(CN(C(c4c(F)ccc(N)c4)=O)C3)CC2)snc2ccccc12 C1(CNC(c2c(C)snn2)=O)CN(C(C2COCC(C)(C)O2)=O)CCCO1 CCC(CC)(CCNC(c1cnc(CO)nc1C)=O)NC(=O)CCC(N)=O CC(C)CCCCCC(=O)N1CC2CC(O)C1C2NC(=O)CC(O)C1CCCC1 c1(C=O)cccc(C(F)F)n1.c1(C(=O)NC2CC(C)C2)ccc(C2CC2)o1 N1(C(C(COC)NC(C)=O)=O)CC2OCCN(C(C3CC4(CC4)CO3)=O)C2C1 C1(NC(CCC)=O)CC2(C1)CC2C(N1CCSC(C)C1)=O N1(C(c2nn(CC)c(C)c2)=O)CCC2C(C1)CN2C(C1COCC1C(F)F)=O C1(C(C)C)CN(C(=O)CN2CCC(CO)CC2)CCN1C(C1CCCC(O)C1)=O c1(CC(C(=O)NCC(C(C)C)NC(c2cncs2)=O)C)ccc(C#N)cc1 c1(C(N(CCC)CC2CC2)=O)cccc(Sc2ccccc2)c1[N+](=O)[O-] C1(CC(N2CC(CCOC(C(=O)NC)OCC)C2)=O)CCCC(C)C1 c1(C(=O)NC)cc(Cl)c(C)c(S(=O)(=O)N2CC(N=[N+]=[N-])C2)c1 Cc1cc([N+](=O)[O-])ncc1C(N1CCN(C(=O)CCCC(N)=O)CC1)=O C(=O)(C(CC(C)C)OC)N(C1CCCCC1O)C(C=C)C1CCC1 c1(OC)cc(C(=O)NC2CCN(C(c3cocn3)=O)CC2C)c(F)cn1 C1(NC(C2C3CC4C(C3=O)C24)=O)CN(C(c2cn(C3CC3)nn2)=O)CCC1 CCC(C(=O)N1CCC(C)(C)C(C(N2CC(OC)C2)=O)C1)C(C)(C)CC C12(CNC(C(COC)COC)=O)CCCC(CN1C(c1cccs1)=O)C2 N1(C(c2c(CC)nns2)=O)CCOC(C(=O)NCC2CC3(CC3)CO2)C1 N1(C(Cn2c(C)ncc2)=O)CCCCC(NC(c2cc(C(C)C)nc(O)c2)=O)C1 C(=O)(N1CC(O)C(O)CO1)C1C2N(C(CCOCCC)=O)C(CC2)C1 N1(C(CN(CCC)C)=O)CCCC(NC(=O)CCCCCc2ccccc2)CC1 CC1(C)CN(C(c2cc(C(N)=O)ccn2)=O)CCC1.C1(C=O)CC(=O)N(O)C1.N CC(CCN(C)C)C(=O)NC(Cc1cc[nH]n1)C(=O)N(C)Cc1cscn1 C1(NC(CC2C(=O)NC(=N)S2)=O)C2CC1CN(C(C1CC3(CCC3)C1)=O)C2 N1(C(CCC(N)=O)=O)CCC(C2CCCN(C(=O)Cc3c(F)cccc3Cl)C2)C1 C1(OC)CCC(NC(=O)C=CCC(C)(C)NC(=O)Cc2cnc(C)s2)C1 N#Cc1c(OCC(=O)NCC=CCNC(=O)C(F)C2CCC2)cccc1Br c1ccccc1.C1(C)(N(C=O)CCO)CCS(=O)(=O)C1.CC(=O)N.C(C)C N1(C(COC(C)=O)=O)CC2(C)CC1(C(N1CC3(CC3)CC1CO)=O)C2 C(=O)(C1=CCc2ccccc21)N1CC(NC(C(C)OCCC#C)=O)C(OC)C1 n1(CC=O)c([N+](=O)[O-])cnc1C.CCS(=O)(=O)N(CC(=O)N(CCC)C)C C1(CNC(C(Cn2cccn2)NC(C2C=C(C)CS2)=O)=O)CN2CCC1CC2 N1(C(C(CCC)OCC)=O)CC2C3CCC(C2C1)N(C(C1CCCCS1)=O)C3 N1(C(CC)=O)CCOC(C(=O)N(CCNC(=O)CSC)CC)C1 C1(OCC)CC2(C1)CC2C(=O)N.c1(C(N2CCCC2)=O)n[nH]c(C)c1Cl.C C12CC(CO1)N(C(=O)CC=O)C2.CC1(C)CCOC1C(=O)N.CC(F)(F)F.C C=CCC(C(=O)N1CC(C=C)(CC(N2CCN(CC=C)CC2)=O)C1)C(C)C c1(OC)cccc2c(C(N3CCN(C(C4OCC4(C)C)=O)CC3CO)=O)n[nH]c12 C(=O)(C(C)C(F)(F)F)NC1CC(C)(NC(Cc2nc(C)[nH]n2)=O)C1 C1(CC(N2CC(N(C)C)C(O)C2)=O)CN(C(=O)CCc2nncs2)CC12CC2 C(C1CN(C(=O)C(=O)N(C)C)CC1C(=O)NCC1(Cl)CC1(F)F)=CC CCC(=O)CCC(=O)N1CCC(CCCNC(c2cc(C(C)C)nn2C)=O)CC1 N1(C(C(=Cc2cn[nH]c2)C)=O)CC(C)CCC1C(=O)NCC(C)(C)C1(O)CCC1 c1(C(=O)NC(CC)CN(C(=O)C(C)NC(N)=O)C)c[nH]nc1C1CC1 C#CCC(CC(F)F)C(=O)NCC1CC(C)N(C(c2cccn3ccnc23)=O)C1 c1(OC)cc(C(C)CC(=O)N(c2ccccn2)C2CCC2)ccc1C C1(CNC(C=C(CC)C)=O)CCC1(C)C.c1(CC=O)cc(C2CC2)on1.N c1(CC(=O)NC(C2CCN(C(=O)Cc3ccsc3)CC2)(C)C)cnccc1Cl N1(C(=O)COC(F)(F)F)CC2CCCC2(Nc2ncnc3ccsc23)C1 c1(C(C)C)cc(Br)ccc1C(=O)NC1CN(Cc2ccc(Br)c(F)c2)C1 c1(CN2C(C(=O)NC(CC(=O)OC)C)CNCC2)cc(Br)ccc1F c1(C=O)cc2c(n1C)CCOC2.C1(NC(C(C)OCCCC)=O)CCC(C)C1.N Cc1cc(OCC(N2CCCC2)=O)cc(C)c1.n1(CC(=O)N(C)C)cc(C)cn1 c1(C(=O)NCCCC(C)NC(C2=C(C)OCC2)=O)cn2nc(C)sc2n1 c1(CC(=O)NC2CN(C(Cc3nnc(C)o3)=O)CC23CC3)ccc2c(c1)CCC2 N1(C(=O)Cc2cnccn2)CC(C2CC2)(C(=O)NC2(c3ncc[nH]3)CC2)C1 C1(NC(C(CCC)O)=O)CCN(Cc2sccc2Br)CC1F c1(C=O)c(-c2ccccc2C)noc1C.C(C)(C)(CO)NC(C(C)SCC)=O.N C(=O)(C1=CCCOC1)NC1C(C(=O)NC(c2cn(C)nn2)C)CCOC1 CC1(CNC(=O)C(CC2CC2)NC(=O)Cn2[nH]cnc2=N)CC2CC2C1 C1(CCCNC(CCc2cnc(C)o2)=O)CCN(C(=O)C(C)C2CCOC2)CC1 C(C)(C)(CCCNC(C1CCCCS1)=O)NC(C1C(C)CCO1)=O Cc1cnc(O)c(CNC(C2(C(C)NC(=O)C(C)C(F)F)CC2)=O)c1 C(=O)(C(CCS(C)(=O)=O)OC)N(CCOC)Cc1c(C)nn(C)c1C N1(C(C(C)OCCCC)=O)CCCCC(NC(c2c(C)nc(O)nc2C)=O)CC1 C1(F)(C(=O)OC)CCN(C(C2CCC(NCc3ccsc3)C2)=O)C1 N1(C(CSCC(c2ccccc2)=O)=O)CC2CCC(C2)C1.C1(C=O)CC(O)C1.N C12(C(NOCC(C(C)C)O)=O)CC(CO)(CN1C(c1sccc1C#N)=O)C2 Cc1ccc(N)c(C(=O)NCC(C2CC2)N(C)C(c2cn3c(n2)CCC3)=O)c1 c1(C(N2CCN(C(C(CC=C)C)=O)CC(O)C2)=O)c(C)nc2sc(C)nn12 Cc1cc(OCC(N2CCCC2C(=O)NCC2CCCOC2)=O)no1 C1(C(=O)NCCCCN(C(C2(C#N)CC(C)C2)=O)C)CC2(COCCO2)C1 c1(C(N(C2CCN(C(C(COC)(C)C)=O)C2)C)=O)c[nH]c2ncccc12 C1(O)(C(=O)NCC(C2(O)CN(C(C(C)SC)=O)C2)(C)C)CCOC1(C)C C1(C(=O)O)CC2CC1CN2OCC.c12ccnc(n1)SC2 N12CCC3CN(CC13)C(=O)CCC(=O)OCC2=O.Cn1cc(OCC)cn1 Cc1cc(C(N2CC(CC(=O)NCc3cccc(F)n3)C2)=O)ccn1 C#CCC(O)C(=O)N1CCC(NC(c2cccc(C)n2)=O)C1C(C)C C(=O)(C1SCCc2sccc21)NC(CNC(c1cccc(OC)c1F)=O)C c1(C(N(C(CCNC(Cc2cnc(C)s2)=O)C)C)=O)cc(C#N)oc1C N1(C(C2C(CC)C2)=O)CC2CCC(C=O)(C2)C1.C(C(C)(C)O)C1CC1.CO C1(C)(NC(C=C(C)CNC(=O)C)=O)CC(O)(CO)C1.C1CCOC1=O.S c1(C(=O)NC(CC#C)C(=O)NC2(CC)CCCC2)nccc(C)c1N C1(NC(c2c(C)scn2)=O)CCCCC1CNC(C1(N(C)C)CCC1)=O c1(NC(C2CC2C(=O)N(CC(F)F)CCO)=O)cccc2c1CCCC2 C1(NC(CCCC)=O)CCCC2CN(C(C3(C(F)F)CCCC3)=O)CC12 C(=O)(CC(C)(C)C(F)(F)F)NCCCN(C(c1cccc(Cl)c1)C)C1CC1 C1(C(N2C(C)(CNC(=O)C=CC3CCCCC3)CCC2)=O)CCC(F)(F)CO1 C#CC1CC2(CC2)CN1C(C1CCN(C(c2oc(C)nc2CC)=O)C12CCC2)=O C1(NC(Cc2ccc(C)o2)=O)CC1C1CCN(C(=O)C=CC2CCCC2)CC1 c1(C(=O)OC)cc(NC(=O)C(=O)N(CC(C)C)Cc2cncs2)ccc1Cl CSC1=C(C(=O)NCC(CO)NC(C2CCCSC2)=O)CCCC1 C1(C(N(CCCNC(c2n[nH]cc2Cl)=O)C)=O)CC2(CCC2=O)C1 C1(C(=O)NCC2(C(=O)OCC)CCC2)CCCNC1 CCC(CNC(c1cc(C(F)F)no1)=O)(CC)NC(=O)CC1CCCCO1 C(=O)(N=c1[nH]onc1C)C1CCC(NC(c2c(C)cc(Cl)cc2)=O)CO1 CC1CCCC(C(N2CCSCC2C(N2C3CCC2CC3)=O)=O)C1 Cc1ccc(C(CN(C)C)NC(=O)COc2ccccc2)cc1.C(=O)C(C)C N1(C(C(C)OC)=O)CCCC(N(C)C(c2cc3occc3s2)=O)CC1 C1(NC(c2ncn(C)n2)=O)CCC(CC(N2CC(C(F)(F)F)C2)=O)CC1 C1(CN(c2ncccn2)C)CCCCN1C(C1(O)CCCC1)=O Cc1nc(N2CC(NC(=O)COC(F)(F)F)CC3(CC3)C2)c(F)c(C)n1 c1ccccc1.c1(C(=O)N)cn(CC2CC2)cn1.C12CC(C1)C(=O)NC2 N1(CC(=O)NC2C=CC(CNC(c3cocn3)=O)C2)CCCS1(=O)=O c1(C(=O)NC2(CC)CCN(C(C3(C)CCCCC3)=O)CC2)cc2cnccc2o1 Cc1cc(=NCC(C)c2cccc(Cl)c2)[nH]c(=NCCc2ccc(C)c(C)c2)[nH]1 C1(CCOC)(C(=O)N)CCN(C(=O)CCc2ccc[nH]2)CC1.CC(O)C(F)(F)F c1(CC(CO)NC(=O)NC(CCCOC)C(=O)N(C)C)c[nH]c2ccccc12 N1(C(c2ncn(C)c2)=O)CCc2cc(CNC(C3CCC4(CC4)C3)=O)ccc2C1 N1(C(C(C)(C)Nc2ccccn2)=O)CCCC(NC(C2(CCO)CC2)=O)C(F)C1 O=C(CCCF)N1CCC(C(N2CC(O)C(F)C2)=O)O1 c1(CC)cccc(CC)c1CC(=O)NC1CCN(C(c2ccc(Cl)o2)=O)C1 c1(C(N2CCC(CN(C)Cc3cc(OC)no3)C2)=O)cc2n(n1)CCC2 C1(N(C(C)C=O)C2CCC2)CCCCC1.c1ccn(C)n1.C(=O)C1CC1.C1CC1 Cc1cc(C(C)(C)C(=O)NC2CCC(NC(=O)C(C)(C)n3cccn3)C2)cs1 CC1CN(C(=O)CC2NC(=O)NC2=O)CCC1NC(=O)C=CCO c1(CC(=O)NC(c2cn(-c3ccc(Cl)cc3Cl)nn2)C)cc(F)ccc1F c1(C(N2C(CNC(CC(CCC)O)=O)CCCC2)=O)cc2ccc(Cl)cn2c1 c1(-c2cc(C(=O)NCC3CN(C(=O)CO)C3)on2)ccc(Br)cc1 n1(CC)ncc(C(=O)NCC2CCCCN2C(=O)C(CO)N(C)C)c1C C(=O)CCCCN1C(=O)CCC1=O.c1(CCOC)nnc(N2CC(O)(C)C2)s1.N N1(C(CC2(C)CCCO2)=O)CCC2CN(C(=O)C=Cc3cccc(CO)c3)CC12 C(=O)(C(C1CCC1)NC)NCCOC.c1cn[nH]c1.C(C)(C)C.C=O.N N1(C(c2c(C)ccc(C)n2)=O)CC2OCCN(C(=O)C=C3CCCC3)C2C1 CC1CCC(NC(c2cnc(=N)[nH]c2)=O)CN1C(c1cc(C(F)F)cs1)=O C1(CCCCC)CCCC1N=c1[nH]c(=NCc2cncc(Br)c2)c2[nH]ccc2[nH]1 C12(C(=O)OC)CC(C(N3CC(CC)C3)=O)(C1)C2.C1(CC=O)CCCO1.N C1(NC(Cn2ncn(C)c2=O)=O)CC12CCN(C(=O)C(C)(C)CC#N)CC2 c1(-c2c(OCOC)c(C)ccc2)cc(C(N2C3CCC2CC3)=O)cc2cc[nH]c12 N1(C(C(C)=C2CCC2)=O)CC2C3CCC(CC3)C2C1.C1(O)(CC(=O)N)CCOC1 C1(C(=O)NCC2CCC(Cn3cc(C(=C)C)nn3)CC2)CC12CCC(C)(C)CC2 C1(C(=O)NC(C2(C(=O)NC3CCC4CCC34)CC2)C)CCCCC(=O)N1 C1(C(=O)NCCC(C)N(C(=O)C=Cc2ncc[nH]2)C)CC2OC(=O)OC2C1 C#Cc1cc(NC(C2CCCCC2NC(=O)C(c2cnn(C)c2)C)=O)cc(F)c1 C(C)(C(=O)N1CC2CC2(CNC(C2CC2F)=O)C1)(C(C)C)OC C1(C(N2CCN(C)CC2)=O)CC2CCCC2N1C(C1CC2(CCC2O)C1)=O N1(C(C(C)NC(C)=O)=O)CCC2CN(C(C3Cc4cscc4C3)=O)CC2CC1 c1(OC)cc(OC)cc(CN2CCOC(C(=O)Nc3ccnc(Br)c3F)C2)c1 N1CC2C(C1)C2(C)C.c1(N(C)C)c(-c2cccc(C(F)(F)F)n2)cccc1Br C1(NC(C=CC=CC)=O)CCCC1NC(c1cocn1)=O.c1ccccc1 N1(C(C(COCC)NC(CC(=O)NCC)=O)=O)CCCC(C)CC1 CCCCCCC(CNC(C)C(C)(C1CC1)OC(=O)CCN)CC C1(O)(C(=O)NC2C(C(=O)NC(CC=C)(C)C)CCC2)CCCCCC1 C1(NC(C2CC(C)CC(C)(C)C2)=O)CN(C(=O)CC)CC1S(C)(=O)=O.C1CC1 c1(C(=O)NCC(C2CC2)NC(=O)CSC(F)F)ccc(C2CC2)s1 c1(C(C)NC(C(c2ccoc2)NC(CCC=CC)=O)=O)ccc(C)cn1 C1(CNC(Cn2cc(C(=O)OC)nn2)=O)CN(C(=O)C(O)CSC)CC1O C1(c2nnnn2Cc2ccccc2)(NCc2c(Cl)scc2)CCC2(CCCCC2)C1 C(C(C)(CO)NC(=O)COCCNC(=O)Cc1nocc1C)OC N1(C(c2c(C)snn2)=O)CC(NC(c2ccn(C3CC3)n2)=O)CC2(CC2)C1 Cc1ccc(C(=O)NCC2C3CC2N(C(c2cccs2)=O)C3)c(C)n1 C(=O)(CCCN=[N+]=[N-])NC(c1ccc(C(C)C)cc1)CNC(c1csc(Cl)n1)=O N1(C(C(C)OC)=O)CC2(C)CC(F)(C1)C2.c1(C=O)cccc(C(N)=O)c1.N C1(NC(=O)C(C2(O)CN(C(C3CC(N(C)C)C3)=O)C2)F)CCC(F)(F)C1 N1(C(c2c(CC)c[nH]n2)=O)CCC2OCCN(C(=O)C(C3CCOCC3)F)C2C1 c1(SC)ccccc1S(=O)(=O)N1CCCC1C(=O)Nc1ccc(C2CC2)c(F)c1 n1(CC)cnc(C(=O)NCC(CNC(=O)CN(CC)CC)CO)c1 c1(C(=O)NC(CC)CN(C)C(c2cc(CCO)on2)=O)ccncc1F N1(C(C(C)CO)=O)CCCC(c2nncn2C)C1 c1(C(=O)NC2C(NC(CCC(C)SC)=O)C2)sc2sccc2c1Cl c1(C(C(=O)NCC(=C)CCNC(=O)COCCSC)C)ccccc1.O N1(C(CNS(NC)(=O)=O)=O)CC(NC(=O)C2=CC3C=CC2C3)C2(CCCC2)C1 Cc1cc(C(=O)NC2CCC(CC(=O)NCC3(C)CCCC3)C2)c(C)o1 N1(C(C(CCC)C)=O)CCCC(O)(CN(C)C(c2ncncc2N)=O)C1 C(=O)(C(CCC(N)=O)n1nnnc1N1CCC(N2CC(C)(C)C2=O)C1)OC c1(CC)ccc(NC(=O)CC2(C)CCN2C(c2conc2CC)=O)cc1O N1(C(C(CC)OCC)=O)CCC2(COC(C)C2)C1.C1(C=O)(C(F)F)CC1.N Cc1cccnc1CC(=O)NCC(CO)(CO)NC(c1ccc(Br)o1)=O c1(OC)cccc(C(N2CC(C)(C(=O)Nc3ccno3)C2)=O)c1OC N1(C(CCc2cc(C(=O)O)[nH]c2)=O)CCCC2C(C(F)(F)F)C12 C(=O)(C(C)(C)C(N)=O)N1C(CN(C(=O)C2=CCCCO2)CC)CCC1 c1(NCCC(=O)N(CCCC)C)ccccc1Cl.N1(CC(=O)N)CCC(C)(O)C1 c1ccc([N+](=O)[O-])c(C=O)c1.C1C=CCN(C(=O)CN(C)S(N)(=O)=O)C1.C CC1(C(=O)NC2C=CCN(C(=O)CCc3ccc(Cl)s3)C2)CCSCC1 N1(C(c2n(COC)ncc2)=O)CCN(C(c2cc([N+](=O)[O-])c[nH]2)=O)CC12CCC2 N1(C(CSCCOC)=O)CCN(C(=O)C(C)C(C)O)CC1C1CCCC1 C(=O)(C1CCCn2nccc21)NC(C1CCN(C(C(CC)(C)CC)=O)CC1)C n1(C(C)(C)C)c(NC(c2sccc2-c2ccccc2)=O)nc2ccccc12 c1(N(C2C(N(C(c3cc(C)sc3C)=O)C)CCCC2)C)nc2ccc(N)cc2s1 N1(C(CC(C)C2CC2)=O)CCCCC1c1cn(CCCN(C)C)nn1 N1(C(C(C)NC(c2ccoc2)=O)=O)CCC(NC(=O)CCC2CC2)CC(O)C1 CCCCC(CC)CC(=O)NC1CCCC1NC(C1CC2COCC(C1)C2)=O CC1OC2CCC1(C(=O)NCC=CCNC(C1CCOC1C1CC1)=O)C2 N1(C(C(C)n2ccnn2)=O)CCCC(F)(CNC(C2CC(F)C2)=O)CC1 N1(C(C2(C(=O)OCC)CC2C(F)(F)F)=O)CC2CCC1C(OC)C2 C(CC(O)C(=O)NC(C1CCN(C(=O)C(=O)N(C)C)C1)C)OC c1(C(=O)NCCC(C(=O)NC2(CSC)CCC2)C)[nH]ccc(=O)c1C Cc1cccc(-c2cnoc2C(N2CCN(C(c3ccnc(C)n3)=O)CC2)=O)c1 C1(C(=O)NCCCCc2cnc[nH]2)CC12CCN(C(c1csc(Cl)n1)=O)C2 N1(C(C2(C)COCCO2)=O)CC2CCN(C(=O)Cn3cnnn3)CCC2C1 Cc1ccc(C(N2CCN(C(c3nc[nH]c4ncnc3-4)=O)C3CC23)=O)cc1C#N C(CCC)c1ccccc1.C(C(=O)N)(C1CCC1)OCC.C(=O)CC1(C)CC1 C1C2CC1N(C(c1ocnc1C1CC1)=O)C2.Cc1c[nH]nc1C1(C(=O)N)CC1 O=C1CCN(CCc2ccc(F)cc2)C(=O)N1CC1CC2CC1C2 C1(CNC(CCCOC)c2nnnn2-c2ccccc2)CCCN(C(=O)OC)C1 c1(C(N(C(CNC(C2C(OC)C2)=O)C)C)=O)cnc2nccn2c1 N1(C(c2cocn2)=O)CCN(C(=O)C(F)=C2CCCC2)C(C2CCC2)C1 CC1(CC(N2CCC3CC23C(=O)NCC#CC#CCO)=O)CCCCC1 c1(NC2(c3n(CCCC)nnn3)COC2)cnn2c1OCC(O)C2 c1(CNC(CC(C)CNC(=O)C(C)c2ccco2)=O)ccccc1C#N Cc1n[nH]c(C)c1CCC(=O)NC1CN(C(C2CCC3(CC3)C2)=O)CC1C N1(C(c2scc(OC)c2)=O)CCCCC12CC(NC(c1cnn(C(F)F)c1)=O)C2 C1(CNC(C2C(CCOC)C2)=O)CCCCN1C(=O)Cc1nocc1C c1(C(N(C)CC2(O)CN(C(c3cc(C)n(C)c3)=O)C2)=O)csc2ccccc12 Cc1[nH]c2ncccc2c1C(=O)NC(C1CN(C(c2ccc(CO)nc2)=O)C1)C c1(NC(CC)CNC(=O)C=Cc2ccco2)ncnc2cnccc12 C12(NC(c3n(C)ncc3)=O)CCC(CC1NC(c1c[nH]nc1Br)=O)C2 C(S(=O)c1cccc(Cl)c1)c1n(C(COC)C2CC2)nc(-c2ccoc2C)n1 N1(C(CCC)=O)CCC2CN(C(=O)CC3C(=O)N(C)N=C3C)CC2C1 C(=O)(C(CCF)NC(c1scnc1Cl)=O)N(C1CCN(CC)C1)CC C(=O)(C1=C(Cl)CCOC1)N1CCCC1.CC(C(=O)N)N(C)C=O.C(C)(C)C.C C1(OCC(N2CCC(OCCNC(C3C(CC)C3)=O)C2)=O)CCCCC1 CC1CCC(CNC(c2cc(CO)[nH]n2)=O)N(C(c2[nH]cc3c2CCC3)=O)C1 C(=O)(C1=CCSC1)NC(C)Cc1ccccc1.c1(CC=O)csc(C(C)C)n1.N C1(CNC(c2csnn2)=O)CC2(CO1)CN(C(C1CC3(CCOC3)C1)=O)C2 C1(CN(C(c2c(CC)nn[nH]2)=O)CC)CCCCN1C(=O)Cn1cnnc1 C12(NC(C=CCN(CC)CC)=O)CC(C(=O)N)(C1)C2.c1cc[nH]c1 c1(C(N(CC)CC)=O)ccc(N)c([N+](=O)[O-])c1.c1(C=O)cc2ccccn2c1.N C(=O)(CN=c1cc[nH]cc1)N1C2(CNC(=O)CSc3nncs3)CCCC2CC1 C1(C(=O)N(CCCOCCN(C(=O)Cn2cncn2)C)C)(CC)CCCC1 c1(NC(c2ccc(NCc3c(C(=O)OC)ccs3)cc2)=O)nccc2[nH]ccc12 CC1(C)CN(C(C23CCC(C2)C3)=O)CC(CNC(c2ccc3sncc3c2)=O)O1 O=C1C=C2CN(C(C3CC(F)(F)CN3C(=O)CCCCCCCO)=O)CCC2S1 CCCCC(C(=O)N1C2CC1CN(C(c1c[nH]c(C#N)c1)=O)C2)N(C)C C1(CC(=O)NCC(CNC(=O)Cn2cnccc2=O)O)CCC(F)(F)CO1 C1(OCC)CC(CO)CN(C(C2CCSC2(C)C)C(=O)NCC2CC2)C1 c1(C(N2C3(CNC(CC(C)C)=O)CCC3CC2)=O)cc2ccccc2o1 C1(NC(C2(CC=C)CCCN2C(=O)CCCF)=O)CCC2(CCC2)CC1 c1(C=O)cc(N)c(Cl)cn1.CC(O)(CNC(c1ncsc1C(F)(F)F)=O)C Cc1nc(C(C)(C)C)sc1C(N1CCOC(C)C1)=O.C(=O)(CCc1nc[nH]n1)N C12(C(CNC(c3cnccn3)=O)NC(C3CC4CC4C3)=O)CCC(CC1)C2 N1(C(C2CCC(=O)NC2)=O)CC2(CCCCN(C(c3cc4ccsc4s3)=O)C2)C1 N1(CC(=O)N=Cc2cocn2)CCC(N=c2[nH]c(C3CC3)nc3c2CCC3)C1 C1(CNC(C2(CNC(COC)=O)CC2)=O)CCN(C(C)=O)C1 C1(NC(C(CNC(c2c(C(C)C)c[nH]c2)=O)C)=O)CCC(=O)NC1=O N1(CCCC)CCCCC1C(=O)N(C)C.C1(O)CN(C(C2CC2C(F)F)=O)C1 c1(C(=O)NC(C(CO)NC(C(C=CCCC)O)=O)C)ccc(C)c(F)c1 N1(C(c2c(C)[nH]c(=N)s2)=O)CCC(C2CN(C(=O)CC3CCC3(C)C)C2)CC1 CCCC(C#N)C(=O)N1CC(CNC(=O)C(F)(F)c2ccccc2)(OC)C1 c1(CC)cccc(CC)c1CC(N1CCC(C)C(NC(=O)CC(CC)OC)C1)=O c1(OCC(=O)NC(CCCNC(C(C)=C2CCCC2)=O)C)ccc(F)cn1 c1(C(N(C(C)CNC(=O)C)CC)=O)n[nH]c2c1COC2.c1n[nH]c(O)n1.S C(=O)(CCC(=O)N1CCCC(CCCCNC(=O)C=C2CCOCC2)C1)N(C)C Cc1cc(NC2CC(NC(=O)C(c3ccc(C4CC4)cc3)O)C2)nc(C)n1 C=CCC(C)(C)C(=O)NC(C)C(C)NC(=O)CCC(F)(F)F Cc1cccc(NNC(=O)C(=O)Nc2ccc(CCC(C)(C)C)cc2)c1 N1(C(CC=CC)=O)CC2CCC1CC2NC(c1csc(-c2ccccc2)n1)=O C1(NC(CN(C)C2CC2)=O)CCCOC1c1ccc(Cl)cc1 N1(C(c2ccn(CCC)n2)=O)CCC(C)CC1CNC(=O)C(C)CSC c1(C(=O)NCC2COCCO2)cc(F)ncc1NCc1cccc(O)c1 CC1=C(C(=O)NC2CCCCC2)CCS1(=O)=O.c1(C(=O)N)cc(C(C)C)oc1C C1(C(N2CC(F)(C(N)=O)C2)=O)CC(NC(=O)Cc2ccc[nH]2)CCO1 CN1CC(n2cc(CN(C)CC3CCCCC3O)nn2)Cc2ccccc21 c1(CN2CCN(C(c3ccc(OC)cc3I)=O)C3C2C3)ccc2nc(C)oc2c1 c1(CC(=O)NCC2CCN(C(CCC=CC(C)C)=O)C2)ccc(Br)c(O)c1 Cc1c(C(N2CC3CC2(CNC(=O)C=C2CN4CCC2CC4)C3)=O)cncc1N C(=O)(C1=CCSC1)N(CCCNC(CSCC(C)C)=O)C c1(C(N2CC(C)C(NC(C3(C)CC4CCC(C3)S4)=O)C2)=O)c(F)ccc(O)c1F c1(C(C)C)cc(C(=O)NC2(C)CC(NC(=O)CCn3cncn3)C2)no1 C#Cc1ccc(C(=O)NCCC(C)(C)C)cc1C.C12(CC(=O)N)COCC(C1)C2 N1(C(Cn2c(C)nnn2)=O)CC(O)CC1CNC(c1ccc(=O)oc1)=O C12(C=O)CC3CC(C1)CC(C)(C3)C2.N1(C(C2CC2)=O)CCC(CC)CC1.CO C(=O)(C1=CC2(CN(C(=O)Cc3ccsn3)C2)OC1)N(CC#C)CCF C1(CCNC(c2nccc(C)c2)=O)CCCN(C(c2ccc(Cl)c(N)c2)=O)CC1 C1(CC)CN(C(C2CCC(NC(C3CCCSC3C)=O)CC2)=O)CC(=O)N1 Cn1ccnc1CC(=O)NCCOCCCNC(C1CC1c1cccnc1)=O C1(C(N(CCCNC(=O)C(N2CCOCC2)C2CC2)C2CC2)=O)CCCC1O c1(C(N2CCN(C(CSCC(=O)OC)=O)CC2C2CC2)=O)ccnc2ccnn12 N1(C(CCC#C)=O)CCCN(CCNC(c2cc(C)n(C(C)C3CC3)n2)=O)CC1 C(CCCC(C)NC(=O)C)NC(C(C=CC)O)=O.C(=O)CCC1CCCC1.N c1(C(=O)NC(C(C)NC(C2(C)CC=CC2)=O)CO)cccn2nccc12 C1CC(O)C1C=O.C1(C=O)(C2CC2)CCOC1.CC(C)(C)OC=O.CC N1(C(C(c2n(C)ccn2)(F)F)=O)CCN(C(=O)CNS(N)(=O)=O)C(CF)C1 C1(F)(C(=O)NC2CN(C(CC(CC)(F)F)=O)C(C)CC2)CCC(F)(F)CC1 C(=O)(CCC(O)C(C)(C)C)NCC1CN(C(=O)CCC2CCCC2)CC(C)(C)O1 CN1CCN(CC(=O)NC(Cc2ccoc2)C(N2CC3CCC2C3)=O)CC1 CCCC(CCC)C(=O)NCc1ncccc1C(=O)NCc1cc[nH]n1 c1(CC(=O)NC(C2CCC(F)(F)C2)C)ccc2c(n1)OCCO2 C1(C(N2CCC(NC(COC(CC)CC)=O)CC2)=O)CC2CCC(C1)C2=O C(=O)(N=c1[nH]nc(C2CC2)n1C)C1C(C)OCCN1C(=O)OCc1ccccc1 c1(CSCC(Cc2ccccc2)OC)cc2ccc(C(=O)O)cc2[nH]1 c1(C(N2CCCC(C(C)NC(CCSCCC)=O)C2)=O)ccc(Cl)cc1O C1(N(C(C(C)(C)CCl)=O)CCN2CCNC2=N)CCC2(CC1)CNC2 c1(C(=O)NC(CC)CNC(=O)C(C)O)cc(Cl)ccc1OCCOC c1(NC(C2(CC)CC(C)(C)C2)c2nnnn2C)ccc(F)c(S(N)(=O)=O)c1 C1CN(C(=O)OC)C(=O)O1.c1(CC2(O)CC(OCC)C2)ccon1.O N1(C(CCCC#CC)=O)CCC2CN(C(c3cccnc3N)=O)CC2C1 Cc1cc(C(N2CCN(C(=O)CNC(C3CCC34CCC4)=O)CC2)=O)cc(C)n1 N1(C(C(CC=C)c2ccccc2)=O)CC2(CCCC2NC(C2CCC2)=O)C1 O=C(C(CO)C(F)(F)F)NC1C2CC1N(C(C1COCCO1)=O)C2 C(=O)(C#CC1CCOC1)NC(CC(C)C)(C)CNC(c1csc(S)n1)=O N1(C(C(C)NS(CCC)(=O)=O)=O)CC2CC(NC(C3CC(O)C3)=O)CC1C2 C1(NC(c2cc(C(=O)OC)oc2C)=O)CN(C(=O)CO)CC(C)(C)C1 N1(C(C2N(C)C(=O)CC2)=O)CCOC2(CCS(=O)(=NC(=O)C3(CF)CC3)CC2)C1 C(CCCCCC(=O)NC1CCOC(C2CCCN(C(=O)CNC=O)C2)C1)SC C(=O)(CS(=O)(=O)C1CCCC1)N(CC(C)NC(CC(CC)(F)F)=O)C CCCCC(CC)C(=O)N1CC2CCN(C(c3cn(C(C)(C)C)nn3)=O)C2C1 N1(C(C(C=CC)O)=O)CCCC12CCCN(C(c1cn(C)c(=O)cn1)=O)C2 CC1CCN(C(c2ccccc2Cl)=O)C(C)C1NC(C12CCOC1CCOC2)=O c1(CN2CCCC(SCC(C(=O)OC)C)C2)cc(Cl)c2c(c1)OCO2 O=CN1CCOCC1C(=O)NC1CCCCC1NC(=O)Cc1cnoc1 CC1C(NC(=O)C(N2CCOCC2)C)CCCN1C(=O)CCCc1ccsc1 C(=O)(C(CC)C(F)(F)F)N1C(C(N2CCC(C=C)C2)=O)CN(C)CC1 c1(C(N2CCCC(CCNC(C(CCCOC)C)=O)C2)=O)cn2cnnc2cn1 CCCC(N)CCCNC(C1CC(=O)C1C(C)(C)C)=O Cc1nc(C)c(C(=O)NC(C)(CNC(=O)C(F)(F)C2CCCC2)CO)o1 CC1(CNC(c2cc[nH]n2)=O)CCN(C(=O)C(c2ccc(C#N)cc2)(C)C)CC1 CC1CCN(C(C23CCCCC2C3)=O)C1CNC(=O)COCC(F)F c1(OC)ccc(C(=O)N(C)CC=Cc2ccccc2)c(F)c1 c1(C(N2CC(NC(C(CC=C)NC(C)=O)=O)C(OC)C2)=O)ccc2c[nH]nc2c1 c1(C(=O)NC2CCN(C(C3(Cl)C(C)(C)C3)=O)CC2F)ccn2cnnc2c1 C1(C(=O)NC(C)CCNC(c2csc(CC(F)(F)F)n2)=O)CCC(C)(O)CC1 CCC(CCC(=O)N(CC(=O)NC)CC)NC(c1c[nH]c(=S)cn1)=O N1(C(=O)CCCc2ccccc2Cl)CCOC2(C1)CN(C(=O)CCF)C2 C(=O)(C(C(F)(F)F)C(F)(F)F)NCC1(C)N(C(C2C(C)(C)C2)=O)CCC1 C1(C(=O)NC2C3CN(C(CSCCC(C)C)=O)C2C3)CCC2C1C2(F)F N1(C(C2C(CNC(c3ccn(COC)n3)=O)CCC2)=O)c2ccccc2CC1C C1(NC(C23N(C(c4c(NC)cccc4)=O)CCC2C3)=O)CNC(=O)C1(C)C CCCCCCNC(c1cc(COC)no1)=O.C1(C(=O)N)CC1C(F)(F)F Cc1cccc2cc(NC(P3c4ccccc4CC3O)C3CC3)cnc12 N1(c2n(CC3(SC)CC3)c(C3CC3)nn2)CCN(CCc2ccsc2)CC1C O=C(C1=NOC2(CCN(C(=O)C3=NNC(=O)C3)C2)C1)Nc1cc(F)c(F)c(F)c1 C(CCCN1CCC1)c1ccccc1.C(=O)(C(=O)N)NCC1(CSC)CC1 C#CCC(C)(CC)C(=O)N1CCOCC(NC(=O)Cc2cncnc2)C1 CS(=O)(=O)CCCN=c1[nH]c2ccc(S(=O)(=O)N3CC=CCC3)cc2s1 C1(CC(=O)NC2CN(C(=O)CCc3ccnc(Cl)c3)C2)CC2COCC12 N1(C(c2csc(C)c2N)=O)CCC(CNC(C2Cc3nccn3C2)=O)C(F)(F)C1 N1(C(C(CC)=CCCC)=O)CCOCC1CNC(=O)CN1CCC(CO)CC1 Cc1csc(C(N2CC(CNC(c3ccccc3Cl)=O)C3CC23)=O)c1Cl C(=O)(CS(=O)(=O)CCO)N1C(CNC(C2C(C(C)C)C2)=O)CN(C)CC1 c1(C(=O)NC(CN(C(=O)CCS(C)(=O)=O)C)(C)C)cc2cc(Cl)cnc2o1 c1(C=O)ccc([N+](=O)[O-])cc1[N+](=O)[O-].CS(=O)(=O)C1(C(=O)NCCCO)CC1 Cc1nc(C(C)NC(=O)CC2CCC2ON)c(C)o1 C(=O)(C(C)CC=CCC)N(CCN(C(CC=CC=C)=O)CC)CC c1(OC)cc(C(=O)NC23CCCC2CN(C(c2nn[nH]c2Cl)=O)C3)cc(F)c1F C1CN(C(=O)CC(C)n2ccc(C)n2)CCO1.C12(CC)CC(C(=O)N)(C1)C2.C C1(NC(C(C)N(C(C)=O)C)=O)CCCC(C(N2CC(F)CC2C)=O)CC1 N1(C(CCN(C(=O)CCC(=O)C2CC2)CC#C)=O)CCC(CF)CC1 c1(C(C(=O)NC(C(C)C)CNC(C2CC(F)(F)C2)=O)C)noc2ccccc12 c1(CC(C)NC(C(C)N(C(=O)C(C)C2(O)CCC2)CCC)=O)ccncc1 c1(NCC2(C)CCCN(C(C3(n4cncn4)CC3)=O)C2)ccnc2ncnn12 c1(NC(=O)OC)ccc(C(=O)NCCC(O)C)cc1.C1(CC=O)CC=CC1 Cc1sc(=O)n(CC(=O)NC2CCN(C(=O)CC3CCCC(=O)N3)CC2C)c1C CC1=C(C(=O)NC2CC(C)C2)C(=O)OC1(C)C.C1(C(=O)N)CC12CCSCC2 c1(C(N2CCN(C(=O)CO)CC2)=O)cccc(F)c1C(F)F c1(C(=O)OC)nsc(=NC(C)C2CC(NC(c3coc(C)c3)=O)C2)[nH]1 N1(C(c2c(C)cc(C)nc2Cl)=O)CCN(C(c2ccsn2)=O)CC(C)(F)C1 C1(C(=O)NCC2(CC)COC2)CSCN1S(=O)(=O)CC1CC2CC1C2 N1(C(CCCCC=C)=O)Cc2occ(C(=O)NC3(C)CC(F)(F)C3)c2C1 Cc1ccccc1CC(=O)NC1(CO)CCN(C(C2(CCN(C)C)CC2)=O)C1 N1(C(Cc2nc(NC(=O)CC3(C)CC3)cs2)=O)CCC2CCCC12OCC c1(OCC(N2CCC(NC(c3cccc(I)c3)=O)C2)=O)cccc(F)c1F N1(C(C(C)=C(C)C)=O)CCC(NC(c2cc(-c3ccncc3)no2)=O)C1C N1(C(=O)C(F)=CC2CC2)CCC(F)(C(=O)NCC2(C3CC3)CCCO2)CC1 C(=O)(C1=CC(O)CCC1)NC1CN(C(COCP(C)(C)=O)=O)CC1O C1(C(=O)NCC(C(C)C)CO)CCC(C)CN1C(C1COCCC1C)=O c1(OC)ccnc(F)c1C(=O)NC1CCN(C(=O)C(C)C(F)F)CC1O c1(COC)nc(OC)cc(N2CCN(CCCNC(=O)C(O)COC)CC2)n1 C=CC(CC)CC(=O)N1CCN(C(c2cc(F)ccc2OC(C)C)=O)CC1CF N1(C(c2cnc3n2C(C)CCC3)=O)CCOCC12CNCCOC2 N1(C(c2csc(C)c2C)=O)CCN(C(C2CC(C)(C)C2)=O)C(C(C)C)C1 CC(CC(=O)NOC1CCCC1)NC(=O)C(C)(C)O Cc1cccc(NC(C2CCCCN2C(c2nccs2)=O)=O)n1 c1(C(C(=O)OCC)NC(c2conc2)=O)ccc(NC(C)=O)cc1Br.C c1(C(=O)NCC2=CCN(C(=O)C(F)(F)C(F)F)CC2)cncc2ccsc12 c1(C2(C(=O)N)CC2)ccc(Cl)cc1.C1(C(N2CCCC2C)=O)(OC)CCSC1 c1(CC(=O)NCC2(CNC(C(C)SC)=O)CC2(F)F)cccnc1F c1(CC(N2C(CCNC(=O)CC3CC3)COCC2)=O)cc2ccccc2s1 c1(C(=O)N)ccc(C=NOC)cc1.C1(NC(CN(CC)CC)=O)CC2CCC1C2 C(CC1CC1)(C(=O)NCC1CC12CCC2)NC(COCC)=O O=C(NN=c1ccc2nccn2[nH]1)NCc1cc(Br)no1 S(=O)(=O)(c1ccc(Br)c2ccccc12)Nc1c(C(=O)OC)ccc(F)c1 c1(NC(c2cc(Cl)ncc2NCc2cn[nH]c2)=O)cc(F)ccc1Br C(=O)(CC(C(F)F)C(C)(C)C)NC1CN(C(C=CCN(C)C)=O)C2C1CCCC2 Cc1cc(O)nc(N2CCC(C(=O)NC3CCC3)CC2)n1.C12C(C)CCN1CC2 C(=O)(C1=NOCC1)NCCC(C)N(C)C(C1CC2CCCC12)=O c1(N(C2CCC(Oc3ccccc3)CC2)C)cc(Cl)nc(Cl)c1 C1(C(N2C(CNC(c3c(CCC)[nH]cc3)=O)COCC2)=O)CCC(C)(C)OC1 C1(N(C(=O)C(C)OCCOC)CC#C)CCN(C(C2(CO)CCCC2)=O)C1 C(N=c1cc(NCc2cc(F)c(Cl)cc2F)nc[nH]1)c1n(C)ccn1 C1(CC)CCN(C(=O)C)CC1.c1(C(C=O)=O)cnn(C)c1.C1(C=O)CC1C.N c1(C(=O)NCC(CCNC(CNCCCOC)=O)OC)ccc(C)c(C)c1N c1(C=O)cccc(O)c1F.c1(C(N(CC)CC2CCOC2)=O)cc(C)[nH]n1.N C1(NC(CC2CC(C)(C)CN2C(C2CC3(CC3)C2)=O)=O)CCC2(CCCC2)C1 c1(C=O)ccc2oc(=O)oc2c1.Cc1cc(Cl)c(C(=O)NCC2CC2)cc1F.N C#Cc1cc(C(N2CCC(CNC(=O)CC3CCOCC3(C)C)C2)=O)ccc1C C1(CNC(C=NOC)=O)CCC(NC(=O)CC(C)NC(C2CCCCC2)=O)CC1 c1(C(=O)NC2C(CNC(CCC(=C)C)=O)C2)ccc2n[nH]c(CCC)c2c1 C(=O)(C(O)C1CCCC1)NCCN(C(=O)CC1(C#N)CC1)CCC CNS(=O)(=O)NCC(=O)NCC(F)CNC(=O)C=C(C)C1CC1 N1(C(CSc2ccc(OCC(N)=O)cc2)=O)CCCOC(CNC(=O)C)C1 c1(C(=O)NC2(CC=C)CN(C(=O)C(O)CCC(C)C)C2)cccn2c(C)nnc12 C1(C(=O)NC2CC(C)(NC(=O)CSc3ccccc3)C2)CCCC(F)C1 C(=O)(C(C)c1cc[nH]n1)NCCOCCNC(C1(COC)CC1)=O N1(C(C(CC(C)C)C)=O)CCC(C2(NC(c3ccc(=O)n(CCF)n3)=O)CC2)C1 C1(NC(c2cn(C(C)C)nc2)=O)CN(C(c2ccc(C(C)(C)C)[nH]2)=O)CC1C c1(CC(N2C(C)CN(C)CCC2)=O)cc2ccccc2c(O)n1 c1(OCCC(=O)NC(CNC(c2c(C)nn(CCO)c2)=O)C)ccc(Cl)cc1Cl N1(C(=O)C=CBr)CC2CN(C(C3CCCCS3)=O)CC(C1)O2 C(=O)(C#CC1CCCOC1)N1CC(C)(NC(CC(CN(C)C)(C)C)=O)C1 N1(C(C)C)C(=O)NC2(CCN(C(=O)NC3CC4(CCOCC4)C3)C2)C1=O C12(C(N(C(C)C(C)(C)O)C)=O)CC1CCN2C(c1cnn(C)n1)=O CCC(CCCC(=O)NCC1C=CCCC1)NC(=O)CCCc1ncco1 C1(CCC(=O)NC2CCC(CNC(c3cc(C)oc3)=O)C2)NC(=O)NC1=O c1(OC)ccc(CC(N2CCCC(C)(C)C2)=O)c(Cl)c1.C(=O)C(C)C(C)(C)O.N Cc1cc(C(N2CC(NC(=O)Cn3[nH]cnc3=N)C3(CCC3)C2)=O)cc(C)c1C C(=O)(C(C)(CO)NC(c1cnncc1O)=O)N(CCCC(=O)NC)C c1(C(N(C2CCCN(C(C3C(C#N)C3)=O)C2)CCF)=O)n[nH]c2c1COCC2 C(CC(=O)N(C)CC1CC1(F)F)(C(F)F)NC(C(C)SC(C)C)=O C1(NC(COC(CC)C)=O)CC(NC(c2cnn(CC(C)(C)O)c2C)=O)CC1O c1(-c2cc(OCCOC)ncc2)cc2c(C(=O)NCC3CCO3)coc2cc1N C1(C(N(CC(C)NC(c2cnc(CC(C)C)[nH]2)=O)C)=O)CCCC1(C)C N1(C(C(C)N(CC)CC)=O)CC(=O)NCC1C(=O)NC1C(O)CC1O Cc1c(C(=O)N(CC)C(C)C)cc(C2CC2)n1C.c1(C(C=O)O)ccccc1.N c1(CC2CC(NC(=O)Nc3cc(C(C)C)c(Cl)cc3)C2)csc2ccc(F)cc12 C1(NC(C2C(=C)C2)=O)CCN(C(=O)Cc2ccccc2C)C12CCC2 C(C(C(=O)N1CC(OCC(F)F)C1)C(C)C)NC(c1cncc(C)n1)=O C1(C(C(=O)NC)OC)CC(F)(F)C1.C1CCC1.C1(C=O)(N(C)C)CCC1 N1(C(c2ccc(NC(C)=O)cc2)=O)CC2CN(Cc3ccc(C#N)s3)C2C1 C1(C(N2C(COC)COCC2)=O)CCC2(CN(C(c3ccc(Cl)cc3Cl)=O)C2)O1 CC(C)(C#CC(=O)NCc1cccc(F)c1F)C.C(=O)(C(O)Cn1cncn1)N N1(C(c2cn(CC)nc2)=O)CCC2CCN(C(C3CCOC(=O)N3)=O)C2C1 c1(N2CC(CC(=O)NCc3cc(C)n(C)n3)OCC2)ncnc2n[nH]cc12 C1(C(N2C(CN(C(C)=O)C3CC3)CCC2)=O)CCCCC1.C1(C=O)CCCO1 C1(C)(NC(C2(CO)CCN(C(C(c3cncnc3)C)=O)C2)=O)CC(C)(C)OC1=O C1(C(N2CCCC(C)C2)=O)CC2(C1)CC1(CCC1)C2.C1(C(=O)N)CC1C(F)F C1(F)(C(=O)NCC(CCNC(C2(CC)CC2)=O)O)CCCCC1 C(=O)(C(C(C)C)NC(=O)C(C1(O)CCCC1)F)NCCc1c(C)ocn1 Cc1ccc(C(C)N(C)C(c2cncnc2C2CC2)=O)c(C)c1 [N-]=[N+]=Nc1cncc(C(N2CCCC(CO)(NC(c3ccoc3Br)=O)C2)=O)c1 C(=O)C(O)CC(F)(F)F.Cc1c(C(=O)NC2(C)CCOC2)nnn1C(C)C.N CC1CN(C(=O)C(C2CCOCC2)=O)CC1CC(=O)NC(C)(C)C(O)CO C#Cc1ccc(C(N2CCN(C(C)C)C(=O)C2)C(=O)NCCCC)cn1 n1(CC(=O)NCCSCC(=O)NC2C(C)(C)CC2)cc(C#N)cn1 C(=O)(C(C)CN(C(=O)CCC1CCC(C)O1)C)NCC(COC(C)C)O Cc1c(CN2CC3CN(C(=O)Cc4ccccc4C(F)(F)F)CC23)cccc1F C=CC1(C(=O)NC(c2nnc(C)s2)C)CCN(C(=O)CC2CC3(CC3)C2)C1 N1(C(C=Cc2cnc(C)s2)=O)CC(NC(=O)C(O)C(C)C)C(C)(C)C1 c1(CC)cc(C)cc(CC)c1CC(=O)OCC1CC(F)(F)C1 C1(C=C)(CC=C)CCN(C(=O)C=Cc2cscn2)CC1.C1(C=O)CCCC(O)CC1 N1(C(c2cccc(OCC)c2)C(=O)NCCCF)CCc2cc(CO)ccc2C1 C1(OC)(OC)CCN(Cc2cccc(O)c2)C1 c1(C(=O)NC2C=CCN(C(C3C(C)(C)CCC3)=O)C2)cnn2cnnc2c1 C(=O)(CN=C(NC1CCCC1)N1CCOC(CF)C1)NCC(C)C Cc1cc(=O)n2nc(CNC3COCc4cccnc43)sc2n1 c1(C=O)ccnc(-n2cccc2)c1.C(C)CCO.C(=O)(C=CC=O)OCC.N C=Cn1nccc1C(=O)NCC(C)(C(C)C)NC(=O)C=CC1CCC1 N1(C(CN(C)C(=O)C2CC2)=O)CCC2(C1)CN(C(C1CCC3(C1)N=N3)=O)C2 N1(C(COCCSC)=O)CCCCCC1CNC(=O)C(C)CC1CCCC1 N1(C(C2CC(C(C)C)C2)=O)CCCC2(CCCN2C(=O)CCc2cn(C)cn2)C1 c1(C(N(C(CNC(CCc2ccnc(C)n2)=O)C)C)=O)cnc(O)n(C)c1=O c1(C(N2CC(C(C)NC(c3oc(CC)c(C)c3)=O)OCC2)=O)c(C)cccc1N C1(NC(COCC(C)C)=O)CC(C(=O)NC(c2ccc(O)nc2)C)=CC1O c1(C(=O)NCC2CCC(NC(C3(Cl)CC3)=O)C2)cc2sc(Cl)cc2s1 c1(C(=O)NC2CCN(C(=O)CC3CCOC3=O)C2)occ2c1CCC2 c1(C=O)ccccn1.C(CC(=O)NCC1(C)CC1)NC(C)=O.C(C)C.N c1(C(=O)NC2CC(C(C)NC(c3ccc(C)cc3C)=O)C2)cnc2cc[nH]c2c1 c1(C(=O)NCC(CNC(CCOCC)=O)CO)cn2c(n1)CC(C)CC2 C1CC2CCC1CC2.CC1(C)CC(C(=O)NCc2cc(C(=O)N)cs2)(CO)C1 C1(C(N(CCNC(C2C(C=C)C2)=O)C2CC2)=O)COCC1C(F)F c1(C(N2CCC(CCNC(C(CC)(C)OC)=O)CC2)=O)cc2c(cc1O)OCO2 N1(C(c2nccc(OC)c2O)=O)CCN(C(C2C(C)C2C)=O)CC(O)C1 C1(NC(CCC(C)SC)=O)CCCCN(C(=O)C2=CCCCO2)CC1 c1(C(N(C2CCCC(NC(Cc3cnc(C)[nH]3)=O)C2)C)=O)cc(Cl)cc(F)c1F c1(CC(=O)NCC(CNC(CC2C(CC)C2(F)F)=O)O)cc(F)ccc1C C1(C(=O)OC)CCN(C(=O)C(C)N(C(=O)Cn2nnnc2C)C2CC2)C1 CC(F)(F)C(F)F.c1(CNC(C2(CC(C)=O)CC2)=O)ccoc1C=O.N c1(C(=O)NCC(CC(=O)Nc2ccc(C)c(C)n2)OC)ccc(C)c(C#N)c1 CCC(C)C(C(=O)NCC1CCC2(CCC2)O1)N(C(=O)CCc1conc1C)C c1(N2CC=CCC(C)(C)C2)ccc(S(=O)(=O)NC2CC2C2CCCCC2)cc1F C1(CCN(C)C)CCCN1C(=O)CCc1cn[nH]c1.N1(CC(=O)N)CC2CC2C1 c1(C(C)OCC)ncc(NC(c2cc(C3CC3)on2)c2nnnn2CC)s1 Cc1c(Cl)sc(Cl)c1C(N1CC(NC(=O)CC2CCCCN2C)C(O)C1)=O C1(CC(=O)N(C(c2ccccc2)CNC(=O)Cc2csnn2)C)C=CCCC1 C12C3CN(CC13)c1cc(ncn1)OC2=O.Cc1ncc(C(C)N(C)C)s1 C1(CC(=O)N)CC(C)(C)CO1.C1(NC(CCNS(CC)(=O)=O)=O)CCCC1 CC1CC(C=O)CCN1C(=O)C=C1CCC1.C1CCCC(C)C1.C(=O)(C)NC C1(C(C)NC(C(CC)SC)=O)CN(C(c2cnn(C3CCC3)c2C)=O)CCO1 Cc1ccc(CNC(=O)C#CCNC(c2occc2C(C)C)=O)o1 C1(CNC(c2c(C)ocn2)=O)CN(C(=O)CC=Cc2ccccc2F)CC12CC2 CC(C)(C)C(CC(=O)NC1C2CCCC1CC2)NC(=O)Cn1c(O)nnc1O C1(NC(CN(C(C)=O)C)=O)COCCC1C(=O)NCC1CC12CC2(F)F c1(C(=O)NC23C(CCN(C(C4(CC)COC4)=O)CC2)C3)cc2cccc(C)n2n1 CC1CN(C(c2ccc(-c3ccccc3)nc2)=O)CC1NS(=O)(=O)C(Cl)(Cl)Cl Cc1ccc(N2CCCC2)c(C(=O)NCC(O)CN(C(=O)CC(O)C(C)C)C)c1 C1(NC(c2c(CC)nccc2)=O)CCN(C(=O)CC2CC2)C(C2CC2)C1 CCC1=NOC(CNC(=O)CC2CN(C(c3cc(O)ncn3)=O)CC2C)C1 C1(N(C(c2c(OC)csc2)=O)C)CCC2CN(C(=O)CC3CCC(=O)NC3)CC12 Cc1ccc(C)c(CNC(C2CC(O)CN2C(=O)CC2CCC(=O)NC2)=O)c1 CN1CCN(c2cc(NC(c3cc(-c4sccc4CO)ccn3)=O)ncn2)CC1 c1(CC(=O)N(C2CN(C(c3nn(CC)c(C)c3)=O)CC2F)C)cc(F)ccc1Cl c1(C(NCC)=O)cc(F)c(F)cc1O.C(=O)(C(C(C)C)NC=O)N1CCCC1.C CC(CN=c1ncc([N+](=O)[O-])c[nH]1)NC(c1ccc2c(c1)CCC(=O)N2)=O c1(C=O)ccc2c(c1)n(C)c(=O)n2C.C(C)(CC)NC(COCCC=C)=O.N C(=O)(CCCCCOC)NC1C(CNC(COCCOC)=O)CCC1 c1(C(CNC(c2csnc2C)=O)NC(CCn2ccc(C)n2)=O)cccc(Cl)c1 N1(C(CS(=O)(=O)N(C)C)=O)CCCC(C2CC2)C1.C1(C(=O)N)COCC(C)(C)O1 O=C(N=c1cc(C2CCCCN2C(=O)Nc2ccccc2Cl)[nH][nH]1)C(Cl)Cl C(CO)(CN=c1ccc(Br)c(S(=O)(=O)N2CCC3(CCCCO3)CC2)[nH]1)N(C)C c1(C(N2CCC(CC=C)(NC(c3cccnc3)=O)C2)=O)ccc2[nH]nc(O)c2c1 c1(C(C)=O)c(C)[nH]c(C(N2CC(NC(c3cnsc3)=O)C3CC23)=O)c1C c1(CN2CC(F)CC(C(=O)NCc3cccc(O)c3)C2)c[nH]c2cc(Br)ccc12 C1(NC(C(CCC)(C)C)=O)CC2(CCCCN2C(=O)CCN2CCCCCC2)C1 c1(C(=O)NCCC2(C(=O)NC3CC(C(=O)OC)C3)CC2)ccn(C)n1 C1(NC(c2cc(C)nn2C)=O)CCN(C(c2cscc2C#N)=O)CCC1CO Cn1cc(NC(C23CC(CN)(C2)C3)=O)cc1C(=O)NCc1sccc1Cl CCS(=O)(=O)CC(C)NC(c1cc(C)c(C)s1)c1nnnn1C1(C)CC1 N(C(=NCCC1CC2(CCC2)CO1)NCC(F)F)CCn1c(CC)nnc1 c1(CNC2C(C(=O)NCc3cccc(F)n3)C2)c(F)cccc1I C=CCC(CC(=O)N(CCC(=O)OC)C)NC(=O)C(C)(C)CCOCC c1(C(CC)(C2CCC2)NCC2CC2c2ccccc2)nnnn1CCCSC C(=O)(C(F)C(C)CC(C)(C)C)N(CCN(C(C1CCC(C)(CC)O1)=O)C)C n1(CCC)nc(C)c(Cl)c1C(N1CCCC(CCO)CC1)C(=O)NC1COC1 n1(CC#C)c(C)cc(C(N2CCC(CNC(=O)CC)C(C)C2)=O)c1C C(=O)(NN1CCC(F)(F)CC1)c1ccc(-c2c(OC)nnc(Cl)c2)cc1 N1(C(c2cc(C)oc2)=O)CCN(C2CCC(NC(=O)COC(F)F)CC2)CC1 N1(C(CC2CC(C)(C)C2)=O)CCCCC(NC(c2cnc(OC(C)C)cn2)=O)C1 C=C(Cl)C(C)(C)C(=O)NC(C)CCNC(c1cc(-c2ccccc2)co1)=O C(=O)(C(C)C1=CCCC1)N1CCN(C(C=CC=CC)=O)CC1CS(C)(=O)=O Cc1c(CNCC2CSC(C(F)(F)F)C2)ccc2c1CCC2 CS(=O)(=O)c1cc(C(N2CCCCC(NC(=O)Cc3ccon3)CC2)=O)co1 C(C(=O)NC1CCCN(C(C)=O)C1)(C(C)OC)NC(CNC(=O)OC)=O Cc1ccnc(-c2cn(CC(F)(F)CNC(=O)Cc3ccc(Br)s3)nn2)c1 N1(C(C#CC2(C)COC2)=O)C2CC=C(C(=O)NC3CCCC34CC4)C1CC2 Cc1ccc(C(=O)NC2CCCN(C(c3cc(N)ccc3O)=O)CC2)c(Br)c1 C(=O)(C(C(C)(C)C)n1cc(C(N2CCCC2)C)nn1)NC(CCCC)COC C1(OCCC)CCCN(C(CCC2CC2C)C(=O)NCC2CCOC2)C1 N1(C(c2c(CC)csc2)=O)CCC2CN(C(=O)COCC(C)(C)C)CC2C1 CC1(CNC(C2(C(N)=O)CC2)=O)CCC(NC(c2sc(Cl)cc2Cl)=O)C1 N1(C(C=CC2(C)COC2)=O)CCCC2(CCCN2C(C2CC(C3CC3)C2)=O)C1 C=C(C(=O)OC(C)(C)C)C(C)(C)C.C1C(C(C)C)C(=O)N1CC1CCC1 Cc1cn(C)nc1C(=O)NC1COCC1CNC(C1(Cl)CC1(F)F)=O N1(C(C(C(C)C)(C)O)=O)CC2(CCCN(C(c3ccc([N+](=O)[O-])c(O)c3)=O)C2)C1 c1(CC)cc(=NCC2C(C)CCCN2C(C2CC3(CCCC3)CO2)=O)[nH]cn1 c1(C(=O)NCCCCC)ccc(CC2CC2)nc1.C(=O)C(C)CC1CCCC1.N c1(OC)cc(O)c(CNC2CCCC2C(=O)NC(C)CF)c(Br)c1 Cc1cc(C(=O)NC2CCC(NC(c3nn(C)cc3Br)=O)C2)ccc1O N(C=CC(=O)C(F)(F)F)C(C1SCCN(Cc2c(OC)ccc(C(C)C)c2)C1)=O C1(C(N(CC(=C)C)C)=O)CCCCC1NC(=O)C(CC1CC1)OC c1(CCC(N2CC(C)(C)C(NC(=O)Cn3nccn3)C2)=O)cnc2n1CCOC2 C(CC(CC)C(=O)NCC1CC1(F)F)=CC.C1(CC=O)CCC(C)(C)CO1 c1(C(N2C3(c4nnc(C(C)C)o4)CCC3CC2)=O)ccc(F)c(F)c1N C(=O)(C(CCF)NC(=O)C=C1CCOCC1)NCc1c(C)noc1 C1(NC(=O)C(c2ccc(F)cc2)O)COC2CN(C(C3(F)CC=CC3)=O)CC12 N1(C(Cc2ccn(CC)n2)=O)CC(OC)CC1CCNC(=O)CCOC c1(-c2cn(Cc3cccc(OC)c3)nn2)cc2ccccc2s1 O=C(CC(O)CNC(c1cncc(Cl)c1)=O)NC(C1CCCC1)CO C1(CN(C)C(C2CN(C3CCOC3)C2)=O)CCC(CNC(=O)C(F)F)CC1 c1(C(N2CCCCC2CNC(C2(O)CCOCC2)=O)=O)cn2cc(F)ccc2n1 CCC(CC)(CO)C(=O)NCCOCCCNC(C1CC(CC(F)F)C1)=O c1(C(N2CCC(CNC(c3c(CC)nco3)=O)C2)=O)cc(N)cc2ccccc12 C(=O)(C1=COCCO1)N1CC(CCC)C(NC(=O)CCc2cn(C)cn2)C1 CN1CC2CN(C(=O)NC3CCc4cccnc4C3)CCN2C1=O C1(NC(C(C(C)C)c2cnc(C)s2)=O)CCC2OCCC2C1 CC1(C)CC(C(=O)NCC2CCCCCC2)CCN1C(=O)CC1CCCC12CC2 c1(C(=O)NCC(C)(C)OCC(=O)NCCc2cncs2)ncccc1F C1(NC(C2C(NC(C(CCOC)OC)=O)CCO2)=O)CCn2nccc2C1 C1(CNC(c2cc(CC)[nH]n2)=O)(CO)CCCN(C(c2ccc(F)cc2F)=O)C1 N1(C(CSc2ccc(C)cc2)=O)CC2CCN(C(C3(C)CC(F)(F)C3)=O)C(C2)C1 CCCCCCC(CNc1ncnc(NC2CCN(OC)CC2)c1C)CC C(C(CNC(=O)CC1CCC(=O)N1C)S(C)(=O)=O)NC(C1CC(C)C1)=O C(CCCCCC(=O)NC(CNC(=O)COC1CCC1)C(C)C)SC c1(C(NCC)=O)cc2n(c1)CCCC2.CC1(C(F)F)CC1C=O.C1CC1.N Cn1ncc([N+](=O)[O-])c1C(=O)NCC(CO)NC(=O)Cc1ccnc(F)c1 C1(C(=O)NCCCOCCNC(CCSCCC)=O)CCCN2CCCC12 N1(C(CC2C(C)=NNC2=O)=O)CCC(N(C)C(c2cc(CO)[nH]n2)=O)C2(CC2)C1 c1(C(=O)NC(N2CCC(C(C)O)CC2)=O)ccn2ccccc12 Nc1cnc(Cl)c(C(N2CCCC(NC(c3ccc(F)c(F)c3)=O)CC2)=O)c1 CC1=C(C(=O)Nc2ccc(C)cc2C)C(c2cn(C)nc2C2CC2)NC(=O)N1C C(=O)(C(F)C(F)(F)F)NCCC(C)CCNC(=O)C(C)(C)CC1CC1 C(=O)(CCC(=O)NC1(C(F)F)CC(NC(c2cnc(C)[nH]2)=O)C1)NC C1(C(=O)OCc2ccc(-c3ccsc3)cc2)CCOC2(CCOCC2)C1 N1(C(C2CCC(CC)CC2)=O)CC(NC(=O)C2=CSCS2)CC2(CCC2)C1 O=C1CS(=O)(=O)CC(C(=O)NC)N1.c1(C(N2CCOCC2)=O)ncc(Cl)cc1F C1(C(=O)NCC(C)(CO)NC(Cc2c(OC)nccc2)=O)CCn2nccc2C1 C12(NC(=O)OC)CCC(C=O)(CC1)C2.C(=O)C1=NOC(C)C1.C(C)C.N c1(CN2CCN(C(C(=O)NC)C)CC2)nc2cc(Cl)ccc2n1CCO C(=O)(C(CO)C(C)(C)C)N1CCN(CCC2CCN(C(C3(C)CC3)=O)CC2)CC1 c1(C(N2CC3CCN(C(c4cnc(CC)[nH]4)=O)C3C2)=O)ccn2c(C)cnc2c1 c1(C(=O)NC(CNc2ncc(C(C)=O)cn2)CC(C)C)ccc(Cl)cc1Cl Cc1cc(F)c(NC(C2CC3(CCN(C(=O)C=CCO)C3)C2)=O)cc1F C(C(CCN=c1nc2scnc2c(NC2CC(COC)C2)[nH]1)OC)OC c1(N2CCN(C(c3ccc(C(N)=O)s3)=O)CC(O)C2)nc2cc(F)ccc2o1 C1(CS(C)(=O)=O)(C(N(CCCC(=O)NC)C)=O)CCNCC1 CC1CC(C(N2CCC(c3nc(C=CC(=O)O)cs3)CC2)=O)CCO1 n1(CC2(O)CN(C(=O)OC(C)(C)C)C2)nccc1[N+](=O)[O-] c1(OCC)ccc([N+](=O)[O-])c(C(=O)NC(C)CC)c1.C(=O)C=O.C(C)C C1(CCNC(C2C3CCCCC23)=O)CC(F)(F)CN1C(c1ncnc(O)c1F)=O Cc1ccnn1C(C)C(=O)NC(C)(C)C1CC1.C(=O)(CCC=CC(C)C)N CCCCC(C(=O)Nc1cnc(C)c(C)c1)NC(=O)Cn1ccc(C)n1 c1(C(C(=O)NC(CC)(C)C)N(c2ccsc2)C)nn(C)c2c1CCC2 O(NC(=O)CCc1cnccc1OC)CC(=O)NCCC=CC C(CCC)(CC(=O)N1CCOCCC1C(C)C)NC(CCC=CCC=C)=O c1(OC)cccc(C(=O)NC(C)CCN(C)C(C2CCNC2=O)=O)c1 CC(CN=c1[nH]cnc(Cl)c1CO)N(C(=O)CCc1cn[nH]c1)C N1(C(C2(CCC)CC2)=O)CC(C)OC2(CCN(c3ccc(C#N)nn3)C2)C1 C(=O)(C(C)(C)C(C)C)NC(CCNC(CCOc1c(CC)cccc1)=O)C c1(C(=O)NC2C(NC(CC(C)CF)=O)CCCC2)cc2c(cc1F)NC(=O)CC2 Cc1ccc(CC(=O)NCC2C(C)CCN2C(=O)CO)cn1 C=CCC(CC)C(=O)NCC1CCCCCN1C(=O)CN(c1ncccn1)C c1(CC(=O)NCC(CO)NC(=O)CCN2CCCC2)c[nH]nn1.C1CCCO1.C C1(CC(=O)N(CCCNC(=O)CCn2ccnn2)C(C)C)CCCN1C CC1(NC(C2CCC(C)CC2)=O)CCN(C(=O)CCF)C1 CC(C)C(F)C(=O)N(C)CCNC(=O)C(C)NC(C1CCCCC1)=O CCCCCCCNC(=O)CC(C)CNC(=O)CC1CCC(=O)N1 c1(OC)ccccc1CN(C)C(C1CC2CC1(C(=O)O)C2)=O C1(NC(C(C)Oc2cccc(Cl)c2)=O)CN(C(=O)C2=CCCO2)CCC1C c1(C(=O)Nc2c(C)nn(C(C)C)c2)cc2cc(Br)cnc2s1 Cc1nc(C2CC2)ncc1C(N1CCCC1(C)CNC(=O)C(C)N1CCC1)=O C1(NC(CN(C)C)=O)CC(NC(c2ccc(SC(F)(F)F)cc2)=O)CC1O C(=O)(C(C)(CC)CO)N1CC(O)(CN(C(C(C)OCC=C)=O)C)C1 CCC#CC(C)(C)NC(C1CCCCC1CNC(c1cncc(Cl)c1)=O)=O CC(CN(C)C)CCC(=O)N(CCC(=O)N(C1CCC(F)(F)CC1)C)C Cc1[nH]c(C#N)cc1C(N1CCOC(C(=O)NCC23CCCC(CO2)C3)CC1)=O C1(NC(C2C(COC)CC2)=O)CN(C(C2SCC=C2C)=O)CC1C Cc1ccccc1CNC(=O)CC1CN(C(C2CCCOCC2)=O)CC1C CN1CCC(=O)NC2CN(C(=O)NCc3cccc4c3CCCC4)CCC12 c1(C(N2CC3C(C(=O)NC(COC(C)=O)CO)(C3)C2)=O)cn2ccccc2n1 N1(C(Cc2nc(C)sc2)=O)CCCC(NC(c2ccc(CN(C)C)nc2)=O)C1 N1(C(Cc2nn(C)c(C(F)(F)F)c2)=O)CCC(F)C(NC(C2COCCO2)=O)C1 c1(NC(CC2CCN(C(C3C(C)(C)C3)=O)CC2)=O)cc(F)c(Cl)cc1Cl O=S(=O)(c1ccc(NCCC2CC(O)C2)cc1Cl)NCC1CN2CCN1CC2 C#CCCN=C(NCCc1nnc(C)s1)NCC(c1cc(C)cc(C)c1)O c1(CC)nc(N2CC=C(CNC(=O)C=Cc3ccc(C)cc3)CC2)[nH]c(=N)n1 c1(C(N2C(CNC(c3nc(C)n(C)n3)=O)C(C)CC2)=O)csc2c1CCCC2 c1(OC)c(F)cc(C(=O)N(C)CCN(C(=O)CC2CCOCC2(C)C)C)cc1Cl CC(C(=O)N1CCC(CO)(CNC(C2CC(F)(F)C2)=O)C1)C(F)(F)C(F)F C1(NC(c2cccc(Cl)c2)CC)CC2(COC(C)(C)C2)C1 c1(COC)nccc(=NCC2CN(C(c3sc(C(C)C)nc3C)=O)CC2(C)C)[nH]1 c1(C(C)C)nc(-c2nc[nH]n2)sc1C(=O)NCCNC(=O)C(O)c1ccsc1 c1(-c2cc(CC(=O)NCC(C)C)no2)ccccc1Cl.C1(C(=O)N)C2COCC12 C1(O)(C(C(=O)N(CCN2CC=CC2)CC)F)CN(C(C2CCOC2)=O)C1.C C(=O)(CC(CNC(=O)CCCC1CCCO1)C1CCC1)NCC c1(NC(c2cccnn2)C)nccc(N(C)Cc2cnccn2)n1 CS(=O)(=O)C1CCCC1C(=O)NCC1(NC(=O)CCCCO)CCCCC1 N1(CC)CC(NC(=O)C(=O)NC)CC1=O.C1CCN(C(=O)CCC2CCC2)C1 Cn1cc(CC(N2CCCC2CNC(c2cnn(C)c2Cl)=O)=O)c2ccccc12 C=CCC(CC)C(=O)NCCC1(O)CCCN(C(=O)Cc2ccccc2Cl)C1 C1(NC(C(=CC2CCCC2)C)=O)C2CC1CN(C(=O)CC1CSCCS1)C2 CC1=NOC(C(=O)NC(C)C(CO)NC(=O)C(C)OC2CCCCC2)C1 N1(C(c2ccc(C)s2)=O)CCOC2(CCN(C(C3CCCCC3C)=O)CC2)C1 C1(CCNC(C(C=CC)O)=O)CCCCN1C(=O)Cn1ccc(Br)n1 N1(C(=O)Cn2nccn2)CC2CN(C(=O)CC3CC34CC4)CC(F)(F)C2C1 C(c1cc(F)cc(F)c1)=CC=O.CC(C)(C(=O)NC1CC1C)C1CCCC1 N1(C(C2(C(N)=O)CC2)=O)CCC(CC(=O)Nc2cc(-c3ccccc3)no2)CC1 Cc1cnnc(O)c1C(=O)NC(C)CCC(=O)N(C)CCC1CCCC1 C=C(C)CCCC(=O)NC1(C)CCCN(C(C2CCC2(OC)OC)=O)C1 Cc1cccc(C(=O)NC2CCCN(C(c3n[nH]c(C(C)C)c3Br)=O)C2)c1O c1(CC(N2C(C(=O)N)CCC2)=O)cnc2c(=O)[nH]ccn12.c1(C(C)=O)ccccc1 CCCCCCNC(=O)CCOCC1CC1.C1(C(=O)N)CCS(=O)(=O)C1 C1(NC(CC2CCC(C)CC2)=O)C2COCC1CN(C(=O)C(C)(C)O)C2 N1(C(C(C2CCN(C(=O)C=Cc3cn(C)cn3)C2)C)=O)CCN(C)C(C2CC2)C1 C1(CNC(c2cn(CC=C)nc2)=O)CN(C(=O)CC2CSC2)CC1C C1(C(=O)NCC2CCN(C(CCN(C)CCO)=O)CC2)CCc2cnn(C)c2C1 C#Cc1ccc(C(=O)NC(C)C(C)NC(=O)CCC2CCCC(O)C2)cc1 Cc1ccc(NC2CCC(c3ccccc3)CC2)cc1F C1(F)(C(=O)N)CC=CCC1.c1(C(=O)NC2CC(C)C2)cccc(C2CC2)n1 c1(CC(N2CCCC(NC(C3(C)CC=CCC3)=O)C2)=O)nc2ncccn2n1 C(=O)(CCOC1CN(C(=O)Cc2cnsc2)C1)NCCN(C)CC N1(C(c2c(C)sc(CC(F)(F)F)n2)=O)CCCC(NC(=O)C(O)C(C)C)CC1 C1(NC(c2c(SC)scc2)=O)CCC(F)(CNC(c2cc(O)ncn2)=O)C1 N1(C(c2c(C)nc(C)o2)=O)CCC2(CCC2)C1.c1(C=O)cc(Cl)c([N+](=O)[O-])[nH]1.N N1(C(C(CCC)O)=O)C2CC1CN(C(=O)C(C)NS(C)(=O)=O)C2 C(=O)(C1=CCC(C)(C)CC1)NC1(C(N2CC3CC(C)C3C2)=O)CCSC1 N1(C(C2C(C)CCC2)=O)CCC(CCNC(=O)COc2cccc(Cl)c2)CC1 C1(C(C)NC(C2C3CC4C(C3)C24)=O)CCN(C(C2CC(C)(C)O2)=O)CC1 C(=O)(C1=NN(c2cccc(F)c2)C(=O)CC1)NC(c1ccccc1C(F)(F)F)C C(CCC(C)(C)C(=O)NC1CN(CC)CC1(C)C)NC(CCN(CC)CC)=O c1(N2CC=CC(NC(c3cc(=O)cc(Cl)[nH]3)=O)C2)ncc2c(n1)COC2 C1(C(N2CCC(O)(CN(C(CN3C(C)CCCC3)=O)C)C2)=O)CCCC2(CC2)C1 c1(C(=O)NCC(CNC(C2CCCN(C(C)C)C2)=O)(C)C)cc(F)cc(Cl)c1 CCCC(CNC(c1cnccn1)=O)C(=O)N(CC(O)CN(C)C)C c1(CCC)c(C(=O)N(C2CCN(C(C3CCOC3)=O)C2)CC)nnn1C C(CC(O)C(=O)NC1(C2(C)CCCN2C(=O)C(F)CC2CCCCC2)CC1)SC C(CNC(c1sccc1-c1ccccc1)=O)(C(C)C)NC(COC(C)C)=O N1(C(c2ncc(C)c(Br)c2)=O)CC=C(CCNC(C2CCCC2O)=O)CC1 c1(C(C(=O)N(C(CSC)C)C)CN)ccc(C)cc1 n1(CC)ncc(C(=O)NCC(CO)Nc2ncncc2Br)c1C c1(OC)cc(C(=O)NC2CC(C)C2)c2c(c1)CCCC2.C(=O)C=C(C)Cl C1(C(N2CC(NC(C(CC)(O)c3ccccc3)=O)C2)=O)CC12CCSCC2 C(N=c1[nH]c(CNC(C)CC(C)C)nc(=N)[nH]1)C1(SCC)CC1 c1(NCc2cc(C)cc(C)n2)ncc(S(=O)(=O)N2CCC(N3CCC3)C2)cc1Cl C1(NC(C(c2n(C)ccn2)(F)F)=O)CCN(C(c2cncc(C#N)c2)=O)CC1F c1(CC)cc(C(N2CC(C)C3CC23)=O)c(C)nn1.c1(CC(=O)N)ccccc1Cl C12(NC(C(CC)=CC)=O)CCC1CN(C(c1cn(C(C)C)nn1)=O)C2 Cc1ccc(C(C)NC(c2cc(CNC(=O)CCN(C)C)on2)=O)o1 C1(C(=O)NCc2cc(Cl)ccc2Cl)Cc2cc(Cl)cc(Br)c2O1 CC1(CNC(c2ccccn2)=O)CCC(NC(=O)Cc2cccnc2)C1 c1(C(=O)NCC(C)NC(=O)CCCN=[N+]=[N-])ccc2c(c1)OC(C)(C)C(=O)N2 N1(C(C(C)(C)OCC)=O)CC(NC(=O)C(c2ccc(O)cc2C)C)CC(F)C1 C1(C(=O)OC)Cc2ccc(F)cc2N1C(C1CCC(C)O1)=O c1(OC)cccc(CN2CCCC2(C)C(=O)NC(c2ccno2)C)c1O Cc1csc(NCC(=O)NC(C)(C)CN(C(=O)CC2CCCC2O)C)n1 N1(C(C2CCC(n3cc(C4(COC)CCCO4)nn3)C2)=O)Cc2nc(C)sc2C1 C1(C=O)CC(N=[N+]=[N-])C1.c1(C(N)=O)ncn(CC(=O)NCC2CCCC2)n1.N N1(C(C(C)C)=O)CC2CC2(CNC(C2(n3cc(Br)cn3)CC2)=O)C1 c1(C(=O)NCC(C)(C)NC(C2C(C)OCCC2)=O)c[nH]c2ncccc12 N1(C(C(CC)C)=O)CCc2c(c(CNC(=O)CC3C=NN(C)C3=O)nn2C)C1 C(=O)(CCC(=O)NCCCOCCC(=O)NCCC1CCCO1)N(C)C CC(C)CC(C(=O)NC(C)(CNC(c1ccc2cncn2c1)=O)C1CC1)C(C)C C(CC(C)C)(C(C)(C)C)NC(c1ccc(OC)nc1F)=O C1(C(N2CCN(C)CC2)=O)CCC2CC(C)CN2C1.N1(CC)CCC1C(=O)NC CCC(CC(=O)NCCN(C(c1n[nH]c(C)c1F)=O)C(C)C)C1CCC1 CC1OCCOC1C(=O)N(C1CCOCC1)CCF CCCN(OC)C(=O)C1CCN(C(=O)Cn2nc(C)cc2C)CC1C C(=O)(C(CC)O)NCCN(CCC)C(C1CC(C=O)C1)=O.c1ccccc1 C1(C(N2CCCCC2CNC(C23CC(CO2)C3)=O)=O)CCc2nn[nH]c2C1 c1(C(N2CCCC(NC(C(C)(C)SC)=O)C2C)=O)ccc2cc(C)ccc2n1 C1(NC(C(C2CCOCC2)C)=O)CCCC1CC(=O)N(C)C(c1nccs1)C Cc1cc(C)c(C(=O)NC2(C3CCCN3C(c3cc(SC)oc3C)=O)CC2)cn1 CC(C)(C(=O)N1CCC2CN(C(=O)C=Cc3ccc[nH]3)C2C1)S(C)(=O)=O C=CCN=c1[nH]cc(C(=O)NC(C)(C)CNC(=O)CCC(CC)CC)s1 C1(C)(NC(C2CN(C(C)C)C2)=O)CCN(C(=O)CC2CCCOC2)CC1 N1(C(C(C)CN(C)C)=O)CC2CCN(C(=O)CCCN3CCCCC3)C2C1 C(=O)(C1=COCCO1)N1CCC(C(CNC(C2(OCC)CCOC2)=O)(C)O)CC1 O=C(C1=NOC(c2ccccc2)C1)N1CCC(CNC(C2(O)CCSCC2)=O)C1 C1(N(C(=O)CCOC)CC)CCN(C(=O)C(C)(C)Oc2ccccc2)CC1 Cc1coc(C(C)C)c1C(=O)NC1CCCC1.C1(CC=O)NC(=O)NC1=O.C c1(C(=O)NCCC2CN(C(=O)CSC3CC3)C2)ccc(F)s1 CC(C)CC(O)C(=O)NC(CCN(C)C(c1c(Cl)cncc1Cl)=O)C(C)C C1(C(=O)NCc2nc(C3CC3)no2)CCCCN1C(=O)C(O)CO CCC(C)(C)C(O)C(=O)N(CCC(N1CCNC(=O)C1CCO)=O)CCO C1(CC(=O)NC(CC)CNC(c2cn(CC)nn2)=O)CCC2(CCOCC2)CO1 c1(C(C(=O)N(CCNC(COCCSC)=O)C2CC2)=O)cccn1C c1(CC(C)NC(=O)CCN(C(=O)CC#N)CCCO)nccn1C Cc1nc2cc(C(N3C4CCC3(CNC(C3C(C)C3C)=O)CC4)=O)c(F)cc2[nH]1 n1(CC(N2CC=CCC2)=O)nc(C)c2cccnc12.C(C(=O)N)(C(C)C)SCC CCC(C(=O)N(CC(=O)NCCN=[N+]=[N-])C)N(C)C C1(C)(CC)CC(NC(=O)C2=CCCC2)CN1C(c1ccc(OC)nc1C)=O N1(c2c(C#N)cncn2)CCC(C2(CNC(=O)CCC3CCCCC3)CC2)CC1 c1(C(=O)NCC2C3CN(C(c4nc(C)n(C)n4)=O)C2C3)cc2n(n1)CCCC2O N1(C(C(c2ccccc2)OC)=O)CCN(C(=O)Cc2nnc(C)s2)CC1C(F)F C(C(C(=O)N)C(C)(C)C)NC(C1CN(C(C)=O)C1)=O.C1CC(F)(F)C1(C)C C12(CC13CCC3)C(=O)N2.C(CC#CCO)SCC(=O)NCc1cn[nH]c1 C(C)(N=c1[nH]c(=NCC2(C)CC2(Cl)Cl)c2c(F)cccc2[nH]1)c1ccnc(C)n1 Cc1cncc(C)c1C(=O)NOCC(=O)NCC1CC(O)C1(C)C C1(NC(c2c(CC)ccs2)=O)CC(C)N(C(c2cncn2C)=O)C1 c1(CC)oncc1C(=O)NC(Cc1ccccc1)CCNC(C1(F)CC1)=O C(=O)(C1CS(=O)(=O)c2ccccc21)N1CC2N(C(CCC(=C)C)=O)C(CCC2)C1 C12(C(N(CCN(C)C)C)=O)CCN(C(c3ncccc3C)=O)CC1C2 N#Cc1ccc(C(=O)NCCCOCCCNC(C2CCCCC2O)=O)s1 C(=O)(C(CN(C)C)C(C)C)NC(CC)CN(C(=O)C(CSC)OC)C c1(C(N2CC3C(NC(C4=C(C)OCC4)=O)(C3)C2)=O)cnc(O)c2cnccc12 C#Cc1cc(C(N2CC(C(=O)N(C)C(c3ccco3)C)C(F)(F)C2)=O)ccc1C CCC(C)(C(=O)NCCC1(NC(c2ccn3nccc3n2)=O)CC1)C(N)=O OC(CCO)(C(F)(F)F)c1nccn1Cc1ccccc1 C#CCC(C(=O)NC1CCCNC1=O)NC(=O)C1=COCC1 c1(Cc2onc(C(CC)Oc3ccc(F)cc3)n2)cccc(OC)c1 c1(C(=O)O)cc(S(=O)(=O)N2CC(NCc3nccs3)C3(CC3)C2)ccc1F C1(C(=O)NC2(CC=C)CN(C(=O)CC(Cl)Cl)C2)CCS(=O)(=O)C1 C1(NC(C(C=C)O)=O)CCOCC1C(=O)NCC1CC(C(=O)OC)C1 c1(C(=O)NCCCC(C)NC(C2CCC(=O)O2)=O)cc(Br)sc1Cl C1(C(=O)NC(C2CCN(C(=O)C(C)C(F)F)C2)C)CCCC(=O)N1C C=C(C)C(C)(C)C(=O)N1CC(CNC(C23CC2CNC3=O)=O)C2(CC2)C1 C(=O)(C1=COCCO1)N(CCCCCC)CCNC(=O)CC1OCCC1C N1(C(=O)CN2CCSCC2)CCN(C(=O)C(C2CCCC2)C2CCCC2)C2CCC12 CC1CCCC1(C)C(=O)N(C1CCC(n2nnnc2O)CC1)C N1(Cc2cnc(C(C)C)s2)Cc2[nH][nH]c(=NC(=O)c3ccnc(C(F)F)c3)c2C1 n1(CC)cnc2c(NCc3cccc(O)n3)[nH]c(=NCC3(C)CCCCC3)nc12 c1(CN2C(CCC(=O)Nc3c(Cl)ccc(OC)c3)CCC2)cc(C)c(C)cc1C N1(C(c2n(CCC)ccc2)=O)CCCC(N(C(=O)CCc2nccs2)CCO)C1 c1(C(=O)NC(C2(CNC(CCOCC#C)=O)CC2)C)ccc2nc[nH]c2n1 C1(C2CC2)(C(N(C2(C(NOCC(=O)OC)=O)CCC2)C2CC2)=O)CC1 C1(NC(c2c(C)csc2)=O)CC2CC(C1)N(c1ncnc(Cl)c1CO)C2 c1(C(=O)NCC2(OC)CN(C(C(C=C)(C)O)=O)C2)c(F)ccc2c1OCC2 N1(C(C(COC)N(C)C)=O)CCC(C(=O)NC2(c3noc(C)n3)CC2)C12CC2 c1(OC)ncc(Cl)c(=NC(CNC(c2cc3cc(Cl)ccc3o2)=O)C(C)C)[nH]1 C12(COC)CC(NC(=O)C(C)CF)(CN1C(c1ccc(C)cc1)=O)C2 Cc1cc(NC(C2(CO)CCCC2)=O)ccc1NC(c1nscc1C)=O C1CN(C(=O)C)CC1C(F)(F)F.c1(C=O)cnn(C2CC2)c1.C1CCOC1.N n1(CC)cnc2c(NCC3C=CCC3)nc(N3CCc4cc(F)ccc4C3)nc12 c1(C(=O)NC2CC2C(=O)N)ccc(Br)c2ccccc12.c1(CC)cccc(F)c1 c1(C(=O)NC2CC(O)(CNC(C(C)C(F)F)=O)C2)ccc2c(c1)OCO2 N1(C(CCCC#CC)=O)CC2CC(NC(c3sc(CO)nc3C)=O)CC2C1 Cc1nc(C2CC2)oc1C(N1CC(C(F)Cn2cc(-c3cncn3C)nn2)C1)=O C(C(C)C(=O)NCCC(C)NC(=O)CC1COCCO1)OC c1(C(=O)NCC#CCNC(c2ccsn2)=O)cc(C(F)(F)F)c[nH]1 c1(OC(=O)OCCNC(C(C)O)C)cccc(C(F)(F)F)c1 N(C(=NCC1CCNC(=O)C1)N1CCC(C(=O)NC2CC2)CC1)CC(C)(C)C N1(C(CN(CC)CC)=O)CC2(CCN(C(=O)C(C(C)(C)C)N(C)C)CC2)C1 N1(C(C=C(C)Cl)=O)CCC2(CC1)CN(C(C1C(C)C1(F)F)=O)C2C(C)C C(=O)(C(C(C)(C)C)OC(C)(C)C)NCCCC.c1(C=O)cccc(Cl)c1N.N C1(C(=O)NC2CC(CCNC(C3CC=CCC3)=O)C2)CC2CCC(C1)S2 c1(C(=O)NCC2(C)COCCO2)cc2cc(Cl)cc(Br)c2o1 C(=O)(C(CC(C)C)N(C)C)NC(C(CO)NC(CCCCOC)=O)C c1(CCC(=O)NC2(CCNC(C3CC4(CSC4)C3)=O)CC2)c(F)cccc1Cl C1(OC)CC(C)CN(C(=O)C(C)N(C)C)C1.C1(C)(C(=O)N)CC(=O)N(C)C1 CC(C)(CNC(c1n[nH]c2c1CCC2)=O)CC(=O)N1CCCC(CO)CC1 N1(C(CC2(CNC(C3SCCS3)=O)CC2)=O)CCCC1c1ccon1 c1(OC)c(C(=O)C(=O)NCC(C)C2CCC2)sc2ccccc12 c1(NC(=O)CN2CCC(F)(c3ccc(F)cc3)C2)nc2ccc(F)cc2s1 O=S(=O)(c1ccc(N2CCC(O)CC2)c(F)c1)NC1CCCOC12CCC2 N1(C(=O)OC(C)(C)C)CCC(C)(NC(=O)CSC2CCCCO2)C1 C1CC2COCC(C1)N2C(=O)C(C)CC1CC1.c1(OC)ncc(C)cc1C=O.N Cn1c(C(=O)NCCOCC2CCC2)ccc1[N+](=O)[O-] C(=O)(C(F)CCC(C)(C)C)N1CCCC(NC(c2c(C)cnnc2O)=O)C1 CON1CCC(C(N2CC(NC(=O)CC(C)n3ccnc3)CC(C)C2)=O)CC1 C12(C(=O)NC3(CNC(C(CC)O)=O)CCOCC3)CCC(OC)(CC1)CC2 O=C(C#CC1CCCO1)NCCNC(C1(n2cccn2)CCCC1)=O c1(C(=O)NC2C(NC(=O)CC3CCOC3=O)CCC2)ccnc(OC2CC2)c1 c1(C(N2CCC(C(C)NC(CC=CCC)=O)C2)=O)ccc(C(F)(F)CF)cc1 N1(C(C)=O)CC2CN(C(=O)CCn3cc(-c4cc[nH]n4)nn3)C(C34CC(C3)C4)C2C1 N=c1cc(C(=O)NC(CNC(C2CCOCC2)=O)C2CC2)nc(Cl)[nH]1 CCCCC(CNC(=O)C(C#N)=CC(C)C)NC(=O)C(F)(F)c1cncs1 Cn1nc(C(=O)NCC2COCC2NC(C2C=CC=CC=C2)=O)c2ccccc12 c1(NC(C2C3CC2N(C(c2cccc(O)n2)=O)C3)=O)nc(Cl)cnc1Br N1(C(c2c(CC)n(C3CCCC3)nc2)=O)CC2CC1CN2C(C1CC(C)(O)C1)=O Cc1cc(C(N2CC(F)CC2C(=O)N(C)Cc2ccsc2)=O)c(C)[nH]1 c1(C(N(C2CN(C(C3CCCO3)=O)C2)C)=O)cc2c(F)c(F)c(F)cc2[nH]1 c1(C(=O)NC2C(CC)CN(C(=O)CCC(C)C)CC2)ccc2nc(=N)[nH]n2c1 c1(C(N2CCC3(CCC(O)C3)C2)C(=O)NCCCOC)cc2ccnc(Cl)c2s1 N1(c2nc(C)c(Br)cn2)CC(C2CCCCN(C(c3ccoc3)=O)C2)C1 N1(C(c2cccc(C#C)c2)=O)CC(C)CN(C(=O)CCOCCOC)C(C)C1 Cc1cc(Br)cc(C)c1C(=O)NC1CC(NC(C2CCC2(C)C)=O)C1 Cc1cc(N2CCOC(C3CCC3)C2)nc(=NCC2CCC23CCOCC3)[nH]1 N1(C(C2(CC=C)CCN(C(=O)C(C)=CC(C)(C)C)C2)=O)CC(C)C(C)C1C c1(C(C)C)cc(C(=O)N)ns1.C1(C(N(CC)C(C)C)=O)OCCC1C(C)C CCCC(O)CCN=c1[nH]c(=NCCn2cc(CSC)nn2)[nH]c2c1CCCC2 CC(=O)CCCC(C)C(=O)NC1C=CC(CC(N2CCCCC2CO)=O)C1 C1(CNC(c2ccn(C)n2)=O)C2CN(C(=O)CC3CCNC(=O)C3)CC12 C1(NC(c2c(C)csc2)=O)CCC2CCN(c3cc(=O)n(C)c(O)n3)C1C2 c1(CC(=O)OC)ccccc1NC(c1cncc(-c2cnn(CCC#N)c2)n1)=O n1(CC)cnc(C(=O)NCC2CC2)c1.c1(C=O)csc(-c2cccs2)n1.C N1(C(C(COC)OC)=O)CC=C(CC(=O)N(C(C)C(N)=O)C)CC1 N(C(=NCC1CCOC1)NCC1CCCO1)Cc1c(C)ncs1 C1(NC(C2CC(SC)C2)=O)COCCC1NC(=O)C=Cc1scnc1C N1(C(C(CCO)N(C)C)=O)CC(C2CN(C(C3CS(=O)(=O)CC34CC4)=O)C2)C1 CC1(C(=O)NCC(c2ccccc2)NC(c2n[nH]cc2Cl)=O)CCCNS1(=O)=O Cc1cc(C(=O)NC2CCCC2(C)NC(=O)CC2CCCO2)cc(F)c1 N1(C(CC(C)O)=O)CC2(C1)CN(C(c1ccc(C(C)(C)C)cc1)=O)CC2C(=O)O C=CCC(C)(C)CC(=O)NCCC1CC1.c1(C(=O)N)ccccc1.C(=O)N C(C)(CC(=O)NC(c1ncc[nH]1)C)NC(C1CC(CC)C1)=O C(=O)(C(C)(C)C(=O)NC1CCCC(NC(=O)C(C)CCCOC)C1)NC C1(CNC(c2c(CC)ocn2)=O)C2CN(C(C3C(F)(F)C34CC4)=O)CC12 C1(C(N2C(CNC(C3C4CCCC34)=O)CC2)=O)CC2(C1)CC1(CCC1)C2 c1(C(N(CC(C)CNC(c2cnsn2)=O)C)=O)ccccc1CCC(F)(F)F C1(c2cn(CC(C)NC(C3CC(F)(F)C3(C)C)=O)nn2)CCC(F)(F)CC1 c1(OC)cccc2c1C(C(=O)N1CCN(C(c3ccon3)=O)CC1)CC2=O Cc1ccc(NC(C)C(N2CC3C(NC(c4c[nH]c(C)c4)=O)C3C2)=O)cc1 c1(C(C=O)(C)F)ccc(F)cc1.C(C)(C(=O)NC1(CC)CCC1)OCC.N CC1(C)C(C(=O)NCCC2COCCN2C(=O)C(=O)N)C1(C)C.c1ncc[nH]1 N1(C(CCC(C)SC)=O)CCC(C2CCCN(C(=O)CC(F)F)CC2)CC1 c1(C(C2(C(CC)C)CC2)NC(CC)C2CCC2)nnnn1CC1CCOCC1 c1(C(=O)NCC2N(C(C(C)P(C)(C)=O)=O)CC2)cccc2nc(O)n(C)c12 C1(CNC(c2nn(C)c(=O)cc2)=O)CCCCN(C(c2csnc2Cl)=O)CC1 c1(C(=O)NCC2(NC(C3C(C)C3C)=O)CCC2)ccc(=O)n(C)c1 C1(CNC(COCC(=C)C)=O)CN(C(c2cccnc2)=O)CCO1.CCCC.S C#Cc1ccnc(C(N2CCC(C(N3CCCC(CC)CC3)=O)C(C)C2)=O)c1 C1(C(N2CCC(Cc3cn(-c4cccc(OC)c4)nn3)C2)=O)CCCCC1(C)N C(CC)(CCCC(=O)O)NC(c1ccc(Cl)cc1)CCCC N1(C(c2c(N)c(F)c(Br)c(F)c2)=O)CCCC2CN(C(=O)CCF)CCC12 c1(C(N2CCC(C)C(NC(=O)COc3cn[nH]c3)C2)=O)c[nH]c2cc(F)ccc12 CC(C)(C)C(CO)C(=O)NCC1(NC(c2cc(O)ncc2F)=O)CCCCCC1 c1(CN(C(C(=O)NC2CCOC2)c2nccs2)CC)cccs1 c1(NC(=O)NCC(C)C(F)C(=O)O)c(Cl)ccc2ncccc12 Cc1cc(O)nc(CNC(=O)CC2CN(C(=O)CCNC(N)=O)CCO2)n1 c1(OC)ccccc1C(C)C(=O)NCC1CCCN1C(=O)C(C)SC(F)(F)F c1(OC)ccc2c(c1)CCCN2C(CC1(C#N)CCC1)C(=O)NC1CC1 C1(NC(C2(CC#C)CCN(C(C3CC(C4CC4)C3)=O)C2)=O)CC2(CCC2)C1O C1(CC(C)C)(C(=O)NCC(C)(CO)NC(=O)CN2CCOCC2)CCNC1=O N1(C(=O)Cc2ncncc2Cl)C2CCC1CN(C(C1(Br)CC1)=O)C2 CC(C)S(=O)(=O)CC(=O)NCC(CO)NC(=O)Cc1ccccc1CC(N)=O N1(C(C2C(C#N)C2)=O)CCC2C(C1)CN2C(c1cnc2cccnn12)=O O=C(CCCCCF)N1CC2CC2(CNC(C2(Cl)CC2(F)F)=O)C1 N1(C(CCc2nc(C)c(C)[nH]2)=O)CCOCC(NC(=O)C(=Cc2c[nH]cn2)F)C1 CC1(C(=O)NCCCc2cnccn2)CCSCC1 N1(C(CCCOCC)=O)CC(CNC(C2(C)CCN(C)C2)=O)OC(C)(C)C1 c1(C(N2C(C)C(C(=O)NOCC3CCCC3)CC2)=O)c[nH]c2nccc-2c1 C1(NC(c2c(OC)ccs2)=O)CC(F)(F)CC1NC(=O)CP(C)(C)=O c1(CC(=O)NC(C)CCCNC(C2OCCN(C)C2=O)=O)ccc2ocnc2c1 Cc1cccc(Cn2nc(-c3ccoc3C)nc2C2CC=CCC2C)n1 C=CCC(C)C(=O)N1CC(O)(CN(C(=O)C=CCOC)C)C1 C=C(Cl)CC(C(=O)NOCCCCC1CC1)NC(=O)CC(C)SC N1(C(C(CC(=C)C)OC)=O)CCCCC2(CCN(C(=O)CC(C)(C)C3CC3)C2)C1 C(N(C)N1CC(C(F)(F)F)CC1C)c1onc(COCC)n1 C(N=c1[nH]c(=NCC2OCCC2(C)C)[nH]c2ccccc12)C1(CCOC)CC1 N1(C(c2cc(C)ns2)=O)CCN(C(=O)CCSC(F)(F)F)C2CCC12 CCC(CC(C)C)C(=O)N1CCC1c1cn(-c2cc(C)cc(F)c2)nn1 n1(CC)ncc2c1CC(C(N1CCC(C)(CNC(c3ccccc3)=O)C1)=O)CC2 CC1CN(C(c2cn(C)[nH]c2=N)=O)CC1NC(=O)CC1C=CCCC1 C(=O)(CCCCCNC(C1CC(C#N)(OC)C1)=O)N1CC(C)(OCC)C1 c1(OC(F)F)cccc(NCCC2CC3(CCC3)C2)c1 c1(C(N2CC(NC(CNC=O)=O)C(C(F)F)C2)=O)ccnc2[nH]c(O)nc12 N1(C(Cc2scc(C)c2)=O)CC2CCC2(NC(c2ccc(C)s2)=O)C1 C(CN=c1[nH]c(=NCCCP(C)(C)=O)[nH]c2cc[nH]c12)SCC CCC(C)C(C(=O)OC)Sc1c[nH][nH]c1=N Cc1ccc(F)c(C(=O)N(CCC(=O)NCC(CO)CC(C)C)C)c1 C1(NC(CCC)=O)CCC2(CC1)CN(C(=O)C(COC)NC(C)=O)CCO2 C(=O)(CCCCCN(C)C)N1CCC(C)C1.C1(CC(C)C)(C(=O)NC)CCCC1 CC(C)(C)C(CNC(C1(O)CCCC1)=O)C(=O)NCC(C)(O)C1(C)CC1 C1(NC(Cn2nnc(C)n2)=O)CCC(C)N(C(C2(C3CCCO3)CCC2)=O)C1 C1(C(NOCC=C(C)C)=O)COCC1NC(c1n[nH]c(C)n1)=O Cc1ccc2[nH]cc(CCC(=O)NC(C)CCN(C)C(=O)OC(C)(C)C)c2c1 c1(C(=O)OC)cc(NC(C2CC2C(=O)Nc2ncc(C)cc2Cl)=O)ccc1F CC(C)CC(C)CC(=O)NCC1(C)COCCN(C(c2cn(C)ccc2=O)=O)C1 CC1Cc2cc(CC(=O)NC(C)CNC(=O)C(O)c3ccsc3)ccc2O1 C(=O)CCS(C)(=O)=O.CC1(CC(N2CCCC2)=O)CN(C=O)C1.C(C)(C)C.N Cc1ccc(CC(N2CC=C(CNC(=O)C(F)OC(F)(F)F)CC2)=O)c(Cl)n1 c1(C(N2CC(NC(C=C(C)c3ccsc3)=O)C2)=O)cc(N)cc(O)n1 C1(C(=O)NCCOCCC=C)(NC(=O)CCC2CCCC2)CCCCC1 C(=O)(C(C)(F)C(C)(C)F)N1CC2C(N(C(=O)Cc3c[nH]nc3O)C)C2C1 C1(C(N(CC(C)N(C)C(c2cc(C3CC3)on2)=O)C)=O)CCCC1(F)F c1(OC(C)C)cccc(CN)c1.C12CC(C=O)(C1)C2.c1(CC)cn(C)cn1 C1(C=O)C2CCC(C2)C1C.CCCCOCC1CC1.C(=O)C.C(=O)C.N C(C)(CO)(C(=O)NCC(C)(C1CCC1)NC(=O)C=CCO)OC C#Cc1ccc(F)cc1C(N1CCC(F)C(NC(C2CCC(=O)C2)=O)C1)=O CN1CC=C(CC(=O)Nc2cccc(NC(C3(C)CC3Br)=O)c2)CC1 N1(C(c2[nH]c(C)c(C(C)=O)c2C)=O)CCC(C)N(C(c2cccnc2C)=O)CC1 c1(C2(C=O)CC2)ccc(C(C(=O)N)N(C)C)cc1.c1(CCC)nn[nH]n1.CS N1(C(C(C)C)=O)CCCC(C(=O)NCC(O)CNC(=O)CCc2ccsc2)C1 n1(CCC(=O)NC(CNC)C)nc(O)c2ccccc2c1=O c1(CC)c(C(=O)OCc2cccc(C(F)(F)F)n2)cnc2ncnn12 Cc1nc(C(N2CCC(F)C2)=O)c2ccnc-2[nH]1.C(=O)CN(S(C)(=O)=O)C.N C(=O)(CCCC(OC)OC)NC1CC2(C(C(N3C(CCC)CCCC3)=O)C2)C1 c1(CC(=O)NC2CN(C(C3(C(F)F)CCCC3)=O)CC23CC3)cccc(O)c1F c1(C(=O)NCC(N(C(C=CCCC)=O)C)C2CC2)cnc(NC2CC2)s1 C1(NC(c2cc(C)oc2)=O)CC(NC(c2cc(N)ccc2O)=O)C12CCOCC2 c1(CNC(C2C=CCN2C(=O)C=CC(F)(F)F)=O)cncc(Cl)c1 C(=O)(C1CCCn2cc(C)nc21)NCCN(C(C(CCSC)OC)=O)C(C)C Cc1[nH]nc(C(=O)N(C(C)C(=O)NCC2(C)CCOC2)C)c1O c1(NC(c2cnc(OC)c(C)c2)=O)nc(C2=CCCC2)sc1C N1(C(c2c(CC)cccc2)=O)CC2CN(C(c3ncccc3F)=O)CC12 Cc1nc(C(C)C)oc1C(=O)NC1(C)CN(C(c2cscc2Br)=O)C1 CC1CCS(=O)(=O)CCN1C(=O)NCC1CCCCC(O)C1 c1(C(=O)NCC2C(NC(C3CC(OC)CC3)=O)C2)cc(Cl)c(F)cc1F N1(C(c2cnc(Cl)n2C)C(=O)NCCCCCC)c2ccccc2CC1C Cc1noc(C)c1C(N1CC(O)CC1C(=O)NCCN)=O.c1cccc(F)c1 C1(NC(C2N(C(C3CCCN(CC)CC3)=O)CCCC2)=O)CCC(F)(F)CC1 CC1CCCCCN1C(=O)C=CC(C)(C)NC(c1ccnn1CCF)=O c1(C(=O)OC)cc(C(=O)N)c(F)cn1.c1(C=O)c(Cl)c(C)nn1C.CC(O)C CCC(CC(C)C)C(=O)N1CCCC1(C)CNC(c1csc(COC)n1)=O N1(c2nccc(OCC)n2)CC2(CCCC2NC(c2cnc(C(C)C)s2)=O)C1 C1(NC(c2ccn(C(F)F)n2)=O)CN(C(C2CC3CCC(C2)C3)=O)CC1C1CC1 c1(CC)ncccc1C(N1CC2C(CNC(=O)C(C(C)C)N(C)C)C2C1)=O CN1CCC(N(C)C)(CNC(=O)Nc2ncoc2-c2ccccc2)CC1 C=C1CC2(C1)CC(C(=O)NCCC1(C)CC1)C2.c1(C(C=O)O)cncn1C C1(C(=O)NCC=CC(=O)NCc2cc(OC)no2)CC(=O)N(C)C1 c1(CC(=O)NCC2N(C(C(=O)N(C)C)=O)CCC2)cc(Cl)cc2c1OCC2 C(C)(CC(=O)N1CCC(C(C)(C)C(=O)NCCC2(C)CC2)C1)SC C1(C(=O)NC2C(C)(CC)C2)CCN(C(=O)Cc2cc[nH]c2)C(C)(C)C1 Cc1c(Cl)cnn1CC(N1CCCCC1C(C)NC(=O)CCCC1CCCC1)=O CC(CCC(=O)NC1CN(C(C2(Cl)CC2)=O)CC2(CCC2)C1)S(C)(=O)=O C(c1ccc2c(c1)CCO2)=CC(=O)NC1CN(C(C(C(CC)C)OC)=O)C1 c1(C(=O)NCC(CC)NC(C2(N(C)C)CCC2)=O)cnc2[nH]cnc2c1 CC1=C(C(=O)N2CC(NC(c3ncsc3C)=O)CC(O)C2)SCCO1 N1(C(=O)CN2CC=CC2)CCCN(C(c2oc(Br)nc2C(F)F)=O)CC1 C1(C(=O)NCCc2cc[nH]n2)(NC(C(CSC)O)=O)CCN(C)C1 c1(C(=O)NCCC2(C)CCN(C(C(CCC)OC)=O)C2)c[nH]c(=NCC)s1 C1(C(C)(C)C)C(NC(c2cc(C(F)(F)F)on2)=O)CCN1C(C1CCC1)=O C1(C(=O)OC)CCN(C(CC2CCC(C)(C)O2)C=O)C(C)(C)C1.C1CCCC1.N CC(C)C(CCNC(c1snnc1C1CC1)=O)NC(C1CC2CCC1O2)=O C1(CC)CC(C(N2CCN(C(=O)CCSC)C(CC)C2)=O)CC(=O)N1.C(=O)N C1(NC(=O)CC2CCC3CC3C2)CN(C(c2ccsc2)=O)CCC12CCOCC2 c1(-c2c(N)cccc2)n[nH]c2c1CN(C(=O)CSc1ccc(F)c(F)c1)CC2 C1(C(=O)Oc2n(C3CCCC(OC)C3)ncc2C#N)CCOCC12CCCCC2 C1(C(N(C(C)CO)CCC)=O)CC2CCN(C(C)CCC(=O)O)CC12 C1(CNC(N(C2CC2(C)C)C)=O)CCN(CC(F)(F)F)C1 N(C(=NCc1ccc(OC(F)F)cc1)NCC1CC12CC2)CC1N(CC)CCC1 C1(OC)CC2CC1CC2N(C(c1sc(Br)cc1C)C(=O)NC1(C)CC1)C CC1CC(C)CN1C(=O)CNS(N)(=O)=O.c1(C(=O)N)ccc(N(C)C)cc1 c1(OCC)cncc(C(N2CC(C)(C(=O)NC(C#N)C(N)=O)C2)=O)c1 N1(C(C(CC#C)NC(c2cc(C)[nH]c2C)=O)=O)CCn2ccnc2C1 CN=C(NCC(=O)N(CC)OC)N1CCC(C(c2cccc(Cl)c2)C)CC1 C(CN=c1[nH]c(Cl)ncc1Br)OCCNC(CCN(C)CC)=O c1(CC=O)cccc(Cl)c1Cl.C1(OCC=CC(=O)N(CCC)C)CCOCC1 Cc1cc(C(F)(F)F)ncc1C(=O)NC(CO)C(C)NC(c1snnc1C)=O N1(C(c2c(Br)c(C)n(C)n2)=O)CC2(CCC(C(=O)Nc3cc(Br)ccc3I)O2)C1 C1(C(=O)N(C(C)C(N)=O)C)(COC)C=CCN1C(c1cccc(F)c1)=O N1(C(CC)=O)CCC(C(C)C)C1.C(C)(C1CC1)=CC=O.C(CO)OCC c1(NC(C(=O)OC)Cc2ccc(F)cc2)cccc(C2CC2(F)F)c1 Cc1ccc(-c2nc(COC3CC(F)(F)C3)n(CCCC(F)F)n2)cc1 C1(CC=C)(NC(=O)C(CO)c2ccccc2)CCN(C(C2NC(=O)OC2C)=O)C1 c1(-n2ccc(NC(C(C(C)C)ON)=O)n2)c(F)cccc1F c1(N2CCCC(C(C)NC(=O)CCCN(C)C)C2)nc2cc(Br)ccc2o1 CC1ON=C(C(=O)NC2CCC2NC(=O)C=CC2CCCCCC2)C1C C1(C(=O)NCC(C)(C2CC2)NC(c2c[nH]cc(Br)c2=O)=O)CCOC(=O)CC1 Cc1ccc(Cl)c(CNC(=O)NC2(CO)CC(F)(F)C2)c1 Nc1cc(CNCCC23CCC(CC2)CC3)cc(O)c1 N1(C(C2C(C)C2)=O)CC(NC(c2cnc(Cc3ccccc3)s2)=O)C2CC2C1 c1(C(=O)NCCC(=C)CNC(=O)C(C)S(N)(=O)=O)c(C)cc(C)oc1=O C(C)(C)(CCCC(=O)NCC1CC2CC2C1)NC(C1(Cl)C(C(C)=O)C1)=O.C N1(C(=O)OC(C)(C)C)CCC(F)(NC(=O)NCC2CCC(Cl)CC2)CC1 N1(Cc2c(C)cc(Br)cc2)CC2CCC(NC(=O)CC3CC3)CC2C1 C(C1CNCC1C=O)=CC.C(C)CC.C(C)(C)C.C=O.C(=O)C1CC1.N CC1CSc2ccccc2N1C(C1CCC2C(CC1)C2(F)F)=O c1(C2C(C=O)C2)cccc(C(F)(F)F)c1.C(=O)(CCn1cncn1)N(C)CC c1(N(C(=O)C(O)C2CN(C=O)C2)C)cccc(C(F)(F)F)c1N.C(C)(C)C.O C=CCCCCC(=O)N1CC(CNC(=O)CCc2nc(CCC)no2)C1 CC(C)CCCCCNC(=O)C(C)(C1CC1)N(C(=O)C(F)C(C)(F)F)C C(=O)C(F)(F)CCn1cccn1.C1(CC(=O)NCCCS)CC1(Cl)Cl.CC=O N1(C(c2ccn(C)n2)=O)CC(NC(=O)CC(C)(C)C(F)F)CC12CCCCC2 C(c1cnc(C)nc1O)=CC(=O)NCC1C(NC(C=C(C)Cl)=O)C1 N1(C(C2CCN(S(CC)(=O)=O)CC2)=O)CC(C)CN(C(c2ccoc2)=O)C(C)C1 c1(OC)cncc(Br)c1C(N1CCC1CNC(c1cc(O)cc(Cl)c1)=O)=O c1(C(N(C2CCN(C(C3C(C=C)OCC3)=O)C2)CCC)=O)c[nH]c2ccncc12 c1(C(=O)NCCCCCNC(CC2(OC)CC2)=O)ccncc1C1CC1 c1(C(N2CC(NC(C(C)(C)c3cscn3)=O)C(F)CC2)=O)ccn2nnnc2c1 C(=O)(CC(C(F)(F)F)NC(=O)CNC(N)=O)NC(CN(C)C)CO c1(C(N2CC(CNC(CCC#C)=O)C(C)(C)C2)=O)cc(Br)c(OC)cc1C C1(CC(=O)NCc2nc(C)cs2)CCCCO1.C(=O)(C)N.C(=O)C1CC1 C1(NC(C2CCN(C(CCC=CCC=C)=O)C2)=O)CCC2(CCC2)CC1 C1(NC(C2CCCC(OC)C2)=O)CC2CCC1CC2NC(c1ncccc1C)=O Cn1nc(C(=O)N(CCn2cncn2)Cc2ccccc2)c2c1CCCC2O c1(C(=O)NCC(CNC(CC2C(C)CCCC2)=O)(C)C)cccc2ccncc12 CC1CC(C)N(C(c2cnn(C(C)(C)C)c2)=O)CCN1C(=O)CCN1CCCC1 N1(C(C(C(C)(C)C)N(C)C)=O)CC2(NC(=O)CCCC)CCC1CC2.C(N)(=O)N N1(C(c2c(C(C)C)cco2)=O)CCCC(CC(=O)N(C(C(N)=O)C2CC2)C)C1 N1(C(c2cncc(C)n2)=O)CCC(CC(N)=O)(NC(=O)C(F)C(C)(C)O)CC1 N1(C(CN(CCC)C)=O)CCN(C(=O)C(F)CNC2CC2)CC1CC(F)F.C n1(CC(=O)NC(CN(C(c2cc(C)n(CCO)n2)=O)C)C)ccc([N+](=O)[O-])n1 C(=O)(C(C)CC#N)NC1(C2N(C(=O)NC3C(CC)OCC3)CCC2)CC1 CCCCCC(O)CC(=O)N1CCN(C(=O)CC2(C)CCC2)CC1CCO c1(C=O)ccoc1C(F)(F)F.C(CC(=O)NCC1CC1)NC(=O)NC C1(NC(C(C)c2ccsc2)=O)CCCCN(C(c2cnn(C)c2Cl)=O)C1 Cc1nc(O)[nH]c1C(=O)NC1(C)CCN(C(C2CC2c2ccncc2F)=O)C1 Cn1nnc(NC(=O)NCC2=NOC(C)C2)c1C(F)(F)F n1(CC)ncc(P(C)(C)=O)c1NC(N1CCN(c2ccc(C#N)cn2)CC1)=O N1(C(C2(COCC)CC2)=O)CCOCCC1.C(=O)CC=O.CC(F)(F)F.C C#Cc1cncc(C(=O)N(C2CCN(C(c3cc(C)c(CC)s3)=O)CC2)C)c1 C1(CC=O)(C(F)(F)F)CC(=O)N(O)C1.c1(CN(C(C)C)CC)ccns1 c1(C(=O)NC2C(CNC(CCSCC)=O)C2)cccc(C#CCO)c1 C1(NC(C2CC=CCC2)=O)C2CC3C(C2)C13C(=O)NCCn1ncnn1 N1(C(C2(C)CC=CC2)=O)CCCC(C(=O)NC2CC23CCC3)CC1 C12(CC)CCC1CN(C(c1conc1C1CC1)=O)C2.Cc1ncn(O)c1C(=O)N Cc1cc(C(=O)N(C(C)CCNC(C2(CCO)CC2)=O)C)c2c(C)n[nH]c2n1 c1(NC(C2CCOC2)=O)cc(Cl)c2[nH]ncc2c1 C(=O)(CC(=O)Nc1nc(C(N2CCCC2c2ccncc2)=O)cs1)OCC C(=O)(C1CCCn2cnnc21)N1C2CC(CNC(C3(CC)CC3)=O)C1CC2 c1(OC(C)C)nccc(C(N2CCC(NC(=O)C(O)C(C)C)C2(C)C)=O)c1F Cc1cc(=O)n(C)cc1C(=O)NC1CN(C(=O)C2=NNC(=O)C2)CC1O C(C)(C)(CC(F)C(=O)N1CCC(c2ccco2)C1)NC(c1c[nH]c(=NC)s1)=O C(N=c1[nH]c(=NCC2CC3C(C2)C3(F)F)c2ccccc2[nH]1)c1cccc(O)n1 c1(C(C(=O)N(C2CCS(=O)(=O)C2)CCC)O)ccc(F)c(Br)c1 N1(C(C(=O)N(C)C)=O)CCC2CCN(C(c3cc4c[nH]nc4s3)=O)CC2C1 C(CC(=O)NCC1(F)CCC1)(c1cccs1)NC(C)=O.C1(C=O)CCO1.N c1(C2(C(=O)NC(CNC(C(CC)OCC)=O)C)CCCC2)ccc(Cl)cc1Cl O=C1OC2CC(C(=O)Nc3cccc(Br)c3I)CC2O1 c1(C(=O)NC2CCCCN(C(C3CC(C)OC3)=O)C2)nnc2n1CCCCC2 C(C)(C(C)C(=O)NCC1CCOC1C)NC(c1c(C)noc1)=O N1(C(c2c(CC)noc2)=O)C(C(=O)NC(C)C(C)(C)C)CC2CCCC12 c1(CC(=O)N(CC(CC)NC(c2ccc(N)cn2)=O)C)ccnc(Cl)c1F c1(C(=O)NCC(C2CC2)NC(C2(C)ON=C(C)C2)=O)cc2cn[nH]c2cn1 c1(C(N2CCC(CN(C(C=CC(CC)C)=O)C)C2)=O)c(Cl)ccc(Cl)c1O C1(NC(CCCCOC)=O)CCC2(CC1)CC2NC(c1cc(=O)n(C)cn1)=O C1(CNC(c2c(OC)nn(C)c2)=O)CN(C(c2ccccc2)=O)C(C)(C)C1 C1(NC(COC)=O)CC1C1CCCN(C(c2cc3occc3[nH]2)=O)C1 N1(C(C(C2CCCCC2)OC)=O)CC2CC2(C(N2CCC(C(N)=O)CC2)=O)C1 C1(C(N(CCC(=O)OC)CC)=O)C(C2CC2)CCN1C(=O)Cc1cnsc1 c1(C(N2CCC(CC)C2C(=O)NCCOC2CCC2)=O)c[nH]c2ncccc12 N1(c2ncnc(CC)c2F)C2CCC1C(C)C(NC(=O)CCN1CCCCC1)C2 Cn1cc(SCC(=O)NCC2CCN(C(C3(CO)CC3(F)F)=O)C2)cn1 c1(C(=O)NCC(C)NC(=O)CC2CCC3CC23)c[nH]nc1-c1cnn(C)c1 C1(COC)(NC(=O)CC2CN(C(C3CCC3)=O)C2)CCCCC1.N(C)C Cc1nc[nH]c1C(=O)NCC(c1ccccc1)N(C(=O)C(C)CO)C C=C(C)CC(C(=O)NC1CN(C(c2c(C)nn(C)c2OC)=O)C(C)(C)C1)OC c1(CC(C(=O)O)NC(C(n2ccc(C3CC3)n2)C)=O)cc(F)cc(F)c1F Fc1cc(Br)cc(-c2nc(COc3ccccc3)no2)c1F C1(C(=O)NC(C)CCCCO)CCCCCCN1C(c1cccc(O)n1)=O N1(C(CCNC(COC)=O)=O)CC(F)(F)CC1.C(=O)C(C)(C)c1cnc[nH]1.C c1(C(=O)NCC2CN(C(c3c(C)noc3C3CC3)=O)C2)sc(C)c(Br)c1C C(C1=NOC2CN(C(c3cn(C)nc3Cl)=O)CC12)NC(CC(CC)CC)=O CC(CNC(=O)C(C)(C)C(F)F)C(F)C(=O)NCC1CC12CC2(F)F CCCCCC(C)(C)C(=O)NC1CCCCCCC1NC(=O)C(C)CS(C)=O Cc1ccc(NC(=O)NCC(O)CS(C)(=O)=O)cc1C(F)(F)F C(=O)(C(F)C(C)(C)O)N1CCN(CCN(C(C(C)C2CC2)=O)C)CC1 CCC(C)C(O)C(=O)NCCN(C(c1ccc(C=O)c(C)c1)=O)C(C)C.O O=C(CCCC1(NC(C2CC2(F)Cl)=O)CCC1)NC1CCCC1O c1(C(=O)NC2C(NC(CC=CC=C)=O)CCC2)cccc(Cl)c1C C(=O)(C1=CC2C=CC1C2)NCC1(C)C(C)CN(C(c2c(C)scc2)=O)C1 C(=O)(C1=CCOCC1)N1CC(C(N)=O)(CNC(=O)C(F)C2CCC2)C1 C1(NC(C(C)NC(CC)=O)=O)CN(C(=O)C=Cc2cnn(C)c2)CCC1C c1(C(=O)NCC(CNC(c2n(CC)cc(Cl)c2)=O)O)ccc2c(c1)ncn2C C(CCC1CCC1)(C=O)NC(C(C)=C(CC)C)=O.N1(CC)CC(=O)NC1=O.N C1(NC(C2(OC)CCOC2)=O)CCOCC1C(=O)NCCCCCCO C1(C2CCOCC2)(C(=O)NC(C)CN(C)C(C2CC3(C2)CC3(F)F)=O)CC1 c1(C2CN(C(C(C)=CC)=O)C2)ocnc1CNC(C1CC1C(C)C)=O N1(C(CC(=O)OCC)=O)CC(C)(O)CC1C(=O)NOC(C)CCC(=O)OC C1(C=O)CCOC(=O)CC1.Cc1csc(CC(=O)NCC2(O)CC(C)C2)c1.N CS(=O)(=O)CCCC(=O)NC1C2CC1N(C(c1ccn3nnnc3c1)=O)C2 C1(CC)CC(C(=O)NC(C)Cc2cnn(C)c2)CCN1C(C1CC(O)C1)=O C=CCC(C(=O)N1CC=CC1(C(=O)N=c1ccn(C2CCC2)[nH]1)C)C(C)C C(=O)(C(C)(C)C(C)NC(=O)Cc1cn(C)nc1C)N1C(C(=O)OC)CC1 CC(C)(C)CCC(F)C(=O)N1CC(C)(C)CC1C(=O)NCCCc1cn[nH]c1 N(C(=NCCc1ccccn1)NCc1ncc(Cl)s1)C(C=C)C c1(OC(C#C)C)ccccc1OC(c1ccccc1OCC(=O)NC)=O C(c1cnn(C)c1)=CC=O.C(=O)(C(C)C1CC1)OC.C(=O)C.C(=O)C C1(NC(C2(CC=C)CCN(C(=O)CC(C)O)C2)=O)CCC2(CCC2)C1 C(c1ncc[nH]1)=CC(N1CCC(C2CCCN2C(=O)C(F)=C2CCCC2)C1)=O N1(C(C(C)NC=O)=O)CC(F)(F)CC1C(=O)NC1CC1C N1(c2nc(C)nc(O)c2C)CCC2(CCCCC2NC(=O)C(N)=O)CC1 N1(C(CCNC(c2ccc[nH]2)=O)=O)CC(Nc2ncncc2I)C2(CC2)C1 c1(C(N2CC(NC(c3c(SC)cccc3F)=O)C(C)C2)=O)c(F)ccc(F)c1Cl C(=O)(C1=CC2(CN(C(=O)Cc3csnc3C)C2)OC1)N1CC(C(=O)NC)OCC1 C=C(C)CC(C(=O)NCc1cc(=O)cc[nH]1)NC(=O)C(C)CN(C)C CC1COCC(CC(=O)NCc2cc(C(=O)NCc3nc(CO)n[nH]3)no2)O1 c1(C(=O)NC2CCN(C(C(C(C)C)F)=O)CC2CO)cc2c(=O)cc[nH]c2s1 N1(C(C(OC)OC)=O)CCCC(CNC(C2CC3(C2)CC(O)C3)=O)(OC)C1 Cc1cc(C(N2CCCC2C(C)(C)CNC(=O)CC=O)=O)nnc1C.C1CC1.N c1ccc(F)cc1F.c1(C(=O)NC(C2CCCN2C(=O)CO)(C)C)coc(O)n1 C#Cc1cccc(CC(N2CCC(C(=O)N(C3CCOCC3)C)(CC)C2)=O)c1 C1(C(CNC(c2ccn[nH]2)=O)F)CCN(C(=O)CC2CCCO2)CC1.C1CC1.C C(C(=O)NC(CC)C(C)C)(C(C)C)NC(C)=O.c1cc(C)no1.C(=O)C.N C=CCCC(C)(C)C(=O)NC(C1CCN(C(c2ccnc(CC(C)C)n2)=O)C1)C C1(C(=O)NCCOC)C2CCC(C2)C1NC(c1cc[n+]([O-])cc1)=O Cc1cccc(C(=O)NCC2CCCN2C(C2(C=O)CCC2)=O)c1Cl.C1CC1 N1(C(CCOC(C)C)=O)CC(NC(C2COCCN2C=O)=O)C(C)(C)C1 c1(CC(=O)NCCC2CC(NC(Cc3c(C)n[nH]c3)=O)C2)ccc2nonc2c1 N1(CC)CCC(NC(=O)CC2CN(C(=O)CSC)CC2C)C(C)C1 N1(C(c2cn(CCC)nc2)=O)CCCCC1C(=O)NCc1cnn(C)c1C CC(CN=c1ncc(NC(=O)CS(N)(=O)=O)c[nH]1)c1ccc(Cc2ccccc2)cc1 C1CC(C2CCN(C(=O)C(C)(C)C)CC2)C1.C(C)(C=O)OCC=C.C(C)C.N n1(CC)nnc(C)c1C(=O)NCC(C)N(C)C(c1cc(C#N)cs1)=O c1(C(N2CC(C)C(CNC(c3ccc(CO)cn3)=O)C2)=O)cccn2nccc12 c1(C=O)ccc(F)c2ccoc12.NC(=O)CCNC(=O)C(=O)N.C1CCC1.C C#CCCCCC(=O)NC1C2CC(NC(=O)C(F)C(F)(F)F)CC12 C1(C(=O)NCC(COC)NC(=O)C2=C(Cl)CCOC2)C2Cc3ccccc3C12 N1(C(C(C)Cc2ccccn2)=O)CCC(NC(c2ccns2)=O)CC1C C1(NC(C(CCC=C)(F)F)=O)CCN(C(C2CC23CCOCC3)=O)CCC1(F)F c1(CN(C)Cc2cnc3ccc(Br)cc3c2)nc2ccc(Br)cc2n1C C1(C)(CCC(=O)N(C(C)CNC(c2cncs2)=O)CC)CCC(=O)N1 c1(OC)cc(N)cc(NC(c2ccc(S(=O)(=O)N(C)C)cc2)C)c1[N+](=O)[O-] c1(C(=O)NC2(COC)CN(C(=O)C(C)=C3CC3)C2)cc[nH]c2nccc1-2 CC1CN(C(C2CC3CC3C2)=O)CCC1C.C1(C(=O)N)CC(=O)N(C2CC2)C1 c1(NC(COCCOCC)=O)cnc(Cl)c(Cl)c1C(=O)OC CCCC(CCC)C(=O)N1CCCC1CNC(c1nc(Br)cnc1N)=O CC(C)C(O)C(C)(C)C(=O)NCCCCCCNC(=O)C1=CS(=O)CCC1 c1(C(CNC(c2nccn2C)CC)F)ccc(F)cc1F Cc1nc2c(s1)CCCC2C(=O)NCC(C(C)C)NC(=O)C(C)(C)C(C)C c1(C(N(CC(=O)N(C2CCC(NC(c3ccccc3)=O)C2)C)C)=O)ccccc1 C(F)(C(=O)N1CCCO1)C1CC(CNC(=O)CCOC2CCC2)C1 c1(CC)ccc(C(=O)NC2(C(=O)C3CC3)CC2)cc1F c1(SC)cccc(F)c1C(=O)Nc1ccc(NC(=O)C)c(C)c1.CC(N)=O c1(C(N2CCC(NC(c3cncc(C)n3)=O)C2C2CC2)=O)cc([N+](=O)[O-])c[nH]1 c1(CC(C)NC2CCN(c3ccc(OC)cc3)CC2)cccc(Cl)c1Cl C#Cc1cnc(C(=O)NC(C)(CO)C(N2CCOC(CC)CC2)=O)c(C)c1 C1(NC(C2C(CC)C2)=O)CN(C(c2ccoc2C)=O)CC12CC2 c1(C(=O)NC2CN(C(CCCOCC)=O)C(C)(C)C2)cc2ccccc2n1C c1(C(=O)NCCC(C)N(C(C2C(OC)CCCC2)=O)C)cnc2n[nH]c(C)c2c1 CCCC(CC(=O)NCC1(CC(C)=O)CC1)NC(C1CC(CC)C1)=O c1(C(=O)NCCC(=C)CNC(C2CC(N(C)C)C2)=O)cnc(OC)cn1 C1(NC(c2ccc(C)s2)=O)CCOC2(CCN(C(=O)C(O)CC(C)(C)C)CC2)C1 C(=O)(C1=C(C2CC2C)N(C2CC2)C(=S)NC1c1cc(C)cc([N+](=O)[O-])c1)OC c1(OC)cc(OC)[nH]c(=NC2CC(F)(CNC(=O)C(C)SC(F)(F)F)C2)n1 Cc1cncc(C(=O)NC2CCC(CCNC(=O)C=CCO)C2)c1C c1(C(=O)NCC)ccc2c(C(=O)N(C3CCC4(CC3)OCCO4)C)n[nH]c2c1 c1(CN(C(=O)NCC(=O)N(C)C)CCO)ccc(C2CC2)cc1F c1(C(N2CC(COC)(NC(=O)CCC(C)N(C)C)C2)=O)cc(Cl)ccc1F Cc1ccc(C(=O)NCC2COC(C)C2)nc1.c1(C=O)ccsc1C(F)F.N CCCCC(CNC(=O)C(c1ccccc1CC)(F)F)NC(C1CCOC1)=O C#Cc1ccc(C(=O)NCC(C)NC(=O)C(C)N2CCCC2)o1 C(=O)(CCCCCN(C)C(C12CCC(CC1)CC2)=O)NC(C(=O)NCC)C C12(C(=O)N(C3CCNC3)C3CC3)CC(C1)C(C(F)(F)F)N2 C12(C(=O)NC3(CCC)CC3)CCN(C(C3(NC(N)=O)CC3)=O)CCC1C2 CN1CCC(C(=O)NCCCC2CN(C(C3COCC3C(N)=O)=O)CCO2)C1=O c1(C(=O)Nc2ccc(-c3nn[nH]n3)cn2)nnc(Sc2ccccc2)cc1Br Cc1cc2c(C(=O)NCC3CC(F)(C)C3)cccc2o1.c1(C(=O)N)ccc[nH]1 c1(C(=O)NCC(CC=C)NC(C2(C)CCCS2)=O)cc(=O)c2cc(Cl)ccc2o1 c1(SC)cccc(C(=O)NC(C)C(CO)NC(c2ncoc2Br)=O)c1 C1(F)(C(N2C(C)CN(C(c3ccoc3)=O)CC2)=O)CCCCC1(F)F c1(CC=O)ccc(C=O)nc1.C(C1CCCO1)=CC(=O)N(C1CCC1)C.CO N1(C(c2ccn(COC)n2)=O)C2CCC1CN(C(=O)C(N1CCN(C)CC1)C)C2 C#CCCCCCC(=O)NC1CN(C(=O)CC(CC)C(C)C)CC1n1ccnn1 C1(C(=O)NC(CN(C)C)CO)(NC(c2csc(CO)n2)=O)CC(F)C1 Cc1cccc2cc(C(=O)NCCCC3(NC(C4CC(F)C4)=O)CC3)[nH]c12 C1(NC(CCc2cccc(OCC)c2)=O)CC2CCC1N(C(=O)C)C2.C1CC1.O CCCCC(C)C(=O)N1CCN(C(=O)C(C)C(C)C)CC1CCO N1(C(CCN(CCC)C)=O)CCCC2(CNC(c3ccc(C)cc3C)=O)CC12 c1(OC)ccc(CC(=O)NC2CC(NC(=O)Cn3ccccc3=O)C2)cc1 N1(C(CCOCC#C)=O)CCC(C=C)(C(N2CCCC(CF)C2)=O)C1 C(=O)(C1=CC2(CCOC2)C1)NC1CCC(NC(C(c2ccccc2Cl)(C)C)=O)C1 c1(C(=O)N)ccc2c(C)[nH]nc2c1.C(C(C)C(C)C)NC(c1c(CC)c[nH]c1)=O c1(C(=O)NCC(C)N(C(CNC(CC)=O)=O)C)cn(CCOC)cn1 C(=O)(C(C)(C)C(C)(C)C)NCCCNC(c1ccc(OCC=C)cc1)=O N1(C(C2N(C)CCC2)=O)CCCC(F)(C(N2CCNC(=O)C2)=O)C1 Cc1nscc1C(=O)NCc1cc(C(=O)NC(C)C(C)CO)co1 N1(C(C(C)OC2COC2)=O)CCC2(C1)CN(C(=O)C=C1CCCC1)CC(C)O2 Cc1cc(NC(=O)CNCC(=O)N)ccc1[N+](=O)[O-].c1ccccc1S(C)(=O)=O C1(NC(C(CC(=C)C)NC(=O)C(C2CCCCC2)O)=O)CC2(COCCO2)C1 C1CN(C(=O)Cc2n[nH]c(=N)s2)C(C)(C)C1.c1(N(CC(=O)N)C)ccccc1 N1(C(COCCOC)=O)CCC(N(C(=O)CCC2CCCCCC2)C)C(C)C1 Cc1ccc(C(=O)C(N2CCCC2C(C)(C)C)=O)cc1.C1(C=O)(C(C)C)CC1 N1(CC(=O)NC(C)C(c2cccc(Br)c2)N)CCCOC1=O N1(C(C(c2cncn2C)N(C)C)=O)CC2C3CCC(C(NC(=O)CCF)C3)C2C1 CC1CCN(c2ncc(C(=O)NCC(C3CCCN3C(=O)C(N)=O)(C)C)s2)CC1 c1(CC(=O)NC(=O)NCC(COC)F)cc(C(F)(F)F)cc(F)c1 c1(CCCCCC)nc(CC2CCC(=O)N2)n(-c2cccnc2)n1 C1(CC(=O)NCC(C)C)CC2CC2C1.c1(C(=O)N)conc1C1(C)COC1 CC(C(=O)NC1(CC=CC(N2CC3CCC(C2)O3)=O)CCC1)C(F)(F)F C(=O)C(C#N)C(C)(C)C.C(C)C(C)(C)C.n1(CCOC)cc(C(=O)N)cn1 N1(C(=O)Cc2noc3ccccc23)CC2(CCN(Cc3n[nH]cc3Br)CC2)C1 N1(C(c2cc(C)sn2)=O)CCN(C(=O)CSCc2ccccc2)C2CCCCC12 C1(CC)C(NC(c2cc(C)no2)=O)CCN1C(=O)CCc1c(C)noc1Cl C1(CC(=O)N(CC(C)NC(C(C)NS(CC)(=O)=O)=O)C)CCOCC1.C C1(C(=O)NC2C(C=C)COC2)CC(C)(C)CN1C(=O)CC1COC(=O)C1 S(=O)(=O)(c1ccc(N2CC3CC2CO3)cc1Br)NC(C)CCCCCO N1(C(c2n(C)cc(C(N)=O)c2)=O)CCC2(CC2)C1.C12(CC=O)CCCC1C2.C c1(OCC)ccc(F)cc1OCCC(=O)NCC1C2CCOCC12 CCC(CC(=O)NC(C1CCN(C(=O)CC2(C)CC2)CC1)C)c1ccc(C)cc1 S(=O)(=O)(c1ccccc1N1CCC(N2CC(OC)CC2=O)CC1)N(C)C1CC1 C1(C(=O)NCCOC2CCN(C(c3[nH]cc(CC)c3)=O)C2)OCC2CCCCC12 C(=O)(C(C)(C)CC(=O)OC)N1C2(C(=O)NCC(CC)O)CC(C)(C1)C2 c1(C(=O)NCC(N2CCN(C(C=CSC)=O)CC2)C)ccc(N)c(F)n1 N1(C(C2CN(C(C)=O)C2)=O)CCN(C)C(C(=O)NC2CN3CCC2CC3)C1 CN(C)NC(=O)CCC(=O)N1CCCC1C(C)(C)C.C1(CC(=O)N)CCC(=O)O1 C1(CNC(CC)=O)COCC2(CCN(C(c3c(OC)ccnc3F)=O)C2)O1 c1(OC)ccnc(O)c1C(N1CCC(NC(=O)C#CC2CC2)C(CO)C1)=O c1(C(N2CCC(C)C2)=O)ccc2c(c1)CC2.C(C)(C(=O)N)OCCOC.C C1(NC(c2cc(C)c(F)cc2)=O)CN(Cc2ccc(O)cn2)CC(F)(F)C1 c1(C(=O)NC2CC3CC(NC(C(C=C)(C)C)=O)CC3C2)cnc2n[nH]c(C)c2c1 CCCC(CNC(c1sccc1CC)=O)C(=O)N(C1CCN(C)C1)CC C1(C(=O)NC2CCC(C(=O)NC(C(C)C)CO)C2)CC(=O)CC(=O)N1 N1(C(CN2CC(CC)C2)=O)CCCC(C2CCN(C(c3c(Cl)cnn3C)=O)C2)C1 C(=O)(C1=CCc2ccccc21)N1C(CNC(CC(C)F)=O)CC2(CC2)C1 Cn1nc(C(=O)NCC2CCCC2)cc1C(F)F.C1(CC=O)CCCCCC1.N C1(NC(C2CCCC(C(=O)OC)C2)=O)CC2CCC(C1)N2C.c1c(C)noc1C Cc1cc(C#N)cc(C)c1-n1cc(CN(O)C(C2(C)CCC(C)C2)=O)nn1 NC(=O)CCCCC(=O)NC1CC(C(=O)NCC2(C(F)(F)F)CCC2)C1 N1CCN(C(=O)C(N2CCNC2=O)C)CC1.C(C)(C(=O)NC1CC1)=C(CC)C.C Cc1ccc(C(C)C)c(OCC=O)c1.C(C)C(C)C.C1(CC=O)CC1(C)C.N c1(-n2c(C(C3CCCC3(C)C)NC3(CC)CCC3)nnn2)ccccc1Cl c1(C(N2CCC(CNC(C(CC)C3CCOCC3)=O)C2)=O)cncc2n[nH]cc12 c1(CN(C2CCN(C(C(c3ccccc3Cl)OCC)=O)C2)C)ccnc(Cl)c1 c1(OC)coc(C(=O)NCC2CCC(NC(C3CC(C)OC3C)=O)C2)cc1=O CCC(CCCC(=O)NOCC1CCC1)NC(=O)C(C#N)C(C)(C)C c1(OCC#C)ccc(C(N2CCC(CCCNC(=O)CNC=O)CC2)=O)cc1 N1(C(CCCc2ncc(C)o2)=O)CCC(NC(C2CCC(C)(F)CC2)=O)C(O)C1 N1(C(c2c(CC)n(C)cc2)=O)CC2CC1CN(C(=O)CCN1CCOCC1)C2 c1(CC)nc(C)c(C(=O)NC2CCN(C(=O)C(C#N)CC3CC3)C2C)o1 Cc1cc(Br)c(F)cc1CNC.C1CCC(C=O)CC1.c1cnccc1Cl.C(=O)O N1(C(Cc2cc(C)no2)=O)CC(C)CN(C(=O)C(C2CCCCCC2)F)CC1C C(CCCCC(=O)NC(C)(C(=O)Nc1cnc(Cl)c(C)c1)C1CCC1)=CC Cn1cc(C(=O)NS(=O)(=O)CCc2cccnc2Cl)c2ccncc12 C(=O)(C1=NOC(C)(C)C1)N1C(C)CC(NC(c2ccc(C(F)(F)F)nc2)=O)C1 C1(C(=O)NC(C)CNC(c2cnc(-c3cccs3)s2)=O)CC2CCC1CC2 c1(C(C)(F)F)ccc(C(N2CCN(C(C3(C#N)CC3(C)C)=O)CC2)=O)cn1 n1(N(CC(N2CCOCC2)=O)C(=O)NC(C)CC2CCC2)cnc2ccccc12 c1(CC)cc(C(N2CCCCC2C2(NC(c3ccc[nH]3)=O)CC2)=O)oc1CC Cc1ccc(C(C)C(=O)N(CCCN(C)C)CCNC(=O)C=CBr)s1 CCCCC(=O)NCC(C)(C)CNC(C1CCCCS1)=O.C(C)(C)C.C=O.N N1(C(C)C(=O)NCCCC2CCCN2C(=O)Cn2cnnc2)CCCCCC1 N1(C(c2cn(CC)nn2)=O)CCN(C(=O)C(F)CC(C)C)C2CCCC12 C1(N(C(C)=O)C)CC2CCC(C1)N2C(c1ccsc1C(F)(F)F)=O.C=O.CN c1(C(N2CCN(C(c3cnn(C)c3C#N)=O)CC2CO)=O)ncn2ccccc12 c1(C=O)cncc(Cl)c1.C1(C(=O)NC2(C(N(C)C)=O)CC2)CCC(C)C1.N Cc1cc(C(=O)N(C2CCN(C(=O)CCC3CCCO3)C2)C)cc(C)n1 c1(OC)ccc(N)c(C(=O)NC23CC2CN(C(c2c(C)nn(C)c2C)=O)C3)c1 C1(CNC(C(C)=CC)=O)CCN(C(=O)C(c2ccc(F)cc2)F)CC1(F)F c1(C(N2C(C(=O)Nc3ccc(F)cc3)CCC2)=O)ccc2c(Br)n[nH]c2c1 S(=O)(=O)(c1ccc(Cl)cc1F)N1CC2C(C(=O)NCc3ccsc3)(CC2)C1 C1(C(NCCC)=O)CC12CCCCC2.C(=O)(C(=O)N)NCCOCCCC CCC(CN=C(NC1CCCCC1)N(C)CC1CCCS1(=O)=O)OC C#CC(CCC)NC(=O)CC1(OCc2ccccc2)CC1 C(=O)(C(F)C(C)CNC(c1ccc(C)cc1)=O)N1CC(O)(CCC)C1 n1(C(CC)(C)C)nnnc1C(c1conc1C1CC1)NCCC(O)COC C1(C(=O)NC2(CCCNC(Cc3c(C)scc3)=O)CC2)CCC(O)CC1 Cc1cc(Br)c(C(=O)NCCC(C)N(C)C(C2CN(C)CCO2)=O)s1 c1(C(N2C(C(N3CCC(CN4CCCCC4)CC3)=O)CCC2)=O)cccnc1Cl N1(C(C(C)O)=O)CC2CC(NC(c3cn(C(C)(C)C)nn3)=O)CC2C1 C=CCCCCCCC(=O)NCC1CCCCC1NC(C1CC(F)(F)CS1)=O N1(C(CC2N(C)CC=CC2)=O)CC(C2CN(C(c3cnc4c(c3)COC4)=O)C2)C1 C(=O)(CCC(C)(C)C)NC12CC(CNC(Cn3c(C)cnc3)=O)(C1)C2 c1(CC)ccccc1C(C)N(CC(c1ccc(Br)cc1)O)C(C)C c1(C(N(CC(CC)NC(c2c(F)cccc2F)=O)CC)=O)cc2nc[nH]c2cn1 C(=O)(C(C)C)N.C1(CC(=O)N(CC)CC)CNC(=O)O1.[SH](C)(=O)=O c1(SCC)cccnc1C(=O)NC(C1CN(C(C2(C)CC=CCC2)=O)C1)C CC1(CNC(c2cnc(-c3ccccn3)nc2)=O)CCN(C(C2CC2CF)=O)C1 N#Cc1ccncc1C(N1CCCC1CCC(=O)NC1CCCC(O)C1)=O C1(C(C)C(=O)N2CC(CCO)C2)CCN(C(C2CC(O)C(F)C2)=O)CC1 C1(C(N(CCCNC(=O)C(F)(F)C2CC2)CC)=O)CCC2CCC(=O)N12 C(CCCN=c1[nH]cncc1C)NC(C(COCC)N=[N+]=[N-])=O Cc1c(Br)csc1C(c1nnnn1C(C)C)NCc1cc(-c2ccccc2)on1 Cc1nc2cccc(C(=O)NC3CCCC3NC(c3cnn4c3SCC4)=O)c2[nH]1 C1(F)(CNC(CCOC)=O)CCCN(C(c2ccc(C(F)(F)F)cc2N)=O)C1 Cc1cc(C(=O)NC(CO)C(=O)NCCc2scnc2C)no1 C1(C2CC2)CCN(C(=O)C(C)n2cncn2)C1.c1(OCC)ccc(C(=O)N)cc1 C1(C(=O)NC2CC(CNC(=O)COC3CCC3)C2)CCC2CC12 c1(C=O)cnc2n(c1=O)CCS2.C(=O)(CCC(=O)N(CC)C1CC1)NCCC CC1(C)COCC(C(=O)NCC2CCC(NC(c3ccc(N)c(Cl)n3)=O)C2)O1 c1(C(=O)NC(CNC(CC(CCC)O)=O)CC)sc2ccccc2c1CSC N1(C(C=CSC)=O)CCC2C(C(=O)NCc3cc(C4CC4)no3)C2C1 N1(C(c2cc(SC)oc2)=O)CC(CNC(c2c[nH]c(C)c2)=O)OC(C)(C)C1 N1(C(CCC#CC)=O)CCC(C2CCCN(C(c3c(C)csc3Cl)=O)C2)C1 C1(C(N(CCNC(c2cnc(O)s2)=O)C)=O)CCCC12CC2.c1ccccc1 c1(CC=O)ccccc1S(C)(=O)=O.C(=O)(C(C)(C)F)N(C)CCOCCC c1(CC(=O)NC2(CC)CCN(C(=O)C(O)CC(C)C)CC2)ccc2nonc2c1 C1(NC(C(C)n2cccn2)=O)CN(C(=O)C=CC(c2ccccc2F)=O)CC12CC2 Cc1nc(C(=O)N(C2CN(C(=O)CC(C)C3CCCO3)C2)C)c2ccccn12 C1(CC(=O)NC(CCNC(c2c(C)n[nH]c2)=O)Cc2ccccc2)CC=CCN1C c1(CNC(=O)Cc2cccnc2)cc(Cl)cnc1F C#Cc1cc(C(N2CCC(NC(=O)CCc3ccncc3)C(C)C2)=O)ccc1Cl c1(C(=O)NCC2(C(=O)O)CC(F)(F)C2)cccc([N+](=O)[O-])c1.C(CO)N C1(CC(=O)NCC2CSC2)CCCCC1NC(=O)COCC1CCCC1 C(CC(C(=O)NC1CC2C=CC1C2)NC(c1cn(C(C)C)nn1)=O)=CC C(=O)(C#CCC(C)(C)C)NCCNC(C(c1cccc(C#N)c1)C)=O C(=O)(C(C)(O)C(C)C)NC(CCCNC(C(CC)(F)F)=O)C c1(NC(C)CCCc2cccnc2)ccccc1CC(=O)OC(C)(C)C Cc1nc(CNS(=O)(=O)CC2(C)CCCCO2)cc(O)n1 C1(C(=O)Nc2cccc(OC)c2C)N(C(c2cncs2)=O)CC12CCCC2 c1(C(=O)NC23CCN(C(C4CN(CCC)C4)=O)CC2C3)cc2ccc(C)cn2c1 Cc1nc(C)n(CC(=O)NC(C)CCCCNC(C23CC(C)(CO2)C3)=O)n1 C=CC(C)(C)C(=O)NCC1CCCC(CNC(c2cccn2CCC)=O)C1 N1(C(C2(N(C)C)CCCC2)=O)CCCC(N(C(=O)CC2(C#N)CC2)CCO)C1 c1(C(=O)NC2CC(CCNC(C(C=C)(C)O)=O)C2)cc([SH](=O)=O)ccc1F Cc1cc(C(N2CCC2CNC(c2ccc(C#N)s2)=O)=O)cc(C)c1Cl C#Cc1cccc(CC(N2CCC(CNC(c3ccc(=N)[nH]n3)=O)CC2C)=O)c1 N1(C(C(CC#C)(C)C)=O)CCC2(CC1)CN(C(=O)CCc1ccon1)CC2CO CN1CC2(CCCN(c3nc(N4CCS(=O)CC4)nc4cccnc34)C2)CC1=O C1(CNC(C(CC)Sc2nc(=N)[nH][nH]2)=O)CC2CCC1N2C(c1[nH]cnc1C)=O Cc1cc(Cl)ccc1C(=O)NCC1CCC(C)N(C(=O)C2=CCCSC2)C1 C(=O)(CCCCCn1cc(CN2CCCCCC2=O)nn1)N(C1C(C)CCC1)C CCCCC(F)C(=O)N1CCC(OCCNC(c2cc(OC)ns2)=O)C1 N1(C(c2c(OC)nc(C(C)C)cc2)=O)CCCC(F)(F)C1.c1(C(=O)N)cc[nH]c1 c1(C=O)ccc(F)c(F)c1N.N1(C(CNS(NC)(=O)=O)=O)CCC(F)(C)CC1.N C1(NC(=O)Cc2ccc(C)cc2)CCCN(C(C2(C#N)CC2(C)C)=O)CC1.CC N1(C(C(=O)NC(c2ccncc2)C)=O)CCOCCC1C(C)(C)C C(CC(C)(C)C)(C(=O)NCC(CO)NC(=O)Cc1csnn1)OC C#Cc1cn(C)nc1C(=O)N(C1CN(C(=O)C(C(C)(C)C)n2ccnn2)C1)C C1(CCNC(C(C(C)C)OC)=O)CCCN(C(c2cncc(CO)c2)=O)CC1 C1(N(CC(=O)N(CC(C)N(C(=O)CCOC)C)C)C)CCCC1.C1CCC1 C1(C(=O)NC(C2CCC(C)CC2)CC)CCN(CC)C1C.C1(C=O)CCCCCC1 CC(F)(F)C(C)(C)C(=O)NC1CC(CO)N(C(c2cn(C3CC3)cn2)=O)C1 c1(C(=O)NC2C(CNC(C3=CCCC3C)=O)COC2)ccnc2cc[nH]c12 N1(C(c2ncn(CC)c2)=O)CC(C(=O)NCCCCCC2CC2)OC(C)C1 C(=O)(C1CCCc2n[nH]cc21)NC(CC1CC1)N(C(=O)COC1CCOC1)C N1(C(Cn2cc(-c3cccc(C(=O)OC)c3)nn2)=O)CCCc2ccccc21 C(=O)(C1CCCc2nc(C)[nH]c21)O.N12CCC(CC1)C(=O)CNC(=O)OCC2 Cc1ccc(C(c2nnnn2C2CCCCC2)NCCC2CC(C)(C)C2)o1 c1(C=O)cc2n(c(=O)c1)CCS2.CC1CC(C(=O)NC2CCCC2)CC(=O)N1.N CC(C(=O)N1C(C(=O)NCC2NC(=O)OC2(C)C)CCC12CC2)S(C)(=O)=O Cc1cc(C(=O)NC2CC(F)(C)C2)n(CC(F)(F)F)n1.c1(C=O)ccncn1 C1(C(=O)NCC(CCNC(C(C=C)OC)=O)OC)CCOC(C)C1 C1(C(N2CC(N3CCOCC3)C2)=O)CC2(C1)CN(Cc1c(Cl)cccc1Br)C2 n1(CCOC)cc(C(=O)NCC(C)CNC(c2ncncc2C)=O)ccc1=O C=CCN=C(NCCCC#N)N1CCC(C)(c2ccc(F)cc2)C1 c1(C(N2CCC(N(C(=O)C(=Cc3cccnc3)F)C)C2)=O)cnn2ccsc12 N#Cc1ccc(C(N2CCCC2C)=O)c(Br)c1.c1(CCC=O)ccc(C(=O)O)[nH]1 N1(C(C(c2n(C)ncc2)(F)F)=O)CCC(O)C(NC(=O)C(=C2CCCCC2)F)C1 C=CC1CN(C(c2coc(C(C)OC)n2)=O)CC1NC(c1ocnc1CCC)=O C1(CNC(C(C)O)=O)CN(C(=O)Cc2cc3ccccc3s2)CC(C)(C)C1 C(=O)(CS(=O)(=O)CCO)N1CC(O)(CN(C(CCc2ccc(OC)cc2)=O)C)C1 C(c1ccccc1)=CC(=O)NC1(CN(C(C=COCC)=O)C)CC1 C1(C(=O)NCc2ccncc2F)CN(Cc2cccc(N3CCCC3)c2)CCO1 CC(CCCCn1cc(-c2cccnc2)nn1)NC(=O)COC1(C)CCCC1 N1(C(CC2C(=O)NCCC2)=O)CC(NC(C2(n3cncn3)CC2)=O)CC(F)C1 C1(Nc2ccnc(OC)n2)CC(=O)NC(c2ccccc2)C1 CN1CCC(C(F)(F)F)(NC(=O)NCCCCOc2ccccc2Cl)C1 CC(C(=O)N1CC(O)CC1C(=O)NCc1cnsc1)C(F)(F)F c1(C(N2CCC(N3CCOC3=O)CC2)C(=O)NCCCC)c(Cl)ncn1C C(C)([Si](C)(C)C)NC(N(C(C)Cc1ccsc1)C)=O CC1(N2CCOCC2)CCN(CC2(COCCO)CCCC2)C1 C(C(CO)N=c1ccc2nnnn2[nH]1)NC(C1CCn2c(C)ncc2C1)=O C1(C(=O)NCCNC(c2c(-n3ccc(C)n3)cccc2)=O)CN2CCN1CC2 N1(C(CNC(=O)OCC=C)=O)CCN(C(=O)CCS(C)(=O)=O)C2COCC12 C1(NC(C=CSC)=O)CCC(C)N(C(c2cnc(C(C)(C)C)[nH]2)=O)C1 C1(C(=O)NC(C)CC(C)(C)O)CN(C(=O)CCC2(C)CC2)CC1(F)F N(C(=NCc1cc(C(F)(F)F)co1)NCC(c1ccccc1)(F)F)C1C(C)C1 C1(C(N2C3C(NC(C4CN(CC)C(=O)C4)=O)C(C3)C2)=O)CCCC1S(C)(=O)=O c1(C(N(CCCNC(=O)CC)C(C)C)=O)coc(C(F)(F)F)c1.C(N)=O CC1CCN(C(=O)Cc2cc[nH]n2)C1CNC(c1cn(C(F)(F)CO)nn1)=O c1(C(=O)NCC(CNC(C(COCC)N=[N+]=[N-])=O)C)nc(C)c(C)nc1C c1(C(=O)NCC2(CN(C(CCCCC#C)=O)C)CC2)cn2ccc(C)c(C)c2n1 N1(C(c2cc(OCC)ncc2)=O)CCN(C(c2ncsc2C(C)C)=O)CCC1C CC(C(=O)N1CCC(F)C(NC(c2cnoc2-c2ccoc2)=O)C1)C(F)(F)F c1(C(N2CCC(NC(C(CC)N(CC)CC)=O)(CF)C2)=O)oc2ccccc2c1C Cn1cc(Br)c2c(N3CC4CC4(C(=O)Nc4cccc(Cl)n4)C3)ncnc12 C(N=c1[nH]c2cc(F)c(F)cc2s1)C1(C)CCN(C(C2(C)COC2)=O)C1 C(=O)(C(C)C(F)F)N(CCCC(=O)Nc1cc(C(C)C)no1)C(C)C C1(NC(CCCCSC)=O)CCC2(CC1)CCN(C(c1c(C)ccn1C)=O)CC2 C#Cc1ccc(C(=O)NC2C3CCN(C(=O)CNC(=O)NC)CC23)c(C)c1 C1(NC(C2CCC(C)(F)CC2)=O)CC2CCC1CN(C(=O)CCCC#N)C2 N1(C(C(=O)NC2CC2c2ccc(Br)s2)=O)Cc2c(O)n[nH]c2C(F)(F)C1 c1(C(N2CCC(C(Cc3nn[nH]n3)OCO)C2)C)cccc(Br)c1 c1(C(N2CCCC(NC(=O)C=C3CCC3)CCC2)=O)cc(Cl)cc2c1OCC2 Cc1c(NCCS(N)(=O)=O)ncnc1N1CCCC(NC(C)C)CC1 c1(C(N2CC3CN(C(C45CC(C)C4C5)=O)CC3C2)=O)ccc2oc(O)nc2c1 C12(CNC(C3CCC(=O)N3)=O)CCCC1N(C(c1ccnc(F)c1F)=O)CCC2 C=C(C)C(C)(C)C(=O)NC1C=CCN(C(c2nn[nH]c2C(F)(F)F)=O)C1 Cc1cc(C(=O)NC2CC(C)C2)c(N)c(F)c1.C1(C=O)CCN(CC(C)C)C1 Cc1ccn(CCC(=O)N(C2CCN(C(=O)CN3CC=CC3)C2)CCO)n1 C(=O)(C1=C(Cl)CCCC1)N1CC(C)(CCC(=O)N(CC(O)CO)CCO)C1 C1(C(=O)NC2CCC(N(C(C(C)NC(N)=O)=O)C)CC2)CCOC(=O)CC1 N1(C(C=CC(C)(C)C)=O)CCC2C(CCCN2C(=O)CO)C1.c1ccc(Cl)cc1 N1(C(COC2CC(NC(c3cc(SC)oc3)=O)C2)=O)CCN(C)C(C)(C)C1 C(c1cccc(F)c1)=CC(=O)NCCC.c1(C=O)ccccc1C(F)(F)F.N C1(C(=O)N)CC12CCN(C(C1CCOC(C)(C)C1)=O)CC2.c1(CC)cc(C)on1 S(=O)(=O)(c1cc2nc(O)[nH]c2cc1Cl)N1CCCC(OCC#C)C1 C1(C(=O)OC)CCN(C(=O)CC2CN(C(c3ncncc3N)=O)CCO2)C1C Cc1cnc2n1CCC(C(N1CCC3(CC1)CC3NC(C13CCC(C1)C3)=O)=O)C2 C1(NC(CC2COCC(C)O2)=O)C2CC3C(C2)C13C(=O)N.c1cn(C)cn1.C N1(CC(=O)NC2CC(CNC(C(C)(C)O)=O)C2)CCCCS1(=O)=O c1(CCC(=O)NCC2CC(NC(C3CCC34CCC4)=O)C2)ccc(O)nn1 CCC(C)C(O)CC(=O)N1CC(O)(CN(C(=O)C=Cc2ccccc2C#N)C)C1 Cn1ccnc1S(C)(=O)=NC(=O)CCC(=O)Nc1ccc(Cl)c(Cl)c1 N1(C(C2C(C)C2)=O)C2CCC1C(C(N1CCC(C(C)(C)O)C1)=O)C2 c1(CNC(C2C(C(C)(C)C)CC2)=O)ccc(C(N2CCC2CF)=O)cn1 C1(NC(CC2(C#N)CC2)=O)CCC(NC(=O)C(F)(F)c2cncs2)C1 N1(C(C(=C)C(F)(F)F)=O)CC(NC(=O)C)C2(COC2)C1.C(C)(C)C.C=O N1(C(CNC(=O)OC)=O)CC2CC(NC(=O)C3=CC(O)CCC3)CC(C2)C1 c1(C(C(=O)N2CC(C(C)NC(C3C(C)(CC)C3)=O)C2)(C)C)ccccc1Cl Cc1cc2c(C(=O)NC(C)(C)CNC(=O)CCCC(C)(C)C)cccc2[nH]1 c1(CC)nc(Cl)nc(N2CCS(=O)(=O)C(CC)C2)c1Cl.c1(CC(=O)N)cnoc1 C1(CC)(NC(c2coc(Cl)c2)=O)CCN(C(c2csc(NC=O)n2)=O)CC1 Cc1cc(=NC(=O)C(C)CCN(C2CCCC2)C(Cc2ccccc2Cl)=O)[nH]o1 CC1(C(=O)NCCC2CN(C(c3ccc(C(N)=O)nc3)=O)CCO2)CCNC1=O Cc1nc(C(F)(F)F)c(CN(CC(C)NC(C2CCCC23CC3)=O)C)s1 c1(C(=O)NC2CC(NC(c3nccc(C)c3)=O)C(O)C2)cccc2ccsc12 C(=O)(CCC(O)C(C)(C)C)NC1CCCN(C(c2c(CC)noc2)=O)CC1 S(=O)(=O)(CC(=O)NC1CCCC1)NC.c1(C=O)nn(C2CCOCC2)cc1C.C c1(CC)cncc(C(=O)N)c1.C1(F)CCN(C(c2n[nH]cc2C2CCC2)=O)C1.C C1(NC(c2cc(O)ncn2)=O)CCN(Cc2cc(C(F)(F)F)cc(Cl)c2)CC1O C1(CCNC(C(C)(C)OC)=O)CN(C(=O)C)CC1O.CCN(C)C.C=O C1(N(C(C2C=CCC2)=O)CC)CCCN(C(c2coc(C3CCOCC3)n2)=O)C1 N1(C(CCC(C)=O)=O)CCC2CCCC12C(=O)NCC(O)C(C)O C1(Cc2nnc(N3CCC(OC)C3(C)C)n2CC2CC2)CC2(C1)CC21CCC1 c1(SC(C)C(=O)Nc2ccccc2-c2nn[nH]n2)ccc(Cl)c(Cl)c1 c1(OC)ccc(C(N2CCCC(n3cc(CN(C)C)nn3)C2)=O)cc1OC(F)F C(=O)(CP(C)(C)=O)NCC1(C(=O)NCCCCC)CC1 CC1CN(C(=O)CC2(CO)CCC2)CCC1NC(C1CCOC1)=O c1(C(C)C)ccc(C(N2C3CCC2C(C)C3)=O)c(O)c1.C1(C=O)CCC(=O)N1.N C(N=c1[nH]c(=N)[nH]c(=NC2CCOCC2F)[nH]1)c1ccc(N(C)C)cn1 C(=O)(C1=CC2C=CC(C1)C2)NC(C)CNC(=O)C1=CCOCC1 C(C)(CCCC(=O)NC1CCCN(C)C1)NC(c1ccn(COC)n1)=O C1(CC(=O)NCc2cc(C(N3CC(CC)C3)=O)on2)CCC(C)CO1 c1(C(N(C)CC2CCCN2C(=O)CCC2CCCN2C)=O)[nH]nc2ncccc12 N1(C(C(C(=O)NC)(C)C)=O)CCCC(C2CN(C(C3CC(C)N(C)C3)=O)C2)C1 C(=O)(C(=O)N=c1cc(C)o[nH]1)N1CC(CCNC(C(C)=C2CC2)=O)OCC1 C#Cc1ccnc(C(=O)N(C(C)CC(=O)NCCC(C)(O)C2CC2)C)c1 C12(C(=O)Nc3cccc(NC(=O)CC4CCCOC4)c3)CC(C3COC3)(C1)C2 C=CC(CO)NC(=O)CN(C(=O)CSCCCC)CC(C)C c1(N(C)Cc2nc(C)[nH]n2)nc(=NCC(C)Cc2cccs2)[nH]c2c1CCC2 N1(C(c2cc(Br)c3c(c2)OCCO3)C(=O)NCC)CCCCC2(CCOCC2)C1 Cc1nc(NC(C2CCCC(NC(=O)Cn3ccnc3)C2)=O)c(F)c(Cl)n1 CC1CCN(C(c2ccsc2)=O)CC1CNC(=O)CCN1C(C)CCCC1C N1(CC)CCCC1CC(=O)NC(CNC(=O)C(=O)N(C)C)CCOC Cc1c(N)ccc(C(=O)NC2CCC2NC(C2CC3(CCC3)C2)=O)c1C N1(C(c2c(C)nc(CNC(COc3cc(C)on3)=O)o2)=O)CC2CC2C2CC12 C(N=c1[nH]ccnc1F)C1(C)CCN(C(=O)C=Cc2ccc(C(N)=O)o2)C1 c1(CCC(=O)NC(C(C)NC(=O)C(C)n2cncn2)CO)ccc2[nH]ccc2c1 c1(N(C(=O)C(F)(F)F)C)ccc([N+](=O)[O-])n1C.n12cc(nn1)CCCOCC2 N1(C(c2c(C)scc2)=O)Cc2n[nH]cc2C1C(=O)N1CCC2(CCOC2)C1 C(CC(=O)N)(CC(C)C)NC(C1(CC)CC(C)(C)C1)=O.c1(CCF)ccccc1 S(=O)(=O)(c1ccc(N2CC3(C)CCC3(C)C2)c(F)c1)N(C(c1cccnc1)C)C C1CC(C)CN(C(=O)CC2(C)CC2)C1.c1(OC)ccc(C2CC2C=O)cc1.N Cc1cc(C(N2CCC(C)(NC(=O)C=C3CCC3)C2)=O)oc1C N1(C(=O)NC(c2n(CC)ccn2)C2CCOCC2)CCCC2(CCO2)CC1 C(=O)(CC(C)(C)CCOCCOC)NCC(CCC)C(=O)N(C)CCOC CC(C)N=c1nc2c(ncn2C)c(NCC2Cc3cc(Cl)ccc3O2)[nH]1 C(=O)(C(O)CCCNC(C1(COC)CC(=O)C1)=O)NC(C#C)C c1(C(=O)NCC(CCC)NC(c2cc(C(C)(C)C)no2)=O)cccc2c[nH]nc12 C(C(C)(CC(C)C)NC(c1cc(C)c(C)nn1)=O)NC(C(CC)OC)=O C1(NC(c2nc(C(C)NC(c3nc(CC)sc3)=O)oc2)=O)CC(O)C(O)C1 N(C1c2ccccc2CC1NC(=O)C1CCc2c[nH]nc21)C(C(C1CC1)OC)=O Cc1ccnc2c(C(N3CC(N(C)C(c4cccn5nccc45)=O)C3)=O)cnn12 c1(CC)nn(C)c(CC)c1CC(=O)N.c1(C(N2CCC2)=O)cc(C)cc(Cl)c1 c1(C(N2CCC(C(C)NC(=O)COC3CCC3)C2)=O)cc2nccn2c(O)n1 C1(NC(c2n[nH]c(C)c2Cl)=O)C2CC1CN(C(c1ccc(C(F)F)c(F)c1)=O)C2 CCC(C)C(O)C(=O)NCC1CCCN(C(=O)Cc2cccc(Cl)c2F)C1 N1(C(c2ccc(CC)c(Cl)n2)=O)CCC2CCN(C(c3cc(CO)[nH]n3)=O)CC12 C1(C(=O)NC2CC(C)(NC(c3cnc(O)o3)=O)C2)CC2(C1)NC(=O)NC2=O N1(C(C2=CC(C)(CC)C2)=O)CC(C2CCN(C(c3cccnc3C)=O)CC2)C1 C1(NC(C2N(C(C(CCC)OCC)=O)CSC2)=O)CC2(CCCCO2)C1 CC1(C)CC(C)(CO)CN1C(=O)COC1CCN(C(C2(C3CC3)CC2)=O)C1 Cc1cc(C)c(C(=O)Nc2cccc(OCC3CCOCC3)c2)cc1C N1(C(C(C)(CO)NC(c2nn(CC)c(O)c2)=O)=O)CC2OC(=O)N(C)C2C1 C1CN(C(C2C3CCCC23)=O)Cc2nccn2C1.C(C)(C)C=O.C(=O)NCC.N C(=O)(C(CNC(=O)Cc1ccsn1)CC1CC1)N1CC(C)(CC)C1 C=C(C)C(C)(C)C(=O)N1CCC(O)(CNC(=O)C(C)Oc2cccnc2)C1 CCCCCC(O)C(=O)NCC1CCN(C(c2ncoc2C2CC2)=O)C1 C(=O)(C(O)(C=C)C(F)(F)F)NCC1N(C(C2(CC#C)CCC2)=O)CCC1 C1(F)(C(N2C(C)C(CO)CCC2)=O)CSCC12COC2 CCC(C)(C)CC(=O)NCC1(C)CCCC1NC(c1ccn(C)c1)=O Cc1cn2ccnc(C(=O)NCCCN(C(=O)C=CC3CC3)C)c2n1 CCC(CC)C(C)C(=O)N1CCN(CCN(C)C(c2cc(C)on2)=O)CC1 C1(CNC(CC2(OC)CCC2)=O)CN(C(=O)C2=CCC2)C2(CCOCC2)C1 c1(OC)ncc(C(=O)NCC2(C)CCCN(C(=O)C(C)CC(N)=O)C2)cc1Cl N1(C(C(CCC)C)=O)CCc2nc(CNC(C3C4CCC34)=O)sc2C1 c1(C(=O)NCC2CCCN(C(CC(C=C)C)=O)C2)ccc(Cl)c(C)c1Cl N=c1ncn(CC(=O)NCC2CC2)[nH]1.C1CCOCC1.C(=O)C=CC=O.C c1(C(=O)NC2CN(C(CCc3c(C)cccn3)=O)C(C)C2)c(Cl)nn(C)c1C c1(C(N2CC3(N(C(c4cc(C)cc(C)n4)=O)CC3)C2)=O)nc2c(C)cccc2[nH]1 c1(OC)cc(NC(C2CCCC(NC(c3cncc(O)c3)=O)C2)=O)ccc1Cl Cc1cc(C(=O)NCC(O)COc2cccc(Cl)c2Cl)c(C)n1NC(N)=O N1(C(c2c(CNC(c3cc(C)c(O)cc3)=O)c[nH]n2)=O)CCC(O)C(C)(C)C1 c1(OC)cc(Cl)c(C(=O)NC23CC(C2)N(C(=O)C)C3)cc1Cl.CC(N)=O.S N(C(=NCC(=O)NC1CCC1)N1CCC(CSC)C1)C(COC)C Cn1ncc2cc(C(=O)NC3CC4(CCN(c5ncnc(Cl)c5CO)C4)C3)sc12 C(=O)(C(CC)CCOC)NC1(CO)CN(C(c2c(CC)cccc2)=O)C1 N1(C(C)=O)CCN(S(=O)(=O)NC(c2[nH]nc(C(F)(F)F)c2Br)=O)CC1 c1(C(N(CC(C)(C)NC(c2c(SC)cccn2)=O)C)=O)cc2n(n1)CCOC2 Cc1nc(C(=O)NC(CCF)C(=O)N2CC(C)(C)C2C2CC2)c(C)s1 C1(CNC(CC(=O)N(C)C)=O)CN(C(=O)C(O)Cc2ccccn2)CCN1C C1(NC(=O)CC2CN(C(c3ccc[n+]([O-])c3)=O)CCO2)CC(C2CCC2)C1 N1(CCOC)CC(C(=O)NCC(c2ccncc2)(C)O)CC1=O c1(C(N2CC(n3ncc(NS(CC#N)(=O)=O)c3)C2)=O)ccc2cnccc2c1 c1(C(=O)NCC2CN(C(c3cnc(C)o3)=O)C2)cc(C(C)C)ccc1F c1(CC)nn(C)c(C(=O)NC(C)(C)CCCNC(=O)CC=O)c1Cl.C1CC1 c1(C(N(CC(CNC(c2cnc(C)nc2O)=O)C)C)=O)cnn2c1NCCC2 c1(N2CCCCC(C)C2)[nH]c(=NCCc2cc(O)n(C)n2)nc2sccc12 CC#CCCCC(=O)N1C2CCC1C(CNC(=O)C(C)NC(c1cccs1)=O)C2 c1(CC)ccc2[nH]c(C(N3CCC(O)(C(=O)NC4(C)CC4)C3)=O)c(C)c2c1 c1(OC)cc(CC(N2CCC(O)C2)=O)ccc1O.C1(CC(=O)N)NC(=O)CNC1=O CCC#CC(C)(C)NC(C1CSCCN1C(=O)CCCOC(C)(C)C)=O C1(O)(CNC(C=Cc2c(C)n(C)nc2)=O)CCCN(C(=O)Cc2cnoc2)CC1 C(=O)(C(C)CC1CCCC1)NC1(CC=C)CCOC1.c1(CC=O)cnnn1C.N C1CC2(CCCCN2C(C2CC3CCC(C2)C3)=O)C1.C(CC=O)NC(=O)NC.N c1(C(=O)NCC(C)(C)NC(c2cnn(CC)n2)=O)nc2c(Br)cncc2[nH]1 Cn1cc(CC(=O)NCCCOCCC(=O)NC2CC(SC)C2)cn1 c1(C(=O)NC(CNC(CCC#C)=O)(C)C2CC2)cncc(P(C)(C)=O)c1 N1(C(C2C(C)C2)=O)CCOC(CCNC(=O)CCCc2cccs2)C1 C#Cc1ccc(C(=O)NC2CN(C(=O)CSC)CC2C2CC2)c(OC)c1 N#Cc1cccc(NC(C2(CNC(c3cc(O)ncn3)=O)CC2)=O)c1[N+](=O)[O-] n1(C(C)C)ncc(C(=O)N(C)CC2CCCN2C(C2CCC2)=O)n1 c1(C(=O)NC(C)CC(C)NC(c2n[nH]c3c2CCC3)=O)cc2n(n1)CCCC2O C=CCC(CC(C)C)C(=O)NCC1(C(=O)Nc2cccc(N=[N+]=[N-])c2)CC1 c1(C(N(C2CCN(C(c3cccc(F)c3)=O)C2)C)=O)coc2c1C(O)CCC2 c1(C(N2CC(CCNC(c3cn(CCO)nn3)=O)C2)=O)ncccc1CO c1(OC)cc(C)c(Cl)cc1C(=O)NC(C)CCO.C(=O)C(=O)N=S(C)(C)=O C1(NC(CCCNC(CC(C)SC)=O)=O)CN2CCCC1C2 c1(C(C=O)C2CC2)ccccc1.C1CCC1.C(C(=O)NC)=CC=CCC N1(C(C(=COCC)C#N)=O)CC(C)CN(C(=O)CC2(OC)CC2)CC1C C1(NC(CCC2CC(C)C2)=O)CCC(C(=O)NCCCC(C)CO)CC1 C(=O)(CS(=O)C(F)(F)F)N.c1(OC)cccc(Cl)c1C(=O)NCC=CC c1(C(N2CCC(NC(CC(CC)(C)C)=O)C(F)C2)=O)cnc(N)c([N+](=O)[O-])c1 O=C1CCCC2C(C(N3CCC=C(CNC(=O)C(=C4CCCCC4)F)C3)=O)C12 N1(C(CCOCC)=O)CCN(C(=O)CCOc2ccc(Cl)c(C)c2)C(CF)C1 N1(C(C#CC(C)C)=O)CCC(O)C(NC(C2CCCN2CCC(C)C)=O)C1 c1(NC(CC2N(C(C(C=C)CC)=O)CC(O)C2)=O)cc(C)c(F)cc1C C(CCCCC(=O)NC1CC2(C1)CC(NC(C1CC(SC)C1)=O)C2)OC C1(CNC(c2n[nH]cc2Cl)=O)CN(C(c2cncc(Br)c2)=O)CC1O C1(NC(C(CCC)O)=O)CCC2CN(C(=O)C(F)(F)C3=CCOCC3)CCC2C1 c1(C(C(=O)NCCC#N)N(C2CCCC2C)CC)cnc(C(C)O)s1 S(=O)(=O)(c1cccnc1NCCC1=CCCCC1)NC(C)C(C)S(C)(=O)=O Cn1nnnc1C(C)(CC1CCCCC1)NC1CONC1=O C1(C(=O)NC2C=CC(CO)C2)(NS(=O)(=O)C2CC2)CCOCC1 C1(c2n(CCC3(C)CC3)nnn2)(NCCC(F)(F)F)CCCCC1CCCO C(=O)(CN=c1cc[nH]cc1)NC(COC)CC(N1CC2CSCC2C1)=O N1(CCC)CCCC2C(NC(c3cnc(CC)s3)=O)C(C)(C)C12 C(=O)(C(C)(CO)NC(=O)C(C1CCC1)OCC)NC1(C)CC(=C)C1 C12(C(=O)NCC(=O)NC3CCCC3)CCC(CC1)N(C(=O)C1=CCCCC1)C2 CCCC(C(=O)NCCCCNC(c1cnc(CC(C)C)[nH]1)=O)C(C)C c1(OC)ccc2c(c1)OCCN(c1nccc(=NCC(CCSC)OC)[nH]1)C2 C#Cc1ccccc1CC(=O)N(CCC(=O)NCC(C)(C)CCOC)C CC(C(=O)N1CCCC(C(=O)NCCSC(F)F)CC1)S(C)(=O)=O CC(=NO)C1CC(C(=O)NCC(C)Nc2ncc(F)c(-c3ccsc3)n2)C1(C)C C1(NC(=O)NCCCS(C)=O)CCCC(c2ccccc2)C1 C1(CNC(c2cc(F)c[nH]2)=O)(NC(C2CCC(F)(F)C2)=O)CCCCC1 c1(CCC)nc(=NC2CCN(C(=O)CC3CCC4CC4C3)CC2)s[nH]1 c1(C(N2C(CN(C(=O)CC3CCCC3O)C)CCC2)=O)ccc(NCCO)cc1 C(=O)(C(C)(O)CC(C)C)NC1CC2CC(NC(c3c(C)nncc3)=O)C1C2 C(=O)(N=c1[nH]sc2ncccc12)C1N(C(C(OC)OC)=O)CC2(CC2)C1 C12(NC(C34N(C(c5nc(OCC)oc5)=O)CC(C3)C4)=O)CCC(C1)OC2C C(CC(=O)NC(c1cccs1)C)(C(C)OC)NC(c1cccc(OC)n1)=O c1(CC(=O)NC2(CNC(Cc3n(C)ccn3)=O)CCOC2)cc(Cl)sc1Cl c1(C(=O)Nc2cccc(C(C)=O)c2)cc(Cl)ncc1.c1(C=O)cc(Br)c(C)s1.N C1(NC(c2cnc(OCC)s2)=O)CN(C(=O)C(O)C2CCC2)Cc2nccn2C1 C(c1ccc([N+](=O)[O-])s1)=CC(=O)NC1CCC(NC(C(C(C)O)(F)F)=O)C1 N1(C(C(C)Cn2ccnc2)=O)CC(NC(=O)Cc2ccsc2Br)C(O)C1 O=C1CCc2cc(NC(=O)NCc3cn[nH]c3)ccc21 c1(C(=O)OCC)cc(F)ccc1C(N1CC2CN(Cc3sccc3Br)C2C1)=O n1(CCC(N2C(CCCNC(CNC=O)=O)CCCC2)=O)ccc2ccccc12 c1(C(N2CCCC(C)C2CNC(=O)CCF)=O)cc2nc[nH]c2cc1N Cc1cnn2cc(C(=O)NC(CNC(c3ccc(Cl)cc3F)=O)CO)cnc12 c1(C(C(=O)NCCN(C(C2CC(C)(CC)C2)=O)CC)C)ccc(C)s1 C1(C(N2CC3CC3(CO)C2)=O)(CNC(CN(C2CCC2)C)=O)CCCCC1 CC1(C)CCOC1CCNC(C12CC1CCN2C(=O)CC1CCSC1)=O Cc1cc(C(=O)NC2C=CCN(C(=O)C(c3cccc(C)c3)O)C2)nc(Cl)c1 N1(C(c2c(C)nc(O)[nH]2)=O)CCC2CN(c3c(Cl)cccc3[N+](=O)[O-])CC2CC1 c1(C(N2CCCC(F)(CNS(=O)(=O)CCCCl)C2)=O)cc(Cl)c2cn[nH]c2c1 N1(C(C(=O)Nc2c(C)cccc2C)=O)CCC2CC2CC1.c1(C=O)csc(O)n1.N CC(CC(=O)N1CCCC(N(CCF)C(C2CN3CCC2CC3)=O)C1)C(F)(F)F C(=O)(C(C)(C)CC(=O)N1CC(NC(c2cccc(C)c2C)=O)CC(F)(F)C1)OC c1(COC)noc(CNC(=O)CC2CCC2)n1.C1(C(=O)N)CC(F)C1 C(=O)(CS(=O)C(F)(F)F)N1CCN(C(CNC(Cc2nc(=N)[nH][nH]2)=O)=O)CC1 c1(OC)cccc(C(O)C(N2CCCCC2C)=O)c1.c1(C=O)nc(=O)n(C)[nH]1.N C(C(CC(F)(F)F)NC(C1(c2ncccc2F)CCC1)=O)OC N1(C(CN(C(CC)=O)C)=O)CCC(F)(C(N)=O)CC1.c12ccc(cc1)SCC2=O Cc1cc(C(=O)NCCC(C)NC(c2cccc(C(C)C)c2)=O)ccc1[N+](=O)[O-] C=CC(C)(CC)C(=O)NC(C)C(CO)NC(c1ccc(OC2CCCC2)nc1)=O N1(C(C2C(NC(c3ccoc3)=O)CC2)=O)CCOC(CC2CC2)C1 C1(C(=O)NCC(CC)N(C)CC)(NC(=O)CN(C)C(N)=O)CCCC1 C1(C(=O)NCC(C)CNC(=O)C(C)Cn2ccnc2)CCC(F)CC1 C1(CC)CN(C(C2CCOC(=O)N2)=O)CCN1C(=O)CCCCN1CCOCC1 N1(C(C2CCC(NC)C2)=O)CCOCC(NC(=O)CSCCOC)C1 N1(C(c2c(CC)n(C)nn2)=O)CC2(C=C(C(=O)N(CCC(N)=O)C)CO2)C1 N1(C(C(C(C)O)C)=O)CCN(C(C2(CO)CC(F)(F)C2)=O)CC(C)(C)C1 C(=O)(C(C)C1CCC1)N(CC(=O)NCC(C1CCC1)OC)CC(C)C c1(CC)cc(F)ccc1C(=O)NC1CC(C)C1.c1(C(=O)N)cc(O)ccc1 c12cc(cc(Br)c1)CO2.C1(F)(C(C)(C)C)CCN(C(=O)C2CC2)C1 C1CN(C(c2csc(Cl)n2)=O)C2(CCOCC2)C1.C1(CC)CN(CC(=O)NC)C1 N1(C(C(C)c2cccs2)=O)C(CC(=O)NC(CCO)C(F)F)C2CCCC12 C(=O)(C(C(C)(C)C)OC(C)(C)C)NCC(C)(C)NC(C1CC1F)=O N1(C(C2CCCN(CC)C2)=O)CCN(C(=O)CC(F)F)C(C2CCC2)C1 C12(C(N(C(C)CN(C(=O)Cc3cncn3C)C)C)=O)CCC(C1)C2(C)C C(C(C(=O)NCCCNC(c1ocnc1C)=O)N(C)C)OC C12(NC(C3CCN(C(c4c(C)cn(C)n4)=O)C3)=O)CC1COC2(C)C C(CC(C(=O)N(C1CC(NC(c2[nH]cnc2C)=O)C1)C)NC=O)SC CCN=C(NCCCNC(=O)NC1CCCC1)N1CCCC(C2(C)OCCO2)C1 C1(c2nnnn2C(C)(C)C)(NCCc2n(C(C)C)cnn2)CCOCCC1C C1(C#N)(C(=O)N)CC(F)(F)C1.CN1N=CC(CC(N2CCC(CC)CC2)=O)C1=O C1(NC(c2c(C)cccn2)=O)CCC2CCN(C(=O)C(C)(C)C(C)(C)C)C1C2 C(=O)(C(C#N)C(C)(C)C)N1CC(C(=O)NCCCCCCF)(COC)C1 c1(CC)cc(C(=O)N(CC(C)NC(=O)C=Cc2ccsc2)C)ccc1Cl N1(C(c2cnc(C)s2)=O)CC2CCCC1(CNC(=O)C1=CC(C)(C)C1)C2 S(=O)(=O)(c1cccc(C(N2CCCC(CC3C(NC)COC3)C2)=O)c1)NC N1(CCC)CCCCC1C(=O)NC1CCC(NC(c2cnc(C(C)C)s2)=O)CC1 C1(NC(CC2C(C)(C)C2)=O)CCC12CCN(C(c1ccc(F)cc1)=O)CC2 c1(C(=O)N)ccc2nc(C)sc2c1.C(CCOCC(=O)NC1CC1C)OC C(=O)(C1=C(F)CN(C(C2(C)CCOCC2)=O)CC1)NC(C)Cc1ncn(C)n1 Cc1c(C#N)sc2ccc(NC(=O)NCc3cnc(C(C)C)nc3)cc12 NC(=O)CCCCC(=O)NC1CC(CNC(C2(n3ccnn3)CC2)=O)C1 N1(C(CC2N(C)CCOC2)=O)CCN(C(c2n[nH]c3c2CSCC3)=O)CC(O)C1 Cc1cccc(Br)c1C(N1CC(NC(C2CCN2C2CCCC2)=O)C(C)C1)=O c1(NC(=O)Cc2ccc(C3CCC3)cc2)cccc2c1OCC2 Fc1cc(Br)c2c(c1)N(Cc1nnnn1CC1CCOC1)CCO2 CC#CCCCC(=O)NC(CCN(C(=O)C(C)NS(C)(=O)=O)C)C(C)C C12(NC(C3CCC4(CCC4)O3)=O)CCCCCC1N(C(c1cnsc1)=O)CC2 CC1CCC(NC(=O)CCc2cnn[nH]2)CN1C(=O)CNS(=O)(=O)C1CC1 c1(CC(=O)OCc2nccc(N)c2)c(F)ccc(Br)c1F Cc1ccc(C(=O)C=CC(=O)NCCCN(C)C(C2NC(=O)CC2C)=O)cc1 c1(CC(N2CCC(CNC(c3nc(C#C)sc3)=O)C2)=O)cc(F)ccc1O N1(C(CCCOCC)=O)CCN(C(C2CC(C)(C)C2)=O)C2CC12 C(N=c1nc2sccc2c(N(CC(C)C)CC(C)C)[nH]1)C1(CCC)CCC1 C1(NC(C2C(CCC)C2)=O)CC2CC(NC(c3ccc(F)cc3C)=O)CC12 Cc1nnc2cc(N3CCCC(C4CC4NC(C4CCCSC4)=O)C3)ncn12 C1(C(=O)NCC(C=C)O)CCN(C(C2CC3C=CC2O3)=O)C(CC)C1 N1(C(C(C)=CCC)=O)CC(C(=O)NC2CCCC2O)CC1(C)C N1(C(c2nc(C)c(C#N)cc2)=O)CCN(C(=O)COCCN(C)C)CC(C)(F)C1 n1(CC(=O)NCCC)cnc([N+](=O)[O-])n1.C1(C)(CCC=O)CC1(F)F.CC C(C(CC1CCCC1)C(=O)Nc1cn(C)nc1Cl)NC(CCCNC(C)=O)=O C12(C(=O)NC3CCN(C(C(F)=CCC)=O)C34CCC4)CC(C)(C1)OC21CCC1 O=C(C1=CCOCC1)NC(Cc1cc[nH]n1)C(=O)NC1CCCC1CF C(=O)(C#CC1CCCOC1)NC(C(C)NC(C1(CC(C)C)CCC1)=O)CO c1(C(N2CCC(CC)C2C(=O)NC2C(C)C2C)=O)cc(C#N)oc1C C1(NC(C2(OCC)CCOCC2)=O)CN(C(=O)C#CC2CC2)C2(CCOC2)C1 C1(C=O)CC2CCC(C1)C2.C1(NC(C(C)NS(CC)(=O)=O)=O)CCCCC1.C C12(NC(=O)C(O)CCl)CCCC1N(C(c1cccc3ncsc13)=O)CC2 N1(C(CSCCOC)=O)CC(CNC(=O)Cn2cc(C)cn2)C(O)C1 N1(C(C(C)C)=O)CC2CCC(C1)N(C(c1ncc(C)cc1C)=O)C2.C(=O)(OC)N Cn1cnc2c(NCc3ccc(Cl)cn3)nc(N3CCCC(C#N)C3)nc12 CC(C)C(C(=O)N1CCSCC1CO)NC(=O)C(c1cnn(C)c1)=O C1(O)(CC(=O)N(C)C)COC(C)(C)C1.C1CCCN1C(C1(CCF)CC1)=O c1(C(=O)NCCCC=C)cnc2sc(C)c(C)n12.C(c1ccncc1)=CC(=O)N C1(O)(CCNC(C=CC(CC)=CC)=O)CCN(C(=O)C(O)CCS)CC1 CCCC(C)NC(=O)CCNC(=O)CC1CC1(C)C N1(C(CNC(C=Cc2n(C)ncc2)=O)=O)CC(C(N)=O)C2(CC2)C1 c1(OC)cc(C=CC(=O)N(C2CC3CC2N(C(=O)CCCF)C3)C)ccc1F N1(C(C2(C)ON=C(C)C2)=O)CC2CCN(C(c3ccc(C#N)cn3)=O)CC2C1 N1(C(CC(=O)OCC)=O)CCCC2CN(C(=O)C(c3c(C)n[nH]c3C)C)CCC12 C1(NC(C(CC)CC)=O)C2COCC1CC(NC(c1cc(C3CC3)on1)=O)C2 CC1CC(CC(=O)N(C(C)CNC(c2nncn2C2CC2)=O)C)C(C)O1 C=CC(CCC)CC(=O)NC1(C(=O)NC2CC(CN(C)C)C2)CCCC1C N1(C(CC(C(C)(C)C)NC(CC(CCCC)O)=O)=O)CCn2cc(C)nc2C1 C1(CNC(C(COC)C)=O)COCCN(C(c2cccc(-n3cccn3)n2)=O)C1 C(=O)(CCCC(C)NC(=O)CN=[N+]=[N-])N(CC(=O)N(CC)CC)C C(C(F)(F)C(=O)N1CC(NC(C2CNC(=O)O2)=O)C(SC)C1)OC c1(C(N2CC(NC(C(C)(C)F)=O)C(O)C2)=O)cc(Br)ccc1O C1(C(=O)NCCC(CNC(c2sccc2F)=O)O)COc2ccc(Cl)cc2C1 CN1CC(C(=O)NC(C)(C)CN(C)C(C2CCCS2)=O)CCC1=O C1(NCCN(C(C)C)CC)CCC2(CNC2)OC1 CC(C)(C)CCC(F)C(=O)NCC1(O)CCC1.C1(C=O)CS(=O)(=O)C1.C CC(C)C(CNC(=O)Cn1cc(Br)cn1)NC(c1ccc(C2CC2)o1)=O CC#CC1CCN(C(=O)C(C)(C)CNC(=O)C(C)OCC)C1 N1(C(C2(C)CCC3CC3C2)=O)CC(NC(C2CCCN2C(N)=O)=O)CCC(O)C1 C1(C(=O)NC2(C)CC(NC(c3n(CC)ncc3)=O)C2)CC2(CCO1)CC2 c1(COC)nc(Cn2nnnc2N2CCC(Nc3ncccn3)C2)cs1 c1(C(=O)N)cc(O)nc(Cl)c1.C(C(C(=O)NCC(C)CO)NC(C)=O)OC c1(C(=O)NC2(CO)CN(C(CC3CCC(C)C3)=O)C2)sc2cccc(F)c2c1Cl N#CC1(C(N2CC(F)(CNC(=O)C#CC3CCCO3)C2)=O)CC12CCCC2 Cc1cc(=NC(=O)C(=O)NC2(C3CC3)CCN(C(=O)Cc3cnoc3)C2)[nH]o1 C(=O)(C(=O)CC(C)C)N(CCC(NOCCCCC)=O)CCO Cc1cc(Br)cc2c1CN(C(=O)NCC1(c3ccc(F)cc3)CCCC1)CC2 CC(C)C(O)C(F)(F)C(=O)NCCCN(C(=O)Cc1csc(C2CC2)n1)C C1(NC(c2cn(CCO)nn2)=O)CC2CCC(C1)N2C(=O)Cn1cc(Cl)cn1 c1(CC(=O)NCC2CC(CNC(C3(N(C)C)CC3)=O)C2)sccc1Cl C(=O)(C1=C(Cl)CCC1)NC(C1CCCC1)CNC(C(C)(C)n1cc(Cl)cn1)=O C=CC1CN(C(=O)CCSC)CC1NC(=O)C(C)C(C)(F)F c1(OC)ccc(C(N2CC(CNC(=O)C(F)C3CCC3)CC2C)=O)nc1Cl N1(C(c2c(CC)scc2)=O)CCC(NC(c2c(Cl)c(C)nn2C)=O)C(CO)CC1 CCCC(C(O)C(=O)NCC1(CF)CCC1)NC(=O)CSC(F)(F)F C1(C(CNC(CCSCC(C)C)=O)C)CCN(C(=O)C=Cc2cn[nH]c2)CC1 N1(C(C(C2CCN(C(c3cc(CC)oc3C)=O)C2)F)=O)CCCOCC1C C1(CC)CC(C)CN1C(C1CCC(CNC(=O)CCc2cncn2C)O1)=O C1(c2ccccc2Cl)(C(=O)NC(C)CNC(=O)CC2C=CCC2)CCOCC1 C1(CNC(CCN(C(=O)CCC2CC(OC)C2)CC=C)=O)CC12CCCCC2 Cc1cc(Cl)cc([N+](=O)[O-])c1C(=O)NCCN(C)C(c1ccc(C)n1C)=O CC(C)C(CO)C(=O)N(C)CCOCCNC(=O)C(CC(C)C)n1ccnc1 CCC(C)(CNC(=O)COCCCOC)C(=O)N1CCC(C#N)CC1 C1(OCC)CC(N(C(c2ccsc2Cl)C(=O)NC2CCC2)C)C1(C)C N1(C(c2cnn(C)c2C(F)F)=O)CCOCC(CNC(c2cccc(O)n2)=O)C1 C#Cc1cc(C(=O)OCc2cc(C(=O)O)co2)cc(Br)c1 C(=O)C(C)CC(N)=O.Cc1noc(COCC(=O)NC(C2CCCC2)C)n1.N C1(C(N)=O)CCC(CCC(=O)NC(C)C2CCC2)O1.n1(CCC=O)cc(C)cn1 N1(C(CNC(CCNC(=O)NC)=O)=O)CCCSCC1C.c12ocnc1C2 C=CC1(C(=O)NC2CCN(C(=O)Cc3c(Cl)cnn3C)CC2O)CCCCC1 c1(C(N(CC(=O)NCc2ccn(CC)n2)C(C)C)=O)ccc(C)n1C Cc1coc(C)c1C(=O)NC1CC(N(C(=O)C(C)C)C)C1.[SH](C)(=O)=O.N C1(C(N(C2CN(C(c3cnc(C(C)C)n3C)=O)C2)C)=O)CC1C1CC(F)(F)C1 C1(CN)CCN(S(=O)(=O)NC(=O)C=CC(=O)Nc2ccc(F)cc2)CC1 c1ccc(I)cc1C(F)(F)F.N1(CC)CCN(CCCNCC(C)C)CC1 Cc1ccc(-c2n[nH]c3c2CN(C(c2n[nH]c4cccnc24)=O)C3)c2cn[nH]c12 CS(=O)CCC(=O)NCC1(F)CN(C(=O)CCOc2ccc(Br)cc2)C1 Cc1cc(=O)n2[nH]c(C(=O)NCc3nccc4ccccc34)cc2n1 Cc1ccc(C)c(C(=O)NCC(C2CCCCC2)NC(=O)COCCCF)c1C C(=O)(CCCCC)NC(CC=C)CNC(=O)CCCOc1cccc(C)c1 C1(C(C)NC(=O)C(C)(C)N2CCCCC2)CN(C(=O)CCCN(C)C)CCO1 Cc1c(C(N2CC(NC(c3ccc(F)nc3F)=O)C(C)C2)=O)c(C(F)F)nn1C n1(CC(=O)NCCC(CNC(C(C(C)O)N(C)C)=O)O)nc2c(n1)CCCC2 c1(OC)ccccc1OC(C)C(=O)NC1CC(NC(c2cc(C)ns2)=O)C1 O=C1CCc2c(C(N3CCCC(NC(=O)CC4CC4)C(F)C3)=O)cccc2N1 CCC(C)(CO)C(=O)NC1CCC(NC(c2nc(SC)ncc2N)=O)CC1 C1(NC(c2c(C)n(C)cc2)=O)CCN(C(c2ccc(C(F)F)cc2F)=O)CC1C N1(C(c2c(CC)nc(C)o2)=O)C(C(N2CCCC(C)CC2)=O)CCC12CC2 N1(C(c2cc(C)nc(C)c2)=O)CC2CC3CC2C1C3NC(C1CC2(CCC2)C1)=O C1(C)(CC=O)CC(F)(F)C1.C1(C(=O)NCCOCC)(OC)CCSC1 C(c1cc(OC)c(OC)cc1OC)=CC(=O)N(C(CCNC(CC)=O)C)C Cc1cc(C)c2ncc(C#N)c(N3CCOC(CNC(=O)CSC(F)F)C3)c2c1 N(C1CCc2cc(F)c(F)c(F)c21)Cc1ccc(C(C)C(F)(F)F)cc1 C12(C(=O)NC(CCC)C(C)C)CC(O)(C1)C(c1ccccc1)O2.C(=O)OC c1(C=O)cc([N+](=O)[O-])cnc1N.c1(CC(=O)NC(C2(C)CC2)C)ccns1 CN=c1[nH]cc(C(N2CCC(C(=O)NCC(C)(F)F)C2C)=O)o1 N1(C(C(F)=C(C)C)=O)CC(CNC(C2CCC23CCOCC3)=O)CC12CCC2 Cc1ccc2c(c1C)OCC2NC(=O)C(N1CCC12CCSCC2)=O C1(C(=O)NCCOCCCNC(C2C(C)OC(=O)N2)=O)CCc2nncn2C1 N1(C(CCC2CCN(C(CSCCC)=O)C2)=O)CC2C3CCC(C3)C12 C1C(C)CCCN1C(=O)C1=COCCC1.c1(C(=O)OC)cncc(C(=O)NC)c1 CN1C(=O)OCC1C(N1CCCC(N(C(=O)CCN2CCNC(=O)C2)C)C1)=O CCC(CN(C)C)CC(=O)N(C(C)CCNC(C1(C#N)CC=CC1)=O)C c1(N2CC3C(C(=O)NCc4c(CC)nccn4)C3C2)nc(SC)nc(C)c1Br C1(NC(C(C)C(F)F)=O)CC(C(=O)NC(Cc2ccco2)CO)=CC1O CCCCC(C)CCC(=O)N(C(C)C(=O)NC(C)C)C C(c1cccc(O)c1)=CC(=O)NCC(CNC(C1(C(N)=O)CCC1)=O)F N1(C(CCOC)=O)CCOCC1c1ccc(C(N2CC(CC(C)C)C2)=O)n1C c1(CC)onc(C(=O)NC2CCC(C)C2)c1C.n1(CC(=O)N)ncc(Br)c1C C1(C=O)CN=C2N1C=NN=CS2(=O)=O.Cc1nn(CC#N)c(Cl)c1C=CC(=O)O Cc1nc2ccc(C(N3CCC(COCC(F)(F)F)CC3)=O)cc2n1C c1(N2C(CC(=O)NCC3N(C(C)=O)CCC3)CCC2)ccc(C#N)cn1 C1(C2CC2)CCN(C(=O)C(C)CSC(F)(F)F)C1.Cc1nnc(C(=O)NC)s1 c1(C(=O)NC23CC(C(=O)NCCCN4CCOCC4)(C2)C3)ccc(I)cc1O C(=O)(CCCC#Cc1ccccc1)N(CC(C)NC(=O)C=C1CC1)C CS(=O)(=O)c1cc([N+](=O)[O-])c(C(N2CCC(c3ccc(Br)cc3F)CC2)=O)s1 N1(C(CNC=O)=O)CCN(C(C2(Sc3ccccc3)CCCC2)=O)CC12CCC2 C=C(C)C1OCCC1C(N1CCN(C(C2C(C)(C)OC2(C)C)=O)C(CC)C1)=O C1(C(=O)Nc2c(OCCC)cc(C)c(Cl)c2)COc2cc(Br)ccc2O1 N1(CC)CCCCC1C(=O)N(CCC(=O)NC(c1ncc(C)cn1)C)CCCO C12(CNC(=O)CCc3ccc(Cl)cc3)CCCC1N(C(c1cn[nH]c1)=O)CCC2 C=C=CCC(=O)NCC(CNC(=O)C(C)OCC1CC1)CO Cc1nc2cc(OS(=O)(=O)CCC(F)(F)F)ccc2s1 c1(OC)ccccc1N1CC(NC(c2cccc(OCC(C)C)c2)=O)CC1=O c1(OC)cc(C(=O)NCCO)n(C)n1.C1(C(N(CCC)C)=O)OCC1(C)C c1(C(=O)NC(CC(C)NC(Cc2c(C)con2)=O)C)cnn2c1C(=O)NCC2 CCC(CNC(c1cn[nH]c1)=O)(CC)NC(c1ccc(NC(=O)N)cc1)=O CC(C)C(C)C(C)CC(=O)N1CCC(CN(C)C(c2ccc([N+](=O)[O-])s2)=O)CC1 N1(C(c2n(CC)ccc2)=O)CCC(N=[N+]=[N-])(C(=O)NOCCCO)C1 CC(C)CS(=O)(=O)CC(=O)N1CCC2CCCC12CNC(c1ccsc1)=O CC1CCN(C(C2CC2(C)Br)=O)CC1NC(c1ccc(OC2CC2)cc1)=O Cc1cc(F)cnc1C(=O)NC1CCCN(C(c2nnn(C)c2C(F)(F)F)=O)C1 c1(NC(N2C(CC(=O)NC(c3cn(C)cn3)C)CC2)=O)cnnc(O)c1 c1(C=O)cn(C)ccc1=O.C1(C(N(CC)Cc2cncn2C)=O)(C)CCCO1 N1(C(C(C)CSC(F)(F)F)=O)CCCC2(C1)CN(C(c1cn3c(n1)CCC3)=O)C2 c1(-c2cn(C3(C=O)CCC3)nn2)c(C)nn(C(F)(F)F)c1C.C(=O)C.CC.N c1(N(C(C2C=CCN(C(c3ccc(C)cc3)=O)C2)=O)C)cccc(C#N)c1 C#Cc1ccc(C(N2CCCCC(NC(C3CCCCS3)=O)C2)=O)c(OC)c1 c1(NC(C)=O)ccc2c(c1)OCC2NC(N1CCN(S(C)(=O)=O)C(C)C1)=O C1N(C(c2nc(C3CC3)cs2)=O)CCCC1(C)C.CC(C(=O)N)OCC1CC1 C=C(F)C1(CC(=O)NC2CCCCC2CNC(c2cnsc2C)=O)CCC1 CC(C(C)(C)C)=CC(N1CCC(NC(c2c[nH]nc2C)=O)C1)=O c1(OC)ccc(NC(c2nc(NCc3cccc(OC)n3)cn2C)=O)c(C)c1 c1(C(N2C(CNC(=O)CC3CC4(CC4)CO3)CCCC2)=O)ccc(Cl)c(Cl)c1 C1(C(N2CC(NC(C3CC(C)OC3)=O)(CO)C2)=O)CCCC(F)(F)C1 c1(C(C(N2CC(CC(C)NC(=O)CN)C2)=O)=O)cccc(N)c1.c1cnc[nH]1 c1(C2CCC(NC(C3(c4ccncc4)CC3)=O)C2)cc(F)cc(F)c1 c1(CC)nnc(C)cc1C(=O)NC(CNC(=O)CC1(C=O)CC1)CC N1(C(c2c(C)n(C)nn2)=O)CC2(CNC(c3cncnc3)=O)CC(F)(C1)C2 C1(CC)(NC(c2ccnc(F)c2N)=O)CCN(C(C2(C)CC=CCC2)=O)CC1 c1(CN(C)CC2CCCN2C(C2CCCC(F)(F)C2)=O)cc(F)ccc1F C(=O)(C1CN(C(=O)CCc2ccoc2)Cc2nnn(CC3CC3)c21)NC(C)CO CC(=NO)C1CC(C(=O)NCCNC(=O)Cc2cnc3n2CCOC3)C1(C)C CC(C)C(CNC(C12C=CC(CC1)C2)=O)C(=O)N(C)CC1CC1(F)F CC1CN(C(=O)CC2CC3CC3C2)C(C)CN1C(c1cc(C#N)cn1C)=O C(CN=c1[nH]c2ccc(F)cc2s1)(CC(C)C)NC(CCCOCCC)=O C1(C(N(CCCCO)C)=O)CCN(C(C2(N(C)C)CCCC2)=O)CC1(C)C c1(C(=O)NCC(C(C)C)(C)NC(=O)C(O)Cc2ccccn2)cnc(Cl)cc1N C1(C(N(CC#C)CC2CC2)=O)CCN(C(C2CC2=C)=O)C1CC C1(c2cn(CCC(=O)OC)nn2)CC12CCN(C(c1csc(Br)n1)=O)CC2 n1(CC)ncc(C(N2CCCC2C2(NC(=O)CCC3CC3C)CC2)=O)c1Br c1ncnc2[nH]cnc12.Cc1n[nH]cc1C(=O)NCC1CC(NC(=O)CS)C1 c1(CC)cnc(C(N2CCC(N(C(=O)C(C)Oc3cccc(F)c3)C)C2)=O)nc1 C1(C(=O)NC(C)(C)CCO)(NC(c2c(COC)ncs2)=O)CCCCC1 c1(C=O)cccc2[nH]ccc12.C(=O)C(C)N(C)C.C(=O)(CC)N(CC)CC.N C1(NC(CCC(C)SC)=O)CCC12CCCN(C(c1cccn3cnnc13)=O)C2 CC1CC(C(N2CCC3(C2)CN(C(c2cccn(O)c2=O)=O)C3)=O)CCS1(=O)=O c1(C=O)ccc2c[nH]nc2n1.c1(SCC)cccnc1C(=O)NCC1CC1.N N1(CC(=O)NC)CCC(NC(=O)CCCOc2ccc(C)c(C)c2)CC1C CC(C)CC(C(=O)NCC(C)N(C(=O)CCOCC(F)F)C)N1CCCCC1=O c1(C(N2CCC(NC(CC3ON=C(CC)C3)=O)C2C)=O)ccc(OC)c(OC)n1 CC1(C(N2CCCC(CNC(=O)CCc3ccncn3)CC2)=O)CCCC1(F)F c1(OC)ccc2c(ccn2CC(=O)N(CC(O)CN(C)C(C2CCOC2)=O)C)c1 N1(C(CC(C)n2ccnc2)=O)CCN(C)CC1C(N1CCC2C(O)CC12)=O CC1CCN(C(=O)CCc2csnn2)CC1CNC(c1cnoc1C1CCC1)=O N1(C(CC(C)O)=O)CCC2C(CCN2C(c2cc(F)cc([N+](=O)[O-])c2)=O)C1 c1(C(N(C2CCN(C(C3CCC4(C3)N=N4)=O)C2)CC)=O)cc(C)oc1C N1(C(C2C(=C)C2)=O)CCc2sc(C)nc2C1.C1(C=O)CN(S(C)(=O)=O)C1.N c1(C(=O)NCC2CC(OC)CN2C(C2CCC2)=O)nn(C)c2c1CCCC2.C C(CCC)N(C(CC1(COC)CC1)=O)C.C(=O)(C(C1CCC1)C1CCC1)N C1(NC(c2cc(Cl)ns2)=O)(CO)CN(C(c2csc(C3CC3)n2)=O)C1 c1(NC(c2cc3ccccc3s2)=O)nc2ccc(O)cc2s1 CN1C(=O)Cc2cc(NC(C3CC34CCN(C(c3ccc(Br)s3)=O)C4)=O)ccc21 C1(c2n(CCOC)nnn2)(NCc2c(Br)nnn2C)CCC2CCC12 N1(C(COCC(=O)OC)=O)CC2CC2C1.C1(C(=O)N)CCN(C2CC2)CC1 C1(C(N2CCC(c3cn(-c4cc(F)cc(Cl)c4)nn3)C2)=O)COCCC1(F)F Cc1cc(CC(N2CC(CNC(=O)C(C)OC3CCCC3)C2)=O)sn1 C(=O)(C1CCCn2c(C)cnc21)NC(CC=C)CNC(c1cccc(F)c1O)=O c1(CNC(Cc2scc(C)c2)=O)nc(C)c(C(=O)NC2CC(CCO)C2)o1 CC(C)CCCCNC(C1CCC(NC(=O)Cc2nc(=N)[nH][nH]2)C1)=O c1(C(N2CCC(N(C(C(CC=CC)CC)=O)C)C2)=O)cc2[nH]nnc2cc1OC c1ccccc1.C(CC1CC1)(C(=O)NCC1CC1NC(=O)C)OC.N C(=O)(C(F)(F)C1CCOCC1)NCCCCN(C)C(C1(Cl)CC1)=O C(CCSC)(C(=O)NC1(CNC(=O)CCCN2CCCC2)CCOC1)OC c1(C(=O)NC2COCC2NC(c2cc(O)nc(O)n2)=O)ccc2c(c1)CCO2 c1(C(=O)NCCC2OCCCN(C(C(C)C(C)(C)C)=O)C2)ccc(F)c(F)c1F C1(C(=O)OCC(C)(C)NC(C)=O)CCC(F)(F)C1 Cc1cn(CC(=O)NCC(CO)NC(C2CCCN2C)=O)c2ccccc12 c1(CC(=O)NC2CCCN(C(C3N(S(C)(=O)=O)CC3)=O)C2)c(F)cccc1F c1(NC)snc(C)c1C(=O)NC1CCCC1.C(=O)CCN(S(C)(=O)=O)C C1(OC)CN(C(=O)CCSC2CCCC2)CC1.C1(CC=CC=O)CCOCC1 C12(CC(=O)N(CCn3cc(C4(C)CCCC4)nn3)C)CCC(C(=O)O)(CC1)CO2 Cc1nnc2n1CC(C(=O)NC1(CO)CCN(C(c3ccc[nH]3)=O)CC1)C2 c1(C(=O)NCC2(F)CCN(C(CC(C)OC)=O)C2)ccc(F)cc1.C(C)=O c1(C(N2CCCN(C(c3ccccc3)=O)CC2)=O)ccc2c[nH]nc2c1 c1(C(=O)NC2C(NC(=O)C=CC3CCC3)CCC2)cccc(-n2ccnc2)c1 C(=O)(CCN(OC)C(=O)C=CCOC)NC(C1CCCC1)CC C1(CNC(CCCOC)=O)(CO)CCCN(C(c2cc(C)sc2N)=O)C1 N1(C(C(C2CCN(C(c3c(OC)scc3)=O)C2)(C)C)=O)CCSCCC1C N1(C(C2(CC#C)CCCC2)=O)CC(C)C(C)C1.c1(C=O)cccc(C(C)=O)c1 N1(C(C(CC)(C)OC)=O)CCC2(CC1)OCCC2NC(C1CC2(CCOC2)C1)=O n1(CC)nc(C)cc1C(=O)NCC1C=CCN1C(=O)CC1C=CCC1 CCCC(CCCNC(c1cccc(OC)c1C)=O)NC(c1ccsc1)=O C1(NC(CC2OCCN(C(c3c(CC)oc(C)c3)=O)C2)=O)(CO)CCCCCC1 C1(C(N(C2CCOC2)CC)=O)CC12CC(NC(C1CCSC1)=O)C2 C1(C2(O)CCN(C(C3CC4CCC3C4)=O)CC2)(NC(Cc2n(C)ccn2)=O)CC1 CC1CN(C(c2c[nH][nH]c2=N)=O)CCC1NC(c1cnnn1-c1ccccc1)=O N1(C(C(F)=CCC)=O)CCC(C2(NC(c3cn(C4CCCC4)nn3)=O)CC2)C1 C(=O)(C1Cc2ccccc21)N(CC(C)NC(=O)CCCCC(F)(F)F)C c1(C(=O)NC2CC(NC(c3c(SC)csc3)=O)C2)ccnc(C)c1 c1(C(=O)NC(C2(C)CC2)CN2CCOCC2)ccc2c(c1)CCOC2 c1(C(=O)NCC(CC)NC(=O)C(c2ccccc2F)C)c(C)ccn1C CCCC(C)(CC)NC(=O)CC1(C)CCN1C(=O)CN1CCCCCC1 c1(CCC)ccc(C(=O)NCC(C)NC(C2CC2(C)C(F)F)=O)cc1 C(=O)(C1=CC2CCCCC12)N(CCCNC(c1ccc(CC)c(CC)c1)=O)C N1(C(C2C(CCC)C2)=O)CCN(C(=O)CC(C)(C)O)CC1c1nccn1C C1(C=O)CCS(=O)(=O)C1.C1(N2CC(C(N(CCC)CC)=O)C2)CCOCC1 Cc1nn(CCC(=O)NC2CC(CNC(C3CCC34CCCO4)=O)C2)c(C)c1C c1(C(N2CC(C(C)NC(=O)CC3CCC(F)(F)C3)C2)=O)cccc2c1ncn2C c1(NC(C2(C(C)C)N(C(C(CC)COC)=O)CCC2)=O)ccc(F)cc1CO c1(C(N2CCC(NC(c3cnco3)=O)C(CO)C2)=O)oc2ccccc2c1Cl c1(CNC(CC)=O)ccc2c(c1)CCCC2NC(=O)C(=Cc1c[nH]cn1)F CC1(C)CC(C(=O)NCc2nocc2C=O)=NO1.C1CCCCC1C(N)=O.N CCCCCCC(=O)N1CCCC(N(C)C(C2CC3(CC3)CN2C)=O)C1 CC(C)CC(O)C(=O)NC.C1(O)CCCN(C(=O)C=CC(c2ccccc2)=O)C1 C(CCC(C)C)(C(=O)NCC1CC2(CC2)C1)NC(C(C)OCCC=C)=O C1(CC(=O)NCc2c(C(C)C)noc2)CCCCN1C(C1CC=CCO1)=O c1(C(=O)NCC2CC(C)C2)ccc(-n2cc(C3(O)CSC3)nn2)cc1 CCCC(CCCNC(C1(c2cccc(F)c2)CC1)=O)NC(=O)COC CCCCCC(F)C(=O)N1CC(C(N2CC(O)(c3nn[nH]n3)C2)=O)C(C(C)C)C1 C1(C(C=O)C)CCN(C(c2oc(C)cc2C)=O)CC1.C(C)(C)(C1(C)CC1)OC C(=O)(CCC(=O)c1ccc(Cl)cn1)NCCCN(C(C1CCC(C)C1)=O)CCO Cc1cc(CC=O)n(C)n1.C(=O)(C(C)CC1CCCO1)N1CC(C=O)C1.CC.N c1(C=O)cc(N)cc(F)c1.Cc1[nH]nc(C(C)C)c1C(=O)N(C)CCO.CC CC(C)C(F)(CNC(C1CC1C(F)(F)F)=O)C(=O)NCCN1CCCC1 N1(C(C2(CC)CCCC2)=O)CC2=C(C1)CN(C(c1cc(F)n(C)n1)=O)C2.CC N1(C(C(C)C2CCCC2)=O)CCC2(CCC2NC(c2nc(Cl)ccc2N)=O)CC1 C(=O)(C1=NOC(C)C1C)NC(CCC)CC(=O)Nc1cnn(C)c1OC C#CC1(C(=O)NC2CCC(C)(C)C2)CCN(C(=O)CNC=O)C1 N1(C(CCN(CCC)C)=O)CCCC(F)(F)C1.n1(CC(=O)N)cc(C2CC2)cn1 N1(C(c2c(CCC)n[nH]c2)=O)CCC2(CC(NC(=O)Cc3cccc(Cl)c3)C2)C1 c1(NC(CCc2c(C)cc(Br)cc2)=O)cc(Cl)nc2cnccc12 C1(NC(CC2CC(=O)OC2)=O)CCC2CN(C(c3snc(Cl)c3Cl)=O)CC2C1 c1(-c2nc(C(C(C)O)N)on2)cc(OC(C)(C)C)cc(Br)c1 c1(C(N2CC(CNC(CCCCC)=O)OCC2)=O)cnc(C2CCCC2)[nH]c1=N C1(NC(CC2CC(OCC)C2)=O)CCC(C)N(C(c2cccc(SC)n2)=O)C1 Cc1ccncc1C(=O)NCC(C(C)(C)C)NC(=O)CC(C)n1cccc1 c1(C(=O)NC(C)CNC(=O)Cc2c(F)cccc2Cl)cc2ccc(Cl)cc2[nH]1 C(=O)(C(F)(F)C(C)(C)O)N1C(CNC(CCc2nc(C)c(C)[nH]2)=O)CCC1 C(=O)(C(C)CC(C)C)N(C)Cc1n(CC)ccn1.c1(C(=O)N)cnc(C)nc1C c1(OC)ncc(C(=O)NCc2cncs2)cc1-c1ccnc(C)c1 C(=O)(C(C)C(C)NC(c1cccnn1)=O)N(CC(C)C)CCO C1(OC)CCC2(C(=O)N(C)CC3CC(F)CN3C(=O)Cc3ccsc3)CC12 C(C(C)CO)NC(N1CC(=C(C)C(F)F)C1)=O.CCC=O.C(C)(C)(C)C=O C(=O)(C(C)CC(=O)OC)NCC(C(=O)NCC(COC)(F)F)N(C)C c1(C(N2CC3C(N(C(c4nnn(CC)c4C)=O)C)C3C2)=O)cc(=O)c(OC)c[nH]1 c1(CN(C(CN(CCC)C(c2cc(Cl)cs2)=O)=O)C)ccncc1C N1(C(c2c(C(C)C)sc(Cl)n2)=O)CCC(C)C(C)C1.C(=O)(CCc1ccco1)N c1(C(=O)Nc2c(C)noc2)cnc(C(C)C)n1C CON(CCC(=O)NCc1ccc(F)c(O)c1)C(=O)Cc1cn[nH]c1 c1(C=O)cc(O)ccc1C.C1(CCOC)CCCN(C(C2C(C)C2(C)C)=O)C1.N C(=O)(C1CCCc2cc(O)ccc21)NC1C(NC(C=CCOC)=O)CCCC1 N1(C(NOCC(=C)C)=O)CCc2cc(S(=O)(=O)NC)ccc21 N1(C(C2(OC)CCOCC2)=O)CCC2(CC1)CC(NC(C1CCOCC1C)=O)C2 c1(C=O)csc(S(C)(=O)=O)c1.c1(SCC)cccc(CC(=O)N)c1.C1CC1 c1(C(N2CCCC(NC(c3c[nH]c(=NC)o3)=O)C2)=O)c([N+](=O)[O-])cnn1C C1(C)(C(=O)NC(C2C(C(N(C(CC)CC)CCC)=O)C2)C)COCCO1 C1(CC(=O)NCC(CNC(COC)=O)C)CCn2cncc2C1 C1(CNC(c2c(C)csc2)=O)CCC(NC(=O)CC2CC=CCC2)CC1 C=CCCCCCNC(=O)C(Cc1ccco1)NC(=O)C(CC)CC c1(C(=O)NCC(CO)NC(c2ccc(S(C)=O)cc2)=O)cnc2ccccc2c1 C1(C(=O)NCCC(O)CO)CCC(CNC(c2nc(Cl)cs2)=O)CC1 CC1(C)CC(NC(=O)CC2CCCCCC2)CN(C(=O)C2=CCOC2)C1 C1(OCC)CC(CNC(=O)C(C)N(C(=O)C(C)c2ccsc2)CC)C1 CC1CC(C(=O)NC2CCC2)N1C=O.C1(C=O)(CCF)CC1.C(C)(C)C c1(COCC(=O)NC(c2ccc(Cl)cc2)Cc2cnccn2)ccc(F)cc1 C(=O)(C1=CCCC(C)(C)C1)NC1C(CNC(C(C(C)C)OC)=O)CCC1 c1(OC)ccc(C(=O)NC2(CCNC(=O)C(C)C(C)O)CC2)c(Br)c1F N1(C(c2n[nH]c(C)c2C(F)(F)F)=O)C2CCC1C(CNC(c1nccs1)=O)C2 C1(c2cn(CCCN(C(C3(COCC)COC3)=O)C)nn2)CCCCC1O C1(CNC(CC=C)=O)CCN(c2ccc3nnnn3n2)CCC1(F)F c1(OC)cc(CNC(=O)C(C)C(C)NC(=O)CCc2ccncn2)ncn1 c1(C(C(=O)N(CCCNC(=O)CC)CC)(F)F)cccc(Cl)c1F.C=O.N CC(C)C(CN(C)C)C(=O)N1CCC(CO)(C)CC1.C1(C(=O)N)C2CCCCC12 N1(C(=O)NC2CCCC2O)CCOC2(CCCCCC2)C1 Cc1cncc2cc(C(=O)NCC3CC3NC(C3CCc4ncnn4C3)=O)sc12 C12(C(=O)NCC(C)N(C(C(C(C)C)O)=O)C)CCC(O1)c1ccccc12 c1(C(N2CCCC2C2CC2)=O)cnc(S(C)(=O)=O)s1.C(C=O)N(CC)C Cc1ccc(CSCCC2CN3CCC2CC3)c(C(C)C)c1 S(=O)(=O)(c1ccc(=NCC(C)CCC)[nH]c1)NC(CC)(C1CC1)C1CC1 c1(OCC=C)ccc(Cl)nc1C(=O)NCC1CC1.c1(C=O)cc[nH]n1.N C(CC(C)C)(C(=O)N1CCCCC1CF)ONC(c1cc(CC)sn1)=O CC1(F)CN(C(C23CC(C2)C3)=O)CCN(C(C2(C3CC3)CCC2)=O)C1 c1(C(N2CCC(C)(NC(c3ncn(C)c3)=O)C2)=O)ccc2c(c1)ncn2C Cc1nn(CC(=O)N(C)CC2CN(C(c3cnnn3C)=O)CCO2)c(C)c1C N1(C(C(=O)NCC(C)C)=O)CCCC(C(N2CC(CO)C(O)C2)=O)CC1 C(=O)(C1=C(c2cscn2)N(C)C(=O)NC1c1ccc(SC(F)(F)F)cc1)OCC C(=O)(C1=CCCOCC1)NC(C1CCCC1)CNC(c1ccc(N)cc1)=O C1(NC(CCOCCC)=O)C2COCC1CC(NC(C1CC(=O)OC1(C)C)=O)C2 N1(C(C(CC)N(C)C)=O)CCC2(CCCN2C(C2CC(S(C)(=O)=O)C2)=O)CC1 Cc1cc(=NC(=O)NC2SC(=S)N(C)C2=O)[nH]n1-c1ccccc1Br C(=O)(C(C)CC(=O)N1CCN(C(c2ccc(-n3ccnc3)nn2)=O)CC1C)OC c1(C=O)ccc(C#N)[nH]1.C(=O)(CCOC(C)C)N(CC=C)CC1CC1 C(=O)(CC(C)C(=O)NC1CC(NC(c2cn(C3CCOC3)nn2)=O)C1)OC C=C1CCC(C(=O)NC(C2CN(C(C3(C)CC(F)C3)=O)CCO2)C)CC1 c1(C(=O)NC(C2CNC2)C)cccc2c1CCOC2 S(=O)(=O)(c1ccn(C)n1)N1CCN(C(c2cc(C)[nH]c2C)=O)C2C1C2 N1(C(=O)C(O)CC(F)F)CC2CCC1CN2C(=O)Cc1c(F)cccc1Cl Cc1cccc2[nH]cc(CCC(=O)N(C3CN(C(C4CC(F)C4)=O)CC3O)C)c12 c1(OC)nc(C)ccc1C(=O)N(C1CCC(NC(c2nccc(Cl)c2O)=O)C1)C C=CC(C)C(C)C(=O)N(C1CCN(C(c2cnn(CCC(C)C)c2C)=O)CC1)C c1(C(=O)NCC2N(C(CCCC)=O)CCCC2(C)C)ccc(N)c2ncccc12 c1(C(=O)Nc2ccc(OCC)c(F)c2F)cccc2c1CNCC2 N1(C(C(N2CSCSC2)C)=O)CC(NC(=O)C(C)(C)F)C2(COC2)C1 N1(C(=O)Cc2nncs2)CCN(C2CCN(C(c3csc(Cl)c3)=O)CC2)CC1 CC(C)CCCCCC(=O)N1CCC2CC12C(N1CCn2ncnc2C1)=O C12(CNC(=O)CCN3CCC(F)C3)CC1CN(C(=O)Cc1ccccc1C)C2 c1(NC(C2CN(Cc3ccc(Br)c(F)c3)CCC2O)=O)ccnc(Br)c1[N+](=O)[O-] CCN(OC)C(=O)CCC(C(C)C)NC(=O)C(C)(C(C)C)OC S(=O)(=O)(CCC(=O)N)NC.C1CCN(C(=O)CC2C=CCC2)C1c1ccccc1 C(=O)(C1=C(Cl)CCC1)N.C1(C(C)(O)C)CCN(C(c2sccc2C2CC2)=O)CC1 C1(C(=O)OCC2CCC(OC)C2)(OC)CCCCC1 N1(C(CC2(N(C)C)CC2)=O)CCOC(CCCNC(=O)Cc2ccnn2C)C1 N1(C(c2ncc(C)c(C)c2)=O)CC2CCC1CC2NC(C1CCC(F)(F)CC1)=O c1(C(=O)NC2C(C)CN(C(c3ccn(C)c3)=O)CC2C)cc2cccn2c(O)n1 C(=O)(C(C)CC(F)(F)F)NC(CC1CN(C(c2cc(OCC)n[nH]2)=O)C1)C C(=O)(C(CNC(c1ccc(F)cc1)=O)CC(C)C)NCCN(CC)CC N1(C(c2c(C)ncnc2)=O)CC2CC(C1)CN(C(c1cc3cccnn3n1)=O)C2 C=CC1(O)CCN(C(=O)CC2(C)CCN(C(=O)Cc3ccn(CC)n3)C2)C1 c1(C(=O)NCC(C)CN(C)C(C2CC2(F)F)=O)cccnc1O Cc1onc(C(=O)N(C)CCOCCN(C(=O)CO)C)c1I C(=O)(CC(C(F)F)C(C)(C)C)NCC(C(C)C)NC(c1n(OC)cnc1C)=O c1(C(N2C(C(=O)NC(c3ccc(Cl)c(Cl)c3)C)CCC2)=O)cnc(O)c(Cl)c1 O=C1COc2c(C(=O)NC3CC(NC(c4cnc(O)o4)=O)C3)cccc2N1 C(=O)(C1=CS(=O)CCC1)NC(CCN(C(c1ccc(OC)nc1C)=O)C)C(C)C C(CC(O)CC(=O)N(C(C)CNC(c1cc(-c2csc(C)n2)cn1C)=O)C)SC Cc1cc(F)ccc1C(O)C(=O)NCCNC(C1CCCN(c2nccs2)C1)=O CC(C)CCC(O)C(=O)N(CCN(C)C(c1ccc2c(c1)CC2)=O)C(C)C c1(OC)c(C(N2CCC(NC(=O)COc3ccsc3)CC2C)=O)cccc1F C#CCC(C(=O)NCC1CC1C1CCC1)NC(c1ccnnc1C)=O c1(C(=O)OC)cc(OC)cc(C(=O)N)n1.C1CCN(C(=O)C=C2CC2)C1 C(=O)(C#CC1CCCO1)N1CCN(C2CN(C(c3c(C)nc(N)cn3)=O)C2)CC1 C=C(Cl)C(C)(C)C(=O)NC1CCC(CNC(=O)C(C)O)CC1 n1(CC=O)ccc2nc(O)nc(O)c12.N1(C(CC)=O)CC(O)(CC)C1.CCS Cc1cc(C(=O)NCCCCC(C)NC(=O)CCc2cncs2)c(C)[nH]1 N1(C(C(CC)SC)=O)CC(CNC(c2cc(C3CC3)on2)=O)C2(CC2)C1 N1(C(c2cc(N)nc(Cl)c2)=O)CCS(=O)(=O)C(CC)C1.C1(C=O)CC1CF C12(C(=O)NC3CC4CC(NC(c5c(C)cco5)=O)C4C3)CCC(F)(CC1)CC2 C1(NC(c2cn(CCC)nn2)=O)CCCCCC1NC(c1cnn(C)c1SC)=O Cc1c[nH]cc1C(=O)NCC1CC1NC(c1ccccn1)=O c1(CC(=O)NC(CN(C)C(c2csc(S)n2)=O)(C)C)cnc2cccnn12 Cc1cc(O)cc(C)c1C(N1CCOCC(NC(C2(CC(F)F)CCC2)=O)C1)=O N1(C(COCCSC)=O)CCC(O)(CCNC(=O)C(=O)NCC)C1.S c1(OC)ccc(OC)c(C(N2CC3CCC2C3NC(c2sccc2F)=O)=O)c1 C(=O)(C(F)C(C)(C)O)NC(C1CN(C(c2c[nH]nc2C2CC2)=O)C1)C C=C(Br)CCC(=O)NC1COCCC1NC(c1sc(CO)nc1C)=O c1(C(=O)NC(CCCOC)C(=O)NC(C)(C)C)ccc(-c2nn[nH]n2)c(I)c1 c1(CCNC(C2(F)CN(C(C3N(CCC)CCC3)=O)C2)=O)ccc(O)cn1 C(N=c1nc(-c2ccccc2)[nH]c(=NC2CC3CC3C2)[nH]1)C1CCCN(C)C1=O C1(O)CCN(C)CC1.N1(CC(N2CC(C(C(=O)N)OC)C2)=O)CCOCC1=O.C C1(NC(c2cnn(CCO)c2)=O)CN(C(c2cc(C(F)F)cs2)=O)CC1C1CC1 N1(C(C(C)SC)=O)CC2CN(C(c3cc(C(N)=O)cs3)=O)CC(C1)O2 c1(OCC)cc(C(N2CCC(NC(=O)C(C)(C)COC)C2)=O)ccn1 N1(C(C2CC(OC)C(OC)C2)=O)CCN(C(=O)CC2(O)CCC2)CC1C c1(C(C2CCCN(c3nc(Cl)ncc3F)C2)=O)cc([N+](=O)[O-])cnc1O CCCC(CC)C(=O)N1CCCC1(C(N1CCN(C2(C)CC2)CC1)=O)C(C)C C1(C(N(C2CCC(NC(CC(C)F)=O)CC2)C)=O)CCc2nn[nH]c2C1 C1(CNC(C2(OC)CCCCC2)=O)CC2CC(C1)N(C=O)C2.C(C)(C)C.O N1(C(C2CC23CCOCC3)C(=O)NCCCC)CC(C)C(N=[N+]=[N-])C1 c1(C(N(C2CC(NC(CN(CCOC)C)=O)C2)C)=O)ocnc1C C1(O)(CN(C(CC(CC)C2CC2)=O)C)CCN(C(=O)CCc2ccn(C)n2)CC1 C1(CNC(=O)C2=C(Cl)CCC2)CCC2(CCC2)CN1C(C1CCC1(F)F)=O C1(NC(c2ccn(C)c2)=O)C2CCN(C(=O)CCNc3ccccn3)CC12 N1(C(C(CCC)NC(C)=O)=O)CCc2[nH]nc(C(N3CCC(CO)C3)=O)c2C1 N1(C(C=Cc2ccc(C)s2)=O)CC2CCC2C1.N1(CCC(=O)N)CCCS1(=O)=O c1(C(N2C(CNC(c3cn(C)c(=O)cn3)=O)CC(O)C2)=O)cc2n(n1)CCCC2 C=CC1(C(=O)NCc2ncn(CC)n2)CCN(C(=O)C=CC2CCC2)C1 C12CCCC13CCN(CC3)C2.c1(C(=O)OC)ncc(C(=O)OC)cc1N N(C(=NCC(C)C1CCC1)NCC1CCOC1)Cc1cccc(SC)c1 C1(C)(C(=O)NC(CN(C(=O)Cn2cccc2)CC)C)CCCCC1 c1(CNC(C(C2CCN(C(CC(CC)C)=O)CC2)C)=O)cc(O)ccc1C N1(C(C2(CC#C)CCC2)=O)CC2CC(NC(c3c(C)cnnc3O)=O)CC2C1 Cc1ccnc(Cl)c1C(=O)NC(C)CCC.c1(C=O)[nH]c(=N)sc1C(F)(F)F c1(CC)c(NC(C2(C)CN(C(c3cn(CC)nc3C)=O)C2)=O)cnn1C C(CN=C(NCC1CC12CC2)NC1CC1C(F)F)c1ccc(OC)cc1 C(CC(O)C(=O)NCC1(C(=O)NC2COCC2CO)CCCC1)SC N1(C(C(N2CCN(C)CC2)C)=O)CCCC(NC(c2ncn(C)n2)=O)CCC1 C1(NC(CCN(C(=O)C(=C2CCCCC2)F)C)=O)C(=O)OCC1(C)C C1(NC(Cc2c(C)nc(C)nc2O)=O)CC2CCC(C1F)N2C(C1CCO1)=O C(=O)(C1CCCn2ccnc21)N(CC(C)(C)NC(=O)CCCc1ccccn1)C c1(C(C)C)ccoc1C(=O)NCC(C)NC(C1CCOC1C)=O c1(SC)ccc(-n2cc(C3CC3C(=O)C(F)CC3CCOC3)nn2)cc1 C(=O)(C(C)CC(N)=O)N1CCC(N2CCC(NC(CCC=CCC=C)=O)CC2)C1 N1(C(C(C)SC(F)(F)F)=O)CCC2(CNC(c3c(C=O)cnn3C)=O)CCCC12 C1(NC(=O)Nc2c(CC)nccc2C)CCCC(C2CC2)C1 c1(C(=O)NC2CCCN(Cc3c(N(C)C)cccc3)C2)ccn2ncnc2c1 C(=O)(NN1CCP(C)(=O)CC1)c1ccc(Sc2c(C)cc(Cl)cc2)cc1 c1(C(=O)NC2(CO)CCCN(C(C3N(N=O)CCC3)=O)C2)ccc2c(c1)CCC2 CCCCCCCCC(F)C(=O)NCC1CN(C(c2cc3sccc3cn2)=O)C1 c1(C(=O)NC23CC(CNC(CC(C)F)=O)(C2)C3)ccccc1.N(C)(C)C C(=O)(C1c2ccc(Br)cc2CCN1CC)C(CCOCC)=O.OCC O=C(C1=COCCC1)NC1CC(C(N2CC3C(C2)C3(F)F)=O)C1 c1(C(=O)NC2CCC(=O)N(C)C2c2cnn(C)c2)ccn2ncc(Cl)c2n1 CCC(C(=O)NCC1(Sc2ccc(Br)cc2)CC1)C(C)(C)CC c1(C(CSCc2c(C)ccc(OC)c2Br)=O)ccc([N+](=O)[O-])cc1F CON1CCC(NC(C2(CNC(C3(C(=O)O)CC=CC3)=O)CC2)=O)CC1 C(CCCCCCC(=O)N(C)CC1CCCN(C(c2ncn(C)n2)=O)C1)SC c1(C(N2CCCC(C)(CNC(CC3CN(C)C3)=O)C2)=O)cnn2c1CCCC2 C1(CNC(C2CCN(C)C2=O)=O)N(C(=O)C2=CCCSC2)CCCC1(C)C C1(C(=O)NC2C3CC2N(C(=O)CO)C3)CC1C1CC(F)(F)C1.C1CCCC1 N1(C(CCC(C)SC)=O)CCN(C(c2cc(C(F)F)[nH]n2)=O)C(C2CCCC2)C1 C(=O)(CC(CC)C(C)C)NCCN(C(C(CC=C)C)=O)CCOC(C)=O c1(C(N2CCCC(CCC)(NC(=O)C(O)CC)C2)=O)ccnc2ccc(O)cc12 c1(C(=O)NCCC(C)NC(c2coc(Cl)n2)=O)cc(Cl)cc([N+](=O)[O-])c1 N#Cc1c(F)ccc2[nH]c(C(N3CCC3CNC(=O)CCN3CCC3)=O)cc12 N1(C(CC2(SC)CN(C(c3c(CCC)[nH]cc3)=O)C2)=O)CCCCC(CO)C1 c1(OC)cccc(OC)c1CC(N1CC(CCO)(NC(=O)C(O)CSC)C1)=O C12(CNC(c3c(C)onc3)=O)CC1CN(C(C1CC(N(C)C)C1)=O)C2 c1(C(=O)OC)ccc(C(N2CC(C)CC2C)=O)c(F)c1.C(=O)(CC(F)(F)F)N N1(C(CNC(CC)=O)=O)CC2(C(=O)NC(CC)CC)CC1CCO2 c1(C(N2CCCCC2)=O)cc(C#N)cn1C.C1(CC)(COC)CC(C(=O)N)C1 N1(C(CC(C)SC)=O)CCc2ccc(C(=O)N(C)CC3CCC3)nc2C1 C(=O)(CCCC(F)(F)F)NC1C(C(=O)NC2CC(C)OC(C)C2)OCC1 c1(N(CC(C)NC(CCC(C)SC)=O)C)nc(C)nc2n[nH]cc12 CC(CC(=O)NC(Cn1cncn1)C(=O)NCCN1CC2CC2C1)C(F)F Cc1sc(Br)c(C(=O)Nc2nc(-c3cc(Cl)cc(Cl)c3)no2)c1C C(=O)(CC(C(=O)OCCSCC)N1CCCCC1)OC.CCC(=O)C(C)(C)C C1(NC(c2cc(CC)n(CCO)n2)=O)CCN(C(C2CCOC(C)C2)=O)C(C)C1 Cc1cc(C)c(C(=O)CN2CCCC(C(=O)N)C2)c(C)c1.c1nc(C(=O)O)co1 CCS(=O)CC(=O)NC(c1ccccc1F)CNC(c1nccnc1OC)=O N1(C(C2(N(C(CN(C(=O)OC)C)=O)C)CC2)=O)CCCC(C)(C)C1C C1(NC(c2ccc(C)o2)=O)CN(C(=O)CC2COCCO2)C2(CCCCC2)C1 C(c1ccccn1)=C(C)C(=O)NC(C)CC1CN(C(=O)C(F)n2cccn2)C1 Cc1cc(-n2cccn2)nc(N(C)CC)n1.C12CCCN1C2.C(=O)C(C)C1CCC1 C1(OC)CCC12CC(C(=O)NCC(C)N(C(=O)CCC(=O)N1CCOCC1)C)C2 N1(C(C2CCC23CCCO3)=O)CC2(CCN(C(C3CC4CCC3CC4)=O)CC2)C1 C1(NC(CCCOCC)=O)CCC2CCN(C(=O)CN3CCS(=O)(=O)CC3)C12 c1(C(=O)OC)cc(CC(N2CC(CO)(NC(c3cscc3Cl)=O)C2)=O)cs1 Cc1nc(C(F)(F)F)c(C(=O)NCCC2CC2)s1.C1(C)(C=O)CCC1.C Cc1c(C(=O)NC23CC(C2)C3)[nH]c2ccc(F)cc12.C1(C(=O)N)CC2CCC12 c1(SC)ccccc1C(=O)N(C1CN(C(=O)Cc2cccc(C(C)C)c2)C1)C C1CN(C(C2C(C(F)F)C2(C)C)=O)CC1O.n1(CCC(C)C)cc(C(=O)N)nn1 N1(C(C(CCC)N(C)C)=O)CC(F)(F)CC1CNC(=O)C(C1CCOCC1)F N1(C(CC=CC=C)=O)CC(C(=O)NC2CCC(C(=O)OC)C2)C(C)C1 c1(C(N2CC3(CC(CNC(c4cccnc4S)=O)C3)C2)=O)ccc2occc2c1 Cc1ccc(NC(C2CCN(Cc3ccc(F)c(C)c3F)CC2O)=O)c(C)c1C Cc1cc(C=O)c(C)n1CC(F)(F)F.C(=O)(C(O)C(F)F)N(CC)C(C)C c1(C(=O)NC2CN(Cc3ccc(OC)cc3C)C2)ccc2c(c1)NC(=O)CO2 C=CCCCCC(=O)NCC(C(=O)N(C)CC1CCCC1)N(C)C c1(C(N(CC(C)N(C(COc2cn(C(C)C)nc2)=O)C)C)=O)nc(=N)cc[nH]1 Cn1cc(CC(=O)NC2(CO)CCN(C(C3(CN(C)C)CC3)=O)C2)c(Cl)n1 c1(CNC(=O)NCc2cccc(Cl)c2)nnc2n1CCNC2=O C(=O)(CCCCC(F)(F)F)NC1C(NC(CSCCC(C)C)=O)CC1 c1(NC)ccc(C=O)cc1F.C1(C=O)CCCN1C(=O)CC1CC1.C1CC1.N c1(CC(N2CCC(C(C)NC(C3CCOCC3)=O)C2)=O)cccc(F)c1O c1(OC)c(C(c2nnnn2CC(F)F)NCC(C)(C)C(F)F)cccc1Br c1(C(N2C(CNC(C(C=C)(C)CC)=O)C(C)(C)CC2)=O)cc2c(F)cccc2s1 C1(NC(c2nc(C)sc2)=O)COCCC1NC(=O)CC=CC(C)(C)C N1(C(CCCCN(C)C(c2cnn(C)c2N)=O)=O)CCSC2CCC12 CC(C(=O)NCC1(F)CCN(C(c2ccc(Cl)c(N)c2)=O)C1)C(F)(F)C(F)F C1(C(=O)NCCNC(c2cnn(-c3ccccc3F)c2)=O)CCC2(CCC2)OC1 N1(C(C(CC)N(C)C)=O)CC(C(N2CC(N3CCCC3=O)C2)=O)C(F)C1 Cc1cc([N+](=O)[O-])ccc1C(=O)N(C1CN(C(=O)C(O)CN2CCCC2)C1)C Cc1ccc(C(C)C(=O)NC(CNC(=O)CCF)C(C)C)cc1 C12(C(N(CCOCCCNC(CC(CC)SC)=O)C)=O)CCC(F)(CC1)CC2 C1(Cc2scc(C)n2)CN(Cc2nc(Br)co2)CC1C N1(CC)CCC(N(C(=O)CSCC(F)F)C(c2cccc(Cl)c2)=O)CC1 C1(c2nnnn2C2CC(F)(F)C2)(NCCOCC=C)CCN2CCCCC2C1 CC1CC(C(=O)NC23CC(NC(c4ccsc4Cl)=O)(C2)C3)CCO1 c1(CN2CC(CC)N(C(c3[nH]cc(C)c3C)=O)CC2)cc(F)cc(C#N)c1 O=C1CC2(CCN(C(C3CC(C4CC4)=NO3)=O)CC2)C(O)CN1 Cc1c(C(N2CCCC2c2cccs2)C(=O)NC(C)(C)C)cnn1C C1(NC(c2nncc(C)c2)=O)CN(C(c2ocnc2C(F)F)=O)C2CCCCC12 C1(C2(C)CC2)(C(N(CCCn2cc(CC(COC)O)nn2)C2CC2)=O)CC1 CCC(N)C(=O)CN1CC(N(C)C(=O)OC(C)(C)C)C(F)C1 N1(C(CC(=C=C)C)=O)CCCC(NC(c2cnoc2CC)=O)CC1 Cc1ccnc(NCC(CNC(c2cc(C)n(C)c2)=O)C(F)(F)F)c1[N+](=O)[O-] N1(C(C2CCC(CC)O2)=O)CC2CC1CN(C(=O)Cc1cnn3ccccc13)C2 C1(C(=O)NC2CCCN(C)C2)CC(N=[N+]=[N-])CN1C(c1cn(C)cn1)=O C1(CNC(C(CC=C)NC(=O)CCCN(C)C(C)=O)=O)CCOCC1(C)C c1(C(N2CC(C3(NC(C(C(C)(C)C)O)=O)CC3)C2)=O)cnn2cccc(Cl)c12 C12(NC(c3nccc(C(N)=O)c3)=O)COC(C1)CC2.C(=O)CCc1ccsc1.N Cc1c(C(=O)NC(C)C(C)NC(C2(n3cccc3)CCCC2)=O)ncn1C N1(C(CCSCC)=O)CCC(NC(=O)Cn2nnc(-c3ccccc3)n2)C12CC2 N#CCCCC(=O)NC1CCC(CNC(=O)CCCc2ccc(Br)cc2)C1 N1(C(CCOCCOCC)=O)CCN(C(=O)C(C)n2cccn2)CC1C(F)F C=CCCC(C(=O)N(CCCOC)CCO)NC(=O)C(=O)C(C)(C)C N1(C(C2(C)C(C)(C)C2(C)C)=O)CCOCC(F)(C)C1.c1(CC(=O)N)nc[nH]n1 c1(OCCCNC(=O)NCCc2nc(CC)on2)cccc(C#N)c1 Cc1c[nH]c(C#N)nc1=NC1CCC2CN(C(=O)CCC(C)(C)F)CC12 CCC(C)C(CNC(c1cn(CCNC(=O)C(C)(C)CF)cn1)=O)OC n1(CC)cc(C(=O)NCC2C=CCN2C(=O)CCc2cncn2C)nn1 N1(C(C(C2CCCC2)OCC)=O)CCC(C)N(C(c2ccc(Cl)nn2)=O)CC1 c1(CC)ccc(F)cc1C(=O)NC1CC2CN(C(=O)Cc3cnn(C)c3)CC12 c1(C(C)C)ccc(C#N)c(NC2CN(C(=O)CC3CC4CCC3O4)C2)n1 C1(C(=O)NC(C2CCN(C(C(C)=CC)=O)C2)(C)C)CC2OC(=O)OC2C1 C#CCCN=C(NCCC(C)OC)N1CCC(O)(c2cccc(C)c2)CC1 N1(C(COCCOCC)=O)CC=CC(NC(C2CCCN2N=O)=O)C1 C#Cc1ccc(C(=O)N(C(C)CCNC(c2[nH]ccc2C2CC2)=O)C)c(O)c1 c1(N(CC(CN(C(Cc2nc(C)[nH]n2)=O)C)O)C)ccnc2ncnn12 Cc1csc(C)c1C(N1CCOC(C(=O)NCC(O)CN(C)C)C1)=O c1(OC)cccc(C(F)F)c1C(=O)NCC(CO)NC(c1c(C)[nH][nH]c1=N)=O c1(C(=O)NC2C(NC(C(CC(C)C)O)=O)CC2)cc([N+](=O)[O-])ccc1Br C1(NC(C2(O)CC2)=O)COCC1NC(C1(c2cccnc2)CC1)=O c1(C(N(CCCNC(C2CCCS2)=O)CC)=O)cnc(C)c(C#N)c1 C1(C(N(CC)C2CC2)=O)CCC([N+](=O)[O-])CC1.c1(CC)cc(C=O)oc1.N Cc1nc2ccccc2cc1C(=O)NCCCNC(c1c(Cl)cnn1C(C)C)=O CC1=NOC(CC(=O)NCC2(O)CC(NC(=O)CSC3CC3)C2)C1 c12cc(ccn1)NC2=O.C=C1CC(C)C1.C12CC(C1)CCNC2=O.C=O C1(NC(C(C(C)O)C)=O)CN(C(=O)C(C2CCCCCC2)O)CCC1C(F)(F)F c1(C(N2CC(CCNC(C3(CC)CCC3)=O)C(C)C2)=O)cc2c(o1)CCCC2 C(=O)(CN=c1[nH]c(C)cs1)N1CC2(CCC(CNC(CCC(C)OC)=O)O2)C1 C1(OC(C)(C)C)CC(NC(N2CCCCC2)=O)C1(C)C.N1(C=O)CCOCC1.N c1(OC)cc(F)ccc1C(=O)N.C1C(O)C(O)CN1C(c1cc(F)c[nH]1)=O.C N1(C(C2(CCCC)CC2)=O)CC2C(C(=O)NCC3CN(C4CC4)C3)C2C1 C(C(C)C(=O)N(C1CCCC1)CC)SC.C(=O)CC(c1ccccc1)C1CC1.N c1(CC(=O)N(C(C)CNC(=O)C=CC2CCCO2)C)ccccc1Br N1(C(C)(C)C)CCC(NC(c2ccc(Br)cc2)c2nnnn2CCCF)C1=O C1(NC(C(=O)NC(C)C)=O)CC2CCC1CC2NC(C1CCCC(=O)N1)=O c1(C=O)ccc2c(c1)CCOC2.C1(CNC(CC(=O)OC)=O)CC12CCC2.C C(=O)(CCCC(=O)NCCC1CC2(COC2)C1)OCC c1(C(N(C(C(=O)N(C(C(C)SC)C)C)C)C2CC2)=O)cc(C)cc(O)n1 C1(N(C)C)(CC)CCN(C(C2CCC3CC23)=O)C1 C(c1ncco1)=CC(=O)NCCC(C)NC(c1c[nH]nc1-c1cnn(C)c1)=O Cc1cc(O)n2ncc(C(N3CCCC(C)(CNC(=O)C4=CSCS4)C3)=O)c2n1 C1(CCC)CN(C(=O)C=Cc2ccc(CC)o2)CCN1C(C1CC12CCCC2)=O C1(C(=O)OC)CCC(NCCS(C)(=O)=O)CC1(C)C c1(C(=O)NCC(C2CCC2)NC(C2CC3C=CC2CC3)=O)ccc2nsnc2c1 C(CN=[N+]=[N-])(C(=O)NCCC1CC=CC1)NC(c1ccn(C)n1)=O N1(C(CCOCCC)=O)C2CCC1CN(C(C1(CC)CCCCO1)=O)C2 N1(Cc2c(I)cn(C)n2)CC2CS(=N)(=O)CC2C1 Cc1cc(N)cnc1C(N1CCCC(NC(c2ncsc2C(F)(F)F)=O)C1)=O C1(NC(C(CC=C)C)=O)CCN(C(c2c(C)n[nH]c2C)=O)CC(C)(C)C1 c1(C(N2CCC(C=O)C2)=O)ccc(S(=O)(=O)N(C)C2CC2)o1.C(C)(C)C c1(CC(=O)N(C2CN(C(=O)CC3(C)CC3(Cl)Cl)C2)C)ccc2c(c1)CCCO2 c1(N(CC(CNC(C(CC)CCOC)=O)C)C)nc(C)cc(C#N)n1 C1(NC(=O)CCCc2ccccn2)CN(C(=O)CC2CC2C2CC2)CC1O c1(CC)ncc(C(=O)NCCCN(C(=O)Cc2cncs2)C)c(C)n1 Cc1ccc(C(N2CC3=C(C2)CN(C(=O)CC2CCC(C)C2)C3)=O)c2c1CCC2 c1(OC)ccc2[nH]c(=NCCF)[nH]c(=NC(C)COC3CCCCC3)c2c1 C(=O)(C(C)(COC)CO)N1CC(CC(=O)NCC(CCC)(C)O)(OC)C1 c1(OC)cccc(F)c1-c1cc(C(=O)OC(c2ccc[n+]([O-])c2)C)n[nH]1 Cc1cccc(C(N2CCCOC(CNC(=O)C(C)N=[N+]=[N-])C2)=O)c1C C(=O)(C1=C(C(C)CC)N(CC2CC2)C(=O)NC1c1sc(C)nc1C)OCC O=C(N=c1[nH]oc2cc(Br)cnc12)Nc1cccc(Cl)c1S(=O)(=O)C(F)F Cc1c(Cl)ccnc1C(N1CCCC(CCNC(C2SCCCS2)=O)C1)=O C1(NC(c2ccsc2)=O)C2CC3CN(C(c4ccc5sccc5c4)=O)C1C3C2 c1(CC)nc(-c2cc(CC3CC3)c[nH]2)n(Cc2ccccc2C(C)C)n1 N1(S(CC(=O)OC)(=O)=O)CCc2nc(NC(=O)CN3CCC(C)CC3)ccc2C1 n1(CCC(=O)NC2CC(C)N(C(=O)CC3CC3)CC2)cc(Br)c(O)nc1=O c1(CCNCc2ccc(OCCCCCC)cn2)cn2cccnc2n1 N1(C(C=CCCC)=O)CCC2C(NC(=O)CCC(C)N(C)C)CC12 C1(NC(CN(C(C)C)C)=O)CCN(C(=O)Cn2cccc(N)c2=O)C12CC2 Cc1cc(C(=O)NC(C)CCCNC(c2conc2C(C)(C)C)=O)c(C)s1 C1(NC(c2noc3c2CCC3)c2n(CCOCC)nnn2)CCc2nncn2C1 c1(C(N2CC(C(=O)NC3C(C)CCC3C)OCC2)=O)cccc(O)c1F Cc1cc(C)c(S(=O)(=O)NC2CN(C(c3cscc3Br)=O)CC2C)c(C)c1 N1(C(C(=O)NCC2CCCCO2)=O)CCC(O)(c2ccc(Br)cc2)C1 C(C)(CC(F)(F)F)(c1ccccc1)NC(CC(C)(C)c1ccc(C(=O)O)cc1)=O N1(CC(=O)N(C2CCN(C(c3c(SC)cnn3C)=O)C2)CC)CCCCC1CC c1(C(N(C)CCNC(=O)Cc2csc(Br)n2)=O)ccccc1CC#N c1nnc(C)n1C.C(C(C(=O)NCC(C)CN(C(=O)CNC)C)OC)OC.C c1(CN2C(C(=O)OC)CC3(CCC3)C2)nc2ccccc2nc1C C1(CNC(C2C=CCN(C(Cc3cc(C)no3)=O)C2)=O)CCCCC1(C)C c1(C(N(CC(CNC(C(C(C)C)C)=O)O)C)=O)ccc2occc2c1 C1(OCC(=O)NCCOCCC(=O)N(C(CC)CO)CC)CCCCC1 C(c1ccc(F)cc1)=CC(=O)NC1CCC(NC(CC2CCC(C)C2)=O)CC1 c1(C(N2C(C(N3CCC(C4CCC4)C3)=O)CC(O)C2)=O)ccc2[nH]ccc2n1 C(CNC(c1c[nH]nc1Cl)=O)(C(=O)N(C)CC1(O)CCOC1)OC N1(C(CCC(=O)OC)=O)CCC(NC(c2cncc(C(F)F)c2)=O)CC1C N1(C(C(c2cccc(C)c2)F)=O)CC(NC(C2CC2(C)C)=O)CC1(C)C c1(C(=O)NCC(C2CCCC2)NC(C2C(C)C2C)=O)cccc2sncc12 C1(C(C)C)CN(C(=O)CCCOc2ccccc2)CCN1C(c1cnn(C)c1)=O Cc1nc2cccc(C(=O)NC3CS(=O)(=O)CC3)c2[nH]1.c1(C=O)cn(C)cn1.N C12(NC(CC(CC)O)=O)CCCC1N(C(=O)Cc1cccc(C(N)=O)c1)CCC2 C(CCC(C)(C)C)(C(=O)NC1CCOC1)N1CCCC(COC)C1 CC(C)C(F)C(=O)NC12CC(NC(C3CN(C4CCOC4)C3)=O)(C1)C2 c1(C2C(NC(N(CC(CCC)C)C)=O)C2)ccc(C(F)(F)F)cn1 C1(NC(CCOCC)=O)COC2(CNC(=O)CCC(C)N(C)C)CC1C2 C(CC(F)F)(C(=O)NCC1(F)CC(CO)C1)NC(C1C(C)CC1)=O S(=O)(=O)(c1ccc(N(CC(C)CO)C)cc1Br)NCCC(OCC)OCC c1(SC)ccc(C=CC(N2CCC(NC(C3CCC=CCCC3)=O)CC2)=O)cc1 C1(C(=O)NCC2(C(N3CCC(CC)C3)=O)CC(C)(C)C2)CCCCC1CC c1(CC)ncc(CNC(C2(NC(=O)CCc3ccno3)CC(F)C2)=O)s1 C(=O)(CCCC(F)(F)CO)NC1C(C)N(C(c2ccc(O)cc2F)=O)CCC1 c1(C(N2CCOC(CO)C2)=O)cc(-c2ccc3c[nH]nc3c2)cc2[nH]ncc12 c1(C(=O)NC(C)CC2CN(C(=O)CN(C3CCSC3)C)C2)cncc(F)n1 CCC(C)C(O)C(=O)N(CC)C1CC1.c1(CC)ccccc1.C(=O)C.C(C)=O C1CCC1(C)C.c1(OC)nc(C(=O)NC)co1.c1(C2C(C=O)C2)ccnn1C C1(C(=O)NCc2cn[nH]c2)(CNC(C=C(CCC)C)=O)CC12CCC2 c1(CC)nc2ccccn2c1C(N1CCC(C)C(NC(=O)OC(C)(C)C)C1)=O C(c1cccc(F)c1F)=CC(=O)NC1C(N(C(C(CO)N(C)C)=O)C)CCCC1 N1(C(c2c(C)onc2CO)=O)CC2(C1)CN(C(=O)Cc1ccccc1)CCO2 O=C1CC(CC(=O)NCC2(NC(=O)C3=CC4C=CC3C4)CCCC2)=NN1 c1(NC(C2CCCN(Cc3ccc(F)cc3)C2)=O)cc2oc(=O)sc2cc1O C1(C(=O)NCCC=C)CCCN(C(C)CCn2cccn2)CC1 C1(CCC(=O)NCCN(C(C)C)C(C2CCCS2(=O)=O)=O)CCCC(O)C1 c1(C(=O)NCCC(C(C)C)NC(C(CCCC#C)C)=O)ccc2nc(C)[nH]c2c1 C1(NC(C(C2CC2)NC(C2C3CN(C)CC32)=O)=O)CCCCC12CC2 N1(C(CC=CCC)=O)CCCC(C(=O)Nc2nccc(I)n2)CC1 c1(C(=O)NCCC2CN(C(CSCCC)=O)C2)cc2c(nc1N)CCCC2 N1(C(C2CCN(c3n(C)ccn3)C2)=O)CCCC(NC(=O)Cc2cc[nH]n2)C1 CCC(C(=O)NCCN(C(=O)CC1CCC1)C(C)C)C1CCOCC1 O=C(C(O)CC(F)(F)F)NCC1CC2CN(C(=O)C3=CCCCC3)CC12 c1(C(N2CCC(COC)(NC(=O)CC(C)SC)CC2)=O)c(N)sc2c1CCC2 C12(NC(c3cccc4c3SCCC4)=O)CCCCC1N(C(c1cncs1)=O)CC2 c1ccc(Cl)nc1.CC(C)(O)CN(CC(C)(C)O)C(C1CC1C(=O)N)=O c1(OC)nc(C)c(Br)cc1-c1noc(-c2cn(-c3cccc(Br)c3)nc2C)n1 CC(C)CC(O)CC(=O)NCC1C2CN(C(c3cnn4ccsc34)=O)CC12 C1(O)(CCNC(c2cc(Cl)c(Cl)s2)=O)CCN(C(c2cnc(Cl)[nH]2)=O)C1 C1(NC(C2C(C=C)C2)=O)CN(C(=O)CCc2cnccn2)CC1SC N1(C(C(CCSC)O)=O)CC(C2CCCN(C(C3CC(=O)N3)=O)C2)C1 c1(C2C(C(=O)NC(CNC(c3c(C)nn[nH]3)=O)C)C2)ccc(Cl)cc1 CCCC(=O)NCCC1CCN(C(=O)CC(C)C2CCCO2)C1.N1(C=O)CCOCC1 c1(C(N(C2CCN(C(C3CCSC(C)C3)=O)CC2)CC)=O)cnn(CC)c1Cl C=C(C)CC(C(=O)NCC(C)(C)n1cccn1)NC(C1CCS(=O)CC1)=O c1(C(N(C2CC(C(=O)NCC(C)(C)C3CCCO3)C2)C)=O)ccc(Cl)cc1 C(CC(C(=O)N(C(C)CSC)C)NC(C1CCC(=O)CC1)=O)OC C(=O)(C(C)C(C)C)NCCN(CCCCCC)C(=O)COC1CC=CC1 Cc1ccnc(NC(C2CCN(Cc3ccc(C(F)(F)F)cn3)C2)=O)c1F N1(CC)CCC(N=c2cc[nH]cc2S(=O)(=O)NC2CCS(=O)(=O)CC2)CC1C c1(CC)c(NC2CCC(NC(=O)C=Cc3cscn3)CC2)nc(C)nc1Cl CCC(C)(CC)C(=O)N(C1CCCN(CCn2cccn2)CC1)C c1(C(N(C)C)=O)cccc(C(N2CC3C(NC(C4(C)CCCO4)=O)C3C2)=O)n1 c1(C(=O)NCCC2(C(=O)NC(CCC=C)(C)C)CCCC2)c[nH]c(C#N)c1C CC1(C)CCC(C(=O)NCC2C3CN(C(c4csc(C5CC5)n4)=O)CC23)O1 C#CCC(C)(CC)C(=O)NCc1cc(C(N2CC(N=[N+]=[N-])C2)=O)n[nH]1 N1(C(c2ccn(C)n2)=O)CCN(C(=O)C(F)(F)Cl)CC1C(F)(F)F C1(CC(=O)NC(C2CC(NC(C=CCC)=O)C2)C)OCCC1(C)C c1(C(C(=O)NC2CN(C(Cc3ncc(C)o3)=O)CC2C)C)cc(F)cc(F)c1 C(CC(C)C(=O)N(CC(C)(C)CNC(c1cnc(SC)s1)=O)C)OC C(=O)C(C=O)C(C)(C)C.C1(C)CCN(C(C2(c3ncco3)CC2)=O)C1.CC.O c1(C(C(=O)NC(C)(C)CC)N(CCCC)CC)cn2ccc(Br)cc2n1 N1(C(C(CC)O)=O)CCCC12CCN(C(=O)COCC(C)C)C2 n1(CC)cc(C(=O)N(CCC)C(C)C)c(C)n1.C1(C=O)CN(C(N)=O)C1 c1(C(C)NC(=O)NCC(c2cccc(OC)c2)(C)C)nnc2ccccn12 C(=O)(CC1OCCc2ccsc21)NCC(CO)NC(c1cc(CC)c(F)cc1)=O c1(N2CCCC(OC(C)C)C2)nc(N2CCCC(OCCO)C2)c2ncsc2n1 N1(C(C)=O)CCCC(O)(C(=O)Nc2cn(C3CCOC3)nn2)C1 C1(CN(C(=O)CC2CNC(=O)C2)C)CCCN(C(=O)CCc2cscn2)C1 CCC(C#N)(CC)C(=O)NCC(C(C)(C)C)NC(c1cnc(OC)c(C)c1)=O N1(C(=O)NCC(C)(C)C(F)(F)F)Cc2ccccc2C(O)C1 c1(C(=O)NC2CCC(NC(C3C4CC4C4CC34)=O)CC2)cccc(=S)n1O c1(CCC)nc(C(=O)NC(CNC(c2coc(C(F)F)n2)=O)CC)co1.C C(=O)(CC(CCC)CCC)NC(CC(=O)N1CC(CCCCC)C1)COC C(=O)(C(C)C(O)C(C)C)NCC1OCCN(C(C2(C)CCN(C(C)=O)C2)=O)C1 c1(C(N2CCC(CNC(c3cnc(C(C)=O)s3)=O)C2)=O)cncc(Cl)c1 c1(C(=O)NC2CN(c3nnc(COC)s3)C(C)C2)cc(F)c(F)cc1F C1(CC)C(C(=O)NCc2cn(C)cn2)CCN1C(C1CCN1C)=O C(=O)(CCCCC1CC1)N1CC(C)(CCC(=O)NCCSCC)C1 N1(C(C(C=C)CC)=O)CCC2(CC1)CC2C(=O)Nc1cnc(OC)cc1F CC1CCN(C(C2CC(F)(F)CS2)=O)CCN1C(C1CC(=O)NC(=O)N1)=O CCC(CN(C)C)C(=O)N(CCC(=O)NCCN(C)C(=O)C1CC1)CCO C(=O)(CC1OCCc2ccsc21)N1C(C)C(NC(C2CC23CC3)=O)CCC1 C(=O)(CC1OCc2ccccc21)N(CCC)CCNC(c1c[nH]c(=NCC)s1)=O c1(-c2cn(Cc3ncc(N(C)C)cn3)nn2)cc(C(F)(F)F)cc(Br)c1 N1(C(C(C(C)C)NC(C)=O)=O)CCC2CCN(C(=O)Cc3cscn3)CC2C1 Cc1cc(S(=O)(=O)N2CC(C)CCC2C(=O)N(C)C)cnc1C(F)(F)F c1(C2C(C(=O)NCc3c(CC)c[nH]n3)C2)cncc(C)c1 CC(C)CCC(C)N(C(=O)C(C1CCOC1)NC(=O)Cc1cnoc1)C c1(C(N(CCC(C)NC(=O)C=CC(C)(C)C)C)=O)cc2c([nH]1)CCOC2 Cc1nncc(C(=O)NCC(C2CCN(C(C3(C)CCC(C)C3)=O)CC2)O)c1C c1(C(C(=O)NCC)N(C)C)ccccc1Cl.CC1=NOC(C=O)C1.C1CC1.N C1(NC(C(C(C)C)NC(C)=O)=O)CC2CC1N(C(=O)CO)C2.C(C)(C)C c1(C(=O)NCCC(=O)Nc2ccc(C)cc2Cl)cc(F)c(F)c(Cl)c1 c1(C(N(C2CCN(C(C(C3CCCCCC3)C)=O)C2)C)=O)ccc2c(n1)CCO2 C1(CC(=O)NCCCN2CCN(CC(=O)OC)CC2)CC(C)(C)C(=O)N1 c1(OC)c(C(=O)NC(C)(C)C(=O)NCCC2CCCC23CC3)cnn1C C1(NC(CC2(C)CCCC2)=O)COC2(CCN(C(c3cc(Cl)ccc3F)=O)C2)C1 N1(C(c2n(C)c(S)nc2)=O)CCN(C(C2COC3(CCC3)C2)=O)CC1CO C1(CC(=O)NC2C(CNC(CC(=O)OC)=O)COC2)CC2(CCC2)CO1 c1(CC)ccccc1CC.C(=O)C(F)=C(C)C.C(=O)C.C(C)C.C(C)=O Cc1cc(F)c(C(=O)NC2CCCN(c3ncc4ccsc4n3)CC2)c(F)c1 C=CC(CC)C(=O)NC(C)CCC(=O)NCc1nc(CO)n[nH]1 N1(C(C(CC=C)C)=O)CCN(C(=O)CCN2CCNC(=O)C2)CC1CC1CC1 c1(C(N2C(CCCNC(C(COC)O)=O)CCCC2)=O)cn2cccc(Cl)c2n1 C(=O)(C1CCc2nnc(C)n21)OCC12CCC(C(=O)OCC)(C1)CO2 CC(C)C(C)CNC(=O)C(C(C)C)n1cnnc1.C1(=CC(=O)N)CCOCC1 N1(C(=O)C2=CCCS2)CCOC2(CCN(C(C3CCC4(C3)N=N4)=O)C2)C1 N1(C(C=Cc2ccc(C)s2)=O)CC(C)C(F)(F)C1.C(=O)(C(F)(F)C(C)O)N C1(CNC(c2n(CC)nnc2)=O)(C)CC12CCC2.C1(C(=O)N)CCOC1 CCC(CC)CC(=O)NC1CN(C(C2(c3ccc(C)cc3)CC2)=O)CC1SC N1(C(CCCN(C(c2ncn(CC)c2)=O)C)=O)CCOC(COC(C)=O)C1 C12(CNC(C=CSC)=O)CCCCC1N(C(=O)C(O)Cc1ccccc1)CC2 NC(=O)CC(C(=O)NC1(C(F)(F)F)CC1)NC(C12CCCCC1C2)=O Cc1ccc(F)c(C(=O)NCCCCC(C)NC(C2CCC(C)(C)OC2)=O)c1 C1(CCC(=O)N(C2(CC(=O)NCCS(N)(=O)=O)CC2)C)CCCCC1 c1(C(NNC(=O)Nc2ccn(C)n2)=O)cc(CN2CCOCC2)ccc1[N+](=O)[O-] C(=O)(C(C)(CC)C(N)=O)NCC(CCCC)NC(=O)C(C)(C)c1cncs1 Cc1cncc(CCNC(=O)C(C2CC2)NC(=O)CCC2CCC2)n1 c1(C(=O)NCCN(CCC)C(c2ccn(COC)n2)=O)c(Cl)oc2ccccc12 c1(C(C)C)ccc2cc(C(N3CCOC4CC34)=O)ccc2c1 C(=O)(C1=C(F)CN(C(c2cccc(O)c2F)=O)CC1)NCCNC(COC)=O C1(NC(=O)COc2ccccc2Br)CC2CC1N(C(=O)CO)C2 C1(C(N(CC(N2CCCC2)C)C)=O)CCN(C(=O)Cc2ccccc2O)C1(C)C C1CN(C(C2CC3(C2)CC3(F)F)=O)CCC1C(F)(F)F.Cc1ccc(C=O)s1.N c1(C(=O)OCC)ccc2c(c1)CC(NC(c1c(Cl)cc(F)cc1Br)=O)C2 O(C=CC(=O)NCC1(F)CC(NC(=O)Cn2nnc(C3CC3)n2)C1)CC C1(n2c(-c3cncc(O)c3)nc(-c3ccccc3F)n2)CCCCCCC1 N#Cc1ccc(O)c(C(=O)NC2CC23CC(NC(C2CN4CCN2CC4)=O)C3)c1 N1(C(c2ccn(C)n2)=O)CCC2(C(=O)Nc3ccc(F)c(F)c3)CC2C1 Nc1ccc(C(N2CC(NC(C3(C4CC4)CC3)=O)C(n3ccnn3)C2)=O)c(Cl)c1 c12ncc(C#N)c(n1)S2.N1(CC(=O)NC(CN(CC)CC)C)CCOCC1 C=CCC(C)(C)C(=O)N1CCC(N(C(=O)C(C#N)C2CC2)CCO)C1 N1(C(C2C(c3n(C)ncc3)C2)=O)CCC2(CCCN2C(c2cnsn2)=O)CC1 Cc1cc(C(=O)NC2CCCC2NC(C2CC(n3ccnn3)C2)=O)n(C)n1 c1(CN2C3C(C(=O)Nc4c(C)ccnc4Cl)C(C3)C2)cc(Br)c([N+](=O)[O-])s1 C=CCC(C(=O)NCC1(CNC(=O)CCc2nc(=N)[nH][nH]2)CC1)C(C)C c1(C(N(CC(C)NC(C2(n3cnnn3)CC2)=O)CC)=O)cnc2n1CCCC2 c1(C(=O)NC2(C)CCN(C(c3ncc(Cl)s3)=O)C2)cc(F)c(F)c(F)c1F C1(CNC(CCCC(=O)NC)=O)CC2CCC1N(C(C1(F)CCOC1C)=O)C2 c1(OC)c(F)cc(C(=O)NC2CCCN(C(=O)C(C)n3cccc3)C2)cc1Cl Cc1ccc(CC(=O)NCC(C)CNC(=O)C(c2cncnc2)C)cc1 c1(C(=O)NC2CCCC(NC(c3cc(OC)ncc3)=O)C2)cc(C)cc(N)c1 CCC(CNC(=O)C(C)N(C(=O)CC1CCC(=O)CC1)C1CC1)CC(C)C c1(C(=O)NCC2C(NC(=O)Cc3ccsc3)C2)cc2n(n1)CCCO2 c1(C(N2CCC(NC(C(C(C)(C)C)SC)=O)C2C)=O)nc(N)cc2ccccc12 c1(CNC(CN(CCC)C(C2CNC(=O)C2)=O)=O)ncccn1 c1(OC)c(Cl)ccc2[nH]c(C(=O)NC3(C)CCC3)cc12.C(=O)(C(C)(C)C)N c1(C(N2CC3C(CNC(c4c[nH]c(=NC)s4)=O)(C3)C2)=O)cnn2ccc(O)nc12 C(=O)(C(C)C(C)C)NCCCN(C(C1CC2CC2C1)=O)CC.C(C)=O.N CCCCC(CC)C(=O)NCCN(CC(C)O)C(c1cc(CC)on1)=O N1(Cc2c(Br)c(C)n(C)n2)CCC(F)(F)C(Nc2cc(-n3cncn3)ncn2)C1 N1(C(c2c(C)[nH]nc2Cl)=O)CCC2(CCC(CNC(C3CC=CC3)=O)OC2)CC1 c1(C(=O)OC)ccccc1OC(C)CNC=O.C1CCN(C(N)=O)CC1.N N1(C(C2(CCC=C)CC2)=O)CC2(CCC2)C1.C1(CC(=O)N)C=NN(C)C1=O N1(C(c2n(CCC)ccc2)=O)CCN(C)C(C(=O)NC(c2snnc2C)C)C1 c1(OC)cncnc1C(=O)NC(C)Cn1cc(CNC(=O)C(C)O)nn1 c1(C(=O)NC2CCC(CNC(CCc3cc(C)on3)=O)C2)cc(C)cc(F)c1N N1(C(CCP(C)(C)=O)=O)CCC(C2CC2)C1CNC(C1CCOCC1)=O C(=O)(CS(=O)(=O)CCO)N1CCCC1(C)C.Cc1ccccc1SCC(=O)N.C N1(C(C(C)(C)F)=O)CC2CC(C(=O)NCC(c3cccs3)O)(C2)C1 C(=O)(C(C)S(N)(=O)=O)N1C(CNC(C2N(C(C)C)CCC2)=O)CCCC1 n1(CC)c(C(=O)NCC2CC2C(=O)NCC(O)C(N)=O)cnc1O C1(CC(N2CCN(CCCNC(COCCC#C)=O)CC2)=O)NC(=O)CNC1=O CC(C(=O)NCC1(C)CC(NC(c2cocn2)=O)C1)C(F)(F)F.C1CC1 c1(C(=O)NCC2(O)CN(C(CCSc3n(C)ccn3)=O)C2)csc2cccnc12 c1(C(=O)NCC2CCN(C(CCC(CC)OC)=O)C2)cnc2c(c1)NC(=O)CN2 c1(C(=O)NCC(CC)C)ccc2nncn2c1.C(=O)CC1CC1C(F)(F)F.N C1(NC(C2C3CN(C(C4CCCC4F)=O)CC23)=O)CC2(CCCC2)C1 Cc1ccc(C(N2CCC3CCC23C)=O)cc1S(N)(=O)=O.C1(C=O)CN(C)C1.N C(C(=O)NCCCOCC)(C1=CCCSC1)N1CCC(CC)(CO)C1 CC(C)CC(C(=O)N)C(C)C.C1(CC(N2CC(O)(CC)C2)=O)COC(C)(C)CO1 c1(C(N(CCCCO)CCCC)=O)ccc(NC(c2cccc(Br)n2)=O)cn1 c1(C(N2CC(CNC(CCOCC#C)=O)C2)=O)ccc(S(=O)(=O)CC)cc1 C1(CNC(CCCC#C)=O)CN(C(c2cc(Cl)ccn2)=O)CCC1(F)F c1(CNC(C(C2COC2)NC)=O)ccc(OC2CCOC2)nc1 c1(CC(=O)NCC2(F)CN(C(C3C(C#C)C3)=O)C2)cn(C)nc1Cl c1(C(=O)NC(c2ncc[nH]2)C)cnn(-c2ccncc2)c1C(F)(F)F c1(OC)cc(Cl)ccc1C(=O)C(N1CC2C(C(=O)NC3(C)CC3)C2C1)=O N1(C(Cc2ccc(N)cn2)=O)CCC(CC(=O)O)CC12CC2 c1(C(C)(C)C(=O)NCC2CCN2C(=O)Cc2ccon2)ccc2c(c1)OCO2 C1(CN(C)C(C2C=CC=CC=C2)=O)CCC(NC(C2(O)CC2)=O)CC1 c1(C(=O)NC2CN(C(c3c(C)cncc3)=O)CC2C)cnn2c1C(C)CCC2 c1(CNC(CCOC2CN(C(C(C)OC(C)=O)=O)C2)=O)nc(CO)n[nH]1 c1(OC)c(C(N2CCC(CNC(c3cc(C)cs3)=O)CC2)=O)csc1Cl Cc1nc(C(=O)NCCNC(c2occc2C2CC2)=O)nn1C n1(CC=O)ccc2nc(O)nc(O)c12.C(CC(C)(C)C)NC(C(CSC)C)=O.N CC(C)CC(F)C(=O)NC1CCC(NC(c2cc(C(N)=O)cs2)=O)CC1 N1(C(C2C(C)CCN2C(=O)CCc2cnn[nH]2)=O)CC2(C=CCO2)C1 C1(N(C(COC2CCCC(C)C2)=O)C)CN(C(=O)C)CC12CC2.CCN(C)C.S N1(C(C(C)n2cccn2)=O)C2CCC1C(CNC(=O)C=C1CCCCC1)C2 C#Cc1ccc(C(=O)N(C)CCN(C(=O)C(C)S(C)(=O)=O)C(C)C)cc1C C1(C(=O)NC2CCN(C(C)=O)CC2)C2CCCC2CN1C(=O)C(O)CC(N)=O c1(C(=O)NC2C(NC(C(c3ccc(F)cc3)C)=O)C2)cn(C)c(=O)nc1O Cc1c(C(=O)NCC(C)N(C(=O)CCc2ccc(O)nn2)C)cccc1[N+](=O)[O-] CC1=CCC(C)(C(=O)NCC2(F)CCN(C(c3cc(C#N)cs3)=O)CC2)CC1 N1(C(C(C2(O)CCC2)NC(C(CC2CC2)OC)=O)=O)CCCC(F)(F)CC1 C(=O)(C1c2ccccc2CN1C(c1cc[nH]n1)=O)Nc1cc(C)c(F)cn1 N1(C(C(COC)COC)=O)CC2(CC2)CC1C(=O)N.C1CCN(C2CC2)C1=O C(=O)(C1=C(Cl)CCCC1)N1C(CNC(=O)CCCC2CCCC(=O)N2)CCC1 N1(C(CCNC(CC(C)C)=O)=O)CC(NC(C2CCC(=O)CC2C)=O)CCC1C C(=O)(C1=CCCN(C(=O)C(F)(F)Cl)C1)NCC1N(C(C)=O)CSC1 CC1(C)COC(C(=O)NCC2CCCN2C(=O)C(c2ccc(Cl)s2)=O)C1 N1(C(CCc2cnc(C)o2)=O)CCC(CC(C)NC(c2cnc(S)n2C)=O)CC1 c1(C(c2n(C)nnn2)NCC2COC(=O)C2)cc2cc(Br)ccc2o1 C(=O)(C1CSc2ccccc21)NCC(CNC(CC=CCC)=O)(C)O C1(CC(=O)NC(c2cccnc2)Cc2ccc(C)cc2)CCC2(CCNCC2)O1 c1(CCC(=O)N)ccc(F)c(F)c1.c1(OC)ncccc1CC(=O)NC1CCC1 c1(CCC(=O)NCCC(CCNC(c2ccc(C)nn2)=O)C)ccc(Cl)c(C)c1 C1(CC(=O)NC2C(OC)C(O)C2)N(C(c2ccncc2O)=O)CCC1(C)C N1(C(Cc2nnc(C)s2)=O)CC2CC(NC(C3(C)CC(C)C3)=O)C2C1 N1(C(c2c(C)[nH]c(C)c2C)=O)CCC2(CCC2NC(=O)CN(C)C2CC2)CC1 C1(NC(C2CCC(C(N)=O)C2)=O)CCCCC1NC(c1cnc(C2CC2)s1)=O C1(NC(COC(C)C)=O)CN(C(c2ccccc2CCC(F)(F)F)=O)CC1C C1(O)(CCNC(C(C(=O)OC)C)=O)CCN(C(=O)COC2CCC2)CC1 c1(C(CC)(C)C)n[nH]c(=NC(CNC(C2CC(C(C)C)=NO2)=O)C2CCC2)o1 C1CN(C(C2COC3(CCC3)C2)=O)CC1(C)C.c1(C(=O)OC)cc(C=O)cs1.N N1(CC)CC(CNC(=O)CC2(NC(c3cc(C)co3)=O)CC2)CC1=O c1(C(=O)NCC2N(C(CC3(C=C)CC3)=O)CC2)cc(O)nc(OC)n1 CCCS(=O)(=O)CC(=O)NC1CCC(N(C(=O)CCN(C)CCO)C)C1 C(=O)(C1=C(C)CCCC1)N(CCCCN(C(COc1c(CC)cccc1)=O)C)C CCC(CC)C(C)C(=O)N(C1CCCN(C(C2CC(=O)C2C)=O)CC1)C C1(=C(CNC(c2csc(-c3ccoc3)n2)=O)F)CCSCC1 CCCC(C#N)C(=O)NC(CCN(C)C(c1cc(COC)oc1C)=O)C(C)(C)C C(CCCCC(=O)NCC1(O)CCSC1)N(C(C(N1CCNC1=O)C)=O)C CC(C(=O)N(CC(O)CN(C)C(C1CN(C)CCO1)=O)C)C(C)(C)C c1(CN(C2CN(C(CC=C)=O)C2)C(=O)O)ncc(F)c(OC)n1.C(C)(C)C c1(OC)cc(-c2cc(C(=O)Nc3cc(O)nc(O)n3)cnc2OC)cnc1F C1(NC(C2(COC)CC(=C)C2)=O)CCN(C(=O)CCn2ccc(C)n2)CC1.C N1(C(CCN(CCCCC)C)=O)CCN(C(C2CC3(C2)CC3F)=O)C2CCC12 CC(C)(CC#N)CS(=O)(=O)N1CCC1c1ccc(Br)cc1 CC1CCCc2c(C(=O)NCCCCCCN(C)C(c3cc(Cl)ns3)=O)cnn21 C(=O)(C(C)CC(C)C)N1CCC(NC(C2(C(=O)OCC)CC2)=O)(CO)C1 c1(N2CC(C)OC3(C2)CCOC3)nc(=NCCCN2CCC2)[nH]c2c1CCCC2 Cc1ccc(C(N2C(C(=O)NC3(CO)CC(C)C3)CCC2C)=O)c(C)c1 c1(C(C(=O)NC2C(C)CN(C(C3CCC4(C3)N=N4)=O)C2)O)cccc2c1OCC2 c1(CNC2CC(CC(=O)NCc3cnccn3)C2)ccc(F)c(F)c1 C(C)(C)(CC(F)C(=O)NCc1nnc(C)s1)NC(CCC(C)OC)=O C(c1ccc2ccccc2c1)=CC(=O)N(CCC#N)CC(=O)OCC1CC1 O=C(CCC(=O)Nc1nccs1)NCCC1CN(C(=O)CO)CCO1 N1(C(C(c2cccnc2)NC(CCCCCOC)=O)=O)CC2(CC(CO)CO2)C1 C12(NC(CC3N(C(c4ccc(N)cn4)=O)CCC3)=O)CC=CC(C1)OC2 c1(CC(=O)NC2(CNC(=O)C(O)C3CCC3)CCCCC2)cc2ccccc2o1 [N-]=[N+]=Nc1cc(C(=O)NCc2ccnn2Cc2ccccc2)ccc1O c1(C(N2CCC(NC(C3N(C(C(C)C)=O)CCC3)=O)C2)=O)cc2c([nH]1)CCCC2 Cc1noc(C)c1C(C)C(N1CCC(C)C1)=O.c1(C(=O)N)cccc(C(F)F)c1 N1(C(CCC#CC)=O)C(C)CC2CN(C(=O)Cc3csc(-c4cccs4)n3)CC12 C(=O)(CC1=CCCCC1)NCC1(NC(Cc2cccc(C(N)=O)c2)=O)CCOC1 CCC(CC)(CCNC(C1(C)CC(F)C1)=O)NC(=O)C(C)Cc1ccccc1F Cc1ccc(CNC(=O)C(C2CC2)N(C)C(C2CC3(CCC3)C2)=O)cc1O C(CC(CC)C(=O)NCCCCNC(c1n[nH]c(C)c1F)=O)=CC C1(NC(C=Cc2cncc(C)c2)=O)CC2CCC1CN(C(=O)Cc1cscn1)C2 n1(CC(C)(C)CO)nc(CC2CC2)nc1-c1cc(-c2ccncc2)on1 n1(C(CC)CC)ncc(C(N2CCC(CF)(NC(c3ccco3)=O)C2)=O)c1C C1(C2CCN(C(C3CCO3)=O)CC2)(CNC(CCC(C)(C)C)=O)CCOCC1 c1(C(=O)NC2CCN(C(c3c(C)cc(O)nc3)=O)C2)cnn2c(C)cccc12 C=CC(C)N=C(NC1CC(Oc2ccc(OC)cc2)C1)N(C)Cc1ncc(C)s1 CCC(C(=O)NC1CC(N(C(=O)CCc2nncs2)C)C1)C(C)(C)CC c1(C(N2CCC(CNC(C3(CC#C)CCOC3)=O)C2)=O)cnn(C)c1N Cc1cc(CC(=O)N(CCN(C)CC2(C(N)=O)CCCC2)C(C)C)nn1C C(CC(C)(C)C(=O)N(C1(CO)CC1)C)NC(C(C)=CC1CC1)=O c1(OC(C)C)nc(N(C2CCN(C(=O)Cc3c(F)cccc3F)C2)C)ncc1Br CP1(=O)CCN(CC(=O)NC2CCCC(NC(c3ncc(F)cc3N)=O)C2)CC1 N1(C(COCCCC)=O)CCC(C)(C(=O)NCC2CC2CCC)CC1 C1(C(=O)NCC2C3CCC(C3)N2C(=O)C(F)F)CCCC(F)(F)CC1 n1(CCC)ccc(C(c2nnnn2CCSC)NC2CCCCC2)n1 C(=O)(C(C)CC(F)(F)F)NCC(CC)NC(=O)C=Cc1cocn1 c1(CC)occ(C(F)(F)F)c1C(=O)NCC(C)CO.c1(C=O)ccc(N)cn1 C(CC1(O)C(=O)Nc2ccccc21)NC(c1ccon1)=O c1ccccc1Cl.C1(COCC(=O)N(C(C)C)CC)CCOCC1.C(=O)C c1(C(N2CCC(C(C)NC(C3CC(C)(C)CO3)=O)CC2)=O)nccc2[nH]ccc12 C1(C(N2CC(CN(C)C(C3(C4CC4)CCCO3)=O)OCC2)=O)CN2CCN1CC2 c1(C(N2CCN(C(C3CCCC3)=O)C3C2C3)=O)cc2cc(F)ccc2s1 C(C)(CNC(C1(CC(C)C)CCC1)=O)(C(C)C)NC(CN(C)CC)=O Cc1ncc(C)c(=NCC2CCCC(NC(=O)CC3CCC4(CCC4)CO3)C2)[nH]1 c1(C(N2C(C(=O)NCCC(O)C3CCCC3)CC2)=O)ccc2cc[nH]c2c1 c1(OC)ccc(Cl)c(CC(=O)NC2CC(CCNC(c3c[nH]nc3F)=O)C2)c1 c1(CN=c2[nH]cc(CCNC(=O)CO)s2)ccnc2ccccc12 c1(NCC2C(C)C2)[nH]c(=NCCc2cc(F)cc(Br)c2)nc2c1cnn2C(C)C N1(C(C=CC)=O)CC(NC(=O)C(C)(C)COC(C)C)CC12CCCOC2 CC(C)C(C(=O)N(CC(C)CO)C(c1sc(Cl)cc1Br)=O)N1CCCCC1 CS(=N)(=O)C1CN(C(=O)CCCCNC(C2CC2C2CC2)=O)C1 CCCCC(CC)CC(=O)NC(C)(CNC(c1cnc(C2CC2)nc1C)=O)CO C1CCC(O)C1.c1(C=O)oc(C)nc1C.C(C(=O)N)OCCOCCOC N1(C(C2N(C(C)C)CCCC2)=O)CC2(CC(NC(=O)CSC(F)(F)F)C2)C1 c1(C(N2C(CC(N3CCOCC3)=O)CCC2)=O)cncc(OC(F)F)c1 CC(CCCCNC(C12CC3CC1C2C3)=O)NC(c1csc(C(F)(F)F)c1)=O N1(C(C=CSC)=O)CC(CO)C2(C1)CN(C(C1CC13CCC3)=O)C2 C(=O)(CCCCC(C)(C)OC)N1CC(N(C(c2ccc(COC)c(F)c2)=O)C)C1 CC1CCN(C(=O)CCCCCNC(c2ccc3cccnn23)=O)CC1(C)C c1(C(CNC(c2cnsc2)=O)NC(C2CC2C(F)(F)F)=O)ccccc1 N1(C(CNC(CN(C)C)=O)=O)CCC(NC(c2cc(CO)[nH]n2)=O)C12CC2 C1(C)(CNC(C=COCC)=O)CN(C(=O)COCc2ccccc2)CC1C c1(C(=O)OC)cccc(C(N2CCC(NCC34CCN(CC3)C4)C2)=O)c1F C1(C(N2CCC(O)(CCNC(=O)Cn3cc(C)cn3)C2)=O)(OC)CCSCC1 N1(C(C(SC)SC)=O)CC2CCC(C1)N2C(=O)C(c1ccccc1)n1cccn1 C(=O)(C#CC1CCCC1)N1CCN(C(c2cc(=N)[nH]cc2Br)=O)CC1CO N1(C(Cn2ccc(C)n2)=O)CC2CCCC2(CNC(=O)CCCn2cncn2)C1 c1(C(CNCC2N(CCC)CCCC2)(C)C)ccc(OC)c(OCC(=O)O)c1 C1(NC(c2ccoc2Br)=O)CC(NC(c2cnoc2C2CC2)=O)C(O)C1 Cc1c(F)ccc2[nH]c(C(=O)NC3CCC3NC(=O)C(C)(C)CC(C)C)cc12 C1(C(=O)O)CN(C(c2cc(Cl)cc(Cl)c2)C(=O)O)Cc2nccn2C1 CCC(C)(C)CC(C(=O)NC(C)(C)C)N1CCOCC12CCSC2 C(C)(CN=c1nc2c(ncn2C)c(NC(c2ccc(F)c(C)c2)C)[nH]1)OC c1(OC)cc(Cl)c(C(N2CC(C)C(C)C2)=O)cc1Cl.C1(CC=O)COC(=O)C1 CC1=CCCN(c2nnc(-c3ccc(C)s3)n2CC(=O)OC(C)(C)C)C1.CCO C=CCCCC(C(=O)NN(CCC)C)NC(=O)OC(C)(C)C.c1ccccc1.S C1(C(N2CC(NC(C)=O)C2)=O)CSCCN1C(=O)CC(C)N(C)C C(N=c1[nH]c(N2CCC(CNS(C)(=O)=O)C2)nc(=NC)[nH]1)C1(CCC)CCC1 CCC1=C(C(=O)NCC2CCCN(C(C3(C)CCCCC3(F)F)=O)C2)CCCO1 C(C)(CC(C)C(F)F)NC(C(COCC)NC(=O)Cc1cnns1)=O CC(C)C(C)(O)C(=O)N1CCN(C(C23CCC(F)(CC2)C3)=O)C(CC(F)(F)F)C1 C1(F)(C(=O)NCCCCCOC)CCN(C(=O)C2=CCCSC2)CC1 c1(C(N(CCCCNC(C2(C=O)CCC2)=O)C)=O)ccc(C#N)o1.C1CC1 Cc1nc(C=O)cc(O)n1.C(c1nc(C)c(C)[nH]1)=CC(=O)N(CCC)CCC C(=O)(C1CCCn2cnnc21)NCCOCCN(C)C(C1C=CCS1)=O C(=O)(C(CNC(c1ccc(CO)s1)=O)C(C)C)N(C1CCN(C)CC1)CC c1(C(=O)NCC(C)(C(C)C)NC(CCCOC)=O)cc(OC)cc(Cl)c1O N1(C(C(=O)Nc2nnn(C)n2)CSc2ccc(F)cc2)CCC(F)C(O)C1 c1(OCC=C)cccnc1C(N1CC(NC(=O)C(CC)CO)CC1C)=O c1(CN2CCC(NC(CNc3cc(C)c(F)cc3N)=O)C2)c(F)c(F)cc(F)c1F N1(C(C)C)CCN(C(=O)C(C2CC2)NC(c2cccc(O)n2)=O)CC1 Cc1nc(Cl)ccc1C(=O)NC1CC1C=O.c1ncc(C(F)(F)F)c(Cl)n1.N N1(C(CS(C)(=O)=O)=O)CC2CCCC1(CNC(=O)C(=O)Nc1ccccc1)C2 N1(C(C2(C)CCC(=O)NC2)=O)CC2CC(O)C1C2NC(c1cnc(N)cn1)=O N1(C(=O)CC2CCCC3CC23)CC2CCC1CN2Cc1nnnn1C1CC1 c1(C(=O)NC(CN(C(=O)CC2(OC)CCC2)CC)C)cnc2n1CCS2 C(=O)(C#CC1CCOCC1)NC1CN(C(c2c(OCC)c(F)ccc2)=O)CC1F c1(OC)cc(CNC=O)ccc1F.c1(C=O)cc(C=O)co1.C(C)(C)C.O c1(CC)cc(C(=O)N(CC(C)NC(=O)C(C2CCC(=O)N2)C)CC)no1 CC(C)C(F)(F)CC(=O)N1CCCC1CNC(c1cc(O)ccc1Cl)=O c1(OCC(=O)NC2C=CC(NC(CSc3n(C)nnn3)=O)C2)ccccc1 C1(CNC(=O)CSc2cn[nH]c2)CC(C(=O)NCc2cncnc2)CO1 c1(C2(NCc3nc(CCC)on3)CCC2)ccc(C(=O)OC)cc1OCC C(=O)(C#CC1CCCCO1)N1CCC(CC=C)(NC(=O)CCCC(=O)NCC)C1 N1(C(c2n[nH]nc2C)=O)CCN(C(=O)Cn2cc(Cl)c(C)n2)CC1C(C)C.C C1(CCCC=O)CCCC(=O)N1.c1(COC)ccc(C(=O)NC2CCC2)s1.C N1(C(C2C(C)(C)C2)=O)CCCC1(C)CNC(c1cn[nH]c1)=O C1(CC)(OC)CN(C(=O)C=Cc2cn[nH]c2)C1.C(=O)C(C)(C)C1CCOC1.N c1(C(=O)NCCC(C)(C)NC(=O)CC2CCCO2)c(Br)nc2n1CCCC2 Cc1cc(C(N)=O)ccc1NC(=O)C(N1CC(C(F)F)C(N)C1)C CC1(F)CCN(Cc2cn(-c3cc(C4CC4)[nH]n3)nn2)CC1 c1(C(=O)NCCC2(O)CCN(C(C3(F)CCCCC3)=O)C2)cc2n(n1)CCOC2 C1(CC)(NC(C2CC(OC)C2)=O)CCCN(C(=O)COC(F)F)C1 CN1CCC(CC(N2CCCCC2C(=O)NCC2(C)COCCO2)=O)CC1 N1(C(c2cccc(C)c2F)=O)CCC(C2(NC(=O)C(O)C3CCCC3)CC2)CC1 N1(C2N(C(C(n3cc(-c4cc(F)ccc4N)nn3)C)=O)CC2)CC2C=CC1CC2 CCCCCCCCN(C(=O)C(C1(O)CCC1)NC(=O)C(C)C1CCCC1)C c1(C(C(=O)NCCNC(C(c2ccc(F)cc2)CC)=O)C)ccccc1F C1(NC(c2ccc(F)s2)=O)CCOCC1NC(=O)C(O)Cc1ccccn1 C#Cc1ccc(C(=O)NCc2ccc(C(=O)NC(C(N)=O)C(C)C)cc2)cc1 C1(C(=O)NC2CC(NC(CCCOC)=O)C23CCC3)CCCN2CCCC12 c1(OC)ccc(C(=O)NCCOC(C)(C)C)cc1C.c1(C=O)c[nH]nc1C.N N1(C(c2c(OC)c(Br)ccc2)=O)CC2CN(Cc3csc(C(C)C)n3)CC2C1 c1(NC(C(C)(C)CCl)c2n(CCC(=O)OCC)nnn2)ccc2oc(Cl)cc2c1 N1(C(C=Cc2c(C)nccc2)=O)CCC2(CC1)CN(C(=O)C(F)=C1CCCC1)C2 C1(C(N2CC(CC)(NC(C3CC3C(F)F)=O)C2)=O)CCCC(CF)C1 C(c1nc2ccccc2o1)=CC(=O)N(C1CCCN(C(C(CC)C(C)C)=O)C1)C N1(C(=O)CCn2cnc([N+](=O)[O-])c2)CCOCC12CC(O)(C(F)(F)F)C2 N1(C(Cn2nc(C)oc2=O)=O)CC2(CCC2)CC1C(=O)NCc1ccsc1C N1(C(c2cn(C)nc2)=O)CC(c2ccccc2)C(F)(CSc2cncc(Br)c2)C1 c1(CNC(CC2(C#N)CCC2)=O)ccc(CNC(C2C3CCCC23)=O)cc1 N1(C(C(C=C)CC)=O)CCOC2CN(C(=O)CN3CSCC3=O)CC12 N1(C(c2c[nH]c(=NC)o2)=O)CCN(C(C2CCC(N(C)C)C2)=O)CC1C N1(C(CC2C(C)(C)C(O)C2)=O)C2CCC1CC(CNC(=O)COCCO)C2 CN1CCC(CCC(=O)NCCCN(CCO)C(c2cc(C(F)(F)F)n[nH]2)=O)C1 C1(N(C(c2cn(CC)nc2)=O)C)CCN(C(c2c[nH]ccc2=N)=O)CC1C c1(NC(C)CC2C=CCC2)nc2c(s1)CCC2 C1(NC(C2(CF)CCN(C(C3C=C(C)CS3)=O)C2)=O)CCc2ncnn2C1 C1(C(N2CC(O)(CC=C)C2)=O)N(C(=O)CC2CCOC2)CCCC1(C)C c1(N(CCN(C(C2=CC(C)(CC)C2)=O)C)C)c(F)cccc1[N+](=O)[O-] c1(NCC(C)(C)NC(CCc2n(C)ccn2)=O)c[n+]([O-])ccc1[N+](=O)[O-] c1(C(=O)NC(CNC(=O)CC2CCCO2)CO)ccnc(O)c1F Cc1nn(C(C)C)cc1C(=O)N.c1(C=O)ccc(Br)nc1.C1CC1.C(C)(C)C C1(NC(C(CCC)NC(C2CC=CC(O)C2)=O)=O)CN(C)CC1(C)C C(c1ccc(O)c(O)c1)=CC(N1CCC(CC)C1)=O.C1(C=O)(CCF)CC1.N N12CC(CO)CN(CC1)C(=O)CCC(=O)N(C)C(C)C2=O.NCC.CCO.C Cc1nc(N2CCC(C(=O)Nc3cc(Cl)c(Cl)cc3C)C(O)C2)c2c[nH]nc2n1 C1(NC(C(F)=CCC)=O)CC2(C1)CCC2.C1(C=O)CC(O)CN1C(N)=O N1(C(C(c2ccoc2)NC(c2nc(C)sc2)=O)=O)CCSCC1C1CC1 C(CCC(C)CC(=O)NC1(C)CC(NC(c2c(C)[nH]c(C)c2C)=O)C1)=C(C)C c1(C(=O)NC2CC3N(C(C(CC)O)=O)C(CC3)C2)ccc2c(c1)CNC2=O c1(OCC=C)c(C(=O)NC2CC(F)C2)cccc1C.C(=O)C(O)CC1CC1 N1(C(C(CC)CN(C)C)=O)CCCC(CO)(NC(=O)CN2CC3CCC2C3)C1 N1(Cc2ccc(N(C)CCO)cc2)CCC2(CC2C(N2CCNC(=O)CC2)=O)C1 N1(C(c2c(C)cccn2)=O)CCN(C(C2CCc3ncsc3C2)=O)CC2(CC2)C1 C=C(C)CC(C(=O)N(CCO)OC)NC(=O)C(C)Cn1ccnc1 C(=O)(C1=CNC2=NCCCN12)N1CCC(NC(c2cc(Cl)c[nH]2)=O)(CF)C1 c1(C(N2C(CNC(C(COC)(F)F)=O)C=CC2)=O)sc(C)c(Br)c1C Cc1cccc(SCc2nc(-c3nc[nH]n3)nn2C23CC(C2)C3)c1 CC(C)(C#N)NC(=O)CCOC1CN(C(=O)C=CCO)C1 C1(CCC)COCCN1C(C1CC=CCC1NC(C1COC(=O)N1C)=O)=O C(=O)(C1=C(F)CN(CC2CC(=C3CCC3)C2)CC1)N(C)CCN1CCCC1=O Cc1cc2n[nH]cc2cc1C(N1CCCC(O)(CNC(C2CNC(=O)C2)=O)C1)=O c1(CN2C(C(=O)NC3(C)CC3)C3CCC2C3)cccc(S(C)(=O)=O)c1 Cc1noc(C)c1CN(C)C(C1CC(=O)CN1C(C1(N(C)C)CC1)=O)=O C=CCC(CC(C)C)C(=O)NC1(C(=O)Nc2cc(C)c(O)cc2C)CC1 CC1(C(=O)NCCc2cccnc2)CCN1Cc1ccc(CO)o1 c1(C(C(=O)NCCC2CN(C(CC3C(COC)C3)=O)C2)C)cnccn1 N1(C(c2[nH]cc(C(C)C)c2)=O)CCC2(NC(=O)Cc3cccc(C#N)c3)CC2C1 Cc1nc2n(c(=O)c1CCNC(=O)C(N1CCN(C(C)CO)CC1)=O)CCCC2 c1(C(=O)NCC(C)CNC(=O)Cc2cn[nH]c2)ccc2c(n1)CCCN2 c1(C(N(C(C(=O)NCC(CC)(O)CC)CC(F)F)C)=O)cnn2cccc2c1 c1nc(Br)n(C)n1.C(C(=O)OCC1CC1)(c1cccs1)NC(C)=O Cc1cc(=O)n(C(=O)CC2CCC2)c(=S)n1S(=O)(=O)CCOc1ccccc1Cl c1(C2(NC(=O)NCCC3(O)CCCOC3)CC2)cccc(Br)c1Cl S(=O)(=O)(c1cc(C(F)(F)F)ccc1F)NC1CN(C(c2ncc(C)s2)=O)CC1O c1(OC)ccc(Br)c(CN2CC=C(CNC(C3OC(C)CC3C)=O)CC2)c1 Cc1nc2cc(Cl)cc(C(N3CC(C)C(C)(C)C3)=O)c2[nH]1.C1(C=O)CC1(F)F.N C1(C(C)NC(c2cc(C(F)F)[nH]n2)=O)CN(C(=O)CN2CCCNC2=O)CCO1 C1(C)(C=O)CC(O)CN1C(=O)CC1(N(C)C)CC1.C(=O)(CCC)O.CC c1(CC)nc(C)c(CC(=O)N(CCC)CC)c(C)n1.C(=O)C(Br)=C(C)C.N c1(NCc2cc(OC)c(N)cc2)nc(C)c2ccccc2n1 N1(C(CNC(CC)=O)=O)CCC2(CC1)CC(C)N(C(c1cc(OC)cnn1)=O)C2 C1(C(N2CCC(C(C)C(=O)N(C3(c4ccnn4C)CC3)C)C2)=O)CCN(C)CC1 CCCC(C)(C)C(=O)NCCNC(C1CN(C(c2nccc(F)c2Cl)=O)C1)=O CCC(CNC(C1CCCOC1)=O)(CC)C(=O)NCc1c(C)ccnc1C C(=O)(CS(N)(=O)=O)NC(c1ccc(F)cc1)CNC(C(C=C)C)=O C1(CC(=O)NCc2ncoc2C2CC2)CN(C(=O)CC2OCCCO2)CCO1 C1(CNC(c2cc(CC)nn2C)=O)C(C)CCCN1C(c1nccc(C)n1)=O CC(CCC(=O)NC(CCO)C1CCC1)NC(C1CC(OC2CC2)C1)=O c1(OC(C)C(N2CCC(CNC(=O)CO)C2)=O)ccc(F)cc1.c1ccsn1 c1(OC)cc(C)sc1C(=O)NCCC(C)(C)C.c1(C(=O)N)cc(CC)on1 C1(CCNC(c2cc(Cl)cnn2)=O)CCCN(C(=O)C(O)CC2CCCCC2)C1 C(=O)(C1=NN(C)C(=O)CC1)NC1C(NC(CCCCOC)=O)CCC1 CCC(CCCC(=O)NC(c1nnnn1C)C)NC(=O)C(O)Cn1cncn1 C1(N(CCC)C(C2CC2C#N)=O)CCN(C(C2CC2c2ccoc2)=O)CC1 C1(C(=O)NC(CC)CNC(c2ccccc2)=O)OCCCC1c1ccccc1 Cc1ccc(C)c(C(=O)NC2(C(=O)NCC(C)C(F)(F)F)CC2(C)C)n1 N1(C(C(=O)NC2CC=CCC2C(F)(F)F)=O)CCC2(CC1)CCC(F)(F)C2 c1(OC)cc(F)cc(C=CC(=O)N(CCC)C)c1.c1(C(=O)N)ncnc(O)c1Cl S(=O)(=O)(c1c(C)noc1C)N1CCCC(C(=O)NC(c2cc(C)oc2C)C)C1 c1(C=O)c(C)ccc(F)c1O.C1(CNC(c2cnn(CC)n2)=O)CCCCC1.N C1(C(=O)NC(CNC(Cc2c(C)nn(C)c2)=O)(C)C2CC2)CC12CCSCC2 N1(C(C(C=C)C)=O)CCCC(O)(CNC(=O)C2=NOCC2)CC1 Clc1ncccc1CN1CCCCC1Cn1ccnn1 N1(C(C2(CCC)CC2)=O)CCC(C(F)(F)F)CC1.C(=O)(CCC(=O)C1CC1)N CC1(C)C(NC(=O)CCS(N)(=O)=O)CCN1C(c1c[nH]cc(F)c1=O)=O N1(C(CCSCCC)=O)CCN(C(=O)CCc2ccc(N)cn2)CC(C)(F)C1 N1(C(C2(C=C)CC2)=O)CCC(O)(CNC(C2C(C)(C)C2(F)F)=O)CC1 CC1(C)CC(C)(CNC(=O)Cc2cnccn2)CN1C(c1cscn1)=O c1(C(=O)NCCNC(C2CC(C(=O)OC)C2(C)C)=O)ccc2ncnn2c1 Cn1nc2ccc(Br)cc2c1CN1CCC(CNC(C2(Br)CCC2)=O)C1 C12(NC(c3n(CC)ccn3)=O)CCCC1(F)CN(C(=O)C(O)CC1CCCC1)C2 c1(OC)c(F)cc(C(=O)NC(C)CNC(C23CCCN2CCC3)=O)cc1Br c1(NC(C2CC(NC(C3C(C)C3)=O)C2)=O)cccc(C#C[Si](C)(C)C)c1 c1(OC)nc(C)ccc1C(N1CC(O)(CCNC(c2occc2C)=O)C1)=O.S c1(C(=O)NCC2N(C(c3c(CCC)n[nH]c3)=O)CCC2)cc2cccc(F)c2o1 CC(C)C(C)CC(=O)NCC(C)(C)NC(C1CC1c1ccccc1)=O CC(C)C(C(=O)NC1CCCN(C(=O)Cc2cocn2)C1)n1ccc(C2CC2)n1 N1(C(c2cnc(Cl)cn2)=O)CC2CC(N=c3[nH]c4cc(Cl)ccc4s3)CC1C2 c1(C(N(C(C)CC)C)=O)cc(S(N)(=O)=O)cs1.C1(C=O)CCN(C(N)=O)CC1 C1(C(=O)NC2C(CC(C)C)C2)CCC2(CCCC2)N(C(=O)O)C1.C(C)(C)C c1(SC)ncc2c(n1)CN(C(C1CC3(C1)CN(Cc1ccc(I)o1)C3)=O)CC2 Cc1ccc(Cl)c(O)c1C(N1CCCOC(CNC(c2cncnc2C)=O)C1)=O c1(CC(N2CC(NC(C3CC(=O)NC3)=O)C3(C2)CC3)=O)ncn2c1COCC2 N1(CC(N2CC(C(N3CC(O)(COC)C3)=O)(CC)C2)=O)CCOCC1=O C12CCCC(CN(C(C3(O)CC(C)(C)C3)=O)C1)C2.c1(C(C)C)nc(C=O)cs1.N C(=O)(CCS(=O)(=O)NCC)NC(CNC(CC(C=C)C)=O)CO.c1ccccc1 CCCC(CCC)CC(=O)NC(C1(O)CN(C(C2CN3CCN2C(C)C3)=O)C1)C N1(C(C(CCC)(C)O)=O)CCC(C)N(C(=O)CCC(CC)CC)CC1 n1(CC(N2CC(CNC(C(C)(O)C3CCC3)=O)C2)=O)cc(Br)ccc1=O c1(C(=O)NC2C3CCCCC23)ccc(C)nc1.c1(C(=O)N)c[nH]cc1C1CC1 CC1(C)CCOC1CCNC(C1(NC(c2ccsc2)=O)CC(CO)C1)=O Cc1ncc(CCC(N2CCS(=O)CC2c2ccccc2)=O)c(O)n1 N1(C(C(CC)NC(N)=O)=O)CCN(C(c2c[nH]nc2OC)=O)CC(C)C1 C1(C)(NC(C2CN(C(C)=O)C2)=O)CCN(C(=O)CCCC2CC2)CC1 c1(C(=O)NCC2CN(C(c3c(C)cc(Cl)cc3)=O)CC2C)nccc2n[nH]cc12 c1(Cc2cnc(NC(C(C)NS(CCCCC)(=O)=O)=O)s2)cccc([N+](=O)[O-])c1 c1(OC)nc(-c2cc(OC(C)C)cnc2F)ccc1C(=O)NCCCC(F)(F)F C(=O)(C1=CC(C)(C)C1)N1C(CNC(C(N2CCC(C)C2)=O)=O)CC1 C#CCCCCCC(=O)NCC(C1CCC1)Nc1ccc([N+](=O)[O-])cn1 C1(CC=O)CC(F)(F)C1.c1(C(N(CCC)CC)=O)cc(-c2ccccc2)[nH]n1 c1(NC(C2(OC)CCC2)=O)cnc(CNC(C(C=C)CC)=O)nc1C c1cccc(S(C)(=O)=O)c1.N1(C(c2cc(C)oc2C)=O)CC(=O)NC(C=O)C1.N C12(C(=O)NC(c3ccc(O)nc3)C)CC(CN1C(=O)C(C1CCOCC1)O)C2 c1(OC)ccc(C(C(F)(F)F)N(C(c2sccc2S)=O)Cc2ccco2)cc1 C#CC1(O)CC(C(N2CC=CC(NC(=O)C(F)OC)C2)=O)C1 c1(CC(=O)N)cc(C)ccc1O.C1(OC)CC(C)N(C(C2OCCC2(C)C)=O)C1 C(CCC(C(=O)NC1CC(C)CCC1O)NC(=O)C1=CCCCO1)OC c1(COC)ccc(C(=O)NC2CC(CNC(C3CCC(C)S3)=O)C2)cc1 Cc1c(F)ccc(C(N2CC(C)OC(C)(C)C2)C(=O)Nc2ccccc2Cl)c1Cl C=CCCCCCCC(=O)N1CCC(N2CCC(NC(=O)C=CSC)C2)CC1 N1(C(c2c(CCC)n(C)nn2)=O)CC(C)N(C(c2sc(C)c(C)c2C)=O)C(C)C1 C1(C(=O)NCC(C)NC(C2CC(N3CCOCC3)C2)=O)(CC)CCCC1 c1(C(=O)NCC(CN(C(=O)CSS(C)(=O)=O)C)O)ccn(CC(F)F)n1 CCC(C(=O)OC)C(=O)N1CCC(C(=O)NCCc2cnn(CC)c2)(CC)C1 N1(C(c2c(COC)cccc2)=O)CC(C)CN(C(c2cnc(C#N)s2)=O)CC1C C(=O)(C1=CC2(CN(C(c3cnc(Cl)s3)=O)C2)OC1)N1CCC(C)(NC(C)=O)C1 C(=O)(C1=CCCC(C)(C)C1)NCCCN(C(=O)CC(=O)N)C(C)C.C1CC1 c1(C(=O)N)c(C)nn2ncccc12.CCC(C(=O)NC(C)(C)CO)NC(C)=O c1(C(=O)NCCCC2N(C(C3ON=C(C)C3)=O)CCC2)ccc(F)cc1C1CC1 C1(CNC(CN2CCC(C)C2)=O)CN(C(=O)CC(=O)NCC2CC2)CCCO1 c1(C(N(CC(CC)NC(CNC(C(CC)C)=O)=O)C)=O)cccc2[nH]cc(Cl)c12 C1(CC#C)CCN(C(=O)CCC2CSCCN2)C1 C(C)(C1CCCc2ccccc21)NC(COC(C(C)=C1CCCC1)=O)=O c1(C(N)=O)cccnc1NC(C1CCC(NC(c2ccc(CO)cc2)=O)C1)=O C(=O)(C(O)C(C)(C)C)NCCCC1N(C(CNS(CCCC)(=O)=O)=O)CCCC1 Cc1cc(C(N2CC(F)CC2CC(=O)N(C2CCCOC2)C)=O)cnn1 C1(NC(C2(NC(C(C)c3cc[nH]n3)=O)CCCC2)=O)CC2CC1C(O)C2O c1(C(=O)NC(C=C)C)nc(CNC(=O)C(CC)NC(N)=O)oc1C CC1=C(C(=O)NC2COCCC2NC(c2cc(Br)cn2C)=O)CCC1 CC1(C(=O)OC2CCCC2c2ccc(F)cc2)CC2CC2C1 n1(CC)cc(NC(C2(C)CCCN2C(=O)CC2(CC)CCC2)=O)c(C)n1 c1(OC)ccc(C#N)cc1CN1CCC(NC(C2(N(C)C)CC2)=O)CC1C c1(C(=O)NC(CC)CNC(=O)CC2C=CCCC2)ccc2cccnc2c1F Cc1oc([N+](=O)[O-])cc1C(N1CCCCCC1CNC(=O)CCC(C)(F)F)=O c1(C2(Nc3ccc(C(=O)NCCOC)nc3)CC2)cc(C)cnc1O c1(SC)ccc(NC(C2(NC(c3cc(C)on3)=O)CCSC2)=O)cc1 C(=O)(CC(O)CC(C)C)NC1CC2(CC(C(=O)NC)C2)C1 N(C1CCCc2ccoc21)C(C1CC(CNC(C2C(C)CCCC2)=O)C1)=O CCC(C)CC(=O)C(=O)NCCOCC(=O)NCc1ccc(C)cc1C c1(C(N(CCNC(C2C(C)CC2)=O)C2CC2)=O)cccc(N)c1 C1(CN(C(c2c(CCC)nco2)=O)C)C2CN(C(c3csc(Cl)c3)=O)CC12 C1(NCc2cn(C(C)C)nc2Br)CC(C)CN(Cc2ccc(C(=O)O)cc2)C1 c1(C(N(C)C(C2CCC(C(F)(F)F)CC2)=O)=O)cc[n+]([O-])cc1 c1(CC)cccc(CNC(=O)C(CC2CCC2)NC(C2(C)CCOC2)=O)c1 CCC(C)C(C(=O)N=c1ccn(C)[nH]1)N(C)C(C1CCN1CC)=O N1(C(C=COCC)=O)CCC2(CC(NC(=O)C(=O)Nc3ccc(C)cc3)C2)C1 C(C(C)(O)C(C)CC)NC(C1CCCC(NC(C2(OCC)CC2)=O)C1)=O N(C1CCOc2c(Cl)cc(Cl)cc21)C(C(C)C(C)(F)F)=O c1(CN2C(C(=O)OC)CSCC2)cc(OC)c(OC)cc1F C(CC(=O)NC1CCC2(CC2)C1)(C(F)(F)F)NC(C(CC(C)C)=O)=O c1(C(=O)NC(C(C)C)CCN(C)C(c2ccccn2)=O)cccc2nsnc12 C1(c2n(C)ccn2)CN(C(C2(CO)CCC2)=O)CC1NC(c1ccon1)=O c1(C(N2C(C(C)NC(=O)C=Cc3nccs3)CCC2)=O)coc2cc(O)ccc12 C1(C(=O)NCC)(C(C)C)CCN(C(=O)Cn2cccc2)C1.CCCCSC.O CCC(C)CC(CO)NC(=O)CC1CCCCC1.C1(CC(=O)N)CC(N(C)C)C1 C(=O)(CC(F)(F)C(F)F)NC(CC(=O)NC(CC#C)CC(=O)OC)C(C)C c1(CC(=O)NCc2cc(CC)[nH]n2)c(C)cccc1Br.C(=O)C(C)C(C)C.N c1(CNC(C2(NC(C(C)CC3CCC3)=O)CC2C)=O)c(F)cncc1F N1(C(C2CCN(C)C2=O)=O)CCCC(NC(C2CC(C)(F)C2)=O)CC1 C1(C2CCCN(C(c3cc(C)ccn3)=O)C2)(NC(CCNC(C)=O)=O)CC1 CC(C(=O)N(C1(C(N)=O)CC1)C)P(C)(C)=O C1(C(N2C3CC(C3)C2)=O)CCCCN(C)C1=O.Cc1ncc(C=CC(=O)NC)s1 C=CCC(CC)C(=O)N1CC(CCNC(c2sc(C)cc2Br)=O)(OC)C1 C=CCC(CC=C)C(=O)NCC1(O)CCN(C(=O)Cn2cnc([N+](=O)[O-])n2)CC1 n1(CC)c(CSCCS(=O)(=O)N(c2ccccn2)C)nnc1SC N1(C(C(C)SC)=O)CC(C)(C)CC1CNC(=O)C(C)O.C1CCCCO1.C N1(C(C(C2CCC(=O)N2C)C)=O)CCN(C(C2CN(C(=O)CC(F)F)C2)=O)CC1 CCC(C(=O)NCC1(CO)CCN(C(=O)COc2ccccc2Cl)CC1)C(C)C CCC(CC(C)C)C(=O)NC1CC(C)N(C(c2ccc(C(OC)OC)o2)=O)C1 c1(NC(C(CCNC(C2N(CC)CC2)=O)O)=O)ccc2cnccc2c1 c1(N2C3C(NC(c4c(C)nc(C)s4)=O)(CCC3)CC2)ncnc2c1CCCC2 c1(C(=O)NC(C(C)C)CNC(=O)C=CC(N2CCOCC2)=O)cccc[n+]1[O-] C(=O)(C(C)CC(F)(F)F)N1CCCC(C)(C(N2CCC(C(C)C)CC2)=O)C1 C(=O)(CCN(OC)C(=O)Cc1cccc(C#N)c1)NC(CC=C)CC C1CCC2(CN(C(=O)CC3CCC(O)C3)C2)O1.N1(CCC(=O)N)CCC(F)C1.C N1(CC(=O)NCC(C)N(C(=O)CC2(C#N)CCOCC2)C)Cc2ccccc2C1 c1(NC(C(C(C)C)CN(C)C)=O)ccnc2ncnn12 C1(C(=O)NCc2cccc(CN(C(C)=O)C)c2)CC2CCCCCCC12 c1(OC)ncnc(OC)c1C=O.C1(CC=O)CNC(=O)C1.CC(C)C1CC1.N C(=O)(C1CCc2cccc(=O)n21)N1CC(C)N(c2cc(F)c(Br)cc2F)CC1 Cn1oc(C(=O)NCC(CNC(=O)Cc2cncc(Br)c2)CO)cc1=O Cn1ncc2cc(CC(N3CC(NC(C45CCC(C4)C5)=O)CC(O)C3)=O)ccc12 C1(C(=O)NCCCN(C(=O)C=CBr)CC2CCCC2)CC(=O)N1 Cc1cc(O)nc(Cc2cn(C3CCCC(N4CCCC4=O)C3)nn2)n1 C1(C(=O)NCC(C(N2C(C=C)CC2)=O)O)CC2CCC1CC2 Cc1cc(C)n2ccc(C(=O)NC(c3ccc(Cl)cc3)C(C)C)c2n1 c1(C(N2CC(NC(CCC(C)C)=O)C(n3ccnn3)C2)=O)ccc2nsnc2c1 C(C(CC(C)C)C(=O)N(CC(C)C#N)CC)NC(CCCC(=C)C)=O c1(-c2c(CN(C)C)nc[nH]2)nc(-c2ccncc2)nn1C1CCOCC1 C1(OC)(CNC(c2cnn(C3CCCC3)c2C(F)(F)F)=O)CCCC(C)C1 Cc1cc(C(=O)NC(Cn2ccnn2)C(=O)NCc2ccns2)nc(O)c1 C1(C(=O)OC)CCOCCN1C(CCC1CC=CCC1)C(=O)NC1CCOC1 c1(C(=O)N)cc(C)n(C2CC2)c1C.Cc1cc(C(N2CCC(CC)C2)=O)c(C)s1 c1(C(C)C)nc(NCCC2CCCC(C)(C)C2)cc(=NC2CC(=C3CCC3)C2)[nH]1 c1(CC(N2CCC(C(C)(C)NC(CCCOCC)=O)C2)=O)cnn2c1OCCC2 N1(C(C=Cc2c(C)ncs2)=O)CCC(NC(=O)CCn2ccnn2)CC1C1CC1 C=C(F)C1(CC(N2CC3CC2C3C(=O)NCc2cnn(C)c2O)=O)CCC1 C1(CN(CCOC)C(c2scc(OC)c2)=O)CCN(S(C)(=O)=O)CC1.O N1(C(c2nccc(C#C)c2)=O)CCC2(C1)CN(C(c1cn(C)c(=O)nc1O)=O)C2 C1(C(N2CC(N(C(CC(CC)C)=O)C)C3(C2)CC3)=O)Cc2ccccc2C1 CCC(CC)CCCC(=O)N1CC(n2cc(CNC(=O)C(C)C(F)(F)F)nn2)C1 C(C)(N=c1cc(C)nc(C)[nH]1)C1CCN(C(C(C2CCOC2)OC)=O)C1 Oc1nc2ccc(CSCCCNC3CCOC3)cc2n1CCc1ccccc1 C1(CC(=O)NCc2ccc(C(=O)OC)cc2)CCC(C(F)(F)F)N(C)C1 CCCCCCC(CC)C(=O)NC1(CF)CCN(C(=O)CC2CC2(C)C)C1 CCC(C)CCC(=O)N1CCCC(CCNC(c2cnc(=N)[nH]c2)=O)C1 C(=O)(C1=C(Cl)CCCC1)N.c1(OC)ncncc1NC(C1(C)CC12CCC2)=O N1(C(Cc2nc(CC)sc2)=O)CCC(C)(CNC(=O)C(C)=CC2CC2)C1 C12(C(N3CC(CNC(c4cc(C(F)F)[nH]n4)=O)OCC3)=O)CCC(C1)OC2 Cc1c(Cl)sc(Cl)c1C(=O)NC(C1CCCN1C(=O)CCc1cn[nH]c1)C N1(C(=O)NC(c2cccc(Br)c2)C#C)CC2COCC(C(=O)OC)(C1)C2(F)F C1(C#CC(=O)NC(CCC(C)C)C(=O)N2CCCC2CCOC)(CC)COC1 C1(C(C)C(=O)N(C2CCCC2)C)CCN(C(C2(N(C)C)CC2)=O)C1 c1(C=O)ccc(C#N)cc1C.C1(C(=O)N)(COCC)CC1.C1(CC)CC1 C1(NC(c2cc(C(C)C)on2)=O)CCCCCN(C(=O)C2=CC(O)CCC2)C1 C(=O)(C1=CCCCC1C)NCC(C(N1CCC(C2CC2)C1)=O)OC C1(C(=O)NC2CC2)CC2(CCN1C(c1ccccc1CCF)=O)CC2.C1CC1 Cc1cccc(OCC(=O)NCCC2CSCCN2C(C2CC2(C)C)=O)c1 C(=O)(C(C(=O)NC1CC(C)N(C(c2ccc[n+]([O-])c2)=O)C1)C(C)C)OCC N1(C(C(CC(C)C)NC(CCCCCSC)=O)=O)CCn2ncc(O)c2C1 C=CCC(C)(C)C(=O)NCC1(C(F)F)CCN(C(=O)C(C2CCCCCC2)O)C1 CC1CC(NC(=O)Nc2ccc(-c3nnco3)cc2)CN1C1CC1 C1(CNC(C(CC)(C)F)=O)CC2(CO1)CN(C(=O)C)C2.c1ccc(Cl)cc1C.O N1(C(C2C(CC)CCC2)=O)CC(F)(F)CC1CCNC(=O)CC.C(=O)C c1(C(=O)OC)ccc(C)c(C=O)c1.C1CN(C(=O)Cc2csc(C)c2)CC1F.N Cc1sncc1C(N1CCC1C(=O)NCCOCC(N)=O)=O CC1CCN(C(c2ccc(C3CC3)o2)=O)CC1N(C(=O)C1=CC(C)(C)C1)C N1(C(C=Cc2c(C)cccn2)=O)CCOC2CN(C(C3C(C)(C)C3(F)F)=O)CC12 N1(C(C=CS(C)=O)=O)CC2CCN(C(c3ccc(OC(F)F)cc3)=O)CC(C2)C1 c1(C=O)cc(F)cc(Cl)c1O.C1(C(NCCC)=O)CS(=O)(=O)CC12CC2.CC CCCC(C)C(=O)N(C)CC1CN(C(=O)CC(c2cccc(OC)c2)C)C1 N1(C(=O)CSC2CC2)CCCCC1C1CCCN1c1nc2ccc(O)cc2s1 c1(OC)cccc2cc(C(=O)NC3CC3NC(=O)C=CC3CCCO3)[nH]c12 N1(C(C2CCN(C)C2)=O)CC2CCC(C1)C2CC(=O)NCc1cocn1 N1(CCN(CCC)CCC)C(=O)CN(CCOC2(CC)CCSC2)C1=O c1(OC(=O)NC2(c3cccc(F)c3Br)CC2)cc(OC(F)(F)F)ccc1Br c1(C(N2CCC(O)C2)=O)cc2c(F)cc(Cl)cc2[nH]1.C1(C=O)(C(F)F)CC1.C CCCCC(O)C(C)C(=O)N1CC2CC2(C(=O)NCC2(C)CCCS2)C1 CC1(CO)CC(NC(C2(CNC(=O)CC3CCCCC3)CC2)=O)C1 N1(C(Cn2c(C)ccn2)=O)CC2CC1CCC2NC(c1cn(C)c(=O)cn1)=O C12(C(=O)NC3CC(C)N(c4ccnc(C(N)=O)n4)C3)CCCC(C1)OC2 c1(NC(C2CCN(C(c3cn(CC=C)nc3)=O)C23CC3)=O)cccc(C#N)c1C C#CCC(C)(CC)C(=O)N1CCCC1CNC(=O)CCCc1cc(C)no1 C1(C(NNC(=O)c2cccc(CN3CCSCC3)c2)=O)Cc2cc(Cl)ccc2O1 C1(CC)C(NC(=O)C2=COCC2)CCCN1C(c1cc(C2CC2C)on1)=O C(=O)(C(CC(F)F)NC(C1C=CCS1)=O)NCC1(N(C)C)CCCC1 c1(NC)snc(C)c1C(=O)NCC1CCN1C(=O)CCNC1CCC1 C=CC(C)(C)C(=O)NCC(CNC(=O)CN1CCC(F)(F)C1)OC N1(c2c(C#N)nccn2)CCC2(CCCC2CNC(c2cc(Cl)no2)=O)CC1 CS(=O)(=O)c1ccccc1-n1nc(-c2nccs2)nc1Cc1csnn1 Cn1ncc(C(=O)NCC2COC(CNC(c3ccc(O)nc3)=O)C2)c1Br C(=O)(CCCCCO)OC.c1(N(CC)CCNC)nnnn1C1CCC1.C(C)C C(c1ccc(COC)s1)=CC(=O)NC1CN(C(C2CCC(CC)O2)=O)C1 CS(=O)(=O)c1ccc(CN2CC3OCCN(C)C3C2)cc1.C1CN1 c1(C(=O)NCC(CNC(CC(C)n2ccnc2)=O)(C)O)ccc(F)c(Cl)c1F C(=O)(C(C)C(C)COC)N(CCOC)CCNC(=O)C(C)(C)SC C1(NC(Cc2c(C)cnn2C)=O)CCCC12CN(C(C1CCC(F)(F)C1)=O)C2 C#CCC(C)(C(=O)N1CC(OCCCC)C1)NC(=O)C(C)OC Cc1c(C(=O)NCC2CC2)sc2[nH]cnc(=O)c12.O(CP(C)(C)=O)CC=O c1(CC(=O)N(C(C)C)CC)cc(OC)c(O)cc1F.C(=O)CCc1nncs1 N1(C(CC(C)c2ccco2)=O)CCOC2(CCN(C(=O)C3=NOCC3)C2)C1 c1(C(=O)NC23CN(C(C4N(C(C)C)C(=O)CC4)=O)C(C2)C3)cccc2nc[nH]c12 c1(C(C)OC)nc(-c2cc(=O)cc[nH]2)n(-c2cccc(NC(C)=O)c2)n1 CC1(C)CC(C(=O)Nc2cc(O)cc(F)c2)CN1C(=O)CCCC1CCC1 C1(O)(CNC(c2ncc(C(F)F)s2)=O)CCN(C(=O)CO)C1.CC(F)F C1(NC(CN(C(=O)OC)C)=O)CC(C)C12CCC2.n1(CC=O)cccn1.N C(CCC(O)C(=O)NCC(F)(F)Cl)NC(=O)C=Cc1nccs1 C12(NC(Cc3n(C)ncc3Cl)=O)CCCC1N(C(=O)C1=CS(=O)CCC1)CC2 C(=O)(CCCCCCCO)N1CC2N(C(c3cc(C)c(Br)cc3C)=O)C(C2)C1 C12(NC(c3c(SCC)cccn3)=O)CCCCCC1N(C(=O)C(C)COC)CC2 N1(C(c2c(CCC)[nH]cc2)=O)CCCN(C(c2c(C)noc2C2CC2)=O)CC1C N1(C(=O)OCCC)CCN(N(CC2CC2)CCCO)CC1 C(=O)(C1=CC2CCC1C2)N1CCC(C(C)NC(C2CN(C(C)C)C2)=O)CC1 c1(C(=O)NCCC2(OC)CN(C(C3(C#N)CC3)=O)C2)ncc2ccccn12 C(=O)(C(C)(C(F)(F)F)c1cc[nH]n1)NCCC(C)NC(=O)Cn1nccn1 C1(C(N(C)Cc2c(C)ccnc2)=O)CN(C(c2c(C)nn(C)c2C)=O)CC1(C)C C=CCC(C(=O)NCC1CCCN1CCC)NC(=O)CC1CCCC(C)O1 c1(C(N2CC(CNC(C3CCCO3)=O)C(O)C2)=O)n[nH]cc1[N+](=O)[O-] N1(C(C(C)OCC=C)=O)CC2(CCOCC2C(=O)Nc2ccon2)C1 C(CCCC(=O)NC1CC(F)CN(C(=O)C(C(C)C)SC)C1)(OC)OC C(=O)(NNC(=O)CCCO)c1ccc(CC#N)cc1 CC1CCC(C(=O)NCC2CCCCN2C(=O)CCCc2ccncc2)CC1 c1(C(N2C(c3cn(Cc4occ(C)n4)nn3)CC2)=O)cc2oc(Br)cc2[nH]1 c1(CC)nn2c(=O)cc(Cc3cnn(C(C)C(=O)N4CCCC4)c3)nc2s1 C(CCC(F)(F)F)NC(=O)COCCF.c1(CC=O)cccc(C(F)(F)F)c1 Cc1cc(Br)ccc1CCC(N1CCC(N(C)C(C2CC2C)=O)C1)=O c1(C(=O)NC2CC(C)(NC(C(C)NC(CC)(C)C)=O)C2)ccncc1C CC(C)(C)C(C(=O)N1CC(O)(CCNC(c2ccon2)=O)C1)N1CCNC1=O C12(C(=O)Nc3c(C(=O)NCC(C)C)nn(C)c3)CCC(F)C1CC2 Cc1cc(C(=O)NCC2CCN(C(c3cc(C)n(CCO)n3)=O)C2)c(Cl)cc1F c1(C(N(C(CCNC(Cc2c(C)nc(S)s2)=O)C)C)=O)ccc(N)c(C)c1C c1(C(=O)NCCC(C)NC(C2COC(=O)O2)=O)cnn(C)c1C(F)F C(=O)(C1=C(Cl)CC1)NCC(CCNC(CN(c1ccncc1)C)=O)O c1(C(N2C(COC)CN(C(=O)C(C)C(C)C)CC2)=O)ncnc2sccc12 CC1C(=O)N(C)CN1C(=NCCc1cn(C)cn1)NCc1ccc(F)cc1 C#CC(C(C)C)NC(=O)NC(C)CCCO C=CCCCC(C(=O)NCC1CC1)NC(C1CN(C(=O)NC)C1)=O CCC(CC)(C(=O)NC(C)C1CC1)c1ccccc1.C(c1cn[nH]c1)=CC(=O)N C(CN=c1[nH]c(=NC2CCS(=O)(=O)C2)[nH]c2cc[nH]c12)(c1ccc(Cl)cc1)OC N1(C(CC2CC(NC(C(CC)N(CC)CC)=O)C2)=O)CC(O)C(F)C1 Cc1cc(C)n2c(NC(N3CCC(NC(C4COCCO4)=O)CC3)=O)nnc2n1 CC(CCCCNC(=O)CC1CCC(=O)N1C)NC(=O)C(F)(F)CC1CC1 N1(C(C2C(CC)CCC2)=O)CCC12CN(C(c1cc(C(F)(F)F)ccc1F)=O)C2 N1(C(CC2CC(CC)C2)=O)CCCCC1CN(C)C(c1nnn(C)c1N)=O C1(C(=O)NC(c2ccc(Br)cc2)C(F)(F)F)CC(O)CNO1 CC(C)(C)C(C#N)C(=O)N1CCC(n2cc(Cn3cncn3)nn2)C1 c1(C(N(C2CCN(C(c3cn(C)c(O)n3)=O)C2)C)=O)cc2ccncc2cc1F Cc1coc(C)c1C=CC(=O)NC1CC(CNC(=O)C(C)C(F)F)C(O)C1 CC1CN(C(c2ccc(CO)o2)=O)CCN1C(=O)CC1(C#N)CCC1 N1(C(c2cc(OC)ns2)=O)CCN(C(C2CCCCCCC2)=O)CC(C)(F)C1 C1(C(F)(F)F)(C(N(C2CCN(CCC(=O)O)CC2)CCO)=O)OC2CCC1CC2 CCC(C)C(O)C(C)C(=O)N1C2CCCC1COC2 CCCCC(CCCC)N=c1nc(N2CCC(CF)CC2)c2cccc(F)c2[nH]1 N1(C(c2nc(O)[nH]c(=O)n2)=O)CC2CCCCC2(CNc2cc(O)ncn2)C1 c1(C(=O)NC(COCC)C(=O)NCc2csnc2OC)cnc(=N)[nH]c1 n1(CCC=O)cc(Br)ccc1=O.C(C(=O)NCC1CC1)=CCN(C)CC O=S(=O)(c1cc2sc(N3CCCC3)nc2cc1Cl)NC1CCCC(F)C1 C(=O)(C(O)C(C)(C)C)NC1CC(OC(C(=O)NCCN(OC)C)C(C)C)C1 N1(C(C2=CC(O)C(NC(CP(C)(C)=O)=O)C2)=O)CCc2ncncc2C1 N1(C(Cc2n(C)cnc2)=O)CCC2(CC1)CC2C(N1CCCC(CCO)CC1)=O Cc1cnn2cc(NC(=O)CC3CS(=O)(=O)CCN3)cnc12 C(=O)(N=c1nc(OC)[nH]n1C)NC(C1CCCOC1)COC N1(C(CCCOCCOC)=O)CCC(CC(C)NC(C2(F)CCOCC2)=O)CC1 Cc1cnc(NCc2cc(C)sc2C)c(S(=O)(=O)N2CCCC(C)C2CCO)c1 C1(C)(C(N(C)C)=O)C2Cc3ccccc3C12.Cc1sccc1CC(=O)NC1CC1 N1(C(c2c(CC)cccc2)=O)CCCCCCC1Cc1nn[nH]n1 CN1CCC(NC(c2cn(Cc3cccnc3)nn2)=O)CC1.C(C)(C)C.C=O.C c1(-c2c(OC)cc(F)cc2)cccn2ncc(C(=O)NCc3ccc(I)cc3)c12 c1(C(N2C(CNC(=O)Cc3c[nH]nc3O)CC2)=O)cc(F)cc([N+](=O)[O-])c1Br NS(=O)(=O)c1csc(C(=O)NC2(CO)CN(C(c3nccn4nccc34)=O)C2)c1 C1(C(=O)NC2CC(NC(c3cc(CO)[nH]n3)=O)C2)CC12CCCCCC2 Cc1cc(C(=O)NC2CC(N(C)C(C3CN4CCCC4CO3)=O)C2)ccc1C#N c1(C(C)(C)C)cc(Br)ccc1N=[N+]=[N-] C(=O)(C(CNC(=O)Cc1cncn1C)C(C)C)N1CCC(OCC=C)CC1 N1(C(C(c2n(C)ncc2)O)=O)CCN(C(c2ccnn2C2CC2)=O)CC(C)(C)C1 Cc1ccc(C(=O)NC2CCCC(NC(c3[nH]c(O)nc3C)=O)C2)c(Cl)c1 N1(C(CC2CC(C)OC2C)=O)CC(NC(c2ccc(C(C)(C)C)s2)=O)CCC1C C1(NC(C(C)N(C(=O)C(C2CCC2)OCC)CCC)=O)CC(C)CCC1O c1(CC)nn(C)cc1C(=O)NC(CNC(C1CCCCO1)=O)CC c1(CC(=O)N(C2CCCN(C(C34CC(O)C3C4)=O)CC2)C)c[nH]c2ccccc12 C1(CC(N2C(CNC(C3CCC=CO3)=O)CC2)=O)CC2CCC(C1)C2 N1(C(C(CC)C#N)=O)CC(NC(=O)Cc2cncc(F)c2)CC(F)C1 c1(C(N(C2CC3CC2CN3)CC(c2ccc(C)cc2)C)=O)cc(F)cc(Br)c1F Cc1cc(C(=O)NCC(O)CNC(c2conc2C2CC2)=O)c(N)c(Cl)n1 c1(NC(CN(C(C(C)CC2CCCC2)=O)C2CC(C#N)C2)=O)cccn2ccnc12 c1(CC(=O)Nc2scc(C)n2)ccc2oc(O)nc2c1 C=Cn1nncc1C(=O)NCC1CCCN(C(c2[nH]c(C)nc2CC)=O)C1 N1(C(=O)OC)CCCC(N=c2nc3sccc3c(NCCCn3ccnc3)[nH]2)C1 C(=O)(N=S(C)(=O)c1cnn2c1CN(C(=O)CC(F)(F)F)CC2)c1cc(C)on1 CCC(CC)CC(=O)NCC1(OC)CCN(C(c2cc3[nH]ccc3s2)=O)C1 Cc1[nH]nc(C(=O)NCC2CCC2NC(c2cc(O)n(C)n2)=O)c1[N+](=O)[O-] CC1C(C)N(C(c2cnn3c2CCCC3)=O)CCN1C(=O)CCc1ccnn1C c1(-n2cc(C(CC)OC)nn2)cccc(C(=O)NCC(C)(CSC)CO)c1 N1(C(c2c(C)noc2)=O)CCC2(CCCCC2NC(=O)CC(C)NC(N)=O)C1 N1(C(C(C)C(C)O)=O)CC2(CC(NC(c3cnn4cccnc34)=O)CO2)C1 c1(C(=O)NCCCN(C(C(CC=C)OC)=O)CCO)cc(F)c(C)cc1N C=CCC(CNC(=O)CC1CCC(O)C1)NC(=O)CC=C CCC(C(=O)NCC(C)(CNC(C1CC1C1CC1)=O)OC)N(C)C C(=O)(C1=NOC(C)C1)NCC(C)(C1CCC1)NC(c1scc(C)c1Br)=O O=C1CN(c2ccc(C(=O)NCC#CCNC(c3cnc(Cl)s3)=O)cc2)CCN1 Cc1coc(C)c1C=CC(=O)NC1CCN(C(=O)C(F)n2cccn2)C1 c1(C(N2CCCC(NC(C(CC)SC)=O)(COC)C2)=O)cc(F)c(F)cc1OC N1(C(c2cc(C)c(O)cc2)=O)CCOC2CN(C(C3CC(C(F)(F)F)C3)=O)CC12 C#CCCCC(=O)NCC(C)(C)Cn1cc(CN(S(C)(=O)=O)C)nn1 C(=O)(C(C)C(CC)CC)N.C1(CC(N2CC(CC=C)C2)=O)C=CS(=O)(=O)C1 C(=O)(CCC(=O)c1ccccc1)NCC(CN(C(=O)C=CS(C)=O)C)O C=C(C)C(C)(C)C(=O)NCC1CC(C)CN(C(c2ccc(Cl)o2)=O)C1 c1(NCC2(C(C)(F)F)CCC2)ncccc1S(=O)(=O)NC1(CO)CCC1 CC(C1OCCc2sccc21)NC(=O)Nc1nc(C2SCCCS2)cs1 CC(C)CCC(C(=O)NC1CC2(C1)CC21CCC1)NC(=O)CSC1CC1 CC1(NC(=O)C(O)C2CC2)CCN(C(C2(Cl)CC2(C)C)=O)CC1 Cc1cc(C(N2CC(CNC(C3(Br)CC3)=O)C(C)C2)=O)nc(C)c1 CC12CN(C(=O)C(F)(F)C(F)F)C(C(N3CCC3C3CCCC3)=O)(C1)C2 N1(C(CCOCC#C)=O)CCC(C(CO)NC(=O)CC2C=CCC2)CC1 C1(CNC(c2ccc(Cl)cc2)=O)CC2(CCN(C(=O)C3CC3)CC2)C1 C1(CCOC)(NC(c2cccc[n+]2[O-])=O)CCN(C(=O)CC2CCC3CC23)CC1 N1(CC(=O)N(CCOC)Cc2ccc(Cl)cc2)CCC(C)S(=O)(=O)CC1 CC1=NOC(C(N2CC(NC(=O)Cc3ccco3)C(C)C2)=O)C1C C1(C(=O)N)CC2CCCC(C1)C2=O.CN1CCC(=CC(=O)NC2(C)CC2)CC1 CC(C)(CCC(=O)N1CCC(n2cnnn2)C1)NC(C12CSCC1C2)=O c1(C(=O)OCc2cnn(Cc3ccccc3)c2)nccc2nc[nH]c12 C=C(C)C1OCCC1C(N1CCCC(NC(=O)Cc2scnc2C)CC1)=O N1(C(CCc2ccc(C)cc2)=O)CC2(C1)CN(C(C1CCC(C#N)C1)=O)CCO2 C(=O)(C1CCCc2cncn21)NC1C(CC)CN(C(=O)C(C)NC(C)(C)CC)C1 C(CCC(C)(C)C(=O)NC(CCCC)CCCC)NC(C1CC(=C)C1)=O N1(C(C2C(OCC)C2C)=O)CCCC(C2CCN(c3nn4cc(C)nc4s3)C2)C1 n1(CCOC)ncc(C(=O)NCC2(F)CCCC2)c1C.C(=O)C(C)(C)F.N CCC(C)(CC)C(=O)N1CC2CC2(CNC(c2cc(C)oc2C)=O)C1 C(=O)(C1=CCCSC1)NCC(C)NC(c1c[nH]nc1[N+](=O)[O-])=O CC1CC(NC(=O)CCc2cn[nH]c2)CCN1C(=O)CC1CC(=O)C1 c1(NC(=O)CC2CC(OC(F)F)C2)ccc(F)cc1[N+](=O)[O-] C#CCC(O)C(=O)N(C)CCC1CCCCN1C(C1C2CC3C(C2)C13)=O N1(C(C(c2cccc(OC)c2)(C)C)=O)C2CCC1CC(N(c1ccncn1)C)C2 c1(CC(N2CCC(NC(C3CCCC(C(N)=O)C3)=O)C2)=O)ccc(C)nn1.C C1(C(=O)N(CC(O)CN(C(=O)Cc2cc(C)cs2)C)C)C=CCC1.COC Cc1cccc(CC(=O)N(C)Cc2ccccc2CNC(=O)CCC2CC2)c1 N1(C(c2cncc(C)c2)=O)CC(NC(c2ccn(C(C)(C)C)n2)=O)CC(C)C1 N1(C(CCCC2C(C)C2)=O)CCCC(O)(CN(C)C(c2cccnn2)=O)C1 c1(C(C)C)nc(N(C)CC2CCCN2C(C2C(C)(C)C2(C)C)=O)cc(Cl)n1 c1(C=O)cnc2cccc(C)n12.C1(NC(C2C(CC)C2)=O)(C)CCCCC1C.N N1(C(C(CC)C(C)C)=O)CCC2(CC1)CN(C(C1(C)CS(=O)(=O)C1)=O)CC(C)O2 c1(OC)ccc2[nH]cc(C(C)CNC(=O)CSc3ccc(C#N)cc3)c2c1 C(C1(C)CCOCC1)=CC(N1C(C)CC(C)C1)=O.C(=O)(CC)N.C(=O)C=CCl C1(C(N2CC3C(NC(Cn4nnc(C)n4)=O)C(C3)C2)=O)CC2CCC(C1)C2O CC(C)C(O)C(F)(F)C(=O)N(CCCCNC(=O)C(F)C(C)(C)O)C c1(C(=O)NC2CCCC(NC(c3n(C(C)C)nnc3)=O)C2)cc2sccc2[nH]1 N1(C(C2CN(C(N)=O)C2)=O)CCC2(CCC(NC(C3CCOCC3)=O)C2)CC1 c1(-n2cc(CNC(=O)CC3(CO)CCC3)nn2)cncc(F)c1 C12(NC(CCSC)=O)CCCC1N(C(c1cncc(NS(C)(=O)=O)c1)=O)CC2 C1(CC(N2CC(CC)C2)=O)Cc2cc(F)ccc2O1.CC1(C(=O)N)CNC(=O)C1 C1(C(N2CCC(NC(=O)NC)CC2)C(=O)N)CCOC(C)(C)C1.CCC1CC1 CC(C)C(C(=O)N1CCCC1CN(CC(Cl)=CCl)C)N(C)Cc1ccccn1 N1(C(c2n(CCC)nc(C)c2)=O)CC2(C1)CN(C(=O)C(C)CCO)CC(C)(C)O2 C1(C(N(CCNC(CS(=O)(=O)NCC)=O)CC)=O)CC2CCCCN2C1 Cc1cc(C(=O)NCC(C2CC2)NC(=O)CC(C)c2ccccc2)c(C)s1 c1(C(N2CC(F)(C(N3CC4CC3C3CC43)=O)C2)=O)n[nH]c2ccccc12 C1(NC(C(C)n2cccn2)=O)CCCCCN(C(C2(C)CCCCC2)=O)C1 N1(C(C)=O)CCCN(Cc2ccc(-c3ccccc3C(F)(F)F)c(F)c2)C(C)C1 C(=O)(CC(C)(C)CC(=O)N1CCCC1C(C)NC(c1nnsc1C)=O)OCC Cc1cc(N2CCN(c3ccncc3)CC2)nc(=NCc2ccc(N)cc2Cl)[nH]1 CCC(CC(=O)N1CCC(C(=O)N(C)Cc2cncs2)C1C)C(F)F c1(C=O)cccc(C(N)=O)c1.C1(CNC(C(C2CCCC2)SC)=O)CCCC1 Cc1sc2ccc(Br)cc2c1C(=O)NC1(CC(=O)O)CCCOC1 c1(N2CCC(=CBr)CC2)nc2c(c(=NCC3CC4(CCC4)CO3)[nH]1)CSC2 C1(C)(C(=O)NC(CCCC)CNC(=O)C=Cc2ncc(C)[nH]2)CCC(O)CC1 C1CN(C(C2(c3ccnc(Cl)c3)CC2)=O)CC(C)(C)C1.C(CC(C)C=O)=CC.N CC1=C(C(=O)N2CC(CNC(C3CC(OC4CC4)C3)=O)C(C)C2)CCCO1 C1(CC=C)(NC(C2CCC2C)=O)CCN(C(=O)CCN(S(C)(=O)=O)C)C1 C1(C)COCCN(C(c2c[nH]c(=N)o2)=O)C1.c1(CC(C)C)ccc(C(=O)N)s1.C N1(C(C(CC#C)(C)CC)=O)CCCC2(CCCN2C(c2cc(F)n[nH]2)=O)C1 c1(C(N(CC(CC)NC(C2ON=C(CC)C2)=O)CC)=O)cc(SC)ccc1Cl c1(OC)cccc(CC(=O)N)c1F.C1(CC(=O)N(CCC)C2CC2)CC1(Cl)Cl n1(CC(=O)N(CC(N)=O)C)cc(CCC2CCCN2C)nn1 Cc1nc(CC(C)C)sc1C(=O)NCC(C)C1CC1.c1(C=O)cn(C)nc1Cl.N C1(NC(C(c2cccnc2)C)=O)CCC2(CC1)CN(C(c1ccsc1)=O)C2 c1(CC)c(C(c2nnnn2Cc2ccccc2)NC2CSC2)cnn1C c1(OCC(C)CNC(=O)NCCOc2cccnc2)ccccc1Cl c1(OC)cccc(C(=O)NCC(C)NC(=O)Cc2cccc(OC(F)F)c2)n1 c1(C(=O)NC2CC(NC(c3c(C=C)cnn3C)=O)C2)cc2ccncc2cc1F N1(C(C2(OC)CCN(C(=O)Cn3cc(CO)nn3)C2)=O)CC2(CCCC2)C1 C1(NC(c2c(C(N(C3CC4CCC3O4)C)=O)n[nH]c2)=O)CCC=CCC1 N1(C(C(C)n2ccnc2)=O)C2CCC1CN(C(=O)C(C)(F)F)CC2 CN(C1CCOc2ccc(F)cc21)C(=O)CCc1nc2ccccc2o1 CC(C)CC(CNC(C1CC(O)C(F)C1)=O)C(=O)NC1CC2C(C1)C2(F)F O=C(C1=CC2CCC=CCCC12)NC1CCCN(C(C23CC(C2)S(=O)(=O)C3)=O)C1 O=C(C1=CCC(NC(C2CC3CC3C2)=O)C1)NCc1ccc(F)cc1 N1(C(C(C)(C)Br)=O)CCC2C(CNC(=O)CC3NC(=O)NC3=O)C2C1 c1(CC(=O)NCC=CCNC(c2cccc3cncn23)=O)ccc2ccoc2c1 c1(C(=O)N)cc2c(s1)CCC(C)C2.c1(C(=O)NCCCC)cc(Cl)ccc1OC CC(C)C(CCNC(=O)CSC(F)(F)F)NC(c1n[nH]cc1C1CC1)=O C=CC(C)(CC)C(=O)NCCCOCCCNC(=O)CCN1CCC(F)C1 CC1=NOC(C)(C(=O)NCCC2CCN(C(C3CCCS3)=O)CC2)C1 C1(C(N2CC(O)(C(C)NC(CCSC)=O)C2)=O)CC2C=CC1CCC2 C1(NC(=O)CC23CCCC2C3)CCC(CNC(C2CC3C=CC2O3)=O)CC1 C(=O)(CC(C(F)F)n1cccn1)NCC1CN(C(Cc2cnc(C)[nH]2)=O)C1 N1(C(CCc2n(C)ncc2)=O)CCC(C)(C)C1CC(=O)NCCCc1ccco1 N1(c2c(C)cnc(C#N)n2)CCC2C(CCCN2C(c2cc(=O)cc(Cl)[nH]2)=O)C1 c1(C(=O)NC(CC=C)CNC(=O)C(=Cc2cnn(C)c2)C)ccc2cnoc2c1 c1(C(N2CC(C(C)NC(c3cc(O)no3)=O)OCC2)=O)c(O)nnc2c1CCC2 C1(NC(=O)C2CC2)CCN(C(=O)Cc2ccc(O)nc2)CC1O C1(CC)CN(C(=O)C(c2cnn(C)c2)=O)CCN1C(=O)C(CC)SC c1(OC)ccc(CC2CN(C(c3sccc3C)=O)C2)cc1 c1ccc([N+](=O)[O-])cc1.N1(C(CC=CC=C)=O)CC(NC(=O)CO)CC(C)C1 N1(C(Cc2c(C)n[nH]c2)=O)CCC(C)(C)C1C(=O)Nc1cccc(NC=O)c1 CCCC(CCC)=CCNC(C1CC1C(=O)N(c1ccc(Cl)cc1)CCC)=O CC(C)S(=O)(=O)C1CCN(c2cc(NCC3(N4CCOCC4)CCC3)ncn2)C1 c1(CC(=O)OCC(C)NCC2CCC(CC)CC2)ccc(OC)cc1Cl C=CCN=C(NCC1(C2=CCOCC2)CC1)N1CCC(c2cccnc2)C1 C1(CCNC(CCCC)=O)C(C)CCCN1C(=O)Cc1cc(C)cc(C)c1 c1(CCNC(C(N2CCC(c3cccc(N)c3)CC2)=O)=O)cc(Br)ccc1I c1(OCC(=O)NCC)cccc(CO)c1.C1(C=O)CC2CCC1C2.CC(F)F.N N1(C(c2c(CCC)nco2)=O)CCCC(C2CCN(C(=O)CCCOC)C2)C1 C1(N(CCCC)C(c2cc(OC)no2)=O)CCN(C(c2ccc(Cl)cc2)=O)CC1 C1(NC(c2cc(C(C)C)on2)=O)CCN(C(c2csnc2C2CC2)=O)CC1O CN1CC(C)(C)CC1C(=O)NCC1CCCCS1(=O)=O C1(NC(C(C)(C)c2cc[nH]n2)=O)CN(C(=O)CCn2ccnc2)C(C)(C)C1 CC(C)C(C)(CNC(C1(CO)CCCCC1)=O)NC(=O)C(O)C1CCCC1 C1(NC(c2cc(F)ccc2F)=O)CCN(C(=O)CCc2ncc[nH]2)C(C2CC2)C1 c1(OC)cc(C(N2CCOC(C(C)NC(=O)CCCCCSC)C2)=O)cc(F)n1 Cc1cc(C)c2sc(NC(=O)OCCC3CCCC(C)C3)nc2c1 C=CCC(C)(CC)C(=O)NCC1CC(NC(=O)C(O)CCc2ccccc2)C1 N1(C2CCN(C(C(=O)NCCOC)C3CC3)CC2)CC(C)CC(C)C1 Cc1cc(C(=O)NC2CC3(C2)CN(C(c2n[nH]cc2C2CCC2)=O)C3)cc(C)n1 C=CCC(CC(=O)N1CCCCCC1CCO)NC(=O)CC(=O)OC(C)(C)C C1(NC(c2cc(C(N)=O)[nH]n2)=O)C2CC3C1C3C2C(N1CCC2CC12)=O N1(C(CC2(C)N(C(C(CCC)F)=O)CC2)=O)CCC(O)CC1CC c1(OCC)cc(C=O)oc(=O)c1.C(C)(C)CO.C1(CC=O)C(C)C1(F)F c1(N2CCC(NC(C(C)NC(=O)NC)=O)(CF)C2)ccn2ccnc2n1 CCCCC(CC)CC(=O)N1CCN(C(=O)CCC(C)CC)CC1CO C1(C(=O)NCC(CCC)OCC)CCCCN1C(C1CC1C(=O)OC)=O C(C(CCN=c1[nH]c(=NCc2cc(Br)ccc2C)[nH]c2c1CSC2)OC)OC C(C(=O)NC1CN(c2ncco2)C1)(C(C)CC)N(C(CCN(CCC)C)=O)C C1(CNC(C(C)OC)=O)CC2(CC2)CN1C(c1ccncc1)=O.N(C)C.C C(=O)(CCC(C)C)NCC(C)(C)NC(C1CC(c2ccccc2)(CC)C1)=O S(=O)(=O)(c1ccc(NC2CC(CN(C)C)C2)c(F)c1)N1CCC(C)C1CO c1(CC)c(C(=O)NCCC2CCN(C(=O)CCn3cnnn3)C2)ccn1C c1(CC)noc(C)c1C(=O)NC1CN(C(=O)CSc2nncn2C)CC1F CCC(CC)C(C(=O)NCC(CNC(c1sccc1-n1cnnn1)=O)OC)OC N1(C(c2c(C)nc(-c3ccc(OC)cc3)s2)=O)CC2CCCCN2CC1C N1(C(c2c(CSC)scc2)=O)CCC(NC(=O)C2CC2)C(F)C1 C(=O)(C#CC(C)(C)O)N1CCC(C)C1C(N1CCC(C)(C#N)C1)=O n1(CC)cnnc1CCNC(=O)CCCNC(=O)C(O)C1CCCC1 N#CC12CC(C(N3CCCC3CC(=O)Nc3cccnc3C(F)F)=O)(C1)C2 N1(C(c2ccc(SC)cc2)=O)CC2CCC1(CNC(=O)C=CC1CC1)CC2 c1(C(N2CCCC2(C)C)=O)ccc(N)c(C)c1C.C1(C(=O)NC)(OC)CCSC1 c1(C(=O)NCC(C)NC(C(C(CC)(F)F)(C)C)=O)cc2c(nc1O)CCCC2O CCCC(C(=O)NCC1(Cl)CC1(F)F)NC(c1ccoc1Cl)=O [SH](=O)(=O)c1cc(C(N2CCN(C(=O)CC34CCCC3C4)CC(O)C2)=O)co1.CN CC1CC(NC(c2sccc2C2CC2)=O)CCN1C(c1ccc(N)cc1F)=O C(=O)(CCCC(F)(F)F)N1CCC(C(N2CCC(OC(C)=O)C2)=O)C1 C=CCC(C(=O)NCCc1cccnc1F)NC(=O)C=CC1CCCCC1 C1(C(=O)NC(C2CN(C(c3n[nH]cc3F)=O)CCO2)C)CCC(C)(O)CC1 c1(C(=O)NCC2(C)CCCN2C(=O)CCC2CCC2)cccc2nc(O)ccc12 c1(CC)ccc(C(=O)NCC2CN(C(c3cc(OC)ns3)=O)CCC2C)cc1Cl c1(C(N)=O)ccc(NC(C2CCCC2)=O)c(N(C)C)c1.C1(F)(C(=O)N)CC1 c1(C(=O)NC2CC(NC(=O)Cc3cnco3)C2)ccccc1C1CCC1 c1(NCC2OCC(CNC(C(C)(F)F)=O)C2)cccc(F)c1[N+](=O)[O-] CC1CCC(C)(C(=O)NCC=CC(=O)NCC2=CCCCC2)C1 c1(OC)cc(O)c(NC(=O)C(C)CCCc2ccccc2)cc1OC c1(CC(=O)NCC(CN(C(c2cc(C)sn2)=O)C)C)ccc(C)c([N+](=O)[O-])c1 C1(CNC(=O)C=C2CCC2)CCCC(NC(C2CCOCC2)=O)C1 C1(F)CCCC1.C1(C=O)CC2C=CC1O2.Cc1noc(COCC(=O)N)n1.C N1(C(C(CC)C)=O)CCN(C(=O)C(C)(C)COC)CC1CC(=O)NC CCCC(C)(C)CC(=O)N1CC(NC(c2noc(C)c2[N+](=O)[O-])=O)C(F)C1 C1(CNC(C2N(C(CC=C)=O)CC2)=O)CCCN(C(=O)C)C1.c1ccccc1.O N1(C(c2ccc(CC)o2)=O)CC=CCC1C(N1CC(C(=O)OC)(CC)C1)=O C1(C(=O)NCCCCSC)CCC2CCC1N2C(C1CCC1)=O C=CCC(CNC(=O)Cn1ccnc1C)C(=O)N1CCC1CC Cc1ccc2c(CC(=O)NCC3CCCC3NC(=O)C(CO)N(C)C)c[nH]c2c1 Cc1cc(O)c(C(=O)NC2CC(CCNC(c3cnncc3C)=O)C2)cc1Br N1(C(C2CCOC2)=O)CCC2=C(CCC(=O)N2)C1.CC(C)(C)OC=O.CC.N C1(O)(C(C)NC(=O)CCCn2cccn2)CCN(C(c2cnc(O)s2)=O)C1 C(CC(=O)NC1CCCOC1)(C(F)(F)F)NC(c1ccc(C(C)=O)o1)=O C(C(CC(=O)N(C1CCCC1O)C1CC1)C1CCC1)NC(=O)C=Cc1ccc[nH]1 N1(C(CC=C(C)C)=O)CCCC2(C1)CN(C(C1CC(C)OC1=O)=O)C2 C(=O)(C(C)CCC(C)(C)C)N1CCCN(C(c2c(C)ccc(OC)c2)=O)CC1 C1(NC(C2(CC)CCN(C(=O)Cn3nccc3C)C2)=O)C2CCCC1CC2 N1(C(CC(C)(F)F)=O)CC(C)(C)CCC1(C)C c1(SC(c2ccccc2)C(=O)NC(CCCCC)C)c(C)ccc2cccnc12 C(=O)(C(CC(C)(C)C)NC(=O)CC1CCC(=O)C1C)NCCCCCC(C)C Cc1cnoc1C(=O)N(CC(C)O)CCNC(C1(c2ccccc2)CCC1)=O n1(CC(=O)N)ccc(O)nc1=O.N1(C(C2C(C)C2C)=O)CCC(C(F)F)(C)C1 C12(CC(=O)NCc3n[nH]c(C)c3C)CCC1CN(C(=O)C(C)(F)c1ccon1)C2 c1(C(c2n(CC)nnn2)Nc2ccc(F)nc2)cc(C)c(F)c(C)c1 N1(C(Cc2nc(C)sc2Cl)=O)CCC(NC(=O)COCC2CCC2)C(O)C1 CC(C)CC(=O)NC1CN(C(c2ccn(-c3ccncc3)n2)=O)C1 c1(NC)ccc(CC(=O)N(C)CC2C(C(=O)NCCC#C)CCCC2)cc1 N1(C(C(CCC)(F)F)=O)Cc2[nH]nc(C(N3CCCC3C)=O)c2C1 N1(C(CCC2(C)CN(C(C3(CO)CCSC3)=O)C2)=O)CCn2c(O)nnc2C1 Cc1coc(C(N2CCC(C3CCCN3C(=O)Cc3ccccc3)CC2)=O)c1C C#Cc1cccc(C(=O)NC(C)CCNC(=O)CC(O)CCC)c1Cl N1(C(C2(C(C)C)CCC2)=O)Cc2ccccc2CC1CNC(c1cccnn1)=O N1(C(c2ccc(C#C)cc2F)C(=O)NCCCF)CCCc2ccsc2C1 C=CCC(CC)C(=O)N1CCCC1CNC(=O)COc1cc(C)ccc1Cl CC(C)CC(C(=O)N1CCOCC1)Nn1c(N2CCC2)nnc1SCS(C)(=O)=O C1(O)(C(=O)NCC23C(CN(C(CC(CC)(C)C)=O)C2)C3)CCCC(C)(C)CC1 Cc1cc(C(=O)N(C2CCN(C(c3[nH]c(O)nc3C)=O)C2)C)oc1Br C1(C(N(C2CCCN(C(C3CC(O)C3)=O)C2)CC)=O)C2CNC(=O)C12 c1(CNC(C=CC(C)NC(CCOCC#C)=O)=O)ccccc1C#C N1(C(Cn2c(C(=O)OC)cnc2)=O)CCC2(C1)CN(C(c1cscn1)=O)CCO2 C(=O)(C#CC1CC1)NCc1cc(C(=O)NC(c2cccs2)CC)on1 c1(C(N(C)CC2CCN(C(=O)C(c3cccn3C)=O)CC2)=O)cn2c(n1)CCC2 C1(CNC(c2c(CC)cco2)=O)C2CCC(C2)N1C(C1(C)CCOCC1)=O N1(C(CC2CCCC(C)C2)=O)CC(C2(N=c3[nH]nc(C(F)F)o3)CC2)C1 c1(C(N2C(C(=O)NC3(c4ccc(O)cc4)CC3)CCC2)=O)cccc2c1CCC2 c1(C(N2CC(NC(C3CCC3)=O)CC(C)C2)=O)ccc(C#N)c(Cl)c1 C1(O)(CNC(c2sccc2Cl)=O)CCN(C(c2ccc(CO)cn2)=O)CC1 c1(C(CNC(c2ccsc2)C)O)ccc(C#N)cc1 c1(C(=O)NCC2C(NC(C(CC(C)C)F)=O)C2)cc2cccc([N+](=O)[O-])c2[nH]1 C#Cc1cn(C)nc1C=O.C1CN(C(C2CCC(=O)N2C(C)C)=O)CC12CC2.N N1(C(c2c(C)cc(Br)o2)=O)C2CCC1(c1cn(C3CC(O)C3)nn1)CC2 CC1CN(C(C2(CO)CC2)=O)CC1CNC(c1ccc(NCCF)cn1)=O C=Cc1ccc(C(=O)NCc2ccsc2C(=O)NC2(C)CC=CCC2)cc1 C(=O)(C1CCCc2c[nH]nc21)NC1C(NC(Cc2c(C)ccc(Br)c2)=O)C1 N1(C(C(C)N2CCC2)=O)CCC(C(F)(F)F)C(NC(=O)C=Cc2cnccn2)C1 Cc1ccc2c(C(N3CCC(N(C)C(C4C5CC6C(C5=O)C46)=O)C3)=O)n[nH]c2c1 C1(c2nc(-c3cc(C)cc(F)c3)nn2CCC2CC2)CCCN(CP(C)(C)=O)C1 CC(CC(=O)NC1CCC(CNC(=O)Cn2cnccc2=O)C1)P(C)(C)=O N1(C(C(COC)COC)=O)CCCC12CCN(C(c1c(C)cc(C)cc1O)=O)C2 C1(CNC(C2C(C)C2)=O)CCC(CNC(C2(C)CCN(C)C2)=O)CC1 N1(C(c2n[nH]c(C)c2C)=O)CCC2(CC1)CN(C(=O)CC1CC1)CC(C)O2 C(=O)(CCCCC(=O)OC)NCCOCCOCCCNC(C(C=C)CC)=O N1(C(COC2CN(C(CC=CC=C)=O)C2)=O)CCSC2CCC12 C#Cc1ccc(C(N2CCCN(C(=O)Cc3cc(C4CC4)no3)CC2)=O)c(C)c1 Cc1ncccc1NC(=O)C(C)C(C)NC(C1(CC(C)C)CC1)=O c1(OC)ccc(C(C)=CC(N2CCN(C(c3occc3C)=O)CC2CO)=O)cc1 C1(NC(c2nc(CC)sc2)=O)CC2CCC1N2C(=O)CO.c1ccccc1C.C Cc1cc(C(=O)NCCCC2CCCCN2C(=O)C2CC2)ccc1Br C(CCCC(C)NC(=O)CCF)NC(C1N(C(CCC)=O)CSC1)=O c1(C(=O)N)ccc2c(c1)OCC(=O)N2.C1(NC(C(CC)O)=O)COC2(C)CC1C2 c1(OCC)cccnc1C(=O)NCC(O)CNC(=O)CCSC N1(C(CCc2c(OC)cccc2)=O)CCC(NC(C2(C(C)C)CCC2)=O)C(C)C1 c1(C(=O)NCC(C)N(C(CC(C)SC)=O)C)ccccc1N1CCCC1 c1(C=O)cccc2c1OCC2.Cc1c(C(=O)NCC2CCC2)noc1C1CC1.N CN1CCNC(=O)C12CCN(S(=O)(=O)c1cnccc1F)CC2 N1(C(COCCCN(C)C)=O)CC(CC(N2CCC(C)(CO)C2)=O)C2(CC2)C1 C1(C(N2CC(NC(CCCCC=CC)=O)(CO)C2)=O)CC2CCCCC2O1 N#CC1(C(=O)NCCc2cccc(Br)c2)CCc2ccccc2C1 c1(OC)cnccc1C(=O)NCCC1CCN(C(=O)C(C)CSC(F)(F)F)C1 C1(O)(CNC(C2CCO2)=O)CCN(C(c2cn(CCO)nn2)=O)C1 C1(C#N)(C(N(CCCCC(=O)NC(C(C)(C)OC)C)C)=O)CC2CC2C1 C1(NC(c2c(C)nco2)=O)CN(c2ccc(C#N)c(C)n2)C2CCCCC12 c1(OC)ccc(C)c(CN2CCOCC2C(=O)Nc2ccc(F)nc2F)c1 N12CC(C(F)C1)NC(=O)CCOCC(C)=CC2=O.C1(OC)CCCOC1 N1(C(CCc2cc(C)no2)=O)CC(CNC(c2ccc(Cl)cc2)=O)C2CC12 CC(F)(F)CC(=O)NCC1CC(O)(C)C1.c1(C=O)nnn(-c2ccccc2)n1 c1(CN2C(CCC)CCC2)ccc(=NCc2ccsc2)[nH]c1 C1(C(=O)NC(C)C(=O)N2C(C=O)CC2C)(COC)C=CCC1.C=O.O C1(CC(=O)N(C(CC#C)C)C)CN(C(=O)CSCCCC)CC12CC2 CC1CCC2(CCC2)CN1Cc1cccc(OC(F)F)c1 C#CCC(C)(CC)C(=O)NCC1CCN1C(=O)C(=O)NCC1CC1 NS(=O)(=O)c1ccsc1C(N1CCOCCC1)=O.C1(C=O)CC(C(F)(F)F)C1.N C(C(C(=O)NCCC(C)OC)NC(C1CC1C(N)=O)=O)OC CC(C)CC(C)C(=O)N1CCCC(F)(C(N2CC(N3CCNC3=O)C2)=O)C1 c1(CNCC(C)Oc2cccc(OC)c2)cccc([N+](=O)[O-])c1F N1(C(c2nc(CC)sc2)=O)CC(CNC(c2cnccc2Cl)=O)C(C)C1 c1ncccc1[N+](=O)[O-].c1(OC)nc(C(=O)NCC2(C)CCCC2)cc(O)n1.N c1(OC)ccc(F)cc1CC(=O)NCC#CCNC(C1(OC)CC1)=O C(CS(=O)(=O)N=c1nc(-c2ccccc2C(F)(F)F)[nH]s1)c1c(C)cccc1 C(=O)(CC(C(F)F)NC(c1cc(Cl)n(C)n1)=O)N1C(C)(COC)CCC1 c1(C(=O)NCc2ncc(C)cn2)cccc2c1CN(C(c1cc(C)[nH]n1)=O)CC2 c1(C(=O)NCC(C)N(C(=O)Cc2ccnn2C)C)ccc([N+](=O)[O-])o1 C12(NC(=NCC(=C)CC)NCC3CCOC3)CCC(C1)OC21CNC1 CCCC(CC)CCC(=O)NCC(CC(=O)N1CCC2CC12)C1CCC1 C1(NC(CN(C(COC)=O)C)=O)CCN(C(=O)C(CO)C(F)(F)F)CC(O)C1 Cc1ccc(C(N2CCN(C(C3CC3CC(C)C)=O)C(C3CC3)C2)=O)c(=O)n1C c1(OC)c(C)cc(CN2CC3CC(NC(C4CC4(C)C)=O)CC3C2)cc1C C1(CC(=O)NCCN2CCCCC2)CCC2(CCC2)CO1.C(=O)(C(F)C1CC1)N c1(C(=O)N)cc(Cl)cc(C)c1C.N1(C(c2nc(OC)oc2)=O)CC(CC)C(C)C1 c1cc(F)c(F)c(Cl)c1F.c1(OC)cc(NC(C2CC2C=O)=O)c(C)cn1.N C1(C(N)=O)(NC(NNC(C(CC)C)=O)=O)COc2ccccc2C1 c1(C(=O)NC2C(C)N(CCn3cccn3)CCC2)cccc2[nH]ncc12 C(=O)(CC1=CCN(C(c2cc(C)c(F)cn2)=O)CC1)NC(COC)COC N1(C(c2cc(C)[nH]c2)=O)CCCC2(CCN(C(=O)CC3(O)CCOCC3)CC2)C1 Cc1cc(F)sc1C(N1CC(CO)(NC(c2cc(-c3cccs3)[nH]n2)=O)C1)=O Cc1nc(C(=O)NC(C(O)CO)C2CC2)sc1C c1(OC(C)C)ccc(N)c(C(=O)NC(C2CCCC(C)C2)C)c1 c1(C(=O)NCC(CC)NC(C2(C)CC2(Cl)Cl)=O)cnn(CCCOC)c1 C1(NC(c2ncccn2)=O)(CNC(c2ccccc2SC(F)F)=O)CCCCC1 c1(CC)ccc(C(C)=CC(=O)N(CC(C)NC(C2CC23CCC3)=O)C)cc1 N1(C(C2CN(CC(C)C)C2)=O)CCCC(CO)(NC(=O)CCS(C)(=O)=O)C1 C#Cc1cccc(C(=O)NCC(C)NC(c2cnn(C3CC3)c2Cl)=O)c1 c1(C(N(C(C)C)Cc2cccs2)=O)cc2n(c1)CCC2 c1(CC=O)cc(F)ccc1F.C1(C(N(CCCO)C)=O)C2CCC(=O)C12.CC C1(OC)CCN(CC(N2CCC(C(C)(C)C(=O)NCCC3CCSC3)C2)=O)C1 C=CCC(C)C(=O)N1CCCCC1C1(NC(=O)O)CC1.OCP(C)(C)=O C1(CNC(C(C)N(CC)CC)=O)CN(C(=O)CCS)CCO1.CC(N)=O N1(C(C2CC2)=O)CCC(C2CC2)C1.c1(C(N(CC=O)C)=O)ccccc1.CO N1(C(C(F)=CC)=O)CC(OC)CC1CCNC(=O)C(c1ccccc1)C c1(OC)ccc(C(N2C3CCC2(C)CC3)=O)c(F)c1.C1(C=O)CC1(C)C(F)F N1(C(CC(C=C)CC)=O)CC2CC1CCC2NC(C1(C)C(C)(C)C1(C)C)=O Cc1ccc(C(=O)NCC2(C)CN(C(=O)C(F)C(F)(F)F)CC2C)nc1O C1(CCC)CCCN(C(=NCCC(C)=O)NCCOC)C1 C(=O)(C#CC1CCCC1)NCC1CCC(CNC(CSCC)=O)CC1 C1(CCC)CCC(CC(=O)NCCSCC)CC1.c1(C=O)ncc(C(F)F)s1 c1(OC)cc(C(N2CC(NC(c3cnco3)=O)CC(O)C2)=O)cnc1O c1(C(N(CCNC(C2CCC3(CCC3)OC2)=O)CC)=O)sc2nccnc2c1N C1(C=O)CCS(=O)(=O)N1.C1COCC1.c1(C(=O)NN2CCCC2)ccc[nH]1.N C1(CN(C(=O)CCC2CCC2)C)COC(=O)N1.C1(C)(CC=O)CCOC1.N N1(c2nc(Cl)nc(C)c2Cl)CC(C2CCCN(C(c3ccc(F)nc3)=O)C2)C1 C(C(=O)N1CCC(CNC(c2ccon2)=O)CC1)(C(C)C)N(CC)CC.C N1(C(C2CC(CF)C2)=O)CC2CC(C1)N(C(c1ccnc(Cl)c1O)=O)C2 c1(N2CCC(C=C)C2)cc(NCC2CCCCCC2)nc(C(C)C)n1 Cc1cn2c(n1)CCC(C(N1CC3C(NC(=O)COc4cccnc4)C3C1)=O)C2 N1(C(CC2C(C)(C)CCO2)=O)CC(NC(=O)COCP(C)(C)=O)CC12CCCC2 C#CCCC(O)C(=O)N(CC(C)(C)CNC(c1ccc(Cl)cc1NC)=O)C N1(C(c2cc(OC)ns2)=O)CCC2(CC1)CC(NC(c1csnc1Cl)=O)C2 C1(NC(C=CC=CC)=O)COC2(CCN(C(=O)C(C)(C3CC3)O)CC2)C1 c1(CC(N2CC(CC)C2)=O)ccc(C2CCC2)cc1.C(=O)(CCC1CCOC1)N c1(C(=O)NCC(C)N(C(c2nnc(C)s2)C)C)ccc2cnccc2c1 C1(NC(C(C)N(C(C)=O)C)=O)C2CN(C(=O)Cc3ccc(Br)nc3)CC12 c1(C(N(C2CCN(C(C(CC)F)=O)CC2)CCO)=O)cnc2sc(C)c(C)n12 N1(C(C2(C#C)CC2)=O)CCC(NC(C2C=CC=CC=C2)=O)C(CC)C1 N1(C(c2c(C)nn(CC)c2C)=O)CC2ON=C(C)C2C1.c1(C(=O)N)ccc(Cl)s1 c1(C(N(CCNC(=O)C(C)C2CCCO2)CC)=O)nc(C(C)(F)F)cs1 Cc1onc(C(=O)N)c1[N+](=O)[O-].C1(C)CCCN1C(C1CC1c1nc[nH]n1)=O.C Cc1cc(F)c(C(=O)NC2CN(C(=O)Cn3[nH]cnc3=N)C3(CCC3)C2)c(F)c1 c1(CCCC(=O)NCC(CNC(=O)C(C)C2CCC2)OC)ccc(O)cc1 c1(C(CC)C)ccccc1N1CC(C(=O)Oc2nccnc2SC)CC1=O c1(C(N2CC(NC(c3cc(C)sc3)=O)C(CO)C2)=O)ccc2c(c1)COC2 c1(C(N(C2CCN(CC#CC)CC2)CC2CC2)=O)oc2ccccc2c1C C1(C#N)(C(=O)NCCN(C(=O)C(C2CCCCC2)O)C)CC1(C)C c1(OC(C(=O)NC(c2cccc(C(C)C)c2)C)C)ccc2c(c1)CCC(=O)N2 CCC(N=c1ccnc(NC(c2ccc(C)cc2)CC)[nH]1)c1cccc(OC)n1 C(=O)(C(C1=CCCCCCC1)N1CCOCC1C(=O)OC)NCC Cc1nnc2n1CCC(C(=O)NCC1(O)CN(C(=O)COC3CCOC3)C1)C2 C1(CC(=O)NCCC(CC)CO)N(C(C2OCCC2(C)C)=O)CCC1(C)C C(=O)(C(O)C(C)(C)C)N(CCCN(C(c1[nH]cc(C(C)=O)c1C)=O)C)C n1(CC)cnc2c(NCC3CCC4CC34)[nH]c(=NCc3cc(C)cc(Cl)c3)nc12 c1(-n2cc(CNC(=O)NC(C(=O)OC)CF)nn2)cccc(C)c1 c1(C(=O)NCC(=O)NCC(C)C)ccc(CNC(=O)CC(Cl)Cl)nc1 C=CC(C)(O)C(=O)NCC1(F)CCC1.C1(c2cccnc2)(C=O)CCCCC1.N C(=O)(N=c1cc(C)n(CCC#N)[nH]1)Nc1ncc(CCC)s1 c1(OCC(=O)NC(C#C)CCC)c(C)occc1=O c1(C(N(C2CCC(NC(C3(CO)CC3)=O)C2)C)=O)ccccc1 Cc1cnc(O)cc1NC1CCN(C(=O)C(O)C(C)C)C1 C1(CNC(=O)Cc2ccco2)CCCN(C(c2cc(-c3ccco3)[nH]n2)=O)CC1 N#Cc1cc(NC(C2CCC3(CCC3)C2)=O)ccc1F c1(C(=O)NCC(C)NC(CCC=CC)=O)cn(C)nc1-c1ccccc1Cl N1(C(CCc2c(C)cccc2)=O)CC2CCCCC2(NC(=O)C(C)C#N)C1 C(CC(N=c1[nH]c2c(F)cc(Cl)cc2s1)C(C)C)NC(C(=CC1CCCC1)C)=O Cc1ccc2c(Cl)c(C(N3CCC(c4ccccc4)(CO)C3)=O)sc2c1 N1(Cc2cnc(C)o2)CCCC(C(C)NC(c2nocc2C)=O)C1 C1(C)(C(N2C(CNC(CCCCCN(C)C)=O)CCC2)=O)CCC(=O)N(C)C1 N1(C(CSCCOC)=O)CCCC2C1CCCN2C(c1ccc([N+](=O)[O-])n1C)=O C(=O)(CC(C)C(F)(F)F)NC(C1(C(N2CCCC(OCCC)C2)=O)CC1)C c1(CCC(N2C(CNC(c3n(CCC)ncc3)=O)CC2)=O)cccc(C)c1.O C1(F)(CNC(c2cc(C)ns2)=O)COCCN(C(=O)Cn2cccnc2=O)C1 c1(C(N2CCC(C(O)C(F)(F)F)CC2)C(=O)NCC)cn2cc(F)ccc2n1 C1(C=O)CN(S(N)(=O)=O)C1.C1(OC)CCCCC1C(=O)NC1CCCCC1.C C(=O)(C1CCc2ccccc21)NCC(C)CN(C)C(c1cc2c(o1)CCCC2)=O C1(C(C(=O)NCC(CC)NC(c2cnn(C)c2)=O)F)CCCCC1 CC(C)(C)CC(F)C(=O)NC1CCOC(C(=O)Nc2cnn(C(F)F)c2)C1 c1(C(N2CC3N(C(C(CCCOC)C)=O)C(CC3)C2)=O)cc2cccc(Cl)c2s1 N1(C(c2ccn(CCC)n2)=O)CC2C(CNC(=O)CC3CC(OC)C3)C2C1 N1(C(CNC(CC)=O)=O)CCN(C(=O)C(C)(C)NC(=O)C(F)(F)F)CC1.C Cn1cc([N+](=O)[O-])cc1C(=O)NC1CCCC1(C)CNC(=O)C#CC1CCOC1 c1(CNCC2N(C(c3cnc(OC)c(F)c3)=O)CCCC2)c(F)cc(O)cc1F c1(C(=O)NC2CCC(CNC(=O)CSCc3cscn3)C2)cncnc1C CP(C)(=O)CN1CC(C(=O)NC2(C)CC(NC(c3c[nH]ccc3=O)=O)C2)C1 C(=O)(C(C#N)C(C)(C)C)NC(CNC(C1(OCC)CCC1)=O)CO CCCCCC(CC)C(=O)NC1CCC12CN(C(c1cnc(C(C)=O)s1)=O)C2 CCCCC(C)C(=O)N1CC(O)(C(F)C(=O)NCc2ccoc2)C1 N1(C(c2c(C)nco2)=O)C(C(=O)N(C)CC2CC2C)CCC1C(C)C c1(C(N2CCC(NC(C(n3cc(Cl)cn3)C)=O)C2)=O)cnc2nc(O)ccc2c1 c1(C(N2CC(C(=O)Nc3c(C#N)nc(C)o3)C2)=O)ccc([Si](C)(C)C)cc1 N1(C(C(C)NC(=O)NC)=O)CCC(C)C1.c1(C=O)csc(C(C)(F)F)n1 N1(C(c2c(C)c(C#N)ccc2)=O)CCCC12CCN(C(=O)CC1CC1(Cl)Cl)C2 c1(C(N(CC(C)N(C(C(CC)O)=O)C)C)=O)csc(C)c1C C1(NC(C(CCOC)C)=O)CN(CC2CC(F)(F)C2)CCC1C c1(NC(C2C(NC(c3ccc(OC)nn3)=O)CCCC2)=O)c(Br)ccnc1C C(=O)(CCCCCF)NC12CC(NC(c3ccc(C(N)=O)s3)=O)(C1)C2 N1(C(C(CC)CC(F)F)=O)CCC(C2CCCN(C(=O)CCCCN(C)C)C2)C1 C1(NC(c2ccsc2)=O)COC2(CCCN(C(c3cc4cn[nH]c4cn3)=O)C2)C1 C#Cc1ccc(C(=O)NC(C(=O)NCCN(CC)C(C)C2CC2)C)cc1 Cc1ccc(OCC(N2CC(NC(c3ccc(F)cc3O)=O)C(O)C2)=O)cc1C C1(C)(CNC(C2CC(O)(CC#C)C2)=O)CCN(C(C2CSCN2C)=O)C1 c1(CC)cc(C(=O)NC2(CCNC(C3CC3C)=O)CCCC2)cn(C)c1=O Cc1cnc(CCNC(=O)NC(c2ncc[nH]2)c2cncs2)cn1 C(=O)(C(F)CC(C)(C)NC(c1ccc2[nH]ccc2c1)=O)N(C(C#C)C1CCC1)C N1(C(c2cc(C(N)=O)no2)C(=O)NC2(C)CC2)CCC(CN(C)C)CC1 c1(C(=O)NC(C)CN(C(=O)CC2CCNC2=O)C)cnc2c(c1)CCOC2 c1(C(=O)NC2C=CC(CNC(=O)CSc3ccccc3)C2)cnc2n1CCS2 O=C(C1=CSCCO1)N1CCC(Cn2cc(C3(O)CCCCC3)nn2)C1 c1(N2CCC(n3cc(Cn4ncc(C)c4)nn3)C2)ccc2c(c1)NC(=O)CO2 c1(C(C)OC)nc(C(=O)NCCc2ocnc2)co1.C(=O)C(F)C1CCC1.C N1(C(C(CN(C(=O)CCC(CF)CF)C)(C)C)=O)CCC2(CNC(=O)C2)C1 c12ccc(cc1)NC(=O)CO2.N1(C(COC)=O)CC(OC)C(C(F)F)C1 c1(C(CC(=O)NCCCCNC(Cc2c(C)nc[nH]2)=O)O)ccc(F)cc1 c1(C(N2CCCC(NC(CSc3ccc(C)cc3)=O)C2)=O)cccn(C)c1=O CC(C)CCCNC(=O)CC12CC(C1)C2.C1(C(=O)N)CSCN1C(C)=O C1(NC(c2c(SC)csc2)=O)CCCCN(C(=O)CC#N)CC1 C1(OC)CC(CNC(c2cnnn2C)=O)N(C(C2CC=CC(O)C2)=O)C1 C1(C(=O)NOCC(C)(C)C)(CC=C)CCN(C(c2[nH]nnc2CC)=O)C1 c1(C(=O)NC(C)CN(C(=O)CN2CCC2C)C)c[nH]c2cccc([N+](=O)[O-])c12 C1(C(=O)NC(c2ccnn2C)CC)CCN(C(C2(C)CCOCC2)=O)CC1O c1(C(N2CCC(c3ccccc3F)C2)=O)ccc(OCC2(CO)CC2)cc1F c1(C(=O)Nc2ccccc2)nnn2c1CN(C(=O)Cc1ccc(O)cn1)CC2 C(=O)(CC1=NN(C)C(=O)C1)N1C2CCC(CC)(C2)C1.Cc1cccc(C(=O)N)c1 C(C(C)(C)CC(=O)NC1(CO)CCCCC1C)NC(CC(C)(C)OC)=O C(=O)(C(C#N)C(C)C)N1CC(CC(=O)N(C2CC2(C)C)C)(OC)C1 c1(-c2onc(-c3c(C)c(Br)c(O)nc3)n2)cn2c(n1)C(=O)N(C)CC2 c1(C(=O)NCCCNC(C=C(C)c2ccco2)=O)ncn2c1CCCC2 CC(CS(C)=O)NC(=O)CCCNC(=O)Cc1ccsn1 C1(NC(COC(CC)C)=O)CC2CC1N(C(=O)Cc1csc(COC)n1)C2 Cc1cn(C)nc1C(N1CCC(c2cnn(C)c2)C1)=O.C1(C)(C=O)CC1(F)F.N c1(C(c2nnnn2CCC2CC2)NC2C(C)(C)C2)ccc2nccnc2c1 c1(C(N2CCC(O)(CNC(C3CC(O)C3)=O)C2)=O)cnc2cc(Br)ccn12 N1(C(C2N(C(C)(C)C)CC2)=O)CCCC(CO)(NC(C2CCOCC2)=O)C1 C1(NC(C(C)NC(C)=O)=O)(CO)CCCN(C(=O)N(C)C)C1.C1CCC1 N1(C(C(C=C=C)C)=O)CCC2(CCCN2C(c2cn3cccc(F)c3n2)=O)CC1 C1(NC(C(C)(C)OC)=O)CC2CCC1N(C(=O)Cn1ncc(Br)c1C)C2 c1(CC(=O)NCCCC(C)NC(c2c(C)c(Cl)cnc2)=O)ccc2c(c1)OCO2 C1(C(=O)NC(C2CCOC2)CNC(c2cccs2)=O)(COC)CC=CC1 C(=O)(CCC(C)NC(c1nocc1Cl)=O)N1CC(OC)C1 Cc1cc(C(N2CCCN(C(c3cncn3C)=O)C(CO)C2)=O)n2nccc2n1 C12(C(=O)NCC(C)N(C(=O)C=Cc3cnn(C)c3)C)CCC(=O)N1CCS2 C1(C(=O)NC(CN(C)C(c2ccccc2)=O)(C)C)CCCCC1O.C(C(N)=O)O N1(C(C2CC(C#N)C2)=O)CC2(CCC2)CC1CNC(c1cnco1)=O c1(C(N2CC(F)(CNC(CC3CCC(C)C3)=O)C2)=O)ncc(Br)cc1O C1(NC(C(=O)NCC)=O)CC12CCN(C(C13CCC(OC)C1CC3)=O)CC2 C1(NC(C2(C(=O)NC)CCC2)=O)COCC1.C1(CC=O)CC(C)(C)C1.N Cc1cnc2cc(C(N3CCOC(CNC(=O)C(C)C(F)(F)F)C3)=O)ccn12 C(=O)(C(O)(CC)c1ccccc1)NCC1CN(C(CC(=O)NCC)=O)C1.O CC(O)(CNC(=O)Cc1ccsc1Cl)CNC(C1CC1[N+](=O)[O-])=O C1(C(=O)NCC2(CNC(c3cc(Br)ccn3)=O)CC2)COCCOC1 c1(C(N(CCCNC(C2CCCCN2C)=O)CC)=O)csc2c1CCCC2 C(=O)(CC(F)(F)C(F)F)N(C)C.C(C(=O)N1CCC1)(C(F)(F)F)OC(C)=O CCC(C)(CC)C(=O)N1CCCC1CN(C)C(C1CCC(CSC)CC1)=O C(C)(CCCC(=O)N(C1CC(O)C1(C)C)C)NC(c1oc(CC)c(C)c1)=O C=CC1(CC(=O)NC2CCCCC2CC)CN(C(=O)C(C)(C)OCC)C1 C=CCCCCCC(=O)NC(C1(O)CN(C(C2(C)CC(F)(F)C2)=O)C1)C Cc1cc(OC(C)C(=O)NC(C)(C)CCNC(=O)CS(C)(=O)=O)ccc1Cl C(=O)(C(O)CC(F)(F)F)N1CCCC(NC(Cc2n[nH]c(=NC)s2)=O)C1 c1(C=O)ccc(F)c(O)c1F.c1(C(N(C(C)(C)C)CC)=O)cc(C2CC2)on1 CCCCC(O)C(C)C(=O)N(CCC(=O)N(CC(C)C(=O)NC)C)CC c1(C(=O)NC23CN(C(C4(C)CCCCO4)=O)C(CC2)C3)cc(Cl)cc([N+](=O)[O-])c1 C=CC1(C(=O)NCCC(Cl)Cl)CCN(C(=O)CC(C(=C)C)OCC)CC1 N1(C(c2cncc(NC(c3cc([N+](=O)[O-])cs3)=O)c2)=O)Cc2ccc(O)cc2C1 c1(OCCCC)ccc(C(=O)NNC(=O)CN(c2ccccc2)C)cc1OC c1(CC)ccc(OC)c(C(N2CCN(C(c3cccn3C)=O)C(C)C2)=O)c1 c1(C(N2CC(NC(c3ccccc3)=O)C(O)CC2)=O)cnn2c1OCCC2 Cc1cc(C(=O)NCC(C)NC(c2cnn(C)c2C(C)C)=O)cnn1 c1(CNC(C(CC)NC(C2CC2c2ccoc2)=O)=O)cc(C)sc1C c1(OC)ccc2occ(C(=O)NC3CCN(C(=O)C4=CSCS4)CC3)c2c1 C(N=c1[nH]cnc2ccsc12)C12OCC(CSc3c(C)cnn3C)(C1)C2 C(=O)(C1=C(F)CN(C(=O)C(c2ccnn2C)O)CC1)N1C(C=C)CCC1 N1(C(COCCOC)=O)CCOC2CCN(C(c3cc(F)cc(Cl)c3N)=O)CC12 Cc1ccc(C)c(C(=O)N)c1N.C12(C(N3CCC(O)C3)=O)CC(C)(CCO1)C2.C N1(C(C(C2CCCC2)OC)=O)CCN(C(C2(O)CCOCC2)=O)CC1CC1CC1 C=CC(C)(C)CC(=O)N1CCC(NC(=O)CN2CSCC2=O)C(C)C1 C1(C(=O)NCC(COC)OC)CCCCN(C(c2ncccc2O)=O)C1 C12(C=O)CCC(CC1)CC2.C1(C(=O)OC)CCCC1C(=O)N.CCC1CC1 N1(C(c2cc(C#N)cc(C)n2)=O)CCC2(CCN(C(C3CC(C)C3)=O)C2)C1 Cc1cc(Cl)ccc1NC(=O)CCC1CCCC1.c1(C(=O)N)cnc(C2CC2)o1 C1(C(N2CC(C)CC(CC)C2)=O)CC2CC1CN(C(=O)C(F)C1CCC1)C2 N1(C(c2c(C)nc(CC)o2)=O)CC(C)CCC1CNC(c1coc(Cl)c1)=O CCC(C(=O)N(CC(O)CNC(=O)C(F)(F)c1nccs1)C)n1cccn1 c1(N2CCCC(C(=O)Nc3c(OC)cccc3OC)C2=O)c(C)cc(Br)cc1C Cc1nn2c(c1C(N1CC3CCC3(NC(C3CCCOC3C)=O)C1)=O)CCCC2 c1(OC)ccc(C(=O)NC(C)C2CCC2)c(Cl)n1.c1(C=O)ccc(Cl)nc1O.N CCCC(C(=O)NCC(C)CNC(c1cc(C(C)=O)on1)=O)c1ccccc1 N1(C(CC)C(=O)N2CC(NC(c3conc3C3CCCO3)=O)C2)C(=O)CCC1=O N1(C(C(COC)(C)O)=O)CC2CC(NC(=O)CC3CCCC(C)C3)CC2C1 c1(CNC(CC2C(C)(C)CC2)=O)cccnc1C.c1(C=O)cc[nH]c(=N)c1.N C(C(C)(C)CC(=O)O)NC(C(Cc1ccc(OCC)cc1)C)=O C(C(=O)Nc1ccccc1O)(C(C)(C)O)NC(C=Cc1ccc(C)o1)=O N(C(=NCCN(c1ccc(F)cc1)C)NC1CCCCC1C)CC(=C)CC c1(CC)nccn1C.C1(N2C(=O)CN2C)CCN(Cc2ccc(C)[nH]2)C1 CC1CC(C(N2CCC(CC(N3CCCC3)=O)C2)=O)C1.C1(C)CCCC1 C(c1cc(F)c(F)c(F)c1)=CC=O.CC1(C(=O)NC2CCC2)CCNC1=O.N N1(C(c2n(C)c(Cl)cn2)=O)CC2CC1CCC2NC(C1CCc2nncn2C1)=O CCC(F)(F)C(=O)N1CCC(C(C)NC(=O)COc2ccon2)C1 CC1CN(C(C2CC23CC(C)(C)C3)=O)CCN1C(c1ccn(C2CCCC2)n1)=O O(NC(=O)C(C)(C)C=C)CC(=O)Nc1ccc(C#C)cc1 c1(C(N(CCNC(C(CCC)NC(C)=O)=O)CC)=O)c[nH]c2cccnc12 c1(OC)c(C(=O)NCCCCCCNC(=O)Cc2cc(C)[nH]n2)cnn1C c1(C(=O)NC2CN(C(C(CC=C)C)=O)CC2C(F)F)cc(Cl)cc([N+](=O)[O-])c1O O=S(=O)(c1cccnc1NCC(c1cccnc1)O)NC1CC(F)(F)C1 C(=O)(C(CCCC)C(C)C)N1C(C#C)CN(C(=O)CN2CCC(F)CC2)CC1 Cc1nc(C(N2CC(NC(C3CCCCN3C)=O)CC2(C)C)=O)ccc1Br C1(C(N2CCC(NC(C=CC=CCC)=O)CC2)=O)CC(C)(C)OC1(C)C.C C(=O)(C1=CC(O)C(NC(=O)Cn2ccnn2)C1)NC1C(C)(C)CC1 O=C(C1CC(O)c2ccccc21)Nc1cnc2n1CCC2 C(=O)(CC(C)(O)COC)N1CC(=C(CNC(C=C(CC)CC)=O)F)C1 C(=O)(C1=CCC2CCC1N2C(C1CCCC1)=O)NC1CN(C)CC1(F)F c1(N2CCC(CNC(CCCN(C)C)=O)C(F)(F)C2)ncnc2c(Br)c[nH]c12 C=CCC(C(=O)NC(C)CCSCC)NC(c1ccsc1OC)=O C12(CNC(Cc3cn(CC)nn3)=O)CCCC1N(C(c1ccc(C)cn1)=O)CC2 N1(C(CCCCSC)=O)CCN(C(c2cccc(N)c2F)=O)CCC1C CC(CC(=O)NCC=C1CCN(C(=O)OC(C)(C)C)CC1)C(F)(F)F CC1C(C)N(C(c2cc3cscc3s2)=O)CCN1C(=O)CCn1ncn(C)c1=O CC(C)C(CNC(=O)CN1CCSCC1)NC(=O)C(c1ccccc1)C1CC1 c1(-c2cn(CC3OCCN(C(CCCC4C(C)=C4)=O)C3)nn2)cc(C)nc(C)c1 C(=O)(CS(=O)(=O)C1CCCC1)NC1(C)CCC(NC(C2CCCC2(C)C)=O)CC1 C(CN=c1[nH]c2c(c(=NCC3CC3(Cl)Cl)[nH]1)COCC2)C1CCN(C)C1 Cc1cc(C(N2CCC(C(C)NC(=O)CNC(N)=O)C2)=O)c(O)c(C)n1 C=C(C)CCC(=O)NCCOCCN(C)C(c1cn(C(C)C)cn1)=O C(=O)(CS(=O)(=O)CCO)NC(C1CCN(C(C2CC3CC(=O)C2C3)=O)C1)C NS(=O)(=O)c1coc(C(=O)NC2CCC(C)C2)c1.C1(O)(CC=O)CCOC1 c1(OC)c(C)ccc(F)c1-c1ccc(CNC(c2cnccc2OC)=O)nc1 c1(C(=O)NCC(C2CC2)NC(C2(F)C(C)C2)=O)c(-n2cccn2)cccc1F C=CCC(CC(C)C)C(=O)NCCC1CC1.c1(C(=O)N)cc(C(C)=O)ccc1O c1(C(C)C)ccc(C(=O)N(C)CC)s1.c1(C=O)csc(C(C)(C)C)n1.CC.O c1(CNC(=NCCN(CC)CC)NCc2ccc(Cl)o2)ccc2c(c1)CCO2 C1(C(N(Cc2c(C)cccc2)Cc2ccccc2)=O)C2C3CC4C1C1C2CC3C41 N1(C(CCCCOCC)=O)CCN(C(=O)CCc2nc(C)no2)CC(C)(C)C1 CCCCCC(CC)C(=O)NC1(CN(C)C(C2CCOC(C)(C)C2)=O)CC1 c1ccc([N+](=O)[O-])cc1.C1(C(C)NC(=O)C(C)(C)N)CCCN(C(=O)CCF)C1 n1(CCC(=O)OCc2ccc3c(Cl)csc3c2)c(=O)oc2cc([N+](=O)[O-])ccc12 c1(CNC(COCCOCC)=O)nc(C)cs1.c1(CC=O)nc[nH]n1 c1(C(N2CC=CC(NC(c3ccc(C(F)(F)F)s3)=O)C2)=O)n[nH]c2c1CCSC2 c1(C(=O)NCC2CCCC2)ccc2nc[nH]c2c1.c1(C(=O)N)cn2c(n1)SCC2 c1(C(=O)NCC(C)NC(c2csnc2Cl)=O)ccc(NS(C)(=O)=O)nc1 c1(N2C(C(=O)Nc3ccc(O)nc3)CNCC2)ncnc2c1oc1ccccc21 C(CCOC)(C=O)NC(c1n(CC#C)ccc1)=O.C(CN(C)C)CC(C)C.N CC(C)C(O)CC(=O)NCCC1CCN(C(=O)CCCOC(C)(C)C)C1 C1(OC)CN(C(c2ccccc2Cl)=O)CCC1NC(C1CC(C2CC2)C1)=O N1(C(CSc2nc(C)[nH]n2)=O)CCN(C(=O)C=C2CCOCC2)C2CCCC12 C(=O)(C(F)C1=CCCCC1)N1CC(O)(CCNC(C2N(C(C)C)CCC2)=O)C1 c1(C(N(CCC(C)NC(C=CC(C)C)=O)C)=O)cc2c(s1)CCOC2 c1(C=O)sc(-c2ncc[nH]2)nc1C.C1(NC(C=C(COC)C)=O)CC(C)C1.N Cc1ccccc1CCC(=O)NCCN(C)C(C1CC1c1ccc(F)cc1)=O C1(CNC(CC2(OC)CCC2)=O)CC(C)(C)CN1C(C1CCC12CCC2)=O CC(C)CC(C)CC(=O)N1CCCC1(C)CNC(c1cn(C)nc1C(C)(C)C)=O Cc1oc(S(C)(=O)=O)cc1C(=O)NCCOCC1(O)CCN(C)CC1 c1(CC(N2C(C)CC(NC(C3(C(C)C)CCC3)=O)C2)=O)cc(F)ccc1O CC(C(=O)NCCCOCCC(=O)NC1CC(CC2CC2)C1)n1cccn1 C1(NC(C(COC)C)=O)CCS(=O)(=O)C12CN(C(c1ccc(Cl)cn1)=O)C2 Cc1cc(C(N2C(C(=O)NC(C)(C)C)CC2C)=O)cn1C N1(CCCCCCC)CCC2(CCCN(C(C3CCC(=O)N3C)=O)C2)C1 C1(C=O)CC(=O)N(c2cn[nH]c2)C1.CC(C(F)F)=CC(=O)N(C)CC1CC1 N1(C(c2ccc(C(C)=O)c(F)c2)=O)CC2(CCCN(C(=O)C(F)CC3CC3)C2)C1 N1(C(=O)CC2OCCO2)CC(C(=O)O)C2(C1)CN(C(c1cc3sccc3s1)=O)C2 CC1CCC=C1C(=O)NCC1CCC(C(=O)Nc2cscc2C2CC2)O1 c1(OC)ccc(C)cc1C(=O)NC1CCC(C)C1 N1(CC(N2CC(O)(CC)C2)=O)CCOCC1=O.C(CC1CCC1)(C(=O)N)OC Cc1nccnc1C(N1CCC(C(C)C(N(C)C[Si](C)(C)C)=O)C1)=O c1(C(=O)NC2C(OC)CN(C(c3cnc(C)[nH]3)=O)C2)nn(C)c(C)c1Br N#Cc1cccc(C(N2CCOCC(NC(c3cscc3Br)=O)C2)=O)c1F Cc1cc(F)c2c(c1)CCN(c1cc[nH]c(=NCCCCN3CCCC3)n1)C2 Cc1ccc(C(=O)NCC23CCC(CC2)N3C(=O)C(C)n2cccc2)cc1F N1(C(COCc2onc(C)n2)=O)CC(NC(=O)CC)C2(CCC2)C1.C(N)=O C1CN(C(C2C3CC4C(C3)C24)=O)CC(C)(C)O1.CC1CCCN1CC(=O)NC n1(CCC)ccc2ccc(C(=O)NCc3cnn(CC(F)(F)F)n3)cc12 CC1CN(C(=O)CCc2cscn2)CC1NC(c1ccn(C2CC2)n1)=O C(=O)(CCCCC(C)=O)NC(CC(=C)C)C(=O)NCc1cccc(F)c1O N(C1CCCn2nccc21)C(C(CC=C)NC(c1cn(C)c(=O)n1C)=O)=O C=C1CN2C(=O)CCC2(C(N2CC3CC3(NC(=O)Cn3cc(Cl)cn3)C2)=O)C1 C1CC(C2CC2)C1.C1(C=O)(CNC(c2ocnc2C2CC2)=O)CCCO1.N c1(C(C(=O)NC(C)C)N(C(CCC)C#N)C)cc(C)sc1C C1(OC)CN(C(C2CC3CC3N2C(C2(C)CCN(C)C2)=O)=O)CC1OC CC1(C)CN(C(=O)C=Cc2cncs2)CCC1C(=O)NCC(F)C1CCC1 CCC(C)(O)C(=O)NCCC(C)(C)NC(C1CC(=O)N(c2nccs2)C1)=O CCC(CC)CCNC(C1CC1OC(C)=O)=O.C1(C=O)CCC2CC2CC1.N c1(-c2ncc(C(=O)Nc3ccsc3C(F)(F)F)s2)ccccc1F c1(C(=O)OC)cccnc1N1CCC(C(C)NC(c2occc2C)=O)C1 C1(C)(C(N2CC(C=C)(O)C2)=O)CC(O)CN1C(c1cnc(CC)nc1)=O CCC(CCC(=O)NCC1(CC(=O)Nc2ccc(Cl)c(O)c2)CC1)OC c1(C(=O)NC(CNC(c2cnn(C)c2C2CC2)=O)CO)coc2c(Cl)cccc12 C(CC(O)CC(=O)N1CCN(C(=O)C2=CC(C)(C)C2)C(C(C)C)C1)SC C1(C(N2CCC(OCC(=O)NC(c3nccs3)C)C2)=O)(CC)CCCCC1 N1(C2CCN(C(C3(CC)COC3)=O)C2)CCN(C(C2(COC)CC2)=O)CC1 CS(C)(=O)=NCC(=O)N1CCC2(NC(=O)CNC(=O)N)CC2C1.C1CC1 CC1(C)CC(C(N2CCCC(O)(C)C2)=O)CC(C)(C)C1.C1(Cl)(C=O)CC1(C)C NS(=O)(=O)c1cc(C(=O)NC(CNC(C2CCC(F)(F)CC2)=O)CO)co1 C1(CCC)(NC(C2(C3CCCCO3)CC2)=O)CCCN(C(c2ccncc2)=O)C1 c1(C(CC(=O)NC2CCC2)NC(C)=O)ccc(Cl)cc1.C(=O)C(F)C1CC1.N c1cccc(OC)c1Cl.c1(C(c2n(CCSCC)nnn2)N)ccnc(Cl)c1 C(CC(C)C)(C(=O)N1CC(CNC(=O)CCc2cc[nH]n2)C(O)C1)OC C1(OC)CN(C(=O)C(c2ccoc2)NC(c2ccc(C)[nH]2)=O)CC1(C)C c1(C(N2CCC(S(C)(=O)=O)CC2)C(=O)NCC)cnc2ccc(Cl)cn12 CC1OCCC1(C)C(=O)NCC1(F)CC(NC(c2c[nH]cc2Br)=O)C1 c1(CNC(C2C=CCN(C(C(c3cccnc3)OC)=O)C2)=O)ncc(C)cc1C C1(CNC(COC)=O)COC(C(F)(F)F)CN1C(c1cc(C)n(C)c1)=O c1(C(=O)Nc2c(C(=O)OCC)c(C)c(Cl)cn2)ccn2cc(C)nc2c1 CCCCC(CC)CC(=O)NC1CC2CC(NC(=O)CS(=O)(=O)C3CC3)C1C2 CC#CCC(C(=O)NC(c1cncn1C)CO)NC(C1CC12CCCCC2)=O c1(-n2ncc(C(N3CC(NC(=O)Cn4cnc(Br)c4)C3)=O)c2)ccc(F)cc1 c1(CCC(=O)NC(CN(C(c2ccn(C(C)C)n2)=O)C)(C)C)ccccc1O C(=O)(C(C)(C)C(C)NC(c1occc1CC)=O)NCCOCC#C c1(C(N2C(C)CC(CNC(C34CC3C4)=O)C2)=O)cccc(Cl)c1Cl c1(OC)c(C(=O)NCC2CCCC2NC(=O)C(N)=O)ccnc1Cl c1(OC)cc(NCC(C2CC2)N(C(=O)CS(N)(=O)=O)C)c(Cl)cc1[N+](=O)[O-] c1(C(N2CCC(CNC(c3cc(C)ncn3)=O)C2)=O)cc2oc(Cl)cc2[nH]1 c1(C(=O)NCCN(C)C(C2CC(=O)N(C3CC3)C2)=O)cnn2ccn(C)c12 N1(C(N(C)C)=O)CC(C(=O)N(C)CC2CC2)C1.C(=O)C(F)C1CCCC1.N CCC(C)CCCCC(=O)N1CC(CNC(c2nc(C)nn2C)=O)CC(C)C1 c1(C(N2C(CCNC(C3CC3C3CC3)=O)CCC2)=O)cccn2cnnc12 c1(C(N2CCN(C(C3(CCCC)CCC3)=O)CC2)=O)nc(C)c(C)nc1O c1(C(=O)N)ccccn1.C1(C(N(C(C)C)CC)=O)CC(OC)C1.C(C)=O C(=O)(C(O)CC(F)(F)F)NC(CC(=C)Cl)C(=O)NC12CC1COC2(C)C C1(NC(CCOC)=O)CC(NC(c2cncc(F)c2Cl)=O)C12CCOCC2 n1(CC)nc(C(N2C(C(=O)NOC3CCOCC3)CCC2C(C)C)=O)cc1O C1(O)(CC)CCN(C(=O)CN(C(=O)C)C)CC1.c1(CC)cc(C=O)on1.N Cc1nc2sccn2c1C(=O)NCCNC(=O)CCC=O.c1nnc(C(C)C)s1 Cc1nc(C(=O)NC(C2CC(NC(=O)COCCCC(C)C)C2)C)sc1C C1CN(C(=O)Cc2cccs2)CCCO1.Cn1cc(C(=O)NC)c(C(C)(F)F)n1 Cc1cnccc1C(=O)NCC1CCCC1NC(=O)CCC1CC1C C1(N(C(c2cc(OC)nn2C)=O)C)CN(C(=O)CO)CC12CC2.c1ccccn1 Cn1nc(C(=O)NCCC2CCC(NC(=O)COC(F)F)C2)cc1C1CC1 c1(C(=O)NC2C(NC(=O)CN3C(=O)CCC3=O)C2)c(F)cc(Cl)cc1Br C#Cc1ccccc1CC(=O)NCC1(F)CN(C(=O)C(O)CC(F)F)C1 N1(CC#C)CCOCC1C(=O)N(CCC)Cc1ccccc1OC Cc1cc(Br)ccc1C(=O)N(C(C)C1CC1)C.c1(C(=O)N)cnnn1C1CC1 Cc1cccc2c1OC(C(N1CC(CNC(C3CC=CCO3)=O)CC1C)=O)C2 c1(C=O)cc(Cl)c(N)cc1F.C1(C(N(C(C)C2CC2)C)=O)CCC(C)(C)O1.N C12(C(N3CCC(NC(C=CCC)=O)C3c3ccccc3)=O)COCC(C1)OC2 N1(C(C(C)=CCC)=O)CCC(CCC(N2CC(CO)C(CCC)C2)=O)CC1 c1(C(N2C(C(C)NC(=O)C(C)n3cccc3)CCC2)=O)ccn2nccc2n1 CCCCCC(C)(CC)C(=O)NCC(C1CC1)NC(C1(CO)CCC1)=O C(=O)(CC(C)(C)C(=O)N(C)C)N(CC(C)NC(C1COCCC1(F)F)=O)C N1(C(CC#N)=O)CCC2C(CCN2Cc2ccc(O)cc2O)C1 Cc1cc(C(=O)NCCC2CC2)c(-n2cccc2)s1.C(=O)C(F)CC1CCC1 C1CCCCC1.c1(C=O)c(C)ncn1C.C1(C)(C(=O)OC)CC(C(=O)N)C1.C C(N=c1nc(C(F)(F)F)[nH]s1)C1CC(C)N(C(c2cn(CC(N)=O)nn2)=O)C1 C12(CNC(c3c(C)n[nH]c3)=O)CCCC1N(C(=O)Cc1nnc(S)n1C)CCC2 C12(C(=O)NC3CCN(C(c4cc(C#N)[nH]c4)=O)CC3O)CC3CC1(CO)CC3C2 C1(F)(C(=O)OC)CN(C(=O)CCC2(NC(C3CCCS3)=O)CCCC2)C1 C(=O)(CCCCC(C)C)NC1CN(C(CNC(CCC)=O)=O)CC12CC2 n1(CC(CC)O)cc(COCCCCCNC(C2(CO)CC2)=O)nn1 Cc1cc(I)ccc1C(N1CC(F)(F)CC1C(=O)Nc1cc(Br)cc(Br)c1)=O N1(C(C=C(C)C)=O)CC2CCCC(CNC(=O)CC3CC3(Cl)Cl)C2C1 N1(C(C2(C)CN(C(c3ccc(OC(C)C)cn3)=O)C2)=O)CCC(C)(C)C(O)C1 c1(C(N2CC(N(C(C3CCC(C)C3)=O)C)C2)=O)c[nH]c2nccc-2c1 C1C2CN(C(C3C(C)(C)C3(C)C)=O)CC12.c1(C(C)(C)C(=O)N)ccccc1Cl.C C1(CC=O)CCC(=O)NC1=O.CC1CCCN1C(c1cnn(C(C)(C)C)c1)=O.N Cc1nnc2n1CCCC2C(=O)N1CCC2(NC(c3ccnn3C)=O)CCCC12 C(CCC(C(=O)NCC(F)(F)C(C)C)NC(c1ccc(=N)[nH]n1)=O)OC C1(NC(COCC)=O)CCN(Cc2ccc(O)c(Cl)c2)CC1F C1(C(=O)NC(C(=O)NCCOC(F)F)c2ccco2)CCC1(F)F c1(COC)ccc(C(N2CC3CC3C2)=O)cc1.c1(C2C(C=O)C2)ccncc1.N CN(S(N)(=O)=O)CC(=O)NC1CC(C)C1.c1(C=O)cc(C2CCOCC2)on1 c1(-c2nc(CN(C(c3cccc(Cl)c3)C(C)C)C)sc2)ccc(S(C)(=O)=O)cc1 c1(C(N(C(C)C)CCN(C)C)=O)ccc2c(n1)CN(C(=O)CC(C)(F)F)CC2 Cc1ccc2oc(C(N3CCC4(C3)CN(C(=O)CC(C)C(F)(F)F)C4)=O)cc2c1 C1(C(=O)NCC(C(C)C)NC(c2cn(C)c(=O)cn2)=O)CC2CCC(C1)N2C C1(N2C(C(=O)OC)CCCC2)C2CCC1CN(C(c1cnn(C)c1)=O)C2 N1(C(c2nc(C)c(C)o2)C(=O)NCc2ccco2)CC(C)C12CCOCC2 C1(C(N2CC(NC(C3C(C)C3C)=O)(CO)C2)=O)CCc2nnn(C)c2C1 c1(C(N2CC(n3cc(C(C)O)nn3)C(C)C2)=O)c(C#N)ncn1C C1(CN(C(C(=O)NCCCC)C)C)CCCN1C(c1ccsc1C)=O Cc1noc(C)c1-n1nc(C2CCC(C)CC2)nc1-c1cc[nH]c1 Cc1cc(Cl)cc(C(=O)NCC(O)CN(C)C(C2CC(C3CCC3)C2)=O)c1N c1(NC(C2CCCC(NC(c3ccc(O)cc3F)=O)C2)=O)cccc(Cl)c1F c1(C(N(C2CCCC2)C)=O)cc2n(n1)CC1(CC1)C2.C(CC(=O)N)SCCCC c1(CN2CCN(C3CCN(CCC(=O)OC)C3=O)CC2)ccc([Si](C)(C)C)s1 C#CCCC(=O)NC1(C(N2CCC2c2ccccc2)=O)CCC1 C(CCCC(C)(C)C(=O)NNC(=O)c1cccc(OC)n1)NC(C1C(=C)CC1)=O c1(CC(=O)N)c(F)cccc1F.c1(CC)cccc(C(N2CC3C(C)C3C2)=O)c1 C(=O)(CS(=O)(=O)C(C)C)N1CC(CNC(c2occ(C)c2)=O)C(O)C1 Cc1cc(C#N)nc(NC2CS(=O)(=O)CC2NC(=O)C(C)(F)C(C)(C)F)n1 CCCCC(C(=O)N(c1cccc(O)c1)C)NC(=O)CC1CC2CC2C1 CC1(C)CN(C(C2CCC(N)C2)=O)CCN1Cc1cc[nH]c(=N)c1 C(=O)(CC(C)(O)CCC)NC1(CCNC(C2C(=C)CC2)=O)CCCC1 Cc1csc(C(=O)NC2CC2CNC(c2cc(F)c[nH]2)=O)c1Cl n1(CC(=O)NCCN(C(C2C(CC)C2)=O)C)c(=O)cc(C)c2ccccc12 Cc1nc(O)nc(O)c1CC(=O)NC.C1CCN(C(C2(n3ccnn3)CC2)=O)C1 Cc1c(C(=O)NCC(CC(=O)NCC2C3COCC23)C2CCC2)[nH]ccc1=O c1(COC(C)=O)ccc(-c2ccc(C(N3CCCCC3CCO)=O)nn2)cc1 CC(C(=O)NC1CCN(C(C2CSC2)=O)CC1C(N)=O)C(C)(C)C c1(CC(N2CCC(NC(=O)CCSC(F)(F)F)C(F)C2)=O)cnc2cccnn12 N1(C(C(C)C#N)=O)CCC(C2CC2)C1CNC(c1cnc(Cl)c(Cl)c1)=O C1(c2cc(CNC(C(C)=C3CCCC3)=O)on2)CCN(C(C2CC2C#N)=O)CC1 c1(C(=O)NC(c2ccc(CO)cc2)C)ccnc(-c2cncc(F)c2)c1 c1(C(N(C2CN(C(c3ccc[nH]3)=O)C2)C)=O)ccc2c(c1)CCC(C)N2.COC C1(C(N(C)CC2OCCN(C(c3cc(OC)ncc3)=O)C2)=O)CCCCN1N=O N1(C(c2ccco2)=O)CCN(C(c2cncc(C(F)F)c2)=O)C(CCO)C1 C1(C(N2CC(F)(C(=O)NCc3c(OC)cncc3)C2)=O)CNC(=O)CC1C C(=O)(C(C)(C)CC)NCc1onc(CC)n1.C(=O)(CN(C1CCC1)C)N C1(C(=O)NCC2N(C(C(COC)OC)=O)CC(OC)C2)CN(C)CC(C)O1 CCCCC(C)C(=O)N(C1CCN(C(=O)CS(=O)(=O)NC(C)(C)C)CC1)CCC c1(C(=O)NC2CC(C(N(CC)Cc3cccnc3)=O)C2)c(C)ccn1C N1(C(C2N(CCC)CCC2)=O)CC(C)CC(C)(C)C1.c1(C(=O)N)ccc(C)n1C c1(OC)n[nH]c(NC(=O)CC2CN(C(C3CC=CCC3)=O)C2)c1C#N n1(CC=O)nc2n(c1=O)CCCC2.N1(C(C(C)OCC)=O)CCSCC1CC.N C(CC(N)=O)(C(=O)NCC1CC=CC1)NC(CC1CC(OC)C1)=O N1(C(C(CC=CC)C)=O)CCC2(CC2C(N2CC(O)(c3cc[nH]n3)C2)=O)C1 C1(C)(C(=O)OCC)CN(C(=O)CSc2nnsc2N)C1 C(=O)(C#CC1CCCO1)NCC1CC(NC(C(CCOC)C)=O)C1 N1(C(C=CC=CC)=O)CCC2CCN(C(=O)CC3CCC(=O)C3)CC2C1 N(C1c2ccccc2CCC1OC)C(c1cc(OC)cc(CC)c1)=O C1(CNC(CN(CC(C)(C)C)C)=O)(CO)CCCN1C(=O)C1=C(Cl)CC1 C1CCCN2C(C)C(=O)NC(=O)C(C(=O)C2)CCO1.C(C)(C)(C)OC C#CCC(CC#C)C(=O)NC(CNC(=O)CC1CCCN1CC)C(C)(C)C C(=O)(C(C(C)(C)C)c1ccccc1)N1CCN(CC(C)NC(=O)C2=CCC2)CC1 C(=O)(CCCCn1ccnn1)NC1C(Cn2cc(-c3c(C)nsc3)nn2)CCC1 C=C(Cl)CCC(=O)NC(C1CCN(C(c2oc(CC3CC3)nc2C)=O)C1)(C)C N1(C(C=C(C)C)=O)CCC2(CC1)CN(C(c1cnn(C3CC3)c1)=O)CC2CO c1(C(N2CC3C(NC(=O)CC4CCC4)(C3)C2)=O)ccc(F)c2cnccc12 CN=c1[nH]c(=NCc2n[nH]c(C)c2C)[nH]c(=NCC(CO)OC)[nH]1 C1(CCOC)(C(=O)NC2CC(C)N(C(C3CC(O)C3)=O)C2)SCCCS1 C=C(C)C(CC(=O)NCc1cc[nH]c1C(=O)NC(c1ccncc1F)C)O.C C1(NC(CCCCOC)=O)C2CC3CN(C(c4cnc(C5CCC5)s4)=O)C1C3C2 c1(C=O)ccc(O)c(Cl)n1.C1(CC(=O)N(C(C)C2CC2)C)CC(C)(C)CO1 c1(CCC2CN(C(CCSC)=O)C2)ccccc1-n1cc(CCOCCO)nn1 C1(NC(c2coc(C3CC3)n2)=O)CN(C(c2cnc(C3CCC3)s2)=O)CC1O c1(OC)cccc2cc(C(=O)NC(C)C(CO)NC(c3ccc(CO)o3)=O)oc12 C1(CNC(C2(C)CCOC2)=O)CCCC2(CCN(C(=O)Cc3cc[nH]c3)CC2)O1 c1(C(C=O)O)cc(F)cc(F)c1.n1(CC)cc(Cl)cc1C=O.C(C)C1CC1.N CC(C)(F)C(=O)NCCC1CCN(C(C2OCCC2Cn2ccnc2)=O)C1 C1(NC(CNC(Cc2c(C)nn(C)c2)=O)=O)CCCN(O)C1=O N1(C(c2c(CC#N)ccs2)=O)CCCC(NC(c2ccc(Cl)o2)=O)CC1 n1(CC(N2CCC2)=O)ccc([N+](=O)[O-])n1.c1(C(=O)N)cc(C2CC2)ns1.C C(=O)(C1=CCCS1)N1CC(CN(C(=O)CC(c2cccc(F)c2)O)C)C1 C1(CCC(N2C(CNC(C(C)(C)F)=O)C(C)(C)CC2)=O)CCC(C2OCCO2)O1 C1(NC(C2(CCC)CC2)=O)CCCC(C(=O)NCc2cc(=O)cc[nH]2)CC1 c1(C(=O)NC(CC(C)NC(c2cc(C)sn2)=O)C)ccsc1C#N C=CCC(CC(C)C)C(=O)N1CC(O)CC1CNC(=O)C(O)Cc1ccccc1 C(=O)(C(C)CC(F)(F)F)N1CCN(C(C(C)=C(CC)C)=O)CC1CC(F)F C1(CC)COC(C)CN1C(C1(F)CCN(C(=O)C=C(C)C2CC2)CC1)=O C1(NC(C(COC)N(C)C)=O)CCCN(C(C2(CF)COC2)=O)CC1 C(=O)(CCCC(C)C)N1C(C)(CNC(C(CC)OC2CCCCC2)=O)CCC1 C1(C(N(C)CCOC)=O)CCC2(CC2)N1C(C1(C#N)CC1)=O.C1CC1 c1(C(=O)NC2CN(C(C(COC)COC)=O)C2)cc(I)ccc1C C1(CCCCNC(C(CC)N(C)C)=O)CCN(C(c2nc(OC)c(C)s2)=O)CC1 N#Cc1ccc2c(c1)CCN(C(=O)CC1CCCN1C(c1ccc(F)cn1)=O)C2 C1(C)(C(N(CCN(C)C)CCO)=O)CC(O)CN1C(=O)C1=CC(C)(C)C1 N1(C(C(NC(C)=O)=Cc2cccs2)=O)CC(NC(=O)C#CC(C)C)CCC1C Cc1nc(O)ccc1C(=O)NCCCC1CCCN1C(C1CCCS(=O)(=O)C1)=O N1(C(CC(C(C)=O)(C)C)=O)CCC(CNC(=O)CCOCC(C)C)C12CCC2 CC(C)C(O)C(=O)NC1COCCC1NC(=O)Cc1ccc(Cl)cn1 c1(C(=O)NCCCN(CC(C)C)C)c(C)cnn1C.N1(CC=O)CCCC1.N c1(NCC(CC)OC)cc(C)c(S(=O)(=O)NC(C)Cc2cccnc2)cn1 C12(NC(c3scc(C#N)c3)=O)CCN(C(=O)COc3ccc(F)cc3F)CC1C2 c1(N(C)C)ccc(C(=O)NC)cc1.C1(O)CCN(C(=O)C=CC2CCOCC2)C1 c1(C(=O)NCc2cccc(NC(COCC)=O)c2)cc2cccc(Br)c2o1 C1(NC(c2cc(C)cc(C)n2)=O)CCCC12CN(C(=O)Cc1cnc[nH]1)C2 CC1CN(C(c2ccccc2N(C)C)=O)CC1CC.C1(C)(C=O)CC(C#N)C1.N C1(C(N(CCC(N2CC3(CSC3)C2)=O)C)=O)CCCC2(CC2)C1 C(=O)(C1=CCCN(C(C2CCCOC2)=O)C1)NCCn1c(C)cc(C)n1 C1(CNC(COC)=O)CC(O)CN1C(C1CCC1(F)F)=O c1(N(C(C(c2ccccc2)OC)=O)C2CC(N)C2)ncnc(C(F)(F)F)c1Br C1(C(=O)NCCN(C(C2CCN(C)CC2)=O)CC)CC2(C1)CC1(CC1)C2 CC(C)(CC1CC1)C(=O)NC(C1CCCC1)C#N Cn1nc(Br)cc1S(=O)(=O)N1CCCC(C2(C)COC(=O)N2)C1 c1(CNC(C23CC2CN(Cc2ncccc2Br)C3)=O)cnc2ccc(Cl)cn12 C1(CNC(c2c(C)ccnc2)=O)CCN(C(C2(C)CCNC2=O)=O)CCC1(F)F C1(NC(Cc2c(C)cccc2)=O)CN(C(=O)Cn2cncn2)C2(CCCOC2)C1 CN1CCN(C(=O)NC2CC2c2cccc(Br)c2)C(C2CC2)C1 C12(NC(C3CC4C=CC3O4)=O)CCN(C(=O)CC3CN4CCC3CC4)CC1C2 c1(CNC(C(C(C=C)C)C)=O)nc2c(s1)CN(C(c1n[nH]cc1CC)=O)CC2 C#CCC(C)(C(=O)N1CC(S(C)=O)C1)NC(=O)CC(C=C)CC c1(SC)ccc(C(N2CCC(N3CCC(CN(C)C)CC3)CC2)=O)cc1 Cc1cc2ccccc2cc1C(N1CC(NC(C2CCC(=O)O2)=O)C2(CC2)C1)=O Cc1cccc(C(C)C)c1-n1nc(-c2ccoc2)nc1C1CC(CF)C1 N(C1CCOc2c(F)ccc(F)c21)C(=O)Nc1n(C(C)C2CC2)ncc1 c1(C(=O)NC(C(=O)N(C)CC2CCCO2)c2ccoc2)cccn2cncc12 Cc1cc(NC(=O)CCN(C(c2cn(C)c(C)n2)=O)C(C)C)ccc1O c1(N2CC(CC(C)C)OCC2)nc(=NCC=CCl)[nH]c2c1CCCC2 C1(OC)CC2C1CCN2C(=O)C(C1CC1)N(C)C(C1CNC(=O)O1)=O C1(C(N2CC(C(C(=O)NCC3(C#N)CCCC3)OC)C2)=O)CCCCC(=O)N1 c1(C(N2CCOC(c3nc(C4CC4)no3)C2)C(=O)NC)nc(C(F)(F)F)oc1C c1(C(=O)N)cnc(C2CC2)[nH]c1=N.c1(SC)cccc(C(=O)NC2CCCC2)c1 c12cccc(c1)C(=O)N2C1(C(=O)O)CC1C.c1(C(C2CC2)OC)nc[nH]n1 C1(C)(CNC(c2cnc(C)o2)=O)CCC(NC(=O)CN2CCOCC2=O)CC1 C12(NC(c3n[nH]cc3[N+](=O)[O-])=O)CCCC1N(C(c1cc([N+](=O)[O-])c[nH]1)=O)CC2 c1(C(=O)NCC2(F)CC(CNC(C3C=CCC3)=O)C2)ncccc1Br C1(NC(c2c(C)cc(C)o2)=O)CCCC(NC(=O)C=CC2CCCC2)CC1 c1(C(=O)OC)cc(CNC2CN(C(=O)C(O)C(C)C)CC23CC3)ccc1F N1(C(CS(=O)(=O)NC)=O)CCCCC(NC(c2ccn(C3CCOCC3)n2)=O)C1 Cc1oc(C(=O)NC2CC(C)(CNC(=O)C(O)c3ccsc3)C2)cc1CO c1(C(C(N2CCN(C(C(CC=C)CC)=O)CC2)=O)(F)F)ccc([N+](=O)[O-])cc1 C=CCCC(F)(F)C(=O)N1CC(NC(=O)CN2CCCCCC2)C(SC)C1 C#Cc1ccc(C(=O)NC)c(C)c1.n1(CC(N2CCC2)=O)nc(C)n(C)c1=O C1(N(C(CC=C=C)=O)Cc2ccccn2)CCN(C(=O)COCC(=C)C)CC1 Cc1ccc(CCC(=O)NC2(C)CCN(C(C34CCC(C3)C4)=O)C2)nc1 c1(C(=O)NCC(CNC(C2C(COC)CC2)=O)OC)cc(O)nc(O)n1 C1(NC(CN(CCOC)C(C2C=CCC2)=O)=O)CCC(=O)NC1(C)C C(Cc1ccccc1)(C(=O)NC(c1cn(-c2ccccc2)nn1)(C)C)N(C)C CN=c1[nH]cnc2cc(C(=O)NCCNC(=O)CN3C(=O)CCC3=O)ccc12 C(C(=O)N1CCCc2nncn21)OC(C(CN(C(CCC(CC)CC)=O)CC)C)=O C1(SC)CN(C(c2ccc(-c3ccco3)cc2)=O)CC1N c1(NC(=O)NCC2(CCC=C)CC2)ccc(S(=O)(=O)NC(C)C)cc1 C1(CCOC)(NC(=O)C2=CCCC2)CCN(c2nc(C(=O)OC)cc(C)n2)CC1 C1(CCn2cc(CS(C)(=O)=O)nn2)CCC2(CC1)COC2.C(C#N)N C1(C=O)CCS(=O)(=O)CC1.c1(CC)sc(=N)[nH]c1C(=O)N.C1(F)CCC1 C(=O)(CCC(=O)C(C)(C)C)N1CC(C(C)C)N(C(c2cnc(F)c(Cl)c2)=O)CC1 c1(C(=O)NCCCCN(C(CC(C)c2ccncc2)=O)C)cc2ncccc2o1 c1(OC(C)C)cccc(C=CC=O)c1.C1(CC=O)CC(C)(C)C1.CC(O)C c1(CCCCC)cn(C2CC3(C(=O)NC(C)(C)CN4CCCC4)CC23)nn1 N1(C(c2ccnc(C)n2)=O)CC23CCCC2(C1)CN(c1ncnc2scnc12)C3 Cc1ccc(NC(C2C(C)CCN2C(c2ccoc2C)=O)=O)cc1O C(C)(c1ccccc1F)=CC(=O)NC1CCC(NC(C(C)OCC#C)=O)C1 C1(OC)CC(NC(C23CCCC2CCC3)=O)CN(C(=O)C(=CC2CCCC2)C)C1 C(CNC(C1(O)CCSC1)=O)(CC(=O)NCc1cnc(C)[nH]1)OC Cc1cc(Br)ccc1C(=O)NC(C1CCN(C(c2ccc(Br)cc2Br)=O)CC1)C C1(N(C(c2ccc(C)cn2)=O)CC2CCCCC2)COC2(CCNCC2)C1 CC1CN(C(c2ccnn2CC(F)F)=O)CC(C)C1NC(C1CC(C)(C)C1)=O C(=O)(CCCN(C)N=O)NC(CCC1N(C(CCC(CC)C)=O)CCCC1)(C)C C(=O)(C(C(C)OC)NC(=O)CC(C)O)NC CCC(C)CCN=c1[nH]c(N2CCC(c3cccc(Cl)c3C)C2)nc2c1CSC2 CC1(C)Cc2cc(C(=O)NC3C4CC5CN(C(=O)CC(F)(F)F)C3C5C4)sc2C1 C(=O)(C(C)C(C)S(C)(=O)=O)NC1CC(C)(NC(CCCCCCC)=O)C1 C(=O)(CCC(C)(C)F)N1CCC(N(C(=O)CC2CC3CC3C2)C)CC1 C1(C(=O)OC)C2CN(C(C3OCCC3NC(C3(CF)CC3)=O)=O)CC12 C12CCC3CN(CC13)C(=O)Cc1cn(nn1)C(=O)N2.c1(CC)cccc(NC)c1 c1(C(=O)NCCC2(OC)CN(c3cc(Cl)nc(C)n3)C2)c(C)cc(C)nc1Cl C1(C)(C(=O)NCC(C2CCC2)OC)C=CCN1C(=O)C=CC1CCCC1 C(C(C)NC(c1ccnc(C)c1)=O)(C(C)C)NC(CSCC#C)=O C(=O)(C#CC(C)(C)C)NC(C)CS(N)(=O)=O.C1(C=O)CC(=O)CC12CCC2.N C(C)(C1=CCN(C)CC1)NC(C1CCN(C(c2ccc(C)cc2C)=O)C1)=O C(CC(O)C(=O)N(C(C)C(=O)OC)C1CC1)NC(c1n(COC)ncc1)=O c1c(C)cccc1Cl.Cc1ccn(CC(C)C(=O)N2CC(CNC(=O)CO)C2)n1 CN1CCC2(CCN(C(C3CCc4nc[nH]c4C3)=O)CC2)C1.C12CCCN1C2 N1(C(C=C(C)C)=O)CCC(O)C(N(C)C(c2cc(C(F)(F)F)n[nH]2)=O)C1 N1(C(c2cc(CC)n(C)n2)=O)CCN(C(C2(C)CC2C)=O)CC2(CC2)C1 C(CC(C(=O)NC1(c2nc[nH]n2)CC1)NC(=O)C(Cl)Cl)OCC c1(C2(CNC(=O)NCCC3(CC4CC4)CC3)CC2)ccccc1 C1(OC)C(C)(C)CN(C(c2cnn(C)c2C)C(=O)NC2CCOC2)C1(C)C c1(C(=O)NCC2(CNC(c3nc(C)sc3)=O)CCCC2)cc(C#N)no1 CC(CC(=O)N1CCC1C(=O)N(C1CCC2(CC1)CC2)C)C(F)(F)F CC(C)C(O)C(C)C(=O)NC1CCC(NC(=O)CO)C1.C1CCC(F)(F)CC1 C=CC1CCCN(C(c2coc(CNC(=O)CC3CC4(CC4)CO3)n2)=O)C1 n1(CC)nc(CNC(=O)NCCCc2cccs2)c(C)n1 CC(C)(O)C(C)(C)CNC(C1CC(F)CCN1C(C1CCCC(CF)C1)=O)=O C(CCO)(C(F)(F)F)NC(C(C)CN(C(=O)CC1OCCO1)C)=O C1(CC(N2CCCCC2)=O)CCCC2(CC2)C1.c1(C(N(CC)C)=O)[nH]ncc1Cl O=C1CCc2cc(C(=O)NNC(=O)Nc3ccc(C(F)(F)F)cn3)c(O)cc2N1 Cc1cc(C(=O)NCC2(NC(c3coc(C)n3)=O)CCCCC2C)nc(O)c1 c1(OC)cc(N2CCC(NC(=O)C(=Cc3ccco3)C)C2(C)C)nc(OC)n1 N1(Cc2cn(C3CCN(C(c4cn(C)nc4)=O)C3)nn2)Cc2cccc(F)c2C1 C#Cc1cccc(C(=O)NCC2CN(C(c3coc(C(C)=O)c3)=O)C2)c1Cl.O Cc1c(CNC(=O)C(C)(C)C2CCN(C(=O)C(F)C(C)C)C2)cccc1O CCCC(C)CC(=O)NCCCC(C)NC(=O)Cn1nc(C(=O)OC)cc1C CC(C)(C(=O)NCC1CC(NC(c2snc(Cl)c2Cl)=O)C1)C(F)F N1(C(CCn2ncc(C)c2)=O)CCCC2(CCC2NC(=O)C=C2CCN(C)C2)C1 N1(C(C(C)OCOC)=O)CCCC(COC)(NC(=O)Cc2cncnc2)C1 c1(C(N2CCCC(C)C2CNC(=O)CN2CCCCC2)=O)cc2nc[nH]c2cn1 N1(C(CC2CC(=O)C2)=O)Cc2ccccc2CC1CNC(=O)C1=C(Cl)CCOC1 c1(OC)ncc(C(=O)NCC(C)CNC(C2(CC(F)F)CC2)=O)c(C)n1 N1(C(C(C)OCC(F)(F)F)=O)CCCCC(Cn2cc(C3CCCN3C)nn2)C1 Cc1c(C(N2CCN(C(C3CCCOC3)=O)CC2)=O)nnn1C C1(C(N2CCC(CNC(c3cn(C(F)F)cn3)=O)C2)=O)CCCS1(=O)=O C1(C(=O)NC2CCN(C(COCCC#C)=O)C2)C2CC3C(C2)C13 CCCCC(C)C(C(=O)NCCC)N1CCCC(C)(CC)C1 N1(C(C(CC=C)(C)C)=O)CCC2(CCC2)C(NC(c2cc3ncccn3n2)=O)C1 C1(NC(C(C(C)C)F)=O)CCN(C(=O)Cc2ccc(Cl)nc2)C12CCC2 c1(C(N(CC(C)N(C)C(C2CC(O)C2)=O)C)=O)cccc2c1CCCCC2 c1(SC)cn(C)nc1C(=O)NCC1(F)CCCC1.C(=O)(COC(F)F)N CCC(CC(=O)NCC1(C(=O)NCCN2CCCC2)CCCCC1)SC C=CCCCCCC(=O)NCC(C1CCCN(C(c2sc(=N)[nH]c2C)=O)C1)(C)O C1(CNC(=O)Cn2ccnn2)CN(C(C23CCCC2C3)=O)CC1(F)F S(=O)(=O)(c1ccc(F)cc1Cl)N1CCC(C(=O)NCc2ncc(CCO)s2)C1 N1(C(c2cc(C(F)(F)F)ns2)=O)CCC(F)(c2cn(Cc3cccs3)nn2)C1 C1(C(C(=O)NC(C)(C)C)N(C(C=C)C)C)CC2C(C1)C2(F)F C1(C(F)(F)F)(C(N(CCC(C)NC(C(C)SCC)=O)C)=O)CCOCC1 N1(C(c2ccc(C)nn2)=O)CCC2CN(C(C3(C)CC3)=O)CCC2C1 N1(C(c2cc(C)ns2)=O)CC(C)CCC1CNC(=O)Cc1ccsc1 c1(OCCC)cc(C)ccc1C(=O)NCc1cc(-c2ccccc2)on1 CC1CC(NC(C2CSC2)=O)CCN1C(c1ccccc1C(C)(C)C)=O CCC(C)C(O)C(=O)NC(C1CCN(C(c2cc(C)cnc2C)=O)CC1)C C#Cc1ccc(OC)c(C(=O)NC23CC(C2)C3)c1.C1(C(=O)N)CC12CCCC2 C1(NC(CCc2cc(C)[nH]n2)=O)CCCN(C(=O)CCOC2CCCOC2)CC1 c1(C(=O)NC(C)C(C)(C)NC(c2nccnc2N)=O)ccc(-c2cc[nH]n2)cc1 C1(C(N2C(C(C)(C)C)CCCC2)=O)CN(C(=O)CN2CCSCC2)CC1(F)F CCCCCCC(C)C(=O)N1CC2CC1(C(=O)N(CC(C)O)CCO)C2 C1(C)(OCCNC(CNC(COc2ccn(C)n2)=O)=O)CC2CCC1C2 C1CCC2(CCC2)C1.c1(CC=O)ccc(F)cc1F.C(C)(C(=O)NC)=C(C)C c1(C(N2CC3CCC(C2)N3C(C2CC(O)C(F)C2)=O)=O)cc2cccnc2s1 C(CC1OCCc2ccccc21)NC(C12CCC(c3ccccc3)(C1)C2)=O C(N=c1[nH]nc(-c2ccc(F)cc2)o1)c1ccc(NC(C)=O)s1 c1(CC)ncc2c(n1)CCC(C(N1CCC(NC(=O)C(C)=C3CCC3)CC1)=O)C2 O=C(Cc1ccc2nonc2c1)NN=c1[nH]nc(C(F)F)s1 C1(C(=O)NCC2(CCC)CC2)CC(C)(C)CN1C(=O)Cn1ccnn1.C c1(C=O)ccc2c(c1)COC2.C1(NC(C2CC(SC)C2)=O)CC(F)(F)C1.C C12(CCNC(CCC=CC)=O)CCC(CC1)N(C(c1cc(Br)no1)=O)C2 Cc1cc(C(F)(F)F)ccc1S(=O)(=O)Nc1cccc2c1ccn2C C1(CNC(=O)NCC2(CO)CCNC2)CC2(C1)CC2F.c1ccccc1.C c1(C(N2C(CNC(C(COC)NC(C)=O)=O)CC2)=O)cnc2[nH]ncc2c1 Cc1cccc(C(N2CCC3CC23CCN2CCOCC2)C(=O)NC2CCC2)c1 c1(OCC)ccc(C(=O)N(C2CSC2)CC)cn1 c1(C(N2CC(C(C)NC(CCC(=O)NCC)=O)C2)=O)c[nH]nc1[N+](=O)[O-] C=CCN=c1[nH]cc(C(=O)Nc2ccc(C)c(OC)c2)s1 Cc1noc(C2CC2)c1NC(=O)NCCN1CCCC1C(=O)NC(C)C c1(C(=O)NCCC2CC(C(N(CC(CC)C)CC)=O)C2)cc(Cl)c[nH]1 C(CCOCCO)(C(=O)NC(C1CCOC1)CO)NC(=O)CCCF C1(C(=O)NC2(CC(C)C)CC2)C(C)CN1C(=O)CCc1cccnc1 c1(C(=O)NC(C2OCCN(C(c3nc(C)oc3)=O)C2)C)cc(C)c(N)cc1Cl CC1CCN(C(c2cc(Cl)cs2)=O)CC1C.c1(C(=O)N)cc(C(F)(F)F)nn1C C=CC(CCC)CC(=O)NC(CC(=C)C)C(=O)NCCOC1CC1(F)F c1ccc(C(=O)NC2C=CS(=O)(=O)C2)cc1.c1cccc(Cl)c1.C=CC(=O)N O=C(C1=CS(=O)CCC1)NCCOC1CCN(C(=O)CSc2ccncc2)C1 N1(C(Cc2c(C)ncs2)=O)CCCC(CCNC(C2(CO)CCCO2)=O)C1 N1(C(c2c(OCC)scc2)=O)CCC2CC1CN(C(=O)C(C)Cc1ccco1)C2 C(N=c1cc[nH]cc1S(=O)(=O)NCCCCC(C)(F)F)C1C(CCC)CCC1 C(=O)(C1CCc2ccccc21)NCC(CNC(c1cncc(N=[N+]=[N-])c1)=O)O c1(C(=O)NCC(CNC(CCC(=C)Br)=O)C)ccc2sncc2c1 N1(C(c2c(C)c[nH]c2)=O)CC(C(=O)N(CC(C)(C)C)CC(C)C)C(F)C1 c1(C(N2CC(C(=O)Nc3ccccc3Cl)C2)=O)ccc(F)c2occc12 C(=O)(Nn1cccn1)c1c(CN(C(CS(CC)=O)=O)CC(F)F)cc[nH]1 c1(N2CC(CNC(Cc3cn(C)nc3)=O)C(F)(F)CC2)ccc([N+](=O)[O-])c(O)n1 c1(C(=O)NC2(CCOC)CCN(C(C3CCOC3)=O)C2)ccc2cccnc2c1 N1(CC2C(C(N(CC#C)C)=O)C2)CCN(C(=O)C(C)=CC(C)(C)C)CC1C N1(C(CCC)=O)CCCCC1C(=O)NCC(C)NC(=O)C(F)(F)CF c1(C(N(C2CCN(C(C3ON=C(CC)C3)=O)C2)C)=O)ccc(OC)c(Cl)c1OC c1(-c2nc(-c3c(C)occ3)nn2C(c2ccc(Cl)cc2)C)cc2c[nH]cnc-2n1 Nc1ccc(C(N2CC(NC(=O)Cn3cc(CO)nn3)C3(CC3)C2)=O)nc1Cl c1ccc(Cl)c(Cl)c1.S(=O)(=O)(C1CC1)NCC(=O)N(CC=O)C1CC1 c1(C(=O)NC2CN(C(C3C(CC)CC3)=O)C(C)(COC)C2)cnc2[nH]ncc2c1 C#CCCC(O)C(=O)N(CC(CC)NC(C1(c2ccccc2OC)CCC1)=O)C C1(C(=O)OC)CN(C(c2cc3n(c2)CCOC3)=O)CC(C)(C)S1(=O)=O C#CCCC(C(=O)NCc1ccnn1C(C)C)NC(C1CC2CC2C1)=O N1(CC)CCCC(C(=O)NC2(C(=O)NCC(O)CC(C)C)CCN(C)C2)C1 C1(NC(CC(C)(C)OC)=O)CN(C(=O)C2CCc3nccn32)C2(CCOCC2)C1 n1(CC=O)cccc(C)c1=O.C1(CNC(C2(C#C)CC2)=O)COC(C)C1.N C1(C(N2CC(OCCCCC)C2)=O)COCCN(C(C2CC3CCC2CC3)=O)C1 C1(C(=O)NC2CC(C(C)NC(C(CCSC)O)=O)C2)CCC=CCCC1 C(C(CC(=O)NC1CC2C=CC1C2)NC(=O)Cc1ccoc1)OC Cc1cc(N)c(C(=O)NC2CCCN(C(=O)C=CCN3CCOCC3)C2)cc1C C1CC2CN(C(=O)CN3CC(C)(C)C3)CC12.c1(C(C)C)nnc(C=CC=O)o1 Cc1nn(C)c(C)c1C(N1CCC(N(C(=O)Cc2ccc(Br)cn2)C)C1)=O c1(OC)cc(C(N2CC3CC2(CNC(=O)C(C)SC)C3)=O)c(F)c(Cl)c1 Cc1cc(=NCc2ccc(N)cn2)[nH]c(N2CCc3n[nH]cc3C2)n1 CC1(C)C(NC(=O)CSC2CC2)CC1CNC(=O)CCC(N)=O C(C(O)CC(=O)NCC=CBr)NC(C(CC)=CCCC)=O CON1CCC(C(=O)NCC=CC(=O)NC(c2cnn(C)c2)(C)C)CC1 c1(NC(c2ccc(OCC(=O)N(C)C)cc2)=O)cc(F)c(C(F)(F)F)cc1F N1(C(c2c(CC)cccc2)=O)CCC(C)C(NC(c2cc(Br)cs2)=O)C1 CCC(CC(=O)NC(Cc1ccco1)C(=O)N(CC(O)C1CCC1)C)SC C1C2CCCCCC12.C1(C=O)(CNC(C2CC(O)C(F)C2)=O)CC2(CC2)C1 CCCC(C)(O)CC(=O)NC(CO)C(=O)NCc1cccnc1 N1(C(C(C2CCC2)OC)=O)CC2(C1)SCCC2NC(c1nsc2ccccc12)=O c1(OC)oc(C)nc1C(=O)NCC(CNC(=O)COC1CCCCC1)CO C1(C)(SC)CN(C(C2CC(CNC(C3CCC3)=O)C2)=O)C1.C(C)=O.N C1(C=O)CCC(=O)N(CC(F)(F)F)C1.c1(CC)nc(C)c(C(=O)NCC)s1 C1(C(C)C)CN(C(C2CCCN2C(c2ccccc2)=O)=O)CC(=O)N1 N1(C(CCC(C)OCC)=O)CCC2CCCC12C(N1CCC2C(C1)C2(F)F)=O Cc1c(Br)ccc(F)c1CNC(C1CCCO1)C1CC1 c1(C(=O)NCC2CCN(C(=O)COCCF)C2)ccn2c(Br)cnc2c1 n1(C(C)(C)C)nnc(C(N2CCC(NC(c3cccnn3)=O)C2)=O)n1.C1CC1.C C(C)(CNC(=O)C(c1ccc(O)cc1)OC)(CC(C)C)NC(CCC=C=C)=O C1(C(N(CC(CC)C)C)=O)C2CCCC2CN1C(=O)C=Cc1ccoc1 C1(C(C)C)CCc2[nH]nc(C(=O)N(CCNC(C3CCSC3)=O)C3CC3)c2C1 O=C1CC(C(N2CCCC3(NC(C4CCSC4)=O)CC3C2)=O)C2CCCCC2N1 C1(C(N(CC)C2CC2)=O)CC(S(N)(=O)=O)C1.C1(CCCC)(C=O)CCC1 S(=O)(=O)(c1c(Cl)cccc1Cl)NCC1CCCN(C(c2cccc(OC)n2)=O)C1 C=C(C)C(C)(O)C(=O)NC1CCC(N(C(=O)C(=Cc2ccc(F)cc2)C)C)CC1 C(C)(CO)(C(F)(F)F)C(C1CCC(COCC)CC1)=O.C1CN(C2COC2)C1 c1(CNC(C2(COC)CCCO2)=O)cccc(C(N2CCC3CC3C2)=O)n1 C1(CC)CN(C(=O)CS(=O)(=O)CCOC)CCC1N=c1[nH]c(Cl)nc2[nH]ccc12 N1(C(c2cc(C)on2)=O)CCCC2(CNC(c3ccc(C(=O)CF)cc3)=O)CC12 C(=O)(CCCC(C)(C)NC(c1sccc1CO)=O)NC(c1ccccn1)C c1(C(N(CC(CC)NC(=O)CN2CC3CC3C2)C)=O)ncc(Cl)cc1Cl C1(CNC(CNC)=O)CCCC(NC(=O)C)C1.c1ccc(Cl)s1.C1CCC1 O=C(CC1OCc2cc(Cl)ccc21)NC1(O)CCc2ccccc2C1 C1(F)(C2CC2)CCC1.C(C(=O)N)(C1CCCC1)N.C(=O)C.CC(=O)C=O c1ccc(O)c(I)c1.c1(CNC(C2CC3CC3N2)=O)cnc(C(F)(F)F)cn1 N1(C(C2N(CCC)CCC2)=O)CC(NC(=O)CCCOC)C2(CC2)C1 C(=O)CC(C)C(F)(F)F.N1(C(c2n(CC(C)C)ncc2)=O)C2CCC1C(C)C2.N CN(CCCC(=O)NC1CCN(C(C2CCC(C)(C)C2)=O)C12CC2)N=O N1(C(C2(CC)COC2)=O)CCCC12CCN(C(c1ccc(C(N)=O)cc1)=O)C2 O=C(O)CC1CN(CC(O)COc2c(F)cccc2F)Cc2ccccc21 C(=O)(C(CC(F)F)N(C)C(C1CC(C)(C)CO1)=O)N1CC=C(C)CC1 C1(COC)CC(C)N(C(=O)CCC#N)C1.c1(C(=O)N)csc(C)c1C1CC1 C1(OCC(=O)N(CC(C)NC(=O)Cc2ccon2)C)CCN(C)CC1 C(=O)(C1c2c[nH]nc2CN1C(=O)CCCC1CCCC1)NCC(c1ccsc1)C CN=c1nc(C(=O)NCC(O)C)cc(C)[nH]1.c1(C(=O)N)ccoc1C(F)(F)F C1(CNC(c2ccc(CCC)s2)=O)CC(NC(=O)CCCOC)C12CCC2 N1(C(=O)CCOC2CC2)CCC(CO)(NC(C2C3CCCCC23)=O)C1 c1(NC(C=CC(C)(C)NC(c2ccco2)=O)=O)cccc(CCF)c1 N1(C(C(CSC)C)=O)CCN(C)C(C(=O)N(C(CF)CF)C)C1 C#CCCCCC(c1nnnn1CCCC)Nc1ccc(OC(F)F)nc1 Cc1c(C(=O)NC2CCN(CCC)C2)cccc1O.C1(C)(CC(=O)N)CC1(Cl)Cl c1(C(=O)NC2CN(C(C=CC)=O)C3C2C3)ccc(N=[N+]=[N-])cc1 C(CCO)(CC(C)C)NC(C1(CCNC(c2ccc(C(C)=O)o2)=O)CC1)=O C12CCCC1CN(C(c1cc(Cl)c(C)cn1)=O)C2.C(C)(CCC(=O)NC)OCC C=CCCCCC(=O)NCC(CC1CC1)C(N1CC2(CC=CC2)C1)=O N1(CC(N2CCN(C(CC(C)CF)=O)CC2)=O)CC(=O)Nc2ccccc21 C1(O)(CC(=O)N(C2CCC(NC(C3(F)CCC3)=O)CC2)C)CCCOC1 N1(C(c2c(NCC)scn2)=O)CC2CCC(N(C(=O)CC(C)CC(C)C)C)C2C1 C1(C(N(C)CC2OCCN(C(CNS(CC)(=O)=O)=O)C2)=O)CC2(CCOC2)C1 N#CC1=C(C(=O)N)CCC1.C1(F)CCN(C(C2CCOC2C(F)(F)F)=O)CC1.C c1(C(=O)NCC2COCCN(C(c3c(C)onc3O)=O)C2)[nH]nc([N+](=O)[O-])c1Cl c1(OC)c(C(=O)NCC2(C(=O)N(CCO)C3CC3)CC=CC2)cnn1C N1(C(CC(C)CN(C)C)=O)CCN(C(C2C=CCC2)=O)CC1CO C#CCC(O)C(=O)NC1CCN(C(=O)C(C(C)C)C2CCC2)C1 c1(CC)nc(O)c(C(N2CCC(NC(=O)CC(CC)C3CC3)CC2C)=O)cc1C c1(OC)ccc2cc(C(=O)NCC(C)NC(c3cc(Br)cs3)=O)ccc2c1 C(=O)(C(C)(F)C(=O)OCC)N1CC(NC(c2c(CCC)n(C)nc2)=O)C(C)C1 c1(CN2C(COC)CCCC2)cnc2sc(Br)cn12 C1(NC(C(C(C)C)(C)C)=O)CC2CCC1N(C(c1cn3ccnc3s1)=O)C2 C=CC(C)(CCOC)C(=O)NCc1cscn1.n1(C(C=O)C)ccc(C)n1.C c1(CC(=O)NCC(C)(C)N(C(C)=O)CC)nc(C2CC2)c(C)s1 C1(CC(=O)NCC(CN(C(C(C(C)C)C(C)C)=O)C)O)COc2ccccc2O1 Cc1ccc(OC(C)C(=O)NC(C)CCNC(c2cnns2)=O)cc1 C1(NC(CCCCCC)=O)CCOC12CCN(C(C1CC=CCO1)=O)CC2 C(CCC)(C(=O)N1CCC(CO)(NC(=O)Cn2nccn2)C1)=CCC C1(C(N2CC=C(CNC(c3cnc(C(C)C)[nH]3)=O)CC2)=O)CCCC12OCCO2 Cc1cccc(CCC(=O)NCC#CCNC(=O)CC2CCCCO2)c1 C1(NC(COC(C)C)=O)CCCN(CC(=O)N(C)Cc2ccccn2)C1 C1(C(N2CC(F)CC(NC(C3CC(=C)C3)=O)C2)=O)CCCCC1C1CC1 C(=O)(C(C)Cc1cnco1)N(CCNC(=O)CC1CCSC1)CC C(CC(C)C)(C(=O)NC1CC(CC)C1)OC.c1(C(=O)N)cnc(CC(C)C)[nH]1 CCCCCCC(=O)N1CC(CC(F)C(=O)NCC(CC)CO)C1 C(C)(CCC(=O)NOCC1CC2C=CC1C2)NC(C1=CCCC1C)=O N1(C(C2CCC(C)C2)=O)CC2CC(C=O)(C2)C1.C1(CC2CCC2)CCC1.C n1(CCCC)nc(C2CCCC2)nc1-c1cccc(CCCc2ccccc2)c1 N1(CCCCNC(=O)NCCc2c(C)n[nH]c2)CC(C)OC(C)C1 c1(C(N2CCC(NC(C(CSC)O)=O)C2C2CC2)=O)ccc2c(c1)C(=O)OC2 Cn1ncc2c1CCC(C(=O)NC1CC1CNC(c1ccc3c[nH]nc3c1)=O)C2 c1(C(=O)NCC2(C)CCCN(C(C3CCC(C)C3)=O)C2)cnc2ncnn2c1O c1(C(N2C(C(=O)Nc3ccnnc3)CC3(CC3)C2)=O)cnc2[nH]ncc2c1 Cc1ncc(CCNC(=O)Cc2cn(C)nn2)s1.c1(C=O)ccn(C(C)C)n1 C1(NC(c2nncc(C)c2)=O)CCCN(C(=O)Cc2ccnc(C)c2)C1C c1(C(N2CC3CN(C(c4cccc(OC)n4)=O)C3C2)=O)cc(Br)cc(F)c1O C(=O)(CCCCCC#N)NC1CC(CNC(c2c(NC)cc(Cl)cc2)=O)C1 C(=O)(C1CC(=O)Nc2ncccc21)NC1(CC=C)CCN(C(C2CCCO2)=O)C1 c1(SC)cccc(S(=O)(=O)NC2CCCN(C)C2c2ccccc2)c1 CC(C)CCCCC(=O)N1CCCC(CNC(C2CC(=C3CC3)C2)=O)C1 C1(CNC(=O)NC(c2cc(Cl)ccc2Cl)C2CC2)COC2(CCOCC2)O1 C1(NC(c2c(CC)nc(C)o2)=O)CCC(C)N(C(=O)CS(=O)(=O)NC)C1 C12(C(=O)O)CCCC1CC(NS(=O)(=O)Cn1cccn1)CC2 CCCCC(C(=O)NCCCN(C(=O)C(C)(c1cccs1)NC(C)=O)C)C(C)C Cn1ccc(CCC(N2CC(C)(C(=O)NCC3CCCOC3)C2)=O)n1 C1(C2CN(C(c3conc3C3CCC3)=O)C2)(NC(c2cnc3sccn23)=O)CC1 N1(C(c2c(C)nc(-c3c(Cl)cccc3Cl)s2)=O)CCN2C(=O)CCCC2C1 N(C(=NCCCN1CCOC1=O)NC1CCC2(C1)OCCO2)CC(C)C N1(C(CNS(NC)(=O)=O)=O)CC(CNC(c2cccc(=S)n2O)=O)CCC1C CC(CNC(=O)CCNC(=O)CCNC(=O)C=CCl)CC1CCC1 C1(C(N)=O)CN(C(C23COCC2C3)=O)C1.c1ccccc1.C(C(=O)N)=CC Cc1cc(F)cc(C(N2CCC(NC(=O)CCCCC3CC3)CC2)=O)c1O N1(C(C2OCCC(C)C2)=O)CC2(C(=O)NCC(O)CCO)CCC1CC2 C1(C(N2CCC(C(=O)O)CC(C)(C)C2)=O)C2CC3C4CC5CC3C1C(C5)C4C2 Cc1cc(N2CCC(NC(=O)NC(C3CCN(C)C3)C)C2=O)n(C)n1 C1(CCC(=O)OCCCC(=O)NC)CCN(C(=O)C(C)CCOC)CC1 Cc1cc(C(N2CC(CNC(c3c[nH]c(C#N)c3)=O)C(O)C2)=O)cc(C)c1Cl c1(CC)cc(C(=O)NC2(C)CC(NC(=O)CC3CCCN(C)C3)C2)ccc1O CC#CCCCC(=O)NC1CCN(C(=O)C(c2ccccc2F)F)C12CC2 C1(C(N2CCC(C)(CNC(C3CC=CC3)=O)C2)=O)CCCCC12OCCO2 c1(C2C(CNC(C(=O)N(CCC(=O)NC)C)=O)C2)cccc(OC)c1 c1(OC)cccc(C(=O)NCC(C)(C)CNC(C2(Cl)CC2(F)F)=O)c1N N1(C(C=C(C)CNC(C2CCC2C#N)=O)=O)CCOC(C)CC1 C1(NC(CC2C3CN(C(C(C=C)(C)C)=O)CC32)=O)CCC(C2CC2)C1 Cc1coc(C)c1C=CC(N1CCC12CN(C(C1CCC3CC13)=O)C2)=O CC1CN(C(=O)Cn2cc(C3CC3)nn2)CCC1NC(c1ccc(Cl)c(Cl)c1)=O c1(N2CCC(CC)(CC)C2)ncnc2c(Br)nn(C)c12 CCC(C)CCC(O)CC(=O)N1CCN(C(c2nn(C)c(Cl)c2Cl)=O)C(C)C1 c1(C=O)nc(C)c(N)cc1C.C#Cc1cncc(C(=O)NCC2(F)CCC2)c1.N c1(C(N2CCC(C(C)NC(c3cc(CO)on3)=O)C2)=O)ccc(Cl)c(F)c1 c1(NC(CCC)C)[nH]c(=NC2CCCC(F)(F)C2)nc2scnc12 Cc1cc(C(N2CCC(C(=O)NCC3(F)CCOC3)(C(C)C)C2)=O)nnc1O C1(C(N(CC(=O)NCC(F)F)C)=O)CCC2(CCC2)O1 c1(C(=O)NC2C(CNC(CCC(C)(C)C)=O)C2)c(F)ccc(N)c1Br c1(C(N2CCOC(C)C2CO)=O)cc(Cl)ccc1Cl C(=O)(CN=c1cc[nH]cc1)N(CCC(C(C)(C)C)NC(=O)CCN1CCC1)C c1(CC(=O)N(CC(C)NC(=O)CCc2cn[nH]c2)C)cccc(Br)c1F C1(N(C(C2CCC2)=O)CCO)CCN(C(=O)CC2CC(F)(F)C2)CC1.CNC c1(CNCC2N(C(C3(F)CC3)=O)CCOC2)ccc(O)c(F)c1 c1(C(C)N(C)C(c2cncn2C)=O)ccccc1F.C(=O)C(C1CC1)C1CC1.N C1(C(=O)NC2C(CNC(=O)Cc3ccco3)CCC2)CCCCC1O CC1(C)CCCCC1=CC(N1CCC(F)(C)CC1)=O.C1(C=O)CC2(CC2)CO1.N CC1CN(C(c2ccc3c(n2)CCC3)=O)CCCN1C(=O)C(O)Cc1cnc[nH]1 C(=O)(CCC(=O)C(C)(C)C)NC(C(=O)NCC(CO)OC)c1cccs1 CC1(C)C(NC(=O)C2CC2)CCN1C(=O)Cc1cccc(O)c1 c1(C(=O)NCC2C3CN(Cc4cc(C)on4)CC32)ccc2nc[nH]c2n1 C(=O)(CCCC(C)c1cccc(OC)c1)NCC(CN(C(C(CC)F)=O)C)(C)C N1(C(C(C(C)C)n2cccc2)=O)CCN(C(=O)COc2cccnc2)C(CO)C1 c1(C(=O)NCC2C(C)CCN(C(=O)C(N)=O)C2)nn2ccccc2c1Br c1(C(=O)NCC2(C(C)NC(CCOC)=O)CC2)cc2ccccc2c(O)n1 C(=O)(CC(CCC)CCC)NC1(CC=C)CCN(C(c2cncn2C(C)C)=O)C1 CC(C)(C)C(CN=c1[nH]cnc2cccc(Br)c12)NC(c1c(Cl)ccnc1F)=O C1(C(N(CCN(C(=O)C(c2cnn(C)c2)=O)C)C)=O)CCCN1C1CC1 C=CCC(C)(CC=C)NC(=O)CC1CCCCC1NC(=O)C(C)(O)C1CC1 C1(NC(C(CSC)C)=O)CCN(C(c2cnc(C)c(C#N)c2)=O)CC(O)C1 C1(CNC(c2c(OC)nsc2)=O)CCCCC1NC(=O)CC1CC=CCC1 c1(C2C(C(=O)NC(C3N(C(C)=O)CCC3)C)C2)ccc2c(c1)OCCO2 c1(CCNC(C2(F)C(C)C2)=O)ccc(F)cc1.c1(C2(C(=O)N)CC2)cc[nH]n1 c1(C(N2CCN(C)CC2CNC(=O)Cc2ccon2)=O)nc2cc(F)ccc2s1 N1(C(C(n2ccc(C)n2)(C)C)=O)CC(O)(C2CCN(C(C3CC3(C)C)=O)CC2)C1 C(=O)(C#CC1CCOC1)NC(C(=O)NCCc1cc(C)ncc1)Cc1cn[nH]c1 C(CC(C)C)(C(N)=O)NC(C1(NC(c2c(OC)cccc2)=O)CCCC1C)=O CC1CC(C(=O)N(C(CF)CF)C)CCN1C(=O)COC1(C)CCCC1 c1(NC(c2c(OC)nccc2)=O)cc(Br)ccc1NC(=O)CC(C)(F)F C(=O)(C1=C(Cl)CCCC1)N1CCOCC(CNC(c2cn(CCC)nn2)=O)C1 N1(C(C2(CNC(c3cnc(C)n3C)=O)CC(=C)C2)=O)CC2CC1CN2CC c1(C(C(=O)NCCOC)N(C)CCC2CCCN2C)cccc2cnn(C)c12 CC1(C(=O)NCc2ncccc2C(=O)NCC2CC2(Cl)Cl)CC=CCC1 CCC(C)(C)C(O)C(=O)N1CCC(NC(=O)C(C)CF)CC1C C1(NC(C=CSC)=O)CC2CC(C1)N(C(c1ccsc1Br)=O)C2 CC(C)C(C)C(C)CC(=O)N(C1CC2CCC(C1)N2C(=O)COC(C)(C)C)C C(=O)(C1=CN=C2N=CNN2C1)NC(CCCC)CNC(=O)CCc1nccn1C N1(C(C(C)OCCOC)=O)CC2(CCC2)C1.c1(C=O)ccccn1.C(C)=O C1(C(=O)NCC(C#C)CC2CC2)(CC=C)CCN(C(=O)Cc2ccnn2C)C1 c1(NCCCNS(C)(=O)=O)[nH]c(=NC2CCCc3cnccc32)nc2sccc12 N1(C(C(COC)COC)=O)CCC(F)(CNC(=O)CC2CCC(O)C2)CC1 C1(C(N(CCCCC(=O)NC)C)=O)CN(C(c2ccc(F)s2)=O)CC1(C)C C1(CC(=O)NC(CNC(Cc2nnc(C)s2)=O)(C)C)CC2(CCCC2)CO1 CC1CC(C)CN1C(c1cc(C(F)(F)F)cs1)=O.c1(C(C(=O)N)O)cccnc1 c1(OC)cc(OC)cc(C2CCN(C(=O)NCCC(=O)NCC(F)(F)F)C2)c1 CC1(C)CN(C(c2ccc(Cl)nc2O)=O)CCC1NC(=O)Cn1cnccc1=O C1(CCC(=O)NCC2C(NC(Cc3nc(C)oc3)=O)CC2)CCC(O)CC1 c1(CC)cc(C(=O)N(C2CCN(C(c3sc(Br)cc3Br)=O)C2)C)n(C)n1 c1(C(=O)NCC(C)=CC(=O)NCCS(C)(=N)=O)cccc2[nH]ccc12 N1(CC)OCC(NC(c2ccn(CC)c2)=O)C1=O.C1(Cl)(C(=O)N)CC1(F)F C1(CC(=O)NCCC2CCN(C(CCc3n(C)cnn3)=O)C2)CCS(=O)(=O)C1 N1(C(C2(CCNC(CC(CCC)C)=O)CC2)=O)CC2(CNC(=O)OC2)C1 c1(NC(CC2CCN(Cc3cccc(OC(C)=O)c3)CC2)=O)cnnc(O)c1Cl C1(C=O)CCCC2C1C2(F)F.c1(CC)cc(C(=O)NCC2(CC)CC2)n[nH]1 C1(OCCNC(CC2(C)CC2F)=O)(CNC(=O)C2=CCCC2)CCOCC1 C1(C)(CNC(CC(C)OC)=O)CCN(C(C2CCCN(C(C)=O)C2)=O)C1 C(=O)(C1=C(Cl)CCCC1)N.Cc1coc(C(C)C)c1C(=O)NCC1COCC1 c1(CN(C(c2ccccc2)CN2CCCC2)C2CC2)n[nH]c2c1CNCC2 C(=O)(C(C(=O)N1CCOCC1CN(C(=O)CCN1CCCC1=O)C)OC)OC c1(C(=O)NC(C)(C)CNC(C2CCC3(CCC3)C2)=O)nccn2cnnc12 N1(C(C)=O)CCCC(C(=O)NC2(CC)CC2)C1.C1(Cl)(C(=O)N)CC12CCC2 Cc1cc(F)cc(C(=O)NC23CC(NC(c4cccc(F)c4)=O)(C2)C3)c1N C=CCC(O)(CC=C)C(C)NC(C1CCCN(C(=O)Cc2ccc(I)cc2)C1)=O c1(NC(C2N(C(c3nnn(C)c3C(F)F)=O)CCCC2)=O)cccc(N=[N+]=[N-])c1 N1(C(CCCN(C(C)C)C)=O)CC(C)CN(C(=O)Cn2ccccc2=O)C(C)C1 N1(C(=O)OC(C)(C)C)CCC12CC(C(N1CCN(C(=O)CCCO)CC1)=O)C2 C12CCC(C1)N(C(c1cc(C)nn1-c1ccccn1)=O)C2.C(C(=O)N)SCC C(=O)(CCCC(C)NC(=O)C(C)(C)N(C)C)NC(c1ccccn1)C CC(C)(C#N)CCC(=O)N1CCC(OCC(N2CC(C)(CF)C2)=O)C1 N1(C(CNC(N)=O)=O)C2CC=C(C(=O)N3CCc4nncn4CC3)C1CC2 C(C(=O)NCC1(C(N2CCC2(C)CC)=O)CC=CC1)(C(C)C)OCC C(=O)(C(F)(F)C(F)(F)F)N1CCN(CC2CN(C(Cc3ccn(C)c3)=O)C2)CC1 N1(C(C(=O)NCCCC)CC)CCCN(CC(c2ccccc2)O)CC1 N1(CC(=O)NCC2CCN(C(c3csc(-c4ccncc4)n3)=O)C2)CCOCC1 c1(C(=O)NCC2CN(C(CC3(CC(=O)OC)CC3)=O)C2)ccncc1F C(=O)(CC(C)(O)c1ccccc1)NCCC1(NC(CC(C)SC)=O)CCC1 C=CCC(CC(=O)N1CCC(C(N)=O)C1)NC(=O)Cc1cncn1C c1(C(N2CC3C(CNC(C(C)(O)C4CC4)=O)(CC3)C2)=O)cnn2c1OCCC2 c1(OC)cc(C(N2CC(=O)NC(=O)C2)C(=O)NC2CCCCC2)oc(=O)c1 CCC(C)C(C(=O)NCC(CNC(c1cnc(C2CC2)o1)=O)CO)N(C)C C1(C(C)NC(CC2CC(=C)C2)=O)CCCN1C(c1cscc1C)=O c1(OC)cccc(CCNC(C23CSC(C2)C3)=O)c1.c1(C=O)n[nH]c(C)c1O c1(C(=O)NC(CC)(C)CCNC(=O)COC)ccnc2cc[nH]c12 O=C(C1=CCCN(C(C2CC23CCOCC3)=O)C1)N1CCC(CO)C1 c1(C2N(C(c3c(CCC)n[nH]c3)=O)CCC2)ccc(-c2nn[nH]n2)cc1 C1(C(C)Nc2cn(CC)nc2)CN(N(C)CC2CC2(C)C)C1 C(C(C)CC(=O)NCc1ccc(C(N2CCC(OCC(C)C)C2)=O)s1)OC C1(CC)C(C(N2CC(C#N)C2)=O)CCN1C(=O)Cc1ccsc1 N1(C(C2N(C)CCOC2)=O)CCOCC(C(=O)NCCn2cnccc2=O)C1 C1(NC(c2cnc(OC(C)C)nc2)=O)CCC(C(F)(F)F)NC1=O C(=O)(C1CCCc2c[nH]nc21)NC1C(C)(C)CN(C(=O)C2=COCCC2)C1 C(=O)(C(C)C(C)S(C)(=O)=O)N.N1(C(C2C(C(=O)OC)C2)=O)CCCCC1C C(=O)(C1=CC2CCCCCC12)N(CCCNC(C1(C)CSC1)=O)CCO c1(C(C)OC(CC(c2ccc(C)cc2)C)=O)ccc2c(c1)CC(=O)N2 C1(CC(=O)N(CCCC)C)CCN(C(=O)Cn2ccc(C)c2)C1(C)C C12(OC)CCC(C(N3CC=C(CC)CC3)=O)(CC1)CC2.C1(C)(C(=O)N)CCCS1 c1(C(N(C(CNC(C(=Cc2cnc[nH]2)C)=O)C)C)=O)cccc(C2(C)CCO2)c1 N1(C(C2N(C(CC(CCOC)(C)C)=O)CCCC2)=O)CCc2ccc(F)cc21 Cc1csc(C(=O)N(C)CCNC(c2c[nH]nc2F)=O)c1Cl c1(OC)c(C)cc(C(N2CCN(C(=O)C(C)c3cncs3)CC2CO)=O)cc1C C1(C(=O)NCCOC(C)(C)CNC(=O)C(C)(Cl)Cl)C(F)(F)C12CC2 C1(C(=O)NCC(CNC(C(CC=CC)CC)=O)C)CC(C)(C)OC(C)(C)C1 c1(C(=O)NCC(CNC(CCNC(=O)NC)=O)C)ccc(Cl)c(F)c1N C1(CC=C)(NC(=O)CSC)CCCN(C(c2ccccc2-c2nnc(C)o2)=O)C1 c1(C(N(C(C(=O)N(C)CC2CCCN2C)CC(F)F)C)=O)cccn2nccc12 Cc1cc(=NC(C)CNC(=O)C2=CC(C)(C)C2)nc(-c2cccs2)[nH]1 C1(C(N2CC(C(C)NC(=O)CS)C2)=O)COc2cc(F)ccc2C1.c1cccs1 N1(C(=O)Nc2ncc(CC(C)C)s2)CCCCCC(S(C)(=O)=O)C1 n1(CC(N2C(C(C)(C)C)CCC2)=O)[nH]cc2c(=O)ncnc1-2.C1(C=O)CSC1.N N1(C(=O)CSN2CCOC2=O)CCC(C(N2CC(F)C2)=O)C(c2ccccc2)C1 c1(CCC)noc2ncc(C(=O)NC3CCCN(C(=O)CC4CSC4)C3C)cc12 c1(NCC2CC(Sc3ccccc3)C2)cnc2c(c1)CCO2 C1(NC(C(CCC)N(C)C)=O)C2CCN(Cc3cn(C(C)(C)C(=O)O)nn3)CC12 C(=O)(C1=CCOC1)N(C1CCCN(C(=O)CC2CCCS2(=O)=O)C1)C N1(C(c2ccc(C)s2)=O)CCCC(C)(CNC(=O)Cn2nc(C)cc2C)C1 N1(C(c2cc(C)c(Cl)cc2)=O)Cc2ccnn2CC(NC(C2CC(C)(C)C2)=O)C1 Cc1c(C(=O)NCC(CNC(C2(C)CCCOC2)=O)S(C)(=O)=O)cncc1F C1(NC2(P(C)(C)=O)COC2)CC2CC3CC(C2)C1C3 C1(C(=O)N)C2C3CCC(C3)C12.C(CCCCNC(=O)C=CC(C)C)N(C)C N1(C(C2(C)CN(C)C(=O)CC2)=O)CC(C2CCN(C(c3nnsc3N)=O)CC2)C1 c1(C(N(C(=O)CSC2CC2)Cc2ccccn2)=O)ccc(Br)cc1 N1(C(C2C(OC)CN(C(C3(C)CCC(=O)C3)=O)C2)=O)CC2(CCC(=O)NC2)C1 C1(CNC(C2C(C)C2)=O)CCC2CN(c3cncc(Cl)n3)CCC2C1 N1(C(c2ccc(C(C)C)s2)=O)CCC(N(CCO)C(c2ccnnc2O)=O)CC1 C12CCOC(C1)SC1(C3CCC23)CC1.c1(SC(C)(C)C)cc(C2CCC2)no1 CCC(C)CC(C(=O)N(C)CCC1CCCN1C)NC(=O)C(C)SC C(=O)(CP(C)(C)=O)NCC1CC(NC(CCC2CCC(C)O2)=O)C1 C12(C=O)CC3CC(C(=O)N1)C2C3.c1nc(C=O)co1.CC=CC.COC C=C(Cl)CCC(=O)OC(c1ccc(-n2cccn2)cc1)C c1(-c2ccc(C(N3CCC(N(C(=O)C=CCF)C)C3)=O)o2)ccc(N)cc1 N1(C(c2c(C)ncs2)=O)CCC(C2CC2)CC1.C(=O)C(C)(O)C1CC1.COC c1(CC(=O)NC(CNC(C(C(=O)OC)C)=O)(C)C(C)C)cnc(Cl)cc1C N1(C(=O)C2=CSCS2)CCC2CN(C(=O)COCCF)CCC2C1 CC1CN(C(=O)C(F)(F)CC2CC2)CC1NC(=O)CN(C1CCCC1)C CCCCCCC(CC)C(=O)N1CCC(CCCCNC(=O)C(O)C2CC2)CC1 Cc1cc(C(N2CC3CC3(CNC(C3CCC(C(C)(C)C)O3)=O)C2)=O)ncn1 C1(C(=O)NC(C)(C)CF)CCOCC1NC(c1ccc(N)cn1)=O CC(CNC(=O)C=C1CCCCC1)C(F)C(=O)NCCCO N=c1[nH]c2cc(C(=O)NCC3CN(C(c4c(F)cc(F)cc4Cl)=O)C3)ccc2s1 c1(C(=O)NCC(CC)(C)NC(=O)CCn2cccn2)cnc2scc(C)n2c1=O c1(C(=O)NCCN(CCC)C(c2ccsc2C(F)F)=O)ncn2c1CCC2 c1(C(=O)NC2(C)CC(NC(c3c(C)nc[nH]3)=O)C2)noc2c1CC(C)CC2 c1(C(=O)NCC(C(=O)OC(C)(C)C)O)cc(Cl)sc1Cl c1(C(=O)NCC2CCCN(C(C(CCCC)C)=O)C2)cnc2cnccc2c1 CC(C)CC(C(=O)NC1CCCCC1(F)F)N(C)C(C1CC1Cl)=O c1ccc2c(c1)OCC2Cn1cc(CN2CCCNCC2)nn1 c1(OC)ccc(CC(=O)NC2C3CN(C(=O)CC4(O)CCOC4)CC23)c(Cl)c1 c1(OC)cc(CN2CCC(NC(c3c[nH]nc3-c3cccs3)=O)C2)sn1 N1(C(CC(COC)C)=O)CCCC(C)C1CNC(=O)C=Cc1cccnc1C c1(CNC(CC2CCC(NC(c3cn(CC)nc3)=O)C2)=O)ccccc1Cl C(c1ccccc1Cl)=C(C)C(=O)NCC(C)(C)CNC(=O)C1=COCCO1 c1(CC=O)cccc(C(F)(F)F)n1.c1(C(N(CCC)C(C)C)=O)ncn(C)n1 C1(C(N2CC3CC(NC(Cc4c(C)con4)=O)C3C2)=O)CCCC1S(C)(=O)=O Cc1nc(CO)ncc1C(=O)NC1CN(C(=O)C(C2CC2)N(C)C)CC12CC2 Cc1nc2cc(C(N3CCN(C(=O)CC(C)C)C4CC34)=O)ccc2o1 C1(NC(c2cc(F)c(F)cc2F)=O)CCC2(C1)CN(C(c1sc(Cl)nc1Cl)=O)C2 CC(CC(=O)N(CCCCC(=O)NC1CC1C1CCOCC1)C)C(C)(C)C c1(C(N(C(C(=O)NCC(COC)O)C)C2CC2)=O)ccc(Cl)cn1 C1(C(N(C(CC)CC(=O)N(C(C)CC(F)(F)F)C)C)=O)CC2C(C1)C2(C)C C=CCCCCCCC(=O)NC(C1CCN(C(C2CC3C=CC2C3)=O)CC1)C c1(C(=O)NCC(=C)CCNC(=O)C(F)=CC2CC2)cccn2cc(C)nc12 N1(C(C2CC(C)OCC2)=O)CCC2(CC1)CCN(C(=O)C1=COCC1)CC2 c1(C(N(CCC)C)=O)cnc(C2CCC2)nc1O.C1(C(=O)O)CC1C=O.CC C1(C(=O)NCCC(=C)CNC(=O)C(CC)n2cccn2)CCC(C(N)=O)CC1 C#Cc1cc(C(=O)NC(CC(=C)C)C(=O)N2CCCC(NC(C)=O)C2)ccc1C C1(NC(CCCOC)=O)(CNC(=O)C(C)Sc2nncn2C)CCCCCC1 N1(C(C2CN(C)C(=O)N2)=O)CCC2CN(C(c3cc(N)cc(F)c3)=O)CC2C1 c1(C(N2CC(NC(CCS(C)=O)=O)C2)=O)cccc2nc(C(F)F)sc12 c1(C(N2CC(F)(C(=O)Nc3cc(O)cc(O)c3)C2)=O)ccc(CO)cc1F c1(NC(C2C(C(=O)Nc3cccc(C(=O)OC)c3)C2)=O)nc(C)ccc1O C=CC1OCCCC1C(=O)Nc1cccc(NC(C2CC(O)CN2C)=O)c1 C=C(F)C1(CC(=O)NCC2CCC2C(=O)NC(C)C2CC2)CCC1 c1(C(N2C3CC(N(C)C(C4CC45CC5)=O)CC2CC3)=O)c(F)ccc2nc[nH]c12 C=CC1(C(=O)N(C)OCC(=O)OC)CCN(C(c2sccc2C)=O)C1 O=C(CCCC(F)(F)F)N(CCO)CC1CCN(Cc2ccccc2)CC1(F)F C(CC(C(=O)NCCn1ncnn1)NC(=O)CCCn1cccn1)SC c1(C(N(C(C)CNC(C2CCCSC2)=O)C)=O)cc(=O)c(Br)c[nH]1 c1(C(=O)NC(CNC(c2cn(CCC)nn2)=O)C2CC2)cncc(N)c1C Cc1ncc(CCC(=O)NCCCN(C)C(C2CCC(N(C)C)C2)=O)c(O)n1 C1(NC(c2cc(C)no2)=O)CCOCC1C(N1C2CCC1CC2)=O CCCCC(CNC(c1cnncc1C)=O)NC(c1cnn(CCO)c1CCC)=O C(=O)(C1CCCc2n[nH]cc21)NC(CNC(c1c(Cl)ccc(SC)c1)=O)C(C)C CCC(C(=O)N1CCC(CN(C)C(c2c[nH]c(C(N)=O)c2)=O)C1)n1ccnc1 N1(C(C2CCN(C)C2)=O)CCC2(CC1)CCN(C(c1cc(S(N)(=O)=O)co1)=O)C2 c1(C(=O)NC(CC)CN(C)C(C2(CC)CCCCO2)=O)ccc(F)c(Cl)c1F C1(NC(CCCOCC)=O)CC2CCC1N(c1nc(Oc3ccccc3)cs1)C2 C1(NC(=O)Cn2cncn2)CCN(C(=O)C(F)C2CCC2)C12CCC2 c1(C(=O)NC(Cc2c(OC)cccc2)(C)C)ncc(Br)cc1O C1(c2ccc(COC)o2)COCCN1CC(=O)Nc1cc(C)nn1C Cn1c(C(=O)NC2C3CN(C(C4(C)CCSCC4)=O)CC23)cc2occc12 c1(NC(c2n(CC)ncc2)c2nnnn2-c2ccccc2C)ccc(Br)cc1OC C(CC(C(C)C)NC(c1cc(Cl)c(Br)s1)=O)N(C(C(CC)OC)=O)C N1(C(c2c(C)csc2)=O)CCC(CNC(C2CC(F)(CF)C2)=O)C12CCC2 CC(c1ccc(F)cc1)=CCNC1(C(=O)NC(C)(C)C)CCCC1 c1(OC(C)C(N2CCCC(CNC(=O)C3=CCCS3)CC2)=O)cc(F)cc(F)c1 c1(C(N2CCC(NC(C3Cc4nccn4C3)=O)C2)=O)ccc2c(c1O)CCCC2 C1(C=O)CCn2nccc2C1.n1(CC)cc(CC(=O)NCC2CC2C)cn1.N C=CCC(CC)C(=O)NC1CCCN(C(=O)CCCOc2ccc(C)c(C)c2)C1 Cc1ccnc(C(=O)NCCNC(=O)CCN(CC(F)(F)F)C)c1Br N1(C(C2(CCCC)CC2)=O)CCCC(NC(=O)C(CC)n2cncn2)CCC1 C(CCCN(CC)CC)NC(CN(CC#C)C(C1CC1F)=O)=O N1(CC(=O)N(CCCCNC(C2CCC(=O)N2)=O)C)CCCC(C(N)=O)C1 Cc1cc(C(=O)NCC(C)NC(C2(C)CCC(=O)C2)=O)c2c(C)noc2n1 CN1CCOCC1C(=O)NC1CCN(C(=O)Cc2ccccc2)CC1 C1(CNC(C(C)(C)C2CCC2)=O)CCCN(C(C2CCCC23CC3)=O)C1 C1(NC(c2cn[nH]c2)=O)CC2CN(C(c3cnc(Cl)cn3)=O)CC12 C=Cc1cc(C(N2C3CCC2CC(N(C(=O)C=CCOC)C)C3)=O)cc(F)c1 N1(C(CN2CC(CC)C2)=O)CCC2(CC1)CC2CNC(=O)C(CC)CCOC C(=O)(C1=C(c2ccc(Br)s2)N(CC)C(=S)NC1c1c(C)nn(CC)c1C)OCC Cc1cc(C(C)NCc2ccc(OCC3CCC3)cc2)cc(C)c1 N1(C(CC(C(C)C)NC(=O)C=Cc2ccc[nH]2)=O)CCCC2(CCCO2)C1 C1(CCC=O)CCCN(C(=O)C(C2CC2)C2CC2)C1.C(CC)N(CCC)C C1(CN(C(c2ccnc(OC)n2)=O)C)CN(C(c2nccnc2C)=O)CC12CC2 c1(C(N(C(CCNC(C(C=C)C)=O)C)C)=O)cc(C)c2n[nH]cc2c1 C12(NC(CC3(C(=C)F)CCC3)=O)CCC(C)(CC1)OC2.c1(C(=O)N)ccco1 C(CC(C)N=c1cccc(S(=O)(=O)N(C)CCOCCOC)[nH]1)OC c1(CCC(=O)NCC(C)CNC(=O)C(C)CC2CCCC2)cnc2ncccn12 c1(C(N(C2CCN(C(=O)COCC3CCC3)C2)C)=O)ccc(O)c(F)c1F c1(OC)cc(C(N2CC(C)(NC(=O)CCc3ccncn3)C2)=O)n(C)n1 CCCCC(CNC(C1(OC)CC1)=O)NC(c1ccnc(N)c1)=O.C1CCCC1 c1(CN2CCCN(C(=O)C3=CC4CCC3C4)CC2)ncccc1[N+](=O)[O-] C1(CNC(C2CCC(=C)CC2)=O)CC2(CCC2)CN1C(=O)C1=CCCCO1 C1(CC)CC(CC(=O)NC2CCC(NC(=O)Cc3n[nH]c(C)n3)CC2)CCO1 c1(CC)c(C(N2CCC(N(C)C(c3ccc(N)cn3)=O)C2)=O)csc1C c1(OC)c(C)cc(C(=O)NC2CC2NC(c2ccn(C)c2)=O)cc1C Cn1ncc2c1CCCC2C(=O)NC1CCNC(=O)CC1 N1(C(C=CC=CCC)=O)CC2CC(C(N3CCCCC3)=O)(C2)C1.N(C)(C)C C1(C(=O)NC2CC(NC(C3(CSC)CCC3)=O)C2)CCCC12CC2 CCCC(C)(O)CC(=O)NN1CCCC1C(N1CCCC1CNC(C)=O)=O C1(NC(CCC2CCN(C(C3CC3C(F)F)=O)CC2)=O)CCCC1C1CC1 C1(NC(=O)NC2(CN)CC2)CCc2nn(CCO)cc2C1 N#Cc1ccc(NC2CC3CN(C(=O)CC4CCCCC4(F)F)CC23)cn1 C=CC(CC)CC(=O)NC(C)(C)C(C)NC(c1sc(CC)nc1C)=O CC(C)(C)C(=O)C(=O)N1CCCC1C1CCCN(C(=O)C2=CCSC2)C1.C(=O)N C1(CCNC(C2C(C)(C)CC2)=O)CCCCN1C(c1n[nH]cc1Br)=O C1(NC(c2cnc(C)n2C)=O)CN(C(=O)C(O)Cc2cnc[nH]2)CC1(C)C Cc1c(Cl)ccc(C(=O)NCC2(NC(=O)Cn3c(C)csc3=O)CC2)c1O C(=O)(C1CCc2c[nH]nc21)N1CCN(C)CC1.CC(C(=O)NC)OCCN(C)C C1(C(N2CCC2)=O)CCCN(CC(F)F)C1.c1(CC(C)C)cc(C(=O)N)n[nH]1.C c1(C(N(C(C)CCNC(c2ccc[nH]2)=O)C)=O)ccc(=N)[nH]n1 C(=O)(C(CCS(C)=O)N(C)C)NCC1N(C(C2CN(C)C2)=O)CCC1 c1(CC(=O)N)c(C)cc(O)cc1C.c1(C(N(CC)CC)=O)cn(C)c(C)n1 CCC(C)(C)C(O)C(=O)N1CCC1CNC(c1nncs1)=O C(=O)(CCCCSC)N(C(CC)CNC(=O)CC1CCCC1O)C CC1(C)COCC(NC(C2CCC=CC2NC(c2ccc(C(N)=O)[nH]2)=O)=O)C1 C12(CC(=O)N)CCC1CN(C(C1CC3(CC3)C1)=O)C2.Cn1nccc1C(O)C Nc1cnc(Cl)cc1C(=O)NCC#CCNC(=O)CC1CCCNC1=O N1(CC(=O)NC23CC(n4cc(-c5cccs5)nn4)C2C3)CCOCC1 C#CCC(O)C(=O)NC(c1nocc1C(=O)NCC(F)CO)C c1(NCC2CCCCN(C)C2)cc(=NCC2SCCS2)[nH]cn1 N1(C(COCCCC)=O)C2CCC1CC(N(C)C(c1cnc(OC)cn1)=O)C2 c1(COC)ccc(C(=O)N)cc1F.C1(CC(N2CCC2)=O)NC(=O)CNC1=O C=CCCC(CC(C)C)C(=O)N1CC2CCCC2(NC(C2CN(C(N)=O)C2)=O)C1 N1(C(CN(CCC)C(c2ccc(O)cc2)=O)=O)CCC2(CCOC2)C1 C(CC(C)C(=O)NC(c1cccnc1)C(=O)NC1CC=CCC1C)=CC Cc1ccc(C(N2CCC(CN(C)C(C3CN(C)CC3C)=O)CC2)=O)c(O)c1 c1(NC(C2C(NC(C(C)Cc3ccccc3)=O)C2)=O)cc2ccccc2[nH]1 Cc1cccc(C2(C(=O)ON)CC(NC(=O)C(c3ccc(I)cc3)C)C2)c1 C(=O)(CC(CNC(=O)CC1OCCCO1)OC)NCCC=C=C CC(C)CC(C)C(=O)NC1CN(C(C2CCCC(=O)CC2)=O)CCC1C c1(C(=O)NCCOCCCNC(C(C(C)O)C)=O)cnc2cnccc2c1 N1(C(C(C)SCC)=O)CCC2C(NC(c3ccc(-c4csc(C)n4)cc3)=O)C12 c1(CC)cc(C(N2CCC(C(C)CNC(C3CCCSC3)=O)CC2)=O)c(C)o1 C1(C(=O)N)CC12CCCC2.CCCCCN(CCC(=O)NC1CC(C)C1)CCC C1(NC(C(C)(F)F)=O)CCCCCN(C(=O)CN2CCCCC2=O)C1 Cc1cc(C(=O)NC23CC(C2)C3)ccc1[N+](=O)[O-].N1(CC=O)CC2CC2C1.N C1(C(N(CCC(C(C)C)NC(c2c(OC)ccnc2)=O)C)=O)Cc2nccn2C1 c1(C(=O)NC2C3CC(NC(CC(C)CN(C)C)=O)CC32)occ2c1CCCC2 C(=O)(C(CCCC)NC(=O)CC(C)(O)COC)N(CCCCC)CCO c1ccc(C=CC(=O)NC)o1.c1(C=O)cc(C)n(C2CC2)n1.C1CC1.CC c1(C(N2CCC(N=[N+]=[N-])C2)=O)ccc(Cl)c(Br)c1N N1(C(CNS(CCCC)(=O)=O)=O)CC2CCC2(CC)C1.C(=O)C(F)(F)C(F)F.N Cc1ccc(O)c(C(=O)NCC2CCCC2C(=O)N)c1.C1CCN(C(C)C)C1 CCCN(OC)C(=O)C1COCCC1NC(=O)CCc1cccnc1 c1(C(N2CC(CC(C)NC(C3(C)CC=CCO3)=O)C2)=O)cnn2cccc(Cl)c12 c1(OC(C)C(=O)OC)cc(C#N)ccc1Oc1cc(F)ccc1N N1(C(C(C)OCCC=C)=O)CCN(C(c2cc(F)ccc2C)=O)CC12CC2 C12(CNC(C(c3n(C)ccc3)=O)=O)CC(CCO1)N(C(=O)CC1CCC1)C2 c1(OC)ccc(C(=O)C(=O)NC(CNC(=O)C#CC(C)C)C2CC2)cc1Cl CC1CCn2c(C(=O)NCCCOCC)cnc2C1.C1(C=O)CC(C)(C)CO1.N C(=O)C1=C(Cl)CCOC1.C1(NC(=O)CNC(C2CCC2)=O)CCC(C)C1.N C(=O)(CCC(F)(F)C(F)(F)F)NC1CN(C(C(C)O)=O)CC1O N1(C(c2[nH]cc(CC)c2)=O)CC2CCC(C1)N(C(c1cncc(C(C)=O)c1)=O)C2 Cc1cc(CNCC(C)NC(=O)OCc2ccccc2)c(C)[nH]1 N1(C(CCCC)=O)CCOCC1.C1C(C)(C)OCC(=O)N1.C1C(=O)N1 C(=O)(CS(=O)(=O)C1CCCC1)N1CCC(NC(c2c(C)csc2)=O)CC(C)(C)C1 C(=O)(C(O)CC1CCCC1)N1CC(OCC(=O)NCC(COC)O)C1 N1(C(C(CCC2CCC2)NC(c2c(C)snc2)=O)=O)CC2(C)CCC2(C)C1 C=Cc1cncc(-c2ccc(OC3CCCC3)cc2)c1 c1(C(=O)OC)c[nH]ccc1=NC1CC2CN(C(c3cn(C4CCC4)nn3)=O)CC12 c1(C(=O)NCC(CNC(C(C)(C)OC)=O)F)coc(=O)c2ccccc12 CCCC(O)C(=O)N(C(CC)CC(=O)NCC#CC(F)(F)F)C N1(C(CSCCN(C)C)=O)CCCC(C(=O)N(C)Cc2ccsc2)C1 c1(C(=O)NC2(C)CN(C(c3cc(CC)[nH]n3)=O)C2)ccc(C2CC2)c(C)c1 Cc1ccc2nsnc2c1C(=O)NCC1CN(C(c2coc(CO)c2)=O)CC1C N1(C(c2cc(Cl)c(Cl)c(Cl)c2)C(=O)NCCOC)CCc2cc(Cl)ccc2C1C c1(CC)c[nH]nc1C(=O)N.C1(CC)CNC(=O)C1.C1(CC=O)CCC1.C1CC1 c1(C=O)cn(C(F)F)c(C)n1.C1(OC)CC(C(=O)NCC2CC2)C1.C CCCCCC(O)C(=O)N(C1C2CN(C(C3C4CCC3(C)C4(C)C)=O)CC12)C Cc1cc(C(=O)NC2(CNC(C3CCC4(CCC4)C3)=O)CCOC2)c(C)cn1 C12(CC(=O)N(C)CC)CCC1CN(C(=O)C#CC(C)(C)O)C2 C1(NC(C2(C)CCCCC2)=O)CC2CCC1N(c1nnc(C(F)F)o1)C2 N1(C(C2N(C(C(c3cn(C)nc3)O)=O)CCCC2)=O)CCOC2(CC2)C1 N1(C(c2c(NC)cnnc2)=O)CCCC12CCN(C(=O)C(C)(C)COC)C2 C1(C(N2CC=CC2)=O)Cc2c(F)cccc2C(=O)O1.C(CC)(C(=O)NC)=CC C=CC(C)(C)CC(=O)N1CCCC(N2CCN(CCC(C)F)CC2=O)C1 C(=O)(C(C)(CC)C(F)F)N1CC2(C1)C(=O)N2.c1(C(=O)OC)sccc1SC C1(C(F)(F)F)(C=O)CC(C)(C)C1.N1CCOC(C2CNC2)C1.C1(CC)CCCO1 c1(C(=O)NCCOCC(=O)NCC2C=CCCC2)cccc2cncn12 C12(COC)CCN(C1)C2=O.C1CCCN1C(N)=O.C(=O)(C)N.C1CCC1 C1(CNC(c2c(C)nc[nH]2)=O)C(C2CC2)CCN1C(=O)C(c1ccccc1Cl)C Oc1c(-c2ccnc(O)c2-c2nccn2C2CC3CCC2C3)ccc2ccccc12 N1(C(c2ncc(Cl)cc2Cl)=O)CCC(C2CN(Cc3cc(O)ccc3Cl)C2)CC1 C1(C(=O)NCC(C)(C)OCC)CCCN(C(c2ccc(OC)o2)=O)C1 c1(C(C(=O)NCCCN(C(=O)CC(C)N(C)C)CC)O)ccccc1F c1(C(N(CCCC)C)=O)ccc(S(N)(=O)=O)s1.C=CC(C(=O)N)c1ccccc1 C1(F)(CNC(C2CC(CC(F)F)C2)=O)CCN(C(C2CC(O)C2)=O)C1 C#CCC(C(=O)N(CCC)OC)NC(=O)C(C)(O)CCN(C)C CCC(CCC(=O)NC(CCN(C)C)C(=O)NCc1oc(C)nc1C)OC n1(CCCC)ncc(C(=O)NCC#CCNC(c2cccs2)=O)c1C.C1CC1.C CCC(CC(=O)N1CC(C(N2CCN(C)C(C)C2)=O)C2(CC2)C1)C(F)F Cc1cccnc1C(=O)N(C1CCN(C(c2cccnc2C(F)F)=O)C1)CCO N1(C(CNC(c2onc(CC)n2)=O)=O)CCCC(C)C1 C(=O)(C(O)CNC(=O)C(CC1CCC1)NC(=O)Cc1cnnn1C)NC C1(NC(c2cc(CC)c(C)cc2)=O)CN(C(=O)C(N)=O)CC1C1CC1 C1(CCC(=O)OC)CCCN(C(C)=O)C1.C1C(O)CN1CC.C(C)(C)C CC1CC(NC(=O)C(=O)Cc2cccs2)CN1C(=O)C(C)C1CCCO1 C#CCCN=C(NCC(Cc1ccccc1)CO)NCC1CCCO1 Cc1cc(C#N)c(O)nc1C(=O)NC1CCCC12CCNCC2 CCCC(C#N)C(=O)NCC(C)C1CC1.C1(C=O)CC(CC=O)C1.C(C)(C)C C1(CN(C)C)CCCN1C(c1cc(CNC(=O)CC)cs1)=O.CC(N)=O.S C(=O)(C(CNC(C1CCC(=O)C1)=O)C(C)(C)C)NC1(CCC)CCNC1=O Cc1cc(CC(=O)NCCCCCNC(C2(C(C)C)CC2)=O)cs1 C1(C2CCN(C(=O)C(C)(C)OC)C2)(NC(C(CC)c2ccccc2)=O)CC1 C1(C(=O)NC2CC(NC(CC3CC(=C)C3)=O)C(O)C2)CC(=O)N(OC)C1 Cc1nc(C(=O)NCCC2CCCCN2C(=O)Cc2cnoc2)sc1C c1(C(=O)NC(CC)C(=O)NC(C)C(=O)NC(C)(C)C)cc[nH]c2nccc1-2 N1(C(C2C(NC(C3=C(C)OCC3)=O)C2)=O)Cc2ccc(Cl)nc2C1 N1(C(C(C=C=C)C)=O)CC2C3CCC(C2C1)N(C(=O)Cc1ccc(Cl)cn1)C3 C1(NC(=O)CCOCC2CNC2)CCCC(C(F)(F)F)C1 C1(CC(=O)NC(C2CCCCC2)CC)C2CN(C(c3nscc3C)=O)CC12 c1(NC)ccc(S(N)(=O)=O)cc1NC(c1ccc2c(F)cccc2c1)=O C1(C(=O)N)CCS(=O)(=O)C1.c1(C(N(CCC)C)=O)conc1C1(C)COC1 C(=O)(CCCC(F)(F)CO)NC12C(CN(C(C(C)CC(F)F)=O)C1)C2 C1(Cn2cc(C(CSCC)C)nn2)CC(F)(F)CN1C(=O)CC1(C)CC1 C1(c2cccc(F)c2)(NC(c2ccsc2)=O)CCN(C(=O)CC2C=CCCC2)C1 c1(C(=O)N)cc(C)c(C)c(C)c1.C1(NC(C(C)(C)OCC)=O)CCCCC1 C1(C(=O)NCC2CC(CN(C)C)C2)(NC(=O)C)CCSC1.c1ccsc1 C1(NC(CCCC2C(C)C2)=O)CCC(NC(c2nc(C(C)(C)C)no2)=O)CC1 c1(CC(=O)NCC(CO)NC(COC(C)=O)=O)cc(C2CC2)nn1C C1(NC(C=CCOC)=O)CCN(C(=O)Cc2cccc(C(C)(C)C)c2)CC1 Cc1cc(C(=O)NC(C2CN(C(C3CC3(C)C)=O)CCO2)C)c2cnccc2c1 C1(NC(C2CC(C)(CC)C2)=O)CCOC12CCN(C(=O)C1=NNC(=O)C1)CC2 Cc1cc(C(=O)NC(C)CNC(=O)Cc2cnco2)c2c(n1)CCCC2 CCCCCCC(C)C(=O)NCC=C1CCN(C(C2CCOC2)=O)CC1 c1(C=O)ccc(-n2ccnc2)cc1.C(CC1CC1)(C(=O)N(CC(O)C)C)OC.N c1(C=O)cnn2c(=O)cc[nH]c12.C1(C(=O)N)(COC)CC1(F)F.C1CCCC1 N1(C(C(C(=C)C)(C)C)=O)CCC2(CCCC2NC(c2cc(C)c(C)nc2O)=O)C1 N1(C(CC#N)=O)CC2(CCCCN2C(c2nc3ccccn3c2Br)=O)C1 S(=O)(=O)(c1ccc(N)c(Br)c1)N1CCCC(C(=O)OCC)(C(C)C)C1 C1(C(C)S)CC(Cc2cn(CCCCCO)nn2)CC(=O)N1.C(=O)C(C)(CC)CO c1(CC(=O)NC(COCC)C(=O)NC(C)C(C)F)ncccc1C C(CCC(=O)N(CC(C)C(=O)NC(CO)C1CCC1)C)OCC CS(=O)(=O)c1nccc(NC2(CNC(C3Cc4ccccc4C3)=O)COC2)n1 c1(COC)nc(NCC2CC2(Cl)Cl)cc(=NC(C)c2nc(O)n[nH]2)[nH]1 c1(OC)cccc2c(=O)c(C(=O)NCC(=O)N(C)C(c3cccnc3)C)c[nH]c12 C(c1cc(Cl)ccc1Cl)=CC(N1CCCC(C(C)NC(=O)Cn2cnnn2)C1)=O CCCC(C(=O)OC)NC(=O)CCn1cc(-c2ccc(OC)nc2)nn1 Cc1ccc(C=CC(=O)N(c2ccc(Br)cc2)Cc2ncc[nH]2)c(C)c1 c1(C(N2CCC2)=O)c(Cl)ccnc1C.c1(COC)nocc1C(=O)NCC.O C1(C(=O)NCC(CNC(C2CCCO2)=O)OC)CC2(C1)CC(F)(F)C2 C1(C(N(CCCO)CC#C)=O)C(C)CCN1C(C1C2CN(C)CC12)=O C1(C(C)NC(c2cc(C)ns2)=O)CCCCN1C(c1cnsc1)=O C1(NC(Cc2ccc(OC)c(Cl)c2)=O)CC2CCC(C1)N2C(C1CC(C)=NO1)=O c1(C(=O)NCC2C(NC(C=C(C)C(F)F)=O)CCC2)nccc2cc[nH]c12 c1(CC)cnoc1C(N1CC(C)(OCC(=O)NCCc2c[nH]nc2O)C1)=O c1(CC(=O)NC2C(C)(NC(C3CC(C)OCC3)=O)CCC2)ccc2ccoc2c1 N1(C(C=CC)=O)CCC2(CCC2)CC1.c1ccc(F)cc1.C(=O)C=CC=O.N c1(C(=O)OC)cc(F)ccc1CC(=O)NC(CN(C(=O)C)C)(CO)CO.S N1(C(C(CO)N(C)C)=O)CC(NC(=O)C)CC(C)(C)C1.C1CCCC1.C(=O)O N1(C(c2c(C)n(C)cn2)=O)CCC(NC(=O)CN2CCOCC2=O)C(F)C1 C1(C)(C=O)CCOCC1.C1(CNC(COCCCOC)=O)C(C)C1(F)F C(c1cnc[nH]1)=C(C(=O)NCC(CC)NC(C1(C)CCCO1)=O)C c1(OC)cccc(C=CC(=O)NCC2CC2)c1.c1cccnc1.C(=O)C.C N1(C(C(C=C)C)=O)CCCCC1CCC(=O)NCCCN(CC(C)C)C N1(C(c2c(C)cc[nH]2)=O)CCN(C(c2n[nH]c3c2CCC3)=O)C(C2CC2)C1 N1(C(C2N(C)C(=O)OC2)=O)CCN(C(=O)CCc2cnoc2)C(CC(F)(F)F)C1 C(=O)(CCCCCCNC(C1CCCC1)=O)NC(C)Cc1nncn1C N1(C(C2N(CC)CCOC2)=O)CC(C)N(C(c2cc3sccc3[nH]2)=O)C(C)C1 c1(CC(=O)NCCN(C(=O)OC(C)(C)C)C2CC2)c(F)cccc1Br c1(-c2c(C(=O)Nc3ccc(C(N(C)C)=O)cc3)n[nH]c2)ccc(S(C)(=O)=O)nc1 C1(CN(C(C)=O)CC)CCCN(C(=O)C=Cc2cnccn2)C1 N1(C(C(C(C)(C)C)O)=O)CCC2(CC1)CN(C(C1OCC1(C)C)=O)CC2CO c1(C(N2CCN(C(Cc3c(C)n[nH]c3)=O)CC2)=O)cc2c(ccn2C)s1 N1(C(C2C(C(C)C)CCC2)=O)CCC(O)C1C(=O)NCC(=O)NC1CCCC1 CC1(C)CC(NC(C2(C#N)CC23CCCC3)=O)CN(C(c2c[nH]c(Br)c2)=O)C1 c1(C(=O)NC(C)C(C)NC(c2ccnn2C2CCCC2)=O)cnc(C(F)F)s1 c1(C(N(CCCCC)CC2CCCCC2)=O)ccc(C)s1 CN1C(=O)CC(C(=O)COC(=O)CCCCc2cccs2)C1=O N1(C(C(C)(C)C)=O)CCC2C(C1)NC(=O)CN2C(=O)COc1ccsc1Cl Cc1cc(CNC(=O)CN2C(=O)CCC2=O)oc1C(N1CC(N=[N+]=[N-])C1)=O C12(CC=O)CCC(CC1)CC2.n1(CC(=O)N(C(C)C)C)cnc([N+](=O)[O-])c1 C(=O)(C(C)(C)C(C)O)NCC1N(C(C2CCN(CCC#C)CC2)=O)CC1 C(=O)(C(C)(C)S(=O)(=O)C1CC1)N1C2CC(CN(C(CC)=O)C2)C1.C=O.CN Cc1c(CC(=O)NC2CC(CNC(=O)CC3CCCC3)C2)oc2ccccc12 C(=O)(C(C)(C)N=[N+]=[N-])NCCCC(CO)NC(CC1CCC(C)CC1)=O c1(C(=O)NCC(C)CC(=O)NCC(C)(O)CCO)cccc2ccnn12 c1(C(C)C)cc(C(=O)N(C(C)C)C)cc(F)c1.N1(CC=O)CCC(C)(C)C1.N Cc1ccc(NC(=O)C(CC(F)F)N(C(=O)CC2CCCCO2)C)c(C)n1 C1(CNC(C2(OC)CCSCC2)=O)CCC12CCC2.C1(O)(CC=O)CCCC1 c1(C=O)cc2c(cn1)NC(=O)CO2.c1(CC)cc(C(=O)NC(C)CC)c(C)o1 C(=O)(CCS(=O)(=O)NC(=O)OC(C)(C)C)NC1C(SCC)CCCC1 C1(C=O)CCS(=O)(=O)C12CCC2.C1C2CN(C(=O)C=CC3CCCC3)CC12.N N1(C(C2CC3(CCC3)C2)=O)CC2CCC(C1)N2CC1CCS(=O)(=O)CC1 C1(C(=O)NC2CN(C(C(C)O)=O)C2)CNC(=O)CC12CCOC2 C12(N(C)C)CCC(C(=O)NC3CCC(NC(c4nncs4)=O)C3)(CC1)CC2 C1(C)(NC(C(C)OC2CCCCC2)=O)CCN(c2cc(F)ncn2)C1 c1(CC)n[nH]c(=NCc2ccc(CNC(=O)CO)c(F)c2)o1.c1ccccc1 N1(C(C2N(C(COCC(=O)OC)=O)CC=C2)=O)CCCC(CF)C1 C=CCC(CNC(=O)C(C)NC(C)=O)C(=O)NCC(C)(O)C1CCC1 C1(CNC(C2(SC)CCC2)=O)C(C)CCCN1C(=O)C.CCN(C)C.S CCCCC(CNC(=O)CCCCc1cnn[nH]1)NC(C12CC(CC)(CO1)C2)=O c1(OC)ccc(C(=O)NCC2CCCCN2C(=O)C(F)F)c2c1CCCC2 N1(C(c2n(CC)nc(CN)c2)=O)CCCC(N)(CO)C1 C1(NC(C(C)OCC=C)=O)C=CCN(C(=O)C(c2cncn2C)=O)C1 C(=O)(C1=C(CF)N(CC2CCCO2)C(=O)NC1c1cc(C)n(C)c1C)OC Cc1ccc(C(=O)N(CCCCCC(=O)N2CCC(F)(CO)C2)C)c(C)c1 C1CCN(C(C2(C)CCCN2C(C)=O)=O)C1.c1(CC=O)cncnc1.COC N1(C(C2CCC(C)O2)=O)CCCC2(CNC(c3ccnn3C)=O)CCCC12 C(CCCCC(=O)N(CC(CC)NC(C1CCC1c1nc[nH]n1)=O)C)OCC CCS(=O)(=O)C1CCN(C(c2nc(Br)sc2C)C(=O)NCCC#N)C1 c1(C(=O)NCC(C)CN(C(=O)C(C)n2cccn2)C)cnn2c(Cl)cccc12 N1(C(C(COC)C)=O)CC2CN(C(=O)Cn3c(C)ccc3C)CC2C1 C1(NC(CC(CC)SC)=O)CCN(C(c2cnc(C3CC3)nc2)=O)CC1F N1(CC(N2CC(C(C)NC(C)=O)OCC2)=O)C(=O)C(=O)N(C)C1=O N1(c2c(C)c(N3CCC(c4ncc[nH]4)C3)ncn2)CC(O)CC2(CCCC2)C1 CC1(O)CCC(C(=O)NC2CCOC(C(N3CCC(CO)C(O)C3)=O)C2)CC1 CCC(C)(C)CCCC(=O)NCC(CC1CC1)C(=O)NCC1CC2CCC1O2 c1(C(=O)NCCN(C(C2CCc3ccnn3C2)=O)CC)ccc2c(c1)nnn2C c1(CC)cc(N2CCCCC2CCNC(C2CCC(C)(C)O2)=O)ncn1 C1(CNc2cc(N(C(c3ccc(Cl)cc3)C)C)ncn2)COC2(CCCCC2)O1 Cc1cc(C)c(C(=O)NCCN(CCc2ccccc2)C(c2snnc2C)=O)s1 C1(C(N(C(CN(C(Cc2c(C)ccs2)=O)C)C)C)=O)CN2CCN1C(C)C2 C1(C(N(CCCF)CC)=O)C2CCN(C(c3nc(Cl)cs3)=O)CC12 N1(C(C(C=C)CC)=O)CC(F)(F)CC1C(=O)NC1C=CCCC1 C(C(C(=O)N(C1CN(C2CC2)C1)C)NC(C1CC1(Cl)Cl)=O)OCC C1(N(c2cccc(C(N)=O)c2)C(C(C)NC(C=C)=O)=O)CCNCC12CC2 C1(CC)COCCOC1.CC(C)C(=O)N(CC(=O)NCC1CC(C(=O)N)C1)C N1(C(C(C2CCN(C(C3(n4cccn4)CC3)=O)CC2)C)=O)CCC(CO)C(O)C1 CC(C)CC(C)CNC(c1ncccc1Cl)=O.C12(C=O)CCCC1(C(N)=O)C2.N C1(C(N2CC(NC(c3cc(Cl)ccn3)=O)C(O)C2)=O)CC2CCCC(C1)C2 C1(NC(C2(OCC)CCCC2)=O)CCN(Cc2cn(CC)nn2)CC1 C(CC(C)C(=O)NCC1OCCC1C(=O)N(CCCC(C)O)C)=CCC c1ccc(S(C)(=O)=O)cn1.c1(C(CN)N(C(=O)Cc2ccco2)C)ccccc1 Cc1nnc(C2CCCN2CC(C)CC2CCCC2)o1 C1(OC)CCN(C(=O)CC(C)NC(=O)Cn2ccc(C)n2)CC1(C)C Cc1cc(C(N2CCC(NC(C3CC4CC4CC3C)=O)C2(C)C)=O)nc(O)n1 C=CCCN=C(NCc1cc(C)ccn1)NC1CCOC(CC(C)C)C1 N1(C(c2cc(C)ns2)=O)CCCN(C(c2ccc(C)c(C(F)(F)F)c2)=O)CC1C c1(C(N2CC3CCC2C3)=O)cc2c(s1)CCS(=O)(=O)C2.O=CC=CC1CC1 C=CC(C)(CCOC)C(=O)N1CCC(N(C(=O)CN2CCCCC2)CCC)CC1 c1(OCC)cc(C(=O)NC(COC)CNC(=O)C=C(C)C)on1 c1(C2(OC)COC2)ccc(C(=O)NC2(c3ccccc3)CCNCC2)cc1 c1(C(N(CCCNC(C2(SCC)CC2)=O)C)=O)ccc2cnnc(O)c2c1 C(CCC(C)(C)C)N(C(=O)CC(C)CN(C)C)C.C(C(F)(F)F)=CC=O.N C1(C2CCN(C(C3(C)CCOC3)=O)C2)(NC(c2c(OC)c(Cl)sc2)=O)CC1 c1(CC(=O)NC(C(C)NC(c2ccc(SC)cc2)=O)C)cc(F)ccc1Cl Cc1[nH]nc2c1CC(C(=O)NCC(CO)NC(c1ccsn1)=O)CC2 Cc1nc2cc(-c3csc(NCc4ccc([N+](=O)[O-])cc4)c3)ccc2s1 c1(C=O)c([N+](=O)[O-])cnn1C.N1(CC)CCOCC1CC(=O)NCC(C)(O)C.N Cc1onc(-c2ccccc2)c1C(=O)NCCCN(C)C(C1C2CCC(=O)C12)=O N1(C(CCS(N)(=O)=O)=O)CCC2CC2(C(=O)NCc2ccc(CO)o2)CC1 c1(CC(N2CC(C)(NC(C3CC4CC4C3)=O)C2)=O)c[nH]c2cccc(F)c12 N1(C(C2C(C)C2)=O)Cc2ccccc2C(CNC(=O)C2Cc3ccc(Cl)cc32)C1 c1(CC(N2CCC(NCc3cccc(F)c3)CC2)=O)ccccc1C(=O)O Fc1cc(F)c(CCNC2(COCSc3ccccc3)CC2)c(F)c1 C1(CC(=O)N(C2CC(NC(C3C4CCCOC34)=O)C2)C)CCCNC(=O)C1 C1(C(=O)Nc2csnc2C2CC2)CCC(n2cc(CCCCO)nn2)C1 C(C(CC1CC1)C=O)NC(C(C)(C)OC(C)C)=O.C1CCC1.C(C)=O.N N1(C(=O)C=Cc2ccc[nH]2)CCCC(N(C(=O)C(C2CCOCC2)F)CCF)C1 C1(CC)(CO)CCCN(C(=O)C(=O)N2CC(C(F)C=O)C2)C1.CC.C1CC1.N C(=O)(CC(C(F)(F)F)NC(=O)C1=C(Cl)CCC1)N1CCCC(C)C1 n1(CC(N2C3C(NC(C(CC=CC)C)=O)C(C3)C2)=O)cc([N+](=O)[O-])c(C)n1 C1CCCC(=O)N1.C1(CC#C)(C(=O)N(CC(=O)NCCOC)C)CCOC1 CCN=c1[nH]c(C)c(C(=O)NCCOCCN(C(=O)Cn2ncnn2)C)s1 C1(NC(c2c(CC)nns2)=O)CC2C(NC(=O)CCCn3cccn3)C2C1 C(C(C)(C)CC(=O)NCC1CCC1NC(c1c(O)cccc1Cl)=O)N(C)C C1(C=O)C(C#N)C1(C)C.C1(CNC(CSCCOC)=O)CC(F)C1.C N1(C(C(C)OCCOCC)=O)CCOCC(C)C1.c1(C=O)sc(C)cc1C.N c1(NC(CNC(C(C(C)C)N2CCCC2=O)=O)C2CCC2)cccc(F)c1C#N C1(C)(CC)C=C(C(=O)N2CC(NC(c3ccc(F)cn3)=O)CC(F)C2)C1 N1(C(Cc2cc(C)[nH]n2)=O)CC(NC(=O)CCc2c(F)cccc2Cl)CC(C)C1 Cn1c(C(=O)NC23CC(C)(C2)C3)cc(Cl)c1Cl.c1(C=O)cnc2sccn12.N c1(-c2ccc(C(=O)OC)s2)cc(=O)n2cccc(OC)c2n1.C12CCN(CC1)C2 c1(C(N2CC(CNC(C(C(C)C)NC=O)=O)OCCC2)=O)cccc2nc[nH]c12 c1(C(N2CCCC(NC(C3CC(n4ccnc4)C3)=O)C2)=O)ncc(Cl)cc1Cl O=C1CCC(C2(C(=O)NC(CNC(=O)Cc3cnoc3)CO)CCC2)CN1 Cc1cnc2n1C(C(=O)NC1CC(NC(c3ccccc3C(C)C)=O)C1)CCC2 C1(C(N2C(C(=O)NC)CC2)=O)C(C2CC2)CCN1C(=O)CCCCC#N C(=O)(CCCC(=O)N1CC(CC(=O)NC2CCCCC2C#N)CC1(C)C)OCC c1(NC(CC2(C)CN(C(C3CN(C)C(=O)C3)=O)C2)=O)c(O)cccc1Br C1(CNC(CC2(C)OCCO2)=O)CCN(C(=O)Cc2csnn2)C1(C)C C#Cc1ccc(C(N2CC(NC(=O)Cc3ccc(C)cc3F)CC(F)C2)=O)nc1 c1(OC)ccnc(F)c1C(=O)NCC(CO)NC(=O)CCc1cncc(O)c1 C(CS(=O)(=O)CC(=O)NC1CC(C(F)F)(NC(C2CCCSC2C)=O)C1)OC c1(C=O)cc2c(C)nn(C)c2s1.CCCCNC(C1(NC(C)C)CC1)=O.N CC(C)C(C)C(=O)N1CC2CC1C2CNC(=O)C(C)(C)Cc1cnn[nH]1 C=C(Cl)CC(C(=O)N1CC(O)CC1CO)NC(C1CCC(C)(C)OC1)=O c1(C(=O)NCCC(C)N(C)C(C2CC(C)N(C)C2)=O)ccnc(N(C)C)c1 c1(C(=O)N)cc2c(s1)CN(C)CC2.c1(C(C)=O)ccc(C(=O)NC(C)CC)[nH]1 C1(C(=O)NC(c2cnc(C)s2)C)CCCN(CC2CCCCO2)C1 C1(CCOC)(NC(=O)CC(=O)N(C)C)CCN(C(c2ccc(F)nc2)=O)C1 C(=O)(C(C)(C)C(F)F)N1CCC(F)(CNC(c2cnn(C(CC)C)c2C)=O)C1 C1(C(=O)NCC(CCC)NC(=O)C2=CCCOCC2)Cc2nc(C)cn2C1 C#CCC(CC(=O)NC1(c2noc(C)n2)CC1)NC(=O)C(=O)C(C)CC CCP1(=O)CCN(C(=O)C(=O)N2CC(n3cc(Br)nn3)C2)CC1 N1(C(CCOC(CC(C)C)C)=O)CC2CCN(C(c3cn4c(n3)SCC4)=O)C2C1 c1(C(N2CCN(C(c3c(C)c(Cl)ccc3)=O)C(C)C2)=O)ccc(C#N)c(Cl)c1 c1(CCCC)nc(Cc2ccncc2)nn1-c1ccc(Cl)cc1 CC1CCCc2cc(C(=O)NCC3CC(F)CN3C(C3CCCC(=O)O3)=O)nn21 Cc1cc(C(=O)N(C(CNC(c2cncc(N(C)C)c2)=O)C2CC2)C)nnc1C c1(N(C2(c3cccc(Br)c3)CCC2)C)ncnc(C(=O)O)c1F O=C(NNS(=O)(=O)C1CCOC1C1CC(F)(F)C1)C1OCCC1C(F)(F)F c1(C(=O)NCC(CNC(c2c(C)ncc(C)c2)=O)C)ccn2c1CCCC2 C=CC1CCCN1C(CC1CCC1)C(=O)NCCNC(=O)O.C(C)(C)C c1(C(C#N)N(C(C)COC)CCOCC)ccc(Cl)c(Cl)c1 C(=O)(CCCC(=O)C1CC1)N.C1CC12CCC2.CN1CC(O)(CNC=O)C1 O=C1CCCCC(C(=O)NC2CC(C(N3CCOC(C#N)C3)=O)C2)N1 C1(C(=O)OC)C(F)(F)C12CC(NC(=O)NC(C(N)=O)C1CCCC1)C2 CCC(C)C(C)C(=O)N1CCC(CCNC(=O)Cc2cc(OC)no2)CC1 C1CC2CCC(C1)N2C(=O)CC1COC(C)(C)C1.Cc1cnc(C(=O)N)c(C)c1 C=CC(C)(O)C(=O)N1CC(OC2CCN(C(c3ccccc3C)=O)CC2)C1 C(=O)(C(F)CCC(C)(C)C)N1C(C)CC(CNC(CCCCN(C(C)C)C)=O)C1 C1(NC(C2CCCN(CCC)C2)=O)CCN(C(c2csc(CO)n2)=O)CC1C C1(CNC(CCCOCC=C)=O)(CO)CC=CCC1.C(C)(C)C CCC(CC(=O)NCC(C(=O)N(CC(O)COC)C)C(C)(C)C)CC(C)C N1(C(Cc2nc(C)sc2)=O)CCC2(C1)CN(C(=O)C(C)(C)C(F)F)CC(C)O2 c1(C(N2CCC(C)(C(=O)NC3(C)CC(C)(C)C3)C2)=O)ccc(F)cc1O c1(C(C=O)O)ccc(C#N)cc1.C1(N(C)C)(C(=O)NCCC2CC2)CCC1.C c1(CNCC2OCCN(C(c3c(C)ccc(Br)c3)=O)C2)ccc([N+](=O)[O-])c(O)c1 C1(NC(CC(C)SC)=O)CC2CCC1CC2NC(c1cc(C)c(C)[nH]1)=O c1(OC)ccc(C)c(C(=O)N(C2CCN(C(C3(C)CCCO3)=O)C2)CCO)n1 CCCC(C(=O)NC(CNC(=O)C(O)C1CCC1)CC)c1ccc(Cl)cc1 c1(C(N2CC3C(CNC(C(=O)NCC)=O)(C3)C2)=O)cnc2cc[nH]c2c1 N1(c2ccnc(OC)n2)CCC=C(c2cnc(Nc3cnncc3C)c(C)c2)C1 c1(C(CC)C)ccc(C#N)c(NC2CCCN(C(=O)CNC(C)=O)C2)n1 N=c1cc(C(=O)NCC(CNC(c2ccc[nH]2)=O)C(F)(F)F)c(Br)c[nH]1 N1(C(C2(C)CC2)=O)CCC2(CCC2)C(NC(=O)C(Cc2ccccc2F)OC)C1 N1(C(CNC(=O)NC)=O)CCCC12CCCCCC2.C1(C(=O)N)CC(C(F)F)C1 CC1=C(C(=O)NC2CC(CNC(=O)C=CBr)C23CCC3)SCCO1 C1(NC(c2snc(Cl)c2Cl)=O)CC12CCN(C(=O)Cn1cccc1)CC2 C1(C=C)(C=O)CCOCC1.C1(CC)(CNC(C2CC2)=O)CCC(=O)N1.C C1(CC=C)(NC(C2ON=C(C)C2C)=O)CCN(Cc2cccs2)C1 C(=O)(C(CC(C)C)n1ccnc1)N(CCC(C(C)C)NC(CCSCCC)=O)C CCCCC(CNC(C1CCC(C)CC1)=O)NC(C1CCC(C)(CC)O1)=O N1(C(c2scc(COC)c2)=O)CC(O)CC1CNC(=O)Cc1ncoc1C CN1CC(N(C(=O)C(C)(CO)NC(c2cnncc2O)=O)C)CCC1=O C1(C(=O)NC2CCCC(NC(=O)CC3CC3)C2)CCn2c(O)nnc2C1 C(=O)CCCC.CCC(CNC(c1ccco1)=O)NC(=O)C(C)NC(N)=O CC1=NOC(=O)C1CCC(N1CCC(CNC(c2ccc(Cl)cc2)=O)C1)=O c1(NC(C2CSC2)C)ccc(S(=O)(=O)NCC2(C3=CCOCC3)CC2)cc1Br Cc1c(C(=O)NCC(C)(C2CC2)NC(C2CC2[N+](=O)[O-])=O)cccc1[N+](=O)[O-] C(=O)(C(CC)(CC)OC)NCC(=O)NCC(C(CC)C)O C12(NC(c3cnc(C)[nH]3)=O)CCN(C(=O)CN3CC=CC3)CC1C2 CCC(CC(=O)N1CCCC(OC)C1)N(C)C(c1occc1C(=O)OC)=O CC1(C)OCCOC1C(=O)NCCC(O)CNC(c1coc2c1COC2)=O Cc1ccc2nsnc2c1C(N1CCC(C)(C)C(CNC(c2cnsc2)=O)C1)=O Cc1csc(=NCC(=O)N2CCC(Cc3cn(C4CC(F)C(=O)N4)nn3)C2)[nH]1 c1(C(=O)NC2CCN(C(c3cc(Cl)cs3)=O)C2)cc2cncn2c(O)n1 Cc1cn(C)nc1C(=O)N(CC)C(C)C.C1(C=O)CCCC1c1nncn1C.N c1(OC)cc(C(N2CC(C)(NC(=O)C(C)C#N)C2)=O)ncc1Br C1(CNC(C2(CC)CCOC2)=O)CCCCN1C(=O)CCCOC(C)=O C(C(C(=O)O)c1ccccc1)NCC(C)Cn1ccc(C(F)(F)F)n1 c1(C(=O)NCCCN(C(=O)CC2CCNC2=O)CC)cc2ccncc2s1 C1(C(N(CCCCNC(=O)CC2CC=CCC2)C)=O)CC(C)(C)OC1(C)C N1(C(CCC#C)=O)CCC2(CCCN(C(c3scnc3C(F)F)=O)C2)C1 Cc1cnccc1-c1ccc(C(=O)N(CC(F)(F)F)CC2CCCO2)s1 c1(C(=O)N)cc2n(n1)CCOC2.C1(C(=O)OC)(C(=O)NCCCC)CCOCC1 c1(C(=O)NC(CC)CNC(=O)CNC(c2cncs2)=O)cc(C)nn1C Cn1nccc1C(=O)NC1CC(n2cc(CNC(C3CCCC3)=O)nn2)C1 C1(CC(=O)N(C(C)C=O)C2CC2)(CC)CCC1.CC(C)(C)C1(O)CCC1.N [SH](=O)(=O)c1cnn(C)c1.C=C(C)CC.C(C1CCC1)=CC(=O)N.C(=O)C c1(CNC(CSCCC)=O)ccc2c(c1)CCN(C(C1CC13CC3)=O)C2 N1(C(C=C(CCC)C)=O)CC2(CCC2NC(c2oc(C(F)(F)F)nc2C)=O)C1 c1(CC)c(N2CCC(NC(C3CCCOCC3)=O)C2)nc(C2CCC2)nc1Cl c1(C2(C(N(CC)CC)=O)CC2)ccc2c(c1)OCO2.C1(C=O)CC12CC2.N CC1(C)CN(C(=O)Cn2cncn2)CC1NC(c1cc(C2CC2)nc(O)c1)=O C(=O)(CCC(=O)NC1CCCC1)OCC.c1(C2(C=O)CC2)cccc(C)c1.N c1(OC)ccc2c(c1)N(C(=O)NCC1CNC(=O)O1)CC2C c1(C(N2CCC(n3cc(CC(=O)OC)nn3)CC2)=O)ccnc2c(Br)cccc12 N1(C(Cc2ccc(NC(C)=O)cc2)=O)CC2CN(C(=O)Cc3ccccc3F)CC12 C1(C2CCN(C(=O)C(O)C3CCC3)CC2)(NC(C2CCCCCS2(=O)=O)=O)CC1 C12(CNC(CN(C)C3CC3)=O)CCC1CCN2C(=O)Cn1cnnn1 N1(C(CCCOCC=C)=O)CC(NC(C2(c3ccccc3)CC2(C)C)=O)CC1C c1(CC=C)cccc(C(=O)NC2CN(C(=O)C(C3CCC3)OCC)CC2)c1 c1(C(=O)NC(C(=O)Nc2cn(C)nc2)CC2CCOCC2)nccc2[nH]ccc12 CCC(F)(F)CC(=O)NC1CC2CC1N(C(c1ccnc(OC)c1F)=O)C2 c1(OC)cc(C)c(C(=O)NC2CCN(C(=O)C(C#N)C(C)C)C23CC3)cc1Br C1(OC(C)=O)CCN(C(=O)C(C2CCN(C(c3ccc(C#N)o3)=O)C2)F)CC1 C1(C(N2CCC(CN(C(=O)C[SH](=O)=O)CC)CC2)=O)COC2(CCC2)C1.N C12(CCCC1)C(=O)N2.C1(C(=O)NC(c2nccs2)C)CCSCC1 c1(C(N2CCCC(CNC(CCCOC)=O)C2)=O)ccc2oc(O)nc2c1 N1(C(C(=O)NC)CCC2CC=CCC2)CCCC2(CC1)CNC(=O)C2 c1(C(C(=O)O)NC(C=CCCC(C)C)=O)ccc(OC(C)C)cc1 c1(OC)ccc2occ(C(N3CCN(C(=O)C=C4CC4)CCC3C)=O)c2c1 c1(C(N2C(C(=O)Nc3cnc(C)s3)CC(O)C2)=O)n[nH]c2ccccc12 N1(C(C2CCCOC2)C(=O)NCC=C)CCCCC1C1CNC(=O)C1 c1(C(=O)NC(CNC(C2C(C=C)C2)=O)C(C)C)c(Br)c(C2CC2)nn1C N1(C(c2cnn(CC)c2C)=O)CCCN(C(C23CCC(C2)C(C)(C)O3)=O)CC1C c1(C(N2CCCC2)=O)cn(C)ccc1=O.c1(C(N(C)C)=O)nccnc1C(N)=O C(=O)(C(C)CC(C)(F)F)N1CC(CCNC(C2OCCN(C(C)C)C2)=O)C1 c1(NC(c2scc(C(=O)Nc3cn(COC)nc3)n2)=O)cncc(O)c1 N1(C(CS(CC)=O)=O)CC2CCC1C2NC(c1ccn(C(C)C)c1C)=O C(=O)(C(C)(C)C(C)(C)C)N1CC(C)C(C)C1.c1(C(=O)N)cnn(CC(F)F)n1 n1(CC)cc(CN(C2CC2)Cc2c[nH]nc2C(F)(F)F)c(C)n1 N1(C(CC(C)SC)=O)CCCC1(C(=O)NC(c1nn[nH]n1)C1CC1)C(C)C N1(C(C2(C)CC(C)C2)=O)CCC(F)C(NC(c2cccc(CC(F)(F)F)c2)=O)C1 C12(NC(C3(C)CCCN(C(c4cnn(C)c(=O)c4)=O)C3)=O)CC3CC(CC1C3)C2 CC1(C)CCN(C(C2CC(O)C2)=O)CC1NC(c1cc2nc[nH]c2cn1)=O c1(C(N2CCC(NC(c3cc(Cl)ncc3Cl)=O)C2)=O)ccc2nc(O)[nH]c2c1 c1(C(=O)NCCCCCCNC(C2C(C)(C)NC(=O)C2)=O)cc2nccnc2[nH]1 S(=O)(=O)(c1cccnc1)NCC(=O)NCCCC.C1(C=O)COC(=O)N1.N C1(NC(C2CC(OC)C2)=O)CCCC(NC(=O)CSc2ccccc2)C1.O Cc1c(C(=O)NCC2CN(C(=O)Cn3cc(Br)cn3)CC2C)nn(C)c1N C1(O)(CC=C)CN(C(C2CCCN2C(=O)C(C)NC(C)(C)CC)=O)C1 N1(C(CCC(=O)OC)=O)CCCC(N(c2cc(SC)nc(SC)n2)C)CC1 CCC(CC)CC(F)C(=O)NC(C(=O)Nc1ccc(SC)nc1)C(C)OC N1(C(c2c(Cl)cnc(CC)n2)=O)CCC2(CCN(C(C3ON=C(C)C3C)=O)C2)C1 c1(C(N2C(C(=O)Nc3n(C)nnc3)CCC2)=O)ccc2[nH]c(=O)ccc2c1 N1(C(C(c2ccc(C)s2)C)=O)CC2(CNC(=O)Cn3cnnc3O)CC1CCO2 C1(CCN(c2c(C)c(N)ncn2)C)Oc2ccccc2NC1=O CC(CNC(c1ccc(C(F)C(F)(F)F)cc1)=O)S(C)(=O)=O N1(C(c2cc(C)n(C)c2)=O)CCCC(C)C1CNC(=O)Cc1nncs1 CCC(C)(C)C(C)CC(=O)N(CCCOCCNC(=O)Cc1ccsc1C)C C1(NC(CCc2cc(C)on2)=O)C2CCC1CN(C(=O)C(C)CC(C)C)C2 c1(NCc2c(-c3c(C)cc(OC(C)C)nc3)ncc(Cl)c2)cccc2nc(O)[nH]c12 C(=O)(C(C)(CO)NC(=O)C(O)CS)N1CC(OCC(=O)OCC)C1 C(=O)(C(CN(C)C)C(C)C)N1C(CC(N2C(COC)C=CCC2)=O)CCC1 CN1CC=C(CC(=O)NC23CC2CN(C(c2cc(C4CC4)on2)=O)C3)CC1 c1(C(=O)NCCO)cncc([N+](=O)[O-])c1.C1CCN(C(=O)Cc2cnc[nH]2)C1 C1(NC(C2CCC(OC)CC2)=O)C2CCCN(CC(=O)NCCOC)C2C1(C)C N1(C(CCC#C)=O)CC2CCC1C(NC(c1ccc(=O)n(CCOC)c1)=O)C2 c1(CC(=O)Nc2ccsc2C(=O)NN2CCC(O)CC2)cc(F)cc(F)c1F C1(CNC(C(CCC)=CCC)=O)C(C)CCCN1C(=O)CO.c1ccccn1 c1(C=O)nnc2ccccn12.C1(CCOC)(C(=O)NC2CC(C)C2)CCC1.N CCCCCCC(C)C(=O)N(CC(O)CN(C)C(c1nc(Br)c[nH]1)=O)C N1(C(c2cn(CCC)nn2)C(=O)NCC2CCOC2)Cc2cc(Cl)c(Cl)cc2C1 Cc1cc(C(N2CC3CC3(C(=O)N(CC(C)(C)O)CC(C)(C)O)C2)=O)nn1C N1(C(C=C(C)C)=O)CCC2(NC(=O)CCC=CBr)CCCCCC12 c1(C(=O)NC2CC(NC(C3C(C)(C)C3(C)C)=O)C23CCC3)snc2ccccc12 c1(CN2C(=O)CC(C(=O)NC(C#C)CC3CCOCC3)C2)c(F)cccc1F C1(F)(C(=O)NC(CC)C(N)=O)CCCN(C(c2cccnc2OC)=O)C1 N1(C(C#CC(C)C)=O)C(C)CC2CN(C(=O)CCF)CC12 O=[N+]([O-])c1cc(Br)ccc1.N12CC3CCC(C1)C3C(=O)OCC2.C1(S)CCCCC1 C(C(C(=O)NCC(c1ccco1)O)N(C)C)NC(C1C(CCOC)C1)=O C12(OC)CCC(C(=O)N)(CC1)C2.C12CC1CN(C(C1CCC(=O)N1)=O)C2.C C(=O)(C1=NOC2COCC12)N1CC(CC=C)(C(N2CC(SC(F)F)C2)=O)C1 c1(C(C)NC(C2C3CC2N(Cc2cnn(C4CC4)c2)C3)=O)ncc(Cl)cc1Cl N1(Cc2c(C(C)C)cccc2)CCC(NC(=O)CC2CCCS2(=O)=O)C(O)C1 C(=O)(C#CC(C)(C)CNC(c1ncc2ccccn12)=O)NC1(C(C)C)CC1 c1(C(=O)NC(C2CCN(C(C3CC(C)(F)C3)=O)CC2)C(C)C)ccnc(S)c1 Cc1cc(C(=O)CCC(=O)NCC2CCN2C(=O)CC(C)(C)F)c(C)s1 C1(C(=O)NC(CC(C)NC(=O)Cc2nccs2)C)CCC=CCC1 C(CCCCCNC(c1cnn(C2CCC2)n1)=O)NC(c1n(C)ccc1)=O Cc1ccc(C=CC(N2CCN(Cc3cccc(I)c3O)C3CC23)=O)cc1 N1(C(CC(CC)C)=O)CCN(C(c2cc(Br)cnc2O)=O)C2(CC2)C1 C1(C(N(C)CCNC(=O)CCc2ccncn2)=O)C2CC2C2CC12 S(=O)(=O)(CCCS(=O)(=O)NCC1CC1C)N1CC(C)(OC)C1 N1(C(C2CCN(CCC)CC2)=O)CC(NC(c2cccc(F)c2O)=O)CC(F)C1 c1(NC(C)C)cccc(C(N2CCC(NC(=O)C)C2)=O)c1.c1cccc(F)c1.S CC(C)C(C(C1CCC1)NC(=O)C1CC1)NC(=O)C(F)=CCCF C1(CNC(c2c(C)onc2)=O)CC2CCC1N(C(c1cnc3ncccn13)=O)C2 C1(CNC(CSCC#C)=O)CN(C(c2cc(-c3ccccc3F)no2)=O)CC1O Cn1ccc2cccc(C(=O)NCC34CCCCC3CN(C(=O)C=CCO)C4)c12 c1(CN2CC3N(C(c4cc(OC)ncc4Br)=O)C(C3)C2)c[nH]c2ccc(Br)cc12 Cc1cc(C(=O)NCC(=O)N(CC(C)N(C)C(c2scnc2Cl)=O)C)cc(C)c1 c1(N(C)C)ccc2c(c1)CN(C(=O)Cc1ccc(Br)s1)CCC2 C(=O)(C(C)(C)CCCNC(C1CCC(O)CC1)=O)NC(C)CC(F)(F)F N1(C(c2c(C)cc(C)nc2Cl)=O)CCN(C(=O)CC2CCC3CC23)CC(C)(F)C1 C1(CC#C)CN(C(c2cnn(C(C)C)n2)=O)CCO1.C1(C(=O)N)CCCCC1C C(=O)(CS(=O)(=O)CCC(F)(F)F)N1CCC(C)(NC(c2cc(C)ncc2C)=O)C1 C(C(C)(C)CN(C(=O)CSS(C)(=O)=O)C)NC(C=CC=CCC)=O C1(C(N2CCC(CC=C)(C(=O)NCC3CCC(C)C3)C2)=O)Cc2nccn2C1 c1(C(=O)NCC2CCC(NC(=O)CCc3nccs3)C2)cccc2[nH]ncc12 C(=O)(C1CCc2c[nH]nc21)NC1(CNC(c2ccc(C)n2C)=O)CCOC1 CS(=O)(=O)c1cc(CN2CC(N3CCN(C(=O)C(Cl)(Cl)Cl)CC3)C2)ccc1F c1(C(=O)NC2C3CN(C(CCCCOCC)=O)C2CC3)cc(Cl)cc(Cl)c1N C1(NC(C(C)(CO)OC)=O)CC2CC1N(C(c1ccc(O)cn1)=O)C2 CC1=C(C(=O)N(C2CN(C(c3cnn(CC(F)(F)F)c3)=O)CC2(C)C)C)CCO1 C=C(C)CCC(=O)NCCCC1CCCN1C(c1nccnc1C)=O c1(C=O)c(C)nn2c1CCCC2.C(C)(C)(C)OC.N1(CC(=O)N)CCC(C)C1 CC(c1cccs1)=CC(N1CC2CC2(CNC(C2CSCCS2)=O)C1)=O C1(C)(C=O)CCOC(C)C1.N1(C(C2(CCOCC)CCC2)=O)CC(F)C1.C N1(c2cc(NC(c3c(Cl)cccc3Cl)C)nc(C)n2)CC2C3C=CC(CC3)C2C1 C1(CC(=O)NC2(C)CC(NC(C(C)CO)=O)C2)COC2(CCC2)CO1 C1(NC(C2CCCCC(=O)C2)=O)CC2CC(C1)N(C(c1cnccn1)=O)C2 C1(NC(C2(CC(C)C)CC2)=O)CN(C(c2ccccc2)=O)CC1F.C1(O)CC1 c1(CCC(=O)NCCC2(NC(C3CC(SC)C3)=O)CC2)ccc(F)cc1 c1(C(N2CCN(C(C(C=CC)O)=O)CC2C)=O)cc2c(cnn2C)nc1C C(C)(C)(CC(C)C)NC(C(CC)OC)=O.c1(C(=O)N)cc(C)c(C(N)=O)cn1 c1(C(=O)NC(C)CC(=O)NCCC(C)N(C)C(C2(Cl)CC2)=O)cc(Cl)ccn1 Cc1cncnc1N(CC(C)NC(=O)CSC(F)F)C CCC(C)(C(=O)N1CCCC(C)(NC(=O)CCc2cc(C)no2)C1)C(N)=O N1(C(CCC=CC)=O)C2CCC1CN(C(=O)C=Cc1cnn(C)c1C)CC2 c1(C(=O)NCc2ccnc(C(=O)NC3CCCC3(F)F)c2)cc(F)cc(F)c1 c1(C(N2CC(O)CC(NC(CCNC(N)=O)=O)C2)=O)cccc2c1CCCC2 c1(C(N(CC(=O)Nc2cccc(OC)c2)CC(C)C)=O)cnn2c1NCC(C)C2 C1(CN(C(=O)Cc2cscn2)C)CN(C(=O)C(F)(F)c2cscn2)CCO1 Cc1nc(O)nc(C)c1C(=O)NC1COCCC1NC(=O)CCS(C)(=O)=O c1(CC(=O)N(C2(CC(=O)NC3CN(C(C)=O)C3)CC2)C)n[nH]c(C)n1 c1(C(N2CC3C(CNC(=O)CO)(C3)C2)=O)ccc2c(c1)OCCCO2 C1(NC(C(n2cc(C)nc2)(C)C)=O)C2CN(C(C3C(Cl)(Cl)C34CC4)=O)CC12 C1(CC=C)(NC(C2CCC(C)O2)=O)CCN(C(C2(COC)CC2)=O)CC1 N1(C(Cc2c(C)nn(C)c2C)=O)CCC(F)(F)C(NS(=O)(=O)C2CC2)C1 c1(NC(C2N(Cc3c(O)cc(C)c(Cl)c3)CC=C2)=O)ccc2c(C)nn(C)c2c1 N1(C(c2cc(C(=O)OC)on2)=O)CCC(C)C(NC(c2nc(C)oc2C)=O)C1 C(c1cncs1)=CCNC(C1CC(c2nn[nH]n2)C1)=O c1(C(=O)NCCCOCCN(C(=O)C(F)C2CCC2)C)cnn2cccnc12 O=C(CCCCc1ccc(Cl)cc1)NCCN(C1CCCC1)C(C1CCSC1)=O C1(C(=O)NC(CCC=C)CO)CN(C(c2nccc(C)c2F)=O)CC(C)O1 N1(C(c2cccc(C)c2)=O)CCC2CN(C(=O)C(O)C(F)F)CC12 C12(CNC(C(CC)SC)=O)CCC(C)(CC1)OC2.c1(C=O)cnc2sccn12.N N1(C(c2ncn(C)c2)=O)CCC(CNC(=O)CSc2ccncc2)C1(C)C c1(CCCC=C)ccc(C(=O)N)cc1.C1C2CC1N(C(C13CCC(C1)C3)=O)C2.C c1(OC)cccc(CN2CC(NC3CCN(C)CC3)CC(F)C2)c1OC c1(C(N2CC(NC(C(COCC)C)=O)C(S)C2)=O)cc(C(F)F)cc(C)c1 c1(NC(C2C(NC(c3c(O)cccc3F)=O)C2)=O)cc(Br)cnc1I c1(CN2CC(CNC(C3(C)CC3)=O)C2)ccc([N+](=O)[O-])cc1 C1(CCNC(=O)Nc2ccc(OCC3CCCO3)cc2)CC12CCOCC2 C1(O)(CNC(C=C(CCC)C)=O)CCCN(C(=O)C(c2cccc(O)c2)(C)C)C1 CCC(C)C(C(=O)N1CC(F)(CO)C1)NC(=O)C=Cc1cncn1C C(C(C)NC(c1ccnc(-n2cccn2)c1)=O)(C(C)C)NC(c1c(C)n[nH]c1)=O C(CC(=O)N(C1CC(C(=O)NCCC(=O)N(C)C2CC2)C1)C)=C(C)C C1(NC(CCc2cccc(C)c2)=O)CN(C(c2cn(C(F)F)cn2)=O)CC1(C)C C1(CNC(C(C2CCCCC2)OC)=O)CCCN(C(c2sccc2C)=O)C1 Cc1ccc(N)cc1C(=O)NC1(CCNC(c2cccnc2)=O)CC1 C1(C(N2CCN(C3CN(C(c4cn(C)nc4)=O)C3)CC2)=O)CCc2nncn2C1 Cc1nc(CNCCc2cccc(C#N)n2)cc(=NCCOCCS(C)(=O)=O)[nH]1 C(=O)C(C)C(F)(F)F.c1ccccc1.CCCCNC(=O)CO.C(=O)C.C c1(-c2nc(CNCC(CC)NC(=O)OC(C)(C)C)sn2)ccc(Br)cc1 C1(C(=O)NC2CC2NC(=O)C(F)(F)c2cncs2)CCc2[nH]nc(O)c2C1 C1(O)(CCNC(C(C=C)(F)F)=O)CCN(C(C2(F)CCOCC2)=O)CC1 c1(SCC(=O)NCCCNC(C2CC(SC)C2)=O)ccncc1.C1CC1 c1(CC(N2CCN(C(c3c(CC)ncs3)=O)C3C2C3)=O)cn2cc(F)ccc2n1 N1(C(C(c2ccn(C)c2)C)=O)CCCC(CNC(=O)CS(C)(=O)=O)C1C Cc1csc2ccc(C(=O)NCC3CCCCN(C(C4CCCO4)=O)C3)cc12 N1(C(C2C(C(=O)N)C2)=O)CCC(CCC)CC1.c1(C=O)nnn(C)n1.C#CC C1(NC(CSCC=C)=O)CCN(C(=O)COC)C(C)C1.c1ccnc(O)c1 Cc1nc(O)nc(O)c1CCC(=O)NC(C)C1CC1.C1(C=O)CC(C)(C)O1.N C(C(C)C(=O)N1CCC(CCNC(=O)CC2(OC)CCCC2)C1)OCC c1(C(=O)NCC23N(C(C4CC(C)(C)O4)=O)C(CC2)CC3)cnn2cccc(Cl)c12 C(=O)(C1CCc2c[nH]nc21)N(CC(O)CNC(=O)Cc1ccc2nonc2c1)C C1(NC(C2C(NC(C(CSC)O)=O)CCO2)=O)CCCC(C)(C)C1 C1(CC(=O)NC(C(C)C)C2CC2)CCCN(C(c2cc(Cl)n(C)n2)=O)CC1 Cc1cccc2nc(CCC(N3CCN(CC(=O)N=c4cco[nH]4)CC3)=O)[nH]c12 C=CC1CCCCN1C(c1c[nH]nc1C1CCCCN1C(C12COCC1C2)=O)=O c1(C(=O)NC(CNC(c2c(OC)ccs2)=O)CO)sc2ccc(C)cc2c1C c1(C(N2CCCC(CNC(c3cc(OC)ns3)=O)C2)=O)cc(N)cc(F)c1 c1(C(=O)NC(CN(C(C2N(C(C)=O)CCCC2)=O)C)C)cc2ncccc2o1 c1(OC)c(C)csc1C(=O)NC1(C)CN(C(=O)C=Cc2cnn(C)c2)C1 CC1CCCn2ncc(C(=O)N(CCO)CC3CCCN3S(C)(=O)=O)c21 c1(OC)cncc(CNC(=O)CCCCNC(=O)Cc2ccc(O)cn2)n1 C1(NC(Cn2c(C)ccn2)=O)(CNC(C2CCCCC2F)=O)CCC(C)(C)CC1 C1(C(=O)NCCC(=C)CNC(=O)Cc2cnc[nH]2)CCCC(C(N)=O)C1 C#Cc1cncc(NC(=O)CCCCCN(C)C(C2CCNC2=O)=O)c1 C(CNC(=O)CC1CCOC1)(CC(=O)NCCc1ccc(C)cc1)OC Cc1ccc([N+](=O)[O-])cc1C(=O)NCC1CCN(c2ncncc2F)C1 CN1C(=O)OC2CN(C(C3CCCCN(C(=O)C(C)(C)C(C)(F)F)C3)=O)CC12 C1(CC)(CC)CC(NC(=O)Cc2ccnn2C)CN1C(C1CCCN1C=O)=O C1(C(C)NC(C2CS(=O)(=O)C2)=O)CCN(C(=O)CN2CCCC2C)CC1 N1(C(C(CC)NC(N)=O)=O)CCCC(CCNC(=O)CCC=CC(C)C)CC1 C(=O)(CCC(C)(C)F)NCC(C1CCN(C(Cc2cc(C)no2)=O)CC1)(C)C C#Cc1cc(NC(C2CC(OC)CN2C(=O)C(CC)n2ccnc2)=O)cc(F)c1 C(C1=CCN(C(=O)C(F)(F)CN(C)C)CC1)NC(C1C(OC)CCCC1)=O C=C(CNC(C1CC1C(C)C)=O)CCNC(=O)C(C)Cc1ccccn1 c1(C(N2CC=CC(NC(C3C(OCC)C3C)=O)C2)=O)ccc2ccccc2c1F C1(NC(c2cc(C(=O)OC(C)(C)C)no2)=O)CC2(C1)CC2F C(=O)(C(F)CC1CN(C(=O)CCN(C)C)C1)NCCCOCCCC c1(CCC(=O)NC(CCCOc2cc(C)c(Cl)cc2)C)nc2c(O)ncnc2s1 C(=O)(CCCCCN(C)C)NCC(CN(C(C(C)C(N)=O)=O)C)(C)C C1CN(C(C2(c3ccno3)CC2)=O)CC1(F)F.C(C(=O)N)OCCOCC C1(NC(=O)Cc2csc(C3CCCC3)n2)CN(C(=O)CCCF)CC12CC2 c1(C(C)(C)C)cc(=NCCCOCCNC(C23CCCN2CCC3)=O)[nH]cn1 C(=O)(C1CCc2nccn21)NC(C(=O)NC(c1onc(C)n1)C)CC(N)=O C1(CNC(c2csc(C3CC3)n2)=O)COCCN(C(c2csc(Cl)n2)=O)C1 C1(NC(C2(CC)CC2(F)F)=O)CCCCN(C(=O)CCCc2ccccn2)C1 C1(C(N(C)C)=O)C2CCN(C(=O)C)CC12.C1C(=O)N1.C1(CC)CCC1.C=O c1(CC)nc(C)sc1C(N1CCCC(CNC(=O)CC2(C)CCOC2)C1)=O CC1CCN(C(C2(c3ccno3)CCC2)=O)CC1NC(c1cc[n+]([O-])cc1)=O S(=O)(=O)(CCC(=O)NCCCC(C)NC(C1CC1C(F)F)=O)NC Brc1cncc(-n2nc(C3CSC3)nc2-c2cn(C3CCCC3)nn2)c1 c1(N2CCC(CNC(CCC3C(C)=NOC3=O)=O)C2)ncccc1[N+](=O)[O-] C(CC(CC)C(=O)NC1CC(C)CN(C(c2nc(C)oc2OCC)=O)C1)=CC C=CC(C)(C)CC(=O)NC1CC1NC(c1ncc(C(F)(F)F)cc1N)=O C(=O)(CCC1=CCCCC1)NC1CC(N(C)C(C2(C)COC(=O)C2)=O)C1 C1(C(=O)NCCCCC#C)(COC)C=CCN1C(c1ccc(C#N)[nH]1)=O c1(C(=O)NCC2CCCC(NC(CSC)=O)C2)cc(F)cc2nn(C)cc12 CCCCC(C(=O)NC1C2CC3CN(C(=O)C=C(C)C4CC4)C1C3C2)C(C)C N1(Cc2cnc(CC)s2)CCCC(C(=O)Nc2ccc(N(CC)CC)cc2)C1 c1(C(C(=O)NCCCSCC)N(C(C)CSCC)C)cnn(CC)c1 C(=O)(CC1CCc2ccccc21)N1CC(COC)N(C(=O)CCCC(C)=O)CC1 c1(C(=O)NCC2(NC(c3n(CC#C)ccc3)=O)CCC2)cc(O)nn1C c1(NCC2C(C)(C)CCCO2)ccc(S(=O)(=O)N2CC(F)CC(F)C2)c(Cl)c1 C(=O)(C(CO)C(C)(C)C)N1CC(CCC)N(C(=O)Cc2nocc2CC)CC1 c1(C(C)=O)cc(C(=O)NC2C=CCN(C(=O)C(C)CC3CCCC3)C2)oc1C c1(C(=O)NC23CC(NC(c4cn(C)nc4Cl)=O)(C2)C3)cc(O)cc(F)c1 C(CC(O)C(=O)N(C1CCCC1(F)F)C)NC(c1cc(SC)oc1)=O C1(C(=O)OC)N(C(C2CCC2NC(=O)CC(O)CN(C)C)=O)CC1(C)C c1(C(=O)N)ccncc1C.c1(C(N(CCOC)CC)=O)sccc1-n1cnnn1 Cc1ccc(C(=O)NCC(C2CC2)NC(=O)C=CSc2nc[nH]n2)cc1Br c1(CCC)ccc(CC(=O)NCC(C)CNC(=O)C(n2nc(C)cc2C)C)cc1 c1(OC)ccc2[nH]nc(C(=O)N(C(CNC(c3conc3C)=O)C3CC3)C)c2n1 C(=O)CCC(C)C.C1(CNC(=O)C)CC(C)CO1.N1(C(=O)OC)CCC1 N1(C(CCCC)=O)CCN(C(=O)CCOc2ccc(F)c(F)c2)C(CC(F)F)C1 N1(C(C2OCCC(NC(c3cn(CC=C)nc3)=O)C2)=O)CCc2ncccc21 Cc1oc(Cl)nc1C(=O)N(CCCNC(c1cnc(C2CCC2)s1)=O)C c1(C(=O)NC2(C(=O)NC(c3cccnc3)CC)CC(O)C2)cnc(C)nc1C N1(C(C2OCC(=O)C2)=O)C2CCC1CC(CNC(C1(F)CC1)=O)C2 N1(C(Cc2cc(C)no2)=O)CC2(CC(NC(c3cnc(O)o3)=O)C2)C1 C1(CNC(CCCOCCOCC)=O)CCN(C(C2CC=CC2)=O)CC1 C1(C2CCCN(C(c3ccnc(OC)n3)=O)C2)(NC(C(CCC)C(C)C)=O)CC1 CCCC(C)(O)CC(=O)NCC1(C)CCCN(C(c2occc2COC)=O)C1 c1(C2(C)C(C(N3CC(NC(Cc4cc(C)no4)=O)C3)=O)C2)ccccc1F c1(C=O)ncc(F)cc1F.C1(NC(CN(C)C(=O)C2CC2)=O)CCC1C.N C1(CC)CN(C(=O)CCOC2CCCC2)CCC1NC(c1c(Cl)n[nH]c1C)=O C1(OC(NOC(C)C(=O)N)=O)(CO)CCN(C(=O)C(C)(C)F)CC1.C(C)(C)C NC(=O)CC(O)C(=O)NCCCn1cc(CCCNS(C)(=O)=O)nn1 CC1CCC(NC(=O)C=Cc2ccccn2)CN1C(=O)CS(C)(=O)=O N(C1CCCc2ccoc21)C(C1C(NC(=O)C2CC2)CCCC1)=O C(=O)(C(F)(CNC(C1OCCC1(C)C)=O)C(C)C)NCCC(=O)OC C(C)(C)(C(=O)NCC(C)CNC(=O)Cn1ccc(=N)[nH]1)SC N1(C(C(C)=CC)=O)CCCC2(CNC(=O)CCc3ccc(Cl)nc3)CCCC12 C1(NC(C2CCC2(F)F)=O)CN(C(C2(F)CCC2)=O)CC1O N1(C(C(C)CC(N)=O)=O)CC2(CCN(C(=O)C(C)n3ccnn3)C2)C1 c1(OC)ccc(Br)nc1NC(c1csc(C(=O)Nc2csnc2C)n1)=O C#CCC(CC(F)F)C(=O)NC(C)CCC(=O)NCc1ccc(CO)o1 C(=O)(C(C)(F)C(=O)N1CC(CNC(c2coc3c2COC3)=O)C1)OCC C#CCC(C)(C(=O)NC(C)C(F)F)NC(c1cc(C(N)=O)co1)=O CC(CCC(=O)NCC1CCC(CO)O1)NC(=O)COCC(F)F c1(-c2ccc(C)cc2CN2CCCC(CO)C2)ccc(C(=O)O)c2c1OCO2 C(CN=C(NCC1CC1CF)NCC(C)(C)CC(C)O)OCC C(CC)(CCCC(=O)NCCc1ncccc1C)NC(C1(CCC)CC1)=O c1(-c2nnc(N3C4CC(C)(OC4)C3)n2CC2CC2)cnc2ccccn12 CCCCCCC(F)C(=O)N1CCOCC(NC(=O)CCOCCCCCC)C1 N1(C(C2(C(F)(F)F)CN(C(=O)CC3CCC3)C2)=O)CCOC2CCCCC12 Cc1c(CC(=O)NCC2CCOC2)cnn1C.n1(CC=O)ccc(C(F)F)n1.N CC1CC(CNC(=O)CC2CSCCS2)CN1C(=O)CC(C)c1ccco1 CCC(C#N)(CC)C(=O)NCC1CCCN1C(c1ccc2cncn2c1)=O c1(NC(C(C(C)NC(c2c(C(C)C)onc2)=O)C)=O)ccc2c(c1)CCO2 N1(C(CCC=C)=O)CCN(C(c2ccn(-c3ccc(Cl)cc3)n2)=O)CCC1C CC1CNC(=O)CN1C(=O)CNC(=O)CNC(c1ccc[n+]([O-])c1)=O Cc1cc(C(=O)NC(C)(C)CCNC(=O)CCCN2CCCC2)c2c(c1)CCO2 N1(C(C(COC)NC(C)=O)=O)CC2CN(C(c3cc4c(ccn4C)[nH]3)=O)CCC12 C1(C(N2CCC(CCNC(C3CNC(=O)C3)=O)C2)=O)(OC)CCCCCCC1 Cc1ccc(Cl)c(C(=O)NCCC2CN(C(C3(CO)CCOCC3)=O)CC2C)c1 Cc1ccncc1C(N1CCOCC1C(N1CCC(SC(F)(F)F)CC1)=O)=O N1(C(C2C(CC)C2)=O)CC(NC(c2cccn2C2CCCC2)=O)C2CCCCC12 C1(OC)CN(C(=O)C(CCC2CCC2)NC(C2CSC2)=O)CC12CC2 CC(C(=O)N1CC(F)CC1CNC(=O)CSc1nnnn1C)S(C)(=O)=O Cc1c(Br)cc(C(N2C(C(N3CCN4CCCC4C3)=O)CC3CC23)=O)cc1Br CC1CCN(C(c2nccc(Cl)c2O)=O)CC1CNC(=O)CCc1nccn1C C(N=C(NCC(F)F)NC1CCOCC1)c1ccccc1.CC1CCCC1 c1(CN(CCN(C(CCOC)=O)C)C)c(Br)cnn1C c1(C(=O)OC)ccn(CC(=O)NCC2(Cn3cccn3)CC2)n1 Cc1cc(C(=O)NC(C)(C)CNC(C2CC2(C)C)=O)c(C)n1C C1CN(C(=O)Cc2cc(C)cc(F)c2)C(C)(C)C1.c1(CC)nc(C(=O)N)cs1 c1(N(C2CCCC2n2cccc2)C(N(CC)C)=O)cncc(C)c1C.C1CC1 N1(C(C(C)=C2CCC2)=O)CCCC(C2CCN(C(C3OCCC3(C)C)=O)C2)C1 C=CC(C)(CC)C(=O)N1CC(CNC(=O)C(c2cccnc2)C)(COC)C1 C(=O)(CCCCCNC(c1cncc(F)c1C)=O)NC(CCC)CO C1(CNC(c2cnc(C(C)=O)s2)=O)CCN(C(C2CC23CCCC3)=O)C(C)C1 C1(CNC(CCOCCOCC)=O)COCCN1C(C1CC(=O)NC1)=O N1(CCC)CCN(C(c2ccc(CNC(=O)C3=CCCC3)cc2)=O)CC1 C1(CCN(C)C(c2cnc(N)cn2)=O)CCCCN1C(=O)CC1(O)CCCCC1 C1(CNC(c2cc(F)cnc2O)=O)CC2COCC2N1C(=O)C1=CCC1 CS(=O)(=O)C1(C(=O)N)CCC1.c1(CCC(N2CCCC2)=O)ccc(F)c(F)c1 C(=O)(CC1=CCN(C(=O)C(C)S(N)(=O)=O)CC1)NCC(CCC)OC C(CN=c1ccc(C#N)n[nH]1)(C1CCCCC1)NC(c1c(CC)nco1)=O C(=O)(C1NCCc2cc(C#N)ccc21)N1CC(C)OC2(C1)CCOCC2 c1(OC)c(C(=O)NCCC)ccc(Cl)c1C.c1(C=O)ccc(C(F)(F)F)nc1.N Cc1ccc(F)c2[nH]c(C(=O)NC(C)CNC(C3CC(O)CN3C)=O)cc12 C1(NC(C(=O)NCCC(N)=O)=O)CCCCCC1.c1(C(=O)N)c(N)cccc1F C(=O)(C(CCN(C)C)NC(=O)C1CC1)NCC=C(C)C C(=O)(C(F)C(C)C(F)(F)F)NC(C)CC(C)NC(=O)C(C)n1cccc1 C#Cc1nc(C(N2CC(F)CC2CN(C(=O)CNC(=O)CC)C)=O)cs1 C(CC=O)(C(C)C)NC(c1ccc(OC)s1)=O.C(CC1CC1)CC1CC1.N C(C(C)C(C)C(=O)NC12CC(NC(c3ccc(N)c(N)n3)=O)(C1)C2)OC C(=O)(C1=CCCSC1)N(C1C2CN(C(c3cccc(OC(F)(F)F)c3)=O)CC12)C C(CC(O)C(C)C)NC(C(Cn1cncn1)NC(c1ccc(CC)s1)=O)=O N=c1[nH]c2ccc(C(=O)NC34CC3CN(C(C3CC5(C3)CC5(F)F)=O)C4)cc2[nH]1 c1(CCNC(=O)CC(O)C(Cl)(Cl)Cl)ccc2c(c1)OCCO2 N1(C(CC(C)N(C)C)=O)CCC2(CC2C(N2CCCN(CCO)CC2)=O)C1 c1(C(=O)NC2C(CNC(Cc3cccc(CC)c3)=O)CCC2)cc(Cl)nnc1Cl N1(C(CC(C(C)C)O)=O)CCC2(CC1)CC(NC(C1CCC(=O)N(C)C1)=O)C2 c1(CC)c(C(=O)NC(C)CNC(C2(C)CCCCO2)=O)cccc1C c1(C(=O)NC23C(CN(C(=O)CN4CC5CC5C4)C2)CCC3)nccc2occc12 Cn1nc2c(c1C(=O)NC1CCC1)CN(C(=O)CC1(C)CC1(F)Cl)CC2 Cc1c(C(=O)N(C2CCN(C(=O)C(CO)N(C)C)C2)CCO)sc2cncn12 Cc1nc(C(C)(C)C)c(C(=O)NC2CC(CC)C2)s1.c1(C=O)ncc(F)cn1 Cc1ccc(N(C(=O)C)C(=O)CN2CCC2)cc1.C(C(F)(F)F)N.C(C)C C(=O)C(C)(C)C#N.CC(C)(C)Cc1ccccc1.C1(C=O)CN(C(N)=O)C1.N N1(C(C2C(C=C)C2)=O)CCC2(CC1)CC(NC(C1CN(C(=O)NC)C1)=O)C2 CCC(O)C(F)(F)C(=O)N(CC(C)NC(=O)CSc1ccccc1F)C C1(NC(C2C(C)=C2)=O)CCN(C(=O)CN2CCCC(C)C2)CCC1CO N1(C(CNS(CCCOC)(=O)=O)=O)CCN(C(=O)CN2CC=CC2)CC12CC2 N1(C(C2CC2)=O)CC2CC1CN2C(C1CCC(C(F)(F)F)CC1)=O.CC(C)O Cc1cc(C(N2CCN(C(=O)CN(C)C(N)=O)C3CC23)=O)c2ccc(F)cc2n1 C=CCONS(=O)(=O)c1cnn(CCOc2ccc(Cl)cc2)c1C c1(C2C(NC(C3(NC(C(C)c4ccco4)=O)CCC3)=O)C2)ccnn1C C1(NC(C(CSCC)NC(C2CC2(F)Cl)=O)=O)(CO)CC2(CCC2)C1 C1(C(N(CC(=O)OC)C)=O)CCN(C(=O)CC2CC2)CC1C n1(C(C)(C)C)cc(C(=O)NCC(C2CCCCC2)NC(c2cnsn2)=O)cn1 C(=O)(CCCC(F)(F)F)NCCCCC(=O)NCC1(CC)CCC(=O)N1 N1(C(c2cncc(OCC)c2)=O)CCOCC(NC(C2(CCF)CC2)=O)C1 C1(C=O)COc2cc(Cl)ccc2C1.C1(C(=O)NCCC2(C)CC2)CCCCS1.N N1(C(CC(C)c2ccco2)=O)CCOCC1CN(C)C(c1nnc(S)n1C)=O N1(C(C(C2CCOC2)NC(c2c(C)oc(CO)c2)=O)=O)CC2CCCC(O)C2C1 C=CCC(CC(=O)NCCCC(O)CO)NC(=O)C(C)NC(=O)OC C1(F)(CNC(C(C)(C)OC)=O)CCN(C(c2ccccn2)=O)CC1.C(CF)O c1(NC(C2C(C(=O)Nc3cnc(F)c(Br)c3)C2)=O)ccc2c[nH]nc2c1 CCCCC(O)C(=O)N1CC(NC(c2cnc(-c3cccs3)s2)=O)C(F)C1 C(=O)(C(O)c1ccco1)NCCN(C(=O)Cn1cncn1)CCC C1(NC(c2c(CC)onc2)=O)CCN(C(c2cc(Br)sn2)=O)C12CC2 C(=O)(CS(=O)(=O)CC(=O)N1CCC2CCN(C(=O)CN(C)C3CC3)C2C1)OC C1(NC(C(C(C)C)O)=O)CCC2CN(C(=O)CSCCC(F)(F)F)CC2C1 C1(N(C(CCC=C)=O)C)CN(C(=O)COC2CCCC2)CC1O C1(C(=O)NCCN2CCC(NC(CC(CC)CC)=O)CC2)CN2CCC1(C)CC2 c1(CCC(=O)NCC(CC)NC(C23CC(F)(C2)C3)=O)ccc(F)c(F)c1 C(=O)(C(C)(C)CCF)NCCSCC(=O)N(C1CCC(OC)CC1)C c1(C(=O)OC)cc(C(N2CC(C)(NC(C3CCCCN3C)=O)C2)=O)ccc1Cl C1(CC(=O)NC(C2CN(C(C=C(C)C3CC3)=O)C2)C)CCCOC1 C(CC(C)C(=O)N(C)CCN(C(c1ccn(CCC)n1)=O)C(C)C)=CC c1(C(N2CC3C(N(C(C(CC=C)(F)F)=O)C)C3C2)=O)cc(C)c(Cl)cc1F C1(NC(c2cn(C)nc2Cl)=O)CCC(O)CN(C(=O)C(O)CC(F)(F)F)C1 N1(C(C(CCCC)(C)F)=O)CCC(NC(C2CCC(C)(C)O2)=O)C2(CCC2)C1 C(C)(C(=O)N1CC(OCC(=O)NC2(CF)CC2)C1)SC(C)C C=CCCN=C(NCCCN1CCCC1=O)NCC(C)C=C c1(C(=O)NC2CC3N(C(C4CC(=O)OC4)=O)C(CC3)C2)nc2n(c1Cl)CCCC2 N1(C(C(CC=C)CC)=O)CCC2CN(C(=O)CC3(N(C)C)COC3)CC12 C(=O)(C1=NN(C)C(=O)CC1)N1CCC(C)N(C(c2ccc(S(N)(=O)=O)[nH]2)=O)CC1 N1(c2cc(NCc3cc(CC)no3)ncn2)CCN(C)c2ncccc2C1 c1(CC)c(C(N2CC3CC3(NC(C3CC(CC)(CC)C3)=O)C2)=O)csc1C C(=O)(C1CNC(=O)c2ccnn21)NC1C(NC(CN=S(C)(C)=O)=O)CCCC1 c1(OCCC(N2C(CNC(c3c(C)n(C)nc3)=O)C=CC2)=O)ccc(Cl)cc1Cl C(C#Cc1cn(C2CCCc3cccnc32)nn1)NC(c1c(CC)nco1)=O N1(C(C2CC(C#C)(O)C2)=O)CCCC2(NC(c3cnc4n3CCC4)=O)CCCC12 C(C(=O)NCc1cccc(NC(=O)C(C)C(F)(F)F)c1)(C(C)(C)C)OC N1(C(c2n(CCC)ccc2)=O)CC(C)C(N=c2ccnc(Cl)[nH]2)C1 N1(C(C2CC(NC(C3(CC#C)CCCC3)=O)C2)=O)CCCC(CC)CC1 C(=O)(C1=CC2C=CC(C1)C2)NCC.C(c1ccccn1)=CC(=O)N(C)CC Cc1cc(Cl)cc(C(=O)NC(C)(C)CCCNC(c2cccn(C)c2=O)=O)c1N c1(C(=O)NC2CC(C)(NC(=O)Cc3cc[nH]n3)C2)cc2c(nn1)CCOC2 c1(C(=O)NCCCN(C(C(CC)n2cccn2)=O)CC)c(C)c(C)cc(C)c1C C(=O)C(O)CC(N)=O.c1(C(N(C)CC2CCC(C)CC2)=O)ccc(F)cc1F.N C12(NC(c3c(C)cncn3)=O)CCCC1N(C(=O)CN(C(=O)C(C)C)C)CC2 n1(CC)c(C(=O)NC(C)C2CC2)cnc1O.n1(C(CC=O)C)nc(C)cc1C.N c1(CCC)c(C(=O)NC2C=CCN(C(C34CCCCC3C4)=O)C2)nnn1CC CC(Cn1ccnc1)C(=O)NCc1ccsc1C(=O)NCCC1CCCCC1 C1(C(N(CCCC)CCCC)=O)CC(C)CN(C(=O)Cn2cnc(=N)[nH]2)C1 C1(C)(CNC(C=CCC)=O)CCC(NC(c2nn(CC)nc2C)=O)C1 O=S(=O)(c1cccnc1NCCCCN1CCC1)NC(c1c(Cl)cccc1Cl)=O.C CN1CCC(N(C(=O)CN(C(C2(C)CC3CC3C2)=O)CC2CC2)C)CC1 C1(C(N(C(C(=O)OC)C)C)=O)CCN(C(C2CCC(N(C)C)C2)=O)CC1(C)C C1(NC(C2C(C)(C)C2)=O)CN(C(C2(c3ccc(O)cc3)CC2)=O)CC1C#N N1(C(C2(OC)CCOC2)=O)CC(CNC(=O)CC)CC(C)C1.c1ccccc1.O C(=O)(CC(CC#N)c1ccccc1)NC(C(C)C)CCNC(C1C2COCC12)=O C1CC1C1CCCC1.c1(NC=O)ccc(C23CC(C2)C3)cn1.C(=O)C1CC1.C CCCCC(F)C(=O)N(CCCCC(=O)NCC(CO)C(C)(C)C)C c1(C(=O)OCC)cnn(C)c1C(=O)N(C)CC.c1(CC(=O)N)ccoc1 Cc1nc[nH]c(=NCCC2CCCCN2C(=O)C2CCCc3scnc32)c1C#N c1(CNC(=O)NC2CCC(C#N)C2)cc(F)ccc1-c1ccoc1 Cn1nc(C(=O)O)cc1-c1ccc(CN2CC3CC3C2C(=O)O)s1 c1(OC)ccc(F)c(C(=O)NCCC2CC2)c1F.c1(C=O)c(Cl)cccc1Cl.N C1(OCC(N2C(C(C)NC(=O)Cn3cnnc3)CCC2)=O)CCN(C)CC1 C1(CC(N2CCC(CC3CC3)CC2)=O)CN(C(C2CCCO2)=O)CC12CC2 N1(C(c2cc(C(C)(C)C)no2)=O)CC2CCOC2(CNC(C2CC(O)C2)=O)C1 CCCC(CC)CCC(=O)N1CCC(CCC(=O)NCC2CCCC(=O)N2)C1 N1(C(CN(C(COC)=O)C)=O)CCCC(C)C1.c1(C(=O)N)cccnc1C(F)F N1(C(COCC)=O)CCCC(CCNC(=O)C(c2ccccc2F)C)CC1 c1(CC)nc2ccccc2c(C(=O)Nc2ncc(OCC(F)(F)F)cc2C)c1C c1(C(=O)NCc2nccc(C(=O)OC)c2)cnn(C)c(=O)c1 c1(C(=O)NC2(C)CN(C(CC(C(F)(F)F)OC)=O)C2)ncnc2cc(Br)ccc12 N1(C(c2c[nH]c(=N)o2)=O)CCC2(CC(C(N3CCC4(CC4)C3)=O)C2)C1 c1(C(N2CC3C(CNC(Cc4cc(CC)no4)=O)(C3)C2)=O)cnn2cccnc12 CCC(C)C(O)C(=O)N1CC(C)C(C)C1.C1(C#N)(C(=O)N)CC1C(F)(F)F CCCCC(C)CCC(=O)NCC1(C)CC(F)(F)CN1C(=O)Cc1sccc1C C(CC(=O)N(C1CCCOC1)CC)(C(C)CC)NC(C(C)NC(CC)=O)=O C(=O)(C1(C)CCc2ccccc21)NCC(N=c1ccn(C(CCC)C(=O)O)[nH]1)=O Cc1coc(C(=O)NC2CCCC2NC(=O)CC2CC2(Cl)Cl)c1 c1(COC)cn(C(C)CNC(=O)CC2(F)CCC2)nn1.c1ncon1 Cc1ccc(C(c2nnnn2C2CCCC2)Nc2nc(Br)cs2)cc1 C12(C(=O)NC(CCC)C3CC3)CC(CO)(CN1C(=O)C(C)=CC1CC1)C2 c1(C(=O)NCC2(C)CCCO2)ccnc(CNC(=O)C=CC(F)F)c1 C1(CC)CN(C(=O)CC2CCOC2)CCN1C(=O)CCOCc1ccccc1 C1(C=O)CC(O)C(F)C1.CC(C)(C)OC=O.C1(CC=O)CC1.C1CC1.N c1(C(=O)NC(C(C)NC(=O)CCCc2ncco2)C)cncc(F)c1Cl c1(C(N(CCCNC(Cc2nc(C)oc2)=O)C)=O)cccc(-n2nnnc2O)c1 c1(C(=O)Nc2sc(NCCNC(C)=O)c(C)n2)ccc2cn(C)nc2c1 c1(CC)c(C(=O)NC2CC(NC(C3(CC)CCCCC3)=O)C(O)C2)nnn1C C=CCC(CC=C)C(=O)N1C(C(=O)NCCN(CCCC)C)CC1C N#CCCCCC(=O)NC1CCN(C(C2CC(N3CCCC3)C2)=O)CC1 C(CC(=O)NNC(=O)c1ccccc1)c1nn(C)c(-c2ccc(Cl)cc2)c1 c1(C(=O)NC(CNC(=O)C=CCO)C2CC2)cc(Br)c2nccnc2c1 C1(NC(CCC2OCC(C)(C)C2)=O)CCSC12CN(C(c1n[nH]c(=N)[nH]1)=O)C2 N1(C(C2CCCCCN2C(=O)CN2CSCC2=O)=O)CCc2ccsc2C1 N1(C(C(=O)N(C)Cc2ccc(O)nn2)=O)CCC2(CC(O)c3ccccc3O2)C1 S(=O)(=O)(c1ccc(C#N)c(N2CCOC(C3CC3)C2)c1)NCCC(C)N(C)C c1(C(N2C(CNC(C(CC)CO)=O)CC3(CCC3)C2)=O)cccc2c1COCC2 C1(C(=O)NCCn2ccc(=O)cc2)CC2CCC1N2C(C1(CO)CCOC1)=O C1(C(N2CCC2(C)C(N2CCCC2CC2CC2)=O)=O)(OC)CCOC1 C1(C(=O)NC2(CO)CN(C(C3C(C)CCC3)=O)C2)CCC(NC(N)=O)CC1 CC(O)C(F)(F)C(=O)NCCC1(O)CCN(C(=O)CS(C)(=O)=O)CC1 Cc1c(C(=O)N(CCCN(C(=O)C(C)C#N)C)C)cnn1CC(F)F C1(C(N2CC3(CC(NC(CSCC)=O)C3)C2)=O)CCOC2(CCCCC2)C1 C1(C(=O)NC(c2cncc(F)c2)C)CC2(CCCC2)C1 c1(OC)nc(C(=O)NC2CCCC2NC(C2(C)CCSCC2)=O)ncc1F CC1CN(C(=O)Cn2cnc(C#N)n2)CCC1NC(=O)CCCC1CCC1 c1(CC(=O)N(c2cc(C)ncn2)CC2CCCN2)cc(F)ccc1F c1(C(N2CC(NC(Cc3c(C)n[nH]c3)=O)C(CO)CC2)=O)ccccc1S(C)=O c1(CNC(CCCSC)=O)cccc(CN(C(=O)C(C)OCC(C)C)C)c1 c1(C(N2CC(NC(c3n(C(C)C)ccc3)=O)C(C)C2)=O)cnn2ccn(C)c12 C(=O)(C(=O)C(C)(C)CC)N1CC(O)(CNC(C(CC)Sc2ccccc2)=O)C1 C1(CC=C)(NC(c2cc(OC)n[nH]2)=O)CCCN(C(=O)CCSCC)C1 C1(C)CCC(=O)N1C.C1(C=O)CC=CC1.C1(OCC)CC(C(=O)NC)C1 C(=O)(C(CC)Oc1ccccc1)NC(CNC(CCSCC)=O)CC C(=O)(CCC1=CCCCC1)NC1(CC)CCCN(C(=O)CC2NC(=O)NC2=O)C1 CC1(C)CC(CC(N2CCC(NC(C3CC(F)C3)=O)C2)=O)C(=O)O1 C1(OC)CC(C(=O)NCCCOCC(F)F)N(C(=O)CC2CCCC2)C1 C1(C(N(CC=C)C(C)C)=O)CN(C(=O)CCCOCC)CC1(F)F N1(C(CCC2CCC(=O)N2)=O)CCC2(CCN(C(=O)CCOC3COC3)C2)C1 CC(CCC(C)(C)C)C(=O)NCCCC1CCCN1C(C1OCCCO1)=O N#Cc1ccc(NC(c2cc(F)ccc2N)=O)cn1 Cc1cnc2c(C(N3CC4OCCN(C(=O)CC5CCC5)C4C3)=O)c(C)nn2c1 C(=O)(C1=C(SC)CCCC1)NCC1N(C(C(C2CCCCC2)OC)=O)CC(F)C1 C1(C(N2CCC(NC(C(=O)NC3CC3)=O)C2)=O)CCCS(=O)(=O)N1 c1ccc(F)cc1Cl.C(=O)(CCCNC(N)=O)N(C1CCN(C(=O)CO)C1)C C1(NC(N2CCCN(Cc3ccccc3)CC2)=O)CCC(O)C(O)CC1 c1(C(CCO)NC(C2N(C(C)=O)CC2(C)C)=O)cccc([N+](=O)[O-])c1 CC1=NN(c2ccc(C(N3CC4CC4(NC(C4CCC4)=O)C3)=O)cc2)CC1 C=CC(C)C(C)C(=O)N1CC(C(C)(C)O)(CNC(c2ccnnc2C)=O)C1 C=CC1CCCCN1C(=O)COC1CC(NC(=O)C(CC)OC(C)=O)C1 c1(CC(=O)NCC(CC=C)NC(=O)Cn2cc(Cl)cn2)cc[nH]c(=N)c1 C(=O)(CC(O)C(C)CC)N1C(C)(C(N2CCC(NC(CC)=O)CC2)=O)CCCC1 c1(C(=O)NC(C)C(CO)NC(c2ccc(N)cc2O)=O)cnc2ncccn12 N1(CCCC)CCOCC(C(N2CCCC(c3noc(C)n3)C2)=O)C1 C#CCC(C(=O)N(C1COCC1OC)C)NC(=O)CCCN(C)C c1(C(C(=O)O)NCc2ccc(CSC(F)F)o2)ccc2c(c1)OCCO2 N1(C(c2cc(OC)ns2)=O)CC(NC(c2cnc(OC)s2)=O)CC2(CC2)C1 C=CCC(CC(C)C)C(=O)NCC1(CCNC(C2CC(OC)C2)=O)CC1 c1(OC)nc(C)cc(=NC2CCCCCN(C(=O)Cn3cc[n+](C)c3)C2)[nH]1 C12(CNC(c3ncn(C)n3)=O)CCC(CC1)CN2C(=O)CC1CCCC(=O)N1 C1(NC(C2CCS(=O)(=O)C2)=O)CCCC12CN(C(=O)CO)C2.C1CC=CC1 C1(OCc2cn(-c3c(NS(C)(=O)=O)ccc(Br)c3)nn2)CCCC(F)(F)C1 C(C)(CCCNC(c1ccc(C(C)C)s1)=O)NC(COCC)=O C1(C(=O)NC(c2ccc(C)cn2)C)CCOCCN1C(c1cc(C)c(C)cn1)=O c1(C(=O)NCC(C)(C)O)nnc2ccc(-c3cccc4ccoc34)cn12 c1(CNC(c2ccn(C)n2)=O)n[nH]c2c1CN(C(C1C3CCCC13)=O)CC2 C1(N)(C(=O)OC)CC(C(=O)NC2(c3ccccc3)COC2)C1 O=C1CC(=O)NC(C(N2CCC(CCC(=O)NCC3CCCOCC3)CC2)=O)C1 N1(C(CC2(OC)CCCCC2)=O)CCN(C(C2(C)CC2C)=O)C(C)C1 C1(NC(C(CC(C)C)NC(c2n(C=C)ncc2)=O)=O)CCOC2(CCC2)C1 C1(C(N(CC(=O)OC)C)=O)(C(C)C)CCCN1C(=O)CC1CCC(=O)N1 C1(NC(C(C)n2cnnn2)=O)CC(C)(NC(=O)CC2(O)CCCC2)C1 C1(CC(=O)NC2CN(C(c3cnn(C(C)C)c3Cl)=O)CC2O)OCCCC1(C)C c1(C(N(CCCCNC(CC2C(OC)CC2)=O)C)=O)csc(-c2cccs2)n1 C1(CC)CCN(C(=O)CC2CC(SC)C2)C1CNC(C1CCN1C)=O C=CC1(CC(=O)NCCCC(C)CO)CN(C(C2(CCCC)CCC2)=O)C1 O=C(C1=NOC2(CCC2)C1)NC(C(=O)NCc1nnc(O)o1)C1CCOC1 CC(C)CC(C(=O)N1CCC(C(=O)NCCN2CC=CC2)C1)C(N)=O C(c1ccc(F)c(F)c1)=C(C)C(=O)NCC(=O)Nc1ccc(OC(F)F)c(C)c1 CC1CN(C(=O)CCc2cncs2)CC2(CCN(C(=O)CCc3ncco3)C2)O1 C(=O)(CC(CNC(=O)CC1(C)OCCO1)C1CCC1)N1CC(C)(CC=C)C1 C1(C(N2CCC(Cn3cc(C4(CO)CC4)nn3)C2)=O)CCc2nccn2C1 c1(C(N2CCCC2)=O)ccc(C(C)C)c(C)c1.C(=O)(CC(C)(C)C)NCC.C c1(C(N2CC(COC)N(C(=O)CC(C)(C)F)CC2)=O)ccc2cccc(Cl)c2n1 CC(C)S(=O)(=O)CC(=O)NCCC(C)(C)C.c1(C=O)cccc(C2CCC2)c1.N N1(C(CC(=O)OCC)=O)CCCC(O)(CNC(c2c[nH]cc2C)=O)C1 C(=O)(C(CC(C)C)NC=O)N1CCCC1.C(=O)(C(C)(F)F)N(CCC)CC c1(C(N2CC3(CCN(C(C(CC#C)C4CC4)=O)C3)C2)=O)cc2c(nc1N)CCC2 C(CC#CC)(C(=O)NC1COCCC1C)NCCSCC=C.CCC.CC(F)F.O C(=O)(C(C)(F)C(=O)N1CCCC(C(=O)NCCN2CCOC(C)C2)C1)OC N1(C(CC2ON=C(CC)C2)=O)CCC2(CC2C(=O)NCCc2cccs2)C1 c1(COC)cccc(C(=O)NCCCC2CC2)c1.c1(C(=O)N)csc(Cl)n1 N1(C(C=CCC2(NC(c3csc(F)c3)=O)CCC2)=O)CCSC2CCC12 C(=O)(C(F)C(F)(F)C(F)(F)F)N1CC(C)N(C(=O)C2=CCCS2)CCC1 Cc1ccc(C(=O)NC2(CNC(=O)CNC(=O)C3CC3)CCCC2)[nH]1 N1(C(c2nccc(OC)c2)=O)CC2CCCC2(Nc2snc(Cl)c2C#N)C1 C1(NC(C(CC)NC(N)=O)=O)CN(C(c2cc(C#N)c[nH]2)=O)Cc2nccn2C1 C1(NC(C(C)(C)C)=O)COC2(CNC(=O)CCn3ccnc3)CC1C2 CC(C)C(C(=O)N1CCC(NC(=O)C(CO)N(C)C)CC1)c1cccc(Cl)c1 Cc1cccc(C(N2CCOCC2CNC(c2cn(CC(F)(F)F)nn2)=O)=O)c1 C1(NC(=O)Nc2nc(CC)c(C(C)(C)C)s2)CCC2C(C1)C2(F)F N1(C(=O)CC2CC(F)C2)CCC2CCN(C(c3cncc4[nH]ccc34)=O)CC2C1 C1(NC(C2CCN(C(CC)=O)C2)=O)CCN(C(=O)CC(C)C(C)C)C(C)C1 c1(CCC(=O)NC2CCCN(C(c3c[nH]c(=O)cn3)=O)C2)ccc(Cl)nc1 c1(C(=O)NCCCN(C(=O)C(CCOC)OC)CC)cnc2c(c1)CCC2 Cc1cc(C#N)nc(N(C2CC23CCNCC3)C(c2cnc[nH]2)=O)n1 C1(NC(=O)C(F)CC2CCOC2)(CF)CCN(C(=O)C=CC=C(Cl)Cl)C1 c1(C(N2CC(NC(CC(CC)(F)F)=O)C(O)C2)=O)ccc2c(c1C)CCC2 C(=O)(C1SCCc2ccccc21)N1CCC(CNC(CCC(C)(F)F)=O)C1 C(=O)(N=c1cc[nH]cc1Cl)c1ccc(NC(CC(=O)OC)=O)cn1 C(c1ccccc1)=CC=CC=O.Cc1ccn(CC(=O)N)n1.C1(=CC)CC1 C#CCC(CC(=O)OC)NC(=O)CC1CC(F)CN1C(c1cccc(C)c1F)=O N1(C(=O)NC23C4C5C6C4C2C6C35)CCc2nc(-c3ccccc3)ncc2C1 C(=O)(C(O)C(C)CC)N(CCCC)Cc1cn(-c2cncc(C(=O)O)c2)nn1 CC(C)(CCNC(c1cc(C2CC2)[nH]n1)=O)C(=O)N1CCCC(F)CC1 CCCC(CCCNC(c1nsnc1O)=O)NC(c1ccn(CC)c1C)=O N1(C(c2c(CC)non2)=O)CC(C(=O)N)C(F)(F)C1.C1CC(=O)N(C)C1.C CCCC(C)C(=O)N1CCC(CO)(NC(c2sc(-c3cnn(C)c3)nc2C)=O)C1 N1(C(c2ccnc(C(C)C)n2)=O)CCC(C2(NC(=O)CN3CCC(C)C3)CC2)C1 C(=O)(C(=O)CC(C)CC)N1CCCC(C(C(=O)N(CCCO)CCC)(C)C)C1 CC(C)(C)C(C)(O)CNC(c1coc(C)n1)=O.C1(C=O)CC2(CC2)C1.C c1(C(=O)Nc2ccc(CC(=O)Nc3ccc(Br)c(O)c3)cc2)cc(F)cc(F)c1 CC(C)C1=NOC(CNC(=O)NC2(CO)CC3CCC2C3)C1 N1(CCOC)CC(CNC2CCNC(c3ccccc3)C2)CC1=O Cc1c(C(N2CCCC2CCC(=O)Nc2ccc(SC(C)C)cc2)=O)cccc1Cl c1(OC)ccc(C(=O)NC2(CCO)CN(C(C3CC4CCC3CC4)=O)C2)c(O)c1 c1(OC)ccc(C)nc1-c1nc(-c2cncs2)nn1CCCCO C(=O)(C1=C(C)OCC1)N1CC(C=C)C1 Cc1ccc(CC(=O)NC2CC(C(=O)NCCOCC(C)(C)O)C2)cc1 N1(C(C(CC)(C)OC)=O)CC2CC(NC(c3c(C)ccnc3C)=O)C1C2 CCC(C)(CNC(C1CCC(C#N)CC1)=O)C(=O)NCCn1cc(CO)nn1 C1(N(C(=O)CNC=O)C)CCN(C(c2cncc(N)n2)=O)CC12CC2 c1cccc(Cl)c1Cl.CC1OCCC1CC(=O)NCCOC1CN(C(=O)C)C1.N C1(CC(=O)NC(CC(C)NC(c2c(COC)ncs2)=O)C)CCCCC1.O C1(COC)CN(C(=O)OC(C)(C)C)CCN1C(=O)Nc1cc(Br)ccc1O N1(CCC)CCC(C(N2CCC2CNC(C2(c3cncs3)CC2)=O)=O)CC1 C1(CCC)(NC(=O)C(O)C(C)SC)CCN(C(=O)CCc2ccc(C)s2)CC1 c1(C(N2C(CNC(c3ccc4nncn4c3)=O)CC2)=O)cc([N+](=O)[O-])ccc1Cl N1(C(CC2C(C)CCO2)=O)CCC2CCCC12C(=O)NCCc1cn[nH]c1 CC#CCC(CO)NC(=O)CNC1CC(NC(=O)C(C)(F)c2ccon2)C1 C#CCC(C)(C(=O)NCC(O)C1CCC1)NC(=O)Cc1sccc1C CC1CN2CCN1CC2C(N1CC(O)(CN(C)C(c2cc3occc3s2)=O)C1)=O N1(C(C2CC2F)=O)CC2CCCN(C(c3cc4nc[nH]c4cn3)=O)C2C1 c1(CNCC2(NC(c3ccc(=O)oc3)=O)COC2)c[nH]c2cccc(O)c12 C1(NC(c2ccc3cc[nH]c3n2)=O)C2CC3CN(C(=O)C4=CSCS4)C1C3C2 C(=O)(CCN(OC)C(=O)CCc1cccs1)NCC1(CC)CCC(=O)N1 C(=O)(CCC(C)NC(C1CCCC1)=O)NCC CC(C(CO)NC(C1CC1c1cn[nH]c1)=O)NC(c1cnco1)=O c1(N2CCC(NC(=O)CC3CCCCO3)C(F)C2)nc2ccc(F)cc2o1 N1(C(C(C)SCC)=O)CCC(NC(=O)Cc2cocn2)C(F)C1 C(=O)(C(C(C)C)NC(=O)Cn1cccnc1=O)NC(CC=CC)CO c1(C(C)C(=O)NCC2CCN2Cc2ccsc2)ccc(F)cc1 C1(OC(C)C)CC2CCC1(CO)C2.c12ccc(c(Cl)c1)c(=O)[nH]2 c1(-c2nc(-c3oc(C)c(-c4ccccc4)c3)on2)cc(F)c(F)c(F)c1 C1(C(=O)NCC2CCN2C(=O)CCc2cccs2)CC(c2ccncc2)=NO1 c1(CC)ccnn1C.C1(C(=O)NOCC(=O)NC)CCCCC1CNC(C)C C1(NC(CCC=C=C)=O)CCN(C(c2cn(C)nc2-c2ccoc2)=O)CC1C N1(CC2C(CC(C)(C)C)C2)CC2(C=C(C=O)CO2)C1.C(C(F)F)C(C)(C)C C1(F)(C(=O)NC2C(F)CCN(C(c3cc(C)[nH]n3)=O)C2)CCC(F)(F)CC1 CC1CCN(C(C2CCCCS2)=O)C1CNC(c1cncnc1C1CC1)=O c1(C(N2CCC(O)(CNC(CC(C)OC)=O)CC2)=O)cc(=O)n(C)cc1Br C=C(C)C(CC(=O)NC(C)C(C)(C)C(=O)NC1C(O)CC1O)OCC C(=O)(CC(C)O)N(C(C)C(=O)N(C1CC(CO)C1)C)CC c1(CCC)c(C(=O)NC(C2CCN(C(=O)Cc3cnsc3)C2)C)cnn1CCO C(=O)(NNc1c(Cl)cc([N+](=O)[O-])cc1Cl)C1CC(NC(=O)OC(C)(C)C)C1 N(C(=NCC(C(C)C)OCC)NC1CCC1)C(C#C)COC c1(C(=O)OC)cc(C(N2CCCC2CCNC(=O)C(CO)N(C)C)=O)cs1 Cc1[nH]nc2ccc(C(=O)NCC(C)(CO)NC(C3CC3CC(C)C)=O)cc12 N1(C(c2c(C)onc2Br)=O)CCCCC(NC(c2cc(C#N)no2)=O)C1 c1(CC(N2CCC(OCCNC(C(C)OC)=O)C2)=O)sc2ccccc2c1C c1(OC)ccncc1CC(=O)NC(C)CC(C)NC(c1ccc(OC)nn1)=O CS(=O)c1cccc(C(N2CC(F)(F)CC2CNC(=O)C(F)C2CCC2)=O)c1 C(=O)(C1Cc2ccccc21)NCCCNC(=O)COCCc1ccc(Cl)s1 N1(C(CC(=C=C)C)=O)CCC(C)C(NC(=O)Cc2cccc(OC)c2)C1 C1(OC)CC(NC(C2CCN(C3CCCCC3)C2)=O)CN(C(C2CC23CC3)=O)C1 c1(CNC(C2C(=C)CC2)=O)ncoc1C1CN(C(C2COC(=O)C2)=O)C1 c1(C(N2CC(NC(c3n(CC)ncc3)=O)C(F)C2)=O)cc([N+](=O)[O-])cc(C)n1 N1(C(C(COCC=C)N(C)C)=O)CCN(C(=O)C(CCOC)OC)C2(CCC2)C1 c1(C=O)ccc2c(n1)CCCN2.C(CCCNC(=O)C(COC)N(C)C)OC.N CC(F)CCS(=O)(=O)NC1(c2cccc(C(=O)N(C)C)c2)CC1 c1(C(N(CCN(C(C2C(C=C)C2)=O)CC)CC)=O)cc(Br)c(C)cn1 C1(C(=O)NC2C(NC(C(C)(C)N(C)C)=O)CC2)CC12CCOc1ccccc12 C1(NC(C(=O)OCC)CCCOC(C)(C)C)COc2cc(O)ccc2C1 n1(CC)cnnc1CCNC(C1CN(C(=O)CNC=O)C1)=O.c1ccccc1 C(C(CC1CCCC1)C(=O)N1CC(CO)(CO)C1)NC(Cn1ncc(C)c1)=O N1(C(c2nc(C)sc2)=O)CC=C(CCNC(=O)CC2CC(C)OC2C)CC1 N1(C(C(CC=C)OC)=O)CCCC2C1CCCN2C(=O)C(C)=C(C)C C(=O)(C(C(C)C)OC1(OCC)CCOC1)N1CC(CCCCC)C1 C1(F)(C(=O)NC(c2nc[nH]n2)CC)CCN(C(c2cc(C)no2)=O)CC1 c1(N2CC(CO)N(c3cc(-n4cncn4)ncn3)CC2)ncnc2n[nH]c(I)c12 c1(CC(N2CC(NC(=O)CC34CCCC3C4)C(C(F)F)C2)=O)cc(F)ccc1O C=C(C)CCCC(=O)NCC(CC(=O)NCc1ncoc1C)C1CCC1 C#CCC(C)C(=O)NC1CCN(C(=O)C=CCOCC(F)(F)F)C1C C12(CCOCC1)C(=O)NC1CCC(C1)C(=O)N2.C(C(C)OCCO)SC c1(C(N2C(C)C(NC(C3(O)COC3)=O)CCC2)=O)cccc2ccnn12 Cc1noc(C)c1CNC(CC1CCCCC1)CC(=O)N.C1CC1C(C)(F)F c1(CC=O)ccc2n[nH]cc2c1.C1CC(F)(F)C1.C(CC)N(C(=O)C)CC.N C(CN=c1[nH]c2c(F)cccc2o1)(C1CCCC1)NC(=O)C1Cc2ccccc21 C(=O)(C(C)(C)NC(=O)CC1CC=CC1)NCC1C(C(C)C)C1 C(=O)(C1CCc2ccccc21)NCC(C)NC(c1cnn2cc[nH]c(=O)c12)=O N1(C(C2C(C(=O)OC)C2)=O)CCN(C(=O)CC(C)SC)CC1 C12(NC(c3cc(C)oc3)=O)CCCN(C(=O)CCn3cccn3)CC1C2 C(CCC(=O)NC1CC(C(F)F)C1)OCCOC.C1(C=O)CC1(C)C.N c1(C(=O)N)ccc(O)c(N)n1.C1(CNC(C2(OC)CCC2)=O)CCCCC1 N1(C(c2cn(CCN(C)C)nc2)=O)CCC2CN(C(=O)CCCC#N)CC2CC1 C(=O)(CC(CC(N)=O)c1ccc(F)cc1)NCCNC(CCC1C(C)(C)C1)=O C(=O)(C1=C(COC)N(CC(C)C)C(=S)NC1c1ccc(F)cc1)OCC CCCCCCCCNC(=O)NCCSCC1(O)CCOC1C.c1(C)ccccc1 c1(OC)ncc(C(N2CCOCC(NC(=O)CSC)C2)=O)cc1C C1(C(=O)NC2CC(C)N(C(=O)C=C3CCSCC3)C2)CCCC12CCOCC2 c1(C(N2C(CCNC(C3C(C)OCCO3)=O)CSCC2)=O)cc2cn[nH]c2cn1 Cc1ccc(C(=O)NCC2(F)CN(S(=O)(=O)CCCCl)C2)c(C(F)(F)F)c1 N1(C(c2cnc(C)[nH]c2=N)=O)CCC(C(N2CC(O)C(O)C2(C)C)=O)C(C)(C)C1 C1(NC(C(C)NC(CC)=O)=O)CN(C(=O)CC2(C)CC2)CC1C N1(C(C2(CC)COC2)=O)C2CCC1CC(CNC(=O)CC1CCN(C)C1)C2 C1(NC(C(C=C)O)=O)CC=C(C(=O)NCCN2CCCCC2C)C1 CCCC(CC(C)C)C(=O)N1CCCC(N(C)C(c2cc(C3CC3)no2)=O)CC1 c1(C(=O)NCCNC(c2cc(N)c(O)c(F)c2)=O)cnc2n1CCCCC2 Cc1c(C(N)=O)cccc1C(=O)N.C1CCN(C(C2CC3CC3C2)=O)C12CC2.C Cc1cc(C(=O)NC(C(=O)NC(C)CS(C)(=O)=O)C2(C)CC2)nc(O)n1 c1(NC(c2c(CNC(=O)C=Cc3cc[nH]n3)c[nH]n2)=O)ccc(O)c(Cl)c1 C(=O)(C1=CCOCC1)N1CCC(CC)C1C(=O)NCc1ncnn1C c1(CN(C)C)ccccc1.n1(C(C)C(=O)N2CCCC2)cc(C2CCN2C)nn1.S c1(C(=O)NCC(C)(C)CNC(C2CCCC2(C)C)=O)cc(F)c(Br)cc1F c1(C(=O)NC2C(CNC(C(c3ccccc3)SC)=O)C2)cn(C)nn1 N1(C(C2CCC(OC)CC2)=O)C2CCC1(CNC(C1CCCCS1)=O)CC2 C1(COCC)CC2C=CC1CC2.c1(CNCC)cc(C(F)F)cs1 c1(C(N(CC(C)NC(CC(CCCC)O)=O)C)=O)cc(C)n(NC(N)=O)c1C CC(C)S(=O)(=O)C(C)C(=O)NC1CC2CCC1N(C(=O)C(O)CC(N)=O)C2 N1(C(Cc2cc(C)[nH]n2)=O)CCC2(NC(=O)C=CC=C(Cl)Cl)CCCC12 c1(OC)ccc(C(=O)NCC2CCN(C(C3(CO)CC3)=O)CC2C)c(F)c1F c1(OC)cnccc1C(N1CCC(N2CCN(C(=O)CCNC(N)=O)CC2)C1)=O Cc1ccc(CNC(c2c(C)nn(C)c2F)=O)cc1Cl C#Cc1ccc(C(N2CC(CNC3CCC(c4ccccc4)C(C)C3)C2)=O)cc1 c1(C(N2CC(O)(CNC(CN(C(C)=O)C)=O)C2)=O)c[nH]c2c(Cl)cccc12 C(CC(C)CCNC(=O)CC1CSC1)NC(C1(NC(C)=O)CCC1)=O C1(NC(C2(CC)CCNC2=O)=O)CCC(C)N(c2ccnc(C(=O)OC)n2)C1 C1(CNC(c2c(OC)nsc2OC)=O)CCC2(CN(C(C3CCC3)=O)C2)O1 c1(C(N(CC(C)N(C(=O)CCCn2cccn2)C)C)=O)noc2cc(F)ccc12 C1(CNC(Cc2c(C)ocn2)=O)CCN(C(=O)C=Cc2cccc(F)c2)C1(C)C C(=O)(C1CNC(=O)c2ccccc21)N(CCNC(C1CCCCNC1=O)=O)CC c1(C(=O)NC(C2CCCN(C(=O)C(F)=CCCF)C2)C)cc(Cl)n(C)n1 c1(C(N2CCC(NC(=O)CN3CC4CC4C3)C2)=O)cccc2nonc12 c1(C(N2CCN(C(C3(C)CCSCC3)=O)CC2)=O)cnc2nccnc2c1 C1(NC(c2c(=N)c(Br)c[nH]c2)=O)CC2CC(C1)CC(F)(F)C2 Cc1ccc2c(c1)C(C(=O)NC(C)CN(C(=O)C=CC1CC1)C)OCC2 CC1(C)C2CCC1(C)C2C(N1CCC(C)(CNC(c2cc(Cl)c[nH]2)=O)C1)=O C1(C(N(C2CCN(C(CC3CCC3)=O)C2)CCO)=O)CS(=O)(=O)CC(=O)N1 CC1CCC(CNC(C2(C(F)F)CC2)=O)CN1C(c1ccc(CO)cc1)=O C1(C)(NC(C(c2cccc(Br)c2)C)=O)CCC(NC(c2cnc(O)o2)=O)CC1 c1(C(=O)NCCOCCNC(C(CC=C)C)=O)cccc2c1CCS2(=O)=O CC1CCC(F)(F)CN1C(=O)C(C1CC=CCC1)NC(=O)C(Cl)Cl C1(CNC(C(COCC)(C)C)=O)CN(C(=O)C(Cl)=CCl)CC(C)(C)C1 N1(C(CC(C)OC)=O)CCCCC(CNC(c2cscn2)=O)CC1 S(=O)(=O)(c1cn(C)c(Cl)n1)Nc1cc(C(=O)NC)n(C)n1 CCC(CCCC(=O)NC1CC2(COCCO2)C1)NC(=O)C(C#N)(CC)CC C1(C(N(C2(C(=O)NC(c3nnnn3C)C)CC2)C)=O)COCCN1C C1(CC(=O)NC(C2CCN(C(=O)C=C3CCN(C)C3)C2)C)CCOC1=O C=CCCC(CC(C)C)C(=O)NC1CC1NC(C1CCC(CCC)CC1)=O C1(C(N(C(C)(C)CC(=O)NCCC2CCC(=O)N2)C)=O)CC(=O)C12CCC2 c1(C(N(C(CCNC(CCC(C)CN(C)C)=O)C)C)=O)ncnc2c1CCCC2 c1(N2CCC(C(C)C)C2)nc(=NCc2cc3c(s2)CCC3)[nH]c2c(F)cccc12 N1(C(C(=O)NC)c2ccns2)CCCC(C(=O)NCCOC)C1 c1(NC(CCCC=C)C)cc(S(=O)(=O)N2CCN(CC(C)O)CC2)ccc1C#N C1(N2CCCC(CNC(=O)CN3CCCC3=O)C2)CCc2ccccc2C1 N1(C(C(C(C)OC)NC(=O)CC(F)(F)F)=O)CC2(CCC2)CC1CO c1(CC(=O)NC2CCN(C(C3CC3C(F)F)=O)CC2O)cc(Cl)cc(Cl)c1 N1(C(c2nn(C)c(Cl)c2Cl)=O)CCCC2(CC2)C1.C1(S(C)(=O)=O)(C=O)CC1.N n1(CC)ncc(C)c1C(N1CCOC(CCCNC(C2CC3CC3C2)=O)C1)=O N#Cc1cc(C(=O)NCCCN(C(=O)CCC2CCC(=O)N2)CCO)ccc1Cl Cc1ccc(C(=O)N(CC(C)(C)C(=O)NC(C)(C)CCCO)C)nc1O c1(C(=O)OC)cccc(O)c1NC(C1CC(C)CN1C(=O)C1=CCCCO1)=O C1(C(=O)Nc2cn(C)nc2)CCOCC1NC(c1cnn(C)c1)=O C(C(F)(F)C(=O)N1CC(CC(F)C(=O)NC2CCCC(O)C2)C1)OC C(=O)(C(O)C(C(C)C)OC)N1C(C)(CCC(=O)NCCCCCOC)CCC1 C1(C)CCN(C(c2cnc(C3CC3)o2)=O)CC1.C#CC1C(C(=O)NC)C1(C)C c1(C(=O)NCCCCCNC(C(C=CC)O)=O)cc2ccc(Cl)cn2c1 CC1(C)CC(C)CN1C(C1CC12CCOCC2)=O.C1(CC(=O)N)CC2(CC2)C1 C1(C(=O)NCC2(O)CCN(C(=O)Cn3cncn3)C2)CC12CC(F)(F)C2 N1(C(c2c(CC)ccc(F)c2)=O)CC2CCC(C1)N2C(C1CN(C)CCO1)=O N1(C(Cn2c(N)ccn2)=O)CC=C(CNC(=O)C(F)CC2CCCCC2)CC1 C(=O)(C(=O)CCC(C)(C)C)NC(C)CN(C(=O)CC12COC(C)(C1)C2)C c1(C(=O)NCC(CNC(=O)CC(F)(F)F)O)cc2ncc(Br)cn2n1 C=CCC(C(=O)NCCC1(O)CCN(C(c2cc(CC)nc(O)c2)=O)C1)C(C)C CC1(C(=O)NC2CC(F)(F)C2)CCCN(C(=O)CC2CCCC2)C1 Cc1cc(C(=O)NC2(CNC(=O)CCn3ccnn3)CCC2)cnc1O C1(C(=O)Nc2cc(C)c(F)cc2)CN(C(=O)C=CCBr)CCC1(F)F C(C(C(=O)NCC(C)(F)F)NC(c1cnsc1)=O)OC(C)C C(=O)(CC(=O)NC(CC1CCC1)C(=O)NC1(CO)CC1)N(C)C N1(C(c2c(C)cnnc2)=O)CC2CC(NC(C3C=CCS3)=O)C(C2)C1 C(CS(=O)(=O)CC(=O)NCCCCC(N1CC2CCCCC2C1)=O)OC c1(C(=O)NCC2N(c3ncc(C#C)cn3)CC(C)(C)C2)ccc2c(c1)ncn2C c1ccc(CS)cc1.C1(C(C)(C2CC2)OC)CC(NCCNC=O)C1 c1(C(=O)NCC2C(C)CCCN2C(=O)C(F)C(C)(C)O)cccc2ccnn12 C=CCC(CC(C)C)C(=O)N1CC=CC(NC(c2ccc([N+](=O)[O-])cc2F)=O)C1 c1(C(=O)NC2C3CN(C(C4(CC)CCCCO4)=O)C2C3)c[nH]c2nccc(Cl)c12 C1(C(=O)Nc2ccnc(OC)c2Cl)CN2CC3CC2(CO1)C3 Cc1cc(C#N)c[nH]c1=NC1CC(C(C)NC(=O)C(F)(F)CN(C)C)C1 C(CN=c1[nH]c(=NCC2(C)CCCCCCC2)c2ncccc2[nH]1)SC c1(C(=O)NC2CC(CCNC(C3(N(C)C)CC3)=O)C2)cc(F)cc(Cl)c1N C(=O)(C1=C(Cl)CCC1)NCC(C)(C1CCC1)NC(c1ncccc1F)=O C(=O)(CCC1=CCc2ccccc21)N1C(CNC(=O)C2=CCC2)CC1 S(=O)(=O)(c1ccc(NC2CCN(CCCO)CC2)c(Cl)c1)NC.CC1CC1N c1(OC)nscc1C(=O)NC1CCC1CNC(C12CC(F)C1C2)=O c1(C(=O)OC)ccccc1S(=O)(=O)N1CC2C(C(N3CCC(C(C)O)C3)=O)C2C1 n1(CCC(N2CCCC(N(C3CCCNC3=O)C)C2)=O)ccc2ccccc12 C(=O)(C1=CCCCO1)NC1CC(CNC(C)=O)OCC1 O=C(N=c1cc[nH]cc1Cl)C1CCCN(C(=O)C=CC2CC2)CC1 CCCCCC(O)C(C)C(=O)N1CCCC(CNC(=O)C(C)c2ccco2)CC1 C1(CC)CN(C(c2cnco2)=O)CCC1CNC(C1CCC1(OC)OC)=O C1(O)(CC)CCCN(C(=O)CC2CCN(C)C2)C1.c1(C(C)C)scnc1C(=O)N c1(CC(=O)NCC(C)(CO)NC(c2cc(C)ncc2)=O)ccc(C)c(Br)c1 Cn1c(=O)nc(O)c2cc(C(=O)N=c3cc4n([nH]3)CC(O)CO4)cnc12 C1(CNC(Cc2c(C)ocn2)=O)CN(C(=O)C(C)CN(C)C)C2CCCC2O1 N1(C(c2c(C)cccn2)=O)CCC(F)(C(N2CCC2C(C)O)=O)CC1 c1(C(=O)Nc2ccc(-c3c(C)nn(C)c3)c(F)c2)ccnc2c1OCO2 C1(C(N2CC(CC)C2)=O)CCCCC1CC(F)(F)F.C1CC=CC1.C(=O)(C)N O=S(=O)(CCCN=c1ccnc(NC2CCCOC2)[nH]1)C(F)F C(=O)(CC(C)C(F)(F)F)NC(c1ccnn1C)C(=O)NC(C(CC)(C)C)C CCCC(CCC)C(=O)NC(CC)CCC(N1CC2(C1)CC(C)(C)C2)=O C1(C(N2CC(OC)C(NC(=O)CCN3CCC3)C2)=O)CCC(=O)N(C)C1 C=CCN=C(NCc1c(C)nn(C)c1N1CCOCC1)N1CCCC(O)(COC)C1 CCC(CCCC(=O)N(CCCC(C)(F)F)C)NC(c1cccn2ccnc12)=O C1(CC)CN(C(=O)C=CC(c2cnn(C)c2)=O)CCO1.c1(CC=O)ccoc1 C1(C(N(CC(C(C)C)C)C)=O)C2CN(C(=O)CC3CC(F)(F)C3)CC12 c1(C(N2CC(O)(C(C)NC(CNC(C(CC)C)=O)=O)C2)=O)c[nH]c(=O)cn1 Cc1ccc(C(=O)NC2CC(C(=O)NCc3ccncc3)C2(C)C)cn1 C#CCC(CC(=O)NCCC(=O)NO)NC(c1csc(C)c1C)=O [nH]1nc(C(N2CCC(C(F)(F)F)C2)=O)c(C)n1.C(=O)CN(C)C(C)C.CC n1(CCCC)nnnc1C(c1coc(C)n1)NCCCSCC(C)C c1(OC)cc(CC(=O)NCC(C)(O)CNC(C2CNC(=O)C2)=O)ccn1 N1(C(c2c(OC)ccc(C)c2)=O)CCCC2C1CCCN2C(=O)C#CC1CC1 C(=O)(C(O)CC(N)=O)N(CCC(=O)N(CCC(F)(F)F)CC)CC=C N1(C(C=C(C)C(C)C)=O)CC2C3CCC(C2C1)N(C(C1CC1C1CCCO1)=O)C3 c1(CCC)[nH]ccc1C(=O)NC1(C)CC1.c1(C2C(C(=O)N)C2)ccccc1 c1(C(=O)NC(CSC)(C)C)oc(CO)cc1C.c1(CC(=O)N)ccsc1.CC N1(C(c2cnc(SC)s2)=O)CCCC(CO)(NC(c2n[nH]c(C3CC3)n2)=O)C1 O=C1CCN(Cc2cscc2Cl)C(=O)N1Cc1nc(C2CC2)cs1 C#CCC(C)(C(=O)NC1CCCCC1(C)C)NC(C1CC(=O)C1(C)C)=O N1(C(C(C)OCCC#C)=O)CC(CNC(c2cccnc2)=O)CC12CCOCC2 C(CCC(C)(C)C(=O)NCC1CCC12CCC2)OC.C(=O)(CCC(C)(C)C#N)N C1(COC)CN(C(=O)CCF)CCN1C(=O)CCCc1cnn[nH]1 CN1CCN(C(=O)OC(C)(C)C)C(CC(=O)NCCCCN2CCCC2)C1=O C12(NC(C=C=C(C)C)=O)CCCCCC1N(C(=O)Cc1ccc(F)cc1)CC2 C1(C)(CCNC(CCCC2C(C)C2)=O)CCN(C(c2nnn(C(C)C)c2C)=O)C1 CCCCC(C(=O)NCC1CN(C(C)C)C1)NC(=O)CCCn1cccn1 Cc1c(Cl)cc(C(=O)NC2(CC(F)(F)F)CC2)cc1Br c1(NC(=O)Nc2ccc(CCCC#C)cc2)cc(C)c(I)c(C)c1 Cc1nccc(CCC(=O)NC(Cn2cccn2)C(=O)NCc2csc(C)n2)n1 CC(C)CC(=O)C(=O)N1CCC(C)C1CNC(=O)C#CC1CC1 C=C(C)CC(C(=O)NC1(CCNC(c2cnc(SC)n2C)=O)CCOCC1)OC c1(C(=O)NC(C2(CNC(c3csc(O)n3)=O)CC2)C)cccc(N)n1 CC(CC(F)(F)F)C(=O)NCC1COCCN(C(c2cc(C#N)no2)=O)C1 N1(C(C2CC(OCC)C2)C(=O)NCC2CCOC2)CCNC(=O)C1CC CCC(C)C(C(=O)N1CC(OC(F)F)C1)NC(c1sccc1C#N)=O CC1CN(C(C2CCOCCN2C(=O)CNC(=O)C(C)(C)C)=O)C(C)C1C CC(CN(C(=O)CC1CC2CCC1O2)C)C(=O)NOCc1ccccc1 C(=O)(CCCC(=O)N1CCC(CO)C(NC(C2(CC)CCOC2)=O)C1)NCC c1(C(=O)NCCCC(C)NC(CC2CC(CC)C2)=O)c(C)cnn1C CC1(CNC(=O)CC2CCC2)COCCN(C(c2cc(-c3ccco3)no2)=O)C1 N1(C(C2(OC)CCC2)=O)CCCC(NC(c2ccnn2CC2CCC2)=O)C1 CC(C(C)(C)C(=O)NC(C)CF)NC(=O)COCC1CC1 N1(C(C(=C)F)=O)CCC2(CC(C(=O)Nc3ccc(OCC)cc3)=NO2)C1 Cc1ccc(C(=O)N(C2CCCN(C(=O)C=Cc3cccnc3C)C2)C)c(C)n1 CC1CN(C(c2ccco2)=O)CC1NC(=O)CCNC(c1ccsc1)=O c1(CNC23CCC(n4cc(-c5c(C)ocn5)nn4)(CC2)C3)cc2ccccc2[nH]1 Cc1oc(S(C)(=O)=O)cc1C(N1CC(NC(c2ccoc2C2CC2)=O)C1)=O C(=O)(CC(C)NC(C1CC(N(C)C)C1)=O)NCC(C=C)O n1(CCC(=O)NC2C(CNC(C=NOC)=O)C2)cnc([N+](=O)[O-])c1 N1(C(C(=O)NCCSC)c2nccs2)CCCCC1.N1(C)CCOCC1.C(C)=O Cc1ccccc1C=CC(=O)NCC(O)CCNC(c1cc(O)cs1)=O c1(C(=O)NC(C2CN(C(C3(C(C)C)CC3)=O)C2)C)cc(Br)cc(Cl)c1F CC1C(N=c2cc[nH]cc2S(=O)(=O)NCC=C(Cl)Cl)CCS1(=O)=O N1(C(c2c(C)nccc2)=O)CC(CNC(=O)CNc2ccccn2)CC1(C)C CC(C)CC(C(=O)NOCC1(C)CC1)ONC(C1(F)CCOC1)=O N1(C(C2(C(C)C)COC2)=O)CC(O)CC1C(=O)NC1CCCC1C CC(C(C)C1(C(=O)O)CCC1)NC(=O)CC1CC(C(C)(C)C)C1 N1(C(C2CC(C)CN2C(=O)CN2CC3CC3C2)=O)CCS(=O)CC1C C1(C(C(=O)NC(c2ccnn2C)C)C)CCN(C(=O)CC(C)N(C)C)CC1 C1(C(=O)OCC2C(C)(C)CCO2)N(Cc2ccccc2)CC12CCOCC2 CC(C)(F)C(C)(F)C(=O)NCC12CCC(CC1)OC2.c1(C=O)cccnc1.C N1(C(C(n2c(C)cc(C)n2)C)=O)CCN(C)C(C)C1.c1(C=O)nc(C)c(C)s1.N Cc1cc(=NCCC(O)C2CCCC2)[nH]c(=NCc2ccc(Cl)c(C)c2)[nH]1 N1(c2ccnc(C)n2)CC2CC(CN(Cc3c(Br)ccc(C(F)(F)F)c3F)C2)C1 N1(C(CCOCC#C)=O)CC2C=CC1C(C(=O)NOCC1(C)CCC1)C2 N1(C(C(CC)C#N)=O)CCC2CCN(C(c3cc4ccnc(Cl)c4[nH]3)=O)C2C1 n1(CC(CC)(CC)CO)cnc2c(N3CCC34CCS(=O)(=O)C4)ncnc12 C=CCCC(F)(F)C(=O)N1CCC(N(C)C(c2sc(=N)[nH]c2CC)=O)CC1 c1(C(=O)OCC)cc(C(=O)N(CC(C)C)C)[nH]c1C.C1(C=O)CCN(C)CC1 C1(NC(Cc2ccc(SC)cc2)=O)CCCCN(C(=O)CCCCCO)C1 N1(C(C2C(=C)CC2)=O)CCOC2(C1)CN(C(=O)C=Cc1ccccc1)C2 C(N=C(NC1CCCCC1)NC1CCC2(CC2)C1)C1C(C)(C)C1C(F)F O=S1(=O)CCCC(NC(=NCCc2cccs2)NCC2(F)CCCCC2)C1 Cc1nc2ccnn2c(C)c1C(=O)NC1CC1NC(C1CC1C1(C)COC1)=O N1(C(C2(C)N(C(C3(N(C)C)CCCC3)=O)CC2)=O)CCOC(C#N)C1 C1(CNC(CCCCOC)=O)CN(C(c2cc(Br)co2)=O)C2CCCC2O1 c1(NC2CN(C(C(C=C)(C)O)=O)CC2(C)C)ccnc2nc(C)nn12 C(=O)(CCC(=O)N1CCC(O)CC1)N.C(C(O)C)N(C(=O)CC1CC(=O)C1)C CC1(C)CCCN(C(C2CCC(n3cc(CCS(C)(=O)=O)nn3)CC2)=O)S1(=O)=O N1(C(c2cc(C)nnc2O)=O)CCCN(C(C2CC(=O)C2C)=O)C(C)C1 N1(C(c2cc(C)ns2)C(=O)NCC2CCOC2)CCc2sc(Br)cc2C1 C1(NC(CCOCC)=O)CCCN(C(=O)CN2CCC(CO)CC2)CCC1 Cc1c(C(N2CCN(C(c3cc(CO)[nH]n3)=O)C3CC23)=O)sc2cccc(F)c12 c1(C(N2CC=CC(NC(COCCCC(C)C)=O)C2)=O)cc2ccccc2[nH]1 C1(NC(c2ccc(N)c(Cl)c2)=O)CN(C(C2C=CCC2)=O)C2(CCC2)C1 c1(C(=O)NC2COCCN(C(c3ncc[nH]3)=O)C2)coc2cc(O)ccc12 c1(C=O)[nH]c(C)c(C)c1C.C1(OC)CN(C(c2ncsc2C(F)(F)F)=O)C1.C N1(C(C(=O)NC(c2nncs2)C)=O)CC(N)CC(O)C1 Cc1ccc2c(c1)CN(C(=O)CC(C)CNC(=O)CCc1cn(C)nn1)C2 C1(CNC(CN(C)C(c2cccs2)=O)=O)CCCCCN1C(=O)CC(F)F N1(C(CC2(COC)CC2)=O)CCC(O)(C)C1.C1(CCC=O)CCN(C)C1.N O(N=C1CCCCCC1)CC(=O)Nc1c(OC)ccc(NC(=O)COC)c1 CC1CCC(CNC(=O)C(C)(C)O)CN1C(=O)CCC(=O)Nc1nccs1 Cc1ncncc1C(=O)NCc1ccc(CCNC(=O)C(C)C2CCOC2)cc1 c1(NC(CCCCNC(C)=O)=O)cc(C)cnc1F c1(C(N)=O)ncc(C(=O)NCCOC2CN(C(=O)CC3CCOC3)C2)s1 Cc1[nH]cc(C(=O)NC(C2(O)CN(C(=O)CC(C)F)C2)C)c(=O)c1Cl C(=O)(CCCC)NCC(N(C(C(c1ccccc1F)C)=O)C)C1CC1.C(N)(=O)N C12CCCC(CC1)C(=O)NC1(CC1)CC(=O)N2.c1cccc(Cl)n1.COC C12(C(N(C(C)C)C)=O)CC(CC(F)F)(C1)C2.C(c1cc[nH]c1)=CC=O CCCC(C)C(C)NC(C1(NC(C2CCS2(=O)=O)=O)CCOCC1)=O c1(C(C)CC(=O)NC2CCC(=O)NC2Cc2ccccc2)c[nH]c2ccccc12 c1(C(N(CC(=O)NC(c2ncc(C)o2)C)CC2CC2)=O)cc(O)ncc1F CCC(C)(C)C(O)C(=O)N1CCC(NC(c2cc(C)c(Cl)s2)=O)C(F)C1 CC1(C)CN(C(C2CC(=O)NC(=O)C2)=O)CC1NC(=O)CCN1CCC1 CC(C)C(C(C)NC(=O)COc1ccc(Br)cc1)NC(c1ncn(C)n1)=O N1(C(c2cnc(C)o2)=O)CCC2(CCCC2CNC(=O)CCC(C)N(C)C)CC1 c1(C(=O)NCCC2N(C(c3c(C)noc3)=O)CCOC2)cnc2n1CCC(C)C2 Cc1cc(C)c(C(=O)NCC(C)N(C)CCN2CCCC2=O)c(C)c1 N1(C(CCOCCOC)=O)CC2CCC1CN2C(C1CCC(C)=C(C)C1)=O c12ccc(cc1)o2.C1(C(N2CCC(NCC)CC2)=O)CC2CCC(C1)S2.OC c1(OC)cc(Cn2nnnc2C(C2COC(=O)C2)NCC(C)SC)ccc1Cl N1(C(C(C)(C)c2cc[nH]n2)=O)CCN(CCCNC(C2(C)CCC(=O)C2)=O)CC1 O=C(CCOCCO)NCCCN(C(=O)Cc1ccoc1)C1CC1 c1(-n2cnnn2)ccc2c(c1)CCC2.C12(CO)CCC(C)(CC1)C2.C1CC12CC2.S C(CCN=c1[nH]nc(-c2ccccc2)s1)CCC.C1(CCC)CCCCN1C(=O)C(C)C CC1CCN(C(c2ccc(C(N)=O)o2)=O)CC1C.C1(C2CC2)(C(=O)N)CCC1 N1(C(COCC)=O)CC2CCC2(CNC(=O)Cc2ccccc2)C1.CC.O N1(C(Cc2n(C)ccc2)=O)CCC2(CC1)OCCCC2NC(=O)C=CC(C)(C)C c1(C(=O)NC2C(NC(CCN(C)CC)=O)COCC2)[nH]c(C)c(C(C)=O)c1C N1(C(C(CC(C)C)(C)C)=O)CC2CCOCC2(NC(c2cnc(C(C)C)[nH]2)=O)C1 c1(C(=O)NCCC(C)NC(c2ccc(O)cc2F)=O)cccc(P(C)(C)=O)c1 CC1CCC(NC(c2scnc2Br)=O)CN1C(c1ccoc1)=O c1(C(C)C)nnc2cc(N3CC(NC(c4ccc(F)c(F)c4)=O)CC3C)ncn12 c1(C(N2CCC(c3cccc(OC)c3)(C)C2)=O)ccn2cnc(Br)c2c1 C12(CNC(CSCC(C)C)=O)COC(C)(C1)C2.c1(C=O)c[nH]nc1Br.N c1(SC)cc(Cl)ccc1C(=O)NC1CC1NC(=O)Cc1cnoc1 C12(C(N(CC(=O)NC(COC)CO)CC(C)C)=O)CCCC1C2(F)F N1(CC(c2cc(Cl)sc2Cl)=O)CCC(F)(F)CC1C(=O)O N1(C(c2cnc(C)s2)=O)CC(C)CCC1CNC(=O)C=Cc1cccs1 C=CC(C)(O)CC(=O)NCC(C1CCCC1)NC(c1cccnc1OC(F)F)=O C1(NC(c2cc(C(C)C)[nH]n2)=O)CN(C(=O)CC2CC2(Cl)Cl)C2(CCC2)C1 c1(C(=O)NCC(CNC(C(COC)(C)C)=O)CO)c(C)ccc(Cl)c1F n1(CC)nc(C(=O)NCC2CCN(Cc3cnoc3C)CC2)ccc1=O C(C)(C(N=c1[nH]nc(CO)s1)C(C)C)NC(c1ccc(C)nn1)=O c1(C(CN(C(C)(C)C)C)C)cccc(Br)c1 C1(C(=O)NC(C=CC(=O)N(CC(CCC=C)O)C)(C)C)CC2CCC(C1)C2 C1(NC(C(C)=C2CC2)=O)CCN(C(c2cccc(N)n2)=O)C(c2ccccc2)C1 C=C(Cl)CC(C(=O)Nc1ccc(O)cc1C)NC(=O)C(C)c1ccsc1 C1(OC)CC(C)CN(C(c2cc(CNC(=O)Cc3ccon3)ccn2)=O)C1 C(C1CCN(C(c2nnn(C)c2N)=O)CC1)=CC(=O)N(C)CC1CC1(C)C C#CC1(C)CCCN(C(=O)C(C)(C)NC(=O)Cc2cnccc2C)C1 c1(SC(C(=O)NCCCN(C(=O)C2=CCCS2)CC)C)ccc(N)cc1 C1(CNC(C(CC=CC)NC(=O)Cn2ccnc2)=O)CC12CCCCC2 C1(C(N2CC(C)(NC(c3occc3C3CC3)=O)C2)=O)CNc2ccnn2C1 C(=O)(CS(=O)(=O)C1CC1)N.C1(C(C)C)CCCN1C(c1ncc(C(F)F)s1)=O N1(C(c2c(C(C)C)cco2)=O)CC2(NC(=O)CC3SC(=N)NC3=O)CCC1CC2 Cc1sccc1CC(=O)NCCCN(C(=O)CCC1CC(F)(F)C1)CCO N1(C(c2nn(CC)nc2C)=O)CC(NC(c2n[nH]cc2C2CC2)=O)CC(C)C1 C#Cc1cc(C(N2CC3CC3(C(=O)NCCCF)C2)=O)ccc1C C1(NC(C2(CC=C)CC=CC2)=O)Cc2ccccc2N(C(=O)CCS(C)(=O)=O)C1 c1(C=O)cccc(F)c1C1CC1.C1(CNC(=O)CSC2CC2)CCOCC1 N1(C(C(C)NC(C)=O)=O)CCC2(CCC2NC(c2ncccc2F)=O)CC1 C1(CC(=O)NCC2CCN(CC(=O)NC(CC)C)CC2)CCC(F)(F)CC1 N1(C(Cc2nnc(C)s2)=O)CCC(F)C(NC(=O)CCCOC(C)C)C1 N1(C(C(COCC)C)=O)CCN(C(=O)C(C2CC2)OC)CC1C1CCC1 Cc1cc(C(=O)N(C2CCN(C(C3CCOCC34CCC4)=O)C2)C)c(O)c(C)c1 C1(NC(C(CC)=O)=O)CN(Cc2ncccc2C(F)(F)F)CC1O C(c1cccc([N+](=O)[O-])c1)=CC(N1C2CC(C2)C1)=O.CCC(COC)C(=O)N CS(C)(=O)=Nc1ccc(C(=O)NCC(F)CNC(=O)CC23CCCC2C3)s1 C12(C(N3CCC(N(C)C(C4CC4(F)F)=O)C3)=O)CC3CC(CC(C3)C1)C2 C(=O)(C(O)CC(F)(F)F)N1C(C(=O)NC2C(C)(C)C2)CC2CC21 c1(C(N2C3C(C(=O)Nc4ccc(C)nc4F)C(C3)C2)=O)cc(Br)c(C)cc1O c1(C(C)C)cc(C(=O)N(C2CN(C(=O)CC(C)n3cc(Br)cn3)C2)C)on1 C12(NC(C(C)OCC)=O)CCCC1CN(C(=O)CCc1c(Cl)cccc1Cl)C2 C1(C(=O)NCC2CCC=CCC2)(CNC(Cn2c(C)nnn2)=O)CCCCC1 C#CC1CCCC(NC(C2(CNC(=O)CN3CCCCC3C)CCC2)=O)C1 N1(C(CCCCC=CC)=O)C2CCC1CC(CNC(=O)CS)C2.c1ncc[nH]1.C N1(C)CCC2CCCCCC12.C1(NC(=O)OC(C)(C)C)CC2(C1)NC(=O)NC2=O C(=O)(C#CC(=O)NCC1CCN(C(=O)CC2CCC(=O)O2)CC1)N(C)C c1(C(=O)NC(CNC(C(C=CCCC)O)=O)CC)cccc(C(N)=O)c1N Cc1cnc(C=CC(=O)NCC)[nH]1.c1(C=O)ccsc1C(F)F.C1CC1.N C1(C(N(C(c2ccc(F)cc2)C(=O)O)C)=O)CCCC(O)C1 c1(COc2ccc(CCC(=O)OC)cc2)ccc(Cl)nc1.C(=O)(C1CC1)N CC1CC=C(C(=O)NCC2(F)CC(C)C2)CC1.c1(C(C=O)O)ccc(F)cc1 N1(C(C=O)C)CCCC(O)C1.C1(C(=O)NCCOCC)(COC)COC1 C(CCN=C(NCc1ccsc1C)N1CCC(c2ccccn2)C1)SC CC1CN(C(C2CCCOCC2)=O)CC(C)CN1C(c1nccc(Cl)c1F)=O C#CC1(C)CCCN(C(=O)CCOCCCNC(c2nccc(C)c2N)=O)C1 C12(C(=O)NCC(C(C)C)OC)CC(CN(C(C3CC4(CCC4)CO3)=O)C1)C2 Cc1ccc2nc(C(N3CCCN(C(=O)CSC(C)(C)C)CC3C)=O)ccc2c1 c1(OCC)ncccc1C(C)NC(C1C(C(=O)OC)C1(C)C)C c1(C(CO)NCCS(=O)(=O)NC)cc(C)ccc1C C1(NC(c2ccn(C(C)C)n2)=O)CN(C(=O)C=CC2CCOC2)C2(CCCC2)C1 c1(C=O)cc([N+](=O)[O-])c(C)s1.c1(OC(C(=O)NCCCC)C)ccc(F)nc1 S(=O)(=O)(C1CCOCC1)NCC1CCN(C(c2ccc(C(C)(C)C)s2)=O)C1 c1(C(CC)(C)C)ccc(C(=O)N(C2CCN(C(C3CCSCC3)=O)CC2)C)cc1 C1(CNC(C2CC2c2ccccc2)=O)CCN(C(c2cnsn2)=O)C1 C1(OC)CC2(C1)CC(C(=O)N)C2.c1(C=O)ncnc(C)c1C.C(C)C(C)(C)C CC1CC(NC(c2coc(CNC(c3ccnn3C)=O)c2)=O)CCO1 C1(NC(c2c(C)cccc2)=O)CC(F)CN(C(c2cc(=O)n(C)o2)=O)C1 c1(C(N(C2CCCN(C(C(C)CC3CCC3)=O)C2)C)=O)cccc(=S)n1O N1(C(CSC(C)=O)=O)CC(C(=O)Nc2cc(Cl)cnc2C)CC(F)(F)C1 C1(C(=O)NC2CC(NC(C3(C)COC3)=O)C2)CCC=CCCC1 c1(OC)cc2c(cc1C(=O)NC1C3CN(C(C4(C)CCCN4C)=O)CC13)CCC2 c1(OC)ccc2c(c1)CC(C(=O)NC1CCCCC1NC(=O)C#CC(C)C)CO2 c1(CC(N2CCC(NC(c3nc(C)oc3C)=O)C2)=O)cn2ccccc2n1 c1(NC2C3CN(C(C(N4C(C)CCC4C)C)=O)CC32)ccnc(C#N)n1 c1(C(N2CCC3C2C3)=O)ccc(=O)n(C2CC2)c1.O=C(CCn1cccn1)N.C N1(C(c2c(CC)nn[nH]2)=O)CCOCC1CC(=O)Nc1ccc(C)nc1 C1(C(N2CC(CNC(COCC=C)=O)OCC2)=O)CCCCCS1(=O)=O C1(C(=O)NC(C(=O)N(C(C(N)=O)C2CC2)C)CCF)CC(=O)C12CCC2 N1(C(c2ccc(C(C)C)cn2)=O)CCOCC(NC(C2(C)CCOC2)=O)C1 N1(CC(=O)N(C(C)C=O)CCC)CCCC1=O.C1(CC2CC2)C(=O)N1.N C1(C(=O)NC(C(C)NC(c2ccc(Br)s2)=O)CO)CCCCC(C)(C)C1 N1(C(C2(CC=C)CCCN2C(=O)C(CC)C(C)C)=O)CCC12CCCC2 C1(NC(c2c(C)cccc2)=O)CCC(C)N(C(=O)CCCc2cccs2)C1 N1(C(CCCC=C)=O)CC(C)(C)CCC1CNC(=O)Cn1ccnc1CCC C=CCCCC(C(=O)NCc1cnc(COC)[nH]1)NC(C1CCC(C)(C)C1)=O C1(C(=O)NC(C(=O)NCCc2n(C)ccn2)Cc2cc[nH]n2)CCCCC1(C)C CCC(COC)(CC)C(=O)N(C)CCN(C(C1CNC(=O)CC1C)=O)C(C)C C(C(C)(O)C(F)(F)F)NCC1CC(C#N)(OC)C1 C1(C(=O)NC2CCN(CCCNC(C(CSC)(C)C)=O)C2)CCc2cnnn2C1 C(=O)(CC(C)CC(=O)NCC(C)=CC(N1CCC(OC)C(C)(C)C1)=O)OC C(c1nc2ccccc2s1)=CC(=O)NC(C)CCNC(C1SCCS1)=O Cc1cccc(C)c1OCCN1CCOCC1CO N1(C(C=CC=CCC)=O)CC(NC(c2cc(OC)nn2C)=O)CCC1C C1(O)(C(=O)NCCCN(C(C(c2c(C)n[nH]c2C)C)=O)C)CCC(C)CC1 c1(C(C=O)N(C)CCC2CC2)cc(F)c(F)c(F)c1.c1(OC)ccccc1.C c1(C(=O)OC)ccc(O)c(NC(c2nccn2C)=O)c1.C(=O)C(=O)C(C)C.N C(C(C)(C(=O)N1CCOC(CN(C)C(c2cncc(OC)n2)=O)C1)OC)OC C1(NC(c2c(C)[nH]cc2)=O)CCCCC1NC(=O)CCc1cncc(F)c1 C1(NC(CC2CCC(OC)CC2)=O)CCC12CN(C(c1cc(C3CC3)no1)=O)C2 CC(CCCc1ccccc1)C(=O)N(CCCNC(=O)C)C(C)C.C(N)=O.N C(CN=c1[nH]n2cc(C)nc2s1)(C1CCCCC1)NC(C1(CC)CC1(F)F)=O C1(C(=O)NCCNC(=O)NCC)CCC(C)(C)C1.C(=O)C#CC(C)C CC(C(=O)NN(c1ccccc1)c1ccccc1)N(C)Cc1ccccc1 Cc1cccc(C(=O)NCC2CCN2C(=O)COc2ccccc2F)c1 C1CN(C(=O)C=C(C)C2CC2)CCC1C.[nH]1nc(C=O)cc1C(F)(F)F.CC c1(C(=O)NC(CNC(c2ccc(O)cn2)=O)C2CC2)ccc2ocnc2n1 CCCCCCCCN(C(=O)C(n1cc(CN2CCCC2C(=O)O)nn1)C)C Cc1cc(C(=O)N(C2(CN3CCC(N4CCCC4)C3)CSC2)C2CC2)nc(O)n1 CCCCCC(O)C(=O)N1CC(F)(C(N2CCCC(C#N)C2)=O)C1 C1(NC(C2(C(N(C)C)=O)CC2)=O)CN(C(c2ccc(CO)o2)=O)C2CCCC12 C(CCC(C)C(=O)NC1COCC1NC(c1c(Cl)n[nH]c1C1CC1)=O)OC N1(C(c2c(C)csc2)=O)CCC=CC1C(=O)NCC1(C)CCCCC1 CC(C)(C)CC(F)C(=O)NC1CCC(C(=O)NC2(C)CS(=O)(=O)C2)C1 C(CNC(=O)C=CI)(C(C)(C)C)NC(C1C(C)C1)=O c1(C(=O)NC(CC)CNC(=O)CCc2cncn2C)ccc(CC(=O)NC)cc1 C(C1CCCCC1)=C(C(=O)NCC(C1CCC1)NC(c1cc(Br)no1)=O)F N1(C(C(COC)OC)=O)CC2CC2(NC(c2cc(Cl)c(Br)[nH]2)=O)C1 c1nc(NCC2CCC3(CCC3)CC2)cc(=NCC23CC(CN2C2CC2)C3)[nH]1 c1(OC)c(C(=O)NC2CCC(NC(c3[nH]nnc3C)=O)C2)cccc1Br c1(NC(CN(CC(C)C)C(c2ccon2)=O)=O)ccc(Cl)cc1 N1(C(C=CSC)=O)CCN(C(=O)Cn2cnc(C(F)(F)F)n2)CC1C N1(C(Cn2cc(C(=O)OC)nc2)=O)Cc2cnc(Cl)cc2C1 Cc1ncc(Br)cc1NC(c1nc(-c2ccc(Oc3ccccc3)cc2)cs1)=O C(=O)(C(F)(F)C(F)F)N1CC(C(N)=O)C1.[nH]1nc(C2CC2)cc1C=O.CC c1(C(=O)NCC2(OC)CN(C(=O)C3=CCCC3)C2)ccn(C2CC2)c1C CC1CN(C(c2cc(Br)n[nH]2)=O)CCC1NCc1ccc(-n2cccn2)cc1 CC(C(=O)NCCCCCC(=O)N1CCN2CCC1C2)S(N)(=O)=O CCCCC(C)(F)C(=O)N1CCN(C(C2CCC(C(C)(C)O)CC2)=O)C(C)C1 C(CO)(C(C)NC(C1CCOC1)=O)NC(C(C)SCCCC)=O CCCCCCC(F)C(=O)NC1(CNC(c2cc(C3CCC3)no2)=O)CCOC1 C1(CN(C)C(C2CSCCN2C(c2cn(C)cn2)=O)=O)(CO)CC(C)(C)C1 c1(-c2c(C)csc2)ccc2cc(C(=O)Nc3cccc(C(C)O)c3)cn2c1 C=CC1(C(=O)Nc2cccc(F)c2O)CCN(C(=O)C(CCC)OC)C1 C(=O)(C(F)(CNC(=O)CCC1CCCC1)C(C)C)NCc1cc(C)c(C)nn1 CCC(CC(C)C)C(=O)NC1CN(C(=O)CC#N)CC1N=[N+]=[N-] N1(C(CCCSC)=O)CC2COCCC2(NC(=O)CSCc2cccnc2)C1 c1(NC)ccccc1C(=O)NC.c1(C=O)ccnn1CCN(C)C.C1CC1 C(=O)(C1CC(=O)Nc2ncccc21)NC(C)CNC(c1ccc(C(F)F)cc1)=O c1(C(=O)NC2CC(N(C(Cc3c(C)ccs3)=O)C)C2)ccc(N)c(F)n1 C1(CNC(CCCOCC=C)=O)CCC2(CCC2)CN1C(c1coc(C)c1)=O c1(C(N2CCC(C(C)(C)C)C2)=O)cc2nn[nH]c2cc1F.C(C(=O)NC)=C(C)Cl CCCCCCC(C)CC(=O)NCC(O)CN(C)C(c1cc2n(c1)CCCC2)=O CC1CC(NC(=O)CC2(O)CCOCC2)CN1C(=O)C=Cc1nccs1 C1(C(=O)NCC(CC=C)NC(c2ccc(F)s2)=O)CC2(CCOCC2)CO1 N1(C(C(C)NC(C)=O)=O)CC2CCC2(NC(=O)CN2CCOC2=O)C1 C1(C(=O)NCC(O)CC)(OC)CCCOC1.C1(C=O)CCC1.[SH](C)(=O)=O.N C(=O)(CC(CN(C)C)C(F)F)NC.N1(C(COCCCOC)=O)CCCCC1.C Cc1ccc(C)c(C(N2CCC(C)(CC(=O)N(C)Cc3ocnc3C)C2)=O)c1 c1(C(=O)NC(C)CCC(=O)NCCc2ncnn2C)nccc2[nH]ccc12 C=CC1(C(=O)NC2CCN(c3ccc(C)cc3)C2=O)CCCN1 Cc1ccn(C)c1C(N1CC(NC(C2CC2C(C)C)=O)C1)=O C(C)(C(C)C(=O)NCc1cc(C2CC2)n[nH]1)NC(Cc1cnc(C)s1)=O C1(NC(c2ccc(-c3nn[nH]n3)cc2O)=O)CCC2(CCCNC2)C1 c1(C(=O)NCC2CCC(NC(C(CN(C)C)(C)C)=O)C2)cccc(O)c1Cl c1(C(N2C(CC)C(NC(=O)C=CC(C)(C)SC)CC2)=O)cc2ccccc2o1 n1(CC)c(C(N2CC(=C(F)C)C2)=O)cc2ccccc12.C(=O)C1=NNC(=O)C1 C(=O)(CCC(F)F)N.C1(COC)(C)CCC1.C1(Cl)(C=O)CC1C(C)=O c1ccc2c(c1)CN(CC1CCCOC1)c1ccccc1S2 C1(CC)CN(C)CCCN1C(C1(C)CCCN(C(=O)CCCC(C)(C)C)C1)=O C(=O)(C(C)(F)C(=O)NC1CC(CC(=O)NC(C)C(C)SC)C1)OC c1(C(N2C(C(C)(C)NC(c3c(CC)nns3)=O)CCC2)=O)cccc(C)c1F C1(C(N2C(C)CC(NC(Cc3c(C)noc3C)=O)C2)=O)CN(C)CCN(C)C1 C12(C(N3CC(CNC(c4c(C)n(CCC#N)nc4)=O)C3)=O)CCOC1CCOC2 CC(CNC(c1cccnn1)=O)C(=O)NC(C)(C)CC1CCOC1 C(C(CC(F)(F)F)NC(c1cc(O)ccc1Cl)=O)NC(C1(C)CC1)=O C1(C(N(CCC(C)NC(=O)CC2(O)CCC2)C)=O)CN(C(C)C)CCO1 C(CCCC(=O)NCc1ncoc1CCNC(c1sccc1)=O)OC.C1CC1 Cc1cc[nH]c1C(=O)N(C)CCN(C(=O)C(C)NS(C)(=O)=O)C(C)C c1(C(N2CC(NC(=O)C#CC3CC3)CC(C)C2)=O)ccc2c(c1)NC(=O)CCS2 c1(C(N2CCC(C)(CC(=O)N(CCC=C)CC)C2)=O)ccc(F)c(O)c1 CC(C)C(C)C(=O)NCC1CCCN1C(C1(C)CCC1)=O C1(NC(C2CCN(C)CC2)=O)CCN(C(=O)C2=CC3CCCC23)CC1(C)C C1(NC(c2cccc(Cl)c2Cl)=O)CC2CCC(C1)N2C(C1(F)CCOC1)=O C1CCC(=O)N(C)C1=O.Cc1nc(O)sc1C(=O)NC(Cc1cc[nH]n1)C=O.N N1(C(CC(C(CC)(C)C)C)=O)C2CCC1c1ccccc12 C1(CNC(CN(CCC#C)C)=O)CC(NC(=O)CCc2ccccc2F)CCO1 c1(NC(CC(C)N)C)ccnc2cc(C(F)(F)F)ccc12 CCC(C)CC(C)C(=O)N1CCC(C)(C)C1C(=O)NC1(C(=O)N(C)C)CC1 c1(C(C)C)ccc(NC(C2CC(C)N2C(=O)CCc2cccnc2)=O)cn1 C1(CC(=O)N(C(CO)CO)CC)CC(NC(=O)CC)C1(C)C.C1CCOCC1 C(=O)(C(CNC(=O)C=CCC)C(C)C)NC(CC#C)CCOC c1(NCC)cncc(C=O)c1.C(C)CC(C)C.C1(C=O)CC1C(F)(F)F.N Cc1cc(F)c(C(=O)NCC=CCNC(c2cccn3ccnc23)=O)cc1Br Cn1cc(CCCNC(C2CCOC2CNC(=O)CN2CCCC2=O)=O)cn1 c1(OC)cc(C(=O)Nc2cc(C(=O)Nc3cccc(I)c3)n(C)c2)cnc1Cl c1(C(N2CC(CCc3cn(CC4C(=C)CC4)nn3)C2)=O)ccc(C2CC2)cc1 C1(C(C)NC(=O)CCC2COCCO2)CCN(C(=O)Cn2ncn(C)c2=O)CC1 N1(C(c2cc(OC)no2)=O)CCCC(C(C)C(=O)N2CC(CC(C)C)C2)C1 N1(C(c2nnc(C)s2)=O)CC2CCCCC2(CNC(C2(C)CCCCC2)=O)C1 CCC(CNC(=O)CCCN(C(=O)CC1CCCO1)C)(CC)CO N1(C(=O)CC2CC2(Cl)Cl)CCCN(C(=O)C2=CCS(=O)(=O)C2)C(CO)C1 c1(CC(=O)NCCCC)cc(OC)c(O)c(OC)c1.C1(C=O)CC(O)CN1C.N C1(C(N(CC(=O)OC)CC#C)=O)CC2CC2N1C(=O)CC1CCCO1 Cc1cccc2cc(C(N3CCN(C(c4ccc(I)c(Br)c4)=O)C4CC34)=O)[nH]c12 c1(C(N2CCOC(c3ccc(F)cc3)C2)C(=O)NCC)ccc2nc(C)sc2c1 N1(CC)CCN(C(=O)C(n2cc(CC(C)O)nn2)C)CC12CCOC2 CC1CN(C(c2cccc([N+](=O)[O-])c2)=O)CC(C)N1C(c1cc(Cl)cc(Br)c1)=O C1(Cc2c(C)cccc2)CN(N2CCOC(Cc3ccccc3)C2)C1 O=C1CCCC(CCC(N2CCOC(CNC(c3cc(O)ncn3)=O)C2)=O)N1 N1(CC(=O)N(C)C)CC(=O)NC1=O.n1(CCCC)nccc1C(N1CCCC1)=O O=S(=O)(c1ccc2nc(N3C4C=CC(C4)C3CO)sc2c1)N1CCSC1 C=CC1(C(=O)NCC2CC(F)(F)CN2C(c2ncc(C)s2)=O)CCCCC1.O Cc1c[nH]nc1C(=O)NC1(C2CCCN2C(c2coc(Cl)n2)=O)CC1 C(c1ccc2c(c1)OCO2)=CC(N1CCC(C2CCCN2C(C2CCC2)=O)C1)=O C1(C(=O)N)C2C3CC4C1C1C2CC3C41.CC(C(=O)NC1CC(C)C1)N(C)C CC(C)=C=CC(=O)NC(C)(C)CC=CC(=O)NCCSC(C)(C)C c1(C(N2C(CNC(C(COC)OC)=O)CCC2)=O)ncn2c1CCCCC2 c1(C(C)C)oncc1C(=O)NCC1CC(C(=O)N)C1.c1(C2CC2)ccoc1 C(c1ccc(Cl)s1)=CC(=O)N(CC(CC)NC(c1cncnc1)=O)C c1(C(C(=O)NCCC(C)NC(C2CCCO2)=O)C)cccc(O)c1 C(=O)(C1CCc2nccn21)NC1(c2ccccc2)C(C)(C)C1 C1(NC(C(C)(C)F)=O)CCCC(NC(C2(C)CCNC2=O)=O)C1 c1(OC)nc(=NC(CNC(=O)C(C)NC(N)=O)C(C)C(C)C)[nH]c2[nH]cnc12 N1(C(C2(CC#C)CC2)=O)CCC(C2CCN(C(c3cc(Br)nn3C)=O)C2)C1 c1(C(C)C)ncncc1C(N1CC(CNC(c2c[nH]nc2Br)=O)C1)=O C(=O)(CCCS(C)(=O)=O)NC1CC(CNC(C2CCC(C(C)C)CC2)=O)C1 N1(C(CCCC=C)=O)CC2CCN(C(c3ccc(C)c(O)n3)=O)CC12 CC1c2ccccc2OC1CC(N1CCCC(CNC(=O)C2=CCOCC2)C1)=O C(CC1CCC1)(C(=O)N1CSCC1C(=O)NCC(c1cn(C)cn1)O)OC C1(C(=O)NCCN(C(=O)C)CC)C2(CC2)C12CC2.c1nnc(S)s1.S C1(C#N)(C(=O)NCC2N(C(C(CN(CC)CC)F)=O)CCC2)CCCCC1 N1(C(Cc2c(C)occ2)=O)CC(NC(=O)CC2CCC2)C(C(F)F)C1.C1CC1 N1(C(C(CC)(F)F)=O)CC(CNC(=O)C(C)CCCOC)OC2CCCC12 C#Cc1cccc(C(N2CCC(C(F)F)(CNC(=O)CC3CC3)C2)=O)c1.O C1(NC(c2ccc(CCO)cc2)=O)CC2CC1CN(C(c1cccnc1)=O)C2 N1(C(C(C2(O)CCC2)NC(CCCOCCC)=O)=O)CCC2(CCO2)C1 c1(C(=O)NCCC(=C)C)ccc(F)c(CC)c1.c1(C=O)nocc1C(C)C.N C1(C)(NC(CCc2nc(C)c(C)[nH]2)=O)CCN(C(C2CC23CCOC3)=O)CC1 C(C(CO)C(C)(C)C)NC(C1CC(C)(NC(Cn2ncc(C#C)c2)=O)C1)=O c1(SC(C)C(=O)NCC2(NC(=O)Cc3nc[nH]n3)CC2)nncn1C C(=O)(C1=NOC2(CCOC2)C1)N1CC2C(NC(C=Cc3c(C)nccc3)=O)(C2)C1 CCCC(C)(O)CC(=O)N1CCC(O)(CCNC(=O)Cc2nccs2)CC1 c1(C(=O)NC2(CCNC(C3CCCOC3)=O)CC2)ccc(C(O)CF)cc1 c1(SCC(=O)OC)cc2c3ccnc2cc1N3.c1(C(=O)OC)ccccc1 C1(NC(CN(C(C=CC(C)C)=O)C)=O)CC2CC1OC(=O)N2 Cc1cc(NC(=O)CC2CCCCC2O)ccc1NC(=O)CC1CC1 C(C(C)(C)C1=CCCC1)NC(=NCCN1CCN(C)CC1)NCC1CCCCO1 C1(CC(=O)N)NC(=O)NC1=O.C1(N(C(=O)C(F)C2CCC2)C)CC2CCC1O2 N1(CCC(=O)NCC(C)CNC(C2(N(C)C)CCC2)=O)CCOCC1=O CCCCC(CN=c1nc(O)c2ccccc2[nH]1)NC(C1CC(SC)C1)=O C(C(N=[N+]=[N-])C(=O)NCC(O)CC(N1CC2(CCN2C)C1)=O)OCC C#Cc1ccc(OCC(N2CCC3CN(C(=O)C(F)C(C)C)CC23)=O)c(OC)c1 C=CCC(C)(C)CC(=O)N1CCC(C(C)NC(=O)C(c2ccc(F)cc2)C)CC1 CC1CN(C(c2cnccc2Cl)=O)CC1NC(=O)COCc1cccc(Cl)c1 C1(CC(=O)NCCCCCCNC(=O)CCn2ccccc2=O)CCCCC1O C1(C(=O)NC2(C)CN(C(C(CC)NC(C)=O)=O)C2)CC2(CCC2)C1 C1(NC(=O)NC2CN(c3ncc(CC)cn3)C2)CC2(C1)CC21CC1 c1(C(=O)NC(C)CC(C)NC(=O)Cc2cccc(C3CC3)c2)ccc(Cl)nn1 c1(C(=O)NCCC2CCC(C)O2)nc2ccccc2nc1O N1(C(c2cc(OC)cc(C(=O)OC)n2)=O)CCCC2CCCC12.C(=O)(C(N)=O)N N1(C(C2C(C)C2)=O)CCC(C)(C)C(NC(c2nn(C)c3c2CCC3)=O)C1 CCCCCC(CCCCC)C(=O)NC1CC1NC(=O)C(C)(O)C1CC1 c1(NC(CC(C)(C)C2CCCCC2)=O)sc2c(c1C#N)CCCC2 C12(C(=O)NCC3N(C(c4cscn4)=O)CCN(C)C3)CCOC1CCOC2 C1(NC(c2c(CC)c[nH]c2)=O)CN(C(c2ccc(C)nc2N)=O)CC1(C)C c1(OC)ccc2c(c1)C=C(C(=O)NCCC)CO2.c1(C=O)cnn(C2CC2)c1.N Cc1ccc(N)cc1-c1cn(C2COCC2Oc2ccccc2)nn1 C1(CNC(c2sccc2Cl)=O)CCC2CN(C(C34CC(F)(C3)C4)=O)CCC2C1 C(=O)(CCC(C)CN(C)C)N(C1CN(C(c2ccc(OC)cc2)=O)CC1O)C N1(C(C(CSC)C)=O)CC(CNC(c2csc(C(C)(C)C)n2)=O)C(C)C1 C1(NC(C2CC23CCN(C(C2CCCC(O)C2)=O)C3)=O)CC2CC1C(O)C2O C1(NC(Cn2c(C)ncc2)=O)CCN(C(=O)C(C2CCOCC2)O)C12CCC2 CON(CCC(=O)NCC(C)(C)C(C)O)C(=O)C(C)c1ccnn1C CN1CC(C(=O)NC23CC2CN(C(c2ccc(Cl)cc2)=O)C3)CC1=O Cn1nnc(CNC(=O)CC2CCOC2=O)c1C(=O)NC1CCNC(=O)C1 C1(CNC(C(C)=CC2CC2)=O)CCCC12CCN(C(c1cnsc1)=O)CC2 N1(C(c2cc(OC)ncc2)=O)CCOC2CN(C(=O)CCC(N)=O)CC12 CC12CCC(C)(O1)C(C(=O)NCCNC(=O)COc1ccccc1)C2 Cc1nc2[nH]ccc2c(=NCCCCCCN(C(=O)C(C)CCN(C)C)C)[nH]1 C1(C(N2C(C(=O)Nc3ccc(OC(C)C)nc3)CC2)=O)CCC2CCC(=O)N2C1 O=C1CNc2nc(C(N3CC4=C(C3)CN(C(c3ccc(Cl)s3)=O)C4)=O)ccc2N1 C1(C(=O)NC(C)(C)CCCO)CCC2CCC1N2C(=O)C1=CCSC1 C(c1ccc(Cl)cc1)=CS(N1CC(C#N)(C(=O)OC)C1)(=O)=O C1(CNC(C2CCC(=O)N2)=O)COCCN1C(=O)Cc1ccccc1Br c1(NCC2CCC(OC)CC2)[nH]c(=NCc2cccs2)nc2c1cnn2C N1(C(CCCCC(OC)OC)=O)CCCC2(CCN(C)C2=O)C1 N1(C(c2n[nH]c(C)c2C)=O)C2CCC1CC(NC(c1cc(C(N)=O)cn1C)=O)C2 c1(CC(=O)NC2C(C)N(C(=O)C=C3CCC3)CCC2)n[nH]c2c1CCCC2 C1(CNC(CN(C2CC2)CC)=O)CCCN1C(=O)CC1CCCC1O.C c1(C(=O)NCCCC=C)cn2cc(C)sc2n1.c1(C=O)nnn(C(C)(C)C)n1.N C1(C(c2n(CCC)nnn2)NCC2(C)CCCC2)CC(C)(C)OC(C)(C)C1 Cc1nc(NCc2nnc(C)n2C)cc(=NCC2CCCS(=O)(=O)C2)[nH]1 C1(NC(C(CC)COC)=O)CCOC12CCN(C(C1(Br)CC1)=O)CC2 c1(C(=O)NCC(CNC(c2ccc(CO)cc2)=O)O)cc(Cl)cc(Br)c1 c1(C(N2CCCC(NC(C(CC)F)=O)(CO)C2)=O)cn(C)c(=O)n(C)c1=O C1(NC(C2CCC(OC)C2)=O)CCC(NC(=O)CC(C)N2CCCC2=O)CC1 c1(C(=O)NCC(CNC(c2c(C)nc(C)s2)=O)C)ccc2ccn(C)c2c1 Cc1ccc(O)c(C(=O)NC2CC23CC(NC(C2OCCCC2(C)C)=O)C3)c1 C1(C(=O)OC)(CNC(COCC)=O)C=CCN1C(=O)CNC=O N12CCC(O)C(C1)C(=O)N(CC(C)(C)C)CC(O)Cn1cc(nn1)C2.CO CC1C(=O)NCCN1C(c1cccc(-c2ccnc(C(=O)O)c2)c1)=O c1(NC(C)Cc2cnccn2)nccc(-n2cccn2)n1 N1(C(Cn2c(C)c(Cl)cn2)=O)CCC(NC(c2cc(Cl)n(C)n2)=O)C(C)C1 N1(C(c2c(C)cc(F)cn2)=O)CCc2c(CNC(=O)C=C(Cl)Cl)cccc2C1 C(=O)(C(CCc1ccsc1)N1CCC(N2CC(=O)NC2=O)CC1)NCC(=C)C C(=O)(CCC(C(C)C)NC(c1cccc(O)c1F)=O)N(CCCCC)CCO CCCCC(C(=O)N1CCN(C(c2ccon2)=O)CC1CC(=O)NC)C(C)C C1(NC(c2cc(C)[nH]n2)=O)CN(C(=O)C(C)(C)Cc2cnn[nH]2)CC12CC2 C(CN=c1[nH]c(=NCCc2cnccn2)[nH]c2cccnc12)N1CCC(OC)C1 C1(F)(CNC(C(C(C)C)O)=O)CCN(C(=O)CC(O)c2ccccc2)CC1 c1(C(N2CCCC(CC=C)(NC(=O)CC=CCC)C2)=O)cccc(Cl)c1[N+](=O)[O-] c1(C(N2C(CNC(C3CCC(=O)N3)=O)CCC2)=O)ccc(OC(F)F)cc1 c1(NC(=O)NC(C(C)SC)C)ccc(F)c(I)c1Cl C1(CNC(C(CC(C)C)N(C)C)=O)CC2CCC1CC2.c1(C(=O)N)cnn(C)c1 c1(C(=O)N)cnn2ccnc(C)c12.N1(C(CSCC#C)=O)CCC(CCOC)C1 Cc1ccc(CO)cc1NC(C1(F)CCN(C(c2cnsc2)=O)C1)=O C#Cc1cc(NC(C2(C#C)CCN(C(C3CCC(C)(C)C3)=O)CC2)=O)ccc1C Cc1ncc(C(N2CC3CCC3(CNC(C3(F)CCC3)=O)C2)=O)c(C)n1 C(=O)(C(C)C(=O)OC)N1C(CN(C(c2csnc2C)=O)CC)CCC1 c1(C=O)ccc(F)c(F)c1F.N1(C(C(C(C)C)N(C)C)=O)CC2(CCC2C)C1.N C1(NC(c2ccncc2)=O)CN(C(C2(C3CCC3)CC2)=O)CCC1CO C(=O)(C(C)S(N)(=O)=O)N1C(CC(=O)NCC#CC)CCC1 c1(C(=O)NC(CC)Cn2cncn2)nnc(S)n1C.C12(CC1)C(=O)NC2C CCC(CN(C)C)C(=O)NCC1(F)CN(C(c2cc(N)ccn2)=O)C1 C#CCC(CC(F)(F)F)NS(=O)(=O)NCC(C)C C1(OC)CCCC(C(=O)NCCCCNC(c2c[nH]cc2C)=O)C1 Cc1cnc(C(=O)NCC(C)(C)CC(=O)N2CC3CC3(CO)C2)cc1C CC(CO)CCNC(CCSC)(c1nnnn1C1CC(F)(F)C1)C1CC1 C1(CC(=O)NC(CC)C)OCC2CN(C(=O)C(c3ccc(C)cc3)C)CCC12 c1(C(=O)NC(C(C)NC(C(C2CC2)OC)=O)(C)C)ccc(N)c(N)n1 c1(N2CC(CCCCNC(C(C)CC3CCCC3)=O)C2)ncc2ncn(C)c2n1 Cc1cccc(-n2ncc(C(=O)NCCN3CCC3)c2C)c1 C(CC(C(=O)N=S1(=O)CCNCC1)NC(=O)OC(C)(C)C)c1nc(C)sc1 CCC(C(=O)NCCC(C)NC(=O)C(C1(OC)CCOCC1)(F)F)C(F)(F)F c1(C(=O)NCC2(NC(c3cnc(CC)s3)=O)CCCC2)csc(C#N)c1 N1(C(COc2cc(C)on2)=O)C(C)C2CC1C2NC(=O)C(C)(C)C1CC1 C1(CN(C)C(c2cnc(O)s2)=O)CC(F)CN1C(C1CCCN1C=O)=O C#Cc1cccc(C(N2CCCC(C)(CNC(=O)C(C)C3CCC3)C2)=O)c1 S(=O)(=O)(c1c(C)c(C)cc(C)c1C)N1CCCC(CC)(NC(C2CCCN2)=O)C1 c1(SC)ncc(Br)c(N2CCC3(CC3C(N3CCCC(O)C3)=O)C2)n1 c1(C(C)=O)ccc(C(N2CC(CN3CC(C)OC(C)C3)CC2(C)C)=O)cc1C#N c1(CC)cc(C)ccc1C(=O)NCC(C1CC1)NC(C1(C)CCCN1C)=O N1(C(C2(CCCC)CCC2)=O)CC2CCCC2(NC(=O)CCc2cc(Cl)cs2)C1 C12(C(=O)NC(C3CN(C(=O)CC=C(Cl)Cl)CCO3)C)CC=CC(C1)OC2 C=CCCCC(C(=O)NC(c1nnc(O)o1)C)NC(=O)C(F)C(=O)OCC N1(C(c2cnc(CC)s2)=O)CCC(CNC(=O)CCc2cc(C)on2)C(C)C1 C12(NC(CC3(CC)CCC3)=O)CCCC1N(C(C1CC(C(=O)O)C1)=O)CCC2 c1(C(N2CC(NC(C3CC(=O)NC3)=O)C(O)C2)=O)cc(Br)c(F)cc1F C(=O)(C(CCCC(=O)OC(C)(C)C)N(C)Cc1ccoc1)NCCSC c1(C(N2CC3C(NC(C(C)NC(N)=O)=O)(CCC3)C2)=O)cc2cc[nH]c(=O)c2s1 c1(C(=O)NCC(C)(CO)NC(=O)COC2CCCCCC2)cn2ncccc2n1 CCCCC(C)C(=O)N1CC(CC(C)(C)CNC(C2(OCC)CCOC2)=O)C1 C1(CCNC(C2COCCOC2)=O)CSCCN1C(c1ccnnc1)=O S(=O)(=O)(c1cccnc1NCC12CCCC(CO1)C2)N1C2CN(C)C(C2)C1 c1(C(N2CCN(C(c3ccc(C)s3)=O)C(CO)C2)=O)cncc2c(Cl)cccc12 c1(C(N2CC(NC(C3C4CCCC34)=O)CC(C)(C)C2)=O)ccc2ncccc2c1 C1(C(C)(C)NC(C=C(CC)C)=O)CCCN1C(=O)COCc1ncno1 CCC(CC(=O)NCCC(C)N(C)C(c1cnc(SC)nc1O)=O)C(F)F C(C)(CCCCCO)NC(CC(C)N(C(CSCCCC)=O)C1CC1)=O C1(C(N2CCC(C(=O)NC3CCN(C)C3)(OC)C2)=O)CC2(C1)CC(C)C2 Cc1cnc(F)c(C(=O)NC2(CNC(=O)C)CCOCC2)c1.c1ccccc1.O N1(C(c2ccc(C#N)cc2)=O)CC2(C1)CN(C(C1CC13CC3(F)F)=O)CCO2 c1(C(N2CCN(C3CC3)CC2)=O)ccc2nc(-c3cnc4n[nH]cc4c3)sc2c1 Cc1cc(F)c(C(=O)NC(CNC(=O)CN2CCN(C)CC2)CO)cc1F c1(C(N2CC(CNC(=O)COC3CC=CC3)C3C2C3)=O)ccc2scnc2c1 CCCC(C(=O)N1CCCC1(C)CNC(=O)CCSCC(C)C)C(C)C C(CCCC(=O)NCC(C)CC(=O)NCC1CCC1)(OC)OC N1(C(C)(C)C)CC(C(=O)NCC2COCCN2C(C2CCC(F)CC2)=O)CC1=O c1(CC(=O)NCC(=C)CCNC(=O)C(c2cccnc2)C)c(C)ncnc1C C1(COC(C2C3CCC(O3)C2C(F)(F)F)=O)CC2(C1)CC(F)C2 CC(C)(C#N)CC(=O)NC(CC(F)F)C(=O)NCC(O)CC(F)(F)F N1(C(CN(C2CCSC2)C)=O)CC(NC(=O)C=CBr)C1 C(C)(C)(C(C)(C)CO)NC(C1(F)CCN(C(CCNC(=O)NC)=O)C1)=O c1(CC)nc(=N)[nH]cc1C(N1CCC(C(C)(C)NC(C2CC=CCO2)=O)C1)=O N1(C(C2CC=C(C)CC2)=O)CCC2(CCC2NC(=O)C(F)CC(C)C)CC1 c1(CC(=O)NCCNC(=O)CC(C(F)F)n2cccn2)ccc([N+](=O)[O-])cc1Cl C12(C(N3CCN(C(C4Cc5cccnc5C4)=O)CC3)=O)CCCN1S(=O)(=O)CC2 CC1CCN(C(=O)CN2CCN(CCO)CC2)CC1NC(C1CN(C)C(=O)N1)=O C(=O)CCCn1ccnn1.C(C)(C)CN(C(=O)C=CCC1CCC1)C.CO c1(C(N2CCCC(N(c3nccc(OC)n3)C)C2)=O)ccc(=O)n(C)c1 c1(CNC(C(C)SC)=O)cc(C(=O)NCc2[nH]cnc2C)co1 N1(C(CC(CC)C)=O)CC2N(C(=O)C(O)CCN(C)C)CCC2(C)C1 Cc1c(C=CC(=O)NCCCCC(C)(C)NC(C2CCC(F)C2)=O)cnn1C C1(C(=O)NC2CCN(C(c3cc(C)sn3)=O)C23CC3)CCCC12CCOCC2 c1(C(=O)NC2C(CNC(C=NOC)=O)CCC2)cc(O)ccc1[N+](=O)[O-] C1(N(C(C2C(CCC)C2)=O)C)CCCCN(C(c2cnc(NCC)c(Cl)c2)=O)C1 C(CCNC(c1cnoc1)=O)(C(C)C)NC(c1c(CC)noc1)=O C(=O)(CC(CN(C)C)C(F)F)NC1C(C)N(C(=O)C2=CCCCO2)CC1 c1(N2CC(CN(C)C(C3CCC(=O)N3)=O)C2)nc(Cl)ncc1C(N)=O N(C1c2ccccc2CCC1F)C1CCN(CCCO)CC1 c1(C(=O)NCC2N(C(CSCCN(C)C)=O)CC2)ncsc1C(=O)O C(CCN=c1cc2c(n[nH]1)CCC2)OCC c1(C(N2CC(NC(C3CCN(C(CC)=O)C3)=O)C(C)C2)=O)cc(OC)nc(Cl)c1 C1(NC(CCc2ccc(C#N)cc2)=O)CCCC12CCN(C(C1CCC1)=O)C2 C1(CNC(CCOCCC)=O)CCCCN(C(=O)C=Cc2cscn2)C1 C(CN=c1[nH]c(=NCC2CCCS2)[nH]c2cc(C)ccc12)c1cc(OC)ncc1 C(C(C)CN=c1cccc(S(=O)(=O)N2CCn3cc(C)nc3C2)[nH]1)OC CC1CCN(C(=O)CCN2C(=O)CCC2=O)CC1C.C(=O)C(C)(C)CN(C)C C#CCC(C)(C(=O)NC(c1ncc(C)[nH]1)CC)NC(=O)CC1CCC(C)CO1 C(=O)(CC(C(C)C)C(C)C)NC1CC(CNC(C2(CC)CC2)=O)OCC1 C1(C=O)CC2CCCC(C1)N2.CC1CC(CS(C)(=O)=O)CN1CC.C(C)(C)C.N C(=O)(CCCCCC#N)N1CCC(O)(CN(C(COCCC#C)=O)C)C1 C1(NC(CP(C)(C)=O)=O)CC(NC(c2ccn3ncccc23)=O)C12CCOCC2 Cc1ccc(S(=O)(=O)N(CC=O)C)cc1.C12CC(C1)N(C(=O)C)C2.C(N)=O c1(-c2cn(CC3CN(C(C4COCC4c4ccccc4)=O)C3)nn2)cccc(Cl)n1 Cn1nc(C(N2CC(CNC(=O)CC3CC4CC4C3)C2)=O)cc1.C1CC1.C c1(C(N(C2CCN(C(=O)C3=CC(O)CCC3)CC2)C)=O)ccc2c(c1)COC2=O C1(C)(OC)CN(C(=O)CC2CCCN2C(=O)Cc2cn(C)nn2)C1 C(=O)(CCC(C)(C)[N+](=O)[O-])NC(CNC(c1ccc(OC)s1)=O)C Cc1cc(Cl)c(Cl)cc1C(=O)NCCC(O)CNC(=O)C(C)Cc1ccco1 c1(C(N2CCC3(CN(C(CN4C(C)CC4)=O)C3)C2)=O)ccccc1S(C)(=O)=O C(CCC(=O)N1CCC(C(C)NC(c2csnc2Cl)=O)C1)=C(C)C Cc1ncnc(C)c1C(=O)NC1(C(F)F)CCC1.C1(C(=O)N)CCNC(=O)C1 c1(C(=O)NC(C2CCN(C(c3[nH]cc(C)c3)=O)C2)C)cccn2ncnc12 Cc1cnc(C(=O)NC2(C)CC(NC(=O)C(F)F)C2)c(Br)c1 c1(CCN(C(=O)C(CC2CCCC2)NC(=O)CC2COCCO2)C)cnccn1 C(C1CN(C(c2ccc(F)cc2F)=O)CC1C(=O)N(C(C)CCSC)C)=CC Cc1c(O)ccc(C(=O)NCC2CC2)c1C.c1(C=O)cc(C2CCC2)no1.C c1(OC)ccc(C(=O)N(C2COC(C)(C)C2)C)cc1S(=O)(=O)NC(C)C C1CC2(CCN(C(c3ccon3)=O)CC2)C1.N1(CC)C(=O)CCC1CC(=O)N.C C1(NC(c2c(C(C)C)nco2)=O)CC2CC1CN(C(=O)CC1CCCC1)C2 N1(C(C(CC2CC2)OC)=O)CCC(C)(C)C1CC(=O)NC(c1cccs1)C C(N=c1[nH]cnc(Cl)c1C)C1N(C(c2n(CC(=O)OC)cnc2C)=O)CCCC1 CC(C)C(CNC(=NCCc1ccc(F)cc1)NC1CC1C)C(C)C C(C#Cc1cccnc1)NC(C1(NC(=O)C(O)C(F)(F)F)CCSC1)=O C(C1CCN(C(C2CCSC2)=O)CC1)=CC(=O)NCC1C2CCCCC12 N1(C(C2C3CCC(C3)N2C(=O)Cc2ccc(O)cn2)=O)CCCC2(CCCC2)C1 NS(=O)(=O)CC(=O)N1CCC1CNC(=O)CCc1ccc(C(F)(F)F)cc1 c1(C(=O)NCC(C)NC(CSCCC)=O)ccc(CC)c(Cl)c1 C(=O)(C(O)CC(N)=O)N(CCCCCCNC(C1(C)CCNC1=O)=O)C C#CCCCCCC(c1nnnn1C)Nc1cnc(C(C)C)nc1 c1(NC(c2c(NC(CC(C)c3ccccc3)=O)c[nH]n2)=O)cncc([N+](=O)[O-])c1 CCCS(=O)(=O)C(C)C(=O)N(CC(C)NC(=O)Cn1c(C)c(C)sc1=O)C CCCC(CC(=O)N(C(C)CC)C)NC(=O)C(C)(COC)COC Cc1nc(NC(C)Cc2ccncc2)cc(=NC(C)c2cnc(C)s2)[nH]1 C(=O)(C(C)(C)C(=C)C)NC1C(NC(CC(=C)C)=O)COC1 c1(C(N(CC(C)CNC(=O)Cc2cn[nH]c2)C)=O)cccnc1CO c1(CCNC(=O)CC2(c3ccc(Br)cc3)CC2)cc(F)c(F)c(F)c1F C=CC(C)(O)CC(=O)N1CCN(C(c2cc(C3CC3)cs2)=O)CC1C(F)F N1(C(c2c(OC)cc(F)cc2)=O)CC2CN(C(c3ccc(Br)c(O)c3)=O)CC2C1 N1(C(CN(C(C=CCCC(C)C)=O)C2CC2)=O)CCC(CO)C(C)C1 C1(CC(=O)NC2CCC(N(C(CC(C(C)C)O)=O)C)CC2)SC2=NCCN2C1=O c1(C(=O)NCCCCN(C)C(C2CC3CCC2NC3=O)=O)cc2cnn(C)c2s1 C1(CC)CN(C(=O)CCS)CCN1C(=O)CC(C)(C1CCC1)N(C)C.CC(C)C Cc1cc(CNC(=O)CC2(C)CCN(C(c3ccc(=N)[nH]n3)=O)C2)ccc1F CC1CN(C(=O)Cc2csc(C3CC3)n2)CCN1C(=O)C=Cc1ccc(F)nc1 N1(C(C2(NC(=O)CNC(=O)C3CC3)CC(O)C2)=O)CC2CCC(O)CC2C1 C1(NC(C2CC2c2ccc(Br)s2)=O)C2CCC1CN(C(c1cccnc1)=O)C2 C1(C(N2C(C)CC(CNC(=O)C=CCF)CC2)=O)CCc2nc[nH]c2C1 N1(C(CCCCCSC)=O)CCC2(NC(C3CCCC3O)=O)CCCCCC12 CC(C)C(C(CO)C(C)C)NC(=O)C(=O)Nc1ccc(Cl)cn1 N1(C(CCCCOCC)=O)Cc2[nH]nc(C(N3CCC(O)CC3C3CC3)=O)c2C1 c1(C(=O)NCC(N2CCN(C(c3[nH]cc(C)c3)=O)CC2)=O)cnn2ccsc12 C1(N(C(Cc2nc(C)[nH]n2)=O)CC2CC2)CCN(C(C2CCC3CCC23)=O)CC1 C1(C#CC(=O)NCC23CC2CN(C(=O)Cn2cnc(Br)c2)C3)(CC)COC1 C(=O)(C1Cc2ccccc21)N1CCC(CC(=O)NCCc2cccc(C)c2)C1 C1(NC(c2cncc(C(C)(F)F)c2)=O)CCN(C(=O)CC2OCCO2)CC1F c1(C(=O)NCCNC(Cc2c(OC)ncc(Br)c2)=O)ccn2ncnc2c1 C(=O)(C(O)CC(N)=O)N(C)C(C1CCCCC1)=O.C(=O)C.C(=O)C1CC1.N C(C(F)(F)C(F)(F)F)OCCC(=O)N(CC(C)NC(C1CCCCO1)=O)C c1(OC)ccc(Cl)cc1S(=O)(=O)NC1CC(NC(c2ccc(Br)nc2F)=O)C1 c1(C(N(CC(CC)C)CC)=O)ccc(CNC(C2(C)CC2C)=O)nc1 c1(CC(=O)OC)ccc(NCC(C(C)(C)C)NC(c2sc(C)cc2)=O)nc1 C12(CNC(=NC)NCC3CC(c4ccccc4)C3)CC(CO)(CO1)C2 c1(C(F)F)ccc(-n2nc(C3CCCCC3)nc2C(C)Oc2cccnc2)cc1 c1(C=O)c(C)cc(=O)oc1C.c1(C(N(CCOC)CC)=O)csc(C)c1C.N C1(NC(C(C)O)=O)CCCN(C(C2(C)CC2C)=O)C1 O=C(C#CC1CC1)NCC(C1CCOC1)NC(c1cccn1C1CC1)=O C(c1ccc(C(F)(F)F)cc1)=C(C=O)F.C(CCC)OC.C(=O)C=C1CC1 Cc1ccncc1C(=O)NC1CCN(C(c2cnc(S)n2C)=O)C1 C=C(C)CC(C)C(=O)NCC1CN(C(C2CC(C(=O)OC)C2)=O)CCO1 C(=O)(C(F)C(C)C(F)(F)F)N1C(C)C(NC(=O)CCc2nccn2C)CC1 n1(CC=O)nc(C)c(C=NO)c1C.C(C(C)(C)C)NC(C1(CC#C)CC1)=O c1(C(=O)NC2CCN(C(Cc3nc(NC=O)sc3)=O)C2)cnc2n1CCOC2 CC(CN(C)C)CC(=O)N1CCC(N2CCC(NC(C3CC4CC3C4)=O)CC2)C1 c1(C(=O)NC2CCCC(NC(C(COC)(F)F)=O)C2)c(C)cccc1C c1(C(=O)NC2CCCN(CC)C2)ccc(Br)cc1CC#N C12(CNC(C3N(CC)CCC3)=O)CCCC1N(C(=O)C(C)n1cccc1)CCC2 N1(C(c2n[nH]c(C)c2Br)C(=O)NC2CC(F)(F)C2)CCC2NC(=O)CCC2C1 N1(C(C(n2c(C)cc(C)n2)C)=O)CCN(C(=O)C(C)(C)C2CCC2)CC12CCC2 Cn1cc(C(=O)NCCCN2CCN(C(C3(C)CC3)=O)CC2)c(C(F)(F)F)n1 C1(C(N(CC(=O)NCC)C)=O)CCCN1C(c1sccc1C(=O)OC)=O C1(C(=O)NCC(c2ccccc2)NC(c2cc[n+]([O-])cc2)=O)CC2CCCCC12 C(=O)(C1=C(C#N)CCC1)N1CCN(C(c2ccc(C3C(C)(C)C3(C)C)cc2)=O)CC1 Cc1nc2nccc(NC(CNC(=O)C=Cc3ccccc3Cl)CO)n2n1 C(=O)(C(CNC(C1CCCC1O)=O)C(C)C)N(C(CCC)C)C C1(CNC(c2ccc(C(C)=O)nn2)=O)COC(C)(C)CN1C(=O)CCS(C)=O c1(OC)cccc(O)c1C(N1CC(NC(=O)C(C)Cc2ccc(F)cc2)C1)=O CC1Cc2cc(CCNC(=O)C=Cc3ccc(N(C)C)cc3)ccc2O1 C#CCCCCC(=O)N(CC(C)(C)NC(=O)C=C(C)c1cnn(C)c1)C N1(C(CCCNC(N)=O)=O)CCCC(C(F)C(=O)NC(CO)CO)C1 N1(C(=O)CCCCCF)CC(CO)C2(C1)CN(C(c1cn(C3CC3)nn1)=O)C2 c1(C(=O)NC2C(NC(Cn3ccc(C)n3)=O)CC2)c(F)ccc(F)c1F CC1CC(CC(=O)NC2CCNC2=O)CN1C(=O)Cc1ccon1 c1(C(N2CC(CN=c3[nH]nc(C)o3)OCCC2)=O)c[nH]c2cccc(F)c12 N1(C(C2C(COC)CC2)=O)CCN(C(=O)CCC(C)OC)C2CCCCC2C1 c1(C(N2CCOCC(NC(C3CC(O)C3)=O)C2)=O)cc2ccc(O)nc2s1 C1(CNC(N2C(C)CC(C)C2)=O)CCC2COCCC2O1 C=CCC(CC)C(=O)NC1CC1CNC(c1noc(C)c1I)=O C(=O)CS(=O)(=O)C1CC1.c1(OC)ccc(OCC(N2CCC(C)C2)=O)cc1C.N c1(COC)nc(NC23CCN(CC2)C3)cc(=NC2CC3CCCC3C2)[nH]1 n1(CC)cc(CNCC2(C(=O)Nc3cc(Cl)ncc3I)CC2)c2cccnc12 C1(C(=O)NC2C(CCC)CN(C(=O)C(COC)OC)C2)CCN(OC)CC1 C(=O)(C(F)C(C)(C)O)N1CCC(CC=C)(NC(=O)C(C)C)C1 n1(CC)nnc2c(NC3CCCCCN(C(=O)CC4CC=CCC4)C3)ncnc12 Cc1ccc(C(=O)NC(CO)C(C)NC(=O)Cc2cn[nH]c2)cc1-n1cccc1 C1(CC(=O)NC2(C#C)CC2)CC2(C1)CN(C(=O)C(C)(O)CC)C2 c1(C(=O)NC2(C)CCN(C(C(CC#C)C)=O)C2)cc(C)c2nc(C)cn2n1 CC(Cn1cccn1)C(=O)NC1CCC(NC(=O)CCC2(C#N)CCC2)C1 c1(C(N2CCCN(C(C(C)C#N)=O)CC2)=O)ncc2c(F)cccn12 c1(CC(=O)NCCCC2(NC(C(C(CC)O)C)=O)CC2)cn2cccc(C)c2n1 O=S(=O)(c1cccnc1N1C2CCC1CC1(CC1)C2)NC1CC=CCC1 N=c1cc2c(n[nH]1)CCN(C(c1ccnc3c(I)cnn13)=O)C2 c1(CC(N2CCN(C(CNC(=O)Cc3ccoc3)=O)CC2)=O)ccc2occc2c1 C1(NC(C(C)c2ccco2)=O)CCCC12CN(C(=O)CCC(=O)N(C)C)C2 Cc1ccc(C(=O)N(CCC(=O)NC(CO)C2(O)CC2)CCO)n1C c1(C(N2CCCC(N(C)C(c3nn(C)cc3N)=O)C2)=O)cnn2c1CC(F)(F)C2 C1(CNC(C=CC2(C)COC2)=O)CCCCCN1C(=O)CSC(F)F C(=O)(C1=C(C#N)CCC1)NC1C2(C(=O)NCC(CC)CO)CCC(C1)C2 Cc1nccc(C(=O)NCC2C=CC(NC(=O)CC3CCCC(C)O3)C2)n1 CCC(CC(=O)NC1(CO)CCN(C(=O)CC2NC(=O)CNC2=O)CC1)C(C)C Cc1cc(C(=O)N)c(O)nn1.C1(O)CN(CC(=O)N(C2CCCCC2)C(C)C)C1 C1(CNCC2CC(c3n(C)ncc3)CC2O)CCCC(F)(F)C1 N1(C(C(C)SC(C)C)=O)CCN(C(=O)C(c2cnn(C(C)(C)C)c2)=O)CC1.C C1(C(=O)NCC(C)(C)NC(C2CC(C)(C)C2)=O)CC(c2ccccc2)=NO1 c1(C(=O)N)cc(N)cc(O)c1C.N1(C(c2[nH]cc(CC)c2)=O)CCC(C)C(C)C1 N1(C(CNC(C)=O)=O)CCC(N(CC(C)C)C(c2cnc(C)nc2)=O)CC1 C(C(=O)N(C)CCN(c1ncc(Br)cn1)C)(C(C)C)OCC(C)C C(=O)(C(F)C1=CCCCC1)N(C1CCCN(C(c2c(C)cc[nH]2)=O)CC1)C C1(n2cc(C(=O)NC(C)Cc3nncn3C)nn2)CCCN(C(=O)C2CC2)C1 N1(C(C2CC(OC)C2)=O)CCC2(CNC(C3(F)CCCCCC3)=O)CCCCC12 C1(NC(CCNC(N)=O)=O)CCN(C(=O)C=C2CN3CCC2CC3)CCC1(F)F CC(CC(F)(F)F)C(=O)N1CCOC(c2ccc(Cl)s2)C1 C1(O)(C(N)=O)CCCN(C(=O)NC2CN(C(C3CCC3)=O)C2)C1 c1(C(=O)NCCN(C(=O)CCC2CCCC(O)C2)CC)c(F)cccc1F.O c1(CC)cc(NC(c2c(CNC(C3CCC(F)C3)=O)cnn2C)=O)cnc1C C(=O)(C1=CC2CCCC12)N1CC(C)(N(C(C2(c3cccc(C)c3)CC2)=O)C)C1 C=C1CCN(C(=O)C(CC)n2cncn2)C(C(=O)NCC(O)CCCC)C1 CCC(C(=O)NC1CCCN(C(c2ncccc2N(C)C)=O)C1)C(C)(C)CC C=CC1(C(N2CC3CC3(CNC(c3ccc(Cl)c(F)c3)=O)C2)=O)CCOCC1 C12(NC(C(C)OCCC=C)=O)CCC(CC1)N(C(C1CC1COC)=O)C2 c1(CC=O)ccc([N+](=O)[O-])cc1.C(CC(C)C)C(=O)N1CC(=C(F)C)C1.CO c1(C(=O)NCC(CN(C(C2CCC(OC)C2)=O)C)C)ccc2n[nH]cc2n1 c1(CCC(N2CCC(N(C(c3cnc(CC)s3)=O)CCO)C2)=O)ncccc1C CCC(C)C(C)(O)C.c1(C(NCCC(=O)N)=O)ccco1.C1CC1.N(C)C Cc1nscc1CC(=O)NC1CCOC1C(=O)NCC1(CCO)CCC1 c1nc(Cl)c(Br)nc1Br.c1(C(=O)OC)ccnc(C(=O)NC2CC2C=O)c1.N C1(CNC(C2(NC(c3c(CC)ncs3)=O)CCC2)=O)CC(O)C(O)C1 c1(C(=O)NC(CCN(C(c2c(CC)con2)=O)C)C)ccc2c(c1)nc(C)n2C c1(C(=O)N)occ(C)c1C.C(=O)(CCCNC(c1ccco1)=O)N(CCCC)C N1(C(C)C)CC(C)(CNC(=O)NC(C2(O)CCC2)(C)C)C1=O C(CC(C)CC)(C(=O)N1CCCOCC1C)NC(C(CCC)C#N)=O c1(C(N2CC(=O)N(Cc3ccccc3)CC2)=O)cc2ccc(Br)c(Cl)c2s1 N1(C(C2CCCC(=O)N2)=O)CCCCC(NC(=O)CCOc2cccc(F)c2)C1 CC1(C)CC(=O)CCC1C(=O)NC1CC1CNC(c1ccnc(S)c1)=O c1(C(=O)NC2CCC(NC(CCc3c(C)ncs3)=O)C2)cnn2c1CC(F)(F)C2 C1(C#N)(C(=O)NCC(C)N(C(=O)CCc2ccc(Br)nc2)C)CCCCC1 Cc1ccc(C(=O)NCC2CCCN(C(=O)C(O)CN(C)C)C2)c2c1CCCN2 n1(CC)ncc(C(=O)NC(Cc2ccoc2)C(N2CCC(O)(C)C2)=O)c1C.S C1(N(C(CSCCOC)=O)C)CCCN(C(c2conc2C2CCCC2)=O)CC1 c1(NC2C(C(=O)Nc3nc(C)nc(Cl)c3)CCCC2)ncnc2c(Br)c[nH]c12 C(=O)(CCC(O)C(C)(C)C)NC1C(C)CN(C(C2CN3CCN2CC3)=O)CC1 C1(CC(C)NC(C(C)OCC#C)=O)CC2CCC(C1)N2c1nccc(C)n1 N1(C(C(=O)NCC=C)=O)CC(NC(=O)OC(C)(C)C)CC12CCC2 c1(C=O)ccnc(Cl)c1O.C1(OC(C)(C)C)CC(C(=O)NC(C)C2CC2)C1 c1(CC)cc(N2CCN(C(=O)C(=O)NC3(C(N)=O)CCOC3)CC2)ncn1 N1(C(c2c(CC)cco2)=O)CC(C)C2(CC2)C1.c1(C(=O)N)cc(CCO)on1 C1(CCNC(C(N2CCOCC2)C)=O)CN(C(c2cccs2)=O)CCO1 N1(C(c2ncn(CC)c2)=O)CC(C(=O)NC2(C3CCCCC3)CC2)CC(C)(C)C1 CC1CCC(N2CCC(C(=O)NCCC3CCCS3)CC2)CC1 C1(NC(c2cc(COC)sc2)=O)CC2CCC1N2C(c1cccc(=O)n1C)=O c1(C(N(CCCN(C)C(C2CC3(C2)CC3(F)F)=O)C)=O)cc(O)c2ccoc2c1 C1(NC(=O)C2=CCOC2)CC2CN(C(c3ncc(F)cc3F)=O)CC2C1 N1(C(CCCC)=O)CCC(O)C(NC(C2(C)CC2(Cl)Cl)=O)C1 N1(C(C(c2ccccc2F)=O)=O)CCC2CCN(C(c3csnn3)=O)CC12 N1(C(C(C)C(=O)OC(C)(C)C)=O)CC2CC(C1)CN(C(=O)CCc1cncs1)C2 N1(C(C(C)=C2CC2)=O)CC(O)CC1CNC(C1COCC1(C)C)=O N1(C(C2CC3(CC(=C)C3)C2)=O)C(C)CC2CN(C(=O)CC3(C)CC3)CC12.O c1(C(N(C2CN(C(=O)Cc3cnns3)CC2F)C)=O)cc(F)ccc1C(F)F Cc1c(C(=O)N(CC(O)CN(C)C(C2CCCOC2)=O)C)cnc2ncnn12 C1(CC)CN(C(=O)C(C2CCN(C(=O)CCOC3CC3)C2)C)CCO1 c1(CC)ccccc1CC(N1CC(NC(=O)CCC(N)=O)C(C)C1)=O c1(CC(=O)NCC)cc(F)cc(S(N)(=O)=O)c1.C(=O)C=CC.CC c1(C(=O)NCCNC(C(C)N2CCC2)=O)cc2c(nn1)OCCS2 c1(C(N2CCC(O)(C(C)CNC(=O)Cc3csc(S)n3)C2)=O)cccc(F)c1N C1(NC(C=CS(C)=O)=O)CN(C(=O)C(=O)NCC2CC2)CC2(CCC2)C1 CC1=C(C)CC(C)(NC(=O)CC2COCCN2C(c2scnc2Cl)=O)CC1 C(C1=NOC2CN(C(=O)CC#N)CC12)NC(Cn1cc(C)c(O)nc1=O)=O CC1(C)CN(C(c2cc([N+](=O)[O-])c[nH]2)=O)CC1NC(=O)CCCc1ccccn1 C1(NC(C2(CSC)CCC2)=O)CCCCC1NC(=O)C(O)CF c1(CCC(=O)NCC2CC2NC(=O)CCn2cncn2)csc2ccccc12 c1(C(=O)NCC(CC)NC(=O)COc2ccnc(C(=O)O)c2)ccccc1C C(C(F)(F)CCC(=O)N1CC=CC(O)C1)n1cc(CC(C)C)nn1 c1(C(N2C3CC(NC(c4cc(C(F)F)cs4)=O)C2CC3)=O)cc2ccccc2s1 CC(C)(CC(F)C(=O)NCCP(C)(C)=O)NC(=O)CC1C=CCCC1 C1(N(C(c2c(C)snn2)=O)C)CCCN(C(=O)C(F)(F)C2CCCCC2)C1 N1(C(C2CC(CNC(C(CC)N(C)C)=O)OC2)=O)CCC(C)CC1C CN=C(NC1CC(O)C12CCC2)N1CCC2=C(COC2=O)C1 c1(OC)cc(C=CC(=O)NCC(=O)NNC(=O)c2cccs2)cc(Cl)c1OC n1(C2CC(CC)C2)c(-c2sccc2C)csc1=Nc1cccc(Cl)c1C N1(C(CCC#C)=O)CCCN(C(c2cncn(C)c2=O)=O)C(C(C)C)C1 N1(C(CCCCCC)=O)CC(NC(C2CC(C(=O)OC)C2)=O)C2(CCC2)C1 C1(C(=O)NCC(C)CNC(c2cnc3[nH]ccc3c2)=O)CCc2ncncc2C1 C1(C(=O)NCc2ccc(F)cc2)CC12CCN(C(C1CN3CCC1CC3)=O)CC2 CN1CCN(C(c2cc(Cl)ns2)=O)CC1CNC(=O)CCN1CCOCC1=O CC(C)C(CN(C)C)C(=O)N1CC(C)C2(CC2)C1.c1(CC=O)ccc(Cl)cn1 C1(N(C(c2c(C)snc2)=O)CCO)CCN(C(=O)CC)CC1.C(=O)C(C)(C)C.N N1(C(C(n2ncc(C)c2)C)=O)CC(F)(F)CC1CNC(c1n[nH]cc1C)=O CN1CCN(CC(=O)NC(Cn2cncn2)C(N2CCC3CCC23)=O)CC1 CCC(C)C(CO)NC(C1CN(C(c2cscc2Br)=O)CCN1)=O c1(CN2CCC3(CN(S(CC)(=O)=O)C3)CC2)cc2ccccc2nc1O CC1Cc2cc(C(=O)NC(C)CCCNC(C3(O)CCSC3)=O)ccc2O1 c1(C(=O)N)ccc2oc(O)nc2n1.Cc1cc(C(=O)N(CC)C(C)C)nc(C)c1 C(C)(CSC)(C(=O)NCC1(C)CCCOC1)NC(CC1CC(SC)C1)=O N1(C(c2nc(C(C)C)oc2)=O)CCC2(CCCCC2NC(C2CC2F)=O)CC1 N1(C(C=C(CCC)C)=O)CCOC2(CCCN(C(=O)C(CN(C)C)C(C)C)C2)C1 N1(C(c2n(C)cc(Cl)c2)=O)CCC2(CC1)CC2C(=O)NCC(CO)C(F)(F)F N1(C(C(C)C(C)(C)C)=O)CC2CCC1CC2NC(=O)CN1CC2CCC1C2 N1(C(c2scnc2C(F)F)=O)CCN(C(=O)CC2CCOC2)C(CO)C1 C=C(Cl)CCC(=O)N1CC(C(C(=O)NCC(C)(O)CCC)OC)C1 Cc1ccc(=O)n(CC(N2CC3C(NC(=O)C=C4CCN(C)C4)C3C2)=O)n1 c1(SC)nc(C)c(CCC(=O)NCC2CCCN2C(=O)CCC(C)OC)c(O)n1 N(C1CCCOc2ccc(F)cc21)C(N1CC2(CC(CO)C2)C1)=O C#CC12CC(CN1C(C1CCCC(NC(=O)C(Cl)Cl)CC1)=O)C2 C1(CC)COC(C)CN1C(=O)CC1(OC)CN(C(c2ncc[nH]2)=O)C1 Cc1cccc2c(C(=O)NCC3(O)CCN(C(=O)CCc4ccsc4)C3)c[nH]c12 C12(C(=O)OC)CCCC1(C(=O)N(C)C)C2.c1(C(N2CCCC2)=O)ncncc1F N1(C(c2cc(C)sc2Br)=O)CCc2c(O)noc2C1 C12(OC)CCCCC(C(=O)NC(C)CCCNC(C3CCCCO3)=O)(C1)C2 c1(OC)ccc(C(N2CC(C(C)NC(=O)CCc3cncnc3)C2)=O)cc1F C(=O)(C1=NNC(=O)C1)N(C)CC1CCCN(C(C2CCN(C(CC)=O)C2)=O)C1 C=CCCCC(C)(C)CN=c1[nH]c(=NC)[nH]c(=NCc2cccc(OCC)c2)[nH]1 CC(C)(CN=C(NCC1(C)CCOC1)NC1CCC1)CS(C)(=O)=O c1(NC(C2N(C(CCCOC(C)=O)=O)CCC2C)=O)cc(C)cc(Cl)c1 c1(N2CCC(C)C(NC(=O)C(C)O)C2)ncnc2c1nnn2CC1CC1 N1(C(C2(COC)CCC2)=O)CCCC(N(c2nc(C3CC3)ns2)C)C1 c1(CC)cccc(C)c1C(=O)NC1CCN(C(c2cc(C(N)=O)c[nH]2)=O)CC1O C(=O)(C(CC(C)C)ONC(C1(C)CCC(=O)NC1)=O)N1CC(CC)(CC)C1 N1(C(C(C)=O)=O)CCC2(COCCN2C(=O)C(C)Oc2cccnc2)C1 C1(C(N2CC(NC(c3c(SC)snn3)=O)C2)=O)CC2C=CC1C2 N1(C(C(CC=C)CC(C)C)=O)CCC2(CCCCN(C(=O)COCC)C2)C1 CCCC(CNC(c1cc(=O)cc[nH]1)=O)C(=O)N1CC2CC2(CO)C1 N1(C(CC2(NC(CNC(=O)OC)=O)CCC2)=O)CC2CCCCC2C1C Cc1cc(C#N)cnc1C(=O)NCC1C2CCC12c1ccccc1 Cc1cc(C(N2CCOC(CCNC(=O)C)C2)=O)nc(C(F)F)n1.CC(C)C.S C(=O)(CC(O)CNC(C1CCN1C(=O)Cn1cnc(C#N)n1)=O)OC N1(C(c2n(C)ccc2)=O)CC2CCN(C(c3ccc4c(n3)CCO4)=O)CC(C2)C1 N1(C(c2c(C)cc(CNC(CN(C(C)=O)C)=O)o2)=O)CCCC(F)(CO)C1 c1(C(N)=O)nc(NC(c2ccnc(C)c2)=O)ccc1Br.n1(CC(=O)N)nccn1 Cc1ccc(CC(=O)NC(C)CCCCNC(c2sc(C)cc2Cl)=O)c(F)c1 N1(C(Cc2c(C)cc(Cl)cc2)=O)CCC(NC(=O)CC(C)(C)F)CC(O)C1 c1(C(CNC(=O)C(O)Cn2cncn2)NC(=O)CCC2CC2)ccc(F)cc1 CC1(C)CNC(=O)OC12CN(C(=O)CCC1=CCCCC1)C2 CC1CC(F)(F)CN1C(=O)CC1(C#N)CC1.c1(C=O)occc1C1CC1.C C(=O)(CC(C)C(=O)NC(C1CC=CCC1)C(=O)NC1CCN(CCCO)C1)OC C(=O)(C1=C(Cl)CCC(C)C1)NCCOCCNC(c1c(C)ccc(F)c1)=O C=CC1(C(N2CCC(N=[N+]=[N-])C2)=O)CCN(C(c2cccc(OC)c2)=O)C1 N1(C(C2CC(Cl)(Cl)C2)=O)CC2CC(C1)CN(C(C1CC(n3cnnc3)C1)=O)C2 C1(NC(=O)C(O)c2ccco2)CCOC(CNC(C2CCOCC2)=O)C1 c1(OC)oc(C)nc1C(N1CC(CO)(NC(=O)CN2CCCCCC2)C1)=O C1(C(=O)N)CCCCN1S(C)(=O)=O.C=C(C)CC.c1(CC=O)cc(C)on1 C#Cc1cc(C(=O)NC2CCN(C(=O)C(c3ccccc3F)O)C2)cc(Br)c1 C(=O)(CC1OCCc2sccc21)NC(C)CN(C)C(c1cccc(C#N)c1)=O CP(C)(=O)C1CCC(NC(=O)C(N2CCC(c3ccc(F)cc3)CC2)=O)C1 c1(NC(C(=O)NCc2nc(Cl)cs2)=O)ccc2nonc2c1 C1(CC)CN(C(c2cnc(C(C)(C)C)[nH]2)=O)CCN1C(=O)CCc1cc(C)on1 c1(C(=O)NC2CN(C(C3C=CC=CC=C3)=O)CC3CC23)cn2cc(Cl)cnc2n1 CC1CCCn2cc(C(=O)NC3CC(CC)C3)nc21.C1(C)(C=O)CCC(=O)N1.N c1(C(N2CCCC(C)(NC(c3nccc(C)c3)=O)C2)=O)c(C)cc(O)cc1C C=CCC(CC(F)F)C(=O)NCCC1CCCCN1C(c1cc[n+]([O-])cc1)=O C#Cc1ccc(C(=O)NC2CC3CC2CN3C(=O)C=Cc2ccc(C)s2)cc1F Cn1nnc2c(C(=O)NC3CCN(C(c4sc(F)cc4Cl)=O)C3)cccc12 CCC(CCOC)C(=O)N(CCNC(C1CC(C)(C)CCO1)=O)CC c1(CC(=O)N)cn2cc(F)ccc2n1.c1(C(N(C(C)C)C)=O)ccc(=O)n(C)n1 N1(C(C2CC(C)CC(C)C2)C(=O)NC2CCCCC2)CCC2CS(=O)(=O)CC12 c1(CCN(C(C(=O)NC(CSC)C)C)CCc2ccccc2)ccccc1 C1(OC)(CNC(=O)Nc2ccccc2CCN=[N+]=[N-])CCCS(=O)(=O)C1 CC1CN(C(=O)CC2(CO)CC2)CCC1C(c1ccco1)=O Cc1coc(C(=O)N(C2CCN(C(=O)CC3CCCN3C)C2)CCO)c1C C12(CNC(c3ccc(Cl)cn3)=O)CC(CN1C(C1CC3CCCC13)=O)C2 N#Cc1csc(C(c2nnnn2C2COC2)Nc2ccc(-c3ccno3)cc2)c1 N1(C(CSCCOC)=O)CC(CNC(c2ccc(S)o2)=O)OC(C)(C)C1 c1(CCC(=O)NCC(CC=C)NC(=O)C#CC2CC2)ccc(Cl)c(OC)c1 N1(CCCC)CCCC(C(=O)NC2(C)CC(NC(=O)COCC(F)F)C2)C1 CC(CC(=O)NC1CCN(C(c2ccnn2CC2CC2)=O)CC1F)CC(C)(C)C N1(C(CC2N(CC)CCOC2)=O)CCC(CNC(C2CCCSS2)=O)C12CC2 C1(NC(c2c(CC)occ2)=O)CC2CC(NC(C3(C)CCCO3)=O)CC2C1 C12CCN(C1C)C2=O.C1(CC)CN(C(=O)CC2(COC)CCC2)CC1C c1(COC)cc(C(=O)NCC(CC(C)C)NC(=O)C)n(C)c1.C(C)C.S N1(C(COCC(=O)NC)=O)CC(C)(NC(=O)CCc2cn[nH]c2)C1 Cc1cc(F)c(Cl)cc1NC(C1CC1C(=O)Nc1cncnc1I)=O N1(C(c2cnn3c2CC(CN)CC3)=O)CCC[Si]2(CCCC2)CC1 CCCC(C)C(=O)NC1CCN(C(c2coc(Cn3cccn3)c2)=O)C1 c1(C(=O)NC(C(C)C)CCN(C(=O)CS(=O)(=O)N(C)C)C)cccc2cnnn12 C1(NC(CC(=C)C)=O)CN(C(c2cn(C3CCCCC3)nn2)=O)CC12CC2 C1(C(=O)NC(C2CN(C(C)=O)C2)C)CCC(C(F)(F)F)NC1=O C1(C2CCC(=O)CC2)(NC(=O)NC(c2cccc(C3CC3)c2)C)CC1 c1(OC)ccc2c(C(=O)NCC3CCCN3C(=O)CCC(C)C)n[nH]c2c1 CC1CCCN(C(=O)COc2cncc(Cl)n2)C1CC.C1(F)(C=O)CC=CC1.N N1(C(CSCC=C)=O)CC2CC1C2CNC(C1CCOC(C)C1)=O C(=O)(C1=NOC2COCC12)N1CC(NC(c2ccc(F)o2)=O)C2(C1)CCC2 C1(C(=O)NCC(C)C)CCN(C(=O)Cc2ccc(O)cn2)CC1 N1(C(Cc2cn(CC)nn2)=O)CCN(C(c2cc(C3CCOC3)[nH]n2)=O)C(C)C1 c1(OC)c(C(N2CCN(C(c3nnc(O)cc3O)=O)C(CO)C2)=O)cccc1Cl n1(CCNC(c2cccc(-c3nn[nH]n3)c2)=O)nnn(C2CCCC2)c1=O c1(C(=O)OC)cc(C=O)n(C)n1.c1(C=O)nnn(C)c1C(F)F.C(C)CC S(=O)(=O)(c1cnc(O)c2ccccc12)NC(NNC(N=c1c(C)cn(CC)[nH]1)=O)=O N1(C(=O)NCC2CCN(Cc3ccccc3)C2)CCN(c2ccncn2)CC1 C1(C(=O)Nc2cn(C3CCCC3=O)nn2)CCNC2(CCOCC2)C1 C1(NC(C(CN(C)C)(F)F)=O)CN(C(C2CC23CCCC3)=O)CC1N=[N+]=[N-] C1(C(C)(C)NC(CCN(C)CC)=O)CCN(C(=O)CCc2ccncc2)C1 c1(C(NC(C)C)=O)ccc2c(c1)COC2=O.c1(C=O)cn(C(C)C)cn1.CC c1(C(=O)NCCCN(C(C2CCC(C)S2)=O)CCO)ccc(CO)cn1 CCCC(CCCNC(C1CCS(=O)(=O)C1)=O)NC(=O)Cn1cccnc1=O C(=O)(C(C)Cc1cccnc1)NC(C(C)NC(CC1CC(OC)C1)=O)C N1(C(C(CC)C)=O)CCCCC(NC(c2ccnn2CC2CC2)=O)C1 C(=O)(C#CC(C)C)NCC(CCC)NC(c1cc(O)n(C)n1)=O CC(C(F)(F)C(F)F)c1nc(-c2cccc(C(F)F)c2)nn1Cc1cccc(Cl)c1 c1(C(N2C(C(N(C3CCO3)CC)=O)CC3CC32)=O)ccc(C(F)(F)F)cc1 N1(C(C2OCCN(C(C)C)C2)=O)CCCN(C(c2cc(N)ccc2F)=O)CC1C Cc1csc(C(=O)NCC(c2ccccc2)CNC(c2ccc(O)nn2)=O)c1C Cn1cc(C(N2CCC2CNC(=O)CCc2cccc(O)c2)=O)c(=O)c(Br)c1 N#Cc1cc(C(=O)NC2CCCCC2C)co1.C(=O)C(F)(F)F.C(=O)(C)N CC1C(NC(=O)C(F)C(C)(C)O)C(C)CCN1C(=O)COCC1CCOC1 C1(NC(c2cscc2Br)=O)CN(C(C2CC3(CCC3)C2)=O)CC1(F)F c1(C(N(CCC)CC)=O)ccc2nc(C)[nH]c2c1.c1(C=O)cc(C(C)C)no1.N c1(C(N2CC3C(CNC(c4cc(C)sc4)=O)C3C2)=O)ccc2ccn(C)c2c1 c1(CN2CC(C(=O)NCC(=O)NC)SCC2)c[nH]c2cc(F)c(F)cc12 C(=O)(C(C)CCO)NC(C1CCN(C(=O)CCC2CCCOC2)CC1)C c1(C(=O)N)cn2c(n1)CCCC2.c1(CC)cc(C(=O)N(CC)C(C)C)cs1 C(=O)(CCC(N)=O)N.C1(OC)CCCC(C(N2CC(O)(C)C2)=O)C1.C(C)=O C1(C(N2CCC(OC)C2)=O)C2CCC1CN(C(C1CC1C1CC1)=O)C2 c1(C(C(=O)NCC(C)CN(C(=O)CCCc2cccnc2)C)O)ccccc1 N1(C(C2C(C3CN(C(C(C)Cn4cccn4)=O)C3)C2)=O)C2CCC1CC1(C2)N=N1 CCCCCC(C)(c1nnnn1Cc1ccco1)NCc1cn(C)cn1 c1(NC(CC2C(C(=O)NC(CCOC)COC)C2)=O)cc(C(N)=O)oc1C c1(C(N2C(C(N3C(CC(C)C)CCC3)=O)CNC(=O)C2)=O)cnn2cccc2c1 C=CCCCC(C)NC(=O)C(C)(C1CC1)N(C)C(C1CCN1C(C)(C)C)=O Cc1cc(C(=O)NCC2CN(C)CCN2C(c2cnn(C)c2)=O)nc(O)c1 C(c1ccn(C)c1)=CC(=O)NC(c1cccnc1)C(=O)N(CCCCOC)C N1(C(CCC)=O)CCCCC1CC(c1ccccc1)NC(c1cnsn1)=O N1(C(C(CC=C)(F)F)=O)CC2=C(C1)CN(C(=O)C(c1ccc(Cl)s1)C)C2 N1(CC(=O)NCC2(O)CN(C(c3cc(Cl)sc3Cl)=O)C2)CCc2ccccc21 c1(NC(C(C2CCN(C(Cc3cncc(C)c3)=O)C2)C)=O)cc(C)c(F)cc1F C(=O)(CCC(C)(C)[N+](=O)[O-])NC1CN(C(C(CC=CCC)C)=O)CC12CCC2 c1(C(=O)OCC)ccc(S(=O)(=O)N2CCCC(C)(N)C2)cc1.C1COCCO1.C N1(CCNC(CCOC)=O)CCC(NC(=O)CSc2ccc(O)cc2)CC1 C(=O)(C(C)(C)O)NCCCNC(C1(C(N(C)C)=O)CC1)=O.C1CCCC1 C1(NC(C(C)NS(C)(=O)=O)=O)CN(C(c2cncc(Cl)c2)=O)CC12CCC2 N1(CC(N2CCN(C3(CC4CC4)CC3)CC2)=O)C(=O)NC2(CCCC2)C1=O c1(CNCC2(C(=O)NC(CC)C(=O)OC)CC2)cnnc(-c2ccccc2)c1 C(=O)(C(C)S(=O)(=O)C(C)C)NCC(CC)(CC)NC(=O)C1=NOC2COCC12 C(=O)(C(F)(F)C1=CCOCC1)NC1C(NC(=O)CC2C=CCCC2)CC1 C(=O)(CCC1=CCc2ccccc21)N1CC(C)N(C(=O)Cn2cnnn2)CC1 N1(C(COCC(=O)NC)=O)CCC2CCCC12.c1(C=O)cn[nH]c1.C1CC1.N CCCCCC(=O)N1CC2CC2(NC(=O)CCCOc2ccccc2)C1 C1(NC(c2c(Cl)cn(C)n2)=O)CC2CCC1CC2.C1(C(=O)N)CC(=O)OC1(C)C C(COC(C)(C)C)(C(=O)OC(C)(C)C)N(C(=O)C(F)(F)F)C CC1(C)CC(NC(=O)C2=CCCCC2)CN1C(=O)C(O)CF C(C(N=[N+]=[N-])C(=O)NNc1ccc([N+](=O)[O-])cc1)OCC C(=O)(CCCCC=C)N1CC(CC(=O)N(CC#C)CC2CCCO2)(OC)C1 CCCCCS(=O)(=O)CC(=O)NCC(C)(C1CCC1)NC(=O)CS(=O)CC N1(CC(=O)N(CCCN(C(C2(CCOC)CCCC2)=O)C)C)CCC(C)CC1 CC1(C)CC(=O)NCC1C(=O)NCC1(O)CCN(C(=O)Cc2cnns2)C1 C1(C(=O)NC2CC(C(C)NC(C3CCSC3)=O)C2)(COC)CCOCC1 c1(C(=O)NCCCNC(C(CC)NC(C)=O)=O)cnn2c1N(C)CC2 C12(C(N(CCCCCC)C)=O)CCN(C1)S(=O)(=O)C2.C1(C(C)C)(C=O)CC1.N c1(COC)nc(CCNCc2ncc(Br)s2)cs1 c1(CCNC(=O)NC2CCN(c3ccncn3)C2)nc(-c2ccccc2)cs1 N1(C(C#CC)=O)CCN(C(=O)CSc2ccccc2OC)CC1CC Cc1cc(C(=O)NC2(C)CCN(C(=O)CN3CC4CC4C3)CC2)c(O)nn1 c1(CC)ncc(C(=O)NCCc2cncs2)cn1 c1(OCCC)ccc(C(=O)NCC(C)NC(C2CCCCC2O)=O)cc1N C1(CNC(C2(CC=C)CCOC2)=O)CCCCN1C(c1cc[nH]n1)=O S(=O)(=O)(c1ccc(NS(C)(=O)=O)cc1)NC(CNC(CC=C)=O)(C)C Cc1cc(C(N)=O)c(NC(C2CC(O)CN2C(C2CCCC2C)=O)=O)s1 c1(CN(C)CC2N(C(CCc3c(C)cccn3)=O)CCC2)cc(Br)ccc1C C1(CC(=O)NCC(N2CCCCC2)C)CC(NC(=O)C(=O)N(C)C)C1(C)C C=Cn1nccc1C(N1CC2CC1(C(=O)NC(C)(C)COC)C2)=O N1(C(CCCOC(C)=O)=O)CCC=C(C(=O)N2CC(O)(C(C)C)C2)C1 C1(OC)CC(F)CN(C(C23CC2CCN3C(=O)CCn2cccn2)=O)C1 C1(CC)(NC(=O)CN(CC(C)(C)C)C)CN(C(=O)C(Cl)=CCl)C1 C1CN(C)CCN1C(=O)CNS(N)(=O)=O.c1(NC(C)=O)nc(C=O)cs1.N Cc1cnc(C)c(C(=O)NC2CC(NC(=O)CN3C(=O)CSC3=S)C2)n1 N1(C(C(C)NC(CC)=O)=O)CCN(C(c2oc(CC)cc2C)=O)CC1CCO C(CCN=C(NCC1CN(Cc2ccccc2)CCO1)NC1CC1C(C)C)SC N1(C(CCN(CCC)C)=O)CCN(C(=O)C(S(C)(=O)=O)C2CC2)CC(O)C1 Cc1cc(CC(=O)NCC(C)CNC(c2ccc(C3CCC3)nc2)=O)ccc1O C1(NC(CNC(=O)Cn2cnnc2)=O)CCCC1NC(=O)C(O)C1CCCC1 Cc1cc(CN(C2CCN(CC(F)(F)F)C2)C(=O)NC)ccc1F.C1CCCO1 CCCCCCN(C(=O)C(O)Cc1cn(C)cn1)CCNC(c1nsnc1O)=O C1(NC(C=C(COC)C)=O)CC12CCC(NC(c1ccc(Cl)o1)=O)CC2 CC1=C(C(=O)N2C3CCC2C(C(N2CC4COCC4C2)=O)C3)CCC1 CCCCCCCC(=O)N1CCC(NC(c2c(OC)noc2C2CC2)=O)C1C C1(CNC(c2c(CC)nc(C)o2)=O)CCC2CN(C(c3ccco3)=O)CCC2C1 c1(OC)cncc(C(C(=O)NCc2ccccc2)N(C)C(C2CCOC2)C)c1 c1(C(N2CC(NC(C3(C(C)C)CNC(=O)C3)=O)C2)=O)csc2cc(Cl)cnc12 N1(CCNCC2C(=C)C2)C(=O)NC(C)C1=O N1(C(c2cnc3c(c2)CCC3)C(=O)NCCCSC)CCC(C2CNC(=O)C2)C1 C(=O)(C#CC1CCCO1)N1CCC(NC(=O)COc2ccc(F)cc2)(CO)CC1 n1(CC)cc(CC(=O)NC2CCCC2NC(c2cccs2)=O)c(C)n1 c1(CC)ccc(C(=O)NCC(CC)NC(c2cnoc2C2CCC2)=O)c(O)c1 c1(NC2CCCCN(C(C3(CC)CC3)=O)C2)nc(C)cc(C)c1C(=O)OC c1(CNCC2N(CCOC)CCC2)c(OC)ccc2c1CCC2 c1(C(=O)NCCC(CNC(=O)C(=O)NC)O)nc2ccccc2nc1O.C1CC1 C#CCC(C(=O)NC)NC(=O)CCNC(c1cccc(-n2ccnn2)c1)=O C(=O)(C(C#N)C(C)C)N1CC(CC=C)(C(=O)Nc2cn(CC)nc2C)C1 C1(NC(C(CC)OC)=O)(CF)CCN(C(c2ncsc2C)=O)C1 C1(CNC(C)=O)CCC(C)CN1C(c1sc(SC(F)(F)F)nc1C)=O N(C1CCc2cc(CNC(c3cnc4cccnc4c3)=O)ccc21)C(CSC)=O c1(C(N2CC=CC(NC(C3(C(C)(C)C)CCC3)=O)C2)=O)ncc(F)cc1N c1(C(=O)NCC2N(C(C(c3cccnc3)OC)=O)CC=C2)cc(C)nnc1O c1(C(=O)NC2(CC=C)CCN(C(=O)C(C)C(CC)CC)C2)cnc2[nH]cnc2c1 CCC(CC)CCCNC(=O)C(C)CNC(=O)CN(C1CCCC1)C N1(C(C2(COC)CCCCO2)=O)CCCCC(NC(c2nccn2C(C)C)=O)C1 C#CC(C)(C)C(=O)NCCN(C(=O)Cc1csc(CC)n1)CC N1(C(=O)CSC(F)F)CCC(C(=O)NCc2cnsc2)(CO)C1 N1(C(CCOCC#C)=O)CC2CCN(C(c3[nH]c(O)nc3C)=O)C2C1 c1(CC)ccc(C)c(NC(N2CCN(c3ccc(C(F)(F)F)cc3)C(=O)C2)=O)c1 C1(NC(CCc2cnc(C)s2)=O)CC(C)CN(C(c2ccc(C(N)=O)nc2)=O)C1 c1(C(N2CCCN(C(CCCCC)=O)CC2)=O)ncnc2c1c(Br)cn2C C(=O)(C(CO)C(F)(F)F)NCCOC1CCN(C(C(C#C)(C)C)=O)CC1 c1(C(=O)NCC(C)(C)NC(C2CCN(CC)C2)=O)ccc(C)cc1O c1(OC)ncc(C(N2CCN(C(c3cc(=O)n(C)o3)=O)CC2CCO)=O)cc1C C(=O)(C(C)(O)C(F)(F)F)N1CCC(C(=O)NC2(CC=C)CCC2)C1 c1(CC(=O)NCC(C)N(C(c2ccc(CC)nc2)=O)C)ccc(O)c(F)c1 N1(C(CCCCCSC)=O)CCCC1C1CCCCN1C(=O)Cc1cnnn1C c1(N(CC(CNC(CC(C)(C)OC)=O)C)C)c(C#N)nnc2ccccc12 N1(C(C2N(C(C(COC(C)=O)C)=O)CSC2)=O)CC2CCC(O)C(O)C12 C(c1ccccc1)=C(OC)C(=O)NC1CC(NC(c2nnn(C)c2C)=O)C1 c1(C(N2CC(CO)C3(CC3)C2)C(=O)NC)cc(C(C)C)ccc1F N1CCN(C(C2CC(O)CN2C(C)=O)=O)CC1.c1(C(=O)OCC)ccc[nH]1.C c1(C(N2CC3(C)CC2(C(=O)NCC2CCCC(F)C2)C3)=O)cccc2[nH]ccc12 c1(C(N(C2CN(C(C3CCCS3(=O)=O)=O)CC2O)C)=O)cncc2cccnc12 c1(CC)nn(C)c(NC2C3CN(C(=O)C(=O)Nc4ncc[nH]4)CC23)c1[N+](=O)[O-] C1(CC)CCCN(C(=O)C(C)N(C)C(C)=O)C1C(=O)N.c1cccc(C#N)c1 C1(NC(C2CCC(C)(C)OC2)=O)CCC2CN(C(C3CCC(F)CC3)=O)CC2C1 N1(C(=O)OC(C)(C)C)CC2C(C(F)(F)F)CC2(NCC(C2CCCC2)=O)C1 C1(CC(=O)NC)CN(C(=O)C(C)OC)CCN1C(c1ccc(OC)c(Cl)c1)=O C1(C(=O)NCCCCCCNC(Cc2c(SC)cccc2)=O)CC(=O)OC1(C)C C1(NC(C2C3CCCC23)=O)CN(C(=O)C=CCO)CC2(CC2)C1 c1(C(=O)NCC(C(C)(C)C)NC(CCCSC)=O)cc2ccncc2s1 C(=O)(C#CC1CCC1)N1CCC(C(C)NC(C(C)CC2CCCCC2)=O)C1 CC#CCC(C(=O)NC1(CCC)CC1)NC(=O)CCCC1CCCO1 C=Cc1ccc(C(=O)NC2CCCCC2CNC(=O)C(C)O)cc1.C1CCCC1 CC(CC(=O)NCC(C(=O)NCCc1nccs1)N(C)C)C(F)(F)F C1(CNC(C(CC)OC)=O)CN(C(c2cc(SC)cc(Cl)c2)=O)CC1(F)F C1(C(=O)NC2CC(C)N(C(=O)CCC=CBr)CC2)CCC2(CC1)CC(O)C2 c1(C=O)ccc2c(n1)NCC2.c1(SC)ccccc1CC(=O)NCCC1CC1.N Cc1c(Cl)c(C(=O)NC(CNC(c2cccc(O)n2)=O)C2CC2)nn1C N1(C(C2CN(S(CC)(=O)=O)C2)=O)CCC2(CC1)CN(C)C2.c1cc(O)cc(=O)o1 Cc1cnc(C(=O)NC2(CCCNC(c3ccc(F)c(C)c3)=O)CC2)c(C)c1 Cc1cc2c(cn1)CCN2C(=O)Nc1cnc(COC(C)(C)C)s1 c1(SC)cc(C(N2CC(NC(=O)CC3(C)CC3)CC(O)C2)=O)cc(Cl)c1 Cc1ccc(CCC(=O)NCC2CC3CC3N2C(=O)C2=CCSC2)c(C)c1 C(=O)(C1=CCCOCC1)N1CC2(C(CNC(C3(C)CCC(O)CC3)=O)CC2)C1 Cc1cn2cc(C(=O)NCC3CCCCN3C(C3CCCN3C)=O)sc2n1 c1(C(N2C3CN(C(c4cc(C)[nH]n4)=O)C(C3)C2)=O)c(Cl)ccc2c1OCO2 N1(C(C(CC)(COC)CC)=O)CCCC2(CCCN2C(=O)C(C2CCC2)OC)C1 c1(OCC)ccc(O)cc1C(N1CCCCC1C(=O)Nc1ccsc1)=O c1(C=O)cnc(O)n(C)c1=O.C(C(C)(C)C(=O)NC1CCCCC1)OCC.C c1(C(=O)NC2C(CNC(CC(C=C)C)=O)COC2)cc2c(OC)cc(Cl)cc2[nH]1 C(CCC(=O)NCC(CC)NC(=O)C(C1CCC1)OC)=CC C(=O)(CCCCC(C)=O)N1CCC(C(=O)NCc2c(OC)nn(C)c2)(CF)C1 C=C(Cl)CCC(=O)NCCC(Cc1ccccc1)NC(=O)C(COC)OC c1(CC)cccc(C(=O)NCC(C)(C)NC(C2CC(O)C2)=O)c1 N1(C(C=Cc2ncn(C)c2)=O)CCN(C(c2cncc3[nH]ccc23)=O)C2(CC2)C1 c1(C(=O)NCCCNC(C2C(C=C)OCC2)=O)ccc2c(C)noc2c1 C1(NC(C2CC(OCC)C2)=O)CC2(C1)CC(C=O)C2.C1(C)CC=CC1.N N1(C(C2N(C(CCN(C)CC)=O)CC3CC32)=O)CC2(C1)OC(=O)NC2C c1(C(=O)NC(CC)CNC(=O)CC(C)n2cccc2)cc(F)cc(C)c1C C1(OC)CC(CNC(=O)C(Cl)=CCl)N(C(=O)Cc2cncc(C)c2)C1 C1(NC(=O)CCN2CCC(O)CC2)COCCN(c2nnc(C(F)F)s2)C1 c1(C(=O)Nc2cc(O)ccc2F)ccc(Cl)nc1N=c1ccnc(C(F)(F)F)[nH]1 C(=O)(CC1=NNC(=O)C1)N.C1(CCOC)CCN(c2ccc(C(F)(F)F)cn2)C1 c1(N2CC(C)C(NC(=O)Cc3csc(C4CC4)n3)CC2)c(Br)cncc1[N+](=O)[O-] C(=O)(CCCS(N)(=O)=O)N1CC(CCCCNC(CCC2CCN(C)CC2)=O)C1 N1(C(CC2CCCO2)=O)CCOCC(C)(C)C1.C(C)(C(=O)N)OCCOCC c1(CN2CC(N3CCN(C(c4cncs4)=O)CC3)C2)c(F)ccc2occc12 N1(C(C(CC)C(C)O)=O)CC2CC(NC(c3cn(CCCOC)cn3)=O)CC1C2 N1(CCCNC(C2CC(C)(O)C2)=O)CCN(C(=O)Cc2cccc(O)c2)CC1 N1(C(C(C)Cc2cnco2)=O)CC(NC(c2ccccc2C(N)=O)=O)C(F)C1 c1(C(N(C2CCN(C(C3(C#N)CCOCC3)=O)C2)C)=O)cnn2c1OCC(O)C2 c1(C(N2C(C)CC(NC(c3c(C)noc3C)=O)C2)=O)cnn2ncccc12 C(=O)(C(CCSC)NC(C1CCC2CC12)=O)NCCOC CC1=CCC(N=c2[nH]c(N3CCOCC3)nc(=NCCOC(F)F)[nH]2)CC1 c1(C(=O)NC(CC(C)NC(COc2cc(C)on2)=O)C)ccc2nc(C)sc2c1 N1(C(C2CCC(=C)CC2)=O)CC2(CC2)CC1C(=O)NC1CCC(CO)C1 C1(NC(C(C)OCC=C)=O)CC(C)CN(C(=O)CCOC(C)C)C1 Cc1ccc2ncc(C(N3CC4CC3CC4NC(=O)C3=CCCCO3)=O)cc2c1 C1(C(=O)NCCC=CC=C)CCC(C)N(C(c2ccc(C)o2)=O)C1 C1(C=O)CC2OC(=O)OC2C1.Cc1cn(C(C)C)cc1C(=O)NCC(C)(C)C C(=O)(C#CC(C)(C)CNC(C1(C)CCCC1)=O)N(CC(CC)OC)C C1(CC(N2CC(O)(C(C=O)F)C2)=O)CC2(CCC2)C1.C1(CC)CCCSC1C.N C(N=c1cc[nH]c(=NCCCCc2ccc(Cl)cc2)[nH]1)C1CCCCC(F)(F)C1 c1(C(N2C(CNC(CCC(C)(C)C)=O)COCC2)=O)cc(C#N)c(N)cc1O c1(C(=O)NC(c2cnn(C)c2)C(=O)NC(CN(C)C)CCO)sccc1C#N N1(C(Cc2nc(C)sc2)=O)CC(CNC(=O)C2=CCCC2C)CC(C)C1 Cc1cc(C)c(C(=O)NCCCC2(NC(=O)C(F)CC3CC3)CC2)cc1C N1(C(C(c2cccc(C#N)c2)C(C)C)=O)CC2(CCC2)CC1C.C(=O)(C1CC1)N C1(CCC(=O)N2CC(N3CCN(C(c4cnco4)=O)CC3)C2)CCCC(O)C1 N1(C(CS(CC)=O)=O)CCC2(CCC2)C(CNC(C2CCC(C)(C)O2)=O)C1 c1(CNC(CCC2CCN(C(C(n3ncc(C)c3)C)=O)C2)=O)cc(O)ccc1C c1(CC(=O)N(C2CCN(C(=O)C3=CCCC3)C2)CCC)cccc2ccncc12 C(=O)(C1CCCc2scnc21)N1CC(C2(CNC(C3COC3)=O)CC2)(O)C1 c1(N(CCCCCC=C)C)nc(N(CC(=O)OC(C)C)C)c2c(n1)COC2 C1(CNC(c2cnc(S)nc2)=O)CCN(C(=O)CCCc2ccc(F)cc2)CC1 c1(C2C(NS(Cc3cccc(C)c3)(=O)=O)C2)ccc(C#N)cc1 c1(C(=O)NC2(C(=O)OCC)CC2(C)C)ccc(CC#N)cc1.C1CC1.C c1(C(=O)NC2CC(C)N(C(=O)COc3cnn(C)c3)C2)cnc2sccn2c1=O c1(C(=O)NCCC(CNC(C2(SC)CC2)=O)O)coc2ccc(Cl)cc12 C1(NC(c2cccc(C(=O)NC)n2)=O)CCN(C(c2nocc2C)=O)C(C)C1 C=CC(CC(=O)N(CC(C)(C)CNC(=O)CCC(=O)NC)C)c1ccccc1 N1(Cc2ccc(-c3cnc(C(C)(C)C)nc3)cn2)CCN(CC(=O)O)C(=O)C1 N1(C(c2c(C)[nH]c(C#N)c2)=O)CCC2(CC(NC(c3cccc(=O)o3)=O)CO2)C1 CN1CCCCC1C(N1CCCCC1C1CCN(C(C2(C)CC(F)C2)=O)C1)=O C1(F)(CNC(C2C(C)(C)CC2)=O)CCC(C)C1.c1(C=O)ccc(F)cc1.N CC(C)CC(CC(C)C)C(=O)NCC1C(C2CC2)CCN1C(c1n[nH]cc1Br)=O S(=O)(=O)(c1sncc1Br)N1CCC(Br)=C(C)C1 Cc1cc(C(=O)NCC2CCCN2C(=O)CCc2nnc(C)n2C)n2ncnc2n1 c1(OC)ccc(C(=O)NC2CC2C(=O)Nc2onc(C)c2C)cc1N(C)C N1(C(C2C(C)C2)=O)CCN(C2CCC(NC(C3CCC(=O)N3)=O)CC2)CC1 C(=O)(C#CC1CCCCC1)N.C1(C)(COC)CCCN1C(=O)C=Cc1cn[nH]c1 N1(C(CC(C=C)c2ccc(OC)cc2)=O)CCC(CC)(NC(C2CC2F)=O)CC1 C(C(=O)NCC1(C#N)CCOCC1)(C(C)CC)N(C(CCCCOCC)=O)C c1ccc([SH](=O)=O)cc1F.C1(CCC2CCCO2)CCN(C)C1.C(CN)OCC C1(NC(C(CC)(C)O)=O)COC2(C1)CN(C(=O)Cc1cncc(O)c1)C2 C12(C(N(C)CC3CCC(CNC(C(C)C)=O)CC3)=O)CC1COC21CCC1 c1(C(N(CCCNC(=O)CCc2ccon2)C2CC2)=O)cnn2c1CCCC2 c1(SC)ccsc1C(=O)NC1CCN(C(C2C(C)C2C)=O)C1 c1(CC)cc(OC)ccc1C(N1CC(O)C(O)C1C)=O.C(=O)(CCC(N)=O)N c1(C(C)C)nccc(C(=O)NCC2CCN(C(c3cncc(C(F)F)c3)=O)C2)n1 C1(C=O)CCC2CC1CO2.c1(C(C)(C)C)n[nH]cc1C(=O)NCC(C)C1CC1.N c1(OC)ccccc1C=CC(=O)NCC(C)C1CC1.c1(C=O)nc(Cl)sc1Cl.N N1(C(C(C(C)(C)C)O)=O)CC2(C(N3CCC4CCCC4C3)=O)CCC1CC2 n1(CC(=O)NC2(C)CCN(C(C(C)=C3CCC3)=O)C2)cnc2c(cnn2C)c1=O O=C1CC(=O)CC(C(=O)NCCC(F)Cn2cc(CO)nn2)C1 C1(NC(CCCC(=O)NCC)=O)CCCC2CN(C(c3cc(C#N)c[nH]3)=O)CC12 C(=O)(C1=CCOCC1)N(c1ccc(Cl)cc1)C1CCN(C(C2C(C)C2)=O)CC1 c1(CC)cc(C(N2CCC(C)(NC(C3C4CC5C(C4)C35)=O)C2)=O)ccc1F N1(C(CC(C(C)OC)NC(c2cscc2C)=O)=O)CCC12CCN(C)C2 CC(C)S(=O)(=O)C1CCN(C(=O)NCC2CC3CCC2C32CC2)C1 N1(C(C2C(OCC)C2)=O)CC2(CCCN(C(c3c(Br)ccc(N)c3F)=O)C2)C1 N1(C(c2c(CC)noc2)=O)CC2CCC(NC(=O)CC(C)O)(C2)C1 Cc1ccc(O)c(CC(=O)NC(C)CC2CN(C(=O)Cc3ccc(O)nc3)C2)c1 C1(CN(C(CCCN(C)C)=O)C)CN(C(=O)C(F)(F)C2CCOCC2)CCO1 C1(C(=O)NC2CCCC2C(=O)Nc2cnc(O)c(Br)c2)CCc2ccccc2O1 c1(C(N(CCN(C(=O)CCCN2CCCC2)CC)CC)=O)cc[nH]c(=O)c1 C1(C2(O)CN(C(=O)CC)C2)CC1.c1(C(C)=O)cccc(C(=O)N)c1.C(N)=O N1(C(CP(C)(C)=O)=O)CCN2C(=O)C(NC(c3ccnc4[nH]nnc34)=O)CC2C1 C1(C)(C(=O)NCCNC(c2nc(OC)nc(O)c2)=O)Cc2ccccc2NC1=O c1(CNC(C=COCC)=O)n[nH]c2c1CN(C(c1ccc(C)c(C)c1N)=O)CC2 N1(C(c2ccc(O)nc2)=O)CCC2(CC1)OCCC2NC(C12CCC1C2)=O Cc1cc(C(=O)NC2CC3CN(C(=O)Cn4nc(C)cc4N)CC23)nc(O)n1 c1(-c2n(CCOCC)c(N3CC=CC(OC(C)(C)C)C3)nn2)cnc(Cl)cc1C C(=O)(C1=CC2CC3CC(C2)CC1C3)NC1(CO)CN(C(c2n(C=C)ncc2)=O)C1 CC1CCCc2nc(C(=O)NCC3(CNC(c4cscn4)=O)CC3)cn21 C1(C(N(C)CCOCCNC(=O)C=C2CCC2)=O)C2CCCCCC12 CCCC(C)(CCC)C(=O)NC1CC(NC(c2n[nH]c3ccc(Cl)cc23)=O)C1 C(C)(CO)(C(=O)NCC1(CO)CCN(C(C23CCCC2C3)=O)C1)OC C(CNC(=O)C=C(Cl)Cl)(C(C)C(C)C)NC(C1CC(OC)(OC)C1)=O C(C)(C(C)C(=O)NCCCCN1CCCC1)NC(C=C(C)C(C)(C)C)=O CC(O)C(F)(F)C(=O)N1CC=C(CNC(c2cnc(C3CCC3)s2)=O)CC1 c1(NC(CC#CC)CO)ccc(S(=O)(=O)NC2CCCC2COC)c(Br)c1 c1(OC)cc(C)cc(C(N2CCC(NC(c3csnc3OC)=O)C(C)C2)=O)c1O CC1CCN2N=C(C(=O)NC(C)(C)CCNC(C3CC4CCC3O4)=O)NC2=N1 N1(C(C2(C(N(C)C)=O)CC2)=O)CC=C(C(=O)NCC2CCCO2)C1 C1(CNC(COCc2onc(C)n2)=O)C2CN(C(C3CC3(Cl)Cl)=O)CC12 O=C(C1=NN2CCCN=C2N1)NC1CCN(C(C2CCCSC2)=O)C1 C(CC1C(=O)Nc2ccc(F)cc21)NCC1(OCC)CCOC1(C)C Cc1cc(C(N2CC(NC(c3nn(C)nc3C)=O)CCC2C)=O)cc(C)c1C#N N1(C(C2(CC=C)CC2)=O)CCCC2(CCN(C(=O)C=C(CC)CC)C2)C1 N1(C(c2ncsc2)=O)CCN(C(=O)C)C2CS(=O)(=O)CC12.O=CC1CC1.N C12(C(=O)NC(CC)CNC(=O)Cc3cccc(Br)c3)CC(C1)OC2(C)C.C N1(CC(=O)NCCN(C(C2CCC3CCC2O3)=O)CC)CCCCC(O)C1=O CC1(NC(=O)Cc2cccc(F)c2F)CCCN(C(c2c(N)cccc2F)=O)C1 c1(COCC)nc(Cn2cc(CCC3CCCCO3)nn2)c(C)s1 c1(OC)cccc2c1OCC2NC(CC(=O)O)c1nccs1 N1(C(c2[nH]c(=NC)sc2)=O)CCCN(C(=O)C2=CC(C)(C)C2)CC1CO N1(C(c2c(F)ccc(OC)c2)=O)CCOCC12CCOC2 N1(CC(N2CC(N(C(=O)Cn3cc(N)cn3)C)C2)=O)CCCNC1=O C1(C(NC)=O)CC(C2CC2)=NO1.C(C)(C(C(=O)N1CCOCC1)N(C)C)OC.C C(=O)(C1OCCn2ccnc21)N1CCC(F)(CNC(C2(C)CC(=C)C2)=O)C1 c1(CC(=O)NCC2OCCN(C(C(CSC)OC)=O)C2)cc(F)ccc1F Cc1ccc2c(CC(=O)NCC3(NC(C4OCCOC4(C)C)=O)CC3)coc2c1 C(=O)(CCC(=O)NC1CCCC1(C)CNC(c1ncn(CC)n1)=O)OCC Cc1nnccc1C(=O)NCCC(C)CCNC(=O)CCC(=O)N1CCOCC1 C1(NC(c2c(CC)n(C)nc2)=O)CN(C(=O)Cc2cn(C)nn2)CCC1C C(N=c1[nH]c(Cl)nc(C)c1F)C1(CC#C)CCCC1.c1(CC=O)c(O)ncnc1O C1CC(C)CN(C(=O)C)C1.c1ccc(Cl)c(F)c1.C(=O)(CC(=O)N)NCC#C C1(C)(C(=O)Nc2c(C)nsc2)C=CCN1C(=O)C(Cl)Cl C1(C2CC2)(CNC(C(CNC(COCCCOC)=O)C)=O)CCC1 C=C(Cl)CC(C(=O)N1CCCC(O)CC1)NC(=O)CSC N1(C(C2CCCC(C)CC2)=O)CCc2ccc(-c3nn[nH]n3)cc2C1 N1(C(CC2CCC(NC(c3c(F)cccc3F)=O)C2)=O)CC2COCC(C2)C1 N1(C(c2cnc(C)s2)=O)CCCN(C(=O)C(F)(F)C(C)O)CCC1 c1(CN2CCN(C)C(C3COC3)C2)cc2c(cc1Br)OCCO2 C1(NC(CCOC)=O)CCC(C)(CNC(=O)C2=C(C)CC2)C1 N1(C(C(C)CO)=O)CC(CNC(=O)CCN2CCOC2=O)CC12CCOCC2 c1(OC)cc(N)c(C(=O)NC2CN(C(c3cc(C)ccc3Cl)=O)CC2C)cc1F c1(CC)ccc(C(=O)C(=O)NC(C)C(N)c2ccco2)s1 C1(C=O)CC(F)(F)CN1C(=O)CC=O.C(=O)(C(C)CC)OC.C(C)(C)C.N Cc1nnc(N2CCC(C(=O)N(C)CCO)CC2)c2ccccc12 C1(C(=O)NCCCCC(N)=O)CN(C(=O)C(=O)N)CC1C1CC1.CC.C(C)=O C(=O)(C1=C2CCN=C2NC=C1)N1CCCC(N(C(c2sc(C)cc2Cl)=O)CC)C1 C1(NC(c2scc(C)c2)=O)CC2CCC1CN(C(=O)CCCc1ccccn1)C2 N1(C(c2nccc(CC)c2)=O)CCC2(CC(NC(=O)C3=COCCO3)CO2)C1 C1(O)(C(=O)NCC(C)NC(=O)C(C)(C)N2CCCC2)CCSCC1 c1(CC)cncc(C(=O)NC(CO)C(=O)NCCC(O)CC)c1 Cc1ccc(F)c(C(=O)N(CC(C)CNC(c2occc2F)=O)C)c1Cl CCC(C)(CCNC(c1snnc1C)=O)NC(=O)CN(S(C)(=O)=O)C c1(C(=O)NC2CCN(C(c3scc(OC)c3)=O)CC2F)cn2cnnc2cn1 CCCCC(C)(F)C(=O)N1CC2CC2(CNC(=O)CC2(C)CCCCC2)C1 N1(C(CCS(=O)(=O)NC)=O)CCCC12CCN(C(c1ncsc1C)=O)C2 C(=O)(C(F)C(F)(F)C(F)(F)F)NCCC(CNC(Cc1ccc(C)o1)=O)(C)C CCCCCC(C)CC(=O)N(C)CCOCCNC(=O)CCC(C)C.C(C)(=O)O c1(C(N(C(CNC(COCCOCC)=O)C)C)=O)cc(C)cn2ccnc12 c1(-n2ncc(C(C(=O)NCC(F)F)N(c3cccnn3)C)c2)ccc(F)cc1 N1(C(C(C(C)C)C#N)=O)CC2CC(C1)CN(C(=O)CC(C)(C(F)F)N(C)C)C2 C(C(=O)NC(C1CCN(C(c2cnc(C)o2)=O)CC1)C)(C(C)(C)C)OC c1(C(N2C3(CNC(C4C(=O)NCC4)=O)CC(C2)C3)=O)ccc2c(n1)CCCN2 C1(C(=O)NC(C2CCCN(CCC(C)F)C2)C)CS(=O)(=O)CC(=O)N1 C(=O)CC(C)CC(C)C.Cc1c(C(N)=O)cccc1C(=O)NCC1CCC1.C C1(CNC(=O)COC2CCOC2)CCCCN(C(=O)Cc2cccnc2)C1 N1(C(c2ncc(C)nc2)=O)CCC2CCN(c3nccnc3F)CC2C1 C12(C(=O)NC3C(OC)COC3)CC(CO1)N(C(=O)C(C1CCC1)OC)C2 CCCCC(C)C(=O)NCC1CCCCCN1C(c1scnc1CC)=O CC(C)CC(C)(O)C(=O)NC1CC(OCC(=O)NC2(C)CCC(C)C2)C1 N1(C(CCCC(=C)C)=O)CC2CCCN(C(c3cc(C(=O)OCC)n[nH]3)=O)C2C1 CC1=C(C(=O)NCCCC2CCN(C(C3OCCO3)=O)CC2)S(=O)(=O)CCO1 C1(C(=O)NCCOCCC#C)CC(N=[N+]=[N-])CN1C(=O)C(O)C=CC C1(NC(CC(C)c2cnn(C)c2)=O)CC2(CCN(C(=O)CCSC(F)(F)F)C2)C1 C(=O)(C(CC(C)C)C(C)C)N1CCCC(COC)C1.c1(C=O)cn(C)c(O)n1.N N1(C(Cc2nc(C)[nH]n2)=O)CCC(C(=O)NCCC(F)CN=[N+]=[N-])C12CCC2 C(=O)(C(C(F)(F)F)C(F)(F)F)N1CCC(CC)CC1.CCC(C)(COC)C(=O)N c1(CN2C3CN(C(=O)Cc4cccc(F)c4)C(C3)C2)c(F)ccc(Br)c1F c1(CSC)ccc(C(=O)NC2CCC2)o1.c1(C=O)c[nH]nc1C1CCCO1.N Cc1cccc(C(F)(F)C(=O)NC2CCCC2NC(=O)CO)c1.c1nc[nH]n1 C(CCP(C)(C)=O)NC(C(COC)NC(=O)C(C)C1CC1)=O CCC(C)C(C)C(=O)N1CCCN(C(=O)Cc2cccnc2)CC1 c1(C(C)NC(C23CC(c4ccccc4)C2C3)=O)ccc(-n2ccnc2)cc1 c1(CC(=O)N)cccc(C#N)c1.CC(C)C(C(=O)NC1(C)CC1)n1cnnc1 C1(CNC(C(F)OC)=O)CCN(C(=O)C(C)OCCc2ccccc2)CC1F c1(C(N2CC(CCNC(C3(C)CCCOC3)=O)C2)=O)csc2ncnc(O)c12 CC(C(=O)N(C)CC1CN(C(=O)Cc2ccco2)CCO1)S(C)(=O)=O N1(C(C2(NC(=O)NC)CC2)=O)CCC(=CCNC(=O)CCC)CC1.O c1(N2CCC(OCC=C)C2)nc(N2Cc3c[nH]nc3CC(C)C2)nc2ccsc12 C(=O)(C1CCCc2ncnn21)N1C2C(NC(C(C)CC(C)(C)C)=O)CC(CC2)C1 N1(Cc2cnc(C)s2)CC2CC(NC(c3ccc4c(c3)COC4)=O)CC1C2 N1(CC(C)O)CCC(CNC(c2ccc(C(=O)O)cc2)CC#N)CC1 C1(C(=O)Nc2scc(C(C)C)n2)CN(C(=O)C(C)(C)CCl)CCS1 c1(C(N2CC3C(CC(=O)O)C3C2)C(=O)NCCOC)cccc2nnn(C)c12 C1(N(C2CCCC2)C(CCc2ccc(C(=O)OC)[nH]2)=O)CCCN(C(C)=O)C1 C1(C(=O)NC2CCC(NC(c3c(C)sc(O)n3)=O)CC2)CCCCC1(C)C C1(NC(=O)C=Cc2cn[nH]c2)CCCC(O)CC1 N1(C(C2N(CC)CCC2)=O)CC2C=CC1C(C(=O)NC(C)(C)C(C)O)C2 c1(NCc2c(OCC#C)cccc2)cc2c(cc1Cl)NC(=O)CO2 c1(C(N2CC(NC(CC(CC)C(F)F)=O)C(C)C2)=O)ccc2sc(=N)[nH]c2c1 C1(CCOC)CCN(C(=O)CC)C1.c1(C(=O)N)cnc(C(F)F)nc1.C(C)C C1(NC(C2CCCOCC2)=O)CCSC12CN(C(c1c(F)cc(F)cc1Cl)=O)C2 N12CC(C3(CC3)C1)N(C)C(C)CC2=O.C1(n2cc(SC)nn2)C2CC3C(C2)C13 c1(C(=O)NCC(C(=O)O)Cc2ccc(C(F)(F)F)cc2)ncn2cc(Br)sc12.C C1(C(C)C)CN(C(c2ccccc2CO)=O)CCN1C(=O)CC1CC=CC1 N1(CC(=O)Nc2c(C)cco2)CCCCC1COC(=O)NC(C)(C)C C(=O)(C1=C(F)CN(C(c2nc(=N)cc[nH]2)=O)CC1)NC(C1CC1(C)C)CC c1(C(N2CCC(C)(C(=O)Nc3snc(C)c3C#N)CC2)=O)cccc2nsnc12 c1(C(N2C(CNC(CCCc3cc(C)no3)=O)CC2)=O)cnc2n1C(C)CCC2 C1(C(N2C(C)CN(C(C3CC3C)=O)CC(C)C2)=O)CC12C1CC3CC(C1)CC2C3 N1(C(C2C(COC)C2)=O)C(CNC(c2ccncc2F)=O)CC2CCCC12 CC1CCC(NC(c2cc[nH]c2C2CCCC2)=O)CN1C(=O)CC1CCCOC1 CC#CCCC(=O)N(C1CCN(C(=O)COC)CC1)CC1CC1.c1nccn1C N1(C(CCCOC(C)C)=O)CC2(CO)CC1(C(N1CC3(C1)CN(C)C3)=O)C2 c1(C(N2CCCC(NC(C(C)(C)C(N)=O)=O)C2)=O)cc2cc(Cl)ccc2s1 CCCC(C=O)NC(C)=O.C1C2CC1N(C(c1ccc(C(F)(F)F)nc1)=O)C2.N N1(C(c2c(C)coc2C)=O)CCN(C(c2ccn(C(F)(F)F)n2)=O)CC1C N1(C(Cn2ncc(C#C)c2)=O)CCN(C(c2cc3sccc3[nH]2)=O)C(CC)C1 C1(NC(=O)CC2COCCN2C(=O)COC2CCCCC2)CCC=CCCC1 N1(c2ncn(C)c(=O)c2)CCC2(CCCN(C(c3c[nH]c4cnccc34)=O)C2)C1 C1(OC)(CNC(=NCc2ccsc2)NC(c2ccccc2)C)CCCSC1 CC(C)C(CC1CCC1)C(=O)NC1CN(C(C2(N3CCCC3)CC2)=O)CC1C Cc1cccc2c(=O)c(C(=O)NC3CC(C)C3)c[nH]c12.C(=O)(C(=O)N(C)C)N N1(C(c2ccc(Nc3c(C(C)C)cccc3)cc2)=O)CCC(C)(O)C(C)(O)C1 c1(CC(=O)OCC2Cc3nccn3C2)ccc(OCc2ccncc2)cc1 C#CC1(C=C)COCCN1C(c1cc(OC)c(OC)c(Cl)c1)C(=O)NC C1(CNC(C(C)C2CCCO2)=O)(NC(=O)C)CCC(C)(C)CC1.c1nc[nH]n1 c1(C(=O)NC(CNC(CC2N(C)C(=O)CC2)=O)C2CCC2)c(N)cccc1F C(CCCCC(=O)N(C1CC(C(N2CCOC(CCO)C2)=O)C1)C)OC C(=O)(C1c2ccccc2C2CC1C2)NC1CCCC(CNC(C(C=CC)O)=O)C1 Cc1cc2scc(CC(N3CC4CC(NC(c5c(C)ncn5O)=O)C3C4)=O)c2s1 CC1C(N(C)C(C2C(C)CN2C(c2cnn(C3CC3)c2)=O)=O)CCCC1C c12cn(nn1)C2.C1(CNC(=O)CC2(CO)CC2)COCCO1.C1CC12CCC2 Cc1cc(NC(=O)C(C2CCC2)NC(=O)C=Cc2cc[nH]c2)c(C)cc1F C(N=c1[nH]c(=NCCN(C)C2CC2)[nH]c2ccc(Cl)cc12)c1c(C)ccnc1C C(=O)(C(F)C(=O)NC(CCF)C(=O)N(C(C)C)Cc1ccco1)OCC C(=O)(C(C)(CSC)NC(=O)CCc1ccncn1)NCC.c1cncn1C N1(C(C(c2ccc(OC)c(F)c2)C)=O)CCC(NC(=O)C=C(C)Cl)C12CCCC2 CC1CCC(CC(=O)NCCSCC(N2CCC(OCC3CC3)C2)=O)CC1 N1(C(C2C(CC)CCO2)=O)CCOCC1CN(C(=O)C=CCO)C CCCCCCOCC(N1CCCC1CNC(C1(OC)CCOC1)=O)=O c1(C(=O)NC(CC)CNC(c2ncccc2C)=O)cccc2nc(O)n(C)c12 c1(C(=O)NCc2occ(C(N(C(CC#C)C)C)=O)c2)cn(C)c(=O)n1C N(C1CCC(NC(c2cc(F)c3[nH]nnc3c2)=O)c2ccccc21)C(C=CC)=O C(C(=O)NNC(=O)C(C)(C)CCCCNC(C1CC1Cl)=O)Nc1ccc(C)s1 N1(C(c2nc(CCC)oc2)=O)CCC(O)(C(C)NC(c2ccc(C)o2)=O)C1.C C1(NC(CCCC=C)=O)C(C)CN(C(=O)Cc2cc3ccccc3s2)CC1C c1(C(N2C(C)CC(NC(C(C(C)C)NC=O)=O)C2)=O)ccc2c(c1)CC(C)O2 c1(C(=O)NCCN(C(c2sccc2F)=O)CC)ncsc1C(F)(F)F CCCC(C(=O)NC1(C)CCN(C(c2cccc(-c3cnco3)c2)=O)C1)N(C)C c1(C(N2CC(C)C(CNC(C34CCC(CC3)OC4)=O)C2)=O)ccc([N+](=O)[O-])s1 Cc1ccc(CC(=O)NC(C2CN(C(c3ccc(C4CC4)s3)=O)C2)C)cc1C N1(C(C2(CC#C)CCN(C(c3cc(Cl)no3)=O)C2)=O)CCC(C)(C)C1C c1(NC(C2N(C(c3cc(C(C)=O)on3)=O)CCCC2)=O)cccc(F)c1O c1(C(=O)NCCC(=C)CNC(=O)Cc2ccnn2C)cncc(C(N)=O)c1 c1(C(N2CC(NC(C(C(C)(C)C)OC)=O)C(F)CC2)=O)c(N)ccc(F)c1C C1(C(N(C(C)C(=O)NCC(C)(C)C)CC)=O)COC(=O)N1C c1(CC(=O)N)cccc2nonc12.c1(C(N(C(C)C2CC2)C)=O)ccc(F)cn1 N1(C(C(C)S)=O)CCC(C(=O)Nc2sccc2C(C)C)C1C(C)C C1(CCNC(C=CSC)=O)CCCN(C(C2CCCN2C)=O)C1 N1(C(C2C(C)C2)=O)CCc2c(-c3cc(F)c(CO)c(F)c3)cccc2C1 N1(C(C=Cc2ccc(CC)o2)=O)C2CCC1CN(C(c1ncnc(C)c1C)=O)C2 CC1CN(C(=O)C(c2ccc(Cl)nc2)(F)F)CCCN1C(=O)Cc1csc(=N)[nH]1 C1(c2n(CCCOC)nnn2)(NCC(C)CO)CC(C)(C)OC(C)(C)C1 C1(C(N2CC3(CN(C(c4cccc(OC)c4)=O)C3)C2)=O)CCOCC12CCCC2 c1(OC)c(C(=O)NCC(CNC(c2coc(Cl)n2)=O)CO)cccc1F c1(C(=O)NC2CC(CNC(C3(C)C(C)C3)=O)C2)cc(Br)c(F)cc1N c1(C(N2CCC(O)(CNC(c3csc(S)n3)=O)C2)=O)cc(F)cc2cnccc12 Cc1cc(NC(C2COCCN2C(=O)C(C)Cn2cccn2)=O)ccc1I CCC(CC)(C(=O)N1CC(CC(=O)NC(c2cccc(Br)c2)CO)C1)C(=O)O C1(NC(C2CC(O)CN2C(C2CCC=CCCC2)=O)=O)CCCC(O)C1O C1(C(N2CC(CC(C)NC(=O)Cc3nc[nH]n3)C2)=O)(CC)CCCO1 c1(OC)ccc(Cl)c(F)c1C(=O)NC1CC(N(C)C(C2CCCOC2)=O)C1 c1(C(N2CCN(C(c3c(OC)scc3)=O)CC(O)C2)=O)[nH]nc2ncnc(O)c12 C(=O)(C#CC1CCCO1)N1CC(OCCNC(c2cc(COC)[nH]n2)=O)C1 Cc1nc2ccnn2cc1C(=O)NC(C)C1CC1.C1(CC=O)CCN(C)C1=O.N C1(NC(=O)CCF)CCC2(CC1)CCN(C(c1cc3n(n1)CCCC3)=O)C2 c1(N(C(C)=O)C)ccc(C(=O)N(C)CCNC(c2cccnc2C)=O)cn1 C=CC1CCN(C(=O)C(C)=C(C)C(c2ccc(Br)cc2)=O)C1 c1(C(n2cc(-c3cnn(C)c3C#N)nn2)CC)ccc(Cl)c(Cl)c1 n1(CC(=O)OCC)ncc(C=O)c1N.C1(C)C(=O)N1.C1CCC1.C(C)C c1(CC)cc(CC(=O)NCCC2CCCN2C(=O)Cc2nnc(C)o2)n(C)n1 C1(O)(CC(N2C(CCNC(c3cn(C)nn3)=O)CCC2)=O)CCCCC1 c1(C=O)oc(C=O)cc1C.C1(CC)CCC2CC12.C12(CC1)C(=O)NC2.N C1(NC(CCCC(C)C)=O)COC2C(NC(c3c(Cl)csc3Cl)=O)COC12 C12(NC(C3CCC(C)CC3)=O)CCC(C(=O)NC3C(O)C4CCOC34)(CC1)C2 N1(C(CC2(C=C)CCOCC2)=O)CC2OCCN(C(=O)CC(C)(C)CCC)C2C1 C1(C(=O)NC(C)(C)CCCNC(c2ccnn2CC(F)F)=O)COCCC1(F)F C12(C(N3CCOCC(NC(=O)CC4CC5OCCC5O4)C3)=O)CCCCN1CCC2 c1(CC(=O)N(CC(C)(C)NC(c2c(C)con2)=O)C)c(C)nn(C)c1C N1(C(COCCOCC#C)=O)CCC(N(C(=O)C(CC)N(C)C)CC)C1 N1(C(C)=O)CC(O)CC1C(=O)NCCCN(C(=O)C(C(C)C)n1ccnc1)C C12(NC(=O)Cc3ccc(Cl)cn3)CCN(C(=O)Cc3cnccn3)CC1C2 C(C(COC)C(=O)N1CCC(NC(C2CC(=C3CCC3)C2)=O)C1C)OC C1(C(=O)NCc2nc(C)[nH]n2)C2CC1N(C(=O)CS(C)(=O)=O)C2 c1(C(=O)NCC(C)NC(=O)C=Cc2ccncc2)cccc2ccc(O)nc12 C1(CC(N2CCCCC2CCO)=O)COCCN1C(c1ncsc1Br)=O C(=O)(C1CCc2c[nH]nc21)N1C(CCN(C(C=CC=CCC)=O)C)CCCC1 c1(CC(N2CCC(OCCCNC(=O)CC(F)F)CC2)=O)csc2ccccc12 c1(-n2cc(CC3CCN(C4(c5c(CC)cc[nH]5)CC4)C3)nn2)cc(F)cnc1Br C=CC(C)(O)C(=O)N(CCNC(=O)COc1ccn(C)n1)C1CC1 C(=O)(C(C)NC(=O)C=CCN(C(=O)C(O)C1CCC1)C)NC(CC)C c1(C(=O)NCCC(C)NC(C2CCSC2)=O)cccc(N2CCCS2(=O)=O)c1 c1(CN2C(C(=O)Nc3nnc(Cl)cc3C(=O)O)CSCC2)cc(F)cnc1Cl c1(C(=O)NCc2cccc(C)n2)cn2c(n1)CCN(C1CCNC1(C)C)CC2 N1(C(=O)C=Cc2cncs2)CCC2(CCN(C(c3cnc(O)c(Br)c3)=O)C2)C1 c1(C(=O)NCC2CCN2C(C2CC2c2cccnc2)=O)ccc2c(n1)CCO2 c1(C(=O)NC2CN(C(CC(=C)Br)=O)CC2C)cc2cc(Cl)ccc2[nH]1 C(=O)(Nn1cnc2ccccc12)C1(C(=O)NC)CC1.N12C3CCC1CC(C3)C2=O c1(C(C)=O)ccc(CNC(c2nnc(O)nc2O)=O)nc1C C1(NC(C=CSC)=O)CCC(N(C)C(C2CCN(CC(F)(F)F)C2)=O)CC1 N1(C(c2c(C)cccn2)=O)CCN(C(=O)CNC=O)C(c2ccc(F)c(F)c2)C1 CC1(C)CC(CO)CN(CC(C)(C(F)(F)F)NC(=O)OC(C)(C)C)C1 CC(C)CC(C(=O)NC1CC(NC(c2ccoc2Cl)=O)C1)C(N)=O Cc1ncc([N+](=O)[O-])n1CC(=O)NC1CCC(C)N(C(c2ccncc2O)=O)C1 N(C(C(=O)NCCO)=Cc1cccs1)C(C)=O.C(C1CCC1)=CC=O.CC c1(C(=O)NC2C(NC(C(C)NS(C)(=O)=O)=O)CCCC2)noc2ncccc12 N=c1[nH]n(CC(=O)NCCNC(=O)CC2CCCO2)cc1Br Cc1cc(C(N2CC3C(NC(c4ncncc4F)=O)C3C2)=O)sc1Br C(=O)(CCC(C)(C)F)N(C(CC(F)F)C(=O)NC1CCN(C(N)=O)C1)C CC1CCc2[nH]nc(C(=O)NCC(C)(C)CCNC(=O)CCCC(N)=O)c2C1 C=CCN=C(NCC1COC(=O)N1)N1CCC(CSc2ccc(C(N)=O)cc2)C1 Cc1nc2[nH][nH]cc-2c(=Nc2nc(Cl)ccc2C(=O)Nc2cnnc(Cl)c2Cl)n1 CN1CCC(C(=O)NC2CCCC(NC(c3ccccc3)=O)C2)C1=O.C(N)=O.N N1(C(CNC(CC)=O)=O)CC(O)CC1C(=O)N(C)Cc1ncc[nH]1 Cc1cc(NC(C2CN(C(c3c(I)ccnc3Cl)=O)CCC2O)=O)c(Br)cc1F C12(C(=O)NCC(C)CNC(=O)CCC3CCC(=O)NC3)CCC(CC1=O)C2 N1(C(C(C)C2CC2)=O)CCN(C(C2(CO)CCOCC2)=O)CC1c1cnn(C)c1 C(=O)(CC(C)(C)O)NC(C1(O)CN(C(=O)CC2CCOC2)C1)C C1(NC(C(C)=C(CC)C)=O)CC2CC(C1)CN(C(=O)CN1CCC(C)(C)C1)C2 c1(NC(COC(C(CC=C)CC=C)=O)=O)c(C)ccc2ncccc12 c1(OC)ccc(OCCCS(=O)(=O)NC(=O)C(C)=CCN)cc1.C1C(=O)N1 N1(C(CN2CCN(CC)CC2)=O)C2CCC1CC(NC(=O)CCCCCO)C2 C1(C)(C=O)Cc2ccccc2C1.N1(C(C)C)C(=O)CCC1C(N1CCC1C)=O.N CCC(C)CCCC(=O)N1CC(CNC(c2coc(C(C)C)n2)=O)C(F)(F)C1 C(=O)(C(C(C)C)NC(=O)CC1CCCCC1)NCc1c(CC)c[nH]n1 c1(C(C)=O)cc(N2CCC(NC(C3CC(C)CC(C)C3)=O)C(O)C2)nc(C)n1 c1(C(=O)OCC)cc2ccccc2c(NC(C2CCCCCCC2)=O)n1 CCC1=C(C(=O)Nc2cccc(-c3nc(S(C)(=O)=O)n[nH]3)c2)CCCO1 c1(CC(=O)N(C(C)(C)C)CC2CCCO2)ccc(Br)cc1 CC1CN(C(C23CCC(CC2)OC3)=O)CCC1N(C)C(c1cccs1)=O c1(CC)cc(CC)[nH]c(=NCCNC(C2CC(=O)N(C3CCCC3)C2)=O)n1 CCC(C)CCCC(=O)NC(CO)C(C)NC(C1CCS(=O)CC1)=O N1(C(C(C)OCC2CC2)=O)CCCC2(C1)CN(C(c1cccc3c1CCO3)=O)C2 c1(C(N2CC3C(CC)(CC3)C2)=O)cc(F)c(F)c(F)c1.C1(C=O)CC1.CO.C C1(C(=O)NCCCOCCCNC(c2n(C)nc(Cl)c2)=O)CCc2nc[nH]c2C1 N1(C(C(C2CC2)SC)=O)CC2CCC(CNC(c3cnc4ccnn4c3)=O)C2C1 N1(C(C2CCCC2O)=O)CC(CO)C2(C1)CN(C(C1CCCC3C1C3(F)F)=O)C2 CC(C)CCCN(C(=O)CSCC(N)=O)C.c1(CC=O)cnn(C(F)F)c1 N1(C(C(C)(C)C#N)=O)CCC2(CCCC2C(=O)Nc2ccc(O)cc2[N+](=O)[O-])C1 C(=O)(CC1=CCCCC1)NCCC1(CNC(CC2C(C)(C)OCCO2)=O)CC1 C1(OC)CC2CC1CN(C(C13CC1CCN3C(c1cnn(CCF)c1)=O)=O)C2 C1(C(N(CC(O)CNC(=O)CCCC2CCC2)C)=O)CCS(=O)(=O)N1 N1(C(C)=O)CCc2ccccc2C1CC(=O)NCCNC(=O)CC1=NNC(=O)C1 c1(C(N2CC(C(N3CCC(C(N)=O)CC3)=O)SCC2)=O)cn2ccc(Br)cc2n1 C1(N(C)C)CCCN(C(c2ccc(I)s2)C(=O)Nc2ccccc2)C1 c1(C(=O)NCC(CNC(c2ncc(NC)nc2)=O)C)cccc(C)c1C c1(CC(N2CCN(c3nnc(C)o3)C(C(C)C)C2)=O)ccn2nnnc2c1 C(C(C(=O)NCC1(C)CCC1)OC)OC.c1(CC=O)cc(C(C)C)no1 CC1CC(NC2(c3nnnn3CCOCc3ccccc3)CCCSC2)CCS1 c1(CC=O)nsc2ccccc12.c1(SC)cccc(C(=O)NCC(C)=CC)c1.N N1(C2CC(OC)C2O)C(=O)NC(Cc2csc(C(C)C)n2)C1=O.c1ccccc1 c1(C(=O)NC(C(C)NC(CCc2scc(C)n2)=O)C)csc2c(O)ccnc12 c1(C(=O)NCCCC(C)NC(=O)Cc2cncnc2)ccc(-c2nccs2)cc1 C1(C#N)(C=O)CC(F)(F)C1.CC1CN(C(c2cccc(C(N)=O)n2)=O)CC1.C C1(CNC(C(C)(O)C2CC2)=O)C2CN(C(=O)Cn3ccccc3=O)CC12 C1(C)(CNC(CCc2n(C)ncn2)=O)CN(C(=O)CCc2ccccn2)CCO1 c1(C(C)C)cccc(C(=O)NCC2CCC(NC(=O)CC3CC3C)CC2)n1 N1(C(CCC(=C)C)=O)CCC2(CC1)CC(NC(=O)CCc1ccc(F)c(F)c1)C2 c1(C(=O)NC(CNC(c2n(C)c(S)nn2)=O)C2CCC2)cccc2c1OCO2 CC1(C)CC(NC(=O)CC2CCN(C(=O)CC3COCCOC3)C2)CCO1 c1(OCCNC(=O)OCC(F)F)cccc2cnc(Cl)cc12 C1(NC(=O)CSc2ccccn2)CCN(C(=O)C(F)C(F)(F)F)CC1CO CCCCC(C(=O)N1CC(C(=O)Nn2cncn2)CC1(C)C)C(C)C N1(C(c2ccc(=N)[nH]c2Cl)=O)CCN(C(=O)C(=O)NC2CC2)C2(CCC2)C1 C1(NC(C2CC(=O)N(C3CCCC3)C2)=O)CCCN(C(c2ccccc2O)=O)C1 N1(C(CC(C(C)C)OCC)=O)CC(NC(=O)C(C)(C)CSC)CC2(CC2)C1 Cc1scc(C(=O)NC2C3CC2N(C(c2cc(-c4ccco4)c[nH]2)=O)C3)c1C C1(CNC(c2ccc3c(c2)CCO3)=O)CC2COCC2N1C(C1(O)COC1)=O CCCCCCC(C)C(=O)NC1CCCC(NC(C2CCSC2)=O)C1 C1(CNC(CSC)=O)N(C(c2ccc(N)c(Br)n2)=O)CCC1(C)C C12(CNC(C3CC(SC)C3)=O)COCCN1C(=O)CN(C(c1csnn1)=O)C2 CC(C)(CNC(C1C2CC3C(C2)C13)=O)CC(=O)NC(C(F)F)C(C)(C)C c1(C(=O)NC2CN(C(c3cc(CC)nc(O)c3)=O)CC2C)c(C)ccc(C)c1O Cc1c[nH]cc(C(=O)NCC2CCCCN(C(C3CCC(N=[N+]=[N-])C3)=O)C2)c1=O n1(CC)ncc(C(N2CCC(C(C)NC(C3(C)CC3)=O)C2)=O)n1 N1(C(C=Cc2n(C)ncc2)=O)CCOC2CCN(C(=O)CCn3cncn3)CC12 c1(C(=O)NCCn2ccc(C(C)=O)n2)cc(F)cc(F)c1O c1(C(=O)NCC(CC(C)C)(C)NC(C2CCCC2(C)C)=O)cnn2cnnc2c1 C1(C(=O)NC(C(C)C)CNC(=O)Cc2ccccc2F)Cc2ccccc2CO1 N1(C(C(C)O)=O)CC2(C1)CN(C(c1cccc(C(N)=O)c1)=O)C2 Cc1ccc(CO)c(NC(C2CCC(O)CN2C(c2cn(C)ccc2=O)=O)=O)c1 N1(C(C2C(CC)CCC2)=O)CC2(C1)CN(C(C1CN(C)C1)=O)C2 C1CC2(CC2)CN1C(=O)CCCc1ccc(Cl)cc1.C(C)(C(=O)N)NC(C)=O Cc1ccc(Br)c(CN2CCCC2C(=O)NCC2CCC(CN)C2)c1F Cn1c(=O)[nH]c(N2CCN(c3cccc(F)c3)CC2)c(C#N)c1=O n1(CC=O)ccc2c(F)cccc12.c1(C(=O)N(C)CC2(C)COC2)cscn1 C(=O)(C(C(C)C)NC(=O)CCCC#N)N1CC(OC(CC)=O)C1 C(=O)(CCCS(N)(=O)=O)N1C(CNC(Cc2cc(OC)ncc2)=O)COCC1 n1(CC(=O)N)ccc(=O)n(C)c1=O.C(CC)(C(C)C)NC(C=C(CCC)C)=O C1(NC(C=NOC)=O)CC(C(F)(F)F)CN(C(c2ccc(C(C)(C)C)[nH]2)=O)C1 CCCC(CCO)NC(=O)C(CNC(=O)CC(C)(C)OC)CC1CCCC1 CC1CCC(C(N2CCCCC2C)=O)CN1C(=O)CCN(C)C N1(C(C2(C)CC=CC2)=O)CC2C=CC1C(C(=O)NC1CC(n3ccnn3)C1)C2 C1(C(=O)NC2(CNC(CC(C)C)=O)CCC2)CCOCC1C Cc1cc(=NC(=O)CC2CCCN(C(c3c(C(F)(F)F)coc3C)=O)C2)[nH][nH]1 c1(C(N2CCC(C)(NC(c3csc(C(F)F)n3)=O)C2)=O)ccn2nccc2c1 n1(CC=O)ccc2ccccc12.C(C(C)=CC(=O)NCCC1(C)CC1)OC C(C)(C)(CC(=O)N1CCCC(CC(=O)NCc2nc(C(C)C)n[nH]2)C1)OC c1(C(C)=O)ccc(-c2cn(CC3C(C)C3(F)F)nn2)s1.c1(CC=O)cncs1 c1(C(C)=O)cc(C(=O)NCC(C)CNC(c2[nH]nc(OC)c2Cl)=O)c(C)o1 c1ccc2ncn(C)c2c1.C1(N(C)C)CC(C(=O)OC(C)(C)C)CN(C(=O)N)C1 C(=O)(CC1CC(=O)c2ccccc21)N1CCC(O)(CNC(C2(CC)CC2)=O)C1 N1(S(CCCC)(=O)=O)CCC(O)C(C(=O)Nc2cc(C3CC3)nn2C)C1 N1(C(c2cccnc2Br)=O)CC2CCCC(C1)N2C(=O)COC1CCOC1 Cc1cccc(CCC(=O)NCC(C)CN(C(=O)Cn2cnnn2)C)c1 C1(c2n(C(C)(C)C)nnn2)(NCC(C)(F)C(C)(C)F)CC2CCC(C1)S2 c1(Oc2ccnc(OC)c2F)cc2n(n1)CCCO2 N1(C(C(CC#C)O)=O)CCC2(CC1)CCN(C(C1COC(=O)N1)=O)C2 n1(CCC)nccc1C(=O)NC1CC(N(C(=O)Cc2ccsc2Cl)C)C1 c1(C(=O)N)c(C)cc(C)nc1O.N1(C(C2C(=C)CC2)=O)CCC(CC(C)(C)C)C1 Cc1c(C(=O)NC2CC(CNC(=O)C3=CCOC3)C2)c(C)n2ccncc12 C1(NC(CCc2cc(C)on2)=O)CC2(C1)CC2NC(c1cc[nH]c1)=O CC1CCCN1C(=O)CC1CC=CC1.S(=O)(=O)(C(F)F)N1CC(C(=O)N)C1 Cc1nc(N(C)C)sc1C(=O)NCC.c1(C=O)cc[nH]c1C1CC1.CCC.O C(=O)(CC(C)(C)C)NC(C)C(N1CCCCC1C)=O.c1(C=O)ccnc(Cl)n1.N C(=O)(C(C)C(O)C(C)C)N1CCC(O)(CNC(C2(CC#C)CCCCC2)=O)C1 c1(OC)ccc(CC(=O)NC2CN(Cc3scc(Br)c3Br)CC2F)c(Cl)c1 c1(OCCN(C)C)nc(N(C(=O)C(C)(C)F)Cc2ccccc2)ns1 N1(C(c2cc(CC)no2)=O)CC(NC(=O)C(C)OC)C(CC(C)(C)C)C1 c1(CC)ccc(CCC(=O)NCC2CCCN2C(c2cnnn2C(C)C)=O)cc1 C1(C#N)(C(=O)NC(C)CC(C)NC(c2scnc2C(F)(F)F)=O)CC1(C)C C(c1cc(F)ccc1F)=CC(=O)N(C1CC12CCNCC2)Cc1ccsc1 c1(CC)ccc(F)cc1C(=O)NC1CS(=O)(=O)CC1NC(=O)CCCCC#N CCC(C)CCC(=O)NCC1CCC(NC(c2conc2C2CCC2)=O)C1 c1(C(N2CC(NC(C(C(CC)O)(F)F)=O)C(C)C2)=O)c(O)cnc2ccccc12 C(c1c(Cl)cccc1Cl)=C(C(=O)N(C1CCN(C(C(CC=C)CC)=O)CC1)C)C CC1CN(C(C2CC(N)CCO2)=O)CCC1(F)F C1(C(=O)N)C2CC(O)C(C2)N1C(=O)C1=CCCCCC1.c1(OC)cccc(C)n1 S(=O)(=O)(c1cc(C(C)C)no1)N1CCCC1.Cc1nc(N)sc1C(=O)O c1(N(C(=O)NCC(C)C2CCC2)C)cccc(F)c1F.c1ccccc1 c1(C(=O)NC(C(CC)C)C(=O)NCC(n2ccnn2)C)cc2cccn2cn1 C(C(COC)CC(=O)NCC1CN(C(=O)Cc2csc(C(C)C)n2)C1)OC Cc1cc(N2CCC(CF)(NC(=O)CCCNS(C)(=O)=O)C2)nc(C)n1 Cn1nc(C(=O)NCC2COC2)c2ccc(-c3ccc(I)cc3)cc12 C1(NC(C(CCOC)C)=O)CC2CC1CC2C(=O)NCC1(C(C)C)CC1 N1(C(c2c(C)con2)=O)CCC(CNC(=O)C#CC2CCCOC2)C(F)(F)CC1 c1(SC(C)C(=O)NCCCCNC(=O)Cn2cn[nH]c2=N)ccccc1 c1(NC(C2CCCC(CC)N2)=O)cc(F)cnc1Br Cc1ccc(=NCCC(=O)NC23CCCC2N(C(C2CSC2)=O)CC3)[nH]c1 CC(C)CC(CNC(=O)C(F)CC1CCC1)NC(C1CCC1)=O.C1CC1.C N1(C(C(=O)NCC)=O)CCC2(CCCCC2)C1.c1(C(=O)N)oc(C=O)cc1C c1(NC(N(C2CCCCC2)C(C#C)(C)C)=O)ccc(-c2cccc(OC)c2)cc1 C(=O)(C(F)(F)C(F)F)N1CC(CC(=O)NC2CN(C3CC3)CC2C)(OC)C1 c1(C(N2CCC(N3C(=O)CCC3=O)C2)=O)cc(OC2CCCC2)ccc1Cl c1(C(N(Cc2cn(CC3(CC#N)CC34CCC4)nn2)O)=O)ccc(F)cn1 C12(NC(c3c(Cl)cnc(C(C)C)n3)=O)CCCCC1N(C(C1OCCO1)=O)CC2 C1(C(=O)NC(C2(O)CN(C(CCCCCOCC)=O)C2)C)CCOC2(CCC2)C1 Cc1cccc(C)c1CC(=O)NCC1CN(C(C2CCC=CCC2)=O)C(C)(C)C1 c1(C(=O)NC(c2ccc(C)cc2)CNC(C(CC)F)=O)c(Cl)ccc(F)c1N C1(NC(c2c(C)nsc2N)=O)CCCCCN(C(c2cccn3cncc23)=O)C1 Cc1nc(O)ccc1C(=O)NC(CO)CCCNC(C1(C#N)CC1(C)C)=O CS(=O)(=O)c1nccc(N2CCC(F)(F)CC2C(=O)NCCN2CCCC2)n1.C Cc1cccc(Br)c1C(=O)NCC(C(C)C)NC(=O)CSc1nncn1C CC1OC2(CNC(=O)Cn3nc(O)ccc3=O)CC1C2.c1(C(=O)N)ccoc1 N12CCCC1(C)C2=O.CC(O)CC(=O)N1CCCC1C(=O)NCCC(F)(F)F c1(C=O)snc(O)c1Cl.C1CCC(CC)C1.CC(C)(C)OC(=O)C=CC=O C(C(C(C)C)NC(=O)CC1(NC(=O)C(C)C2CCC2)CCC1)OC CC(C)CC(F)(F)C(=O)NCCCCC(C)NC(C1CCCCC1(C)C)=O C1(OC)CC2CC1CN(C(c1occc1CNC(=O)C#CC(C)(C)O)=O)C2 C1(C(N(C(C=C)C2CC2)C)=O)(OC)CCN(C(C2CC23CCCC3)=O)C1 C1(CN(C(CC2CCC(C)O2)=O)C)COCCN1C(=O)C=CSc1ccccc1 c1(CC)cc(C)c(C=O)o1.C1(CC)CCCN1C(c1cnn(C2CCC2)c1)=O.N C1(C(N(CC(CN(C(C2(CCCC)CC2)=O)C)O)C)=O)C2CCCCC12 C(CC(COC)NC(C1(NC(=O)C(F)F)CC1(C)C)=O)OC n1(C(C2(C)CC2)C)nc(-c2ccccc2)nc1C1CCN(C)C1=O c1(C(=O)NC(CC(C)C)CNC(C2CC(F)C(=O)N2C)=O)cccn2ccnc12 Brc1ccc2ncnc(NCC3CCCCC3c3ccccc3)c2c1 C1(OC)COCCC1CNC(c1ccoc1CC(N)=O)=O C1(NCc2cc(OC)ccc2)CCCCN(CC)C1=O.N1(CCOC)CCOCC1 N1(C(c2c[nH]cc2C(F)(F)F)=O)Cc2cccnc2N2CC(O)CC2C1 C1(C=O)C(C)(C)C1(F)F.c1(OCC)sccc1C(=O)NCC1CCC1 c1(CC(=O)NCC2CCCN(C(=O)C=Cc3ccoc3)C2)nc2c([nH]1)CCCC2 c1(C(N2CCC(CNC(C3CC4C=CC3C4)=O)CC2)=O)cc2c(F)cccc2[nH]1 Cc1nc(C(N2CCC(=CC)CC2)=O)cn1C(F)F.C1(C)(CC=O)CCC1.N CCC(C)C(C(F)(F)F)NC(=O)Nc1nc(C)c(C)s1 c1(NC(CN(C(C(C)N2CCC2)=O)C)C)snc(Cl)c1C#N N1(C(c2cc(C)ccc2F)C(=O)NC(CC)C)CCC(OC)C12CCC2 c1(C(N2CCCCC(CNC(C=CC=CCC)=O)C2)=O)sc2nccn2c1C CC(=O)C(C)CC(C)C(=O)N1CCCC(C(=O)Nc2cccc(C)c2)C1 C(=O)(C(O)CCN(C)C)NC(C1CCN(C(c2coc(Br)c2)=O)C1)C c1(C(=O)NC2C(CNC(C(CCC)(C)C)=O)CCCC2)cc2ccnc(Cl)c2[nH]1 C1(NC(CCN(C)CC)=O)CCCN(C(c2cnc(N(C)C)c(Cl)c2)=O)C1C c1(C(=O)N)cc(S(=O)(=O)NC)c[nH]1.N1(C(CC2C(C)(C)C2)=O)CCC(C)C1 c1(C(=O)NCC2N(C(c3ncn(CC)n3)=O)CCC2)cc([N+](=O)[O-])cn1C Cc1ncncc1C(=O)NC1CCC(NC(C2CC2C2CC2)=O)C1 C(=O)(CCO)NC(C)CN(C)C(c1cc(CCn2cccn2)on1)=O.C(N)=O Cc1[nH]c(=N)nc(O)c1CCC(=O)NC1CCCC1.C(=O)(C(F)CC1CCC1)N C1(C(=O)NCC2CC(NC(c3cc(C)c(N)cn3)=O)C2)CCc2nc[nH]c2C1 c1(CN2CCC(N(C(=O)OC(C)(C)C)CCO)C2)ccc([N+](=O)[O-])cc1F CC1CCN(C(=O)CSCC=O)C1.c1(CCC=O)cccc(O)n1.C(C)(C)C C(C1=CCCN(C(C2CC(CCO)C2)=O)C1)NC(c1ccc(CO)s1)=O C1(C(=O)NCCC(O)CNC(=O)C(F)(F)CO)(OC)CCCC(C)(C)CC1 c1(CC(=O)N(C2CCCC2)CC)ccnc(Cl)c1F.C(CCC(=O)N)NC(N)=O C=CC(C)(C)CC(=O)N1CCCC1CC(=O)NC1CCN(CC2CC2)CC1 c1(C=O)nc2cnccc2s1.C1(NC(C(C2CCC2)OC)=O)CCC(F)(C)C1.N c1(C(=O)NC(CCCC)CNC(c2ccc(C#N)o2)=O)cnc2[nH]cncc1-2 c1(C(N2C(C)(C(=O)NCCCCC(F)(F)F)CC(O)C2)=O)cccc2occc12 N1(C(CNC(c2cccc(C)c2F)=O)=O)CC(C2=NOC(C)C2)C1 N1(C(C(C)NC(C)=O)=O)CC(CC)C(C)C1.C(c1ccccc1)=CC(C=O)C C1(NC(C=Cc2n(C)ccc2)=O)CC2CC(NC(=O)CCO)C1C2.C1CCOC1 Cc1ccc(N)c(C(=O)NCC2CC2NC(=O)Cn2nnc(=O)[nH]2)c1F C1(CC)CNC(=O)CN1C(C1C2CCC(C2)N1C(=O)C(O)c1ccco1)=O CS(=O)(=O)c1csc(C(=O)NC23CC2CN(C(c2ccn4nccc4n2)=O)C3)c1 C1(C)(CNC(CC(C)OC)=O)CCC(NC(C2(N(C)C)CCCC2)=O)CC1 c1(C(=O)NCC(C(C)(C)C)NC(c2ncc(Cl)s2)=O)ccc2c(n1)OCCO2 c1(OC)cc(C(=O)NCCC(C)NC(=O)C=Cc2nc(C)co2)cc(Cl)n1 CC(C)=C=CC(=O)NC1(C(=O)NOCC(C)(C)C)CCN(C)C1 c1(C(N(C2CN(C(c3cnc(C(N)=O)cn3)=O)C2)C)=O)cc2nc(Cl)ccc2o1 CC(CC1CCCCC1)C(=O)N(CCCCNC(=O)C(N1CCC(C)C1)=O)C S(=O)(=O)(c1cccc(C(N2C3CCC2C(N)C3)=O)c1)NC(CC(C)C)CC(=O)O Cc1cc(CCCC(=O)NCC2(NC(C3CCCN3C)=O)CC2)on1 c1(C(N2CC(C)C(n3cc(CCC(C)(C)O)nn3)C2)=O)cc2ncc(Br)cn2n1 N1(C(=O)OC(C)(C)C)CCN(C2CCCC2C)CC1.c1(C=O)sc(F)cc1Cl.N c1(C(C(=O)N)NC(C(C(C)C)SCC)=O)c(C)cccc1Br.C1(CCF)CC1 c1(CC=O)cc(F)cc(F)c1.c1(CC)cc(C(=O)N(CC(O)C)C)c(C)o1.N N1(C(C(N2CCC(c3ccno3)CC2)=O)=O)CCc2cccnc2C1 C1(C(=O)NC2CN(CCC)C2)CCC2(CC2)N1C(=O)CCCC#N C1(CC(=O)NCC=CCNC(CCC#CC)=O)CCc2ncc(Br)n2C1 N=c1[nH]c(O)ncc1N1CCN(C(c2cc(C(F)(F)F)cc(F)c2)=O)CC1 N1(C(C2C(CO)C2(F)F)=O)CCOC(C2CC2)CC1 C(=O)(C1=CCCCO1)N(CC(=O)NCCCCCNC(C)=O)C(C)C c1(C(C)C)c(C(N2CCOC3(C2)CN(C(=O)C=CCO)C3)=O)cnc2ncnn12 c1(CC(N2CCC(NC(C(CC)CO)=O)(CF)C2)=O)csc2nc(C)cn12 N1(C(c2cc(CC)[nH]n2)=O)CC2CCC1C1CN(Cc3csc(C)n3)CC21 C1(NC(C2C(C)(C)CCO2)=O)C2CC1CN(C(=O)C(=O)NCC1CC1)C2 c1(C(c2n(C)nnn2)NCc2ccc(C(C)(C)C)cc2)ccc2ncc(I)n2c1 C#Cc1ccc(F)cc1CNC(=O)C(=O)NC1CNOC1 C1(NC(c2oc(C)c(CO)c2)=O)CCC2(CCN(C(=O)CCC(N)=O)CC2)C1 N1(C(C2C=C(C)CS2)=O)CCC(C2CC2)C1CNC(C1CC(O)CN1C)=O CCCCCC(O)C(=O)NCC1(C(N2CCCC(C#N)C2)=O)CC12CCC2 CCCC(C)(O)CC(=O)N(C1(C(=O)NOCC(O)CO)CCC1)C1CC1 c1(C(N2CC3(CN(C(=O)C(F)C(F)(F)F)C3)C2)=O)ccc2c(c1)C=CS2(=O)=O C(=O)(C(C)(C)CCF)NCC(C(CC)C)O Cc1cc(C)c(C(=O)N)s1.N1(C(C2CC=CC2)=O)CCOC(CC(=O)N(C)C)C1 C1(NC(c2n(C=C)nnc2)=O)CCN(C(=O)CCNS(=O)(=O)CC)CC1F C1(NC(C(COC(C)C)NC(CCN(CCC)C)=O)=O)C2CCCOC12 C1(N(C(C2CCCN2N=O)=O)CC)CCCN(C(=O)CCc2scnc2C)CC1 C1(C(=O)NCCOCCN(C)C(c2c[nH]c(=N)s2)=O)CCC2(CC2)C1 c1(CCNC(c2cccc(OCCC)c2)c2nnnn2C)nnc2n1CCOC2 N1(C(=O)Nc2c(OCCOC)nccc2)CCCC(C#N)C1 C1CCCCN1C(=O)CCc1nc(C)no1.C(C)(C(=O)NC)NC(=O)NC.C c1(CCCNC(c2n(CC(=C)C)nnn2)c2ncc[nH]2)cc(OC)cc(OC)c1 C1(OC)(CNC(c2cscc2)=O)CCN(C(c2csc(C(F)F)n2)=O)C1.S C1(CNC(C2(C)CC(=C)C2)=O)C2CN(c3ncc(Cl)cn3)CC12 N1(CCC)CCCC1C(=O)N(C)CC1CCN(C(c2cnnn2C)=O)C1 C1(C(N2CC(Cc3ccoc3)C2)=O)CCN(C(C23CC(F)(C2)C3)=O)CCO1 N1(C(c2c(CC)cc[nH]2)=O)CCCCCC1C(=O)NCC#CC(F)(F)F C1(NC(C2(c3ccccn3)CCC2)=O)CCCC1CO C1(NC(C2N(C(C(CCC)C)=O)CCCC2)=O)COC2(CCC2)C1 c1(C(=O)NC2(CO)CCN(C(C3CC(C)(C)C3)=O)CC2)c[nH]c2nccc-2c1 N1(C(c2ccc(F)c(C)c2Cl)=O)CCCC2(C1)CN(C(C1CC3C=CC1C3)=O)C2 c1(C(=O)NCC(C)C)cc(S(N)(=O)=O)cs1.C12(CC=O)COC(C1)C2 C#CC1CCCN1C(c1c[nH]nc1C1CCCCN1C(=O)CN=[N+]=[N-])=O C1(NC(CCC=C)=O)CCN(C(=O)CN(C)CC)CC(C)(C)C1 C1(C(N(C(C)C)CCF)=O)CC12CC(NC(=O)COC1CCCOC1)C2 N1(C(c2cc(C)n(-c3cc4nc(=O)ccn4[nH]3)c2C)=O)CCN2C(=O)NCC2C1 c1(C(=O)NCCN(C)C(c2c(Cl)csc2Cl)=O)cccc2ncccc12 N1(CC(=O)N(CC(O)CNC(C23CCC2CC3)=O)C)CCCCCC1 c1(NCC(CC=C)(C)CO)ccc(S(=O)(=O)N2CCCC(COC)C2)cc1Br C1(CC(=O)NC(C(C)C)(C)CNC(c2cc[nH]c2)=O)CCC2(CCC2)O1 N1(C(c2c(CCC)n(C)nn2)=O)CCCC(NC(c2nc(C)oc2C)=O)C1C C(=O)(C(F)CC(C)(C)C)N1CC(C(C)NC(=O)CCN2CCCC2)OCC1 c1(C(N(C(CNC(C23CC(CC(C)O2)C3)=O)C)C)=O)ccn2ncnc2c1 C(=O)C(CCO)N(C)C.c1(NC(C(=O)NCCOC)=O)cnn(CC)c1.N c1(C(N2C(C)CC(NC(CCN(CCC)C)=O)C2)=O)cc(N)c(C)cc1Cl c1(C(N2CCN(C(C=C(CCC)C)=O)C3C2C3)=O)ccc2c(c1)COCC2 C1(C(N(C)CCOCC)=O)CCC(C)CC1.C(=O)C(Cc1ccsc1)NC=O C1(CNC(C=CC=CC)=O)CCN(C(c2ccnn(C)c2=O)=O)C12CCC2 C(=O)(C(CO)NC(c1nccn1C)=O)NC(C)CCc1cn[nH]c1 c1(C(C)C)ncc(C(N2CC(NC(=O)CC3COC(=O)C3)C(C)C2)=O)cn1 C1(c2ccc(OC)cc2)CCN(C(=O)OC(C)(C)C)CC1NS(C)(=O)=O c1(C(=O)OC)ccoc1.[nH]1cc(C2CCCN2C(C2(N(C)C)CCC2)=O)nn1.C c1(C(N2CCC(C)(C#N)CC2)=O)cn2c(n1)CN(C(C1CCC=CO1)=O)CC2 C1(CC(=O)NCC2(C(=O)NCCC3CC(C)C3)CC2)CCOC1(C)C Cc1ccc(C2(CC(=O)N=c3cc[nH][nH]3)CC2)c(F)c1F.C12(CCC1)CC(=O)N2 C1(CC(=O)NC(c2cccc(Cl)c2)(C)C)COC2(CCC2)CN1 N1(C(=O)CC2CSCCO2)CCCC2CN(C(C34CCC(C3)C4)=O)CCC12 C1(NC(CC2(C=C)CC2)=O)CN(C(=O)C(CCC)=CCC)C(C)(COC)C1 c1(Cn2cc(CC(CC)(C)O)nn2)ccc(C(=O)NCC2(C)CCCS2)cc1 C1(C(N(C(COC)C)C)=O)(CO)CCCN(C(c2cc(C)nn2C)=O)C1 C#CC(C)(C)C(=O)N1CCC(C(F)C(=O)NCCCC(C)(F)F)C1 c1(SC)cc(C(N2C3CCC2C(CNC(=O)C(CO)C(C)C)C3)=O)ccc1F CC1C(NC(C2CC2(Cl)Cl)=O)CCCN1C(c1ncc(C(F)(F)F)n1C)=O c1(C(=O)Nc2ncc(-c3ccc(Cn4cccn4)cc3)cn2)c(O)cccc1F c1(NC(c2ccc(C)c(C)n2)=O)ccc2c(Br)nn(C)c2c1 C1(C(N2CCC(C(C)(C)O)C2)=O)CCC2CCC1N2C(C1CC2(CCO1)CC2)=O C1(O)(CNC(C(C)c2cccs2)=O)CCN(C(c2cnoc2C2CC2)=O)C1 CCC(CC)CCCNC(C1(Cc2cc(C)nc(C)c2)CCCCC1)=O c1(COC(Cn2c(CCCC)ncc2)=O)cc(=O)oc2cc(O)c(O)cc12 C(CCC(=O)NCC(C)OC(F)F)NC(CC=CC)=O c1(N2CC(C)C(NC(c3cccc(F)c3I)=O)C2)ncc2[nH]ccc2n1 C12(CC)CCC1CN(C(=O)C=Cc1ccoc1)C2.c1(OC)c(C(=O)N)csc1C c1(NC(C)CNC(c2cnco2)=O)cc(=O)n(C)c(=O)n1C C1CCN(C(C2(C)CCN(C)C2)=O)CC1.C1(CC(=O)NC)(COC)CCCC1 N1(C(CCC=CC)=O)CCN(C)CC1C(=O)NCC1CC1Cl C1(C(N(C(C(=O)NCCCOCC=C)C)CCC)=O)CCN(C)CC1 C(CCCC(C)NC(c1cc(O)ncn1)=O)NC(CN(CCOC)C)=O N1(C(c2c(OC)ccs2)=O)CC2CC(C1)N(C(=O)CNc1ncccn1)C2 c1(C(=O)N)ccnc(C(F)(F)F)c1N.C(=O)(C(C)Cc1ccco1)NCCCC c1(C(N2CCCC(NC(=O)NCCOC)C2)=O)nc2ccccc2[nH]c1=O c1(C(N2CCCOC(C(C)C)C2)C(=O)NCCSC)cc(F)c(F)c(F)c1F C1(C(C)C)CCC(C(=O)NC2CCC(CNC(c3ccn(C)c3)=O)CC2)CC1 N1(C(C2N(C)C(=O)NC2)=O)CCC(CNC(C2CC=CC2)=O)C(F)(F)CC1 N1(C(CCCOCCC)=O)CCCOC(CCNC(=O)CCCNC(=O)OC)C1 Cc1cc(NC(C2CCC2c2nncn2C)=O)ccc1NC(=O)Cn1cnnc1 C1(C=O)CCCCC1c1nc(S)n[nH]1.C(CO)(CC)NC(CNC(=O)OC)=O C1(C)(CNC(c2nnn(C)n2)=O)CCCN1C(=O)CCC1CCCC(=O)N1 c1(CC)ccnc(C(=O)NCCCNC(=O)CN(C2CCCC2O)C)c1 C1COCCC1C(=O)N(C)CCn1cncn1.C1(C=O)COC1.C1CC1.CO.C C1(CN(C(=O)CC2CCC(NC=O)C2)C)CCC(F)(F)CO1.C(C)(C)C CS(=O)C=CC(=O)N(CCNC(c1ccc(NC=O)cc1)=O)C1CC1 N1(C(CC2(C=C)CN(C(c3c[nH]nc3CCC)=O)C2)=O)CCC12CCC(O)CC2 C1(CC(=O)NCCC2CCCCO2)CCCN(C(c2scnc2C2CC2)=O)CC1 c1(C(=O)Nc2ccc(OCCF)cn2)nnc2c(F)cccn12 c1(C(N2CC3C(CNC(CC=C=C)=O)C3C2)=O)ccc2c(C)cc(Cl)nc2c1 c1(OC)cc(C)c(C(=O)N)c(C)c1.C1CN(C(=O)CC2CCC2)CC(C)(C)C1 N1(C(C(CSC)OC)=O)CCCCC(n2cc(-c3cccnc3F)nn2)C1 c1(COC(CCN(CCCCOC)C)=O)ccc(C)c2[nH]c(C(=O)OC)cc12 c1(C(N(C2CCN(C(=O)C(CO)CC)C2)CCC)=O)sc(N(C)C)nc1Cl.C c1(COC)cc(C(N2CCN(C(C3(n4cncn4)CC3)=O)CC2)=O)n(C)c1 C(CN=c1[nH]ccc(=NCC(C)(C)c2ccccn2)[nH]1)NS(NC)(=O)=O C(=O)(C(C)CC(C)C)N1CC(CC(=O)NCCCCN(CC)CC)(OC)C1 Cc1cc(C)c(C(=O)NCC2CCCN(Cc3nc(=O)n(C)[nH]3)C2)cc1C C1(F)(C=O)CCOC1.C(=O)(C=O)NCCOCCOC.CCCCC.N N1(C(=O)CCc2ccnc(Br)c2)CC2C(C(F)(F)F)CC2(C(=O)O)C1 c1(N2C(c3cccc(F)c3)CC(C)C2)c([N+](=O)[O-])cnc2ccccc12 c1(OC)cccc(-n2cc(CNC3CCC4CC4C3)nn2)c1 c1(SCCOC)ccc([N+](=O)[O-])cc1NC(C1CCC(CCC(C)C)CC1)=O C1(NC(C(CSC)O)=O)CCC(C(N2CC(CO)(OC)C2)=O)CC1 C1(C(C)CNC(C2(C)CCCS2)=O)CCN(C(=O)Cc2c(Cl)cnn2C)CC1 C=C=CC(C)C(=O)NCC12COC(CNC(c3cnnn3C)=O)(C1)C2 C1(C)(C(N2CCC(NC(C(C)C)=O)C2)=O)CC(c2cc(Cl)cc(Cl)c2)=NO1 C(=O)(C(O)CCCNC(C1CC(C)(F)C1)=O)N1CCC(OCC#C)CC1 Nc1ncc(C(N2CC(NC(C34CC(C3)S(=O)(=O)C4)=O)C(O)C2)=O)cc1Cl c1(C(=O)NC(C(N2CCC(C)(CCC)C2)=O)(C)C)nc(C)ccc1C C1(C(=O)OC)CC(=O)N(C2CN(C(C3CC34CC4)=O)C2)C1 C(=O)(CCC(C)(C)NC(=O)C(C)n1cncn1)NCCc1nnc(C)s1 Cc1c(C(=O)NCCC2(O)CN(C(C3CCOC3)=O)C2)ccn1C(C)C Cc1cc(NC(c2cscc2C(F)F)=O)cc2c[nH]nc12 N1(C(C2CCN(C(C)C)CC2)=O)CC(C2CCCN(C(C3(C)CC3(F)Cl)=O)C2)C1 C1(C(=O)NC(C(=O)NCCC)Cc2cn[nH]c2)CC=CC(O)C1 C(CS(=O)(=O)c1ccc(NC(=O)CCc2c(F)cccc2Br)cc1)OC C(=O)(CCCCC(=O)N1CCC(C)C1CNC(c1cc(=O)cc[nH]1)=O)NC C(=O)(C1CCc2nnc(C)n21)N(CC(C)N(C(c1c(C)cc(SC)o1)=O)C)C CC(CC(=O)NCC1CC(NC(=O)CN2CCC(C)(C)C2)C1)C(F)F C1(O)(CNC(C=NOC)=O)CCCN(C(C2(C)CCN(C(C)=O)CC2)=O)C1 CC1CCC=C1C(=O)NCC1CC(C(=O)N(C)Cc2cccs2)CO1 C1(C(=O)NCC(CC)CC)CCN(C(c2coc(COC)n2)=O)CCO1 N1(C(C(COCC)NC(=O)C(O)Cn2cncn2)=O)CCCC(CCF)C1 C1(N=[N+]=[N-])(C(=O)NC(C(C)(C)OC)C)CCOCC1 n1(CC=O)cc2ncccc2n1.C1(CC=O)C=CS(=O)(=O)C1.C1(CC)CC1.N c1(C(CC)C)ccc(C(=O)NCC2CCN(C(c3nscc3N)=O)C2)cc1 c1(C(=O)NC(CCOC)CNC(=O)CC(=O)Nc2nccs2)ccc(O)cc1 C1(C(=O)NCC(=C)C)(SC)CN(C(=O)CC2CCC3CC23)C1 CC(C)(C(=O)NC1CC(NC(=O)CCC2OCCO2)C1)C1CCCCO1 c1(CNC(COCCNC(C(C=C)OC)=O)=O)c(C)nnn1CC C(C)(CNC(c1sccc1Br)=O)(CO)NC(C1C(COC)C1)=O c1(COC)ccc(C(CC(=O)O)NC(=O)C(C)C2CC2)cc1 CC1CC(CO)CN(C(=O)C(C)(C)CNC(=O)CC2CCOC2C)C1 C(c1cccc(Cl)c1)=C(C=O)C.C1(C(=O)NCC2CCC2)(OC)CCOCC1 O(NC(=O)CCCNC(=O)NC)CC(=O)NC(C#C)CC(C)C c1(CC)cc(C(N2CCCC2C2(C(=O)N(C3CC(SC)C3)C)CC2)=O)on1 N1(C(CC=CC=C)=O)CCC(N(C(=O)CC=C(C)C)CCCC)CC1 CC1(C(=O)NC2CC(NC(=O)CC3CCCCCC3)CC2O)CCC(F)(F)C1 C(=O)(CC(C)(C)C)N1CCC(N(C(COCC#C)=O)CCC)C1 c1(C(N2CC(CC(=O)OCC)C2)=O)ccc2nc(C(F)(F)F)[nH]c2c1 C1(C(N2C(CNC(CN(CC)CC)=O)COCC2)=O)CCC12CCOCC2 N1(C(COC(C)C)=O)CCC(NC(=O)C(C)NC(N)=O)CC1C C(=O)(CC(CN(C)C)CC)N(CCC)CCNC(c1cc(Cl)no1)=O C12(C(N3CCCCC3)=O)C3CC(CC13)C2(F)F.c1(C(=O)N)ccc(F)c(F)c1 C(=O)(CC(C)(C)C(F)F)NCCN(CCC)C(C1(C)CC1)=O.C1CCC1 c1(CN2CC(=O)N(CC3CCN(C(C)C)C3)C2=O)cccc2ccoc12 CC(C)C(CNC(=O)C(O)CC1CCCC1)NC(=O)CC(C)F N1(C(C(C)OC(C)=O)=O)CCCC1(C)CNC(=O)CC(C)n1cccn1 c1(C(N(CCN(C(C)C)C(C2CCSCC2)=O)C)=O)cnc2ccccc2c1 N1(C(C(C)c2ccsn2)=O)CC2(CCCN(C(c3ccc(CO)c(F)c3)=O)C2)C1 C(=O)(C(CO)C(F)(F)F)N1C(CC(=O)NCCC(C(=O)OC)C)CCCC1 C1(NC(c2ccc(F)cc2)=O)Cc2ccccc2C1NC(C1(F)CC=CC1)=O C=CCCCCC(=O)N1CCC(CNC(=O)CSCc2ccc(Cl)cc2)C(C)C1 n1(CCCNC(c2ccc(C3CCCCC3)o2)=O)cc(CC2CC(F)(F)C2)nn1 CCCCC(CNC(c1nnn(-c2ccccc2)n1)=O)NC(=O)C(C)C(C)O c1(NC(C2(C(F)F)CCNCC2)=O)cnc(C(F)F)nc1O C1(CS(=O)(=O)N(C(C)(C)C)CC2(C)CC2(F)F)CCS(=O)(=O)C1 c1(NC2(C(N(C)C)=O)CC2)nc(NC(=O)C(C)(C)C)ncc1Cl C1(NC(c2cc(OC(CC)C)ncc2)=O)CCN(c2nnc(C#N)s2)CC1F Cc1cc(O)cc(C)c1C(=O)NCCCNC(=O)CC1CCC(O)C1 c1(C(=O)NCCc2cccc(O)c2)cn2cc(-c3c(O)cccc3O)ccc2n1 C1(NC(C2C(C)CCO2)=O)CC(C(=O)NOCC(O)C(C)(C)C)C1(C)C CC#CCC(C(=O)NC1CCOC(C)(CC)C1)NC(c1c[nH]nc1Cl)=O c1(OC)cc(C=O)cc([N+](=O)[O-])c1.C1CN(C(C2(C)CCC(=O)C2)=O)CC1C.N C1(C(N(C)CC2CC3(CCC3)C2)=O)CCC2(CC2)N1C(=O)C1CC1 N1(C(C)=O)CCc2cc(-c3cc(C(=O)NCc4cccc(C)n4)ccn3)ccc21 c1ccc(S(=O)(=O)N(C)C)cc1.C=CC1CC(c2nnnn2CCC2CC2)(N)C1 C1(NC(=O)C=Cc2cccnc2)C2CC3CN(C(=O)CC4OCCO4)C1C3C2 C1(NC(C(c2ccccc2)C)=O)CC(NC(C2(C(F)F)CCC2)=O)CC1O CC1CCCCC1NCC(=O)N.N1(CC(N2C(CCC)CCC2)=O)CCNC(=O)C1 CC1(F)COCCN(N2CCCC(C3(C)OCCO3)C2)C1 c1(CC(=O)NCC2CC2)cc(F)ccc1F.c1(C=O)csc(-c2cn[nH]c2)n1.N c1(C(N(CCN(C(CSCC)=O)C(C)C)C)=O)nc(-c2ccccc2)oc1C C1(NC(=O)C2CC2)(CO)CCCN(C(=O)C(c2ccc(Br)cc2)O)C1 c1(C(N(C2CCC(NC(c3c(C)nccc3Cl)=O)C2)C)=O)cccn2nccc12 CC1(C)CC(C)(CNC(c2csc(Cl)c2)=O)CN1C(=O)CCc1ccccn1 CC1CC2CN(C(=O)C(c3ccco3)NC(c3cnnc(O)c3)=O)CCN2C1 C1(C(N(CCCNC(C2CC(F)(CF)C2)=O)C)=O)CC2CCCC(C1)C2 N(C1CCCc2cc(CN)ccc21)Cc1c(C)cc(O)cc1C N1(C(C(C)NC(=O)C2CC2)=O)CC2CCN(C(=O)C(C)N(C)C)CC12 C1(CCOC)CCN(C(c2cc(C#N)c[nH]2)=O)CC1.c1(C(=O)N)cccc(=O)o1 C1(CCNC(CCOCC)=O)CCN(C(=O)CCC)CC1.c1(C=O)ccsc1.N C1(CC(=O)NCCc2cccc(Cl)c2)(CCN)COCCO1 N1(C(C)C)CCCC1C(N1CC(C)(OCC=O)C1)=O.CC(O)CC1CCCC1.N Cc1cc(F)ccc1C(=O)NC1CCN(C(=O)CCCF)CC1c1ccccc1 N1(C(C=CCC)=O)CCC2(C1)CN(C(=O)C(c1ccc(Br)cc1)CC)CCO2 C1(C(N(CCN(C)C(c2ncn3c2CCCC3)=O)C)=O)CC2CCC(C1)C2(F)F CCC(C)C(C)C(=O)NCCC(=O)NCCc1cnco1 N1(C(=O)C=CC=C(Cl)Cl)CCC2(CC1)CC2NC(=O)C(O)Cc1cnc[nH]1 N1(C(C2CC2C2CC2)=O)CC2OCC(C(N3CCn4ncnc4C3)=O)C2C1 C1(OCC)CCC(C(=O)NCCCC2CCCN2C(c2cc(Cl)ns2)=O)CC1 CCCCN=C(NCC(CC1CCCC1)OC)NC1CCN(CCOC)C1 C1(C(=O)NC2CCC(NC(CC(=C)I)=O)C2)COCCOC1 C1(NC(C2(CCC=C)CCCC2)=O)CN(C(=O)CC(C)SC)CCC1(C)C C=C(C)CCCC(=O)N1CCC(N(CCCC)C(C2Cc3nncn3C2)=O)CC1 C12(C(=O)NCCCN(C(=O)C(C)CCOC)CC)CCCC1C2(F)F C1(NC(C(C2CCCC2)OC)=O)COCC1n1cc(CC2(O)COC2)nn1 c1(SCC(=O)NCC2CC2C(=O)NCC(O)Cn2cccn2)nc[nH]n1 c1(C(N2CC3C(C(N4CCC(OC5CC5)CC4)=O)(C3)C2)=O)cnn2cccc2c1 C1(C)(C(=O)Nc2cn(CC)nc2)CCN(C(c2nn(C)cc2C)=O)C1 C(=O)(CCCNC(c1cnn(C2CC2)c1)=O)N(C(C(C)SC)C)C c1(C(=O)NC(CNC(C2(C=C)CCC2)=O)(C)C)cc2c(s1)CCC(C)C2 c1(OC)ccc(Cl)cc1C(=O)NCC1(F)CN(C(C2(C)CCCO2)=O)C1 C1(NC(C2(CSC)CC2)=O)CC2CN(C(=O)CSc3nnnn3C)CC2C1 c1(C(=O)NCC2CC(NC(COC)=O)C2)cc(Br)n2c1CCC2 N1(C(c2n(CC)c(O)nc2)=O)CC23CCCC2(C1)CN(C(c1c[nH]nc1Cl)=O)C3 c1(C(=O)NCCc2cnc(C)o2)n[nH]c2c1CN(C(c1ccc(C#N)s1)=O)C2 c1(NC(C(=O)NCCCC2C(C)C2)=O)cccc(Cn2cc(Cl)cn2)c1 Cc1cnc2n1C(C(=O)N1CCCC1CCNC(C1(F)CCC1)=O)CCC2 C1(C(N(CCCN(C)C)CCNC(c2nc(C)sc2)=O)=O)CC12CCCCC2 N1(C(C(C2CC2)SC)=O)CC2C(NC(c3ccc(-c4ccco4)o3)=O)C2C1 N1(CC(=O)NC2CCC(CN(C(=O)C=C(Cl)Cl)C)CC2)CCn2ccnc2C1 c1(NC2C(NC(=O)C3=CCCCCC3)CS(=O)(=O)C2)nc2ccc(Br)cc2o1 C1(CC)(NC(=O)C2=COCCO2)CCN(C(=O)CCc2c(C)ncnc2O)CC1 N1(C(C(C)Oc2ccccc2Cl)=O)CCCC(O)(CCNC(c2cocn2)=O)C1 C1(NC(C2=CC(C)(C)C2)=O)CCC12CCOCC2.N1(C2(CC=O)CC2)CCCC1 C1(NC(CCC)=O)CC(C)CN(C(c2ccccc2Sc2ncccn2)=O)C1 C(C)(C)(C(C)CC(=O)N1CCC(C)(CC)CC1)NC(C(CCCC)O)=O C1(NC(CCc2cnc(C)o2)=O)CCCC(NC(=O)CC2CC2(C)C)C1 c1(C(N)=O)ccc(Cl)cc1C(N1CCCCC1CC1CCCN1)=O.C1(=O)CN1 C1(NC(c2c(OC)cccc2Cl)=O)CCN(c2ncc(C)c(OC)n2)CC1(C)C C1(C(=O)NCC(Cc2ccccc2)NC(c2coc(O)n2)=O)CC2CCC2C1 Cc1cccc(-c2cn(C3CCCCC3N(C(=O)C(C)C(=O)O)CC(C)C)nn2)n1 C1(C(=O)NCC(C)NC(C23CC(CC(F)F)(C2)C3)=O)OCCOC1C Cc1oc(-c2ccccc2)nc1CN(C)CC1CCCN(C)C1.N1COCC1(C)C CCC(C)C(C(=O)NCCn1cc(CCN)nn1)NC(N)=O.[SH](C)(=O)=O N1(C(C)=O)CC2CC2(C(=O)N)C1.C1CCCN(C(=O)Cc2cccc(C)c2)C1.C C(=O)(C1=CCC(NC(C2CCN(C)C2)=O)C1)NC(C(=O)OCC)C C#CCCCCCCC(=O)N(CC(CC)NC(c1cnn(CCC)c1)=O)CC c1(C(N(CCOC)CCNC(=O)C(C)N(C)C)=O)cc(Br)c[nH]1 N1(C(CC)=O)CCC(C(F)F)(CNC(c2ccnnc2C)=O)C1 C(C(=O)NN1CCCC1C(N1CCCC1CCCO)=O)n1ccc(C)n1 C1(C(C)C(=O)NCC2(CCO)CCC2)CCCN(C(c2cnc(N)cn2)=O)C1 C1(C(N(C)CC2(C)CC2)=O)CCCN(C(C2CC2C2CC2)=O)C1 c1(C(N2CC(NC(C(c3nccc(C)c3)(C)C)=O)C2)=O)ncnc2c1ccn2C N1(CC(=O)N(CCN(C(c2cc(C)oc2)=O)C)C(C)C)CCC(C)(O)C1 C(CC(C)(C)C(=O)N1CC2CC(NC(c3cc(C4CC4)ccn3)=O)C1C2)OC N1(C(C2N(C(COC3(C)CCC3)=O)C3C(O)CC2C3)=O)CCN2CCCCC2C1 N1(C(c2nn(C)c(O)c2)=O)CC2CCN(C(c3cc(F)c[nH]3)=O)CC(C2)C1 C(=O)(CC1=CCOCC1)NC(CCC)CNC(C1CC(C2CC2)=NO1)=O C1(C(=O)NCCNC(c2c(C)cc(C)nc2)=O)CC12C(=O)Nc1ccccc12 C1(NC(C(COC)(C)C)=O)CCN(C(c2c(N)cc(C)cc2F)=O)CCC1CO Cc1c(C(=O)NC(C)CCCNC(=O)C(c2cncnc2)C)cccc1N n1(CCSC)nnnc1C(c1cc(C)no1)NCCCCCc1ccccc1 N1(C(c2cc(C)sn2)=O)CCCCC1CCNC(c1[nH]ccc1C1CC1)=O c1(C(=O)NCC2C(NC(c3ncccn3)=O)C2)cc(Cl)cnn1 Cc1c(C(=O)NCCCN(C(=O)C(O)Cc2cnc[nH]2)C)cnn1C(C)C C1(CNC(c2c(C)ccnc2C)=O)(C)CC2CCCC2C1.c1(C=O)ccsc1.N c1(C(=O)NC2C(NC(C3(C#C)CCC3)=O)CCOC2)ccnc2ncnn12 CS(=O)(=O)C1CCN(C2CC3CCC(C2)N3C(c2ccc3nncn3c2)=O)CC1 c1(C(=O)NCCC(C(=O)O)OC(C)(C)C)cc2cccn2cn1 CCC(CC(=O)NC1CC2(C1)CC2NC(c1cnn(C)n1)=O)CC(C)C CCC(CC)C(F)C(=O)N1CC(NC(C2(C)CCC3CC3C2)=O)CC(F)(F)C1 N1(C(=O)CCOc2ccccc2)CCN(Cc2ccc(O)cn2)C2CC12 Cc1cc(C(=O)NCC2CN(C(c3ccc(CSC(F)F)o3)=O)C2)ncc1F C1(C(=O)NCCC=C=C)C(C)CCN1C(=O)Cc1cc(C)nn1C C1(NC(CCc2cccc(OC)n2)=O)CC(NC(=O)CSC)C12CCC2 n1(CCC)nc(-c2ccoc2C)nc1CCCC(=O)N(C)C C1(CNCc2n(C)ncc2)CCC(C(=O)Nc2nc(-c3ccncc3)cs2)CC1 CC1(C)CC1(C#N)C(N1CCC(F)(CNC(=O)C=CS)C1)=O.c1ccco1.C C1(F)(CNC(C2C(=C)CC2)=O)CCN(C(c2cnn(C(CC)CC)c2C)=O)CC1 c1(CC(=O)NC2(CF)CCN(C(c3nccnc3Cl)=O)C2)ccccc1F N1(C(CN(C(C(C)C)=O)C)=O)CC(N(C)C(c2occ3c2CCC3)=O)C2(CC2)C1 CN1CC(CC(=O)NC2CCCN(C(=O)C=Cc3ncco3)C2)c2ccccc21 c1(C=O)ccccc1S(C)=O.c1(CNC(COCCC(C)C)=O)csc(C)n1 C1(OC)CC2(C(=O)N(C3CCN(Cc4cn(-c5cccnc5)nn4)C3)C)CC12 C1(NC(CN(C2CC(c3c[nH]nn3)C2)C)=O)CC2CCC1C2.C1CC(F)(F)C1.C C(=O)(C(C)CC(C)(C)C)N.c1(C(C)OCC)nc(C(=O)N(CCCC)C)cs1 C1(C)(C(=O)NCC2CCC(NC(CC(CC)C)=O)CC2)CCCC1(F)F C1(C(=O)OC)CCC(C(=O)N(C)CC)CC1.c1(CCC=O)nc(C2CC2)no1 Cc1cc(NC2CCCC(NC(c3ncn(C(C)(C)C)n3)=O)C2)ncc1[N+](=O)[O-] N1(C(CC(C)c2cnn(C)c2)=O)CC(CNC(=O)CO)CC1C.CCN(C)C Cn1ncc2ccc(C(=O)NC3CCC(CC(=O)Nc4cnns4)CC3)cc12 C(=O)(CC(F)(F)C(F)F)N(C1CN(C(c2c(C)nc(C(C)C)s2)=O)CC1F)C CCCC(CCC)CC(=O)N(C1CN(C(=O)C(=Cc2cccnc2)F)C1)C Cc1nnc2c(C(=O)NC3(CNC(=O)CC(C)C(C)(C)C)CCOC3)cccn12 N1(C(=O)OCC(C)(C)C)CCc2ncnc(N3CCCC(C4CCO4)C3)c2C1 Cc1cc(CN2CCN(C(=O)Cn3nc(C)c(C)c3C)CC2)cc(F)c1 Cc1nc(C(N2CC(NC(=O)C(C)N3CCC3)CC(F)C2)=O)ccc1C#N C#Cc1ccccc1CC(=O)NCc1cc[nH]c1C(N1CCC(O)C(F)C1)=O N1(C(Cc2cn(CC)nc2)=O)CCN(C(=O)CC2CCC3(CCC3)O2)C2CCCC12 C1(NC(CCCC#C)=O)CN(C(=O)Cc2ccc(Cl)c(C)c2)CC12CCC2 Cc1coc(C)c1C(N1CC(NC(=O)C(C)Cc2ccco2)CC1C)=O Cc1c(F)cc(-c2noc(-c3cc4sccc4n3C)n2)cc1F C(=O)(C1CCCc2c[nH]nc21)NCC(C1N(C(CCCOC)=O)CCC1)(C)C C1(C(N(C2C(C)CCC2)CCc2ccccn2)=O)CCCN(CP(C)(C)=O)C1 Cc1nccc(C(N2CCCC2CNC(=O)CCc2ccccc2C)=O)n1 c1(CCC(N2CCCC(C(=O)Nc3ccc(F)cc3F)C2)=O)cn2ccsc2n1 c1(C(N(C2CN(C(c3ccc(C(N)=O)cc3)=O)C2)C)=O)cc(N)cc(O)n1 N1(C(C2N(CC)CCCC2)=O)CCN(C(=O)Cc2cn3ccsc3n2)CC12CC2 Cn1nc(C(C)(C)C)cc1CN1CCC(CC(=O)N(C)C)CC1 C1(NC(C=C(CCC)C)=O)CN(C(=O)C(n2ccc(C)n2)C)CCC1F c1(C(N2CC(NC(C(COC)NC(C)=O)=O)C2)=O)cc(C)oc1C c1(-c2cn(C3CC(NC(C(c4cccc(C)c4)C)=O)C3)nn2)ccc(Cl)cc1F N1(C(CSCC#C)=O)C2CCC1CC(N(C(=O)CCc1cncs1)C)C2 c1(OCC(=O)N)ccc(F)cc1.C1(C(F)F)CCN(C(C2(O)CCSC2)=O)C1 CC(C)(CN1CCN(C(=O)NC2CCCC2c2ccccc2)CC1)C(=O)O CC(C)(O)CCCNC(C1CCN(C(C2(C)CC2(C)C)=O)CC1)=O C(=O)(C1=CCC2(COC2)OC1)N1CCN(C)CC1CNC(=O)C(C)(C)N(C)C c1(CC)nc(C)ncc1C(=O)NC1C2CN(C(=O)C3=COCCO3)CC12 C1(C(=O)NC(C(=O)NCCOC(=N)O)Cc2cnc[nH]2)CC(=O)CCO1 C(C)(C(=O)NC1CC1CNC(=O)Cc1c[nH]nc1C)(c1ccccc1)OC c1(NC(=O)NC(CC)COC(C)(C)C)cccc(C2CNC(=O)C2)c1 C(=O)(CC(C)(C)F)NCC1CC(NC(c2cc(OC)ns2)=O)C1 C(C1=NOC2CN(C(=O)CC3(CO)CC3)CC12)NC(c1cn(C)nc1)=O C(=O)(CCCC(F)(F)F)NC1C(CNC(C(C)(C)c2cscc2Cl)=O)C1 Cc1cc(C(=O)NC2(C)CN(C(c3cccc(C(F)(F)F)n3)=O)C2)ccc1Br CC1C(C)N(C(c2cc3c(ccn3C)[nH]2)=O)CCN1C(c1csc(O)n1)=O C1(NC(CCSCCC)=O)CN(C(c2cocn2)=O)C2CC12 N1(C(c2c(CC)cncc2)=O)CCC2CC2(C(=O)N(CC(C)(CO)CO)C)CC1 C1(NC(CCC#N)=O)CCC2CN(C(=O)C=CC(F)F)CC12 CC1(C)CCC(C(=O)NC2CC(F)C2)(NC(c2cc[nH]c2)=O)C1 C12(CC)CN(C(C3CCCCO3)=O)C(CNC(C3CCCC3C3CC3)=O)(C1)C2 c1(NC(c2cc(-c3cc4ccccc4o3)cnc2F)=O)cc(F)c(F)cc1F C1(CC=C)(NC(=O)CC2(O)CCC2)CCCN(C(C2CCC(OC)CC2)=O)C1 c1(OC)cccc(C(N2CC(CNC(c3ccc(C)cc3O)=O)CC2C)=O)c1Cl CC(C)CCC(=O)NCC1CC(O)CN1C(C1CCC1O)=O.c1cc(Br)cs1 C1(C(N2CC(NC(CCC(=O)NCCC)=O)(CO)C2)=O)C(F)(F)C12CCC2 N1(Cc2cc(C)cc(Br)c2)CCc2ccc(C(=O)Nc3c(C)csc3C)cc2C1 C(=O)(CCS(=O)(=O)c1ccccc1)N1CCC(NC(c2ncn(CC)c2)=O)C1C C1(C#N)(C(N2CC(C(C)NC(CC3(OC)CCC3)=O)C2)=O)CC2CCC1CC2 CCCC(C(=O)NCC(O)C)c1cccc(Cl)c1.C1(CC=O)C(C)(C)C1(C)C.N CCCCC(O)CCC(=O)N1CC2(CCN(C(c3cc(O)ccc3O)=O)C2)C1 N(C(=NCC1CCCN(C(=O)OC)C1)N1CCc2ccccc2C1)C(CC)CC C1(NC(c2c(OC)n[nH]c2)=O)C2CC3CN(C(=O)C(O)Cn4cncn4)C1C3C2 C1(C(N2CCOC(CNC(C3(F)CCCCC3)=O)C2)=O)CCOC2(CCCC2)C1 C1(C(=O)NCCCC(=O)NCc2c(C)nns2)CCCC(F)C1 Cc1c(C(N2CC3CCC2CN3C(=O)C(O)C2CC2)=O)[nH]c2c1C(=O)CCC2 c1(NC(C(=O)N(CC(CC)(F)F)C)=O)ccc(C#N)c(Cl)c1 CC(CC(=O)O)C(=O)N1CCC(c2cn(-c3cncc(Br)c3)nn2)(N(C)C)CC1 N1(C(c2c(CC)c[nH]c2)=O)CC2CCCCC2(NC(=O)C(c2ccc(C)o2)C)C1 c1(C(=O)NCCC2CCN(C(c3ncn(C)c3)=O)C2)cccc2oc(O)nc12 C=CCC(CC(=O)N1C2CCCC1CC2)NC(c1cncn1C1CC1)=O c1(OCC(=O)NCCCOC)ccsc1C(=O)Oc1ccccn1 c1(C(=O)NC2C(CNC(CCCC=C)=O)CC2)ccc(Cl)c2ccccc12 N1(C(C(=O)Nc2c(OC)ccc(F)c2)=O)C2CCC1CC(CCF)C2 c1(C(=O)O)cc(F)cc2c1CN(Cc1cc(I)cc3c1OCC3)CC2 N1(C(COCCCOC)=O)CCC2(COCC(CNC(c3cn[nH]c3)=O)O2)C1 CCCCCC(F)C(=O)NCC(CCC)NC(C1(C)CCC(=O)NC1)=O C=CC(C)(C)CC(=O)NCCC1CCOC1.c1(C(=O)N)scnc1C(C)(C)C C1(NC(C2COCCN2C2CCCC2)=O)CC2CC1CN(C(c1cnco1)=O)C2 N1(C(COC2CCN(C(c3nccc(C#C)c3)=O)C2)=O)CCC2CCCC2CC1 c1(OC)coc(CN2CCC(C)(NC(=O)Cc3cccnc3)CC2)cc1=O CC(C)CC(O)C(C)C(=O)NCC1(O)CN(C(C2(N(C)C)CC2)=O)C1 c1(C(=O)NC2(C)CCN(C(CC(C)(C)F)=O)C2)cc2cccnc2nc1N C1(CC=C)(NC(=O)CO)CCN(C(C2CC3CCC3C2)=O)C1.C1(C)CCCC1 C(=O)(C(C)CC(C)C(C)=O)NC(C(C(=O)N(CCN(C)C)CC)(C)C)C Cc1nn(C)cc1C(=O)N(C)CC1CCCC(NC(=O)COCC(F)F)C1 N1(C(C(C2CCCC2)OC)=O)C2CCC1CC(C(=O)NC1C(=O)OCC1CO)C2 N1(CC)CCOCC1CC(=O)NCC(CC(C)C)NC(c1coc(C)c1)=O Cc1cccc(CC(=O)NC2CC3(C2)CC3C(N2CCC(O)(CO)C2)=O)c1 N1(C(C(C(C)C)N(C)C)=O)CC2CCCC2(NC(c2ccnn2CC(F)F)=O)C1 C(C1CCN(C(c2cncc(Cl)c2)=O)CC1)=CC(=O)N.c1(C(C)C)cc(C)no1 c1(CN2CCN(C(C(C(C)C)n3cnnn3)=O)C(C)C2)nc2ccccc2s1 c1(OC)cc(=O)n(C)cc1C(=O)N.C1CCCCC1.C(=O)C=CC(C)C.C c1(NC(c2cc(O)n[nH]2)C)nccc(=NCCNc2cccnn2)[nH]1 CCC(C)CCC(=O)NCC1(C(C)NC(C2CC(OC)C2)=O)CC1 c1(C(=O)NCC2OCCN(C(CC(C)C3CC3)=O)C2)cc(F)c(Cl)cc1F c1(C(C)NC(C(=O)N(CC(CC)C)C)=O)cccc(OC(F)F)c1 N1(C(CC(=C)Br)=O)CC2CCCC2(NC(C2CCC(C(N)=O)CC2)=O)C1 C#Cc1ccc(C(=O)NCC(C2(O)CCN(C(=O)CP(C)(C)=O)C2)C)c(F)c1 C12(C(=O)NC(CN(C(C(C)O)=O)C)Cc3ccccc3)CCC(CC1)O2 C(=O)(C(CO)C(C)(C)C)NC(C(N1C(C)CCC(C(N)=O)C1)=O)Cc1cnc[nH]1 CC(C)CC(CC(=O)N1CCOC(CC(N)=O)C1)NC(=O)CNc1ncccn1 c1(C(N2CCC(CC)C2C(=O)N(C)CC)=O)cc([N+](=O)[O-])c[nH]1.C(C)=O.N n1(CC(=O)NCCNC(c2cccc(C)c2)=O)cnc2cc(C)c(C)cc12 c1(CCCC(=O)NCCC(C)(C)NC(C2COCCO2)=O)ccc(Cl)cc1 c1(CCNC(CN(C(CCn2cnc(=N)[nH]2)=O)C2CC2)=O)ccc(O)nc1 N1(C(C(CC2CC2)OC)=O)C2CCC1CN(C(=O)CCCCCSC)C2 C(=O)(C(C)(C(F)(F)F)NC(c1ccc(C#N)s1)=O)OCC C(=O)(C(C)Cc1cccnc1)NCCC(C)N(C(=O)Cc1ccn(C)n1)C CC(C)CCCNC(c1cccc(C2(C)CC2)c1)=O.C1(C(=O)N)CC(C)CCO1 C1(C(=O)NCC(CC)NC(=O)C(O)Cn2cncn2)CC(F)C(=O)N1 c1(C(=O)NCC2(F)CCCN(Cc3ccn(C)n3)C2)cc2[nH]ccc2cc1Cl Cc1ccnc2c(C(N3CCN(C(c4cnsn4)=O)CC3CC3CC3)=O)cnn12 c1(C(C(=O)OC(C(C)C)C#N)O)ccc(C(F)(F)F)cc1 C1(CC(N2CCC2)=O)CCCS(=O)(=O)C1.C(C1CCCN1C)=CC=O.C=CC c1(CCC(=O)NCCC(C)N(C)C(C2CN(S(C)(=O)=O)C2)=O)nncn1C C1(NC(CONC(c2ccc(C)nn2)=O)=O)CC(CO)C12CCC2 c1(C(N2CC(C)CCC2)=O)ccc2[nH]nc(Cl)c2c1.C1(C(C)C)(C(=O)NC)CC1 C(c1cccc(Cl)c1)=CC=O.CC(C)(C)C(=O)NCC=O.C1(CC)CC1.N C(C(N)=O)(C(C)CC)OC(C1CC(CC)(CC)C1)=O c1(C=O)ccc(N)c(Cl)c1.c1(OCCC)ccc(OCC(=O)N)cc1.C(C)C c1(CN(C(C2N3CC(C)N(CC3)C2)=O)C)cnn2c1CN(C(=O)C=CI)CC2 C1(CNC(c2ccncc2)=O)CC12CCN(C(c1n[nH]c3c1CCCC3)=O)CC2 c1(-c2cc(C(=O)NCCCN(C(=O)Cc3sccc3Cl)C)n[nH]2)ccc(F)cc1 c1(CCC(=O)NCC(C(C)C)NC(=O)C=CC2CCOC2)cccnc1Cl CCS(=O)(=O)CC(=O)NC1CCN(C(c2cc(Cc3ccccc3)on2)=O)C1 C1(CNC(c2cnc(CC)s2)=O)CN(CCOCC2CCC2)CCCO1 C12(NC(c3cncc(C(C)C)c3)=O)CCC(CN(C(C3(C)CCC3)=O)C1)C2 CCCCCC(O)C(=O)NCC(C)CN(C)C(c1cnn(C(C)(C)C)c1)=O N(C1CCCc2cccnc21)(C(=O)C(CCC)OCC)CCC Cc1sc(C(N2CCC(O)(C(C)NC(=O)Cn3nccn3)C2)=O)cc1Br C12(C=O)C3C4C1C1C2C3C41C.CC1CN(C(C2(C)CCCN2C)=O)CC1CC.N N1(C(C(=O)Nc2cccc(N3CCCCCC3)c2)=O)CC2CC(O)CC(C2)C1 CCC(CC)CCC(=O)NC1CN(C(C2CN(C3CCOCC3)C2)=O)CCC1C n1(CC(=O)NC2(C)CN(C(=O)CC3CC34CC4)C2)[nH]cc2c(=O)ncnc1-2 c1(OC)ccc([N+](=O)[O-])cc1C(=O)NCC(F)CNC(c1cocc1C)=O C1(CCOC)(NC(c2cscc2Br)=O)CCN(C(C2CCOCC2)=O)C1 c1(C(N2CC(CNC(C3(CCOC)CCC3)=O)OCC2)=O)nccn2ccnc12 CC(C(=O)N(CC(O)C)C)O.CC(F)(F)F.C1(CS(C)(=O)=O)(C=O)CCC1 C=CCC(CC)C(=O)NC1CC(CCC(=O)NCC(F)(F)C(N)=O)C1 CC1(C(=O)N2CCC(NC(c3ccc(F)c(F)c3)=O)C(O)C2)CCn2ccnc21 CC1(C)OC2(CNC(C3C4COCC34)=O)CC1(NC(C1CC1F)=O)C2 C1(NC(C(C)=C(C)C)=O)CCOC(C(=O)N(C)Cc2c(C)noc2C)C1 Clc1cccc2c(CN3CCN(Cc4cccs4)CC3)cncc12 c1(NC(CCC2CCN(C(CC3C(C)(C)C3)=O)C2)=O)cncc(C#N)c1 N1(C(=O)CCN2CCOCC2)CCC2(C1)CN(C(c1ccncc1Br)=O)CCO2 CC(=NO)C1CC(C(N2CC(C)(NC(=O)CCn3cccn3)C2)=O)C1(C)C c1(C(c2nnnn2C2COC2)NC(CCC)CC)ccc(Cl)c(F)c1 c1(SCCC)cccc(C(=O)NC(C)(C)C2CC2)c1.c1(C=O)nncn1C.N c1(C(=O)NC2C(NC(c3c(Cl)cn(C)n3)=O)CCCC2)ccc2nccn2c1 N1(C(C=Cc2scc(C)n2)=O)CC(C)CN(C(=O)C2=COCCO2)CC1C Cc1nnc2n1CCCC2NC(c1ccc(CN=[N+]=[N-])o1)=O C1(NC(=O)Cc2cnoc2)CC(C(=O)NCC2CC23CC3(F)F)CC1O.C C1(CNC(C2N(Cc3ccc(C)cc3)CCCC2)=O)CCC2(CC1)CC2 N1(C(CCOCC#C)=O)CC(O)CC1CNC(=O)C(F)n1cccn1 C1(C2CCN(C(c3cn4c(n3)CCC4)=O)CC2)(NC(C2CC(C)OCC2)=O)CC1 c1(C=O)cc2c(s1)CCCNC2=O.C1(C)(NC(COCCOC)=O)CCC1.N n1(CC(=O)NC2C(NC(=O)CN3CCC(O)CC3)CC2)sc2ccccc2c1=O CC1CCC(NC(=O)Cn2cnc(N(CC(F)F)C)c2)c2ccccc21 C1(N(C)C)CCOC(C(N2CC(CNC(=O)CCCc3cccnc3)C2)=O)C1 C1(NC(c2ccc(Cl)o2)=O)CC2CN(C(c3cnccc3C(F)F)=O)CC2C1 C1(c2n(-c3c(C)cc(Br)cc3)nc(CCN(C)C)n2)CCCC(C)(C)CC1 C1(O)(CC)CCN(C(=O)Cc2cccnc2Cl)C1.c1(OCC)n[nH]cc1C=O.N C(=O)(Nn1ccnn1)C1CCN(C(C2CCC(C)O2)=O)CC1 N1(C(c2cnc(C)c(N)c2)=O)CC2(C1)SCCC2NC(=O)C(C)CC(C)(C)C C(=O)(C(C(C)(C)C)NC(N)=O)N(CCNC(c1cc(C(C)C)no1)=O)C N1(C(C2CCCC(C3CC3)O2)=O)CCC2(CCCN2C(c2ns[nH]c2=O)=O)CC1 c1(C(c2nnnn2C(C)(C)C)NCCOC)nc(C)ccc1OC C1(CNC(c2cnc(S)nc2)=O)CCCCN(C(C2C=CCC2)=O)CC1 c1(C(CNC(=O)C(=O)NCC(C)(O)Cn2cc(Br)cn2)OC)ccccc1Cl C1(C(=O)NC2(CC=C)CCOC2)CCOCCN1C(c1cncs1)=O C1(NC(CC(n2ccc(C)n2)C)=O)COC2(C1)CN(C(C1CC13CCC3)=O)C2 C(C(C)(C)CC(=O)N1CC(=O)CC1C(=O)NCC1CCOC1)OC Cc1oc(C(=O)NC(C)Cn2cc(C3CC3)nn2)cc1CC1CCCCN1C c1(OC)cc(Br)c(C)cc1NC(c1cn(C)c2ncccc12)=O Cc1cc(CNC2CN(C(c3cc4occc4[nH]3)=O)CC23CC3)cc(O)c1 C(=O)(CCCCc1cnn[nH]1)NC(C1CN(C(=O)C(c2ccnn2C)O)C1)C CN=c1[nH]c(C(=O)NC2CC2CNC(=O)C(C)Cc2ccccc2F)cs1 C=C(C)CCCC(=O)NC1CCCN(C(=O)COCCC)C1CC C(=O)(CCCCCCBr)N(C)CC1CN(C(=O)Cc2ccc(Br)cc2)C1 c1(C(N2CC(C(=O)Nc3cnc(C)c(F)c3)OCC2)=O)cc(F)c(F)c(Br)c1F c1(CC(=O)NCCCN(C(C2CN(C)CCO2)=O)CC)sc(C)cc1C c1(C(=O)NCC(CC=C)NC(=O)C)cnc2c(C)c(Cl)ccc2c1.C(C)CC.O CCC(C)(C)C(C(=O)NCCCC1(NC(C2CCC(C)CC2)=O)CC1)OC Nc1c(C(=O)NCCC2CCN(C(C3CC4CCCC34)=O)C2)sc2ncccc12 c1(C(=O)NCC2C(C(N3CC(NC(C)=O)C3)=O)CCO2)[nH]ccc(=O)c1C c1(CCC)no[nH]c1=NS(=O)(=O)CCCCS(=O)(=O)N(C)CC1CCSCC1 C(C(C)(C)C1=CCCC1)NC(C1CC(C)N1C(c1ccccc1Cl)=O)=O C1(NC(C(C=C)O)=O)CN(C(C2CC(C(F)(F)F)C2)=O)CC2(CCC2)C1 C(=O)(C1=CC2CCCCC12)N1C(CNC(=O)Cc2cccs2)CC1 CCC(c1ccccc1)=CC(=O)NC1CCC1NC(c1ccc2scnc2c1)=O c1(C(=O)Nc2c(OCC)nccc2)sc(=NCc2ccccc2C(=O)O)[nH]c1C C(CO)(C(=O)NC1CC(NC(C2(CO)CCCC2)=O)C1)NC(C(C)C)=O N1(C(C(CCCC)NC(=O)CCSCCCC)=O)CCOC2(CCC2)C1 C1(C)(C(=O)NC(c2ncn(C)n2)C)CCN(C(C2CC3CCC3C2)=O)C1 c1(C(=O)NC(CC)CNC(C2CCCOCC2)=O)c(Cl)nc2ccccn12 c1(C(=O)NC2CC3CN(C(C(C)OC)=O)CC2C3)[nH]c2ccccc2c1C c1(C(=O)N)cc2n(n1)CCCO2.CCCC(C(=O)NC(C)(C)CC)NC(C)=O C=CC(CC)CC(=O)N1CC(OCCC(=O)Nc2cnc(F)nc2)C1 C1CCCN(C(=O)Cn2cnccc2=O)CC1.C(C=O)OCCOCCOC.N C1(C(=O)NCC(CCCC)NC(c2ncccc2SCC)=O)CCCCS1(=O)=O CC(C)CC(O)C(=O)N1CCCCC(NC(c2cnc(C3CCOC3)s2)=O)C1 c1(CN(C(CN(C(COCCOC)=O)C(C)C)=O)C)ccco1 Cc1cc(F)cnc1CNC(=O)NC(C)CC1CC1 Cc1nnc2n1CC(C(=O)NCC1(O)CN(C(c3c[nH]c4nccc-4c3)=O)C1)C2 c1(C(N(CCN(C(C(CCC)N(C)C)=O)C)C)=O)cc(O)cc(F)c1 C1(CNC(=O)CC2CC(=O)N2)CCCCN(C(c2csc(-c3ncc[nH]3)n2)=O)C1 C(=O)(C(C)(C)CC(=O)NC1CC2CCC1(C(N1CC(C)C1(C)C)=O)C2)OC c1(C(N(CCCNC(C2(C)CC2)=O)C)=O)c(C(F)F)cccc1Br N1(C(CC2ON=C(C)C2)=O)CCC(NC(c2nc(C)ncc2Cl)=O)C(C)C1 Cn1cc(C(=O)NCCC2CCN(c3ccncn3)CC2)c(C2CCCC2)n1 c1(CC(=O)NC(C)CC2CN(C(C3CCC(=O)N3)=O)C2)cnn2c1OCCC2 CCCCC(CC)C(=O)N1CCC1C(=O)NCCn1ncnn1 N1(C(C(CCOC)NC(C2CC2C(=O)OC)=O)=O)CCn2ncnc2C1 c1ccc(F)c(F)c1.c1(OCC)cccc(C(N2CC3CN(C(=O)N)C3C2)=O)n1 N1(C(Cc2nc(C(C)(C)C)sc2)=O)CC2CCN(C(=O)CS)C2C1.CCN(C)C c1(C(=O)NCC(C)OC)c(C)n[nH]c1C.c1(C2(C=O)CC2)cc(C)no1.N C1(NC(C(CC)N(C(=O)CC2COCC2O)C)=O)CCC(C2CC2)C1 CC1CCC(NC(=O)CN2CC=CC2)CN1C(c1c[nH]nc1F)=O c1(C(=O)NC(c2cc(C)on2)C)ccc(=O)[nH]c1.c1cn(C(C)C(=O)O)nn1.C N1(C(=O)C(O)C(F)(F)F)CCC2(CCCN2C(=O)C2=NOCC2)CC1 N1(C(C(N2CCSCC2)C)=O)CCN(C(C2CC3CCC2CC3)=O)CC1C(F)F CCC(C)(C)C(O)C(=O)NC1CC(C)(NC(C2CC23CCOCC3)=O)C1 N1(C(Cc2cc(C)ns2)=O)CC(CNC(=O)C(C)n2cccn2)C(F)(F)C1 N1(C(CCNC(N)=O)=O)CCN(C(=O)COCCOc2ccccc2)C2CC12 N1(C(c2ccc(C)[nH]2)=O)CC(NC(=O)C(F)OC(F)(F)F)CC1C c1(C(=O)NC2CCCC(NC(C(C=C)O)=O)C2)cnc(O)c2ncccc12 C(=O)(C(O)CCCNC(=O)C(C)n1cccc1)N1CC(C)(COC)C1 N1(C(CC2CC(=C)C2)=O)CC(NC(=O)C=Cc2cccs2)C2(CCOCC2)C1 C1(C2(O)CN(C=O)C2)(CC)CC1.C12(O)CN(C1)C(=O)C2.C(C)(C)C.CO C=CC1(CC(=O)NC2CCCC2(C)N(C)C)CN(C(=O)CC2(C)CC2)C1 CC(C)CC(O)C(=O)NC1(CO)CCN(C(c2cncc(C(C)(F)F)c2)=O)C1 N1(CC)CCC(CN(C(=O)CCNC(c2ncccc2CN)=O)C)CC1 c1(COC)ccc(C(=O)N)o1.C1(F)CCC1.C1(C=O)CSCN1C(C)=O c1(CN2CC(F)(C(=O)Nc3cc(CC)no3)C2)c[nH]c2cccc(C)c12 Cc1nc(C(=O)NC2CCN(C(c3cnn(C)c3N)=O)CC2F)c(=O)[nH]c1C c1(NC(C23C(CN(C(c4c(C)cn(C)n4)=O)C2)C3)=O)ccc(F)cc1O C1(NC(C(c2ccccc2)C)=O)CC2CCC(C1F)N2C(C1(O)CCC1)=O CC1(C)CN(C(C2CCCN2N=O)=O)CC1NC(c1csc(-c2ccco2)n1)=O c1(C(=O)Nc2cc(C(=O)OCC)c(O)cc2)cc2[nH]ccc2cc1-c1cnoc1 C1(NC(COCC(=O)NC)=O)CC2CCC1N2C(=O)C(c1ccccc1F)C [N-]=[N+]=Nc1ccccc1NC(C1CCN1C(C1C=CCCC1)=O)=O C1(CC(=O)N(C2(C(=O)N(C3(C4CC4)CC3)C)CC2)C)CCCSC1 C=CCC(C)(CC)C(=O)N1C2CCC1C(NC(c1ccon1)=O)C2 C(=O)(C(C)=Cn1ccnn1)NCC1CCN(C(C(C(CC)C)N(C)C)=O)CC1C c1(CC(=O)Nc2ccc(Oc3ccc(CC)c(I)c3)cc2)ccc2[nH]ccc2c1 c1(NC)c(C(=O)N(CC(C)NC(=O)C(C)c2cncs2)C)cccc1F N1(C(COC)=O)CC(CNC(c2nnn(-c3ccc(Br)cc3)c2C)=O)CCC1C c1(C(=O)NC2CCCCN(C(C3CCCC(F)C3)=O)C2)ccn2ccnc2n1 CC(C)C(O)CC(=O)NCC1C(C)CCN1C(C1CC(n2ccnn2)C1)=O Cc1cccn2cc(C(N3CCN(C(=O)C(C)(C)C4CC4)CCC3C)=O)cc12 c1(OC)cccc(C(=O)NCCCCCN(C(=O)CCc2ccccc2)C)c1F Cc1noc(Cl)c1CCC(=O)NCC(C1CC1)NC(c1coc(C#N)c1)=O c1(CNC(CN(CCC)C(C2CCC(C)C2)=O)=O)cc(C)ncn1 C1(NC(c2ccc(CC)nc2)=O)CC12CCC(NC(=O)C(C)COC)CC2 c1(CC)cccc(C(=O)NC)c1.C1CCCC1.c1(CC=O)cnn(C(C)C)c1 C(=O)(CCC(=O)N1CCOCC1CN(C)C(c1conc1C1CCC1)=O)N(C)C C=CC1(C(=O)NCCc2cncs2)CCN(C(c2cnc(Cl)s2)=O)CC1 c1(C(N2CCC(OC)(CNC(C3CCCSC3)=O)C2)=O)ccc(C#N)nc1O CC(C)C(C)CC(=O)NC(C)CCCCNC(=O)C(C)(C)CC1CCOC1 C1(CNC(CN(CCCOC)CC2CCCC2)=O)CC=CCC1 c1ccc(S(C)(=O)=O)cc1.C1(OC)CC2(C1)CC(C(C=O)NC)C2.C1CC1.N C1(C)(CCC)CCN1C(=O)C(C)OCCNC(=O)C(C)OCCC(C)C Cc1ccc(C)c(OCCC(=O)N(C2CCCCO2)Cc2cc3c[nH]nc3s2)c1 C(=O)(C(=O)N=S(C)(C)=O)N(C1CC(NC(c2c(C)cccc2O)=O)C1)C CCCC(C(=O)N(CC(=O)NCCS(=O)(=O)CC)CC(C)C)C(C)C C1CC2(C1)CCC2.c1ccc(C=O)o1.C(=O)CC.C(C)(C)C.C(CS)OC N1(C(CNC(C(C)C)=O)=O)CCN(c2ncc(Br)c(N3CCOCC3)n2)CC1C C(=O)(C(COC)CC(C)C)NC1(C)CCCN(C(c2n[nH]c(CC)c2Cl)=O)C1 c1(C(N2CC(CNC(C3(CC)CC3(F)F)=O)C2)=O)cc(N)cc(O)c1 Cc1cccn2c(C(N3CC(NC(=O)C(F)(F)CC4CCCO4)C3)=O)cnc12 N1(C(c2cc(CC)no2)C(=O)NC2CCCC2)CC(CO)C2(CC2)C1 C1(O)(NC(COC2(C)CN(C(=O)C(F)C(C)(C)O)C2)=O)CCCCCC1 NC(=NCC1CC1)NC1CC12CC2.C1(C(=O)NCC)CCC1.C1COC1.C C(=O)(C(C#N)C(C)C)N1CCC(CC#C)(C(=O)NCC2CC2C2CCC2)C1 C(=O)C#CC1(C)CCCO1.c1(OCC)ccccc1C=CC(=O)NCC(F)C.N c1(C(N2CC(C)(C(=O)NCCOCC)C2)=O)ccc(N(C)CCO)cc1.C c1(C(=O)NC(CN(C(c2cc(CC(C)C)[nH]n2)=O)CC)C)cc(Cl)ccn1 CCC(CC)CCNC(=O)CN1CCC(O)CC1.c1(C2C(C(=O)N)C2)ccoc1 C1(O)(CC(=O)Nc2c(CC)cncc2)CCN(C(c2ncc(Br)cc2C)=O)CC1 N1(C(CSS(C)(=O)=O)=O)CC2(CCN2C(=O)CCCCC2CCCCC2)C1 c1(C2N(c3n(CCCC)c(-c4nc(CO)cs4)nn3)CCC2)ccc(Cl)c(Cl)c1 C(CC(=O)N1CC2CC(C1)C2)(C(C)C)OCC.c1(C=O)ccc(C2CC2)o1.N C1(C(=O)NCC2(C)C(C)(C)C2)CN(C(=O)Cn2cc(CO)nn2)CCO1 C1(C(N2C(C)C(NC(c3cnn(C)c3)=O)CC2)=O)COCC2(CCC2)O1.C1CC1 CCCCCCCC(=O)NC1CCCN(C(c2c(C(C)(C)C)nsc2N)=O)C1 CC1CCC(F)(F)CN1C(=O)C(C)(C(F)F)c1ccccc1 c1(C(=O)N)cc(C)nc(C(F)(F)F)n1.C=CCCCNC(c1ccc(F)s1)=O c1(C(=O)NCC(C)NC(=O)CO)nn(-c2ccccc2F)cc1O N=c1[nH]cc(CN(C(=O)NCC(C2CCNCC2)O)C2CC2)s1 c1(CC)cccc(C(N2CC(NC(C3CCSCC3)=O)C3CC23)=O)c1N N1(C(c2ccc(COC)cc2)=O)CC2CCOCC2(NC(c2cc(C)on2)=O)C1 N1(C(C2(NC(C(C3CC3)OC)=O)CC(O)C2)=O)CCC(C2CCC2)CC1 C#CC1(O)CCCN(C(=O)CCN(C(=O)CC=CC=C)CCCO)C1 C(CCC(=O)N(C)C)(c1nnnn1C1CC1)NC(C(C)NC(N)=O)=O C1(NC(c2nccc(OC)c2)=O)CCN(C(c2cnnc(Cl)c2)=O)CC12CCC2 n1(CCOC)cc(C(=O)NC2CCC(NC(C3CCCSC3)=O)CC2)c(C)n1 N1(C(CSCC=C)=O)CCC(F)(C(N2CCCC(COC)C2)=O)CC1 C#CCC(C(=O)N1CC(CS(C)=O)C1)NC(C12CCCC1C2)=O c1(-c2cn(C3CCC(NC(CC(CC)SC)=O)C3)nn2)cc(F)cc2nn[nH]c12 c1(OCC)cccc2c1OCC(C(=O)N(CC(C)C)C)C2.C(=O)C1=C(Cl)CC1.N C(=O)(C(C)(C)C(C)O)N.C1(CC=CC(=O)NCC=CCCC)CCC1 N1(CC)CCC(N(C(=O)C(C)(C)Nc2cccc(-c3nn[nH]n3)c2)CC)CC1C N1(C(CS(=O)(=O)N(CC)CC)=O)CCCC(C)C1C.C(=O)CCC(C)(C)F c1(COC2CCCN(C(=O)Cc3cn(C4CCC4O)nn3)C2)csc2nccn12 C1(NC(c2ccc(C(C)=O)[nH]2)=O)CCC(NC(c2cc(F)n[nH]2)=O)CC1 O(NC(=O)C(C)N(C(=O)C(C)CN(C)C)C(C)C)CCCOCC c1(C(=O)NCCN(CCC)C(c2cscc2Cl)=O)cnc(C(C)C)[nH]1 CCC(C(=O)N)Sc1nc(C)no1.C1C=CCN1C(=O)CCc1cnc(O)[nH]1.C N1(C(C(CNC(C)=O)(C)C)=O)CCC(O)(C)CC1.C12(C=O)CCC(CC1)CO2 N1(C(C2CC(C)(F)C2)=O)CCCC(NC(=O)Cc2cccc(C#N)c2)CC1 c1(C(C)O)ccc(C(=O)NC2CCN(C(c3cn(C4CC4)nn3)=O)C2)cc1 C1(C(=O)NC(CNC(CC(C)(C)C)=O)CO)CC(=O)c2ccccc2O1 c1(N2CCC(CCC)C2)nc(N(C)CCc2ncc(C)s2)c2c(n1)CSC2 c1(C=O)c(C)nn(C)c1N.N1(S(CC)(=O)=O)CCCC1C(=O)N.C1CCC1.C C(=O)(C(CCS(C)=O)N(C)C)c1scc(-c2ccc(C)s2)n1.C12CCCC1CN2 N1(C(C(CC)c2cccnc2)=O)CC(N(C(=O)CCC(C)(C)F)C)C2(CC2)C1 N1(S(CCCC)(=O)=O)CC(NC(=O)CCNC(=O)C(=O)CC)C(C#N)C1 Cc1ccc(F)c(C(N2CC(F)CC2CC(=O)N(C2CCN(C)C2=O)C)=O)n1 c1(C(=O)NC2C(NC(CSC(C)C)=O)C2)cc(Cl)c(F)cc1Cl C#Cc1ccc(O)c(CNC2CC3CCC2N(C)C3)c1 C(=O)(C1=C2CCCN=C2NN1)NCC1OCCCN(C(CNC(=O)NC)=O)C1 c1(C(=O)OC)c(C)[nH]c(C(=O)NC2C3CN(C(C4CCC4)=O)CC23)c1C CC1CC(NC(C2CC(C)(C(=O)O)C2)=O)CN1C(c1csnn1)=O C1(N(C(C(SC)SC)=O)C)CCC(NC(=O)Cn2nnc(C3CC3)n2)C1 NC(=O)CCCCC(=O)NCCC1(O)CN(C(C2(Br)CC23CCC3)=O)C1 c1(C(=O)NCC2CC(NC(CCCC)=O)C2)c(C)cc(C)c([N+](=O)[O-])c1C c1(CC)ccc(C)c(NC(C2CN(C(=O)C(C)c3ccco3)CC23CC3)=O)c1 CC1(C)CCCC(O)(C(N2CCC(NC(=O)C(F)(F)CO)C(F)C2)=O)CC1 N1(CC(=O)N(CCN(C(C)C)C(C2CCCOC2C)=O)C)CC(=O)NC1=O N1(C(c2ccn3ccccc23)=O)CCC(C2CCCN(C(=O)C(O)C3CC3)C2)C1 CN=c1[nH]c(=NC(CC(N)=O)C2CC2)[nH]c(=NC2CCN(C(C)(C)C)C2)[nH]1 c1(COC)cc(C(=O)NCCc2cn(CC(C)(C)O)nn2)n(C)c1 Cc1nc(C2CC2)nc(O)c1C(=O)NC1CCCCN(C(=O)CO)C1.C1CCC1 Cc1cc(F)c(C(=O)NC(C)CCN(C(=O)CC2(C#N)CCC2)C)c(Cl)c1 c1(NC(CC(CC#C)NC(c2csc(C#N)c2)=O)=O)cc(O)c(C)cc1C C1(C)(NC(C(CC(C)C)N(C(C(C(CC)C)=O)=O)C)=O)CCCCC1(C)C C1(C(=O)NC2C(NC(CCC3CC(C)C3)=O)CC2)CC(O)C12CCC2 N1(C(C=CC(=O)N(C)C)=O)CC2CC(C1)C2NC(C1C=CCC1)=O C1(NC(=NCC=C)NCC(F)C(F)(F)F)CN(C(=O)OC(C)(C)C)CC12CCC2 n1(CCCC)nc(C)c(C(=O)NC2CCN(Cc3nc(C)cs3)CC2)c1Cl C(=O)(CCP(C)(C)=O)N1CCC(C(C)NC(C=COc2ccc(OC)cc2)=O)C1 C1(O)(CNC(c2cccc([N+](=O)[O-])c2)=O)CC(N=c2[nH]nc(-c3ccon3)s2)C1 C1(C(=O)N)C2CC1N(C(C1CCCC1)=O)C2.C1CC1C(F)(F)F.C1CC1 C1CCCN(C(c2cscc2C(F)(F)F)=O)C1.n1(COC)nccc1C(=O)N.C N1(C(c2cn(C)c(=O)n2C)=O)CC2(CCC(CNC(=O)CC3CCCC3)O2)C1 CCCCC(CC)CC(=O)N1CCC(OCC(N2CC=CC2CF)=O)C1 Cc1nc(NCCS(=O)(=O)CC2CCC2)cc(=NC(C)c2cnn(C)c2C)[nH]1 c1(C(N(CCCN(C(=O)CCOC2CCOC2)C)C)=O)ccc2oc(O)nc2c1 CC1(C)CN(C(=O)Cc2cnc[nH]2)CC1CNC(c1ccc(N)c(O)c1)=O Cn1nc(C2CC2)cc1-c1ncccc1C(N1CCC(Br)C1)=O c1(SC(C)C(=O)NCC2CN(C(=O)CCCN(C)C)CCO2)ccc(F)cc1 C1(C(=O)N(C2CCNC2=O)C)(COC)C=CCN1C(c1c[nH]c(=N)o1)=O c1(OC)cc(C(N2CC(O)CC2(C)C)=O)c(NC(C2CCCN(C)C2)=O)cn1 c1(OC)cc(C)cnc1C(N1CC(NC(=O)CC2(OC)CCCC2)C1)=O C1(CC)CCC1C(=O)NOCC(N1CC(COC)C1)=O C=CC1CCCN(C(C2OCCC2CNC(=O)CC(F)(F)CC)=O)C1 C1(NC(C(CO)NC(C(C)C)=O)=O)CC2(C1)CN(C(c1cnsc1)=O)C2 CC1CC(NC(c2cccc(N)c2O)=O)CCN1C(c1cc(F)cnc1O)=O Cc1c(CN(C)CC2CCCN(c3ncc4[nH]ccc4n3)C2)[nH]c2ccccc12 N1(C(CSCC(=O)OC)=O)CC2(CC(NC(C3CC4CC3C4)=O)CO2)C1 N1(C(c2c[nH]c(=N)o2)=O)CCN(C(=O)CSCC(N)=O)C2(CCC2)C1 C1(C(=O)NC(C2CCCCC2)CNC(C2(SCC)CCC2)=O)CCOC1C c1(C(=O)NCC(CO)NC(c2cnc[nH]2)=O)n[nH]c2c1COCC2 N1(C(c2ccc(CC)[nH]2)=O)CCC(C2CC2)C1CNC(=O)C(C)C(C)C C1(C(=O)NCC(C)(C)SC)CCCCC1(C)NC(c1ncncc1N)=O CC1CN2CCN1CC2C(=O)NCC1CCN(C(=O)CC(F)(F)Cl)CC1 CCC(C)C(O)C(=O)NC(C1CCN(C(=O)CC2(C)CCC2)CC1)(C)C C=C1CC2(C1)CC(C(N1CC(F)CC1CNC(c1cc(Br)c[nH]1)=O)=O)C2 C1(CC#C)CN(C(=O)C(COC)NC(c2ncoc2C)=O)CCO1 c12ccc(cc1F)CC(=O)N2.C1(C(=O)OCC)CCCC1N(C)C c1(N2C(CNC(C=CC)=O)CC(F)C2)cc(C(C)C)nc(C)n1 c1(C(=O)NC2CC(CNC(=O)CCC3CCOC3)C2)cccnc1-n1cccn1 C1(NC(CC2N(C(CCC(C)(F)F)=O)CC2)=O)C(=O)OC2CCCC12 C1(C)(NC(C(C)OCC2CCCO2)=O)CC(NC(=O)C)C1.c1ccncc1 CS(=O)(=O)C1CCCC1C(=O)NCCC1CCCC1.C1(C=O)CCC=CCC1.N C1(COC)CCN(C(C2CC(=O)CN2C(c2nc(C)c(C)s2)=O)=O)C1(C)C C1(OC)CCCCC1n1cc(CCC2(O)CN(C(=O)COC(C)=O)C2)nn1 CN1CC2OCCN(C(=O)C(C)(CO)NC(=O)C(F)n3ccnc3)C2C1 CCC1=NOC(C(=O)N(CC(C)NC(=O)Cc2ccncc2Cl)CC)C1 CCC(CC(=O)NC1CC=CCC1C(=O)N=c1cc(C)n(C(C)C)[nH]1)CC(C)C C1(NC(c2cnc(-c3ccoc3)s2)=O)CCCC(NCc2cn(C(C)C)nn2)C1 c1(C(N2CCCN(C(=O)OCc3ccccc3)CC2)C)cccc2ccccc12 N1(C(c2cnc(CC)nc2)=O)CCCC(CC)C1C(=O)N(CC(C)(F)F)C c1(NC(C)=O)ccc(C(=O)COC(c2ccnc(C)c2Cl)=O)cc1F C1(O)CCCOC1.C1(CCC=C)(C(=O)N)CN(C(=O)C(C)Cn2cccn2)C1.C c1(C(=O)NC2C(NC(C3(OC)CCC3)=O)COC2)ccc(Br)c(Cl)c1 c1(C(=O)OCC)cnn2c1OCC(NC(=O)Cc1cn(C)nc1Cl)C2 N1(C(C(C)SC)=O)CC2(CCC2NC(=O)C(=Cc2ccc(F)cc2)C)C1 Cn1nnc(C(N2CCC(F)(CNC(c3cc(C(F)(F)F)cs3)=O)C2)=O)c1N Cc1nc(C(=O)NCCC2(C)CCN(C(=O)C3=CCOC3)C2)cc(O)n1 CS(=O)(=O)C1CC(C(=O)N)C1.C1CCCCN(C(=O)C=CC(F)(F)F)C1.C Cc1ccc(C)c(C(N2CC3(CCC3NC(=O)C(C)NC(N)=O)C2)=O)c1 C1(CC(=O)NC)CN(C(=O)C=C(C)C(F)F)CCN1C(c1cccnn1)=O C1(CC=O)NC(=O)NC1=O.C(C)(C)(C1CCC1)NC(COCCCC)=O.N C1(OC)CCN(C(=O)C=Cc2ccn(C)c2)C1.C(=O)C(C)Cn1ccnc1.C C1(NC(C=CSC)=O)(CNC(=O)CN2C(C)CCC2C)CCCCC1 c1(C(=O)N)nccc2cccnc12.N1(C(CNC(C)=O)=O)CCC(C(F)F)(C)C1 C(N=c1cc(NCCN(C2CC2)CC)nc(C)[nH]1)c1cc(CC)ncc1 C(=O)(C(CC(C)C)SC)N(CC(CC)NC(C1(S)CC1)=O)CC.C(C)=O C1(c2nnc(C)o2)COCCN1C(CC1(C#N)CC1)C(=O)NCCCF Cc1ccccc1CNC(C1CCC(C2CC2)N1C(=O)CC1CC1)=O c1(C(N(C2CCN(C(=O)C=CS(C)=O)CC2)CCCC)=O)cccc(C)c1N CCCCS(=O)(=O)CC(=O)NCC1(O)CCCN(C(c2nocc2C)=O)C1 N1(C(C(CCC)=CCC)=O)CC2CCCC1C2C.c1(C=O)csc(C(N)=O)n1.N c1(C(=O)NC2CC(C(N3CC(O)(CC=C)C3)=O)C2(C)C)cc2ccccc2[nH]1 C=CCCC(C(=O)NCCC(=O)N(C)C)NC(=O)C(C)CC(=O)OC CC(C)(O)CCC(C)(c1nnnn1CCC1(C)CC1)NCCc1ccns1 N1(C(c2c[nH]c(=NC)s2)=O)CCN(C(c2cccc(CSC)c2)=O)C(C)CC1C C(C(C)(C)CNC(=O)CCCN(C)C(C1CCCS1)=O)OC N1(C(C2CC(OC)C2)=O)CCCC(F)(C(=O)NCCc2ccc(C)s2)C1 c1(C(C)(C)C)ccc(C(=O)NC(C)(CNC(c2cnc(S)[nH]2)=O)CO)nc1 C(CCCC1CC1)(C(=O)Nc1ccccc1)N1C(C(=O)OC)CC(O)C1 C(=O)(C(C)(C)CCCNC(=O)CCCF)NCC1N(CC)CCC1 Cc1nc(C(C)(C)C)sc1C(=O)NCC(C)(C)C(C)C C1(NC(C(C(C)C)NC=O)=O)CCN(C(c2nccc(N)c2Cl)=O)CCC1CO CN1CCCC(F)(C(=O)NC2CC(CNC(c3ccccc3O)=O)C2)C1 c1(CN=C(NC(C)C2CC2)NCc2cccc(F)n2)c(F)cc(F)cc1F C1(F)(C(=O)OCC)CN(CC(=O)NCC2CCN(CC)CC2)CC1C1CC1 n1(Cc2cncc(C(C)C)c2)c(-c2ccc(Br)o2)csc1=Nc1ccnc(F)c1 c1(C(N2CC(C(=O)O)CC(C)C2)=O)cc2n(n1)CCCC2 Cc1cc(CN2CC(=O)N(CC(=O)NC3CCCCCC3)C2=O)cc(F)c1 CC1C(C(N)=O)CCCN1N1CCC(O)C(O)CC1 C1(C(=O)NCC=C)(COC)C=CCN1C(=O)CN(C)C(N)=O C1(NC(CC=C)=O)COC2(CNC(c3c[nH]c(-c4ccccc4)c3)=O)CC1C2 c1(CCC(=O)N)ccc2[nH]ccc2c1.N1(C(C(C2CC2)OCC)=O)CCC(F)C1 C(=O)(C(C)(C)C(F)F)N1CC(NC(c2cc(CCOC)on2)=O)(CO)C1 C1(C(=O)NCCC2CCCN(C(=O)Cn3cnnc3)C2)CC2(CCCCO2)C1 N1(C(C(CCC)NC(=O)C(C)=C2CCCC2)=O)CCCC(C)(N(C)C)C1 c1(-c2cn(CC3C(NC(C(CC)n4ccnc4)=O)C3)nn2)cccc(C#N)c1C N1(C(C2N(C(C3(C)CCSCC3)=O)C3(CC2)CC3)=O)CC2(CCC(O)CC2)C1 N1(C(CNC(CC(C)C)=O)=O)CC(NC(C2CC(N(C)C)C2)=O)CC1(C)C CCC(C)C(C(=O)NCc1ncc(C)[nH]1)N(C)C(C1CC1c1ccco1)=O.C N1(C(c2nc(Cl)sc2Cl)=O)CC2CN(C(C3CC(O)C3)=O)CCC2(CO)C1 N1(C(CSC)=O)CCCC(CCNC(=O)C(N2CCOCC2)C)C1 C1(C(=O)NCC2CCN2C(c2cnn(C3CC3(F)F)c2)=O)(OC)CCCC1 Cc1cc(COC(C2CC(=O)N(c3ccccc3C(C)CC)C2)=O)cc(F)c1 C1(C(N2CCC(C(CO)NC(C(C)(C)SC)=O)CC2)=O)CCC=CCCC1 C1(C)(C(=O)NC(CC#C)CO)CN(C(=O)CCC2(C#N)CCC2)C(C)(C)C1 N1(Cc2ccc(C)s2)CC2CC1C2C(=O)Nc1cc(C2CCCCC2)no1 c1(C(N2C(C(C)NC(C3CCN(C)C3=O)=O)CCC2)=O)cc(Cl)c(Cl)[nH]c1=N c1(NC(c2c(OCC)cccn2)=O)cccc(F)c1C(=O)N.c1ccc(Cl)s1 c1(C(N(CCCNC(C2(COCC)CC2)=O)C)=O)c(Cl)sc(Cl)c1C C1(C(N2C3(CNC(CSC(C)C)=O)CC(C2)C3)=O)C2CCCC(F)(F)C12 c1(C(=O)NCCC2CN(C(c3c(Cl)ccc(C)c3)=O)C2)cnc(O)c2ccsc12 C1(O)(CN(C(C(CC)OC)=O)C)CCN(C(c2sc(OC)nc2C)=O)C1 n1(CCOC)cc(C(=O)NC(C2CCN(C(C3CC3(F)F)=O)C2)C)ccc1=O c1(C(N2C3(CN(C(c4cscc4Cl)=O)C3)CC2)=O)cn(CCO)c(=O)nc1O N1(C(C(C)(C)S(C)(=O)=O)=O)C2CCC1CN(C(c1cn(C(C)(C)C)cn1)=O)CC2 N1(C(C=C(CCC)C)=O)CCC(O)(C(C)NC(C2CC2C2CCCC2)=O)CC1 c1(OCCOC)ccc2nc(NC(c3cncnc3-c3ccccc3)=O)sc2c1 Cc1ccc2c(c1)CC(C(=O)NCCOC1CCN(C(c3cscc3C)=O)C1)O2 CCC(C(=O)NC1(CCNC(=O)Cc2cncnc2)CCC1)C1CCOCC1 N1(C(c2cc(CCC)[nH]n2)=O)CC(CCNC(=O)CC2=CCCC2)OC(C)C1 C1(C(=O)NC(C2CCN(C(=O)C(CO)N(C)C)C2)(C)C)CCCN1C1CC1 C1(SC)CCCC1C(=O)N(CCC)C1CC1.c1(C(=O)N)nnsc1C(F)F N1(C(CN(C(C)C)C)=O)CCN(C(c2csc(-c3ccccn3)n2)=O)CC1CO C1(C)(C=O)CC(F)(F)C1.c1(C=O)ccn(CC)c1.C1(CCOC)CC1.C C=C(C)CN=C(NCC1COCCO1)N1CCc2ccc(Cl)cc2C1 C1(F)(C(=O)NCCOC(=O)C2CC2)CN(C(=O)CC2CCCO2)C1 N1(c2nccc(OC)n2)CC(C)CN(C(c2cc(C(F)(F)F)n[nH]2)=O)CC1C CC1CCC=C1C(=O)N1CC(CNC(=O)Cc2cc(O)nc(O)n2)C(C)(C)C1 N1(C(CC(CCC)O)=O)CCC(NC(=O)C(n2ccc(C3CC3)n2)C)C12CCC2 c1(CC)ccc([N+](=O)[O-])cc1C(=O)NC1CN(C(c2coc(C)c2)=O)CCC1F N1(C(=O)CC2OCCCO2)CCOC(CNC(C2(C(F)F)CC(F)(F)C2)=O)C1 N1(C(C2CCN(CC)C2)=O)C2CCC1CC(NC(=O)C1=CCCCC1C)C2 c1(CC(=O)NCC2N(C)CCN(C(CC=C)=O)C2)c[nH]c2cnc(Cl)cc12 CC1CN(C(=O)CCCC2CCC2)CC(C)N(C(=O)COC2CCN(C)CC2)C1 C(CNC(=O)CCc1nc(C)c(C)o1)(CC(F)(F)F)NC(C(CSC)O)=O C1(CC(=O)NC2CCCCO2)CCN(Cc2cscn2)C1 N1(C(CC2C(C)CCCC2)=O)CC(CNC(C2(CF)CC2)=O)C(F)(CO)C1 c1(OC)ccc(C)c(C(=O)NCC2CCCCC2)c1.C(c1cncs1)=CC=O N1(C(c2csc(Cl)n2)=O)CCCC(NC)C1.N12CCCC1CN(C)C(=O)C2=O Cc1ccc(C(=O)NCCC2(O)CCCN(C(C3(O)CCSCC3)=O)C2)c(C)n1 CC(C)CC(=O)C(=O)N(C1(C(=O)NCc2nn(C)cc2CO)CC1)C C(=O)(C(C)(C)C(F)F)NC(C(C)C)CCN(C)C(c1c(Cl)cnn1C)=O Cc1nc(C(=O)NC(CCN(C)C(c2ccn(C3CC3)n2)=O)c2cccs2)n[nH]1 C(CC(C)C(=O)N(C)CC=CC(N1CC(CC)(CO)C1)=O)=CC c1(C(N2CCC(O)C2)=O)cnc(O)c(C)c1.C1(C(=O)N)(CC)CC(C)(C)C1 N1(C(C2CC(=O)NC2)=O)CCC2(C1)CN(C(=O)CCc1cnco1)C2 C1(C(C)C)(CNC(=O)Nc2ccc(C(c3ccccc3)C)cc2)CCCC(=O)N1 C=CCC(CC=C)C(=O)N1CCN(C(=O)CC2CCSC2)C(CCC)C1 c1(N2CCC(N(C(=O)C=Cc3cnn(C)c3)CCC)C2)nc2cc(Br)ccc2o1 C1(c2nnnn2CCC2CC2)CCS(=O)(=O)CC1.CC12CCC(CO1)C2.C1CC1 c1(C(N2C3C(NC(C4OCCCO4)=O)C(C3)C2)=O)cc2ccc(Cl)cc2[nH]1 C1(C=O)CC(=O)CN(C=O)C1.c1(C(=O)OC)noc(C)c1C.C(C)(C)C Cc1cc(=NCC(C)N(C)C(c2ccc(Cl)nc2Cl)=O)[nH]c(CC2CC2)n1 c1(C(N2CCC(C(N3C(CC)CCC3)=O)CC2)=O)cccc(Br)c1F c1(C(=O)NC2CCC2)cnc(O)c(Cl)c1.C(=O)CS(=O)(=O)N1CCCCC1.C c1(C(N)=O)ccncc1NC(=O)CC1CC(NCc2cnc(Cl)s2)C1 C(=O)(CC(CC)SC)NC1CCN(CCCN(C(C2CC(CC)C2)=O)CC)C1 C1(NC(C2(C)CCN(C(C)=O)C2)=O)CCC(C)N(C(c2cc(O)ccc2N)=O)C1 C=C(C)C(C)(C)C(=O)NCC1CC(C)N(C(c2nccnc2Cl)=O)C1 C1(C)(COC)CCN(C(=NCC2CC2)NCc2ccccc2N2CCOCC2)C1 N(C(=NCCC1CCS(=O)(=O)CC1)N1CCC(n2cc(C)cn2)C1)C(COC)C C(=O)(C1=CCCCCC1)N(C1CCN(C(C(C(=O)OCC)OC)=O)C1)CC N1(C(CC(CC2CC2)NC(c2ncc(C)c(C)c2)=O)=O)CC2(CC(C)CO2)C1 N1(C(C(C)OCC2CC2)=O)CCC(O)(C)C1.c1(C=O)coc(C(N)=O)c1 C1(S(N)(=O)=O)(C(=O)NCCN(C(=O)C(C)CF)CC(C)O)CCCC1 N1(C(C(=O)NC(CC)C)C(C)CCC=C(C)C)CC(C)Oc2ccc(Cl)cc21 N1(CCC(=O)NCCOCCCNC(c2c(CC)con2)=O)CCCCCC1 N1(C(C(CCC)N(C)C)=O)CC2(CCCC2)C1C(=O)NCC1(O)CC2CCC1O2 C1(NC(=O)CC2CC3CCC2CC3)(CF)CCC(F)(F)CC1.C12CN(C1)C2=O C1(C2CCN(C(=O)C=CS(C)=O)C2)(NC(CCc2cn(C)nc2)=O)CC1 c1(CC(=O)N(C(C(CC)C)=O)CC(C)C)ccc(F)cn1 C#Cc1ccc(CC(=O)N(C2CN(C(C34CCC(CC3)C4)=O)CC2F)C)cc1 C1(CNC(CN(CCC#C)C)=O)CC(F)(CNC(C2CC2(C)C)=O)C1 N1(C(C2C(CC)N(C(c3ccnn3CCF)=O)CC2)=O)CCC2(CCC(O)C2)C1 C(CCS(C)(=O)=O)(C(=O)N1CCCC1C)OC.c1(C=O)cc(C)c(C#N)[nH]1.N Cc1c(C(N2CCC(C(C)(C)C(=O)NCCC3CCCCO3)C2)=O)ncn1C N1(C(Cc2cn(CC)nc2)=O)CCC2CN(C(c3cc[nH]c3C)=O)C(C)C12 N1(C(c2cc(C)cc(Br)c2)=O)CCC2(CC1)CN(C(=O)C(O)C1CC1)CCO2 c1(C(=O)NC2CC(NC(c3cncc(C#C)c3)=O)C2)cc2sc(Cl)cc2s1 C(CCC(C)C(=O)NCCCN(C)C(C1(C)CCOC1)=O)OC N1(C(C(C(=O)OC)C)=O)CC2CCC(C1)C(NC(=O)C1=NOC(C)C1)C2 C1(NC(CN(C)C)=O)CCC12CCN(C(=O)CN1CC(=O)NC1=O)CC2 S(=O)(=O)(c1ccc(Cl)s1)N(C(c1ccccc1)=O)Cc1ccns1 N1(C(c2ccc(C(F)(F)F)cc2)C)CCC(O)C(C=O)C1.C(C)(C)CCl.CC.N C1(NC(C(C)n2ccnc2)=O)CN(C(C23CCN(CC2)C3)=O)CC1F C1(C(N2CCC(C(=O)NC(C(C)(C)C)CO)C2)=O)CCc2ccccc2O1 C=CCC(C)(C)C(=O)NC1CCCOC1C1CCN(C(C2(O)CC2)=O)CC1 N1(C(C(C)=CC2CC2)=O)CC2(NC(c3cc(O)ncn3)=O)CCC1C2 C1(C(=O)Nc2cccc(OCF)c2)(NC(C(C=C)C)=O)CCCC1C N1(C(C2(CC(C)C)CC2)=O)CCC2(CCC2)C(NC(c2csc3nnsc23)=O)C1 c1(C(N2CC(C)(CCC(=O)NC3C=CC(CO)C3)C2)=O)cnnc(O)c1 S(=O)(=O)(c1ccc(F)c(C(=O)O)c1)N1C(C=O)CC1.N#Cc1cc(Br)ccc1.N CC1(C)CC=C(c2cccc(NS(=O)(=O)Cc3ccc(Cl)cc3)n2)CC1 N1(C(c2cc[nH]n2)=O)CCCCCC(Nc2ncc3c(n2)COC3)C1 Oc1cc(CN2CCCCC2c2ccc(O)nc2)cc(Br)c1 C(=O)(CCCCC(=O)NCC(C)(C)CNC(=O)CCC1CC1(Cl)Cl)NC c1(N(C(=O)CC#N)C(CN(CCCC)C)=O)cc2nc(C)cc(C(F)(F)Cl)n2n1 C(=O)(C#CC1CCOCC1)NC1CCN(C(c2oc(CC)c(C)c2)=O)C1C c1(SC)cncc(C(N2CCOC(C(C)NC(c3ccoc3Br)=O)C2)=O)c1 CCCCC(O)C(=O)NC(C1CCCC1)C.c1(C(N(CC(=O)N)C)=O)ccoc1 c1(OCCC)cccc2c1OCC2NC(N1CCCC(S(C)(=O)=O)CC1)=O C1(CN(C(=O)C)CC)CCCN(C(c2cnn(CCN)c2)=O)C1.C1CC1 Cc1cnc2cc(C(=O)N(C)CC3C4CN(C(=O)C(C)CF)CC34)nn2c1 C(=O)(C(CCCC#N)N1CCCCC1)NCCC(=O)OCC.C(=O)(N(C)C)N Cc1snnc1C(N1CCC(OCC(=O)NCC2CC2(F)F)C1)=O C#CC1CCCN1C(=O)CN(C(C1CC1C#N)=O)C1CC1 c1(C(=O)NCC(C)CN(C(=O)C(CCO)N(C)C)C)nc2ccccc2[nH]c1=O c1(C(N2CCC2)=O)ccc([N+](=O)[O-])c(C)n1.n1(CC)nnc(C(=O)NC)c1C N1(CC(C)C)N=C(C(=O)N2CCC(CC3CC3)CC2)CCC1=O N1(C(C#C)=O)CCCC1C(=O)Nc1cnn(-c2ccccn2)c1 C1(C(=O)NCC(C)N(C(=O)COC2CCOCC2)C)C(C)(C)C1(F)F N1(C(CCN(C(Cc2ccn(CC)n2)=O)C)=O)CCC2(CCC(O)C2)C1.C1CC1 c1(CN(C(C(N2CCC(C(CC)CC)CC2)=O)=O)CC)ccc2c(c1)CCO2 CC(C)CC(=O)N1CCC(CCNC(=O)C(O)Cc2ccccn2)C1 C1CC2(CCC2)CN1C(=O)C(C)(C)O.c1(CC)ccc(C=CC(=O)N)o1.C N1(C(c2cccc(OCCC)c2)=O)CCN(C(=O)C(=O)NCC(F)F)CC1C C#CCCCC(C)C(=O)N(CCCC(=O)NC(C)(COC)CO)C c1(CC)cc(C(=O)NC2CCCC2)no1.c1(CC=O)ccn(CC(F)(F)F)n1 N1(C(CN(C(C)C)C)=O)CC(C)N(C(c2ccnc(C(F)(F)F)c2F)=O)CC1C c1(C(C)C)cccc(CC(=O)NC2CC(C(=O)NCCc3cccnc3)C2)c1 C1(NC(C(C)OCc2ccncc2)=O)(CO)CCCN(C(c2sccc2F)=O)C1 c1(C(=O)NCC(c2cccc(C)c2)NC(=O)C(C)(C)C#N)nccc(Cl)c1C Cc1cc(CC(N2CC(NC(=O)CN3CCS(=O)CC3)CC2(C)C)=O)ccc1O N1(C(c2ccc(C(C)C)s2)=O)CC2CCCC(NC(=O)Cc3cnccn3)C2C1 CC1CCC2(CC1)OCC(CNC(c1cccc(-c3noc(C4CC4)n3)c1)=O)O2 CC(C)(C)CC(=O)NC1CC(NC(c2csc(CC(F)F)n2)=O)CC1O Cc1cnc(NC(=O)CC2CC(NCc3cccc(C(F)(F)F)c3Cl)C2)cc1F c1(C(N2CCC(N(C(C3CCCN(C)C3)=O)CC)C2)=O)cc2c(s1)CCCC2 C(N=c1[nH]c(N2CCN3CCCCC3C2)nc2c(F)cccc12)c1n[nH]c(=N)o1 N1(C(C2CCC(C)(C)OC2)=O)CCC2(C1)CN(C(=O)CC1CCCCC1(C)C)C2 N1(C(c2c(C)oc(C(F)(F)F)n2)=O)CCCC1(C)C.C1(C=O)CC1C(C)C.N N1(C(CCCC#C)=O)CCCC2(NC(=O)Cc3ccnnc3O)CCCC12 CC(CN(C)C(c1ccc(Cl)s1)=O)C(=O)N(CC(N)=O)C C(=O)(C#CC1CCCCO1)N1CCCC(CCNC(C2C3CCCC23)=O)C1 N1(CC(=O)NC(CNC(C(COC)N(C)C)=O)(C)C2CCC2)CCCNC1=O C1(CCNC(=NC)NCC(c2cc(F)ccc2F)C(F)F)COCC12OCCO2 C#Cc1ccc(F)cc1C(N1CCC2(C1)CN(C(=O)CC1(C)CC1)C2)=O c1(C(C)C(=O)NC2CCC(CNC(=O)C3=CCC3)C2)ccc(F)c(Cl)c1 c1ccc2c(c1)CCO2.C1(C2(O)CCC2)(C(=O)NCCSCC(=O)N)CC1 c1(C(=O)NC2CCCC(NC(C(C)C)=O)C2)cc(=O)c2ccc(Br)cc2o1 C1(C(=O)NCC2(CNC(C(C)(C)CO)=O)CCCC2)CCCCC1(C)C C1(CC(=O)NC2(CC(=O)NCCOCC)CC2)OCCCO1 C1(CC)CCN(C(C2COCCC2C)=O)C1CNC(c1sc(F)cc1C)=O C1(NC(c2c(C)n(C)nc2)=O)CC2CCC(C1)N2C(c1cnn2cccc2c1)=O c1(C(=O)NC(CN(C(=O)Cc2ccco2)C)(C)C)cnc2c(c1)NCC2 C1(NC(CC(CC)OC)=O)CC2CC(NC(=O)C(=O)NC(C)C)CC2C1 c1(C(=O)NCCCN(C(c2sc(Cl)c(Cl)c2N)=O)CC)cnc(C)cc1C Cc1nc(CC(C)C)c(C(N2CCCCC2C)=O)s1.C(=O)(C(C)N1CC(C)C1)N c1(C(=O)NC2CCN(CCCCC)CC2C)cc2c(C)ccc(F)c2[nH]1 C1(C(=O)NC2(C)CC=CC2)(CC)CCCN(C(=O)CCOC)C1 C#CCCCCCC(=O)NC1(CNC(=O)COC2CCCOC2)CC1 N1(C(C(CCC)CNC(c2cccc(CC)n2)=O)=O)Cc2cccc(C)c2C1 Cc1nnc2n1CC(C(N1CC(NC(C3SCCCS3)=O)C1)=O)C2 N1(C(CCNC(C)=O)=O)CCCCCC(NC(C2(Cl)CC2(C)C)=O)C1 c1(NC(C2CC(NC(c3ccc(F)nc3)=O)C2)=O)ccc(I)c(Cl)c1 c1(C(N(CCNC(c2cscc2CC=O)=O)CC)=O)cccn(C)c1=O.O c1(OCC(=O)NCCOCCCNC(CC2C(C)CC2)=O)cccnc1 CC(C(=O)Nc1ccccc1Cn1cccn1)S(=O)(=O)c1ccc(F)cc1 N1(C(c2cc(CCC)[nH]n2)=O)CC2(CC(CNC(c3sncc3C)=O)C2)C1 C(=O)(N(CCC(=O)NC1C2C=CC(C2)C1CO)OC)c1c(CC)oc(C)c1 C(CC(C)C)(C(=O)NC(C1CCN(C(C2CNC(=O)O2)=O)CC1)C)OC c1(OC)cccc(C(=O)Nc2c[nH]nc2C(=O)Nc2cncc(Br)n2)c1 C1(C(F)(F)F)(C(N2CCC(CCNC(CC3CN(C)C3)=O)C2)=O)CCCCC1 C1(CNC(C(C)C2CC2)=O)CCCCCN1C(c1cccc(Cl)c1Cl)=O C12(C(N3CCCC3c3ccco3)=O)CCNC1CCOC2 N1(C(c2c(Cl)cn(CC)n2)=O)CCN(C(C2(C)C=CCCC2)=O)CC1C C1(C(=O)NC(C)CCCNC(=O)C(C)O)CCC(C(F)(F)F)CC1 CN1CCC(C)(C(N2CCC(CO)C(NC(c3c[nH]ccc3=N)=O)C2)=O)CC1 Cc1cc(NC(C(N2CCCc3ccccc32)=O)C(C)C)c2c(c1)CCO2 c1(C=O)ccc2c(c1)C(C)CO2.C1(CC)CCOC1C(=O)NCC1CC1.N C1(NC(C2CC(OC)C(OC)C2)=O)CCC(C)N(C(=O)CCc2ccccc2)C1 c1(CC(=O)N(C)CC2(O)CCCN(C(C=C(CC)C)=O)C2)coc2ccccc12 N1(C(c2ccc(C)cc2F)=O)Cc2ccnn2CC(NC(C2CCC2(C)C)=O)C1 C(=O)(CCCC(=O)OC(C)(C)C)NCC(CC)C.C12(C=O)CCCC1C2(F)F CCCCC(C(=O)N1CC2(C(=O)NC3CN(C4CCC4)C3)CC1CCO2)C(C)C N1(C(C23CC(C)C2C3)=O)CCN(C(C2CCS(=O)CC2)=O)CC1CC(F)(F)F c1(N(C2CCN(C(C3CC(C)SCC3)=O)C2)C)cc(Cl)nc(C(F)(F)F)n1 c1(C(=O)N)cnn(C)c1N.c1(C(=O)OCC)cc(C(=O)NCCCCC)[nH]n1 C(=O)(CCCC(C)(F)F)NC1C(CNC(CC(=O)OCC)=O)C1 C1(CNC(C2(C)COCCO2)=O)CCCCN(C(c2sccc2Br)=O)C1 C=CCC(CC)C(=O)NC(CNC(C1(C)CC1)=O)C(C)C.c1cccc(Cl)c1 C=Cc1cncc(C(N2CCOC(C3CC3)C2)C(=O)NC2CC2)c1 C(=O)(C1CCCc2cccnc21)N1CC2(N(C(c3cnc(C)s3)=O)CC2)C1 C(=O)(C(C)C(C)(F)F)N1CC(C)(NC(COC(CC)C)=O)C1 c1(COC)cc(C(N2CCCCC2C2CN(C(=O)C)C2)=O)n(C)n1.C=O.N C(=O)(CC(C1CC1)C1CC1)NC1C(CNC(C2(C)CCC2)=O)C1 C(=O)(C1CCc2cc(F)ccc21)NC1CCN(C(c2cncc(C)c2Cl)=O)C1 C(=O)(C(C)C(=O)N1CCC(C(N2CC(S(C)=O)C2)=O)(C(C)C)C1)OC N1(C(CCCOCC)=O)CCOCC1.c1(CC(=O)N(C)C)cccc(C(N)=O)c1 C(C(C)CSC(C)(C)C)NC(C1CC(SCC)C1)=O C1(NC(=O)CNC(c2cscn2)=O)CCN(C(C2(F)CCCCC2)=O)CC1O N1(C(CCNC(=O)OCC)=O)CCC(NC(=O)CCC(C)SC)C(C)(C)C1 Cc1cc(C(=O)NCC2CN(C(=O)COC3CC=CC3)C2)sc1Cl c1(C(=O)NCC(C2CCCC2)N(C(C)=O)C)ccc(C(C)(C)C)nc1 c1(C(N2C(CNC(C3C(C)(CC)C3)=O)CC(F)C2)=O)ncn2ccccc12 C1(C(=O)NCCC(C)C)CCC(S(C)(=O)=O)CC1.c1(C=O)cccc(=O)o1.N C=C(C)C1OCCC1C(=O)NCCN(C(=O)CC1CCCN1C)CCC N1(C(=O)OC(C)(C)C)CC(O)CC12CN(C(C1CN3CC4CC3(CO1)C4)=O)C2 c1(C(N2CCC(NC(C3C(C(=O)OC)C3)=O)C2)=O)cc(Br)c(C)cc1C N1(C(C(C2CCOCC2)OC)=O)CCN(C(=O)CC(C)(C)OC)C2CC12 c1(C(C)C)cc(N2CC(NC(c3cnn(C4CC4(F)F)c3)=O)CC2C)ncn1 C(=O)(C(CC)C(C)(C)CC)NC1CCN(C(C=CCC)=O)CC1OCCC c1(NC(C)C)ccc(C(=O)NCCC(C)NC(c2cccs2)=O)cc1.C1CC1 C(=O)(C1CCC(=O)c2cccn21)N1CCC(N(C(=O)C=Cc2ccsc2)C)CC1 c1(NC(=O)NCC23CCCC2C3)ccc(-c2cc[nH]n2)cc1 CCCC(C(=O)NC1(C(N2CCCOC(CC)C2)=O)CSC1)C(C)C C12(C(N(CCN(C(C(CSC)O)=O)C(C)C)C)=O)CCC(N=[N+]=[N-])C1C2 C1(CCNC(COCCN(C)C)=O)CCN(C(=O)COc2ccsc2)C1 CC#CCCC(=O)NC(C)CCCNC(=O)C(C)NC(N)=O.C(CCC)S C1(C(=O)NCc2cccc(Cl)c2)CN(C(=O)C#CC2CC2)CCC1O c1(NC(=O)NCc2nc(COc3ccccc3)co2)csc2ccc(Br)cc12 CCCCC(COC)NC(C1CC(=O)N(c2ccccc2Br)C1)=O N1(C(COCc2onc(C)n2)=O)CCC(NC(=O)CC(C)(C)O)C(CO)CC1 N1(C(c2ccn(CC)n2)=O)CCC2(CCN(C(=O)CC3CCOC(C)(C)C3)C2)C1 C1(C(N2C(C(=O)N)CCC2)=O)CCC2(CC2)N1C(=O)C(C)c1ccsc1.CC c1(OC)ncccc1S(=O)(=O)N(C1CCN(Cc2cccc(Br)n2)C1)C c1(C(C)NC(CN(C(CNC(CCC)=O)=O)CC)=O)nnc(C)s1 c1(C(C(=O)NCC(CNC(=O)COc2ccsc2)O)F)ccc(F)cc1 C(=O)(C(Cn1cncn1)N1CCOCC1)NCc1n(C(C)(C)C)nnn1 CCCCC(CC)C(=O)N1CCCC1CNC(C1(c2ccno2)CCC1)=O N1(C(C(C2CN(C(C(C)OCC=C)=O)C2)O)=O)CC(CO)C1(C)C C1(C(=O)NC2C(CNC(C(N3CCOCC3)C)=O)CCC2)CC12CC(C)(C)C2 Cc1cc(C(=O)NCC2(O)CCC2)c(F)c(Br)c1.c1(C(=O)N)cc(C)no1 c1(C(NCCC)=O)cccc(S(C)(=O)=O)c1.C1(C=O)(C(N)=O)CCC1.C N1(C(c2c(OC)n[nH]c2)=O)CC(C(=O)NC(C2CCOC2)(C)C)C2(CC2)C1 c1(C(N2CC(O)(C(C)NC(c3cc(OC)no3)=O)C2)=O)nccc2cc[nH]c12 CN1CCCC2(CCN(C(c3ccco3)=O)C2)C1=O c1(N)cnccc1.C1(NC(C(C)NC(C(C)OCC(C)C)=O)=O)CCCC1 CC(C)C(C(=O)NCCC(C)N(C)C(c1csnn1)=O)N1CCCC1=O N1(Cc2cc(OC)c(I)cc2)CC(C(=O)NCc2cnc(Br)s2)CC(F)(F)C1 C(=O)(N=c1cc2ccccn2[nH]1)C1(OC)CCN(C(c2ccc(CO)s2)=O)C1 N1(C(c2c(C)oc(Cl)n2)=O)CC=C(C(=O)NCC2=CCCC2)CC1 N1(C(c2cc(CC)no2)=O)CCN(C(C2(C)CCCCCC2)=O)C2(CCC2)C1 C1(C(C)C)CCC(C(=O)NC2CC2NC(=O)C2CC2)CC1 Cc1nn(C(C)C)c(C)c1CN(C)C(=O)NC1(C(C)O)CC1 CC1CCN(C(c2cn(C)cn2)=O)CC1N(C)C(c1nccc(N)c1Cl)=O Cc1cn2cc(C(=O)NC3C4CC3CN(C(c3cn(CCO)nn3)=O)C4)sc2n1 C1(CC(=O)N(C(C)CCNC(c2cccn2C)=O)C)CC2(CCO1)CC2 C12(CNC(C3C(=O)NCCCC3)=O)CCCCC1N(C(=O)C=CBr)CC2 c1(CSC)nc(C(N2CCC3CC23)C(=O)NCc2ccco2)cs1 N1(C(=O)NCC(=O)Nc2ccc(-c3cscn3)cc2)CC2CNCC2C1 C1(NC(c2ccc(C)o2)=O)C2CCCN(c3cc(CC4CC4)ncn3)C2C1(C)C C1(C(C)C)CCC(C(=O)N(C)CC2CCN(C(C3CCC(C)C3)=O)CC2)C(=O)N1 CC1C2CC(C2NC(c2ncc(F)cn2)=O)N1C(=O)CC1CCC(=O)N1 c1(OC(C)C(=O)NC2CC(NC(c3ccc(F)cc3)=O)C2)ccc(F)cc1 c1(C(=O)OCc2ncccc2-n2cncn2)cc([N+](=O)[O-])ccc1.C(F)F c1(OC)c(Cl)cc(C(N2CCN(C(=O)C=CCCC(C)C)CC2CO)=O)cc1Cl c1ccc2c(c1)OCCC2NCc1cc2ncnn2cn1 N1(C(C)=O)CC2CCN(Cc3cc(Br)cc(C#N)c3)C2C1 c1(COC)c(C(=O)NCC2CC(NC(=O)CC)C2)cnn1C.C(C)=O c1(CC(=O)NCC2N(C(C3(C)C=CCCC3)=O)CCC2)cccc2cccnc12 Cc1cc(NC(=O)Cn2cc(-c3ncc(Cl)cc3C)nn2)cc(Br)c1 Cc1cccc(C=CC=O)c1.c1(CC(=O)NCC(C)C)nc([N+](=O)[O-])n[nH]1 C1(CC)CN(C(=O)C(C)(C)C2CCCCC2)CCC1NC(c1cc(C#N)c[nH]1)=O N1(C(Cc2nnc(C)s2)=O)CC2(CC(NC(=O)CC(=O)N)CO2)C1.CC(F)(F)F N1(C(c2ocnc2C(F)F)=O)CCC2C(CCCN2C(=O)C=Cc2ncc[nH]2)C1 c1(C(N2CC(CC(=O)NCC3CC4C=CC3O4)OCC2)=O)cc2cccn2cn1 C1(C)(NC(CN(C)CC)=O)CCCCC1C(=O)N(C1CC=CC1)C c1(NC(N=c2[nH]nc(SCCC(C)C)s2)=O)ccc2c(c1)CNC2=O CCC(=O)CCC(=O)N1CCCC(C(=O)NC2(C(N)=O)CCOC2)CC1 C(CS(=O)(=O)CC(=O)N1CCC2C(C1)CN2C(c1ccc([N+](=O)[O-])[nH]1)=O)OC N1(C(C=NOC)=O)CC2CC(NC(C3(CCO)CC3)=O)C2C1 N1(C(C(c2ccccc2)OC)=O)CCC2(CC1)CN(C(c1n[nH]cc1F)=O)C2 c1(C(=O)NC(CC)CNC(c2cnc(O)n2C)=O)ncc(Cl)cc1O CCC(COC)C(=O)N(CCCNC(C1COCCO1)=O)C CC(C)CCCCCC(=O)NCC1CC1CNC(c1csc(Br)n1)=O CN1CCc2ccc(C(N3CCN(C(=O)CC(F)(F)F)CC4(CC4)C3)=O)cc21 c1(C(=O)NCC2(F)CC(NC(CC(C=C)C)=O)C2)ccc2nccn2n1 N1(C(C(C)n2cccc2)=O)CCOCC(F)(CNC(c2ccc(=O)oc2)=O)C1 c1(-c2onc(C(c3ccc(Cl)cc3)OC)n2)cccc2ncsc12 c1(C(=O)NCCC2(O)CCN(C(c3n(CC)nnc3)=O)C2)cccc(Cl)c1.C Cc1cc2ncc(C(=O)NC(C)(CNC(=O)C(F)n3cccn3)C(C)C)cn2n1 C(=O)(C(C)(C)CC(=O)NCC(C)C)OCC.c1(CC=O)c(C)n[nH]c1C.N c1(OC)c(C(=O)NC2(C)CCOC2)ccnc1Cl.C12(CC(=O)N)CCCC1C2 C(=O)(C(C)(C)C(C)(C)C)NCCC1(O)CCN(C(c2nn(C)c(Cl)c2)=O)C1 c1(SCC(=O)NCCC2CCCN(C(=O)CC3(O)CCOC3)C2)cccc[n+]1[O-] c1(CN2CC3(C(C(=O)Nc4ccc(C(=O)OC)cn4)C3)C2)c(Cl)ccnc1Br c1(C(=O)NC(CN(C(=O)C(C)OC)CC)C)nc2ncccn2n1.C1CC1 c1(C(=O)NC2CCN(C(C(C=C=C)C)=O)C2C(C)C)ccc2c(c1)NC(=O)CO2 C(=O)(N=c1ccn(CCF)[nH]1)C1C(CNC(C(C)(C)OC(C)=O)=O)CCC1 Cc1cc(CC(N2CCCC2CC(=O)NCCNS(C)(=O)=O)=O)on1 c1(OC)cccc(C(CNC(C2(C)CCSCC2)=O)NC(c2ccoc2Cl)=O)c1 c1(CCC(=O)NC2CC(NC(c3cnc(C)o3)=O)C2)cc(Br)ccc1F N1(C(C2(CC)CCN(C(=O)Cc3ccsn3)C2)=O)CCc2nncn2CC1 CC1(C)CN(C(=O)CCC2CC2(C)C)CC2(CN(C(=O)C(C)(O)C3CC3)C2)O1 C1(O)(CCNC(C2CCC(CC)O2)=O)CCN(C(c2nnc(S)n2C)=O)C1 C(=O)(CC(C)C(C)(C)C)N1CCOCC(C(=O)NC(C(=O)OCC)CC)C1 C1(C(N(C2CCOC2)CC#C)=O)CC2(CCN(C(c3nnc(O)nc3O)=O)C2)C1 c1(C(C)C)cc(C(N2CCN(CCNC(C3CC4CC3C4)=O)CC2)=O)n(C)n1 C(C(N=c1ccnc(N2CCCN(C(C)(C)C)CC2)[nH]1)c1ccccc1)OC C1(C)(C(=O)NC(C)CCNC(c2cc(Cl)ccc2N)=O)CC(C(F)(F)F)=NO1 C(C(C(=O)N(C1CC2CCC1O2)C)C(C)C)NC(CCN(C)CC)=O C1(C(=O)NC2C(NC(C3CNC(=O)N3)=O)CCCC2)CC12CCC(F)(F)CC2 C1(NC(CCc2n(C)ncc2)=O)CCCC(NC(=O)C(C)(C)O)C1 CC1(CN2CC3C(Cc4ccccc4)C3C2)CCOC2(CCC2)C1 N1(C(C(CC)F)=O)CC2CC(NC(=O)CCCc3ccc(OC)c(OC)c3)C2C1 CCN=C(NCC1CC1C(F)F)N1CCCC(O)(c2ccc(Cl)cc2)C1 C1(NC(c2ccc(C(F)(F)F)[nH]2)=O)CC2CN(C(=O)C3=CCCCO3)CC2C1 C1(NC(CN(CCOC)C)=O)CC2CN(C(c3cnc4ccccn34)=O)CC2C1 CCC(CC)C(=O)N(CC(C)C)C.C1(CC(=O)N)CCN(C=O)C1.C(C)(C)C C1(CC=O)CCC(F)(F)CC1.c1(C(C)NC(=O)C=CCF)ccc(F)cc1.N c1(C(N(CCNC(C(C)(C)OCC)=O)C)=O)cc(N)c(Cl)c(O)n1 Cn1cc(Br)c2c(N3CCC(C)(C(=O)NCc4ccc(Cl)cn4)CC3)ncnc12 C1(CC(=O)NCC2(SC)CCC2)CC(F)CN1C(c1cc[nH]c(=N)n1)=O Cc1cc(F)cc2[nH]c(C(=O)NC3CC3NC(C3CCCS3(=O)=O)=O)cc12 C(=O)(NNc1cccc(F)c1OC)NCCOCP(OC)(=O)OC c1(CC)ccnc(N2CCCCC2)n1.C1(NC=O)CCCC1.C12(C=O)CCC1C2.N Cc1cc(NC(C2CC(F)CN2C(c2ccn(C(C)C)n2)=O)=O)c(C)cc1O C1(OC)CC(C(=O)NCc2ccccn2)N(C(=O)CN(C)C)C1.CC(F)F Cc1ccc(-n2nc(-c3cccc(F)c3)nc2C2CCC2F)cc1 C1(N(C)C(c2ccn(C3CC3)n2)=O)CCC2CN(C(c3cnc(N)cn3)=O)CC12 c1(NC(C(N2CCC(OCC)C2)=O)=O)cccc(C(C)(F)F)c1 CCCCS(=O)(=O)CC(=O)N1CCC(NC(c2c(C)cc(Cl)cc2C)=O)C(C)C1 C(=O)C(C)(F)C(=O)N1CCC(C(C)(C)C)C1.C1(C=O)CN(C(C)=O)C1.C C1(C(=O)NC(CNC(Cc2n(C(C)C)cnn2)=O)(C)CO)CC=CCC1C C1(C(=O)NC2C(C)(C)COCC2)CC2(CCN1C(c1ccc(=N)[nH]c1)=O)CC2 Cc1cc(=NCCN2CC3CC3C2)[nH]c(NC2CCN(c3cccnc3)C2)n1 N1(C(C2(CNC(c3c(C)noc3N)=O)CC2)=O)CCCC(O)(C(C)C)C1 C1(COC)CC12CCN(C(=O)Cc1ccccc1O)CC2 C1(C(=O)NC(C(C)NC(c2ccc(F)cn2)=O)(C)C)CCS(=O)(=O)C1(C)C Cc1cc(C(N2CCC2CNC(=O)CCc2cc(C)on2)=O)n2nc(C)cc2n1 c1(C(N2CC3(CC(CNC(c4n(C=C)ncc4)=O)C3)C2)=O)c[nH]c2nccc-2c1 C(=O)(C(O)CCS(C)=O)NC1C2CN(C(CCCCN(C)C)=O)CC1C2 c1(C(=O)NC(C(=O)NCC(C)(C)C2CC2)C2CCOC2)ncccc1Cl C(c1ccncc1)=C(C)C(N1CCOCC1CNC(=O)CCc1nc(C)no1)=O C(CCC(CO)NC(C1(C)CCNC1=O)=O)NC(C(n1ccc(C)n1)C)=O c1(C(N)=O)cc(C(=O)N(C2CCCC2)CCCNC(C2CCC(F)C2)=O)co1 C=CC1(CC(=O)NCCCOC(F)(F)F)CN(C(=O)CC2CCOCC2)C1 C1(NC(CN(C(C)=O)C)=O)CCCC12CN(C(c1ccc(C(F)(F)F)nc1)=O)C2 c1ccccc1.C1(C=O)OCCC1C(C)C.C1(C(=O)NC)(CSC)CCC1 c1(OC)cc(Br)cnc1C(N1CCC(C)C1CNC(c1ccc[nH]1)=O)=O c1(CC(=O)NCC2(F)CCN(C(C3C(OC)CC3)=O)C2)cc(O)ccc1 N1(C(c2ccc(C(C)C)cc2)=O)CCCCC(NC(c2cc(O)nn2C)=O)CC1 c1(N2CCC(C(F)F)(F)C2)cc(=NCCc2nnc3ccccn23)[nH]cn1 N1(C(C(CSC)OC)=O)CCC(C(N2CCC(C)(N(C)C)C2)=O)(CO)C1 CCCCC(C(=O)NCCCC(C)C)NC(N)=O.c1(C(=O)N)cnc(N(C)C)o1 N1(C(c2nc(C)sc2)=O)CC2C3CCC(C(NC(C4CC=CCO4)=O)C3)C2C1 N1(C(c2cc[nH]n2)=O)CCN(C(c2ccc(Br)cc2F)=O)C2CCCCC12 C(C)(C)(CC(=O)NCC(C1CCCCC1)O)NC(c1c(C)nns1)=O c1(C(C=O)C)cc(C)cc(F)c1.CCS(=O)(=O)N1CC(C(=O)N(C)CC)C1.N C1(NC(c2c(OC)csc2)=O)CC2C1CCN2C(c1ccsc1SC)=O c1(C(=O)NC2C(NC(=O)CCSC(F)(F)F)CCCC2)cc2n(n1)CCCC2O CCCC(=O)NCC(=O)NCC.C(=O)(CN(C)C(C)C)N(CC)C.CC CC1(NC(=O)C2=C(Cl)CC2)CCN(C(c2cc(-c3ccccc3)ns2)=O)C1 N1(C(COCCC=C)=O)CCC(C=C)(C(=O)N(C)Cc2cnc(C)s2)C1 CC1COCC(CC(=O)NCC2CC(C(=O)NCCN3CCNC(=O)C3)C2)O1 CCC(CC)CC(=O)N1CCC(CNC(=O)C(C2CC2)N(C)C)(OC)C1 C1(NC(c2cn(CCC)nc2)=O)CCN(C(C)C(=O)NC(N)=O)C(C)C1 C(=O)(CC(C)C)N(c1cnnn1C1CN(C(C)=O)C1)C(c1cncn1C)=O.C CCCC(C(O)C=O)NC(C1(CCN(C)C)CC1)=O.C(C(C)(C)C)=CC.N c1(C(COCCNCCC(=O)N(C(C)C(=O)OC)CCC)C)ccccc1 C1(C(=O)OC)CN(C(=O)CNS(=O)(=O)c2ccc(Cl)s2)C(C)(C)CO1 c1(C(N2CC(NC(C34CCC(CC)(OC3)C4)=O)C(C)C2)=O)cc2n(n1)CCCO2 c1(C(c2n(C(CC)(C)C)nnn2)NCC2(F)CCOCC2)c(F)cc(Br)cc1F C1(C(C)CNC(=O)CSc2ccncc2)CCN(C(c2ccnnc2S)=O)CC1 c1(N(CC(=C)C)C)nnc(Cc2csc(C)c2)n1CC1CC1 C1(NC(C2CCN(C(C(C)(C)CC3CC3)=O)CC2O)=O)CC2CCCCCC12 C(CN=c1c(C#N)c[nH]c2c(F)ccc(F)c12)OCCNC(C1CCN(CC)C1)=O C1(C(N2C(C)(COC)CC2)=O)N(C(=O)C(CC(C)(C)C)OC)CCCC1(C)C N1(C(c2cc(C)nnc2)=O)CCC2(NC(=O)CNC(=O)CC(F)(F)F)CC2C1 c1(CC(=O)NC(CNC(C(n2ncc(C)c2)C)=O)(C)CO)ccc(F)c(Cl)c1 CCC(C)C(C(=O)NC(c1ncc(C)cn1)C)N(C)C(c1ncccc1N)=O c1(C(CCN(C(=O)NCC(C)O)Cc2c(C)ccs2)O)cc2ccccc2[nH]1 C1(NC(c2cnc(C)s2)=O)COC2(CNC(=O)CC3CCCO3)CC1C2 O=C(C1=CC2CCCCCC12)NC1CN(C(C23CCC(F)(CC2)CC3)=O)C1 C1(NC(C=CCNC(c2c(C)nc(O)s2)=O)=O)(CO)CCCCC1C C(=O)(CC(O)CC(C)(C)C)N1CCC(C#C)(C(=O)NC(C)CC)C1 c1(C(=O)OCC(=O)NCc2ccc(CC)s2)cc(F)cc2ccncc12 CC1CCNC(=O)C1NC(=O)CN(C(c1ccc(N)cn1)=O)CC1CC1 N1(C(=O)NC(C)CN2C(=O)CCC2=O)CCN(CCC(C)F)CC1C CCC(C)CCCC(=O)N1CC(NC(=O)CCc2cnn(C)c2)CCC1C C1(C(N(C)CC2(NC(=O)CCc3cnoc3)CC2)=O)CNC(=O)CC1(C)C c1(C=O)c(F)c(C)cc(N)c1F.C(=O)(CC(C)CN(C)C)NCCC(=C)C.N N1(C(CNC(C(CC)C)=O)=O)CC(NC(c2cc(Cl)ns2)=O)CC12CCCC2 c1(C(=O)NC2(C(=O)NCCC=CCCC)CCCC2)cnn(C)c1C CC#CCCCC(=O)N1CC(CCNC(c2cccc(-c3nnc(C)o3)c2)=O)C1 CC(C)(C(O)CO)NC(c1ncoc1CNC(=O)Cc1ccon1)=O c1(CC)cc(C(=O)NCC(C)NC(c2cnc(C)cc2C)=O)ccc1F C(C(=O)NNC(=O)NCc1ccc(-c2ccco2)cc1F)c1c(CC)cccc1 C1(C(N2CCCC(O)C2)=O)CC2CCC1N(C(=O)Cc1cscn1)C2 C1(COC)CN(C(=O)C)C1.c1(C=O)csc(C2CCCO2)n1.CCN(C)C CC1(C)C(NC(=O)Cn2cc(-c3cnc(Cl)s3)nn2)C1CO C(=O)(C1=CCC2CCC1N2C(=O)CC(C)C)Nc1c(C)nc(Cl)cc1.C(N)(=O)N C1(CC)CN(C(c2ccc(NC(C)=O)cc2)C(=O)NC2CC2)CCO1 O=C(CC(F)(F)C(F)F)NCC(O)C(N1CCCC(CO)C1)=O c1(C(=O)NC2COCCN(C(Cc3cc(C)on3)=O)C2)cccc2ccsc12 C(=O)CS(=O)(=O)c1ccc(Cl)cc1.C(c1cocn1)=CC(=O)NC1CC(C)C1 CS(=O)(=O)c1cc(NCC2CCCN2C(C2CC23CCOC3)=O)ncn1 Cc1ccc(S(=O)(=O)CC(=O)N2CCOC3CN(Cc4csc(C)n4)CC23)cc1 CC1CN(C(c2c(C3CCC3)cnn2C)=O)CC1NC(=O)CCC1CC1(Cl)Cl c1(CC(=O)N(C(C)CCNC(C2Cc3nncn3C2)=O)C)nc2c([nH]1)CCCC2 c1(C(N2CCN(C(C=C(CCC)CCC)=O)CC2)=O)cc2n(n1)CCNC2=O c1(OC)cc(-c2cn(CCOCCNC(c3ccccc3)=O)nn2)sn1 C(=O)(C1=NOC2COCC12)N1C(C(=O)NC(CO)CCO)CCC1 c1(N(C2CCC2)C(C23CC2CCCN3)=O)ccc(C(F)F)cc1 c1(OCC)ccnc(N2CCCC2CNCc2ccc(C(F)(F)F)cc2)n1 O=S(=O)(c1ccc2nc(N3CC4CC(O)CC4C3)sc2c1)NC1CCSC1 c1(NC(c2c(COC)noc2)=O)sc(-c2cccs2)nc1C N1(C(C)=O)CSCC1C(=O)NC(C)(C)C.C1(C(C)(F)F)(C=O)CCC1.N N1(C(CCS(CC)=O)=O)CC2(CCCN(C(=O)CNC(C)(C)C)C2)C1 C(=O)(C#CC1CCCCO1)NCC1CCN(C(CN2CCN(C)CC2)=O)C1 C1(CNC(c2c[nH]cc2C2CC2)=O)CCN(C(=O)CC2CCCC2(F)F)CC1 Cn1cc(CC(=O)NC2(CCCCNC(=O)Cc3ccnn3C)CC2)nn1 C(CC(CNC(C1SCCCS1)=O)NC(c1c[nH]nc1-c1ccsc1)=O)OC C1(CC(=O)N(C(C=C)C)C)C2CN(C(=O)CP(C)(C)=O)CC12 C1(C(=O)NCC(C(=O)OC)O)CSCCN1C(c1n[nH]cc1Cl)=O N12CCN(CC1)CCC(=O)OCCC2.C(=O)C(F)(F)F.CCCC.CCCSCC c1(C(=O)Nc2cncc(C(=O)OCC)c2)c(C)cc(C)nc1OC1CCC1 C(=O)(C(C)SCCCC)NCC1C(CC(=O)NCCCC)C1 CC1CN(C(=O)COc2cn[nH]c2)CCCN1C(=O)C=Cc1cccnc1 N1(C(C2CCC(N(C)C)C2)=O)CCC2C(C1)NC(=O)CCN2C(c1ccoc1)=O CC(C)(C)CC(F)C(=O)N1CCCC1C=CC(=O)NCCCN1CCCC1 c1(C(NC(=O)CN2CCOCC2)=O)ccc(C(F)(F)F)cc1I.C1(O)CNC1.C C(C)(C(F)(F)C(F)F)NC(CCCOc1cccc(OC)c1)=O C(c1ccc(F)c(F)c1)=CC=O.CC1(C)C(NC(=O)C(N)=O)CC1C.N Cc1cc(F)c(CNC2CC(C)(NC(=O)OC(C)(C)C)C2(C)C)nc1Cl c1(-n2ncc(C(=O)NC(CCNC(C3C(C=C)C3)=O)C)c2)ccc(OC)cc1 CCC(C)C(C(=O)NCCCN(C)CCc1scnc1C)N(C)C c1(OC)cc(C)sc1C(=O)NCC(CCNC(c1nccn1C)=O)OC N1(C(C2(COC)COC2)=O)CCC(C)C(NC(c2ccc(Cl)cc2C)=O)C1 N(C1CCCc2ccccc21)(C(=O)CC12CC(C1)C2)C1CC1 C1(C(=O)NC2CC3(CC(C)C3)C2)COC2(CCN(Cc3ccccc3)CC2)C1 c1(OC)ncc(C(=O)NC(CNC(=O)C)C(C)C)cn1.CCN(C)C.S N1(C(CN(C)C)=O)CCCC1CN(C)C(C1(CC(=O)N)CCCC1)=O.C1CC1 c1(C(N(C2CC2)CC2(NC(=O)CSc3nc[nH]n3)CC2)=O)scnc1Cl c1(C(=O)NCCCC)ccc2cc(C(=O)NNc3cccc(C(F)(F)F)n3)[nH]c2c1 C(=O)(C1CCc2c[nH]nc21)N1CC(NC(CCC(=C)C)=O)(COC)C1 CCC(CC)C(C)C(=O)N1CCCC1C(C)NC(=O)CN1CC(=O)N(C)C1=O C1(C(=O)NC(C(=O)OC)C2CC2)CC2(CCC2)C1.c1(C=O)ccccc1 C(=O)(C(O)C(C(C)C)OC)N(CCC(=O)NCC1CCCN(C)C1)CC C1(C(COC)(C)C)CCN(N(Cc2ccnn2C)C2CC2)CC1 c1(C(N(CC(C)N(C(=O)CC2COCC(C)(C)O2)C)C)=O)cnn2c1OCCC2 CCCCC(C)C(=O)N(CCCCN(C)C(C1(C)CNC(=O)C1)=O)C C(=O)(C1CCCc2scnc21)N1CC(CNC(c2c(C)cno2)=O)N(C)CC1 CC(C)(C#N)CC(C(=O)NC1CC1)N1CCCC1c1c(F)cccc1F c1(OC)ccc(-c2nc(CC3CCCN(C)C3)n(CCCO)n2)cc1Cl N1(C(C2CCCC(OC)C2)=O)CCN(C(c2ccc(C3(C)CC3)cc2)=O)CC1C c1(NC(C23CN(C(C4(C)COC(=O)N4)=O)C(C2)C3)=O)ccc2occc2c1 C(=O)(CCC(=O)c1cccnc1)NCC1CN(C(CC2ON=C(C)C2)=O)C1 C=CCC(F)(F)C(=O)NC1CC(NC(c2ccnn2C)=O)C1 c1(C(N(C(C)CNC(=O)C2=CC(O)CCC2)C)=O)cc2cc(F)cc(F)c2[nH]1 N1(C(C2C(C)=CCS2)=O)CC2CCCC(CNC(=O)CCCC3CCCO3)C2C1 C(CCCC(=O)N1CCC(OCCNC(C2NC(=O)OC2C)=O)C1)OC C1(NC(C2CC2(F)F)=O)CC2CC1N(C(c1cc[nH]c1-c1ccccc1)=O)C2 c1(C(=O)NC2CN(C(C3C(C)C3)=O)C3(C2)CCC3)ccnc2c(C(N)=O)cnn12 N1(C(CC)=O)CC2(COCC2)C1.C1(CS(N)(=O)=O)(C=O)COC1.CC(=O)N N1(C(c2nc(OC)nc(O)c2)=O)CC2(CCN(C(c3nnc(C(C)C)s3)=O)C2)C1 CCCS(=O)(=O)C(C)C(=O)N(CCCNC(c1ccccn1)=O)C.C(C)(=O)N C1(NC(N(CCOCC=C)C)=O)CCc2ncsc2C1 C1(F)(CNC(C2C(C)CC2)=O)CC(CNC(c2cccs2)=O)C1 N1(C(C2C3C(NC(CNS(CC)(=O)=O)=O)C4C(C3)C42)=O)C2C=CCC1CCC2 c1(SC)cccc(C(=O)NC(C)CCNc2cc(-c3cccc(Cl)c3)ncn2)n1 CCC(C#N)C(=O)N1CC(NC(=O)CC(C)(C)OC)C(C)C1 CC1COCCN1C(=O)Oc1cccc(OC2CCC2)c1 C(=O)(C1=NN(C2CC2)C(=O)CC1)NC(CCCNC(c1c(C)scn1)=O)C O=C(C#CC1(C(F)(F)F)CC1)NCC1CN(C(=O)CCN2CCC(F)C2)C1 C1(C(=O)Nc2ccc(OC)cc2F)C2CC(O)C(C2)N1C(c1cscn1)=O N1(C(C2(F)CCN(C(CC3C=NN(C)C3=O)=O)C2)=O)CCC2(CCC(O)C2)C1 C#Cc1ccc(C(N2CCC(C)C(CNC(=O)Cc3ccc(O)nc3)C2)=O)cn1 Cc1cc(F)ccc1CNC(C1CC(C)CN1C(c1ccn(C)n1)=O)=O CC1CCC(C(=O)N(CC(C)NC(c2ccn(C)n2)=O)C)C1 c1(NC2C(C)CN(C(c3ccncn3)=O)CC2)ncnc2sccc12 C1(C)(C=O)CCNC(=O)C1.CC(C)(C)C(=O)N1CCC1.CC(C)(C)OC=O N1(C(COCP(C)(C)=O)=O)CCC2CCN(C(C3CC(Cl)(Cl)C3)=O)CC2C1 C1(CNC(C(C(C)C)CO)=O)CC2(CCOCC2)CN1C(=O)CC(O)C1CC1 CC1CCN(C(=O)Cc2ccn(C)n2)CC1N(C(=O)C1=C(Cl)CCC1)C CCCCCC(C)(C)C(=O)NCC(c1ccccc1F)NC(=O)CCC1CCC1 C(=O)(CCC(C)(C)F)N1C(CNC(C2C(C)C2)=O)C(C)CC1 N1(Cc2cc(Cl)c(OCC#C)c(Br)c2)CC2CC3(CCC3)C2C1 c1(CC)c(C(=O)NC(C2(O)CCCCC2)C(N2CC=CC2CF)=O)nnn1C Cc1c(C(=O)NCCCC2CC2)c(C(F)(F)F)nn1C.C1(CC=O)CCCC1 CC1(C)CC(C(=O)NC2(c3ncccn3)CC2)CN(C(C2(C#N)CC2)=O)C1 Cc1c(C(=O)NC(C)CN(C(=O)CCC(F)F)C)[nH]c2ccc([N+](=O)[O-])cc12 N1(C(C(CC)(C)C#N)=O)CCCC(O)(CNC(C2(N3CCCC3)CCC2)=O)CC1 N(C1c2ccccc2CC1NC(c1cc(Cl)on1)=O)C(=O)CC1CC2(CCC2)C1 C1(S(C)=O)(CNC(C(c2ccco2)NC(COC)=O)=O)CC1 C#CC(CC)(CC)NC(=O)CCC1(C)CN(C(c2nnn(CC)c2C)=O)C1 C1(NC(=O)C(F)CC2CCOCC2)CCCCC12CCCN(C(=O)C=C(Cl)Cl)C2 C(N=c1[nH]cncc1I)C1(F)CC(NC(C2CCN(C(=O)NC)CC2)=O)C1 Cc1c(C(=O)NC(C)C(C)(C)NC(=O)CCn2cccc2)oc2c(F)cccc12 CN1CCC(O)(CC(N2CC(N3CC(NC(=O)C4=CCCS4)CC3=O)C2)=O)CC1 Cc1ccc(CNC2(c3nnnn3C3CC3)CC3(C2)OCCO3)c(=O)n1C N1(C(CC2C(C)C2)=O)CCOC2(CCC(NC(=O)COCC3CCC3)CC2)C1 C1(C(N2CCCC(NC(c3cnns3)=O)CCC2)=O)COc2cc(Cl)ccc2C1 N1(C(CC2(C(=C)F)CCC2)=O)CCC(O)(c2cn(CC(C)O)nn2)CC1 C(=O)C1=CCCCO1.c1(C(N(C(C)C2CC2)C)=O)cn(C)nc1-c1cccs1.N n1(CC(=O)NC2(CC)COC2)ncc2ncccc12 Cn1nnc2ccc(C(N3CC4CC(NC(c5coc(Cl)n5)=O)CC3C4)=O)cc12 N1(C(CC2CC(F)(F)C2)=O)CCCN(C(=O)CN(C)C(N)=O)CC1.CCO c1(CC)[nH]nc(C(=O)NCc2cncc(C(N3CC(C)C(C)C3)=O)c2)c1C c1(C(N2C3C(NC(C(C)N(C)C)=O)C(C3)C2)=O)cc(=N)[nH]c(Cl)n1 c1(C(N2CCC(NC(c3cc(O)nc(O)n3)=O)C(F)C2)=O)cc2cnccc2o1 c1(C(C(=O)NCC=C)N(CC(C)SC)C)cc(C2CCC2)[nH]n1 Cc1cccc(C(=O)NC2CC(NC(C3CCCCC3C)=O)C2)c1O CCC(C(=O)NC1CCC(CC(N2CCC2(C)C(=O)NC)=O)C1)n1cncn1 c1(C(=O)OC)sccc1S(=O)(=O)NC1CCCC1.c1(C=O)ccn(C2CC2)n1 O=C(C(O)C1CCc2ccccc21)N1CCC(S(=O)(=O)C(F)F)C1 C1(C(=O)OC)CC(C)CN(CC(=O)NC(=O)NC(C)CC(C)C)C1 c1(C(N(C(C)CCNC(C2CC2CF)=O)C)=O)cc(C#N)ccc1Cl C1(NC(C(Cn2ccc(C)n2)C)=O)CC2(C1)CN(C(C1CCCC1F)=O)C2 c1(CC(=O)NC(C)C(C)NC(C2CCCCC2O)=O)n[nH]c2ccccc12 C1(NC(C2N(CC)CCCC2)=O)CN(C(c2cc([N+](=O)[O-])c[nH]2)=O)CC1C1CC1 N1(C(c2nn[nH]n2)CC)CCC(O)(COCc2nnnn2C2CC2C)CC1 CCCC(C(=O)OC)C(=O)N1CC=CC(C(=O)NCC(C)(C)OC)C1 c1(CC(N)=O)ccccc1CC(=O)NCCC1CCN(C(C2CCC(F)C2)=O)C1 C1(CC(N2C(C)CC2(C)C)=O)CC2CCC1N(C(=O)OC(C)(C)C)C2 N1(C(C(C)=C(C)C)=O)CCN(C(c2cc(C3CC3)[nH]n2)=O)CC1CO n1(CC(=O)NCC(CC=C)NC(c2cn(CC)nn2)=O)c([N+](=O)[O-])cnc1C C(C(F)(F)CCC(=O)NC1CCOC1(C)C)n1cc(CCN(C(C)(C)C)C)nn1 c1(C(=O)NCC(C2CCCCN2C(=O)CC)(C)C)cncc(O)c1.C(N)(=O)N N1(C(CC=C=C)=O)CC(C)CCC1C(=O)NC1(C)CC(N(C)C)C1 N1(C(C(C)CSc2ccccc2)=O)CCC2(NC(=O)C=CCO)CCCC12 Cc1ccc(S(=O)(=O)C2CCCCC2NC(=O)Cc2cnoc2)cc1 CC(F)(F)CCCC(=O)NC1CCCN(C(c2ccccc2NC(N)=O)=O)C1 C(=O)(C(C)(C)CCCNC(c1ccn(C(F)F)n1)=O)NCCc1ncn(C)n1 C1(CCNC(CNC(C)=O)=O)CC(F)(F)CN1C(C1CCC(C)(C)OC1)=O C1(NC(C2C(CC)C2)=O)CC1C1CCCN(C(=O)C(C)=O)C1 c1(CC)cc(N)c(C(N2CC(CNC(c3ccoc3)=O)C(C)C2)=O)cc1F.C C1(NC(=O)CC2(CNC(C3CC34CC4)=O)CC2)CCCCC12CC2 C1(C2(NC(C3CC3F)=O)CC2)CCCCN1C(=O)CC(C1CC1)C1CC1 C(=O)(C#CC1CCCC1)N(C(C)C(=O)NCc1cc(C)ccc1F)CC c1(OCCC(=O)NCC2CC(O)CN2C(=O)CSC(F)F)ccc(F)cc1 c1(C(N(C2CCCN(C(=O)C3=NNC(C(F)(F)F)C3)C2)C)=O)ncc(Cl)cc1F C1(NC(c2cc(Br)n[nH]2)=O)CC12CCN(C(=O)CC1CCCC1O)CC2 CCC(C)C(CC(=O)N1CCCC(OC2CC2)C1)NC(c1nocc1C)=O c1(CC(=O)N(c2c(OC)ccc(Cl)c2)C)ccccc1S(C)=O CC(C)C(O)C(=O)NCCCNC(C1COCCN1CC(F)F)=O C1(NC(C2C(C#C)C2)=O)CCCCN(C(c2ccc(Cl)cc2SCC)=O)C1 C1(N(C(c2cnccc2)=O)C)CC(C)CC(C)C1.C1(C(=O)N)(OC)CC(C)C1 C(=O)(C(C)S(=O)(=O)C(C)C)N1C(CC)CCC1.c1(SC)ccc(C(=O)N)cc1 N1(CC=O)CC(=O)NC1=O.Cn1cncc1CC=O.C(C)(C)Cn1cccn1.N c1(C(N2C3CC(NC(C4(CC=C)CC4)=O)C(C3)C2)=O)ccc2scnc2c1 N1(C(CC2(OC)CC2)=O)CCC(C)N(C(=O)COC(F)(F)F)CC1 Cc1nc(C)c(CC(=O)NC(C)CCNC(C2(C(C)C)CCC2)=O)s1 C(=O)(CCP(C)(C)=O)N1C(C(=O)NCCc2n(C)c(=O)on2)CCC1C(C)=O c1(C(C(=O)NCC2CCCO2)N(C(CC)C)CCSC)cnc(C2CC2)[nH]1 c1cnn(C)c1Cl.c1(CC)ccc(C(=O)N(C2CCN(C(=O)CC)C2)CC)[nH]1 C1(C(N2C(CCNC(C(C)(F)F)=O)CSCC2)=O)Cc2cccc(F)c2O1 c1(SCC)cccc(C(N2CCC(NC(=O)C(C)OCOC)C2C)=O)c1 N1(CC)CC(C(N2CCN(C3CCCN(C(=O)C(C)(C)F)C3)CC2)=O)CCC1=O c1(NC2(c3onc(C)n3)CC2)ccc(CNC(=O)OC(C)(C)C)cc1Cl N1(C(c2ccc[nH]2)=O)CC2CC2C1.C(=O)(CCC1CC1(C)C)NC(C)(C)C.C C1(C#CC(=O)NCCCCC(CO)NC(=O)Cn2ccc(C)n2)(CC)CC1 N1(C(=O)CC2CCC(C3CC3)O2)CCC(N=c2[nH]nc(-c3ccccc3)o2)C1 C1(NC(C2C(=C)CC2)=O)CCN(c2ccnc(C#N)n2)CC1C c1(NC(C(N2CC(CC)(CC)SCC2)=O)=O)ccc2c(c1)CCO2 N1(Cc2ccc(NC(CN(C(C)=O)C)=O)cc2)CCCN(S(=O)(=O)N(C)C)CC1 C1(CC)CCCC(NC(c2nnnn2-c2ccccc2C)C2(CC#N)CC2)C1 c1(C(CNC(C2CC2F)=O)NC(c2cnccc2Cl)=O)ccc(O)cc1 C(=O)(C(C)S(N)(=O)=O)N1CCCC(CNC(c2cc(C)c(C)[nH]2)=O)C1 C=CCC(CC(=O)NCC(C)(C)CC=C)NC(C1CC1OC(C)=O)=O C(=O)(C(F)C(=O)NC1CC1CNC(c1cccnc1OC)=O)OCC c1(OCC)ccc(NC(=O)NC(CC(C)C)C2CC2)cc1 C1(C(C)NC(C(F)=CCC)=O)CCCN(C(c2cncc(OC)n2)=O)C1 C1(C(=O)OCC)OCCNCC1N(C(C)C(C)(C)C)C(c1cncnc1)=O C=C(C)CC(C(=O)N(CCCCC)C(C)C)NC(C)=O.C(=O)CC.C(N)=O C(C(C)C(C)(F)F)NC(C1(NC(C=C(COC)C)=O)CC(F)C1)=O C(=O)(C(O)CCS(C)=O)NC(C(C)C)CCN(C)C(C1CC2CCC1CC2)=O c1(C(N2CCCCCC2C(=O)OC)C(=O)NCCC)ccc(Br)c(F)c1 C1(NC(C(CC)n2ccnc2)=O)CCOCC1NC(c1ccc(SC)cc1)=O C1(C(C(=O)N(CCCC)CCCC)(C)C)CCCN(C(C2C3CC(=O)CC23)=O)C1 C1(N2CC(C=O)C2)CCOCC1.c1(C(=O)N(CC(O)C)CCO)coc(Br)c1.N C#CC1CN(C(=O)C(CO)NC(=O)CCN(CC)CC)CC1O C(=O)(CC(C)C(=O)N1CC2(C(=O)NC3(c4ncc(C)o4)CC3)CC1CO2)OC CCC(CC)C(C)C(=O)NCCC1CCCN(C(c2cncc(Cl)c2)=O)C1 N1(C(C2C(NC(COC(C)C)=O)CCCC2)=O)C(C)CCCC1C O=C(CCc1cn[nH]c1)NCCC(=O)N1CCC1C1CCCC1 C1(NC(C(C)OCC)=O)CCCCC1C.C(=O)C(C)(C)C.C(=O)CC.N c1(C(=O)OC)c(Cl)nc[nH]c1=NCC1CCCCN1C(c1cccnc1CO)=O C12(C(=O)Nc3c(C(C)C)ccnc3)CCC(N)(CC1)C2 Cc1nnc(CC(=O)NC(C)C(CO)NC(c2coc(Br)c2)=O)o1 C(=O)(CCC(C)(F)F)NC(CNC(CN(CCOC)C)=O)C c1(C(N2CCN(C(CC3CCN(C)C3)=O)CC2)=O)c[nH]cc(F)c1=O c1(CNCC2CCCC2)nccn1CCC1CCCO1 c1(C(=O)N)cn(C)nc1C(C)C.n1(CC#C)cccc1C(=O)NC(C)CC C1(CNC(C(C)c2ccsc2)=O)CCN(C(C2(C#N)CCCC2)=O)CC1C1CC1 CC1CCCC(C(=O)NCCCCCCNC(=O)CC2CC=CC2)C1 c1(OC)ccc2c(c1)CC(C(=O)NCCN1CCC(N)C1)O2 c1(C(=O)Nc2nnc(N3CC(C)(C)C3c3ccco3)s2)c(O)cccc1F C1(NC(=O)C=C2CCCC2)C2CC3CN(C(C4CC5(CCOCC5)C4)=O)C1C3C2 c1(CC(=O)NC2C(NC(c3c(C)scc3)=O)COC2)ccc(-n2ccnc2)cc1 C(c1ccc(F)c(F)c1)=CC=O.c1(C(c2cc(F)ncn2)=O)ccc(F)cc1F N1(C(c2cnc(C)s2)=O)CCC(C(=O)NCCn2ncnn2)C12CCC2 C1(CNC(C2C(C)C2)=O)C(C(=O)N(CC(F)F)C)C1(C)C c1(C(N2CC(COC)C2)=O)c[nH]c2ccc(F)cc12.C1(C=O)CC(CCO)C1.N n1(CCC)nnnc1C(c1cnccn1)NC1(C(=O)N(C)C)CC1 N1(C(COc2cccc(CC=C)c2)=O)CC2CN(C(=O)C(C)CC=C)CCC12 c1(C(CC(=O)NCC2(O)CCN(C(=O)CN3CCOC3=O)C2)O)cccc(F)c1 n1(CC)nc(C)cc1C(N1CCOC(c2cn[nH]c2)C1)C(=O)NCCSC Cn1cc(C2=NOC(C(=O)NCC(C)(C3CC3)NC(C3CCOC3)=O)C2)cn1 CC(C)CS(=O)(=O)CC(=O)NCC1CCC1(C)C.C1(CC=O)OCCC1(C)C C1(CNC(C2C(C)CC2)=O)CCC(NC(C2CCCN(CC(F)F)C2)=O)CC1 c1(NC(C2CCCN(C(c3ccccc3C(F)(F)F)=O)C2)=O)cc(Br)cc(Cl)n1 C1CC2CC(C1)N(C(=O)C=C1CCC(C)CC1)C2.c1(CC)ccc(C(=O)N)o1 N1(C(Cc2nc(C(C)C)sc2)=O)CCC(NC(c2ccc(N)cc2Cl)=O)CC1C CC1=C(C(=O)NCC2CC(F)(F)CO2)C(C)(C)CCC1 c1(C(=O)NC2CN(C(CCC#C)=O)CC2O)cc(OC)nc(F)c1 N1(C(C2(C(N)=O)CC2)=O)CCC(C(F)C(=O)NC2(C(O)CO)CC2)C1 c1(OC)ccc(C(N2CC=CCC2C(N2CCC(OCC(N)=O)C2)=O)=O)nn1 C(=O)(C1CNC(=O)c2ccnn21)N(CCN(C(CCN(CCC)C)=O)C)CC.O Cc1cc(C)c2c(c1)N(C(c1csc(C)c1C)C(=O)NC1CC(F)(F)C1)CC2 C(=O)(C1OCCn2ccnc21)NCC(C1CCN(C(c2ccns2)=O)CC1)(C)O C12(C(N3C(CNC(c4cc(C)n(C)n4)=O)CC3)=O)CCCC1CC(=O)CC2 CCCC(C(O)C(=O)N)NC(=O)C(=O)NCC1CC1.c1ccc(C)cc1F.C c1(C(=O)NCC(CC=C)NC(C2(CF)CC(F)(F)C2)=O)ccncc1NC CCCC(C)(CCC)C(=O)N1CCC(CN(C(C2CCCC2SC)=O)CC)CC1 N1(C(=O)NCCC2CC2C2CC2)CCc2cc3c(cc2C1)CCCC3 c1(C(=O)NCC(C)N(C(C(C)O)=O)CC)ccn(CC=O)c1.C(C)(C)C C1(NC(C(CCC)C)=O)CCN(C(c2ccccc2)=O)C1(C)C N1(C(CC2C(NC(c3ccc(Cl)o3)=O)CCC2)=O)CC2CCC1CC2 N1(C(C(C)=CC2CC2)=O)CCC(C(C)CNC(c2ccnc(CO)c2)=O)CC1 N1(C(C2CC(C)(C)C2)=O)CC(O)CC1C(=O)NC1CCN(C2CC2)C1 S(=O)(=O)(c1ccc(Br)cc1NCCc1cc(C2CC2)no1)NC1CC(=O)NC1 N1(C(c2cccc3nsnc23)=O)CC2(CCOCC2C(N2CCCCC2)=O)C1 C(CC(=O)NCCn1ncnn1)(C(F)(F)F)NC(C=C(C)C(C)C)=O C=CC(C)CC(=O)NCC1C(C(=O)NC(C2(OC)CCC2)C)C1(C)C N1(C(C2C(CCOC)C2)=O)CC2(NC(=O)C(c3ccc(Cl)s3)C)CCC1CC2 N1(C(CC2(NC(C(C(CC)C)O)=O)CC2)=O)CC23CCC2(COC3)C1 Cc1cc(C(=O)NCc2ccccc2CN(C)C(C2CNC(=O)C2)=O)ccn1 c1(C(C)NCC2CCCN2C)ccc(I)cc1O c1(C(N2C(C(N3CC(C)(C)C3)=O)COCC2)=O)c(F)cccc1F c1(CC)nccnc1C(N1CCC(NC(=O)C(c2ccc(C)cc2)=O)C1)=O N1(C(c2ccc(CC)[nH]2)=O)CCN(C(c2ncncc2F)=O)CC1C C(=O)C(C)CCN(C)C.C=C1CC(C(=O)NCc2conc2)(COC)C1 C1(C(N2CCC(F)(CNC(c3cnsn3)=O)C2)=O)CC(=O)c2ccccc2O1 Cc1cn2cc(C(=O)NC(C)CN(C)C(C3CC4COCC4C3)=O)sc2n1 c1(C(CC(=O)NC(C2CCN(C(c3cc(=O)cc[nH]3)=O)C2)C)C)ccc(N)cc1 CC(C)(CCNC(c1cc(C(F)F)[nH]n1)=O)C(=O)NC(CN1CCCC1)CO N1(C(CC2CCCN(C(C)C)C2)=O)CCCN(C(C2CCCN2C=O)=O)CC1 c1(NC(c2c(NC)c3c(s2)nccn3)=O)cccc2cccc(Cl)c12 C=CCCC(F)(F)C(=O)NC1CN(C(c2cnc(CCCC)s2)=O)CC1C=C c1(CCN(CCC(=O)NCCc2nc(C3CC3)no2)CC)ccc(F)cc1 C(=O)(C(CC(C)C)NC(=O)CC(C)c1ccco1)NCC1(C#C)CCC1 c1(C(=O)NC2C(NC(C3(CC#C)CCOC3)=O)CC2)n[nH]c2cc(Br)ccc12 C1(C(=O)Nc2n(C)nc(C3CC3)c2)CC12CCN(C(c1cccnc1)=O)CC2 C1(C(CNC(Cc2cnc(C)s2)=O)C)CCN(C(C2CC(O)(C(F)F)C2)=O)CC1 C1(C(=O)NCCCCNC(CC(C)C2CC2)=O)CNC(=O)CC1(C)C N1(C(CCCCOCC)=O)CC(C(=O)NC(C2CCOC2)CO)C(C)(C)C1 c1(C(=O)NC(C)CCCCNC(C2CC(=C(F)F)C2)=O)csc2c1CCCC2 N1(C(C(c2cccnc2)NC(C(CCC)F)=O)=O)CCOC2CCC12 c1(C(N(C2CN(C(C3(C)CCCOC3)=O)C2)C)=O)cc2c(o1)CCCC2 C1(NC(COC(C)C)=O)CC12CC(NC(C1CCCOCC1)=O)C2 c1(OC)cc(CCNC(C2NCCC(O)C2O)=O)ccc1O c1(-c2nnco2)ccc(F)cc1.C(=O)CC1CC1.C(=O)(C)NCCOC.O N1(C(c2cccc(CC)c2)=O)CCC(CO)(NC(=O)Cc2ncoc2C)CC1 C1(C(N2CC3CC3C2)=O)C2(CCC2)C12CCC2.C1(C=O)CC(C(F)F)C1.CO CC1(C)CN(C(=O)Cc2cnccn2)CCC1NC(c1cc(Br)c[nH]1)=O c1(CC)cccc(C(=O)NC2C=CCCC2C(=O)NCc2ccc(C)s2)c1 c1(C(N2CCC(CN(C)CCN3CCCC3)CC2)=O)cccc2c1OCC2 C12(CNC(CCC=C=C)=O)CCCC1CN(C(=O)CCc1c(C)n[nH]c1C)C2 C1(c2n(CCOCC)nnn2)(NCCCCN(C)C(C)=O)CCOCC1CC c1(C(N2CCC(C(C)NC(=O)C(Cl)(Cl)Cl)CC2)=O)c(Br)ccc(F)c1F C1(CN(C(=O)Cc2cccnc2)C)CN(C(C2CNC(=O)N2)=O)CC12CC2 Cc1cccc(CC(N2CCCC2C2(NC(c3[nH]cnc3C)=O)CC2)=O)c1 C1(C(N2CC(OCCNC(c3c(C)snc3)=O)C2)=O)CN2CCC1CC2 C(CC1CC1)(C(=O)NOCC1(CC2CC(F)(F)CO2)CCC1)OC CCCCC(O)C(C)C(=O)N1CC(CNC(c2ccc(F)s2)=O)C2(CC2)C1 c1(N2C(=O)CC(C(=O)N(C3CCCC3)C3CCC3)C2)cc(F)cc(F)c1 O=C(CC1=CCCCC1)N1CCC(F)(C(N2CC(O)(C3CC3)C2)=O)C1 n1(C(C)C)cnc(C(=O)NC(c2cn(CC(=O)NC3CCC(=O)N3)nn2)C)c1 C1(NC(C2=NOC(C)C2)=O)CCC2CC1CN2C(C1Cc2cscc2C1)=O c1(C(N2C(C3(NC(CCC(C)(C)C)=O)CC3)CCC2)=O)ccc(S(C)(=O)=O)[nH]1 CC1CCN(CCOCCO)CC1NC(=O)CCCCN(C)C C1(NC(c2cncn(C)c2=O)=O)CCN(C(=O)CCC2CCC(=O)N2)C12CCC2 c1(C(C)=O)cncc(C(=O)NC2(C)CCN(C(=O)C(=Cc3ccccc3)C)C2)c1 CCC(CCCO)NC(c1c[nH]nc1CNC(c1csnc1C)=O)=O C1(C(=O)NCC(CN(C)C(c2cn(C)c(=O)cn2)=O)O)CCc2nnnn2CC1 C1(C)(CC)CCC(C(=O)NCC(C)CNC(=O)C(c2ccc(C)cc2)F)O1 N1(C(C(C)(C)OCC)=O)CCCCC1.c1(C(NC)=O)sc(C(F)(F)F)nc1C C#Cc1cn(C)nc1C(=O)NCC(C)C(F)(F)F.c1(C=O)cc([N+](=O)[O-])c[nH]1 N1(C(c2c(C(C)(C)C)cccn2)=O)CCCCC(CNC(=O)CC2CSC2)C1 c1ccccc1.c1(C(N2CCC(OC)C2)C(=O)NC)ncc(CC)o1.C(C)=O C12(NC(COCCN(C)C)=O)COC(C1)C(NC(=O)CN1CCOCC1)C2 C1CC2(CCN(C(c3cscn3)=O)C2)CO1.Cc1cc(=O)n(C)nc1C(=O)NC Cc1c(C#N)nn(-c2ccccc2)c1NC(C1(C)CCNC1=O)=O C1(CNC(C(COC)OC)=O)CCN(C(=O)CCCc2sccc2C)C12CCC2 C(=O)(C(CC(C)(C)C)OC)NC1CC(OC)CN(C(CCS(=O)(=O)NC)=O)C1 c1(OC)ccc([N+](=O)[O-])c(N2CCC(C)C(NC(c3c(C)ncn3C)=O)C2)n1 c1(C(=O)NCC2CC3(CN(C(CCCC(N)=O)=O)C3)C2)c(F)cc(F)cc1F C1(CCN(C(c2c(CC)[nH]cc2)=O)C)CCCCN1C(=O)C(C)N1CC(C)C1 C(C1=CCN(C(c2csc3nccn23)=O)CC1)NC(c1c(Br)cn(C)n1)=O C(=O)(C(N)CCCCCC1OCCO1)NC(CCC)CCO c1ccc(C#N)cc1F.Cc1csc(C(C)C(=O)NC2(C)CN(C(=O)CN)C2)n1 C1(CC)C(CO)CCCN1C(C1CC12CCOCC2)C(=O)NCCC1(C)CC1 Cn1ncc(C(N2CC(C3(NC(C45CC(CO)(C4)C5)=O)CC3)C2)=O)cc1=O Cc1cc(C(=O)NC(C)CCCC(=O)N(CC(O)C(F)(F)F)C)cc(O)n1 C(C)(C(=O)N=S(C)(=O)CCC1CC(N)C1)c1nc(C)[nH]n1 N1(C(CC2CCC(NC(CC(CC)C)=O)C2)=O)CC(C2(C)CC2)C1 CC1CN(C(C23CC(CO)(C2)C3)=O)C(C)CN1C(c1ccc(CO)s1)=O CCCCCC(O)C(=O)N(C1CCCN(C(c2csc(C(F)(F)F)c2)=O)C1)CC Cc1ncccc1CC(=O)N(C(C)CCNC(=O)CN1CCC1)C c1(C(=O)NCCCCCCNC(CC2N(C)CCC2)=O)cc(N)ccc1O N1(C(c2c(Cl)cnc(C)n2)=O)CC2CCN(C(=O)CNC(N)=O)CC2C1 N1(C(C2(CC=C)CC2)=O)CC2CCC(NC(=O)CC3CC3(Cl)Cl)CC2C1 C1(CNC(=O)CC2CCOC2)CCN(C(C2(F)CCC2)=O)CC1C1CC1 C=CCCCCCC(=O)NCc1ccc(C(=O)NC(CC)C(N)=O)o1 C1(C(=O)N)(OC)CC(C)C1.C1(C(C)(C)O)CN(C(=O)C)C1.c1ccon1 c1(NC(C2(N(C)C(C3CC(C#N)C3)=O)CCC2)=O)cncc(C#N)c1 c1(C(C)=O)cccc(NC(C2CC2NC(C2CC(C)(C)C2)=O)=O)c1O C(=O)(CC(C)C(C)(C)C)N1CC(N(C(c2c(C)scc2)=O)C)C2(C1)CC2 c1(C(N2C3CC(CNC(C4CC(=O)NC4)=O)C2CC3)=O)cc2cc(O)ccc2[nH]1 c1(C(=O)NC(CCNC(C(C)OC2CCCCC2)=O)(C)C)ccc2ncsc2c1 C1(CCC)CN(C(c2sccc2OC)=O)CCN1C(c1cn(C)c(=O)n1C)=O C1(CSC)CCCN1C(=O)CC1CCN(C2CCC(C)C2)C1 C12(C(=O)NCC3(O)CCN(C(c4c(C)c[nH]c4)=O)C3)CC=CCN1CCC2 C1(C)(C(N(C2CC(=C)C2)C)=O)CC(O)CN1C(=O)CC(C)F c1(NC(C2CC(C)CN2C(=O)CC2CCCC2)=O)cnc(O)nc1O CN1CC2C(C(=O)NC3(CCC)CC3)C2C1.c1(C=O)ccc(C(N)=O)nc1.N c1(C(N2CCC(N(C(C(C)n3cccc3)=O)C)C2)=O)cc(F)cc2ccoc12 c1(C(=O)NCC(C)(C)CNC(=O)Cc2ccns2)oc2ccccc2c1C Cc1ccc(C(=O)NC(c2ccnn2C)C(=O)N(C(C)C(C)C)C)cn1 N1(C(C(CC)C)=O)CCN(C(=O)CCc2cnc(C3CCC3)o2)C2CCC12 C1(C(=O)NCC(O)C(F)F)CCC(OCC2CCCC2)CC1 N1(C(C=C(C)C(C)C)=O)CCc2[nH]nc(CNC(=O)CC3CCNC3=O)c2C1 CC1=C(C)CC(C(=O)NCCC2(O)CN(C(=O)C(F)C3CC3)C2)CC1 N1(S(c2ccc(C(=O)O)cc2)(=O)=O)CCC(Cc2ccccc2)C2(CCC2)C1 c1(C(=O)NCC2CCC(NC(=O)CN3CC=CC3)C2)cc2c(nc1O)CCC2 c1(-c2nc(-c3c(O)nc(C)c(I)c3)on2)cc(Cl)cc2c1OCC2 CCC(N=c1[nH]c(N2CCCN(CCO)CC2)nc2c1SCC2)C1CCCOC1 C(CCN=C(NCc1cccc(NC(C)=O)c1)NCC(c1cnn(C)c1)O)SC Cc1c(C(=O)NCC(F)CNC(=O)CCc2c(F)cccc2F)cccc1F C1(NC(c2scc(C(C)=O)c2)=O)CN(C(c2ncn(C)n2)=O)CC1C C12(C=O)CCC(C1)OC2.c1(CCC)nc(C)c(C(=O)NCC2CC2)o1.N C1(CC(C)C)(C(=O)NCC(CN(C(C(CC)n2ccnc2)=O)C)C)CCNC1=O c1(C(N(CCC(C)NC(C(CCC)O)=O)C)=O)cnc(C)nc1-c1ccncc1 FCCCN=C(NCc1csc(C(F)(F)F)n1)NCC1CCC(F)(F)CC1 N1(C(=O)C=CCO)CCC2CCCC(C1)N2C(c1cc2ccc(Cl)cc2[nH]1)=O N1(C(C(C(C)C)SCC)=O)CCC2(CC1)CC2C(=O)N(CC)OC C(=O)(CCC(C)NC(c1ccnn1C1CC1)=O)NC(CC)C(=O)N(C)C N1(C(C(C(C)C)OC)=O)CCC(NC(=O)Cn2cc(Cl)cn2)CC(O)C1 C1(C(N2C(C(N(C)C)=O)CC2)=O)CCN(C(C2CC3(CC(=O)C3)C2)=O)CC1O C(=O)(C(N)CC(=O)N1CCCC(c2ccc(Br)cn2)C1)OCC=C C1(CCO)CN(Cc2cn(C3CCOC3)nn2)CCO1 c1(C(=O)OC)cncc(-n2cc(C3CCCCN3C(C3(C)COCCO3)=O)nn2)c1 C1(CC(=O)NC2(C(=O)NC)CC2)CC(C)(C)CN1C(c1c[nH]nc1Cl)=O C=C(C)CCC(=O)NCC1CC(NC(C2CC2C(C)(F)F)=O)C1 C(=O)(C(O)CCC(C)C)N(C1C2CN(C(C=Cc3ccc(OC)cc3)=O)CC21)C c1(C(=O)NC2CC(CNC(CC(C)CF)=O)C2)ccc2n[nH]cc2c1 c1(CN(C)C(C2CCN2C(=O)CC2CCCCO2)=O)ccccn1 C(C)(CO)(C(=O)NCC1(NC(C2CC2C(N)=O)=O)CCC1)OC.O c1(C=O)ccc(C#N)c(C)n1.C12(OC)CCC(C(=O)NCCC(C)C)(CC1)C2 Cc1ncc2c(n1)CNC2C(=O)Nc1cccc2c1CCC2N N1(C(CCN(CCC)C)=O)CCC(C(C)(C)NC(=O)CC2CCN(C)C2)CC1 c1(C(N2CC(C)(NC(C3CCc4ncsc4C3)=O)C2)=O)cc2cc(O)ccc2[nH]1 c1(C(=O)OC)ccc(-c2cn(CCNC(C3CC4CC3CO4)=O)nn2)cn1 C(c1ccc(Cl)cc1F)=CC(N1C(C)(C)CCC1)=O.C1(O)(CC(=O)N)CCOC1 CCC(C(=O)NC(C(NC1CCCc2ccoc21)=O)C1CCCC1)C(C)(C)CC C1(NC(Cc2cc(C)ns2)=O)COC2(CCN(C(c3ccc(C(C)C)s3)=O)C2)C1 C(CC)CC#C.C12CN(C1)C(=O)CO2.C#CCOCCNCCN.O N1(C(CCC(=C)Cl)=O)CCC2CN(C(=O)CCSc3ccc(OC)cc3)CC12 C(=O)(CCCCC(F)(F)F)NC(C)CCCNC(C1CC(Cl)(Cl)C1)=O N1(C(C(CC#C)C)=O)CCCC2(CCN(C(c3ncc(Br)cc3N)=O)CC2)C1 CC1(C)CC(CNC(=O)C(=Cc2c[nH]cn2)F)CN1C(c1cncc(F)c1)=O N1(C(Cc2c(C)nc(S)s2)=O)C2CCC1C(NC(=O)CC1CCC1C)C2 C1(OC(C)(C)C)CCOC1COC(c1c[nH]c(=N)o1)=O CCCCC(CC)CC(C(=O)NCC)N1CCCC1c1cccc2ccccc12 CC(CC(=O)N(C)CC1CCN(C(C2COC2)=O)CC1)CC(C)(C)C N1(C(c2n(CCC)ncc2)=O)CCC(NC(c2cc(C)nnc2O)=O)C12CCC2 C12(C(N3C(C)CN(C)CC3)=O)CCCC1CCN2C(c1cscn1)=O N1(C(C2=CCCC2(C)C)=O)CCCC12CCN(C(=O)CC(F)(F)C(F)(F)F)C2 Cc1ccc2ccc(C(=O)NC(C)(CNC(=O)C(C)SC(C)C)CO)nc2c1 C(=O)(CC(F)(F)F)N.C1(C)(C(NC)=O)CC=CCO1.N1(C(CC)=O)CC(O)C1 C1(CC)(CNC(C2CCN2C(=O)CC2C=CCCC2)=O)CCCC1 C(=O)(C#CC(C)(C)CNC(=O)C(C)O)NC1C(C)CN(C)CC1.C1CC1.C c1(CC(=O)NC2C3CN(C(CC=CC)=O)C(C3)C2)coc2ccccc12 c1(OC)cccc2[nH]c(NCC(n3ccnc3C(C)C)C)cc12 C#Cc1ccc(C(=O)NOCC(=O)NC2CCCC2C#N)cn1 n1(C(C(=O)OC(C)C(=O)ON)Cc2ccccc2)c(S)nc2ccccc2c1=O N1(C(CC(C)N(C(c2c(C)cns2)=O)C)=O)CCC2(COC(C)C2)C1 N1(Cc2ccc(CCC)o2)CCC(O)C(C(=O)NC2CNC(=O)C2(C)C)C1 N1(C(C(=Cc2cnc[nH]2)C)=O)CCC(NC(=O)C(=O)CCC(C)C)C2(CCC2)C1 C12(CN(C)Cc3cn(-c4cn(CCC=C)nc4)nn3)CC(C1)C(CO)O2 N1(C(C2C(CC)OCC2)=O)CC2(C1)SCCC2NC(=O)C(F)=CC1CC1 [N-]=[N+]=NC1CC(C(N2CC(CC(F)C(N3CCOC(CC4CC4)C3)=O)C2)=O)C1 c1(C(N2CC(C)N(C(=O)CCc3nc[nH]n3)CCC2)=O)ncccc1S(C)(=O)=O c1(C(=O)N)ccc(C(F)(F)F)c(O)n1.C12(C=O)COCC1C2.C1(CC)CC1 C1(NC(=O)NC2CCCC(C(F)(F)F)C2)CCCCNC1=O c1(CNC(N2CCCN(CCF)CC2)=O)ccc(O)cc1I C1(Cn2ncc(NC(=O)NC(c3ccc(F)cc3)C)c2)CCc2ccccc2C1 N1(C(COC(C)=O)=O)CCCC1C1CCCN1C(=O)CC(F)(F)F N1(C(CC(=C)C)=O)CCCC2(CCCN2C(=O)CCCC(=O)NCC)C1 C1(C2CC2)(C(=O)NC2C(NC(C(C=C)C)=O)CCOC2)CC(=O)C1 Cc1[nH]c2ccc(Cl)cc2c1CCNc1nnc(CF)s1 C(=O)(CN(CC1CCCO1)N(C)Cc1ccccc1C#N)OCC c1(OC)ccc(CC(N2CC(NC(c3cccnc3C)=O)CC(F)C2)=O)cc1O C1(NC(C(N2CC(C)C2)C)=O)CN(C(=O)CCc2cncnc2)CCC1CO C=CCN=c1[nH]c(C(N2CC(C)(NC(c3cn(C(F)(F)CO)nn3)=O)C2)=O)cs1 C1(NC(C(C)O)=O)CCN(C(C2(n3cc(Br)cn3)CCC2)=O)C1(C)C c1(CN2C(C(=O)Nc3c(Cl)nc(C)c(C)n3)CC2)ccc([N+](=O)[O-])cc1O C1(C(=O)Nc2cc(OC)c(O)cc2)CCCC2CN(C(=O)CC3CCC3)CC12 N1(C(c2cc(CCOC)on2)=O)CC(NC(=O)Cc2ccns2)C2CC12 C#Cc1cccc(C(=O)NC2CC2NC(=O)C(C)(c2cccs2)N(C)C)c1 C(=O)(C(F)CC(C)(C)C)NCCCN(CCCNC(C(C)C(F)(F)F)=O)C c1(C(C)(C)C)cc(NCCN2CC[Si](C)(C)CC2)n2ncnc2n1 N1(C(CCOC)=O)CCC(O)(CCNC(c2cc(Br)ccn2)=O)CC1 C1(C(N2CCC(CC(C)NC(c3nonc3N)=O)CC2)=O)CCCCC1C1CC1 C12(NC(CNC(C)=O)=O)CC(CNC(c3ncccc3O)=O)(C1)OC2C c1(CS(C)(=O)=O)nc(-c2cccc(Br)n2)n(CCCCO)n1 N(C(=NCCSc1ccc(Cl)cc1)NCCn1cncn1)CC(CCC)C C1(C(=O)N(CC(C)(C)C(=O)NCCN2CCC3CC23)C)(CC)CCNC1=O c1(CC)cnc(C(=O)NCCC2CC2)nc1.c1(C(=O)N)[nH]ccc1C1CC1 N1(C(C2C(C)C2)=O)CCC2(CC1)CC2NC(=O)Cc1cnn(C(F)F)c1 c1(N2CCC(C)S(=O)(=O)CC2)nc(=NCCSC(F)(F)F)[nH]c2c1SCC2 C(=O)(C1CCc2c[nH]nc21)N1CCCC(C(=O)NC(CCC(C)C)C)CC1 c1(C(=O)NCC2(CNC(CCN3CCN(C)CC3)=O)CC2)nccc2occc12 N1(C(c2ccc(CCC)cc2)C)Cc2ccc(CNCC(C)C)cc2C1 Cn1ncc2c(C(=O)NCC3(F)CCN(C(=O)Cn4cc(Cl)cn4)C3)ccnc12 c1cc(C)ccc1O.N1(C(C(=O)NCC)=O)CCC(C(=O)NC)(C(C)C)C1 c1(C(=O)NCCC(C)(C)NC(C2CC(C)(CC)C2)=O)cnncc1NC N1(C(=O)CCc2ccncn2)CCCCC(C2CN(c3cc(F)ncn3)C2)C1 N1(C(C2(CN(C)C)CC2)=O)CC2CC1C2C(=O)N(CCCF)C CC1CN(C(=O)CN2CC(=O)N(C)C2=O)CC2(CCN(C(=O)CCC3CC3)C2)O1 C(C)(c1cccs1)=CC=O.c1(CCC)cc(C(=O)N)n[nH]1.C(C)(C)C1CC1 c1(COC)nc(NCCCS(C)(=O)=O)cc(=NCc2nccc(=N)[nH]2)[nH]1 c1(C(N2CC(C)(NC(C(C(C)C)O)=O)C2)=O)cnc2c(Br)cccn12 c1(SCC)ccccc1C(N1CCN(CCNC(=O)C(O)C2CCCC2)CC1)=O O=C(C1=COCC1)N1CCC(CCNC(C2(Cc3ccncc3)CC2)=O)C1 c1(C(C)C)nc(C(c2cnn(C)c2)NC(=O)NCCC2CCCC2)no1 c1(N2C3CCC3CC2=O)cc(F)c(C(N)=O)c(F)c1.C1(NC)CCCCC1.CO C(=O)C1=NOC(C)(C)C1.c1(C(C)NC(CC(=O)OCC)=O)ccccc1.N S(=O)(=O)(c1cccc(Cl)c1)NCCC(C(OCC)OCC)O.C(CCCO)N O(N1CCC(CC(=O)N(C2CCCCN(C(=O)C(C)S(C)(=O)=O)C2)C)CC1)CC N1(C(COCCC#C)=O)CC2(C)CC2(C(F)(F)F)C1.C1(C=O)CCOCC1.N c1(C(=O)NC(C)CC(C)NC(C2CCCCS2(=O)=O)=O)cc2c(nc1O)CCC2 C(=O)C(F)(F)c1csc(Cl)c1.CC(C)(C)OC=O.C1(C=O)CC1.CC.N c1(CN2C(C(=O)NC(CCCC)CO)C(O)CC2)c(F)ccc(Br)c1OC c1(C(=O)O)cc(Cc2ccccc2)nn1CC1CCCN(C(=O)CCC(F)F)C1 N1(C(C2N(C(=O)OC(C)(C)C)C(=O)CC2)=O)CC2CCC(C1)O2 Cc1cc(NC(C2CC3(CCC3)C2)=O)cc(C#N)c1.c1(C(=O)N)c(C)n[nH]c1C C12(C(=O)Nc3cnc(C)s3)CC1CN(c1ccnc(NCc3ccccc3)n1)C2 Cc1nc(C)c(-c2cn(-c3cccc(C(=O)N(CC(N)=O)CC(N)=O)c3)nn2)s1 Cc1cc(Br)c(F)cc1NNC(=O)NCc1c(C)cc(Br)cc1F C=C(C)CCC(=O)N1CCC(NC(=O)CCc2ccc(OC(F)(F)F)cc2)C1 C1(CC(=O)NC2C(C(=O)NCCC(=O)NC)CC2)OCCCO1 C(=O)(C(C)(C)C1=CCN(C(C2CCCCCC2)=O)C1)NCCc1ncc(C)nc1 c1(C(N2CC3(CCN(C(C4(C)CCN4)=O)C3)C2)=O)cc(=O)c2cc(F)ccc2o1 N1(C(c2c(CC)c[nH]n2)=O)CCC(C)(CC(=O)NC2C=CCCC2)C1 C(=O)(C1=CCCCCC1)N1CCN(C(CC(C=C)(C)C)=O)CC1c1nccn1C c1(CN(C(c2ccccc2)=O)Cc2ccccc2)cccc2c1CCN(CCl)C2 C(=O)(CCCC(F)(F)F)N1C(C(C)C)(C(N2CCOC(C)(C(C)C)C2)=O)CCC1 CCC(C)(C)C(C)NC(=O)C(Cc1ccco1)NC(=O)C(c1ccccc1)C c1(C(=O)OCC)cnc(N2CCCC(C(C)NC(c3cc(C)[nH]n3)=O)C2)cn1 N1(C(C)C)CC(C(=O)NCCCCNC(C2CC2(Cl)Cl)=O)CCC1=O C=CCCCCC(=O)NCC1(C)CCCN1C(c1cccc(O)c1Cl)=O C1(NC(c2cc(C)[nH]c2)=O)CC(NC(c2ccncc2F)C(C)C)C12CCC2 C1CCC(C(F)F)C1.N1(C(C(=O)NCC2CC2)=O)CCCC(c2ncc[nH]2)C1.O N1(C(CC(C)C)=O)CCCC12CCN(C(C1CCc3nnnn3C1)=O)CC2 N1(CC)CC(C(=O)NC(CNC(=O)CC2=CCCC2)C(C)(C)C)c2ccccc21 N(C(=NC1CCCC1)NC1CCOc2ccccc21)CCC1C(C)(C)CCCO1 C1(CNC(=O)C2=CCOC2)CCC2(CCC2)C1NC(c1ccc2n[nH]cc2n1)=O C1(NC(C(CSC)C)=O)CCC(C)(CNC(c2nnn(C)c2C)=O)CC1 C(=O)(C(C)C(F)(F)F)NCC(CCCC)NC(c1cnccc1C(F)F)=O C1(N)(CC(=O)NC2CC(C[Si](C)(C)C)C2)CCCCC1 C1(NC(c2c(CC)cno2)=O)CCC(NC(=O)C(C)(C)O)CC1 C1(CC(=O)NCCCN(C(=O)CC2CCSC2)C)COCCO1 C(c1cnc[nH]1)=CC(=O)NCCN(C(=O)C(C)OCCC(C)C)CC c1(C(=O)NC(CCCC)CNC(=O)CCCC(C)=O)c(C)nn2c1CCCC2C C(C)(C)(C(=O)NC)NC(=O)OC.C1CCN(C(=O)CCN(C)CCO)C1 c1(C(N2CCC(CCNC(C3CC3Br)=O)C2)=O)c[nH]c2nc(Cl)ccc12 N1(C(c2n(CC)ccc2)=O)CC2(C)CN(C(C3(c4nccs4)CC3)=O)CC2(C)C1 C1(CC=O)C=CS(=O)(=O)C1.C1(NC(COCCN(C)C)=O)CC(C)C1 N1(C(c2ccc(N)cn2)=O)CC2CC(NC(C3(N4CCOCC4)CCC3)=O)C1C2 C=CC(C)(C)C(=O)NC1CCC1C(=O)NC(C)COC Cc1sccc1COC(=O)C(c1ccccc1)NC(N)=O C1(C(N(CC(=O)NCC)CC)=O)CN(C(=O)C)CC1(C)C.C(C)C.O N1(C(C(=O)NCCOCC)C2COC2)CCCC(C)(O)C1 C(=O)(C(O)C(F)(F)F)NCC(C)(C1CCC1)NC(c1cccc(C)c1)=O c1(NC(C2CCCN(Cc3cc(O)cc(O)c3)CC2)=O)cc(O)nc(O)n1 C1(C(=O)NCCCN(C(=O)CCSC2CCCC2)CC)CCCCC1(F)F C1(NC(c2cc(-c3ccco3)on2)=O)CN(Cc2ccc(Br)[nH]2)CC1F c1(C(=O)NC2C(NC(CN(c3cnc(C(F)(F)F)s3)C)=O)C2)ccccc1 N1(Cc2ccc(C)c(F)c2F)CCc2c(C(=O)NCC(F)CO)n[nH]c2C1 N1(C(c2c(C)cc(CC)o2)=O)CCC(CO)(CNC(=O)CO)CC1.CCF C1(CNC(CCC(=O)OCC)=O)CN(C(c2sncc2C)=O)CC12CCC2 c1(C(C2CCSCC2)NCCC(F)F)nnnn1CC1CCCO1 C(C(=O)NN1CCCOC1=O)(n1cc(C(C)NC)nn1)c1ccccc1 N1(C(c2cc(C)cc(N)c2)=O)CC2(CCC(C)O2)C1.C(=O)C(F)OC(F)(F)F.N N1(C(c2ccc(OC)s2)=O)CCC(O)(C(=O)NCC2CCCC2)C1 c1(CNC(c2cccc(C)c2)c2ccccc2)ccc(S(C)(=O)=O)cc1F c1(C(=O)NC(CC)CN(C)C(c2cc(OC)ns2)=O)sc2ncccc2c1Cl n1(CC=CC)ncc(C=O)c1Br.CC(C)C.C(=O)C=CC=O.C1CC1.N CN1CCCCC1C(N1CCC(C(C)(C)NC(C23CCC2CC3)=O)C1)=O c1(C(N2CCC(NC(=O)Cc3cccs3)C2)=O)cc(Cl)ncc1OCC(F)F Cn1cc(C(=O)NC2CC3C(NC(=O)CN4CCCC4C)C3C2)n(C)c1=O c1(NCC2OCC(CNC(CS(C)(=O)=O)=O)C2)ccc(CN)c(Cl)c1 c1(C(N(CC(C)(C)O)CC)=O)cc(=O)cc[nH]1.C1(C)C(=O)N1C1CC1 Cc1ccc(C(=O)NCC(C(=O)NCCC2COC(C)(C)C2)N(C)C)nc1 c1(CC(N2CC3C(NC(c4cccc(C#N)c4)=O)C3C2)=O)ccc2occc2c1 CC1CN(C(=O)CCCOc2cccc(F)c2)CC1NC(C1(Cl)CC1)=O C#Cc1cc(C(=O)NC2CCN(C(=O)C3=NOC(C)C3C)C2)ccc1C C1(C(N2CC(C)(NC(c3ccn(CC)n3)=O)C2)=O)CCC(C)NC1=O c1(NC(C2CCOC2)CC)ccc(S(=O)(=O)NCCNC2CCCC2F)cc1Br c1(C(N(CCNC(C2(C)C(CC)CCC2)=O)CC)=O)cccc2c1nc(O)n2C C(CN=c1[nH]cnc2cc(Br)ccc12)C1N(Cc2c(O)c(F)ccc2F)CCC1 N1(C(c2cccc(NC)n2)=O)CC(NC(=O)CC(F)(F)C(F)F)CC(F)(F)C1 C(=O)(CCCC(CC)CC)N(CCC)CCNC(c1cc(Br)ccn1)=O c1(C(CCO)NC(C2CCN(C(C=COCC)=O)C2)=O)ccc(Cl)cc1 Fc1ccc2c(c1)CC(NCCCOC1CCOC1)CO2 C(=O)(C(O)CC(F)F)NCC1CCN(C(C2CN(C)C(=O)N2)=O)CC1.C1CC1.C Cc1cc(C(N)=O)sc1CNC(=O)CC(C)NC1CCC(C)C1 C1(NC(C2(C)CCSCC2)=O)CS(=O)(=O)CC1NC(c1cccnc1)=O c1(C(N2CC(CC)OCC2)=O)cn(C)c(=O)n1C.c1(CC(=O)N)cccc(Cl)c1 Cc1cc(CN(C)CCN(C)C(c2cc(Cl)no2)=O)sn1 C(=O)(CCCC(C)c1ccccc1)NCCC(C)NC(C1(C(F)F)CC1)=O C(=O)(C(C)(C)CCNC(c1ccns1)=O)NC(C1CC1(C)C)CC Cc1cccc(-c2cc(C(N3CC4CC4(CNC(C4CCCO4)=O)C3)=O)on2)c1 c1(CC=O)cccc2cccnc12.n1(CCC)cc(C(=O)NCC2CC2)cn1.N c1(C(N2C(CNC(c3c(C)snc3)=O)CCC2)=O)ccnc(NC2CCCC2)c1 N1(CCNC(c2cnc(CC)[nH]2)=O)CCCN(C(C2(C)CCC(O)CC2)=O)CC1 c1(C(=O)NC)ccc(-c2nccn2CC2(C)CC2)cc1-c1cnc(=N)[nH]c1.O c1(C(N2CCN(C(C(C=C)(C)C)=O)CC2CO)=O)ccc(F)c2occc12 c1(C(=O)NC(CN(C(C(COC)C)=O)C)C)cc2ccc(OC)nc2[nH]1 CC(CC(=O)NCC1(O)CC(C(N2CCC(C)(C)CC2)=O)C1)C(F)F c1(-c2n(C(C3CCOCC3)C)nc(C3CN(C)CCO3)n2)cc2ccccn2n1 C1(NC(C=NOC)=O)COCCC1NC(=O)COc1cn[nH]c1 c1(CNC(C2(C)CCCN2C(=O)C2CC2)=O)cc(O)ccc1Br N1(C(c2cccc3cnsc23)=O)CCC2CC(C1)CN(C(C1C3COCC13)=O)C2 c1(OC)ccc(CCCC(=O)N2CC(CC)C2)cc1.C1(C)(C(=O)N)CC2(CC2)C1 N1(C(C(COC)C)=O)CCCCC12CC(NC(c1ccnnc1O)=O)C2 CC1(C)CC(CNC(=O)C)N(C(=O)CCc2ccnc(Cl)c2)C1.C1CC=CC1 C#CC1(C(=O)NCC2Cc3nccn3C2)CCN(C(c2cc(CC)[nH]c2C)=O)C1 C1(NC(Cc2cc(=N)[nH]cc2)=O)CC(NC(=O)CCC(F)(F)F)C12CCOCC2 N1(C(C(CSC)(C)C)=O)CCCC(NC(C2CCCCO2)=O)CC1 CC1C(C)N(C)CCN1C(=O)CCN(CCCO)C(=O)CC1CC2CCC1O2 C1(CNC(c2csc(O)n2)=O)CCN(C(=O)CCN2CCC(F)C2)CC1(F)F C1(NC(CCCCC)=O)CC2CN(C(c3cc4n(c3)CCSC4)=O)CCN2C1=O CC1CN(C(c2cnn(CC(F)(F)F)n2)=O)CCCN1C(=O)C(C)n1cccn1 n1(CC=O)cc(C#N)cn1.C1(CCC)CCCC1C(=O)NC12CC(C1)C2.N C1(c2cn(C(CNC(CNC(CN(C)CC)=O)=O)C)nn2)CCC(C)=CC1C C(=O)(C(C)(C)C(=O)NCC1CCCCO1)OCC.c1(C=O)nn(C)cc1C C1(CNC(CCC2CC(OC)C2)=O)CC(O)CN1C(=O)CSCC(C)C c1(-c2cn(CCC(N3CCC(COC(F)F)C3)=O)nn2)cc(F)c(Cl)c(F)c1 C1CN(C(=O)CC2CC=CC2)C2(CCC2)C1.c1(SCC(=O)NC)ccccc1 CC(C)CCCN(C(=O)COc1ccccn1)C.C(c1c[nH]cn1)=C(C(=O)N)F CC1CCCC(C(=O)NCCOCC(N2CC(C(=O)N(C)C)C2)=O)CC1 Cc1nc(N2CCOC(C(=O)Nc3cnc(Br)nc3)C2)nc2ccccc12 c1(C(N(C(C)CNC(=O)C=C2CC2)C)=O)csc2ccc(Br)cc12 N1(C(CC(CC)(F)F)=O)Cc2ccc(CNC(C3CCSC(C)C3)=O)cc2C1 C1(C(N(CCCF)CC)=O)CN(C(C2CCC(C(N)=O)C2)=O)CC1F C(N=c1cc(Cl)nc[nH]1)C1N(C(C2CC(C)SCC2)=O)CCCC1C N1(c2nc(C(C)(C)C)nc(Cl)c2)CC2CCCC(NC(c3ccoc3Br)=O)C2C1 C1CN(C(C23CCCC2(C(N)=O)C3)=O)CCO1.C1(C(=O)N)(CN(C)C)CC1 c1(C(N2CCC(O)(CN(C(C(CCOC)C)=O)C)C2)=O)ccc2cc[nH]c2c1 C1(O)(CC)CCN(C(c2sc(=N)[nH]c2C)=O)C1.C(C)(C)(C=CC=O)SC.N CCC(CC(=O)NC(c1nc[nH]n1)C1CC1)NC(=O)CCC(C)SC c1cccc([N+](=O)[O-])c1.C(C)(C(=O)NC1CCC1)N(C(C)=O)C.C(=O)CC.N C(=O)(C1=NOC2(CCN(C(C3CCN(Cc4cnccn4)CC3)=O)C2)C1)NC Cc1ccn(C)c1C(=O)NC1CC1c1cccc(Cl)c1 C1(C(=O)NCCc2ccc(C)cc2)(COC)CCC(=O)CC1 c1(C(N2CCCC(C)(CNC(CCSC)=O)C2)=O)cc(Cl)c(N)c([N+](=O)[O-])c1 C(=O)(C1=NN(C(C)C)C(=O)CC1)N(CCCC)C.C(C)(C(=O)N)N(C(C)=O)C C1(OCC)CCC12CCC2.c1(C(c2nnnn2CC(F)F)N)ccc(C)c(I)c1 C#CC1(O)CC(C(=O)NCC(CCCC)NC(=O)Cc2ccn(C)n2)C1 C1(C(=O)NC(CC(=O)OCC)C)CCC(C)CN1C(=O)C(C)C(C)(C)C c1(C(CC)NC(C2COCCN2CCCNC(C)=O)=O)cc(C)ccc1C c1(OC)ncnc(OC)c1C(=O)NC1CC2(C1)CC2NC(=O)CCCCC.S CCCC(C)(C)CNC(=O)C(C1CC=CCC1)NC(=O)COCCF c1ccc(F)c(F)c1.C1(CNC(=O)CN2CC3CC3C2)CCN(C(=O)C)C1.O C12CCCCCN1C2=O.Cc1ccc(-n2cc(CCN3CCOCC3)nn2)cc1 c1(C(=O)NC(CNC(c2noc(CC)c2C)=O)C(C)(C)C)ccc2nc[nH]c2n1 c1(C(=O)NCC23CC2CN(C(c2cncc(CO)c2)=O)C3)cc2cnccc2o1 CC1(C)OCC2CC12C(=O)NC.C1CCCCN(C(=O)C)C1.C1CC(F)(F)C1 CC1CN(C(c2ncc(F)cc2F)=O)CCC1CNC(C1C=CC=CC=C1)=O c1(CC(N2C(C)CCC2)=O)noc2ccccc12.C(C(COC)C(=O)NC)OC C=C=CC(C)C(=O)N1CC(O)(C2CCCN2C(=O)CCS(C)=O)C1 N1(C(c2cc(OC)no2)=O)CCC(NC(c2cnc(S)n2C)=O)C(O)C1 c1(C=O)cc2ccccc2[nH]1.O=C(C1CC1)NCCOCC.CC.CC.O N1(C(C=CC(CC)=CC)=O)CC2CC(NC(=O)CCc3ccncc3)CC1C2 Cc1cc(C)c(C(N2CCCC2(C)CNC(=O)CC2(CO)CC2)=O)o1 N1(C(c2c(C(C)C)c[nH]n2)=O)CC(CNC(c2nc(Cl)cs2)=O)OC(C)(C)C1 c1(OC(CC)C)ccc(-c2nc(-c3cscn3)nn2CCC2CCCCC2)cc1 C1(NC(c2c(C)n(C)nn2)=O)CC(NC(c2ccc(F)c(CO)c2)=O)C12CCC2 N1(C(C2(C#C)CC2)=O)CC2(CCCC2NC(=O)C#CC2(CC)COC2)C1 n1(CC)nccc1C(C(=O)NCCCC1CC1)N(C)Cc1cnco1 CC1CC(=O)Nc2ccccc2N1C(N1CCCC1(C)CCc1ccccc1)=O c1(C(=O)NC2CN(C(c3c(C)nc(C)s3)=O)CC2F)cc(I)ccc1Cl CC(C)CC(F)C(=O)N(C(C)CN(C(=O)C(c1ccc(Cl)cc1)=O)C)C c1(C(=O)NCC2C(C)CCN(C(c3nc(CN)cs3)=O)C2)nccc2occc12 N1(C(C(C)CC2CCCCC2)=O)CCCC(C)C1CNC(C1CCCN1C=O)=O C=C(CNC(C1CCCCN1C(c1cnc2cc[nH]c2c1)=O)=O)c1ccccc1 C(=O)(C(C)(C)C(C)(F)F)N(C(C(c1scc(C)n1)(F)F)=O)CC=CC=O N1(C(c2cccc(NC)c2)=O)CC2CCC(C)C2C1.C1(CC(=O)N)CC2CC2C1 Cc1ccc(C(=O)NC2CCCC(NC(=O)CCc3cncs3)C2)c(N)c1F c1(C(=O)NC(C)C(C)(C)NC(C2(F)CCCCC2)=O)ccc(-n2cncn2)cn1 C1(NC(CC(CCC)CC)=O)CC(N=c2cc[nH]cc2[N+](=O)[O-])C12CCC2 C(C(=O)NCC1C2CN(C(=O)CCCc3ccc(F)cc3)CC12)(C(C)C)OC CCCS(=O)(=O)CC(=O)N1CCN(CC(C)NC(=O)CCCC#N)CC1 N1(CC(N2CCC2)=O)C(=O)CC(C)(C)C1=O.n1(C(C)C)cnc(C(=O)N)c1 C12(C(N)=O)CCCC1(C(=O)NC1CC1NC(c1ncccc1F)=O)C2 C1(CCC)CCC(C(=O)NC(C2(O)CCN(C(c3ncn(CC)n3)=O)C2)C)CC1 C1(C(N(CC(C)(C)NC(=O)C(C#N)C2CC2)C)=O)CCC(C)(C)O1 C1CC(O)C12CCC2.C1(CC(=O)N)CN(C(=O)Cc2coc(C(F)F)n2)CCO1 Cn1c(C(=O)NC2(C)CCN(C(=O)CC3CCCOCC3)C2)cc(Cl)c1Cl c1(C(N2CC(CCCC)C2)=O)n[nH]cc1C(F)(F)F.C(C=O)=CCNC.CC CC(C)(C)C(C(=O)N1CC2C(NC(C3CCCO3)=O)C2C1)N1C(=O)CCC1=O CCCC(C(=O)NC1CN(C(C2CCC3CC23)=O)CC1SC)OCC c1(CN2CCC(C(=O)Nc3ccnnc3)CC2)ccc(-c2cnoc2)c(F)c1 Cc1cc(C(=O)NC(C2CN(C(c3cc(=O)n(C)o3)=O)C2)C)c(F)c(Br)c1 N1(C(C(OC)OC)=O)CCCC2(NC(c3cnn4ccn(C)c34)=O)CC2C1 C1(CC)CN(C(C23CC(CC)(CO2)C3)=O)CCC1.C(c1cncs1)=CC=O.N C(=O)(CC(C)(C)CC(=O)OC)N1CCCC(C)(NC(COCCC)=O)C1 c1ccccc1.N1(C(C=O)C2CC2(C)Br)CCN(C(=O)C=C(C)C)CC1.CC c1(-n2ccc(C=O)n2)ccccc1C.C(C(=O)NCC1CC1)=CC=CCC c1(C(N(C2CC(NC(=O)C=C3CCSCC3)C2)C)=O)cc2ccccc2c(O)n1 N1(C(c2n(CC)ccc2)=O)CCC(N(C(=O)CCn2ccnc2)CC(C)C)CC1 C1(C(=O)NCc2cn[nH]c2)CN(C(C2CC(F)C2)=O)CCS1 c1(C=O)cnc2ccnn2c1.CC(C)C(C)(C)C(=O)NC1CC2(C1)CC(C)C2.N CC(C1OCCc2sccc21)NC(=O)Cn1cc([N+](=O)[O-])c(-c2ccc(F)cn2)n1 C=C(C)C(C)(C)C(=O)N1CCCC1.C(=O)(C(O)CC1CCCC1)NC1CC1.C C1(N(C(C2(COC)C=CCC2)=O)C)CCCN(C(c2csnn2)=O)CC1 C1(NC(CCOCC)=O)CCC(NC(=O)CC)CC1.c1(C(=O)N)ccccc1 C(c1cscn1)=CC(=O)NC1(C(=O)NC(c2ccco2)CO)C(C)C1 C1(CC(N2CCCCC2)=O)CC(F)(F)C1(F)F.c1(C(=O)N)ccsc1C(F)F n1(CC)ncc2c1CCC(NC(=O)CCCOC(F)F)C2 CC1=C(C)CN(C(C(C)=Cc2ccc(Br)s2)C(=O)NC2(C)CC2)CC1 C(=O)(CCCCCNC(=O)C(C)CC1CC1)NCC(C)C N1(C(C(c2cccs2)SC)=O)CCCCCC1(C)C(=O)O C(c1ccccn1)=CC(=O)N.c1(C(C)C)cc(C(N2CCC(C(C)C)C2)=O)on1 c1(C(N2CC3CCCC3(CNC(C3(Br)CC3)=O)C2)=O)cc2cccn2cn1 Cc1c(NCCCN2CCCC2)nc[nH]c1=NCc1cccc(Cl)c1F CCCCCCCCC(C)C(=O)NCC1(NC(C2(NC(N)=O)CC2)=O)CC1 N1(C(COCC(=O)NC)=O)CC(O)CC1(C)C(=O)NC12CC(C)(C1)C2 c1(OCCNC(Cc2c(OC)nccc2)=O)c(C)cc(C)cc1C c1(NC(C2(C)CCCN2C(c2ccc[nH]2)=O)=O)ccc(Br)c2ccncc12 C1(C(N2C(CNC(C(F)=CCC)=O)CCC2)=O)CCC(C)CC1 c1(C(=O)NC(Cc2ccc(Cl)cc2)CO)ccc(C(F)(F)F)c([N+](=O)[O-])c1 N1(C(CC2C(C)CCO2)=O)CCOC2(CCN(C(=O)OC(C)(C)C)CC2)C1 C1(CC(N2CC(C=C)C2)=O)CC(NC(=O)CC2(OCC)CC2)C1(C)C Cc1ncc2n1CC(C(=O)NC1CC(CN=c3[nH]nc(C(F)(F)F)s3)C1)CC2 C1(NC(c2cc3ccsc3s2)=O)COC2(CCN(C(=O)CC3OCCCO3)C2)C1 c1(CC)cnc(C(N2CCC(C(C)NC(C3CCC3)=O)C2)=O)nc1.C1CC1.C CC1(O)CCCC1NC(C1(NC(C2CCCSC2)=O)CSC1)=O [SH](=O)(=O)c1ccc(C=O)cc1.C(=O)(C(Cc1ccnn1C)NC(=O)N)OC c1(C(=O)N)ccc2c(c1)COC(=O)N2.c1(CC)cnoc1C(=O)NC(C)CO CC1(C)C(NC(=O)CC2CNC(=O)O2)CC1CC(N1CCOCC1)=O C(=O)(C1CCc2c[nH]nc21)N1CC(C)C(CNC(C2CCCC3(CCC3)O2)=O)C1 c1(C(=O)NCC(CC=C)NC(=O)C(C)COC)cc(Br)cc(CC)c1N C=CCC(CC(C)C)C(=O)NC1(C)CCN(C(C2(CS(C)(=O)=O)COC2)=O)C1 C1(C(=O)NCCCOC(C)C)CC(F)(F)CN1C(c1sccc1F)=O C(CC)(C(=O)NCC(C1CCC1)NC(=O)C(C)(C)F)OCC CC(C)C(CNC(C1(C(C)C)CCC1)=O)NC(=O)C(C)Sc1nncn1C N1(C(CCC2CCN(C(C3C4CC(=O)CC43)=O)CC2)=O)CCC2C(C1)C2(F)F N1(C(CCCCOCCC=C)=O)CCN(C(=O)CN2CC3CC3C2)C(C)C1 OC1C2COC1CN(c1cc(NCCOC3CC3(F)F)ncn1)C2 N1(C(CC2CCCC(C)O2)=O)CCCC12CCCN(C(=O)CCCC(N)=O)C2 C1(NC(C(=O)NC2C(CCCC)CCC2)=O)CCCN(c2nccn2C)C1 C1(CC(=O)NCCCCN(C(C2(C)CC(=C)C2)=O)C)C(=O)NN=C1C CC1(C)CC(C(=O)NC2CCCC2(C)C)CN(C(C23CSCC2C3)=O)C1 C1(N(C(C2C(CCC)CCC2)=O)C)CCCN(C(C2CCN(C(C)=O)C2)=O)C1 N1(C(C2CC2)=O)CCC(C2(O)CN(C(=O)C)C2)CC1.C(C)(C)C(F)(F)F.C c1(C(=O)NC(CCN(C(c2c(CC)cc[nH]2)=O)C)C)cc(O)n(C)n1 C(CCCCCNC(c1n[nH]cc1C1CCC1)=O)NC(C(C)(C)F)=O C1(C)(C(N(C)CC2N(C(C3CCC(CC)O3)=O)CCC2)=O)CC2CCC(C1)S2 C1(NC(Cc2cn(CC)nn2)=O)CCCCCN(C(=O)Cc2cc(C)oc2C)C1 N#Cc1ccc(CC(=O)NC(C(N2CCC(CSC)CC2)=O)c2ccco2)cc1 CC1C(NC(C2CC(=O)N2)=O)C(C)CCN1C(=O)C1=CCS(=O)(=O)C1 c1(C(=O)NC2C(NC(c3ccc(C)s3)=O)CCOC2)cccc2ncccc12 N1(C(c2cc(OCC)n[nH]2)=O)CCC(CC(=O)O)(OC)C1.C1CN(C=O)C1 C1(O)(CNC(CC(CC)O)=O)CCCN(C(=O)CC2CCCN2CC)C1 N1(C(=O)OC(C)(C)C)CCN(C2CCCN(C(=O)C=Cc3cn[nH]c3)C2)CC1 CCC1=NOC(CC(=O)N(CC(O)CNC(=O)C(c2cnn(C)c2)=O)C)C1 C1(C#CC(=O)NC(C2CCN(C(c3cc(N)cc(O)c3C)=O)C2)C)(CC)COC1 c1(C(=O)NC2CCN(C(CC3OCC(C)(C)C3)=O)C2)cc(Br)n2c1CCC2 C=CCC(CC)C(=O)NCc1ccoc1C(N1CCOC(C)C1CO)=O CC1(C)CCC(=CC(=O)NCC2(C)CN(C(c3sccc3C)=O)CCO2)CC1 N1(C(C(C)c2ccsc2)=O)C(C(=O)NOCC2CCOCC2)CC2CCCC12 c1(CNc2cc(C(N3CC(C(=O)OCC)OCC3)=O)n(C)c2)cc(F)ccc1I C(CC(O)C(F)(F)F)NC(C1(C(C)C)CCCN1C(c1ccccc1CO)=O)=O C1(C(N(C2CCN(C(CCN(C)CC)=O)CC2)CC)=O)CCCC(C)(C)C1 C(=O)(C1=C(F)CN(C(=O)C2=CCCC2C)CC1)N(C(C)CC(F)(F)F)C C(=O)(CCCCCN=[N+]=[N-])N1CCC2(C(NC(C3C(OCC)C3)=O)C2)CC1 C1(CC(N2CCC(CC=C)(NC(=O)CCCOC)C2)=O)CC2(CCC2)CCO1 c1(C(=O)NC2(CCNC(C3(Cl)C(C)(C)C3)=O)CC2)cccc2c1CCCN2 C1(CC(=O)NCC=C(C)C)CCCN1C(C1CC1Cl)=O CCC(O)C(C)C(=O)N(CCCNC(c1cccc(OC(F)(F)F)n1)=O)C CC(C)CC(C(=O)N1CC2CC1CN2Cc1ccc(C#N)cc1)C(N)=O c1(C(=O)NCC(CC(=O)OC)C(C)C)cc2ccc(Cl)cc2c(O)n1 N1(C(C2C(c3ccc(C)c(C)c3)C2)=O)CCN(C(C2(C(C)C)CC2)=O)CCC1C C(CCOC)(C(=O)NCCC1CC(C)(C)C1)NC(Cc1cn(CC)nc1)=O C1(NC(c2c(CCNC(Cc3c(C)ncs3)=O)n[nH]c2)=O)CN(C(C)C)CC1C C=CC1(CC(=O)N(CC(C)NC(=O)COC2CC2)CC)CCCCC1 C1(C(=O)NCC2N(C)C(=O)CC2)CC2(C1)C(F)(F)C21CC1 C1(C=O)Cc2cc(C)c(C)cc2O1.C1(CNC(C2(CCCC)CC2)=O)CCC1 C(=O)(CC(O)CC(C)(C)C)N(C1CC1)CC1CCN(C(CCOCC)=O)CC1 N1(C(COCCC)=O)CC(C(=O)NCc2csc(C)c2)C2(CC2)C1 C1(NC(CC=CC=C)=O)CN(C(c2cc3occc3[nH]2)=O)C2CCCC12 c1(C(N)=O)cnc2c(C(N3CCCC(NC(c4nocc4Cl)=O)C3)=O)cnn2c1 CCCC(C(=O)NCC(C)(C)C)NC(c1ccn(C2CC2)n1)=O N1(C(CC(C)(C)C2CC2)=O)CCOC(C(=O)Nc2cnc(F)nc2)CC1 CC(CN(C)C)CC(=O)N1CCC2CC12C(=O)NC(C)Cc1ccnn1C C1(NC(C)=O)CN(C(C2(c3ccccc3F)CCCC2)=O)CC2CC12 N1(C(CC=CC)=O)CCC(C2CCN(C(c3ccc(SC)c([N+](=O)[O-])c3)=O)C2)C1 CC(CCc1ccccc1)CC(=O)N1CCCC1C(O)C(=O)O CCCC(CC(C)C)C(=O)N1CCC2(CC1)CC2CNC(=O)CC(C)(C)C(F)F CC(C)(CCCC(=O)NCCCSCCO)NC(C1CC(=O)NC(=O)N1)=O C(C(C(=O)NCC(C)CO)NC(C)=O)OC.c1(C=O)cnc(-c2ccoc2)s1 N1(C(=O)Cc2ccccn2)CCN(C(=O)CC2CC2(Cl)Cl)C(CCO)C1 C1(C(=O)N)CCCCCC1(F)F.N1(C(C2(CC(C)C)CC2)=O)CCC(C)(C)CC1 c1(C(N2CC3(C(CNC(CCC)=O)CC3)C2)=O)c(O)cc(=O)n2c1COCC2 N1(C(C(CC)(C)C#N)=O)CC2CCC1(CNC(C1CCC(=O)N1)=O)CC2 c1(C(=O)NCCC(C)NC(c2c(CC)onc2C)=O)ccc(O)c(N)c1 Cn1cccc(C(=O)NCC2CCCN(C(c3cncn3C(F)(F)F)=O)C2)c1=O c1(CC)cc(C(=O)NC2CCCCC2)nn1CCO.C1(C#N)(C(=O)N)CCCC1 CC1CN(C(c2ncccc2C(F)(F)F)=O)CC1NC(=O)Cc1c(Cl)cnn1C c1(C(=O)OC)ccccc1CC(=O)N.C(=O)(C(C)(C)c1cccs1)N(C(C)C)C C1(c2cn(CC(C)C)nn2)CCCCN1C(=O)C(c1ccc(Cl)cc1)(C)O c1(C(N(CCCNC(CCC)=O)C2CC2)=O)sc(-c2ccccc2)nc1C(C)C CCC(C)(C(=O)N1CCN(CCNC(c2csc(-c3ccco3)n2)=O)CC1)OC Cc1cc(C)cc(S(=O)(=O)NC2CC(C(=O)NC3CS(=O)(=O)C3)C2)c1 N1(C(C2(C)CCCN(C(CC(C(C)=O)C)=O)C2)=O)CCc2sccc2C1 C(=O)(CN1C(=O)CCOc2ccccc21)NCC(C)CNC(=O)C1=CCCOC1 c1(C(=O)NCC23CC(NC(CCC)=O)(C2)C(C)O3)cc(Cl)c(O)c(Cl)c1 Cc1ccc(O)c(CNC(C2CN(C(=O)CCN(C)CCO)CC(C)O2)=O)n1 C(=O)CCC(C)S(C)(=O)=O.C(=O)(C(C)(C)C(=O)NC)OCC.C1CC1 c1(OC)ccc(NC2(c3nnnn3C(C)(C)C)CCN(C=O)C2)c(Cl)c1 n1(CCC(=O)NCCC)sc2ccccc2c1=O.C(=O)C(C)(C)C.C(=O)(C)N c1(OC)cnc(Cl)c(NC(=O)C=CC=Cc2ccccc2)c1 c1(NC(N)=O)ccccc1C(=O)NCC1CCC(NC(=O)C2=CCCS2)C1 CC1OC(C)C(C)C1C(=O)NCC=CC.C(=O)(C(=O)Cc1cccs1)N C12(CSC)CC(C(N3CCOC(C(C)NC(=O)C4=CCCC4)C3)=O)(CO1)C2 CCCCC(=O)C(=O)N(CC(C)(C)CNC(=O)CC1(C)CC1(Cl)Cl)C C1(C(N(C)Cc2ccncn2)=O)CC(C)(C)CCN1C(C1CC2OC1C1CC21)=O N1(C(c2c(CC)nc(C)[nH]2)=O)CCN(C(c2cc(F)ccc2Cl)=O)CC1CCO c1(CC=O)cccc([N+](=O)[O-])c1.c1(C(C)OCC)ncc(C(=O)N)s1.CC C12(C(N(C(COC)C)Cc3cccc(Oc4ccccc4)n3)=O)CCCCC1C2 CC1CC(CNC(c2ccc(CO)c(F)c2)=O)CCN1C(c1cncn1C)=O C(=O)(C1CCCc2cc(C#N)ccc21)NCCN(C(C(COC)COC)=O)C C=CC1(C(=O)NC(c2n[nH]c(CC)n2)C)CCN(C(=O)C(C)C2CC2)C1 C1(C(N(CC(=O)NCC(=C)CC)C2CC2)=O)C2CCCCC12 c1(CC)ncnc(CC)c1C(=O)NCC1CC(O)CN1C(=O)CC(O)CC C(=O)(CC(C)CNC(C1C=CCCN1C(c1ccoc1)=O)=O)OC CCC(CCOC)C(=O)NC1CN(C(c2cc(C3CC3)nc(O)c2)=O)CC1F c1(C(=O)NCC(CNC(c2n[nH]c(C)c2Cl)=O)(C)O)cn(C)c2ccccc12 c1(CC(=O)NCC(C(C)(C)C)NC(C(C)C(C)O)=O)ccc(F)c(Cl)c1 CCC(C)(O)CCNC(=O)C(C(C)C)NC(=O)CCNC(N)=O c1(OCC(=O)NC(CNC(CCCC=C)=O)CO)ccc(S(N)(=O)=O)cc1F N1(C(C(CNC(C2C3C4CCC(C4)C23)=O)N(C)C)=O)CC2CCC(O)C2C1 N1(C(C2(CCCC)CCC2)=O)CC2CN(C(c3c(N)cccc3Cl)=O)CC2(C)C1 c1(C(N2CC3=C(C2)CN(C(C2CCCSC2)=O)C3)=O)ncnc2c1OCCO2 C1(NC(c2c[nH]nc2-c2ccc(Cl)s2)=O)CCCC1.C1(CC=O)CC12CC2.C N1(C(C(CC#C)NC(=O)CC2CCCNC2=O)=O)CCCC(C2(C)CC2)C1 N1(c2ncnc(C)c2F)CC2CCC1C1CN(C(c3ccc([N+](=O)[O-])o3)=O)CC21 C1(CC(N2CCC(CC(C)C)C2)=O)(OC)CN(C(=O)CC2(O)CCCC2)C1 C(=O)(C(F)(F)C(O)C(C)C)NCC1C(OC)CCC1 n1(CC)cnc2nc(=NCc3cc(Br)ccc3F)[nH]c(NCCCCCCO)c12 c1(OCCOC)ccc2c(c1)CCN(c1nnc(C3CCCN3C)n1C)C2 C1(C(=O)NCC(c2ccccc2)CNC(c2c(C)onc2)=O)CCCN1C=O N1(C(C(CC#C)O)=O)CCC(NC(=O)CCCOCC=C)C(C)(C)C1 C1(CCC(=O)OCC(O)Cc2ccccc2)CCC(F)(F)CC1 CN1C2CCC1CN(C(C1CC(O)CN1C(C1C=CCS1)=O)=O)C2 C1(=CCNC(Cc2nc(C)sc2)=O)CCN(C(=O)CCC2CCC(=O)NC2)CC1 C1(NC(CCC=C)=O)CC2CCC(C1F)N2C(=O)CCc1ccc(=N)[nH]c1 n1(CC)cc(CC(=O)N(CC=C)CCOC(C)=O)cn1 C1(C(=O)NCC(CNC(C(C)n2cccc2)=O)O)CC2(CCOCC2)CO1 C1(NC(Cc2[nH]n(CC(C)C)c(=O)c2)=O)CCN(C)C12CCCN(c1nnco1)C2 C(C(N=[N+]=[N-])C(=O)NC1(C)CCN(C(c2cc(C)c(F)cn2)=O)C1)OCC CCC(C)(CC)C(=O)NCC1CN(C(c2cccnc2C(F)F)=O)CC1(C)C C1(NC(CC=C)=O)CC2CCC1CN(C(c1ccc(C)c(OC)c1)=O)C2 c1(C(=O)NCCNC(c2c(C)ncnc2O)=O)ccc2c(c1)n(C)c(=O)n2C Cc1cc(CC(=O)NC2CCCCN(C(C3(CO)CCOCC3)=O)C2)cc(C)c1 N(C(=NCc1nc(C(F)(F)F)cs1)N1CCC(F)(F)C1)CC(N1CCCCC1)(C)C N1(C(c2ccc3occc3c2)=O)CCN(Cc2ccccc2)C2(CCCCC2)C1 Cc1cnc(NC(C2CCC2)C)c(S(=O)(=O)N2CCN(C(C)C(F)(F)F)CC2)c1 N1(C(C(CCCC)NC(c2ccncc2F)=O)=O)CC(C)OCC(C)(C)C1 O=S1(=O)CCC(CN=C(NCC2(c3ccccc3)CCCCO2)NC2CCC2)C1 N1(Cc2cccc(C)n2)CC(C(=O)Nc2cc(Cl)cnc2Cl)CC(F)C1 CC(C)(CCCCNC(C1CC12CCCCC2)=O)NC(c1cnccn1)=O C1CN(C(c2cc(F)cc(F)c2)=O)CC(F)(F)C1.C(C(=O)N)NC(=O)NC c1(C(CC)=O)ccc(C(=O)N(CCNC(C2CC2C(N)=O)=O)CC)cc1 Cc1n[nH]c(=NC2CCC(NC(=O)CC3COCC(C)(C)O3)CC2)s1 Cc1cccc(C(=O)NC2CCCCN(C(=O)COCc3ccccn3)C2)c1F c1(OC)ccc(C(=O)NC(C)CC(C)N)c(N)c1Cl n1(CC)cnc2nc(N3Cc4cccc(Br)c4C3)nc(N3CC4CCCC4C3)c12 C#CCCC(O)C(=O)N(C1CCN(C(c2ccncc2C)=O)CC1)CCOC c1(OC)ccc(NC(C2(c3ccc(-c4ccc(CO)o4)cc3F)CC2)=O)c(C)c1 Cc1cc(C(=O)N(C2CCN(C(=O)C(F)(F)C3CCCC3)C2)C)c(C)nc1C C1(C(=O)NCC(N(C(=O)CCc2cn[nH]c2)C)C2CC2)CCOCC12CCCC2 C1(NC(c2c(CNC(=O)CSC3CC3)n[nH]c2)=O)CC2CC1CC2CO c1(OC)c(F)cc(F)c(N2CCC(C)C(NC(=O)C(C)C3CCC3)C2)c1[N+](=O)[O-] C1(C=O)CC(O)C(F)C1.c1(C(=O)NC2(C(C)(F)F)CCC2)coc(C)n1.N Cc1cnc(C)c(NC(=O)C(CC2CC2)NC(=O)CC2CCOC2=O)c1 C1(NC(C2(C#C)CCC2)=O)CCN(C(c2cncnc2C)=O)CC1CO c1(SC)cccc(C(N2CCC(n3cc(CCCCO)nn3)C2)=O)c1C c1(C(N(CC(CN(C(=O)C)C)O)C)=O)ccc(CO)nc1.c1cncc(Cl)n1.O N1(C(C2(C(C)C)CC2)=O)CCOC(CCNC(c2ccon2)=O)C1.C1CC1.C Cc1cnc(C(=O)NC2(CN(C)C(c3cc(Cl)cnc3O)=O)CC2)c(C)c1 c1(C(N2CCC(N(C(=O)C(=O)Nc3ncc[nH]3)CC)C2)=O)ccnnc1Cl C1(C(=O)NCc2n(CCC)cnc2)CCCCCN1C(c1cc(C)nnc1O)=O N1(C(=O)CC2CCN(C(c3ccc(F)c(Cl)c3F)=O)C2)CC2CCCCC2C1 c1(C(N2CCN(C(CCS(N)(=O)=O)=O)CC2)=O)ccc(Cl)c(Cl)c1Cl c1(C(=O)NCC(C)(CO)NC(C2CCN(CC(C)C)C2)=O)cc(Cl)sc1Cl C12(C(=O)NC(C(C)NC(=O)CC3CCOC3)CO)CCCCN1CCC2 c1(N(C)Cc2ncc(C)nc2)cc(N2CCN(C3CCCOC3)CC2)nc(C)n1 Cc1ccnc2c(C(=O)NC3CCCCC3NC(C3COC(=O)N3)=O)cnn12 c1(OC)ccc(CC(N2CCCC2)=O)cc1Cl.C12(C(=O)N)CC(CN1C1CC1)C2 Cc1cc(S(N)(=O)=O)sc1C=O.C1(C)(C(N(CC(C)(C)C)C)=O)CCCC1O Cc1cccc(C(N2CC(F)CC2CNC(c2ccc(C(N)=O)o2)=O)=O)n1 C(CC(CC)(CC)NC(=O)C(c1ccccc1)C)NC(c1ccn(CCC)n1)=O c1(C(N2CCC2)=O)cc(S(N)(=O)=O)c(C)cc1C.C(C)(C)(C=O)OC(C)=O c1(NC(C2CCN(C(CCCOC(C)(C)C)=O)C2)=O)ncccc1C(F)(F)F CS(=O)(=O)n1cc(NC(C2CC2C(=O)Nc2nccnc2Cl)=O)cn1 N1(C(c2nncc(OC)c2)=O)CCC(C2CC2NC(=O)CC2=CCCCC2)CC1 c1(C(=O)N)cncc2nc(C)[nH]c12.c1(SC)cscc1C(=O)NC1CCC1C C1(CC(=O)N(CC(O)CN(C)C(C2(CF)CC2)=O)C)CC2CCC1CC2 c1(CN2C(C(N3CCC(SC)CC3)=O)C(O)CC2)cc(Cl)cc(Br)c1 C1(C#N)(OC)CC(C(=O)N(CC(C)C(=O)Nc2ccc(F)nc2)C)C1 Cc1c(-c2cn(CC(C34CCC(C3)OC4C)=O)nn2)cncc1Br c1(C(N2CC3C(C(=O)Nc4cc(C(C)C)no4)(C3)C2)=O)cc(F)cc(Br)c1F C#Cc1cc(C(=O)NCC(CNC(=O)C(C)(C=C)CC)CO)cc(N)c1 CCCCC(F)(F)C(=O)N1CCC(CNC(=O)C(=O)NCC(F)(F)F)C(O)C1 Cc1cc(C(F)(F)F)ccc1C=CC(=O)Nc1ccnn1CC(C)C C(c1ccc(Cl)cc1Cl)=CC(=O)NC1(CNC(C(N)=O)=O)CCCCC1 C1(CC(=O)N(C)CC2C(C)C2)N(C(C2CC(C3CC3)=NO2)=O)CCC1(C)C c1(-c2n(CC=C)nc(-c3ccnc(N(C)C)c3)n2)cc(F)c(Cl)cc1OC C1(C#N)(C(NC)=O)C(C#N)C1(C)C.C1(C=O)CCN(CCF)CC1.C1CC1.C CC1(C)CN(C(=O)CN2CCCCC2)C(CNC(=O)Cc2cncnc2)CO1 N1(C(c2c(OCC)oc(C)n2)=O)CCCC1(C)C.C1(CC=O)CC=CCN1C.N O=C(C1CCc2c[nH]nc21)NCC=C1CCN(C(c2c[nH]cc2Br)=O)CC1 c1ccc(C=O)cc1.C1(CC=CC=O)CCCC1.CCC.C(=O)OCC.N C(=O)C1=CCc2ccccc21.c1(C(C)C)ncsc1C(=O)NCC1CC1C.N c1(N(C(C(CCOCC)NC(c2nccn2C)=O)=O)C)cccn(C)c1=O c1(C(N2CC3CN(c4cc(N(C)C)ncn4)C3C2)=O)ncc2ccccn12 N(C(=NC)N(C)Cc1cccs1)CC(CC)(C)OC Cc1cc(Cl)ccc1-n1cc(CC2CCCN2C(=O)COC2CCOC2)nn1 c1(C(N2CCCC2(C)C)=O)cc(N)c(Cl)c(O)c1.Cc1nc(C)c(C(=O)N)s1 c1(C(C)=O)ccc(Br)c(C(=O)N(C)CCNC(=O)C(C)(C)C)c1 c1(C(CC)C(=O)NCCC(C)N(C)C(c2n[nH]cc2OC)=O)ccc(OC)cc1 c1(C(=O)NCC(N(C(C(CC=C)C)=O)C)C2CC2)cc(OC)c(OC)cc1F c1(N2CCCC(CNC(c3n(C)c4c(c3)scc4)=O)C2)nc(Cl)nc2[nH]cnc12 C1(NC(=O)CCN2CCCC2)CCCC1CNC(=O)CC(C1CC1)C1CC1 C(CCS(C)(=O)=O)(C(N)=O)c1cc(Nc2ccnc(S(C)(=O)=O)c2)nc(C)n1 C1(N(C(CSCC)=O)C)CCN(C(c2ccc(C#N)o2)=O)CC1C N1(C(C2N(C)CCC2)=O)CCN(C(=O)CCc2n[nH]c3c2CCCC3)CC(O)C1 C(C(CC(C)C)C(=O)N1CCC(c2cnco2)C1)NC(c1c(CC)nc(C)o1)=O N(C1CCc2ccc(Br)cc21)C(c1ncccc1-c1cccc(F)c1)=O c1(OC)ccc(S(C)(=O)=NC(=O)c2ccn3cc(C)nc3c2)cc1 CC#CCCCC(=O)NC1CN(C(C2(C(F)F)CCOCC2)=O)CCC1C C(=O)CC1=NN(C)C(=O)C1.C(=O)(CS(=O)(=O)C1CC1)N(CCC(C)F)CC n1(CC)nc(C)cc1C(=O)NC1CCCC1NC(=O)C=Cc1c[nH]nc1C C(=O)(C(F)(F)C1(O)CCC1)NC1(NC(C(N2CCOCC2)C)=O)CC1 C(=O)(C1Cc2ccccc21)N1CCC(F)(C(=O)NCC2C(C)(C)COC2)CC1 C(=O)(CC(C)(O)CCC)N1CC(CCNC(CCC#C)=O)C(C)C1 c1(C(=O)NC2CC(OC)CN(C(=O)C(C)O)C2)cc2c(s1)-c1ccccc1OC2 c1(C(N2C(CN(C(CC(C=C)(C)C)=O)C)COCC2)=O)ccnc2[nH]ncc12 C1(NC(C2CC(OC)(OC)C2)=O)CN(C(c2oncc2C)=O)CC1C1CC1 C#CC1(C(=O)NCC2CCN(C(C3CC4CC4C3)=O)C2)CCCC1 C1(CNC(CCC(=C)C)=O)CC(NC(=O)Cc2c[nH]nc2C)C12CCC2 CC1(C)CCN(C(C2(F)CCOCC2)=O)CC1.C1(C(=O)N)CC(S(C)(=O)=O)C1 N1(C(c2ccc(C#N)s2)=O)CCN(C(=O)COC(F)(F)F)C2CCCCC12 O=C(N=c1cc(C(F)(F)F)cn[nH]1)C1CCCC(NCc2ccnc(Cl)c2)C1 N1(C(C(=O)N(C)C)=O)CCC2CN(C(c3cc(-c4ccco4)no3)=O)CCC2C1 C(=O)(C1=NN2CC(C)CN=C2N1)N1C2CN(C(c3c(C)scn3)=O)C(CC2)C1 O=C(C1=NOC2COCC12)NCC1COCCN1C(c1cccc2c[nH]nc12)=O C(CC(C(=O)NCC(c1ccccn1)(F)F)NC=O)SC c1(C=O)cc(N)cc([N+](=O)[O-])c1.N(S(=O)(=O)N(C)C)CC=O.C(C)C.C O(P(=O)(Cn1cc(C2CC2)nn1)OCC)CC.C1(C)(C(=O)N)CCC(C)C1 N1(C(C(C)OCC#C)=O)CC(NC(c2nc(OC)ccc2F)=O)CC1(C)C Cc1cccc2ncnc(N3CCC(N(C(=O)C(C)n4ccnc4)C)CC3)c12 C1(NC(=O)CCc2nncn2-c2ccccc2)CCN(C(=O)COC2CC2)CC1 C1(NC(c2n(C)ncc2C2CC2)=O)CC(O)CN(C(c2cscc2F)=O)C1 c1(CC(=O)NC(CCC)CNC(=O)CC2CC3CC3C2)ccccc1OC c1(C(N(C)CCNC(=O)CC2CCC(O)C2)=O)ccc(F)c2cnccc12 C12(CNC(C=NOC)=O)CCCCC1N(C(C13CC1COC31CCC1)=O)CC2 c1(C2CC(NC(C(=O)N(C3CCNC3=O)CC)=O)C2)ccccc1 c1(C2CC2)ccc(C)c(C)c1.c1(C=O)cc(C(=O)NC(C)C)c(C)o1.CO C12(NC(C3CCCN(CCC)C3)=O)CCCC1CN(C(=O)COC1CCOC1)C2 Cc1cc(F)ccc1C(N1CC(C(=O)NC2CCCNC2=O)OC(C)C1)=O N1(C(c2c(CC)con2)=O)CC2(CCOCC2)CC1CC(=O)O C(=O)(C1=CCCCCC1)NCC(CNC(CC1C(C)C(=O)CC1)=O)CO C1(CNC(C=C2CCC(C)CC2)=O)CN(C(c2cncs2)=O)CC1(F)F N1(C(C(c2cccs2)NC(C2C(C)CC2)=O)=O)CC(=O)N2CCCC2C1 C(c1ccc(F)c(Cl)c1)=CC(N1C(CC)CN(C(=O)CC2CC=CCC2)CC1)=O N1(Cc2cn(CC3C(NC(CS(N)(=O)=O)=O)CCC3)nn2)CCc2ccccc21 N1(C(CCC(C)C)=O)CCC(C2CCN(C(C34CCCN3CCC4)=O)C2)C1 C1(CNC(CCc2cc(OC)no2)=O)(NC(=O)Cc2ccco2)CCOCC1 n1(C(C)C)cc(C(=O)N)nn1.c1ncoc1C1CN(C(=O)C(C)C2CCC2)C1.C CC1(C)COCCC1C(=O)NC1COCC1NC(c1coc(C)n1)=O.C1CC1 c1(OC)cc(C)ccc1C(=O)NC1(C)CCCN(C(=O)CCCc2nccs2)C1 Cc1c(C(=O)NCC2CC3(CCC3)CCO2)ccc2c1NCCO2 C(=O)(C1=CCC2(COC2)OC1)N1C2CCN(C(C3CCC(C)(C)C3)=O)CC1CC2 C(=O)(C#CC1(C)COC1)NC1CCCC(C(N2CC=CC(OC)C2)=O)CC1 c1(CCC)nsc(N)c1C(=O)NCCCCC(C)NC(=O)CCc1cnccn1 c1(-n2cc(CN3C(CS(N)(=O)=O)CCC3)nn2)ccn2ccnc2c1 C(CCNC(=O)Cn1ccnn1)(C(C)C)NC(COCC(C)C)=O.CCO C(=O)(C(C)n1cccn1)NCCC1(CNC(C=CCOC)=O)CC1 C1(C(=O)N(C)CCN(C)C(C2CCC2c2ccccc2)=O)CC(F)(F)C1.CC Cc1cc(C)c(C(=O)NCC2C(C)CCN2c2ncncc2I)c(O)n1 c1(C(N2CCC(C)C2)=O)cc(F)c(F)cc1N.c1(COCC)nc(C=O)cs1 c1(C(=O)NCCSCc2cn(C3CC=CC3)nn2)ccc(C2COC2)cc1 C1(CCC(N2CCC(C)C2)=O)CCCCN1C(C1CCN(C)CC1)=O N1(C(COC)=O)CCCC1(C)CNC(c1ccccc1N1CCCC1)=O N1(C(CC2ON=C(C)C2)=O)CCOC(CNC(=O)CCCCN2CCCCC2)C1 O=C1NCC2C(C(=O)NCC3CCCN(C(c4occc4Br)=O)C3)C12 C=C1c2ccccc2C(=O)N1CC(=O)NC1(CCO)CCC(C)(C)CC1 c1(Cc2cn(C3CCN(C(c4cc(C)oc4)=O)C3)nn2)cn2ccccc2n1 C(CC(C)(C)C(=O)NCC1CCCCN1C(c1c(C)nsc1Br)=O)OC c1(C(N(C(CNC(C=C(CC)C)=O)C2CC2)C)=O)ncoc1C1CCC1 c1(C(N2C(C(=O)NCCc3ccn(CC)n3)CC2)=O)ccc(F)cc1C c1(OC)cccc(C(C)NC(C2CCCC2)CO)n1 c1(CC)ccc(C(=O)NCCC2CCN(C(=O)C=Cc3ccco3)C2)c(O)c1 C(=O)(C(CC1CCC1)N1CCC1(C)c1ccccc1)NCCC(=O)OCC.O CS(C)(=O)=NCC(=O)NC1CC(NC(c2cnc(C3CCOC3)s2)=O)C1 c1(Cn2cc(CCNC(=O)OC)nn2)nc(C)oc1C c1(CC)cnc(O)c(C(N2CCCC(C(N3CCOCC3)=O)C2)=O)c1 C(=O)(C(C)(C)C#N)NC(c1ccccc1)CNC(c1ccc(CC)[nH]1)=O N1(C(CCc2cc(C)no2)=O)CC(NC(=O)C(C2CCCCC2)O)CC(C)C1 N1(C(C2(CC)CNC(=O)C2)=O)C2CCC1CCC2.c1(C=O)cnc(N(C)C)o1.N CCC(C)CCCC(=O)NC1CN(C(C2CS(=O)(=O)C2)=O)CC1(C)C C(C(C)(C)C1=CCCC1)NC(c1n(CC=C)nnn1)(CCOC)C1CC1 Cc1nc(CO)ncc1C(N1CC2CC1CC2NC(c1nccn1C)=O)=O C1(C(N2CCN(C(CCC(=O)NCCC)=O)CC2)=O)CS(=O)(=O)CC(=O)N1.C C=CCCC(C(=O)NCCCNC(=O)OC)NC(=O)C(C)O N1(C(C(CSC)O)=O)CC2(CCOCC2)CC1CNC(=O)CCc1ccsc1 C1(C(=O)NC(c2nc[nH]n2)CC)CC=CCC1NC(=O)C1=CCSC1 N1(C(C(C)OCCC(C)C)=O)CCCOC(C)C1.C(c1cccn1C)=CC(=O)N N1(C(CC2CC(=C)C2)=O)CCC(NC(=O)CC2CCC(C(=O)NC)CC2)C1.C Cn1cc(CCC(=O)NC(CNC(=O)C(C)(C)C2CCCC2)CO)nn1 N1(C(C2(C#C)CCN(C(=O)C(F)C(F)(F)F)C2)=O)C2CCC1CC(=C)C2 N#Cc1c(O)csc1C(=O)N.c1(C(CC(=O)N2CCC2)N(C)C)ccc(F)cc1 CC(C)(C(=O)N=c1cc2n([nH]1)CCCC2)C1CCCN(C(c2csc(O)n2)=O)C1 N1(C(C2N(C(c3ccc(OC)o3)=O)CCC2O)=O)CCN(CCO)C(=O)C1 CC1CCCC1(C)NC(=O)CCNC(c1cnnc(O)c1)=O C(N=c1cc[nH]cc1S(=O)(=O)N1CCCC(N(C)C)C1)c1c(OC)c(C)ccc1 N1(C(c2c(CC)noc2)=O)CCCC(NC(c2nc[nH]c2C(C)(C)C)=O)C1C Cn1nnc2c(C(=O)NCCC3CCC3)ccnc12.C1(C)(C=O)CNC(=O)C1.N C12(N(CCCC3CC(C)C3)C(C)=O)CCN(C(=O)CCc3ccncn3)CCC1C2 C(=O)(CCCC(=O)OC)NCC(CC)(C)NC(c1cncc(OC(F)F)c1)=O C1(C(=O)NC2CN(C(C3(N(C)C)CCOCC3)=O)C2)(OC)CCCOC1 C(C(CC1CC1)C(=O)NCC(O)C(C)(C)O)NC(Cc1n(C)nnc1)=O CS(=O)c1cccc(C(=O)NC(CNC(c2c(F)ccc(F)c2N)=O)CO)c1 C1(OCC)COCCC1NC(=O)CC1CC(NC(=O)O)C1.C(C)(C)C n1(CC(=O)N(CC=C)C(c2ccccc2)C)cc(CCCC(=O)OC)nn1 C1(OCCNC(C(C)=C2CCC2)=O)CCN(C(c2ncncc2F)=O)CC1 c1(C(N2C3(CN(C(=O)CSc4ccncc4)C3)CC2)=O)ccc(O)c(O)c1O C(=O)(C1CCc2cccc(O)c21)N1CCC(NC(CNS(CC)(=O)=O)=O)(CF)C1 N1(C(CCC(CC)CC)=O)CCC2CCC(C1)N2C(=O)C(C)CC(C)(C)C C1(COC)(NC(=O)C(C)O)CCN(C(C2CC(C)(O)C2)=O)CC1.C1CC1 N1(C(C(CCC)O)=O)CC2(C1)C(NC(C1CCC3(CC1)CC3)=O)CCS2(=O)=O N1(C(CCCC#C)=O)CCC2CCN(C(c3cc(N(C)C)ccc3N)=O)CC12 C(=O)(CCC(F)(F)C(F)(F)F)N1CC(CNC(=O)Cn2ncnn2)N2CCC1C2 c1(CC(=O)NCC(CN(C(C2CC(OC)C2)=O)C)(C)C)ccccc1C C(=O)(C1=CCCOCC1)N1CCC(C(CNC(C(C)=C2CCCC2)=O)(C)C)CC1 CC1(C)OCCCC1NC(=O)CCC(=O)c1cccs1 C(C(=O)NCc1cc(C(=O)NC2COCCC2O)cs1)(C(C)C)NC(C)=O c1(C(=O)NC2CCN(C(C(CC#C)C3CC3)=O)C2)ccc(S(N)(=O)=O)c(O)c1 CCCC(C(=O)NC(CO)C(=O)NC1(C)CCSC1)C(C)C C#CCCC(O)C(=O)N(CCNC(=O)C(F)OC(F)(F)F)CC c1(C(N2CCC(C(C)C)CC2)=O)cc(Cl)c(F)cc1N.C1(CCC)CC1C(=O)N c1(CC(=O)NCCC2CN(C(C3(C=C)CCC3)=O)CC2C)ccc(O)cc1Cl C1(C(N2CCCC(OC)C2)=O)CCN(C(c2cc(F)cnc2Cl)=O)CC1O N1(C(c2[nH]c(=NC)sc2)=O)CC=C(CCNC(c2sc(C)c(C)c2C)=O)CC1 N(C1CCCc2ccccc21)CCc1nc(C(C)(C)C)sc1.C(C)N CN1CC(C(N2CCCCC2CNC(=O)CCOC2CCOCC2)=O)NC1=O N1(C(c2n(C)nnc2)=O)CCN(C(C2(Cl)CC2)=O)CC2CCCCC12 Cc1cc(=NCCCS(C)=O)[nH]c(=NCCCN2CCN(S(C)(=O)=O)CC2)[nH]1 C(N=c1[nH]c(NC2COCC2F)nc2c1COC2)C1(N(C)C)CCCCC1 N1(C(c2c(C)occ2)=O)Cc2[nH]nc(C(=O)NC(C)Cc3nccn3C)c2C1 N1(c2cc(C)ncn2)CCC2(CNC(c3ccc4c(c3)CCO4)=O)CCCCC12 N1(C(C(n2cc(C3(CC)CC(F)(F)C3)nn2)C)=O)Cc2cccc(OC)c2C1 CC(C)C(C)(O)C(=O)NC(C1CN(C(c2csc(O)n2)=O)CCO1)C N1(C(C(CC)NC)=O)CCOC(CNC(C2(OC)CCC2)=O)C1.c1ccccc1.C C1(C(F)(F)F)(C(N2CC(O)C2)=O)CCC(F)C1.Cc1cc(C(=O)NC)n[nH]1 C(C)(C(C(=O)NCC1CC2CCC1O2)NC(C1CSCC(=O)N1)=O)OC CCCCCCCCC(=O)N1CCC2(CC2C(N2CCC23CCCOCC3)=O)C1 c1(SCC)ccc(C(=O)NC2CCC2)cn1.C(=O)C(C)(C)N1CCCCC1.C N1(C(c2c(CC(N)=O)occ2)=O)CC(C2CN(C(c3cccc[n+]3[O-])=O)C2)C1 C1(CC(=O)NC2CC(C)(C(=O)N(c3ccccc3)CCO)C2)CC(=O)NC1=O CC(=O)C(C)CC(C)C(=O)NC1CCCC(CC(=O)N(C(C)CN(C)C)C)C1 C1(C(=O)NC(CC(C)NC(c2nccc(C)c2)=O)C)CCC2(CC1)COCCO2 CCC(C)CC(=O)N1CC(CNC(c2cc(=O)cc[nH]2)=O)C(C)C1 N1(C(C(CN(C)CC)C)=O)CCOCC(C(=O)N(C2CC2)Cc2nccn2C)C1 C1(CCOC)(NC(c2nnn(C)n2)=O)CCN(C(c2cc(Cl)ccc2Cl)=O)CC1 CC1(C)CN(C(C2CCCN(C3CC4CCC3C4)C2)=O)CCN1CC1CCOC1 N1(C(CN(C2CCC2)C(C2CCCC2C2CC2)=O)=O)CCC2(C=CCO2)CC1 N1(C(c2cccc(C)n2)=O)CC2CCCC2(NC(c2ccc(F)cc2F)=O)C1 CN1CCCC1CCNC(C1(NC(=O)CCc2nc[nH]n2)CC(F)C1)=O C1(C(N(CCN(C)C)CCO)=O)N(C(c2cccnn2)=O)CCCC1(C)C C#CC1(F)CN(C(=O)C=C(C)CNC(=O)Cc2cc[nH]n2)C1 c1(C(=O)N)cncc(C#N)c1.Cn1cnn(CC(=O)NCC2(C)CCCC2)c1=O CCCCC(C)CCC(=O)NCC(CCC)C(=O)NCC(O)C(F)(F)F C1(OC)CCC2(C(=O)NCC(C)NC(=O)Cn3nnc(=N)[nH]3)CC12 C1(C(N2C(C=O)CCC2C(C)C)=O)CC(C)(C)CCO1.C(=O)(CCO)O.CC C#Cc1ccccc1CC(=O)NCC=CC(=O)N1CCC1 N1(C(c2c(C)onc2C2CC2)=O)CC2CCC1CC2NC(=O)CC(C)O CC1CN(C(c2cnc(O)c(F)c2)=O)CCC1NC(=O)C(F)F CC(C)CCCCCC(=O)NC1CC(F)CN(C(C2CC3(CCC3O)C2)=O)C1 C1(NCc2cccc(C)c2Br)CCC2(C1)CN(C(c1ccc(O)c(C#N)c1)=O)C2 N1(C(=O)COc2ccccc2)CCN(S(=O)(=O)CCCCl)C2CC12 CC1CN(C(=O)CCN(C)CCO)CCN1C(=O)CCc1cncn1C c1(OC)ccc(Br)c(NC(C2CC3(C2)CN(C(c2cc(C)ccc2F)=O)C3)=O)n1 CC(c1ccccc1)=CC(=O)NC1CCC(NC(c2cccc[n+]2[O-])=O)C1 c1(N2CCC(CCOC)(NC(=O)C(C)SC)C2)nc(Cl)nc2ccc(Cl)nc12 C1(C(=O)NCC2CN(C(C3(F)C4CCCC34)=O)CCO2)CCCCS1(=O)=O C1(C(=O)NC2CCN(C(c3cn(CCCC)nc3C)=O)C2)CCc2ncnn2C1 CC1Cc2cc(N)ccc2CN1C(C1CC(CN2CCCS2(=O)=O)C1)=O C1(C(NOCC(=O)OC)=O)CCN(C(=O)C#CC2CCCC2)CC1(C)C N1(C(c2cnc3c(c2)COC3)C(=O)NCC=C)CCC(C)CCC1C(C)C N1(C(=O)C(F)CC2CNC2)CCCC(F)CC1 N1(CC(=O)NCC(C)NC(=O)C(C)C2CCCO2)CCOCC1=O c1(N(C(=O)CCc2c(C)nn(-c3ccccc3)c2C)CCC)ccc([N+](=O)[O-])cc1 C(=O)(CCCCCC(C)C)NCC(CC=C)NC(C12CSCC1C2)=O C(=O)(C(C)(C)CC)NC1CCN(CCNC(CC2(C(=C)F)CCC2)=O)CC1.S c1(C(N2C(CC(=O)NCC(CC)(O)CC)CC(O)C2)=O)cc(C)ncc1C CS(=O)(=O)c1ccccc1CN1CC2(CC(NC(=O)CCc3ccoc3)C2)C1 C(=O)(C(F)CC(C)(C)NC(=O)CC1CCCO1)N(CCC#C)CC c1(C(N2CCCC2)=O)cc(C)c(C)nc1C.C1(C(=O)N(C)C)(COC)CCC1 c1(CN(C(=O)CC2CCCN(C(c3cncs3)=O)C2)C)ccc(C#N)cc1 C1(NC(N(CCCOC)C)=O)CCN(Cc2ccnc(SC)c2)CC1 c1(C(=O)NCc2cnc(CC)[nH]2)ccc(C)cc1.c1(CC=O)cccnc1.N N1(C(=O)NC(C)Cc2ccccn2)CC2CCC1(C(=O)O)C2 CC(C)(C)CC(C)(C)C(=O)NC1CCN(C(=O)CC2CCC3(CCC3)O2)CC1 C1(C)(CNC(C(n2cc(Cl)cn2)C)=O)CCCN(C(C2CCCCS2)=O)C1 c1(NCC(CO)OC)cc(S(=O)(=O)N2CCC(CC(F)(F)F)C2)ccc1C#N C1(C(CN(C(C(C)=C2CCCC2)=O)C)C)CCN(C(=O)CC2CC(C)(C)C2)CC1 Cc1ccc(F)cc1C(=O)Nc1nn(-c2ccccc2)cc1Br Cc1nccc(C(N2CC(NC(c3sc(N(C)C)nc3Cl)=O)CC2C)=O)c1C CC(C)C(C)CC(=O)NCC1(CC(=O)NCc2ccc(O)cc2F)CC1 c1(C(c2n(CCC)nnn2)NCC(CC)OC)ccc2c(c1)CCO2 C1(CC(=O)NCC(C)N(C(c2cc(Cl)cs2)=O)CC)CCC12CCC2 Cc1cc(OCC(=O)NC(C)C)cc(C)c1Cl.c1(CC=O)nc([N+](=O)[O-])n[nH]1 C1(NC(C(CC#C)C2CC2)=O)CCN(C(=O)C=C(C)C2CCCCC2)CC1CO CCC(F)(F)C(C)(C)C(=O)N1CC(O)(C(C)NC(=O)C(C)(C)C2CC2)C1 C=CCC(CC)C(=O)N1CC2C(CC(=O)N(CC(N3CCCC3)C)C)C2C1 Cc1ccc(C(=O)N(C2CN(C(=O)C=C3CCCC3)C2)C)c(C(C)C)n1 C=C(C)CC(C)C(=O)N1CCCCC(CNC(C2(CC)CCC2)=O)C1 C1(CC(=O)O)CN(C(=O)CN(CC(C)C)C(C2CC2(C)C)=O)C1.CC C(=O)(C1CCOc2c(F)cccc21)NC1CC(CNC(C2OCCN(C)C2)=O)C1 N1(C(C)=O)CCC(CN(C)C(C2CN(C(=O)C(C)C)C2)=O)C1 C(CCCCCCC)c1ccc(NC(=O)NCCN(C(COCC=C)=O)C)cc1 Cn1cc(CC(=O)NC2CCCC2NC(c2nc[nH]c2C(F)(F)F)=O)c(Cl)n1 C1(C(=O)NCCNC(C(C(C)(C)C)c2ccccc2)=O)Cc2cccnc2C1 c1(OC)ccc(C)c(OC)c1C(=O)N.C1C2CN(C(=O)Cn3cnnc3O)CC12 C(CC(=O)NC1COCCC1NC(c1coc(Cl)c1)=O)(C(N)=O)NC(C)=O N1(CC)CC(C(N2CCC2CC(=O)NCc2cccnc2O)=O)CC1=O C1(NC(C2C(C)OCCC2)=O)CC2CC(C1)N(C1CCN(C3CCC3)C1=O)C2 c1(NC(C2(CO)CCN(C(CCCCC)=O)C2)=O)cn(C)c(=O)cc1C N1(C(C2N(C)CCCC2)=O)CC(C2CC2)(C(N2CCC(CC3CC3)C2)=O)C1 CC(N)(Cc1ccc(OC(F)F)c(F)c1)C(=O)N1CCCCCO1 c1(N(C)Cc2ncc(Br)cn2)nc(Nc2nccn2C(F)F)nc2c1ncn2C C(N=c1ncc(I)c[nH]1)C1C(NC(C2C(CC)OCC2)=O)CCC1 N1(C(CC(OCC)O)=O)CC(NC(=O)CC2CC3C=CC2C3)CC(C)C1.C C(=O)(C(C(=O)O)C(=O)NC(=O)OC(C)(C)C)OC.c1(CC)ccccc1 C=CCC(CC(=O)NC(CO)C(C)C)NC(=O)CCC(C)(C)N(C)C c1(C(=O)NC2C(NC(C(F)=CC)=O)CC2)ccc(OCC)cc1 CCC(CC)C(C)C(=O)N1CCCN(C(=O)CCc2ccc(N)cn2)CC1CO C(=O)(CCCCCC(C)O)N1C(CN(C(COCCC(C)C)=O)C)CCC1 c1(C(=O)NCC2(O)CCN(C(CCC3C(C)(C)C3)=O)CC2)nccc2ccsc12 C(=O)(C(C)CC(C)(F)F)NCCC(C)N(C(c1c(C)nc(C)o1)=O)C N1(C(c2cn(CCOC)nc2)=O)CCN(C(C2(CCF)CCC2)=O)CC1 N1(CC)CC2(CC(Nc3ccc(C(=O)O)[nH]3)C(O)C2)C1C(C)C C(=O)(C#CC1CCCC1)NCC1CCN(C(C(c2cccc(C#N)c2)C)=O)C1 c1(OCC(C)C)ccc(Cl)cc1NC(C1C=CCNC1)=O C1(C(=O)NC2CN(C(C(C)NC(N)=O)=O)C2)CC(S(C)(=O)=O)C1 c1(C(=O)N)csc(C(F)F)n1.C(=O)(C(=O)N(CC(C)C)C)NCCOC c1(NC(=O)NCC2CC(=C)C2)ccc(OCC)c(OC2CCCC2)c1 c1(C(=O)NC2CCC(NC(C(CCC)OC)=O)CC2)cnc2c[nH]nc2c1 CN1C2CCC1CC(C(N1CC3CC(O)C3C1)=O)C2 c1(NCCC(CCC)C)ncc(S(=O)(=O)NC2(C3CC3)CCCCCC2)cc1Cl C1(NC(C2CC(C)=C(C)CC2)=O)CN(C(c2sncc2C)=O)C2(CCOCC2)C1 Cc1ccc(COC(=O)CCC2CCCN(C(=O)OC(C)(C)C)C2)cc1C c1(CNC(c2nnn(C)n2)c2nnnn2C)c(F)c(F)c(Br)c(F)c1F N1(C(CC2(OC)CCCC2)=O)CC2CC2(NC(=O)C(C(C)C)c2ccncc2)C1 c1(C(=O)N)cnc2[nH]nnc2c1.C1(CC(=O)NC2CCCC2C)NC(=O)NC1=O CC(C)C(O)CC(=O)N1CCCC(NC(=O)CC2(N(C)C)CCC2)CC1 N1(C(c2c(C)scn2)=O)CCCCC12CC(NC(C1(F)CC=CC1)=O)C2 C12(C(=O)NC(CC(C)NC(c3cncc(CC)c3)=O)C)CCCCC1OCC2 c1(NC(C2CN(C(c3ccc(C#N)cc3)=O)C2)=O)c(F)cc(Cl)cc1F CCC(C)CCC(=O)NCCN(C(=O)Cc1ccc(F)cc1C)CC N1(C(C(CC=C)(C)C)=O)CCC2(CCCC2NC(c2cnc(O)n2C)=O)CC1 C1(NC(CC(N)=O)=O)CCCC(NC(=O)CNc2ccccn2)C1 c1(NC)nc(C)ccc1NC(C)(CNC(=O)C)C(C)C.c1n[nH]c(O)n1.S c1(N(C(c2cc(SC)nn2C)C(=O)NC)CCC)ccc(Cl)cc1 c1(OC)ccc(C#N)cc1NC(C1(C)CCCN1C(c1cnccn1)=O)=O c1(C(=O)NC2(CC=C)CCCN(C(=O)CCCCC)C2)nn(C)c(=O)cc1C C(CS(=O)(=O)CC(=O)N1CCC(N(C)C(c2cn(C3CCOC3)nn2)=O)C1)OC Cc1cc(COC(=O)COc2ccsc2Cl)cc(C)c1Br C(=O)(C1=CC(O)CCC1)N1CCC(NC(c2c(C)n(CC(F)(F)F)nc2)=O)C1 c1(C(N(CCC(=O)NCC2CC(C(C)C)C2)CC=C)=O)cc(Cl)cs1 N1(C(C=CC=CC)=O)CC2CC(NC(c3ccc(OC)nn3)=O)C(C2)C1 N1(C(=O)NCC2OCC(CC(N)=O)C2)CC2CCN2C1 Cc1cc(C(N2CCCC2C(C)(C)C(=O)NC2CNC(=O)C2)=O)c[nH]c1=N C1(C(=O)NCCC(C)N(CCC)C)(C)CC2(CC2)C1.c1(C=O)cc[nH]n1 N1(C(C2CN(C(C)=O)C2)=O)C2CCC(C(=O)NC)C1CC2.C1CC[Si](C)(C)C1 O=C1COCC2(CN(C(=O)C(CC3CCC3)NC(c3csnn3)=O)C2)N1 N1(C(c2c(Cl)ncc(C)c2)=O)CCC(O)(C2(NC(=O)C3=CCCCC3)CC2)CC1 c1(C(C)N(C(=O)C(n2cc(CN3CCNC3=O)nn2)C)C)ccc(Cl)c(Cl)c1 N1(C(C(C2CCC2)OCC)=O)CCN(C(c2cc(C)nnc2O)=O)C(CC)C1 c1(C(N(CCC(C(C)C)NC(COCCCC)=O)C)=O)csc2nccn12 N1(C(c2cn(CCC=C)nn2)=O)CCCC(COC)(NC(=O)C)C1.C(C)CC c1(C(N2CCC(C)(NC(CCn3ccc(C)n3)=O)C2)=O)cc(O)ccc1Cl Cc1n[nH]cc1C(=O)NC1CCC1NC(c1c[nH]nc1C)=O C(=O)(C(C(C)(C)C)OC)NC(C(=O)NC(CN(CCCC)C)C)CN(C)C CCCCCCC(F)C(=O)N1CC(C)(NC(C2CCC2C(=O)OCC)=O)C1 c1(C(N2C3(CNC(CC=C=C)=O)CCC3CC2)=O)cc2c(OC)cccc2s1 c1(C(=O)NC(C(C)NC(=O)COCP(C)(C)=O)C)cncc2[nH]ccc12 CC1CCCCC1(C)C(=O)NCC(C)(C)CNC(c1cnn2ccsc12)=O C#Cc1cnn(C)c1C(N1CC2CCC2(C)C1)=O.c1(C=O)coc(C(F)F)n1.N C12(C(=O)N)CCN(CC1)CC2.C(CC(C(C)C)NC(C12CC(C1)C2)=O)OC Cc1c(Cl)cnn1CC(N1CCCC1CNC(C1CC1C1CC1C)=O)=O c1(C(N2CC(F)CC(NC(C3CC3(Cl)Cl)=O)C2)=O)nccc2n[nH]cc12 N#Cc1cccc(C(=O)N)c1.C1(O)CC(C=O)C1.C1(CC2CCC2)CCC1.C C1(CNC(CC23CC(C)(OC2)C3)=O)CCN(S(C)(=O)=O)CCC1(F)F Cc1nc(-c2nc(-c3sccc3Br)no2)ccc1-c1cnn(C)c1 CC(C)(C)C(=O)C(=O)N1CC(F)(C)C1.c1(C(=O)N)ccc(C(F)F)c(Cl)c1 N1(C(c2cc(C)sc2N)=O)C(C(=O)N(C2CC(C)(C)C2)C)CCC12CC2 Cc1cccc(Cl)c1C(N1CCCC(NC(c2nc(Cl)cs2)=O)CC1)=O C1(C(N(C)CC)=O)CC(C)(C)CCN1C(=O)CCC1CCOC1 C(=O)(C(C)(C)CC(C)C)NCC=CC(=O)NCCC c1(C=O)ccc(C(C)(C)C)cn1.C1(NC(COCC(C)C)=O)CCCC1C C12(NC(CCOCC)=O)CCCN(C(c3ccc(-c4ccsc4)nc3)=O)CC1C2 Cc1ccc([N+](=O)[O-])c(NCC2CCCN2C(c2c(O)nnc(C)c2C)=O)c1 Cc1ccc(CC(=O)NCc2ccoc2C(N2CCC(CC(C)(C)C)C2)=O)s1 c1(C(=O)NC(CCNC(CCC=C=C)=O)(C)C)cnc2[nH]c(C)nc2c1 c1(C(=O)N)ccc2c(c1)C(=O)NC2.c1(C(N(CCC)CC)=O)snc(O)c1Cl C1(CN(C(=O)Cc2cncnc2)C)CN(C(=O)C(F)(F)c2nccs2)CC12CC2 N1(C(C=COCC)=O)CC(CNC(=O)CNC(C2CCCC2)=O)C(O)C1 Cc1cc(C)c(C(N2CCCC(C)C2)=O)cn1.C(=O)(CC1(C(F)(F)F)CC1)N C1(NC(C(C=C=C)C)=O)CC2(NC(=O)COc3c(C)ncnc3C)COC1C2 c1(C(=O)NC(C)C(C)(C)NC(c2cscn2)=O)cc2c(Cl)cccn2n1 N1(C(c2ccsc2)=O)CCN(C(=O)C(C)=CC(C)(C)C)CC1C(F)F.CO.C C1(c2cn(CCC(=O)OC)nn2)CCN(Cc2cc(C(C)C)cc(O)c2)C(C)C1 C=CCC(C(=O)NC(C)CCCNC(=O)Cn1nc(C)ccc1=O)C(C)C O=C(CC1=CCCC1)N1CCC(OCCNC(c2cc3cscc3s2)=O)CC1 C1(CCNC(c2ccc(-c3cn[nH]c3)cn2)=O)CN(C(c2cscn2)=O)CCO1 C1(CNC(COCCOC)=O)COC(C)C1.n1(CC=O)nnc(=N)[nH]1 CC1(C)CC(O)(C(=O)NCC2CCCCC2)C1.c1(C=O)ccc(C(F)F)cn1 CCS(=O)(=O)CCN=C(NCC1CCN(C2CC2)CC1)NCC1CCC1 c1(C(=O)NCC(CC)NC(=O)C(O)(CC)c2cccs2)cc(Cl)cc(Cl)c1 C1(CC)CN(C(=O)CCc2cn[nH]c2)CCC1CNC(c1ccsc1)=O C1(CC(=O)NCC2(C)CCCO2)CCCCC1.c1(C=O)ccc(C(N)=O)[nH]1.N c1(OC)cnc(C(=O)NCC2CC2C)cn1.c1(C(=O)N)ccc(=N)[nH]n1 Cc1cc2c(-c3ccc(C(=O)Nc4c[nH]nc4C)nc3)ncnc2[nH]1 N1(C(C(C)NC(CC)=O)=O)CC2(CO)CC1(C(N1CC(O)(C3CC3)C1)=O)C2 C1(C)(COC)CN(C(=O)CC2CCCC2NC(=O)Cc2ccoc2)C1 N1(C(c2n(CC=C)ccn2)=O)CCC2(CCCCN(C(=O)C(C)C3CCC3)C2)C1 c1(C(=O)N)cc(S(N)(=O)=O)sc1Cl.Cc1nnccc1C(=O)NC(C)C(C)C N1(C(CCCc2scc(C)n2)=O)CC2CC(C1)N(C(c1ccsn1)=O)C2 c1(C(N2CCN(C(C3CCC3)=O)CC2CC(F)(F)F)=O)ccc2cc[nH]c2c1 c1(C(N(CCNC(c2c(OC)cc(C)cc2)=O)C)=O)ccn2ccnc2n1 CC1CCCCN1C(=O)CS(=O)(=O)NC.C1(C=O)CCN(C(=O)C2CC2)CC1 C1(C)(NC(CCCCN(C(=O)CN(C)C2CC2)C)=O)CCC(C)(C)C1 C1(CCCNC(CSCCCC)=O)CCCN1C(=O)Cc1c[nH]nc1C c1(C(N(CC(C)NC(=O)C(c2nc(F)ccc2Cl)C)C)=O)cc2n(n1)CCCO2 C1(N(C(C(C)CC2CCC2)=O)C)CCN(C(C2CN(C3CCCCC3)C2)=O)CC1 C1(NC(C(CCC)C)=O)CCC(O)CN(C(=O)CC(C2CC2)C2CC2)C1 c1(OCC)cccc(C(=O)NC(CNC(c2cc(C)co2)=O)CO)c1Cl C1(F)(CNC(C2(CC#C)CCCC2)=O)CCCN(C(=O)C(CC(=C)C)O)CC1 c1(OC)ccc(C)cc1C(=O)NC1CC(NCc2ccc(C)o2)C1 c1(C(CN(C(N(c2nc[nH]n2)CCC)=O)C(C)C)O)ccoc1 N1(C(C23C(CN(C(=O)Nc4ccc(CC)cc4)C2)C3)=O)CCC(F)(C=O)CC1 C(=O)(C(C)CC(C)(C)C)NC(CCCC(=O)NCc1c(OC)nn(C)c1)C C1(C(=O)NC2(CC=C)CCOC2)CN(C(=O)C(N2CCCCC2)C)CCN1C c1(C(=O)NC2C(C(=O)Nc3cc(C)c(O)cc3C)C2)cccc2ncccc12 C1(O)(C(C)NC(=O)C(=O)N(C)C)CN(C(=O)C(F)(F)c2ccccc2)C1 CC(C)(C)C(O)C(=O)NC(C)(CNC(=O)COc1cn[nH]c1)CO C1(C(N(CC(CCC=C)O)C)=O)CC(N=[N+]=[N-])CN1C(C1CS(=O)(=O)C1)=O N1(C(C23CCN(C(CC(CC)C)=O)CC2C3)=O)CCC2SC(=O)C=C2C1 Cc1cc(C(=O)N(CCCNC(c2cc(S(C)(=O)=O)co2)=O)C)cc(C)c1Cl c1(C(=O)NCC(C)CN(C(=O)C(C)(C)N(C)C)C)cc2c(Cl)nccc2s1 Cc1cncc(C)c1C=O.C(S(C)(=O)=O)C1(CC(=O)NCCC)CC1.C N1(C(CSC)=O)CCC2CN(C(=O)COCC(c3ccccc3)C)CC2C1 O=C1OC(CNC(c2scnc2Cl)c2nnnn2C2COC2)CC12CC2 C1(C(=O)NCC2OCCN(C(C(C)SCCCC)=O)C2)Cc2ccc(C)cc2S1 c1(CC)cc(C(N2CC(F)CC2C(=O)N(C)CCc2ccccc2)=O)nn1C C1(N(C)C)CCC(N=c2[nH]c(=NCC(C)(C)C3CCCO3)[nH]c3c2CCC3)CC1 N1(C(Cc2nc(C(=O)O)sc2)=O)C2CCC(C2)C1C(N1CCC(Cl)C1)=O c1(C(N(CC(O)CN(C)C(C2CCC(F)C2)=O)C)=O)cc(C2(C)CC2)n[nH]1 C1(NC(C(=O)NCCOCC)C)CC2(CCCCC2)C1.C(c1cnc[nH]1)=C C1(NC(CC(C)SC)=O)CCN(C(c2[nH]c(C)nc2C)=O)CC(C)(C)C1 Cn1cc(C(CO)NC(C2CC(NC(=O)Cc3cnsc3)C2)=O)cn1 c1(C(=O)NC2(CNC(c3cc(C)sn3)=O)CC2)cc2cc(Br)ccc2o1 C1(NCC(C(c2n(-c3c(C)cccc3)nnc2)(C)C)=O)CCCCC1C#N N1(C(CCCOC(C)(C)C)=O)C2CCC1(CNC(=O)CCC1CCOC1)CC2 C1(N(C(C(c2ccccc2)C)=O)CCO)CCN(C(=O)Cn2cnnc2O)CC1 N1(C(c2n(C)c(Cl)cn2)=O)CC2(CC(NC(c3cc4cscc4s3)=O)CO2)C1 c1(C(=O)N)ccc2nn[nH]c2c1.C1(NC(c2ccncn2)=O)CC2(C1)CC(C)C2 c1(NC2CCN(CC)C2)nc2ccccc2nc1N(CC(=O)NCC(F)(F)F)C C(=O)(CC(C)(C)C)NC1CN(C(c2cc(C)nnc2)=O)CC1CO.C(N)(=O)N N1(C(C2CSC2)=O)CC23CCCCC2(C1)CN(c1nnc(C2CC2)s1)C3 c1(OC)ccc(C(N2CC(O)(C3CCCN3C(C3CC(O)CN3C)=O)C2)=O)nc1 C12(NC(c3c(C)nc(CC)s3)=O)CCCCCC1N(C(c1nncn1C)=O)CC2 c1(C(c2nnnn2C(C)(C)C)NC2CC(CC)OCC2)c(F)ccc(NC)c1F N1(C(=O)OC(C)(C)C)Cc2nccc(C(N3CC4OCOC4C3)=O)c2C1 C1(C(N(CC(CC)O)C)=O)CCC2(CC2)N1C(=O)CC1CCOC1 C1(NC(CCNC(CC(CC)OC)=O)=O)CC2CCCCN2C1 CC(CCC(C)(C)C)C(=O)N1CC(C)C(F)(F)C1.N1(CC(=O)N)CCC(O)CC1 c1(CNC2CCC(CC(=O)NCC3CCO3)CC2)c(O)cccc1O C=C=CC(C)C(=O)N1CCCC(CCNC(c2ccc(SC)o2)=O)C1 C12(NC(C3C(C)(C)C3)=O)CCC1CN(C(=O)CN1CCCCC1=O)C2 Cn1cnc(C2CCNCC2)c1NCc1cscc1Br c1(C=O)cc(F)ccc1N.Cc1ccncc1CSCC(=O)NCC1CC1.C O=C1CCc2ccc(C(N3CCOCC3CNC(C3CC4CC3C4)=O)=O)nc2N1 c1(CC)cc(Br)ccc1C(N1CCN(C(=O)COc2ccccc2C)C2CC12)=O N1(C(CC(=O)NCC)=O)CC2CC(NC(c3cccnc3OC)=O)C1C2 C(=O)(NNc1cc(O)c(Cl)cc1F)c1cc(OC)c2c(n1)cccc2 Cc1ccc(C(=O)NCC2CCCN2C(=O)Cc2cn(C)nc2C)c(Br)c1 C12(C(=O)OC)CCC(C(=O)N(CCO)Cc3ccsc3Br)(CC1)O2 N1(C(C(CCCC)O)=O)CCC(C)N(C(=O)Cc2ccn(C3CCCC3)n2)CC1 C1(C(=O)NCCCCCNC(c2csc3nnsc23)=O)C2CC3CC(C2)CC1C3 c1(C(=O)NCCN(C(=O)C(C)OCCOC)CCC)cc(F)ccc1F N1(C(c2ncc(CC)s2)=O)CCC(OCCCNC(=O)C(C)CSC)CC1 C1(CCOC)CCCCN(C(c2csc([N+](=O)[O-])c2)C(=O)NC(C)C(=O)OC)C1 N1(C(Cn2ncc(C#C)c2)=O)CCC2CN(C(=O)CC(C)(C)OC)CCC2C1 c1(C(=O)NC2(C)CN(C(c3cnoc3C3CCC3)=O)C2)cc2c(cc1Cl)OCO2 Cc1nc(CNCC2(C(=O)N(C)Cc3cnco3)CCCC2)sc1C CC1CNC(=O)CN1C(=O)C(Cc1cc[nH]n1)NC(C1CCCCC1)=O C1(F)(C(N(C)Cc2cn[nH]c2)=O)CCCN(C(=O)CCc2ccccc2)C1 [N-]=[N+]=NCCCC(=O)N1CCC(CCNC(C2CCCN2C2CCCCC2)=O)C1 Cc1cc(CNC(c2nnnn2C2CCOC2)C2CC=CC2)sn1 C1(C(=O)OC)CN(C(=O)CO)CC1O.c1(C(N2CCCC2)=O)cc(C)c(C)[nH]1 C1(CNC(c2c(CC)noc2)=O)CC(C(=O)NC(CCO)c2ccco2)=NO1 c1(OCCC)ccc(C(=O)NC(C)C(C)NC(c2nccnc2C)=O)c(O)c1 Cc1ccccc1C(C)C(=O)NCCC1CCCN(C(c2nc(=O)n(C)[nH]2)=O)C1 Cc1ccc(C(N2CC(NC(=O)CC3(C)CC3)CCC2C)=O)cc1C(C)(C)C C1(NC(c2cc(C)no2)=O)CCCCC1NC(=O)C(F)(F)c1cncs1 N1(C(C2(C)C(CC)CCC2)=O)CCC(O)(CNC(c2nc(Cl)ccc2Cl)=O)CC1 C1(O)(CNC(CCC#C)=O)CCCN(C(=O)CCC(C)(C)N2CCOCC2)C1 CC(F)(F)C(F)C(=O)NCCn1cc(C(=O)NC)nn1.c1ccc(C#N)cc1 CCCCCCC(C)NC(C1CCN(C(=O)CCc2nncs2)C1)=O c1(C(C(=O)NCC(F)F)N(CCCCCCC)C)c(C)nn(C)c1C N1(C(c2ccc(OC)nn2)=O)CCN(C)C(CNC(C2CCCCC2C)=O)C1 C1(NC(C2(CCC)CC2)=O)CN(C(C2(COC)CCCCO2)=O)CC12CCC2 C1(C(=O)NCCNC(c2c(C)cc(O)nc2)=O)CCCN2CCCC12.C1CC1.C N1(C(=O)Cc2ccc(Cl)c(Cl)c2)CC2(CCN(C(C3CC34CC4(F)F)=O)C2)C1 c1(N2CCC(C(C)(C)NC(CSCCCC)=O)CC2)nc2cccc(C)c2o1 c1(N2C(CCCNC(C3CC(C(C)C)OCC3)=O)CCC2)ncc(C#N)cc1Cl c1(CNC(COC(CNC(C(N2CCOCC2)C)=O)(C)C)=O)ncc(F)cc1F c1(C(=O)NCC(CNC(C2N(C)CCC2)=O)F)cc(C2CC2)nnc1O C1(NC(Cc2ccc(C)cc2)=O)CN(C(c2nn(C)cc2Cl)=O)CC1C1CC1 c1(C(N(C)C)=O)ccc(C(C)(C)C)cc1.C(c1nc[nH]n1)=CC=O.C1CC1 c1(OC)cccc(C2(C(N3CCC3CNC(C3CCOC3=O)=O)=O)CC2)c1 C1(NC(C2CCCSS2)=O)CCN(C(=O)Cc2cnns2)CC1F c1(NC(c2c(C)ccs2)=O)ncc(C)cc1Cl.N12CCC(O)(C1)C2=O C1(NC(C2CCC3CC23)=O)C2CC1N(C(c1cc(C3CCCC3)[nH]n1)=O)C2 c1(CCC(N2C(CCNC(c3ccnc(C)n3)=O)CCC2)=O)c(C)ncnc1O C=CCC(C)(CC=C)NC(=O)CC1(NC(=O)C2=C(C)OCC2)CCC1 C1(CCCCNC(c2cccc(CO)n2)=O)CCN(C(=O)Cc2ccsn2)CC1 C1(NC(C(C#C)(C)C)=O)CC2CN(C(c3cc(Cl)c(F)c(Cl)c3)=O)CC2C1 C(=O)(C(C)CC(F)F)NC1(CF)CCN(C(CN(CCCCCC)C)=O)C1 C1(C(=O)NC(c2ncccn2)C)C2CCC(C2)N1C(=O)CCc1cn(C)nn1 CC1CCC2(CC1)CCC(COC(=O)CCc1cc(Br)ccc1F)O2 O=C1CC2CC(C(N3CCC4(NC(C5CCCCCC5)=O)CC4C3)=O)C1O2 C(C(C(=O)N1CC2(NC(c3cncs3)=O)CCC1C2)C(C)(C)C)OCC=C.O c1(C(C)NC(c2scc(C)c2)c2nnnn2C2CC2)cccc(C)c1C c1(OCC)ccccc1C(=O)NCC1CCC1.C1(CC(=O)N)CCCSC1 O=C1CCC(C(=O)NC2C3CC2N(C(c2ccccc2[N+](=O)[O-])=O)C3)=NN1 C1(NC(=O)CC2C(NC(c3ccoc3Cl)=O)CC2O)CC2CCCCC12 C(=O)(C(O)CC(F)(F)F)NC1(CC)CCN(C(c2ccc(CO)c(F)c2)=O)CC1 c1(OC)c(C(N2CCC(C)(NC(=O)CCCC(N)=O)CC2)=O)c(C)nn1C CCCC(CNC(=O)OC(C)(C)C)C(=O)N1CCOC(CC)(CC)C1 CC(O)CCC(=O)NCC1(CCNC(c2ccnc(N(C)C)c2)=O)CC1.C c1(-n2ccc(C)n2)ccc(C(=O)NCCNC(=O)Cc2ccc(F)cc2)cc1 c1(OC)cccc(C(=O)N(C2CCN(C(=O)C(F)(F)CN(C)C)CC2)C)n1 C12(NC(C3CC(F)C3)=O)CCC1CN(C(c1cc(N3CCOCC3)ncn1)=O)C2 Cc1nn(C)cc1CCC(=O)NCC1(C(=O)Nc2cccc(F)n2)CC1 C(CCC(C(=O)N(CCF)CCOC)NC(=O)C(C1(O)CCCC1)F)OC Cc1nc2n(n1)CC(C(N1CC(F)(F)CC1C)=O)CC2.c1(C=O)ccn(C)c1.N C1(OC)(CNC(N2CCC(CN3CCCC3=O)C2)=O)CCOC(C)(C)C1 N1(C(C)=O)Cc2nccn2CC(NC(c2c(C)cc(C)nc2S)=O)C1 c1(C(=O)NC(C2CCCN2C(=O)C=CCO)C)ccc2ncnn2c1 c1(NC(N2CCCC(OCCCC)C2)=O)cc(C)ccc1COC c1(C=O)cc2n(n1)CCO2.C1(O)(CNC(C=CCOC)=O)CC(C)C1 c1(C(=O)NC2CCCN(C(C(CC)n3cccn3)=O)CC2)cc(C)c(N)cc1Cl C(C1CCCCCC1)=CC(N1CCC(NC(=O)CCCc2cccs2)(CF)C1)=O C1(NC(C(C)=CC)=O)CS(=O)(=O)C2CN(C(=O)CC3CCCN3C)CC12 CC(CNC(=O)CCC(N)=O)CC(=O)NCCN1CCOCC1C C(CSC)(CN=c1[nH]c(=NCc2ccc(Cl)nc2C)[nH]c2c1COCC2)OC c1(CC(N2CC(NC(C3OCC(C)C3)=O)C2)=O)cc(F)c(F)cc1F C(=O)(C(F)(F)C(O)C1CC1)NCC#CCNC(C(C(C)C)O)=O c1(C(=O)NC2CCCN(C(=O)C3=COCC3)C2)ccn2ncc(Br)c2c1 C1(NC(CNS(CC)(=O)=O)=O)CCCN(C(C2CCS(=O)CC2)=O)CC1F C=CCC(C(=O)N1CC(N2CCCC2=O)C1)NC(=O)Cn1nnnc1C C1CCCN(C(=O)C(CO)N(C)C)C1.C1(C(N(C2CC2)CC)=O)CCSCC1 C(=O)(C1CCc2cc(F)ccc21)N1C2(CN(C(C=C(C)C(C)(C)C)=O)C2)CC1 C(CCCCCCCCO)c1nc(C(CCC)CC)on1 N1(C(C2N(C)CC2)=O)CC(CNC(c2cc3cccn3cn2)=O)CC(F)(F)C1 C1(CC)C(C(=O)Nc2cnccc2C)CCN1C(c1cc[nH]c1)=O C(=O)(C(C)CC(C)(C)C)NCC(CC=C)NC(c1ccnn1C1CCOCC1)=O CC(C)C(CO)C(=O)NCCCCC(C)NC(c1cncc(N(C)C)n1)=O N#Cc1c[nH]c(=NC(=O)C2CC2C(N2CCC3(C2)CC3(F)F)=O)cc1F N1(C(C2CCC(OC)CC2)=O)CCCC2(CCCCC2NC(C2CCCS2)=O)C1 C1(CNC(C(N2CCC(O)CC2)C)=O)CN(C(c2cnns2)=O)CCCO1 C=C1CCN(C(=O)CC2CC(F)(F)C2)C(C(=O)NCCC(O)C(=O)OC)C1 C1(NC(C2CCC(CNC(CCNC(C)=O)=O)O2)=O)CC(C)OC1=O c1(C(=O)NC(CN(C(=O)Cc2cccs2)CC)C)cccc2ncccc12 C1(C(C)C)CCCCCC1NC(=O)N(C)C.N12CCC(C1)n1cc(nn1)C2 C1(CC(C)(C)C)CCCCN1S(=O)(=O)CC1CC12CC2 c1(C(C(=O)OC)NC(C2(CC(F)F)CCC2)=O)cccc(Cl)c1 c1(Nc2c(C(=O)Nc3cc(C)cc(C)n3)n[nH]c2)ncnc2cnn(C)c12 c1(CC(=O)NC2C(C)CN(C(=O)CC3CCOC3(C)C)C2)ccc(C#N)nc1 CC1=CCC(C)(C(=O)NCCCN(C)C(c2cc(F)n[nH]2)=O)CC1 CCCC(O)CC(=O)NCC1(CCC)CCCC1.C(=O)CN(C)C(=O)C1CC1 N1(C(c2ccc(C(N)=O)nc2)=O)CCC2(CCCC2NC(=O)CC)C1.C1CC1.O CCC(CNC(c1cccn1C(C)C)=O)(CC)NC(=O)CC(C)(C)F c1cc2nccnc2c(NC2C3C4CCC(C4)C23)n1 c1(C(C)(C)OC(C)=O)cn(CC(C)(C)CNC(C2CCS2(=O)=O)=O)nn1 C1(CC(=O)OCC)CCC(C)N(C(=O)C=CC=O)C1.c1ccc(F)cc1.N c1(C=O)coc(S(=O)(=O)N(C)C)c1.CCCCC.C1(C(=O)N)CC1.N(C)C N1(C(CCCC(C)=O)=O)CCC(C)(C)C(C(=O)NCCC2CCCC(C)C2)C1 C1(Cc2scc(C(=O)OC)n2)(NC(=O)C(S)C(C)C)CCC(C)(C)CC1 c1(C=O)nc(C)n(C)c1C.Cc1cc(C(=O)NCC2CC2)nn1C(F)F.N c1(C=O)cccc(C(F)F)c1F.C1(C(N(C)CC2CC2)=O)CC(=O)N(O)C1 c1(C(c2n(C3(C)CC3)nnn2)NCC2CC23CCCC3)cnc2n1CCC2 C1(C)(C(N(CCNC(C(OC)OC)=O)C)=O)CCOC1 C1(CNC(c2c(C)ncn2O)=O)CCCN(C(C2(C)CCCOC2)=O)CC1 c1(C(=O)NCC2(O)CN(C(C3CCC(C)(C)CC3)=O)C2)ccc2nc[nH]c2n1 N1(C(c2n(C)nnc2)=O)CCCC2(CC(NC(c3csc(C(N)=O)n3)=O)CO2)C1 N1(C(CCC=C)=O)CCCC(C)(C)C1C(=O)N1CCCCCO1 c1(OC)cccc2nc(NC(=O)NCC3CC(=O)NC(C)C3)sc12 N1(C(CCc2ccc(C#N)cc2)=O)CC2CC1CN(C(=O)CC(O)C1CC1)C2 c1(C(=O)NCC(C)(C)NC(C2CC(n3cccn3)C2)=O)ccc2ccccc2n1 C1(N(C(CCC2CCC2)=O)C)CC(C)OC(C)C1.C(C=O)(C1CCC1)OCC.N c1(OC)cc(OC)nc(N(CCC2CCCNC2)C(c2ccc(Br)cc2I)=O)n1 c1(C(=O)NCC2CN(C(CCC(=O)OC)=O)C3C2C3)cc2cccc(Cl)c2s1 C1(C(=O)Nc2cccc3c2OCC3)CCC2(CCN(C(C3(F)CCC3)=O)CC2)O1 N1(C(C=C=C(C)C)=O)CC(O)CCC1C(N1CC(S(C)(=O)=O)C1)=O C1(CNC(C(C)(O)C2CC2)=O)(NC(=O)C(O)Cc2cnc[nH]2)CCOCC1 c1(OC)cc(C(=O)NCC2(C(N3CCC(C(C)(C)C)C3)=O)CCC2)[nH]n1 c1(C(N2CCC(NC(CN(CC)CC)=O)CC2)=O)nn(C)cc1S(N)(=O)=O C1(C(=O)OC)CCN(C(=O)C2CCC(NC(=O)CC3CCC(=O)CC3)C2)O1 C(CC(C(=O)NCCN(C1CCCC1)C(C1CCC1C)=O)OC)OC N1(C(c2c(CCC)onc2C)=O)CCC(C)(C)C1.C12(CC(=O)N)CCCC1C2 N1(C(C2N(C(C(CC)CN(C)C)=O)C(C)C2)=O)CCC(F)(F)C(F)C1 C1(C(N(CCC)CCC)=O)COCCC1NC(=O)C=Cc1cncn1C Cc1c(C(=O)NCCC2CSCCN2C(=O)C(N)=O)[nH]c2cc(F)cc(F)c12 C(=O)(C1=CCCO1)N(C)Cn1cccn1.CC(CC(=O)N1CCCC1)c1ccncc1 c1(C(=O)N)cnc2c(cnn2CCC(C)C)c1.C(C(O)C(=O)NCC(C)C)SC C=Cc1ccc(C(N2CC3C(CNC(=O)CS)C3C2)=O)cc1.c1cnn(C)c1 C(=O)(C1COc2ccccc21)N(C)CC1(NC(C2CC3CCCCC23)=O)CC1 Cc1cc(C)c(C(N2CC(CNC(C3(CO)CCC3)=O)C2)=O)c(S)n1 CC1CCN(C(c2cn(C)nn2)=O)C1CNC(c1cc(-c2ccccc2)ns1)=O c1(C(N2CCC(CC(=O)N(CC(C)O)CCO)C2)=O)cc(F)c(F)c(F)c1F C#CCC(C(=O)OCC)NC(=O)C(CNC(c1cnccc1C)=O)OC O=C1CCC(C(=O)NC2CCCC2NC(=O)C(c2ccc(F)cc2)F)CN1 N1(C(C2C(CC)N(C(=O)COCCCOC)CC2)=O)CC(F)(F)CC1CO C(C1c2ccccc2CCN1C(c1cnn2c1CCCC2)=O)NC(C=C(C)C)=O c1(C(NC2CCN(C(=O)C=CC(C)C)C2)=O)ccc2[nH]ccc2n1.C(C)=O c1(C(=O)NC2CN(C(c3nc(COC)sc3)=O)C2)c(C)n[nH]c1C(F)F O=C(C(CCc1ccccn1)N1CC=C(Br)CC1)NCc1ccccc1 c1(C(=O)NC2CC(CNC(C(C(=O)OC)OC)=O)C2)cccc2c1OCC2 c1(N2CCOCCC2)ncnc2sccc12.C1(N(C)CCO)CCNC1 N1(C(CCC2N(C)CCC2)=O)CCCC(C)(C)C1C.S(S(C)(=O)=O)CC(=O)N c1(C(N2CC=CC(NC(COC3(C)CCC3)=O)C2)=O)cc(F)c(F)c(F)c1N c1(C(=O)NCCN(C(=O)CC2(COC)CCCC2)CC)cc(C)sc1C C1(CC)CN(C(=O)CCOCC(C)(C)C)CCN1C(c1cncc(O)c1)=O Cc1cc(C(=O)NC2CCC(N(C(=O)C(F)C3CC3)C)CC2)sc1C N1(C(c2cc(OC)ncn2)=O)CCC(C=CC(=O)NC)CC1.C1(C)CCCCC1 c1(C(=O)NC2CCN(C(CCCC=C)=O)CC2CO)cc(Cl)cc2cccnc12 N1(C(CCCNC(=O)OC)=O)CCCC2(C)CCCC12.C(=O)C.[SH](C)(=O)=O c1(CC(N2CC(CNC(C=C(C)Cl)=O)C(C)C2)=O)cc(Br)ccc1C c1(OC)ccc(OC)c2nc(Cl)c(CNCCC(c3ccc(Cl)c(Cl)c3)O)cc12 N1(C(CSc2n(C)ccn2)=O)CC2CN(C(C3CCC=CCC3)=O)CC2(C)C1 c1(OC)cccc(OCC(=O)NCCC(C)NC(=O)CC2C=CCCC2)c1 c1(C(CNC(c2n(CCOC)nnn2)c2cnc(SC)s2)C)cccc(F)c1 C1(NC(CC(C=C)C)=O)CCC2(CCN(C(=O)CCn3nc(C)cc3C)CC2)C1 C1(C(=O)NC2CCN(C(=O)CN(C(=O)COC)C)C2)(CC)CC1(F)F N1(C(Cc2ccc(C)cc2)=O)CCCC2CCN(C(c3cc(C)ns3)=O)CC12 c1(CONC(c2ccn(CCNC(C3CCS3(=O)=O)=O)c2)=O)cccc(O)n1 C1(C(N2CCC(NC(CCc3ncc(C)[nH]3)=O)CC2C)=O)CN2CCCN1CC2 c1(C(=O)NC2C(Nc3c(OC)cncn3)CCCC2)cccn2c(O)nnc12 c1(C(=O)NC2(C)CN(C(c3c(-c4nc(C)sc4)c[nH]c3)=O)C2)ccc(C)c(C)c1 C1(CNC(c2cccc(-c3nc(O)n[nH]3)c2)=O)CCCN(c2ncc(Br)cn2)C1 c1(C(=O)NCCCC=C)cc(-c2cccs2)n(C)n1 CC(C)CC(CNC(=O)CC1(O)CC1)NC(=O)C(C)Cn1cccn1 C1(C(N(C(C)C(=O)NC2CC(Cl)C2)CCC)=O)CCC(C)(C)OC1 c1(C=O)nn(C)c(=O)cc1C.N1(CC)CCOC(C(=O)NC2CC23CCC3)C1.N CCCCC(=O)C(=O)N(CCCCCC(=O)NCC1CC(=O)N(C)C1=O)C Cc1nc(CNC(=O)C(F)(F)CO)oc1C(=O)NCCc1cncn1C C12(NC(c3ccnc(S)c3)=O)CCC(CN(C(C3CCC3(F)F)=O)C1)C2 C12(C=O)CC(C1)C(C(F)(F)F)O2.C(=O)(C=CCO)N(C)CC.CC.O c1(-n2cc(C3N(C(C4CC(C)SCC4)=O)CCC3)nn2)ccccc1[N+](=O)[O-] C=CCC(CC)C(=O)NCCC1CN(C(=O)CCSC2CCCC2)CCO1 C(Cc1cn[nH]c1)(C(=O)NCC1CCC1)NC(=O)Cc1csnn1.C1CC1 C1(C(=O)NCC2=C(C)CCC2)CCC(C)CN1C(c1cc(C)cc(C)c1)=O CC1CCN(C(=O)CN2CCC(CO)CC2)C(C)C1NC(=O)CC1CCCC1 c1(OC)ncccc1-c1nc(NC(c2[nH]nnc2C)=O)cs1 c1(N2CCC(C(=O)OC)C2)cccc(NC(=O)Nc2nccc(OC)n2)c1 N1(C(C(CSC)(C)NC(=O)CC2CC2(C)C)=O)CCC2(CNC(=O)N2)C1 N1(CCC(=O)NC(c2cn(C(c3ccccc3)C)nn2)C)CCOC1=O Cc1nc2cncc(C(=O)NC3(C)CN(C(=O)CC45COC(C)(C4)C5)C3)c2[nH]1 N1(C(c2c(C)cccn2)=O)CCC(C)C(NC(=O)Cc2cnccn2)C1 CCC(C#N)(CC)C(=O)NC1C=CC(CNC(c2cc(C)c(F)cc2Cl)=O)C1 C12(CC(N3CC(NC(Cc4ncc(CC)[nH]4)=O)C(C)C3)=O)CCCN1CCC2 C(=O)(C#CC1CCCCO1)NC1CC2(CN(C(CCCN(C)C)=O)C2)OC1 O=[N+]([O-])c1ccc(Cl)cc1OCCNc1cnn(-c2ccccc2)c1 CC1CCCCN1CCC(N1CCCC(NC(=O)CSCc2cccs2)C1)=O C(=O)(C1CCCc2ccnn21)NC(C(C)NC(c1cccc(F)c1F)=O)CO Cc1cnc(N2CCC3CC23)c(S(=O)(=O)NC(C)CCCCO)c1 C(=O)(C(C)(C)S(=O)(=O)C1CC1)N.N1(CC)CCOC(C(N2CC=CCC2)=O)C1 c1(N(C)C)cnc(C(=O)NCC2CCN(C(C3(CC(F)F)CC3)=O)C2)cn1 C1(C(=O)NCC2CCN(C(CNC(CC)=O)=O)C2)CC2(C1)CC(O)C2 C1(C(=O)OC)CC2CC1CN(C(c1[nH]cnc1C)C(=O)NCCCC1CC1)C2 CC(C)(C(=O)NC1CN(C(c2ccc(-c3ccccn3)o2)=O)C1)C1CCOCC1 c1(OC)ccc2c(c1)OCC2CC(=O)OCC1CC(Cl)=NO1 C1(C)(NC(C=C(CCC)C)=O)CCN(C(C2(C)CCC2)=O)C1.c1cccc(F)c1 C(=O)(C1=Cc2ccccc2OC1)NC1CC2CN(C(c3c(C)ocn3)=O)CC21 C1(O)(C(=O)NCCC(=C)CNC(=O)CCSCCC)CCCC(C)(C)C1 C12CCC(CC1)N2.C1(N(CC)CC)CCN(S(C)(=O)=O)C1 C(CC(=O)N1CC(CN=[N+]=[N-])C1)(C(C)(C)C)NC(CC=CC(C)(C)C)=O N1(C(=O)CN2CCS(=O)CC2)CC2CCCC(C1)N2C(=O)C1=CS(=O)(=O)CCC1 N1(C(C=C(C)C)=O)CCC(C2CCCN2C(=O)Cc2cncnc2)C1 c1(C(=O)NCCn2cc(-c3cn(CCSCC)nc3)nn2)cc(NC)ccc1Cl C1(F)(CNC(C2(CC#C)CC2)=O)CCCN(C(=O)CC=CC)C1 C(=O)(C1=CC2(CCN(C(=O)C=CCO)C2)C1)NC(Cc1c(C)noc1C)C Fc1ccc2c(c1)OCCCC2Nc1cc(NC2CCC3(CC3)C2)ncn1 Cc1ccc(C2CC2C(=O)NCC2CCN(C(c3ccc(C)s3)=O)CC2)cc1 c1(CC)cccc(C(=O)NC2CN(C(=O)C(c3ccccc3)C)CC2SC)n1 c1(OC)ncc(C(=O)NCC)c(C(F)F)n1.C1(CC=O)CC(=O)NC1=O.N Cc1cc(C)c(C(=O)NCC(C)(O)CNC(C2CC23CC3)=O)c(N)c1 c1(C(=O)NC2CCN(C(C3(CC#C)CCCC3)=O)C2)ccc2nccnc2c1 c1(C(=O)NCC2C(C)CCCN2C(C2CCCC2(C)C)=O)cc2c[nH]cnc-2n1 N1(C(c2cnc(C)n2C)=O)CCC(C)(C)C1CC(N1CCCC(CC(C)C)C1)=O C1(C(N(C(C)CNC(c2ccc(=N)[nH]c2)=O)C)=O)CC12CCC1(CC1)CC2 N1(C(c2cn(-c3c(C)cccc3)nc2)=O)CC2CC1CN(C(c1cnsc1)=O)C2 C1(C)COCCN(C(C2COC2)=O)C1.c1(CC(C)C)cc(C(=O)NC)cc(O)n1 N1(C(C=C2CCC(C)C2)=O)CC2C(CNC(C3CC3)=O)C2C1.c1ccccc1 C#CC1CCCC(CNC(C2CN(C(=O)CSc3cn[nH]c3)CCN2C)=O)C1 c1(C(=O)NCC(CC(C)C)NC(=O)CC(C)(C)C)nnc(O)cc1O CC(O)C(C(=O)N1CCC(NC(C2(C)CC2)=O)C1)N(C)C c1(C(N2CCC3(C2)CC3)=O)c(O)nnc(C)c1C.C(=O)(C(C)C(=O)N(C)C)OC N1(C(CC(C(C)C)C)=O)CCC2(CCCN(C(C3(C(C)(F)F)CC3)=O)C2)C1 N1(C(c2ccon2)=O)CC2(CCC2NC)C1.C(C)(C)(C)OC(C)C.C=O c1(C(N2CCC(C)C(NC(C3SCCS3)=O)C2)=O)[nH]nc2cnccc12 C1(C(N(C2CCN(CC(=O)NC3CCCCC3)C2)C)=O)CCc2cncn2C1 CC(CC(=O)N1CC(F)(C(=O)N(C2CCOC2)C2CC2)C1)n1cccc1 C1(C(N2CCC(F)(CO)C2)=O)(NC(C(NOC)=O)=O)CCc2cc(Br)ccc2C1 C(C(C)(CC(C)C)NC(c1cn(C2CC2)nc1C)=O)NC(C(OC)OC)=O Cc1cc(C)c(C(=O)NCCC2CCC(NC(=O)C3=CCCCO3)C2)cn1 C1(C(=O)NCC(CCOC)O)COc2cc(F)ccc2O1 CCC(CC)(C(=O)N1CC(=C)CC1C(=O)Nc1cc(Br)cc(Cl)n1)C(=O)O N1(C(C(C)SC(C)C)=O)CCC2(CCCN(C(c3nc(Cl)cs3)=O)C2)CC1 CC1C(C=CC(=O)NC)C1(Cl)Cl.N1(CC=O)CCS(=O)CC1.C1CCCC1 c1(C(=O)NC2CCN(C(C(C)CCO)=O)CCC2CO)cccc2cnccc12 c1(CN(C(C)C(C)OC)C(CC)C)cccc(Br)c1C c1(CC)nc(O)c(C(N2CCC(COC)(NC(c3ccoc3)=O)C2)=O)cc1C C1(N(C(=O)CC2CCOC2)CC)CCC(NC(=O)Cc2cc(C)on2)CC1 C1(C(N(CC)CC2CCOC2)=O)CCN(C)C1.N1(CCC(=O)N)CCOCC1 CCC(CC(=O)NC1CCC(F)(CNC(=O)CCc2nc(=N)[nH][nH]2)C1)C(C)C c1(C(N(C2CCN(C(=O)C=CC(C)C)C2)CCC)=O)cccc2cnsc12 C1C(C(=O)NC(C)C(C)C)NC(=O)C=CC(=O)O1.CCOCC C1(C2CCC2)(C(=O)NC2CCCN(C(C(CN(CC)CC)F)=O)C2)CCC1 c1(CC(N2CC(NC(CSCC)=O)CC3(C2)CC3)=O)c[nH]c2c(O)cccc12 Cc1cc(Br)ccc1CCC(=O)NCCN(C(=O)C(C)c1ccon1)C C(=O)(C1=CC2(CCOC2)C1)N1CC(NC(C2CCC(C(N)=O)CC2)=O)C2(C1)CC2 c1(OC)ccc(C(F)F)cc1C(=O)NCC1CCC1.C1(C=O)CC(C)CO1 CN1CCC(C(N2CCC(CO)(CNC(C3(C(F)F)CCC3)=O)C2)=O)CC1 CCCC(C(C)(C)C)NC(C1(CNC(=O)CCCOC)CC2(CC2)C1)=O C1(NC(C(C)=CC2CC2)=O)CC12CCN(C(=O)C(N1CCCCC1=O)C)C2 c1(C(N2C(C)CC(NC(c3c(C)cnc(F)c3)=O)C2)=O)cnc2n1CCOC2 N1(C(c2nc(OC)oc2)=O)CCC(O)(CNC(C2CCS2(=O)=O)=O)C1 c1(OC)ccn2ncc(C(N3CC(N4CCC(C(=O)O)CC4)C3)=O)c2c1 C1CC(C)CN(C(=O)CN(C(=O)CC2CC(N(C)C)C2)C2CCC2)C1.CO N=c1cc(C(N2CCC(CCNC(C3CCCC3)=O)CC2)=O)c(Br)c[nH]1 C(=O)(C(CC(C)C)C(N)=O)NC1CCN(C(c2c(OC)c(C)ncn2)=O)CC1F c1(C(=O)NCC2OCCN(C(COCC=C)=O)C2)cc2n(n1)CCC2 C1(OC)(OC)CCSCC1NC(N1CCC2CC1CO2)=O N1(C(c2ccn(C)n2)=O)CCC(N2CCC(N(CCO)CC3CCC3)CC2)CC1 C1(C(=O)NC(c2ccncc2)C)CN(C(C2(Cl)CCC2)=O)CCN1C C1(CNC(C(C)c2ccco2)=O)CN(C(=O)CN(C2CCC2)C)CCO1 c1(C(c2nnnn2CCC)NC2C(C=C)COC2)ccc2c(F)cc(F)cc2n1 C(=O)(C1=CC2CC(C1)CC2O)N(C1CCN(C(c2c(CC)nc(C)n2C)=O)C1)C c1(N2CCCC(CSC)C2)nc(=NCC2CCC=CO2)[nH]c2cccnc12 Cc1cc(N)ccc1C(=O)NC1CC(C)N(C(=O)Cn2cc(CO)nn2)C1 CC(C)(C(=O)NCC)N1CCCC1.c1(CC(N2CCC2)=O)cc(C2CC2)no1 C1(OC(C)(C)C)COCC1C(=O)NC(=O)CC1CCC2CC12 N1(C(C(C2CC2)OC)=O)CCC(C)(NC(C2(NC(N)=O)CC2)=O)CC1 Cc1ccn(CC(=O)N(C2(C(=O)NC3CCCC3C)CC2)C)c1 C#CC1(O)CC(C(=O)NCc2ccnc(C(N3CCC(C(C)O)CC3)=O)c2)C1 c1(NCCC2C(C)C2)ccn2ncc(S(=O)(=O)NCCN(C)CCO)c2n1 c1(OC)cccc(NC(=O)CC2C3CCCC3N2C(=O)C(C)(C)CCSC)c1F C1(C(=O)NC(CC2CN(C(CCC(=O)OC)=O)C2)C)CCn2nncc2C1 N1(C(C(CSC)OC)=O)CCOCC1CC(=O)NCC(O)C(C)(C)O c1cc(C(N)=O)[nH]n1.n1(C(C)C=O)cc(CC(C(=O)O)C2CC2)nn1.C(C)(C)C Cc1cc(C)c(C(=O)NC2CC(CCNC(=O)CC)C2)c(C)n1.C1CCOC1 C1(NC(C=C(C)C(F)F)=O)CCCCCC1NC(=O)C(F)C(C)(F)F C1(C(=O)N)CC(c2cn(C)nc2C)=NO1.C1(OC)CC(C(=O)NCC(C)C)C1 C1(NCc2cc(C(F)(F)F)c(Cl)nc2)CCNC2(CCCC2)C1 CCC(C)C(C)N=c1[nH]nc(Cc2cccnc2)s1 C1(C(N2C(CC(=O)N)COCC2)=O)C2CC3C(C2=O)C13.c1(CCC)ncnn1C CC1CCN(C(c2ccc3[nH]ncc3c2)=O)CCN1C(=O)CNc1ncccn1 C12(CNC(CCCNC(C)=O)=O)CCC1CCN2C(=O)CCCC.C(N)(=O)N C1(C(C)(C)NC(C(C)=C(C)C)=O)CCCN1C(=O)C(F)CC1CCOC1 CC(C)CC(C)CC(=O)N1CC2CC2(CNC(c2scnc2C(F)(F)F)=O)C1 C1(C(N2CCC(=CCC)C2)=O)CCS(=O)(=O)CC1 N1(C(c2nc(Cl)cs2)=O)CC2CCCN(C(c3coc(CO)c3)=O)C2C1 c1(CC)nn(C)c(C)c1CC=O.c1nnc(C(F)(F)F)s1.N1CCC1.C1CC1 C1(c2ccc(Br)cc2)(CN(C2(CC)CC2)C)CCCCC1 CC(C)CC(C)(CNC(c1csnn1)=O)NC(=O)CCc1nc(C2CC2)no1 CC1=C(C(=O)NC2CS(=O)(=O)CC2NC(C2CC23CCCCC3)=O)COCC1 n1(CC=O)[nH]cc2c(=O)ncnc1-2.C1(NC(C2C(C)C2)=O)(C)CCOCC1.N c1(C(=O)OC)cc(C=O)c(C)s1.c1(C=O)nc(C(C)C)oc1C.CC(F)C.N c1(NC(c2nnc(O)n2C)c2n(CCOCC)nnn2)ccc(Cl)cc1CO C(C(C(=O)N1CCCCC(NC(c2cnoc2C2CCC2)=O)C1)C(F)(F)F)OC c1(N2CCCC(CN(C(c3cc(SC)oc3)=O)C)C2)ncc(C)c(SC)n1 c1(CCCC(N2CCC(NC(C=C(C)C(F)F)=O)C2)=O)c(F)cccc1F CCC(COC)C(=O)NCC1CCCN(C(c2sc(C(F)(F)F)nc2C)=O)C1 CC1CN(C(=O)CCc2c(Cl)cncc2Cl)CCC1NC(=O)C=Cc1ccoc1 N1(C(C23N(C(C(CC(CC)C)=O)=O)CCC2C3)=O)CCC2CCC(C1)N2C C(=O)(C1=CCC2CCC1N2C(=O)C(C)N1CCCC1)NCCC=C=C N1(C(C(C)OCC#C)=O)CCCC1CCC(=O)NC(C)(C)C c1cccnc1.c1(CCC(=O)NCC2(CN(C(=O)C)C)CC2)ccccn1 C(=O)C(C)(C)S(=O)(=O)C1CC1.CC1CCCC(OCC(=O)N)C1.C1CC1.C Cc1cc(O)ccc1C(=O)NCC1CCCCN(C(c2ncnn2C(C)C)=O)C1 C1(NC(c2c(C)nc(C3CC3)o2)=O)CCN(C(C2(C)CCC(O)CC2)=O)CC1C c1(NC(=O)NC(c2ncc(C(=O)OC)s2)C)cc(S(C)(=O)=O)ccc1F C1(NC(c2n(CCC)ncc2)=O)CCN(C(=O)CCC(=O)N(C)C)CC1F Cc1cc(NC(=O)CC2CC3(CC3)CN2C(=O)CC(O)C(C)C)cc(O)c1 c1(C(CSC)NC(N(C2CCN(S(C)(=O)=O)C2)CC)=O)ccccc1.O Cn1cnc2c(C(N3CCC(OC4CCOCC4)C3)=O)cccc12 c1(CC(=O)NCCCNC(c2c(C)occ2)=O)ccc(F)cn1.C1CCCC1.C C(=O)(C(C)(C)CCNC(=O)C(C)NC(C1(C2CCCO2)CC1)=O)OC c1(C(=O)NC(C2(O)CN(C(c3cc(C)ns3)=O)C2)C)cn(C)c(C(F)F)n1 C1(OCC(=O)NCC2(C)CCCC2)CCCOC1.C12(C=O)CC(C1)C2.N C#CCCC(C(=O)NC(C)CCC(F)(F)F)NC(c1cc(COC)[nH]n1)=O C(=O)(CCCCC)NC1C(NC(c2ccc(C(=O)OC)nc2)=O)C1.C(N)=O C(=O)(C#CC(C)(C)C)NC(CC)(C)CNC(c1ccon1)=O C1(CNC(C2(CCOC)CCCC2)=O)CC(C)CCN1C(c1cnc[nH]1)=O N1(C(CC2C(CC)C2)=O)CCC(C(C)(C)NC(c2cn(C(C)C)cn2)=O)C1 C1C(C2CC2)CCN1C(c1ccc(=NC)[nH]c1)=O.C(C)(C=O)NC(=O)NC.N C1(C(N(CCNC(=O)Cc2csc(-c3ccoc3)n2)CC)=O)CCCCC1O C(c1ccccc1Cl)=CC(=O)NC1C(NC(c2csc(C)c2C)=O)CCOC1 N(C)(C(=NCCCCl)NC1CSCC1C)CCNC(C)=O C1(C)(C(N(CC)CCO)=O)CCCN1C(=O)C.c1(C=O)cc(C)oc1C.C C1(NC(CC(C)F)=O)CN(C(=O)CCc2ccc(C(F)F)cc2)CC12CC2 N1(C(CC=C(C)C)=O)CCC2CCC(C1)N2C(C1CC(C)(C)CCO1)=O n1(CC)ccc2c(C(N3CCC4(CCSC4)CC3)=O)cccc12 c1(C(N(C(CCNC(c2c(CCC)nns2)=O)C)C)=O)ccnc(CC)c1 CC1OCCN(C(C23CC(CO)(CN2C(C2C4CCCOC24)=O)C3)=O)C1CO c1(CC)cccc(C(=O)N(CC(=O)N(CC(CC)OC)C)CC)n1 C1(C(C)NC(C2(CO)CCCO2)=O)CN(C(=O)C)CCO1.c1ccc(F)cc1.O C(c1ccc(Cl)cc1F)=CC(=O)NC1CCN(C(c2cccc3ccnn23)=O)C1 c1(C(=O)N)cc(O)cc([N+](=O)[O-])c1.C(C(C(=O)NC1COCC1)N(C)C)OC Cc1nc(C(=O)NCC2CCCN2C2CCCCC2)nn1-c1ncccn1 C=C1CCN(C(C2CCN(C(C)C)C2)=O)C(C(N2CCC(CCO)C2)=O)C1 C1(NC(C(C)CN(C)C)=O)CC2CCCC2C1.C(=O)C=CC=O.C1CC1.N C(CCC(=O)N(CCCn1cc(C(C)(C)OC)nn1)C1CC1)N(C(=O)OC)C N1(C(C2C(CCC)C2)=O)C2CCC1C(NC(c1ccc(F)c(C)c1)=O)C2 N1(C(CCN(CCCCC)C)=O)CC2(CO)CC(c3ccc(F)cc3)(C1)C2 c1(C(N(CCCNC(c2cc(-c3ccco3)on2)=O)C)=O)nnc2ccccn12 c1(C=O)cc(S(N)(=O)=O)n(C)c1.C=CCC(F)(F)C(=O)N1CCC(C)C(C)C1 C(=O)(C1=CC(O)CCC1)N1CCC(O)(CNC(C(=O)NCC)=O)CC1 Cc1ccnc2c(-c3cccc(CN)c3)cccc12 c1(C(N(CCCNC(C2(O)CCC(CC)C2)=O)C)=O)c(C)ccc(OC)c1N C(=O)(C(C)(C)CC(F)F)NCCCCCNC(c1cc(C)[nH]c1C)=O O=C(CC1=CCCC1)NC(CC1CCCC1)C(=O)NCCOC1CCC1 CC1CCCCN(C2CNC(c3nc(C(=O)OC(C)(C)C)no3)C2)C1 N1(C(CC(C)NC(C(CC)NC(C)=O)=O)=O)CC(C)c2ncccc21 N1(C(c2c(CNC(c3ccc(O)c(F)c3)=O)ocn2)=O)CCC2CCCC2CC1 N1(C(c2c(OC)n[nH]c2)=O)CCN(C(=O)C)CC1.N1(CC=O)C(=O)CCC1=O N1(C(Cn2c(=O)sc(C)c2C)=O)CCC(C)N(C(c2cc(C#N)no2)=O)CC1 C(=O)(C(C)(C)CC(C)C)N1CCC(CC=C)C1.C1(C=O)CCCN1C(=O)CC C1(CNc2ncc(C)cn2)COCCN(C(C2CCN2C(C)(C)C)=O)C1 C1(CC)CC(C(=O)NCC2CCN(C(=O)CCC3NC(=O)NC3=O)C2)CCO1 C(=O)C(C)(C(F)F)c1ccccc1.C1(NC(C=CC=CC)=O)CCCCC1.N C1(NC(C2C(C)=CCS2)=O)CC(C(N2CC(N(C)OC)C2)=O)C12CCC2 N1(C(COCCC)=O)CC2(CCCC(C)O2)C1.c1(C2C(C=O)C2)cccnc1.N C(=O)(C1=C(C)CCOC1)N1C(CCOC)CN(C(C2SCCCS2)=O)CC1 CCCCC(O)CC(=O)NC1CC2(C1)CC2C(=O)NC1CCCC1(F)F C(=O)(C1=COCCC1)N(CCOCCN(C)CCC1CCOC1)C C(C)(C)(CCC)NC(C(C1CCCO1)OC)=O.C(=O)(CC=CC(C)(C)C)N N1(C(c2cc(C(=O)OCC)on2)=O)CCCC(C)C1.C1(CC=O)C=CCC1 C(=O)(C(O)C(F)(F)F)NC(C(N1CC(=CCC)C1)=O)C1CC1 C1(C#N)(C(N2CC(F)(CNC(CN3C(C)CCC3C)=O)C2)=O)CCOCC1 N1(c2cc(C)c([N+](=O)[O-])cc2)CCOC2(CCC(NC(c3cscn3)=O)CC2)C1 Cc1ccc2oc(C(=O)NCCC3CCN(C(C4CC5C=CC4C5)=O)C3)cc2n1 N(C(=NCCCN1CCCC1)NC1COCC1F)C(C)Cc1ccccn1 c1(C(N2CC(C3N(C(CC4(C#N)CC4)=O)CCC3)(O)C2)=O)cc(F)ccc1Cl c1(C(=O)NCCc2n(CC)cnn2)ccncc1.C(=O)CN(C)C1CC1.C C1(O)(CNC(C2(OCC)CCC2)=O)CCCN(C(=O)C(O)CF)CC1 C#Cc1c[nH]nc1C(=O)Nc1cccc(CNC(C2(CC#C)CCCCO2)=O)c1 N1(C(C2N(C)CCOC2)=O)C2CCC1C1CC1C2.C1(C(=O)N)CN(S(N)(=O)=O)C1 c1(C(=O)NC2CC(C)N(C(=O)CCC(C)(C)O)C2)c(F)cc(C#N)cc1F c1(N2CCC(CNC(N(CC)CC3CCN(C)C3)=O)C2)cccc(Cl)c1 Cc1cc(C(=O)NCC)ccc1S(C)(=O)=O.C1(C)(C=O)C(C)(C)C1(C)C.N N1(C(c2c(N)c(F)cc(F)c2)=O)Cc2ccnn2CC(NC(c2cn[nH]c2)=O)C1 C1(N(C)C(c2cnon2)=O)CCN(C(=O)CCc2ccc(O)cc2)CC1 C1(OC)CC(CCNC(c2occc2C2CC2)=O)N(C(=O)C=CSC)C1 c1(CC=O)scnc1-c1ccccc1.c1(C(N(CCC)CC)=O)csc(Cl)n1.N c1(OC)cccc2c1CCC(Nc1ccc3c(c1)C(=O)NC3=O)C2 O(NC(=O)C(C)C(C)NC(c1cc(C)sn1)=O)C(COC)COC c1(C(=O)NC(C2COCCO2)C)cc2c(cn1)OCCO2 N1(C(C2C(C)=CCS2)=O)CCC(C(=O)NCCc2cc(C)n(C)n2)C1(C)C C#CCC(C)(CNC(C1C2CC1N(C(c1cccnc1CC)=O)C2)=O)CO n1(CCC)ccc(=NC(=O)C(C)=CC2CC2)[nH]1.C12(CCC1)C(=O)NC2 CC1CC2CC2CC1C(=O)NCC1CCCN(C(C2(C)CS(=O)(=O)C2)=O)C1 c1(CNC(c2ccc(C(F)(F)F)cc2)(C)C)nccc2ccccc12 CC1CCc2[nH]c(=NC3CCC(C)(C)C3)nc(N3CCC(F)C3)c2C1 N1(C(c2c(CNC(C3(C)CCCC3)=O)occ2)=O)CC2OCC(CO)C2C1 C#Cc1cccc(C(=O)NCC2(O)CC(NC(c3ccc(Cl)cc3)=O)C2)c1F N1(C(C2CC(C)C2)=O)CC2CN(C(=O)Cc3ccno3)CC(F)(F)C2C1 N1(C(C(CC=C)C)=O)CC2(C1)CN(C(c1cncc(C3CC3)c1)=O)CCO2 C1CN=C2NC3=C(C(=NCCS1)N2)SCC3.C1(OCC)CC1 c1(CNC(CN(C(C2CCOC2)=O)CC)=O)cnccn1 [SH](=O)(=O)c1cccs1.N1(C(CCSCCC)=O)CCCC1CN(C(=O)CC)C Cc1cccc(CC(N2CCC(O)(C(C)CNC(=O)Cn3ccnc3C)C2)=O)c1 C1(C(=O)NCCOCC(=O)NC2(C(N)=O)CCC2)(CO)CCCCO1 C(=O)(CCCCSC)NC12CC(CNC(C3C(CC)CCC3)=O)(C1)C2 C(=O)(C(C)(C)CO)NC1C(CNC(CC(C)N2CCCC2=O)=O)COC1 c1(C(N(C2CCCN(C(C(CC#C)CC#C)=O)C2)C)=O)c[nH]c2cccc(F)c12 CCC(CNC(c1ccccc1)c1nnnn1C(C)(C)C)C(C)(F)F.C(CO)O N1(C(c2c(CC)nc(C)s2)=O)CC(NC(c2ccco2)=O)CC(F)(F)C1 N1(C(C(Cc2c(C)nc[nH]2)O)=O)CC(CNC(c2ncc(F)cn2)=O)C(O)C1 C=CC(C)(CCOC)C(=O)NC1CC(C)CN(C(c2cnnn2CC)=O)C1 c1(C(=O)NC(C(C)OC)C)ccc(-c2ccc(CN(CCC#N)C)cc2)cc1 C1(CCC(=O)NC(c2ccccc2)C(=O)N(CC=C)CC)CCCN1C C1(NC(C=CCOC)=O)CCC2(CCN(C(c3cc(C)n(C)c3C)=O)C2)C1 c1(-c2cccc(NCc3cc(OC)c(Cl)cc3)n2)cc(F)c(F)c(F)c1 CCCC(CC)CC(=O)NCC1(O)CCN(C(C23C4C5C6C4C2C6C35)=O)C1 C1(NC(=O)NCC(C2CCC2)NC(=O)NC2CC2)COCC1C1CC1 c1(C(N(C(CC(F)F)C(N2CCC(CO)C(O)C2)=O)C)=O)cn(C)c(=O)cn1 C(CN=c1nc(N(C)Cc2ccoc2)c2c([nH]1)CCCC2)C1C(C)CCO1 C(=O)(C1=C(C)OCCC1)NCC(CC(=O)NC(c1ncccn1)CC)C N1(C(C2CC23CCN(Cc2c(Cl)ccc(F)c2F)C3)=O)CCc2ncncc2C1 c1(C=O)ccc(C(=O)CF)cc1.N1(C(=O)N)CCCC1.O=CC.C1(CC)CC1 N1(C(CCCC2CCC2)=O)CC2CC(N=c3nc(C4C(C)(C)C4(C)C)[nH]s3)C2C1 O=C1CCCC(C(=O)NC2CCOCC2C(N2C(CO)CCC2CO)=O)C1 Cc1ccc(C(=O)NC23CC(CNC(=O)CC4CC4)(C2)C3)nc1C c1(CC(=O)NCC(C)=CC(=O)NCCCc2cn[nH]c2)cn(C)nc1C C1(C(N(CCCCN(C(C=C(COC)C)=O)C)C)=O)SCCCS1 Cc1cccc(O)c1C(N1CC2CC(NC(=O)Cc3c(C)nn(C)c3C)C2C1)=O c1cc(C(c2nnnn2CCCF)NCC2CCCCO2)c2c(c1)CCOC2 C(C)(C(C(=O)NC(C)Cc1cccs1)NC(c1c[nH]c(=N)o1)=O)OC c1(C(=O)NCC(CC)NC(C(CC)O)=O)cc2cnn(C)c2s1 c1(OC)nc(=NCC2CN(C(C3(O)CCOC3)=O)C2)nc(OC)[nH]1 S(=O)(=O)(c1ccc(CNC(C2(C#N)CC(C)C2)=O)cc1)NCC N#CC1CC12CCN(C(C1CCN(C(=O)c3sccc3CO)O1)=O)CC2 C1(CCC)CN(C(c2n[nH]cc2OC)=O)CCN1C(=O)CCc1ncco1 N1(C(C(C)(C)C(F)F)=O)CCCN(C(c2cocn2)=O)C(CO)C1 c1(C(N(C)Cc2cccc(OC(F)F)n2)=O)nc(Br)ccc1N N1(C(CCCc2onc(C)n2)=O)CCC(NC(=O)C(c2cscn2)N(C)C)CC1 CC(C)CS(=O)(=O)CCC(=O)NC1CCCC1NC(c1cscn1)=O C(CCCCCNC(=O)C=CC(C)CC)N(C(c1c(CC)onc1)=O)C N1(C(=O)Nc2cccc(C)c2)CCC2CN(C(c3c[nH]c(C)c3)=O)CCC12 c1(C(N2CCCC(C)(NC(C3OCCC(C)C3)=O)C2)=O)ccc2c(c1)C=CCC2 c1(C(N2CCC(N(C(CCN(CCCCC)C)=O)C)C2)=O)cncc(C2CC2)c1 C1(C(=O)NC(C(N(OC)C)=O)C)N(C(=O)C(C)OC)CC12CCCC2 O=C1CCC(C(=O)N)CN1.c1cn(C2CCN(C(=O)CSC(F)(F)F)C2)nn1.C Cn1ccc(=O)c(C(=O)NC(CC(=O)NCC2(Cl)CC2(F)F)C2CC2)c1 C12(C(N3C(C(C)O)CC3)=O)CC(CCO1)N(C(=O)C(C)n1ccnc1)C2 n1(CC)nc(C(C)C)cc1C(=O)NC(C)CO.c1(C(=O)N)ccc(C#N)[nH]1 N1(C(C2(C)N(C)CCC2)=O)CC(C)CC(C)(C)C1.c1(C=O)cc(C(N)=O)co1.N n1(CCS(C)(=O)=O)nc(Cc2ccc(Br)cc2)nc1-c1cnnc(O)c1 C#CCC(C(=O)NC1CCN(C(=O)CNC(=O)C)C1)C1CC1.C(C)=O.N C1(C(=O)NCC2CC(SC)C2)C=CCCN1C(=O)CC1CC(C2CC2)C1 C12(CN(C(C(C3CCN(C(=O)C(O)C4CC4)CC3)C)=O)C)CCC(CC1)C2 c1(-c2cc(C)c(F)nc2)ccc2nc(C(N3CC(NC(=O)C(C)C)C3)=O)cn2c1 Cc1cc(NCC=CCNC(=O)C2=CCCCC2)n2nc(C)nc2n1 c1(C(=O)NCC2C(NC(c3ccc(CC)o3)=O)C2)oc(C)nc1CC c1(NC2C3N(C(c4ccc(C#C)cn4)=O)C(CC3)CC2)cnc2ccccc2n1 N1(C(CC)=O)CCC(c2cncn2C)C1.N(C)(S(N)(=O)=O)CC=O.C#CC.O C(=O)(CS(=O)(=O)CC)N1CCC(C(=O)N)(COC)CC1.C1CCC(O)C1.C C12(CC(=O)NCCC3N(C(C4C(C)CCC4)=O)CCC3)COC(C)(C1)C2 Cc1cc(C(=O)NC2CCC2CNC(=O)CCCn2cc(C)cn2)cc(O)c1 C(=O)(C(O)C(C)C)N.c1(N(CC(N2CCC2C)=O)C(=O)OC)ccccc1 CC1CC(F)(F)CCN1C(c1n[nH]c2c1CN(C(=O)CC1CCSCC1)C2)=O C(=O)(N=c1ncnc2[nH][nH]cc1-2)c1c(-c2cc(OC)c(CO)cc2)cncc1F C1(C(c2ccccc2)C(=O)COC(c2ccccc2)C2CC2)CS(=O)(=O)C1 c1(OC)cc(-c2nc(CCO)nn2Cc2ccccn2)ccc1OCC(=O)OC Cc1cnc(C=CC(N2CCSCC2CCNC(=O)Cc2cscn2)=O)[nH]1 C1(NC(C(C)n2cccc2)=O)C2CC3C(C2)C13C(=O)NCc1ncccn1 c1(NC(C)Cc2cc(Br)ccc2F)c2c(nc3ncnn13)CCOC2 c1(C(N2CC(NC(c3cnc(C)[nH]3)=O)C(C)C2)=O)ccc2c(c1)OCC(=O)N2 c1(C(N2CCC(OCC3CC3)C2)=O)cnn2c1CN(C(C1(Br)CCC1)=O)CC2 N1(C(C(C)(C)C)=O)CCCC(n2cc(C(N3CCOCC3)C3CC3)nn2)CC1 c1(C(N2C(CNC(c3c(N)cc(Cl)nc3)=O)CCCC2)=O)occ2c1CCCC2 Cc1ncnc(C(N2CCN(C(C3CSCCS3)=O)C(CCO)C2)=O)c1C CCCC(C)CC(=O)NCC(C)CN(C(=O)Cc1ccc(C(=O)OC)nc1)C Cc1nccc(C(=O)NCCOC2CCN(C(=O)CCC(=O)NCC)C2)n1.S c1(C=O)ccncc1C(F)F.c1(C(C)C(=O)NC2(CC)CC2)ccc(Cl)cc1.N CCC(C)CC(=O)NCC1(C)CCN(C(c2cc(C(F)F)no2)=O)C1 n1(CCOCC)nc(CCOC)nc1-c1csc(Br)c1C C1(C(=O)NCC(C#C)(C)C)CCCC(NC(C2(CC)CNC(=O)C2)=O)CC1 C1(C=O)CC(C)(C)CCN1C(c1cnc(O)c(C)c1)=O.C(C)(CC(C)C)OC.N N1(C(C2C(C(=O)OC)CCO2)=O)CCC(CCNC(=O)CC(C)F)CC1 Cc1cc(=O)c(C(=O)NC2CCN(CCCc3c(F)cccc3F)C2)cn1C Cc1ncc(C2=CCNCC2)cc1NC(c1ccccc1-c1nc[nH]n1)=O Cc1c(C(=O)O)cnc(OCCC(=O)OC2CCCN(S(C)(=O)=O)C2)c1C c1(C(N(C(C(=O)OC)COC(C)C)C)=O)sc2ncc(Br)cc2c1N c1(C(N2C(C)CN(C(=O)CCCCCBr)CC2)=O)ccc([N+](=O)[O-])c(Cl)c1 Cc1cc(Br)ccc1C(=O)NC1C=CC(C)C1.c1(CC(=O)N)c(C)cnn1C c1(OC)nc(C)ccc1-c1ccc(NCc2cc(C)nn2C)nc1 c1ccnn1C.C(CNC(=O)CO)(CC)N(C(=O)C=O)CCC.C(C)C C1(CC=O)CCC(=O)NC1=O.C1(CC#C)(C(=O)N(CCC)CC)CCCO1.N N1(c2c(OC)c(Cl)ncn2)CCC2C(CCCN2C(=O)COCCCC(C)C)C1 N1(C(COCc2onc(CC)n2)=O)CCC(n2cc(C3(O)CC3)nn2)C(O)C1 c1(OC)ccc(C(O)CN2CCC(CC(=O)NCCSc3ccccc3)C2)cc1 N1(C(C2CC(C)CN2C(=O)C(C)CC(F)F)=O)CCCN(CCO)CC1 CC(CC(=O)NC1(CCNC(=O)C(CO)c2ccccc2)CC1)C(C)(C)C N1(C(C2CCNC2)C)CCC(C(c2ccccc2)=O)CC1.C(=O)CCc1ccsc1.C N1(C(C(CC)C(C)C)=O)CC2CC(C)N(C(c3csc4cncn34)=O)C2C1 C1CC(C)(C)CN1C(=O)CCn1ccnc1.C1(C(=O)N)(COC)CCC1.C C(CCCCCNC(C1CC1c1ccco1)=O)N(C)C(C1(C(F)F)CCCO1)=O c1(NC(c2cccc(O)c2F)=O)cc(Br)ccc1-c1nn[nH]n1 CC(C(=O)NCCC(=O)NC1CC1)(C1CCC1)NC(=O)CCC1CCCCO1 c1(C(C=O)N(C2CCS(=O)(=O)C2)CC=C)cc(F)cc(F)c1.c1ccccc1.N C1(C(=O)NCC2COCCN2C(c2cc(O)cc(Cl)c2)=O)Cc2ccccc2O1 c1(CC)cc(C(=O)NCCCCC(C)NC(C2OCCC2(C)C)=O)ccn1 C1(CNC(C=CC(C)C)=O)CN(C(=O)C)CC1O.c1(C=O)cc(Cl)ccn1 CC1CN(C(=O)C(O)CC(F)(F)F)C(C)CN1C(=O)CC1CCSC1 C1(O)(CC)CCN(C(=O)C(F)n2cccn2)CC1.O=CCNC(=O)C1CC1.N Cc1ccc2c(c1)SC(C(=O)NC(C)CN(C)C(c1cc(F)c(C)cc1F)=O)C2 c1(C(=O)Nc2ccc(C(C)O)cc2)cc2c(-c3c[nH]nc3C(F)F)cncc2s1 C1(C(N(C2CN(C(c3cc(=O)n(-c4ccccc4)[nH]3)=O)C2)C)=O)C2CCCOC12 N1(C(c2c(C)coc2)=O)CC2CC(NC(=O)CCCNC(N)=O)C2C1 C(=O)(C(CCOC)NC(=O)Cc1cccnc1F)NCC(=O)NCC=C c1(C(N(C2CCC(NC(c3ccccc3)=O)C2)C)=O)cc(=O)cc[nH]1 CC1CCCn2cc(C(=O)NCC(C3CCCC3)NC(=O)C(C)(C)C)nc21 Cc1ncc(C(N2CCCN(CCNC(c3csc(C)c3)=O)CC2)=O)c(C)n1 c1(CC)nncn1NC(=O)c1ccc(NC(c2ccccc2)=O)nc1C c1(OC)ccc(CC(N2CC(NC(=O)C(N)=O)CC(C)C2)=O)cc1OC C1(NC(c2cnc(C(C)(C)C)o2)=O)CN(C(C2(O)CCSC2)=O)CC(F)(F)C1 N1(C(Cc2nc(C)[nH]n2)=O)CCN(C(C2CCCN2C(C)C)=O)C2COCC12 c1(NC(C)=O)ccc(Cl)c(C(=O)N)c1.C1(C=O)CC12CCCOC2.C(C)(C)C c1(CNC(c2ccccn2)C)nnnn1Cc1ccco1 C1(C(N2CCC3CN(C(c4c(CC)ccs4)=O)CC32)=O)CCc2ncncc2C1 Cc1ccc(N(C(=O)CC2CC=CCC2)C(=O)CN2CCC(N(C)C)CC2)cc1 C(=O)(C1=CCC(NC(=O)C(F)(F)C(C)O)C1)N(CC#C)CCF c1(C(=O)NCCN(C(=O)CC2CCC(C)CC2)CCC)cn2ncccc2n1 N1(c2nccc(OC)n2)CCN(C(c2ccn(-c3ccccc3)n2)=O)CCC1C C=CCC(CNC(=O)C#CC1CCOC1)C(=O)NOCCOCCF N1(C(C(CC(F)F)NC(=O)CCCF)=O)CCC(C2CCC2)CC1 c1(C(=O)NCC(C)N(C(C2CNC(=O)C2)=O)CC)c(C)nn(C)c1C c1(C(N2C(C)CC(CNC(CCCOC)=O)C2)=O)cc2c(C)ccc(C)c2[nH]1 C(=O)(C1CC(=O)c2cccc(OC)c21)NCC(CNC(C1(C=C)CCC1)=O)O c1cn(C(C)C)nc1C=O.C1(C(CC)NC(=O)N)CCCCCC1.C1CC1.C N1(C(c2c(C)cnnc2)=O)CC2CC(C1)CN(C(=O)Cn1cnc(C(N)=O)n1)C2 C(=O)(C1Cc2ccccc21)NCCCCC(C)NC(c1ccn(CC(C)C)n1)=O c1(C(N2C3(CN(C(C4(C(C)C)CCC4)=O)C3)CCC2)=O)ccc(Br)c([N+](=O)[O-])c1 Cc1ccc(F)c(C(N2CCC2C(=O)NOCC2CC2)=O)c1 N1(C(c2c(C)n(C)nc2)=O)CC(CC(=O)NC(c2ccncn2)C)C2(CC2)C1 C(=O)(C#CC1CCCO1)N(C(C)C)CCNC(=O)COc1cc(F)ccc1Br n1(CC(N2CCC(C)(C)C2)=O)ccc2ccccc12.c1(CC(=O)N)n[nH]c(=N)s1 C1(C(N(C2CCCN(C(=O)Cn3ncn(C)c3=O)C2)C)=O)CCCCC1(F)F C1(C(C)N(C(=O)CCCn2cc(-c3cnc(O)nc3)nn2)C)CCN(C)CC1 c1(C(=O)NC2CCC(C)(CNC(C3C=CCS3)=O)CC2)cccc2ccnn12 N1(C(c2c(C(C)C)ocn2)=O)CC=C(c2ccncc2)CC1 c1(C=O)cc(S(N)(=O)=O)c(C)s1.CCC(C(=O)NC12CC(C1)C2)SC.C C1(CNC(CN(C(=O)CCn2cc(C)cn2)CCC)=O)CCCC1N(C)C c1(C(=O)NC(CNC(C(CSC)OC)=O)(C)C2CCC2)ccc(N)cc1F N1(C(C2C(CC)C2)=O)CC2(C(=O)NC3(C)CCC(C)C3)CCC1CC2 c1(C(N2C(CNC(c3ncccn3)=O)CC2)=O)ccc(N2CCOCC2)nc1 C(=O)(CCN1CCCO1)N1CCC(C(N(CC(C)O)C)=O)CC1 N1(C(c2ccc(C)o2)=O)CC(N(C(=O)C(=CC2CCCCC2)F)C)C(F)C1 N1(C(c2c(Cl)nc(OC)s2)=O)CCN(C(C2(S(C)(=O)=O)CC2)=O)CC1CO c1(C(=O)NCC(CNC(c2ccc(OC)nn2)=O)O)cc(F)ccc1Br C(CC(C)(C)C)(C(=O)N1CCN(Cc2cn(Cc3csc(Cl)n3)nn2)CC1)OC N1(C(CN2CCCC(CC)C2)=O)C(CNC(=O)CC(F)(F)F)CC2COCC12 N1(C(=O)CC2CCCCC2)CCC(N(C(=O)C(F)n2cccn2)CC2CC2)CC1 C1(C(=O)Nc2cc(CCC)no2)CC2(C1)CN(C(c1nccnc1Br)=O)C2 S(=O)(=O)(c1c(Cl)cccc1Cl)N1CC(C)C(NCc2ncc[nH]2)C1 c1(C(N(CCCN(C(=O)C2=CCCS2)C)C)=O)cc(Cl)c2c(c1)OCCCO2 N1(C(C(C=C)CC)=O)CC2CCC2(CC(=O)Nc2cnc(Cl)c(C)c2)C1 C(=O)(CCCC(=O)N1CCC(CO)(NC(=O)CCCc2cncs2)C1)NCC C1(C=O)CN(C)CC(C)O1.C#CC(CNC(C1(C)CC1)=O)CC1CC1.N N1(C(c2c(C)sc(Cl)c2)C(=O)NCC2CCCO2)CCc2c(ncn2C)C1C C1(NC(c2nc(CCCC)sc2)=O)CCN(C(=O)C=CCF)C1C(C)(C)C C1(CNC(CCc2n(C)ccn2)=O)CCCN(c2cnc(C#N)cn2)CC1 c1(CCC(=O)NCC(CO)NC(C(CC)SC)=O)c(C)nc2nnnn2c1C N1(C(c2c(CC)nn[nH]2)=O)CCC2OCCN(C(=O)CC3CCCC3)C2C1 CCN=c1cc(-c2nc(-c3ccco3)n(CCn3c(C)csc3=O)n2)cc[nH]1 C(CC(F)F)(C(=O)NC(c1ncn(C)n1)C)NC(C=NOC)=O N1(C(C2(OCC)CCCC2)=O)CCC(NC(=O)CC(O)CN(C)C)CC(O)C1 C1(CN(C)C(c2ncn(C)n2)=O)CCCC(NC(=O)CCOC2CC2)C1 c1(C(=O)Nc2nc(C)c(I)s2)[nH]nc2ncc(-c3cccc(C(F)(F)F)c3)cc12 c1(C(N(C)CC2CCN(C(C(CC)(C)O)=O)C2)=O)ccc(C)cc1SC C1CN(C(C2(F)CCS(=O)(=O)C2)=O)CC12CCOCC2.C1(F)(C(=O)N)CCC1 c1(C(=O)NCC2CC(NC(c3c(C)ccc(Cl)c3)=O)C2)cc(C)c(C)cc1N c1(NC(CC2N(C(C3C(OC)C3)=O)CCOC2)=O)ncc(F)cc1Cl C1(C(N2C(C(=O)NC)CCCC2)=O)CC2CN(C(=O)C(=O)NC3CC3)CC2C1 O=C(CCC1CCCO1)N=c1ccn(C2CN(C(=O)CN3CCCC3=O)C2)[nH]1 N1(C(C(C=C)(F)F)=O)C(CC(=O)NC(C)CC#CC)C2CCCC12 N1(C(CCNC(=O)OC)=O)CCCC(NC(C2(O)CCCCCC2)=O)C(F)C1 c1(C(=O)NC(C(CO)NC(c2c(CC)nn[nH]2)=O)C)cnc2c(c1)nnn2C N1(C(c2c(OC)cc(C)cc2)=O)CC2CN(C(c3ccc(F)o3)=O)CC2C1 N1(C(c2ccc(C(C)O)cc2)=O)CCC2CN(C(C3(F)CCCC=C3F)=O)CC12 N1(C(C(C)N=[N+]=[N-])=O)CCC(C2(NC(C3CC4(C3)CC4(F)F)=O)CC2)CC1 c1(OC)ccnc(OC)c1C(=O)NC1CN(C(c2ccc(O)cc2)=O)C1 S(=O)(=O)(C(C)CN=c1nc(N2CCCC(CO)C2)c2c([nH]1)CCCCC2)NC c1(OCc2c(Br)cc(CC)s2)c(Br)cc(F)cc1[N+](=O)[O-] CCC(O)C(C)C(=O)NC1(CNC(=O)CCc2cc(F)ccc2F)CCCCC1 n1(CC)nc(C(=O)NC2CCN(C(c3cn(C(C)(C)C)nc3C)=O)CC2)cc1C c1(C(N2CCC(C(C)NC(CC=CCC)=O)CC2)=O)ncc2ccccc2c1N C1(CC(=O)NCCC)C(C)(C)C1(C)C.C1CCN(C(=O)C)C1.C1CCCOC1 c1(C(=O)NC(C2CCCC2)CNC(C(CCN(C)C)O)=O)c(Cl)nn(C)c1Cl C1(C(CNC(=O)Nc2c(C)noc2)=O)CCCC(C)C1 CC(C)CS(=O)(=O)CC(=O)N.C1CC(F)(F)CN1C(C1CN(C2CCC2)C1)=O CC1(C)COC(C(=O)NC2CN(C(=O)Cc3ccsn3)C(C)(C)C2)CO1 CC(C=CC(=O)NC1CSC1)NC(=O)COCCN(C)C c1(C=O)cc([N+](=O)[O-])c[nH]1.c1(CC)c(C(=O)NC)csc1C.C1CCC1(C)C C=CCC(C(=O)Nc1cnn(CC)c1C)NC(=O)CC1(OCC)CCC1 C1(N(C(c2c(OCC)ccs2)=O)CC)CCCCN(C(=O)CC(O)CC)C1 C1(C(N2CCCC2)=O)(COC)CCCOC1.C(C1CCCC1)=C(C(=O)NC)C.C c1(C(=O)NCC(Cn2cc(-c3cc[nH]n3)nn2)OC)ccc(C(=O)O)s1 C1(C(N2CC(C)(C)C(NC(c3cccc(O)c3)=O)C2)=O)CCCC(F)(F)CC1 C1(C(=O)NC2(CNC(=O)C(=CC3CCCCC3)F)CC2)CC2CCC(C1)C2O c1ccc(C(=O)N(C)C)nc1.c1(C(C)=O)c[nH]c(C(=O)NOC)c1.N1CCNC1=O c1(Nc2cncc(C(=O)NCCN(CC)CC)c2)ncnc(CO)c1F c1(C(=O)NCCNC(C2(Cl)C(C)(C)C2)=O)cnc(-c2ccncn2)nc1O c1(C(=O)NC(C)C(N2CCCN(C3CC3)CC2)=O)ccc2n[nH]cc2c1 C=C=CCCC(=O)NCCC1CCCN(C(C2(C(=O)OCC)CC2)=O)C1 O=C(C1=NOC2COCC12)NC1CCCC(NC(=O)Cn2cnccc2=O)C1 C1(N(C)C(c2ccc3c(c2)CC3)=O)CCCC2CN(C(C3CCC(O)C3)=O)CC12 c1(NCC2(C)CC=CCC2)nc(N2CCC(C(F)C(N)=O)CC2)nc2sccc12 O=C(C1CCCCc2ccccc21)NCCCCCN=c1[nH]c(C2CC2)nc(=N)[nH]1 C(=O)(C(C(C)NC(c1sc(C)cc1C)=O)C(C)C)NCC(=O)OCC#C N1(C(=O)CS(=O)(=O)CCO)CCC2(CC1)CC(NC(C1(CO)CC1(F)F)=O)C2 N1(C(CCCCN(C)C)=O)CCC2CCCN(C(=O)CCn3ccnn3)C2C1 c1(C(=O)NC2C(NC(COCCCCCC)=O)CCC2)cc(OCC)ncc1Br C1(NC(=O)Cc2cnccn2)COC2(CCN(C(c3cccnn3)=O)C2)C1 N1(C(c2cc(=NC)[nH]cc2)=O)CC(C(=O)Nc2cnc(SC)nc2)C2(CCC2)C1 Cn1cc(C(=O)NCC2CN(C(=O)CCn3ccnc3)C2)c(=N)[nH]1 Cc1onc(-c2ccccn2)c1C(=O)C=Cc1ccc(Cl)s1 C1(NC(c2c(C)cc(=N)[nH]c2)=O)C(C)(C)C(NC(=O)C(C)C(F)F)C1(C)C C1(NC(C(CC)C2CCOCC2)=O)CCCN(C(C2(c3cccnc3)CC2)=O)C1 c1(-c2scc(CC(=O)Nc3ccc(Cl)c(O)c3)n2)c(Cl)cccc1Cl C1(NC(CSCCOC)=O)C(C)(C)C(NC(c2n[nH]cc2Cl)=O)C1(C)C N12CCC(F)(F)C(C1)CCC2=O.C(CCCN=[N+]=[N-])C1C(OC(C)(C)C)C1 CCC1(CNC(N2CCOCC2c2ccc(O)cc2)=O)OCCc2ccccc21 N1(C(C2CC(C#C)(O)C2)=O)CCCC(CC)CC1.C(c1nc(C)cs1)=CC(=O)N C#Cc1ccc(C(=O)NCC2CC3(CC3)CN2C(=O)C(C)COC)cn1 N1(C(C2CC(OC)C2)=O)CCN(C(=O)Cc2csc3nc(C)cn23)CCC1C c1(C(=O)NCC2CCCN2C(=O)C(O)C2CC2)cccc2c1CCCCC2 N1(C(Cc2cn(C)nc2)=O)CC2CC(C(=O)NC3CCCCCC3F)(C2)C1 C12(NC(c3cnc(-c4cccnc4)s3)=O)COC(CS)(C1)C2 c1(C(=O)NCC(CNC(c2ccc(CC)[nH]2)=O)O)ncncc1C N1(C(CCCCC)=O)CCC2(CCC(NC(=O)C(C)C(C)(F)F)CC2)CC1 CCC(C(=O)NCC1(F)CCCN(C(=O)COc2ccsc2)C1)C(F)(F)F c1(CNC(c2csc3cccnc23)=O)ccc2c(c1)CCCO2 CC12CC(CCO1)N(C(=O)C(F)CC1CN(C(=O)Cn3cccc3)C1)C2 N(C1CCCc2cc(F)ccc21)(C1CC1)Cc1cc(C#N)c(F)cc1F C(=O)(C(C)CC(C)(C)C)NCC(CO)NC(C(C)=CC1CC1)=O CC1CC(N=c2[nH]c3c(c(=NCc4ncc5c(n4)CCC5)[nH]2)COCC3)CCS1 N1(C(c2cncn2C)C(=O)Nc2c(OC)cccc2)CCC(C2CCC2)C1 c1(OC)nc(=NCC(C)CNC(=O)COC2CCCC2)[nH]c2[nH]cnc12 c1(NC(N(CC(c2ccc(O)cc2)O)C)=O)c(C2CC2)nc2sccn12 N1(C(C2(C#N)CC2)=O)CC(N=[N+]=[N-])CC1C(N1CCCC(CC(N)=O)C1)=O C(N=c1nc(N(CC2=CCSC2)C)c2c([nH]1)COC2)c1cc(C)sc1C N1(C(c2ccc(CC)c(N)c2)=O)CCC(NC(c2nn(C)nc2C)=O)CC(O)C1 C1(NC(CC2C=CC(NC(c3c(CC)ocn3)=O)C2)=O)CCCCC12CC2 C=C(C)CN=C(NCC(O)(COC)COC)N1CCSC(c2ccccc2)C1 c1(SC)ncc(C(=O)NCC(C2CC2)NC(=O)C=Cc2ccc[nH]2)n1C Cc1c(N)ccc(C(N2CC3CC2CN3C(C23CCC(CC2)C3)=O)=O)c1C CCC(CC)C(F)C(=O)N1CC(OCCNC(=O)C(C)C2(O)CCC2)C1 C1(C(=O)NC2CC3CN(C(C(C=C=C)C)=O)CC2C3)Cc2ccccc2CO1 N1(C(C2(CC=C)CN(C(c3cnncc3OC)=O)C2)=O)CCCC2(C)CCCC12 C1(NC(C2CCC(=O)N2)=O)CN(C(c2cc(F)cc(F)c2)=O)C2(CCOCC2)C1 c1(OCC)cc(CONC(=N)Cc2ccc(F)nc2)ccc1[N+](=O)[O-] C=C(CNC(=O)C(C)O)CCNC(=O)Cc1n[nH]c(C)n1.CC(F)(F)F N1(C(C2CC(C)(CC)C2)=O)CCC(CC)CC1.C1(CC(=O)N)CC2C=CC1C2 Cc1cc2nc(Cl)nc(N3CCC(NC(C4(F)CCOC4)=O)C(O)C3)c2s1 C1(C(=O)NCC(C2CCN(C(c3c(SC)csc3)=O)CC2)C)Cc2cscc2C1 c1(C(=O)NCCC2CN(C(=O)CCOC3CCC3)C2)c[nH]nc1C(F)F Cc1c(C(N2CC(NC(c3ccc(Cl)cc3F)=O)C2)=O)cn2[nH]cnc(=O)c12 C(C(C)CC(F)(F)F)NC(C(CCOCC)NC(c1ccco1)=O)=O C=CCC(C)(C)CC(=O)NC1(C)CN(C(=O)C(c2ccccc2Cl)C)C1 C(=O)(C1CCCc2ncccc21)N1C(CNC(=O)Cc2cocn2)CC(F)(F)C1 CCC(CCC(=O)NCc1ncnn1C)NC(C1(SC)CC1)=O N1(C(c2ccc(CC)s2)=O)C2CCC1CC(NC(c1c(N)cc(Cl)cc1F)=O)C2